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216,c1(C(N(CCCNC(=O)C2CC2)CC)=O)nc(C(C)C)ncc1Cl 217,C(C(C(F)(F)F)N1CCN(C(c2ccoc2)=O)CC1)NC(C1CNC(=O)N1)=O 218,C(=O)(CC1(C(=O)NCCNC(C)=O)CC1)N(CCC)CCOC 219,Cc1cc(-n2cc(CNC(=O)Cc3csc(-c4ccncc4)n3)nn2)ccc1F 220,CC1(C)CC(CNC(=O)COC2COC2)N(C(C2CCC2)=O)C1 221,N1(C(CC(C)O)=O)CC2(CNC(c3csc(-c4ncc[nH]4)n3)=O)CC1CO2 222,C1(CCNC(=O)CCc2cccs2)CCCCN1C(c1coc(C(F)F)n1)=O 223,C(=O)(C(CC(C)(C)C)NC(=O)CC(C)(F)F)N(CC(CN(C)C)O)C 224,N1(CCC(=O)NCC(=O)NCCO)CCCC1=O.C12C(C1(F)F)C(=O)N2 225,C(CC(C(=O)N1CCC(OCCC)CC1)NC(C1CCOC1(C)C)=O)=CC 226,c1(COC)nc(NCCCc2c[nH]c(=N)s2)cc(N(CCCC2CCOC2)C)n1 227,C(=O)(C(C)(C)CCCN=[N+]=[N-])N1CCC(C(NC(C(CC#C)O)=O)CC)C1(C)C 228,C=CCCCC(C(=O)NCCN1CC2CC2C1)NC(C1CCCOCC1)=O 229,c1(C(=O)NCC(CC(C)C)NC(c2cc(CC)oc2C)=O)csc2ccccc12 230,CCC(C)(F)C(=O)N1CC(NC(=O)Cc2cc(-c3ccc(Cl)cc3)on2)C(C)C1 231,C1(NC(C2C(C=C)OCC2)=O)CC12CCN(C(c1ncoc1CC)=O)CC2 232,C=CC(C)(C)C(=O)NCC(c1ccccn1)Sc1ccc(Cl)cc1 233,C(CCC(=O)N(C1CC(C#N)C1)CC(=O)NC(c1nc(C)no1)C)NC(=O)OC 234,CC(C)C(CC(=O)NC1(C)CCN(C(C2(c3cccs3)CC2)=O)C1)C(C)C 235,c1(NC(C2CCN(CCC)CC2)=O)ccc(I)nc1Cl.N1(CC)CCOCC1 236,Cc1ccc2sc(C(=O)NCCCCN(C(=O)C(O)CC3CC3)C)c(C)c2c1 237,c1(OC)cc(CN(CC(c2ccccc2)C)C(C)C)c(O)cc1F 238,C(C(C(=O)NC1CCC1)N(C)C(C1(S(C)(=O)=O)CC1)C)(C1CCC1)OCC 239,c1(NC(=O)OC(C)(C)C)cccc(CSCCCCCC2CC2)c1 240,c1(C(N2CC(CC3CC3)CC(C)C2)C(=O)NC(CC)C)cccn2ccnc12 241,N#CC1CN(C(=O)C(C)Oc2ccccn2)CC1NC(c1ccnc(Br)c1)=O 242,c1(C(=O)NCC(CN(C)C(c2c[nH]nc2C2CCC2)=O)O)cnccc1N(C)C 243,C(C(N=c1[nH]c(N2CCOC(c3cnn(C)c3)C2)nc2c1SCC2)C1CC1)OC 244,Cc1nn(CC(=O)NC(C)(CNC(C2CC2(Cl)Cl)=O)CO)c(=O)o1 245,n1(CC)ccc2cc(CN3CCN(C(CCC(=O)OC)=O)CC3C(C)C)ccc12 246,CC(C)CCC(C(=O)NC1CC2(C1)CC21CCC1)NC(=O)CN(C1CCCC1)C 247,N1(C(c2cn(C(C)C)nn2)=O)CCC(C)(NC(=O)CCC2OCCO2)C1 248,Cc1cc(NC(C2OCCC2(C)C)=O)ccc1NC(=O)C(C)C(C)C 249,c1(NC(C2(OC)CCN(C(=O)OC(C)(C)C)C2)=O)nc2cc(Br)cnc2[nH]1 250,c1(C(N(CC(CNC(Cc2cc(C)on2)=O)O)C)=O)cn2cc[nH]c(=O)c2n1 251,c1(OC)cc(C#N)ccc1C(=O)NCC1CC1CNC(C1(C#N)CC1)=O 252,CC1(O)CC(CNS(=O)(=O)CC2CCCOC2)C1 253,N1(C(c2c(CC)nc(=N)[nH]c2C)=O)CC2CCC1CN2C(=O)CC1OCCC1C 254,N1(C(C(C)(C)CC#N)=O)CCC(C(=O)NC2CC3CC4C(C3)C24)C(C)(C)C1 255,Cc1cc(F)ccc1C(=O)NCCC(O)CNC(C12CCCC1(C(N)=O)C2)=O 256,c1(CCNC(C(=O)NCCC2ON=C(C)C2)=O)c[nH]c(=N)nc1O 257,C1(C(N(CC(=O)Nc2ccncc2Cl)C)=O)CCCCCCC1 258,C1(NC(C2CC3CCC(C2)S3)=O)CC2CN(C(=O)C(F)(F)C3=CCCC3)CC12 259,CC(Cc1nccn1C)N=c1[nH]c(=NCC2(C)CCOC2)[nH]c2c1COCC2 260,C(=O)(CCCCNC(=O)Cc1cc[nH]c1)N1C(C(=O)OC)C=CC1 261,Cc1ccc(Cl)c(C(=O)Nc2ccc(C(=O)Nc3ncnc(Cl)c3Br)cn2)c1 262,CC(CC(F)(F)F)C(=O)NC1CCCC(N(C(=O)CSc2cccc(Cl)c2)C)C1 263,CC(C)(CCCC(=O)N1CCC(O)(CC(N)=O)C1)NC(=O)Cc1ccc(O)cn1 264,CCC(CC)(C(=O)NC1CCC(CNC(c2cc(N)ccc2O)=O)CC1)OC 265,c1(N(C(c2ccc(C(N)=O)cc2)C(=O)NCCCOCC2CC2)C)ccc(Cl)cc1 266,C1(N(c2cccc(F)c2O)C(COCCC=C)=O)C2CC3CN(C(=O)CO)C1C3C2 267,N1(C(C(C2CCOCC2)SC)=O)CCC(C2(NC(C3CC3(C)C)=O)CC2)C1 268,c1(OC)ccc(CNCC2CCC(NC(=O)Cc3ccc(C)cc3C)CC2)c(Cl)c1 269,N1(C(CCNC(=O)OC)=O)CC=CC1(C)C(=O)NCCc1ccc(O)cn1 270,C=CC(CC)CC(=O)NCC1CCCCN(C(=O)Cc2ccccc2O)C1 271,N1(CC(=O)N(CCCC)CC2CC2)CCC(C(=O)N(C2CCCO2)CC)CC1 272,C(=O)(CCCCCF)N(CCOCCOC)CCCC(C)O.C1C(=O)N1 273,C1(CC)C(=O)N(C)CCN1C(C1COCC1NC(c1cc2ccccc2[nH]1)=O)=O 274,CN1CCC(C(=O)NC2(CCNC(=O)CC(=O)Nc3nccs3)CCC2)C1=O 275,C1(C)(C(N2CCC(C(C)NC(c3ccc(C)o3)=O)CC2)=O)CCCNS1(=O)=O 276,c1(S)ccc(CCF)cc1.C1(N(C)C)C=CC(C(=O)NC(CNC=O)C2CC2)C1 277,c1(C(=O)NCCCCNC(c2ccc(F)cn2)=O)cc([N+](=O)[O-])cc([N+](=O)[O-])c1 278,C(C)(CO)(C(=O)NCCCc1nncn1C)NC(C(C)C1CC1)=O 279,C=CC(CC)C(=O)NC(c1ccccc1)C(=O)NCC1CCN1CC 280,N1(C(c2cc(C(C)(C)C)on2)=O)CCCC2CCN(C(=O)C3=CCCS3)CC12 281,c1(C(CNC(Cc2nc(CC)[nH]n2)=O)O)cc(Br)ccc1OC 282,S(=O)(=O)(c1ccc(Cl)c2ncccc12)N1C2CS(=O)(=O)C(C2)C1 283,C(CN=C(NC(c1cc(Br)ccc1F)C)NC1CCCCC1)OC(C)C 284,CCC(C(=O)NCC(C(=O)NCC(c1ccsc1)C)C(C)(C)C)C(C)(C)CC 285,N1(C(C=C(CC)C)=O)CC2CC(NC(=O)CN3C(C)CCC3C)CC(C2)C1 286,C(=O)(C1=CC2CCCCCC12)NC1(C)CCN(C(=O)CC2CC(=O)C2)C1 287,C(c1ccco1)=C(C)C(N1CC(CF)(NC(c2cnn(CCF)c2)=O)C1)=O 288,c1(C(=O)NCC2CCCN(C(CC3CC(CC)C3)=O)C2)ccc(=N)[nH]c1OC 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307,Cc1ccc(F)c(C(N2CC3CC2C3NC(=O)COC2(C)CCOCC2)=O)c1F 308,CCCC(O)(CCC)CC(=O)NC(CCC(=O)O)c1cccc(OCC(=O)NC)c1 309,c1(NC)ccc(C(=O)N(C)CC2CCCN(C(=O)Cn3ncccc3=O)C2)nc1 310,CC1(C(=O)NCCCC2CCCN2C(=O)CCCN2CCOC2=O)CC2CCC1C2 311,N(S(=O)(=O)N(C)C)CC(=O)N(CCNC(=O)Cc1cnccn1)CC 312,c1(CC(=O)NC(C2CCCCN2C(c2cccnc2CO)=O)C)ccc(O)nc1 313,N1(CCCCCc2cn(CCCNCC)nn2)CCN(C(=O)C(C)O)CC1.CC 314,S1(=O)(=O)C2=CC=C(C(F)=C2)N1.C12(CN3CCC(ON)C3)CC3CC1C2C3O 315,C=CCCCC(C(=O)NCc1cc(C)on1)NC(c1cc(C)c(C)[nH]1)=O 316,c1(C(N2CCN(C(=O)CC3CC34CC4)CC2C2CCC2)=O)cncc2c[nH]nc12 317,C1(C)(OC)CCCN(C(=O)Cn2cc(C3(O)COC3)nn2)C1 318,CC1(CNC(=O)CC2CC2(Cl)Cl)CC(F)(F)CN1C(C1CCOC1)=O 319,c1(C(N2CCCCC(NC(C(CC=C)(F)F)=O)C2)=O)cccc2c1NCC2 320,C(=O)(C(=O)C(C)(C)C)N1CC(CNC(CN2CC(C)(C)C2)=O)(OC)C1 321,N1(C(C2C(C)(C)COC2)=O)CCc2[nH]nc(CNC(=O)CC3(C)CCCO3)c2C1 322,c1(OC)ccc(F)c(C(N2CCN(C(=O)Cc3csc(NC=O)n3)C3CC23)=O)n1 323,O=C(C#CC1CCCCC1)N(CCCNC(C1(C(F)(F)F)CCCCO1)=O)CCO 324,c1(C(=O)NCC(C)NC(c2ccn(C)c2)=O)cc2cccnc2s1 325,N1(CC2CCC(C)O2)CC2CC(NC(=O)CCc3ccnn3C)CC1C2 326,Cc1nccc(N2CCC(C)(C(=O)Nc3cccc(C(=O)N(C)C)c3)C2)n1 327,C1(CCC)CC(C(=O)Nc2csc(-c3cc(Br)cs3)n2)CCO1 328,C1(CN(C)C(C2(O)CC2(C)C)=O)CN(C(=O)C=CC2CCC2)CCO1 329,N1(C(CC2(NC(C(CSCCCC)O)=O)CCC2)=O)CCCC(C)(C#N)C1 330,N1(C(c2cc(OC)n[nH]2)=O)CC2CC1(C(=O)NOCCC(C)O)C2 331,c1(C(=O)NCCNC(CC(C)SC)=O)c(C)nn(CCO)c1C 332,c1(C(=O)NC(CCOC)CNC(=O)C(C)c2cc[nH]n2)nn2c(c1C)OCCC2 333,FCCN=c1[nH]c(N2CCCC2c2ccccc2)nc2c1CCC2 334,c1(C(=O)NCCC(C)NC(CCn2ccc(C)n2)=O)cc2c(s1)CCCNC2=O 335,N1(C(C=CCCC=C(C)C)=O)CC2CCC1CN2C(=O)Cc1ccccc1C 336,c1(C(N2CC(C)(NC(C3(C(F)(F)F)CC3)=O)C2)=O)ccc(=O)n(CC(F)F)n1 337,CC(C(=O)OC(C)(C)C)C(=O)NC1CN(C(c2ccc[n+]([O-])c2)=O)CC1C 338,c1(NCCC)[nH]c(=NCC2CCN(c3ccccc3)CC2)nc2c1cnn2C 339,C=CCCCC(C(=O)NCC1(COC)CCCC1)NC(=O)CC(C)C(=O)OC 340,CC1(C)CC(C(=O)NC(C2CCCC2)CNC(c2cc[nH]c2)=O)CC(C)(C)O1 341,c1(CC(=O)NCC(=O)O)cnn2c1CN(C(=O)CC1Cc3ccccc3O1)CC2 342,c1(SC)ccc([N+](=O)[O-])c(C(N2CC3CC(C2)CN(C(C2CC2C)=O)C3)=O)c1 343,c1(C(=O)NC(CCC)CNC(=O)C(C#N)C(C)(C)C)cc2c(=O)[nH]c(C)cn2n1 344,c1(C(N(CC(C)NC(C(CC=C)c2ccccc2)=O)C)=O)csc([N+](=O)[O-])c1 345,c1(NC(=O)CC2(O)CN(C(c3ccc[nH]3)=O)C2)cnc2ncnn2c1 346,N1(C(c2cc(CC)on2)=O)CCN(C(=O)COCC(=O)OC)C(CF)C1 347,N1(C(c2nnc(CC)s2)=O)CCCC(C2CC2NC(C2CCCO2)=O)C1 348,C1(CNC(C2CC(=C)C2)=O)C=CC(NC(=O)C(CC2CCCC2)OC)C1 349,c1(C(N2C3CC(NC(C(C=C)O)=O)CC2CC3)=O)csc2ccc(Br)cc12 350,Cc1ccc(C(=O)NC(CNC(c2ccc(C#N)s2)=O)CO)c(=O)n1C 351,C#Cc1ccccc1CNC(=O)C(C)(C)NC(c1coc(CO)c1)=O 352,N1(C(C2CN(C)C(=O)N2)=O)CCC2(C1)CN(C(=O)CC1CN3CCN1CC3)C2 353,C12(C(N(C(CCNC(c3cnc(C)n3C)=O)C)C)=O)CC3CC(CC(C3)C1)C2 354,C1(C2(NC(CSCC(C)C)=O)CC2)CCCN1C(=O)Cc1cc(C(F)(F)F)n[nH]1 355,N1(C(CC)=O)CCc2nc(CNC(c3ccc4ccccc4n3)=O)sc2C1 356,C1(OCCOC(C2(C)CC2(F)F)=O)CCS(=O)(=O)C1 357,C(=O)(CCCSCC1CCCO1)N(C(C)(C)CNC(c1ccccc1)=O)C 358,CCCC(C(=O)N(C)C(c1cn(-c2ccc(SC)cc2)nn1)C)S(N)(=O)=O 359,CCCC(C(=O)OC)C(=O)NC12CC(CNC(=O)Cc3coc(C)n3)(C1)C2 360,N(C1c2cccc(Br)c2CC1(F)F)C(c1c(OCC(C)C)nccc1)=O 361,CC1(CO)CN(Cc2cc(-c3cccnc3)nn2C2CC2)CCO1 362,c1(OC)ccc(F)cc1C(=O)C(=O)NCC(C)N(C(=O)C1=C(C)OCC1)C 363,c1(OC)cncc(CCC(=O)NC2CN(C(=O)C#CC3CC3)CC2O)c1 364,C(=O)(C1=C(Cl)CCOC1)NC(c1ccccc1)C(=O)NCc1cn(CC=C)nn1 365,C(=O)(CC(C)CC(=O)OC)NC1(CC(=O)NC2(CC(=O)OC)CC2)CC1 366,C(CN=c1[nH]cnc(C)c1C#N)C1N(C(CCC(=O)OC)=O)CCCC1 367,c1(CC(N2CCC(NC(CCC3C(C)C3)=O)C2C)=O)c[nH]c2cnccc12 368,C(=O)(C(O)CNC(c1sccc1CO)=O)N(CCOCCOC)C 369,C1(C(N(C(c2ccncc2)C)C)=O)C2CC(O)C(C2)N1C(C1CN(C)CCO1)=O 370,CCC(C)C(C)C(=O)N1CCCC1CN(C(c1cn(C(C)C)cc1C)=O)C1CC1 371,C(=O)(C(CNC(C1(CNC(C2C3CCC(F)C23)=O)CC1)=O)C(C)C)NC 372,N1(CC(N2CCCN(C(C3C=CCC3)=O)CC2)=O)CCCC(C(F)(F)F)C1=O 373,N1(C(C(C2CCCC2)OC)=O)CCC(C)C(CNC(=O)C=CCF)C1 374,O=C1NCC2CCCN(C(=O)C(O)C3CN(C(c4cncnc4O)=O)C3)C12 375,C=CC(C(=O)NCCn1cc(C(=O)N(C2(SC(C)C)CC2)C)cn1)OC 376,C(=O)(C1CCCn2c(C)cnc21)NCC1CCN(C(C2CC(=C)C2)=O)CC1(F)F 377,C(=O)(C1=NOC(C)C1)N(C1CCCN1C(=O)Cc1csc(NC=O)n1)CC 378,Cc1onc(Br)c1CC(c1noc(Cc2nncn2C2CC2)n1)C.N 379,c1(OC)cccc2c(C(N3CCN(C(=O)C(Cl)=CCl)CC3C(C)C)=O)cccc12 380,C(=O)(CCCCC(N)=O)N(C1CN(C(=O)C2=NOC(C)(C)C2)CC1(C)C)C 381,C1(C(=O)NCCc2c(C)nc[nH]2)CCN(C(C2(C)CC2)=O)CCO1 382,N1(c2nnc(C(N)=O)s2)CCOCC(CNC(=O)C(C2CC2)C2CC2)C1 383,C(=O)(C1Cc2cccc(Br)c21)Nc1c(F)ccc(C(=O)OC)n1 384,c1(C(N2CCN(C(c3c(C)ncs3)=O)C3C2C3)=O)cc(=O)c2ccccc2o1 385,N1(C(c2c(C)nc(C3CC3)s2)=O)CCN(C(=O)CC2(O)CCC2)CC1C(C)C 386,C1(NC(c2cc(C)ncc2)=O)CCC(O)CN(C(c2ccc(S(C)(=O)=O)s2)=O)C1 387,N1(C(CN(CC)CC)=O)CC(NC(c2cc(C#N)cs2)=O)C2(CC2)C1 388,c1(C(=O)NC2C3CN(C(C4COC4)=O)CC23)cccc2c1OCC2 389,c1(OCC(=O)NC2CCC(N(C(Cn3ccc(C)n3)=O)C)C2)ccc(F)cc1Cl 390,n1(CC)cnc2c(NCCS(=O)(=O)CC)nc(N3CCC(CCO)C(C)C3)nc12 391,C1(CC)C(=O)NCCCN1C(=O)C(c1ccnn1C)NC(=O)CC1CCSC1 392,CC(CN(C)C(C1(N(C)C)CCC1)=O)C(=O)NCCc1cscn1 393,N1(C(C(C)OC)=O)CCC2(CCC(NC(=O)CN3CCCCCC3)CC2)CC1 394,C1(C)(CNOC)CC(C(C(CCC2CN(C(CC=CC)=O)C2)=O)=O)C1 395,CCC(CC(=O)NC1CC(C)(NC(c2ccc(OCCOC)o2)=O)C1)SC 396,n1(CC)c(=N)[nH]c2cc(C(=O)NC3CC3NC(=O)CC(C)CCOC)ccc12 397,CC(CN(C)C)CC(=O)N1CC2C(NC(C3(C(=O)NC4CC4)CCC3)=O)C2C1 398,C1(F)(CNC(c2noc(CC)c2C)=O)CCCN(C(C2CC2(F)Cl)=O)CC1 399,Cn1ncc(CC(=O)NCCC(O)CNC(=O)CC2(N3CCCC3)CC2)n1 400,c1(C(C(N2C(CNC(C3(C=C)CCC3)=O)CCC2)=O)OC)cc(F)c(F)c(F)c1 401,C1(CNC(C(C)(C2CC2)NC(C)=O)=O)CC(C)(C)CN1C(C1CCC(C)C(C)C1)=O 402,CC(CCN(CCCN1CCNCC1)C)CC(F)(F)F 403,C1(NC(c2nc(N(C)C)oc2)=O)CCSC12CN(C(=O)CC=C(Cl)Cl)C2 404,c1(SCc2c(C)nn(-c3cccc(Cl)c3)c2Cl)cn(CCO)c(=O)nc1O 405,C(=O)(C1CCCc2ncnn21)N1CCN(C(C2CN(C)C(=O)C2)=O)CC1 406,n1(CC)nc(C(N2CC3C(C(=O)NOCC=CCl)C3C2)=O)cc1C(=O)O 407,C1(C(C)NC(c2csc(Cl)c2)=O)CCN(C(C23CC2CNC3=O)=O)CC1 408,C(=O)(C(C)(F)C(=O)OC)N1CCC(N(C(=O)CCF)CC)C1 409,CCCCC(O)C(C)C(=O)NCC1(O)CCN(C(=O)C=Cc2ccncn2)CC1 410,CN1N=C(CC(=O)N2CCC(F)(F)C(CNC(C3(O)CCSCC3)=O)C2)CC1=O 411,c1(C(=O)NCC2(O)CC(NC(CCCCC=C)=O)C2)cccc2c1OC(C)(C)C2 412,C1(NC(C(CO)NC(C(n2ccc(C)n2)C)=O)=O)CC(CO)C2CC12 413,CCCCC(C(=O)NCC1CCCCS1)NC(c1cccc(C#N)c1)=O 414,c1(CCC)c(C(=O)NC2(CO)CCN(C(=O)Cn3ccc(C)c3)C2)nnn1C 415,CCCC(C(=O)NCc1cccc(Cl)c1)OCC1CCCCN1C1CCCCC1 416,CC(C(=O)OC(C)(C)C)C(=O)N1CCC(CN(C)CCc2ccnn2C)C1 417,Cn1cnc(C(=O)NC2CN(C(=O)CC3C=CCCC3)C2)cc1=O 418,C1(C(=O)NCC(C)NOC(c2cc(CC(=O)N(CC)CC)on2)=O)CC=CCC1C 419,N(C1CCc2ccccc21)C(C(CNC(c1ncnc(C)c1C)=O)O)=O 420,C12(C(N3CCC(CNC(CC(C)N(C)C)=O)C3)=O)CCC(=O)N1CCS2 421,C(=O)(C1CCc2cccc(O)c21)N1CCC(CC)(NC(C2CC(C)CO2)=O)CC1 422,C1(CNC(CSCC)=O)CC2(CCOCC2)CN1C(C1(C2CCCCO2)CC1)=O 423,C1(NC(c2c(C)cc(CC)o2)=O)CCCC12CN(C(=O)CCCc1ccsc1)C2 424,c1(CN(C(c2ccncc2Br)C)C)cc(-c2ncnn2C)ccc1O 425,S(=O)(=O)(c1cccnc1)NCC(=O)NC1CCN(C(=O)C(O)CC2CC2)C1 426,c1(C(F)(F)F)cc(F)cc(F)c1NC(=NCCC1CCC1)NC(C)(C)CC(F)F 427,N1(C(CS(CC)=O)=O)CC2CCCC2(NC(C23CC(COC)(CO2)C3)=O)C1 428,C1(NC(c2c(C)cno2)=O)C=CCN(C(=O)Cn2cccc2)C1 429,O=C1NC(C(=O)NCC2CCN2C(=O)Cn2cnccc2=O)CCO1 430,C(Cn1cccn1)(C(=O)NOCc1nc[nH]n1)NC(C1CCCC(=O)N1)=O 431,c1(C(C(=O)NC2(C)CC(NCc3nn(C)c(C(F)F)c3)C2)=O)ccc(Cl)c(Cl)c1 432,c1(C(N(C2CCCN(C(=O)CC3CC=CC3)C2)C)=O)cn(C)c(=O)cn1 433,C1(NC(CC2C(NC(C3N(C)CC(F)C3)=O)CC2O)=O)CC(C)(C)OC1=O 434,C(N=C(NC1CCOCC1)N1CC(O)C2(CC2)C1)C1(O)C(C)(C)CCC1 435,N1(CC(C)NC(c2nc(CC)sc2)=O)CCN(C(c2nnsc2C)=O)CC1 436,N1(C(c2c(CCC)nco2)=O)CCC2(CC1)CC2C(=O)NC1(C)CCCC1(C)C 437,c1(C(=O)NC(CN(C(C(C)Cc2cnn(C)c2)=O)C)(C)C)cc2n(c1)CCOC2 438,C1(C(=O)Nc2n(CC)nnc2C)CN(C(C)=O)CC(F)(F)C1.C1(=O)CN1C(C)(C)C 439,C1(NC(CCSCCCC)=O)CCCCC1CNC(c1ccn(C)c1CC)=O 440,N1(C(C(C(C)C)n2ncc(C)c2)=O)CC(NC(C2CC23CC3)=O)C2CCCCC12 441,c1(NCC(C(C)(C)O)(C)C)ccc2c(c1)C(=O)NCCC2 442,c1(C(N2CCOCC(F)(CNC(=O)CC34CC(C3)C4)C2)=O)cccc2c[nH]nc12 443,c1(C(c2nnnn2C(C)(C)C)CC)cc([N+](=O)[O-])ccc1C.C=CCC(N)CC1CCOC1 444,CCCC(C(=O)NCC1CN(C(=O)CCc2ccn(C)n2)CC12CC2)S(N)(=O)=O 445,C1(C(=O)NC2C(CNC(c3cccc(CO)c3)=O)C2)CCOC2(CCCCC2)C1 446,c1(COC)cccc2sc(NCc3sc(C(F)(F)F)cc3Br)nc12 447,c1(-n2c(C(C3C(Cl)C3)NCc3cc(F)ccc3Br)nnn2)ccc2c(c1)OCO2 448,c1(C(=O)NC2C(CNC(c3cnn[nH]3)=O)COC2)coc2ccc(Cl)cc12 449,CC(C)C(CO)C(=O)N(CC(C)CNC(=O)CC1CC2CCC1C2)C 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468,N1(C(C(c2cc(O)no2)C)=O)CCC(CC(=O)CCn2ncc(C)c2)CC1 469,N1(C(C(c2cccc(OC)c2)(F)F)=O)CC(NC(c2nncs2)=O)CC(O)C1 470,C=C(Cl)CC(C(=O)N1CCC(SC)C1)NC(=O)CC1CCC=CCC1 471,c1(C(c2ccccn2)NCc2cccc(F)c2)cccc2ccccc12 472,C1(CCC)(NC(CCN(C(=O)C(O)CN(C)C)CC=C)=O)CCCC1 473,c1(CC2N(C(=O)OCCC(C)C)CCSC2)c2c(nn1C)CCCC2 474,C=CC1CN(C(c2ccc(F)c(O)c2)=O)CC1NC(C1CCCS1)=O 475,N1(C(CC)=O)CCC(C(=O)NCCC2(Cc3ccon3)CCCC2)C1 476,c1(C(=O)NCCNC(c2cc(CCCCC)[nH]n2)=O)c(F)cncc1Cl 477,c1(N2CCC(c3ccc(C(=O)OC)cc3)CC2)cc(F)c(OC(F)F)c(F)c1 478,C1(NC(Cc2c(C)ocn2)=O)CCCCN(C(C2CC2c2ccco2)=O)C1 479,c1(OC)ccc(C(C)(C)C(=O)Nc2c[nH]nc2Nc2cnc(I)cn2)cn1 480,C1(CNC(c2c(SCC)cncc2)=O)COCCN(C(C2(C)CCCN2C)=O)C1 481,C1(CNC(C(C)N2CCC2)=O)CC2CCC1N(C(=O)CC(C)c1cccnc1)C2 482,c1(OC)ccc(Cl)cc1C(N1CCN(Cc2cn(-c3ccccn3)nn2)CC1)=O 483,Cc1c(C(N2C(CC(=O)Nc3ccc(Br)cc3I)CCC2)=O)cc(Cl)cc1Br 484,C(C)(CCCC(C)C)NC(CC1(C=C)CN(C(=O)C=Cc2ccc[nH]2)C1)=O 485,Cn1ccc2cccc(C(N3CC(F)CC3C(=O)Nc3cccc(N)c3)=O)c12 486,C(=O)(CCCCC(=O)NC1CC(CC(=O)NC2CCOC2)C1)NC 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631,CS(=O)(=O)c1ccccc1NC(=O)CCN1CC(O)(c2ccncn2)C1 632,c1(C(N2CCC(N(C(c3cnns3)=O)CC)C2)=O)[nH]c(=N)sc1C(F)(F)F 633,C1(COC)CN(C(c2ccc(Cl)cn2)=O)CCN1C(c1ccc(F)c(CO)c1)=O 634,CCC(CC)C(=O)N1CC=CC1(C(=O)NC1C(C)C1(C)C)COC 635,c1(OC)ccc(OC)c(CCC(=O)NC(C)CN(C(=O)C(C)C2CCCO2)C)c1 636,N1(C(C2(CC)CCN(C(=O)CC=C(Cl)Cl)CC2)=O)CC2(COC(=O)C2)C1 637,C1(C)(CNC(COCC#C)=O)CCN(C(=O)CN(C2COCC2O)C)CC1 638,C(=O)(C(C)C(C)(C)c1ccccc1)NC1(C(C)NC(=O)CC(=O)OC(C)(C)C)CC1 639,N1(C(C(CC#C)C)=O)CC(NC(=O)C(CC)C2CCOCC2)CCC(O)C1 640,Cc1nn(C)cc1C(=O)N(O)Cc1cn(Cc2[nH]nnc2C)nn1 641,Cc1ccc(C(N2CCCC(NC(c3ccn(C)n3)=O)C2C)=O)c(F)c1Cl 642,c1(C(=O)NCC2CN(C(CC3C(C)=NN(C)C3=O)=O)C2)ccc2c(C)[nH]nc2c1 643,C(=O)(CC(CC)C1CC1)NCC(CNC(C(C)(C)OCC)=O)(C)F 644,C1(CNC(C2CCCCC2)=O)CN(C(C2CC3CCC(C2)C3O)=O)C2(CCC2)C1 645,C(=O)(C1=CC2CC(C1)CC2O)NC1N(C(CCC(=O)N(CC)CC)=O)CCCC1 646,C1(CNC2(C)CC(NC(N(C)C)=O)C2)OCCCC1c1ccccc1 647,N1(C(C2(C(C)C)COC2)=O)CC2OCCN(C(=O)C(F)CC(C)C)C2C1 648,C(=O)(C(C(=O)N1CCC(C(C)NC(c2coc(C)c2)=O)C1)C(C)C)OCC 649,C1(NC(c2c(CC)nns2)=O)(CF)CCN(C(C2(OC)CC(CF)C2)=O)C1 650,Cc1cc(NC(c2cnn(C)c2C2CC2)c2nnnn2CCC(N)=O)cc(F)c1 651,CC(CCC(=O)NCCCC(O)CO)NC(=O)C(C1CCOCC1)=O 652,CON(CCC(=O)N1CCC2(COC(=O)N2C)C1)C(=O)C(CC(C)C)N(C)C 653,N1(C(c2c(CCC)n(CC)nn2)=O)CCC(NC(C2(CC(F)F)CC2)=O)C(C)C1 654,C1(NC(c2n(C)nc(O)c2)=O)CCC2(CC1)CN(C(=O)C1=CS(=O)CCC1)C2 655,CCCC(C(=O)N1CCC(NC(c2cc(C)n(C)n2)=O)C1)NC(N)=O 656,c1(C(N2CCC(N(C(C=C(C)C(F)F)=O)C)C2)=O)cc(OC)cc(OC)c1N 657,CC(C(=O)N1CCC(CC2CC2)CC1)C(C)NC(c1ncccc1Cl)=O 658,c1(CC)onc(C)c1C(N1CC2CC2(CNC(=O)CCCc2cccs2)C1)=O 659,Nc1cccnc1C(=O)NCC1CN(C(=O)COCCN(C)C)C2CC12 660,Cc1c(CN2CCCC(C(=O)NCCC(C)CCO)C2)cnn1C 661,C(C(C(=O)NCC1(C)CC2(CCC2)C1)C(C)(C)C)NC(C(CCC)(C)O)=O 662,C(N=c1ncnc(C(=O)O)[nH]1)C1CN(C(c2snnc2C2CC2)=O)C1 663,Cc1c(F)ccc(Cl)c1C(=O)NCCCCNC(=O)C=Cc1ccc(Cl)cc1 664,N1(C(c2cc(COC)no2)=O)CC(NC(=O)CNC(C)=O)CC2(CC2)C1 665,n1(CC)nc(C(=O)NC(C2CN(C(=O)CC(F)F)C2)C)c(Cl)c1Br 666,[N-]=[N+]=NC1(C(N2CCC(O)(C(N)=O)C2)=O)CCN(C(C2CC(O)CN2C)=O)C1 667,N1(C(C2(NC(C(C)c3ccsc3)=O)CC(F)(F)C2)=O)CCCC(C)(C)CC1 668,Cc1nc(C2OCCC2C(=O)NCCCC(C)O)n[nH]1 669,N1(C(=O)Cc2cc[nH]n2)CCN(C(C2CS(=O)(=O)CCO2)=O)C(CC2CC2)C1 670,C12(NC(c3n(C)nc(C4CC4)c3)=O)CCCC1CN(C(=O)C(C)(C)CF)C2 671,c1(O)ccc(C)nc1.C1(CCCC)CCN(C(=O)CCN(CCN)C)C1 672,c1(OC)nc(C)ncc1C(=O)NC1CCCC(NC(=O)CSc2n[nH]c(O)n2)C1 673,c1(OC)cccc(C2(CNC3OCCC3F)CCC2)c1 674,c1(C(N2CCN(C(C34CCCC3C4)=O)CC2CCO)=O)ccc(F)cc1[N+](=O)[O-] 675,CCC1=NOC(C(N2CC3CC3(CNC(=O)C(F)=C3CCC3)C2)=O)C1 676,CCCC(C(=O)NC(c1ncccc1F)C)NC(c1csc(Cl)n1)=O 677,N1(C(=O)Nc2scc(COC)n2)CC2CC(C(=O)OC)CC2C1 678,Cc1cc(=NC2CS(=O)(=O)CC2N2CCCCCC2)nc(-c2ccncc2)[nH]1 679,c1(C(=O)NC(CN(C(c2cnc(O)s2)=O)CC)C)cc(C(C)C)cnc1C 680,C(c1ccccc1OC)=CC(=O)NCC(CNC(c1cc(CCC)nn1C)=O)O 681,N1(C(COCC(C)C)=O)CC=CC1(C)C(N1CCC1CC(C)C)=O.C 682,c1(C(=O)NCC2(F)CCCN(C(CN(C(=O)OC)C)=O)C2)cn(C)c(C)cc1=O 683,C1(NC(C2N(CC)CCC2)=O)(Cc2nnc(-n3ncc(CO)n3)s2)CCC1(C)C 684,CC(CS(C)(=O)=O)C(=O)NC1CN(C(c2cc(O)c(O)c(O)c2)=O)CC1C 685,CN1C(=O)OCC1C(=O)NC(C)(CNC(C1CC1C(N)=O)=O)c1cccs1 686,CCCC(C(=O)N1CCC(CNC(=O)CCCOCc2ccccc2)CC1)OC 687,n1(CCN(C(C(C2CC2)OC)=O)C(C)C2CC2)cc(C2CC2)nn1 688,C1(CNC(c2ccc(CC)[nH]2)=O)CCN(C(c2ccnn(C)c2=O)=O)C12CCC2 689,O=C(CC1CCN(C(c2ccnc(S)c2)=O)CC1)N=c1cc(Br)[nH][nH]1 690,c1(CC)cc(C)c(CCC2(O)CN(C(C3(Cc4cccc(C)n4)CCCC3)=O)C2)o1 691,Cc1nc(N2CCCC(C)(CNC(C34CCCC(C3)OC4)=O)C2)cc(C#N)n1 692,c1(N2CC(COC)OCC2)nc(=N)nc(N2CCC(OCc3ccccc3)C2)[nH]1 693,C=CCC(C(=O)N1CC=CC1)NC(=O)CCCN.C1C(=O)N1C(C)C.OC 694,N1(C(CC=CC=C)=O)CCOC(CC(=O)N(C(C)CCCC)CC(C)C)C1 695,c1(OC)ccc(Cl)c(Cl)c1C(N1CCCC(C)(NC(=O)CC(C)C2CC2)C1)=O 696,C(CCN=c1[nH]c(C)cc(=NC2CCC(C)(C)CC2)[nH]1)N(S(CC)(=O)=O)C 697,CCCC(CCCNC(c1c[nH]nc1-n1cnnn1)=O)NC(=O)C(O)CCSC 698,c1(NC(c2nnnn2C(c2cc(C(C)(C)C)no2)SC)C2CC2)nn(C)cc1N 699,c1(CC(=O)NC2(CO)CN(C(CS(CC)=O)=O)C2)cc(F)ccc1F 700,CCC1=C(C(=O)NCC(=O)NCC(N2CCC2CO)=O)CCCO1 701,C1(C(=O)NCC2C(C(=O)NCC3(CC(=O)OC)CC3)C2)CCCCN1C 702,C1(C(N2CCCC2C(=O)NOCP(C)(C)=O)C(=O)OC)(CC=C)CCOC1 703,Cc1nc(NC2CN(C(C3CC=CCO3)=O)CCC2C(F)(F)F)c(C)c(O)n1 704,C1(NC(C(C)NC(N)=O)=O)CN(C(=O)CSc2cccs2)CC1C 705,c1(CC(C)N(C(=O)NC(C2(O)COC2)C)C)ccccc1F 706,c1(CC)cc(C(=O)NC2C3CN(C(c4cc(C)c(Cl)cn4)=O)CC23)ccc1F 707,CC1CC(NC(=O)C=CCF)CN(C(c2ccc(C(F)F)c(Cl)c2)=O)C1 708,c1(C(=O)NCCCC2CCN(C(C3CCCC3)=O)CC2)c(O)cc(F)cc1F 709,N1(C(C(=C)CC(=O)OC)=O)CCC2(CC1)CCN2C(c1cc2sccn2c1)=O 710,c1(NC(=O)OC(C)(C)C)ccc(C(=O)NCc2cc(Br)ccn2)cc1Br 711,c1(NC(C(C)N(C)C(c2ccc(SC3CC3)nc2)=O)=O)cccc2ccoc12 712,C(=O)(C(CC(C)CC)NC(C1CC2CCC1CC2)=O)N1CCN(CCC#C)CC1 713,N12CCN(CC1)C1CCN(CC1)C2=O.C(CC(N)=O)(N(C)C)N(C)C.C(CO)N 714,c1(C(=O)NC(C)C(C)(C)NC(C2CCC2C(C)(C)C)=O)ccc2cn(C)nc2c1 715,Cc1ncc(Cl)cc1NC(C1CCC(C2CC2)N1C(c1c[nH]nc1Cl)=O)=O 716,N1(C(C(CCCC)O)=O)CC2CCCC(C1)N2C(c1[nH]cnc1CC)=O 717,C1(NC(C(=O)OC)C2C(C(=O)OC)C2)COCCO1 718,C1(C(N2CCC(COC)(NC(=O)CCOCC(C)(C)C)C2)=O)CCCC(C)(C)O1 719,C1(NC(C(C)Sc2ccccn2)=O)CCCC12CN(C(=O)Cn1cnnc1)C2 720,N1(C(COC)=O)CCC(Cn2cc(C(c3ccc(F)cc3)O)nn2)CC1 721,N1(CC2CC(NC(CSCCCC)=O)C23CCC3)CC(C)OC2(CCNCC2)C1 722,O=C(C(O)CC(F)F)NC(Cc1cc(Cl)cnc1Cl)CO 723,N1(C(C2(C)CC2)=O)CCC2CCCC(C1)N2C(c1ccc(N)c(N)n1)=O 724,O=C(CC(C(F)F)n1cccn1)N1CC(NC(=O)CC2CC(F)C2)C(C(F)F)C1 725,c1(OCCOCC)ncc(S(=O)(=O)N2CCC(F)CC2C(=O)NC2C3CNC23)s1 726,C=C(C)CC(C(=O)N1CC(C(N)=O)C2(CC2)C1)NC(c1sccc1C#N)=O 727,C1(C(C)NC(c2cccs2)=O)CN(C(c2c[nH]nc2Br)=O)CCO1 728,c1(C(=O)NC2C3(CC(NC(C(C)CN4CCCCC4)=O)C3)C2)cccc(N)c1F 729,C1(CC(N2CCCC(OCC=C)C2)=O)C2CCCC2N1C(=O)C(C)C 730,C1(C(=O)NCCCN(C(CC(C)OC)=O)C)COc2ccc(Cl)cc2C1 731,C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)N1CC(N(C(C=C(CC)C)=O)C)C(C)CC1 732,C1(COC)CN(C(C2(N(C3CC3)C(c3cocc3C)=O)CCC2)=O)CCS1 733,N1(C(C2N(C(c3ccc(CC)[nH]3)=O)CC=C2)=O)CCn2cc(C)nc2C1 734,C1(c2nnnn2CC2CCOCC2)(NC(CCSC)C)CC2(C1)OCCO2 735,CC(C)C(C(=O)N(C1CC(NC(=O)CCCn2ccnc2)C1)C)c1ccccc1 736,C1(C(=O)NCc2csc(C3CC3)n2)CC=CCN1C(=O)CCc1nncs1 737,N1(C(c2cn(CC)nc2)=O)CCN(C(=O)CCOc2ccc(F)cc2)C(C)C1C 738,C1(C(=O)NCCC(C)NC(=O)CCc2cncc(F)c2)CC(S(C)(=O)=O)C1 739,C(=O)(C#CC1CCCOC1)NC1(C)CCN(C(c2c(C)nc(C)o2)=O)CC1 740,S(=O)(=O)(c1cccc(C(=O)N(CCNC(=O)C(C)O)CCO)c1)N(C(C)C)C 741,CCC(C(=O)NCCCC(C)NC(c1ccc(C)nc1N)=O)C(C)C 742,C1(CC(=O)OC)CC(OC2(CCC)CN(C(c3ccc(CC)o3)=O)C2)C1(C)C 743,N1(C(C2CC(C)CN2C(c2c(Cl)cnn2C)=O)=O)CCC(=O)N(C)CC1 744,C1(CNC(CCOCCOC)=O)CN(c2cc(-n3cc(C)cn3)ncn2)CCO1 745,Cc1ccc(=N)[nH]c1C(N1CCN(C(=O)C=Cc2cccnc2)CC1CO)=O 746,C1(C(C)NC(C(F)OC)=O)CCN(C(c2ccccc2OCF)=O)CC1 747,C1(C)(NC(C2CCCN(C(C(C)NC(CC)=O)=O)CC2)=O)CCC2(CC1)CC2 748,N1(C(c2cc(CC)oc2C)=O)C2CCC(C2)C1C(=O)NC1(C)CCCOC1 749,c1(NC(=O)C(=O)Nc2nnc(C(=O)OC(C)C)s2)ccc(OC(F)(F)F)c(Cl)c1 750,c1(OCC)nc(NCCC(C)NC(=O)C(CO)c2ccccc2)ncc1Cl 751,C1(C(=O)N(C2CCC(NC(=O)C(C)NC=O)CC2)C)(OC)CCCCC1 752,N1(C(c2c(C)nncc2)=O)CCC(CO)(CNC(C2CC(C)(C)O2)=O)CC1 753,N1(C(c2c(C)sc(Cl)n2)=O)CC(CNC(=O)COCC(C)C)C2(CCC2)C1 754,Cc1cccc(CCC(=O)NCC23CC2CN(C(=O)Cn2cnnc2)C3)c1Br 755,c1(NC(CNC(C2(C)CCC(C)C2)=O)C2CC2)cc(=O)n2cc(Cl)ccc2n1 756,n1(CC(C)NC(CCN(CC=C)C)=O)ccnc1C 757,C1(NC(C(=O)NC(CC(=O)OC(C)(C)C)c2ccccc2)=O)CCCC=C1Br 758,C1(CN(CCNC(C)=O)C)CCc2nnc(Br)n2C1.N12CCCC1NC(=O)C2=O 759,C#CCC(C)(C(=O)NC(c1cnc[nH]1)C)NC(C1CCCC(=O)CC1)=O 760,c1(N2CC(F)CC(C(=O)Nc3cc(C(F)(F)F)no3)C2)ncnc2c(Br)csc12 761,C1(C(N2CC3(CN(C(C(C4CCOC4)OCC)=O)C3)C2)=O)CCc2ccnn2C1 762,C1(C(=O)NCCCCNC(Cc2nc(-c3ccc(C)o3)sc2)=O)COCC(C)O1 763,C(=O)(CCCCCC(C)(C)C)NCC1(OC)CCN(C(CC=C=C)=O)C1 764,N1(C(C=C(C)C)=O)CCCC2(CCN(C(c3c(Cl)ccc(Cl)c3O)=O)CC2)C1 765,C1(NC(CCC(C)N(C)C)=O)CC2(C1)CC(NC(C1CCC1C)=O)C2 766,Cc1cc(C(=O)NC2CCC2CNC(c2cn(CC(F)(F)F)nn2)=O)n[nH]1 767,c1(CC(=O)NCC(CN(C(C(C2CCCC2)OC)=O)C)O)cccc2occc12 768,C(=O)(C1=CCCCCC1)NC1CC(N(C)C(C2CC23CCOC3)=O)C1 769,C1(C)(CNC(C(COC)O)=O)CCCN(C(=O)CCCOC2CCOCC2)C1 770,C1(C2CCCN(C(=O)Cn3nc(C)ccc3=O)C2)(NC(COCC#C)=O)CC1 771,c1(NC(C)=O)c(C(=O)NCCNC(=O)CC2(C)CC(C)=NO2)cccc1[N+](=O)[O-] 772,Cc1cnn(C)c1-c1cn(CCCC(=O)NC2CNCC2C#N)nn1 773,C(=O)(CCS(=O)(=O)CC(C)C)NC(CC)CNC(C1CCOC1C(F)(F)F)=O 774,N1(C(c2c(CC)nccn2)=O)CCC2(CC1)CCN2C(=O)CCC1CCOC1 775,C1(CC)CCN(C(C2CCCC(OC)C2)=O)C(C(=O)NCCn2nncc2C)C1 776,c1(C(=O)NCCOC2CCN(C(c3c(OC)cncc3)=O)C2)cnc(O)c(C)c1 777,C1(C)(C(N2CC(F)(CNC(C(C(=O)OC)(C)CC)=O)C2)=O)CC2(C1)CC(F)(F)C2 778,N1(C(C=CC)=O)CC2(CCN(C(=O)Cc3sc(Cl)c(Cl)c3OC)CC2)CC1C 779,C1(C(=O)NC2(CO)CN(C(CC3(C)CCC3)=O)C2)CCC(C(C)(C)C)CC1 780,CCC(F)(F)C(C)(C)C(=O)NC1CCCCCC1NC(=O)CC1CCN(C)CC1 781,Cc1cnc(C)o1.C1(=O)C(=O)OCC(=O)N(C)C(C2CC2)CN1.C(C(F)(F)F)S 782,C1(C(=O)NC2CC2O)CCN(C(C2CC2(Cl)Cl)=O)C1 783,C#CCCN=C(NCC(C)C(C)C)NC1CC1(c1cc(C)oc1C)C 784,Cc1cccc(COC(C)C(=O)NCCN(C)C(c2csc(C3CC3)n2)=O)c1 785,C1(NC(C2CCS(=O)(=O)C2)=O)CC2CN(C(C3(n4ccnn4)CC3)=O)CC12 786,C=CCCCCC(=O)N1C2CCC1C(C(=O)N(C)CC1CCCOC1)C2 787,Cc1cc(Br)oc1C(N1CCC(Cn2cc(CC(O)C3CC3)nn2)CC1)=O 788,S1(=O)(=O)C2=CNC(=NC(CCO)N1CCCc1c(C)cccn1)C=C2.C1(C)CC1 789,C1(NCCN(C(CC(CNC(C)=O)(C)C)=O)C(C)C)COc2ccccc2C1 790,c1(CCNC(=O)CCC2(NC(C3CCCCO3)=O)CCC2)ncccc1F 791,C1(OC)CCC(C(N2CCC(C(=O)NCCO)C2)=O)S1.C1(=O)CCOCCN1 792,N1(C(C2C(C)(C)CC2)=O)CC(O)CC1CNC(c1cncc(N)c1)=O 793,N1(C(C=CCC)=O)CCN(C(c2ccc(C(C)(C)C)cc2C)=O)C(CCCC)C1 794,CCCCC(C)CCC(=O)N1CCCC(NC(=O)COCC2CCCC2)CCC1 795,C1(C(=O)NCC(C2(O)CN(C(c3cc(C)[nH]n3)=O)C2)(C)C)CCC(=C(F)F)CC1 796,N1(C(C(C=C)OC)=O)CCCC12CCCN(C(=O)C=C(CC)CC)C2 797,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC1CCN(C(CSCC(=O)OC)=O)C(C)C1 798,c1(C(N2CCCN(C(Cc3c(C)cnn3C)=O)CC2)=O)nc(C)n2ccccc12 799,c1(C(=O)NC23CCN(C(c4ccc(Br)o4)=O)CC2C3)ccc2occc2c1 800,CCN=C(NCCN(C)C(=O)NC1CCC(C(=O)NC2CC2)C1)NC(C)(C)C 801,c1(OC(C(=O)NCC2C(CNC(CCC=CCC=C)=O)C2)CC)cccc(C)c1 802,c1(NCC)ccccc1C(N1CCCC(N(C(=O)CSC)CCOCCO)C1)=O 803,c1(C(N(C2CN(C(CSCC=C)=O)CC2F)C)=O)cc(Cl)c(F)cc1C 804,c1(C(N(C(CNC(c2c(C)nn(C)n2)=O)C)C)=O)nc2ncccn2n1 805,C1(F)(CNC(C2(OCC)CCOC2)=O)CCCN(C(=O)C=Cc2ccsc2)CC1 806,C(CC(C(C)(C)C)NC(=O)CC(C)c1cnn(C)c1)N(C(=O)CCNC(N)=O)C 807,C1(NC(c2n(C)c(SCCO)cc2)=O)CNCCS(=O)(=O)C1 808,Cc1ncc(CC(N2CCC(N(CCO)C(C3CCC3)=O)C2)=O)[nH]1 809,Cc1cccc(C(N2CCC(N=[N+]=[N-])(C(=O)NCC3(O)CCOC3)C2)=O)c1C#N 810,CCC(C(=O)N1CCC(OCC(=O)N(CC(=O)N(CC)CC)C)C1)OC 811,c1(NC(C2(CCNC(c3ccc(OC)s3)=O)CC2)=O)cnc(C)c(C)c1 812,N1(C(C2C(CC)CCN2C(c2ccc(N)cn2)=O)=O)CCC2(CCCO2)CC1 813,N1(C(CC2CC(C)N(C(c3cc(N)cc(F)c3)=O)C2)=O)CC2(CCC(=O)NC2)C1 814,N1(C(CC(C)F)=O)CC2CC(NC(c3c(C(C)(C)C)nsc3N)=O)C1C2 815,N1(C(CSCCOC)=O)CCCC2C1CCN2C(c1ccc2ccn(C)c2c1)=O 816,c1(C(C)C)ccc(C(C)N(CC(C)(C)CNC(C2(C)CNC(=O)C2)=O)C)cc1 817,C(=O)(C(F)(F)C(F)(F)F)NC1(C)CN(C(=O)CCOCc2ccccc2)C1 818,C1(NC(c2ccc(Br)o2)=O)CC2CCC(C1)N2C(=O)CC1CCCc2ccccc21 819,C1(CNC(CO)Cc2ccccc2Cl)C=CCCCCC1 820,c1(C(c2n(C(CC)C)nnn2)Nc2cnn(CCC(=O)OC)c2)ccncc1Br 821,CCC(C)(C)CC(=O)NC12CCC1CN(C(=O)C(C)(O)C(C)C)C2 822,C1(N(C(CN(CC)CC)=O)C)CCCC2CN(C(=O)CCc3cn(C)nn3)CC12 823,c1(C(N(C2CCN(C(=O)CCN3CCOCC3)C2)C)=O)cccc2c1OCO2 824,Cn1ccc2cc(NC(C3CN(Cc4ccc(I)c(F)c4)CCC3O)=O)ccc12 825,c1(C(=O)NCCCC(C)NC(c2c[nH]ccc2=N)=O)cccc2c1CCOC2 826,C(CS(=O)(=O)CCNC(C1CCC(O)C1)=O)OC 827,C(=O)(C(CCCc1ccccc1)N1CCC(NC(N)=O)CC1)NCC=C 828,c1(C(=O)NC2C(F)CCN(C(c3c(C)n(C)nc3)=O)C2)n[nH]c2c1CSCC2 829,Cc1nccc(C(=O)NCc2cc(C(=O)N(C3CCCC3C)C)n(C)n2)n1 830,c1(C(=O)OCC(=O)OCCO)cc2ccc(NC(OC(F)F)=O)cc2[nH]1 831,N1(C(C2(COC)C=CCC2)=O)CCN(C)C(CNC(=O)CC(F)(F)Cl)C1 832,c1(C(C)NC(=O)NCC2CC(=O)CCC(=O)N2)cc2ccccc2[nH]1 833,c1(C(N2CC3C(CNC(CC4(OCC)CC4)=O)(C3)C2)=O)cc(C(N)=O)n(C)n1 834,C(=O)(C(F)(F)CC(C)C)N1CCCC(CC)(NC(c2ncccc2Cl)=O)C1 835,c1(C(=O)O)ccnc(C2CCN(CCCN3CCOC3=O)C2)c1 836,N1(C(c2cc(C)c(Cl)s2)=O)CC(N(C(=O)CCc2ccc(=N)[nH]c2)C)C(C)(C)C1 837,c1(CN2C(CC(=O)Nc3ncc(C)cc3C)COCC2)ccc2nc(C)oc2c1 838,C1(NC(Cn2ncc(C)c2)=O)CCC(C)N(C(=O)Cc2cncn2C)C1 839,C12(CNC(c3cnc[nH]3)=O)CCCC1N(C(C1CCCN1C1CC1)=O)CCC2 840,c1(OC)ccc2cc(C(=O)NCC3CN(C(c4nc(O)nc(O)c4N)=O)C3)sc2c1 841,CC1CCC(C)(C(N2CCN(C(=O)CCc3cncc(F)c3)C(CO)C2)=O)CC1 842,N1(C(C(C)N(C(C)=O)C)=O)CC2C(CN(C)C(c3cc[nH]c3C3CCC3)=O)C2C1 843,N12CCCC3(CCCC13)NC(=O)C2=O.c1(C(=O)Nc2ncc[nH]2)cc(O)no1 844,n1(CC(=O)NC(C)(CNC(C2CC3CC3C2)=O)CO)nnc2ccccc2c1=O 845,Cc1[nH]c(C)c(NC(N2CCC3CC(C(=O)OC(C)(C)C)C32)=O)c1C 846,c1(C(N2CCC(O)(C(C)NC(C(CC)O)=O)C2)=O)cnc2ccccn2c1=O 847,C#CC1CC(C(OCS(=O)(=O)CC)OCC)(NC(C)C(=O)OC)C1 848,Cc1cc(F)c(C(N2CCN(c3ncc4cn[nH]c4n3)C(C#N)C2)=O)cc1F 849,c1(C2C(C(=O)NCC(C)NC(Cc3nc(C)sc3)=O)C2)ccnc2ccccc12 850,C(=O)(C(C)C(O)CC(C)C)NC(CC=CC)C(=O)NCC1OCCC1(C)C 851,c1(C(=O)NCC(C)NC(c2c(SC)cccc2)=O)cnn2c(C)ccnc12 852,C(=O)(C1CCCc2n[nH]cc21)N1CC(CNC(CCCN(C)C)=O)C(C)(C)CC1 853,c1(C(=O)OC)ccc(OC)c(OC(c2cccc(C(=O)OC)c2)=O)c1Cl 854,c1(COC)nn(C)c(Cl)c1C(N1CCC(F)C(NC(=O)Cc2cc(C)no2)C1)=O 855,c1(C(=O)NCC(CN(C)C(C2COC(=O)C2)=O)(C)C)cccc[n+]1[O-] 856,c1(C(N2CCCC(CNC(CC(=C)C)=O)CC2)=O)cc2cncn2c(O)n1 857,c1(C(=O)NCC(CCC)C(=O)NCc2scnc2C)n[nH]c2ccccc12 858,CC1CCCC(C)N1C(=O)CCc1ccc(C(N2CCN(C=O)CC2)=O)cc1 859,c1(CCCC(N2CCN(C(CC)=O)CC2CCO)=O)cc(OC)c(OC)c(OC)c1 860,c12ccc(cc1)C(=O)NC1(CC1)CO2.C1(C(CCCC)=O)CN(CC2CCC2)C1 861,c1(C(=O)NC2C(NC(=O)CCN3CCOC3=O)CC2)ccc(OC2CCC2)cn1 862,O=C(C1SCCc2sccc21)NCC1CN(C(c2cn(C3CC3)nn2)=O)C1 863,N1(C(CC2CCC(=O)O2)=O)CC=C(C(=O)NCC2C3CCCC23)C1 864,c1(CC(=O)NC2C(C(=O)NCCCCCN(C)C)CC2)ccnc(O)c1 865,c1(C(N(C2CCCC(NC(C3CCCCC(=O)N3)=O)C2)C)=O)nnc(O)cc1O 866,C1(CNC(C2C(C)C2C)=O)CCC2(CCN(C(C3(C#N)CC3)=O)CC2)O1 867,c1(OC)cc(COC(F)(F)F)ccc1O.c12c(ccnc1F)NC1CN(C1)C2=O 868,C1(CC(C)C)(C(=O)NCC2(NC(=O)CC(C)(C)C)CCOC2)CCNC1=O 869,c1(OCC)ccc(-c2c(-c3nccn3C3CNCC3C(F)(F)F)n[nH]c2C)cc1 870,C1(OC)CC2CC(C(N3CC=C(CNC(=O)C(N)=O)CC3)=O)CC12 871,N1(C(c2on(C)c(=O)c2)=O)CCC(NC(=O)CCc2ccccn2)CC(C)(C)C1 872,N1(C(CC2CN(C(C(C3CC3)OCC)=O)C(C)C2)=O)CC(=O)NC2(CC2)C1 873,N1(C(CCc2onc(C)n2)=O)CC(CNC(C2CCCC(C)O2)=O)CC1C 874,C(=O)(C1=Cc2cc(F)ccc2OC1)N(CCNC(c1c(C)sc(C)c1C)=O)CC 875,c1(NC2C(C)CN(C(C=C(C)C(F)F)=O)CC2C)cc(C)ccc1[N+](=O)[O-] 876,C1(C(=O)NCCOCCCNC(c2cn(CCC)nc2)=O)CCCCN(C)C1=O 877,C(=O)(C(CC(C)(C)C)NC(c1occ2c1CCC2)=O)Nc1cn(CC)nc1C 878,C1(C(N2CCC(C)(N(C)C)C2)=O)CN(C(C2CS(=O)C2)=O)CC12CCC2 879,C(C1=CCCN(C(=O)CC2(C(F)(F)F)CC2)C1)NC(=O)C=Cc1cn[nH]c1 880,C1(NC(=O)C(CC2CCC2)NC(C2CCOC2)=O)CC12CCCC2 881,N1(OC(c2cn(-c3cccc(OC)c3)nn2)=O)C(=O)NC(C)(C2CCOCC2)C1=O 882,CC1(C)CCCCCC1c1nn[nH]n1.C1(=O)C(C(F)(F)F)Cc2cn(nn2)CC1=O 883,C1(C(=O)Nc2c(C)nccc2)C2CC(CC2F)N1C(=O)C1=NNC(=O)C1 884,N#Cc1c(CN2CC3CC2CN3S(=O)(=O)Cc2ccc(C#N)cc2)cccc1Cl 885,N1(C(=O)OC)CCC(C(=O)NCC2CCN2C(c2ncsc2C(C)C)=O)CC1 886,N1(C(C2(CC)CCN(C(C3CC4C=CC3CC4)=O)C2)=O)CCC2(CCCCC2)C1 887,C1(CCC)(NC(=O)CC2CC(O)CN2C(c2cccnn2)=O)CCNC1=O 888,N1(C(COCC(=O)NC)=O)CC(NC(=O)CSC2CCCCO2)C(CO)C1 889,C1(CNC(C(=O)NC(C)C)=O)CC2(CCC2)CN1C(C1CCCC1C(C)C)=O 890,c1(C(=O)OC)ccc(C(N2CCS(=N)(=O)CC2)C(=O)Nc2ccccc2)cc1C 891,c1(OC)cc(-c2cn(CCN(C(=O)CCn3ccnn3)C)nn2)ccc1F 892,C1(C(C)=O)C(C(=O)N(CC(=O)N(C2CCCS2)C)C(C)C)C1(C)C 893,c1(C(=O)NC2CCC(NC(C3(COC)CCOC3)=O)C2)c([N+](=O)[O-])cnn1C 894,N1(C(CN(S(C)(=O)=O)C)=O)CCN(C(=O)CC2OCCC2(C)C)C2COCC12 895,S(=O)(=O)(C1=CCS(=O)(=O)C1)NCC1C(=O)NCC1 896,C1(CNC(COCC(C)(C)C)=O)CCC(CNC(=O)C=C(C2CC2)C2CC2)CC1 897,N1(C(c2c(C)c(C3CC3)on2)=O)CC2CCCC1C2CNC(=O)Cn1cnnc1 898,Cc1cc(NC(C2CC3CC2CC3O)=O)nc(C)c1.c12cn(nn1)C1CN(C1)C2 899,c1(C(N2CCN(C(CCSCC(N)=O)=O)CC2C(F)F)=O)cc2c(s1)CCOC2 900,C1(C(=O)NC(CNC(C(C)NC(C2CCCC2)=O)=O)C)CCC2(CCCC2)CC1 901,N1(C(C(C(CC)C)O)=O)CC2CCN(C(C3(C)CN4CCC3CC4)=O)CC2C1 902,c1(CN2CC3CN(C(Cc4ccc(OC)nc4)=O)CC32)cc2cc(C)ccc2[nH]1 903,CCC(C)(F)C(=O)NC(C)CNC(C1(Sc2ccccc2)CC1)=O 904,O=C(CC1=CCCC1)NCc1ncccc1C(=O)NC1CCCCC12CC2 905,c1(C(N2CC3C(CNC(Cc4n(C)nnc4)=O)(C3)C2)=O)nnc(O)c(Br)c1 906,CC1(C)CC2CC(C)(CN2C(c2cc3ccncc3[nH]2)=O)C1 907,C1(C(=O)NCc2c(COC)n[nH]c2)CCN(C(=O)CCCN=[N+]=[N-])O1 908,c1(OC)cc(O)ncc1C(=O)NC1CN(C(c2n[nH]c3c2COC3)=O)CC1SC 909,CCC(CC)C(=O)N1CC(O)CC1CNC(c1ccn(-c2cncc(F)c2)n1)=O 910,C(=O)(C(CO)C(F)(F)F)N1CCC(CC=C)(C(=O)NCCCCOC(C)(C)C)C1 911,c1(C(N2CC(CCNC(C(CC(C)C)C)=O)C(C)C2)=O)cc2ccccc2cn1 912,c1(C(=O)NC2CCCCN(C(C3OCCN(C)C3)=O)C2)cncc2ncccc12 913,C#CC1(C(=O)N(C)CC23CCC(CC2)C3)CCN(C(=O)CC(C)C(C)C)C1 914,c1(C(C)Nc2cc(NCc3nccs3)ncn2)cc([N+](=O)[O-])ccc1Cl 915,CCC(CCCC(=O)N1CCC(COC)O1)NC(=O)CCNC(C)=O 916,N1(C(=O)CC23CC(C2)C3)CCC2C1CCCN2C(=O)CCc1cccnc1 917,N1(C(C(CCN(C)C)NC(C(C)OCCOC)=O)=O)CC2CCCCC12C 918,C(CCC(O)C(=O)NC1CCCC(O)C1)NC(c1cc(COC)no1)=O 919,C1(CNC(=O)NC(c2cn(C)nc2C)C(C)(C)OC)CC(F)(F)CO1 920,N1(C(c2c(C(C)C)cco2)=O)CCC(NC(c2cc(Cl)cs2)=O)C(C)(C)C1 921,CC(C)C(C)(C)C(=O)NC1CN(C(C2CCCN(CC(F)F)C2)=O)CC1O 922,CC#CCCCC(=O)NC(C(CCc1ccccc1)OCC(=O)NC1COC1)C 923,Cc1nc(N(C(C2CCC(O)(c3ccccc3)C2)=O)C(C)C)sc1C 924,N1(C(c2c(N)c(F)cc(F)c2)=O)CCC2CN(C(c3ccnnc3)=O)CCC12 925,c1(C(N2C(CCNC(c3c(CC)scn3)=O)CSCC2)=O)cc(F)c(O)c(F)c1 926,c1(C(=O)NCC2(C(C)NC(C(CCCC)O)=O)CC2)cc(Cl)c(OC)c(OC)c1 927,N1(C(c2c(N)cc(C)cc2F)=O)CC(NC(c2cscn2)=O)CC12CCOCC2 928,Cc1nc(C(N2CCC(C)(NC(c3cc(CC(C)C)c[nH]3)=O)C2)=O)c(C)o1 929,CC(C)CC(CNC(C1CCCCC(=O)C1)=O)C(=O)NC(c1nn(C)cc1O)C 930,c1(C(N2C(CNC(C(C)(C)c3sccc3Cl)=O)CCC2)=O)c[nH]c2ccncc12 931,c1(C(N2CCC(N(C(=O)CCNC(c3ccnn3C)=O)C)C2)=O)nnc(S)n1C 932,c1(C(N2CC(F)(CNC(c3cncc(C#C)c3)=O)C2)=O)cc2cc(Cl)cnc2[nH]1 933,C(=O)(C1CCCc2n[nH]cc21)N1CC(CN(C(C(CC)(F)F)=O)C)C1 934,CC1(C)CC(c2nnnn2CC2CCCOC2)(NC(CCO)c2cccs2)CS1 935,C1CCC(O)C(=O)N2CC(C2)C(C)O1.C(F)(C(=O)NCSC)=CCC 936,c1(NC(c2ccc3ncccc3c2)=O)cccc(F)c1[N+](=O)[O-] 937,N1(C(CCc2ccc(C)o2)=O)C2CCC(C(=O)NCCCOCCO)C1CC2 938,c1(C(N(C(C)CCNC(C2CC(O)C2)=O)C)=O)cc(F)c(F)c(C#N)c1 939,CC(C)C(C)CC(=O)NCCCOCCCNC(=O)C(c1cccc(F)c1)(C)C 940,N1(C(CC)=O)CC=CC(NC(=O)CC(c2cccs2)NC(=O)OC(C)(C)C)C1 941,c1(NC(C(CC=C)NC(=O)C(CCC)NC(N)=O)=O)cc(F)ccc1C 942,c1(CC)cc(F)ccc1C(=O)NC1CCN(C(C2CC(F)CN2C)=O)C12CC2 943,C(=O)(C(C)CC(C)(C)C)N1CCC(NC(C(CCCC)O)=O)C1C 944,C1(NC(c2ccc(F)o2)=O)CN(C(C2CC2c2cccs2)=O)CCC12CCC2 945,c1(C(C(=O)NCc2ccco2)N(CC(C)(C)C)CC)nnn(C)c1CC 946,c1(OC(C)C(=O)NC2CCCC2NC(c2cscc2C(N)=O)=O)ccc(Cl)cc1 947,c1(C(N2CCN(C(C(CSC)O)=O)C(C)C2)=O)ccc(Cl)c2cccnc12 948,N1(C(COCCCCCC)=O)CCC(NC(c2cnccc2C)=O)C(C)C1 949,c1(CNc2nccc(NC(C(C)C3=CCCC3)=O)c2)cc(Cl)cc([N+](=O)[O-])c1O 950,C1(CNC(COCCC#C)=O)CCC(NC(c2cc(Cl)cn2C)=O)CC1 951,Cc1oc(C(C)C)nc1C(=O)N(C(C)CCNC(C1(S(C)(=O)=O)CC1)=O)C 952,C12CCN(CC1F)C2=O.c1(CNC(=O)C2CC2)nnc(S)s1 953,CC(CC(=O)NC(CC1CC1)C(=O)NC1(CC(N)=O)CCC1)C1CCCO1 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973,C(C1CCOCC1)=CC(N1CC(C(C(N2C(C(=O)NC)C=CC2)=O)O)C1)=O 974,C(C(C(=O)NCC1(CNC(=O)CSC)CCCC1)OC)OC 975,CCCCC(CNC(=O)Cc1nccn1C)NC(=O)C(CC1CCC1)OC 976,c1(NC2C(C)CN(C(=O)Cc3ccc(O)c(C(=O)O)c3)C2)ncnc2sc(Br)cc12 977,N1(C(C(C)C(F)(F)F)=O)CCC(C2(O)CN(C(=O)CN(C)CC(C)O)C2)CC1.C(C(C)(C)C)N 978,CCC(C)C(CC(=O)NC1(CCO)CC=CC1)NC(=O)COC(C)(C)C 979,c1(OC)c(Br)ccc(F)c1C(=O)NCCNC(=O)C(CC(F)F)C1CCC1 980,C1(CNC(C2C3CNC(=O)C23)=O)COCCN1C(c1scnc1Cl)=O 981,C1(CNC(c2ccc(C(F)F)nc2)=O)CC2CCC(C1)N2C(C12CCC1C2)=O 982,c1(C(C(=O)NC(c2ccn(C)n2)C(=O)OC)C)ccccc1 983,N1(C(C(CC#C)NC(=O)C(C)SC)=O)CCC12CN(C)C2 984,C(=O)(CC(=O)NC1CC(F)(CNC(=O)C(c2ccc(Br)s2)C)C1)OC 985,C(CCCOC)(C(=O)NCC1CN(C)C(=O)N1)NC(c1cn(CC=C)nn1)=O 986,N1(C(c2cc(SC)ncn2)=O)CC(C)N(C(=O)CCc2cccn2C)CC1C 987,C1(C(=O)NC2CCN(C(C)=O)C2)CCN(C(=O)C(F)C(C)(C)O)O1.C(C)(=O)O 988,C1(C(C)C)CCCN(C(C2CCC2NC(c2ocnc2C2CC2)=O)=O)CC1 989,CC(C)C(C(=O)NC(CNC(c1cn(C)nc1Cl)=O)C1CCC1)n1ccnc1 990,C1(N(C(=O)C(C)(F)F)CC)CCCN(C(=O)C(O)c2ccsc2)C1 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1259,c1(-c2cncc(NC(N3CCOCC(O)C3)=O)n2)cc(F)cc2cccnc12 1260,c1(N(C2CN(C(C(C=C)c3ccccc3)=O)C2)C)nc(C)ncc1F 1261,c1(SCc2cn(C)nc2)ccc(C(N2CC(O)CC2CNC(=O)CO)=O)cc1 1262,N1(C(C=CCC)=O)CCC(C)C(CNC(c2cc(C(=O)OC)oc2C)=O)C1 1263,S(=O)(=O)(c1ccc(C(=O)NC2CCC(NC(=O)CC(C)(C)CC3CC3)C2)o1)NC 1264,c1(CCC)cc(C(=O)N(C2CCCC(NC(c3cnc(O)n3C)=O)C2)C)sc1C 1265,c1(CCC)cc(C(N2CC(F)(C(=O)NCC3CC(O)C3)C2)=O)n[nH]1 1266,Cn1nccc1C=CC(N1CC(NC(=O)C(F)C2CCC2)C1)=O 1267,c1(NC(C2CCCC(NC(CCC#C)=O)C2)=O)cnc(Cl)c(F)c1 1268,Cc1cc(CNC(=O)CCC(C)(C)NC(=O)CC(C)(C)C#N)cc(C)c1F 1269,C=CC(C)(CC)C(=O)NCC(C1CC1)N(C(=O)Cc1ccsc1Cl)C 1270,C=C(C)CC(C(=O)NCCc1ccc(F)nc1)NC(C1CCCN1C=O)=O 1271,N1(C(c2cc(C(=O)OC)sc2C)=O)CCCC(C2(NC(=O)CC3C=CCC3)CC2)C1 1272,N1(C(C(C(=O)OCC)CC)=O)CC2CC(NC(=O)C=CC=C(Cl)Cl)CC2C1 1273,C1(N(C(c2c(C)snn2)=O)C)CCN(C(=O)Cc2sccc2Cl)CC1C 1274,Cc1ccc(C)c(CC(=O)NCCCC(=O)NCC2(O)CC=CC2)c1 1275,C1(F)(CNC(Cc2c(C)scc2)=O)CCN(C(c2ccc(C#N)[nH]2)=O)C1 1276,Cc1cn2cc(C(N3CC4CC4(NC(c4cccnc4O)=O)C3)=O)cc(C)c2n1 1277,c1(C(c2n(CCC)nnn2)NCCC2(C)CCCO2)cccc(C(F)(F)F)c1F 1278,C1(CNC(c2c(COC)noc2)=O)CC(F)(F)CN1C(C1CN(C)CC1C)=O 1279,N1(C(c2c(CNC(c3c(=N)[nH]cnc3)=O)c[nH]n2)=O)CCCNC(=O)C12CC2 1280,N1(CCC)CC(C(N2CCCC2CNC(C2(CCO)CC2)=O)=O)CC1=O 1281,CC#CCC(C(=O)NCC(C(F)(F)F)OC)NC(c1ncc(N)cc1C)=O 1282,c1(C(=O)Nc2cc(C)[nH]n2)cc2ncc(-c3cccc(F)c3C)cc2[nH]1 1283,C1(COC)(NC(c2sc(-n3cccc3)nc2C)=O)CCCN(C(=O)C(C)CO)C1 1284,N1(C(c2n(CC(C)C)ncc2)=O)CCN(C)C(CNC(=O)CC2CC2C)C1 1285,c1(C(=O)Nc2cccn(O)c2=O)ncn2cc(-c3cccc(CO)c3)sc12 1286,c1(OC)cnc(Br)cc1C(N1CCCC1C1CCN(C(=O)C(O)C(C)C)C1)=O 1287,Cc1c(F)ccc(C(=O)NC2CC3CC(NC(=O)C(C)C(C)C)CC23)c1C#N 1288,N1(C(C2C(CC=C)C(O)C2)=O)CCOCC1C(=O)NC1CC(=O)N(O)C1 1289,c1(OC)cc(C(N2CC(NC(=O)C(C)CSC(F)(F)F)CCC2C)=O)cc(Cl)c1O 1290,c1(C(=O)OCC)cnc(N2CC(NC(=O)CN=S(C)(C)=O)C2)nc1C 1291,C(=O)(CCC(F)(F)C(F)F)N(C(C)CNC(=O)COCc1nc[nH]n1)C 1292,C1(C)(C(N(CC(C)NC(C23CC(c4ccccc4)(C2)C3)=O)C)=O)CCCO1 1293,Cc1nc2n(n1)CC(C(N1CCCC(CNC(C3(F)CCCCC3)=O)C1)=O)CC2 1294,C1(NC(C=CC(C)(C)SC)=O)CN(C(=O)CN(C2CCC2)C)C2(CCOC2)C1 1295,N1(Cc2n(C)c(-c3ccccc3)nn2)C2CCC1CN(C(C1CCC(O)CC1)=O)C2 1296,C1(c2cn(CC(C(N3CC(C)CC(CC)C3)=O)(F)F)nn2)CN2CCN1CC2 1297,C(CCSC)(C(=O)NCC12CC1CN(C(C1(N(C)C)CCC1)=O)C2)OC 1298,N1(C(C2N(C(CC)=O)CCCC2)=O)CCC(CNC(=O)CCSC)C(O)C1 1299,c1(C(N(C2CCN(C(=O)CCCNC(=O)C3CC3)C2)CCC)=O)cnc(O)n1C 1300,C1(C(N2C(C#C)CC2)=O)CN(C(c2occc2COC)=O)CC12CCC2 1301,c1(C(=O)NC23CCC(CNC(=O)C4=CCCC4)(OC2)C3)cccc2ccsc12 1302,N1(C(CCn2ccc(C)n2)=O)CCN(C(C2CCCC3CC23)=O)C2(CCC2)C1 1303,C1(CCNC(C=C(CC)C)=O)CC(NC(C2CC23CC3)=O)C1 1304,N1(C(CNC(CC)=O)=O)CC2CC(C)N(C(c3csc(C4CCCO4)n3)=O)C2C1 1305,N1(CCC(=O)N(CCCNC(c2ccon2)=O)CCS)CCOCC1.N(C)CCO 1306,CC(C)C(C)C(=O)N1CCN(C2CN(C(=O)C(C)NS(C)(=O)=O)C2)CC1 1307,C(=O)(CC(F)(F)C(F)(F)F)N1CCC(C)(CNC(C(C(C)C)n2cccc2)=O)C1 1308,N1(C(c2cc(C(C)C)on2)=O)CC(NC(=O)Cc2cnco2)C2(CCOCC2)C1 1309,N1(C(CCCc2cc(C)sc2C)=O)CC2CC(NC(=O)C=CCF)C(C2)C1 1310,CCC(CC)C(C(=O)N1CCN(CCNC(C23CC(C)(CCO2)C3)=O)CC1)OC 1311,c1(-n2ncc(C(N(C)C3CC3)=O)c2)ccnc(F)c1.C1(C(=O)NC)(C)CCNC1 1312,C1(NC(C(CN(C)C)(C)C)=O)CC12CCN(C(c1sccc1I)=O)CC2 1313,N1(C(c2c(C)noc2)=O)CCCCC1C(=O)NC(CCO)C(C)C 1314,C1(CNC(=O)C=CC2CCCC2)CN(C(c2cn3c(n2)CCC3)=O)CCC1(F)F 1315,N1(C(COCCN(C)C)=O)CCC(C)(NC(C2CCCN(CC(F)F)C2)=O)C1 1316,C=CCCC(C(=O)NOCC1CC2C=CC1C2)NC(=O)C(CC)NC(N)=O 1317,C1(CN(C(C(CC)N(C(c2ccnn2CCF)=O)C)=O)CC)CCC2(CC1)CC2 1318,c1(N(C=O)CC23CCCCC2C3)ccc(OC(F)F)cc1F 1319,C(CCCCCN(C(=O)CCN1CCC1)C)NC(C(C)C1CCCO1)=O 1320,N1(C(C(c2nccc(C)c2)(F)F)=O)CCC2(CCCC(CNC(=O)CO)O2)CC1 1321,C1(NC(c2cccc(C#C)c2)=O)CC2CCC(C1F)N2C(C1(CF)CC1)=O 1322,Cc1ccc2c(c1)CC(NC(=O)N(C)C(c1cccs1)C)CO2 1323,C1(CNC(c2onc(CC)n2)=O)CC2(CC2)CN1C(=O)C(OC)OC 1324,C(=O)(C1=CCCC1(C)C)N1CCC(O)(CNC(c2sc(C)c(O)n2)=O)C1 1325,C1(c2nnnn2CCCC=C)(C(=O)NC(CN)(C)C)CCCC1C(C)(C)C 1326,N1(C(C=CSC)=O)CCCC(CNC(=O)C(F)(F)C2CCOCC2)CC1 1327,C1(C(N2CC(NC(c3ccc(C(N)=O)nc3)=O)(OC)C2)=O)(COC)CCOCC1 1328,N1(C(C2(C#N)CC2)=O)CCC2C(NC(=O)CSCc3ccccn3)C2CC1 1329,C1(C(=O)NC2C3CN(C(C(C=C)(C)C)=O)C2C3)Cc2cc(C)ccc2O1 1330,Cc1nc2c(o1)CCN(C(=O)C(CCOCCO)NC(=O)CN(C)C)C2 1331,c1(C(=O)NC2C(CNC(c3c(F)ccc(C#C)c3)=O)C2)csc2c(F)cccc12 1332,N1(C(CCC2CC(OC)C2)=O)CCN(C(c2ccc(O)cc2Cl)=O)C(C(C)C)C1 1333,c1(CCC)ncoc1C(N1CC(Cn2cc(-c3cnc(C4CC4)o3)nn2)C1)=O 1334,C1(NC(C=CCC)=O)COC2(CCN(C(=O)CC3(C#N)CC3)CC2)C1 1335,c1(NC(C2C3CC2N(C(=O)CCCn2ccnc2)C3)=O)cnc(Br)nc1 1336,C1(CC)CN(C(c2ccc(Cl)cc2Cl)=O)CCC1NC(c1cnc(C)nc1O)=O 1337,C(CC)(C(=O)N1CC(C(=O)NCC2(CO)CC2(C)C)C1)=COC.C(C)(=O)O 1338,C1(C(CNC(C2CCC2)=O)NC(C2CC(CF)C2)=O)CCCCC1 1339,C(=O)(C#CC1CCOCC1)NC(C1CCN(C(c2cc(Cl)cc(C)c2O)=O)C1)C 1340,C1(C(=O)NCC(C)N(C)C2CC2)CCN(CCN2CCCC2)C1 1341,c1(C(=O)NC2(CC=C)CCN(C(=O)C(O)CSC)CC2)cc2cc(C)ccc2[nH]1 1342,c1(C(=O)NCC2(NC(c3cn(C)c(=O)cn3)=O)CC2)coc2ccc(F)cc12 1343,c1(C(=O)NCC(CC)(C)NC(=O)COCCSc2nccn2C)cc(Cl)ccc1N 1344,C(=O)(C(CC1CC1)C1CCC1)NCCCCN(C(=O)C(c1cccnc1)O)C 1345,c1(NC(c2c(C(C)NC(CC3C(C)OCC3)=O)noc2)=O)ccc(O)cc1Cl 1346,C1(C(=O)NCC2CN(C(C3CC4CCC(C3)S4)=O)C2)CCc2ccnn2C1 1347,C1(OC)CC(NC(c2ccsc2)=O)CN(C(c2cncc(OC(C)C)c2)=O)C1 1348,C1(C(=O)OC)CN(C(C2(F)CN(C(C3CC3F)=O)C2)=O)CCC1O 1349,O=C(CCC(=O)NC1CCC(F)(CNC(=O)CSC2CC2)C1)c1cccs1 1350,CCCC(CCC)CC(=O)N1CC=CC1C(N1CCC(C(C)O)CC1)=O 1351,CC#CCCCC(=O)N(C(C)CNC(=O)C(c1ccc(N(C)C)cc1)C)CC 1352,C1(OC(c2cc(-c3ccccc3Cl)no2)=O)CCCN(c2nccc(Br)n2)CC1 1353,c1(SCCN(C(C(C)N(C(CNC(c2cnc[nH]2)=O)CO)C)=O)C)ccccc1 1354,C1(O)(C(N)=O)CCCN(C(C2CSCCN2C(c2cc(Cl)cs2)=O)=O)C1 1355,c1(C(C(N2C(CNC(CC=CCC)=O)CC2)=O)C)cc2ccccc2nc1O 1356,N1(C(C2C(=C)C2)=O)CC(C(=O)NCCc2c(C(C)C)n[nH]c2)C(C)C1 1357,C1(C(=O)OC)C2C=CC(CC2)C1C(N1CCC(NC(C2CC2c2cnc[nH]2)=O)C1)=O 1358,C1(N(C(C(C=C=C)C)=O)C)CN(C(=O)C(F)(F)Cc2ccccc2)CC12CC2 1359,C1(C(N(CCn2cc(C3(COC)CCOCC3)nn2)C2CC2)=O)CCC(O)CN1C 1360,c1(CSC)cccc(NC(=O)C(c2sccc2NC(=O)OC(C)(C)C)C)c1 1361,C1(C(N(C)CC2CCCC2(C)C)=O)CN(C(C2CC(O)C2)=O)CCC1(C)C 1362,N1(C(C(CC)(F)F)=O)CC2C3CCC(C2C1)N(C(=O)C(c1cscn1)N(C)C)C3 1363,CCC(C(=O)NCC(C(C)C)NC(=O)CCCc1cc[nH]n1)C(C)(C)CC 1364,C1(SCC)CCC(C(=O)NCC2CCCN(C(=O)CC3CCC(C)(C)O3)C2)CC1 1365,N1(C(C(=O)NC2C(C(N(C(CCC)C)C)=O)COC2)C)CCCCC1=O 1366,c1(C(N2C(CNC(CCC#C)=O)CC(F)C2)=O)cc(OC)cc(F)c1 1367,Cn1nnc2cccc(C(=O)Nc3cccc(CSc4ccc(Br)c(O)c4)c3)c12 1368,C12(NC(CC(=O)N(C)C)=O)CCC(CNC(c3cn(C)cn3)=O)(C1)OC2 1369,CCCCC(C(=O)N1CCC(C)C1C(=O)N(C)Cc1cnn[nH]1)C(C)C 1370,N1(C(CCCOC)=O)CCCC2(NC(=O)CN(c3ccccc3)C)CC12 1371,N1(C(CCCC=C)=O)CCN(C(C23CC=CC(C2)OC3)=O)C(CC)C1 1372,c1(C(N2CC(NC(CN(C3CCCC3)C)=O)C(O)C2)=O)c(F)cccc1[N+](=O)[O-] 1373,c1(C(=O)NC2CC3(C2)CN(C(C2CCS(=O)(=O)N2)=O)C3)cc2cccnn2n1 1374,CCC#CCN=c1nc(N2CCC(c3ccccn3)CC2)c2c([nH]1)CCC2 1375,c1(C(=O)NCC(CCNC(C2C(CC)C2)=O)OC)coc2c1C(=O)NCC2 1376,c1(N(C(C(C)C)=O)CC#N)ccccc1[N+](=O)[O-].c12nc(cs1)SCC(=O)N2C(C)=O 1377,CCC(CC(=O)NC(CC(F)F)C(=O)N1CCCC(C(C)C)CC1)CC(C)C 1378,CN1CC=C(CC(=O)NCC2CCN(C(=O)C=Cc3cocn3)C23CCC3)CC1 1379,Cc1cc(Cl)cc(C(N2CC(NC(C3(F)CCC3)=O)CC(C)C2)=O)c1N 1380,C1(C(=O)NC(C)(CNC(c2cc(C(F)(F)F)n[nH]2)=O)CO)COC2(CCC2)CO1 1381,c1(C(=O)NCCN(C(C2=C(C)OCC2)=O)C(C)C)c[nH]c2c(F)cccc2c1=O 1382,C(C(O)CCNC(=O)CCC1CCC(=O)C1)NC(C1(CCCC)CC1)=O 1383,C(=O)(C(CNC(c1ccc(C)c(F)c1)=O)C(C)(C)C)NCC1N(CC)CC1 1384,c1(CC(=O)NCCN(C)C(C2(C(C)(F)F)CCC2)=O)cnoc1 1385,C(=O)(C1=CCCCO1)NC12CC(NC(C3CCCC(C)C3)=O)(C1)C2.C(=O)(C1CC1)N 1386,N1(CC=CCNC(C2C3(CC(NC(C)=O)C3)C2)=O)CCCC(C2(C)CC2)C1 1387,N1(C)CCCC(CCO)C1.C12(CCCC1)C(N1CCC(C)C1)C(=O)N2.C(=O)NC 1388,C(=O)(N=c1ccn(NC(NC(CC)(C)C)=NCc2cc(Br)ccc2OC)[nH]1)OC 1389,C1(NC(C(C)CC#N)=O)CC(F)CN(C(c2nnc(O)cc2O)=O)C1 1390,C(C1=NOC2OCCC12)NC(=O)Nc1cn(C2C=CCCC2)nn1 1391,Cc1ccc(N)cc1C(=O)NCCN1CCCC(C(N)=O)C1 1392,C1(NC(C(C)NC(=O)CCCn2ccnn2)=O)CCC([N+](=O)[O-])CC1 1393,C1(NC(C=C(COC)C)=O)CCN(C(=O)Cn2ncnn2)C1n1cccn1 1394,c1(C(=O)NC(CC)CN(C(=O)CCOc2ccccc2)CC)cccc(F)c1N 1395,N1(C(C2CCC(C)CC2)=O)CCOC2(CCN(C(=O)C=C3CCC3)C2)C1 1396,N1(C(c2n[nH]cc2Br)=O)CCC(C2CC2)C1CNC(C1(CCF)CCC1)=O 1397,c1(C(N(C2CCN(C(CCC(=C)C)=O)CC2)C)=O)c(Cl)cccc1[N+](=O)[O-] 1398,N1(C(C(C=C)O)=O)CCCC2(C1)CN(C(c1cc3n(n1)CC(F)C3)=O)C2 1399,C12(C(=O)NCC3(C(=O)OCC)CC3)COCC1CN(Cc1cnnn1C)C2 1400,C1(C(=O)NC(C=CC(=O)NC2(CC#C)CC2)(C)C)CCCN1C(=O)OC 1401,C(CC(C)(C)C)(C(=O)NC(C)CC1(O)CCC1)NC(C(CCC)C)=O 1402,c1(CC)ccc(C(N2CCC(F)C(NC(c3cc(Br)ccc3Br)=O)C2)=O)cc1Br 1403,c1(C(N2CC(CCOC)(NC(C3CC(CC)(CC)C3)=O)C2)=O)cccc(F)c1O 1404,N1(C(=O)OC(C)(C)C)CCCC(C(O)C(=O)NC2CC2c2ccc(Cl)cc2)C1 1405,c1(C(=O)NC2C=CC(CNC(c3n(CC)ncc3)=O)C2)c(F)cccc1F 1406,C(c1cc(F)cc(F)c1)=CCNCC1C=CC(NC(Cc2c(C)cnn2C)=O)C1 1407,N1(C(CC2CCS(=O)(=O)C2)=O)CCCCC(N(CC(=O)NC)C)CC1 1408,C1(NC(CCn2c(C)csc2=O)=O)CC2(C1)CC(NC(C1(C3CC3)CC1)=O)C2 1409,N1(C(Cc2nc(C)on2)=O)CCC(C(N2CCOC(C)C2)=O)C2OCCC12 1410,c1(C(N(CCN2CCN(C(CC(C)N(C)C)=O)CC2)C)=O)ccc(C#N)cc1F 1411,C(=O)(C1CCCc2n[nH]cc21)N(C(CNC(c1ccc(CC)cc1N)=O)C)C 1412,c1(C(=O)NC(CNC(c2c(C(C)C)nns2)=O)CO)ccc2ncncc2c1 1413,CON(CCC(=O)NCC1CCCC(O)C1)C(=O)Cc1cnccc1Cl 1414,n1(-c2ccc(C)cc2)nc2c(c1NC(=O)C(=O)NCCC(O)C1CC1)CSC2 1415,C1(CC#C)(C(=O)O)CCN(C(C2CCC(N)CC2)=O)CC1 1416,c1(C(N2CCC(C)(CNC(C3CC3F)=O)C2)=O)ccn2c1CCCC2 1417,Cc1nc(C(=O)NCC2CC2CNC(c2ccc(Br)s2)=O)cn1C 1418,c1(OCC)ccc(Br)cc1C(=O)CCCNC1COCCC1c1ccc(F)cc1 1419,C1(C(=O)NC(CCNC(CNC(=O)NC)=O)C)CC(C)CO1 1420,CC(C)(C)CC(=O)NC1CC2C(NC(=O)CCOC3CCCOC3)C2C1 1421,Cc1ccc(SC(C)C(=O)N)cc1.C12(CN(C(C3C(C)CC3C)=O)C1)CC=C2 1422,c1(C(=O)NC(C(N2CC(OC(C)=O)C2)=O)c2ccoc2)coc(CSC)c1 1423,c1(C(=O)NCCC2(NC(=O)Cc3ccccc3F)CC2)nsc2c(Cl)cccc12 1424,n1(CCCC)nnnc1C(CCC1CC=CCC1)NCC(F)=C(C)C 1425,CC1CCN(C(C2(c3cccc(Cl)c3F)CC2)=O)CC1NC(C1(F)CC1)=O 1426,C(C)(CCC(=O)NCC(C1CCN(C(=O)C(C)(C)c2ccsc2)CC1)C)OC 1427,C1(C(=O)Nc2cn(CC#C)nc2)CC2C=CC1N(C(=O)Cc1cnn(CC)c1)C2 1428,c1(CCC(=O)OC)cccc(NC(C2(O)CCN(Cc3cnn(C(C)C)c3)C2)=O)c1 1429,C(N=c1cc(C)nc(Cl)[nH]1)C1CCC(NC(C2(CC)CCCCO2)=O)CC1 1430,C=CC(CC)C(=O)N(C)CCC1CCN(C(=O)CC2CC=CCC2)CC1 1431,C1(C(=O)NCCC(C(C)C)NC(c2ccoc2)=O)CCCCC(C)(C)C1 1432,CC1CCC(CC(N2CC(CC(F)C(=O)N3CCC3(C)C)C2)=O)C1 1433,N1(C(c2c(C)nsc2)=O)CC(N(C)C(c2cncs2)=O)C(F)C1 1434,CCC(CCOC)NC(c1ccccc1)=O.c12nncn1C2 1435,C=CCC(CC(C)C)C(=O)N1CCCC(C)(C)C1CNC(=O)CC1(N(C)C)COC1 1436,c1(CC(C)C(N2CC(NC(c3coc(C4CC4)n3)=O)CC2C)=O)ccccc1F 1437,CC1CCCC1(C)NC(C1(CNC(c2cnn(C)n2)=O)CCCCC1)=O 1438,CC1CCCC(O)(NC(=O)NC2(CNc3ccc(F)cn3)CCC2)CC1 1439,Cc1nc(C(C)C)sc1C(=O)NC1CCC(O)(CNC(C2(Cl)CC2)=O)C1 1440,c1(CC(C(=O)NC)Nc2nc3c(s2)CC(C)(C)CC3)ncc(Br)c2cccnc12 1441,N1(C(C23OCC(C)(C2)C3)=O)CCCC2CN(C(C3(C#N)CCCO3)=O)CCC12 1442,C(C)(C(c1nnnn1C1(C)CC1)Nc1cnn(-c2cccnc2)c1)(C1CC1)OC 1443,c1(NC(=O)Nc2cc(CCCC)sc2C)c(Cl)ccnc1Br 1444,c1(C(N2C(C(N3C(COC)C(O)CC3)=O)CC2)=O)ccc(C)c(C#N)c1 1445,C1(C#CC(=O)N2CCC(NC(=O)COc3ccccc3F)C2(C)C)(CC)COC1 1446,N1(C(C(CC)CC)=O)CCC2(CCCN(C(c3cc(F)c(F)c(F)c3F)=O)C2)C1 1447,n1(CC)cc(NC(C2CC(C)CN2Cc2cnc(N(C)C)cn2)=O)c(C)n1 1448,N1(C(C(C)(C(C)C)NC(C)=O)=O)CCC2(C1)CN(C(c1cc[n+]([O-])cc1)=O)CCO2 1449,C#CCC(C)(C(=O)NCC1NC(=O)CC1(C)C)NC(=O)CCc1nc(=N)[nH][nH]1 1450,c1(C(N2C(CNC(c3ncn(C)n3)=O)CC(OC)C2)=O)cc(Br)cnc1N 1451,c1(C(N2CCCC(C(C)NC(c3cc(C)n(C)n3)=O)C2)=O)ccn2cnnc2c1 1452,c1(OC)ccc(C(=O)NCC2CC(CCOC)CCN2C(C23CC(C2)C3)=O)c(F)c1 1453,c1(C(=O)NCC2(F)CCC(NC(c3c(C)noc3)=O)C2)cnc2ccccn12 1454,n1(CC(N2CCC(N(C(C(CCC)C)=O)C)C2)=O)ncc(C#N)c1Br 1455,C1(C(=O)NC2CCC(C(N3CC(N(C)C)C(F)C3)=O)CC2)CCCC(C#N)C1 1456,c1(C(N(C)CCNC(=O)CCc2cn[nH]c2)=O)ccc(CSC(F)F)o1 1457,C1(C(=O)NCC2C3N(C(C(C)OCC)=O)C(CC3)C2)Cc2cc(C)c(C)cc2O1 1458,CCCCCC(O)CC(=O)NC(CNC(=O)COc1ccccc1C)C(C)(C)C 1459,C(=O)CC1=NNC(=O)C1.C(CC(C)CCNC(=O)CSCCC(F)(F)F)OC 1460,N1(C(c2c(C(C)C)c[nH]n2)=O)CCC2CN(C(c3csc(O)n3)C3CC3)CC2C1 1461,C(=O)(C1=C(C#N)CCC1)N1CCC(OC)(CNC(C2CN(C)C2)=O)CC1 1462,C1(C(C)C)C(=O)N1.C1(CNC(C)=O)C2CN(C(=O)CC(C)CN(C)C)CC12 1463,c1(CC)cc(CC(=O)NC2C=CC(CC(=O)NC)C2)on1.C12CC(C1)CC(=O)N2 1464,C12(CNC(C(C3CC3)OCC)=O)CC(C(N3CCC(CCO)C3)=O)(CCO1)C2 1465,C1(CC=C)(C(=O)NC(c2cnc[nH]2)C)CCN(C(c2ccn(C)n2)=O)C1 1466,C12CCC(CC1)N(CC)C2=O.n1(CCCC)cc(COCC(C)O)nn1 1467,C(=O)(C1=CS(=O)CCC1)N1CCC(C(C)NC(C(C)c2cccs2)=O)CC1 1468,Cc1ccnc2c(C(=O)NCC3CC(NC(c4[nH]cnc4C)=O)C3(C)C)cnn12 1469,O=C(C=CCN(C(=O)CN1CCCCC1)C1CC1)NOCCF 1470,n1(CC)c(C)cc2c1CCCC2NC(c1cc(C(=O)O)ccc1C#N)=O 1471,c1(OC)cc2[nH]ncc2cc1NC(=O)C(=O)NCC1CN2CCC1C2 1472,N1(C(c2ncn(CCNC(C(C)n3ccnn3)=O)c2)=O)CCCCCC1C 1473,N1(C(C2CCSC2)=O)CCc2c(CO)cccc2C1 1474,c1(C(=O)NC2C(CNC(CSC(C)C)=O)C2)coc(Cl)n1 1475,C1(CNC(=O)C(O)CC2CCCCC2)COCCN(C(C2CCC2)=O)C1 1476,C1(OC)CC2(C1)CC(NC(c1cn(CCNC(C3CCC(=O)N3)=O)nn1)=O)C2 1477,C1(NC(Cc2ccc(C)cc2)=O)CCN(C(c2ccc(C)n2C)=O)CC1C(C)C 1478,c1(C(=O)NCC2CC(NC(C3(C)C(CC)CCC3)=O)C2)sc2nccnc2c1NC 1479,O(NC(=O)C(F)CC1CCN1C(=O)COc1cc(C)[nH]n1)C(CC)CC 1480,CC1CCN(C(=O)C(O)Cc2ccco2)CC1CNC(c1ccc(C2CC2)nc1)=O 1481,c1(OC)cc(CN2CCC(NC(c3cccc(F)c3I)=O)C(F)C2)ccc1C 1482,CN1C(=O)C(=O)N(CC(=O)NC2CN(C(C3COC(C)(C)O3)=O)CCC2C)C1=O 1483,C1(C2CCN(C(=O)CCCCC(C)=O)CC2)(NC(c2c(SC)cccn2)=O)CC1 1484,N1(C(=O)C=CSc2nc[nH]n2)CC2(CCCC2NC(=O)C(F)(F)C(F)F)C1 1485,Cc1nccc(Cl)c1C(N1CC(N(C(=O)C(Cl)=CCl)C)C(C)(C)C1)=O 1486,c1(C(=O)NCC2N(C(CC3(C)CC3)=O)CCOC2)cnn2c1S(=O)(=O)NCC2 1487,c1(OC)ccc2oc(C(F)F)c(C)c2c1.n12cc(nn1)CCNC(=O)C2C.CC=CC 1488,Cc1csc(C(=O)NC2(C(=O)NCCCC3CCOC3)CC(O)C2)c1 1489,N1(C(C2(NC(=O)NCC)CCCC2)=O)CCCC(CN(C(=O)C(C)SC)C)CC1 1490,C1(CNC(C2CCC(=C)CC2)=O)CC2CN(C(c3coc(C)c3)=O)CC12 1491,c1(OCCC)cccc(C(N2CC(O)CC2CNC(c2cnnn2C)=O)=O)c1 1492,C(C(C)C(F)C(=O)NCC1CCC(=O)NC1C)NC(CC=CC=C)=O 1493,C12CCN(C13CCC3)C2=O.O=C(CCCOc1ccccc1)NC1CC1 1494,Cc1cc(C)n(CC(N2CC(C)(CCC(=O)NC3(CO)CC(F)(F)C3)C2)=O)n1 1495,C1(CC)CCCC1(C)C(=O)NC1C2CC1N(C(=O)C(N1CCCC1)C1CC1)C2 1496,N1(CCN=c2nc(NC(=O)OC(C)(C)C)[nH]s2)CC2CC3(CCC3)C2C1 1497,N1(CC)CCC(CN(C(=O)C(O)CNC(=O)C(F)=C2CCCC2)C)C1 1498,C1(NC(Cc2cn(C)nc2)=O)CCC2(CC1)CN(C(C1COC(=O)C1)=O)C2 1499,Cc1ccc(C=O)cc1C(=O)NCCNC(=O)C(CC(C)C)n1ccnc1.C(CO)S 1500,c1(C(C)(C)Cc2n(CCOC)nnn2)ccc(OC)nc1.C1(C)(N)CC1 1501,C1(NC(c2ccc(CCC)cc2)=O)C2CCCN(C(C3CC3F)=O)C2C1(C)C 1502,c1(C(=O)NC2C(NC(C3(C(=O)NC)CC3)=O)COC2)[nH]c(O)nc1C 1503,c1(C(=O)NCCCN(C(=O)Cc2ccccc2)CCO)ccc(O)c(Br)c1 1504,N1(C(C(CC)C(C)C)=O)CCC2CC(NC(=O)CCCn3cccn3)CCC2C1 1505,N1(C(C(C)=O)=O)CC2CC(NC(=O)CN3CCOCC3=O)CC1C2 1506,c1(C(N2CCN(C(C3(CF)CC3(F)F)=O)CC2)=O)cc(F)cc(Cl)c1O 1507,C(=O)(C(C)CC(=C)C)NCCCCN(CCCNC(CC=C=C)=O)C 1508,C1(OC)CN(C(=O)C=Cc2csnc2C)CC1CNC(=O)CSCC1CCCO1 1509,c1(C(=O)NC(CC)CNC(=O)C(=O)NC(C)C)sc(C(C)C)nc1C 1510,CCCC(C)CCN=c1[nH]ccc(=NCCc2cc(F)ccc2Cl)[nH]1 1511,CC(C(=O)N(CC)Cc1ccccc1)C(C)NC(c1cccnc1N)=O 1512,c1(CC(=O)NC(CC)CN(C(c2cc(C)ncn2)=O)CC)ccc2nsnc2c1 1513,Cc1[nH]c(C)c(C(N2CCC(CN(C(=O)CCC3CCN(C)CC3)CC)C2)=O)c1C 1514,S(=O)(=O)(c1cc([N+](=O)[O-])ccc1Cl)Nc1c(I)cc(C)c(C)c1 1515,C1(N(C)C)CC(N=c2[nH]c(N3CCc4nc(N(C)C)sc4C3)nc(=N)[nH]2)C1 1516,C(=O)(C(C)(O)CCC)NC(CCNC(c1c(CC)nn(-c2ccccc2)c1)=O)C 1517,N1(C(CC2CC(C)(C)C2)=O)CCN(C(C2(F)CC2)=O)CC1c1cccc(Cl)c1 1518,CN1C(=O)NCC1C(=O)NCCN(C1CCCC1)C(c1ccc(F)cc1)=O 1519,C1(C)(CNC(C(C)C2CC2)=O)CCCN1C(=O)CS(=O)(=O)NC(C)(C)C 1520,C(C)(C)(CCN=c1cc(Cl)nc(CS(C)(=O)=O)[nH]1)NC(C(CC#C)CC(F)F)=O 1521,C(=O)(C#CC1CCOCC1)NC1C(CNC(C2(CC(=O)OC)CC2)=O)CCC1 1522,N1(C(COC)=O)CC(CNC(c2cnn(C(CC)CC)c2C2CC2)=O)C2CC12 1523,C1(CC(=O)NC2CC3(C(NC(CCSCC(C)C)=O)C3)C2)CCCCC1(C)C 1524,C#CCC(C)(CC)C(=O)N1CCCC1CNC(C1(O)CCSCC1)=O 1525,Cc1ccc2c(N(CCCF)C)nc(N(C)CC3CCCS3)nc2c1 1526,C(C)(C(CC(=O)NCCc1ccc(F)nc1)NC(=O)CCN1CCCCC1)OC 1527,C1(NC(CCc2cncc(C)c2)=O)CCN(C(=O)C(C)n2cccc2)C(C)C1 1528,CC(C(C(=O)NCCOCC1CC1)N1CCCC2(CC1)CC2(F)F)C(C)(C)C 1529,C1(CNC(C2C(=C)CC2)=O)CCCCN(C(=O)CSCc2ccccn2)C1 1530,c1(CCC(=O)NCCC(C)N)ccccc1OCC(=O)NC1CCCC1SC.CC 1531,CCCCCC(=O)NCC(C)N(C(=O)Cc1cccnc1)C 1532,Cc1cc(F)ccc1C1CC1C(=O)NC(C)(C)C(C)NC(c1cc2occc2[nH]1)=O 1533,c1(C(=O)NC(CCCNC(c2nc(NC(C)=O)sc2)=O)C)ncnc2cc[nH]c12 1534,N12CCCC(C)(C1)NC(CC1CCOC1)C2=O.C(C(C)O)N(CCO)CC 1535,C1(O)(CNC(=O)C=CC2CCCCC2)CCCN(C(C2CC2C(F)(F)F)=O)CC1 1536,C(=O)(C(CO)NC(=O)CC(C1CC1)C1CC1)N(CC(=O)NCC)CC#C 1537,c1(C(=O)NCCCN(C(CC2CC(CC)C2)=O)CC)ccc(F)cc1C(F)(F)F 1538,N1(C(CC(C=C)CC)=O)CCC(C(=O)NCCc2cccnc2F)C(C)(C)C1 1539,C1(NC(C2C(CC)CN(C(C3(CC)CC3)=O)C2)=O)CC2(CCC2)C1O 1540,C1(C(N2CCN(C(c3cccc(C)c3)=O)CC2C)=O)CC2CCCCN2C1 1541,C1(C(N(C)CC2CCN(C(c3c[nH]c(=N)s3)=O)CC2)=O)CCC(=O)N2CCCC12 1542,Cc1nc2ncc(C(=O)NC(CNC(=O)Cn3cncc3C)CC(C)C)cc2o1 1543,C1(NC(C23CCC(C2)C3)=O)CCCC(NC(C2(Br)CC2)=O)C1 1544,C1(CC(=O)NCCC2CCC(C)C2)CCN(C(=O)C2=NNC(=O)C2)C1(C)C 1545,C#Cc1ccc(C(=O)NCC(O)CCNC(c2c[nH]cc2C)=O)cc1 1546,C(C(N=c1cc[nH]c(-c2ccc(F)cc2)n1)C1CCC1)NC(=O)Cc1cnns1 1547,C1(NC(C(CCF)NC(COCCC)=O)=O)C2CCC(C2)C1C 1548,C(=O)(C#CC1CCCOC1)NC(CNC(Cc1c(OC)ccnc1)=O)CO 1549,N1(C(c2cncc(C=C)c2)C(=O)NC(C)(C)C)CC(=O)N2CCCCC12 1550,c1(-c2cc(C3CC3)cc(C)c2)cccc2c(-c3cnc4[nH]cnc4c3)c[nH]c12 1551,CC(CCC(=O)N1CCC(C)(CNC(=O)COCC(C)(C)C)C1)N(C)C 1552,C1(N(C(c2ccccc2)=O)CC)CCCN(C(C2CCC2(C)C)=O)C1 1553,c1(CC)nn(C)c(Cn2cc(CCNC(=O)CC3OCCC3(C)C)nn2)c1Br 1554,N1(C(CCCSC)=O)CC(NC(=O)C=CC2CCCCCC2)CC(C)(C)C1 1555,c1(N(C2CCNC2)Cc2cc(OC)cc(C)c2)ncnc2ncn(C)c12 1556,c1(OC)nc(C)sc1C(=O)NCC1CCC(NC(c2ccc(C(F)F)nc2)=O)C1 1557,C1(CNC(C(C)(C)SC)=O)CC2CCC(C1)N2C(=O)CCn1ccc(=N)[nH]1 1558,C(=O)(CCCS(C)(=O)=O)N1CC(NC(C(C=C)(C)C)=O)C2C(C1)C2 1559,C1(C(=O)OCC)CC2CCC1N(C(=O)C(=O)NCc1cccc3c[nH]nc13)C2 1560,C1(C(=O)NC2(CCOCC)CC2)CCCN(C(=O)CCCOC)C1 1561,N(C(=NCCC(C)(C)COC1CC1)N1CC=C(CC)CC1)C(C=C)C 1562,S(=O)(=O)(c1cc(C(=O)N(C2CCCOC2)C)oc1C)NC 1563,C12(OC)CCN(C1)C2=O.C1(CC)CC(CNC(=O)CSCCN(C)C)C1 1564,CCCC(CCCNC(C1(O)CCC1)=O)NC(c1cc(CO)n(C)n1)=O 1565,c1(C(N(CCCNC(C2CC2c2cnn(C)c2)=O)C)=O)ncc(F)cn1 1566,CC1(C)CC(NC(C2CC2F)=O)CCN(C(=O)CCc2cc(Cl)cs2)C1 1567,C1(n2cc(-c3cncc(C)c3)nn2)(C(=O)NC2(C(=O)NC)CCC2)CCOCC1 1568,N1(C(C(=O)NCCC)CCC2CCCCC2)CCCC(C2CCN(C)C2)C1 1569,CN=c1[nH]c(C(N2CCN(C(C)CNC(=O)CC3CC34CC4)CC2)=O)cs1 1570,C1(CNC(c2n(CC(C)C)ncc2)=O)CN(C(C2CC2(F)F)=O)CCC1(C)C 1571,c1(N2CC(C)(NC(C3CCC(C)O3)=O)C2)ncccc1C#N.c12ncoc1CCN2 1572,N1(C(C=CC=CCC)=O)CC(CNC(c2c(C)cccc2F)=O)N2CCC1C2 1573,c1(C(=O)NC(CC(C)NC(Cn2c(C)nc(C)n2)=O)C)cc(S(N)(=O)=O)sc1C 1574,Cn1c(C(=O)NCCC2CCCN2C(C2CC2F)=O)c2n(c1=O)CCCC2 1575,c1(N2CCN(C(c3ccn(CC(C)C)n3)=O)CC2C(C)C)cc2nncn2cn1 1576,C1(N(C(C(CCC2CC2)NC(CCC=C)=O)=O)CC)CN2CCC1CC2 1577,C(=O)(C(C)CCCC(C)=O)N1CCC(CCOC)(C(N2CC(C)C(F)(F)C2)=O)CC1 1578,c1(N2CC3CCNC(=O)C3C2)nc(N2CCn3ncc(Cl)c3C2)c2c(n1)CCC2 1579,N1(C(C2N(C(c3cccn3C)=O)CCC(CC)C2)=O)CCCC(C2CCC2)C1 1580,CCC(CC(=O)NC1C2CN(C(c3cccc(N)c3Br)=O)CC12)C(C)C 1581,C(CC(C(=O)NCC1CC2CC2C1)NC(c1cnc(C2CC2)o1)=O)OC 1582,C1(C)(C(N(CCNC(c2nccc(OC)c2N)=O)C)=O)CC(C2CC2)=NO1 1583,Cc1ccccc1CCC(C)NC(=O)NCC1(C(=O)OC)CC(OC(C)(C)C)C1 1584,N1(C(=O)NC)CCCN(N2CCS(=O)(=O)C(CSc3n[nH]c(C)n3)C2)CC1 1585,C=CCCCC(C)(C)C(=O)NC(C)CNC(=O)Cc1ccc(O)c(Cl)c1 1586,CC(CC(=O)NC1CN(C(=O)COC(c2ccccc2)C2CC2)C1)C(F)(F)C(F)(F)F 1587,Cn1nc(C2CC2)cc1C(N1CCC(NC(c2cc[nH]c(=N)c2)=O)C1)=O 1588,c1(OC)cc(CC(N2CCCN(C(C3CC3F)=O)CC2C)=O)c(F)cc1O 1589,S(=O)(=O)(c1cccc(OC(C)(C)C)n1)NCCCC(CCC)Nc1ccccc1 1590,Cc1cccc2[nH]cc(C(=O)NC3CCC3CNC(C34CCC(C3)C4)=O)c12 1591,Cc1ccc2oc(NCC3CCCN(C(c4cnc(F)c(Cl)c4)=O)C3)nc2c1 1592,N1(CC)CC(NC(=O)CCC2CCCN2C(=O)CC2CCC(C)C2)CCC1=O 1593,C1(C)(C(=O)NCCc2c(C)ccnc2)CCCN(C(C2CCN(C)C(=O)C2)=O)C1 1594,c1(C(=O)NCC(CC=C)NC(=O)C(C)SCC)cc(C)nc2ccc(C)cc12 1595,Cc1cccc(NC(=O)CCNS(C)(=O)=O)c1F.C1(=O)CCCCCO1 1596,N1(C(C(C)C)=O)C(C(=O)N(C2CCCN(C)C2)C)C2CC(O)C1C2 1597,N1(C(C2(CC=C)CC2)=O)CC(CNC(=O)C(COC)N(C)C)CC(C)(C)C1 1598,CCC(O)C(C)C(=O)NC1CCCN(C(=O)CSS(C)(=O)=O)C1C 1599,CC1(NC(c2cccc(Cl)c2O)=O)CCC(NC(=O)C(O)c2ccco2)CC1 1600,N(C1CCc2c(CF)cccc21)C(c1ccc(Br)c(Cl)c1)F 1601,N1CC(NC(=O)CCC(=O)Nc2nnc(C)s2)C(O)C1.C(=O)(C1CC1)OC 1602,N1(CCCNC(CC2CCC(C)(C)C2)=O)CCC2(CC1)CSC2 1603,CCC(CC)(CO)C(=O)N1C(C(=O)NCc2cccc(Cl)c2)CC2CC12 1604,C1(O)(CNC(c2cn(CC)nn2)=O)CCCN(C(c2cnc(N(C)C)cn2)=O)C1 1605,c1(C(C)NC(C2(F)CN(C(C(c3ccccn3)C)=O)C2)=O)ccc(Cl)nc1 1606,C1(NC(CC2N(C(C3CCCC(C#N)C3)=O)CCCC2)=O)CCC2(CCCC2)C1 1607,C123CC4CC(C1)CC(C4)(C2)CNC3=O.c1(NC(c2coc(Cl)n2)=O)cncc(Cl)n1 1608,O=C(C1=CC2(CCOC2)C1)NCC1CCN(C(c2nocc2Br)=O)C12CC2 1609,c1(C(=O)NCCCC(C)NC(CC(CC)(C)C)=O)cc2ncccc2o1 1610,CCC(C)CCCCC(=O)NCC(CO)Nc1ncnc2[nH]cnc12 1611,C(=O)(CCS(N)(=O)=O)OCCCNCCC=CCNC(C(CC=C)C)=O 1612,C1(CNC(C(n2cc(-c3nccs3)nn2)C)=O)CC(C2CC2)=NO1 1613,C12(C(C(=O)NCCCCNC(CCCC)=O)=O)CC3CC(CC(C3)C1)C2 1614,Nc1ccc(C(N2CC(NC(C3CC3C3CCC3)=O)C(F)C2)=O)cc1[N+](=O)[O-] 1615,c1(C(=O)NC(C(=O)NC(CCC=C)CO)CCCC)ccc(=O)n(C)c1 1616,c1(C(=O)NC(COC)CC(=O)NCC=CCSC)cc(C)cc(O)n1 1617,c1(C(c2cc3c(cc2)C(=O)CC3)OC)cn(C2CCc3c(F)cc(Cl)cc32)nn1 1618,C(=O)(C(C)CS(C)(=O)=O)N1CC2(CC(NC(CN3CC(CC)C3)=O)C2)C1 1619,C1(CC)CN(C(=O)CCc2ccc[nH]2)CCC1CNC(c1cnc(C)cc1Cl)=O 1620,C(=O)(CCC(F)(F)F)NC(C(C)C)CNC(c1cccnc1N(C)C)=O 1621,C#CC1CCC(C(N2CCC(C#N)(CO)C2)=O)CC1.n12cc(nn1)CC1(CCC1)C2 1622,c1(OC)cc(F)c(C(N2CC(N(C)C(c3cn(CF)cn3)=O)C(F)C2)=O)cc1N 1623,c1(C(=O)NC2CCN(c3ncccn3)C2)ccc2c(c1)CCCCN2 1624,C1(C(N2CC(OC)C(NC(=O)C(C)C3=CCCC3)C2)=O)CCc2[nH]nc(O)c2C1 1625,c1(C(=O)NCCCCC(C)NC(C(C)NC(C)=O)=O)cc(C)c(F)cc1N 1626,CC1c2ccccc2CN1C(N1CCCCC(O)(CNC(=O)NC(C)(C)C)C1)=O 1627,Cc1nc2scc(-c3ccccc3)c2c(=O)n1CCOC(=O)Nc1cccc(Br)c1 1628,Cc1c[nH]cc(C(=O)NC2CCN(CCNC(C3(F)CC3C)=O)CC2)c1=O 1629,c1(C(N(CCCNC(c2c[nH]c(=NCC)s2)=O)C)=O)cc2ccccc2n1C 1630,c1(C(N2C(C(N3CCN4CCC3CC4)=O)CC(=C)C2)=O)cc2nc(C)ccc2o1 1631,C1(C(=O)Nc2ccccc2)CCCN(C(=O)C(=O)NCc2cncnc2)C1 1632,N1(C(c2c(C(C)C)n[nH]c2)=O)CCOC2CCN(C3CC3)CC12 1633,C1(C(N(C2CN(C(C3(CCOC)CC3)=O)C2)C)=O)CCCCC12CC2(F)F 1634,c1(C(=O)NC(C(=O)NCCOCCCC)C2(C)CC2)ccc2n[nH]cc2c1 1635,Cc1cc(F)ccc1CC1(C(=O)NCC(CNC(=O)CC2CCOC2)CO)CC1 1636,C1(C(=O)NCC(C)=CC(=O)NCc2ccncc2Cl)CC=CCC1C 1637,Cc1cc(C(=O)NCc2ccc(CF)cc2)cc(C)n1 1638,c1(C(N(CC(C)(C)NC(=O)CNS(C)(=O)=O)C)=O)ccncc1F 1639,c1(C(=O)NC2CCC(N(C(=O)CNc3cccnc3)C)C2)cnn2ccccc12 1640,C1(F)(C(=O)Nc2ccc(N(C)C)nc2)CCCN(C(C2CCC3(CCC3)C2)=O)C1 1641,CC1CCCn2ncc(C(=O)NC3COCC3N=[N+]=[N-])c21 1642,C1(OCC)CN(C(=O)C(C)SC(F)(F)F)CC1NC(=O)CSCc1ccccc1C 1643,C1(NC(c2cccc(C(=O)NC)n2)=O)COCCN(C(=O)Cc2cc(C)cs2)C1 1644,c1(C(N(C)CCNC(=O)CC(F)(F)c2ccccc2)=O)cccc2oncc12 1645,c1(C(N(C(C)C(=O)NCCF)CCOC)=O)ccc(C)nc1 1646,C1(NC(c2cc(-c3ccncc3)[nH]n2)=O)CC(F)CN(C(c2scnc2Cl)=O)C1 1647,C12(C(=O)NCC3C(CNC(c4ncc(C)cc4F)=O)C3)C3CCC(CC13)C2(F)F 1648,c1(SC)cccc(C(N2CCCC(N(C(=O)C(C(C)O)N(C)C)C)C2)=O)c1Cl 1649,C12(CNC(COCC(=C)C)=O)CC(CO1)N(C(=O)C(C)(C)n1cnc(C)c1)C2 1650,c1(CN(C)CC2COC(c3ccccc3)C2)nc(C(C)(C)O)cs1 1651,C1(NC(c2cnc(C)[nH]2)=O)CCCN(Cc2cn(C3CCCN(C)C3)nn2)C1 1652,Cn1cnc2ccc(C(=O)NCC3CCC(NC(C4CS(=O)(=O)C4)=O)C3)nc12 1653,N1(C(c2c(CCC)n[nH]c2)=O)CC2CC2C1C(N1CCC(CN=[N+]=[N-])C1)=O 1654,C(=O)(C(=O)N=S(C)(C)=O)N1CC(C)(NC(c2ccc(OC3CC3)c(Cl)c2)=O)C1 1655,C12(CNC3C(C(=O)Nc4c(Cl)cc(C)cc4Cl)CCC3)CC3CC(CC(C3)C1)C2 1656,C1(C(N2CCC(=CCC)C2)=O)CCN(C(c2cscc2C)=O)C12CC2 1657,c1(C(N2CCN(C(C=CC=CC)=O)CC2)=O)cc(S(=O)(=O)NCC(C)C)c[nH]1 1658,C1(O)(CNC(c2c(C)nn(C(C)C)c2)=O)CCN(C(C2CC2F)=O)CC1 1659,C1(C(=O)NCc2ccnc(OC)n2)CCN(C(c2csnc2C)=O)C(C)C1 1660,c1(CC)cc(=NC(=O)C2C(O)CCN2C(C2CNC(=O)CC23CCC3)=O)[nH]n1C 1661,C(CC1=CCCCC1)NC(C=CC(C)NC(=O)CC(C)O)=O 1662,C1(C(C)(C)C)(C(C(=O)CCN(C(=O)C=CCl)C2CC2)=O)CCCO1.C(CN)N 1663,N1(C(c2cn(CC=C)nn2)=O)CCOC(C)(CNC(=O)CC=CCO)C1 1664,N1(C(CC2C(NC(C(C)(C)SC)=O)C2)=O)CCN(C2CC2)CC1 1665,CC1(C)C2CN(C(C3COC4(C3)CN(C(c3cnsn3)=O)C4)=O)CC12 1666,C(=O)(CC(C)C(=O)NCCCNC(c1cc(N2CCCC2)ccn1)=O)NC 1667,C(=O)(CC(CN(C)C)C(F)(F)F)N(CCCCNC(C1(CO)CCCCO1)=O)C 1668,C1(C(=O)NC(C2(O)CCN(C(C3CC(O)C3)=O)C2)C)CCc2nnnn2CC1 1669,C#CCCCCCC(=O)N(C1CCN(C(=O)C(C)CSc2ccccc2)C1)CC 1670,c1(C(=O)NCc2ccc(C(N3CCC(COCC)C3)=O)s2)n[nH]c(C)c1Cl 1671,c1(NC(C2CCN(C(=O)NC)C2)=O)cc(F)cc2ccncc12 1672,c1(OC)cncc(C(N2CC(C(=O)NC(c3ccc(OC)cc3)C3CC3)C2)=O)c1 1673,N1(C(C(CCC2CCC2)NC(C2N(C=O)CC2)=O)=O)CC2(CCC(O)CC2)C1 1674,C(=O)(C(C)S(=O)(=O)C(C)C)NCCN(C(c1c(N)sc(C)c1C)=O)C(C)C 1675,c1(C(C)NC(C)=O)c(F)cc(Cl)cc1F.c1(OC)ccc(C2CN2)cc1 1676,c1(C(=O)NC2(C)CC(NC(CCCCC=CC)=O)C2)cc(N)c(C)c([N+](=O)[O-])c1 1677,N1(C(C(CCC=C)NC(c2ccc(N)c(F)n2)=O)=O)CC2CCC(O)C2C1 1678,C(C(=O)N1CCN(C(=O)CC(C)(O)C2CC2)CC1CCO)(C(C)(C)C)NC(C)=O 1679,N1(C(CC(n2c(CC)ncc2)C)=O)CCC(O)(CCNC(c2ccon2)=O)C1 1680,C(C(CO)(CO)NC(=O)Cc1ncsc1Cl)N(C(C(C)CF)=O)C 1681,C1(C(=O)N(C)CCc2cncnc2)(CC)CCN(C(=O)CC2CSCCO2)CC1 1682,C1(NC(c2ccc(C(N)=O)[nH]2)=O)COCCN(C(c2cc3occc3[nH]2)=O)C1 1683,CP(C)(=O)C(O)C(=O)N1CCC(O)(CNC(c2ccc(=O)oc2)=O)CC1 1684,c1(NCCCCCC)ccc(S(=O)(=O)N2CCCC(C)C2CO)cc1C#N 1685,c12ccc(F)cc1CNC2=O.C1(C(=O)NCC2(SC)CC2)(C(F)F)CCC1 1686,C1(CC(=O)NCC2N(C(C(C(C)C)SCC)=O)CC2)CCCCCCC1 1687,S(=O)(=O)(c1cn(C)cn1)NCC(=O)NCC1CC(NC(c2c(C)cc(C)s2)=O)C1 1688,CC1(C(=O)NC2C=CC(CC(=O)NCCc3noc(=O)n3C)C2)CC=CCC1 1689,N1(C(=O)NC2(c3ccccc3)C(C)(C)C2)CCNC(=O)c2c(Br)cccc21 1690,N1(c2nc(C(C)C)nc(Cl)c2)CCS(=O)(=O)C(CC=CCC(=O)NCC#N)C1 1691,C(=O)(C(C)C(O)CCC)N1CC(C)(CNC(C2(C(F)(F)F)CC(=C)C2)=O)C(C)C1 1692,N1(C(=O)NCCCOCCOC)C2CCCC1CC(N)C2 1693,Cc1nc(O)ccc1C(N1CSCC1C(=O)NCC(C)(C)C#N)=O 1694,c1(C(C(=O)N(C2CCN(C(CC(=O)N(C)C)=O)C2)C)(F)F)ccc(Br)nc1 1695,c1(C(=O)NC(C(=O)OC)Cc2cc(C)cc(O)c2)ccc2[nH]cc(C#N)c2c1 1696,C1(NC(c2ncc(C)nc2)=O)CCN(C(=O)C=Cc2ccccc2F)CC1(C)C 1697,CN1CC=C(CC(=O)NC2CCCCC2NC(=O)Cc2c(O)ncnc2O)CC1 1698,C1(C)(C(N(C(C)CCNC(=O)C(Cc2cccs2)C2CC2)C)=O)COCCO1 1699,c1(C(N2CCC(NC(C3C(C(=O)OC)C3)=O)(CF)C2)=O)ccn2nncc2c1 1700,C1(CCC)(NC(C=NOC)=O)CCCN(C(=O)C(c2ccnn2C)C)C1 1701,CC1(C)CCC(CO)N(C(c2conc2CNC(=O)C=CC(F)F)=O)C1 1702,CC1CN(C(=O)Cc2cccnc2Cl)CC1NC(=O)C(O)C1CC1 1703,C1(N(C(=O)CC2CC2(Cl)Cl)CC)CCN(C(=O)Cc2cncnc2O)CC1 1704,CC(C)(C)C(O)C(=O)NC1CCCN(C(=O)CC2CCOC2=O)CC1 1705,c1(C(N2CCC(NC(c3cn[nH]c3)=O)C(O)C2)=O)nccn2nccc12 1706,N1(C(C(C)Nc2ccccc2)=O)CC2CCCN(C(c3cnsc3)=O)C2C1 1707,c1(NC(C(N2CCN(Cc3ccccc3)CCC2C)C)=O)sc2c(c1CO)CCOC2 1708,c1(C(=O)NC2(CO)CCN(C(C3CCC(=O)N3)=O)C2)cncc2ccsc12 1709,n1(C(C(=O)NCC2(C)CCN(C(COC)=O)C2)C)cc2ccccc2n1 1710,C12(C(N3CCC(CCCC)C3)=O)CC(CO1)N(C(=O)CCC(C)=O)C2 1711,Cc1cc(C(N2CCC2C(N2CCC(O)C(C)C2)=O)=O)ccc1F 1712,N1(C(c2sc(C)c(O)n2)=O)CCN(C(=O)CN(C)C(C)C)CC2CCCCC12 1713,N1(C(CCC(=C)Cl)=O)CCCC(CCC)(NC(C2SC3C=CC2CC3)=O)C1 1714,c1(C(=O)NC2CCN(C(CCc3cccc(C)c3)=O)C2C)cc2n(n1)CCC2 1715,c12cc(sc1C)C(=O)N(C(C1CCCCC1)C)C2.C(C)(C)(C)OC(=O)NC1CC1 1716,CCC(O)C(C)C(=O)NCC1CN(C)CCN1C(c1ccc(C(F)F)nc1O)=O 1717,N1(C(CC2CC(OC)C2)=O)CC(CNC(c2ccc(Cl)c(F)c2O)=O)CC12CCC2 1718,CC(C(=O)NC1C=CCN(C(C2CN(C3CCOC3)C2)=O)C1)C(F)(F)F 1719,n1(CC(=O)N(CC(CO)(CO)NC(C2CC(C)(C)CO2)=O)C)cnc([N+](=O)[O-])c1 1720,C(C)(CNC(c1sccc1Cl)=O)(CC)NC(CCC)=O 1721,c1(C(N(C2CN(C(c3c(F)ccc(F)c3N)=O)C2)C)=O)cccn2c(O)nnc12 1722,c1(N(C(=O)CC2CCN(C(=O)Cn3ccnc3)C2)C)nc(C(=O)O)ncc1Br 1723,CCCC(CNC(=O)C=CC(=O)N(C)C)C(=O)NCC1COC(=O)N1 1724,N1(C(C(=O)N(CC)CC2CCC(=O)N2)=O)CCC2C(CCN2C(=O)OC(C)(C)C)C1 1725,c1(CC(=O)NC2C3(CC(NC(C4N(CC)CC4)=O)C3)C2)cccc(F)c1F 1726,N1(c2scc(CC(=O)NC3(C)CC3(F)Cl)n2)C(=O)NC2(CCCC2)C1=O 1727,C1(c2n(C)nnn2)(Nc2ccc3c(c2)CCO3)CC2(CCCCC2)C1 1728,C1(CCO)CC(N=c2[nH]c(=NC3CCC(C4CC4)C3)[nH]c3c2COC3)C1 1729,C(CC(=O)Nc1ccc(CN(C)C)cc1)(C1=CCCC1)NCC 1730,C1(CNC(C(CC#C)O)=O)CCN(C(c2scnc2CC)=O)CC1(F)F 1731,c1(C(=O)NCC(C2CCC2)NC(C(C)SC)=O)cc(C)ccc1Cl 1732,CC(C)CC(CNC(C1CCCN1C=O)=O)NC(=O)C(C)(C)COCC(F)F 1733,c1(OC(C(OCC)OC)=O)cc(C(N)=O)cc(C)c1 1734,CN1CC(C(=O)NCC2CCC(NC(=O)CCCc3ccccn3)C2)CCC1=O 1735,c1(C(N(CC(C)N(C(C(C)OCCC=C)=O)C)C)=O)ccc(Cl)cc1O 1736,C1(C(=O)NC(c2cccnc2)C(=O)N(CCCC)C)CCN(CC)CC1 1737,c1(CC(N2C(CNC(C3(C=C)CCC3)=O)CC2)=O)ccc2c(c1)COC2 1738,C1(CC(=O)NCC(=C2CN(C(c3c(N)nc(Cl)cc3)=O)C2)F)Cc2ccccc2O1 1739,n1(CC(=O)N(C2CCCN(C(c3c(C)onc3Cl)=O)C2)C)ccc2ccccc12 1740,c1(C(=O)NCC2N(C)CCN(C(c3coc(Br)c3)=O)C2)cccn2cncc12 1741,c1(C(N2C(CNC(C(CC(=C)C)C)=O)CCC2)=O)ccc2nsnc2c1 1742,C1(C)(NC(C(C2CCCCCC2)C)=O)CCN(C(c2ncc[nH]2)=O)C1 1743,CCC(C)(C)C(=O)C(=O)N1CCC(C2CCCN2C(c2ccc(Cl)s2)=O)C1 1744,c1(C(=O)NC2CN(C(CN(C)C)=O)C2)cc(=O)cc[nH]1 1745,C(=O)(C1=CC2(CCOC2)C1)N1CCC(CC(C)NC(CC(CC)CC)=O)CC1 1746,c1(C(=O)NCCOCCN(C)Cc2c(OC)ccnc2)ccc2occ(C)c2c1 1747,C1(C2CCCN(C(C3C(C)(C)C3(F)F)=O)C2)(NC(C=C(CCC)C)=O)CC1 1748,c1(OC)ncnc(C(=O)NC(C)CNC(c2cnn(CC3CCC3)c2)=O)c1F 1749,c1(C(=O)NC(C(=O)NC(CC#C)CCOC)CCC)cccc(C#N)c1C 1750,c1(CC=O)c(F)cccc1F.C1(C(N)=O)CN(Cc2nccs2)C1 1751,c1(CNC2C(C(=O)NC(c3cncs3)C)CCC2)c2c(nn1C)CCC2 1752,c1(CNC(C(CC)Br)=O)cc(C)cnc1-c1ccccc1 1753,C1(O)(CC)CCCN(C(=O)C=CCNC(=O)CCn2nc(C)nc2C)C1 1754,Cc1nc2cc(C(=O)N(CC(O)CNC(=O)CC3=NNC(=O)C3)C)cc(O)c2o1 1755,CC(C)CCC(F)C(=O)N1CCCC(C)(C)C1C(=O)NC1C(O)CC1O 1756,C1(S(C)(=O)=O)(NC(=O)NC2(CC(C)C)CC2)CC(F)(F)C1 1757,C(=O)(C(C)CCCOC)NCCCC(C)(C)NC(c1c(CCC)nns1)=O 1758,C#CCCCC(C)C(=O)NCC(C)CNC(c1cc(C(N)=O)[nH]n1)=O 1759,C(C(CC(=O)N(C1(C(O)CO)CC1)C)NC(=O)CCC(C)SC)OC 1760,C(=O)(C1CCOc2ccc(F)cc21)N1CC(CNC(C(Br)=C(C)C)=O)C1 1761,N1(C(C2CC(C)(C)OCC2)=O)CCCCC(NC(C2(CC3CCC3)CC2)=O)CC1 1762,Cc1[nH]c(C#N)cc1C(=O)NCC(O)CNC(C1CC(C)(C)CN1C)=O 1763,CP(C)(=O)CCC(=O)NC1CCN(C(=O)CCCc2csc(=N)[nH]2)C1 1764,Cn1ccc2c(C(=O)NCC3CN(C(=O)C=C4CC4)C3)ccnc12 1765,c1(CC(N2CC(CNC(CCOCC)=O)(COC)C2)=O)ccccc1Br 1766,c1(CC(=O)NC(CNC(c2n(CC#C)ccc2)=O)C2CCC2)cnc(Cl)cc1C 1767,S1(=O)(=O)c2cccc(c2)NC(=O)CN1C.c1(SC)nc(=O)o[nH]1.CC(C)OCC 1768,Cc1cnn(C)c1C(C)(C)NC(C1CCN(C(=O)CCS(C)=O)C1)=O 1769,n1(CC)ncc(C(=O)NCC=CCNC(=O)CC(C)(C)O)c1C(F)(F)F 1770,C12(NC(CC3CCC(C)CO3)=O)CC(CNC(c3cncn3C)=O)(C1)OC2C 1771,C1(C(=O)Nc2c(CC)ncs2)CC12CCN(C(c1ccc(C3CC3)cc1)=O)C2 1772,CS(=O)CCC(O)C(=O)NC1(C)CN(C(=O)Cc2csc(-c3ncccn3)n2)C1 1773,C1(C(=O)NC2CCOC2=O)CCCC2CN(C(=O)C3Cc4ccccc43)CC12 1774,N1(Cc2onc(CC(C)C)n2)CCOC(C)(CNC(C2C3CCC(F)(F)C23)=O)C1 1775,N1(C(c2c(C(C)C)c[nH]n2)=O)CCCC(N(C(=O)CSCC2CCCCO2)C)C1 1776,c1(C(=O)NC(C2CCN(C(c3c(CC)onc3C)=O)C2)C)c(Cl)cncc1Cl 1777,Cc1noc(C)c1C=CC(=O)NC1CC2CC1N(C(c1coc(C(N)=O)c1)=O)C2 1778,c1(CC(=O)NC2CCN(C(C=CC(CC)C)=O)CC2CO)cn2ccccc2n1 1779,c1(OC)ccc(Cl)cc1C(=O)NC(C)CNC(=O)Cc1cccc(F)c1O 1780,CC(CC(F)(F)F)C(=O)NC(CC1CC1)C(=O)N1CC(N2CCC2)C1 1781,c1(OC)c(NC(C2CSCCN2Cc2ncc(C)s2)=O)ccc(Cl)c1Cl 1782,C1(COC)(CNC(=O)CSCCN(C)C)CCCN1C(=O)C(C)(F)F 1783,c1(C(C(=O)NC2(CN(C(COC(CC)C)=O)C)CC2)C)cccc(N(C)C)c1 1784,C1(CNC(=O)CC(CC2CC2)NC(c2ncc(CO)[nH]2)=O)CC2C=CC1CC2 1785,c1(-n2cc(C(C)NC3CN(Cc4ccccc4)C3)nn2)ccc(I)nc1 1786,N1(C(CCC=C=C)=O)CC2CCNCC2C1.C1(C(N2CCNCC2)=O)CCN(CC(C)C)C1 1787,CCCCC(C(=O)N1CCN(C(C2CC3C(C2)C3(F)F)=O)CC1)NC(N)=O 1788,c1(C(N2CC(C)N(C(c3cnc(O)[nH]3)=O)CC2)=O)ccc2c(Cl)cccc2c1 1789,C(=O)(C(=O)NNC(=O)CCc1cccc(C#N)c1)NC(c1ccc(C(F)(F)F)cc1)C 1790,C(=O)(C1SCCc2sccc21)N1C(C(C)NC(c2cc(C)ncc2)=O)CCC1 1791,c1(C(=O)NCC2CC(NC(c3c(CC)onc3C)=O)C2)cc(NC2CC2)nc(C)c1 1792,N1(C(C(C)C)=O)CCCCC1C(=O)Nc1nnc(C(F)(F)F)s1 1793,N1(C(c2c(OC)csc2)=O)CC(CNC(c2cnn[nH]2)=O)OC(C(F)(F)F)C1 1794,C(C1CN(C(C2COCC2C(N)=O)=O)CC1N(C=O)C1CC1)=CC.C1CC=CCC1 1795,c1(C(N2CCN(C(C(C)C(F)(F)F)=O)CC2)=O)cnc2cccc(F)n12 1796,CC(O)C(C)(C)C(=O)NCCCOCCNC(=O)C=CCO 1797,C=CCCC(c1nnnn1C1(C)CC1)(C1CC1)NC(C)CCC(C)C 1798,c1(C(=O)NC2C(NC(c3c(C)ccc(OC)c3)=O)C2)cccc2oc(C)cc12 1799,c1(C(=O)NCC(CN(C(=O)CC2(O)CC2)C)O)n[nH]cc1-c1ccccc1 1800,c1(CN2CCC3CN(Cc4ccc(C(N)=O)cc4)CC32)n[nH]c2cc(Br)ccc12 1801,N1(C(COCCCCC)=O)CCC(CNC(=O)C=CI)C(C)C1 1802,C1(NC(C(C)(C)c2ncco2)=O)CC2CC(NC(c3ccc(F)s3)=O)CC2C1 1803,C1(C(=O)NCC2(CC(=O)NC(C)C(C)(C)C#N)CC2)CC2CC(=O)C1O2 1804,c1(NCC2C(C)CN(C(C3CC(C)(C)C3)=O)C2)ncnc2c1nnn2CCO 1805,C1(C(N2CC(CCCCNC(CN(CCC)C)=O)C2)=O)CC2(C1)CC2C(=O)OC 1806,c1(CC)ccc(C=CC(N2CCCC2CN(C(=O)Cc2ncc(C)o2)C)=O)cc1 1807,N1(C(c2cc(OC)n[nH]2)=O)CCC(C)(CNC(C2CCC(=O)CC2C)=O)CC1 1808,C(=O)(C(C(C)C)NC(=O)OC)NC1CC(C(N2C(CCC)CCC2)=O)C1 1809,C1(OC)CC(C(=O)NC(CNC(c2cn(C(C)C)cn2)=O)C2CC2)CC1OC 1810,Cc1cc(N2CCC(N(C)C(C3C(F)(F)C34CCC4)=O)C2)n2nc(C)nc2n1 1811,C(=O)(C(CNC(c1ccc(C#N)o1)=O)C(C)(C)C)N1CCC(C(=O)NC)C1 1812,C(=O)(C1=CC2CCC=CCCC12)N1CCC(CNC(CNC(N)=O)=O)C1 1813,C1(C(N(C(C(=O)N(CCOC)C)C)C(C)C)=O)COCCN1CC 1814,c1(C(=O)NCC(C)(C)NC(Cc2c(C)noc2)=O)cnc2c(c1)nnn2C 1815,C1(CNC(C(CC)C)=O)COC(C)(C)CN1C(c1cnc(SC)nc1O)=O 1816,C12(NC(Cc3cc(C)no3)=O)CCCCCC1N(C(C1CC(=O)C1)=O)CC2 1817,c1(CNC(C2(NC(c3cc(OC)n[nH]3)=O)CC2)=O)c(CO)cccc1C 1818,CC1CCCCN1C(=O)CCC1CCC1.c1(-c2nc(N3CC3)sc2)ccc(F)cc1 1819,c1(C(N2CC(OC)C(NC(c3c(C)coc3C)=O)C2)=O)ccc(O)c(N)n1 1820,C(C(C)CC(=O)NC(CNC(=O)COC(C)(C)C(F)(F)F)C1CC1)SC 1821,C1(NC(Cc2nc(C)c(C)s2)=O)CC2CC(NC(=O)CC3OCCC3(C)C)CC12 1822,C=CC(CCC)CC(=O)N(CC(=O)NC(CO)C(C)(C)CO)C 1823,C(CC(O)CNC(=O)C(Cn1ccnn1)NC(=O)CC1(O)CCOC1)OC 1824,Cc1ccc(CC(=O)NC2CCC(CO)N(C(=O)CC3CC=CC3)C2)c(F)c1 1825,CC(CC(=O)N(C1CCCN(C(=O)CNC(c2cnc(O)nc2O)=O)C1)C)C(F)F 1826,c1(C(N2CC(CC)C2)=O)cc2scc(Br)c2s1 1827,c1(CC=C)cn(CCC(N2CC(C)(OCC(=O)NC3CCCCS3)C2)=O)nn1 1828,c1(OCC(=O)NC(CNC(C2(CC#C)CCCC2)=O)(C)CO)ccc(F)cn1 1829,c1(C(N2CC(O)(C(C)NC(=O)C=Cc3cncs3)C2)=O)cccc([N+](=O)[O-])c1O 1830,N1(C(CCc2n(C)cnn2)=O)CC2CC2(NC(=O)CCC2CCCOC2)C1 1831,c1(CC(N2C(CNC(C(C)C3CCCC3)=O)CCC2)=O)cc(O)ccc1Br 1832,C1(OC)CN(C(C2(CSC)CC2)=O)CCC1NC(=O)C(O)CCSC 1833,c1(N(CC(C)(C)C)CCO)ccccc1.C(CC=O)OCCO 1834,Cc1nc(C(N2CC3(NC(c4cnoc4C)=O)CC2C3)=O)ccc1C#N 1835,CC1CCCCCN1S(=O)(=O)CC1CC1c1ccccc1-c1ccc(Cl)c(F)c1 1836,C1(C(N2C3(CN(C(C(CCC)CC)=O)C3)CC2)=O)Cc2ccccc2C(C)(C)C1 1837,Cc1cc(C(N2CCC(C(=O)NCC3CCCC3O)(CF)C2)=O)ncc1N 1838,C1(CNC(C(COC)NC(C2CC(CCC)C2)=O)=O)CCC2CC1CO2 1839,Cc1cc(C)c(C(N2CC(C)CC2C(=O)Nc2ccc(C#N)c(Br)c2)=O)cc1C 1840,c1(C(=O)OCC)cc(Cn2cc(-c3ccn(C)n3)nn2)cs1 1841,Cc1cc(S(=O)(=O)NC(C)CCCCCO)c(C)cc1-c1ccnn1C 1842,CC1(CNC(=O)CCc2ncccn2)CCN(C(C2CC(n3ccnc3)C2)=O)C1 1843,C(=O)(CC1C(=O)Nc2ccccc21)NC(C)C(CO)NC(=O)Cc1csc(Cl)n1 1844,C(=O)(CC(F)(F)CS(C)(=O)=O)N1C(CO)CC(NC(C(CC#C)(C)CC)=O)C1 1845,N1(C(C=CCC)=O)CCC(C2CCCCN2C(=O)C(O)Cc2ccccc2)CC1 1846,C12(C(=O)NCC3CCC(NC(c4ccc(Cl)nn4)=O)C3)C=CC(CC1)C2 1847,C(C)(CC(=O)NCC(C1CC1)NC(=O)CC#N)(C(F)(F)F)N(C)C 1848,n1(CC=C)nc(-c2ccoc2C)nc1CCCc1ccc(N)cc1 1849,c1(CN2CC(CC(=O)OC)C2)cc(C(N2CCCC2CC)=O)ccn1 1850,c1(C(N2CC(C)C(N(C)C(C34CC(F)(C3)C4)=O)CC2)=O)ccnc2cc[nH]c12 1851,Cn1cc(CNC(C2CC=CCN2C(=O)C(O)CC2CCCC2)=O)ccc1=O 1852,Cc1cnsc1C(=O)NCC(C)C(=O)NC1CC(CO)C1 1853,CCC(CCCC(=O)N(C)CC1CC(F)(F)C1)NC(=O)Cc1nocc1CC 1854,c1(CC)nnc(CN(C(=O)C=CCNC(=O)Cc2ccc[nH]2)C)o1 1855,CCCC(C)CC(=O)NC1CCCC(CNC(c2c(C)nc(C)n2O)=O)C1 1856,CC1CC(c2nnnn2-c2ccccc2F)(NCCCO)CN1C 1857,c1(C(=O)NC23C(CN(C(C(C)(C(C)C)OC)=O)C2)C3)c(C)nc(C(C)C)nc1O 1858,c1(C(N2CCC(C)(NC(COC)=O)CC2)=O)nccc2cnn(C)c12 1859,c1(C(=O)NC23C(CN(C(C4CC(=O)N(O)C4)=O)C2)CC3)sc2sccc2c1Cl 1860,C1(N(C(=O)CCSc2ccncc2)CC)CCCN(C(=O)CSCC2CCCO2)C1 1861,c1(CC)ccc(C(=O)NC(COC)C(=O)NCC(=O)NCC(F)F)o1 1862,c1(C(N2CCN(CC(F)(F)CO)CC2)=O)ccc2ncsc2c1 1863,Cc1ccc(=O)n(CC(=O)NC2(C)CCN(CCC3CC4CC4C3)CC2)n1 1864,C1(NC(c2c(OC)cccn2)=O)CCCC12CN(C(=O)CC(C)(C)F)C2 1865,O=C(C1=CCCN(C(=O)C(O)Cn2cncn2)C1)NC(C(O)CO)C1CC1 1866,C12(NC(c3ccc(COC)o3)=O)CC1CN(C(C1CCC=CCC1)=O)C2 1867,n1(CC(=O)NCCN(C(C2(OCC)CCCCC2)=O)C)c(C)cc(O)cc1=O 1868,c1(C(C(=O)NC(CC)CNC(=O)C=CSc2ccccc2)C)ccc(O)cc1 1869,CC1CCN(C(c2cc(C(C)(C)C)no2)=O)CCN1C(C1CC1C(C)O)=O 1870,CN1CC(C(=O)NC(C)(C)CCNC(=O)COCC2CCCO2)NC1=O 1871,c1(C(=O)NC(C(=O)NC(CCC)C)Cc2ccccc2)noc2c1CCCCC2 1872,N1(C(C23CCCCC2C3)=O)CC2(CCC(CNC(C(=O)Nc3ccccc3)=O)O2)C1 1873,C1(N(C(C2CC(C)(O)C2)=O)C)CCN(C(=O)C(F)(F)CO)CC12CC2 1874,N1(C(c2c(CC)nc[nH]2)=O)CCCC(O)(CCNC(c2cnc(C3CC3)[nH]2)=O)C1 1875,c1(C2CN(C(=O)NC(CCOC)CN)C2)ccc(Cl)cc1 1876,N1(C(C2CCN(CC#C)CC2)=O)CCC(C(F)(F)F)C(NC(=O)C(C)C#N)C1 1877,C(=O)(C(C)(C)C(C)C)NCC(=O)NCC(N1CCN(C(CCCC)=O)CC1)C 1878,C(=O)(CC(C(F)(F)F)c1ccccc1)NCC(CC)NC(c1ccc(C#C)o1)=O 1879,CC1CCc2cc(C(N3CCOCC3CCNC(c3ccsn3)=O)=O)ccc2N1 1880,C(CN(C(=O)C(c1cccs1)NC(=O)CCn1cncn1)C)(C(C)C)OC 1881,c1(NC(C(C)c2ccsc2)=O)cccc(C(=O)NCC2COC(CC3CC3)C2)n1 1882,CC(C)(C)C(=O)NCC1CCC1NC(C1CCCN1C(=O)Cc1ncc(Cl)s1)=O 1883,Cc1sc(-c2nc[nH]n2)nc1C(=O)NCCCNC(C1CCCC(C)C1)=O 1884,C1(C(N2CCC(Cn3cc(CCN(C)C)nn3)CC2)=O)CC1C1CCCC1 1885,CC1CCC(NC(c2cc(C#N)c[nH]2)=O)CN1C(=O)CCN1CCOCC1 1886,c1(C(N2CCN(C(c3ccc(C)cc3)=O)C3C2C3)=O)ccnc2ccnn12 1887,c1(C(C)(C)C)ccc(CC(=O)NCC2CC2CNC(C2CC=CC2)=O)cc1 1888,c1(OC)ccc(C(N2CC(CCNC(=O)CSC(C)C)(OC)C2)=O)c(N)c1Br 1889,C1(NC(c2cccc(OC)c2)=O)CCN(C(c2cn(C)nc2SC)=O)C1(C)C 1890,CCCC(O)CC(=O)N1CCC(C(C)(C)C)(CNC(=O)CCS(C)(=O)=O)C1 1891,CC(C)S(=O)(=O)CC(=O)N1CCC(=CCNC(=O)CC2CC3OC2C2CC32)CC1 1892,CCC(C)(COC)CNC(C1CCN(C(=O)CCCCN(C)C)C1C)=O 1893,N1(C(C=Cc2ccc(C)o2)=O)CCCC(NC(C2(N(C)C)CCC2)=O)C1C 1894,N1(C(C(CC#C)O)=O)CCC(C(=O)NCC2(OC)CCC2)CC1(C)C 1895,N1(C(=O)Cc2cc(Cl)cc(Cl)c2O)CCC2CCN(C(C3C4COCC34)=O)CC12 1896,C1(C)(C(=O)NCC(CNC(c2c(C)n(C(C)(C)C)nc2)=O)(C)C)COC(C)CO1 1897,CC1(C)CC(NC(C2COCCN2C=O)=O)CN1C(c1cc(C(F)(F)F)no1)=O 1898,C(C)(C(=O)NCC(C)(C)CNC(=O)CC(C)c1ccncc1)(C(C)C)NC(C)=O 1899,C(=O)(CC(C)(O)COC)NC(CC)CNC(c1ncccc1Cc1ccccc1)=O 1900,n1(CC)cnc2c(NC(C)(COC)CCO)[nH]c(=NCCCCCN(C)C)nc12 1901,Cc1noc2ncc(C(N3CCC(NC(C4CS(=O)(=O)C4)=O)C(F)C3)=O)cc12 1902,n1(CC(=O)NC2C(NC(C(CCC)OCC)=O)C2)cc(C)c2ccccc12 1903,Cc1ccc(C)c(C(=O)NCC(CC(C)C)NC(c2cccnc2)=O)c1O 1904,C1(C(=O)N)CCC2(CCN(C(=O)CN(c3cnccn3)C)CC2)C1.CC(C)C(O)CO 1905,c1(OC)c(Cl)cc(C(=O)NC(C)CCCNC(c2c(C)nn(C)c2C)=O)nc1Cl 1906,C(CN=c1nc(Cl)[nH]c(C)c1C#N)C1CCCCCN(C(C(C)SCC)=O)C1 1907,C1(C(=O)NCCCC2CCC2)(CNC(C(C)n2cccc2)=O)CCCCC1 1908,N1(C(C(CCC)CC)=O)CC(NC(c2cc3c([nH]2)CCCC3)=O)CCC(O)C1 1909,c1(C(=O)NCCCN(C)C(C2CCCS2)=O)cc(S(=O)(=O)N2CCOCC2)c[nH]1 1910,C1(NC(c2c(C(N)=O)csc2)=O)CS(=O)(=O)C2CN(C(c3cnns3)=O)CC12 1911,c1(C(=O)NC2CC(CCNC(CC3(OC)CCC3)=O)C2)cncnc1C 1912,c1(CC)cnoc1C(=O)NC1CC(C)(NC(=O)C(C)C2CCCO2)C1 1913,N(C(=NCc1ccc(-c2csc(C)n2)cc1)NC(C)C1CC1)C(C=C)C 1914,CC(C)(CNC(c1sccc1F)c1nnnn1CCC1CC1)CC(F)F 1915,N1(C(C(=O)N(CC(C)N(C)COC2CCCOC2)C)=O)CC(C(F)(F)F)C2(CC2)C1 1916,C(CCC(C)(C)N(C(C1CC1C(C)(C)O)=O)CC)NC(COCCOCC)=O 1917,CC1OC(=O)NC1C(N1CCC1CC(=O)NCC(C)(C)C1CC1)=O 1918,CCC(CC)(CO)C(=O)NC(C1CCN(C(C2(n3cc(Cl)cn3)CC2)=O)C1)C 1919,Cc1cnc2c(C(N3CCN(C(=O)CN4CCC(CO)CC4)CC3)=O)cccn12 1920,C1(C)(C(c2n(CCCSCC)nnn2)NCc2cscc2F)CC2(C1)CC2(F)F 1921,N1(C(C2CCCN(C(C(C(=O)OC)C)=O)C2CC)=O)CCC(O)C(F)(F)C1 1922,C1(C)(CC)CC(NC(=O)CCN(C(C2CC(C)(C)C2)=O)CC2CC2)CCO1 1923,c1(C(N(CC(C)NC(=O)CCC2CCCC2)C)=O)ccc(N)c(Cl)c1 1924,c1(C(=O)NC2CCN(C(c3c(CCC)n(C)nc3)=O)C2C)cc(Cl)ccc1OC 1925,c1(OC)ccccc1C(C)C(=O)N(C1CN(C(c2c(Cl)nsc2Cl)=O)C1)C 1926,c1(C(=O)NCCOC2CN(C(c3c(C)oc(Cl)n3)=O)C2)ccc2c(c1)CC(=O)N2 1927,c1(CC(CC)N(C(C2CCCC23CC3)=O)CC)ccc(F)cc1 1928,c1(C(N(CC(N2CCC(SC(F)F)C2)=O)C)=O)ccc(O)cn1 1929,c1(OC)nc(C)cc2ccc(C(=O)NC(C)CN(C)C(C3C=CCCC3)=O)cc12 1930,c1(C(=O)NC2CC(NC(C=CC3(C)COC3)=O)CC2O)cc2cnccc2o1 1931,C1(CC(C)NC(=O)CN(S(C)(=O)=O)C)CCN(C(=O)C(F)(F)CO)CC1 1932,C1(CNC(C(CSC)O)=O)CN(C(c2ccc3nccn3c2)=O)CCC12CCC2 1933,Cc1scc(-c2cc(CNC3CC(c4ccc(F)cc4)(C)C3)n[nH]2)c1C 1934,CC1CCC=C1C(=O)N1CCC(C(N2CCC(F)CC2)=O)C12CC2 1935,Cc1cc(F)c(C(=O)NC2CCCCC2CNC(c2ncccn2)=O)c(Br)c1 1936,c1(C(=O)NC2CCN(C(CN(C)C)=O)CC2CO)c(F)ccc2occc12 1937,C12(NC(CC(CN(C)C)O)=O)CCCC1(F)CN(C(C1CCCCCC1)=O)C2 1938,C1(n2c(N3CCC4C(F)(F)C4C3)nnn2)C2Cc3cc(Br)ccc3C12 1939,c1(OC)ccnc(O)c1C(=O)N(CC(C)N(C)C(c1cc(C(F)F)[nH]n1)=O)C 1940,CC(C)(CCCCNC(=O)C(O)C1CC1)NC(c1cc(Cl)n[nH]1)=O 1941,C(=O)(C1CCCn2ccnc21)OC.C1(=O)C(C)(C)OCCCN1C(C)C 1942,c1(NCC(CN(C)C)O)ccc(S(=O)(=O)NCc2ccnc(SC)c2)c(Cl)c1 1943,C1(C(=O)NCc2c(C)n[nH]c2)N(C(C2CN3CCC2C3)=O)CCCC1(C)C 1944,c1(C(N2C(C)(CNC(=O)C(F)CC3CC3)CCC2)=O)cccc2c1NCCC2 1945,c1(C(N(CCCNC(C=C(C)C)=O)C(C)C)=O)nncn1C1CC1 1946,C1(OC)(CNC(=O)CC(C)N(C)C)CCN(C(C2CC3(CCO2)CC3)=O)CC1 1947,C1(CCNC(=O)C(O)C2CC2)CCCCN1C(C1CCC(O)CC1)=O 1948,c1(C(N(C)Cc2cc(OC)no2)=O)cc2ccncc2c(O)n1 1949,S(=O)(=O)(c1ccc(NCc2ccns2)cc1Cl)NC(c1ccn(C2CC2)n1)C 1950,C1(C(N2CC=C(C)C2)=O)CCN(C(=O)C(CN=[N+]=[N-])N(C)C)CC1(C)C 1951,c1(OCC=C)ccc(CC(=O)NC2CC(C)(NC(C3CCCC3(F)F)=O)C2)cc1 1952,N1(C(C(C)OCC#C)=O)CCC(C2(NC(c3nc(O)sc3C)=O)CC2)C1 1953,C1(C(N2CCC(Cc3cn(CC(CC)O)nn3)CC2)=O)CCc2ccccc2C1 1954,C1(N(N2CC3CN(S(=O)(=O)CCCCl)CC3C2)C)CCc2nn(C)cc2C1 1955,C(=O)(C(C)(CC)CO)NCC(N1CCN(C(C=CC=CCC)=O)CC1)C 1956,C(CCN=C(NCC(=O)N(C)C)NC1CCC2CC12F)N1CCN(C)CC1 1957,N1(C(C2(OC)CCCC(C)C2)=O)CC2CCCC1C2CNC(c1cc(C)co1)=O 1958,CC1(C)CN(C(c2cccnc2)=O)CC(CNC(=O)Cc2ccc(F)cc2Cl)O1 1959,Cc1cnc(NCC2CCS(=O)(=O)C2)c(S(=O)(=O)NCCCCCF)c1 1960,C1(CNC(C(CN(C)C)(C)C)=O)CCN(C(=O)CN2CCC(C)(O)C2)C12CC2 1961,N1(C(C(C)N(OCC)CC)=O)CCN(C(c2sccc2CO)=O)CC1.C1C(C)S1 1962,c1(C(=O)NCC2CCN(C(C3CN(CCC)C(=O)C3)=O)CC2)cc(C#N)[nH]c1C 1963,C(CC(=O)N1CC2(CCCCC2)C1)(C(F)(F)F)NC(C1CCCCC1)=O 1964,c1(NC(N2C(C)CN(Cc3ccc(Cl)c(Cl)c3)CC2)=O)cn2cccnc2n1 1965,C=C(C)CCCC(=O)NC(C)Cn1cc(CN(C(C)C)C(C)C)nn1 1966,N1(c2c(C#N)cncc2)CC2CN(C(=O)CCC(CF)CF)CC2C1 1967,C1(NC(c2cc(C)c(Br)o2)=O)CC2CCNCC2C1 1968,C12(C(=O)NCCCOCCCNC(=O)Cc3cnsc3)CCCC(CCC1)C2O 1969,CCCCC(C)(C)C(=O)NCC1CCC1NC(=O)Cc1cnccc1C(F)(F)F 1970,C12(NC(Cc3cccc(OC)c3)=O)CCC(CC1)N(C(c1cccc(F)c1)=O)C2 1971,N1(C(C2C(C=C)C2)=O)CC2CCC1CN2C(=O)CNC(=O)OC 1972,N1(C(C=CC=CCCCCC)=O)CCC(CNC(=O)CCF)C12CC2 1973,C1(C(=O)NC2C(CNC(c3sc(CCC)c(C(=O)OC)c3)=O)C2)C(C2CC2)C1(F)F 1974,N1(C(CC=C)=O)CC(C(=O)NC(c2nccc(=N)[nH]2)C)C(F)(F)C1 1975,C=CCCCCCCC(=O)N1CC(C)C1C(=O)NC1CC(O)CC1O 1976,N1(CC)CCCCC(N(c2ccnc(I)n2)C)C1 1977,C1(C(N2CC(CN(C)C(C3SC4C=CC3CC4)=O)C2)=O)C2(CCC2)C12CCC2 1978,n1(CC(N2CC(OCC#C)C2)=O)cc(CNC(=O)CC2(O)CCC2)nn1 1979,c1(C(=O)NCc2cn(CC3C(N)(C(F)(F)F)C3)nn2)ccc(O)c(Br)c1 1980,C1(NC(CCCC#C)=O)CC2CCC1CN(C(C1CCC(F)CC1)=O)C2 1981,c1(C(=O)NCCC2(O)CCN(C(C34OC(C)C(C3)C4)=O)C2)cccc2occc12 1982,n1(C(C(=O)N(CCCNC(=O)Cc2ccco2)CCC)C)nc(C)cc1C 1983,n1(CCC)ncc(C(N2CC(NC(=O)CCc3cnco3)C3CC23)=O)c1C 1984,c1(C(=O)NCC(C2CCC2)NC(c2csc(Cl)n2)=O)ccc([N+](=O)[O-])cn1 1985,C12(NC(C3CC3[N+](=O)[O-])=O)CCC(C1)N(C(=O)CNc1ccc(C(F)(F)F)cn1)C2 1986,C12(CNC(CC(=O)NCCCCC)=O)CN(C(C3CCC3C)=O)CC1CCO2 1987,N1(C(C(C)N(C(C(CCCC)NC(N)=O)=O)C)=O)CCC2(CCC(O)C2)C1 1988,C1(CC=C)(NC(=O)CNC(C)=O)CCN(C(=O)CCC2CCC(C(N)=O)O2)C1 1989,Cc1ncnc(C)c1CC(=O)NCCCNC(C1CC2(F)CC1C2)=O 1990,c1(CC(=O)NCC2N(C(C(CC=C)C)=O)CC2)ccc(Cl)nc1F 1991,Nc1cc(C(=O)NC2CCCCC2NC(=O)CCc2ncccn2)cc(Br)n1 1992,C1(CCC(=O)N(n2cncn2)CC=CC)CCN(C(=O)CN2CCC(C)C2)C1 1993,C1(CC(=O)NCC2CC2NC(=O)Cn2cc(-c3ccncc3)nn2)CC2COCC12 1994,N1(C(C2C3(CCN(C(CC4(N(C)C)CCC4)=O)C3)C2)=O)CCC(C2(C)CC2)CC1 1995,c1(C(=O)NCC2CCN2C(C2COC3(CCC3)CO2)=O)cc2c(Cl)cccc2s1 1996,N1(C(c2nccc(C)c2)=O)CC(CNC(C2CC3(C2)CC(O)C3)=O)OC(C)(C)C1 1997,C1(NC(C(CC)OC)=O)CCCCC12CCN(C(=O)C(O)C(C)CC)C2 1998,c1(OCC(C)C)ccccc1C(=O)NC(CNC(=O)Cc1ccsc1Cl)C(C)C 1999,CCC(CC)(C(=O)N(C)CCSC1(C(=O)NC2CC(OC(F)F)C2)CC1)OC.NC 2000,C1(NC(C=CC=CCC)=O)CCOCC1NC(c1nccnc1OC)=O 2001,C(=O)(CCC(C)(C)NC(c1ccc(F)cc1)=O)NC(C#C)CC 2002,C(=O)(C(O)C1=CCCCC1)N(CC(=O)NC(CCC(C)C)C)C 2003,N1(C(c2cccc(C)c2)=O)CC(NC(=O)CSc2nc[nH]n2)C(C#N)C1 2004,c1(CC)cccc2c1CN(C(=O)C(=O)Nc1ccc(Cl)cc1)CC2 2005,c1(N(C2CCN(C(C3C(C)C3)=O)C2)C)ncc(Cl)cc1[N+](=O)[O-] 2006,CCCC(O)CC(=O)NC(C)(C)C(C)NC(=O)Nc1cc(N2CCCC2)ncn1 2007,Cc1cccn(CC(=O)N(CCNC(C23CCCC2CC3)=O)C(C)C)c1=O 2008,C(=O)(C(C)C(CC)CC)N1CC(CC(=O)NCC(NOCCSC)=O)C2(C1)CC2 2009,c1(C(=O)NCC(C)NC(c2cccn2C)=O)ccc(-c2ccco2)o1 2010,c1(NC(C2(NC(CC(O)CC3CCCC3)=O)CCSC2)=O)cccc(F)c1 2011,C=C=C(C)CC(=O)NC(C(=O)NCCC1CC2C=CC1C2)c1cccs1 2012,CC(CCC(=O)NC1CC(CC(N)=O)C1)NC(c1cnn[nH]1)=O 2013,C1(C(N2CCC(NC(c3c(C)ocn3)=O)C(O)C2)=O)CCc2ccc(F)cc2C1 2014,c1(C(C(=O)NCC(c2ccccc2)NC(C(CC)NC(C)=O)=O)O)ccccc1Cl 2015,Cn1cc(COC(=O)CC2COC(C)(C)C2)c(CCC(F)(F)F)n1 2016,C1(NC(c2n(CC)cc(Br)n2)=O)(CC)CCN(C(C2CC23CC3)=O)CC1 2017,C1(C(=O)NC(c2nccc(O)n2)C)C=CCN(C(=O)Cn2ccnc2)C1 2018,C=CCCC(F)(F)C(=O)NC1CN(C(c2cc3ccccc3s2)=O)C1 2019,Cc1nc2cc(C(=O)NC(C)CCNC(C3CC(C)CC(=O)N3)=O)[nH]c2s1 2020,C(C(C)C(=O)NCCC(C)NC(C1CCC(=O)C1)=O)OC(C)=O 2021,C1(C(=O)NC(C)CNC(=O)Cn2cnnc2)CCCCC12CCC2 2022,N1(C(c2c(C)noc2N)=O)CCCC(C)(C(=O)NC2CC(C(C)(C)C)C2)C1 2023,C1(CNC(c2nocc2Cl)=O)CCN(C(=O)CCn2cc([N+](=O)[O-])cn2)C12CC2 2024,c1(C(=O)NCC(CNC(C2(COC)CCC2)=O)(C)O)cnn(C)c1Cl 2025,C1(NC(C(C(COC)C)C)=O)CCCC12CCN(C(=O)Cn1nnc(=O)[nH]1)CC2 2026,C1(NCCO)CCC2(CCC2)O1.C1(CCC)COCCN1C(=O)C 2027,c1(CC)ccc(C(=O)NCC=CCN(C(C2CCCO2)=O)C2CC2)cc1Br 2028,C1(NC(C(C)OCC#C)=O)CCN(C(=O)CC2C=CCCC2)CC1OC 2029,C1(C(=O)NCC2CCCC(CNC(=O)CCF)C2)CN2CCCC1C2 2030,c1(NC2CCC(C)CC2)ccc(S(=O)(=O)N(C2C(C)N(C)CC2)C)cn1 2031,C1(C(N(CCC(=O)NCC2CCCS2)CCO)=O)C=CCCC1 2032,c1(CNC(C(=Cc2cnc[nH]2)C)=O)cnn2c1CN(C(=O)C(=O)C(F)(F)F)CC2 2033,c1(NC(=O)Nc2c(C)n(-c3ccccc3Cl)nc2)c(Cl)cc(C(N)=O)cc1Cl 2034,O=S(=O)(c1cccc(=NCCc2cnn[nH]2)[nH]1)NC1(C(F)F)CCNC1 2035,N1(C(C2N(C)CC(C)(C)C2)=O)CCC(NC(=O)C2=CC(C)(C)C2)C(F)(F)CC1 2036,N1(C(C(C)(C)c2cscn2)=O)CCC2(CCC2NC(=O)C=Cc2ccsc2)CC1 2037,c1(C(=O)NCC2CCC(NC(CCCC(C)O)=O)C2)ccc(Cl)c2occc12 2038,N1(C(CC(C)(C)O)=O)CCN(C(=O)C=Cc2ccccn2)CC1C1CCCC1 2039,C1(CC)CCC(C(=O)OCCC(=O)NCC(C)C)CC1.c1(N)ccccc1SC 2040,CCCC(C)CC(=O)N(C1CCCN(C(c2sc(N(C)C)nc2C)=O)C1)CCF 2041,C1(CNC(C2CCCC(=O)N2)=O)CCCCN(C(c2cc3c(s2)CCC3)=O)C1 2042,c1(CC(=O)NCCNC(c2c(Cl)csc2Cl)=O)ccc2cccnc2c1 2043,c1(C(=O)NC2C(NC(CC(CC)C)=O)COC2)cnc2c(Br)cccc2c1 2044,C1(OCC)CCCN(C(C(=O)C(c2cccc(C)n2)(F)F)=O)C1 2045,C(CC1=CCCCC1)N(C(C(c1ccccc1)OCCc1c(C)occ1)=O)C 2046,N1(C(CN(C2CCC2)C)=O)CCCC2CN(C(C3(F)CC4(CCC4)C3)=O)CC12 2047,c1(C(=O)NCCCCCNC(c2c[nH]c(=O)cn2)=O)cccc2cnccc12 2048,C=CCC(CN(C(c1ccn(C(C)C)n1)C(=O)NC(C)CC)C)CC(C)C 2049,C(=O)(CS(=O)(=O)C1CC1)NCCOC1CN(C(Cc2c(OC)c(F)ccc2)=O)C1 2050,C1(CC)CCCN(C(c2ccc(OC)cn2)=O)C1C(=O)NCC12CCC(C1)C(=O)N2 2051,c1(CC)c(C(=O)NCC2CN(C(c3csc(COC)n3)=O)CCO2)cccc1F 2052,c1(C(C)C)nnsc1C(N1CC(CCNC(=O)CCc2ncccn2)C1)=O 2053,c1(CC)cc(C(=O)NCCC(C)N(C)C(c2ccc(C#N)o2)=O)ccc1OC 2054,C12(NC(c3cnns3)=O)CCN(C(=O)CCc3cncc(Br)c3)CC1C2 2055,N1(C(c2nn(CC)c(C)c2)=O)CCN(C(=O)C=CCO)CC1CC(C)(C)C 2056,c12c(Cl)ccc-1c2F.N1(CC)CCN(CC2CC2c2cnccc2C)CC1 2057,c1(NC(COC(CCC)=O)=O)cnc(OC)cc1OC.C1(C2CC2)C(=O)N1C 2058,N1(C(C(CC)N2CCCC2=O)=O)CCN(C(=O)CC2CN(C)C2)CC1COC 2059,C=CCC(CC)C(=O)NCC1CN(C(C2CC(N(C)C)C2)=O)CCN1C 2060,c1(C(N(C2CCN(C(C3CN4CCC3C4)=O)C2)CCO)=O)cn2ccccc2n1 2061,C1(C(=O)NCC2(C)CCN(C(=O)CNS(=O)(=O)C3CC3)C2)CC2CC1CC2O 2062,CS(=O)(=O)c1ccccc1C1=CCN(CC(C)(C)C)C1.C1(C2CC2)COC(=O)O1 2063,C(C(=O)NCCC1CCC1)(c1ccns1)N(C)CCOCC1CC1 2064,C1(NC(COCC(=C)C)=O)C=CCN(C(C2(c3ccc(Br)cc3)CCC2)=O)C1 2065,c1(CC)ccc(N)c(C(=O)NC2CN(C(=O)C(O)CC(C)C)CCC2CO)c1 2066,Cn1ncnc1C(=O)NC(CNC(=O)CC1OCCO1)C1CC1 2067,O(C=CC(=O)N1CC(C(C)NC(c2ccc(Br)o2)=O)C1)CC 2068,c1(C(=O)NCC(CO)NC(c2c(C)nn(C(C)(C)C)c2)=O)ccc(N=[N+]=[N-])cc1 2069,C=Cc1cncc(C(N2CCC(N(CCC)C(C3(C)CCNC3=O)=O)C2)=O)c1 2070,C12(CC3(CCC3)C1)CNC(=O)N2.c1(NCC(N)=O)nccc(C(F)(F)F)n1 2071,c1(SC)ccc(CC(=O)NCC2C(CNC(C3CSCCS3)=O)C2(F)F)s1 2072,N1(C(C2N(C(c3cc(C)[nH]n3)=O)CSC2)=O)CCC(O)C(C)C1 2073,C1(C(N2CCC(Oc3nccnc3Cl)CC2)=O)CCCCC12CCC2 2074,N(C1CCCOc2c(OC(C)=O)cccc21)CC(C1CCC1)OCC 2075,C12(CC(=O)NCC3CN(C(c4c(C)occ4)=O)C(C)C3)CCCN1CCC2 2076,C(C(C)(C)CNC(=O)Cn1nnnc1C(C)C)NC(C(C)OCCC#C)=O 2077,c1(C(CC(N2CCC(OCCN3CC(=C(C)C)C3)C2)=O)C)c(C)noc1C 2078,n1(CC(=O)NC2CCn3nncc3C2)nc2ccccn2c1=O 2079,c1(N(C(C(C)NC(CSCCC)=O)=O)C)cc(C)ns1.C(COC)OC=O 2080,c1(C(C)C)nccc(C(N2CCC(C)(NC(C3CCCSS3)=O)C2)=O)n1 2081,c1(COC)cccc(S(=O)(=O)NC(CCc2ccccc2)C(F)F)c1 2082,c1(NC(N2C(OC)C(C)CC2)=O)cnc2sc(C)nc2c1 2083,CCCC(CC(=O)N1CC(CSC2CCCN2)C1)c1ccccc1 2084,Cc1cc(C(N2CC3CC(C(N4CCOC(C(C)(C)C)C4)=O)(C3)C2)=O)cc(O)c1 2085,Cc1nccnc1C(=O)NC1CN(C(=O)NC2(c3nc(CO)no3)CC2)CC1C 2086,c1(CN2CCOCC(NC(C3CCC(=O)NC3)=O)C2)cc(O)c(O)c(O)c1 2087,CC1CC(C(=O)OC(C)(C)C)N(c2ccc(C(=O)O)cn2)C1.C1(C(C)O)C(=O)N1 2088,C1(NC(c2c(C)cn(C)c2)=O)CN(C(=O)C=Cc2c[nH]nc2C)C2(CCOC2)C1 2089,C1(NC(C2N(C(CC(=O)OCC)=O)C(C(C)C)CC2)=O)CCN(C)C(=O)C1 2090,CCCCC(O)C(C)C(=O)N(C(CNC(=O)COC1CC1)CC)C(C)C 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2216,N1(C(C(C(C)C)O)=O)CCC(C)(C)C1C(=O)NC1(CC(C)(C)C)CC1 2217,C1(CC)OCCC1C(=O)NCc1cc(C(=O)NC(C23CC(CO2)C3)C)n[nH]1 2218,c1(C(=O)NCCCCCN(C(=O)CCCN=[N+]=[N-])C)cc2n(n1)CCCC2O 2219,c1(C(N2CC(C(C)NC(c3ccc(CCC)s3)=O)C2)=O)cc2ccc(Cl)cc2[nH]1 2220,C(=O)(CC1=CCOCC1)N(c1nc(C)ccc1C)CCCNC(C(CC#C)(C)C)=O 2221,C(CCN=C(NCCNS(C)(=O)=O)N(CCS(=O)(=O)C1CC1)C1CCC1)SC 2222,C=Cc1ccc(C(N2CC3CCC2C3NC(=O)Cc2ccn(C)n2)=O)cc1 2223,C(=O)(C(O)CC(F)F)NCCCCC1CCCN(C(CCC(C)C)=O)C1 2224,C1(CNC(CC(C(C)C)C)=O)CN(c2nc3cccnc3s2)CC(C)(C)O1 2225,c1(C(=O)NCc2c(-c3c(C)nc(NC)s3)nccc2)cc(C)nc2c1nc(C)n2C 2226,CC(C)(CC#N)C(=O)N1CCC(NC(=O)C(c2ccccc2F)(F)F)C(O)C1 2227,Cc1cc(C(=O)NCC2CN(C(=O)CCCC(C)(F)F)CCC2C)c(N)c(Cl)c1 2228,c1(C(=O)OCCOC(N(C(=O)C(O)Cn2cncn2)C)=O)cnn(C(C)(C)C)c1 2229,c1(CC(=O)NCC2(C)CCC(NC(=O)C(N)=O)C2)ccc2c(c1)OC(F)(F)O2 2230,c1(NC(=O)CCCOCC2C(NC(C(C=C)O)=O)C2)ccc(C)cc1 2231,C(=O)(N=c1ccc(Cl)n[nH]1)C1N(C(c2ccc3ncnn3c2)=O)C2CCC1C2 2232,c1(C(=O)NC(CCC)C(=O)NCCC(C(C)C)N(C)C)cncn(C)c1=O 2233,N1(C(C2CCCN(C)C2)=O)CCC(F)(CNC(c2sccc2C#N)=O)CC1 2234,CC1CCN(C(c2cccc(C3CC3)c2)=O)CCN1C(=O)Cc1ncc(Cl)s1 2235,C(=O)(CCCCCCS(N)(=O)=O)NC(CCNC(Cn1ncc(CC)c1)=O)(C)C 2236,c1(CN2CCOCC(NC(c3ccn(C)n3)=O)C2)cnc2ncccn12 2237,c1(C(C)NCCOCC#C)[nH]c(-c2cccnc2)nc1C 2238,C1(C(=O)NCC2=CCCCC2)CCCCCCN1C(=O)CC12CCCC1C2 2239,C(=O)(CC1=CCCC1)N1C2C(C(=O)NC(C3CCOC3)CO)C(C2)C1 2240,CC(C)(CCC#N)C(=O)NCCC1CC(NC(=O)COc2ccsn2)C1 2241,C=C=C(C)CC(=O)NCC(CNC(c1ccc(OC(C)C)nn1)=O)CO 2242,N1(Cc2nnc(C(C)C)o2)CCC(NC(c2ccc(CO)o2)=O)C(C)C1 2243,C(CO)(C(=O)OCCC1CC(N(C)C)C1)NC(CNC(C(C)C1CC1)=O)=O 2244,c1(NC(C2N(C(c3cc(C)no3)=O)CC(F)C2)=O)cc2nccn2cn1 2245,Cc1nn(C(F)F)c(C)c1CC(=O)NCC1(N(C)C(C2NCC2)=O)CC1 2246,CCC(C)C(F)C(=O)N(CCCCC(=O)NCCC1CCN(C)C1=O)C 2247,CCC(CC)CCC(=O)NC1(C(=O)NC2CCOC(C)(C)C2)CC1 2248,c1(NC(c2ccc(CNC(CCC(C)OC)=O)cn2)=O)ccc2c(c1)OCC2 2249,N1(C(CS(CC)=O)=O)CCN(C(c2cn(C3CC3)nc2C)=O)C2(CC2)C1 2250,N1(C(c2n(C=C)nnc2)=O)CCOC2(CCN(C(=O)CC(C)(O)COC)C2)C1 2251,c1(C(N(C)CC2C3CN(C(C(C=C=C)C)=O)CC32)=O)cc(C)c(=O)n(C)c1 2252,C(=O)(C(C)(C)CC#N)NC(CCOCC)C(=O)NC(C)CCn1cncn1 2253,c1(C(C)NC(C2(C(C)NC(c3cccn3C)=O)CC2)=O)ccnc(O)c1 2254,N1(C(C(C(C)O)NC(C)=O)=O)CCc2ccccc2C(NC(=O)C(C)C(C)O)C1 2255,Cc1ccn2ncc(C(=O)NCCCC(C)NC(=O)CCC3CCOC3)c2c1 2256,Cc1ccc(C(N2CCN(C(=O)C(N3CCCC3)C3CC3)CC2C)=O)c(C)n1 2257,C12(C(N3C(C#C)CCCC3)=O)CCC(CN(C(=O)C(C)OC3CCCC3)C1)C2 2258,O=C(C1=C(Cl)CCC1)NCCCCC1CN(C(C2CC2c2ccnc(Cl)c2)=O)C1 2259,Cc1cc[nH]c(=N)c1C(=O)NCC(C)NC(c1cnn(-c2cccc(F)c2)c1)=O 2260,C(CC(C(=O)N1CCC(CCCF)CC1)NC(c1ccccc1)=O)N(C)C 2261,c1(C(=O)NC(CC)CNC(c2cn(C)nc2O)=O)cc(C)cc2c1CCC2 2262,N1(C(C2(C(=O)NC)CCC2)=O)CC(CNC(=O)C(O)C2CCCC2)C(F)(F)C1 2263,C(=O)(C(CC(C)C)C(C)C)N(CC(C)NC(c1c(C)cc(C)nc1S)=O)C 2264,C1(CC)C(C(=O)NC(c2c(C)noc2C)C2CC2)CCCN1C(C1CCOCC1)=O 2265,N1(C(c2cc(C)no2)=O)CCN(c2nccc(Br)n2)C(C#N)C1 2266,C(=O)(CC(CC)C(C)C)N1CCC(CN(C(=O)C(n2cc(C)cn2)C)CC)CC1 2267,C1(NC(C2(C)CC(=C)C2)=O)CN(C(c2cnn(C(C)C)c2C)=O)CC1C(F)F 2268,c1(CN2C(C(=O)Nc3cc(C)c(Br)c(F)c3)CCCC2)cc(F)ccc1[N+](=O)[O-] 2269,c1(C(=O)NCC2N(C(C3CCN(CC)C3)=O)CCOC2)[nH]cc2c1CCCC2 2270,N1(C(c2cnc(SC)s2)=O)CCC2CCC(C1)N2C(C1CN2CCN1C(C)C2)=O 2271,C(C(C)CN(C)N1CCC(OCC(=O)N(C)C)CC1)c1ccc(C)cc1 2272,c1(CCC(=O)NC2CCCCC2C(=O)NCc2ccnnc2O)ccccc1F 2273,C=C=CC(C)C(=O)NCCN(C1CCCCC1)C(=O)Cc1ccc(C(=O)OC)cc1 2274,N1(C(=O)Cn2cnnc2)CCC2(CCN(C(c3c(F)ccc(F)c3F)=O)C2)C1 2275,c1(C(=O)NC2CCCC(N(C)C(c3conc3C3CC3)=O)C2)cccc(F)c1Cl 2276,C(=O)(CCC(=O)N1CCCC1(CCOC)CO)NC 2277,n1(CC)ncc(C(N2CCCC(CNC(c3cc(F)n(C)n3)=O)C2)=O)c1C1CC1 2278,FC1(F)C2(CCC2)C12CC(CNCC1(c3ccccc3Cl)CCCC1)C2 2279,C1(NC(c2cc(OCC)ncc2)=O)C2CC1CN(C(c1cscn1)=O)C2 2280,CC(CC(=O)N1CC(NC(c2ccc(C(N)=O)[nH]2)=O)C2(CC2)C1)C(F)(F)C(F)(F)F 2281,C1(SC)CCC(C(=O)NC2(C(=O)C(C)OCCN(C)C)CC2)C1.C1(C)CC1 2282,c1(CNC(C(C)OCCOC)=O)cccc(CN(C)C(c2sc(C)nc2C)=O)c1 2283,N1(C(C(CCC)OC)=O)CC2(CCCCN(C(c3cncc(F)n3)=O)C2)C1 2284,c1(C(=O)NCC2C(NC(C34OCC(C)(C3)C4)=O)CCCC2)ccc(O)c(O)c1 2285,C1(NC(C2C(C)OCC2)=O)CCCN(c2ccccc2)C1 2286,c1(C(=O)NCCN(C(=O)C(n2ccc(Br)n2)C)CC)c(C)ncn1O 2287,c1(OC)cc(C)ccc1C(N1CCC(O)(C(=O)NCCC2CC3C=CC2C3)C1)=O 2288,c1(C(=O)NCC2(CNC(c3cc(COC)no3)=O)CC2(F)F)cnc[nH]c1=N 2289,c1(C(=O)NCCCC2N(C(C(C)SC(C)C)=O)CCC2)cc(Br)n(C)c1 2290,c1(C(C(N2CCN(C(c3cc(C)nnc3)=O)CC2)=O)=O)c(C)nn(C)c1C 2291,C1(NC(=O)CC2CC2(Cl)Cl)CN(C(c2cc(F)ccc2F)=O)CC2(CCC2)C1 2292,c1(C(N(CCC(=O)Nc2cnc(COC)s2)CC=C)=O)[nH]ccc1NC 2293,c1(C(N2CCC(C(C)NC(=O)CN3C(=O)CNC3=O)C2)=O)ccc(N=[N+]=[N-])cc1 2294,C(=O)(C(C)(C)CC(=O)N(C)CC1(O)CCN(C(=O)C2=NNC(=O)CC2)CC1)OC 2295,C(Cc1ccccc1)(CCNC(=O)CC1CSC1)NC(C(C)O)=O 2296,N1(C(c2ccc(C(F)(F)F)c(F)c2)=O)CCCN(C(=O)C2=CCCCC2)C(CO)C1 2297,O=C(C1=NOC2(CCC2)C1)NCC1CC2(CC2)CN1C(c1ccc(CO)cc1)=O 2298,c1(C(=O)NCC2CN(C(c3c(C)nn(C(C)C)c3C)=O)C2)cncc([N+](=O)[O-])c1 2299,CCC(F)(F)CC(=O)NCC1(COC)CN(C(c2ccc(Cl)nc2N)=O)C1 2300,c1(CCN(C)C(=O)OC(C)(C)C)nc(-c2cnon2)n(CCCC(F)F)n1 2301,c1(C(=O)NCC2(CN(C(C(C#C)(C)C)=O)C)CC2)nccc(F)c1Cl 2302,c1(C(=O)NCC2(NC(CSC)=O)CCOC2)cc(C2CC2)n(C(C)(C)C)n1 2303,C(C)(C(C)COC)(c1n(CCC)nnn1)NCC(C)(C1CC1)OC 2304,C1(NC(c2c(C)nn[nH]2)=O)CCN(C(=O)Cc2cc(F)cc(Cl)c2)C(C2CC2)C1 2305,C12(C(=O)NCCCC(C)NC(c3ccc(C(N)=O)cn3)=O)CCC(CC1)CO2 2306,c1(C(=O)NCC(C)CN(C)C(c2cc[nH]n2)=O)cc(OC(F)F)ccc1F 2307,n1(CC(=O)NCC(C)(C)NC(CCC(=O)NC)=O)ccc2ccccc2c1=O 2308,C1(CC2C(c3onc(CC(C(C)C)C4OCCO4)n3)CCC2)CCCC(=O)N1 2309,CC1CN(C)CCC1N=c1[nH]c(N2CCc3c[nH]nc3C2)nc2c1CCCC2 2310,C1(CSC2(C)CCCCC2)COC2(CNC2)C1 2311,c1(C(N2CCC3CN(C(c4ccc(OC)s4)=O)CC32)=O)ccc2[nH]c(=N)[nH]c2c1 2312,Cc1sc(Br)nc1C(=O)N(C1CCCN(C(C2CC2F)=O)C1)C 2313,C(C(O)CC(=O)NC(C)(C)CSC)NC(COCCC(C)C)=O 2314,c1(N2C3CC(CN(C(C4C(C)OCC4)=O)C3)C2)ncc([N+](=O)[O-])cc1CO 2315,CC1=CCC(C(=O)NCC(C)(C)OCCNC(c2cnn(CC(F)F)c2)=O)CC1 2316,C1(C(N(CCCNC(CC2(C)CCCO2)=O)C2CC2)=O)CCCC1(F)F 2317,N1(C(c2c(C)nc[nH]c2=N)=O)CCC(NC(c2sccc2Cl)=O)C12CCC2 2318,CCC(CCC(=O)NC(C)CCOC(C)C)NC(C1SCC=C1C)=O 2319,c1(NC(=O)N=c2nc(C3CCOCC3)[nH]s2)ccc2cc[nH]c2n1 2320,c1(NC(CCCN(C)C(C2CCC(C(N)=O)C2)=O)=O)ccc(C(F)F)nc1 2321,C1(C(N(c2nnc(S)n2C)C)=O)CCN(C(c2cnc(Cl)s2)=O)CC1 2322,C1(C(=O)NC(CC#C)C(=O)NC(CO)C(C)O)CC2C(C1)C2(F)F 2323,CC1(C)C(C(N2CC(NC(c3ccoc3Cl)=O)C2)=O)CC1(F)F 2324,N1(C(c2ccc(OCC)cc2)=O)CCC2(CC2)CC1C(N1CC2CC2C2CC12)=O 2325,Cc1noc(Cl)c1CC(N1CCCC(C2CCCCN2C(C2SCCS2)=O)C1)=O 2326,N1(C(C2N(CC)CC2)=O)CC2(C1)CN(C(C1CNC(=O)CC1C)=O)CCO2 2327,c1(C(CCC)C)nc(-c2nn(C)cc2Br)n(-c2cnnn2C)n1 2328,Cc1ccc(C(=O)NCc2ocnc2C(=O)NOCC(C)(C)O)[nH]1 2329,Cc1ccn(C(C)C(=O)NCc2cc(C(N3CC(C)(F)C3)=O)no2)n1 2330,C=CCC(C)C(=O)NC1CC(C(=O)NC(c2nccn2C)C)C1 2331,c1(OC)cc(C(N2CCCC(N(C)C(c3cc(F)cs3)=O)CC2)=O)cnc1O 2332,c1(C(=O)NCC(CC)NC(C2CCCC23CC3)=O)cnn(C(C)(C)C)c1Cl 2333,Cc1nn(CC(=O)N(CCNC(C2(C)CCCC2C)=O)C(C)C)cc1Cl 2334,CC(C)(C(=O)NCC1CCCN(c2ncnc(-c3ccccc3)n2)CC1)C(N)=O 2335,C1(C(C)C)CC(c2nnnn2Cc2ccco2)(NCC2CCS(=O)(=O)C2)CCO1 2336,C(=O)(CCC1=CCCCC1)N(CC(C)NC(=O)CC(C)O)C 2337,N1(C(C(C)OC(C)=O)=O)CC(C(=O)NCCCOCCOCCF)CC(F)C1 2338,S(=O)(=O)(c1ccoc1)N(CC1(C)CCN(C(=O)OC(C)(C)C)C1)CCO 2339,CON(CCC(=O)NC(C)C(F)F)C(=O)C1CC(C(C)(C)C)C1 2340,c1(C(N(CCNC(CC(CCSC)O)=O)C2CC2)=O)cc2ncccn2n1 2341,N1(C(c2cc(C)cc(C)c2)=O)CCN(C(c2nnsc2C)=O)C2CCCCC12 2342,CC1CC(NC(=O)Cc2cc(F)ccc2O)CN(C(c2cc(Cl)c(Cl)[nH]2)=O)C1 2343,C123CC(C1)(C2(F)F)CNC3=O.CCC(C(=O)Nc1nc(C)cs1)SC 2344,C1(CC(=O)NC(CNC(C(c2cccnc2)C)=O)C)CC(F)(F)C1(F)F 2345,C1(CCC)CN(C(=O)CC(C)COCC)CCN1C(=O)C(C)CC1CCC1 2346,c1(C(=O)NCC(C)CNC(c2ccnnc2S)=O)ccc(Cl)c(CCN(C)C)c1 2347,Cc1cc(P(C)(C)=O)oc1C1N(C(C2(n3cc([N+](=O)[O-])cn3)CC2)=O)CCNC1 2348,N1(C(C2C3(CCN(C(C45CCC(C)(OC4)C5)=O)C3)C2)=O)Cc2cncnc2C1 2349,C(=O)(C(C)(CO)NC(c1cnnn1C)=O)N(C(CC(C)C)C)C 2350,c1(CNC(CCN(C)C(C2CCCN2C)=O)=O)ncc(Cl)cn1 2351,c1(C(=O)NC2C(C)N(C(c3csc(C4CC4)n3)=O)CC2)cccc2nn(C)cc12 2352,c1(NC(C(C=C)F)=O)ccccc1NC(=O)CCc1ccc(C)cc1 2353,C(C)(CO)(C(=O)N(C)CC1(CNC(=O)CCn2ccnc2C)CC1)NC(C)=O 2354,N1(C(C2C(CN(C)C)CCC2)=O)CC2CN(C(=O)CN3CCCS3(=O)=O)CC2(C)C1 2355,CC1CCN(C(c2cccc3c2CCC3)=O)CCN1C(c1ccn2c1CCC2)=O 2356,CC1=C(C(=O)N2CCCC2CCNC(c2cnc(O)c(Br)c2)=O)CCO1 2357,C1(C(=O)NCCCCN(C(Cc2nc(NC=O)sc2)=O)CCO)CCC=CCC1 2358,Cc1ccccc1NC(=O)C(C1(O)CCC1)NC(=O)COCCCOC 2359,C=C(C)C1CN(Cc2ccccc2-c2cc(C)c(=O)n(C)c2)CCO1 2360,c1(C(N2C3(CN(CC(C)(C)C)C(CC)=O)CCC3CC2)=O)cc(S(C)(=O)=O)cs1 2361,N1(C(CC2N(CC)CCOC2)=O)CCC(NC(=O)CC2(OC)CCCC2)C(CO)C1 2362,Cc1cccc(N)c1C(N1CC(CCNC(c2ccnn2C(C)C)=O)C(C)C1)=O 2363,CC1(S(C)(=O)=O)CCCN(C(C23CSC(C2)C3)=O)C1 2364,CCC(C)C(C)C(=O)NC(C)Cn1cc(-c2cn(C)nc2C(=O)OC)nn1 2365,c1(CC(CNC(c2sccc2C(F)F)=O)CO)ccc(N2CCCCC2)cc1 2366,CC1CN(C(=O)CCn2ccccc2=O)CC1(C)CNC(=O)C(C)(C)C1CCC1 2367,c1(C(=O)OC)cn(C)nc1C(=O)N(C(C)CNC(=O)CC12CCCC1C2)C 2368,Cc1cc(C)c(C(=O)NCC2C=CCN2C(=O)CN2CCCCCC2)s1 2369,Cc1cc(-c2cn(CCCCCC(=O)N3CCCC(C(=O)O)C3)nn2)nc(O)c1 2370,c1(N2CCC(CCC)C2)nc(N2CCC(C)(c3ccccc3)C2)c2ncsc2n1 2371,C=C(C)CC(C(=O)N1CC(OCCC(=O)NCCc2csc(C)n2)C1)OC 2372,CS(=O)(=O)c1sccc1C(=O)NCC1CC(CNC(=O)Cn2ncnn2)CO1 2373,CS(=O)(=O)C1(C(N2CCCC2CCOC(N2CCCCC2)=O)=O)CCNCC1 2374,N1(C(C(Br)=C(C)C)=O)CCC(C2CC2)(CNC(c2ncnc3c2CCC3)=O)C1 2375,C1(NC(N2C(C)CSCC2)=O)COC2(C1)CN(C(c1ccccc1)=O)C2 2376,N1(C(c2cc(C)c(Cl)s2)=O)CCN(C(=O)Cc2conc2C)C2CC12 2377,N1(C(C2C(C)OCC2)=O)CCC2OCCN(C(c3ns[nH]c3=O)=O)C2C1 2378,c1(C(N2CC(CN(C(CCOC)=O)C)OCC2)=O)cc(Cl)c(F)cc1OC 2379,c1(C(N(C)Cc2cn(CC3CC34CCOC4)nn2)=O)c[nH]ccc1=O 2380,C1(OCC)CC2CN(C(=O)C(CN(C)C)NC(c3c(C)noc3N)=O)CC12 2381,c1(N2CC(C=C)OCC2)cc(S(=O)(=O)NC2CC3(CCC3)C2)ccc1C#N 2382,c1(C(N2C3CN(C(C(C)O)=O)C(C3)C2)=O)ccc2c(O)nnc(O)c2c1 2383,c1(C(=O)NC(C(C)C)CNC(c2cc(Br)ccn2)=O)ccc([N+](=O)[O-])cn1 2384,C1(CC(=O)NCC(CC)N(C)C(c2n[nH]c(C)c2Cl)=O)OCCCC1(C)C 2385,Cc1cc(Cl)cc(C)c1C(=O)NC1CC(NC(=O)CC(C)(C(F)F)N(C)C)C1 2386,C12(CC)CN(C(=O)Cn3cncn3)C(CNC(=O)CN(C)C(C3CC(F)C3)=O)(C1)C2 2387,C1(NC(C=C(C)C(F)F)=O)CN(C(=O)C(C)Sc2ccc(F)cc2F)CC12CC2 2388,C1(C(=O)NCc2ccn(CC)n2)CN(C(=O)C(C)OCCOC)C(C)(C)C1 2389,N1(C(CNC(=O)Nc2ccoc2)C(F)F)CCN(C(=O)CO)CC1 2390,C(C(C)C(F)C(=O)N(CC(C)O)CC)NC(CC1(OCC)CC1)=O 2391,C1(C(N(C2CN(C(C(F)=CC)=O)C2)CC)=O)CCC(C)N(C(=O)OC(C)(C)C)C1 2392,C1(CC(=O)NCC2(NC(C3CCCC3F)=O)CCC2)CCCCO1 2393,C1(CC)C(NC(c2cnc(C(C)(C)CF)o2)=O)CCCN1C(C1CC1(F)Cl)=O 2394,c1(C(N2C(CNC(C3N(N=O)CCCC3)=O)C=CC2)=O)ncnc2ccsc12 2395,N1(C(CC(C(C)C)C)=O)CCCCC12CC(NC(C1(C#N)CCOC1)=O)C2 2396,CC(C)(C)CC(O)C(=O)N1CCN(C(=O)COCCF)C(C(F)F)C1 2397,Cn1ncc2ncnc(N3CCN(C(C4CCSCC4)=O)CC3CO)c12 2398,C(C(C)(C)CNC(C1CCCN1c1nccs1)=O)N(C(C=C(C)Cl)=O)C 2399,Cn1c(O)nc2c(C(N3CC=C(CNC(=O)CN4CC=CC4)CC3)=O)cccc12 2400,c1(CN2CCC(C(=O)NCCCOCCC(=O)OC)C2)cc(C)cc(Cl)c1 2401,c1(C(N(CC(C)CNC(=O)Cc2cccnc2Cl)C)=O)ccnc2c1CC(=O)N2 2402,n1(CC)nncc1C(=O)NCC(CNC(C1CC=CCC1)=O)CO 2403,N1(C(c2c(OC)nsc2)=O)CC(OC)CC1C(=O)NCCO.C1(N)CCCC2CC12 2404,c1(C(=O)NC2CCCN(C(=O)CCc3ccccc3O)C2)ccc([N+](=O)[O-])s1 2405,C(=O)(C#CC1(C)CCCO1)N(C(C)C)CCNC(=O)CCc1nnc(C2CC2)o1 2406,C1(N(C(=O)C(C2CCOCC2)N2CCC2C2CCCC2)C)CCCCC1 2407,C1(C(N2CC(CNC(C3CCC(=O)O3)=O)C2)=O)CCC2CC2CC1 2408,N1(C(C=CC(C)C)=O)CCCN(C(c2cnc(OCC(F)F)c(Cl)c2)=O)CC1C 2409,C1(CNC(C2(CC#C)CC2)=O)CN(C(c2ccc(OCC)nc2)=O)CC(C)(C)C1 2410,N1(C(c2n(C)nc(C)c2Cl)=O)CCC2CCN(C(c3nc(=O)cc(N)[nH]3)=O)CC2C1 2411,C1(CN(C)C(c2cscc2C(F)(F)F)=O)CCCN1C(c1ccnnc1)=O 2412,Cn1cc(CC(=O)NC(CNC(C2COC(=O)N2)=O)Cc2ccccc2)nn1 2413,C(=O)(C(F)C1=CCCCC1)NC(CCNC(c1ncc(CC)s1)=O)C 2414,Cn1cnc(CCC(=O)NCCSCC(N2CC(OCC(N)=O)C2)=O)c1 2415,Cn1ncc(CNc2ccc(C(C)(C)C)cc2)c1F 2416,C1(C)(NC(C)=O)CCN(C(C2CCN(C(C3CC4CC4C3)=O)CC2)=O)C1 2417,C(=O)(CC1=NNC(=O)C1)N1CCC(NC(C(C)OCCOC)=O)C(C)C1 2418,C1(NC(CN(C(C)C)C(C2CCC3CC2CO3)=O)=O)CN2CCC1CC2 2419,n1(CC(=O)NC2CCN(C(=O)C=CC3CCCCC3)C2)nc(Cl)ccc1=O 2420,CCC(C(=O)N1CCCC(CCC(N2CCCC2C(=O)OC)=O)C1)C(C)(C)CC 2421,C(=O)(C1CNC(=O)c2ccccc21)N1CC2C(NC(CCOC)=O)C(C2)C1 2422,C1(C(C(N2CC(N(CC=C)C)C2)=O)C)CCCN(C(=O)C(C)=CCC)C1 2423,CC(CCCCNC(=O)C=CC1CCC1)NC(c1cscc1Cl)=O 2424,C1(C(C)(C)CNC(C23CCC(C2)C3)=O)CCCCN1C(c1cc(Cl)ns1)=O 2425,C1(CCOC2CN(C(CNC(=O)CC3CCCC3)=O)C2)COC2CC1C2 2426,c1(C(N2CCC(C(CC)CC)C2)=O)ccccc1NCC(F)(F)F 2427,c1(C(=O)NC2C(CCC)CN(C(C3CCC(C)O3)=O)C2)ccc(C)c(F)c1 2428,C1(C(F)(F)F)(C(=O)NC2(C)CN(C(CC3C(C)CCC3)=O)C2)CCCCO1 2429,c1(NC(N2C(C(=O)Nc3ncn(CC(C)C)n3)CC2)=O)cc(OC)c(F)cc1F 2430,c1(CC(=O)NC2(CCCCNC(C3CC(CF)C3)=O)CC2)cccc2occc12 2431,C1(C2CC2)(CC(=O)N(CC(CNC(C(C)=CC2CC2)=O)C)C)CC1 2432,N1(C(c2nc(NC(C)=O)sc2)=O)CC2CCN(C(=O)C3=C(Cl)CCC3)C(C2)C1 2433,Cc1oc2ccccc2c1C(=O)NC1CC2(C1)CC(CNC(=O)CC(C)CF)C2 2434,C(CCC(=O)N(C(CNC(c1ccccn1)=O)C1CC1)C)=CCC=C 2435,C12(C(=O)NCc3c(C(=O)NC(C=C)(C)CC)scc3)CC1COC21CCC1 2436,C(=O)(CC(O)CC(C)(C)C)N1CC(NC(CCCOC)=O)C2(C1)CC2 2437,c1(NC)c(C(N2CCCC(NC(C3(C)CCC(F)(F)C3)=O)C2C)=O)cccc1N 2438,C12(C(N3CCC(NC(C4CC5CCCC45)=O)C(F)C3)=O)CCC(F)(CC1)CC2 2439,Cc1nscc1C(=O)N(C(C)C(=O)N(C1CC1(C)C)CC1CC1)C 2440,N1(C(CP(C)(C)=O)=O)CCOC(C(=O)NCC2CCCO2)CC1 2441,C1(C(C(=O)NCCC)N(C2CCCCC2)CCCO)CCN(C)C1 2442,N1(C(C2N(CC)CCCC2)=O)CCCC(C2CCN(C(=O)C(C)CCO)C2)C1 2443,c1(C(N2CCC(NC(CC=C(C)C)=O)C2C)=O)ccc2c(c1)CCC(C)(C)O2 2444,C12C3CN(CC13)C2=O.c1(CC(CC2CC2)OC)cc(C2N=N2)co1 2445,N1(C(CCCSC)=O)CCC(CC(=O)NCCOCC(C)C)CC1 2446,c1(COC)ccccc1C(=O)N(CC(C)N(C(=O)CC1OCCC1(C)C)C)C 2447,S(=O)(=O)(c1ccc(F)cc1)NCCC(N1CCC(n2nncc2I)CC1)=O 2448,c1(CNc2cccc(C(=O)NC(C)C)c2)ccc2ccn(C)c2c1 2449,C(CCC(=O)NCCC(=C)CNC(=O)C(C)NC(=O)CC1C=CCC1)=CC 2450,C=Cc1cc(C(=O)NCCN(CCOC)C(C2(C)SCCCS2)=O)cc(F)c1 2451,c1(N(C(C)C)C)ncc(CN2CCSCC(C)C2)cc1F 2452,C1(N(C(C(CC)C)=O)C)CN(C(=O)Cn2nc(Cl)ccc2=O)CC1(C)C 2453,C(CN=C(NCc1cnn(C)c1)NCCN1CCOCC1)C1CC(C)OCC1 2454,C12(C(=O)NCCNC(c3cccc(O)c3F)=O)CCC(CC1)CC2 2455,C1(C(N2C(C(C)NC(c3cnc(CC)s3)=O)CCCC2)=O)CN2CCN1CC2C 2456,CCC(COC)C(=O)NCC(CC1CC1)C(=O)NCCCCN=[N+]=[N-] 2457,C1(C(=O)NCC(=O)NC(CC2CCC2)C(=O)NCC2CCOC2)CCCCC(O)C1 2458,C1(C(=O)NCC(C)Cn2ccc3cc(F)ccc23)CC2(CCC2)C12CCC2 2459,c1(N(CC(=O)NCC)C)ccc(S(=O)(=O)NC(CO)C2CC2)c(Br)c1 2460,N1(C(CNC(C2(C#N)CC2)=O)=O)CCN(C(C2CC3(CC3)CO2)=O)CC1 2461,c1(C(=O)NCCCCC(C)NC(=O)CN(CC(C)(C)C)C)cccc(C#N)c1Br 2462,C1(NC(c2c(C3C(C)C3)noc2)=O)CC(F)CN(C(=O)Cc2cncs2)C1 2463,c1(C(N(CCCCNC(=O)C(O)c2ccco2)C)=O)sccc1Cl 2464,CC1CN(C(=O)CC2CCN(C(c3ccn4c3CCC4)=O)C2)CC(=O)N1C 2465,N1(C(C(C2CC2)OCCSC)=O)CC(CNC(=O)OC(C)(C)C)C2(CC2)C1 2466,c1(CC)c(N2CCC(NC(=O)CSCC3CCCO3)C(F)C2)nc(C)nc1Cl 2467,N1(C(CC(C)=C(C)C)=O)CCC(C)(CNC(c2csc(-c3ccco3)n2)=O)C1 2468,c1(CC(=O)OC)ccc(CCNC(N2CCOC(CN(C)C)C2)=O)cc1 2469,c1(CNc2ccc(C(=O)NC)cn2)cc(Cl)c(Cl)cc1C.C12CCCN1C(=O)CC2 2470,c1(CC)c(C(=O)NCCC(C)(C)NC(=O)CCc2ncc(F)cn2)csc1C 2471,C(=O)(C1=CCC2CCC1N2C(c1cnc(OC)c(C)c1)=O)NCc1nc(CC)on1 2472,C12CN(CC1C)C(=O)C1(CCSC1)C(=O)OC2C1CCC(=O)N1.C(C)(C)(C)SC 2473,N1(C(CCCNC(C(C)(C2CCC2)OC(C)C)=O)=O)CC=C(C(C)C)CC1 2474,N(C(=NCCN1CCC(C)CC1)N1CCC2(CCCOC2)C1)CCOC 2475,C(=O)(C1=NNC(=O)CC1)N1CCC(O)(CC(=O)Nc2cc(OC)cc(Cl)n2)CC1 2476,c1(CC(C(=O)OCC)OC(c2cnc(OC(C)(C)C)cn2)=O)ccccc1Br 2477,C1(NC(c2ccc(F)c(C(F)F)c2)=O)COCCN(C(C2(C3CCC3)CC2)=O)C1 2478,Cc1cnc(C(N2CCC2CNC(=O)C(c2cccc(F)c2)(C)C)=O)cn1 2479,c1(C(C(=O)NC(C)(C)C)N2CCC2C2CS(=O)(=O)C2)cccc(Cl)c1Cl 2480,C1(C(=O)OC)CC(n2cc(C3(SC)CC3)nn2)CN1C(=O)Cc1cccc(C)c1 2481,c1(CC)nn(C)c(C(c2nnnn2C2CCOC2)NCc2nccs2)c1Cl 2482,Cc1cccc2c1N(C(C1CCCC1NC(=O)CC1(O)CCC1)=O)CC2 2483,c1(NC(=O)NC2CCCC(CN=c3nc(C4CC4)[nH]s3)C2)cnc2[nH]cncc1-2 2484,c1(NC(N2CCC(C(=O)NC)C(O)C2)=O)nccc2c1CNC2=O 2485,C1(C(=O)NC2C(=O)OCC2CO)(NC(C(C(C)C)F)=O)CCc2cc(Br)ccc2C1 2486,O=C1CC(NC(=O)CC2CCN(C(C3(O)CCC3)=O)CC2)CCN1 2487,C(=O)(C(F)(F)CC1CN(C(=O)Cn2nccn2)C1)NC1(CC)CC1 2488,CCCCC(CCCC)NC(=O)C(Cc1ccoc1)NC(c1cccc(C#N)c1)=O 2489,N1(C(c2ccc(C(CC)(C)C)cc2[N+](=O)[O-])=O)Cc2ccccc2CC1C 2490,C(=O)(C1=NNC(C(F)(F)F)C1)NCCCNC(CC1(OC)CCCC1)=O.C1CCS1 2491,c1(C(=O)NC(CC)CNC(=O)CC2CC2C)ccc2nnnn2c1 2492,c1(OC)ncc(C(=O)NCC2(C)CN(C(=O)C(C)N(C)C)CCO2)nc1C 2493,N1(C(CCC2C(C)(C)C2)=O)CC2CC1(C(=O)NC1CCC3(CC3)C1)C2 2494,c1(C(=O)NC2(CN(C(CC(C)(C)SC)=O)C)CC2)cnc2c(C)cccn2c1=O 2495,C1(C(=O)NCC#CCNC(c2c(C)nc(O)cc2)=O)C2CCC(C2)S1(=O)=O 2496,C(CCN(C)C)(C(=O)N1CCOC(C(C)C)C1)NC(c1nc(OCC)oc1)=O 2497,Cc1coc(C2CC2)c1C(N1CCC(OCCNC(C2CC(O)C(F)C2)=O)CC1)=O 2498,c1(C(N(CCCNC(CCOCCCOC)=O)C(C)C)=O)c(Cl)ccnc1F 2499,CCC(CC(=O)NC(C1CN(c2ncccc2C(=O)OC)CCS1)C)C(C)C 2500,N1(C2CN(C(C3(CCC=C)CC3)=O)C2)CC(NC(=O)C(COC)OC)CC1=O 2501,C#CC1CN2CC1N(C1CC1)CC(=O)N1CCCC(C1)CC2=O.SC 2502,C#Cc1ccc(C(=O)NC2(CNC(=O)C(c3ccccc3)C)CC2)nc1 2503,N1(C(C(c2cn(C)nn2)NC(c2ccc(C(C)=O)[nH]2)=O)=O)CC2COCC2(C)C1 2504,CC(CC(=O)NCc1csc(C(N2CC(C3CCCCC3)C2)=O)c1)C(F)(F)F 2505,CCC(CCOC)C(=O)NCC1(C(=O)NC2Cc3nccn3C2)CC1 2506,c1(C(N2C(CNC(C3CCC(=O)C3)=O)CC2)=O)ccc(Br)nc1O 2507,C(c1cc(C)no1)=CC(=O)NCC(C)N(C(CN(S(CC)(=O)=O)C)=O)C 2508,N1(C(CC(C)CNC(=O)CC2(C)CCCO2)=O)CC2(CCOC2)C1 2509,C1(C(=O)NCCC(C)(C)NC(=O)CCS(C)=O)CC(c2cccc(F)c2)=NO1 2510,c1(C(N2CC(N(C(C(C=C)O)=O)C)C(O)C2)=O)nn(C)cc1S(N)(=O)=O 2511,C(=O)(C(C(=O)NC1(CF)CCN(C(c2ncoc2C)=O)C1)C1CC1)OCC 2512,C1(CC=C)(NC(c2cc(CN(C)C)ccn2)=O)CCN(C(=O)C(C)(F)F)C1 2513,C1(CNC(c2nc(OCC)oc2)=O)CN(C(=O)COc2ccn(C)n2)CC1(F)F 2514,CCCC(C)C(CO)NC(c1conc1CNC(=O)C(F)F)=O 2515,C12(NC(C=COCC)=O)CCCC1N(C(c1cncs1)=O)CCC2 2516,c1(SCC)cnc(O)c(C(N2CC(NC(C3(C(C)C)CC3)=O)C(C)C2)=O)c1 2517,N1(C(c2c(C)nns2)=O)CCCC(CC(=O)NCCC2CC(F)(F)C2)CC1 2518,N1(C(C)C)CCCC1CC(=O)N(C(C)CCNC(=O)CCCN(C)C)C 2519,C(N=c1cc[nH]c(=NCCn2cc([N+](=O)[O-])cn2)[nH]1)c1nc(O)sc1 2520,C(CC(F)F)(C(=O)N1CC(=O)NC(=O)C1)NC(c1cnc(C)nc1)=O 2521,N1(C(c2ccc(SC)s2)=O)CCC(C)C(NC(=O)CCC(F)F)C1C 2522,CC1(C2CCCN(C(=O)CC3CCCN(C(c4cn[nH]c4)=O)C3)C2)CC1 2523,N1(C(CNC(C2C=CS(=O)(=O)C2)C)=O)CCCC2(C1)NC(=O)N(C)C2=O 2524,C1(CC)C(NC(C2SCC=C2C)=O)CCN1C(=O)CSCC(=O)OC 2525,c1(C(N2CCCC(C(=O)NCC(C3CCOCC3)OCC)C2)=O)cccc(C)c1O 2526,C1(NC(C(CC#CC)NC(c2cc(CCC)[nH]n2)=O)=O)CCN(C)CC1C#N 2527,N1(C(C2C(CC)OCC2)=O)CC(C2CCCN(C(=O)C(C)(C)C3CCC3)C2)C1 2528,C12CCC(C)CN1C(=O)CN(C1CCC1)C(=O)C(C)S2.C=C(C)COC 2529,C1(CN(CCC2C(O)C=C2)Cc2nnnn2C2CCC2)CCCCN1CC(F)F 2530,c1(C(=O)NC2(C)CCCN(C(CCC(=O)NCCC)=O)C2)cccc2cccn12 2531,C(=O)(CC(C(F)F)n1ccnc1)N(CCC)CCNC(=O)Cc1nc(CC)cs1 2532,C(=O)(N=c1[nH][nH]c2c1CN(S(=O)(=O)CCBr)C2(C)C)c1nc2ccc(OC)cn2c1 2533,c1(C(=O)NC(CN(C(CC(=C)C)=O)C)C)ccc(=NC)[nH]c1 2534,C(=O)(CC(F)(F)C(C)C)N1CC(CCNC(C2N(CC)CCCC2)=O)OCCC1 2535,c1(N2CC3C(NC(Cc4c(C)cc(C)nc4O)=O)C3C2)ncnc2scc(C)c12 2536,O=C(CCCCCc1ccccc1)NC1CC(NC(c2ccc(Cl)cc2O)=O)C1 2537,C=Cc1cncc(C(=O)NCC2CC3CCC2N3C(=O)CC2CC(OC)C2)c1 2538,CN1CCC(C(=O)N(C)CC2CCCN2C(=O)C=CC(=O)NC2CC2)CC1=O 2539,c1(CN2CCCC(NC(c3ccc(CN(C)C)cc3)=O)C2)ccc(F)c(C#N)c1 2540,C1(C(=O)Nc2occ(C(=O)NCc3nc(C)c(Br)s3)n2)CCc2ccccc2O1 2541,C(=O)(CC1OCc2ncccc21)NCCCN(C(C(CCSC)O)=O)C(C)C 2542,c1(CNC(c2ccc(CNC(C3N(CC)CC3)=O)s2)=O)csc(C#N)c1 2543,N1(C(Cn2cc(-c3cc(C)c(OCC)c(C)c3)nn2)=O)CCN2CCCC2C1C 2544,C(C(C)C(=O)NCCC(Cc1ccccc1)NC(c1nscc1N)=O)SC 2545,CC(C)C(C)C(CNC(C1CN(C)C1)=O)NC(=O)C(c1cn(C)nc1C(F)(F)F)=O 2546,N1(C(c2scc(C)c2)=O)CCCCC2(CCN(CCC(N3CCCCC3)=O)C2)C1 2547,CCC(C)CCCC(=O)N1CC2(CC2)CC1C(N1CCC2(CC1)N=N2)=O 2548,C(CCCC(C)NC(C1CC1C#N)=O)NC(C1C(COC)C1)=O 2549,C1(C(=O)NC(CSC)C)CC2CC1CN(C(c1ccc(O)cc1F)=O)C2 2550,C=C(C)C1OCCCC1C(N1CCC1CNC(c1cc(C)cc(O)c1)=O)=O 2551,C(=O)(CC(O)C(C)C)N1C(C(=O)NCC(CC(C)C)C)COCC1 2552,C1(C(N2CC(CF)(NC(=O)C(C)c3cccs3)C2)=O)(CC)CCCCO1 2553,N1(C(c2c(C)nn[nH]2)=O)CCOC(CN(C)C(c2nncn2C2CC2)=O)C1 2554,C1(C(N2CCC(C)(F)C2)=O)N(C(=O)Cc2nc(=N)[nH][nH]2)CC12CCCC2 2555,c1(CC)n[nH]c(CC)c1CC(=O)NCC12CC1CN(C(C1(C)CC(F)C1)=O)C2 2556,C(=O)(C(C)(C)CCCCC)NCC1OCCCN(C(C(CC#C)C)=O)C1 2557,C#Cc1cn(C)nc1C(=O)NC(CNC(=O)C(C)(C)Cc1ccc(Cl)cc1)CO 2558,C(=O)(C(F)CC(C)(C)NC(=O)C=CC1CCCCC1)N1CCC2(CN(C)C2)C1 2559,C1(CNC(C2(C(CC)(F)F)CC2)=O)(NC(=O)Cc2ncccc2C)CCOCC1 2560,N1(C(C(CC)CO)=O)CCC(O)(C2(NC(=O)CCSc3ccccc3)CC2)CC1 2561,C1(CNC(CNC(=O)OC)=O)CN(C(c2cn(C(C)C)nc2C)=O)CC12CCC2 2562,c1(C(C)NC(CCC2CCN(C(CCCOCCOC)=O)C2)=O)c(C)n[nH]c1C 2563,C(=O)(CC(C)C(C)C)NCC(CC(C)C)NC(=O)CN(C1(C)CCCC1)C 2564,C1(C(c2nnnn2C(C)C)NCC2(SC)CC2)CC2CCC1CC2 2565,CN1CCN(C(c2c[nH]nc2[N+](=O)[O-])=O)CC1CNC(C1CCCN1C1CC1)=O 2566,CC1(C)OC2C(NCC=CC3CCNCC3)CC(C(=O)NC3CC3)C2O1 2567,C1(CNC(CCc2cccc(OC)n2)=O)CCCCN(C(=O)CCS(C)(=O)=O)C1 2568,C(CC=C)(CC(=O)N(CC(C1CCCC1)O)C)NC(C(C=C=C)C)=O 2569,C(C(=O)O)(C1=CCC2CC2C1)NC(Cn1cc(-c2ccc(OC)cc2)nn1)=O 2570,Cc1c(C(N2CC(NC(C3(C(F)(F)F)CC3)=O)CC(C)C2)=O)cccc1N 2571,Cc1c(C(N2CC(N3CCN(C(=O)C=CBr)CC3)C2)=O)cnn1C 2572,C1(N(C)C)CCCC(C(N2CCN(C(c3sccc3Cl)=O)CC2CO)=O)CC1 2573,C1(OC)CN(C(C2CC(C)(C)C2)=O)CC1NC(=O)C=CCOCC(F)(F)F 2574,c1(N(CC(CN(C(=O)Cc2ncn3c2CCCC3)C)O)C)ncnc(Cl)c1C#N 2575,C=C(C)CCCC(=O)N1CC(CNC(c2c[nH]cc(Cl)c2=O)=O)C(C)C1 2576,CCC1=C(C(=O)NC2C=CCN(C(C3CCS(=O)(=O)C3)=O)C2)SCCO1 2577,c1(C(=O)NCC(C)N(C)C(C2(C)CCCCO2)=O)ccnc(CO)c1 2578,c1(-c2cc(C(N3C(C)COCC3)=O)sc2)ccc2cc(C3CC3)cn2c1 2579,S(=O)(=O)(C1CN(S(C)(=O)=O)C1)N1C(C)CN(C(c2cccc(OC)c2)=O)C1 2580,N1(C(Cn2c(C)ccn2)=O)CCC2CN(C(c3sccc3SC(F)F)=O)CC12 2581,c1(OC)ccc(F)cc1CN1CCC(CC(=O)NCc2cc3sccc3s2)C1 2582,c1(N(CCC)C)ccnc(C(N2CCC(N(C)C(c3ccc(Cl)s3)=O)CC2)=O)n1 2583,C1(N(c2ncnc(N3CCN(C(=O)C=CCO)CC3)n2)C)CC2CCCCC12 2584,c1(CC)c(C)nn(C)c1Cl.C1(=O)CC(Cc2cn(C3CC3)nn2)N1 2585,C=CCC(C(=O)N1CC(C(=O)NC2(CO)CCC(C)C2)OC(C)C1)C(C)C 2586,N1(C(CC(COC)C)=O)CCC(F)(CNC(C2(C)CCC(C)C2)=O)CC1 2587,C1(=CCC)CN(C(=O)C(C)NC(=O)C(C)SC)C1 2588,C1(NC(CC2(OC)CCCC2)=O)CCN(C(c2nonc2N)=O)CC1C 2589,C1(C(C)C)CN(C(c2cocn2)=O)CCC1NC(c1cnc(C2CC2)nc1O)=O 2590,Cn1ccc2c(C(=O)NC3CCCCN(C(C4CC4C#N)=O)C3)[nH]cc2c1=O 2591,C1(CNC(CCCC=C)=O)(OC)CCN(C(c2ccnn2CCF)=O)CC1 2592,C1(CC)C(F)CCC(c2ccccc2)N1CCOC.c12cnc(C)nc1CO2 2593,N1(C(c2cc(CNC(C(CC)(C)CC)=O)on2)=O)CC(C)CC(C)(C)C1 2594,C1(C(=O)OC)(CCNCCCN(C(=O)CSC)CCSC)CC1 2595,N1(C(c2cn(C)cc2C(F)(F)F)=O)CCCN(C(C2CCCCC2C(N)=O)=O)CC1 2596,c1(C(=O)NC(c2nocc2C(=O)NCC(F)F)C)sccc1C#N 2597,C1(C)(CC)C=C(C(=O)N2CC(CNC(=O)CSc3ccccc3C)CC2(C)C)C1 2598,N1(C(CCC)=O)CCC(C(=O)N(C)C(C2CCOCC2)C)=C(F)C1 2599,C1(OCCC)CCN(C(=O)C(C)(C)C2CCCN2C(=O)CC2CC(SC)C2)CC1 2600,CC(=O)CCCCC(=O)NC1CC=C(C(=O)NCCSCCN(C)C)C1 2601,N1(C(c2c(OC)ccs2)=O)CC(O)(C2(CNC(C3CC(C)(C)CO3)=O)CC2)C1 2602,C1(NC(COCC(=O)NC)=O)COC(C)(C)CN1C(=O)COCC1CCCO1 2603,C1(C(=O)OC)CC(C(=O)OCC2CC2c2ccccc2F)CC(C(=O)OC)C1 2604,c1(C(=O)NC2(C(N(CCC#C)CCOC)=O)CC2C)ncc(F)cc1F 2605,C1(OC(c2ccc(-n3cnnn3)cc2Cl)=O)CCOC2(CCCC2)C1 2606,C12(NC(c3nc(C(C)=O)sc3)=O)CC1CN(C(C1CCC(C)(C)C1)=O)C2 2607,C1(NC(CC=CCC)=O)CCCCC1NC(c1conc1C(F)(F)F)=O 2608,C(C)(CO)(C(=O)N1CC(C(N)=O)(CNC(c2cnn(C)c2Cl)=O)C1)OC 2609,c1(C(N2CCC(OC(C)(C)C)C2)C(=O)NC)cc(-n2cncn2)ccn1 2610,c1(C(=O)NCC(CNC(c2c(C(=O)OCC)c[nH]c2)=O)OC)cnn(CC)c1C 2611,c1(C(=O)NC(CC)CNC(=O)C(C)(C2CC2)OC)cccc2ccc(O)nc12 2612,C(=O)(CCN=c1cc[nH]cc1S(=O)(=O)NC1CCCC1S(C)(=O)=O)N(CC)CC 2613,c1(OC)ccc2c(n1)NC(C(N1CCC(NC(=O)CC(C)CF)C(C(N)=O)C1)=O)C2 2614,c1(C(N(CCNC(CCN(C(C)=O)C)=O)C2CC2)=O)ncc(F)c2ccccc12 2615,N1(C(C(CC2CCC2)OC)=O)CC(F)(F)CC1CNC(c1cc(C)sn1)=O 2616,Cc1cc(C)c(CC(=O)NC2CN(C(=O)C=CC=C(Cl)Cl)CC2O)c(O)n1 2617,C(C(=O)NC1CCN(C(=O)CN2CC(=O)NC2=O)CC1C)(C(F)(F)F)OC(C)=O 2618,CC(C)(C)CCC(C)(C(=O)O)NCc1ccc(NC(=O)OC(C)(C)C)cc1 2619,CC1(C)CCN(C(c2cnc(N)c(Cl)c2)=O)CC1NC(=O)Cc1n[nH]cc1Br 2620,C(=O)(C1CCCCc2ccccc21)NCCN(C(=O)C(C)C#N)CC 2621,CC1(C)CN(Cc2nccs2)CCN1CC1CCC2(C1)CC2(F)F 2622,c1(-n2cc(CCONC(C(C3CCCO3)OCC)=O)nn2)cc2ccccc2[nH]1 2623,C(=O)(CC(C)COC)NC(CC)CN(C(=O)CCn1ccnn1)C 2624,C(CN=c1[nH]c2cccc(C)c2s1)(C1CC1)NC(c1c(OC)cc(C)s1)=O 2625,c1(C(N2C(C)CC(NC(c3cc(F)ccc3F)=O)C2)=O)n[nH]c2c1CN(C)CC2 2626,C1(CN2CCC(C(=O)NC(CC)CC)C2)CC2(CCOCC2)C1 2627,N1(C(CC=C)=O)CC2CCCC2(NC(c2cc(C3CC(F)(F)C3)n(C)n2)=O)C1 2628,C1(NC(=O)NCCCNC(=O)NC)CCN(C(=O)NC)C1 2629,C(CCC)(C(=O)NCCCN(C(C1CC1c1ccn(C)n1)=O)CC)=CCC 2630,C=Cc1cnn(C)c1C(=O)NCC(C)N(C)C(c1nc(Cl)ccc1Cl)=O 2631,N1(CCC=C)CCC2(CN(C(c3nsc4ccccc34)=O)CC(C)O2)C1 2632,C(C(=O)NC(C)(C)C)(C1=CCSC1(C)C)N(CC#C)CC1CN(C(=O)OC)CCO1 2633,C12(C(=O)NC)CCC1CN(c1nccc(O)n1)C2.c1(OC(C)(C)C)ccc(N)cc1 2634,c1(C(=O)NCC2COCC2NC(C2CC2C2CCC2)=O)nccc2[nH]ccc12 2635,C12(CNC(C(CC)N(C)C)=O)CC(NC(=O)CSC3(O)CCCCC3)(CO1)C2 2636,C(CC1CCC1)(C(=O)NCC(N1CC(C)(C)C1)=O)NC(C)C 2637,C=C1CCC(NC(=O)NC(Cc2ccccc2)C(=O)N2CC=CC2)CC1 2638,Cc1cc(F)cc(C)c1C(N1CC2CCC1CN2CC1CCS(=O)(=O)CC1)=O 2639,c1(CC(N2C(CC)C(NC(=O)C(C)CSC)CC2)=O)ccc(C)cc1C 2640,N1(C(C(F)=CCC)=O)CC(C)(C(=O)NC2CC(C)(OC)C2)C1 2641,CC1=C(C(=O)NC2CC2NC(=O)CNC(=O)CC2CCCC2)CCS1(=O)=O 2642,CC1(NC(=O)CCc2c(F)cccc2Cl)CCCN(C(=O)CNS(C)(=O)=O)C1 2643,C#CC1(O)CC(C(=O)N(CCCC(=O)N(CC=C)CCOCCCO)C)C1 2644,C(=O)(C1=NNC(=O)C1)N1CCCC(CNC(=O)C(=Cc2cccc(F)c2)F)C1 2645,c1(N(C)C)cnc(C(N2CCC(C)(CNC(c3ncccc3CO)=O)C2)=O)nc1 2646,N1(C(Cc2nnc(-c3n(C)ccn3)s2)=O)CCCC2CN(C(=O)C#CC3CC3)CC12 2647,C1(C(=O)NC(C(=O)OC(N)=O)Cc2cn(-c3n(C)cnc3)nn2)CC(=O)CCO1 2648,CC1(C)CCN(C(=O)CCc2nccs2)C1CC(N1CCOCC1C1CC1)=O 2649,C1(F)(C(=O)NCC2C=CC(NC(CN3CCC(C(N)=O)C3)=O)C2)CCCCC1 2650,N1(C(c2cccc(C(=O)OC)n2)=O)CCC(NC(C2(CCO)CC2)=O)C(O)C1 2651,c1(C(=O)NC2CC(C)(CC)N(C(=O)C(N)=O)C2)c[nH]c2c(F)cccc12 2652,C1(C(=O)NCCNC(CCCOc2cccc(C#N)c2)=O)CCCCC1C1CC1 2653,N1(c2cc(NCC3CSCCO3)nc(C)n2)CCC(C)C(C)(C)C1 2654,C1(NC(N(C)CC2CCc3ccsc3C2)=O)CCc2cn(C)nc2C1 2655,c1(NC(C(Cc2ccoc2)NC(C(C=C)O)=O)=O)ccccc1F 2656,c1(C(=O)NCC2(C)CCN(C(C(C)=CC)=O)C2)cc(OC)cc(Cl)c1F 2657,C1(C(=O)NCCCC(=O)NO)CCCCCCN1C(c1csc(Cl)n1)=O 2658,c1(CNC(C2ON=C(CC)C2)=O)n[nH]c2c1CN(C(=O)C(C)(C)N(C)C)CC2 2659,c1(C(=O)OC)ccc(CCC(=O)NCC(CC(C)C)Nc2ncccn2)cc1 2660,C1(N(C(c2n(CC(C)C)ncc2)=O)C)CCCC(N(C(=O)C(C)(C)C2CC2)C)C1 2661,C(C)(CO)(C(F)F)C(=O)NC(C)C(=O)NCc1ncoc1C1CC1 2662,C(=O)(CCC(=O)NC(c1ccccc1)CNC(=O)CSCC1CCCCO1)NC 2663,CCC(C)(O)C(=O)NCC1(C)CC(NC(=O)Cn2nccn2)C1 2664,C12C(c3ccccc3)CN1C2=O.C1(SCCOC)OCCC1C 2665,c1(COC)ccsc1C(=O)N(C(C)CCNC(c1ncn(C(C)(C)C)n1)=O)C 2666,C1(NC(C2CCC(C)CN2C(=O)CN2CCCC2)=O)CCn2nnnc2C1 2667,CCCC(O)CC(=O)N1CCNC(=O)C2CC2C1.C(C(C)(C)C)SC1CC1 2668,N1(C(C2(CNC(CC(C)C3CCCO3)=O)CC23CCC3)=O)CCC2(CCCCC2)C1 2669,Cc1cc2[nH]c(C(N3CCCC(NC(c4cc(C#N)no4)=O)C3)=O)cc2o1 2670,C1(NC(C(=O)NC(C)C)=O)CCCCC12CCCN(C(=O)CCC1CCC1)C2 2671,C(CC(C(C)(C)C)NC(=O)Cc1c[nH]nc1O)N(C(=O)C(F)C1CCC1)C 2672,C=C(C)CCC(C)OC(c1ccc(-c2ccncc2C)s1)=O 2673,c1(C(C)=O)ncc(C(N2CCC2CNC(=O)CC(C)c2ccco2)=O)s1 2674,C1CN=C2N=c3ncn(C)c3=C(N2)N1.CC1CO1.C(CN(C)C)OCCN(C)C.O 2675,C1(NC(c2c(CC)c[nH]n2)=O)CN(C(=O)C(F)=C(C)C)CCC1(C)C 2676,c1(CNc2nc(NC(C)=O)c(F)c(Cl)n2)cnn2c1OCCC2 2677,C1(CNC(C(C2CC2)OC)=O)CCCCC1NC(=O)C(C)(C)C1CCCCO1 2678,C12(C(=O)NCC3CC(F)(CNC(c4cnc(SC)[nH]4)=O)C3)CCC(CC1O)C2 2679,C(C(O)CNC(=O)CC1CCSC1)NC(C=C)=O 2680,Cc1cc(S(=O)(=O)N2CCC(F)(NC(=O)OC(C)(C)C)C2)cc(C)n1 2681,C1(CNC(c2cn(C)nn2)=O)CN(C(C2(n3cccn3)CCC2)=O)C2CC12 2682,N1(C(c2c(C)nns2)=O)CCOCC(NC(c2cncnc2C(C)(C)C)=O)C1 2683,N1(C(C(C)CC2CC2)=O)CCN(C(=O)CN2CCN(CC3CC3)CC2)CC1 2684,C(C)(C(C(=O)N1CC(O)CC1C(=O)NCCC1CCCCC1)N(C)C)OC 2685,C1(F)(CNC(c2ccc(N(C(C)=O)CC)cc2)=O)CCC(CNC2CC2)CC1 2686,C1(NC(C2C(C)N(C(c3cn[nH]c3)=O)C2)=O)(CO)CC2CCCC12 2687,c1(C(=O)NC2CN(C(CN(C)CCO)=O)CC2C2CC2)nn(C)c2c1CCCC2 2688,C(C(C)(CC)C(=O)NCCCS(C)=O)NC(C(c1ccc(C)o1)C)=O 2689,Nc1cc(Cl)c(Cl)cc1C(N1CC2C(CNC(c3ccoc3C(F)(F)F)=O)C2C1)=O 2690,O=C(C1=CCCOCC1)NCC1CC2CCCC2N1C(c1cc(C2CC2)on1)=O 2691,C12(CNC(c3c(CC)nc[nH]3)=O)CCCC(CN1C(=O)C1=NOC(C)C1)C2 2692,C1(CNC(=O)NCCC2(c3cccs3)CCCC2)CCN(C2COC2)C1 2693,C1(OC)CN(C(=O)Cc2c[nH]ccc2=O)CC1CNC(=O)CC1CC1C1CCCC1 2694,Cc1cc(CO)oc1C(=O)NC1(CNC(C2CC3C=CC2C3)=O)CCOC1 2695,c1(OCC)cccc(C(N2CC(O)(CNC(C3CCC3C(F)(F)F)=O)C2)=O)c1N 2696,C(CC)(C(=O)N(CC(CC)NC(c1nnc(CSC)s1)=O)C)=CCCC 2697,C1(CCCCNC(C(C)SC(C)C)=O)CCN(C(c2c(C(C)C)cnn2C)=O)CC1 2698,C1(OC(c2c(CN)cccn2)=O)CN(C(=O)NCc2ccccc2)CCC1CO 2699,c1(C(=O)OC)cc(C(=O)N(CC(O)CNC(c2cccnc2)=O)C)cn1C 2700,C1(NC(=O)Cc2nc[nH]n2)CC2(NC(=O)Cc3cnoc3)COC1C2 2701,N1(C(C2(NC(C3CC(CC)OCC3)=O)CC2)=O)CCCC(C)(CO)C1 2702,CCCC(C)CCCC(=O)NC(C)CCN(C)C(c1occ2c1CCC2)=O 2703,c1(C(=O)NC2CC23CCN(C(C2C4CCCCC24)=O)C3)cc2cncn2c(O)n1 2704,N1(C(C(c2cccc(C)c2)(F)F)=O)CC2CC(NC(=O)CC3COCCO3)C2C1 2705,C(=O)(CC(F)(F)C(F)(F)F)N(CCC(C)NC(C1CC(CF)C1)=O)C 2706,N1(C(C(C)(C2CC2)OC)=O)CCN(C(=O)CC2CC3CCC2C3)C(C)C1 2707,c1(CNC(C(C2CCOCC2)C)=O)cccc(C(N2CC3C=CC3C2)=O)c1 2708,CCCC(C(O)C(=O)NCCS(=O)CC)NC(c1ncc(C)cc1F)=O 2709,C1(C(=O)NC2C=CC(C(N(C3CC(O)C3)C)=O)C2)COCC1(C)C 2710,CC(C(=O)NCC1(C)CCCN1C(c1n[nH]cc1Br)=O)P(C)(C)=O 2711,C1(C)(c2cn(CCCCOCC)nn2)COCCN1C(c1nnn(C)n1)=O 2712,C1(C(N2CCC(O)(C(C)NC(C3(CC)CC(C)(C)C3)=O)C2)=O)CC2C=CC1CC2 2713,C1(NC(CC2(OC)CC2)=O)COCCN(C(C2CC3C(C2)C3(F)F)=O)C1 2714,CCCC(C)(O)C(=O)N1CCC(NC(c2cccc(COC)c2)=O)C1 2715,C1(C(=O)NC(C2CCCC2)CNC(=O)CCOc2ccccc2)CC2(CC(=O)N2)C1 2716,Cc1nc(C)c(C(=O)NCC(O)CNC(c2ccsc2)=O)o1 2717,N1(C(C=CC)=O)CCCC(C)(NC(=O)C(C)Oc2ccccc2C#N)C1.C1CO1 2718,C1(NC(CS(N)(=O)=O)=O)CC12CCN(C(=O)CC1(c3ccccc3)CCC1)CC2 2719,C1(CCCC)CCCN(C(=O)NCc2cnc(C(F)(F)F)nc2)C1 2720,c1(OC)cc(C(N2CCC(NC(=O)C(C)C3(O)CCC3)C(C)C2)=O)cc(C)c1 2721,Cc1c(CNC(C2CCN(C(=O)CCNC(N)=O)CC2)=O)cnn1C 2722,C(=O)(N1OC2C=CC1CC2)c1nc(CCNC(CCC2N(C)CCC2)=O)oc1 2723,Cc1ncnc(C)c1OCC(=O)N(CCCNC(C1CCOC1C1CC1)=O)CCO 2724,c1(C(N(CCCCNC(c2cnc(CCC)s2)=O)C)=O)ccc(C)cn1 2725,C1(C(=O)NCCc2ccsc2)CCCCCN1C(C1CC(O)C1)=O 2726,C(N=c1ccc2c([nH]1)CCCCC2=O)C1C(C)CCCN1C(c1cccs1)=O 2727,N1(C(C=C)=O)CCC(C2CCCN(C(C)C(=O)NC3CCCC3)C2)CC1 2728,C1(NC(CSCC(C)C)=O)CN(C(C2(C#N)CCCC2)=O)CC(C)(C)C1 2729,S(=O)(=O)(c1ccc(F)cc1C)n1c(-c2cc(CC)cc(C)n2)nc(C(CCC)C)n1 2730,C(=O)(N(OC)C1CCC1)C1N(C(c2ccc(CC)cc2)=O)C2C(C1)C2 2731,N1(C(C2CCC(C)O2)=O)CCCOC(CNC(=O)CC2(n3cncn3)CC2)C1 2732,N1(C(CN(S(C)(=O)=O)C)=O)CCCCC1CCNC(=O)CC(O)c1ccccc1 2733,CC(C)CC(F)(F)C(=O)NC1CCCC(N(C(=O)C=C2CN3CCC2CC3)C)C1 2734,C(=O)(CC(C)C(C)C)NCCCOCCNC(c1cn(CCOC)nn1)=O 2735,C1(OC)CC(CNC(=O)Cc2ncoc2C)N(C(=O)Cc2ccc(Br)cn2)C1 2736,N1(C(c2c(CC)cns2)=O)CCCCC1CN(C(=O)CN1CCCCC1)C 2737,c1(C(=O)NC2CC2CNC(C2(F)CCC2)=O)c(Br)ccc2ccccc12 2738,CC1CCc2sc(NC3CC4(CCCN(C(=O)COCCN(C)C)C4)C3)cc2C1 2739,C(=O)(C1=CCCCC1C)N(CC(CO)(CO)NC(CC(C=C)(C)C)=O)C 2740,S(=O)(=O)(c1cnc(C(=O)O)s1)NC1(CN(c2c(C)ccc(Cl)c2)C)CCC(F)CC1 2741,C1(CC(=O)NCC2CC(OC)CN2C(=O)C=CC(C)C)CC2(CCCC2)CO1 2742,c1(CNC(C2CSCCN2Cc2ccc(I)o2)=O)cc(Cl)ccc1O 2743,c1(C(=O)NC2(CCCNC(c3cnc(OC)s3)=O)CC2)ccc(F)nc1F 2744,c1(OCOC)cc(-c2ncsc2C(=O)NCCc2ccccn2)c(F)cn1 2745,Cc1nc(C(=O)NCC=CCNC(=O)C(O)c2cnc[nH]2)c(Br)s1 2746,C(=O)(C(C)C(C)NC(=O)CCn1cccn1)NC(c1nc(C)on1)(C)C 2747,C#CCCCCCCC(=O)N1CCC(C(C)C(N2CC=CC2CF)=O)CC1 2748,C1(C(=O)NCCC(=O)NCCN(C)C(C2CCCO2)=O)(NC2CC2)CCCC1 2749,c1(N2CC(O)(CNC(CC(C(C)C)O)=O)C2)ccc(S(=O)(=O)N2CCCC2)cn1 2750,N1(C(C(C)C)=O)CCN(C(=O)CCN(C)CCO)C2COCC12 2751,Cc1cc(Cl)ccc1OCC(=O)NCC(C1CC1)N(C(C1CCCC1(F)F)=O)CC 2752,Cc1c[nH]c(C(=O)NC2CCC(CNC(=O)Cc3cc(Br)cs3)CC2)c1C 2753,Cc1c(C(N2CCCC2CNC(=O)CCC(F)F)=O)c(C(F)(F)F)nn1C 2754,c1(OC)ccc(S(=O)(=O)NCc2cc(C(=O)OC(C)(C)C)ncc2)c(C)c1F 2755,C12(CNC(c3c(CNC(c4ncn(C)n4)=O)ccs3)=O)CCCCC1C2 2756,Cc1coc(C)c1C(=O)Nc1ccccc1.N12CC3C(C3C1)c1cn(nn1)CC2=O 2757,N#Cc1ncc(CN2CCC(Cn3cc(-c4scnc4C4CC4)nn3)C2)s1 2758,Cc1nn(CC(N2CC(NC(=O)Cc3ccc(F)cc3)C3CC23)=O)c(=O)n1C 2759,CCC(CC)C(=O)NCC(=O)NCCC(C)(C)CNC(C1CCN(C(N)=O)C1)=O 2760,Cc1c(O)ccc(C(N2C3CCC2C(CNC(=O)CC(C)NC(N)=O)C3)=O)c1C 2761,C(C1COc2ccccc21)S(=O)(=O)Cc1nnsc1C(F)(F)F 2762,C1(NC(C2ON=C(CC)C2)=O)CCN(C(=O)CNS(=O)(=O)c2cccs2)CC1C 2763,Cc1ccc(C=CC(=O)NCC2CCC(C)N(C(=O)C=CCCC(C)C)C2)nc1 2764,C(CC)(CCCC(=O)N1CCCC(C#N)C1)NC(CCCCCC)=O 2765,C12(C(N(CCCNC(C3(c4n[nH]c(O)n4)CC3)=O)CC)=O)CC(COC)(C1)C2 2766,N1(C(C(C)OCCC=C)=O)C(CNC(c2nonc2CC)=O)CC2CCCCC12 2767,c1(OCC)sccc1C(=O)NCCCN(C)C(C1CCOC1CC)=O 2768,c1(C(N2CCC3CN(C(C45CCC(CC4)O5)=O)CC23)=O)ccc(Br)c2cn[nH]c12 2769,C(=O)(C1=CNC2=NCCC2=C1)NC(C(C)NC(CS(=O)(=O)NCC)=O)C 2770,c1(OC)ccc(Br)cc1CNC1C2CN(C(C3CCCS3)=O)CC12 2771,C1(NC(c2cc(CC)no2)=O)C2CCC(C2)C1C(=O)Nc1cc(C(N)=O)cc(Cl)c1 2772,c1(C(C(=O)NCC#C)NC(=O)C=CC2CCCN2C)ccc(C(F)(F)F)cc1 2773,c1(NC2CC(NC(=O)NC(C3CCCC3)COC)C2)c(C)ncnc1C 2774,C1(CC(=O)NC(CC2CC2)C2CC2)CCCC12CC2.N1(CC(=O)NC)CCCC1C 2775,N1(C(C(C2CCN(C(C3(COC)CCC3)=O)C2)F)=O)CC2CCC2(C(=O)OC)C1 2776,C1(CC)CCN(C(c2ccc(C3CC3)o2)=O)C1C(N1CCNC(=O)C1)=O 2777,c1(C(=O)OC)cc(NC(=O)C(C)n2ccnc2)cc(Cl)c1 2778,c1(COC)nc(NC2CC(C)SC(C)C2)cc(N2CCN(c3cc[nH]n3)CC2)n1 2779,c1(C(N2CC(C(C)NC(=O)C(N3CCCCC3)C)C2)=O)cn2c(n1)CCC2 2780,c1(C(C(=O)NC(C(C)NC(=O)CCc2cccn2C)C)O)cc(F)cc(F)c1 2781,C1(C(=O)NCCC2CCN(C(C3(CC=C)CCOC3)=O)C2)CN=C2N=CNN2C1 2782,C1(NC(c2c(Cl)cc(C)s2)=O)CCN(C(=O)C=Cc2cnccn2)CCC1CO 2783,C#Cc1ccc(C(N2CC(NC(C3CCCC3C3CC3)=O)C(C)(C)C2)=O)cc1 2784,C12(NC(C3CC(NC(=O)CCN4CCOCC4)C3)=O)CCOC(CSC)(C1)C2 2785,CC(CNC(C1CCOC1C1CC1)=O)(CO)NC(=O)COc1cn[nH]c1 2786,C1(C(=O)NC2C(C)CCN(C(C3CCS3(=O)=O)=O)C2)CCC2(CC1)CNC(=O)C2 2787,N1(C(c2ncc(Cl)cc2F)=O)CC(C2CN(C(=O)CSc3nnc(S)s3)C2)C1 2788,Cn1cnc(C(C(F)(F)F)NC(c2cn(CCF)nn2)=O)n1 2789,C(C)(C(CC(=O)NC(C)CCc1cn[nH]c1)NC(=O)CC1CCC=CCC1)OC 2790,C1(CCC(N2CC(C(=O)OCC)CC2(C)C)=O)CCc2ccccc2C1=O 2791,c1(OC(C)C(=O)NCC2(F)CC(NC(c3ccc(CO)o3)=O)C2)cccc(F)c1 2792,N1(C(c2nc(CCCC)sc2)=O)CCC2CN(C(c3cnc(C)cc3Cl)=O)CC12 2793,C(CC(C)(C)C(=O)NC1(C(=O)OC)CC1)NC(c1n(CCC)ccc1)=O 2794,N1(C(c2cc(C(C)=O)on2)=O)CCC(C(N2CC(F)(CO)C2)=O)C12CC2 2795,c1(OC(CC)C)ccc(C(N2CCCC(C(C)NC(=O)CC(F)(F)F)C2)=O)cc1 2796,N1(C(C(N2CCOC2=O)C)=O)CCOC2CN(C(c3ncc(Cl)cn3)=O)CC12 2797,CCCCC(C)C(=O)NCC1(C(=O)NCC2CNC(=O)O2)CC=CC1 2798,C12(CNC(c3c(C)nn(C)c3)=O)CC(CCO1)N(C(=O)COC(C)(C)C)C2 2799,C1(F)(NC(CC2(C)CCN(C(C(C3CCCCC3)C)=O)C2)=O)C(C)(C)C1(C)C 2800,C(CCC(C)(C)NC(=O)C(C1CCCN(C(c2ocnc2C(C)C)=O)C1)C)OC 2801,CC1(NC(C23CC(CN2C(C2CN4CCC2C4)=O)C3)=O)CC2CCC1C2 2802,c1(C(=O)NCC2C3CN(C(C(=O)N(C)C)=O)CC32)ccc2c(c1)COCCN2 2803,C(=O)(C(F)CC(C)(C)NC(=O)C1=NOC(C)C1C)N1CCC(COCC)C1 2804,CC(C)(CCNC(c1cc(C2CC2)nc2ccnn12)=O)S(C)(=O)=O 2805,CCC(C(=O)NC(C)=O)NC(C1CC(O)(CNC(c2cnn(CC)c2)=O)C1)=O 2806,N1(C)C2=NCCC1=CC=C(O)C=CN(C)N=CC=CCCN2C 2807,C(=O)(C(C)(C)C(=O)OC)N1CCC(CC#C)(C(=O)NC(C)CCNC(C)=O)C1 2808,CC1NC(=O)OC12CN(C(=O)C(C1CCN(C(C3CCCCS3)=O)C1)F)C2 2809,C1(C(N2C(CNC(c3cn(CC4(C)COC4)nn3)=O)C=CC2)=O)CC(=O)C12CCC2 2810,CC#CCCCC(=O)N1CCC(O)C(NC(C2CCCC(C)(C)C2)=O)C1 2811,CC(C)C(CO)C(=O)NCC1CC1NC(c1cnn(-c2ccccc2)c1N)=O 2812,C1(CN(C(C2(CC#C)CCC2)=O)C)CN(C(=O)CCc2ccoc2)CCO1 2813,c1(CN2CC(CC(=O)NCc3nc(C)[nH]n3)OCC2)cccc([N+](=O)[O-])c1 2814,C(CNC(=O)Cc1ccsc1Cl)(CC(F)(F)F)NC(=O)CC1(O)CCCC1 2815,c1(CNCCC2(C(=O)NCC(COC)F)CC2)ccc2nc(O)cc(O)c2c1 2816,C1(CN(C)C(C2CC3(CC3)C2)=O)CCCN(C(c2snnc2C2CCC2)=O)C1 2817,N1(C(C2C(=C)CC2)=O)C2CCCC1CC(CNC(c1c(Cl)ccc(F)c1F)=O)C2 2818,Cc1cccc(C(c2ncc[nH]2)NC(=O)N(C)Cc2ccccc2C)c1 2819,C1(C(=O)NC(COC)C(=O)OC)CN(C(=O)COC)CC12CC2.C(C)(C)(CC)N 2820,Cc1nn(CC(N2CC(NC(C34CC(N(C)C)(C3)C4)=O)CC2CO)=O)c(=O)o1 2821,c1(NC(C(c2cncc(C)c2)N(CC2CCOCC2)CC)=O)ccc(C)c(C#N)c1 2822,CC(C(=O)N1OC2C=CC1CC2)C1CCCN(C(c2cccc(F)c2)=O)C1 2823,c1(CC)c(C(N2CCC(CF)(NC(c3oncc3C)=O)C2)=O)cccc1F 2824,c1(C2(C(N3CCOC(Cc4ccc(Cl)cn4)C3)=O)CCCC2)ccccc1F 2825,C1(C(N2CCC(n3cc(CNC(COC(C)=O)=O)nn3)C2)=O)C(C)(C)C1(C)C 2826,CCCCC(C(=O)N1C2CCC1C(CNC(=O)C(C)OCCC(C)C)C2)N(C)C 2827,N1(C(C(CC)COC)=O)CCOC2CN(C(c3cc(C(F)F)cs3)=O)CC12 2828,N1(C(CCCCCCNC(c2ncn(CC)c2)=O)=O)Cc2cccc(C)c2C1 2829,c1(C(=O)NC(C(CO)NC(c2csc(C)c2C)=O)C)ncc(F)c2ccccc12 2830,N1(C(c2sc(C)c(O)n2)=O)CCCC2C1CCN2C(=O)CC1CCOC1 2831,C1(C(=O)NC(CCNC(C(N2CC(C)C2)C)=O)(C)C)CCC(F)(F)C1 2832,CCCC(CCC)=CC(N1CCN(CC(=O)NC2CCOC(C)C2)CC1)=O 2833,FC1(F)CCC2C(Oc3ccc(Oc4ccc(Br)cc4)nc3)C12 2834,N1(C(c2ccc(OC)s2)=O)CCCC(C)(NC(N)=O)C1.N12CC(C1)C2=O 2835,CCC(CC(=O)NCCC(=O)NCC(C)C)CC(C)C.C1(C)C(C)C(=O)N1 2836,c1(NCC2(NC(C3CCCC(F)(F)C3)=O)CCCC2)ncc(Br)c(O)n1 2837,N1(C(C2CN(C(N)=O)C2)=O)CC(C(=O)NCCCN2CCSCC2)C2(CC2)C1 2838,N1(C(=O)NCC(C)N(C)C)CCC(O)(NC(c2cnccn2)=O)C1 2839,C(c1cccnc1)=CC(=O)NC(CNC(C1CCN1C1CCCC1)=O)CO 2840,Cc1ccc(CCC(=O)NCC(C)NC(c2c(C)ccn2C)=O)c(Br)c1 2841,C1(CNC(c2n(CCOC)ccc2)=O)CCCCN1C(=O)Cc1cnccc1C 2842,c1(C(=O)NC(C(=O)N(CC(COC)C)C)(C)CSC)ccc2nccn2c1 2843,c1(C(=O)NCC2(NC(C=C(CC)CC)=O)CCCCCC2)cc(C)c(F)cc1N 2844,N1(C(C(=O)N)COC)CCC(CCc2cncn2C)CC1.CCCCOC 2845,c1(CNC(NC2C(C)C2)=NCc2cnn(C)c2)ccc(Cl)c(C(F)(F)F)c1 2846,c1(COC)nc(C(F)F)cc(=NC(C)C2CCCN2C(=O)C(C2CC2)SC)[nH]1 2847,c1(C(=O)NCC2CCC(NC(CC3(C=C)CCOCC3)=O)C2)c(C)ccc(F)c1N 2848,c1(C(=O)O)cnc2c(c1)N(C(c1nnc3ccccc3n1)=O)CCO2 2849,C1(COC)(CNC(=O)CCCCCN(C)C)CCN(C(=O)CCCCSC)CC1 2850,C1(C(=O)OCC)CN(C(=O)CC2(N(C)C)CC2)C2(CCC2)C1 2851,C1(C(N2CCCC(N(C(C3CCC(=O)O3)=O)CC)C2)=O)CCC(=C(F)F)CC1 2852,CCCC(C)(CO)NC(=O)CCC1CCN(C(c2scc(C)c2C)=O)C1 2853,c1(C(=O)NC2(COC)CCN(C(=O)C=CC(C)(C)SC)C2)cc(C)ncc1C 2854,N(C1CCCn2nccc21)C(CSCCNC(CCC(C)(C)[N+](=O)[O-])=O)=O 2855,c1(CC(=O)NC2CCCN(Cc3ccc(C(=O)O)cc3)C2)ccc(F)cc1 2856,C1(CNC(c2nn(CC)c(O)c2)=O)C2CCCC1N(C(=O)CCC(C)O)C2 2857,N1(C(c2cc(C)nn2C)=O)CCC2CCCC12C(=O)NCCN1CCCC1 2858,C1(C(=O)NCC#CCC)CC2(CCC2)CN1C(c1cc(F)ccc1C)=O 2859,C1(C#N)(C(=O)NC(C)CN(C(=O)CCCN2CCCC2)C)CCS(=O)(=O)CC1 2860,C(C(CNC(c1cnn(-c2ccc(Cl)cc2)c1)=O)C(F)(F)F)NC(=O)C=CCF 2861,C12(C(=O)NC3C4CN(C5CCN(c6c[nH]nc6)C5=O)CC43)CCCC1C2(F)F.CC 2862,C1(C(=O)NCc2ncccn2)Cc2cc(O)ccc2CN1C(c1ccnnc1)=O 2863,c1(NC(C2N(C(c3ccc(OCC)nn3)=O)CCC2C)=O)ccc2c(c1)CCC2 2864,Cc1cc(=NCCc2c[nH]c3ccccc23)[nH]c(=NCC2CCN(C(C)C)C2)[nH]1 2865,C(N=c1cc[nH]c(=NCCN2CCCOCC2)[nH]1)c1ccc(SC)s1 2866,C1(C)(C(=O)NCCC2CCN(C(C(C=C=C)C)=O)C2)CC(OC)CN1C 2867,C(=O)(C1=CCCCC1C)NCC1C(C(=O)NC(C=C)(C)C2CCCC2)CCC1 2868,CCCCC(CC)C(=O)NCCCN(CC(=O)N(C)CC1(C)CC1)C 2869,C1(O)(C(N2CC(NC(C3CCCC3C)=O)CC(C)C2)=O)CN2CCC1CC2 2870,C1(C#N)(C(=O)NCCCCCN(C)C(C2(C3CCCO3)CCC2)=O)CC1(C)C 2871,C#CC1CN(C(=O)CCCN(CC)NC(=O)C=CC(C)(C)SC)CC1OC 2872,CC(C)CC(C(=O)NC1C=CC(C)(C)CC1)NC(c1nn(C)cc1Cl)=O 2873,c1(C(=O)NC2(COC)CN(C(=O)CCN(C)C)C2)cc(C2CC2)nc(O)c1 2874,C(=O)(CC1=NNC(=O)C1)NCCC1CN(C(C2CC(CN(C)C)C2)=O)C1 2875,C1(C)(C(N(CCN(C(C)C)C(C2CCC(F)(F)C2)=O)C)=O)CCCN1C 2876,CC(C)CC(O)C(C)C(=O)NCc1nnn(C)c1C(=O)NC1CN(C)CC1C 2877,CC(CCCCCO)NC(=O)C=CC(C)(C)NC(C1CC(=O)OC1(C)C)=O 2878,N1(C(Cc2scc(C)c2)=O)CCC2C(C1)CN2C(=O)CCCC(=O)OC(C)(C)C 2879,C12(C(=O)NCCC3(C(=O)OC)CCCC3)CC1CN(CC(=O)Cc1nc[nH]n1)C2 2880,c1(CC(=O)NC2C(C)CN(C(C3CC3C)=O)CC2)ccc2c(c1)CCN2C 2881,C1(CC)CN(C(C2CC(OC)CCN2C=O)=O)CCN1C.c1(C)cc(C2CC2)on1 2882,C(=O)(CCN(CCCO)C(=O)C=CCF)N(C)CC1CCCO1 2883,Cn1c(=O)c2ccc(NC(=O)NCC3(CCCO)CC3)cc2n(C)c1=O 2884,N1(C(CCc2c(C)nccc2)=O)CCC(NC(=O)Cc2csc(CO)n2)C(O)C1 2885,N1(C(C(=O)NCCOC)=O)CC2COCCC2(NC(C2CC23CC(F)(F)C3)=O)C1 2886,C1(NC(C2(OCC)CCC2)=O)COCCN(C(c2c[nH]n(CCOC)c2=N)=O)C1 2887,CC1CC(CNC(C2CN(C3COC3)C2)=O)CN1C(=O)CCCCN(C)C 2888,C1(CC#C)(C(=O)NCCCC(N)=O)CCN(C(=O)CCc2cn(C)cn2)C1 2889,C(=O)(CC(C)(C)CNC(C1CCCN1C=O)=O)NC(C)(C)CC1CCC1 2890,CC1=C(C(=O)NC2CN(C(C3(C(F)F)CCCC3)=O)CC3CC23)CCO1 2891,c1(C(=O)NC23CC(NC(C(C)SCC)=O)(C2)C3)cnn(-c2cccc(F)c2)c1C 2892,c1(C(N2CC(N(C(CC=C)=O)C)C(F)C2)=O)[nH]c(C)c(C(=O)OC)c1C 2893,C1(NC(C(=O)NCCC(C=C)C)=O)CC12CCOCC2 2894,CCC(C)CCCC(=O)NCC1(CNC(=O)C(CC)n2ccnc2)CCCCC1 2895,C1(C(=O)NCC=CCNC(CCn2c(C)ncc2)=O)CCc2cnnn2C1 2896,N1(C(c2n(CCC)ncn2)=O)CC(NC(C2CC2OC(C)=O)=O)C2(CCC2)C1 2897,c1(C(=O)NCC(CCOC)NC(=O)CC2CCCN(C)C2)c(C)nnn1C 2898,c1(CN(CC)Cc2ncsc2Br)ccc(C(N2C(CCC)CCCC2)=O)cc1 2899,C1(C(N2CCC(COC)(NC(=O)C=CCOC)CC2)=O)Cc2cccnc2C1 2900,c1(CN(C(=O)C(C)N(C)C(=O)OC(C)(C)C)CC)ccc(C(=O)NC)c(F)c1Cl 2901,N1(C(CCCN(C(=O)CC2CCCC(C)C2)C)=O)CC2CCCC(C1)N2C 2902,c1(CC)nc(N2CCN(C(=O)Cc3ccc(Br)cc3)C(C)C2)c(C#N)cc1C 2903,c1(C(=O)NCC(=C)CCNC(=O)C(F)=C2CCC2)cncc(P(C)(C)=O)c1 2904,C(C)(C)(CCC(=O)N1CC(NC(C2CCCCC(=O)N2)=O)CC1CO)OC 2905,n1(CC#C)ccnc1C(=O)N(CCC)CCNC(C1CC(CC2CC2)C1)=O 2906,N1(C(C2(C#N)CC=CC2)=O)CC(C2CCCN(C(=O)CCCN=[N+]=[N-])C2)C1 2907,N1(C(CCn2ncc(C)c2)=O)CCC(NC(C2(c3cccnc3)CC2)=O)C(O)C1 2908,C1(CNC(=O)CC2CCNC2=O)CCCN(C(C23C=CC(CC2)C3)=O)C1 2909,Cc1ncsc1C=CC(=O)NC1CN(C(=O)C(c2cncc(F)c2)C)C1 2910,C(=O)(C1CCCCn2ccnc21)N1CCCC(CC)(CC)C1 2911,C1(NC(=O)CN(C(=O)Cc2ccsn2)C2CC2)CCN2CCC1C2 2912,c1(C(N(CC(C)O)CCNC(CCCOC)=O)=O)c[nH]c2cc(F)ccc12 2913,c1(C(N2CC(CC3CC3)C2)=O)nccc2occc12.c1cc(C(F)(F)F)ncn1 2914,C1(CNC(c2c(C)non2)=O)CC(F)CN1C(=O)CCc1cccs1 2915,c1(CCC)nc(C)c(C(=O)NC(C2CCCCN2C(=O)Cc2cnc[nH]2)C)s1 2916,C1(C(=O)NCCNC(c2cc3sccc3[nH]2)=O)Cc2ccccc2C(=O)O1 2917,c1(C(C)C)nc(NCc2cc(F)cc(C)c2N)cc(=NC(C)c2nonc2C)[nH]1 2918,c1(C(N2CC(NC(c3cc(C(C)C)[nH]n3)=O)C2)=O)cc(N(C)C)ccc1N 2919,C1(NC(CC2N(CC)C(=O)CC2)=O)CC12CCN(C(=O)CCc1ncco1)CC2 2920,n1(CC)cc(C(N2CC(F)CC2CN(C(c2ccccc2)=O)C2CC2)=O)c(Cl)n1 2921,C1(NC(CCC=C(C)C)=O)CCOC(C(=O)NCCc2c[nH]nc2O)C1 2922,CCC(CCC(=O)NCC(N1CCN(C(=O)Cc2cccnc2)CC1)=O)OC 2923,N1(C(CCC#CC)=O)CCC(C(=O)NCc2ncccc2Cl)C(C)C1 2924,N1(C(C2CCC(NC(C3(OC)CCSC3)=O)C2)=O)CCC2C(=O)NCC2C1 2925,c1(CC(=O)NC2CN(C(C3CC4(CC(=C)C4)C3)=O)CC2F)cccc2sccc12 2926,C(c1c(C)coc1C)=CC(=O)N(C1CN(C(CC=CC=C)=O)C1)C 2927,c1(C(N2CCC(N(C(c3c(CC)c[nH]c3)=O)C)C(C)C2)=O)cc2ccccn2c1 2928,C(=O)(C#CCC(C)(C)C)NCC(C)CCC(=O)NCC(O)C(C)(C)C 2929,c1(CC)ccc(C(N2CCC(N(C(C3CSC3)=O)CC)C2)=O)o1 2930,C(C(=O)O)(C1CCOC1)N(C)CCN(C(=O)CSC(F)(F)F)C 2931,C1(C(C)NC(=O)CSCCO)CCCN1C(C1CC(C)(F)C1)=O.C1(CN)CCCO1 2932,C(=O)(CN1C(=O)COc2ccccc21)N1C(CN(C(=O)C=NOC)C)CCCC1 2933,c1(NC(C(C2C3COCC23)N(C)CCN2CCCC2=O)=O)cccc(Cl)c1 2934,C1(C(N(C2CCOC2)CCNC(CC2C(CC)C2(F)F)=O)=O)CCCCCCC1 2935,C1(NC(CN(C)Cc2ccccc2)=O)CC12CC(NC(C1CCOC1(C)C)=O)C2 2936,Cc1cc(OCC(=O)NCCN(C(=O)CCc2nc(O)n[nH]2)C(C)C)ccc1F 2937,C#Cc1cnc(C(=O)NCC2CCN2C(=O)Cc2cnc[nH]2)c(C)c1 2938,C1(NC(c2cn[nH]c2)=O)CC2(C1)CC(C(=O)NC1(CO)CC(F)C1)C2 2939,CC(C)C(O)C(F)(F)C(=O)N(C)CC1COCCN1C(c1ccc2c(c1)CC2)=O 2940,N1(c2nc(C)nc(O)c2)CC2(CN(C(c3nocc3C)=O)CC2CO)C1 2941,C1(CC(=O)NCCN(C(=O)CC2CSC2)CC)CC=CCC1 2942,c1(CCC)noc(CN(CC(=O)N)C)n1.C(C)(CC#C)CC(F)(F)F 2943,C1(CCCCCNC(C(C)C)=O)CCN(C(=O)C(F)F)CC1 2944,C1(NC(C(F)=C(C)C)=O)CC2CC(C1)CN(C(C1CCCN1CC(F)(F)F)=O)C2 2945,c1(C(=O)NC(CC(C)NC(=O)Cc2ccon2)C)sc2sccc2c1Cl 2946,c1(C(N(CCNC(c2cc(CC)c[nH]2)=O)CC)=O)csc2c1CCC(C)C2 2947,c1(CC)ccc(C(=O)NC(C)CCNC(C2(C)CC2(F)Cl)=O)s1 2948,C1(CC(=O)NC)CN(C(C2CC3(CCCC3)C2)=O)CCN1C(=O)CC(C)F 2949,c1(C(=O)NCCC2(C)CCN(C(=O)CSc3nc[nH]n3)C2)cc(O)nc(O)n1 2950,CC1(NC(=O)CC2(N3CCCC3)CC2)CCN(C(c2sccc2C(F)F)=O)CC1 2951,c1(CCNC(c2ncn(C)c2Cl)c2n(CCOC)nnn2)ccc(C(N)=O)cc1 2952,C(=O)(C(C)(C)CC(=O)NC(c1ccc(F)cc1)CNC(=O)COCCCF)OC 2953,C(c1ccc(C2N(CCSc3ccccc3)CCNC2=O)cc1)=C(C)C 2954,C(=O)(CCC(=O)N1CC2C(CC(=O)N(C)C)C2C1)N(C1CCCOC1)CCC 2955,c1(C(C)=O)c(C)[nH]c(C(N2CC(F)(CNC(C3CCS3(=O)=O)=O)C2)=O)c1C 2956,C(=O)(C(C)(C)CN(C(=O)CC=C(Cl)Cl)C)NCC1CCC(C(=O)OC)O1 2957,C(CCCCC(=O)N1CC(CCONC(=O)N(C)C)C1)n1cc(CCC)nn1 2958,C(CCC(=O)NC(C)CC(C)NC(c1ocnc1-c1ccccc1)=O)OCCC 2959,c1(NC(=O)NC2CC2(c2ccccc2Br)F)ccc2nc(O)oc2c1 2960,C12(C(N(C3CCN(C(C4CCC5(CCC5)O4)=O)CC3)CC)=O)CCOC(C)(C1)C2 2961,N1(C(C2C(CCC)C2)=O)CC(OC)CC(NC(c2cnc(C(C)(C)C)nc2)=O)C1 2962,C1(NC(C(C)SC)=O)CCN(C(C2CC2c2ccccc2Cl)=O)CC1(C)C 2963,c1(C(=O)NC(C2CCN(C(=O)CCC(N)=O)CC2)C)cc(C(F)(F)F)cnc1O 2964,N1(C(CN)=O)CC2CCCC(C1)N2C.c1(CC(=O)CC#C)c(C)noc1C 2965,c1(C(CC)C)nc(C)cc(=NC2CC23CC(NC(=O)C(C)CC(N)=O)C3)[nH]1 2966,C1(C(=O)OCCCC2CCCC2)CC2(CCCC2)CO1 2967,c1(OC)cc(C(N2CCCC(NC(=O)CC3SC(=N)NC3=O)CC2)=O)cc(C)n1 2968,C#Cc1cncc(NC(C2(CNC(=O)CC34CCCN3CCC4)CC2)=O)c1 2969,CN1CC(N(C)C(C2C=CCCN2C(=O)CCCN(C)C)=O)CCC1=O 2970,N1(C(c2ccc(C)s2)=O)CCN(C(=O)CCC2(C)CC2)C(C(F)F)C1 2971,N1(C(CP(C)(C)=O)=O)CC2C3CCC(C2C1)N(C(=O)C=C1CN2CCC1CC2)C3 2972,C(=O)(C1CCCc2nn[nH]c21)NC1CC(C)(NC(c2ccc(Br)c(O)n2)=O)C1 2973,Cc1ccc(CC(=O)NCCCN(CCO)C(C2C(C)(C)C2(F)F)=O)cc1Cl 2974,N1(C(CCCC#CC)=O)CCC2(CCC2NC(=O)CC2OCCC2(C)C)CC1 2975,c1(C(=O)OC)cc2oc(C(N3CCC4C(C(=O)O)C4C3)=O)cc2[nH]1 2976,N1(C(C(CCSC)O)=O)CCCC(NC(C2CCN(C(C)=O)CC2)=O)CC1 2977,NS(=O)(=O)CCC(=O)N1CCCCC1C(=O)NCC1(O)CCSC1 2978,N1(C(C(CC=C)C(C)C)=O)CCC(C2CN(C(=O)CCC3CCOC3)C2)CC1 2979,C1(C(=O)NC2(CO)CN(CC(=O)NC3CCCC3F)C2)C2C3CC4C1C1C2CC3C41 2980,Fc1cc2c(cc1F)C(NC1CC(CC3(C(F)(F)F)CC3)C1)CCC2 2981,Cc1nc(CC(=O)NC23CC(C(=O)Nc4ncco4)(C2)C3)cs1 2982,CC1CCC(C)C1NC(c1c(CNC(=O)CN=[N+]=[N-])nnn1C)=O 2983,c1(-c2cccc(C3C(C)(C)C3(F)F)c2)cccc2nsnc12 2984,Cc1cc(C(=O)NCC(C)(CO)NC(C2CCOC2)=O)nn1-c1ccc(F)cc1 2985,Cc1nn(C)c(NNC(=O)c2nccc3ccccc23)c1C#N 2986,c1(C(N(C)CC2CCN(C(=O)COc3ccon3)C2)=O)ccc(F)c2[nH]ccc12 2987,Cc1ccc(CN(CC(=O)NC(C)CNC(=O)C(C)n2ccnn2)C)cc1 2988,c1(CNC(c2n(CC)nnn2)c2ccn(C(C)(C)C)c2)ccc(C(F)(F)F)cn1 2989,C(CCC[Si](C)(C)C)NC(c1cc(C)c(CC)s1)c1n(C(CC)C)nnn1 2990,n1(CCCC)ccc(C(=O)N(C(CNC(C2CCNC2=O)=O)C2CC2)C)n1 2991,C#CCCCCC(=O)NC1CC(C(C)NC(C23CCCN2CCC3)=O)C1 2992,c1(CNC(=O)Nc2c(OCOC)ccc(Br)c2)cccc([N+](=O)[O-])c1 2993,c1(C(=O)NCC(C2CCC2)NC(C=CCC)=O)cc2cccc(O)c2[nH]1 2994,c1(CC)cc(F)ccc1C(=O)NCC1CN(C(C2CC3C(C2)C3(F)F)=O)CC1O 2995,N1(C(c2nc(C)[nH]n2)=O)CCC2(CCOCC2)C(CNC(=O)CCCC(F)F)C1 2996,C1(NC(C#CC(C)(C)O)=O)CC2CC1CN(C(=O)CCC(C)(C)N1CCCC1)C2 2997,Cc1ncnc(N2CCC(C)(CNC(=O)Cn3cccn3)CC2)c1Br 2998,C(C1CCCN1C(c1csc(Cl)c1)=O)=CC(=O)N(CCSC)C 2999,C1(NC(c2c(CC)ccs2)=O)CC2CN(C(c3c(C)noc3CC)=O)CC2C1 3000,C1(C(=O)NC(C(C)O)(C)C)CCCCCC1NC(=O)CC1OCCO1 3001,C1(NC(c2cn(CCC)nc2C)=O)CC1C1CCCN(C(=O)C(C)(C)C)C1 3002,n1(CCN(C(=O)CSC(c2ccccn2)CC)C(C)C)cc(-c2ccncc2)nn1 3003,Cn1cc(C2OCCC2C(=O)NC2(C)CC(NC(c3ncccn3)=O)C2)cn1 3004,N1(C(=O)Nc2ccc(OCC#C)cc2)CC=C(c2cccc(Cl)c2)CC1 3005,C(=O)(CCCC(=O)NCC1(OC)CN(C(C2CCC3CCC23)=O)C1)NC 3006,CN=c1cc(C(N2CC(C3(NC(C4CC(C)=NO4)=O)CC3)C2)=O)cc[nH]1 3007,C1(CNC(C2(C(=O)NC)CC2)=O)CCCN(C(c2sc(C)cc2Br)=O)C1 3008,Cc1c[nH]cc1C(=O)N(CCCCCNC(c1cn(CC2CCOC2)nn1)=O)C 3009,c1(CC)[nH]nc(C(N2CC(OCC(=O)NC3CC(C(=O)NC)C3)C2)=O)c1Cl 3010,Cc1nc2c(cc1C(=O)NCCC1COCCN1C(=O)C=C1CC1)c(C)nn2C 3011,C1(C(N(CCN(C(Cc2cc(CC)no2)=O)C)C)=O)CC12CCC(=O)CC2 3012,Cc1ccc(C(N2CC3(CCCCC3)C2)=O)c(N)c1F 3013,C(C(=O)NC1(C2CCCN2C(c2nccnc2N)=O)CC1)(C(C)C)SCC 3014,C(=O)(C(C)(O)CC(C)C)NCCC(=C)CNC(=O)COc1cc(C)on1 3015,CCCCC(O)C(=O)N1CCC(CNC(=O)C=C2CCN(C)C2)C(C)C1 3016,c1(OC)c(F)cc(C(=O)NCC2CN(C(C3CN(C)CCO3)=O)CC2C)cc1Cl 3017,N1(CC)CC(C)(C)C2COCC12.C12(C)CCC(O1)CN2C(=O)N(C)C 3018,C#CCCC(O)C(=O)NC(C)CCNC(c1snnc1CC)=O 3019,C1(C(N2CCCC(NC(CCc3ncc(C)[nH]3)=O)C2C)=O)CS(=O)(=O)CC(=O)N1 3020,C(=O)(CCCCC#N)N(C1CN(C(c2c(CC)c[nH]n2)=O)CC1F)C 3021,N1(C(CC)C(C)C)CC2COCC2(C(=O)NC2CCC(C(=O)OC)C2)C1 3022,CCCC(CCCS(C)(=O)=O)C(=O)NCC1(C)COCCN(C(C2COC2)=O)C1 3023,N1(C(C(C(CC)C)N(C(=O)CN2CCCCC2)C)=O)CCN2CC(O)CC2C1 3024,N1(C(c2c(C)coc2)=O)CC2CN(C(=O)C=CC(C)C)CCC2(CO)C1 3025,C1(C(N(CC(C)NC(=O)CCc2ccncc2Br)C)=O)OC2CCC1CC2 3026,CC1C(C)C(C)CN1C(=O)C(=O)N(CC(F)(F)F)Cc1ccc(C(N)=O)c(F)c1 3027,CCC(CCC(=O)NCCN(CC(F)F)C)NC(c1cc(C)ncn1)=O 3028,Cc1cc(=NC(=O)C(=O)NCC2CC(=O)N(CC3CC3)C2)[nH]n1CC 3029,c1(C2C(CNC(=O)NC(C3CCOC3)COC)CC2)ncc(C)cn1 3030,CC(C)CC(F)C(=O)N(C1CCCN(C(=O)CCOCC2CCC2)C1)CCO 3031,C(CC(C)C)(C(=O)N(CC(=O)N(C)OCC(F)(F)F)C)NC(C(CC)C)=O 3032,c1(CCOC(C)=O)ccc(C(=O)NCC2C(NC(=O)CCCF)C2(C)C)cc1 3033,c1(C(=O)NCCN(C(CCn2c(C)ncc2)=O)CC(C)O)c[nH]c(=S)cn1 3034,CCCC(C)CC(=O)N(CCCC(=O)NCCOC1CCOC1)C 3035,c1(N2CCC(NC3CCC(C)C3)C2)ccc(C(F)(F)F)cc1 3036,C(=O)(CC1OCc2ccccc21)NC(CNC(C(=O)NC(C)C)=O)C1CC1 3037,Cc1nnc2n1CCN(C(=O)CC1CCN(CCC(C)C)C1)C2 3038,c1(C(N2C3CCC(CNC(C(CC)COC)=O)(C3)C2)=O)cccc2ccn(C)c12 3039,CC1CN(C(=O)Cc2cc(Cl)ccc2O)CCC1NC(=O)Cn1ccnn1 3040,N1(C(c2cnn(C)c2C)C(=O)NCCCSCC)CC(C)CCCC1C 3041,C1(C(=O)NCC(CC)NC(c2cc(C)on2)=O)(CN2CCCC2)CCCC1 3042,C(C(CC(C)C)C(=O)NCCC(C)CO)NC(CCc1onc(C)n1)=O 3043,c1(C(N2C3C(NC(CS(CC)=O)=O)CC(C3)C2)=O)cn2cccc(C)c2n1 3044,C12(NC(c3cncc(-c4ccoc4)c3)=O)CC1CN(C(C1CCC13CCC3)=O)C2 3045,N1(C(CCC(=O)NC)=O)CCOc2ncc(C(=O)NNC(=O)c3cccnn3)cc21 3046,S(=O)(=O)(c1ccc(F)cc1)NCC(=O)NCC1C(CNC(C(C)N(C)C)=O)C1 3047,C(=O)(CC(C(F)(F)F)n1cccn1)NCC1(CNC(C(C)(C2CC2)OC)=O)CCC1 3048,N1(C(C=C(COC)C)=O)CCC(CN(C)C(C2CC2(F)F)=O)C1 3049,c1(OC)ccccc1C=CC(=O)NC1CCCC1NC(=O)Cc1c(C)noc1C 3050,C1(NC(C2(CC=C)CN(C(C3(O)CCOC3(C)C)=O)C2)=O)CC2(CNC(=O)O2)C1 3051,CC1CCN(C(=O)CCc2cn(C)cn2)C1CNC(=O)Cc1ccc(Cl)nc1 3052,Cc1cc(CNC(C2(O)CCN(C(=O)CC3CCCN(C)C3)C2)=O)cc(O)n1 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3071,N1(C(=O)CCc2cn[nH]c2)CCCC1CN(C(C1(CO)CCCC1)=O)C1CC1 3072,C1(C(N(CC(CNC(c2c(OC)scc2)=O)C)C)=O)CCCC12CCC2 3073,N1(CC(=O)NCCNC(C2C(C)OC(=O)N2)=O)CCC(=O)NC1=O 3074,C1(C(N2C(C)(CC(=O)NC3CCCN3C=O)CC2)=O)CN(CC2CC2)CCO1 3075,CC1CC(C)(C(N2CCCC(O)(CCNC(=O)C3=CCC3)C2)=O)CC(C)O1 3076,c1(CNCC(c2ccc(OC)cc2)NC(C)=O)c(C)cc(C)cc1C.C(=O)(CC)OC 3077,c1(C(C)C(=O)NCC2CCN(C(=O)CC3CCCC4CC34)C2)ccc(Cl)c(Cl)c1 3078,c12nc(C)cnc1NC2=O.c1(N)ccnc(C(F)(F)F)c1.CC 3079,c1(C(=O)NCc2c(CN(C(=O)CS(C)(=O)=O)C)cccc2)cc(N)c(F)cn1 3080,C(=O)(CCCNC(CC(N)=O)=O)C12C(C1)CC(=O)N(C)CC(C)(C)NCC2 3081,c1(OCCC)cccnc1C(N1CCC1CNC(=O)C=Cc1ccc(CC)o1)=O 3082,N1(c2cc(SC)ncn2)CCOCC(NC(c2cscc2Cl)=O)C1 3083,c1(CNc2c(C)ccc(N(C)C)c2)ccnc2c1c(C)nn2C.c1(=O)c(=O)[nH]1 3084,C(=O)(C(Cn1cccn1)NC(C1CCOC1)=O)N(C)Cc1cn[nH]c1 3085,c1(CC)cnc(C(N2CCC(CN(C(=O)Cc3csnc3C)CC)CC2)=O)nc1 3086,Cc1ccnc(O)c1C(=O)NCCNC(c1cn(C)c(-c2ccccn2)n1)=O 3087,c1(C(=O)NC2(C(O)CNC(C3(C4CC4)CC3)=O)CCC2)ccc(CN(C)C)nc1 3088,C1(CN(C)C(C2CN(Cc3ncn(C)n3)C2)=O)CCCC2CC12 3089,N1(C(C(CCC)OCC)=O)CCC2CCN(C(=O)C=Cc3cc(OC)no3)C2C1 3090,C1(C(C(=O)NCC2CCN(C)C2)=O)CCNC1(C)C 3091,c1(OC)nc(Cl)ncc1C(N1CCC(OC)CC1)=O.C12C(C)CCN1C2=O 3092,N1(C(c2c(OCC)scc2)=O)CC2CC(C1)C2NC(=O)CSCCC(F)(F)F 3093,C1(CNC(CCCC)=O)C(C)CCCN1C(c1ccc(CC(C)C)nc1)=O 3094,c1(C(=O)NC2CCCC(n3cc(C(C)NC)nn3)C2)ccc2c(c1)CCCS2 3095,N1(C(COCC(=O)NC)=O)C(C(=O)NC(CO)CCOC)CCC1C(C)C 3096,C1(NC(C23C(CN(C(c4c(OC)cccc4)=O)C2)C3)=O)CCC(C)(C)OC1 3097,c1(C(=O)NC23C(CN(C(CCCC(=C)C)=O)C2)C3)ccc2cncn2c1 3098,N12C(c3ccc(Br)cc3)=CSC1=Nc1cccc(Cl)c1C2C.CC1CC1 3099,C1(NC(CC2(C=C)CCC2)=O)CCN(C(=O)CC2CC(=O)C2)C(C)C1 3100,N#Cc1cc(C(N2CC(NC(c3sccc3F)=O)C3(CCC3)C2)=O)cc(F)c1F 3101,C12(CNC(c3c(Cl)ccc(N)c3)=O)CCCCC1CN(C(=O)CC(F)F)C2 3102,CN1CC(NC(C2CN(C(=O)CN3CCNC3=O)CC23CC3)=O)CCC1=O 3103,C1(N(C)C(C2CC2C2CCC2)=O)COC2(CCN(C(=O)C(C)(C)C)CC2)C1 3104,CCC(C)(C)C(C)CC(=O)NCCC1CC(NC(c2ncc3[nH]ncc3n2)=O)C1 3105,CCCC(C)C(C)NC(=O)CNC(c1ocnc1CC)=O 3106,c1(N(C)C)cc(NC(C2CSCCN2C(c2ccccc2C#N)=O)=O)ccc1Cl 3107,C1(NC(C2CC(C(C)C)C2)=O)CC2CCC(C1)N2C(=O)COCCN(C)C 3108,c1(C(=O)NC(CC(C)NC(c2cc[nH]c2)=O)C)ccc(-c2cnc[nH]2)cc1 3109,C=CCCCC(C(=O)NCC(COC)OC)NC(=O)CCCC(=O)OC 3110,C1(NC(C(C)C2(O)CCC2)=O)COCCC1C(=O)NOCC1CCOCC1 3111,C1(C(N(CC(CCC)O)C)=O)CC(OC)CN1C(=O)CC1CC2(CCC2)C1 3112,C1(NC(C(C)=C(CC)C)=O)CCCN(C(c2n[nH]cc2Br)=O)C1 3113,C1(NC(c2ccc(C)cn2)=O)CCN(C(=O)CN(C)C(=O)C2CC2)C(C)C1 3114,C(=O)(C(=O)CC(C)CC)N(C1CCCN(C(=O)C(CCC)OC)C1)CCC 3115,C(=O)(C(C)CC(C)CC(C)C)NCC1(F)CC(NC(c2nnn(CC)c2C)=O)C1 3116,c1(CN2CC(F)(CC(N3CC4C(C(=O)OC)(C4)C3)=O)C2)ccc2c(c1)nnn2C 3117,C1(C(=O)Nc2cccc(OC3CC3)c2)CCCC(CNC(C2CC2)=O)CC1.COC 3118,C1(CCC)CN(C(=O)CC(CC)SC)CC1C(=O)NC1CC1c1ccccc1 3119,C1(C(N2CC(C)C2C(=O)NCCc2cn(C)nn2)=O)CC12CCCCC2 3120,N1(C(Cn2cc(C(C)=O)nn2)=O)CCC(NC(C2CC23CCOC3)=O)CC1 3121,Cc1ncc(NC(=O)C(C)NC(=O)C(C)C2(O)CCC2)c(C)c1C 3122,c1(CN(C(=O)C(=O)Nc2ccc3nn[nH]c3c2)CCOC)ccc(S(C)(=O)=O)cc1 3123,c1(CC)cc(C(=O)NC(C)C(C)NC(=O)C(C)n2ccnc2)ccc1O 3124,C(=O)(C(F)C(C)CNC(C1CCS(=O)CC1)=O)NCc1c(OC)nn(C)c1 3125,C12(C(=O)NCc3cnc(C)s3)CC1CN(C(C1CCO1)=O)C2 3126,N1(C(CC2C(=O)NC(=N)S2)=O)CCC2CC(NC(=O)C(O)C(N)=O)CCC2C1 3127,c1(C(=O)NC2C(CNC(CNC(C)=O)=O)C2)cncs1 3128,Cc1nc2cc(NC(=O)C(C(C)(C)C)NC(N)=O)cnc2[nH]1 3129,C(CNC(=O)C(F)(F)C(F)F)(CC(F)(F)F)NC(C1CN(S(CC)(=O)=O)C1)=O 3130,C12CCN(C(=NCc3ccc(OC)c(OC)c3C)NC1)C2.OC 3131,N1(CC(CC#C)=O)CCc2ccccc2C1CC(=O)Oc1ccccc1CC 3132,C1(C(=O)NC(C(N2CC(C)=C(C)C2)=O)(C)CN(C)C)CC2(CC(=O)C2)C1 3133,C1(CNC(c2scc(C)n2)=O)CCCN(C(c2cccc(OC(F)(F)F)c2)=O)C1 3134,C1(c2n(CCC(C)=CC3CC3)nc(-c3ccnn3C)n2)CCn2c(C)cnc2C1 3135,C(=O)(CCCCCc1ccc(O)cc1)Nc1cc(C)nn1C(c1cccnc1)C 3136,Cc1ccc(NC(=O)C(=O)N2CC(n3ccc4c(Br)cccc34)C2)cc1[N+](=O)[O-] 3137,N1(C(C=C(C)C)=O)CC(NC(=O)CCCOC(C)C)C(c2ccnn2C)C1 3138,C1(C#N)(NC(CC(C)O)=O)CCN(C(=O)CN2C(=O)CSC2=S)C1 3139,C1(NC(C(CC=CC)C)=O)CC2CCC1C(NC(=O)COc1cc(C)on1)C2 3140,CCCC(C(=O)N1CCC(C)(NC(c2nccn3ccnc23)=O)C1)C(C)C 3141,CC1=CCC(C(N2CCCC2C2(NC(C3CNC(=O)N3)=O)CC2)=O)CC1 3142,CC(C)(C#N)CCCC(=O)NC1CCCC(NC(C2CC23CCSCC3)=O)C1 3143,c12cc(sc1Cl)-c1noc(n1)-c1csc-2n1.c1(C(C)(C)CO)ccccc1 3144,c1(OC)ccc(Br)cc1COC(=O)C(C(C)(C)C)Nc1ccccn1 3145,c1(C(=O)OC(C)(C)C)ccccc1NS(C)(=O)=O 3146,C1(CC(=O)NCCC(C)NC(=O)C=C2CCCCC2)CC2(CCC2)C1 3147,CC(C)C(C(=O)NCC#CCNC(=O)CC1(O)CCC1)c1ccc(F)cc1 3148,c1(COC(C(N2CCCCC2=O)C)=O)nc(Br)nn1C 3149,C1(CCC)CN(C(=O)Cn2nc(C)nc2C)CCN1C(=O)C1=C(Cl)CCC1 3150,N1(C(C2N(C(C3CC3c3ccc(Br)cc3)=O)CCC2)=O)CCN2CC(O)CC2C1 3151,C1(c2scc(C3CCN(CC(C)CC#N)C3)n2)CCCN(C(=O)NC(C)(C)C)C1 3152,C(=O)(C(C)(C)C(C)C)N(C1CCN(C(COCCSCC)=O)C1)C 3153,C1(C(=O)NC(CC(C)NC(=O)C=CC(=O)NC2CC2)C)CC(C(=O)O)C1(C)C 3154,c1(OC)ccc(Br)c(CC(=O)NCCCNC(C2CC3(C2)CC(O)C3)=O)c1 3155,C(=O)(C1=NN(C2CC2)C(=O)CC1)NC(CNC(c1cc(OC)ncc1)=O)CO 3156,C(=O)(CCCCCF)NCCOCCN(C(=O)CC1CC1(Cl)Cl)C 3157,CCCC(C)(O)CC(=O)NC1(C)CCCCC1C(N1CC=CC1CF)=O 3158,CC(CNC(c1csc(O)n1)=O)C(F)C(=O)NCCC1(C)N=N1 3159,N1(C(Cn2ccc(C)n2)=O)CC2(CCOCC2)CC1CNC(=O)C(F)=CCCF 3160,CCC(CC)(CCNC(C1CC1(Cl)Cl)=O)NC(=O)C(O)C1CC1 3161,c1(OC)cccc(-c2cn(C3CN(C(C4(C)CC=CCCC4)=O)CC3O)nn2)c1Cl 3162,C1(C(C2CC2)NC(C2C(C(C)O)C2)=O)CCCN1C(=O)CCN(C)CCO 3163,C1(CC)CC(NC(C2(CNC(=O)CC3CC4CC4C3)CC2)=O)CC(=O)N1 3164,N1(C(COCCCCC)=O)CC(C(=O)NC(C2CCCOC2)(C)C)C(F)(F)C1 3165,N1(CC(c2cc(C)sc2C)CC)CCC2(CCCC2Nc2ccccc2)C1 3166,C1(C(C)NC(c2c(CC)c[nH]n2)=O)CN(C(=O)CCCc2n[nH]c(=N)s2)CCO1 3167,C1(C(=O)NC(C(C)C)CNC(=O)CC2CSC2)CCn2cncc2C1 3168,N1(C(CCNC(=O)NC)=O)CCCN(C(=O)C(C#N)C(C)(C)C)C(C)C1 3169,CC(C)C(O)C(F)(F)C(=O)NCCc1ocnc1CNC(C1Cc2nncn2C1)=O 3170,c1(CCC)ncc(NC(=O)C(CCC2CC2)NC(=O)Cn2cccn2)cn1 3171,c1(OC)cccc2c(CNC(c3nc(C)ccc3Br)c3nnnn3C)cccc12 3172,c1(CC)ncsc1C(=O)NCC1(CNC(=O)CC2CCCC2C)CC1 3173,Cc1cccc2[nH]c(C(N3CCC=C(CNC(C4COC(=O)N4)=O)C3)=O)cc12 3174,c1(CC)cccc(C(=O)NC2(C(=O)NC3(c4ncc[nH]4)CC3)CC2(C)C)n1 3175,C(c1cn(C)nn1)=CC(=O)NC(C(=O)N(CCCC(=O)NC)C)Cc1cc[nH]n1 3176,C(=O)(N=S(C)(=O)c1cccc2cccnc12)c1c(C(=O)OC(C)(C)C)nccc1 3177,C1(CCOC)CN(C(C2CC(C)(O)C2)=O)CCN1C(=O)C=Cc1cnc[nH]1 3178,N1(C(C2C3CCCC(=O)C32)=O)CC2CCCN(C(C34CC(C3)C4)=O)C2C1 3179,c1(NC(=O)NC(C)Cc2cncnc2)nccc2ccncc12 3180,C12(C(=O)NC3CON(CC)C3=O)CCCC1CCN2C(c1csc(F)c1)=O 3181,Cc1cc(C(N2CCC(C)(C#N)C2)C(=O)NC(C)(C)C)cc(Br)c1 3182,N1(C(=O)C2CC2)CCC2CCCC(C1)N2C(c1ccnnc1S)=O.c12ccn(n1)C2 3183,C1(C(=O)NCc2cccc(C(N(C)Cc3cncs3)=O)c2)CCOC(=O)CC1 3184,C#Cc1cncc(C(N2CC(C(C)NC(C3CCS(=O)(=O)C3)=O)C2)=O)c1 3185,n1(CC)nncc1C(=O)NCCC(Cc1ccccc1)NC(C1COC(=O)N1)=O 3186,c1(C(N2C(C)(C(N3CCCC(OCCOC)C3)=O)CC2)=O)ccnc(F)c1Cl 3187,c1(N2CC(CCC)C(CO)C2)cc(S(=O)(=O)Nc2nn(C)cc2Br)ccc1C#N 3188,C1(C(N(C2CCCOC2)C)=O)C2CN(C(c3n[nH]c(=N)[nH]3)=O)CC12 3189,CCC(CCC(=O)N(C1CCN(CC2CC2)C1)C)NC(c1ccnnc1C)=O 3190,c1(C(N(CCNC(C2CC3(CC(C#C)C3)C2)=O)CC)=O)ccc2ncc(=O)[nH]c2c1 3191,c1(OC)cccc2c1CC(C(N1CCOC(CNCc3ccccc3)C1)=O)CO2 3192,C1(C(=O)NC(C)C(C)(C)NC(=O)C=C(C2CC2)C2CC2)CC2CCC(C1)S2 3193,N1(C(c2cnc(SC)s2)=O)CC2CCC(C1)N2C(=O)CN1CCCNC1=O 3194,CCCCCCCCC(=O)N(CC(CC)NC(=O)CC(C)(C)C1CCCCC1)C 3195,C(=O)(C(C)(C)C=O)NCCNC(CCc1cnc(C)o1)=O.C(C)(C)(C)OC(C)=O 3196,N1(C(c2cscn2)=O)CCC2(CCCCN(C(C34CC(C3)C4)=O)C2)C1 3197,N1(C(C(C=C)(F)F)=O)CCCC(CCNC(C2CC3(CSC3)C2)=O)CC1 3198,C1(OC)CN(C(=O)C=C(C)Cl)C(C)(CNC(c2ccc(C3CC3)nc2)=O)C1 3199,Cc1cc(CC(N2CCC(N(C(=O)Cc3ccc(Br)s3)C)C2)=O)c(C)s1 3200,Cc1nc2ccc(C(N3CCCC3CN(C(C3CCCC3)=O)C3CC3)=O)cc2s1 3201,C1(C(=O)NCCC(C)(C)NC(COCC(C)(C)C)=O)CC(S(C)(=O)=O)C1 3202,c1(C(=O)NC(C2CCCN2C(C2CCC(C(F)(F)F)O2)=O)(C)C)cncc(F)c1 3203,C1(C(=O)NC(C)CC(=O)NCCC(O)CO)(Cc2nc[nH]n2)CCOCC1 3204,Cc1cc(CNC(=O)CC2CCN(C(c3ncc(Cl)cc3Cl)=O)CC2)ccc1F 3205,c1(C(=O)NCC2CCCCN(C(=O)Cc3cnco3)C2)cn2cnnc2cn1 3206,C1(C(C)NC(c2ccc(Cl)o2)=O)CCN(Cc2ccn(C)n2)CC1 3207,C1(NC(CNC(C)=O)=O)CCC2CN(C(=O)C(c3ccc(N)cc3)(C)C)CC2C1 3208,C1(C(=O)NCC2CN(C(C3CN(CCOC)C(=O)C3)=O)C2)CC2(C1)CC1(CC1)C2 3209,c1(C2CCN(CC(CC#C)C)CC2)c(C)[nH]c2cc(F)ccc12 3210,c1(C(=O)NC2C3CN(C(C(C=C)(C)CC)=O)C(C3)CC2)ccc2c(c1)CCN2C 3211,C(=O)(NNC(=O)CCc1cccc(Cl)c1)c1ccc(C)cc1 3212,c1(CCC)cc(C(N2CCC(CN3CCC(N)C3)CC2)=O)nn1-c1ccccn1 3213,C1(CC(N2CC3CCC2CC3)=O)C2CCC(C2)N1C(=O)CN1C(=O)CCC1=O 3214,c1(C(=O)NCC(CC)N(C(=O)C(O)c2ccco2)CC)ccnc(C(F)(F)F)c1F 3215,CCCCCCN(C(=O)C=CCNC)CCN(C(=O)CCN1CCC1)C1CCCO1 3216,N1(C(CC=C)=O)CCCC(C)(NC(=O)C(C)OCCOC)C1 3217,N1(C(CSCCC)=O)CCOC2CCN(C(=O)C(C)n3ccnc3)CC12 3218,N#Cc1ccc(C(=O)NCCCNC(c2ccc(-c3cc[nH]n3)s2)=O)o1 3219,c1(C(N(CC(CNC(CCC(=C)Br)=O)O)C)=O)c(C)cccc1Cl 3220,N1(C(c2ccc(Br)cc2Br)=O)CC2CCN(C(c3cccc(F)c3O)=O)C2C1 3221,C=CCC(C)C(=O)N(C)Cc1cccc(CNC(C23CCC2CC3)=O)c1 3222,Cc1oc(S(N)(=O)=O)cc1C(=O)NCC1CCCN(C(C2(C)CNC(=O)C2)=O)C1 3223,CCC(=O)CCC(=O)NCC(=O)NCC(C1CCC1)OC.C1CCCCCC1 3224,CCCC(C(=O)NCCc1cn(Cc2ccc(=O)n(C(C)C)c2)nn1)C(C)C 3225,C(C)(CCCNC(=O)C=CC(N1CCC(C)C1)=O)NC(COCC=C)=O 3226,c1(C(N2CCC(C)(C(=O)NC)C2)C(=O)NCCCSC)ccc(F)c(Cl)c1Cl 3227,c1(C(=O)NC(C(C)NC(C(C)OC)=O)C)ccccc1Oc1ccncc1 3228,C1(c2n(C)cnn2)CCCN(C(=O)CCCNC(=O)OC(C2CCCC2)=O)CC1 3229,CCCCCC(C)CC(=O)NC1CC(N(C)C(c2cocc2C)=O)C1 3230,C1(CNC(C(C)N2CCC2)=O)CN(C)CCN1C(=O)CNC(=O)C(F)(F)F 3231,C1(CCC)(NC(=O)CN2CC(C)(C)C2)CCCN(C(=O)C(C)OC2COC2)C1 3232,C1(C(N2C(C(C)O)COCC2)=O)CCN(C(=O)c2cc(C(C)=O)on2)O1 3233,CCC(C)(C)C(=O)C(=O)N1CCOCC(CNC(=O)CCc2ccc(F)cc2)C1 3234,N1(C(C(C(=O)OCC)F)=O)CCC(CNC(C2(O)CC2)=O)C(F)(F)C1 3235,C1(C(=O)NCCCOC)(CNC(C2CN(C(=O)C(C)OC)C2)=O)CCCC1 3236,N1(C(CCCC#C)=O)CCC2CCN(C(c3cn(C)c(C)n3)=O)CC12 3237,N1(C(C2C(C(C)C)C2)=O)CCC(C2CCN(C(c3cc4sccc4[nH]3)=O)C2)CC1 3238,c1(C(=O)NC2CCN(C(C3C(C=C)C3)=O)C2)cc(OC)cc(NC(C)=O)c1 3239,c1(SC(C)C(=O)NC2CC(CNC(=O)CCc3cncn3C)C2)cccnc1 3240,N1(C(CCC(C)CN(C)C)=O)CC2CN(C(=O)C=CC3(C)CCOCC3)CC2C1 3241,c1(S)ccccc1Cl.C1(C(=O)NC(C(C)NC(=O)COC)CO)CCC12CCC2 3242,CC(C(C)C(=O)NC1(C(O)CO)CCC1)NC(=O)CSC(F)(F)F 3243,N1(C(C2C3COCC23)=O)CC2CCN(S(=O)(=O)c3ccccn3)C2C1 3244,CN1C(=O)CC(C(=O)NCC=CCNC(=O)CCC(N)=O)C1c1cccnc1 3245,CC(C)(C)C(O)CC(=O)N1CC2CC2(CNC(c2cc(F)c[nH]2)=O)C1 3246,c1(C(N2CCN(C(C3CCCN(C)C3)=O)CC2CC#N)=O)ccc(C#N)c(Cl)c1 3247,O=C(CC1=CCCCC1)NCC1CC2(CO1)CN(C(C1CC(F)C1)=O)C2 3248,C(CO)(CCCCNC(c1nnc(C)n1C)=O)NC(C(CC)CC1CCCC1)=O 3249,c1(C(N2CCC(CN(C)C(C3CCCC(=O)N3)=O)C2)=O)cccc(C(C)(F)F)n1 3250,N1(C(C(C)OCCC(C)C)=O)CC2CCC(C1)N2C(=O)CC(F)(F)F 3251,c1(C(N2CCC(CCC(=O)NCC(=O)NCC)C2)=O)c(C#N)ncn1C 3252,C1(C(=O)NCC(CN(C(=O)C(=O)NCC#N)C)(C)C)(CF)CCOCC1 3253,C=C(C)CC(C(=O)NCCC1CC(C)C1)NC(C1CN(C2CC2)C1)=O 3254,N#CC1(C(N2CC3CC2CN3C(=O)C=CBr)=O)CCOCC1 3255,c1(N2CC(NC(=O)C(F)F)C2)cc(Cc2cccc(F)n2)ncn1 3256,C(=O)(C(CCOC)NC(C1(C)CC(C#N)C1)=O)NCCCOCCOC 3257,C(=O)(C(CCCC)N(C)C)N1CCC(C(CNC(CCC=CC=C)=O)C)CC1 3258,c1(C(N2CC(C)N(C(c3cccc4[nH]ccc34)=O)CC2)=O)c[nH]c2cnccc12 3259,N1(C(c2cc(C)oc2)=O)CCN(C(=O)C(n2nc(C)cc2C)C)CC(C)C1 3260,C1(C)(C(=O)NCC2(NC(C(N3CCC(O)CC3)C)=O)CCCC2)COCCO1 3261,c1(C(N(c2ncnc(OC)c2C)C2CNCC2F)=O)cc(Cl)c(Br)cc1Cl 3262,CC1(C)CCc2cc(C(N3CCN(C(=O)Cc4nc[nH]n4)C4CC34)=O)ccc2O1 3263,c1(OC)ccc(-c2cn(CCNC(=O)C(C)(c3cccs3)C3CC3)nn2)nc1 3264,c1(CCC(N2CCN(CCNC(CC3(C)CC3)=O)CC2)=O)c(F)cccc1Cl 3265,C1(C(N(CCC(=O)NC2C=CCCC2)CC#C)=O)CCCC(=O)CC1 3266,C(=O)(C1=NOC2(CCN(Cc3csc([N+](=O)[O-])c3)C2)C1)Nc1cc(C(C)C)no1 3267,c1(C(=O)NC2(C)CCN(C(c3c(C)onc3C(F)(F)F)=O)C2)cn2c(n1)CCC2 3268,CC1Cc2cc(C(N3CCN(C(=O)CC(C)(C)C(F)(F)F)CC3C)=O)ccc2O1 3269,N1(C(C(C(C)C)O)=O)CCC2CN(C(c3cnc4cc[nH]c4c3)=O)C(C)C12 3270,CC1COC(C(=O)N(CC(C)(C)NC(c2cccc(CCO)c2)=O)C)CO1 3271,c1(CC)c[nH]c(C(=O)N(C2CC(NC(=O)CCc3nnc(C4CCC4)o3)C2)C)c1 3272,C1(OCC)COCCC1CC(=O)N(CC(O)CN(C)C1CC1)C.N12CCC(CC1)C2 3273,c1(NCCN(C(=O)CSCC(N)=O)CC)c(C#N)cnc2c(F)cc(F)cc12 3274,C1(C(N2CC3(N(C(C(=C)F)=O)CC3)C2)=O)Cc2ccccc2C1 3275,Cc1[nH]c2ccc(C(=O)NCC(C(C)C)NC(=O)C(C)(C)C3CCC3)cc2c1C 3276,N1(C(C2=CC(C)(C)C2)=O)CCC2CN(C(c3ccc4c(c3)CCOC4)=O)CC2C1 3277,C1(C(=O)NC(c2ccccc2)CC)CC2CCC1C(=O)C2 3278,N1(C(C2(C)CC3C=CC2C3)=O)CC2(CC(NC(c3cc([N+](=O)[O-])n[nH]3)=O)CO2)C1 3279,C1(CC=C)(C(=O)NCC[Si](C)(C)C)CN(C(=O)C(O)c2ccco2)C1 3280,Cc1cc(C(=O)NC(c2nccs2)C)c(C)n1N 3281,C1(CC(=O)NCC2C(C(=O)NCCc3onc(C)n3)C2)C(C)(C)C1(C)C 3282,c1(OCC2CCCN(C(=O)OC(C)(C)C)C2)cc2cc(F)ccc2oc1=O 3283,CN(C)S(=O)(=O)N1CCC(C(=O)NC(C(=O)Nc2ccc(CO)c(F)c2)=O)CC1 3284,c1(OCCF)ccc(-n2nc(CC3CC3)nc2-c2cnn(C3CCCCC3)c2)cc1 3285,c1(C(N2CCN(C(c3c(C)ccc(Br)c3)=O)CC2)=O)cncc2c(Cl)cccc12 3286,C(=O)(CC(C)C(=O)OC)N(C(C(=O)NC1(COC)CCC1)C)C1CC1 3287,Cc1cncc(C(=O)NCC(C)(C)CNC(C2NC(=O)OC2C)=O)c1 3288,C=CC(C)(CC)C(=O)NCC(C)CNC(c1cn2ccnc2s1)=O 3289,C(=O)(CC(C)CCC=C(C)C)NC1(CCOC)CN(C(C2CCCC(C)O2)=O)C1 3290,CN1CCOCC(NC(C2(NC(=O)C(O)CC(N)=O)CSC2)=O)C1 3291,c1(CNC(c2ccco2)=O)nc(N(C)CCOCC(=O)OC)cc(Cl)n1.CCO 3292,CC#CCC(C(=O)N1CCC(N(C)C)CC1)NC(=O)CC1COC(=O)C1 3293,Cc1ccccc1C1(C(N2CCC(C3(NC(=O)CCOC4COC4)CC3)C2)=O)CC1 3294,c1(C(=O)NCC(COC)NC(c2nccc(C)n2)=O)cnc2ccsc2c1 3295,c1(C(N(CC(CC)NC(=O)C(c2cccc(C)c2)C)C)=O)cncc(F)c1C 3296,C(=O)(CS(=O)C(F)(F)F)N1C(CNC(CCc2onc(CCC)n2)=O)CC1 3297,C12(C(=O)NCC(CNC(c3ccccc3C3CCC3)=O)F)CC1CCC2(F)F 3298,C#Cc1ccnc(C(=O)N(CC(C)NC(=O)C(N2CCNC2=O)C)C)c1 3299,c1(CC)cc(C(=O)NC2CCC(N(C)C(c3ccnnc3)=O)C2)cc(F)c1 3300,C1(CC)CC(CC(=O)NC2CC(CNC(=O)CC(C)(F)F)C2)CCO1 3301,c1(CC)cccc(C(=O)NCCOC2CN(C(=O)CC(C)NC3CCCC3)C2)c1 3302,c1(NCC(CCCC)NC(c2cnc(C)s2)=O)cc(=O)n2cc(Cl)ccc2n1 3303,C1(C(=O)OC)(C(=O)OC(c2cc(F)c(OC)cc2N)=O)CC2C(C1)C2(F)F 3304,Cc1ccc(NC(=O)C(N2CCC(C(C)(C)C)CC2)=O)cc1C.N1(C)CCOCC1 3305,N1(C(CSSC)=O)CC(CCNC(c2ccc(CO)s2)=O)OC(C)C1 3306,c1(OC)csc(C(=O)N(CC(O)CNC(=O)Cn2cc(CN(C)C)nn2)C)c1 3307,n1(C(CC)C)ncc(C(=O)OC2CCC2)c1C 3308,N1(C(c2c(OC)c(Cl)ccc2)=O)CCC2(CCN(C(=O)CCNS(C)(=O)=O)C2)C1 3309,C(=O)(C(C)P(C)(C)=O)NCc1c(CCNC(CCNC(CC(C)C)=O)=O)ocn1 3310,N1(C(c2c(C)nsc2)=O)CC(NC(=O)Cc2cc(C3CC3)no2)C(C(F)F)C1 3311,N1(C(c2c(C)scn2)=O)CC2CCOCC2(NC(c2ccc3sccc3c2)=O)C1 3312,N1(c2nc(N3CCC(F)(CO)CC3)nc(OC)n2)CCC2(CC1)CC(CO)CO2 3313,C1(C(=O)OC)C(C(N2CCC(NC(=O)Cc3cscn3)C2)=O)C1(F)F 3314,C(CCN=C(NCC1CC(=O)N(C2CC2)C1)NC1CCSC1)OC 3315,C12(C(=O)NC(C)C(C)n3cccn3)CC1CN(C(=O)C(C)(C)C1CCOC1)C2 3316,C(=O)(C(C)(C)C(C)(C)C)N1CC(N(C)C(c2cnc(Cl)[nH]2)=O)C(F)C1 3317,C(=O)(C(C)S(=O)Cc1cccs1)N(C(c1ccc(Cc2ccccc2)cc1)C)C 3318,C12(C(=O)NC3CCCN(C(C(C)C4CCCC4)=O)CC3)CC(C)(C1)OC21CCC1 3319,c1(OCC(=O)NCC2C(NC(c3c(C)nc(O)[nH]3)=O)C2)cccc(C)c1F 3320,c1(C(=O)NCC2C=CC(NC(C=C(C)Cl)=O)C2)cc(F)c(F)cc1Cl 3321,CC1CC(NC(=O)CCN(C(=O)C2=CCCCC2)CC2CC2)CCC1(C)C 3322,C1(O)(C(C)NC(=O)CCC2CCC(O)CC2)CCN(C(c2ccon2)=O)CC1 3323,C1(C)(C(N(CC(CC)(C)OC)C)=O)CCN(C(=O)Cc2cnccc2C)C1 3324,n1(COC)ccc(C(=O)N(C)CCN(C)C(c2ccn(C(C)C)n2)=O)n1 3325,c1(C(=O)NC(CNC(Cc2nc(CC)sc2)=O)C)c(-c2ccccc2)noc1C 3326,c1(C(N2CCCC(C)(CNC(C3C(C)C3)=O)C2)=O)cc(F)cc2cnccc12 3327,N1(C(CC2N(C)C(=O)CC2)=O)CCC2(CC1)CC2NC(C1(c2cc[nH]n2)CC1)=O 3328,C1(C(=O)NCCC2(O)CCCC2)CCCN(C(c2ccn(CCNC3CC3)n2)=O)C1 3329,c1(C(C(=O)N(C)CCF)NC(CC(=O)OC)=O)c(C)cccc1Br 3330,Nc1cccnc1C(N1CCC(CF)(NC(C2CC3CCC3C2)=O)C1)=O 3331,C1(C(=O)NC(CCN(C(Cc2ccc(COC)cc2)=O)C)C)CC2(CCCO2)C1 3332,c1(CC(=O)NCC2CCCCN2C(=O)OC(C)(C)C)cc(F)cc(F)c1Br 3333,Cc1cccc(C(N2CCC(C)C2CNC(c2cc(=O)cc[nH]2)=O)=O)c1 3334,C1(NC(c2c(C)cns2)=O)CN(C(C2CC2C)=O)C2(CCC2)C1 3335,C1(C(=O)NCc2n(C)nnc2)CCN(C(c2cccc(Cl)c2)=O)CC1(C)C 3336,C1(NC(C2CC(=C)C2)C)CCC(OCC)CC1 3337,c1(C(N2CCN(C(C=C(C)C)=O)CC2c2ccccn2)=O)ccc2c(c1)CCC2 3338,c1(C(N2C(C(N3CC(C(=O)OC)C3)=O)CCC2C2CC2)=O)ccc(N)c(Cl)n1 3339,C1(CC)CN(C(c2ccsc2SC)=O)CCN1C(=O)C(C)CSC 3340,c12cc(on1)NC(=O)C(=O)N2.C(=O)(C(C)(C1CCC1)C1CC1)OC 3341,Cc1oc2ccccc2c1C(=O)NCC1CCCC1NC(c1cc(O)nn1C)=O 3342,N1(C(C2=CC(C)(C)C2)=O)C2CCC1CC(NC(C1(N3CCOCC3)CCC1)=O)C2 3343,c1(C(N2CCC(C)(CNC(C3CCC(C)C3)=O)C2)=O)n[nH]c2cccnc12 3344,N1(N(C(CC)C)C)CCC(=O)N(CC(c2cccc(F)c2)C)C1=O 3345,C(=O)(C(CNC(=O)Cc1nccn1C)C(C)(C)C)N(C)Cc1ccccn1 3346,CC(N=c1[nH]c(N(C)Cc2cnn(C3CC3)c2)nc2c1CCC2)c1csc(Br)c1 3347,c1(C(N(C(C)CCNC(=O)CN2CC3CCC2C3)C)=O)ccc(F)c(N)c1 3348,c1(OC)cc(O)ncc1C(=O)NCCC1(O)CN(C(c2ccc(N)c(N)n2)=O)C1 3349,c1(OC(c2oc(CC)c(C)c2)=O)cc(C2CC2)cc(F)c1 3350,N1(C(C2CC2(Br)Br)=O)CC2(NC(=O)NCc3ccccc3)CC1(C)C2 3351,c1(NC(=O)NCCCC2(NC(CC3(C)CC3)=O)CC2)ccccn1 3352,C1(C(c2n(CCOC)nnn2)NCCCC2CCOCC2OC)CCC(F)(F)CC1 3353,c1(C(=O)NC2C(NC(C3(COC)CCCC3)=O)CCC2)cc2scc(Cl)c2[nH]1 3354,N1(C(c2c(C)scn2)=O)CCCC(C)(C)C1C(N1CCCC(O)C1)=O 3355,c1(-n2cc(CC(=O)OCC)nn2)ccnc(NC(C2CN3CCC2C3)=O)c1 3356,C=C1CC2(C1)CC(C(N1CCN(C(C34C5C6C7C5C3C7C46)=O)C(C3CCC3)C1)=O)C2 3357,C1(CNC(C(c2ccc(OC)cc2)(C)C)=O)CC2COCC2N1C(=O)CC1CC1 3358,CC1(C(=O)NCCC2CCN(C(=O)C(C3CCCCC3)F)C2)CCS(=O)(=O)CC1 3359,C1(O)(CC(=O)NCCC(C)N(C(=O)CCN(C)CCO)C)CCOC1 3360,CC1CC(CCNC(c2csc(C(C)(C)C)n2)=O)CCN1C(=O)Cc1cncs1 3361,Cc1c(-c2cn(CC3CC4(CC4)CN3C(=O)CCC(C)C#N)nn2)cccc1Cl 3362,C1(C(=O)NCCC2CC(NC(c3noc(CC)c3C)=O)C2)CCc2n[nH]cc2C1 3363,N#Cc1c[nH]c(C(N2CC3CC3(NC(c3cc(-c4ccccc4)cs3)=O)C2)=O)c1 3364,CC(C(=O)N1CC(N(C(=O)CNC(=O)C2CC2)C)C1)SC(F)(F)F 3365,C12(CNC(COCC=C)=O)CCC(NC(=O)CCC3CCCCC3)(CC1)CO2 3366,c1(CC(N2CC(C(C)NC(C3COC4CC3C4)=O)C2)=O)cccc(C#N)c1 3367,N1(C(C(CC(C)C)=O)=O)CC2C=CC1C(C(=O)N(C1(C)CC1)C)C2 3368,C=CC(CC)CC(=O)NC(C1CN(C(c2nnc(C(C)C)s2)=O)CCO1)C 3369,C12(CNC(c3cn(CCC)nc3)=O)CC1CN(C(c1sccc1Br)=O)C2 3370,N1(C(c2nc(C)[nH]n2)=O)CC(N(C)C(c2ccc(C(C)(F)F)nc2)=O)C(C)(C)C1 3371,N1(CC=C(CC)CC)CCC(CN(Cn2cc(CC3CCCO3)nn2)CC)CC1 3372,CN1CC=C(C(=O)NCC(C2CCOC2)NC(=O)CC23CCCN2CCC3)C1 3373,c1(CN2CC(C(F)(F)F)(C3CC3)C2)cnn2c1OCC2 3374,C(c1cccc(Cl)c1)=CC(N1CCC(C(C)NC(C(C)(C)OC)=O)C1)=O 3375,CCCCC(CC)(c1nnnn1CC(F)F)NCCS(=O)(=O)NCC1CC1 3376,C1(NC(c2ccc(C(O)CF)cc2)=O)CCN(C(c2cnsc2)=O)CCC1(F)F 3377,N1(C(C=C(C)C(=O)O)=O)CCC(N2CCCC2C(=O)NCC(C)CN)CC1 3378,N1(C(c2ccnc(C)n2)=O)CCN(C)C(C(=O)NC(c2nccc(OC)n2)C)C1 3379,c1(N2C(C)C(NC(=O)CN(C3CCCC3)C)CC2)ccc([N+](=O)[O-])cn1 3380,c1(C(N2C(CN(C)Cc3c(C)ccs3)CCCC2)=O)cnc2c(c1)CCCC2 3381,CC1CC2(C(N3CC(NC(c4cccc(NC5CCCC5)c4)=O)C(O)C3)=O)CC12 3382,CC1CCCN(C(C2CCS(=O)CC2)=O)C1CNC(=O)C=Cc1cncn1C 3383,c1(C(=O)NCC2(C)C(C)CN(C(C(CCSC)O)=O)C2)cc(Cl)c(Cl)cc1N 3384,C1(CNC(CCSCCC)=O)C(C)CCCN1C(c1cc(C2(C)CC2)on1)=O 3385,C(=O)(C1=CC2CCCCCC12)OCC(C(CC)(C)C)=O 3386,c1(C(N2CC(OCC)(CNC(=O)CCc3cc(C)no3)C2)=O)cn(C)nc1CC 3387,N1(C(C2(C)CC(=C)C2)=O)CCC(CNC(c2cnn(-c3nccs3)c2)=O)C(O)C1 3388,C1(C(=O)NCCC(=C)CNC(=O)CSC(C)(C)C)CS(=O)(=O)CN1C(=O)OC 3389,N1(C(=O)OC2CCCCC2)CC=CCC1C(N1CC(N2CCCC2=O)C1)=O 3390,CC1CCCN(C(c2ccc(NCC3CC3)nc2)=O)C1CNC(c1ccsc1)=O 3391,C=C(C)C(CC(=O)NCC(CCOC)NC(=O)Cc1csc(CC)n1)OCC 3392,C1(NC(=O)COc2cccnc2)COCCC1NC(C1CCC(C(F)F)CC1)=O 3393,c1(C(=O)Nc2c(O)ccc(C)c2)c(C)cc(C)c(OC(F)F)c1C 3394,c1(C(N2CCCC2c2cn(C3(C(=O)O)CC3)nn2)=O)cnc(C(F)F)s1 3395,C(=O)(C1=CC2CCCC12)N(C1CCN(C(c2ccc3nncn3c2)=O)C1)CC 3396,C(=O)(CCCCC(=O)OC(C)(C)C)N1CCN(C(C(CC=C)C)=O)CC1COC 3397,CCC(F)(F)C(=O)NCCC1(C(=O)NCC2CC(C)CO2)CCC1 3398,CC1(CNC(=O)Cc2ccc(Cl)s2)CCCN1C(=O)CCc1cocn1 3399,C1(OC)CN(C(c2conc2C(C)C)=O)C(C)(CNC(C2C(C)(C)C2(C)C)=O)C1 3400,C1(C(=O)NCCCC(=C)Cl)CN(C(c2sccc2OC)=O)CC12CC2 3401,c1(CC)cc(F)ccc1CC(N1CCC(F)(CNC(=O)C(O)CCC)CC1)=O 3402,N1(C(C(C)C(F)F)=O)CC(CC(=O)NC2CCC(OCF)CC2)C2(CC2)C1 3403,N1(CC(=O)NC(C)CN2CCN(C(=O)CC3CSC3)CC2)C(=O)NC(C)(C)C1=O 3404,C1(C(N2C(C(=O)NC3CC(C#N)C3)CCCC2)=O)C2CCCC(=O)C12 3405,Cc1nccc(C(=O)NCC23CC(NC(=O)C(C)c4ccsc4)(CO2)C3)c1O 3406,CCCC(CNC(c1cccn1C)=O)C(=O)N(CC)CC1CCCO1 3407,C(=O)(C1=C(C#N)CCC1)N1CCOCC(CNC(Cc2cn(CC)nc2)=O)C1 3408,C1(n2ncc(CC(=O)OC)n2)CCN(C(=O)Nc2cnn(CCO)c2)CC1 3409,N1(C(c2ccc(OC)o2)=O)CC(C)N(C(=O)CCCC#N)CC1C 3410,Cc1cc(=O)ccn1CC(=O)NCCCN(C)C(c1coc(C(F)(F)F)n1)=O 3411,C12(c3cn(C(CC)C)nn3)CC(CN1C(C)=O)C2.C12CCC(CC1)COC2=O 3412,c1(OC)nc(C)ccc1C(N1CCCN(C(C2CC(OC(C)=O)C2)=O)CC1)=O 3413,Cc1cc(S(=O)(=O)NCC(=O)NC2CCCCN(C(=O)CC(C)(F)F)C2)cn1C 3414,C=CCC(CC)C(=O)N1CC2C(CNC(=O)CCSC3CCCC3)C2C1 3415,C1(NC(CC2(OC)CCC2)=O)C2CN(C(C3CCC(N(C)C)CC3)=O)CC12 3416,N1(C(C2C(C(C)C)C2)=O)CCC(OCCCNC(C2(CC#N)COC2)=O)CC1 3417,c1(C(=O)NCC2(OC)CN(C(c3ncoc3C3CCCO3)=O)C2)c(Cl)n[nH]c1C 3418,OC1(CNC(=NCC2CCCSC2)NCC2CCOCC2)CCCCC1 3419,c1(OC)ccc(O)cc1C(N1CC2CC1C2CNC(c1nccn1C(C)C)=O)=O 3420,N1(C(c2c(C)nc(CC)o2)=O)CCN(C(=O)COCC2CCCOC2)C(CO)C1 3421,C(=O)(C1=CCC(C)(C)CC1)N(C1CCN(C(=O)C(O)C(C)OC)CC1)CC 3422,Cc1ncc(NC(C2CCCCN(C(=O)Cc3cccnc3F)C2)=O)cc1C#N 3423,Cc1cc(F)ccc1C(N1CCC(N(CCO)C(C2OCC(=O)N2)=O)C1)=O 3424,N1(C(C(C)(C)NC(N)=O)=O)CC2(C=C(C(=O)NC(C)CC3CC3)CO2)C1 3425,C(CC(=O)NCc1cccc(F)n1)(C(F)(F)F)NC(C(N)=O)=O 3426,Cc1c(F)cc(C(=O)NCC2CC(NC(c3cnn(C)n3)=O)C2)cc1F 3427,c1(CNC(COC(C(C)(C)c2cccnc2)=O)=O)ccc2c(c1)OCCO2 3428,C(CO)(CCCCNC(c1csc(CO)n1)=O)NC(CN1C(C)CC1)=O 3429,CCCCCCCC(=O)N1CCCC(CNC(c2cccc(Cl)c2F)=O)C1 3430,C1(C(N(CCCN(C)CCn2cnccc2=O)C)=O)CN2CCN1CC2 3431,C1(C(=O)NCC=CC(=O)N(CC(COCC)O)C)CCC(C)O1 3432,C1(NC(CCC2N(C(COCC#C)=O)CCC2)=O)CC2C(C1)C2(F)F 3433,CC(C)(CNC(C1CC(F)CN1C(=O)C(O)CC1CCCC1)=O)CCCO 3434,c1(C(=O)NCC(C2CCOC2)NC(C2=NNC(=O)C2)=O)cc(=O)n2nccc2[nH]1 3435,c1(C(N(CCCCN(C(=O)CCc2cocn2)C)C)=O)cc2[nH]ccc2s1 3436,N1(C(c2c(C)nns2)=O)CCN(C(=O)C=C2CCC2)C(C2CCCC2)C1 3437,CCCC(C(=O)N(C)CC1(O)CN(C(c2ccc(F)cn2)=O)C1)OC 3438,C1(C(N2C(CNC(C(C)S(N)(=O)=O)=O)COCC2)=O)CCC2(CCC2)CC1 3439,c1(CC)ccc(OCC(N2CCC(OCCNC(c3cccs3)=O)C2)=O)cc1 3440,C1(C(=O)NC(COCC)C(=O)N2CCC(O)C2)C2CN(C)CC12 3441,CC1(CNC(C2CCC3CC23)=O)CCN(C(=O)CCc2ccon2)CC1 3442,C=CCCCC(C(=O)NC(c1cn(C)nn1)C)NC(=O)C=Cc1cc[nH]n1 3443,Cc1nn(C2CCOC2)cc1C(N1CCCC(NC(C23CCC(C2)C3)=O)C1)=O 3444,C(CNC(C1CCN(CC(C)C)CC1)=O)(C(C)C(C)C)NC(c1cc(C)ns1)=O 3445,C1(NC(C(CC#C)(C)C)=O)CN(C(=O)C(C(C)(C)C)C2CCC2)CCC1(C)C 3446,C1(CC)CN(C(C2C(C)(C)C2(C)C)=O)CCN1C(c1cc(OC)ccn1)=O 3447,C1(C(=O)NC2(C3N(C(c4c(CC)ncnc4)=O)CCC3)CC2)CCc2n[nH]cc2C1 3448,N1(C(c2cc(C)[nH]c2)=O)CC(C)OC2(CCN(C(c3ncccc3F)=O)CC2)C1 3449,N1(C(C(C(=O)NC)(C)C)=O)CCC2(CCN(C(=O)COC3(C)CCC3)C2)C1 3450,C1(C(N2CC(O)(CNC(C(C)CC(F)F)=O)C2)=O)CCCC(F)(F)CC1 3451,c1(OC)c(C(=O)OCC(=O)OC2CCC(=O)N(CC(F)(F)F)C2)cc(I)cc1F 3452,Cc1nc(C)c(C(=O)NCC2(CNC(=O)CCC(=O)N(C)C)CCOCC2)[nH]1 3453,N1(CC#CC)CCN(C(=O)C(CC2CC2)NC(C2CNC(=O)C2)C2CC2)CC1 3454,CN1CCCC(C)(C(=O)NCC(O)CC(=O)NCC2OCCCC2(C)C)C1 3455,N12CC(O)CC1CNC(=O)NCCNC(=O)C2=O.C(C1=CCCC1)=C.C(C)(C)(C)OCC 3456,c1(OC)cccc(COCC(=O)NC2CC(CNC(=O)COC(F)F)C2(C)C)c1 3457,c1(C(N2CCC(C)(CNC(C3C(C)(C)C3)=O)C2)=O)cnc(O)nc1O 3458,N12Cc3ccc(nc3C1)NC(=O)CC(=O)N(CCC)CCCC2.C(C)(C)(C)OC 3459,CC1CN(C(C(=O)OC)=O)CC1C(N1CCC(CN(C)C)C1)=O.C1(CC=O)CC1 3460,CC1CN(C(c2cnncc2Cl)=O)CCCN1C(c1ccc(C(F)(F)F)nc1)=O 3461,N1(C2C(=O)NC2)CCOC(CC(N)=O)C1.c1(CC)nocc1CC 3462,c1(C(N(CC(=O)N(CCCF)C)C(C)C)=O)cnc(C)s1.N(C)CCO 3463,N1(C(CCCc2onc(C)n2)=O)CC2(CCN(C(=O)CN(C)C)CC2)C1 3464,C1(C(N2CCCC2CN(C)C(c2nsnc2O)=O)=O)(OC)CCSC1 3465,S(=O)(=O)(c1cc(NC2CC2C2CC2)nc(Cl)c1)NCc1cc(OC)cc(OC)c1 3466,Cc1nn(C)c(C(=O)NCc2cc(O)nc(CNC(=O)C(C)O)n2)c1Cl 3467,C(=O)(C(C)(C)CC(C)C)N1CC(C)(C(=O)NC2(C(=O)OC)CCCC2)C(C)C1 3468,C1(CCC=C)(C(=O)NCc2cc(COC)on2)CN(C(=O)CCc2cnc[nH]2)C1 3469,C1(NC(C2CC(C)(C)C2)=O)CCC2(CC1)CC2NC(c1cncc(O)c1)=O 3470,c1(C(N(C2CCN(C(=O)Cn3ncn(C)c3=O)C2)C)=O)cnc2c[nH]nc2c1 3471,C1(C#CC(=O)N2CC(c3ocnc3CNC(C3CCC(=O)N3C)=O)C2)(CC)CC1 3472,c1(C(N(CCNC(C(CC)(C)CO)=O)C)=O)cnn2c(C)cccc12 3473,CN1CC=C(C(=O)N(C)CC2CCCN2C(=O)Cc2cncn2C)C1 3474,N1(C(CCCC(=O)NCC)=O)CCN(C(=O)CC2CCCNC2=O)CC12CCC2 3475,C1C(CCC)C(=O)N1.C(=O)(C(F)(F)CF)N1CCC(CNC(=O)OC(C)(C)C)C1 3476,N1(C(C2C(NC(C3CCCC3F)=O)CCOC2)=O)C2C=CCC1CCC2 3477,C(=O)(CS(C)(=O)=O)NCC(C)(C1CC1)NC(CCC=C)=O 3478,Cc1cc(C(N2CCCC2CCNC(=O)CCc2cc[nH]n2)=O)cc(C)c1F 3479,c1(C2OCCN(C(C3C(NC(=O)Cc4ccc(F)cc4)C3)=O)C2)cc(F)cc(Cl)c1 3480,C1(C(N2CC(O)CC(NC(c3c(C)cccc3N)=O)C2)=O)CC2C=CC1C21CC1 3481,c1(OCC)cc(NC2CN(C(C3CCC(OC)CC3)=O)CC2C)nc(C)n1 3482,c1(C(N2C(C(=O)OC)CSCC2)=O)cc2c(C)snc2s1.c12ncc(s1)c(=O)[nH]2 3483,Cc1cnc(C(C)NC(C2CCN(C(=O)Cc3cccs3)C2)=O)nc1 3484,CC1OC(=O)NC1C(N1CC(O)(C(C)(C)CNC(=O)Cn2cnc(C#N)n2)C1)=O 3485,Cc1ccc(-c2nc(CC(N3CC(n4cc(C5CCCC5O)nn4)C3)=O)cs2)o1 3486,c1(CC(=O)NC(CC)CN(C)C(C2CCC(=O)N2)=O)ccc(C2CC2)cc1 3487,N1(C(c2cc(C)nnc2O)=O)CC(C)(CNC(c2csc(Cl)n2)=O)CC1(C)C 3488,CC(C)CC(Cn1cc(-c2cccs2)nn1)NC(C1CC1c1ccccc1)=O 3489,N(C1CCc2ccccc21)(CC(=O)N(C1CC1)CC)C(=O)CN(CCOC)C.CCC 3490,C1(C(C)C)C(NC(C2CC2c2ccn(C)c2)=O)CCN1C(c1cc(Cl)ccn1)=O 3491,CC1CN(C(=O)CSCCC#N)CCC1CNC(=O)Cn1ccccc1=O 3492,N1(C(C2CC(OC)C2)=O)CCC2(CC(NC(=O)CCc3ccnc(Cl)c3)CO2)C1 3493,N1(CC)CCOCC1CC(=O)NC(c1csnn1)CNC(=O)CN(C)C(C)=O 3494,c1(CN(C)C(=O)NC2CC(O)C2)cc2cc(Br)ccc2o1 3495,c1(C2C(C(N3CCC(C(=O)NCC(C)(C)C#N)C3)=O)C2)ccc(C#N)cc1 3496,N1(C(CC(C)SC)=O)CC2(CC(NC(=O)CC34CCCC3C4)C2)C1.C(=O)O 3497,c1(COC)ccc(C(N2CC(Nc3ncc(Br)c(C)n3)CC2C)=O)cc1F 3498,C(CC1=CCN(Cc2ncc(C(C)(C)C)o2)CC1)NC(=O)CCC1CCCCO1 3499,c1(OC)ncnc(OC)c1CC(C)NC(CCC(C)SC(C)C)=O 3500,c1(C(=O)NCC2C(C)CN(C(C34CC5CC3C4C5)=O)CC2)ccn2ccnc2c1 3501,N1(C(N2CCC3C(CCN3Cc3ccccc3)C2)=O)CC(C(=O)O)c2ccccc21 3502,N1(C(C(CCC)=CCC)=O)CCCCC(NC(=O)C(C)N2CC(C)C2)C1 3503,C(CCCC(C)NC(C1CCCSC1)=O)NC(c1ccn(CCC)n1)=O 3504,N1(C(=O)OC(C)(C)C)CC(NCc2coc(C3CCCCC3)n2)C2(CCC2)C1 3505,c1(C(=O)NC(C)CCNC(=O)C(C)OCCN(C)C)cc(Cl)ccc1Cl 3506,C#Cc1cccc(C(=O)NCC2CC(C)N(C(c3cc(Cl)n(C)n3)=O)C2)c1C 3507,c1(C(=O)NC2CC(C)CN(C(C3(O)CCOC3)=O)C2)ccc(S(N)(=O)=O)c(F)c1 3508,Cc1cc(C(N2CC3CC(NC(c4c(C)noc4C)=O)C3C2)=O)cc(O)n1 3509,c1(C2(C)CC2)nc(Cl)cc(=NCC2(C)CCC(NC(C3C=CCCC3)=O)CC2)[nH]1 3510,C1(C(=O)NC(CCC)COC)(COC)C=CCN1C(c1nnsc1C)=O 3511,N1(C(C(C)(C)CF)=O)CCC(CNC(=O)C(c2ccc(F)cn2)(F)F)C(F)(F)C1 3512,C1(C(=O)NCC2CC(NC(C(c3nccc(C)c3)(C)C)=O)C2)CCCS(=O)(=O)C1 3513,Cc1nc2n(n1)CC(C(=O)N(CC(c1ccccc1)C1CCC1)C)CC2 3514,N1(C(CCC=C=C)=O)CCN(C)C(C(N2CC3CCC3(C)C2)=O)C1 3515,C(=O)(C(CCCC=C)NC(=O)C(C1C=NN(C)C1=O)C1CC1)N1C(C#C)CC1 3516,c1(C(=O)NCC(C2CCN(c3snc(SC)n3)CC2)(C)C)cc(C#N)ccc1Cl 3517,c1(C(N2CCCC(N(C(C(CCC)C)=O)CC)C2)=O)c(C)nc(C)n1O 3518,C(CC(=O)NCCC(O)C(F)(F)F)(C(F)(F)F)NC(C(C)c1ccsc1)=O 3519,c1(C(N(CCC(N2C(C)CC2(C)C)=O)CC#C)=O)cc(C#N)n(C)n1 3520,C1(NC(C(c2ccc(OC)cc2C)C)=O)CN(C(=O)C(N)=O)C2(CCCC2)C1 3521,N(C(=NCCc1nnc(C)s1)NCC(c1ccccc1)C)CC(C=C)C 3522,c1(C(=O)OCC=C(Cl)Cl)ccc(C(F)(F)CF)cc1 3523,C1(C(=O)NCCNC(=O)Nc2cccc(N3CCOCC3=O)c2)CCCS1(=O)=O 3524,C(=O)(C1=CCCOCC1)NCC(C(N1CCCC[Si](C)(C)C1)=O)CC1CC1 3525,Cc1cc(C(=O)NC2CC(CNC(c3[nH]cnc3C)=O)CC2O)nnc1O 3526,C1(OC)CN(C(=O)C(F)=C(C)C)CC1C(=O)NC1CC(c2ncc[nH]2)C1 3527,C1(N(C(C)C)C(=O)NCC(C2CCCO2)O)CCN(C)CC1 3528,C#CCC(C(=O)N1CCC(C(F)C(=O)Nc2ccccc2OCC)C1)C1CC1 3529,Cc1cc(C(=O)NC2CCN(C(c3cn(C)nn3)=O)CC2C)ccc1Cl 3530,C(CNC(=O)OC(C)(C)C)(C(=O)N1CCCC1C1CC1)OC(F)F 3531,S(=O)(=O)(c1cccc(N(C(C)COC)C)n1)NCC(CCC)O 3532,c1(C(=O)OC)cc(NC(=O)NC(c2cccc(OC(F)F)c2)C)ccc1F 3533,N1(c2nccc(C(C)(C)C)n2)CC(CNC(=O)CN2CC=CC2)OC2(CCC2)C1 3534,C(C(N)=O)(C(C)(C)C)NC(=O)NCc1cc(C)c(Br)s1 3535,N1(C(C(C=C)O)=O)CCC2(CCC(NC(c3cc(C)c4[nH]nnc4c3)=O)CC2)C1 3536,n1(CCC)cccc1C(=O)NCC=CC.C1(C(N2CC(CO)(C)C2)=O)CCCS1(=O)=O 3537,N1(C(=O)Cc2ccc(Cl)c(C(F)(F)F)c2)CCc2ccc(Br)cc2CC1 3538,c1(CN(C2(CSc3ccccc3)CC(F)(F)C2)C)cn2ccccc2n1 3539,c1(C(N2C(CCC(=O)NC(CC=C)C3CC3)CCC2)=O)ccc([N+](=O)[O-])[nH]1 3540,C(=O)(C1=NN2CCCN=C2N1)N(C(C)CNC(=O)C=CC=C(Cl)Cl)C 3541,C1(CNC(=O)CNC(=O)Cn2cccc2)C2CN(C(=O)CCn3cnnn3)CC12 3542,c1(OC)ccc2c(C)c(C(=O)NC3CCC4(CC3)CC4)[nH]c2c1 3543,c1(C(N(CC(CN(C(=O)Cc2cnoc2)C)O)C)=O)ccn(CCF)n1 3544,C1(F)(CNC(c2nc(CC)oc2C)=O)CCCN(C(c2cc[nH]c(=N)n2)=O)C1 3545,N1(C(C(n2ccc(C(F)(F)F)n2)C)=O)CCCC2CCN(C(=O)C3=COCC3)CC12 3546,C=Cn1nncc1C(=O)NC1(CN2CCN(C(=O)C(C)O)CC2)CC1 3547,c1(CCCN(C)C(C2CC2(C)C)=O)cn(CCN(C)C)nn1 3548,S(=O)(=O)(c1c[nH]ccc1=NC(CSc1nccs1)CO)NCc1cccc(C)n1 3549,Cc1ccsc1CCCC(=O)NCCOCCNC(=O)C(C)C1(O)CCC1 3550,c1(C(=O)NC(CC)CNC(c2cc(C)no2)=O)c(Cl)ccc(Cl)c1OC 3551,C1(CNC(CCCCC=C)=O)CN(C(=O)C(F)(F)C(O)CC)CCC1(C)C 3552,C(=O)(C(C)(CC)C(N)=O)N1CCC(CC=C)(NC(C2CC(=O)NC(=O)N2)=O)C1 3553,CCS(=O)(=O)CC(=O)NC(C)C(C)NC(c1ccoc1C1CCC1)=O 3554,C(=O)(C1CNC1=O)N(C)C.C1(CNC(=O)OC(C)(C)C)CNC(=O)C1 3555,C1(C(=O)NCC(=O)OCCCC)(CO)CCN(C(c2cnn(C)c2N)=O)C1 3556,C1(C(=O)NC(C(=O)N2CC(OCCCCC)C2)CO)COCCN1CC 3557,c1(C(N(CCOC2CN(C(C3C(C#N)C3)=O)C2)C2CC2)=O)ccc2occc2n1 3558,N1(C(CC(C)(F)F)=O)CC2(CCC(NC(=O)CC3NC(=O)NC3=O)CC2)C1 3559,C1(C)(CNC(CNC(=O)OC(C)(C)C)C2CC2)CC2(C1)CC(F)(F)C2 3560,C1(C(=O)NC(CCNC(C(C(C)(C)C)O)=O)(C)C)CC(O)c2ccccc2O1 3561,C(=O)(C1CCc2nccn21)NC(C(=O)NCC)CC1CCOCC1.N12CC(C1)C2 3562,CC1=C(C(=O)NC2CCC2NC(=O)Cn2cncn2)CCS1(=O)=O 3563,N1(C(CC2CCC(NC(C3(SC)CC3)=O)CC2)=O)CCN2C(=O)OCC2C1 3564,c1(C(N2CCN(C(C(c3scc(C)n3)C)=O)CC2C)=O)nn(C)c2c1CCC2 3565,c1(CC)nc(O)c(C(=O)N(C)CCN(C)C(c2oc(Br)nc2C)=O)cc1C 3566,C(CC(F)(F)Cn1cc(CC(C)O)nn1)OC(C(C)C)C#N 3567,C1(NC(CC2(OC)CCC2)=O)CCN(C(C2(OC(C)=O)COC2)=O)C1.C(C)(C)(C)O 3568,CCC(CN(C)C)CC(=O)N1CCN(C(C2CCC(=O)N2C)=O)CC1C(C)(C)C 3569,C(=O)(CCSc1ncc[nH]1)N(CCCNC(c1cnsn1)=O)C 3570,C1(CN(C(C2CC(F)C2)=O)CC)CCCN(C(C2CCC(=O)O2)=O)C1 3571,Cc1cnc(C(N2CC(CNC(=O)C3CC3)C(O)C2)=O)nc1 3572,C#CCCCCC(=O)NCC(C)(O)CNC(c1ccc(Nc2nccs2)cc1)=O 3573,C1(NC(c2ccc(CNC(CC(C)O)=O)cn2)=O)CCCN(C)C1C 3574,c1(C(N2C3C(NC(c4c(N)nc(Cl)cc4)=O)C(C3)C2)=O)cnn2c(=O)cc[nH]c12 3575,C(=O)(CC(C)CC(C)(C)C)N1CC(O)(C(C)NC(C#CC(C)C)=O)C1 3576,C(CCC)(C(O)C(=O)N1CC(OC)CC(O)C1)NC(CC(CC)OC)=O 3577,N1(C(c2c(OC)csc2)=O)CCCN(C(c2ccnn2C(C)C)=O)C(CO)C1 3578,c1(C(=O)NCCC(CNC(=O)C=Cc2ccccc2)O)cccc2ccnn12 3579,C1CC(=O)NCCOCCS1.N1(CC)CCCC1.C1(=O)CCOCCN1 3580,c1(NC2(CO)CN(C(c3sc(NC(=O)OCC)c(C)c3)=O)C2)ccc(C)c(C)c1 3581,C1(=O)CC(C(F)F)CN1.N1(C(c2cc(C)ns2)=O)CC(=O)NCC1c1ccccc1 3582,N1(C(CN(CC#C)C(C2CCC(F)(F)C2)=O)=O)CCC2(CC1)CC2C#N 3583,C1(CNC(c2ccc(OC)nn2)=O)CC2CN(C(c3cc(C)nc(C)c3)=O)CC12 3584,C(=O)(C1=C2CCN=C2NC=C1)N1CCC(N(C(=O)CS(C)(=O)=O)C)CC1 3585,C(N=c1nc(N2CCC3(CCCN(C)C3)C2)c2sccc2[nH]1)c1c(OC)nsc1 3586,c1(CC(N2CCCC(CNC(COCCN(C)C)=O)C2)=O)ccc(Cl)nc1F 3587,CC1CC(COC)CC(C)N1CC(C)(C)CO 3588,Cc1ccc(C(=O)NC2CCC(C)N(C(C3CC4(C3)CC(F)C4)=O)C2)cc1CO 3589,c1(CC)cccc(C(=O)N(C)CCN(C(=O)COc2ccc(C)cc2Cl)C)c1C 3590,N1(C(C2C(OC)COCC2)=O)CCC2(CCNC2)C1 3591,C1(CC(=O)NCC(=C)F)CN(C(c2ccnnc2)=O)C(C)(C)C1 3592,N1(C(COCC(=O)OC)=O)CCC(C(=O)NC(C2CSC2)C)C1C 3593,c1(C(N2CC(C(C)NC(=O)C(C)(C)c3cc[nH]n3)OCC2)=O)cnc(O)c(Cl)c1 3594,c1(C(N2CCC(C(F)C(=O)NCC3CCC(F)(F)C3)C2)=O)cccc[n+]1[O-] 3595,c1(C(N)=O)ccc(C(=O)NC2(CNC(c3cccnn3)=O)CCCCC2)cn1 3596,CN1CCC(NC(C23CC(C(=O)NCC4(C(C)(F)F)CC4)(C2)C3)=O)CC1=O 3597,c1(SC)ccc(C)c(C(N2CCC2CNC(c2ccc(C)c(C)c2)=O)=O)c1 3598,C(C(C)(O)CC(=O)N(C1CN(C(c2c[nH]nc2C)=O)CC1(C)C)C)OC 3599,c1(C(N(C2CCN(C(c3cc(C)c(C)[nH]3)=O)C2)CC#C)=O)ccc(C2CC2)nc1 3600,C1(C)(C(N(C(CNC(=O)CCC2CCCOC2)C2CC2)C)=O)CCCO1 3601,C(=O)(C(C)(C)C(C)(C)O)N1C(CCNC(c2cccc(COC)c2)=O)CCC1 3602,c1(N2CCC3(CCC(O)C3)C2)nc(N2CCC(F)(F)C2)nc2c1CCCC2 3603,c1(C(=O)NC2CC(C(=O)NCCc3cn[nH]c3)C2)nsnc1O 3604,Cc1nc(NC(C2C=CC(=O)N=N2)=O)ccc1Br.N12CCC(O)(C1)C2=O 3605,C(CC(CC)C(=O)NC1C=CCC(C(=O)NCCN(N2CCOCC2)C)C1)=CC 3606,C1(CNC(C2C(C(C)C)OCC2)=O)CCC2CN(C(C3CN(C)CCO3)=O)CC12 3607,C(=O)(C(CNC(c1cc(C2CC2)no1)=O)C(C)(C)C)NC(c1noc(C)n1)CC 3608,N1(C(CC2CCC(=O)N2)=O)CC2(CCC(CNC(c3ccc4c(c3)CCC4)=O)O2)C1 3609,C(=O)(C1=NOC(C)(C)C1)N(CC(=O)NC1CC(OC(C)=O)C1)CCOC 3610,C=CC(O)(C(=O)NC(C)C(C)NC(=O)COC1CC(F)(F)C1)C(F)(F)F 3611,c1(CC)cc(C)c(C(=O)NCC2CC2CNC(=O)CS)o1.c1(O)ccc(C)cc1 3612,C1(CNC(CC(C)C)=O)CC(NC(=O)CCC2CC(C)(C)CO2)C(O)C1 3613,C1(CNC(Cn2c(C)cnc2)=O)CN(C(c2ccnc(OC(F)F)c2)=O)CCO1 3614,n1(CC(=O)N(CCCCCNC(C2CC2Cl)=O)C)ccc([N+](=O)[O-])n1 3615,CCC(CNC(C1CN(C(=O)CCC(C)(C)C)CCN1C)=O)CC(C)C 3616,C(CC(=O)NCCC(O)C1CC1)(C(F)(F)F)NC(C1(COC)CCCC1)=O 3617,N1(C(=O)CC(F)(F)Br)CCC2(CC1)CC(F)CO2 3618,C1(NC(C2N(C)CCCC2)=O)CCN(C(=O)COc2ccsc2Cl)CCC1CO 3619,C=CCC(CC(C)C)C(=O)N(C(C)CCNC(c1nccc2ccccc12)=O)C 3620,N1(C(CC(C)CN(C)C)=O)CC2CCN(C(c3nnn4c3CSCC4)=O)CC2C1 3621,c1(C(=O)NC2C(CNC(Cc3nc(C)sc3C)=O)CCCC2)cccc(Cl)c1N 3622,C1(NC(c2ccc(CC)nc2)=O)CC(O)CN(C(=O)Cn2cc(F)ccc2=O)C1 3623,C(CC(O)C(F)(F)F)NC(C(CC=CC)NC(=O)CC1CCOC1=O)=O 3624,N1(C(C2CC(C#N)C2)=O)CCC2(CC1)CCN(C(C1OCC3CCCCC13)=O)CC2 3625,CCC(C)C(O)C(C)C(=O)NC1CC(CNC(=O)NCCCC2CCC2)C1 3626,N1(C(C2CCCN(C(c3ccn(C(F)F)n3)=O)CC2)=O)CC2CC3CC2C1C3 3627,c1(C(=O)NC(CNC(C(C(C)C)n2cccc2)=O)CO)cn2cnnc2cn1 3628,c1(CC(C)C(=O)NC(C)(C)C)ccc(F)cc1.c12ccc(o1)COCCNC2=O 3629,N1(C(C2(CC#C)CCCOC2)=O)CCC2(CC1)CC2CNC(c1ccc(F)o1)=O 3630,C(=O)(CCN(OC)C(=O)CC1=CCCC1)NCC(=C)C(F)(F)F 3631,N1(C(Cc2nc(C)oc2)=O)CCCC(C)C1CCNC(c1csc(O)n1)=O 3632,C1(F)(CNC(c2c(CC)non2)=O)CCN(C(=O)C(C2CCCCCC2)O)C1 3633,C1(C(=O)NC(CNC(C2CCCN(CC)C2)=O)CC(C)C)CCC(C)(C)OC1 3634,CC1CC2(CCO1)CC2C(=O)N(CCCNC(c1conc1C(C)(C)C)=O)CCO 3635,c1(C(N2CCC(OCCNC(c3c(OC)nccc3)=O)C2)=O)c(C)cnnc1O 3636,N1(C(CCCC(N)=O)=O)CCC2CN(C(c3cccnc3SC(F)F)=O)CC12 3637,N1(C(C2(OC)CC2)=O)CC(NC(C2(c3cccc(Cl)c3)CC(C)C2)=O)CC(C)(C)C1 3638,N1(CC)CC2CN(C(=O)C(CO)NC(c3ccc(F)cn3)=O)CC2C1 3639,Cc1c[nH]c(C(N2CCN(C(=O)CCc3ccc[nH]3)C(C)C2)=O)cc1=O 3640,C(c1cscn1)=CC(=O)N(C1CCN(C(c2sccc2C2CC2)=O)C1)CCC 3641,c1(C(=O)NCC)ccnc(C)n1.C(C(COC)=CC(=O)NC1CC(C(=O)OC)C1)OC 3642,c1(C(N2CC(NC(=O)Cc3cc[nH]n3)C2)=O)ccnn1C1CN(C(=O)OC)C1 3643,c1(C(=O)NCC(CNC(=O)C2=CCCS2)O)coc2c1C(O)CCC2 3644,Cc1nc2cccc(C(=O)NC3CC(NC(c4cc5sc(C)nc5[nH]4)=O)C3)n2n1 3645,CCC(C)C(O)C(C)C(=O)NCC1CC(=O)N1.c1(OC)ccc(OC)cc1O 3646,N1(C(c2cc(CC)no2)=O)CCCC(CNC(C2CN(S(C)(=O)=O)C2)=O)(OC)C1 3647,c1(C(N(CC(C)(C)CNC(=O)Cc2nncn2C)C)=O)cnc2c(c1)ncn2C 3648,N1(C(c2sc(CC)c(C)c2)=O)CCN(C(c2c[nH]nc2F)=O)C2CC12 3649,C12(CCC(F)CC1)CN2.c1(CCC)nc(C)c(-c2nc(C(=O)OC)cs2)s1 3650,Cc1cc(C)c(C(N2CC(NC(c3cncc4ccsc34)=O)CC2C)=O)cc1C 3651,C1(NC(c2n(CC)ccc2)=O)CN(C(=O)C=C(C)C(C)(C)C)CC2(CCC2)C1 3652,N1(C(C)C)CCCC1CC(=O)NC(C)CCCNC(=O)CCc1cc[nH]n1 3653,C1(NC(C=C2CCN(C)C2)=O)CN(C(=O)C(F)=CC2CC2)C2CCCCC12 3654,N1(C(C(CC)C(C)C)=O)CC2CCCC(NC(C3CCCS(=O)(=O)C3)=O)C2C1 3655,c1(C(=O)NC(COC)CNC(=O)Cc2c[nH]nc2C)ccc2n[nH]cc2c1Cl 3656,n1(CC)nccc1C=CC(=O)N(C(C)CCNC(=O)CC1C=NN(C)C1=O)C 3657,c1(C(N2C(CCNC(=O)CCc3cnc[nH]3)CC(OC)C2)=O)c(Cl)c(C)nn1C 3658,N1CCC(CC(=O)C(c2ccc(O)cc2)=O)CC1.CC(C)(C)N 3659,C(=O)(C(O)CCS(C)=O)NC(C1CCCCC1)CNC(CCCCOC)=O 3660,N1(C(CC(C)c2ccco2)=O)CCN(C(=O)CNC(C2CCCS2(=O)=O)=O)CC1 3661,c1(C(N(C2CCCC(NC(c3cc(C)oc3C)=O)C2)C)=O)cnc2n1CCCC2 3662,N1(C(CCSCCC)=O)CCC2CCCC12C(=O)NCC.N12CCC1CC2 3663,Cc1nn(C2CCC2)cc1C(=O)N(C)CCNC(=O)CCc1cccs1 3664,C(=O)(C(CNC(=O)C=Cc1ccncn1)CC1CCCC1)NC1C(CC=C)CCC1 3665,N1(C(C2(CNC(CCOC)=O)CC=CC2)=O)CCC(C)(CCO)C1 3666,Cc1ncccc1NC(C1(CNC(=O)Cc2ccc(Br)nc2)CC1)=O 3667,C(=O)(C#CC1(C)CCCO1)NC(C1CN(C(C2(C)CC(O)CN2C)=O)C1)C 3668,CC1(C)OC(=O)NC1CNC(=O)C(CNC(=O)CSCCC(C)C)CC1CC1 3669,N1(C(CCCC)=O)CCC(C)(CC(=O)NCC2CCCOC2)C1 3670,C1(NC(C(CC)(C)F)=O)CN(C(=O)CCn2ccnc2C)CC(C)(C)C1 3671,N1(C(C(CC)n2ccnc2)=O)CC2(CNC(c3ccc(CSC)o3)=O)CC1CO2 3672,n1(CCNC(CC(C(C)C)c2ccc(F)cc2)=O)cnc2c1CCCC2 3673,C(=O)(C(C(=O)NCC1CCN1C(c1cc(-c2cccs2)on1)=O)OC)OCC 3674,N1(C(c2cnc(C)s2)=O)CCN(CC2CC(F)(F)C2)CC1CO 3675,C(=O)(CC1CCc2ccccc21)N1C(CNC(=O)C#CC2CCOCC2)CC1 3676,c1(C(=O)NCCn2cc(C(=O)NC3CC3C(F)F)cn2)cc2cc(Cl)cnc2o1 3677,CC1CCCN(C(=O)CC(C)(C)C2CCCN2)C1CCOC(CNC(=O)C1CC1)=O 3678,N(C1CN(C(C2(c3ccsc3)CC2)=O)Cc2ccccc21)C(c1c(C)ocn1)=O 3679,Cc1cc(F)cnc1NC(C1(C)CCN1C(c1cc(Cl)c(Br)s1)=O)=O 3680,C1(NC(CCC=C)=O)CC2C(NC(=O)C(C)(C)n3cnnn3)C2C1 3681,c1(N2CCC(NC(c3n(C(C)C)ncc3)=O)C(C)C2)nc2ccc(Br)cc2o1 3682,c1(COCC(=O)NCC(C)(CO)NC(c2cnc(OC)s2)=O)nnc(S)n1C 3683,C1(C(N(CC(C)CNC(C2CCCO2)=O)C)=O)(CO)CC(C)(C)C1 3684,Cn1ncc(C(=O)NCCC2COCCN2C(=O)COCCCN(C)C)c1Cl 3685,n1(CC(N2CC(NC(C3C(C(C)(C)C)CC3)=O)C2)=O)ccc(Br)cc1=O 3686,CC(C)(C(=O)NC1(C)CN(C(=O)CCOCC(F)F)C1)c1cccnc1 3687,N1(C(C2(C#C)CC(=O)C2)=O)CCCC(CC(=O)NCC(C)C(=O)OC)CC1 3688,C=CCCCC(=O)NCC1(CNC(C2CCC(OC(C)C)C2)=O)CCOCC1 3689,N1(C(c2c(C)ocn2)C(=O)NC2CCOC2)CCC(O)C(F)(F)C1 3690,C1(C(=O)NC)CCN(C(=O)C(F)C2CC(O)C2)C1.C12(CCC1)C(=O)NC2.C1CC1 3691,C(=O)(CCS(=O)(=O)N(C)C)N1CCCC(CN(C)C(C2(Cl)CC2(C)C)=O)C1 3692,O(NC(=O)C(C(C)NC(c1cn2c(n1)CCC2)=O)C(C)C)C(C(=O)OC)C 3693,CC(C)(C)C(C(=O)NC1CCN(C(C2CCCCNC2=O)=O)CC1)NC(N)=O 3694,N1(C(C=CC(C)N(C(C=Cc2cc(C)no2)=O)C2CC2)=O)CC(CO)CC(C)(C)C1 3695,C(CCC(C)C)(C(=O)N1CCC(O)(CN(C(=O)CC2CC2C)C)CC1)NC(C)=O 3696,N1(C(C(C(C)(C)C)=O)=O)CC2(CCC(CNC(C3(Cl)CC3(F)F)=O)O2)C1 3697,c1(CNC(C2(C)CCN2C(c2cc(C(C)(C)C)n[nH]2)=O)=O)ccc(O)nn1 3698,c1(NC(NC(CC)CC)=NCCN(CC)CC)cc(O)c2c(CC)n[nH]c2c(=O)c1 3699,c1(C(C)CC(=O)NC2CC(N(C(=O)COc3ccsc3)C)C2)cc(F)cc(F)c1 3700,N#Cc1cc(F)ccc1C(=O)NC1C=CC(C(N2CC3C(C2)C3(F)F)=O)C1 3701,N1(C(CN2CC(C)(OC)C2)=O)CC2CCCC(C1)N2C(C12CC(C(=O)OC)(C1)C2)=O 3702,c1(OCC)ccc(C)cc1NC(C1(F)CCCN(C(=O)CCCF)C1)=O 3703,C=CCC(CNC(=O)C(C)N(C(c1cnccc1OC)=O)C1CC1)CC(C)C 3704,CC(CC(=O)N1CC=CC(O)C1)C(C)(C)NC(=O)Cn1cc(CO)nn1 3705,C(=O)(CC(C)(CN(C)C)C(F)(F)F)NC1CCN(C(C2(C(=O)NC)CCC2)=O)CC1 3706,N1(CCC(=O)NCC(CO)NC(c2c(C)cc[nH]2)=O)CCN(C(C)C)CC1 3707,c1(CNC(C2N(C(c3cc(C)c(F)nc3)=O)C3C(C2)C3)=O)cc2ccccc2[nH]1 3708,c1(C(=O)NC(c2ccc(I)cc2)C(=O)NCC(=C)C)ccc(OC)c(F)c1F 3709,c1(C(N(CCCSC)C)=O)cc(C(N)=O)c[nH]1.C12(CC1)C(=O)NC2 3710,C=CCCN=C(NCc1cc(Cl)cn1C)NC1CCOC(c2ccccc2Br)C1 3711,C1(C(C(=O)NC)N(CCCCCSC)CCOCCOC)CCOC2(CCC2)C1 3712,C=CC1CCN(C(C2(n3cc(C(c4ccccn4)OC)nn3)CCNC2)=O)C1 3713,c1(OC)ccc(C(=O)NC(C2CCCC2)CNC(C2CCCC(F)C2)=O)nc1 3714,C(=O)(CC(C(F)(F)F)NC(=O)COC1CCCOC1)N(C)Cc1cccc(F)c1 3715,Cc1nsc(C(=O)NCCN(C(=O)C(N2CCOCC2)C)C)c1Br 3716,N1(C(CCC(=C)C)=O)CCC(F)(CNC(C2CCC(=O)N2C2CC2)=O)CC1 3717,C1(CN(C(C(C)NC(C=CCOC)=O)=O)C)CCN(C)C1 3718,CC1CN(C)CC(C(=O)NC(C)C(N2CC(O)(CC(N)=O)C2)=O)O1 3719,CCC(CC)C(C(=O)N1CC(O)CC1CNC1(C(C)(C)NCC)CC1)OC 3720,C123COC(C1)(C2)CNC3=O.c1(C(=O)NCCc2ncon2)ccc(CF)nc1 3721,c1(CC)ccc(C)c(C(N2CC3(C2)CN(C(=O)C(c2ccc(Cl)s2)C)C3)=O)c1 3722,N1(C(c2c(OC)n(C)nc2C)=O)C2CCC1CN(C(C1CN(CC(C)C)C1)=O)C2 3723,c1(C(=O)NCCC2N(C(C3(C)C=CCC3)=O)CCC2)ccc2ocnc2n1 3724,C12(NC(C(CCSC)OC)=O)CC1CN(C(c1coc(C)c1)=O)C2 3725,c1(C(c2cccc(C)c2)C(=O)NCCOC)cc(Br)cnc1OC 3726,c1(CC)cnccc1C(N1CCC1(C)CC(=O)N(C(C)CC1CC1)C(C)C)=O 3727,c1(CC(c2cn(CCOC(F)(F)F)nn2)C)ccc(NC2CC3(CC3)C2)cc1 3728,c1(OC)cccc(OC)c1C(=O)NC(C1CCCN(C(=O)C(C(C)C)OC)C1)C 3729,c1(C(=O)Nc2cc(OC)cc(F)c2)ccc2nc(-c3c[nH]nc3C3CC3)sc2c1 3730,CN1C2CCC1CC(=CC(=O)NCC1CCN(c3cc(C(N)=O)ncn3)C13CC3)C2 3731,c1(C(=O)NCCN(C(C2CCC(CN(C)C)O2)=O)CC)c(C)cc(Cl)cc1C 3732,c12ccc(cc1)CN(C1CC1)C(C)(C)c1cn-2nn1.C(=O)(C(C)O)OC 3733,c1(C(N2CC=CC(NC(=O)C3=COCC3)C2)=O)cc2n(n1)CCNS2(=O)=O 3734,CCC(C)(C)CC(=O)NC1(CO)CCN(C(c2csc3cncn23)=O)C1 3735,C1(CC(=O)N(C)CCC2CCCO2)COCCN1C(c1nocc1Cl)=O 3736,c1(C(N(C2CCN(C(=O)CCCC3CC3)C2)CCC)=O)ccc2nc(O)[nH]c2c1 3737,C1(C(=O)Nc2cncc(OC)c2)C2C(CN1Cc1ccc(OC)nc1Cl)C2(C)C 3738,c1(CC(N2CC(NC(CCC(=O)NCC)=O)C(OC)C2)=O)ccc(C)cc1OC 3739,C(=O)(C1CCc2c[nH]nc21)NCC1(C)CCN(C(C(CCCC)O)=O)CC1 3740,C1(NC(=O)CN(C2CCC2)C(C2CCCCS2)=O)CNC(=O)OC1 3741,c1(C(N2CCCC23CCOC3)C(=O)NC)ccc(F)c(C)c1F 3742,N1(C(C2CC(C)N(C)C2)=O)C2CCC(C(=O)NCC3CCC3(F)F)C1CC2 3743,C1(F)(NC(=O)NCC2OCC(CNC(c3cccs3)=O)C2)CCC2(CC1)CC2 3744,c1(C(CC)C)ccc(OC)cc1.c12cccc(c1)NC(=O)NCCO2 3745,c1(C(N(CCNC(=O)C(C)S(N)(=O)=O)CC)=O)c(OC)ccc(F)c1N 3746,C(C(CC(C)C)C(=O)NC1CN(C(=O)Cc2coc3ccccc23)CC1O)OC 3747,c1(OC)cc(OC)cc(S(=O)(=O)Nc2cc(CNC(N3CCC3CO)=O)on2)c1 3748,C#CCC(CC(=O)NCC(C)OC(C)(C)CC)NC(=O)CC(=O)OC 3749,Cc1nn(C)c(Cl)c1C(=O)NCC=CCNC(=O)C(F)C1CCC1 3750,C1(NC(C=C(COC)C)=O)CCC2(CC1)CC2NC(=O)Cn1[nH]cnc1=N 3751,CCCC(CC1CCCCC1)C(=O)NC1CCCC1NC(c1coc(C)c1)=O 3752,C1(NC(c2cn(CCNC(C(C(C)(F)F)F)=O)nc2)=O)CCn2nnnc2C1 3753,c1(C(=O)NC(CN(C(=O)CC(C)CN(C)C)CC)C)ccc2ccnc(Cl)c2n1 3754,Cc1cc(C(=O)NC2CCC2NC(=O)C(C)N(C)C)ccc1O 3755,CC1(C)COC(C(=O)NC2(CO)CCCN(C(=O)COc3cccnc3)C2)CO1 3756,C1(NC(CC(N(C)C)C2CC2)=O)(CF)CCN(C(=O)Cc2cnc[nH]2)C1 3757,c1(CC)cc(C(=O)NCC(C(C)C)NC(c2ccnnc2O)=O)c2c(c1)CCO2 3758,c1(OC)cc(OCC(O)CNC(C2CC3CCCCCC23)=O)ccc1[N+](=O)[O-] 3759,C1(CN(C)C(C23CC(C)(C2)C3)=O)CN(C(=O)C(F)(F)C2CCCC2)CCO1 3760,Cc1ccc(C(C)NCCC(C2(O)CCOCC2)C)cc1C#N 3761,C(c1cccc(F)c1)=C(C(=O)NCC(C)NC(=O)CC1(CC(=O)OC)CCCC1)F 3762,c1(C(=O)NC(C)C)ccc(C(=O)NCC(C)(C2CC2)NC(=O)CCC(C)C)cc1 3763,C(C1CSc2ccccc21)NC1(c2n(CCCSC)nnn2)CSC(C)C1 3764,CC1CC2(CCN(c3ccnc(NC(c4ncc(F)cc4F)C)n3)C2)CO1 3765,C1(C(=O)NC(c2ccccn2)CC)C2CC1N(C(=O)CCc1ccn(C)c1)C2 3766,C(CCCC(C)C)(c1n(C(CC)C)nnn1)NCc1nnn(C(C)(C)C)n1 3767,N1(C(=O)Cc2ccco2)CC2CCCC(C1)N(Cc1ccc3nonc3c1)C2 3768,c1(C(N(C)CCNC(C2(CO)CCOCC2)=O)=O)sc2cccnc2c1Cl 3769,N1(C(=O)CCn2cccn2)C2CCC1CC(C(N1CCC(c3ccon3)C1)=O)C2 3770,c1(NC(C2CC(OC)CN2Cc2cccc(O)c2O)=O)ccc2ncn(C)c2c1 3771,c1(CC(C(=O)OC)NC(=O)OC(C)C)ccc(OC)cc1Br.C1(C(C)C)CO1 3772,N1(C(C(C2(O)CN(C(C3N(C(=O)OC)CSC3)=O)C2)F)=O)CCC2C(OC)C2C1 3773,C1(NC(CCCOC(C)=O)=O)C2CC3C1C3C2C(=O)NC1(C)CCCC1C 3774,C1(NC(C(C2CCC2)OCC)=O)CCN(C)C(c2ccccc2)C1 3775,C1(C(=O)NCCCCN=[N+]=[N-])CN(C(=O)CCOCC2CCC2)CC12CC2 3776,C=CCC(C(=O)NC(C1(O)CN(C(c2cccc(OC)n2)=O)C1)C)OC 3777,CC(C)C(O)C(F)(F)C(=O)NC(C)CC(C)NC(c1cc2nccn2c(O)n1)=O 3778,n1(CC)c(C2CCN(C(=O)NCCOC(C)(C)COC(C)=O)CC2)nnc1O 3779,C(N=c1[nH]c(N(C)Cc2ccc(Br)nc2)nc2c1CSC2)C1(OC)CCOCC1 3780,N1(C(C2N(C(C)=O)CCC2)=O)CCCCC1CCC(C)(C)NC(=O)Cc1cnoc1 3781,C1(C(N2CC(C)(c3nnc(-c4ccccc4)o3)C2)C)CC=CCC1 3782,C1(Nc2cc(N3CCN(C)C(=O)CC3)ncn2)CCC(C2CCCO2)O1 3783,C(=O)(C(C)CC(=O)N1CCC(NC(c2ccc(Cl)cc2F)=O)CC1)OC 3784,c1(C(=O)NCCCN2CCN(C(C3C(OC)CC3)=O)CC2)cccc(=S)n1O 3785,C1(CN(C)C)CCCN(C(c2cnc(CC3C4CCN3C4)s2)=O)C1 3786,N1(C(C(C(C)C)SCCCC)=O)CCC2(CCN(C(c3ncc[nH]c3=O)=O)C2)C1 3787,c1(C(=O)NCC2(C(F)F)CCN(C(C(CC)OC)=O)C2)cc(C)cc(N)c1 3788,CC(C)(C)C(C)(C)C(=O)N1C2CCC1(CNC(=O)C1=CCCCCC1)CC2 3789,Cc1ccc(CCCN(C(C)CNC(C2CCC2)=O)C)c(C)c1 3790,C(C)(C1=CCCOC1)NC(C(c1cn(C)nn1)NC(c1[nH]cc(C)c1)=O)=O 3791,c1(C(=O)NC(C)CC(C)NC(c2n[nH]c3c2CCC3)=O)cc([N+](=O)[O-])nn1C 3792,C1(C(N(CC(C)NC(=O)Cc2cc[nH]c2)C)=O)CC(=O)N(c2ccccc2F)C1 3793,CCC1=NOC(C(N2CC(CNC(C34CCC(CC3)O4)=O)C(O)C2)=O)C1 3794,c1(C(=O)NCC2(F)CCN(C(C(CC)OC)=O)C2)cnc(C)cc1C 3795,c1(C(=O)NC2CC3(C(NC(CN(S(CC)(=O)=O)C)=O)C3)C2)cc(Cl)ccc1F 3796,c1(C(=O)NC(CNC(C2N(C)CCC2)=O)(C)C)ccc2c(=N)[nH]cnc2c1 3797,CC(=O)CCCC(=O)NCC12CC1CN(C(=O)COc1ccc(F)nc1)C2 3798,n1(CC)cc(CN(C(=O)CCCC2CCCO2)C(c2cnc(C)n2C)=O)c(C)n1 3799,c1(NC(=O)Nc2c(SCC)cc(Br)cc2)ccc([N+](=O)[O-])cc1Cl 3800,c1(COCC(=O)NC(C2CCN(C(=O)Cc3nncn3C)C2)C)ccccn1 3801,c1(C(C)C(c2c(-n3cc(C4(N)CC4)nn3)ccs2)=O)cc(C2CCC2)nn1C 3802,CCC(C)(C)CCCC(=O)NC(C)CN(C)C(c1cc[nH]c(=NC)c1N)=O 3803,c1(C(N(CC(=O)N(C(C)C=C)CC)CC#C)=O)cncnc1 3804,c1(NC(=O)NC2(CCC)CCOC2)ccc(C2CC2)c([N+](=O)[O-])c1 3805,C1(C(N2CC(C)OC(C)C2)C(=O)NCCOCC)CC2CC1C1CC21 3806,C(=O)(C1=CCCN(Cc2ccc(O)nc2)C1)Nc1ccc(C#N)nc1 3807,CC1CN(C(=O)COCCF)CCC1CNC(c1ccnn1CC#N)=O 3808,c1(OC)cccc(C(=O)NCCC2CC(NC(=O)C(C)CS(C)=O)C2)c1C 3809,C#Cc1ccc(F)c(C(N2CCCC(NC(C3CCCN3C)=O)C2)=O)c1 3810,N1(C(CCCCCOC)=O)CCC(O)(C2CCN(C(c3c[nH]nc3C)=O)CC2)C1 3811,CN1CC=CCC1C(N1CCC(CC(=O)NCCC2CCCN2C)C1)=O 3812,N1(C(CCC=C)=O)CCCC(C2CCCN(C(=O)CCc3cncc(F)c3)C2)C1 3813,N1(C(C(C)=C(CC)C)=O)CC(O)(C(C)NC(=O)CC2CCC3CC23)C1 3814,CC1CN(C(=O)CC2C=CCC2)C1C(=O)NCC(C)(C)CC1CC1 3815,C#Cc1ccc(C(=O)NC2CCN(C(c3nnc(Cl)cc3N)=O)CC2O)cn1 3816,c1(C(N(C2CCCN(C(=O)CSCC(C)C)CC2)CC)=O)ccc2ccnn2c1 3817,c1(CCC(=O)NC2CCC3CC2CN3C(=O)CCF)cnc2n1CCCCC2 3818,N1(C(C(=O)NCCSCC)c2cccs2)CCOC(C2CC2)CC1 3819,c1(C(C)(C)C)cc(C(N2CCC(C)(NC(=O)Cc3ccoc3)C2)=O)ccc1O 3820,c1(OC)c(C(=O)NC(CNC(C2C3CCCC23)=O)C(C)C)ncnc1C 3821,C(=O)(C(C)COC)NC(C(=O)N(CCC)CCO)c1cccs1 3822,c1(OC)ccc(F)cc1CC1CCCCC1C(N1CCCC(Cn2cccn2)C1)=O 3823,C1(N(C(=O)C(C)C2CCC2)CC)CCN(C(c2csc(C)c2Br)=O)CC1 3824,C12(CNC(C34CC(C)(C3)C4)=O)CC1CN(C(C1(S(N)(=O)=O)CC1)=O)C2 3825,c1(C(N2CCC(F)(CNC(CCOCC(C)C)=O)C2)=O)cc2ccncc2s1 3826,N1(C(c2n[nH]cc2Br)C(=O)NC(CC)(C)C)CCCC(Cn2ccnn2)C1.N(C)C 3827,N1(C(C(=O)NCC)=O)CCC2(CCCN2C(=O)C(O)CC(C)(C)C)C1 3828,n1(CCC(N2CCC(O)(CNC(C3C(C)C3C)=O)CC2)=O)ccc2cccnc12 3829,CC(C)CC(F)C(=O)NC1(C2CN(C(=O)Cc3cc(-c4ccco4)on3)C2)CC1 3830,C1(NC(C(c2cccnc2)C)=O)CC2CC(NC(=O)CCc3cccn3C)C2C1 3831,C=CCCC(C)NC(C1CCCC1CNC(C1CN(C)C1)=O)=O 3832,C1(CNC(c2c(C)cno2)=O)C2CCCC1N(C(c1ccc(O)c(Cl)n1)=O)C2 3833,Cc1nc(OC2CC2)sc1C(=O)NC1CCCC1NC(=O)CSCC(C)C 3834,c1(C(C)NCc2oc(CC)c(C(=O)O)c2)ccc(Br)c(C)c1O 3835,C(=O)(CS(=O)C(F)(F)F)NC(CNC(c1c(CC)ocn1)=O)C1CC1 3836,CC#CCC(C(=O)NCCOc1cnn(C)c1)NC(=O)CCc1cncs1 3837,CCCCCC(O)C(=O)N1CCC2CC12C(=O)NCc1ncnn1CCC 3838,N1(C(C(C=CCCC)O)=O)CC(CNC(C2(C3CC3)CC2)=O)CC1(C)C 3839,C(=O)(C(C(=O)NC(C)(C)C(C)NC(=O)CNC(c1occc1C)=O)OC)OC 3840,c1(C(=O)NCCCOCCNC(C2(CC)CCCO2)=O)cc([N+](=O)[O-])ccc1N 3841,C1(CNC(C(C2CCCOC2)OC)=O)CCCNC12CC2 3842,C1(CC=C)(NC(C2CCS(=O)(=O)C2)=O)CCN(C(C2CCCNS2(=O)=O)=O)CC1 3843,Cc1cc(C)c(C(=O)OCc2ccccc2C)c(Cl)n1.N12CCC(C1)NCC2=O 3844,CC1(C)OC(=O)CC1C(=O)NCCN(CCOCCO)C(C1CC2(CCC2)CO1)=O 3845,c1(C(=O)OC)cccc(Br)c1NC1CCN(C(=O)C(C)CC(F)F)C1 3846,Cc1ocnc1CC(=O)NOCC(=O)NC1CN(C2CC2)C1 3847,N1(Cc2cncc(OC)c2)CCC(C)C(NC(c2ccc3c[nH]nc3c2)=O)C1 3848,CC(C)C(C(=O)NCC1(NC(C2CN(C)C2)=O)CCOC1)c1cnn(C)c1 3849,C1(C(C)C(=O)NCC(O)CNC(c2ccon2)=O)CCC(=O)N1 3850,CC(C)C(CCNC(c1nnnn1C1CCOC1)c1nccs1)N(C)C 3851,c1(OCC(=O)N(CCCN(C(CC(=C=C)C)=O)C)C)ccc(C)cc1C(F)(F)F 3852,C1(C(=O)NCC(CC)(C)NC(=O)CCc2nccs2)CCc2ccccc2C1 3853,C12(CNC(c3ccc(C(C)C)o3)=O)CC(CN1C(C1CCCCO1)=O)C2 3854,C1(CNC(CN(C2CCCC2)C)=O)CC2(CC2)CN1C(c1cn(C2CC2)cn1)=O 3855,Cc1ccccc1OC(=O)CN(C)C(c1cnnn1C(C)C)=O 3856,c1(C(N2C(CNC(C(C)Nc3scc(C)n3)=O)CC2)=O)cc(O)nc(Cl)c1 3857,C=CC(C)(CC)C(=O)N(C1CCN(C(c2ccc(NC(=O)NC)c(Cl)c2)=O)C1)C 3858,c1(C(CNC(=O)CCSCC)O)ccccc1.C(=O)(CCCN(CCOC)CC)N 3859,C12(CNC(=O)CSCC3CCCO3)CC(NC(C3COCC3C(F)F)=O)(C1)C2 3860,C(=O)(CCCCN=[N+]=[N-])NC1CN(C(C(CC=C)(F)F)=O)CC1n1ccnn1 3861,C1(CC(C)C)(N(CCNC(C(C)OCCCCCC)=O)CC)CCNC1=O 3862,Nc1cccnc1C(=O)NCC1C(CNC(c2cnc(C)nc2)=O)CCCC1.C(=O)O 3863,C(=O)(CC(C)C(F)F)NC(C(=O)N(CC(CC)(O)CC)C)COC(C)C 3864,C=CCC(CNC(=O)CCC1(N(C)C)CCCC1)NC(=O)C(=O)NCC1CC1 3865,C1(NC(Cc2nn(C)nc2Br)=O)CN(C(C2CCCN2N=O)=O)CCC1CO 3866,C(CCCCCN=c1[nH]ccnc1C)NC(c1coc(Br)n1)=O.c1(SC)ccccc1 3867,c1(C(=O)NCC2(C#N)CCC2)c(NC(C2CC(=O)N2)=O)sc2c1CCCC2 3868,C=CCC(C)(CNC(=O)CC1(C)CCN(C(=O)COCCCF)C1)CO 3869,c1(CC)cccc(C(=O)N(CCNC(=O)CCc2ccn(C)n2)C2CC2)c1 3870,C#CC1CCCN1C(=O)CC(C)NC(=O)C(O)CN1CCCC1 3871,N1(C(CCSc2n(C)ccn2)=O)CCSCC1CCNC(c1ccc(Cl)nc1)=O 3872,C1(NC(C2(OC)CC2)=O)CC(O)CN(C(c2cnc(C3CCC3)s2)=O)C1 3873,C1(CN(C(=O)COCCOC)CC)CCCCN1C(C1CNC(=O)N1C)=O 3874,Cc1nsc(NCCC(C)NC(C2(CF)CCOCC2)=O)c1C#N 3875,N1(C(C2CN(C)CC2C(F)(F)F)=O)CCCC(NC(=O)C(C)(C)c2cnsc2)CC1 3876,Cc1ccnc2c(C(=O)NC3(CCNC(C4CC45CCOCC5)=O)CC3)cnn12 3877,C1(NC(C(C)CF)=O)CCCCN(C(c2cn(C)c(O)n2)=O)C1 3878,Cc1c(F)cc(C(N2CCC(C(N3CC(C#N)C3)=O)C(O)C2)=O)cc1F 3879,N1(C(c2c(CNC(CCc3cc(C)[nH]n3)=O)c[nH]n2)=O)CCOC2CC12 3880,C1(C(C)C)COCCN1C(=O)NCC1CCCN1Cc1nnn(C)n1 3881,c1(C(=O)NCc2c(CNC(C(F)=CC)=O)ocn2)cc(CC)n(C)n1 3882,c1(C(N(CCN(C(C(C)OCC)=O)C)C)=O)cc(Cl)cnn1 3883,CC1=CCC(N(CC(N2CCN(CCCCCNC(=O)C=CCl)CC2)=O)C)CC1 3884,C1(CNC(c2c(CC)nc[nH]2)=O)CCCN(C(=O)C(CC)N(CC)CC)CC1 3885,c1(N2CC(CC#N)N(C(C3CC3N)=O)CC2)ncnc2ccc(F)cc12 3886,N1(C(C(c2cccc(Cl)c2)CC)=O)CCC(NC(=O)C(C)SC)C(O)C1 3887,C(C(C)(C(=O)NOC1CCCC1)NC(=O)CCc1cc(C)[nH]n1)SC 3888,S(=O)(=O)(c1ccccc1NC(=O)N(C)CC1(O)CCC(C)(C)C1)N(CC)CC 3889,C(=O)(CCCS(C)(=O)=O)NC(CNC(c1c(CC)cc(Cl)cc1)=O)CO 3890,C1(C(N(CC(C)CNC(=O)COCC2CCCO2)C)=O)CCS(=O)(=O)C1(C)C 3891,C#CC1CN(C(=O)C(CCOC)NC(c2cnns2)=O)CCO1 3892,N1(C(C2C(C(=O)OC)CC2)=O)CCC2(CC(NC(=O)C(C)(C)CF)C2)C1 3893,c1(OC)cc(F)c(C(N2CCC(C(C(C)C)NC(=O)C(Cl)=CCl)CC2)=O)c(F)c1 3894,c12ccccc1C(=O)N(C)C2.C1(SC)CCCC1n1cc(CN2CCCC2)nn1 3895,C1(C(N2C(CNC(CC(CC)OC)=O)CC2)=O)CNc2ccnn2C1 3896,C#CCC(CC#C)C(=O)N(C)CC1CCCC(NC(c2cc(C3CC3)on2)=O)C1 3897,C1(C(=O)NCC(CNC(c2c(C)c(N)ccc2)=O)C)Cc2c[nH]cc2S1(=O)=O 3898,C1(NC(CC2(NC(C)=O)CC2)=O)CCCN(C(=O)C(F)(F)C2CC2)CC1 3899,Cc1nnc2n1CCN(Cc1ncc(Br)cc1F)C2.c12c(cccc1F)NC2=O 3900,Cc1c(F)ccc(C(=O)NCC2CC2CNC(C2CCS2(=O)=O)=O)c1Cl 3901,c1(NC(CC(C)Cc2ccccc2C(F)(F)F)=O)cccc([N+](=O)[O-])c1 3902,CCC(O)C(C)C(=O)N1CC(=CC(=O)N(C)CC2(OC)CCC2)C(C)(C)C1 3903,C1(CCC)C(=O)NCCN1C(=O)C(=O)NC(c1ccc(F)cc1Br)C 3904,C1(CNC(C#CC(C)C)=O)CC2(CCOCC2)CN1C(=O)CC1CC(=O)NC1=O 3905,N1(C(C2C(CC)CCC2)=O)CCN(C(c2ccc(NC(C)C)cc2)=O)CCC1C 3906,c1(C(=O)NC2CC(NC(c3ccc(C)n3C)=O)C2)cccn(C2CC2)c1=O 3907,O=C(CCCc1nccs1)NCC(N1CC(CO)C1)=O 3908,C1(OC(C(COC)Cl)=O)CCCN(C(c2ccccc2C)C)C1=O 3909,C(C)(CC(C)(C)C)N(C(c1c(C)csc1)=O)C.C(C=O)=CC=O 3910,CC(C)(CC(=O)N1CC2CC2(NC(=O)Cc2ccc(C#N)nc2)C1)CC(F)(F)F 3911,c1(C(N2CCC(N(C(C3(C#C)CCC3)=O)CC)C2)=O)cc(C2CC2)ccc1Cl 3912,CCC(CCCC(=O)NCC(O)COCC(C)C)NC(c1cc(C(N)=O)co1)=O 3913,C1(NC(CC=CC(C)(C)C)=O)CN(C(=O)C(C)(C)c2cncs2)CCC1CO 3914,Cn1c(C(=O)NCC(O)CNC(C2(C)CC2(F)F)=O)ccc1C#N 3915,N1(C(CCCC)=O)CCC(O)(Cc2n[nH]c(=NCc3occc3C)s2)CC1 3916,CC(CCN(C(=O)CSc1nc[nH]n1)C)NC(=O)Cc1cc[nH]c1 3917,O=C(CN=c1cc[nH]cc1)NC1C2CCN(C(=O)COCCF)CC12 3918,C1(NC(C=C(C)C(C)(C)C)=O)CCCCCN(C(=O)COC2CCN(C)CC2)C1 3919,C=Cc1cc(C(N2CCC(OCCCCC3CN(C(=O)NC)C3)C2)=O)cc(F)c1 3920,c1(C(N2C(CCC)CN(C(c3ns[nH]c3=O)=O)CC2)=O)c(F)ccc(F)c1F 3921,c1(OC)ccc(F)c(CC(=O)N(C2CN(C(c3ncccn3)=O)CC2(C)C)C)c1 3922,C(=O)(C1CCCc2nccn21)NC(CCNC(c1c(CC)ccs1)=O)C 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3941,C12(C(N3CC4C(NC(c5c(NC)scn5)=O)(C4)C3)=O)C3C4C1C1C2C3C41C(N)=O 3942,c1(N2CC3CN(C(CN(C)C(N)=O)=O)CC3C2)nc2cc(F)cc(F)c2o1 3943,N1(C(c2cc(C)on2)=O)CCCC(C2CCN(C(=O)C=C3SCC(=O)N3C)C2)C1 3944,C(=O)(C(CC)(CC)C(=O)OC(C)(C)C)NC(CCNC(C(CC(=C)Br)(C)C)=O)C 3945,c1(C(=O)NC2CC(NC(c3c(NCC)snc3C)=O)C2)ccc(O)nc1C 3946,c1(CC)noc2ncc(C(=O)NC3CCC3CNC(c3ccccc3)=O)cc12 3947,C(N=c1[nH]cnc2cc(F)c(F)cc12)C1N(C(C2(C)CCOCC2)=O)CCCC1 3948,Cc1nccn1CCNC(=O)CCOC1CN(C(c2ccccn2)=O)C1 3949,c1(C(=O)NCC2CN(C(c3[nH]c(=NC4C(C)C4)sc3)=O)C2)ccc2c(c1)CCN2C 3950,C#CCCN(C)N1CCCC(Cc2ccc(Cl)cc2)C1 3951,CCCCCCCCC(=O)N1CCSCC1CCNC(=O)C1=COCCC1 3952,Cc1ccc(SCCC(=O)NCC(C)(C2CCC2)NC(c2cn(C)cn2)=O)cc1 3953,N1(C(CC(CC)C2CC2)=O)CCOCC(F)(CNC(=O)Cn2ccnn2)C1 3954,C12(CNC(c3cc(Cl)cs3)=O)CN(C(c3cccc4nncn34)=O)CC1CCO2 3955,n1(CC(=O)OC)nccc1C(=O)NCCOCCNC(=O)C(O)C1CC1 3956,c1(C(C)=O)ccccc1C(=O)NC12CCNCC1C2 3957,Cc1cnc2cc(C(N3CCCC3CNC(=O)C(C)OC3CCCC3)=O)nn2c1 3958,N1(c2c(C)cc(Cl)cc2)CCCN(C(c2cccc(F)c2C)=O)C(C)C1 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3977,CCCC(C(=O)N(C)CC1(NC(c2ccc3nn[nH]c3n2)=O)CC1)S(N)(=O)=O 3978,CC(F)(F)C(C)(C)C(=O)NCC1(C)CCCN(C(c2ccc(F)cc2C#N)=O)C1 3979,c1(C(=O)NC2C(C)CN(C(c3cnc(O)n3C)=O)CC2)nnn2c1CCCC2 3980,C1(C(=O)NCc2ncc(C)s2)CC12CCN(C(c1n[nH]c(C)c1O)=O)CC2 3981,O=C1CCC(C(=O)NCC2CCCCN2C(c2ccsc2C(F)F)=O)CN1 3982,c1(C(N(CCNC(C2C(CC)CCO2)=O)CC)=O)[nH]c2ccc(F)cc2c1C 3983,CCCC(C(=O)NC1CCCCC1NC(c1cc(F)c(CO)c(F)c1)=O)C(C)C 3984,c1(C(=O)NCCC2CC(OC)CN2C(c2ccns2)=O)cc(Cl)c(F)cc1O 3985,Cc1ccc(OCCC(N2CC(NC(=O)CCC(C)C#N)C3(CC3)C2)=O)cc1C 3986,CCCC(C(=O)N1CC(NC(N)=O)C1)c1ccc(Cl)cc1 3987,c1(Cc2onc(CC(CC)CC)n2)cncc(Br)c1 3988,CC(C)(C)CC(O)CC(=O)NC1CCCC1C(=O)NC(CCO)C(F)(F)F 3989,CCCC(C(=O)N(CCC(=O)NC12CCC(CC1)C2)CC)N(C)C 3990,c1(OC)nc(C(F)(F)F)ccc1-c1nc(C(C)(C)C(C)(F)F)nn1CCCO 3991,c1(C(N(C2CCCN(C(C(CC)O)=O)C2)C)=O)cc(O)cc(N)c1Cl 3992,N1(C(CC2C(CC)CC2)=O)CCN(C(=O)COCCN=[N+]=[N-])CC1C 3993,c1(C(=O)NC2C(CNC(c3n[nH]c(C)c3C)=O)C2)c(C)[nH]c2ncccc12 3994,CCCCC(CC)C(=O)N1CCCC1CCCNC(c1cnc(CC)[nH]1)=O 3995,C1(C(N(C)C(=O)OCC2CCCN2C(C2(C(N)=O)CC2)=O)=O)CC(O)CN1C(N)=O 3996,Cc1nnc(O)c(C(=O)NC2CCC(NC(c3ccc4snnc4c3)=O)C2)c1C 3997,c1(C(=O)OCC2(N3CCOCC3)CCCOC2)nc2ccc(F)cc2s1 3998,c1(C(N2CCCC3(NC(C#CC(C)C)=O)C(C2)C3)=O)n[nH]c2ccc(Br)cc12 3999,c1(CNC(C2CCCN(C(=O)COC3CCCCC3)C2)=O)cc(Br)ncc1F 4000,c1(C(N2CC3C(C(=O)NCC4CCCOC4)C3C2)=O)ccc(Cl)c(F)c1 4001,N1(C(c2ccc(F)c(Cl)c2)=O)CC2CCC1CN2C(C1SC2C=CC1CC2)=O 4002,N1(C(CSC(=N)N)=O)C(CNC(=O)C(c2cscn2)C2CC2)CC2COCC12 4003,C1(CNC(CCC(C)OC)=O)CC2CN(C(C3CCN(CC(C)C)CC3)=O)CC12 4004,Cc1ccc2ccccc2c1C(C)NC(=O)Nc1sc(CC2CC2)nc1C 4005,c1(N2CCC(N(CC#C)C(c3cscc3C)=O)CC2)ncnc2cc(Br)sc12 4006,C1(CCC)CC(C(=O)N(CC(C)(C)NC(=O)C=CI)C)CCO1 4007,c1(NC(C)=O)cccc(COC(=O)NC2(NC(C)(C)C)CCOCC2)n1 4008,C1(N(C(c2ccoc2C2CC2)=O)CCO)C=CCN(C(=O)COCC(O)CO)C1 4009,C(=O)(C(O)CC(N)=O)NC(C)CCC(=O)N(C)Cc1cccc(O)c1 4010,CC1CCC2(CC2)N(c2ncnc(NCc3cnn4c3CCCC4)c2C)C1 4011,c1(CN)n[nH]c2c1CN(C(=O)Nc1cccc(CN3CCNC3=O)c1)CC2 4012,C1(C(=O)NC(CCNC(C(CCCC#C)C)=O)(C)C)CCc2cn(C)nc2C1 4013,C1(NC(Cn2ccc(C)n2)=O)CCN(C(=O)CC2CCC23CCC3)C12CCC2 4014,C(=O)(CCC(=O)NCC1CCN(C(C2COC(C)(C(F)(F)F)C2)=O)C1)NCCC 4015,C1(C(N(CC#C)CCO)=O)(CC)CCCN(C(c2c(OC)noc2C)=O)C1 4016,c1(NC(c2cn(CCNC(CNC(=O)OC)=O)nn2)=O)onc2ccccc12 4017,C(CCC(C)CC(=O)NC1CCN(C(=O)C(CCO)N(C)C)CC1O)=C(C)C 4018,C12(NC(c3c(CC)nn[nH]3)=O)CCCC1CN(C(=O)C=Cc1cccnc1C)C2 4019,C(=O)(CC(F)(F)C(F)F)N1CCCN(C(Cc2ccc(C(C)(C)C)nc2)=O)CC1 4020,N1(C(CCC=C)=O)CCC(CO)(CNC(=O)CCN(C)C(C)=O)CC1 4021,c1(OC)noc(C)c1C(N1CCC(C(C)C(=O)NCC2(C)CCCCC2)C1)=O 4022,N1(C(CC=CCC)C(=O)NC2CC(C(=O)OC)C2)CC2(C1)CC2(F)F 4023,C(=O)(C(=O)CCCC)NC(CC=C)CNC(c1cnc(OC)c(Cl)c1)=O 4024,N1(C(CC(=O)NCC)=O)CCC(C2CC2)C1C(N1CC(C)(N(C)C)C1)=O 4025,c1(C(=O)NC(C)CCN(C)C(C2CCOC(C)C2)=O)cc2c(nc1O)CCC2 4026,c1(C(=O)NCC2C=CCN2C(C2CCCC2(F)F)=O)ccc2c(n1)OCCO2 4027,C1(O)(CN(C(c2n(CC=C)ccc2)=O)C)CCCN(C(=O)C=Cc2ncc[nH]2)C1 4028,C1(NC(C(C)OCCNC(c2ccccc2)=O)=O)CN(C(=O)C(=O)N(C)C)CC1O 4029,c1(C(=O)NCCCCCN(C(c2cc(SC)c(C)o2)=O)C)nc[nH]c2ncnc1-2 4030,c1(OC)ccc(Cl)c(C(=O)NCC23CC2CN(C(=O)CC24CCCC2C4)C3)c1 4031,N1(CCOCCC(C)C)CCC2(CCN(C(c3csc(CO)n3)=O)CC2)C1 4032,c1(CC(N2CCCC(NC(C3(O)CC(CF)C3)=O)C2)=O)cnccc1Cl 4033,C1(CNC(c2n(CCC)ncc2)=O)CCN(C(C2CSCN2C)=O)C12CCC2 4034,N1(C(c2c(C)cc[nH]2)=O)CCN(C(C2CC2CC(C)C)=O)C(C2CC2)C1 4035,C(C(CC(F)(F)F)NC(=O)CCc1cc(F)cc(F)c1)NC(C(CC)NC(C)=O)=O 4036,C1(CC)CC(NC(=O)CCN(C(=O)Cc2cnccc2C)C)CCO1 4037,C(CCC(C)C)(C(=O)NC(c1ccccn1)C)NC(c1c(CC)nccn1)=O 4038,C(=O)(C(C)(O)C(F)(F)F)NCC(=C)CCSc1ccc(C)c(Cl)c1 4039,Cc1ccc(C)c(C(=O)NCC(N2CCC(C)(N(C3CCN(C)C3=O)C)C2)=O)c1 4040,C1(C(=O)NCCC=CC=C)CCCC2CN(C(c3c[nH]ccc3=O)=O)CC12 4041,N1(Cc2onc(C(C)OC)n2)CCCC(CO)(NC(c2cnc(C)[nH]2)=O)C1 4042,C(=O)(C(C1=CCCSC1)N1CCOC(C(C)(C)C)C1)NCC=C 4043,C(N=c1ncc(C(C)(C)O)c[nH]1)C1CC(NC(C2CC(C(C)(C)C)C2)=O)C1 4044,N1(C(c2c(N)cc(F)cn2)=O)CC=C(CC(=O)NC2CC2O)CC1 4045,C1(C(=O)NCC2CN(C(c3c(CC)onc3)=O)C(C)C2)CC2(CC(OC)C2)C1 4046,C(CCC(C)(C)CO)NC(CC1CC(C)N(C(=O)C=CC(=O)N(C)C)C1)=O 4047,C1(NC(c2c(C)ncs2)=O)CS(=O)(=O)CC1NC(c1cnc(C(C)C)[nH]c1=N)=O 4048,C(C(C)(CO)CO)N(C(=O)CC(=O)NCC(=O)NCC1CC1)C 4049,C1(C(N(C2CCOC2)CC#C)=O)CN(C(=O)CCn2cnc(=N)[nH]2)CC1(F)F 4050,c1(NC2CC(C(=O)Nc3nc(C)c(C#N)nc3)C2)ncnc2sc(Br)cc12 4051,c1(SCC2N(C(CC(C)(C)C)=O)CCC2)cc(F)cc(Cl)c1.C1CNC(=O)N1 4052,N1(C(=O)C=Cc2cocn2)CC2CCC(NC(C3(F)CCOC3)=O)C2C1 4053,c1(-n2c(Cc3ccc(OC)cc3C(F)(F)F)nc(CO)n2)cccc2nsnc12 4054,C1(CC)CC2(CCC(NC(=O)NCc3nc(Br)cc(OC)c3OC)CC2)C1 4055,c1(C(C(=O)N(CC(CC)NC(=O)Cc2ccc(C)s2)CC)C)ccccc1C 4056,C1(F)(C(N2CCC(CN(C)C(C3(CF)CCOCC3)=O)CC2)=O)CCS(=O)(=O)C1 4057,C1(NC(CCOCCN(C(=O)C(C)(C)C)C)=O)CCCSC1 4058,N1(C(C=CC)=O)CC2CC(NC(=O)C(C3CCC3)OC)CC1C2 4059,N1(C(C(C)(C)CO)=O)C2CCC1CC(CNC(C1C3CCN1CC3)=O)C2 4060,c1(CC)cc(C(=O)NC2(COC)CN(C(c3cc(Cl)ccn3)=O)C2)ccc1F 4061,ClC1(Cl)CC(N=c2[nH]c3c(c(=NCCCC4CCCCC4)[nH]2)SCC3)CCO1 4062,N1(C(CN2C(C)CCC2C)=O)CC2(CCC(CNC(=O)CCCN3CCC3)O2)C1 4063,C1(C(=O)NC(CNC(C=C(C)C(C)C)=O)CC)CCCOC1CC(F)(F)F 4064,C12(NC(=O)Cc3cc[nH]c3)CCCC1N(c1cc(Cl)nc(C(F)(F)F)n1)CC2 4065,O(N1CCC(N=c2cccc(S(=O)(=O)N3CCCC3C3CCCO3)[nH]2)CC1)CC 4066,c1(OCC)ccc(Cl)c(C(=O)N(C2CCCN(C(C3CC(C#N)C3)=O)C2)CC)n1 4067,C1(C(=O)NC2(C3CCN(C(C(=O)NC(C)C)=O)C3)CC2)CCc2nnnn2CC1 4068,C12(NC(CSCC)=O)CCC(CN(C(=O)CN=[N+]=[N-])C1)C2 4069,C1(CNC(CC2CC(NC(C3OCC(C)C3)=O)C2)=O)OCCC1(C)C 4070,c1(NC(C(N2CC3(C(=O)OC)C(C2)CCCO3)C)=O)cnc2c(C)nccn12 4071,Cc1cc(CNc2cc(F)cnn2)cc(C(F)F)c1 4072,C1(CCNC(C2N(C(CC)=O)CSC2)=O)COCCN1C(=O)COC1CC1 4073,N1(C(C2(C)CC(NC(C3CCN(CC)C3)=O)C2)=O)C2CSCC1C2 4074,Cc1cc2c(Br)cccc2c(C(=O)NCCN(C(c2ccnc(O)c2)=O)C2CC2)n1 4075,c1(C(C)Nc2ccc(F)cc2)ncc2c(n1)CN(Cc1ccc(Br)cc1C#N)C2 4076,Cc1cc(Br)cnc1-n1cc(C2(C(=O)N(C)C)CN(C(=O)C#CC3CCC3)C2)nn1 4077,c1(C(=O)NCC2CC(C(=O)OCC)C2)nc(Cl)oc1C.C12CC1NC2=O 4078,CC1=C(C)CC(C)(C(=O)N(CCNC(=O)CCC#N)C(C)C)CC1 4079,c1(CC)ncsc1C(=O)NCCOC1CCOC1.C1(=O)CCCN1C(C)C 4080,c12ccc(cn1)S(=O)(=O)NC(=O)N2.C=C(COC)C1CCOCC1 4081,Cc1nc(N2CCC3(NC(=O)C4=NNC(=O)CC4)CCCC23)c2ccsc2n1 4082,C1(C)(C(N2CCN(C(COCCCC#C)=O)CC2CF)=O)CC(C(C)(C)C)=NO1 4083,C1(C(=O)Nc2cc(C(CC)CC)no2)C2CN(C=O)CC12.C(=O)(C1CC1)OC 4084,N1(C(c2nc(CNC(CSCC)=O)oc2)=O)CCC2(CCCN2C)C1 4085,c1(CNC(C(C)=CC)=O)ccccc1CNC(c1ccsc1CN(C)C)=O 4086,Cn1cnc(C(=O)NC2COCC2CNC(=O)COc2ccon2)cc1=O 4087,c1(C(N(C)CC2CCCC(NC(C(CC)(C)CO)=O)C2)=O)ccc2cnoc2c1 4088,Cc1ncc(N)cc1C(=O)N(CC(C)NC(=O)C(C)NC(=O)Nc1ccco1)C 4089,Cc1cnc(C(C)NC(=O)CCCC2CN(C(C3CC3(F)F)=O)C2)o1 4090,Cc1nc(N2CCNCC2c2ncc(OC(C)C)cc2F)c2ccccc2n1 4091,n1(CC)nccc1C=CC(=O)NC1CN(C(c2cn(C)nc2O)=O)CC1OC 4092,c1(OC2CCN(C(C3CC3C(F)(F)F)=O)C2)cccc(F)c1 4093,c1(C(=O)NC(CNC(c2c(OC)ccc(OC)c2)=O)(C)C)cn2ncccc2n1 4094,C1(C(=O)OC)CCOC1C(=O)NCCCNC(=O)CC1(C)CCC1 4095,[N-]=[N+]=NC1CN(C(C2(F)CCN(C(c3n[nH]c(O)n3)=O)CC2)=O)CC1O 4096,Cc1ccc(C(N2C3CCC2C(NC(C2CC4CCC2C4)=O)C3)=O)cc1C 4097,C1(CC=C)CCCN1C(=O)CC1CCCN1C(=O)CC(C)NC(N)=O 4098,C(=O)(C1CC=Cc2ccccc21)NC1C2CN(C(C#CC3(C)COC3)=O)C(C2)CC1 4099,Cc1nc(CNC(=O)CCc2cccn2C)oc1C(=O)NC(C)Cn1cnnc1 4100,N1(C(C2CC(C(C)C)OCC2)=O)CCC(F)(CNC(C2CN(C)C2)=O)CC1 4101,c1(OC)cc(OC)cc(C(N2CC(NC(c3cc(C#N)oc3C)=O)C(C)C2)=O)c1 4102,C1(NC(C23CC(C)C2C3)=O)CCN(C(=O)CCC2CC2Cl)CC1 4103,Cc1ccc2c(CC(=O)NC3CCC3NC(=O)CCC3C(=O)ON=C3C)csc2c1 4104,C(=O)(C#CC1(CC)CC1)NC(CC)CN(C(=O)CCC(=O)N(CC)CC)C 4105,C=CCCC(C(=O)N1CCCC(O)(COC)C1)NC(C1CCCN1C1CC1)=O 4106,C1(F)(CNC(C(C=CC)O)=O)CCCN(C(=O)C(F)(F)c2cscn2)C1 4107,C1(C(C(=O)NC2C(CCC)C2)CC)CCN(c2nnnn2C(C)C)CC1 4108,Cc1cocc1C(=O)NC(C1CCCCC1)C(=O)NC1(C)CCSC1 4109,CCCS(=O)(=O)CC(=O)N1CCN(C(c2ccc(CN(C)C)[nH]2)=O)C(C)CC1 4110,Cc1nc(CN2CC(C)CC2C(=O)N(C2CC3CCC2C3)C)c(C)o1 4111,CC1CC(C(N2CC(NC(c3c(Cl)noc3Cl)=O)C2)=O)CC(C)C1 4112,C(=O)(CCCCCCNC(=O)C(O)C(F)(F)F)NCCS(CC)=O 4113,N1(C(C(=O)Nc2ccc(F)nc2)=O)CC2(CCN(C(c3cccnc3)=O)C2)C1 4114,c1(CC)c(C(N2CCCC(NC(=O)C(C)c3ccsn3)C2)=O)cnn1C(C)(C)C 4115,C(=O)(C(CO)C(C)C)N(CCCOC1CN(C(CCC(=O)N(C(C)C)C)=O)C1)CC 4116,N1(C(CC2ON=C(CC)C2)=O)CC2CC1CC2NC(c1cc(-c2ccco2)on1)=O 4117,c1(CC(=O)NC2CC(C)(NC(C3N(CC)CCC3)=O)C2)nc2ccccc2s1 4118,C12(C(=O)NC3C(C(C)C)C3)CCCC1CCN2C(=O)CCCN(C)C 4119,c1(C(=O)NCC2CC(OC)CN2C(=O)CCCC(C)=O)ccc2nnn(C)c2c1 4120,C1(CNC(Cc2c(C)scc2)=O)CC2CCC1N2C(C1(C(N)=O)CC1)=O 4121,c1(N2CCC3(C(CNC(c4cc(C)on4)=O)C3)CC2)ccnc2c1CCO2 4122,C1(C(CC)CO)CCN(N2CCC(N(C(=O)CCc3ccccc3)CC(C)C)C2)CC1 4123,C=C=CCCC(=O)NCC1CN(C(=O)C=C(CCC)CCC)C1 4124,Cc1ncc(Br)c(C(N2CCC(NC(c3ccnnc3O)=O)C(C)C2)=O)n1 4125,C1(S(C)(=O)=O)(C(=O)NC(C)CCNC(c2ccc(F)nc2)=O)CCCCC1 4126,C1(C(=O)NC2CC3CC4C(C3)C24)(CC)CCCN(C(=O)COC2CCC2)C1 4127,C1(NC(C2N(C)CC(O)C2)=O)CCC2(CC1)CN(C(=O)CCF)CCO2 4128,c1(C(=O)NCC(C2CCC(F)(F)CC2)OCC)ccc2n[nH]cc2c1 4129,C(=O)(C#CC1CCCOC1)NCC12C(CN(C(Cn3ccc(C)n3)=O)C1)C2 4130,S(=O)(=O)(c1cccc(=NCCc2cnccn2)[nH]1)N(C(C)CC#N)C 4131,C(CCCCCN=[N+]=[N-])NC(CC1(C)N(C(Cc2c(C)ocn2)=O)CC1)=O 4132,CC1(C)C(=O)CCCN1C(=O)CCOCC(F)(F)F 4133,N1(C(CSCCNC(C2C(OC)CCC2)=O)=O)CCOC2(CCC2)CC1 4134,C1(NC(c2c(C)sc(-c3cccs3)n2)=O)CN(C(C2CCC2C)=O)CC12CCC2 4135,c1(C(=O)NCCCNC(c2nnn(C)c2C(F)(F)F)=O)ccc(C2CC2)nc1O 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4153,n1(CCC2(CNC(c3cnsc3)=O)CC2)cc(CNC(=O)C2CC2)nn1 4154,c1(C(=O)NC2CC3N(C(C(CC)OC)=O)C(CC3)C2)cc2ccccc2cc1F 4155,c1(SC)ncc(Br)c(C(=O)NCC2CC(F)CN2C(=O)C(c2ccccc2)F)n1 4156,c1(CO)ocnc1C(=O)NCC(C1CCOC1)NC(C1C(C(=O)OC)C1)=O 4157,C1(CCCNC(c2c(C)c[nH]n2)=O)CCN(C(c2cccnc2C2CC2)=O)CC1 4158,C12(CCCO1)CC=CC=C2.c1(C(=O)NC)coc(C(=O)OC(C2(CC#C)CCC2)=O)c1 4159,C(C(=O)N=S1(=O)CCC2(C1)NC(=O)NC2=O)c1ccc(CC)[nH]1.C1(S)CC2(C1)OCCO2 4160,N1(C(c2c(CC)ncs2)=O)CCC2CCCC12C(=O)N(CC(F)(F)Cl)C 4161,Cn1nc(C(=O)NCCCNC(=O)CC2(C)CC2)cc1C1CCCO1 4162,c1(C(C(=O)N(CCCCNC(C2(CF)CCC2)=O)C)OC)ccc2ccccc2c1 4163,c1(OC)ccncc1COC(=O)Cc1ccncc1Cl 4164,C1(CNC(C=CC=CC)=O)CCCN1C(=O)C(F)n1ccnc1 4165,N1(C(CC(C(F)F)NC(C2(C)CCC2)=O)=O)CCC(F)(F)C(F)C1 4166,O=C(N=c1[nH]nc(Cl)cc1Br)C1CC12CN(C(c1cn3cc(F)ccc3n1)=O)C2 4167,C(=O)(CCC(C)OC)N1C(CNC(CCCOCC)=O)CCC1 4168,CCC(CC)CCCC(=O)C(C(CNC(C(COC)N)=O)O)=O.C(C)(C)O 4169,c1(C(C(=O)NCCCN(C(C(C)(C)OC(C)=O)=O)C)C)ccc(C)cc1 4170,c1(NCCC2(CNC(C3(OC)CCC3)=O)CC2)cc2nnc(C)n2cn1 4171,C1(C(=O)NCCCOCC)CCCN(C(c2nc(C)sc2C)=O)CC1 4172,C1(CC)CCN(C(C2CC=C(C)CC2)=O)C1C(=O)NC1CN(CC(F)F)C1 4173,Cc1ccc(OC(C)C(=O)N2CCC2CNC(=O)CCC=CC(C)C)c(C)c1 4174,C=CC(CC)CC(=O)NC1C2CCN(C(=O)CN3CCCC(C)C3)CC12 4175,C(=O)(C(O)CCCNC(=O)C(C1CCOCC1)F)N1CCC(OC)C1C(C)C 4176,c1(C(N2CCC3C(C(=O)NC(C(C)C)(C)C)C3C2)=O)c[nH]c2ccccc12 4177,CCCC(C)(CC)C(=O)NCC1(O)CN(C(C2(CO)CC(F)(F)C2)=O)C1 4178,C(C)(N=c1[nH]c(=NCC2SCCS2)[nH]c2c1CSC2)C1C(C)C1 4179,c1(C2(C(=O)NC3CCC(CCNC(c4n(C)nnc4)=O)C3)CC2)ccc(Cl)cc1 4180,c1(C(=O)NC(C)C(C)NC(c2csc(O)n2)=O)ccc(-c2cnnn2C)cc1 4181,C(C(=O)N1CC(c2cc(O)no2)C1)(C(C)(C)C)NC(CC1CCN(C)C1=O)=O 4182,C=CC1OCCC1C(=O)NCCC1CCCN(C(c2scnc2Cl)=O)C1 4183,C1(C(=O)NCc2cc(OC)ns2)CCN(C(N2C(SCC)CCCC2)=O)C12CC2 4184,N1(C(C(=O)NC(C)C)=O)CCC2CCC(NC(=O)CCCC(F)(F)F)C12 4185,C1(C(=O)NCC(c2ccccc2)NC(=O)CC2CCC2)CC2(COC(=O)N2)C1 4186,c1(-c2ccc(C(=O)NCCCCOC)nc2)cccc2nn(C)c(C)c12 4187,C1(NC(COCCCC)=O)CCCC1(C)CN(C(=O)CC1CC1C(F)(F)F)C 4188,C1(NC(C=CC(C)C)=O)C2CCN(C(=O)C(C)(C)c3ccno3)CC12 4189,C1(CC(=O)NC(C2CCOC2)C#C)(OC)CN(C(=O)CCSC)C1 4190,c1(C(=O)NC2CC(C)N(C(C3CC(C#N)C3)=O)C2)cc(Cl)c(F)cc1F 4191,Cc1cc(C(=O)NC2(c3cn(-c4ccc(Br)cc4F)nn3)CCC2)cc(O)c1 4192,CC1CCn2c(C(=O)NCC(C)(C)NC(C3CCCN3C=O)=O)cnc2C1 4193,c1(N(C(c2cccc(F)c2)C)C(=O)NC2CCOC2C(F)(F)F)cccc(Br)c1 4194,Cc1ccc(CC(N2CCC(N(C(=O)COC3(C)CCC3)C)C2)=O)cc1Cl 4195,N1(C(CC(C)C)=O)CCC(F)(CNC(=O)Cc2cccs2)C1 4196,S(=O)(=O)(c1cnccc1N1CCCC(OC(F)(F)C(F)(F)F)CC1)NCCSC 4197,c1(C(N2CCCC(CC(=O)N(C)CCN3CC4CC4C3)C2)=O)cnccc1C#N 4198,C(C(=O)NCC1CC(F)(F)CN1C(c1cc(C2CC2)n(C)n1)=O)(C(C)(C)C)OC 4199,c1(C(=O)NCCCOCCNC(C(C(CC)O)(F)F)=O)c([N+](=O)[O-])c(C)nn1C 4200,C1(CC(N2CCN(C(=O)NCc3n(CC)ccn3)CC2)=O)CCC(F)(F)CC1 4201,CC1(C)CCN(C(=O)CC2CCCC2)C(C(=O)CCc2ccccc2)C1 4202,c1(C(=O)NC2(CCCNC(=O)Cn3cncn3)CC2)coc2c1C(O)CCC2 4203,c1(CCC)cc(C(=O)NC2CCC(NC(C3CC4CC3C4)=O)C2)cc(O)n1 4204,N1(C(Cc2c(C)nccc2)=O)C(C(=O)NCC2(C)CSC(C)=N2)C2CC(O)C1C2 4205,N1(C(C(CC2CC2)OC)=O)CCC(C2CCN(C(=O)C(C)(C)CF)C2)CC1 4206,CCC(C(=O)NC(C)CCCNC(=O)C(=O)NCC)C(C)(C)CC 4207,c1(C(=O)NC2COCC2NC(C2CC2F)=O)cc2occc2[nH]1 4208,c1(-c2ccc(C(N(C(C)(C)C)CC)=O)cc2)ccc(F)c(C)c1 4209,S(=O)(=O)(c1ccc(C=CCC2OCCC2)cc1)NC(C(=O)N(C)CCC1CC1)=O 4210,Cc1ccc(C=CC(=O)NCCC2(C(=O)NC3CCN(C)CC3C)CC2)cc1 4211,C(CC(C(=O)N1OC2CCC1CC2)NC(c1cncnc1C)=O)=CC 4212,Cc1nc2cc(C(N3CC4CC3C4NC(C3COCCN3C)=O)=O)cnc2[nH]1 4213,c1(CCC)ccc(C(N2CC(N(C)C)C(C)C2)=O)cc1.c12ccccc1SC2 4214,N1(C(CC2C(C)C2)=O)CCN(C(c2cnc(Br)s2)=O)C(C)C1 4215,C1(C(=O)NC(C(=O)OC)C)CCC(C)(C)N(C(=O)C(O)c2ccco2)C1 4216,CC(CC(F)F)C(=O)N1C(C(=O)N(CC(=O)NC(C)(C)C)C)CCC1C 4217,N1(C(C=Cc2c(C)ccs2)=O)CCC(C)(C)C(CNC(=O)C(C)C(C)C)C1 4218,c1(C(=O)NCC2CCN(C(C3CSCC(=O)N3)=O)C23CC3)cn2ccccc2n1 4219,N1(C(C2C(C(=O)OC)CC=CC2)=O)CCC2CN(C(=O)C(=C3CCCCC3)F)C2C1 4220,c1(C(=O)NCC(CNC(COCCCOC)=O)C(F)(F)F)cc(C)c(F)c(C)c1 4221,C1(C(N2CC(NC(c3cnco3)=O)C2)=O)C2CCC(C2)C1NC(=O)C1CC1 4222,c1(C(C)NC(C(=O)Nc2c(CC(C)C)cccc2)=O)nc2ccccc2s1 4223,C(C(CC(=O)NCC1CCCN1C(c1cnc2ccsc2c1)=O)C(F)F)N(C)C 4224,c1(C(C(=O)NC(C(C)=O)Cc2ccccc2)=O)c[nH]c2ccc(F)cc12 4225,C12(N(C)C)CCC(C(N3CCCC(NC(C4CCCSC4)=O)C3)=O)(CC1)CC2 4226,C1(NC(CN2C(C)CCC2)=O)CC=C(C(=O)NCCCc2cn[nH]c2)C1 4227,c1(C(=O)OCCOCCCSC)cc(CNC(=O)N(C)C(C)C)ccn1 4228,c1(OC)c(Cl)ccc(Cl)c1C(=O)NC1CN(C(=O)C(C)OC2CCOC2)C1 4229,c1(C(=O)NC2CN(C(C3CC(=O)N(CC4CC4)C3)=O)C2)cc2c(s1)CCOC2 4230,C(C)(C)(CC(F)C(=O)NC1CC(CO)C2CC12)NC(C(n1c(C)ccn1)C)=O 4231,c1(C(=O)NCCCCCNC(Cc2nc(C)[nH]n2)=O)ncnc2sccc12 4232,S(=O)(=O)(c1ccc(N2CCC(NC)CC2)c2cnccc12)N1CC(C)(CC)OCC1 4233,C1(NC(C(C=CC)O)=O)CN(C(=O)CNC(=O)NC2CC2)CC1c1nccn1C 4234,N1(C(C(C)C2(O)CCC2)=O)CCCC(CNC(c2ccnn2C(F)F)=O)C1 4235,Cc1ccc(C#N)c(NC(=O)CC2CN(Cc3ccc4c[nH]nc4c3)CCO2)c1 4236,CCC(CC(F)(F)F)C(=O)N(C)C(C)C.c12cc(Br)c(OC)cc1OC2=O 4237,N(C(=NCCCCl)NC1CCN(C(C)C)C1)S(C)(=O)=O.Cc1nnsc1C 4238,C(C)(C(=O)NC1CCC(n2cc(-c3ccc(C)nc3)nn2)CC1)(C(C)C)OC 4239,c1(C(=O)NCCC(C)N(C(CSCCC(C)C)=O)C)csc(N=S(C)(C)=O)n1 4240,C1(C(=O)NC(c2occ(C(N(C3CCOC3)CC)=O)n2)C)CC(C)N(C)C1 4241,C1(C(=O)NC(CNC(c2ccc(SC)s2)=O)C)CCCN(C)C1=O 4242,c1(COCC(N2CC(O)(C(C)NC(CC=CC=C)=O)C2)=O)ccccc1Cl 4243,c1(NC(c2cccc(C)c2)c2n(CC(=C)C)nnn2)cccc(C(=O)N(C)C)c1 4244,C(=O)(CCCCCS(N)(=O)=O)NCC(C)CNC(c1ccc(CN(C)C)o1)=O 4245,C(=O)(CC1=NNC(=O)C1)NC1CN(C(c2n(C)cnc2)=O)CC(O)C1 4246,Cc1cccc(F)c1C(N1CCN(C(=O)C(c2ccc(Cl)cc2)N)CC1C)=O 4247,N1(C(C(COC)C)=O)CCCC12CCN(C(C1CCC(=O)C1)=O)CC2 4248,c1(CC(C(=O)NC2(CC)CCOC2)C)ccc(OC)c(OC)c1 4249,c1(C(=O)NC2C(CO)CCN(C(C3NC(=O)OC3)=O)C2)cnn2c1OCCC2 4250,[N-]=[N+]=NC1CCC2(C(=O)NC3CC(F)C3)CC12 4251,N1(C(c2cc(C(C)=O)[nH]n2)=O)CCC(C2(NC(=O)CCN(C)C)CC2)CC1 4252,c1(C(=O)NCC2CC3CC3N2C2CCCC2)nc(Br)c2ccccc2n1 4253,C1(NC(c2c(CC)n(C)nc2)=O)CCN(C(=O)Cc2cc(Cl)ccc2Cl)C1(C)C 4254,c1(C(=O)NCC(C23CCC(CC2)C3)NC(CC=C=C)=O)ccc2ncncc2c1 4255,N1(C(C(C)OCCc2ccc(F)cc2)=O)CC2CC2(c2ccccc2)C1 4256,N1(c2cc(C)nc(Cl)n2)CC2CC1CCC2NC(=O)CC(C)C1CCCCC1 4257,CC1CC(C(=O)N(CCC(C)NC(C2CCC(C(F)(F)F)O2)=O)C)CC(C)C1 4258,C1(C(=O)NC2CC(CNC(CC=C(C)C)=O)C2)CCc2ccccc2O1 4259,C12(C(=O)NCCC(C(C)C)NC(=O)C(C)(C)c3cc[nH]n3)COCC(C1)OC2 4260,c1(NC(Cc2ncc(-c3ccc(OC)nc3)cn2)=O)ccc(Cl)nc1Br 4261,C1(C(N2CC(n3ncc(NC(C4CNC4)=O)c3)C2)=O)COCCN1C 4262,N1(C(C(CC)NC)=O)CCSC(C(N2CCC(c3cncc(C)c3)CC2)=O)C1 4263,n1(C(C)C)nnc(C(=O)OCCc2ccc(-c3ccccc3)cc2)c1C(=O)N(C)C 4264,N1(C(C=CC(=O)N(C)C)=O)CCC(C)(C)C1CNC(=O)C=CCF 4265,c1(C(N2CCC(C(C)NC(C3(CO)CCCO3)=O)C2)=O)cc2c(cn1)OCCC2 4266,c1(C(=O)NC2C(CNC(CCCOCC=C)=O)COC2)cncc(F)c1 4267,CC1CN(C(C2CCC3(CCC3)O2)=O)CCN(C(=O)CCc2cn[nH]c2)C1 4268,C(=O)(C(CC(C)(C)C)NC(=O)C1=C(C)OCCC1)N1CC(CCC)C(OC)C1 4269,c1(C(C(=O)NCC(C)(C)NC(c2c(C)con2)=O)O)cc(F)cc(F)c1 4270,S(=O)(=O)(c1ccc(Cl)cc1)N1CCCC(CC=C)(C(=O)NC(C)CO)C1 4271,c1(C(CNC(=O)C2CC2)NC(=O)CC(c2cccc(F)c2)O)cc(F)cc(Cl)c1 4272,C1(C(C)NC(=O)CCCc2cncs2)CCCCN1C(=O)Cn1cnc(C(N)=O)n1 4273,CC1(C)C(C(F)F)(NC2CNC3CC23)CCO1 4274,C1(CNC(C(C)NC(c2ccco2)=O)=O)CC12CCN(C(=O)C=C1CCC1)CC2 4275,CCCC(O)C(=O)N(CC)CC1CCCN(C(=O)C(C)CC2CCCCC2)C1 4276,CC(C)CCN=C(NCC(C)CN1CCOCC1)NC1CCCOC(OC(F)F)C1 4277,N1(C(C2CC(OC)CC2OC)=O)CCC2(C1)CN(C(=O)C(C)(C)CC(C)=O)CCO2 4278,C1(C(=O)OC)CCCCN(N(CCCO)C(=O)C2Oc3ccccc3C2C)C1 4279,C(=O)(CCP(C)(C)=O)N(C(C)C)CCN(C)C(C1(c2cccc(Cl)n2)CC1)=O 4280,CCCCC(F)C(=O)NCC1CCCCN(C(=O)C(N2CCNC2=O)C)C1 4281,c1(C(N2CC(C)(C(=O)Nc3cncnc3O)C2)=O)cc(F)cc(Cl)c1 4282,CC1(CCNC(=O)CC2(O)CCCC2)CCN(C(C23CC(F)C2C3)=O)C1 4283,N1(CC(=O)NC2C(OC)CN(C(c3ccccc3F)=O)C2)CCCCC(O)C1=O 4284,c1(NCc2ccc(OCC)nc2)c(C)nn(C2CC2)c1C(F)(F)Cl 4285,N1(C(c2cc(C)ns2)=O)CC2CCC1C1CN(c3c([N+](=O)[O-])c(C)nn3C)CC21 4286,c1(OC)cc(C)ccc1C(N1CC2CC1C2NC(c1ccnnc1)=O)=O 4287,c1(C(=O)NCCN(CCC)Cc2ccc(O)c(O)c2)cc2cc(C)ccc2s1 4288,CC1COCC(C(=O)NCC(C)CN(C(=O)Cc2cccc(Cl)c2)C)O1 4289,C1(C(=O)NCC2(C(C)NC(CC(=C)C)=O)CC2)CCC2(CC1)CC(=O)C2 4290,c1(C(=O)NCCC2N(C(C(C)C#N)=O)CCCC2)cc(-c2cc[nH]n2)ccc1F 4291,c1(C(=O)NCC2CC(OC)CN2C(=O)CN(C)C(C)C)ccc2c(c1)N(C)CC2 4292,C(CCCCCNC(C1(C(C)(F)F)CCC1)=O)NC(C(=Cc1cccs1)C)=O 4293,c1(C(N(c2cccc(Cl)c2)CC)=O)cccc2c1OC(C)C2 4294,n1(CCC(=O)NCC2CN(C(c3cnccc3Cl)=O)CCO2)cnc([N+](=O)[O-])c1 4295,c1(CN(C)C(C2CCN2C(C2CCCC2O)=O)=O)nccn1C 4296,c1(CC)ccncc1C(N1CC(n2cc(CCNOC(C)=O)nn2)C1)=O 4297,Cc1ccc(CC(=O)NC(C)CNC(C2CC2c2cccnc2)=O)c(Cl)c1 4298,c1(C(=O)NC2CCOC2)cnn(-c2ccncc2)c1.C(C)(C)(C)OC(=O)NCC 4299,Cc1n[nH]cc1C(N1CCC(C(C)(C)NC(=O)C(C)(Cl)Cl)C1)=O 4300,Cc1nc(NC2CN(C(c3ccc(Cl)nc3C)=O)CC2C)c2sccc2n1 4301,C(CCCCNC(C1(n2cc(-c3ccc(C(=O)O)o3)nn2)CC1)=O)N(C)C 4302,N1(C(C(C)=C(C)C)=O)CC2CCCCC2(NC(c2cc(C(N)=O)cc(F)c2)=O)C1 4303,N1(C(c2nc(CC)oc2C)=O)CC2CC1CN(C(C1CCC(C(N)=O)CC1)=O)C2 4304,C(=O)(CC(c1ccccc1)C1CC1)NCCC(C)N(C(CCNC(C)=O)=O)C 4305,N1(C(CCN2CCC(C)CC2)=O)CCC(NC(c2cccc(=O)o2)=O)C(CO)C1 4306,N1(C(C=C(C)C)=O)CCCC2(NC(=O)C3=CCOCC3)CC2C1.C12CCCN1C2 4307,c1(CNC2CC(C(N3CCC(F)C3)=O)C2)cnn(-c2ccccc2)c1 4308,c1(CC(=O)NCCC2CN(C(=O)CCC(F)F)C2)ccc(O)cc1 4309,CCC(C)CCC(O)CC(=O)NC1(CNC(C2CCCN2CC(C)C)=O)CCC1 4310,C#Cc1cc(C(C(=O)NCC2CCOC2)N(CCC#N)C2CC2)cc(Br)c1.C 4311,N1(C(C2C(CC(C)C)C2)=O)CCC(NC(=O)Cc2ccc(C)cc2C)C(C)(C)C1 4312,C(C(CC1CC1)C(=O)N1CCCC1CC)NC(CC1CC(=C)C1)=O 4313,c1(CCN(C)C)ccc(C(=O)NCC(CO)NC(c2occc2C2CC2)=O)cc1 4314,c1(OC)cccc(F)c1CN1CCCCC1c1cn(-c2cccc(C)n2)nn1 4315,c1(C(N2CC(CNC(C3C(C(=O)OC)C3)=O)(CO)C2)=O)c[nH]cc(F)c1=O 4316,CCCCCC=CC(=O)NCCOCCN(C)C(c1cc(C)no1)=O 4317,N1(C(C(CC#C)O)=O)CCC2(CC1)CN(C(c1cc(OCC)no1)=O)CC(C)O2 4318,Cc1ccc(C(N2CCC(CC(=O)NCCn3ccnc3C)C2(C)C)=O)cc1C#N 4319,C1(NC(=O)C=Cc2ccc(C(F)F)o2)CN(C(=O)C(O)C2CC2)CC2(CCC2)C1 4320,C(CC(C)(C)C(=O)N1CCC(OCCO)C1)OC(C(C)SCCCC)=O 4321,Cc1ccc(F)c(NC(C2CCCCCN2C(C2CC23CCCCC3)=O)=O)c1 4322,CC1CCC(N)NC(CC(=O)N)CCCCN2C(CCN1C(C)=O)C2 4323,CCCC(C(=O)OC)C(=O)NC1CC(CNC(c2cc(Cl)ns2)=O)C1 4324,Cc1nn(C)cc1CC(=O)NCC1COCCN1C(C1CC(CC(F)(F)F)C1)=O 4325,C(=O)(C(C)(C)Cn1cccn1)NCC1CN(C(C(C)c2ccsc2)=O)C1 4326,C1(NC(C=C(C)CNC(=O)CC2CCCC3CC23)=O)CC(C(=O)NOC(C)C)N(C)C1 4327,C1(C(=O)NC2CCN(C)C(=O)C2)CC12CCN(C(=O)C#CC1CCOC1)CC2 4328,c1(C(C)=O)ccc(C(N2CCCC2CCc2cn(C(C)(C)C(=O)O)nn2)=O)s1 4329,C(=O)(CCCN(C)C(c1cc[nH]n1)=O)NC(C)CSC(F)F 4330,N1(C(Cc2nc(C)oc2)=O)CCC2(CC1)CN(C(c1n[nH]c(C)c1O)=O)CCO2 4331,C(=O)(C(C)(C)S(C)(=O)=O)NCC1C(C)(C)C1CNC(c1cc2c(s1)CCCC2)=O 4332,C#CC1(O)CCCC(NC(C2(c3ccnc(F)c3)CC2)=O)C1 4333,c1(C(=O)NCC(F)CNC(c2coc(Cl)n2)=O)cccc(N2CCOC2=O)c1 4334,c1(C(=O)NCc2c(C(=O)NC3CC(C)SCC3)occ2)n[nH]c2ccccc12 4335,c1(NC(C2N(C(C(C(C)C)O)=O)CCCC2)=O)cc(Cl)c(Cl)c(Cl)c1 4336,c1(C(C(=O)NC2CC(C)(NC(c3c(CC)scc3)=O)C2)C)c(C)n[nH]c1C 4337,c12ccc(o1)C(=O)NC2.c12ncnn1C2.C(CC(=O)NC(C)C)SCC 4338,Cc1c(C(=O)NCC2CCCCC2NC(=O)C2=CCCCC2)c(C(F)F)nn1C 4339,c1(CC2(CC(=O)NCCCNC(C3C(CC)CCCC3)=O)CC2)ccc(C#N)nc1 4340,C1(N(C)C(c2cc(F)ccc2F)=O)CN(C(=O)CN2CCS(=O)CC2)CC1(C)C 4341,CC1(C)CC=CCN(C(C23CC(CN(C(c4sccc4F)=O)C2)C3)=O)C1 4342,c1(C(N2CCC(O)(CNC(c3c(CC)n(C)nc3)=O)C2)=O)c(C)ccc(C)c1C 4343,CC1CCC(CNC(=O)CC2CS(=O)(=O)C2)CN1C(=O)CCSCC(N)=O 4344,C1(NC(C=C(C)C2CC2)=O)CCN(C(=O)CC2CCCCO2)C12CCCC2 4345,C(CC(C(F)F)c1ccccc1)Cc1nnnn1C1CCCC1.CC(C)CCN 4346,c1(C(=O)NCC2OCCN(C(CC=C=C)=O)C2)nc(Cl)ccc1OCC=C 4347,C(CCC(C)C(=O)NCC12CCC(CC1)N2C(=O)CCC1OCCO1)OC 4348,C1(CNC(c2c(CC)onc2)=O)(NC(=O)COc2cc(C)on2)CCCCC1C 4349,c1(C(=O)NCC(CO)NC(C2SCC(=O)C2)=O)ccc(F)c(Cl)c1 4350,c1(CC)ccc(NC(C2CC23CC(NC(c2cc(COC)[nH]n2)=O)C3)=O)cc1C 4351,c1(C(=O)OC)ccnc(Br)c1.c12ccsc1NC(=O)C1CC(C1)C(=O)NC2 4352,C(=O)(CCC(CF)CF)NC(CC)C(=O)N(C)CCOC 4353,c1(CCCC(=O)NCC(CNC(c2c(C)occ2)=O)CO)ccccc1F 4354,C(CN=c1ccnc(NCc2cccc(N3CCC(SC)CC3)c2)[nH]1)OC 4355,c1(CCCCOC)cn(C(CC2CC2)C(=O)NCc2[nH]nnc2C2CC2)nn1 4356,c1(C(N2CC(C)CC(NC(c3c(CC)noc3)=O)C2)=O)c(Cl)cc(C#N)cc1Cl 4357,C1(NC(C(F)=C(C)C)=O)CC2CCC1CC2NC(c1cc(O)nc(O)n1)=O 4358,N1(C(CC(C)NC(N)=O)=O)CCCOC(CCNC(=O)C(C)(C)CC2CCC2)C1 4359,Cc1cccn2c(=O)cc(CN3CCOC(c4ccc(F)c(Cl)c4)C3)nc12 4360,c1(OCC)ccc([N+](=O)[O-])cc1NC(C1CCCC1NCC1CCCCO1)=O 4361,C1(=O)CCCCCCCC23C(C(=O)OCC)(CN1C2)C3.C(C)(C)(C)OC.C(=O)OC 4362,CC1(C)COCCC1Cn1cc(-c2cccc(C(F)(F)F)c2)nn1 4363,c1(CCC(=O)NC2(c3cn[nH]c3)CN(CCSCC=O)C2)ncccc1C.CO 4364,Cc1cc(=O)oc2cc(NC(C3CC(=O)N(c4cccc(F)c4F)C3)=O)ccc12 4365,n1(CC#C)cccc1C(c1nnnn1C(C)(C)C)NC(c1cnsc1)C 4366,CCC(CC)C(C(=O)NCCCN(C(=O)CCC1NC(=O)NC1=O)C1CC1)OC 4367,C1(NC(c2ccc(C)c(O)n2)=O)CC2CCC1N(C(c1coc(C#N)c1)=O)C2 4368,C=CCC(C(=O)NOCC1CC1)NC(=O)C(c1ccc(O)cc1)CC 4369,C1(C)(C(=O)NCC(C)OCC)C=CCN1C(=O)C(C)C1CC1 4370,C1(NC(C23CC(NC(C(COCC)C)=O)(C2)C3)=O)CC1C1CCCC1 4371,CCC(C)CC(C)C(=O)N(CC(CO)(CO)NC(c1ccnc(OC)c1F)=O)C 4372,c1(C(N(CC(C)NC(C2C(C=C)C2)=O)CC)=O)cccc(OCc2cccs2)c1 4373,C12(C(=O)NCC(CC(C)C)(C)NC(=O)CSC3CC3)CCCN1S(=O)(=O)CC2 4374,C1(COC)(CNC(C2CCC2C#N)=O)CN(C(=O)Cn2[nH]cnc2=N)C1 4375,CC(CC(=O)N(CC(=O)NCc1nc(C(N)=O)co1)C1CC1)n1cccn1 4376,CCCC(CCC)C(=O)N(C)CC1CCN(C(=O)CNC(c2cccnc2)=O)C1 4377,N1(CC(=O)NCCN(CCC)C(C2CCCOC2C(C)C)=O)CCC(=O)NC1=O 4378,Cc1c(NCC2CCOC2)ncnc1N1CCCN(c2ccc(C#N)cn2)CC1 4379,C1(NC(=O)CC2(O)CCOC2)CC2(CCN(c3ncnc(Cl)c3F)CC2)C1 4380,c1(C(C)(F)F)cccnc1NC(=O)NCC1CCN(c2ccccc2F)C1 4381,N1(C(CCCN(C)C)=O)CC2CCC(C1)N2C(c1cc(=O)n(C)o1)=O 4382,c1(C(=O)NCC2CC(n3ccnn3)N(C(=O)CCCF)C2)cccc(Cl)c1 4383,N1(C(C=C(C)C)=O)CCC2CCC(C1)N2C(=O)CC(C(C)C)c1ccon1 4384,N1(C(CC=CCCCCC)=O)CCC2CCCC12C(=O)NC1(C(=O)NC)CC1 4385,C(CC(O)C(=O)N1CCCCC1CN(C)C(c1cccc(C2CC2)n1)=O)SC 4386,N1(C(CNS(NC)(=O)=O)=O)CC2COCC(C1)C2NC(=O)C(C)n1cccn1 4387,C1(C(N2C(CNC(c3ccon3)=O)CC(F)(F)C2)=O)CC2COCC(C1)C2 4388,CC1=CCSC1C(=O)NC1(C)CC(C(=O)NC(C)(CO)C2CCC2)C1 4389,C(=O)(CC(C)NC(=O)C(C)n1ccnc1)N(C(C(=O)NC)C)C 4390,C=CCC(C(=O)NCC1(C)CCCN(C(c2sccc2SC)=O)C1)C(C)C 4391,N1(C(c2cn(CC)nc2C)=O)CC(F)(F)CC1CNC(c1cc(F)ccc1F)=O 4392,c1(C(=O)NC2CCN(C(c3[nH]c(=NC)sc3)=O)CC2C)c[nH]c2cc(O)ccc12 4393,C1(C(N(CC=C)CCO)=O)(CC)CCCN1C(=O)Cn1nc(C)oc1=O 4394,Cc1ccc(CC(=O)NC(C(N2CCOC(CSCCC(C)C)C2)=O)C)cc1 4395,c1(C(=O)NCC2C(NC(c3ccc(F)s3)=O)CCCC2)nccc2ccncc12 4396,C(=O)(NNC(=O)C(C)(C)CCCCNC(C1(C)C=CCC1)=O)C1CC(C)OC1 4397,c1(N2C(C)CC(NC(=O)CC3CCC(C4CC4)O3)C2)ncnc2[nH]ccc12 4398,C1(NC(c2ccc(CC(C)C)s2)=O)CN(C(c2cc(=O)n(C)o2)=O)C2(CCC2)C1 4399,C1(C(=O)NC(C(C)(C)C)CNC(=O)CNC(=O)C2CC2)CCC2C(CC1)C2(F)F 4400,Cc1ccc2c(Br)cnc(N3CCNC(=O)C(F)(F)C3)c2c1 4401,CN=c1nc(N2CCC(OCC(C)C)C2)[nH]c(N(C)CC2COCCO2)n1 4402,c1(OCC)ccc(C(=O)NC(C)C(C)NC(c2cc(Cl)ccc2F)=O)cc1OC 4403,N1(C(CC(C)C)=O)CCC(CNC(C2(CN(C)C)CCOCC2)=O)C(C)C1 4404,N1(C(C2CC(=O)OC2)=O)CCN(C(C2(CF)CC(F)(F)C2)=O)CC1CC(F)(F)F 4405,CCCC(CC)CCC(=O)NC1C=CCN(C(=O)C(C2CC2)SC)C1 4406,C1(NC(CCc2ccnc(C)n2)=O)C2CCC1N(C(=O)Cn1ncc(O)nc1=O)C2 4407,c1(C(N2CC3(C(NC(C(C)=C(C)C)=O)CC3)C2)=O)cc(C)c2n[nH]cc2c1 4408,Cn1c(C(N2CCN(C(c3cccc(CO)n3)=O)CC2)=O)cnc1O 4409,c1(C(C)C)nn(C)cc1C(=O)NCC1CN(C(c2csc(C3CC3)n2)=O)CCO1 4410,C(=O)(C(O)CC(C)(C)C)NC1C(C)N(C(=O)Cc2c(F)cccc2Cl)CC1 4411,C(=O)(C(C)(C)CC(=O)NC1CC(NC(C2CCCN2C(=O)OC)=O)C1)OC 4412,c1(C(N2C(C(C)(C)CNC(C3CC4CC4C3)=O)CCC2)=O)cccc(Br)c1Cl 4413,N1(C(C(CC)C(C)C)=O)CC(NC(=O)C=C(C)C2CC2)CC2(CCC2)C1 4414,c1(C(=O)NCC2C(CNC(C3(C(C)(C)O)CC3)=O)C2)ccnc2[nH]c(O)nc12 4415,n1(CC(=O)NCC(CNC(c2c(CC)nc[nH]2)=O)CO)cc(Cl)c(C)n1 4416,N1(CC(N2C(C3(CNC(C(C)NC(CC)=O)=O)CC3)CCC2)=O)CCNC(=O)C1 4417,C1(NC(=O)C2CC2)CCC2CN(C(C3CC4(CCOCC4)CO3)=O)CCC2C1 4418,c1(C2(C(N(CC(C)(C)NC(CCCOC(C)=O)=O)C)=O)CC2)ccc(Cl)c(F)c1 4419,N1(C(CC(C(C)C)O)=O)CC2CN(C(c3ccncc3-n3cccn3)=O)CC2C1 4420,c1(C(O)N)ncccc1NC(=O)Nc1cn(CC(F)F)nn1 4421,c1(CNC(CN(C(C2CC(OCC)C2)=O)CC)=O)nccc(O)n1 4422,N1(C(CN2C(C)CC2)=O)CCC2(C1)CN(C(c1ccc3nccn3c1)=O)CCO2 4423,N1(C(C(C)OC)=O)CCC(C(C)(C)NC(C2CC2C)=O)CC1 4424,C1(CN(CCC=C2CCN(C)C2)C)CCN(C(=O)Cn2nnc(C3CC3)n2)CC1 4425,C12(NC(CN(C(=O)OC)C)=O)CCC(CC1NC(=O)Cc1sc(C)nc1C)C2 4426,C(=O)(CCC(C)=O)NC(c1cnn(C)c1)C(N1CC(CC)(OC)C1)=O 4427,CC1(C#N)CC(c2nnnn2CC2CCOC2)(NCc2cscn2)C1 4428,c1(CC(=O)NC2C(NC(CC3ON=C(C)C3)=O)CCC2)ccc(=O)n(C)c1 4429,CC1(C)CCC(N=c2cccc(S(=O)(=O)NC3CCC4(CC3)CC4)[nH]2)CC1 4430,N1(C(C2CC(F)(CC)C2)=O)CCN(C(=O)COCC2CCC2)C(CC)C1 4431,Cc1cc(N(CCC(N)=O)C)nc(NC(C)Cn2nccc2C)n1 4432,c1(NC(CC(C)NC(C(CC=C)C)=O)C)ccc(Br)c(C(=O)OCN(C)C)c1 4433,N1(C(Cc2cn(C)nc2)=O)CCOC(CO)C1.c12ccccc1c1cn2nn1 4434,C(=O)(C(CC)C(=O)OC)N1CCC(N(CC#C)C(C2CC(=O)N(OC)C2)=O)C1 4435,N1(C(C=C(C)Cl)=O)CCN(C(C2CCCN2C)=O)CC1c1cc(F)cc(F)c1 4436,Brc1cccc2c1C(NCC1CC1Br)CO2 4437,C1(NC(c2c(C)nsc2)=O)CCN(C(c2cscc2-c2ccccc2)=O)CC1F 4438,c1(C(N(C)CC2CCCN(Cc3ccc(C)cc3Cl)C2)=O)cc(I)cn(C)c1=O 4439,C1(C(=O)NC(CCC=C)C)CCC(NC(=O)C(O)CN2CCCC2)CC1 4440,N1CCC(n2cc(-c3nn(C)cc3C(=O)O)nn2)C(O)C1.C(C(C)(C)C)=C(C)C 4441,n1(CC(N2CC(CC)C(NC(=O)CNS(N)(=O)=O)C2)=O)nc(Cl)ccc1=O 4442,N1(C(CC=CC=C)=O)CC2CCCC1CN(C(c1cc(C)ccc1Cl)=O)C2 4443,C(CCN=c1[nH]cnc(N2CCOCC2)c1Br)c1cncc(OC)n1 4444,N1(C(c2ccnn2CC2CC2)C(=O)NCCCOC)CCC2CCOCC2C1 4445,CCS(=O)(=O)CC(=O)N1CCCC1(C(=O)NC1C=CCCC1)CC 4446,C1(C(=O)NCC2(F)CC(CNC(c3c(C)con3)=O)C2)CCCCC1F 4447,c1(CCC(=O)N(C2CCN(C(c3[nH]cc(C)c3C)=O)C2)CC)ccc(F)cc1F 4448,N1(C(C2(COC)CC=CC2)=O)CCC(C)(CNC(C2COCOC2)=O)C1 4449,C1(C(N2CCC(OC)(CNC(c3cncc(CO)c3)=O)C2)=O)CC(=O)NC(=O)N1 4450,CC1(C)CCC(C(=O)NCC(=C2CN(C(C3(CC4CC4)CCC3)=O)C2)F)OC1 4451,Cc1cc(N(C)Cc2ccc(Br)c(F)c2)nc(=NCCCOC(=N)O)[nH]1 4452,N(C)(S(=O)(=O)N1CCN(CC(=O)NCCOC2CC2(F)Cl)CC1)CC 4453,CCC(CNC(=O)C=Cc1ccccc1C)(CC)C(=O)N1CCC(C(N)=O)C1 4454,N1(C(c2cnc(C(C)C)s2)=O)CCCC(N(CCF)C(C2CCC(=O)NC2)=O)C1 4455,C(=O)(CC(C)(O)COC(C)=O)NCC(C)NC(COCC(=O)OC)=O 4456,c1(NCc2c(C)nn(C)c2Cl)[nH]c(=NC(C)CN2CCCC2=O)nc2c1ncn2C 4457,C(=O)(C(C(C)C)C1CCC1)NCC1(OC)CN(C(c2cnc(O)o2)=O)C1 4458,Cn1ncc(C(=O)OCCc2ccccc2I)c1C1CCC1 4459,c1(C(=O)NC(C)C(N2CCN(C(=O)Cc3cncnc3)CC2)=O)ccc(F)cc1F 4460,C1(OC)(CNC(C2(F)CCN(C(=O)Cn3cnnc3)C2)=O)CCCCC1 4461,C1(O)(CNC(C(N2CCNC2=O)C)=O)CCCN(C(=O)CCc2cnn[nH]2)CC1 4462,C1(C(=O)NC2CC(F)(CNC(C(C)OCC)=O)C2)CC(C)(C)CC(C)(C)C1 4463,c1(C(N2CC(C)(CNC3CCCN3N=O)C2)=O)cc2ccccc2nc1O 4464,C(=O)(C(C(C)(C)O)NC(=O)CC1CCSC1)NCC(CC)CC 4465,c1(C(=O)NCC2CC(F)(CNC(C3(CCCC)CC3)=O)C2)cnn(CC)c1C 4466,C1(C2CCN(C(=O)CN(C)C)C2)(NC(=O)CCNC(=O)Cc2ccccc2Cl)CC1 4467,C1(NC(CCCC)Cc2nccn2C)CCc2cc(C#N)ccc2C1 4468,CC(C)C(CCN(C(=O)CC1C(C)C1(F)F)C)NC(c1cnc(S)n1C)=O 4469,c1(C(=O)NC(C(N2CCC(CN=[N+]=[N-])C2)=O)C2(O)CCC2)cncc(Cl)c1 4470,C(N=c1nc(N2CCC(=NO)CC2)c2c([nH]1)COC2)c1[nH]nc(O)n1 4471,N1(C(C2OCCN(C)C2)=O)CCC2(CC1)CN(C(c1ncccc1N)=O)CCO2 4472,c1(C(=O)OC)ccc(C(=O)NCC2CC2CNC(c2cc(Cl)no2)=O)cn1 4473,O=C(C1CCCc2ccnn21)OCCc1cnc(O)n(-c2ccccc2)c1=O 4474,N12CCOC(C1)CC2=O.C=C1CC(CC(=O)NCC(CC)N(C)C)C1 4475,c1(C(=O)NC(C2CCOC2)CNC(C(C)(C)C(N)=O)=O)csc2c(F)cccc12 4476,CC1CCN(C(=O)CN2CC3CCC2C3)CC1CNC(c1cc(Cl)on1)=O 4477,c1(NCc2n(C)nnc2Br)[nH]c(=NCCC2CCC(O)C2)nc2c1cnn2C 4478,C12CN(CCC1O)C2.C1(C(=O)O)CCCN(c2cccnn2)C1 4479,N1(C(CC2C(=O)NCCC2)=O)CCCC(Cl)(O)CC1 4480,N#Cc1ccc(C(=O)NC2(C(N3CCC3CO)=O)CCSC2)s1 4481,CN1C2(CCNCC2)C(C(=O)Nc2ccc(OCC(C)(F)F)cc2)CS1(=O)=O 4482,C1(CNC(Cc2cc(C)sc2)=O)COCCN1C(c1cnc(C2CCC2)s1)=O 4483,C(=O)(C(CCC(C)C)NC(=O)C=C(C)C(F)F)N1C(CC)CCC1 4484,N1(C(C(Cc2ccsc2)NC(c2cnc(C3CC3)o2)=O)=O)CCC12CCCC2 4485,n1(C(C(=O)NC23CC(NC(c4onc(C)n4)=O)(C2)C3)C)nc(C)cc1C 4486,CCC(C)(CO)NC(=O)COC1CC(NC(=O)CC2CCC(=O)N2)C1 4487,c1(N2CCC(c3cc(F)c(OC)c(F)c3)C23CCC3)ncc2cc(Br)cnc2n1 4488,N1(C(=O)OC(C)(C)C)CCC=CC1NC(=O)OCC12CC(C(C)(F)F)(CO1)C2 4489,Cn1nc(C(N2CC3CCC(C2)N3C(=O)CSC(F)(F)F)=O)c2c1CCSC2 4490,c1(CC(=O)NCC23C(CN(C(CC=C)=O)C2)CC3)ccc(F)cc1[N+](=O)[O-] 4491,C12(C3CCN(C3)C(=O)N1)CC2.C(=O)(CSC(C)(C)C)OC.C1(=O)COC(=O)CN1 4492,C1(CCC(=O)NCC(CO)NC(=O)CSc2nncn2C2CC2)CCC(O)CC1 4493,C1(CNC(C2C(=C)C2)=O)(COC)CCN(C(c2cc(C)ccc2N)=O)CC1 4494,N1(C(C2(C#C)CC2)=O)CCC2(CCCN2C(c2ccc3c(c2)CNC3=O)=O)C1 4495,Cc1cnc(C(=O)N(C2CN(C(c3cnnc(O)c3)=O)CC2F)C)c(Br)c1 4496,N1(C(=O)Cc2ccno2)CCC2CN(C(C3CCCC34CCC4)=O)CC2C1 4497,N12CC(CC(C)C1)C2=O.c1(CCCCC)cn(Cc2cnn(CC)c2)nn1 4498,C(=O)(CCCC(=O)C(C)(C)C)NC(C)C(C)(C)NC(c1c[nH]c(Br)c1)=O 4499,c1(C(N(CCNC(C(C)P(C)(C)=O)=O)CC2CC2)=O)cnc2ncnc(O)c2c1 4500,c1(C(=O)NCCCCCCNC(C(C)c2ccco2)=O)cc2n(n1)CCO2 4501,N1(C(C=CCCC)=O)CCCN(CCNC(C2CCCC(CF)C2)=O)CC1 4502,CCCC(CCCNC(=O)C1CC1)NC(c1ncccc1CC)=O 4503,C1(C2CCN(C(c3ccnc(F)c3)=O)CC2)(NC(C(C(CC)C)O)=O)CC1 4504,C1(C(N2CCC(C(F)F)(CNC(C3CN(C(C)C)C3)=O)C2)=O)CC2C(C1)C2(F)F 4505,C1(N=[N+]=[N-])(C(N(C(C#C)(C)C)C2CC2)=O)CCN(C(=O)CN2CCSCC2)C1 4506,c12cc(ccc1Cl)C(=O)N2.C(=O)(C(O)Cc1ccccn1)N1CCCC1 4507,c1(-n2ncc(CNC(=O)Nc3ncc(C(F)(F)F)s3)c2)ccccc1O 4508,C(=O)(CCCC(C)NC(=O)CN1CCCCC1)NCC(C)C#N 4509,N1(C(C(C)(C)CCC#N)=O)CCN(C(=O)CCC2CCC(=O)N2)CC(C)(F)C1 4510,Cc1cc(CC(=O)NCc2nc(C(=O)N(CC(C)O)C)co2)no1 4511,C(=O)(C1=CCCC1)NCC(CCOC)NC(c1cn(CCCC)nn1)=O 4512,C1(NC(C(c2ccccc2Cl)OCC)=O)CCCN(C(=O)CCF)CC1 4513,CC(N=c1[nH]ccc(C#N)c1[N+](=O)[O-])C1CN(C(=O)CN2CC3CC3C2)C1 4514,CC(C)C(C(=O)NCCc1ccncc1)C(C)NC(C1CC(=O)C1)=O 4515,C(=O)(CCN(CC(=O)OC)N1CCC(=O)N(C)CC1)OC 4516,N1(C(CC#N)=O)CCC2(NC(c3ccc(-c4ccon4)cc3)=O)CCCC12 4517,CC1(C)OC(=O)CC1C(N1CCN(C(=O)Cc2ccc(Cl)s2)C(CF)C1)=O 4518,Cc1ccsc1CC(=O)NCc1cc[nH]c1C(=O)NCC12CC(F)(C1)C2 4519,c1(-c2c(C)ccnc2F)ccc2ccnc(NC(=O)C3=CCCCO3)c2c1 4520,c1(C(=O)NC(C2CCOC2)CNC(c2c(C#N)nc[nH]2)=O)cc2ccccc2o1 4521,n1(CC(=O)N(CC(C)NC(C2C3COCC23)=O)C)nc2n(c(=O)c1=O)CCC2 4522,C(=O)(CCCCCNC(c1cn(C2CC2)nn1)=O)NCC(CCCC)O 4523,C1(NC(C(c2cncn2C)C)=O)C2CC1CN(C(c1ccc([N+](=O)[O-])[nH]1)=O)C2 4524,N1(C(CC(C)C)=O)CCC(CNC(=O)C(O)Cc2cnc[nH]2)C1(C)C 4525,c1(OCC)nc(C(=O)NC2CCCCC2c2cccc(C)c2)ncc1F 4526,c1(C(=O)NCCC2CCC(NC(COC(C)C)=O)C2)cc2c(s1)CCC2=O 4527,C=CCC(C)C(=O)NCC1(C)CC(NC(C2CCCC(CC(F)(F)F)C2)=O)C1 4528,C(N=C(NCC1(C)CCCS1)NC1CCCC1)C1CCN(C(C(C)(C)C)=O)C1 4529,c1(Cn2cc(CC3CCCN(C(CC4(C=C)CC4)=O)C3)nn2)cc(Cl)ncc1F 4530,C1(C)(NC(C(C)CNC(=O)CN2CSCC2=O)=O)CCCCC1(C)C 4531,CCC(O)CC(=O)NC(c1cccc(Cl)c1)CNC(c1cnn(CC)c1)=O 4532,C(CC(C)(C)CC(=O)NCCCN(C(=O)CCCCSC)CC1CCCC1)OC 4533,N1(C(c2cnn(C(C)C)c2Br)=O)CCOCC(CNC(=O)C(O)C(C)(C)C)C1 4534,N1(C(=O)NC(CNC(c2c(C)c[nH]n2)=O)C(C)C)CCN(C(=O)C(C)(C)C)CC1.CC 4535,C12(C(=O)NCCOC3CN(C(C(=O)N(C)C)=O)C3)CCCC1C2(F)F 4536,C1(C(N2CCCC(c3cn(CCCCO)nn3)C2)=O)CC12CCCC2 4537,N1(C(C=Cc2cnc(C)s2)=O)CC2CC(NC(c3cc(C#N)c[nH]3)=O)C1C2 4538,Cn1ncc2cccc(C(=O)NC3CCN(C(c4ccccn4)=O)C34CCC4)c12 4539,c1(C(NNC(NC(c2ccccc2)C)=S)=O)cc(F)cc(I)c1 4540,n1(C(C)C)nncc1C(=O)NCC(C)NC(=O)C(C)(C)c1ccsc1 4541,C1(NC(=O)CCc2ncc(F)cn2)CCCC12CCN(C(c1ccc(Cl)cc1)=O)C2 4542,C(=O)(C1=C(C)OCCS1)N1CCCC(CCC(=O)NC(CC=C)CC(F)F)C1 4543,N1(C(C(C)(C)CS(C)(=O)=O)=O)CCC2(C1)CN(C(=O)CC1COC(=O)C1)CCO2 4544,N1(C(C(CC)F)=O)CCN(C(=O)CCSc2ccc(F)cc2F)C(CC)C1 4545,N1(C(c2cn(C)nc2C(C)(C)C)=O)CCCC(NC(C2(O)CCSCC2)=O)CC1 4546,c1(OC)ccc(O)c(C(=O)NC(CC2(C)CN(C(=O)CC3CCC3)C2)=O)c1 4547,Cc1sc(Cl)c(C(=O)NC(C2(CNC(=O)CCCC#N)CC2)C)c1C 4548,N1(C(CC(C)SC)=O)CC2CCCC(NC(c3ocnc3C(F)F)=O)C2C1 4549,Cc1ccc(C2(C(=O)NCC(C)(CO)NC(c3cc(Br)n[nH]3)=O)CC2)cc1 4550,C(=O)(C1=NOC2(CCC2)C1)NC1C(N2CCN(C(C(COC)C)=O)CC2)CCC1 4551,C1(NC(c2nocc2Cl)=O)CCCC1CNC(C1(C(F)F)CCC1)=O 4552,C(=O)(C(C)(C)C1=CCN(C(=O)C(C2CCCCC2)F)C1)C(CCC=C)=O 4553,C(=O)(C1=NN(C)C(=O)CC1)N1CC(CC=C)(NC(C2(COC)CCCC2)=O)C1 4554,c1(C2(C)C(C(=O)NCC3(C)CCCS3)C2)cccc(Br)c1 4555,C1(C(=O)NCC(=C)CC)C=CCN1C(=O)C(c1cccnc1)C 4556,C1(C(=O)NC(C2CCCCC2)C#C)CCC(NC(c2cscc2C(N)=O)=O)CC1 4557,C(C)(C)(CCCNC(C1CC1F)=O)NC(C(C)CSC(F)(F)F)=O 4558,c1(C(=O)NCCC(CNC(C(C(CC)O)C)=O)OC)cc2cnccc2[nH]1 4559,N1(C(C2(CC)CCNC2=O)=O)CCN(C(C2CCCC(C(N)=O)C2)=O)CC1C 4560,c1(NC(C2(C)CCCN2C(=O)Cn2cccc2)=O)cncc(F)c1I 4561,C1(NCc2ccccc2)CN(C(N2CC(C)(C#N)C2)=O)CCC1F 4562,c1(OC)ccc(Cl)c(C)c1C(=O)NC1CCCCN(C(c2ccc(F)o2)=O)C1 4563,c1(OC)cc(C(=O)NCC2CC(C)N(C(=O)CCC(C)SC)C2)cc(F)c1F 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4689,N1(C(CN(CC#C)C(c2csc(Cl)c2)=O)=O)CCCC(O)C1C 4690,C1(CNC(c2ccc(-c3nc(C)sc3)cc2)=O)CCN(C(=O)C(C)O)C12CC2 4691,C1(NC(CSC(C)C)=O)CS(=O)(=O)C2CN(C(C3C(C)OC(C)C3C)=O)CC12 4692,C1(CC)C(NC(=O)Cc2ncc(C)s2)CCN1C(C1CC1(C)C(F)F)=O 4693,CC1CCN(C(=O)C(F)=CC2CC2)CC1CC(=O)NC(C)(C)CCCO 4694,C(N=c1[nH]c2c(c(=NCc3cocn3)[nH]1)CC(C)CC2)c1c(OC)ccc(F)c1 4695,c1(CC)cc(C(N2CC(O)(C(N3CC(SC(F)F)C3)=O)C2)=O)no1 4696,C1(NC(c2c(C)ccc(N)c2)=O)CC2CCC(C1)C2NC(=O)C1=CCCOCC1 4697,N1(C(c2cnc(C)c(N)c2)=O)CCCC2CN(C(=O)C3=CCN(C)C3)CC12 4698,C(=O)(CC(C)(C)C(=O)OCC)N1CCCC(N(C(C2CCN(CC)C2)=O)C)CC1 4699,C(=O)(C(C)(C)C(C)C)N1CCC(N(C(=O)CN2C(C)CCC2C)CCC)C1 4700,N1(C(C2C(Cl)(C(=O)OC)C2)=O)CCC2C(NC(c3cnn(C)c3F)=O)C12 4701,c1(C(=O)NC(C2(O)CCN(c3nccc(C)n3)C2)C)cnn2cc[nH]c(=O)c12 4702,C(=O)(C(CC)C(C)(C)CC)NC1CCN(C(c2cc(CC)cc(C)c2)=O)C1 4703,N1(C(C2OCCN(CC)C2)=O)CCCC2(C1)C(NC(=O)CCC1CC1)CCN2C 4704,c1(C(N2CCCC(C(C)NC(=O)CC(C)CN(C)C)C2)=O)cc(N)nc(Cl)c1 4705,N1(C(c2ccc(S)cc2)=O)CC2OCCN(S(=O)(=O)c3cccnc3Cl)C2C1 4706,c1(CN2CCC(N3C(=O)CCC3=O)CC2)nc2cc(Br)ccc2o1 4707,c1(CCC(=O)NC(C2CCCC2)CNC(C2CC(N(C)C)C2)=O)cc(F)cc(F)c1 4708,c1(OCC)nccc(C(=O)NCCC(C)CCNC(c2cnncc2O)=O)c1F 4709,CC(C)CC(CNC(C1(NC(=O)COC2CCCOC2)CC1(C)C)=O)CO 4710,N1(C(CNC(=O)OCC)=O)CC(NC(c2nc(C)ccc2O)=O)CC(O)C1 4711,C1(C(N2CCC(CN(C(=O)Cc3ccc(Cl)nc3)C)C2)=O)CCC2CC1C2(C)C 4712,C(C)(C(C(=O)NCC1CCN(CC)C1)C(C)C)NC(c1cn(CCC)nc1)=O 4713,CC1CCN(C(=O)Cc2cc[nH]c2)CC1NC(=O)C=CSc1nc[nH]n1 4714,C12(CCNC(=O)CC3(N4CCCCC4)CC3)CCCC1N(c1ncccn1)CC2 4715,N1(C(C(CCOC(C)(C)C)OC2CCOC2)=O)CC2(CCC2)CC1C(=O)O 4716,Cc1ccnc2sc(C(N3C4CCC3C(F)C(NC(C3CCCO3)=O)C4)=O)c(C)c12 4717,O=C(CN=c1nc(N2CCC(CO)C(F)(F)C2)c2c([nH]1)COC2)NC1CCOC1 4718,C1(NC(C2(S(C)(=O)=O)CCC2)=O)COC2CN(C(c3cnc(C4CC4)[nH]3)=O)CC12 4719,c1(NCC=C(C)C)nc(C)cc(=NCc2cccc(O)n2)[nH]1 4720,c1(CNC(C2N(C(c3cncc(COC)c3)=O)CCC2C)=O)cccc(C)c1O 4721,Cc1cc(C)nc(N(C2(C#N)CCNC2)C(C2CCC(=O)NC2)=O)n1 4722,N(C(=NCCNC1CCC1)NC(c1nccs1)C)CCc1cccc(CC)c1 4723,c1(C(N(C2CCCCN(C(C(C)S(N)(=O)=O)=O)C2)C)=O)csc(=NC2CC2)[nH]1 4724,N1(C(CNC(=O)NC)=O)CCCC2(CNC(=O)C(C)OC(C)C)CCCCC12 4725,C1(NC(c2c(C)n[nH]c2C)=O)CC2CC(NC(=O)C(c3cccc(Cl)c3)O)CC12 4726,S(=O)(=O)(c1cccc(Cl)n1)NCC1CN(C(c2ccccc2)=O)C1 4727,C1(C(=O)NC(C)CO)CC2(CC(NC(=O)C(CO)NC(N)=O)C2)C1 4728,n1(CC)ncc(C(=O)NC2(CNC(=O)C(C)C#N)CCOC2)c1C 4729,CC(C(C)(C)NC(=O)COCC1CCC1)NC(=O)CCC1CCC(=O)N1 4730,Cc1cc(C(N2CCOC(C(N(CCCc3ccccc3)C)=O)C2)=O)nn1C 4731,C(=O)(C1=CSCCO1)NCCN(C(c1c(C)nns1)=O)C 4732,C1(C)(CC)CC(NC(=O)Cc2cc(C)[nH]n2)CN1C(C1(NC(N)=O)CC1)=O 4733,n1(CCCOC)c(N(CCC(=O)OC)C)nnc1C1=C(C)OCCO1 4734,CC1CC(C(=O)N2CC(O)(C(C)(C)CNC(C3CCCC34CC4)=O)C2)=NO1 4735,C1(NC(c2c(CC)ncs2)=O)C2CC1N(C(=O)CCSc1cccc(Cl)c1)C2C 4736,C(CN=c1cc(F)nc[nH]1)(C1CC1)NC(CC(C(C)C)c1ccccc1)=O 4737,N1(C(c2ccccc2Br)C(=O)Nc2ccc(Cl)cn2)CCC2(C1)OCCO2 4738,C1(SC)CN(C(=O)C(=O)N(C)CC2CC(SC)C2)C1 4739,c1(NC(C2N(S(C(CC)Cc3ccccc3)(=O)=O)CCC2)=O)onc2ccccc12 4740,C12(C(=O)Nc3ccccc3-n3cc(C4CC=CCC4)nn3)CCC(F)(CC1)C2 4741,C1(C(=O)NCC2C(CNC(C(CC)OC3CCCCC3)=O)C2)CCC(N(C)C)CC1 4742,c1(OCC(=O)N(N2CCCCC2)CC)ccc(OC)cc1.N1(CC)CCC(CSC)CC1 4743,C(=O)(C1CCc2cc(F)ccc21)N1CCC(F)(CNC(C2CCC(F)C2)=O)CC1 4744,C1(NC(CN(c2ccncc2)C)=O)CC2CCC1CN2C(=O)CCN(S(C)(=O)=O)C 4745,c1(C(N2C(CN(C(=O)C(C)(C)CF)C)CC(F)C2)=O)ccc2c(c1O)CCCC2 4746,C1(C(=O)NC(C#C)C(C)C)N(C(=O)CC2CCC(C)CO2)CCC1(C)C 4747,N1(C(CC(=O)NCC(F)(F)F)=O)CC(O)CC1CNC(C1CC2(CSC2)C1)=O 4748,CC(C)(C)S(=O)(=O)CC(=O)NCC1(O)CN(C(=O)CN2C(=O)CNC2=O)C1 4749,C1(CNC(C2CC23CCOC3)=O)CC2(CC2)CN1C(=O)CN1CCC1 4750,CC1(C(=O)NCC(F)CNC(=O)CCSc2ccccn2)CCCC1 4751,N1(C(c2n[nH]c(C)c2C)=O)CC(NC(=O)C(CC2CC2)CC2CC2)CCC1C 4752,Cc1cc(C(=O)NC2CCC2COC(C2(C)CCC(=O)NC2)=O)ccc1F.C=O 4753,N1(C(CC(C)(C)OC)=O)CCCCC(CNC(=O)Cc2ccc(F)c(F)c2)C1 4754,c1(OC)cc(C(=O)N(C)CCNC(c2c(SC)cnn2C)=O)cc2cn(C)nc12 4755,C(CCCCC(=O)NCC1(CC(=O)O)CCCC1)c1cn(CC(C)OC)nn1 4756,N1(C(c2c(OC)c(F)ncc2)=O)CCC2(CC1)CN(C(=O)CCCC1(C)N=N1)C2 4757,C1(NCC(C2CCCN2C(=O)OC(C)(C)C)C)CCCN(c2ccccn2)C1 4758,c1(N(C(C)C)C(CCCC(N)C2CCCCC2)=O)ccc(C(F)(F)F)cc1C#N 4759,C=C(C)C1OCCC1C(=O)NC1CCN(C2CCN(CCOC)C2)CC1 4760,C1(C(=O)NCC(=O)N(C(C)CO)CC2CCC2)C2CN(C)CC12 4761,c1(OC)cccc2[nH]cc(CC(=O)N(C)CC3(O)CCC(F)(F)CC3)c12 4762,C(=O)(C(F)(F)C(F)(F)F)N1CCC(N(C)C(c2cc(C(F)(F)F)ccc2Cl)=O)C1 4763,C=CCC(C)(C)CNC(C1CCN(C(=O)CP(C)(C)=O)C1)=O 4764,CC1C(NC(=O)Cc2cnsc2)CC2CCC1N2C(=O)C(F)(F)c1cnccn1 4765,N1(C(c2c(C)n[nH]c2)=O)CCN(C(=O)CC=CCO)CC1c1ccnn1C(C)C 4766,N1(C(C)C)CC2CCCCC2(CN=c2[nH]c(N(C)CC3CC3)nc3c2COCC3)C1 4767,c1(C(N2CCOCC2C2CCC2)C(=O)NCC)cc(OC)cc(C2CC2)c1.C(=O)OC 4768,c1(OC)c[nH]ccc1=NC(=O)C(C)C1NC(C)(C)OC1C 4769,C(c1cc(Cl)cc(Cl)c1)=CC(N1CCN(C(C(C)(C)OC)=O)CC1)=O 4770,C1(C(=O)NC2(C)CN(C(c3c(C)ncs3)=O)C2)CCC2(CC1)CC2(F)F 4771,c1(C(N2CCN(C(C(C)SCCCC)=O)CC(O)C2)=O)ccc2ncn(C)c2n1 4772,c1(N2C3(CNC(COC4CCN(C)CC4)=O)CC(C2)C3)snc(Cl)c1C#N 4773,C(CN=c1cc(NCc2ccc(C(N)=O)o2)nc[nH]1)(C1CC1)OC 4774,CCC(C)CC(=O)C(=O)NC(C1CC1C(=O)NCc1ccc(C2CC2)o1)C 4775,C1(CNC(C(C(C)(C)C)SC)=O)CC12CCN(C(c1csc(CO)n1)=O)CC2 4776,c1(N(C(C)=O)C)ccccc1C(=O)NCC(CNC(C1CC(N=[N+]=[N-])C1)=O)CO 4777,CCCCC(C)CCC(=O)NC1COCC1NC(c1cc(Br)cs1)=O 4778,CC1CN(C(=O)CC2CCC(=O)C2C)CCC1C(=O)NCc1cnn(C)c1 4779,C(c1ccc(Cl)c([N+](=O)[O-])c1)=CC(=O)NC1CC2CC1CN2 4780,C(CCCCCNC(=O)COc1ccsc1)NC(c1c(C)snn1)=O 4781,c1(C(=O)NCC2CCCN(C(C(CC3CC3)OC)=O)C2)cc(C#N)n(C)n1 4782,C(c1cncn1C)=CC(=O)N(CCC(=O)N(CC(O)C1CCC1)C)CC 4783,N1(C(CNC(C)=O)=O)CCC2CC1CN2C(c1cccc(C)n1)=O.C1C(=O)N1 4784,c1(SC)ccc(C=CC(=O)NC2CCC(NC(c3ccn(C4CC4)n3)=O)C2)s1 4785,C1(NC(c2c(CC(C)C)cccc2)=O)CCC2(CCN(C(c3ccoc3)=O)C2)C1 4786,CC(C)C(CC(=O)NCC(F)CNC(c1cocn1)=O)c1ccccc1 4787,CCC(CC)CC(F)C(=O)NC1CC2CC1N(C(c1cscc1C(F)F)=O)C2 4788,Cc1cccc(NC(=O)NCC(c2ccc(C3CC3)cc2)(C)C)c1F 4789,C1(C(N2C(N(C(C)C)C)C(C)(C)CC2)=O)CN(C(=O)OC(C)(C)C)C(C)(C)C1 4790,C1(CC(=O)NCC(C)(C)OC)CN(C(C2CC(C)=NO2)=O)CC12CC2 4791,c12cc(c(O)c(C)c1)NC(=O)C(=O)NCC1N(CC=C1)C2=O.C(C)(=O)OC 4792,CCCCC(C(=O)NCc1ocnc1CC)NC(c1cc(C)c(C)[nH]1)=O 4793,c1(CCNC(C=CC(C)(C)NC(c2cc(O)cs2)=O)=O)ccncc1F 4794,C1(CNC(C(C#C)(C)C)=O)CCC(C)N(c2nccc(C)c2C(=O)OC)C1 4795,CCC(C)CC(CO)NC(=O)CC(CC)N(C(=O)CC1CC(=O)NC1=O)C 4796,Cc1nc2ccc(CNC(c3cc(C)c(=O)n(C)c3)=O)cc2o1 4797,C(=O)(C(F)CCC(C)C)NCC1N(C(CC2CCC(OC)CC2)=O)CC1 4798,Cc1n[nH]c(=NC2CCCC(NC(c3cnn(C4CCCC4)c3C)=O)C2)s1 4799,c1(C(N(CCC2N(C(c3c(CC)c[nH]c3)=O)CCCC2)C)=O)c[nH]cc(C)c1=O 4800,N1(C(C(N2CCC(NC(C(C)(C)C)=O)C2)=O)=O)CCCCC1c1cn[nH]c1 4801,C1(NC(CCCC(C)C)=O)CCN(C(c2cc(N)c(Br)cc2F)=O)C12CCCC2 4802,C1(CNC(C2(CCC)CC2)=O)CC2(CCN(C(C3(C)C=CCC3)=O)CC2)C1 4803,c1(C(N2CC(CC3(C(F)(F)F)N=N3)C(C(F)(F)F)C2)=O)[nH]cc2c1CCCC2 4804,c1(C(=O)NCC2C3CN(C(CCCCCC)=O)CC32)cc2n(n1)C(C)CCC2 4805,c1(OC)c(C(=O)NC(Cc2cn[nH]c2)C(=O)N(C2CCOC2C)C2CC2)cnn1C 4806,c1(N(CC=C)CC)cc(OC)c(OC)cc1CC(=O)NC1CC1.C1CC1 4807,N1(C(C(C)OCC=C)=O)CCC(F)(F)C(C(=O)NC2(C)CC(C)(C)C2)C1 4808,C1(NC(C2CC3CCC2C3)=O)CC2CCC1N(CCN1CCCS1(=O)=O)C2 4809,C1(CNC(c2c(C)ocn2)=O)CC2COCC2N1C(c1cc2cccnn2n1)=O 4810,C12(C(=O)NCC3(C(=O)OCC)CCCO3)CC1CN(C(c1cccc[n+]1[O-])=O)C2 4811,N1(C(C(CCCC)O)=O)CC(NC(c2ccncc2)=O)C2CCCC12 4812,c1(C(N2C3CN(C(c4c(CC)scc4)=O)C(CC3)C2)=O)ccnc2c1CC(=O)N2 4813,c1(C(=O)NC(CCCCNC(C(C)SCC)=O)C)cc(O)cc(C#N)c1 4814,C=CCC(C)(C(=O)N1CCC(O)(CCNC(=O)COCC(C)C)CC1)NC(C)=O 4815,C(CC(C)C(=O)NCC1CCN1C(=O)CN1CCCCC1)OC 4816,C1(CCNC(C2CC(Cc3cn(CC4CCOC4)nn3)C2)=O)OCCCO1 4817,CC1CN(C(c2c(F)cccc2Cl)=O)CCN1C(c1ccc(C2CC2)cc1)=O 4818,N1(C(C(C)NC=O)=O)CCOCC12COCCN(C(C1C3C4CCC(C4)C13)=O)C2 4819,N1(C(C=Cc2ccc(C)nc2)=O)CC2(CCN(C(=O)CC3OC(C)(C)OC3=O)C2)C1 4820,C(CCCCC(=O)NC1CCC(C(=O)NCC(C)(C)C2CCC2)C1)SC 4821,c1(C(=O)NCC(C)=CC(=O)NCCN(CC(C)(C)C)C)cnc(C)c(C)c1 4822,CC(C(F)(F)C(F)(F)F)NC(=O)Nc1ccc(Br)c(Cl)n1 4823,S(=O)(=O)(c1ccc(CCC(=O)O)cc1)N(Cc1ccc(C(=O)NC(C)C)cc1)CC 4824,c1(OC(C)C)ncc(C(=O)N(C2CCCCC2)CCC2(CC#N)CCC2)cc1Cl 4825,CC(C)CCCCCC(=O)N(C)CC1(O)CCN(C(C2CNC(=O)C2)=O)C1 4826,n1(C(CC)C)[nH]c(=NC(=O)C(=O)N(C(C)C)Cc2cc(F)c(Cl)cc2F)cc1C 4827,C(=O)(CCCC(N)=O)N(C(C)CCNC(=O)CC1CN(C)C1)C 4828,CCCCCC(O)C(=O)N(CC(N1CC(c2cc[nH]n2)C1)=O)CC1CC1 4829,c1(OC)cc(N2CCC(c3ccc(C)nc3)C2)ncn1.C1(=O)N(C2CC2)CCN1 4830,c1(NCc2nc(C)[nH]n2)nc(N(C)CCN2CCOC2=O)c2ncn(C(C)C)c2n1 4831,C(=O)(C(O)C(F)(F)F)NCC(C)(C)NC(c1cn(C)c(O)n1)=O 4832,c1(N2CCCC(C=C)C2)nc2c(c(=NCC3CCC=CCCC3)[nH]1)CCC2 4833,c1(N2CC(C(C)NC(C3CC3N(C)C)=O)C2)c(C#N)cnc2ccccc12 4834,C1(n2c(C(CCC=C)NCCc3ncco3)nnn2)CCC(F)(F)CC1 4835,c1(C(C)C(=O)NCC2(F)CCN(C(=O)C(C)(C)C)C2)cccc2ccccc12 4836,C(=O)(CC1OCc2ccccc21)NC(C(C)NC(c1n(CC)nnc1)=O)C 4837,C1(C(N)=O)CC2CC(NC(c3cn(C4CCS(=O)(=O)C4)nc3C(F)(F)F)=O)C2C1 4838,C(CC#CCO)(c1cccnc1)NC(=O)NCCC(=O)NC(C)C 4839,N1(C(C2C(C)(C)CO2)=O)CC2CC(NC(=O)CCCc3ccccn3)CC2C1 4840,c1(C(=O)NCCN(C(c2[nH]nnc2C(F)F)=O)CC)cnc(O)n1CC 4841,N1(C(c2c(COC)scc2)=O)CCC(C(F)F)(CNC(C2COCCO2)=O)C1 4842,Cc1noc(N)c1C(N1CCC(NC(c2csc(C(F)(F)F)c2)=O)C1)=O 4843,c1(C(=O)NCCN(C(c2ccc(OC(C)C)cn2)=O)CC)nnc(S)n1C 4844,N1(C(CC(CC)C2CC2)=O)CC(NC(C2CCN(OC)CC2)=O)C2(CC2)C1 4845,CC1CC(C(N2CC(N(C)C)C2)=O)CCN1CC(N1CCC(O)CC1)=O 4846,C1(C(=O)NC2CN(C(c3cccc(C#N)c3)=O)CC(F)C2)CCc2ncnn2C1 4847,S(=O)(=O)(c1ccccc1C)NCCCC(=O)NC1CCC(CNC(C=CC)=O)C1 4848,C12(OC)CN(C(=O)Cc3ccnc(NC(=O)OC(C)(C)C)c3)CC(CO)(C1)C2 4849,N1(C(C(CC)(C)OC)=O)CCCC(CC)(NC(=O)CCc2ccccc2F)C1 4850,CC(C)S(=O)c1ccc(C(=O)NC2CN(C(c3c[nH]c(=N)o3)=O)CC2F)cc1 4851,C1(C(=O)NCC2CCN(C(CC3C(C)(C)C3)=O)C2)CCC(=O)NC1 4852,n1(C(CC#C)CC)c(CSCCOC(C)(C)C)nnc1N=c1ccn(C)[nH]1 4853,c12ccc(cc1)S(=O)(=O)N2.C1(N(C(COC)=O)C)CCCN1.C(CCS)NC(C)(C)C 4854,C1(CC=C)(NC(=O)CC(O)CCSC)CCCN(C(=O)CSCCN(C)C)C1 4855,N1(C(CC(C=C)CC)=O)CC2OCC(NC(=O)CCCCCCC)C2C1 4856,c1(C(N(CCN(C(=O)CSC(C)(C)C)C(C)C)C)=O)nccc2ccn(C)c12 4857,N1(C(C(C)=C2CC2)=O)CC2CC(CNC(=O)COc3ccc(Cl)c(F)c3)C2C1 4858,c1(CC(=O)OCC(c2ccc(Br)cc2)(F)F)cccc2cccnc12 4859,c1(C(N2CC(C(C)NC(c3cnn(C)c3N)=O)OCC2)=O)cc2cscc2s1 4860,c1(C(N2CCCCC(NC(C(CC)(F)F)=O)CC2)=O)cc2c(cn1)NC(=O)CO2 4861,C(CC)(CCCC(=O)NCC(C)(C)CCOC)NC(C1(CCC=C)CC1)=O 4862,c1(C(N2CCCN(S(=O)(=O)CCc3ccccc3)CC2)=O)noc2c1CCCC2 4863,Cn1c(C(N2CC(CO)(NC(=O)C(C#N)=CC3CC3)C2)=O)cc2ccccc12 4864,Cn1cc(C(=O)NC2CCCN(CCCC3CCCCC3)C2)c(O)nc1=O 4865,c1(C(N2CCSCC2C)C(=O)NCCC)cc(C)c(Br)c(Cl)n1 4866,CC1CCC(C)(C(N2CCCCC2CCNC(=O)Cc2cccnc2F)=O)CC1 4867,c1(CCCC)ccc(C(C(=O)NC2CCN(CC(F)F)C2)N(C)CC)cc1 4868,c1(C(N2CC(OC)C(NC(=O)C=CS(C)=O)C2)=O)ccc(C)c(C(F)(F)F)c1 4869,C1(CNC(C(CC)(C)O)=O)CC(C(=O)N2CC(F)(CF)C2)=NO1 4870,c1(-c2n(C(C=C)C)nc(C(C)CC)n2)ccc(C)c(Br)c1 4871,Cc1c(Cl)cc(CN2CC(CC(=O)NCc3c(Br)ccnc3Br)C2)cc1Cl 4872,CCS(=O)(=O)c1ccc(C#N)c(C(=O)Nc2ccnn2Cc2ccccc2Cl)c1 4873,C12(C(=O)NC(c3ccn(C)n3)CC)CC1CCN2C(=O)CC1CC(C)=NO1 4874,N1(C(c2ccc(C(C)(C)C)[nH]2)=O)CCC12CN(C(C1SCCCS1)=O)C2 4875,c1(NC(=O)Nc2c(C)c(N3CCCC3)ccc2)ncc2scc(Br)c2n1 4876,c1(N(CC)CC)ccc(C(CCC)(C)NC2CC3CC23)cc1 4877,CCCCC(CC(=O)N(C(C)CC(C)CC)C)NC(=O)C(F)=CC1CC1 4878,N1(C(CCSCCCC)=O)CC2(CCC(C(=O)NCC3(OC)CCOCC3)O2)C1 4879,c1(NC(c2ccc(-c3cccc(Br)c3)cc2)=O)cc(-c2cccnc2)cnn1 4880,C1(NC(c2c(C(C)=O)ccs2)=O)CCCCN(C(C2CCCC(C)CC2)=O)C1 4881,c1(OCC)ccc(C)nc1C(=O)NCC(F)CNC(C1CC1C(F)(F)F)=O 4882,c1(CC(N2CCCC(NC(CCCNC(N)=O)=O)C2)=O)cc(Br)ccc1F 4883,c1(-n2cc(C3CCN(C(C(c4occ(C)c4)(F)F)=O)C3)nn2)c(C)cccc1Cl 4884,C(CCCC(CO)NC(C1CC2C=CC1C2)=O)NC(c1cc(C)ns1)=O 4885,C1(F)(C(=O)NCC2C(OCC)CC2)CCCN(C(=O)C(C)CC2CCCC2)C1 4886,N1(C(C(C)(C)C)=O)CCC(C(=O)NCCNC(C23CCC2C3)=O)CC1 4887,CN1CCN(C)C(C)C1.C1(NC(=O)CC)CCC1C(F)(F)F 4888,c1(C(N2CCC(O)(C(C)CNC(C3(C(F)F)CCC3)=O)C2)=O)ccnn(C)c1=O 4889,CC1(C(N2CCCC(NC(c3coc(CC4CC4)n3)=O)C2)=O)CC2(CCC2)C1 4890,N1(C(C2CC=C(C)CC2)=O)CCN(C(c2cc(Br)c[nH]2)=O)C(C#N)C1 4891,N1(C(C(C=C=C)C)=O)CC2CCN(C(c3cc(CCN(C)C)on3)=O)CC2C1 4892,c1(C(=O)NC2C3CN(C(C4(n5cncn5)CC4)=O)CC23)c[nH]c2cccnc12 4893,N1(C(c2cnc(C)o2)=O)CC2CCC(NC(c3cccc(F)c3Cl)=O)CC2C1 4894,Cn1c(C(N2CC(F)(F)CC2CCNC(C2CC3(CC3)C2)=O)=O)cccc1=O 4895,c1(NC(C2CC(F)CCN2C(C2C3CCC(C3)C2C)=O)=O)ccc(CO)cc1O 4896,C(=O)(C(O)CC[S+](C)C)N1CCC(NC(c2c(C)oc(CO)c2)=O)C(O)C1 4897,C#CCC(C(=O)N1CCC(CN(C(=O)CN2CCCS2(=O)=O)C)CC1)C1CC1 4898,C1(CNC(C(C2(O)CN(C(C3CCCC(=O)N3)=O)C2)F)=O)CC(O)C12CCC2 4899,C1(C(=O)NCC=CCNC(C(N2CCC(O)CC2)C)=O)CCCC(CF)C1 4900,Cc1cc(C(=O)NC2(c3ccccc3)CN(C(=O)C=C3CCOCC3)C2)n[nH]1 4901,C1(C(=O)NC(C2(C(N3CCOC4CC34)=O)CC(C)(C)C2)C)CCC(C#N)CC1 4902,C1(C(N2C(C(C)NC(=O)CC3CCC34CCC4)CCC2)=O)CCC2(CC1)CC2 4903,N1(C(CS(=O)(=O)NCC)=O)CCCC(NC(c2cnc(C)s2)=O)CC1 4904,C(=O)(CCCCCN=[N+]=[N-])NCCC1(OC)CN(C(C2CCN(C(C)C)C2)=O)C1 4905,Cc1nn(C)c(C)c1CC(C)C(=O)NC(C)CN(C(=O)CN1CCCCCC1)C 4906,c1(C(C)C)conc1C(=O)NC1(CCNC(=O)CC2(C#N)CC2)CC1 4907,n1(CC)cc(C(=O)NC(C)C(C)NC(c2cc(C(F)(F)F)ns2)=O)nn1 4908,c1(C(=O)NC2(C)CC(NC(c3noc(CC)c3C)=O)C2)cc2n(c1)CCC2 4909,c1(C(N(CCN(C(C2CC(C(C)C)C2)=O)CC)CC)=O)ccc2nc[nH]c2n1 4910,N1(C(c2cc(CCNC(c3ccn(CC)n3)=O)on2)=O)CCCC(N=[N+]=[N-])C1 4911,CCCCC(O)C(=O)N(CC(O)CNC(c1ccc(NC(C)=O)cc1F)=O)C 4912,N1(C(CCC)=O)CCOC(CNC(C2CC(C(F)F)C2)=O)C1 4913,c1(CN2CCCC(CN=c3cc(C4CC4)nc[nH]3)(C)C2)cccnc1S(N)(=O)=O 4914,Cc1cc(C)c(C(=O)NC(C)C(C)NC(c2coc(N(C)C)n2)=O)cc1N 4915,CC(CNC(C1CN(CCF)C1)=O)(CO)NC(=O)C(C1CCCCC1)=O 4916,C12(NC(CC3(C)CC3)=O)CC3CC(C1)CC(NC(C1CCCC(O)C1)=O)(C3)C2 4917,Cc1cc(C#N)cc(C(=O)NC2CCCC2CNC(=O)C(C)n2cncn2)n1 4918,c1(C(=O)NCC(C)OCC=C)cccc(S(=O)(=O)Nc2cccnc2)c1 4919,CC1CCCCC1(CNC(=O)CCn1ncn(C)c1=O)NC(C1CC(=O)N1)=O 4920,c1(C(=O)NCCN(CCNC(C2CCCSC2)=O)CC)cccnc1 4921,N1(CC(=O)N(CCCN=[N+]=[N-])CC(C)SC)CC(=O)NCC1C(C)C 4922,N1(C(c2cc(CC)oc2C)=O)CCCCC(CNC(=O)CCc2nncs2)C1 4923,C1(NC(CCC2N(C)CCC2)=O)CN(C(=O)Cc2ccc(=N)[nH]c2)CC12CCC2 4924,N1(C(c2ccc(C#C)c(C)c2)=O)CCC2CCN(C(=O)C3=NOC(C)(C)C3)C2C1 4925,c1(C(=O)NCC(N2CCCC(OC3(C)CCC3)C(F)C2)=O)cc2cncn2c(O)n1 4926,CCCCS(=O)(=O)C(N1CC(CNC(c2[nH]ccc2C)=O)C(O)C1)=O 4927,N1(C(CNC(CCCCC)=O)=O)CCN(C(=O)C(C)CO)CC1C(F)F 4928,C(=O)(CC(C)(C)C)NCCCNCC(=O)NC1C(NC(C(=O)N(C)C)=O)COC1 4929,c1(C(N(C(CNC(C2(Cl)CC2(F)F)=O)C2CC2)C)=O)cnc2c(Cl)cccn12 4930,C1(C(=O)NC(c2nc(C)sc2)C)C=CCN(C(=O)C(F)CC2CCOC2)C1 4931,N1(C2CN(C(COC(C)=O)=O)C2)CC(NC(C2CC2(C)C(F)(F)F)=O)CC1=O 4932,N1(C(CC(C)(C)N(C)C(C2CCC(O)CN2C)=O)=O)CC2CCC1C(O)C2O 4933,c1(C(=O)NC(C2CCOC2)CNC(c2c(C)ccs2)=O)nc2c(s1)COCC2 4934,C(=O)(C1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2)c2ccccc21)OC 4935,Cc1ccc(O)cc1C(N1CC2CC(C1)N2C(c1nc(Cl)ccc1F)=O)=O 4936,N1(C(=O)CC2CC3(CCO2)CC3)CCC2C(C1)CN2C(=O)Cc1cnoc1 4937,N1(C(C2N(C(CC)=O)CSC2)=O)CC(NC(c2ccncc2Br)=O)C(C)C1 4938,CCCCC(C)C(=O)NCC12COC(CNC(=O)CC3COC(C)(C)CO3)(C1)C2 4939,C1(CC)(CNC(=O)C=COCC)CN(C(c2cc(Cn3cc(C)cn3)on2)=O)C1 4940,c1(CN2CC(NC(=O)Cc3cccc(O)c3Br)C2)ccc(Br)c2nsnc12 4941,c1(CC(=O)NCCCCCN(C)C(C23CC2CCC3(F)F)=O)cccc(F)c1F 4942,c1cc(O)ncc1Cl.C1(C(=O)OC)CC(C(=O)NCC2(CNC(=O)C3CC3)CCC2)C1 4943,c1(OC(C)C)ccc(C(=O)NCCCN(C(c2cn(C)nc2Cl)=O)C(C)C)cc1 4944,N1(C(=O)CCOCC(F)F)CCCC(O)(CNC(=O)C(F)(F)C(O)C2CC2)C1 4945,c1(C(=O)NCCSCC)n[nH]c2c1CN(C(c1ncc(C)cc1F)=O)C2 4946,CC1CC2(CCN(C(c3nc(Cl)sc3Cl)=O)CC2)CN1C(=O)C(O)CN(C)C 4947,c1(C(=O)NC2C(NC(c3c(Cl)nc(OC)s3)=O)COC2)ccc(=O)n2c1CCC2 4948,C(=O)(C1=C(C)N(C2CC2)C(=O)NC1C)N1CCCCC(SC)C1 4949,C1(C(=O)NCCC(CCC)C2CC2)CC2(CCC2)CN1C(=O)C1=NOCC1 4950,C(C)(CCN=c1c(Cl)c[nH]cc1[N+](=O)[O-])NC(CCCc1cc(C)no1)=O 4951,c1(NC)ncccc1C(=O)NCC(C)(C1CCC1)NC(c1ncc(OC)cn1)=O 4952,c1(C(=O)NCCC(=C)CNC(=O)C(O)P(C)(C)=O)cc(C)nc2c1cnn2CC 4953,C(=O)(C1CCCn2ccnc21)NC1C(C)C2CCC(C1)N2C(C1CC1F)=O 4954,N1(C(c2nc(C(C)OC)sc2)=O)CCCCCC1CNC(C1CC=CC1)=O 4955,C(C)(CCC(=O)NOCC(=O)NCC1(C(C)C)CC1)OC 4956,N1(C(CC(C)CNC(C2(C)CC(C#N)C2)=O)=O)CC2CN(C)CC2C1 4957,c1(CNC(C2OCCN(C(CCCN(C)C)=O)C2)=O)ccc(F)c(O)c1 4958,c1(NC(C)CCC(F)(F)F)[nH]c(=NC2CSc3ccc(F)cc32)nc2sccc12 4959,CC(CSc1cccc(CNC(=O)C2CC2)c1)CC(=O)N1CCC(C2CCC2)C1 4960,C1(N(C(c2ccn(C(CC)CC)n2)=O)C)CCN(C(=O)COC)CC1C 4961,CC(=O)CCCC(=O)N(C1(CCNC(C2CCC(CS(C)(=O)=O)O2)=O)CC1)C 4962,C1(C(N2CC3C(CNC(COCC(=C)C)=O)(C3)C2)=O)CCC2OCCC2C1 4963,C12(NC(c3ccn(C4CC4)n3)=O)CCCCC1N(C(c1cncc(Cl)n1)=O)CC2 4964,CN1CCOC2CN(CCSCC3CC3OC(=O)NC(C)(C)C)CC12 4965,c1(OC)cccc(C(O)C(=O)NCCCN(C(=O)C(F)C2CC2)CCO)c1 4966,c1(C(=O)NCC2CN(C(CCC(C)C)=O)C2)cn2c(n1)C(C)CCC2 4967,C1(C)(NC(CC2(OC(c3cc(OC)no3)=O)CCC2)=O)CCCC1C 4968,C1(C2CCC2)(NC(C2C=CCCN2C(=O)CCCc2cnn[nH]2)=O)CC1 4969,Cc1cc(C(=O)NC2CCCC2CNC(c2cc(C)n(C)c2C)=O)nnc1C 4970,n1(CC)nc(C)c(NC(C2COCCN2C(c2ncsc2Br)=O)=O)c1C 4971,c1(C(N2C(CCNC(CC(C=C)CC)=O)C(C)CCC2)=O)ccnc2c1CCC2 4972,C1(CC(=O)NC(CC)CO)C=CC(NC(=O)C(CO)N(C)C)C1 4973,C12CN(CCO1)C2=O.C(CCC(=O)N(C)Cc1sncc1Cl)OCCC 4974,C1(O)(C(C)NC(C2(CCCC)CCC2)=O)CCN(C(c2cc(C)no2)=O)C1 4975,C1(CNC(C=CC)=O)CCN(C(c2c(C)noc2-c2ccccc2)=O)C12CCC2 4976,Cc1cnoc1C(=O)NCCn1cc(C(=O)NCC(C2CCCO2)O)cn1 4977,C(=O)(C(C)(C)CC(F)F)NCC1ON=C(C(=O)NC2CN(CC)C(C)C2)C1 4978,C12(C(=O)NCC(COC(C)C)(C)C)COCC1CN(CCCN1CCOC1=O)C2 4979,N(S(=O)(=O)N1CCC(C)CC1)C(c1c(OC)ccc(OC)c1)C 4980,C1(CNC(c2nc(C(C)NC(C3(SC)CC3)=O)oc2)=O)CC(O)C(O)C1 4981,C(=O)(CC(C(F)F)n1ccnc1)NCC1(OCC)CCC1.N12CCCCC1C2=O 4982,c1(-c2cn(CCN(CCN(C(C(C(C)C)OC)=O)C)C)nn2)cccc(F)c1N 4983,C(=O)(CC(O)c1cnc(Cl)s1)NC1CC(CNC(C2C(C=C)C2)=O)C1 4984,C(C(C(=O)NOCC(=O)OC)NC(=O)C(O)CCN(C)C)OCC 4985,CC1(C(=O)NCC(CO)NC(C2CCCCO2)=O)Cc2ccccc2C1 4986,C1(NC(c2cnsc2)=O)CCC2(CCCN(C(C3(F)CCCCC3)=O)C2)C1 4987,C1(NC(c2c(C(C)C)ocn2)=O)CCS(=O)(=O)C12CN(C(=O)C(C)C1CCC1)C2 4988,c1(CN(CCN(C)C)CC2CCS(=O)(=O)C2)cccc(C(C)(C)C)c1 4989,C1(C(=O)Nc2cccc(CC(=O)OCC)c2)CC2(C1)CN(C(=O)C#CC1CCC1)C2 4990,N1(C(c2scc(CC)n2)=O)CCn2c(C3CC3)nnc2C1.c1(CO)ccccc1 4991,C1(NC(CCCc2onc(CC)n2)=O)CCC(C)(CNC(=O)CCC2(C)N=N2)C1 4992,c1(C(=O)NCC2N(C(C3CCC(=O)N3)=O)CC=C2)cc(Cl)cc2cccnc12 4993,N1(C(CCN(C)CC)=O)CCC(NC(=O)CCc2ccon2)C(F)C1 4994,C(=O)(C(C)(C)CO)NCCC1CC(NC(CCCc2cc(C)no2)=O)C1 4995,C(=O)(C(F)C(C)CC(C)(C)C)N(CCC)CCNC(C1CCCN1C(C)=O)=O 4996,c1(NC(CCN(C(C(C)OCC)=O)C2CC2)=O)ccccc1N=[N+]=[N-] 4997,c1(SCC)ccccc1NC(=O)CCN(C)C(C1CCN(C)C1C)=O 4998,c1(C(=O)NC2C(NC(=O)COc3ccsn3)CC2)ncoc1-c1ccon1 4999,c1(C(=O)NC(CC=CC)C(=O)N2CCC(C)(CC)C2)ccc(C)cc1C 5000,C1(COC)(CNC(=O)C(C)(C)N2CCCC2)CN(C(=O)CC2CC(OC)C2)C1 5001,c1(C(C(=O)NC2CCN(C(C(C)N3CCC3)=O)C2)=O)ccc(O)cc1 5002,N1(C(C2(C)CCCOC2)=O)CCC(C2(NC(c3nc4c(s3)CCCC4)=O)CC2)C1 5003,C(=O)(C1CCc2c[nH]nc21)N1C(C(C)NC(c2cccc3nccn23)=O)CCC1 5004,C1(N(C(c2ncsc2Br)C(=O)NCCSC)C)CCCCCC1(C)C 5005,c1(C(N2CC(CC(C)NC(C(CC)C(C)C)=O)C2)=O)cc([N+](=O)[O-])cnc1N 5006,C12(OC)CCC(C(=O)NC3CCC(C)N(C(c4ccon4)=O)C3)(CC1)CC2 5007,C1(NC(C(C)OCCCC)=O)CN(C(=O)C(c2ccccc2)C)CC(C)(C)C1 5008,CC(C)CC(C)(O)CNC(=O)CNC(=O)Cc1ccc(C#N)cc1 5009,N1(c2ncc(C)c(C)n2)CCCC(C)(C)C1CNC(=O)CSc1n[nH]c(O)n1 5010,CCCCCCC(=O)NC1CC2(C1)CN(C(=O)C(C)C(C)c1ccc(F)cc1)C2 5011,C(C)(CNC(C1(C)CCSCC1)=O)(C(C)C)NC(COCc1nnc(C)s1)=O 5012,C(=O)(C1c2ccccc2CN1C(=O)CCCn1ccnc1)N1CC(=O)NCCC1 5013,C1(CNC(c2c(OC)csc2)=O)CCCCN(c2cc(C)nc(CO)n2)C1 5014,c1(C(=O)NC2CC(C)(CC)N(C(=O)C(=O)NC3CC3)C2)cccc(Cl)c1C(F)F 5015,C(N=c1[nH]c(C)cc(=NCC(C)N2CCCCCC2)[nH]1)C1CC(OC)C1 5016,c1(C(N2CCC(N(C(C3CC34CC4)=O)C)CC2)=O)cc(C(=O)OC)cc(Cl)c1O 5017,C(=O)(CC(C)CN(C)C)N1C(CC(=O)NC2(CC)CC2)CCC1 5018,CCC(C(=O)NCCCCN(C(=O)Cn1ccc(Br)n1)C)OC 5019,c1(CNC(C2CC(F)CN(c3ncccn3)C2)=O)cccc(F)c1O 5020,Cc1cc(C#N)nc(NC2CC2CNC(c2cc(-c3cccs3)on2)=O)n1 5021,C1(C(=O)NC2C=CC(CNC(c3ccc(CO)s3)=O)C2)CCC12CCC2 5022,Cc1cc(CN2CCCC(CC3CCNC3)C2)cc(C)c1 5023,C1(N(C(c2nc(CCC)sc2)=O)C)CN(C(C23CCC2C3)=O)CC1(C)C 5024,N1(C(C(CC)C(C)C)=O)CCN(C(C2CC23CC3)=O)C2CNC(=O)CC12 5025,n1(C(C(=O)NCC(CCOC)NC(c2cnn(C)c2C)=O)C)nc(C)cc1C 5026,C(CC(=C)Cl)(C(=O)N=c1cc(C)n(C)[nH]1)NC(COC1(C#C)COC1)=O 5027,C(=O)(C1=NN(C(C)C)C(=O)CC1)NCC1(F)CC(NC(C(CCCCC)O)=O)C1 5028,C1(CNC(CN(CCC)C(=O)OC(C)(C)C)=O)CCC2(CCOCC2)CO1 5029,C(=O)(CCCCC(C)(C)C)N1CCC(N(C)C(c2ccc(F)s2)=O)C1 5030,CCCC(C)(CC)C(=O)NCC1(F)CCCN(C(=O)CSC(C)(C)C)C1 5031,CCCCC(C)CCC(=O)NC(C)CN(C(C1CCC1)=O)CC 5032,c1(C(=O)NC(CCSC)C(=O)NO)ccc2c(c1)OCO2 5033,CCCC(CNC(=O)C(C)(C)c1ccno1)C(=O)N(C)CC1CC1(C)C 5034,C1(NC(C=NOC)=O)(CO)CCN(C(c2c[nH]nc2-c2cnn(C)c2)=O)CC1 5035,C(CCC)(C(=O)NC1CCCC(CN(C)C(c2cccc[n+]2[O-])=O)C1)=CCC 5036,C1(NC(C2C(C(N(CC#C)C)=O)C2)=O)CCCCC1N(C(=O)C=C(C)C(C)C)C 5037,C(=O)(C1=C(F)CN(C(C23CC(F)(C2)C3)=O)CC1)C(C1CC2CCC1CC2)=O.NC 5038,N1(C(CSCc2cccc(C)c2)=O)CCCC12CCN(C(c1ncoc1C)=O)C2 5039,C1(NC(C(C)O)=O)CCN(C(=O)CC(O)C2CCCC2)CC1 5040,O=C1NC2(CNC(N3CC4CC(C3)C(O)(C(F)F)C4)=O)CC3CC1C2C3 5041,C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CC(NC(COCC)=O)C(F)CC1 5042,CCC(C)C(C(=O)NC(CCC1CCC1)C(=O)NCCn1ccc(=O)cc1)N(C)C 5043,Cc1n[nH]c(C)c1C(=O)NCC1CN(C(=O)CCOc2ccccc2F)CCO1 5044,C1(C#CC(=O)N2CCN(C(=O)CC(C)=C(C)C)CC2CC(F)F)(CC)CC1 5045,C1(N(C)C)CCC(C(=O)NCC2(O)CCN(C(c3cccnc3)=O)C2)CC1 5046,c1(OC)cccc(NC(=O)CC2(NC(=O)CC3CC3(C)C)CC2)c1F 5047,c1(CC(=O)NC(C2CCCC2)CNC(C2(N(C)C)CC2)=O)cc(F)cc(F)c1 5048,c1(-c2ccc(C)cc2)nc(=NC2CCCC3CN(C(=O)C(C)SCC(N)=O)CC23)s[nH]1 5049,c1(C(C)C)ccc(C(=O)N(CCCCN(C(=O)C(F)n2cccn2)C)C)cn1 5050,Cc1nc2c(N3CCCC(C(=O)NCc4noc(C)n4)C3)ncnc2[nH]1 5051,C1(NC(c2c(C)nc(Cl)s2)=O)CC2(CCN(C(c3cc(C#N)c[nH]3)=O)CC2)C1 5052,C1(CNC(C(C)CC2CC2)=O)CCCCN(C(=O)CN2CCCCCC2=O)CC1 5053,CCCCC(O)C(=O)NC(CNC(c1ccc(F)cc1C(F)F)=O)CC 5054,C1(COC)CN(C(=O)C=CC(C)(C)SC)CCO1.C(=O)(CN(C(C)=O)C(C)C)O 5055,Cn1ncc2ncnc(N3CC4CN(C(c5cc(I)cnc5Cl)=O)CC34)c12 5056,CC1CCCN(C(=O)COc2cccc(F)c2)C1CNC(c1coc(Cl)c1)=O 5057,C1(C(=O)Nc2cn[nH]c2)CC2(CC2)CN1C(=O)C(=O)Cc1ccccc1 5058,C=C1CC(C(=O)NCCC)(CNC(=O)C(O)C2CCC2)C1 5059,C(=O)(C1CCCc2ccccc21)NC1CCN(C(c2c(C(C)C)cccc2)=O)C1 5060,CN1CC(C)(C)N(c2nnc(C3CCCC3)n2CC2CCC(C)(C)CC2)CC1=O 5061,Cc1cccc2c1C(NC(=O)NC1(CCOC(C)C)CC1)CCC2 5062,C(CC1CCOCC1)(C(=O)NCc1ncsn1)NC(C1CSC1)=O 5063,n1(CC(=O)NCC2CC3(CCN(C(=O)C=CCO)C3)CO2)ccc2c(O)cccc12 5064,C1(O)(C(C(=O)NCc2cn[nH]c2)NC(c2c(NC)scn2)=O)CCCCC1 5065,c1(C(=O)NC(CNC(c2ccc(C#C)cn2)=O)(C)C)cc2cc(C)cc(C)c2[nH]1 5066,CCCC(CCC)C(=O)N1CC2CC2(NC(=O)COc2ccc(C#N)cc2)C1 5067,CC1CN(C)CCCN1C(=O)CCCCN(C(=O)CC1CC(=O)C1)C 5068,C1(C#N)(OC)CC(C(N2CC(F)CC2CN(C)C(c2cnccc2C)=O)=O)C1 5069,c1(CNC(C2CCCN(C(c3cc(C)sc3C)=O)C2)=O)cc(C)c(F)c(C)c1 5070,C1(NC(C(=O)N(C(C)C)Cc2nc(C)c(C(=O)O)s2)=O)CC2(COC(C)C2)C1 5071,C(=O)(C(CC(C)(C)C)NC(c1c[nH]c(=S)cn1)=O)NCCCN(C)C 5072,C1(N(C(=O)CC2CCN(C(=O)C(n3ccc(C)n3)C)C2)CC)(OC)CCNC1=O 5073,Cc1nn2cc[nH]c(=O)c2c1C(=O)OCC(c1cc(C#N)n(C)n1)=O 5074,N1(C(C(CC)COC)=O)CC(C(N2CCCCC2CCOC)=O)C2(CCC2)C1 5075,Cc1nc(NC2CCCC(NC(=O)CCc3cccnc3)C2)c2scc(C)c2n1 5076,N1(C(CS(CC)=O)=O)CCOC2(C1)CN(C(=O)C(C)COC1CCOCC1)C2 5077,c1(C(N)=O)cc([N+](=O)[O-])ccc1N1CCC(NC(c2cc3sccc3[nH]2)=O)C1 5078,c1(N(CCCCC=C)C)nc[nH]c(=NCc2cc(C)ncn2)c1C 5079,C=CCC(CC(F)F)NC(=O)C(F)C(C)CNC(=O)Cc1ccoc1 5080,c1(C(N2CC(C)N(C(C3COC(=O)N3)=O)CC2)=O)nn(C)c2ccccc2c1=O 5081,C1(C)(C(N2CCC(OC)CC2C(C)C)=O)CCCN(C(=O)CSCCOC)C1 5082,N1(C(CSC)=O)CCN(C(c2nnn(-c3ccccc3F)c2C)=O)C2CCCC12 5083,C(C)(C)(CCCCC(=O)NCC(C1CC1)NC(=O)CC1CCCN1C(C)=O)OC 5084,c1(C(=O)NCCN(C(C2CC(C(F)(F)F)C2)=O)C2CC2)cccc2ccnn12 5085,C1(CNC(C2(C=C)CCC2)=O)CCC(C(=O)NCCN(C)CC)CC1 5086,CCCCC(CC)CC(=O)N1CC(F)(F)CC1CCNC(=O)CCOC1CCC1 5087,CCC(C)(C)CC(=O)N(C1CN(C(=O)C#CC(C)C)CCC1C)C 5088,C(CC(C)(C)NC(C1CCN(C(C2CC2c2ccccc2)=O)C1)=O)SC 5089,c1(C(C2CCN(C(=O)NC(c3cc(F)cc(F)c3)C)CC2)=O)cc(N)ccc1Cl 5090,C1(Cl)(C(N2CC(NC(c3cnn(CC(F)(F)F)n3)=O)C2)=O)CC12CCC2 5091,c1(OC)cccc2c(C(=O)OC)cc(SCCC3CNCC3C)nc12 5092,Cc1ccc(Oc2ccc(SC(C3CC=CCC3)=O)cc2)cc1C 5093,c1(C(c2nnnn2CC2CCOCC2)NCC2(CCC)CC2)cc(Cl)no1 5094,C12(C(=O)NCC(CNC(c3cc(SC)nn3C)=O)O)CC(C)(C1)OC2C 5095,C1(C)(CNC(C2N(C)CCN(C)C2)=O)CN(C(C2CCCCO2)=O)C(C)(C)C1 5096,C1(OCCCNC(C23COCC2C3)=O)CCCCC1C(=O)NCCCCOC 5097,C1(CC(=O)NC2CCCC(NC(C=CC)=O)C2)Cc2ccccc2NC1=O 5098,CC(C)(C(=O)NCCN(C1CCCC1)C(=O)CC1CCC(=O)N1)C1CCCCC1 5099,O=C(C1CCCc2ncccc21)NCCNC(c1cccn2nnnc12)=O 5100,C(=O)(C1CCCn2ccnc21)N1CCC2(C(NC(C(C)=CC)=O)C2)CC1 5101,C12(C(=O)NC)CCC(CF)(C1)OC2.n1(C(C2C(C)(C)C2)C(=O)N)cnccc1=O 5102,N1(C(C(=O)NC2CN(C(=O)NC)C2)=O)CCN2C(=O)NCC2C1 5103,C1(CC(=O)NC(COC)C(=O)NCC2NC(=O)NC2=O)COCC(C)O1 5104,N1(C(c2cn(C(C)(C)C)nc2)=O)CCCC(C2CN(C(c3cccnn3)=O)C2)C1 5105,c1(C(N2CCC(n3cc(CSCC)nn3)C2)=O)cc2n(n1)CCNC2=O 5106,C=CCC(C(=O)NC(CO)C(C)NC(=O)CCC(N)=O)c1ccccc1 5107,C(CC(C(=O)NCCC1CCN(C)C1)NC(=O)Cn1ccc(C)c1)OC 5108,C1(CC(N2C(CO)CC(NC(CCC=C=C)=O)C2)=O)CN2CCN1CC2 5109,N1(C(C(COC)N(C)C)=O)CC(C)CN(C(c2c(N)sc(C)c2C)=O)CC1C 5110,c1(C(N(CCOC(=O)NCC(C)SC)CC)=O)cc2c(nc1O)CCCCCC2 5111,c1(C(=O)NCC2(O)CNC2)ccc(F)c(F)c1.C1(C(=O)NC)CC(C)C1n1cccn1 5112,Cc1cc(C)c(C(N2CCC(O)C2C(=O)NCc2cccnc2)=O)cc1Br 5113,n1(CCNC(C=CC)=O)ccc(C(N2CCC(C(C)C)C2)=O)c1 5114,CCC(C)(C)C(O)C(=O)N1CCCCC1CN(C(=O)C(O)CC(C)C)C 5115,N1(C(C(=O)C(C2(CC(C)C)CC2)=O)C)CC(c2cn(CCO)nn2)(C(=O)OC)C1.CN 5116,N1(C(CNC(=O)OC)=O)CC(OC(C)(C)C)CC(NC(c2cc(C(N)=O)co2)=O)C1 5117,C12(CNC(=O)CC3CC=CC3)CCC1CCN2C(=O)C1=COCCC1 5118,C1(NC(CC(C=C)CC)=O)(CNC(c2nn(CC)nc2C)=O)CC2CCC1CC2 5119,N1(C(C=CC(CC)C)=O)CC2CN(C(c3ccc(C(F)(F)F)cn3)=O)CC12 5120,C1(C(=O)O)CC2CCC1N2C(C1(CN)CCOCC1)=O.c1(C)ccc(Cl)cc1F 5121,c1(C(=O)NC(CNC(C2CCN(C(C)C)CC2)=O)C)nsc2ccccc12 5122,C=Cc1ccc(CN2CCN(C(C3CCN(C(=O)CCC)C3)=O)C(=O)C2)cc1 5123,N1(C(C(C2CC(F)(F)C2)OCC)=O)CCC(CN(C(C2CC2F)=O)CC)CC1 5124,Cc1cc(C)nc(SCC(=O)NC2CC(O)(CNC(c3cnccc3Cl)=O)C2)n1 5125,c1(CC(C)C)c[nH]c(C(N2CCC(N(C)C(c3cnn(C)c3)C)C2)=O)c1 5126,c1(C(C)(C)C)ccncc1C(N1CCCCC1CNC(c1cncc(F)c1)=O)=O 5127,c1(C(N2C(CC)C(CO)CCC2)=O)ccc(CO)c([N+](=O)[O-])c1 5128,C1(C(NOCC(C)(C)C)=O)(CNC(C2C=CCS2)=O)CC12CCC2 5129,N1(C(C(C)N(C(C)=O)C)=O)CCN(C(=O)CCCCCN(C)C)CC1CO 5130,N12CCCC1C(=O)NC1CCCC1CNC(=O)C21CCC1.CNC 5131,C1(C(N(CCN(C(c2cnn(C3CC3)c2)=O)CC)CC)=O)CCNC(=O)C1 5132,C1(NC(CC2C(C)CCO2)=O)CC2(CCN(C(c3ccoc3C3CC3)=O)CC2)C1 5133,C1(CC=C)CCCN1C(C1(CNC(=O)CC2CSCCO2)CCC1)=O 5134,Cc1nn(C)c(Cl)c1C(N1CCCC(C)(CNC(=O)C(C)C2CCC2)C1)=O 5135,CC1OC(C)(F)CCN1C(COCC1CCOC1)C(=O)NC1CCC1 5136,Cc1ccc(Cl)c(F)c1C(=O)NCC=CCNC(=O)CCSc1ccccn1 5137,c1(C(N(C2CCN(C(C(F)=CCC)=O)C2)C)=O)ccc(=O)n(C)n1 5138,C1(Cl)(C(=O)NC2CC(NC(C(C)OCC)=O)C2)CC1(C)C 5139,c1(CN2CCCC(CNc3ccc(C(=O)OCC)cc3)C2)c(C)ccc(C)c1O 5140,c1(C(N(CCCNC(C2CC(C3CC3)C2)=O)CCC)=O)ccc2nn[nH]c2c1 5141,c1(OC)ccc(Br)c(CCN(C(=O)C(N)Cc2c(O)cccc2F)C2CC2)c1 5142,C1(CNC(C(=CC2CCCC2)C)=O)CCN(C(=O)CC2(O)CCC2)C12CC2 5143,C(C)(CCCCNC(c1cnc(OC)s1)=O)NC(c1cnc(CCCC)s1)=O 5144,Cc1ccc(-c2cccc(C(N3CC(CCO)C(C(N)=O)C3)=O)c2)cc1 5145,N1(CC(=O)N(CCC(C)NC(=O)COC(F)F)C)CCCC(N(C)C)C1 5146,S(=O)(=O)(c1cccc(NC2COCC2N(C)C)n1)NC(c1nncs1)C 5147,C(=O)(C1CCc2cc(F)ccc21)N1CCC(C2CC2)(NC(CC=C(C)C)=O)C1 5148,N1(C(C(C(C)O)N(C)C)=O)CC(C)(C)CC1CNC(c1sccc1CO)=O 5149,C(=O)(C1Cc2ccc(F)cc21)N1CC(OC)(CNC(=O)Cc2sc(O)nc2O)C1 5150,C1(N(C(CSCc2nc(C)sc2)=O)C)CCN(C(=O)Cc2cccnc2)CC1C 5151,CC(C)(CC(=O)N1CCN(C(=O)CCSCC(N)=O)C2CC12)CC(F)(F)F 5152,C(=O)(C(=O)CC(C)C)N1CC(CC)(NC(=O)Cc2cn[nH]c2)C1 5153,CC(C)C(C)(O)C(=O)N(CCCCCCNC(c1nnn(C)c1C(F)F)=O)C 5154,C1(C(=O)NCCC(C(=O)NCCCCN=[N+]=[N-])OC)CC2(CCCO2)C1 5155,C1(C(=O)NCC(C)(C)O)(CC)CCCN(C(c2csc(CO)n2)=O)C1 5156,c1(C(N(CCCN(C(c2nc(OCC)sn2)=O)C)C)=O)ccc(C#N)cc1F 5157,Cc1n[nH]c(=NC2CCN(C(C3CCCC4CC34)=O)C2)o1 5158,c1(CC(=O)NCC2(OC)CN(C(C3CC3(C)C)=O)C2)ccc(F)cc1C 5159,C(CCC(F)(F)F)(c1ccccc1)NC(=O)NCc1cccc(OC(C)C)n1 5160,C1(NC(C2C(C(C)O)C2)=O)CCC(CNC(c2cnn(-c3ccccn3)c2)=O)C1 5161,Cc1ccc(C(=O)NC(CNC(=O)Cc2ccc(C)nc2)C(C)C)c(N)n1 5162,c1(OC)cc(C(=O)NC2(C3CN(C(=O)C(C)S(N)(=O)=O)C3)CC2)cc(N)c1O 5163,Cc1cnn(C)c1-c1cn(CCN(C(=O)CCC(=O)c2ccccc2Br)CC)nn1 5164,c1(C(=O)NC2(C)CCN(C(c3c(C)cccc3O)=O)C2)ccc2cnccc2c1 5165,C(=O)(C1CCCn2c(C)nnc21)Nc1cncc(-n2c(C)cc(C)n2)n1 5166,C1(C(=O)NCC(C(C)(C)C)NC(C=Cc2c(C)ccs2)=O)CCc2nc[nH]c2C1 5167,CN1CCN(C(C2CCOC2)CNC(=O)COc2cnn(C)c2)CC1 5168,CC1CCC(NC(C2CC3CC3CC2C)=O)CN1C(C)C(=O)NC(N)=O 5169,N1(C(C(c2cccnc2)(C)C)=O)CC2CN(Cc3c(Cl)cncc3Cl)C2C1 5170,N1(C(CCSCCC)=O)CCC(C2CC2)C1CNC(=O)C(F)=C(C)C1CC1 5171,Cc1c(CNC(=O)NC2CCCC(C(C)C)C2)nc2ccccn12 5172,c1(C(=O)NC(C(C)C)CCNC(c2cc3n(c2)CCC3)=O)ccc2nncn2c1 5173,CCCC(C)(O)C(=O)NCCn1ccc(C(=O)NCCC2CC(F)(F)C2)c1 5174,c1(OC)ccc(C=CC(=O)NC(Cc2ccc(S(N)(=O)=O)s2)C(=O)O)cc1F 5175,C12(C(=O)NCC3(OC)CCOC3)COCC1CN(C(C1CCC1C)=O)C2 5176,c1(C(N2CCN(C(C(c3cccc(O)c3)=O)=O)C3C2C3)=O)cc(Cl)cc(Cl)c1Br 5177,CON1CC(CC(N2CCC(N(C)C(C3CC=CCC3)=O)CC2)=O)CC1=O 5178,C=CCCCC(C(=O)NCC1(F)CCC1)NC(C1C2CCCC(=O)C12)=O 5179,N#CC12CCCCCC1CN(C(=O)C(NC1COCc3ccccc31)=O)C2 5180,N1(C(CCC(=C)C)=O)CCC(C)CC1CNC(c1ncc(Cl)cc1O)=O 5181,Cc1cccn2cc(C(N3CC(CNC(=O)CSC(C)(C)C)C(F)C3)=O)nc12 5182,Cc1sncc1C(=O)NCC=CCC(=O)NCCS(C)(=N)=O 5183,c1(CN)cccc(Br)c1OC.CC(Cc1cnc[nH]1)C(=O)NCC1CC1 5184,C(=O)(CCCCC(C)(C)C)N1CCC(F)(CNC(c2c(C)con2)=O)CC1 5185,CC1(NC(=O)CC2CC=CCC2)CCN(C(C2CCC3CCC2O3)=O)CC1 5186,C(Cn1cncn1)(C(=O)NC1CC1CCCCO)NC(c1cc[nH]n1)=O 5187,N1(C(c2ccc(SC)o2)=O)CC(C)CCC1CNC(=O)COc1cnn(C)c1 5188,c1(NCC2CCC(NC(CN3CC(C(=O)OCC)C3)=O)CC2)cc(C)ccc1O 5189,c1(CC(=O)NCCCCCNC(C(CCC)F)=O)ccc(F)cc1C 5190,Cc1cnccc1C(N1CCCC1CN(C)C(c1cnn(CC(F)F)c1C)=O)=O 5191,C1(C(=O)OC)C(F)(F)C12CC(C(N1CCCC(CNC(C)=O)C1)=O)C2 5192,C(CC(C)C)(C(=O)N(CCCCCNC(C1CC12CC(C)(C)C2)=O)C)NC(C)=O 5193,C(=O)(C1=CC2CCCCCCC12)N1CCCC(C)(CNC(c2nsnc2O)=O)C1 5194,C1(C(=O)NCC=CCNC(C2CCCCC2F)=O)CCC(=C(F)F)CC1 5195,c1(C(N2C(C(=O)Nc3ncc(C)cc3I)CC(OC)C2)=O)cc(C)c(C)cc1C 5196,CC1OC2(C(=O)N)CC1C2.c1(CC(CCCN(CC)C2CC2)=O)ccccc1 5197,CC(C)(C)CC(=O)NCC(CCN(CC=CC(=O)N)CCOC(C)(C)C)O 5198,CCCC(CC)C(c1nnnn1CC1CC1)NCc1nnnn1-c1ccccc1 5199,CC1c2ccccc2OC1C(N1CC(NC(=O)COCCF)C(C)C1)=O 5200,N(C(=NCc1cccc(F)c1)NCC12CC(C1)C(C(F)F)O2)C(C)C 5201,CC(C)C#CC(=O)NC1(CCCC(=O)NCC2COCC2O)CCC1 5202,N1(C(C(C)SC(C)C)=O)CCC2CN(C(c3ccoc3Cl)=O)C(CO)C12 5203,c1(CNC(C(=O)NC2(CNC(CC3(C)CC3(F)Cl)=O)CCC2)=O)cccc(F)c1 5204,CN1CCC(N(CC(O)CN(C)C(=O)Nc2occc2Cl)C)CC1 5205,C1(C(=O)NCC(C(C)O)O)CCC2(CC2)N1C(c1cccc(CO)n1)=O 5206,c1(C(=O)NC(C2CCN(C(=O)CC3CC(F)C3)CC2)C)ccnc2ccncc12 5207,C1(C(=O)NC2C(C)(C)C2)(CNC(C2CC(N3CCCC3)C2)=O)CC12CCC2 5208,C1(CNC(CC(C)(C)SC)=O)CCC(C)N(C(c2ccc(F)s2)=O)C1 5209,C(=O)(CCOc1cnns1)N(CCCOCOCC(N)=O)C 5210,CCC(C)(C)C(O)C(=O)NC1CN(C(c2cc(Cl)cc(C)c2O)=O)CC1OC 5211,C1(C(=O)NCC(c2ccsc2)C)CC=CCN1C(c1cccc(CO)c1)=O 5212,c1(C(N2CCC(C)(CNC(Cc3c(C)nsc3)=O)C2)=O)ncc(C2CC2)cc1F 5213,N1(C(C(CCCC)(C)F)=O)CC2(CCN(C(=O)CCCC(=O)NC)CC2)C1 5214,CC1SCCN(C(C23CC(CN2C(=O)C=CCN2CCCC2)C3)=O)C1C 5215,c1(CC(=O)OCC(CC2C(c3cn(C)nc3)C2)O)ccccc1F 5216,N1(C(CC=C=C)=O)CCC2CN(C(c3ccn4nncc4c3)=O)CCC2C1 5217,N1(C(C=CC(CC)C)=O)CC2CCOC2(CNC(c2cc(CC)cc(C)c2)=O)C1 5218,N1(C(C(C(=C)C)(C)O)=O)CCC2(CC1)CC(CNC(=O)CCC(C)C)C2 5219,c1(OCC)cc(C(=O)NCC2CC(NC(C3CCC(COC)O3)=O)C2)[nH]n1 5220,C(=O)(C(CC(C)C)N(C)C(c1c(C)cnn1C)=O)NC(CC)COCC1CC1 5221,Nc1ccccc1C(=O)NCC(=O)NC1CC12CC(NC(C1(COC)CC1)=O)C2 5222,S(=O)(=O)(c1cc([N+](=O)[O-])ccc1Cl)NC1(CC#C)CCCC1 5223,C1(NC(C=CCCOC)=O)CN(C(c2ccncc2OC)=O)C(C)(C)C1 5224,C1(C(C)=O)COCCN(C(=O)C(C(C)C)OC(=O)Nc2cccc(C#N)c2)C1 5225,Cc1c(C(=O)NCCCN(C(C2CCC(=O)O2)=O)C2CC2)c[nH]c2nccc1-2 5226,N1(C(C(CC)C#N)=O)CC2(CCOCC2)CC1CNC(c1cc(F)ccc1F)=O 5227,CCCCC(C)CCC(=O)NC1CCCCC1C(=O)N(C(C)Cn1cnnc1)CC 5228,C(C(CC)(CC)NC(=O)Cc1ncc(C)s1)NC(C(CC)F)=O 5229,C1(CC=C)(NC(=O)C(C)=CC(C)(C)C)CC2CCC(C1)N2C(c1snc(C)c1N)=O 5230,C(=O)(CC(C(F)F)NC(=O)CC1CCCNC1=O)NCC(C)CO 5231,C1(OC)CC(CNC(=O)CC2CC2)CN(C(=O)CC(C)CCc2ccccc2)C1 5232,C1(CC=C)(NC(=O)CC2CCOCC2)CC2CCC(C1)N2C(=O)C=CC(C)=O 5233,C(=O)(CS(=O)(=O)CC(C)C)NC1CCC(CCNC(C(CC(C)=O)(C)C)=O)C1 5234,CC1CCN(C(=O)CCn2ccnn2)C(CNC(C2CCCS(=O)(=O)N2)=O)C1 5235,c1(CCNCc2n(CCCC)nnn2)ccccc1-c1ncc[nH]1 5236,N1(C(C2CC(OCC)C2)=O)CCC2(CNC(=O)Cc3ccc(O)nc3)CCCC12 5237,C1(C(N(CCCN(C(C(C)SCCCC)=O)C)C)=O)CC12CCOCC2 5238,C(CCCC(=O)NCC1CCCN1C(=O)CCCn1cnc(C#N)n1)OC 5239,CCC(C)(C)C(C)(O)C1CCNCC1.OC(F)F 5240,c1(C(N2CCN(CCNC(c3ccn(C)n3)=O)CC2)=O)ccc(C(F)F)c(F)c1 5241,C(=O)(C(C)CC(=O)c1ccc(Cl)cc1)NC(CCNC(c1c(C)cco1)=O)C 5242,C1(NC(COCCCCC)=O)C(C)(C)CN(C(=O)C(C)CC(C)CC)CC1(C)C 5243,N(C1c2ccccc2CC1C)C(C(CC)C)c1nnnn1CCCOC 5244,N1(C(CC(C=C)C)=O)CCC(C(=O)NC(c2nc(=O)o[nH]2)C)C1(C)C 5245,N1(C(c2c(COC)cco2)=O)CC2CC(C(=O)NC(C)(CO)CC(C)C)C(C2)C1 5246,c1(C(=O)NCC2CC(F)(CNC(C3CCC(C)O3)=O)C2)cnc(O)c2ccsc12 5247,c1(C(=O)NC2CCN(C(C3N(N=O)CCC3)=O)C2)ccnc2c1CC(=O)N2 5248,c1(C(=O)NCC(C)(C2CC2)NC(CC2CN(C)C2)=O)ccc2c(n1)OCCO2 5249,C1(C2CC2)(CNC(CCC(C)(F)F)=O)CCN(C(c2cncc3ccsc23)=O)C1 5250,c12cnn(c1)CCNC2=O.N1(CC)CCC(NC(=O)N(C2CCCCO2)C)C1 5251,C(=O)(C(CO)N(C(=O)CN=[N+]=[N-])C)C1CC(C#C)NCC1 5252,Cc1nn(C)c(Cl)c1-c1nc(Cc2cc(-c3cccnc3)nn2CC(F)F)no1 5253,CCC1=C(C(=O)NCC2CC(CNC(c3cc4cscc4s3)=O)CO2)CCCO1 5254,N1(C(CCCN(S(C)(=O)=O)C)=O)CC(NC(=O)C(O)C(C)(C)C)C2(CC2)C1 5255,CCC(CCOC)C(=O)N1CCCC(Cc2ccccc2)CC1 5256,c1(CC)ccc(C)nc1NC(C1(F)CCCN(C(C2CCCO2)=O)C1)=O 5257,CC1CC(N(C(=O)CC2(CNC(=O)COCC(F)F)CC2)C)CC(C)C1 5258,CC1CC(C)CN(CCCC)C1.c1(C2(C=O)CC2)cc(F)cc(F)c1 5259,N1(C(COCCC(C)C)=O)CC2CC(C1)C2NC(c1ncoc1C1CCC1)=O 5260,c1(C(N(C2CCC(NC(Cc3scc(C)c3)=O)C2)C)=O)cc2n(c1)CCOC2 5261,c1(OC)ccnc(C(=O)NCC2(NC(=O)CC3CC(C)=NO3)CCC2)c1 5262,C1(C(N)=O)CCN(C(=O)CC2CCCC(=O)C2)CC1.C12CCC(C3CC3)N1C2=O 5263,c1(CC(=O)NCc2cn(Cc3cccc(Cl)c3)nn2)c(F)ccc(Br)c1Cl 5264,C1(C(C)C)CCCN1C(=O)C(O)CN(C(=O)CC1CC=CC1)C1CC1 5265,C1(CNC(C2C(C=C(C)C)C2(C)C)=O)(NC(c2nnn(C)c2N)=O)CCCCC1 5266,c1(C(N2CCC(C)(NC(C3CN(CC)C(=O)C3)=O)C2)=O)ncnc2cc[nH]c12 5267,c1(SCC)cccc(C(N2CCCC2C2CCCN(C(C3CCCC3)=O)C2)=O)c1 5268,c1(CCOC(C)=O)cc(CCO)ccn1.N12CCCC(C1)Cn1cc(nn1)CS2 5269,O=C(C1=CCCC1)NC1(C2CCCN2C(=O)Cc2n[nH]cc2Br)CC1 5270,CC1CN(C)CC(C(=O)NCC(C)(C)NC(=O)COc2cccc(O)c2)O1 5271,c1(CC(=O)NCCN(C(C2CC(O)C2)=O)C2CC2)cccc2[nH]ncc12 5272,c1(Cn2cc(C(Cc3ccccc3)NCCCCCC)nn2)cccc(Cl)c1Br 5273,Cc1cccc(C(=O)NC2CC2C(=O)NC2CCC(N3CCOCC3)CC2)c1I 5274,N(C(=NCc1cc(CN2CCCC2)co1)N1CCC(COC)C1)C(C=C)C 5275,C1(C)(C(N(C)CC2N(C(c3ncc(C)cc3C)=O)CCC2)=O)CCC(F)(F)CC1 5276,N1(C(CC(C)F)=O)CC(NC(=O)CCOC2COC2)C(C)C1 5277,Cc1cc(CC(=O)OCc2ccnnc2)c(Br)cc1F 5278,C1(COC)(NC(c2nn(C)cc2Cl)=O)CCN(C(c2nccc(C)n2)=O)C1 5279,c1(C(C(N2CCC(N(C(=O)C=CC(C)(C)C)C)C2)=O)(C)C)ccc(Cl)cc1 5280,c1(CC)cccc(C)c1C(N1CCN(C)C(CNC(C2CC(OC)C2)=O)C1)=O 5281,c1(C(N2CCCN(C(=O)C(C3CC3)C3CC3)CC2)=O)cc2c(nc1O)CCOC2 5282,Cc1cnc(C#N)nc1NC1COC2(C1)CN(C(=O)CO)C2 5283,CC(C)(C)C(CNC(C1CCC(F)(F)C1)=O)NC(c1ncccc1Br)=O 5284,c1(CN2CCC(C(=O)Nc3cc(SC)n[nH]3)CC2)ccc(Br)c(C#N)c1 5285,C(=O)(CC(F)(F)CC(=O)NCC(C(C)(C)C)NC(C1CCC2(CCC2)C1)=O)OC 5286,C(=O)(C1=CCC(C)(C)CC1)N1C(CNC(c2c(C)oc(C)c2C)=O)CC(F)(F)C1 5287,C1(NC(c2cc(C)nn2C(F)F)=O)CCC(C)N(C(c2cnccc2Br)=O)C1 5288,Cc1cnc(NCc2nc(=N)n(C)[nH]2)c(S(=O)(=O)N2CCC(C3CCC3)C2)c1 5289,CC1(C)CN(C(=O)CC2CSCCO2)CCC1C(N1CC2(CCOC2)C1)=O 5290,C(C#Cc1cccnc1)NC(=O)COCCNC(=O)CC1COCCO1 5291,N1(C(C2CC(C)(F)C2)=O)CCCC12CCCN(C(c1cccc3c1CCN3)=O)C2 5292,N1(C(CSCCCC)=O)CCN(C(=O)C(C)c2ccsn2)C(CC(F)(F)F)C1 5293,C1(C(N(CCCN(C(CC=CCC)=O)C)C)=O)Cc2cccc(OC)c2O1 5294,c1(C(N2CCC(C)(CNC(=O)Cc3ccoc3)CC2)=O)ccc2nc[nH]c2n1 5295,c1(C(N(C2CCN(C(C3CC3OC)=O)C2)CC)=O)ncccc1C(F)(F)F 5296,c1(C(N(CCN(C(=O)CN2C(=O)CCC2=O)CC)CC)=O)cccc(C2CC2)c1 5297,C1(CN2CC(C(=O)Nc3ccnc(C4CC4)c3)C2)CC12CCCOC2 5298,CCC(CC(C)C)C(=O)NCCC1(NC(=O)CCc2cncs2)CCCC1 5299,Cc1nc2n(c1C(N1CC(C3CCCN3C(=O)CCOC(C)C)C1)=O)CCCC2 5300,n1(C(C)C)cc(C(=O)NCC(C)NC(C2CCN(c3nccn3C)C2)=O)cn1 5301,C1(NC(=O)C(N2CCC(CC3CC3)C2)=O)CCC2CN(C(C3CCOC3)=O)CC2C1 5302,c1(CN2CCCC(CC(=O)NC(CC)C(F)(F)F)C2)cc(OC)ccc1F 5303,N1(C(C2C(OC)C2)=O)CCC1CNC(C1CC(n2ccnc2)C1)=O 5304,c1(C(N2CCCN(C(CCC(CC)C)=O)CCC2)=O)c[nH]c2cc(Cl)ccc12 5305,CCC(C)C(C(=O)NCc1cn(CCCC2C=NN(C)C2=O)nn1)OC 5306,C(=O)(C(C)C(C)S(C)(=O)=O)N1CC(F)(c2cn(C)nn2)C1.c1(CCC)cccnc1 5307,CCCCCCC(F)C(=O)N1CCCC1CN(C)C(c1cncc(OC)c1)=O 5308,c1(OC)ccc(Cl)cc1CC(N1CCC(NC(=O)CCN2CCCC2)C1)=O 5309,C=CCC(CNC(=O)CCN1CCCC1)C(=O)NC1CC(CO)C12CCC2 5310,c1(C(C)=O)csc(C(=O)NCC(C)(C)CN(C(=O)C(F)(F)c2ncccn2)C)c1 5311,N1(C(CCCC#C)=O)CC(C)N(C(c2ccc(C3CCOC3)cc2)=O)CC1C 5312,N12CCC(CC1)c1nc(no1)NC2=O.CC(C(F)F)C1CC1 5313,C#CCC(CC(=O)NCC1CCN1C(C)(C)C)NC(=O)COC1CC1 5314,C1(C(N2CC(n3ccnc3)C2)=O)(CC)CCN(C(c2n[nH]c(C)c2Cl)=O)C1 5315,Cc1cnc(C(N2CCC(CNC(C3CC3(Cl)Cl)=O)CC2)=O)cc1C#N 5316,C1(NC(C(C)SCC)=O)CN(C(=O)C(c2ccc(F)c(C)c2)=O)CCC1O 5317,Cc1ccc(SC(C)C(=O)NC2C3CN(C(=O)C(C)C)CC23)cc1 5318,c1(C(N2CC3CC(CNC(c4n(C)cc(Cl)c4)=O)C3C2)=O)cc2cccnc2[nH]1 5319,c1(CC(=O)NCC(CO)NC(c2ccoc2Br)=O)csc2nccn12 5320,c1(C(=O)NCC2(C(C)NC(C3CC3C(F)F)=O)CC2)cnc2ccccn12 5321,Cc1nn(CCO)cc1C(=O)NCC(O)CN(C)C(C1(C(C)C)CNC(=O)C1)=O 5322,c1(N2CC(CC(=O)OC(C)(C)C)OCC2)c(Br)cncc1[N+](=O)[O-] 5323,c1(C(N(C)CC2N(C(C3(COC)CCOC3)=O)CCC2)=O)ncccc1Br 5324,c1(C(=O)NC(C(=O)N(C)Cc2ncnn2C)(C)C2CCC2)cn2ccccc2n1 5325,CC(CNC(=O)C(C)(C)C1CCC1)C(F)C(=O)NC1(C(=O)N(C)OC)CC1 5326,c1(OC)cc(C)ccc1CC(N1CCNC(=O)C1c1cccc(Br)c1)=O 5327,C1(CC(=O)N(C2CCN(C(C3CC(F)C3)=O)CC2)CCOC)CC2(CCO1)CC2 5328,C(=O)(C(O)CC(=O)OC(C)(C)C)N(C1CCCN(C(c2cc(Cl)no2)=O)C1)CC 5329,C1(F)(CNC(C(C)(C)F)=O)CCN(C(C2CC(c3cccnc3)C2)=O)C1 5330,c1(N2CC3(CCN(C(c4c(CC)nco4)=O)C3)C2)nccc2c1C(=O)OC2(C)C 5331,c1(C(N(CC(CNC(c2c(C)ccc(C)n2)=O)O)C)=O)cc2cc(F)ccc2o1 5332,C1(C(C(=O)NCC#C)NC(=O)CC2(C3CCCC3)CCC2)CCCOC1 5333,C(=O)(C1c2ccccc2C2(CC2)CN1C(=O)N(c1nccs1)CC(C)C)OC 5334,N12CCC3(CCN(C3)OC(=O)c3c(cco3)C1=O)C2.c1(CC)c(Cl)nn(C)c1C 5335,CCCCCC(CC)C(=O)NCC1(CO)CCN(C(c2cc(N)cc(F)c2)=O)C1 5336,c1(C(N(C2CCCN(C(=O)CC34CC(C3)C4)C2)CC)=O)noc2c1CCCCC2 5337,CC1CC(C(N2CCC(O)C2c2ccccc2)=O)N(C(=O)C=CC2CC2)C1 5338,C1(C(N2CCCC(CNC(c3ccc(C)cn3)=O)CC2)=O)Cc2cccnc2C1 5339,C1(C(=O)NC(CC(=O)OCC)C)(C(C)C)CCN(C(=O)C=Cc2cocn2)C1 5340,C(C1=CCCCC1)(c1n(CCOC)nnn1)NCCCC(C)O.c12ccc(cc1)OC2 5341,C1(F)(CNC(c2cnco2)=O)CC2CCC(C1)N2C(c1noc2ncccc12)=O 5342,C(=O)(C(F)C(C)C)NC(C(=O)NC(CN(CC)CC)C)C1CCCC1 5343,CC(C(C(=O)c1cccc(F)c1)NC(C1(CC2CC2)CC1)=O)c1ccccc1Cl 5344,Cc1cccnc1C(N1CC(F)CC1C(N1CCCC(CN=[N+]=[N-])C1)=O)=O 5345,C(CCCCO)N(C)C(c1cc(CNC(=O)CCc2cccn2C)cs1)=O 5346,C1(N(C(=O)C=C2CCC2)C)CCCN(C(=O)CCCC2(C)N=N2)C1.c1cn(C)nn1 5347,C1(CNC(c2c(CC)ncnc2)=O)CCCCN(C(C2COC(=O)N2C)=O)C1 5348,N1(C(C(CC=C)C(C)C)=O)CCN(C(=O)CCS(N)(=O)=O)CC(C)(F)C1 5349,c1(CNC(C(=O)NC(C)C)=O)ccccc1CNC(c1cc[nH]c1C(F)(F)F)=O 5350,N1(C(C(C)(C)n2cccn2)=O)CC2CC2(CC(=O)NC2CC23CCC3)C1 5351,CC1CCC(NC(C2(C)CCC2)=O)CN1C(c1cnn(C(C)(C)C)c1N)=O 5352,N1(C(C(=O)Nc2cc(C(=O)OC)n(C)c2)=O)CCS(=O)(=O)C2(CCCC2)C1 5353,n1(C=O)cc(C(N2CCC2)=O)nn1.C1(CC(=O)NCC2CC(CN)C2)(C(C)C)CC1C 5354,CC(F)(F)CC(=O)NC1CC(C)(CNC(=O)CNC(N)=O)C1 5355,N1(C(C(C)NS(C)(=O)=O)=O)CC(O)CC1CNC(C1CCC(CO)CC1)=O 5356,Cc1cnc2n1CCC(C(=O)NC1CC13CCN(C(c1cc[nH]n1)=O)CC3)C2 5357,c1(C(=O)NCCC2OCCN(C(C(OC)OC)=O)C2)cnn2cccnc12 5358,CCCCC(C(=O)N(CC(CC)NC(c1cnn(C)c(=O)c1)=O)CC)ON=C(C)C 5359,c1(CC(N2C(C(C(=O)NCCC3(OCC)CCC3)(C)C)CCC2)=O)cncnc1 5360,N1(C(C(CCC)NC(C)=O)=O)CCN(C(C2CN3CCN2CC3)=O)C(C(C)C)C1 5361,C12CCCN(CC1)C(=O)COCCn1cc2nn1.c1(Oc2cn[nH]c2)cccnc1 5362,N1(CC(=O)NC2CCC(NC(C3(Br)CC3)=O)CC2)CCNC(=O)C1 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5397,c1(NC(c2cccc(NC(CCc3cncc(C)n3)=O)c2)=O)ccc(Br)c(Cl)c1F 5398,c1(C(c2n(C(CC)C)nnn2)NCc2csc(Br)c2)cnc(C(C)C)c(Cl)c1 5399,c1(OC)ccc(NC(C2(C)CCCN(Cc3cccc(F)c3)C2)=O)c(F)c1 5400,C1(C(N2CC(c3ccco3)C2)=O)CC2CCC1N2C(=O)C(O)CC1CCCC1 5401,CCCCC(C(=O)NC1CCC(NC(c2ccc(F)cn2)=O)C1)C(C)C 5402,C1(C(=O)NCC=CCCC)CC(F)(F)CN1C(=O)C(CC)NC(=O)NCC 5403,CCC(C)CC(C(=O)NCc1cncc(F)c1)NC(=O)CCc1nncn1C 5404,C(=O)(CC(C)(C)CNC(c1cc(Cl)no1)=O)NC1C(C)CCC1 5405,N1(C(C)=O)CC(n2cc(C3(N(c4cccn4C)C)CC3)nn2)C(C)C1 5406,C1(F)(CNC(C(C)OCC)=O)CCCN(C(C2(CO)CCCCC2)=O)CC1 5407,C1(NC(C2(SC)CCC2)=O)CC(O)CN(C(=O)CC2CCC3(CCC3)O2)C1.C(=O)N 5408,C1(C(=O)NCC(CCNC(=O)C=CCF)OC)CCc2nn[nH]c2C1 5409,CC12CC(C(=O)NC3CN(C(C4(O)CCSCC4)=O)CC34CC4)(C1)C(C)(C)O2 5410,N1(C(C(CC=C)(C)C)=O)CC2(CCN(C(C3C=CCS3)=O)C2)C1 5411,C1(NC(C2C(CCC)C2)=O)CC2(C1)CC2NC(=O)COCc1nc[nH]n1 5412,N1(C(c2c(C)nns2)C(=O)NC(C)C(=O)OC)CCC(=Cc2cccnc2)CC1 5413,CC1(C)CC(O)CCN(C(=O)C(C2(C)CC2)NC(=O)CCCC(F)(F)F)C1 5414,CC(C)C(C)C(CNC(=O)Cc1cncc(F)c1)NC(=O)Cc1ccns1 5415,C(=O)(C(C)(C)C(C)(F)F)N1C2CC(NC(CNC(CN(C)C)=O)=O)C(C2)C1 5416,CCC(CC)C(C)C(=O)N1CCN(C(=O)C(=O)NCC2CC2)CC1CC 5417,CC12CCC(C(=O)NC3CC(O)CN(C(c4cn(C(F)F)cn4)=O)C3)(CC1)CO2 5418,C(=O)(CC1=CSC2=NCCN12)NCCCC(C)NC(C1COC(=O)C1)=O 5419,N1(C(C2CCN(C(N)=O)C2)=O)CC2CCN(C(=O)COc3ncccc3O)C2C1 5420,c1(C(N2C(CN(C(CCOC)=O)C)COCC2)=O)cccc(Cl)c1C(F)F 5421,C1(NC(C2CC2F)=O)CCC2CN(CC3N(C)CCCC3)CC2C1 5422,c1(CNC(C2N(c3nnc(C)s3)CCCC2)=O)ccc2c(c1)C(=O)NC2=O 5423,CC1(C#CC(=O)N2CCC(N(C(=O)C(O)c3cnc[nH]3)CCO)C2)CCCO1 5424,c1(C(=O)NCCC2CN(C(C3CC(OC)C34CCC4)=O)C2)nc2c(s1)COCC2 5425,c1(NC(CC(C)NC(C2C(COC)C2)=O)C)cc2c(cc1[N+](=O)[O-])C(=O)NCC2 5426,C1(NC(C=CC=CC)=O)CCSC12CN(C(=O)CSC1CCCCO1)C2 5427,C1(CCNC(C=CSC)=O)CCCN(C(c2ncsc2-c2ccccc2)=O)C1 5428,CCCS(=O)(=O)c1ccccc1S(=O)(=O)CC(C)CC(=O)NCC1CCNC1 5429,c1(C(=O)NC2C(CNC(=O)CCNC(C3CCC3)=O)C2)cnc2ccncc2c1 5430,C#Cc1ccc(C(=O)NCC(O)C(=O)Nc2c(C)nn(C)c2N(C)C)nc1 5431,C1(C(N(CCCN)C(C2(C#N)CC(C)C2)=O)=O)CS(=O)(=O)CC12CC2.CC 5432,CCN=C(NCC12CC(CC1)OC2)NC1CCCC(C(C)C)C1 5433,c1(-n2cc(CN3CCN(C(C4CC(=C)C4)=O)CC3)nn2)ccc(S(C)(=O)=O)nc1 5434,N1(C(CCC=CCC=C)=O)CC(=O)NC1C(N1CCOC(C2CC2)C1)=O 5435,N1(C(C2C(C)OCCC2)=O)CC2(CCN(C(c3nc4c(s3)CCCC4)=O)CC2)C1 5436,C1(CC)C(C(=O)NCC(C)CNC(=O)C=C(C)C(C)C)CCN1C 5437,C12CCCCC1C(=O)NC2.C(=O)(C(C)CC1CCCC1)C(C(C)SCCCC)=O 5438,Cc1c(-n2nnnc2C2CC23CC(C(C2C4CCC(F)(F)C24)N)C3)cccc1Cl 5439,CC(CCCC(=O)N1CCOC(CCF)C1)NC(=O)COCCN(C)C 5440,c1(C(=O)NCCCOCCN(C(c2c(C)cco2)=O)C)cc2cc(O)ccc2[nH]1 5441,C1(C(N(CCCNC(C(C)OC)=O)CCO)=O)CC(=O)NC(=O)N1 5442,C1(NC(CCSCC(C)C)=O)C(C)CN(C(c2ccc(C(C)(C)C)s2)=O)CC1C 5443,C1(C)(C(=O)Nc2c(SC)nccc2)CC(O)CN1C(c1cnn(CC2CC2)c1)=O 5444,N1(C(c2ccc(CC)nc2C)=O)CCN(C(c2nscc2N)=O)CC12CCC2 5445,c1(CCC(=O)NCC2(F)CCN(C(C(C)C(F)F)=O)C2)ccc2cccnc2c1 5446,C(C1CN(C(c2csnn2)=O)Cc2ccccc21)NC(CCC1(C)CC1(F)F)=O 5447,N12CCC(CC1)NC2=O.n1(CC(CC)C)cc(C(C)(C)CC2CCC2)nn1 5448,c1(N2CC(F)CC(OC)C2)nc2cc[nH]c2c(=NCc2ccnc(C)n2)[nH]1 5449,c1(C(N2CC=CC(NC(C(CCC)OC)=O)C2)=O)cc2c(cn1)COCC2 5450,CCC(C)(CNC(=O)CC(C)N(C)C)C(=O)NCC1(CO)CC12CCC2 5451,C(=O)(C(F)(F)C1CCCC1)NC(C1CCCN1C(=O)CSc1n[nH]c(=N)s1)(C)C 5452,C1(N(C)C(c2ccc(C3CC3)s2)=O)CCC(NC(C2CC(=C3CC3)C2)=O)CC1 5453,C1(C(=O)NCCC(C(C)C)NC(c2cc[n+]([O-])cc2)=O)CC(=O)N(C)C(=O)N1 5454,S(=O)(=O)(c1ccc(C#N)cc1C(F)(F)F)N1C(C(=O)OC)CC(OC(C)=O)C1 5455,c1(COCC(=O)NC2C(CNC(C3=C(C#N)CCC3)=O)C2)ccc2c(c1)OCCO2 5456,N1(C(C2CCC(CC)O2)=O)CCCC(O)(CNC(C2CC3C=CC2O3)=O)C1 5457,CC1CCCc2c(OCc3cn(CC4NC(=O)CC4(C)C)nn3)cnn21 5458,N1(C(Cc2cccc(CC)c2)=O)C2CCC1C(C)C(NC(c1nc(C)no1)=O)C2 5459,C(=O)(CCCS(N)(=O)=O)N(CC)CC1CCCCN1C(C1CC2CCC1O2)=O 5460,C(=O)(C(O)C(C)C)NCC(CNC(C1(CS(C)(=O)=O)COC1)=O)OC 5461,Cc1ccccc1CC(=O)N(CC(C)CNC(c1ccc(SC(F)(F)F)s1)=O)C 5462,C1(C(=O)NC23C(CN(C)C2)C3)CC2CCC(C1)N2C(c1cccc(Cl)c1F)=O 5463,c1(C(N2CCC(C)CC2CNC(C2CC2C)=O)=O)cc([N+](=O)[O-])cnc1N 5464,c1(C(=O)NCCC(C)NC(=O)C(C2CCCCC2)=O)cccc2c1COCC2 5465,Cc1nn(C)c(C)c1CNC(C1CC(C)N1C(=O)CCC1CCOCC1)=O 5466,c1(C(=O)NCC(CNC(c2c(C)con2)=O)CO)cc2c(C3CC3)cccc2[nH]1 5467,C(N=C(NCC1CCCCO1)N1CCC(O)CC(C)(C)C1)c1n(C)cnc1 5468,Cc1nccc(C(=O)NC2(CCNC(=O)COc3ccsc3Cl)CC2)n1 5469,N1(C(c2c(C)ncnc2O)=O)CC(C)CN(C(=O)Cc2ccc(F)cc2)CC1C 5470,C(=O)(CC(C)(C)C(=O)OC)NC1(C(=O)NCc2cnc(CC)s2)CCC1 5471,c1(C(C)=O)cc(=NCCCCNC(c2ccc3c(c2)nnn3C)=O)[nH]cn1 5472,C(=O)(CCCCCNC(=O)C(c1nc(C)sc1C)N(CC(=O)NC1CC1)C)OC 5473,CN1C(=O)CCC1(C)CNC(=O)CC(CC1CC1)NC(c1ccc(Cl)o1)=O 5474,Cc1cc(F)cnc1C(=O)NC1COCC1NC(=O)CN1CCCC1CO 5475,N1(C(C2C(C)(C)C2C#N)=O)CC23CCCC2(C1)CN(C(=O)CCOC1CC1)C3 5476,N1(C(C(=O)NCC)=O)CCCN(C(c2ccnc(OCC(F)F)c2)=O)CC1CO 5477,C12(NC(C(C)N(C3CC(CNC(=O)C(O)C4(C)CC4)C3)C)=O)CCCCC1C2 5478,C(C(C(=O)NCC(=O)NCCO)NC(c1ccoc1)=O)NCC(N)=O 5479,N1(C(C2CCCCNC(=O)CC2)C)CCC(C2CCC2)CC1 5480,N1(C(COCC)=O)CCC(CNC(=O)C[SH]=CCOC(C)=O)C(F)(F)C1 5481,C(=O)(C(F)(F)c1ccncc1)N(CC(C)NC(=O)CC1CCC2CC12)C 5482,c1(OCC)ccc(S(=O)(=O)N2CCCC(CNC(c3ccc[n+]([O-])c3)=O)C2)cc1 5483,C(=O)(C(Cl)=CCl)NCCN(C(C)C)C(c1cn(C2CCCCC2)nn1)=O 5484,C1(CNC(CC(=C)C)=O)(CO)CC12CCN(C(=O)COCP(C)(C)=O)CC2 5485,c1(C(=O)NCC2(NC(CCCNC(CC(C)(C)C)=O)=O)CC2)ccc(F)cc1Br 5486,c1(C(=O)NC(C(N2C(CCC#C)CCC2)=O)c2cccs2)ncccc1Cl 5487,N1(CC(C)NC(C2CCN(S(C)(=O)=O)CC2)C)CCc2ccccc21 5488,N(C(=NCC1CC1)N1CCC2(C1)CC(F)(F)C2)Cc1cc2c(cc1)C(=O)CCC2 5489,c1(NCC2C3(C(=O)OC)CCC3C2)c(OC)ccc(C)c1OC 5490,c1(C(N2CCCN(C(C(CC)(C)O)=O)CC2C)=O)cc2ccccc2n1C 5491,c1(C(=O)NCC(CC(=O)NCC2CN(C)CCO2)OC)cc([N+](=O)[O-])c[nH]1 5492,C1(CNC(CCOCC)=O)CCCCC1C(=O)NCCCCOC 5493,c1(C(=O)NC2CC(CNC(=O)CSc3ccccc3)C2)cncc2nc[nH]c12 5494,N1(C(CC(=O)NC(C)C)=O)CC(C(=O)O)OC(C)C1 5495,N1(C(c2cnn(CC3CC3)c2)=O)CC2CCC1CN2C(C12CC3CC1C2C3O)=O 5496,C(=O)(C1=NOC(C)(C)C1)NCC(CNC(c1cc(CC)[nH]n1)=O)OC 5497,CCC(C)C(O)CC(=O)N(CCC(=O)NCC1CC(=O)N(C)C1=O)C(C)C 5498,N1(C(C=C(C)C(F)F)=O)CC2CCC1C(NC(=O)CC1CC3CCC(C1)N3C)C2 5499,C=CC(C)(C)CCC(=O)N1CC(C)CC1C(=O)NCCC(C)(C)COC 5500,CC1CCN(C(=O)CCOCc2ccccc2)CCN1C(=O)Cc1sccc1Cl 5501,C1(C(C)C)CCC(C)CC1OCC(=O)NC1CC(N(C(=O)CN=S(C)(C)=O)C)C1 5502,C1(CNC(=O)C=Cc2ncc[nH]2)CN(C(C2(C3CCC3)CC2)=O)CCC12CCC2 5503,c1(C(N2CCC(c3cccc(Cl)c3)C2)C(=O)NCCCF)cc(Cl)c(Cl)cc1O 5504,N(C1CCS(=O)(=O)c2ccc(Cl)cc21)C(CNC(CCCCC)=O)=O 5505,CC1CCCC(CC(=O)NCCOC2CCN(C(c3cnc(N)cn3)=O)C2)C1 5506,C1(N(C(Cc2c(CC)noc2CC)=O)C)CN(C(c2cnsc2)=O)CCC1C 5507,C(CN=C(NCc1cccn1C)N(C)CC(C)C)c1cccc(CC)c1 5508,N1(C(C2CCCC(NC(c3cnnc(O)c3)=O)CC2)=O)Cc2cccc(O)c2C1 5509,c1(C(=O)NCCCN(C(=O)Cc2cc(C)ccc2F)CC)ccc(N)cc1F 5510,C1(NC(CC)Cc2ccccc2)CCNC(C(=O)OC)C1 5511,N1(C(C(CCC)NC(=O)CCc2ccsc2)=O)CC2CC3CC2C1C3O 5512,N1(C(=O)CC2CN(C(c3cccc(C(F)F)c3)=O)C2)CCC2(CCOC2)C1 5513,Cc1cc(C2CC2)ncc1C(=O)NC1CC(CCNC(C2(C)CCCN2C)=O)C1 5514,N1(C(Cc2nc(C)oc2)=O)CC2CCC1C(CNC(=O)CCCCF)C2 5515,c1(C(N2CC(CC(CNC(CC3ON=C(C)C3)=O)(C)C)C2)=O)cc(C)nc(O)n1 5516,c1(C(N(CC(=O)NCC2CC23CC3)CC#C)=O)cccn1CCC 5517,C(=O)(C(C)(C)C(F)(F)CC)N1CC(CNC(CSCC)=O)C2(C1)CC2 5518,C1(CCNC(COCCCOC)=O)CC2CCC(C1)N2C(=O)C(F)(F)C(C)O 5519,C1(N(C(C2C(C(=O)OCC)C2)=O)C)CN(C(c2cc[nH]n2)=O)CC12CC2 5520,CC1CN(C(c2csc(Cl)n2)=O)CCC1NCc1cnc(C(N)=O)s1 5521,N1(CC)CCN(CC(N2CCC3C(NC(=O)C(C)C4CCC4)C23)=O)CC1 5522,C1(C(=O)NCC2(COC)CN(c3nc(C(C)C)cc(C)n3)C2)Cc2ccncc2C1 5523,c1(C(=O)NCCOCCOCCNC(C2C(=C)CC2)=O)ccoc1C(F)(F)F 5524,C=C1CC(C(N2CC(C)(OCC(=O)OC)C2)=O)(CNC(CO)C(C)O)C1 5525,C1(NC(c2cc(OCC)n[nH]2)=O)C2CC1N(C(C1(C(F)(F)F)CC(F)C1)=O)C2 5526,C1(NC(c2c(OC)cc(O)nc2)=O)C(C)(C)C(NC(=O)C(C)OCOC)C1(C)C 5527,c1(C(=O)NCCCCNC(CSCC=C)=O)ccc2cnc(C)n2c1 5528,CCC(C)(O)C(=O)N1CC(CNC(=O)C(O)Cc2cnn(C)c2)C(O)C1 5529,c1(OCC)ccc(Cl)nc1C(=O)NCC1CC1NC(=O)CCc1cccnc1C 5530,c1(C(C)C(N2CC(O)(C(C)(C)CNC(C3CCSCC3)=O)C2)=O)cncc(O)c1 5531,C(=O)(C1CCc2c(F)cccc21)NC(c1ccc(OC)cc1Br)C 5532,c1(CNC(C(C)C2CCC2)=O)ccnc(CNC(=O)C=CC(F)(F)F)c1 5533,C1(CNC(c2ccc(CCCCCCC)cc2)=O)CCN(C(C)=O)CC1(F)F 5534,c1(C(N(C(CCNC(Cc2ccn(C(C)C)n2)=O)C)C)=O)cnc2[nH]nnc2c1 5535,N1(C(C(CC)OC)=O)CC2CCCC(CNC(=O)CCCN(C)C(C)C)(C2)C1 5536,C=CCCC(F)(F)C(=O)NCC1CN(C(=O)CN2CCC(C)(C)C2)CCC1C 5537,C1(NC(Cc2cccc(CC)c2)=O)CC2CC1N(C(C1CC(=O)N(C)C1)=O)C2 5538,N1(C(Cn2ncc(C#C)c2)=O)CCC2CN(C(=O)CC3CC(F)(F)C3(F)F)CCC12 5539,c1(C(=O)NCC2N(C(CCCC#C)=O)CCC(C)C2)cc(OC)c2c(c1)CC(C)O2 5540,c1(CC)ccoc1C(=O)NC1CCCC1CNC(=O)CC(=O)NC1CC1 5541,Cc1ccc(C(=O)NCC(=O)NCC2(O)CCCC2)cc1.C12C3CN(CC13)C2=O 5542,N1(C(c2c(C)cns2)=O)CCN(C(=O)C#CC(C)(C)C)CC(O)C1 5543,N1(c2cc(OCC)nc(C)n2)Cc2[nH][nH]c(=NC(=O)c3cnn(C)c3)c2C1 5544,C1(C(F)(F)F)(OC(=O)NCC)CCN(C(C23CCCC2CC3)=O)CC1 5545,CC1CCC(C)CN1C(=O)C(=O)NC(c1ccccc1F)c1nnc(CO)s1 5546,C(=O)(CC(CN(C)C)C(F)F)N1CC(O)(CCNC(C=C(C)C2CC2)=O)C1 5547,C1C(CC(C)C)C(=O)N1.C(CC)(CC=O)NC(C=CC(CC)C)=O.OC 5548,N1(C(c2cccnc2O)=O)CC2CC(C1)N2C(=O)CC(O)c1ccccc1 5549,c1(C(=O)NC2CC(C)(C)N(C(c3coc(O)n3)=O)C2)cccc2cnsc12 5550,C(CC(F)F)(C(=O)N1CC(O)(C(F)(F)F)C1)NC(C1C(=C)C1)=O 5551,c1(C(=O)NCC2N(C(C(CC)=CC)=O)CC2)cc2c(cc1N)OCO2 5552,Cc1cccc(C(N2CC=CC2CNC(=O)CC2(c3ccccc3)CC2)=O)n1 5553,n1(CCC)ncc(C(=O)NCC2CN(C(c3sc(C)nc3OC)=O)C3CC23)c1C 5554,c1(CC(N2CC(C)C(C)(CNC(C3(F)CC3)=O)C2)=O)c[nH]c2ccccc12 5555,N1(C(C2N(C(c3coc(C(F)F)c3)=O)CCN(C)C2)=O)CCC12CC(C)(CO)C2 5556,N1(C(C=C(CC)C)=O)CCCC2CN(C(=O)CCS(=O)(=O)NC)CCC12 5557,CC(C(=O)N1CC(C2CC2)C1)C(=O)c1ccccc1F 5558,N1(C(CC(CC)O)=O)CCCCC(C2CN(C(c3cc(C)ccc3F)=O)C2)C1 5559,N1(C(CC(CC)SC)=O)CCC2(C=C(C(=O)N3CCCOC(C)C3)C2)C1 5560,c1(OC)nc(N2CCC(Cc3ccc(F)c(C(F)(F)F)c3)CC2)nc(C)c1F 5561,N1(C(c2cc(C)ns2)=O)CC(C)CN(C(=O)CSCc2c(C)noc2C)C(C)C1 5562,Cc1cc(NC(C2C=CCCC2)=O)ccc1NC(c1cn(CCN(C)C)nn1)=O 5563,C1(NC(CC(CN(C)C)O)=O)CN(C(C2(N(C)C)CCOCC2)=O)CCC12CCC2 5564,C(CC(=O)NC1CCOC1(C)C)(CC(C)C)NC(C(CC)(C)C#N)=O 5565,C12(CNC(C(CC)=CC)=O)CC1CN(C(c1csc(CC3CC3)n1)=O)C2 5566,c12ccc(c(OC)c1)NCC(C)=CC2=O.C1(SCC(=O)OC)OCCCO1 5567,c1(C(N2CC3(CCC3)C2c2ccncc2)=O)nn2c(c1I)CCC2 5568,C1(OC)(OC)CCC(C2(NC(=O)CC(C)(O)COC)CCOCC2)C1 5569,C(N=c1[nH]c(N2CC(=O)NC(=O)C2)nc2c1CCC2)c1c(C)scn1 5570,C(=O)(C1CCCc2nccn21)NC(CCCC)CNC(c1cc(C)oc1C)=O 5571,c1(CN(c2ccccn2)C(C2(O)CC(OC)C2)=O)c(C)c(Br)c(C)c(C)c1Br 5572,C(=O)(C(C)CN(C)C(=O)C1CC1)N(C(CSC)C)C 5573,CC1CC2(CCO1)CC2C(=O)NCC1CCN(C(c2c[nH]ccc2=O)=O)CC1C 5574,N1(C(C)(C)C)CCC(F)(C2CCCN2CC(=O)NC2C3CC4C(C3)C24)C1 5575,O=C1CCCC(c2ccccc2)(CNCCCF)N1 5576,N1(C(=O)C=Cc2ccncc2)CC2(CCN(C(C3CCC4CCC3O4)=O)CC2)C1 5577,C1C(O)C(=O)N1.N1(C(C2C(C(C)(F)F)C2)=O)CC(CO)C1.C(N)=O 5578,C12(CNC(C3C(C)C3)=O)CCCC1N(C(C1CCC1(C)C)=O)CCC2 5579,c1(C(N2CCCN(C(C3CCN(C(C)=O)C3)=O)CC2)=O)ccc(Cl)c(N)c1Cl 5580,C1(C(=O)NCC2=CCN(C(Cc3c(C)ccs3)=O)CC2)CC2C=CC1CCC2 5581,C1(C(N2C(C(C)NC(=O)CC3CCCCN3C)CCC2)=O)CC2OC(=O)OC2C1 5582,C(=O)(C(=O)CC(C)C)NCC1(CCNC(Cc2cn(CC)nc2)=O)CC1 5583,c1(C(N2CC(NC(C(CC=C)C)=O)C(C)C2)=O)cncc(Cl)c1C 5584,C1(N(C(C=CCCC)=O)C)CCCC(NC(=O)CCn2ccnc2)C1 5585,c1(C(N(C(C)(C)CC(=O)NC2CCCC(O)C2)C)=O)ccnc(CO)c1 5586,c1(SCC2CN(C(=O)C=Cc3cccs3)CCO2)ccc2c(C3=CCOC3)cnn2c1 5587,Cc1nc2nc(=S)[nH]n2c(C)c1CC(=O)NC(C)C(C)NC(=O)C(F)F 5588,C12(C(=O)NCCCOC)CCC(NCc3cc(O)cc(Cl)c3)(CC1)CC2 5589,N1(C(Cc2cc(C)no2)=O)CCC(NC(c2cc(Cl)no2)=O)C(O)C1 5590,c1(C(C)=O)ccc(N2CCOC(C(C)NC(c3scnc3Cl)=O)C2)nc1 5591,c1(C(=O)Nc2cccc(C(=O)NC(CC)C)c2)cnc(F)c(C)c1 5592,C(=O)(C1=C(Cl)CCC1)NC1CC(F)(CNC(c2c(C(N)=O)nccc2)=O)C1 5593,Cn1nnnc1SCCOCC1(F)CC(NC(c2ccnn2CCC(F)(F)F)=O)C1 5594,CC(CC(N)=O)C(=O)N1CCCC(N2CCN(C(c3c[nH]ccc3=N)=O)CC2)C1 5595,N1(C(c2ccc(OCC)cc2)=O)CC2(CCC2NC(c2ccc(CO)s2)=O)C1 5596,C1(NC(C=C(C)C(C)(C)C)=O)CC(C)CN(C(c2cnn(CC3CC3)c2)=O)C1 5597,N1(C(C(C)C2CCC2)=O)CCOCC(NC(c2occc2-c2cnn(C)c2)=O)C1 5598,C1(CNC(CC=CC=C)=O)C(CC)CCN1C(=O)C(F)C(C)C 5599,C1(F)(CNC(COCc2n(C)ncc2)=O)CCC(CNC(c2ccsn2)=O)CC1 5600,C(C(=O)NCC1CCCC1NC(=O)CCN(c1ccccc1)C)(C(C)(C)C)OC 5601,C1(NC(c2c(C)onc2CO)=O)CCN(C(c2ccc(N)c(Cl)c2)=O)CC1F 5602,Cc1c(C(=O)NC(C(N2CC[Si](C)(C)C2)=O)C2CCCC2)ccn1C 5603,C(=O)(C1=CC2(CCN(C(=O)CCc3nccn3C)C2)C1)N(CC(=O)NC)C 5604,N1(C(c2c(C)ncn2C)=O)CC(NC(c2ccnn(C)c2=O)=O)CC(O)C1 5605,CC1(C)CC(O)(CC(=O)NCC(F)(C2CCOC2)NC(C23CC(C)(CO2)C3)=O)CO1 5606,CNS(=O)(=O)N1CCC(C(=O)N(CCCN(C(=O)CCNC(=O)CO)C)C)CC1 5607,C1(C)(CC)CC(NC(=O)CCN(C)C(C)=O)CN1C(=O)CCCC 5608,c1(C(=O)NCCNC(C2C(C(N(C)C)=O)CCC2)=O)ncnn2c(Br)ccc12 5609,c1(OC)ccc(OC)c(C(=O)NCC(C)NC(C2(C)CC(C)=NO2)=O)c1N 5610,c1(-c2scc(C(CC)C(=O)OCC(C3CCCCC3)=O)n2)ccc(S(C)(=O)=O)nc1 5611,c1(C(N2CC(C(=O)NCC3OCCN(C)C3)OCC2)=O)cccc2ccoc12 5612,n1(CC(=O)NC(C(C)NC(C2(CCC=C)CC2)=O)C)ccc(=O)cc1C 5613,CC(C)CC(C)CC(=O)NC1CCN(C(=O)C2=CS(=O)CCC2)CC1O 5614,c1(SCC(=O)NC2CC(NC(C3NC(=O)OCC3)=O)C2)cc2ccccc2[nH]1 5615,C(=O)(C#CC(C)(C)CNC(=O)C=Cc1ccc[nH]1)NC(C1CCCO1)C 5616,c1(SCC=C)ccccc1C(N1CC(NC(=O)C(c2cccnc2)O)C(C)C1)=O 5617,C1(C(N2C(CNC(c3c(C)cnnc3O)=O)CC2)=O)Cn2c(C)nnc2CN1C 5618,C1(CN(C(C=CCCC)=O)CC)CCN(C(=O)CCC2CCOCC2)C(C)C1 5619,c1(CC)cnc(C(=O)N(CCCOC)CCNC(=O)CC2C(OC)CC2O)nc1 5620,Cc1ccc(NC(c2cc(NC(=O)Cc3ccc(Br)cc3Br)cn2C)=O)c(I)n1 5621,c1(C(N2CC(O)(C(=O)NCCCCCC(=O)OC)C2)=O)nccc2[nH]ccc12 5622,N1(C(c2cc(C(F)(F)F)cc(Cl)c2)C(=O)NCC#N)CCc2c(Br)cccc2C1 5623,C12(NC(=O)Cc3ccns3)CCC1CN(C(C1CCCOC1)=O)C2 5624,CC#CCCCC(=O)NC1CC(CNC(C2CCCCO2)=O)C1 5625,C(N=c1[nH]c(N2CCC(C(C)C)C2)nc2c1CCCCC2)C1(OC)CC1 5626,C(c1ccc(F)c(F)c1)=CC=CC(N1CCC(C)(NC(Cc2c(C)non2)=O)C1)=O 5627,C1(NC(c2c(CC(C)C)n(C)nc2)=O)CC2CC(C1)N(C1CCC(=O)NC1=O)C2 5628,c1(C(N(CCC)C)=O)cc(SCC(N2CCOCC2CC)=O)ccc1Cl 5629,c1(C(=O)NC(CC)CNC(C2CCC2c2nc[nH]n2)=O)nc2cccnc2s1 5630,c1(C(=O)NC(C)C(c2cccs2)NC(=O)C(F)OC(F)(F)F)cnccc1Cl 5631,N1(CCC(=O)NCCC(O)CNC(c2cnc(C(F)F)s2)=O)CCOC1=O 5632,c1(C(N2CCC(C)(CCO)C2)C(=O)NCCCSC)cc2cc(Cl)cnc2o1 5633,N1(CCOC(CCCCCC)(C)C)CCCc2cc(OC)ccc21 5634,CCN=c1[nH]c(C(N2CCCC2CSCCNC(=O)COC)=O)cs1 5635,c1(COC)ccc(NC(=O)CC2CCCN2C(=O)CNC=O)cc1C(=O)OC 5636,C(=O)(C(C)CC(C)C)N(CCCCNC(=O)C(F)(F)CNC(=O)OC(C)(C)C)CC 5637,c1(C(N(C(CCNC(Cc2cccc(C)c2F)=O)C)C)=O)cc2c(o1)CCCC2 5638,C(=O)(C(Cc1cnc[nH]1)NC(=O)CC1CC1)N(C(CC)C1CC1)C 5639,C1(C(=O)NC2CCN(Cc3nc(-c4ccccc4)no3)C2)CC2CCC1O2 5640,C(=O)(C(C)(O)CNC(=O)CCC1CCCN1C(=O)CCc1cnco1)OC 5641,c1(C(N2CC(O)(CCNC(CNC(C)=O)=O)C2)=O)cncc(N2CCCC2)n1 5642,c1(C(N(CCOC)CCNC(C2CCC(C)CC2)=O)=O)ncc2ccccn12 5643,C(=O)(C(C)(CC)C(=O)NCc1ccc(CCNC(C2CCSC2)=O)cc1)OCC 5644,c1(C(C(=O)NCC2CC(C(=O)OC)C2)N(C2CCSC2)C)cccc2sccc12 5645,c1(OC(C(=O)N2CC(n3cc(N(C)CC)nn3)C2)(C)C)ccc(Cl)cc1 5646,C1(C#N)(C(=O)NCC(C)CNC(=O)CC2(C)CCCC2)CCCC1 5647,N1(CC(=O)NCC2CCCN2C(=O)C=CC(=O)NC2CC2)CCOCC1 5648,N1(C(C2(CC=C)CCCN2C(c2ccc(SC)o2)=O)=O)CC(=O)N(C)CC1C 5649,C(CCN=C(NC(c1cccc(C)c1)C)NC1CC1C1CCOCC1)OCC 5650,N1(C(CC(C)c2cnn(C)c2)=O)C2CCC1C(CNC(c1ccon1)=O)C2 5651,N1(C(C(C2CCOC2)OC)=O)CC=C(C(=O)NC2COCCC2O)C1 5652,c1(C(=O)NC2C3CC2N(C(=O)COC2CCCCC2)C3)ccc2c(n1)CCC2=O 5653,N1(C(C(=O)NCCC(C)NC(C2CN(S(C)(=O)=O)C2)=O)C)CCNC1=O 5654,n1(CC)ncn(NC(=O)C(Cn2ccnn2)NC(=O)Cc2cccnc2F)c1=O 5655,N1(C(C2N(Cc3c(C(N4CCCC4)=O)cn(C)n3)CCC2O)=O)C2CCC1C(N)C2 5656,C1(C(N(CCC(=O)Nc2cncc(CC)c2)C)=O)CC2(C1)CC21CC1 5657,C1(O)(CNC(C2CC(SC)C2)=O)CCN(C(c2scnc2Cl)=O)CC1 5658,C1(O)(CC(=O)NCCS(C)(=O)=O)CCN(C(c2ccc(C#N)cc2)=O)CC1 5659,c1(CCC)sc(NC(c2cscc2C)=O)cc1CC 5660,c1(C(=O)NCCC2(NC(c3cc(C(C)C)no3)=O)CCCC2)cc(N)cc(F)c1 5661,C(=O)(C(C)(O)C(F)(F)F)NCC(CCNC(c1c(F)ccc(CC)c1)=O)OC 5662,C(=O)(CC(O)C(C)C)NCCC1(C(N2CC3C(C(C)=O)C3C2)=O)CCC1 5663,CC1(C(=O)NCC2(CNC(=O)CCF)CCC2)COC(=O)OC1 5664,c1(C(=O)NCC2(F)CCN(C(C(CCC#C)O)=O)C2)ccc([N+](=O)[O-])cc1Cl 5665,C(CC)(c1ccccc1)=CC(N1CCN(C(COC(CC)C)=O)CC1C(F)F)=O 5666,c1(C(N2C(C(N(CC(C3CCC3)OC)C)=O)CC(O)C2)=O)cc2cccnn2c1 5667,Cc1nccc(=NCC2CCN(C(C3(C)CC=CCC3)=O)C2)[nH]1 5668,C1(C(=O)NCC(CCOC)OC)(NC(=O)CC(C)(C)C)CCCCC1 5669,Cc1cc(CNC(c2ncc(F)cc2Cl)c2nnnn2C2CC2)c(C)nn1 5670,N1(C(c2c(COC)noc2)=O)CC2CC(C1)CN(C(=O)C(C)(C)C1CCC1)C2 5671,c1(C(=O)NC(c2cnc(C)s2)C)cc(S(=O)(=O)CC2CC2)ccc1F 5672,c1(OC)ccc(CN2CCN(Cc3cc(Br)cs3)C3CC23)c(C)c1C 5673,CC(C)(C)CC(C(F)(F)F)N1CCCCC1CCNC(=O)OC(C)(C)C 5674,c1(NC(C2CC(NCc3ccnc(O)c3)C2)=O)ccc(Cl)cc1F 5675,Cn1cc(S(N)(=O)=O)c(C(=O)N(CCCNC(C2(C)CC2F)=O)CCO)n1 5676,C#Cc1ccc(C(=O)OC(CCC)C(=O)N(C)C)nc1 5677,c1(C(=O)NC2C(NC(c3ccn(CC)c3C)=O)CCCC2)c(N)cccc1Cl 5678,C(=O)(CCCCC(C)CC)NCCC(=C)CNC(c1cscc1Cl)=O 5679,CCCC(C)(CC)C(=O)NC1CCCC(NC(c2ccc(O)c(C)c2C)=O)C1 5680,N1(C(c2cnc(CCC)s2)=O)CCN(C(c2ccn(CC)c(=O)c2)=O)CC1CO 5681,N1(C(C(C(C(C)C)O)C)=O)CCC2(CC1)CN(C(=O)Cc1cnc(C3CC3)[nH]1)C2 5682,C1(NC(=O)CCc2ccncc2)CCCCC1NC(=O)Cn1cc(Br)cn1 5683,C(=O)(C1CCc2ccccc21)N1C(CN(C)C(C2CC(N=[N+]=[N-])C2)=O)CCCC1 5684,CCCCC(CC)CC(=O)N1CC2CC1CN(C(c1cn(CC)nn1)=O)C2 5685,CC(C(=O)NC1CC(NC(=O)COCc2nnc(S)n2C)CC1O)C(F)F 5686,CCC(CCO)NC(C1CC(CCNC(=O)C=Cc2cc[nH]c2)C1)=O 5687,C12(CNC(C(=O)NC(C)Cc3ccnn3C)=O)CCC(CC1)CN2 5688,CCCCC(CN=c1nc(CC)cc(C)[nH]1)NC(c1n[nH]c2c1CCSC2)=O 5689,N1(C(c2c(CC)nc[nH]2)=O)CC(NC(c2cnns2)=O)C2(CCC2)C1 5690,C1(CC=C)(C(=O)NCC(F)C2CCC2)CCN(C(=O)C(C)(C)C=C)C1 5691,C1(CC(CC(N)=O)N2CCOCC2)CNC(=O)N1C.CCCCSC.OC 5692,c1(OC)cccc(Br)c1C(N1CCC(NC(=O)CC(C)(C)CN(C)C)C(C)C1)=O 5693,Cc1cc2ccc(Cl)cc2c(N2CCOC(c3n[nH]c(-c4ccccc4)n3)C2)n1 5694,N1(C(C2CC(OC)C2)=O)CCN(C(=O)C=C2CCN(C)C2)C2CCCC2(C)C1 5695,Cn1cc(C(N2CC3CC3(NC(=O)CC3CCC3)C2)=O)c(=O)c2cnn(C)c12 5696,Cc1nc(C(F)(F)F)ccc1C(=O)NCC1(NC(=O)Cc2cnc[nH]2)CC1 5697,C(c1cc(F)c(F)c(F)c1)=CC(N1CCCN(C(C2(COC)CC2)=O)CC1C)=O 5698,CCC(C(=O)N(C)CC1(O)CN(C(C2CC(=O)N2)=O)C1)C1CCOCC1 5699,c1(NC2(CO)CCN(C(C3(C(C)C)CC3)=O)CC2)ccc([N+](=O)[O-])c(C#N)c1 5700,c1(OC)ccc2cc1NC2.N12CC3CC1C3NC2=O.C1(NC(C)(C)C)CCCC1 5701,c1(OC)ccc(F)cc1-c1nc(Cc2cccs2)nn1C1CCCC1O 5702,c1(C(N(C2CCN(C(=O)C=CC3CCC3)C2)C)=O)cccc2c1CCCC2 5703,c1(C(=O)NC(C(C)C)CCNC(C2(O)CCOC2)=O)ccc(C#N)c(Cl)c1 5704,N1(C(c2c(C(C)C)scn2)=O)CCC(C)(C)C(NC(=O)CC2C=CCCC2)C1 5705,CC1(C)Oc2ccc(C(N3CCC4C(CCN4C(=O)C(O)C(F)F)C3)=O)cc2O1 5706,N1(C(c2c(C)oc(Br)c2)=O)CC(NC(c2ccnn2C)=O)CC(C)C1 5707,N1(C(CC(=O)OC)=O)CCN(C(=O)Cc2cc(F)cc(F)c2)CC1CO 5708,c1(CNC(CC2CC(NC(=O)C=CC(N3CCOCC3)=O)C2)=O)cncc(O)c1 5709,C(CC(C)C(=O)NCCC1CCCN(C(c2sccc2C)=O)C1)=CC 5710,C1(N(C(C2CN(C(C)=O)C2)=O)C)CN(C(C2(c3ccccc3)CCC2)=O)CC1C 5711,C(CNC(=O)CCCN(C)C(C)C)(C(C)C(C)C)NC(c1c(C)oc(C(C)C)c1)=O 5712,c1(C(=O)NC2C(C)CCN(C(CCOCCCOC)=O)C2)cccn2nccc12 5713,Cc1ncsc1C=CC(=O)NC1CC(O)(CNC(C2CNC(=O)N2)=O)C1 5714,Cc1ccc(Br)c(N)c1C(=O)NCC1(C)CCCN1C(=O)CC(C)C(C)C 5715,c1(C(=O)NCC2N(C(Cn3nnc(=N)[nH]3)=O)CC=C2)cc(Cl)nnc1Cl 5716,c1(CN(C(C2COCC(C)O2)=O)CC)cccc(CNC(c2[nH]nnc2C)=O)c1 5717,C(=O)(CC(C)C(=O)N1CCC(C)C(NC(C2CCCCS2)=O)C1)OC 5718,Cn1cc(C(N2CCC2CNC(C2(C)CCCCO2)=O)=O)c2ccncc12.CC1(C)CC1 5719,C(CCCS(=O)(=O)CCO)NC(=O)NCCc1ccc(-n2c(C)cc(C)n2)cc1 5720,C(=O)(C(C)(C)CC(C)C)NC(COC)CC(=O)N(C)CCC1CCCCC1 5721,C1(NC(C2CCOC2)=O)CN(C(c2ccc(C(F)(F)F)cn2)=O)C2(CCC2)C1 5722,N1(C(Cc2c(COC)cccc2)=O)CC(NC(C2CCOCC2)=O)CC12CCC2 5723,C1(O)(C(=O)NCCCCNC(CCNC(C)=O)=O)CC1(C)C 5724,N1(C(C2CCC(CC)O2)=O)CC2(C)CN(C(c3cnco3)=O)CC2(C)C1 5725,c1(C(N(CC(C)C)CCc2nc(C)sc2)=O)cc([N+](=O)[O-])c(F)c(F)c1Br 5726,c1(C(N2CCN(C(=O)CCc3cncs3)C3CCCC23)=O)n[nH]c2ccccc12 5727,N1(C(CCCC#CC)=O)CC2CC(F)(F)CCC2(NC(=O)CSCC)C1 5728,S(=O)(=O)(c1cnn(C)c1)N.CC(CCNC(=O)C(C)N(C)C)NC(C1CN(C(N)=O)C1)=O 5729,c1(CC)cccc(C(=O)N(CC(=O)NCc2nnn(C)n2)CC2CC2)c1 5730,C(c1cccc(OC(F)F)c1)=CC(=O)NC1(C)CC(NC(C2CCC(=O)N2)=O)C1 5731,C(c1ccn(C)c1)=CC(=O)NC1(CCNC(C(C)OCCCC)=O)CCC1 5732,N1(C(C2(C)N(C(C3OCCC(C)C3)=O)CC=C2)=O)CC(F)CC(F)C1 5733,c1(OC)cc(N)c(Cl)cc1C(N1CCC(C)(NC(=O)C2=CCC(C)CC2)C1)=O 5734,c1(C(=O)NC2(CN(C(CSCCCC)=O)C)CC2)cccc(OC)c1 5735,C(C(=O)NCC1CCCCC1CNC(C1CCC(=O)NC1)=O)(C(C)C)OC 5736,C1(CNC(COCCOCCOC)=O)CCCCCCN1C(c1ccc[nH]1)=O 5737,c1(C(=O)OCC)ccc(Cl)cc1COC(=O)C(F)CC1(c2cc(C)ccn2)CC1 5738,C1(O)(C(C(=O)NCC(CC=C)NC(=O)C(C)(CO)OC)(F)F)CCCCC1 5739,N1(C(c2nc(CCCC)sc2)=O)CCCN(C(c2cc(C)ncn2)=O)CCC1 5740,c1(NCC(=O)N(C2CC2)Cc2cn(C3(C)CCCC3)nn2)cnn2c1CCCC2 5741,N1(C(CCC)=O)CCN(C(=O)C(F)COC=CC(=O)OC)C(c2ccnn2C)C1 5742,CCC(C(=O)N1CCOCC1c1cn(-c2ccncc2)nn1)C(=O)O 5743,Cc1ccc(C(C)(C)CC(=O)Nc2nc(C(C)(F)F)cs2)c(C)c1 5744,c1(CC)noc2ncc(C(=O)N(CCN(c3nnc(C)s3)C)CC)cc12 5745,c1(CNCc2cc(C)nc(O)c2)c[nH]c2cc(Br)ccc12 5746,N1(C(CCN(C(c2ccnc(C)c2N)=O)C(C)C)=O)CCCN2CCCC2C1 5747,CC(CCCCCO)NC(C1CCCC1CNC(=O)Cc1cn[nH]c1)=O 5748,C(C(COC)CC(=O)N1CC(CCNC(C2(Br)CC2(C)C)=O)C1)OC 5749,C(=O)(CC(CCC)NC(=O)C=Cc1ccncn1)NCC(=C)Br 5750,N1(C(=O)Cc2ccc(OC(F)F)cc2)CC2CN(C(c3ccsc3Cl)=O)CC2C1 5751,C#Cc1ccc(Br)c(C(=O)NC2CCCC2CNC(c2cscn2)=O)c1 5752,C1(NC(C(F)=C(C)C)=O)CC2CC1CN(C(=O)C(c1c(C)noc1C)(C)C)C2 5753,c1(N(C2(CC#C)CCOCC2)C(c2ccc(Cl)cc2F)=O)ncnc2[nH]ccc12 5754,Cc1cc([N+](=O)[O-])cc(C(=O)NC2CC3CN(C(=O)CCCCC#N)CC3C2)n1 5755,c1(NC(=O)C(=O)NC2CC(CCc3ccco3)C2)ccccc1 5756,N1(C(c2cc(OC)c(F)cc2)=O)CC2CCC(C1)N2C(c1c[nH]nc1Br)=O 5757,C1(C2CCCCC2)(C(=O)NCC2CC(NC(C3(C#N)CCOC3)=O)C2)CC1 5758,C1(NC(C=CCOC)=O)CCN(C(C2CCC(=O)N2C(C)C)=O)CC1O 5759,N1(C(CCN(C(=O)CC2CCCC2)CCC)=O)CCOC(CN(C)C)C1 5760,c1(OC(C)C#N)ccc(C(=O)NCC2CC2NC(c2cc(CO)ccn2)=O)cc1 5761,c1(C(N(C(C)C)CCNC(C2CC3C=CC2O3)=O)=O)ccc2occc2c1 5762,C(=O)(C(CC)CC(C)C)N1CC(C2CC2)(C(N2C(COC)COCC2)=O)C1 5763,c1(C(=O)NC2CC3CN(C(C(C=C=C)C)=O)C(C2)C3)n[nH]c2c(C)cccc12 5764,N1(C(c2c(C)scn2)=O)CC2OCC(NC(C3CC4(C3)CC(C)C4)=O)C2C1 5765,c1(NC)cnc(C(=O)NCC(C2CCCN2C(C2CCN(C)C2)=O)(C)C)cn1 5766,N1(C(c2c(CNC(c3c(C#N)scc3)=O)noc2)=O)CCOCC(F)(F)C1 5767,CCCCCCC(C)C(=O)NCC12CCC(C1)N(C(=O)CN1C(=O)CNC1=O)C2 5768,C1(C(N(C2CCN(C(=O)C(C)(C)OC)CC2)CC#C)=O)C2CC2C2CC12 5769,N1(C(C2CCC(C)(C)N(C(=O)COCCCF)C2)=O)CCC12CCC(C)CC2 5770,C(CC(=O)N1CCN(C2CC2)CC1)(C(F)(F)F)NC(c1cccc(C)n1)=O 5771,C(C)(C1=CCN(C)CC1)NC(C1C(CC)OCCC1)=O 5772,C12(NC(c3cc(CC(C)C)[nH]n3)=O)CCCN(C(=O)C#CC3CCCO3)CC1C2 5773,N1(c2c(S(=O)(=O)NCCCCOC)cncc2)CCc2c(F)cc(F)c(F)c2C1 5774,c1(C(=O)NCC2(O)CCN(C(COC(CC)(C)C)=O)C2)ccc2c(c1)CC2 5775,c1(C(=O)NCc2cc(Cl)ccc2Br)nn2c(c1C1=CCCCC1)CCCC2 5776,CCCC(C)(C)C(=O)NC1CC(CCNC(=O)COCCOCCO)C1 5777,CCC(C)(F)C(=O)N(C)CCN(C)C(C1(N2CCCCC2)CCCCC1)=O 5778,C1(NC(CS(CC)=O)=O)CCCC2CN(C(c3ccc(N)c(Cl)c3)=O)CC12 5779,c1(OC)ccc2c(c1)NC(=O)C2CC(=O)N1CCOCC1CNC(C1CC1C)=O 5780,S(=O)(=O)(c1ccc(NC(c2cc(C)ccc2F)CO)nc1)N1CCC=C(C)C1 5781,C12(NC(c3c(C)ocn3)=O)CC1CN(C(=O)Cn1nc(C(F)F)cc1C(F)F)C2 5782,c1(C(N2CCC(OCc3onc(C)n3)C2)=O)cccc(F)c1C 5783,Cc1cc(C(=O)NC(CNC(c2cnsn2)=O)CC(C)C)cnc1C(F)(F)F 5784,c1(C(=O)NC(CCCC)CNC(=O)C(C)(O)CCC)cc(S(N)(=O)=O)c[nH]1 5785,N1(C(C2N(C(C)=O)CSC2)=O)CC2CN(Cc3ccc(Cl)cc3C(F)(F)F)C2C1 5786,c1(C(=O)NCC(CNC(C(COC)NC(C)=O)=O)O)sc(C(C)(C)C)nc1C 5787,CC(C)CS(=O)(=O)CC(=O)NC1CC2CC(NC(c3coc(C(F)F)c3)=O)C2C1 5788,C(CS(=O)(=O)C1=NOC(C)(C)C1)N(C)Cc1ccc(CC2CC(=O)NC2=O)cc1 5789,OCCC(N=c1[nH]c(=NCc2snnc2)[nH]c2c1CCCC2)C1CC1 5790,c1(C(=O)NCC(C2CC2)NC(C(C)OCC)=O)ccc(C(F)(F)F)cc1Cl 5791,C1(CN(C(=O)COC(C)(C)CNC(C2CCCCC2O)=O)C)CCCC2CC12 5792,C(=O)(CC1=NNC(=O)C1)NC1CCC(NC(CN(CC)CC)=O)C1 5793,c1(C(=O)NCCN(C(C=CC)=O)CC)cccc(C2CCCOC2)c1 5794,N1(C(c2ccc(C)n2C)=O)CC2CCC1CN2C(c1ccc(-c2ccco2)o1)=O 5795,C1(COC)CN(C(c2cc(CNC(=O)CC3(C)CCC3)[nH]n2)=O)CCO1 5796,C12(CNC(C3(CC=C)CC=CC3)=O)CC(CO1)N(C(=O)CC1(C)CC1(F)Cl)C2 5797,Cc1cccc(C(N2CC(C(O)C(=O)NCCCS(N)(=O)=O)C2)=O)c1 5798,c1(C(=O)O)n[nH]c2c1CCN(C1CC1)C2.C12CCC(O1)c1cc2n[nH]1 5799,S(=O)(=O)(c1cccc(=NCc2cc[nH]c(=N)n2)[nH]1)NCCSCC 5800,Cc1cc(S(=O)(=O)N2CCNCC(NC(=O)C(C)CC(F)(F)F)C2)sc1C 5801,CC1(C)C2CN(CC(N3CCCCCCC3)=O)CC12.C(=O)C1CC1 5802,C1(c2cccs2)CCC2(CC1)CNC2.CC(C)(C=O)Nc1nnco1 5803,C1(S(N)(=O)=O)(C(=O)NC2CCC(N(C(=O)C=CC(F)(F)F)C)CC2)CCC1 5804,c1(C(=O)NCCN(CCC)C(C2CCCOC2C)=O)ccc2nc(S)[nH]c2c1 5805,CC(C)(F)C(C)(F)CNC(=O)CC1CCCN1C(=O)Cc1ccc(F)nc1 5806,C1(Cn2cc(CN(CCCC)C)nn2)CCC(C(=O)O)CC1 5807,c1(NCc2c(C)ocn2)[nH]c(=NC2CCS(=O)(=O)C(C)C2)nc2sccc12 5808,c1(C(=O)OC)ccc(C(N2CCC(N(C(=O)CC(C)c3ccccc3)C)C2)=O)nc1 5809,O=C(Br)CC(=O)NC(c1nc[nH]n1)Cc1ccccc1 5810,C1(NC(C)=O)CCCC(NC(c2ccnc(CC3CCC3)c2)=O)C1.CN(C)CCS 5811,C(=O)(C(C#N)C(C)C)N1C2C(C(=O)NCC(CSC)(C)O)C(C2)C1 5812,C1(CNC(COCCC#C)=O)CCCCN(C(c2csc(-c3ccsc3)n2)=O)C1 5813,C(=O)(C1=COCCO1)NCC1(CNC(C(C(C)C)C)=O)CC1 5814,C1(NC(=O)C=Cc2ccc[nH]2)CS(=O)(=O)CC1NC(c1cc2c(s1)CCC2)=O 5815,C1(NC(c2cc(C3CC3)cs2)=O)CC12CCN(C(=O)CC1CC1(Cl)Cl)C2 5816,c1(OC2CN(Cc3cccc(OCC)c3)C2)ccc2c(C)cc(=O)oc2c1 5817,c1(C(N2C(CNC(CN3CCC(C)CC3)=O)COCC2)=O)ccn2cccc2c1 5818,N1(C(C2CC=C(C)CC2)=O)CCC2CN(C(=O)C=CC(=O)OC(C)C)C2C1 5819,n1(CC(N2CCCC(CN(C)C(c3cscc3F)=O)C2)=O)cc(Cl)c(O)nc1=O 5820,C1(C(=O)NC2C=CCCCC2)CN(C(=O)C(F)(F)CO)CC12CC2 5821,c1(NC(C2(NC(c3ccc4nccn4n3)=O)CC2)=O)ncc2cc(Br)ccc2n1 5822,CCC(C)C(O)C(=O)NCC1CC(C)(C)CN1C(C1COC(=O)N1)=O 5823,C(=O)(CC(CCCC)NC(=O)CCCC(C)SC)NC1CCCC(C#C)C1 5824,c1(C(=O)NC(C)(C)CNC(=O)CC#N)cccn2nnnc12 5825,Cc1ccc(NC(=O)CC(C)F)c(-n2cc(CNCC3CCCC3(C)C)nn2)c1 5826,c1(C(=O)NCC2CCCN(c3ccc([N+](=O)[O-])cc3)C2)coc2c1C(=O)NCC2 5827,C12(C(N3CC4(CCN4C(=O)C4CC4)C3)=O)CCOC1CC(=O)NC2 5828,c1(SCCC(=O)NCCC2(CNC(=O)Cn3cnnn3)CC2)ccccc1Cl 5829,CC1COC2(C1)CN(C(C1(NC(c3coc(CO)c3)=O)CSC1)=O)C2 5830,C1(C(=O)NCCCCN(C(C2(CCOCC)CCC2)=O)C)OCCCC1(C)C 5831,c1(CCC(C)NCc2n(CC)ccn2)cccc(OC(C)(C)C)c1 5832,CC1CN(C(c2ocnc2C2CCC2)=O)CC1CCNC(=O)CCOC1CC1 5833,n1(CC(=O)NCC(C)(CO)NC(=O)CCC2CCCO2)ccc2ccccc12 5834,CC(C)CCCCC(=O)NCC1CCC1C(N1CCC(n2cncn2)C1)=O 5835,C12(C(=O)NC3C(NC(c4ccc(CO)nc4)=O)COCC3)CCC(CO)(CC1)C2 5836,C=CC(C)CCN=c1[nH]c(=NCC2(C)CCOC2)c2sccc2[nH]1 5837,N1(C(C(COC)C)=O)CCC(CC(C)NC(=O)CN2CCNC(=O)C2)CC1 5838,C(CNC(c1ccc(C(F)(F)F)nn1)=O)(CC(F)(F)F)NC(C(C)(C)CO)=O 5839,C(C(C)C(C)C(=O)NCC(C)CN(C(=O)CC=Cc1ccc(F)cc1)C)OC 5840,C1(O)(CNC(C(CCC)OCC)=O)CCCN(C(C2CC3C=CC2CC3)=O)C1 5841,N1(C(c2c(CC)ncs2)=O)CC(O)CC1CC(=O)N(C1CC1)CC(C)C 5842,Clc1cccc(-c2nc(C3CCCCO3)n(-c3ccc(C4CCCO4)cc3)n2)n1 5843,N1(C(CC=C=C)=O)CCN(C2CCN(C(=O)C(C)OCC)C2)C(=O)C1 5844,C1(C(N(c2cccc3c2OCCO3)C)=O)COc2c(cc(Cl)cc2[N+](=O)[O-])C1 5845,C1(C(=O)NCC(F)(F)C(F)F)CC(O)CCN1C(c1cscc1Cl)=O 5846,CCCC(O)CCNC(c1cnc(C2CC2)s1)c1nnnn1C1CC1 5847,N1(C(c2c(C)n(C(C)C)nc2)=O)CC2CC1CN(C(=O)CC1CC3(COC3)C1)C2 5848,c1(C(C(=O)NCC=CCNC(C2CCC(F)C2)=O)(F)F)c(F)cccc1F 5849,N1(CC(=O)NC(CN(C(C(C)CC2CCCC2)=O)C)C)CCCNC1=O 5850,c1(NC(C)CS(C)(=O)=O)nc(N2Cc3cccn3C3(CC3)C2)nc2scnc12 5851,C1(C(=O)N(C)CC2CCN(C(=O)C=Cc3cnc(C)s3)C2)(CC)CCC(O)CC1 5852,C1(=CC(=O)NC2CCC(F)(CNC(C3(C)CCCOC3)=O)C2)CN2CCC1CC2 5853,C(CC(C)(C)CC(=O)N1CCCN(C(=O)Cc2c[nH]c(=N)nc2O)CC1)OC 5854,N1(CC)CCN(CC(N2CCCCC2C(C)NC(=O)C2CC2)=O)CC1 5855,C1(CC=C)(NC(=O)CNc2ccccn2)CCN(C(C2(n3cnc(C)n3)CC2)=O)C1 5856,C1(OCC)CC2CN(C(=O)COC3CCC3)CC12.c12nc(cs1)C(=O)NC2 5857,N1(C(Cn2nnc(C)n2)=O)CCC(C)(C)C(CNC(=O)CC2(C)CCOC2)C1 5858,c1(C2C(CC(=O)NC(c3nc(C)c(C)[nH]3)C)C2)cc(Cl)ccc1F 5859,C1(C(=O)NCC2CCCN(C(C)C)C2)CN(C)CCN1C 5860,CCCCCC(O)C(=O)N1CCC(C2CCCCN2Cc2cnc3occc3c2)C1 5861,c1(N2CCC(O)(C(C)NC(=O)Cc3cccnc3)CC2)ncnn2cccc12 5862,c1(C(N2CCC(NC(C3(C)CCCS3(=O)=O)=O)C2)=O)cc2c(Cl)nccc2o1 5863,c1(C(=O)NC2C3CN(C(C4(SCC)CC4)=O)C2C(O)C3)sc2cccnc2c1Cl 5864,C1(CNC(c2cnoc2)=O)CCN(C(c2cn3ccccc3n2)=O)CC1(F)F 5865,Cc1ccc(C(N2CC(C(F)Cn3cc(C4CCCC4O)nn3)C2)=O)o1 5866,CC1(C)C(N(C(=O)CCc2cnn[nH]2)CCc2ccccc2)CCN1CCO 5867,N1(Cc2n(C)cnc2)C2CCC1CN(C(c1ccc(OC(F)F)c(I)c1)=O)C2 5868,N1(C(=O)C=CC(F)(F)F)CCC2CN(C(c3cnn(C(F)F)c3)=O)CCC2C1 5869,C1(CCOC)CCC(C)N(CCc2ccc(I)s2)C1.c12ccc(cc1)OC2 5870,C=Cc1cc(C(=O)NCC2CCC(C)CN2C(c2nccc(C)n2)=O)cc(F)c1 5871,N1(C(c2cccc(O)n2)=O)CCCC2(C1)CN(C(C1CCC3(CC3)C1)=O)C2 5872,CCCCC(C(=O)NCCC(C)NC(=O)CCCc1cccs1)NC(N)=O 5873,c1(N2CCN(CC)CC2)cccc(NC(c2nc(C3CC3)oc2C)=O)c1C 5874,N1(C(C(=O)NCC(C)(C)OC)=O)CCN(C(C)=O)C2CCCCC2C1 5875,c1(OC)nc(=NC2CC3CN(C(c4cnc(OC)s4)=O)CC23)nc(OC)[nH]1 5876,C1(N(C)C(c2cn(-c3ccc(Br)cn3)nn2)=O)CCc2nnnn2C1 5877,c1(CNC(=O)CSc2ccccn2)cnn2c1CN(C(=O)C=CC1CCC1)CC2 5878,n1(CCC(N2CC3CCC3(NC(C3CCC3)=O)C2)=O)ncc(=O)c2ccccc12 5879,N1(C(C2CCCCCC2)=O)CCCCC1CCC(=O)NC1C(C(N)=O)COC1 5880,c1(OC)nscc1C(=O)NC1COCC1NC(C1CC1(C)C)=O 5881,C(=O)(C(F)(F)C(F)(F)F)NCCCCN(C(=O)CC1(C)CCS(=O)(=O)N1)C 5882,c1(C(N(CC(C)NC(c2cnc(CC)o2)=O)CC)=O)ccc(C(F)F)cn1 5883,N1(C(c2[nH]cc(CC)c2)=O)CCN(C(c2sc(C)cc2OC)=O)C(CC2CC2)C1 5884,CC(=O)CCCC(=O)OC(C(=O)N1CCC1C(=O)OC(C)(C)C)C(C)C 5885,C(=O)(C(O)CC(C)C)NCCN(C(COCC)=O)Cc1noc(C2CC2)n1 5886,N1(C(c2snc(C)c2N)=O)CCC(N=[N+]=[N-])(C(=O)NCC(O)CF)C1 5887,CCC(CC)C(C(=O)NC(C)CCC(=O)NCC(=O)N(C)OCC(F)(F)F)OC 5888,O=C(C#CC1CCCC1)NCCNC(C1CCCC(O)C1)=O 5889,N1(C(C2CC(=C)C2)=O)CC2CC2(NC(=O)Cn2ccnn2)C1 5890,C1(CNC(C2C(CC)OCC2)=O)CCCN(C(c2cnc(C(C)O)s2)=O)C1 5891,Cc1ccc(O)c(CNC(=O)C(c2ccccc2)NC(C2CCN(C)CC2)=O)n1 5892,N1(C(=O)Cc2cn[nH]c2)CC(C2CN(C(=O)CCSc3ccc(F)c(F)c3)C2)C1 5893,C1(C(=O)NC(C)Cn2cc(CN3CC4CC4C3)nn2)CCC(=O)C(C)C1(C)C 5894,C1(CCCNC(C2C(C)C2C)=O)CCN(C(=O)CC2CCC(=O)O2)CC1 5895,N1(C(c2cc(C)no2)=O)CCCC(O)(CNC(c2cc(Cl)ncc2N)=O)C1 5896,C1(CN=C(NCCOC)NCCOC(C)(C)C)CCCCC1(F)F.c1(C)cccs1 5897,N1(C(C(C(C)C)C)=O)CCC(C)N(C(=O)CCCCOCCN(C)C)CC1 5898,S(=O)(=O)(c1ccc(OC)nc1)NC(c1c(CC)cncc1)=O 5899,C12(CNC(=O)Cc3csnn3)CCCC1CCN2C(c1ncccn1)=O 5900,n1(CC(=O)NC(CNC(c2cc(C)c(C)nc2)=O)CO)ncn2nccc2c1=O 5901,C(=O)(CC(C)C(=O)N1CCC(C(N2CC(CO)C2)=O)C1C(C)C)OC 5902,c1(CC)nc(COC)cs1.N12CCC(C1)C2=O 5903,CC(C#N)CN=C(NCC1CCN1Cc1cccc(Cl)c1)NC(C)C 5904,Cc1c(C(=O)N(C2(CF)CC2)C)cnn1C.c12csc(c1)CNC2=O 5905,C(CC(C(=O)NC(C)C(C(C)C)OC)NC(=O)Cn1cc(Cl)cn1)OC 5906,CC12CCC(C)(CN1CCC1CCNCCC1(F)F)C2 5907,N(C1c2ccccc2CC1C)C(c1c(-c2c(C(=O)OC)cccc2)csc1)=O 5908,c1(C(N2C(CNC(C(C)Cc3ccco3)=O)C=CC2)=O)cc2n(c1)CCC2 5909,C(N=c1nc(N(C)CC2(N(C)C)CC2)c2c([nH]1)CCOC2)C1(CCC)CCC1 5910,S(=O)(=O)(c1cnccc1NCC1(CCO)CCC1)NCC1N(C)CCC1 5911,c1(NC(C2C(C(=O)NC3(CC(=O)OC)CC3)C2)=O)cc2ncncc2cc1C 5912,c1(OC)cc(F)c(F)cc1C(=O)NCC(C(=O)NC12CC3CC1C2C3)NC(C)=O 5913,C(=O)(C(Cc1cn[nH]c1)NC(c1cnc(O)o1)=O)N(CCOC)CC 5914,C1(N(C(C(CC)C)=O)C(C2CCCO2)=O)CCN(C(=O)Cc2cccc(F)c2)CC1 5915,C1(NC(CCOC)=O)CCCOC12CCN(C(c1sccc1Cl)=O)CC2 5916,c1(CC)ccc(Br)cc1C(=O)NC(C)CCN(C)C(C1C(C)(C)C1(F)F)=O 5917,CN1CC(NC(=O)NCC23CC(C2)C(C(F)(F)F)O3)Cc2ccccc21 5918,c1(C(=O)Nc2ccnc(O)c2)nc2n(c1Cl)CCN(Cc1cc(Cl)ccc1Br)C2 5919,C1(C)(NC(CN(CC(C)C)C(c2ccn(CCC)n2)=O)=O)CCC(C)(C)C1 5920,c1(CNC2(CC(=O)Nc3cncnc3O)CCC2)ccc(Cl)c(F)c1 5921,C1(NC(C(C)CF)=O)CN(C(c2cc3n(n2)CCC3)=O)CC12CCC2 5922,N#Cc1cncc(C(c2sncc2C#N)NN2CCSC(c3ccccc3)C2)c1 5923,c1(CC(=O)NC(C)CCCNC(C2CCN(CCCO)C2)=O)ccc(F)cc1 5924,Cc1ncc(Cl)cc1C(N1CC(N(C(=O)CC2CC(O)C2(C)C)C)C1)=O 5925,N1(C(C(C)(C)C2CCOC2)=O)CCC(C)(NC(c2cc[nH]n2)=O)C1 5926,S(=O)(=O)(c1cccc(=NCCCOCCO)[nH]1)N1CCC(OCC=C)C1 5927,c1(C(=O)NC2(C(N3CC(COC)C3)=O)CCC2)cncn(C)c1=O 5928,c1(C(=O)NCC)ccc(S(N)(=O)=O)c(NC(=O)C(=O)NC(C)C(=O)OC)c1 5929,c1(C(N2CCC(CN(C(CCN(C(C)=O)C)=O)C)C2)=O)cn(C(C)(C)C)nc1C 5930,c1(OC)cc(C(N2CCC(C(=O)Nc3cccnc3C(F)(F)F)C2)=O)cc(Br)c1 5931,c1(C(=O)NCC2CCCN(C(C3C(C#C)C3)=O)C2)cc2scc(Br)c2s1 5932,N1(C(CCC)=O)CCC(N(C)C(C2CCCN2C(=O)OC2CCC2)=O)C1 5933,CC(C(C)C(=O)NC1CC(NC(C2CCCCC2(F)F)=O)C1(C)C)S(C)(=O)=O 5934,c1(C(C)C)cccc(C(=O)N(C)C(C2CCC(NCC3CC4CC4C3)CC2)=O)n1 5935,c1(OC)ncnc(N2CCN(C(c3ccc(C(F)F)nc3)=O)C(C)C2)c1C 5936,O(NC(=O)C(C1(O)CCC1)NC(c1ccc(O)cc1)=O)CC=CC 5937,C1(c2nnc(C)n2C)CCN(C(=NCC2CC(CO)CO2)NCc2ccco2)CC1 5938,c1(C(N2CCSC(C)C2C)=O)ccc(F)c(-c2ccccc2)c1Cl 5939,CC1CCN(C(=O)CC(C2CCC2)C2CCC2)C1C(=O)NCC1(O)CCC1 5940,C1(C)(C(N2CCC(O)(CN(C(=O)C3=CCOC3)C)CC2)=O)CC(C(C)(C)C)=NO1 5941,C12(C(=O)NCCCn3cc(C(C)(C)NS(C)(=O)=O)nn3)CC(C(F)(F)F)(CO1)C2 5942,c1(C(=O)NCC2(NC(=O)CCc3nccs3)CC2)ccc(C(F)(F)F)nc1 5943,c1(C(=O)NCC(=O)OCC)ccc(C(C)(C)C)cc1.C1(CC)CNC(C)C(=O)N1 5944,c1(CC(C)C)ccc(CN2CC(C)(CNC(C3CCCOCC3)=O)C2)cc1 5945,c1(C(=O)NCC2C(NC(c3n(CC)nc(C4CC4)c3)=O)C2)cccc2c1C(=O)NC2 5946,C1(CC)CN(C(=O)CCc2cccnc2)CCC1N=c1[nH]c2ccc(O)cc2s1 5947,S(=O)(=O)(c1cnn(C)c1)NC(N1CC(C(=O)OC)OC(CO)C1)=O 5948,CC1CC(C(=O)NCC(C)(C)NC(=O)CCc2ccc(F)cc2)=NO1 5949,c1(C(=O)NC2(C3CN(C(CSC(C)(C)C)=O)C3)CC2)nn(C)c2c1COCC2 5950,CC#CCCCC(=O)NC1C=CC(CNC(=O)CCCN2CCCCC2)C1 5951,c1(C(n2cc(C3CCN(C(C4COCCO4)=O)C3)nn2)C)ccccc1F 5952,C1(C(N(CCNC(C(C)CF)=O)CC2CC2)=O)CCc2ccccc2C1 5953,C(=O)(C(F)(F)CCn1cccn1)NC1C(CNC(C2CC=C(C)CC2)=O)C1 5954,c1(NC(C2CN(C(c3c(OC)cncn3)=O)C2)=O)c(C)cccc1[N+](=O)[O-] 5955,C(=O)(C(CC(F)F)N(c1ccc(C)cc1)C)OCC(N1CCC(OC)CC1)C 5956,C1(N)(CO)CCOCC1.C1(c2cc[nH]n2)(CN(C)C)CCOCC1.C12CN(C1)C2=O 5957,c1(OC)cccc2[nH]c(C(N3CC(F)(CNC(C4CCNC(=O)C4)=O)C3)=O)cc12 5958,CC(C(=O)NCCOC(C)(C)CNC(C1CC(=O)NC(=O)N1)=O)C(C)S(C)(=O)=O 5959,n1(CC)cccc1C(=O)NCC(CCNC(c1ccc(CO)s1)=O)OC 5960,C(=O)(C1=CS(=O)CCC1)NC(CC=C)CNC(C1CCCN1C1CCCC1)=O 5961,c1(CNCCN(CCC)C)ccc2c(c1)NC(=O)C2 5962,C(C(=O)N1Cc2ccccc2CO1)C1(NC(COC)=O)CCC1 5963,Cc1ccc(N(C(=O)CC2CCCN2C(C2CC3CC3C2)=O)C)c(C)c1 5964,c1(CN2CC(C#N)C(NC(c3ccc(S)cc3)=O)C2)cc(Br)cc(F)c1F 5965,N1(C(CCCOCCC)=O)CC(C(=O)N(CC(C)CO)C)C(C)(C)C1 5966,N1(C(C2CC(C(=O)OC)C2)=O)CCC(C(=O)NCCCC(C)CO)CC1(C)C 5967,N1(C(CCc2ccc(C)o2)=O)CCOCC1CC(N1CC(F)(F)C1C1CC1)=O 5968,c1(CC(c2ccc(OC)cc2)=O)c[nH]c2ccc(-c3coc(C)c3)cc12.C=O 5969,C(=O)(C1=NN(CCO)C(=O)CC1)NCC(CCOC)NC(C(C)(C1CC1)OC)=O 5970,C(=O)(C1CCCn2c(Br)cnc21)NC(C(CO)N(C)C)=O.C123CC1(C2)C3 5971,C(N=c1[nH]c(NC2CCN(C)C2C)nc2cccnc12)c1c(C)n(C)nc1 5972,Cc1cc(CNC(C2CC(C)N2C(=O)CCC2(C)CC2)=O)ccc1F 5973,CC(C)CC(C(=O)O)NC(C1CCCN(C(c2ccnn2C)=O)C1)=O 5974,c1(C(=O)NCCN(C(c2cc(C(=O)OC)sc2)=O)C)nc(CN(C)C)cc(O)n1 5975,c1(NC(=O)NCc2csc(C3CC3)c2)cc2c(nc1O)CCC2 5976,c1(C(=O)NC2C(CNC(C(C)SC)=O)C2)ccc(-n2cccn2)nc1 5977,N1(C(C(COC)OC)=O)C2CCC1CC(NC(c1ccccc1SC(C)C)=O)C2 5978,C1(NC(C(CSC)C)=O)COCCN(Cc2ccc(F)c(F)c2)C1 5979,CCC(O)C(C)(C)C(=O)NC(c1nc(C(C)(C)C)no1)COC 5980,c1(C(N2CCCOCC2)C(=O)NCCCC(=O)OCC)nc(C)c(Br)s1 5981,C1(CC(=O)NCc2cn[nH]c2)CCN(C(C2CCO2)=O)CC1 5982,N1(C(CCSCCC)=O)CC(NC(c2c(C)csc2Cl)=O)CC1(C)CC 5983,C(=O)(CCCC(=O)NC(CNC(=O)CS)CC)NC(C)C.N1(CC)CCC(OC)C1 5984,C1(C(=O)NCCN(C(=O)CCc2ccn(C)c2)C)CCC(=O)N2CCCC12 5985,N12CC3C(C3C1)NC(C)C2=O.c1(NC(CCOCOC)=O)cccnc1 5986,c1(OC)cc(CCNC(c2scnc2Cl)c2nnnn2C2CCCC2)ccc1Br 5987,Cc1nc(C#N)c2c3c(sc2n1)CCCC3.c1(C=O)ccc2c(c1O)CCC2=O 5988,C1(C)(CN(C(CC2(OC)CNC2)=O)C2CC2)CC=C(C)CC1 5989,c1(N(C)CC2CC2(F)F)cccc(S(=O)(=O)N2CCSC(c3ccccc3)C2)n1 5990,CCCCC(C(=O)NC)NC(=O)CCC=CBr 5991,C(CCCCC(=O)N(C)CC1(O)CCCN(C(=O)CC2CC(F)C2)C1)OCC 5992,C1(C(=O)NCC(CNC(=O)Cc2ccccc2C(=O)O)O)CCC(F)(F)CO1 5993,c1(C(=O)NC(C(=O)NC(C=C)CO)c2ccco2)cnccn1 5994,S(=O)(=O)(c1c(F)cc(F)cc1F)NCc1scc(C(=O)Nc2cccc(Br)c2F)n1 5995,CCCCC(C(=O)NCc1cc(C2CC2)no1)NC(C1OCCC1(C)C)=O 5996,n1(C2CN(C(C(=O)Nc3cccc(SCC#C)c3Cl)=O)C2)c(C)cc(C)nc1=O 5997,c1(C(=O)NC2CN(C(C(C)O)=O)CC2F)cn2ccc(Br)cc2n1 5998,C1(O)(CN(C(C(C)SC(C)C)=O)C)CCN(C(c2n[nH]c(C3CC3)c2Cl)=O)C1 5999,C=CCC(CC)C(=O)N1CCN(C(=O)C(CCSC)NC(C)=O)CC1CC(F)F 6000,C1(NC(CC2(C)CCN2C(c2cnsc2)=O)=O)CC(O)C(O)C1 6001,N1(CC(=O)NC(C(C)NC(C2CCC(=O)O2)=O)(C)C)CCC(C(N)=O)CC1 6002,Cc1cc(C(=O)NC2CC(NC(c3ccc(C)c(C)n3)=O)C2)c2sc(=N)[nH]c2n1 6003,N1(C(c2ccc(C3(C(F)F)CCC3)cc2)=O)Cc2cccc(F)c2C1 6004,Cc1nc(C(=O)NCCC2CCCN2C(=O)CO)ccc1Br 6005,c1(N2CCC(CNC(c3nccc(OC)c3)=O)C2(C)C)ncc2ccccc2n1 6006,c1(C(=O)NC2CCN(C(C(C3CCC3)OC)=O)C2C(C)C)coc(S(C)(=O)=O)c1 6007,C1(C(=O)NCC2=CCN(C(C3CCCCC(=O)C3)=O)CC2)CCn2ncnc2C1 6008,N1(C(CC2(C=C)CC2)=O)CCCC2(NC(C3CCC(C(N)=O)CC3)=O)CC2C1 6009,c1(C(N2CC(NC(C(C)(C)C3CCOCC3)=O)C3C2C3)=O)cc2scc(Cl)c2[nH]1 6010,C1(CNC(c2cscc2C(F)F)=O)CCN(C(C2CC2C(F)F)=O)C1 6011,c1(CC)nn(C)cc1C(=O)NC(C1CCN(C(C2CCO2)=O)C1)C 6012,CCCCC(CNC(C1CC1c1ccncc1F)=O)NC(C1CCCSC1)=O 6013,C(N=c1nc(N2CC3CC2CS3=O)c2c([nH]1)CCCCCC2)C1C(=O)NC(=O)N1 6014,c1c(C)cccc1Br.c1(COC)cn(CC2C=CCN2C(=O)CCC2(C)CC2)nn1 6015,N1(C(C2N(CCC)CCC2)=O)CCCC2(CCCCC2NC(C)=O)C1 6016,Nc1c(F)c(F)cc(C(N2CCN(C(=O)CSC(F)F)C3COCC23)=O)c1Cl 6017,CC(CCC(=O)Nc1cncnc1C(C)C)NC(=O)CC1CC(N(C)C)C1 6018,c1(OCC)ccc(C)nc1C(=O)NC(C)CCNC(c1cc([N+](=O)[O-])c[nH]1)=O 6019,c1(C(=O)NCC2(C(N)=O)CN(C(C=NOC)=O)C2)cc2ccc(F)cc2s1 6020,Cc1cc(F)c(C(=O)NC2CC(CCNC(C3CCOC3C)=O)C2)cc1F 6021,C1(C2CC2)(C(=O)NCCCCNC(=O)C=CCN2CCOCC2)CCC1 6022,C(=O)(C1SCCc2sccc21)N1CCC2(CC(NC(=O)CC=C(Cl)Cl)C2)C1 6023,c1(C(=O)NCCC2(NC(=O)CC3CC4CCC3C4)CC2)ncc(Br)cc1O 6024,C1(C(N(CCNC(c2ccc3nncn3c2)=O)C2CC2)=O)CCc2nnnn2C1 6025,O=C(C(F)C1=CCCCC1)NCC1CCCN1C(C1CC2(CCCC2)CO1)=O 6026,c1(OC)ncc(Cl)c(C(N2CC3(NC(=O)C(C(C)C)SC)CC2C3)=O)c1Cl 6027,c1(N(C)C)nccc(NCC2CC2NC(C2(S(C)(=O)=O)CCC2)=O)c1[N+](=O)[O-] 6028,Cc1nc(CO)ncc1C(N1CCC(N(C)C(c2ncsc2C)=O)C(C)C1)=O 6029,c1(C(N2CCC(C#N)(NC(C(C(C)C)O)=O)C2)=O)cnc2ccccn12 6030,C(=O)(C1=CC2(CCOCC2)C1)NC1CC(C)N(C(=O)C=C2CN3CCC2CC3)CC1 6031,S(=O)(=O)(c1cccnc1NCC1CCCC1C(C)(C)C)N(C1(C)CCCC1)C 6032,C1(C)(CNC(C(c2ccnn2C)NC(Cc2cnc(C)s2)=O)=O)CCN(C)C1 6033,C1(C(=O)NCC2C(NC(c3nc(C(C)=O)sc3)=O)COC2)CCN(CCO)C(=O)C1 6034,C=CCCCCCCCC(=O)N1CCCC1(COC)NC(=O)CC12COCC(C1)C2 6035,N1(C(C(C)CC2CCCC2)=O)C2CCC1CN(C(=O)CN1CC(C)(N(C)C)C1)C2 6036,c1(C(=O)NC(C(C)NC(Cc2c(C)n[nH]c2C)=O)(C)C)cnn2c1OCC(C)C2 6037,c1(CC2(C(=O)NC3CC(O)(CNC(C4CCCO4)=O)C3)CC2)cccc(F)c1 6038,N1(C(CCc2cn(C)nc2)=O)CCC(NC(=O)C=CCN2CCCCC2)C1CO 6039,C(=O)(C(CC(F)F)NC(=O)Cc1cn[nH]c1)N1CCN(C(C)(C)C)CC1 6040,C1(CNC(c2n(C)ncc2)=O)CC2CC1CN2C(c1ccc(C(F)(F)F)cn1)=O 6041,Cc1nn(CC(N2CC(NC(C3(C)CCC3)=O)C(CO)C2)=O)cc1Br 6042,C1(NC(C(n2ncc(C)c2)C)=O)CCCCC1NC(=O)C=Cc1ccoc1 6043,C(=O)(C(F)(CNC(C1CC(C(=O)OC)C1)=O)C(C)C)N(c1cccc(CC)c1)C 6044,N1(C(C=C(CC)C)=O)CCN(C(=O)COC2CC(F)(F)C2)CC1CC 6045,N1(c2cc(NCC3CCN(C)C3)ncn2)CCOC(C)(c2ccccc2)C1 6046,C(=O)(C(C)(C)C(=O)Nc1ccc(F)c(F)c1)NC1CC(C)N(c2ccncn2)C1 6047,c1(C(CC)C)ccc(C(=O)NC2CCC2CNC(C2(O)CC2)=O)c(O)n1 6048,c1(C(=O)NCCNC(C2(OC(C)(C)C)CC2)=O)n[nH]c(=N)[nH]1 6049,C1(C2CC2)(NC(CN(CCC)C(C2CC2C(F)(F)F)=O)=O)CCCC1 6050,c1(NC(c2ccc(OC(F)(F)Cl)cc2)=O)cccc(-c2nc(O)n[nH]2)c1 6051,c1(SC)cc(N(CC(C)C)C(C2CCCOCC2)=O)nc(SC)n1.C1CN1 6052,CCCCC(CN1CCCC(NC(c2n[nH]c(C)c2C)=O)CC1)CC 6053,CP(C)(=O)C1CCCN(C(=O)NCC(c2ccccc2)C2CC2)C1 6054,N1(C(C(C(C)O)NC(C)=O)=O)CC2(CCC2)CCC1CNC(=O)CNC=O 6055,CS(C)(=O)=Nc1nc(C(=O)NC2CCN(C(=O)C=Cc3cnc[nH]3)C23CC3)cs1 6056,C1(NC(C=CC=CC)=O)CC2CCC(C1C)N2c1nccn2nnnc12 6057,C1(C(=O)NCCCN(C(C2CS(=O)(=O)C2)=O)CC)CCC1(F)F 6058,CC1=CCSC1C(=O)NCC(C1CCCC1)NC(C1CCC(C(N)=O)C1)=O 6059,C1(OC)(CNC(c2nc(Cl)c(Cl)s2)=O)CCN(C(c2cnc(C(N)=O)s2)=O)C1 6060,C1(N(C(c2cn(C3CCC3)nn2)C(=O)NCC(=C)C)C)CS(=O)(=O)C12CCOCC2 6061,N(C1c2ccccc2CC1NC(C12CCC(CC1)CC2)=O)C(C(C)C1CCC1)=O 6062,CCCC(CC)C(=O)NC1CN(C(=O)C2=NNC(=O)C2)CC1CC 6063,C1(NC(C(CC)CO)=O)CC2CN(C(=O)C(c3ccccc3F)(F)F)CC2C1 6064,N1(C(C(C)N(C(C2CC(CCC)C2)=O)CCC)=O)CCOC2C(O)CC12 6065,C1(NC(C(CC=C)C)=O)CC(OC)CN(C(c2cc(C)n(CC)n2)=O)C1 6066,C=CCCC(C(=O)OC)NC(C1CC=CCC1NC(=O)C(C)(C)CSC)=O 6067,C1(NC(c2c(OC)csc2)=O)CC2CN(C(c3ccc(CO)s3)=O)CC2C1 6068,N1(C(COCC=C)=O)CCC(CNC(c2cccc(C)c2)=O)C12CCC2 6069,CC1(C)C2CC1CN(C(=O)CC(=O)NCCOCC(F)(F)F)C2 6070,C1(CNC(Cc2c(C)con2)=O)(CNC(c2cc(C)n(C(F)F)n2)=O)CC12CCC2 6071,C1(C(=O)Nc2cnn(CCC)c2C(C)C)C2Cc3c(Br)cccc3C12 6072,C1(C(N(CCCC)CCOC)=O)CCC2(CN(C(c3cnccn3)=O)C2)O1 6073,N1(C(CC(c2scc(C)c2)O)=O)CC=CC(NC(c2ccc(C(C)C)nc2)=O)C1 6074,Cc1ccnc(-c2cn(C3CCC(NC(=O)CN4CCCCCC4)C3)nn2)c1N 6075,Cc1cncc(C)c1C(N1CCCCC1C(C)NC(c1ccc(C#N)n1C)=O)=O 6076,C(CCCCCN(C(=O)CCn1ncn(C)c1=O)C)NC(C1(CC)CC1(F)F)=O 6077,C(=O)(CCN1C(=O)C(C)Oc2ccccc21)NC(C)CCCCl 6078,N1(CC)C(C)(C(=O)OC)c2cc(OCc3cc(Br)c(C#N)s3)ccc21 6079,N1(C(C2CC(OC)C2)=O)CCOC2CN(C(c3nccc(Cl)c3O)=O)CC12 6080,N1(C(C(C)n2cccc2)=O)CCC2(CC2)CC1C(=O)NCCN1CC=CC1 6081,O(NC(=O)C(O)C1CN(C(c2ccc(=N)[nH]n2)=O)C1)CC1CC(=C)C1 6082,C(=O)(C(CCC(N)=O)n1cc(CNC2CCCC2)nn1)NC(C(C(CC)O)C)=O 6083,C#Cc1ccc(CNC(=O)C(C)C(C)NC(=O)CCN2CCOCC2)cc1 6084,n1(CC)c(=O)cnc2ccc(NCc3cc(Br)cc4c3OCC4)cc12 6085,N1(C(C(CC)NC(=O)C(=O)NC2CC2)=O)CCOC(C)(C)C1C 6086,Cc1sc(C(F)(F)F)nc1C(=O)NCC(C(C)(C)C)NC(=O)C(C)OC(C)(C)C 6087,C1(NC(CC2(CC)CCCC2)=O)CCCN(C(=O)C(c2cc(F)ccc2F)=O)C1C 6088,c1(C(=O)NC(CC(=O)OCCC(c2ccccc2)O)=O)cccc(Cl)c1 6089,C=CC(C)(C)CC(=O)N1CCC(CCC(=O)N(CCN(C)C)CCC(C)CCC=C)C1.OC 6090,c1(C(N(CCNC(C(c2c(C)noc2C)C)=O)C)=O)ccc2c(c1)OC(C)(C)O2 6091,C1(C)(C(N(C)CC2CCN(C(C3(C)CCCO3)=O)C2)=O)CCCNC1=O 6092,n1(CC)ncc2c(C(=O)OC(C3CCCCC3)C(=O)OC)cc(C)nc12 6093,c1(CNC(C2C=C(C)CS2)=O)cnc(C)c(C)c1.c12cncc(c1)NC2=O 6094,C=CC(C)(C)CC(=O)NC1CC(C)N(C(=O)C(O)Cc2cnc[nH]2)C1 6095,Cc1cc(C(=O)NCc2nn(-c3ccccc3)c(C)cc2=O)n2ncc(Br)c2n1 6096,Cc1cc(NC(=O)NC2CCCC23CC3)cc(Br)n1 6097,c1(C(=O)NC(CN(C(c2cc(OCC)ncc2)=O)C)C)cc(F)c(N)cc1F 6098,Cc1nccc(NCC2CCCN(C(c3ccc(CCN=[N+]=[N-])cc3)=O)C2)n1 6099,C12(CNC(=O)Cc3cc[nH]n3)CC1CN(C(=O)Cc1cc(Cl)sc1Cl)C2 6100,C1(OC)CC2CC1CN2C(=O)C=Cc1cn(C)cn1.c12cc[nH]c1C(=O)NC2 6101,c1(NCC2N(C(C3CCCS3(=O)=O)=O)CCC2)ncnc2ccc(O)cc12 6102,C(CC(C(=O)NOCC(=C)Cl)NC(C1CC1c1ccncc1)=O)=CC 6103,CC1CCCC=C1C(=O)N1CCCC(F)(C(=O)NC(c2cncn2C)CO)C1 6104,CCCCCS(=O)(=O)CC(=O)NCC1(C)CCCN(C(=O)CC(=O)N(C)C)C1 6105,C1(NC(c2cccc(OC(C)C)n2)=O)CCN(Cc2ccc(Cl)cc2Cl)C(C)C1 6106,c1(OC(C)C(=O)N(CCNC(c2ccc(O)nc2)=O)C2CC2)ccc(Cl)c(Cl)c1 6107,N1(C(Cc2scc(C)c2)=O)CC2CC(C(=O)N(C)C(c3nccs3)C)C(C2)C1 6108,C1(C)(C(=O)NCCCNC(C(C)=C2CCC2)=O)CC2CCC(C1)S2 6109,N1(C(C(COC)N(C)C)=O)CC2(C(N3CC(O)C(F)C3)=O)CC1CCO2 6110,C1(CNC(CNC(=O)NC)=O)CN(C(C2CCCC(=O)C2)=O)C(C)(C)C1 6111,CC1(CNC(c2cnc(NC3CC3)s2)=O)CC12CCN(C(=O)CCC#N)CC2 6112,C1(C(N2C(C(=O)OC)CC2)=O)CCCC(NC(=O)C(=O)N(C)C)C1 6113,C1(NC(CNc2ncc(C)o2)=O)CCCC(N(C(=O)CCSC(F)(F)F)C)C1 6114,C1(CNC(C(CC=C)(F)F)=O)CN(C(c2cnc(C3CC3)s2)=O)CCC1(F)F 6115,N1(C(c2cc(O)cc(O)n2)=O)CCCC2(CCN(C(=O)C(F)(F)C(F)F)C2)C1 6116,N1(C(C=CCN(CC#C)C)=O)CCN(C(C)CNC(C2CC2(Cl)Cl)=O)CC1 6117,CN1CC=C(CC(=O)N2CCC(OCC(N3CC(C4CC4)(CO)C3)=O)C2)CC1 6118,C1(OC)CN(C(=O)C(O)C(F)(F)F)CCC1C(N1CC=C(C)C1)=O 6119,CC(C)(C(=O)NC(CN(C)C(c1coc(Cl)c1)=O)(CO)CO)C1=CCSCC1 6120,N1(C(CS(CC)(=O)=O)=O)CC2CCCC(NC(=O)CSCCC#N)C2C1 6121,CCC(O)C(C)(C)C(=O)NC1CCCC1NC(c1cccc(OC)c1O)=O 6122,C1(CNC(C(C(C)O)(C)C)=O)CCN(C(c2n[nH]c(=N)s2)=O)CCC1(F)F 6123,CC(C(=O)NCCc1noc(CO)n1)(C1CCC1)NC(c1ccc[nH]1)=O 6124,C#Cc1cncc(C(N2CCCCOC(C(F)(F)F)C2)C(=O)NCC=C)c1 6125,CN1C(=O)CCCC1C(=O)NCC1CC(NC(C2(C)C=CCC2)=O)C1 6126,Cc1cc(C(N2CC(NC(=O)Cc3ccccc3)C3CC3C2)=O)c(C)n1C1CC1 6127,C1(CNC(CCNC(=O)OCC)=O)COCCN(C(=O)CC(CC)NC(N)=O)C1 6128,C(C1C(C(=O)NC2CC3CN(C(=O)Cc4ccncc4Cl)CC23)C1(C)C)=C(C)C 6129,C1(NC(c2c(CCC)n[nH]c2)=O)CN(C(=O)CC#N)CCC12CCC2 6130,n1(CC)nc(C)c([N+](=O)[O-])c1NC1CC1CNC(c1ccc(C(C)C)c(F)c1)=O 6131,Cc1cnc(C(=O)NCCC23CCC(C2)N(C(C2(C)CC2)=O)C3)c(F)c1 6132,C(CCCCCC(=O)NCCc1cn(Cc2ccnc(F)c2)nn1)NC(N)=O 6133,Cc1ccc(C(=O)NCC(O)CNC(=O)C2=C(Cl)CCOC2)c2cccnc12 6134,c1(Cc2c(C(N(CC(C)(C)NC(C3CC3C(F)F)=O)C)=O)nco2)ccc(F)cn1 6135,C(=O)(CC(CC)CCCC)NC(CCC)C(=O)NCCS(=O)(=O)NC 6136,N1(C(COCCC(C)C)=O)CC2CCN(C(c3cn(C)c(O)n3)=O)C(C2)C1 6137,c1(C(=O)NCC23CCC2CN(C(=O)CCF)C3)c[nH]ccc1=NC(=O)C(F)(F)F 6138,C#Cc1cc(C(N2CC3CCN(C(=O)C=Cc4ccccc4)CC23)=O)cc(F)c1 6139,CCCCCCNC(CN(C(C1CC(OC(C2CC2(F)Cl)=O)C1)=O)C)C 6140,CCCCC(O)C(C)C(=O)NCCCCCC(C)(C)NC(=O)C(C(C)C)N(C)C 6141,c1(NC(C2CCN(C(CCC=C)=O)CC2O)=O)ccc2c(c1)CCO2 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6160,C1(C(N2CC3(CCC3NC(C3C=CCC3)=O)C2)=O)(CC)CCC(F)(F)CC1 6161,Cc1noc(C)c1C(N1CC2(NC(C3CCC3C)=O)CC1C2)=O 6162,N1(Cc2c(OC)cco2)CCC(F)(F)C(C(=O)Nc2c(OC)cccc2OC)C1 6163,Cc1ccc(C(=O)N(C)CCN(C(c2coc(Cl)n2)=O)C(C)C)nc1 6164,Cc1cccc(F)c1CC(=O)NC1CC(N(C)C(c2c(C)ncn2C)=O)C1 6165,Cc1noc2ncnc(NC(C3CCCN(C(=O)CCn4cnnn4)C3)C)c12 6166,C1(C(N2CC(CCCCNC(C3(COC)COC3)=O)C2)=O)CC2(CC(OC)C2)C1 6167,c1(C(=O)OC)cc(C(=O)NC(C)(C)CCCNC(=O)C=C2CCC2)ccc1F 6168,C1(C)(CNC(c2c(C)ncs2)=O)CCCN(C(=O)CNc2cnn(C)c2)C1 6169,Cc1cncc2cc(C(N3CCCOC(CNC(=O)Cc4csnn4)C3)=O)sc12 6170,N1(C(c2snc(C)c2N)=O)CCCN(CCNC(=O)CC2CN(C)C(=O)N2)CC1 6171,O=C1CCC(C(=O)N2CCC(NC(=O)Cc3cc(C(F)(F)F)cc(Cl)c3)C2)=NN1 6172,C1(C(C(c2nn[nH]n2)C)OC(=O)NC(C)(C)C)COC2(c3nc(C)on3)CC1C2 6173,N1(C(c2c(OC)cc(N)cc2)=O)CCC2CN(C(C3CC3(Cl)Cl)=O)CC2C1 6174,C1(NC(C(C)(C)C2CCCO2)=O)CCCCN(C(c2cc3occc3s2)=O)C1 6175,N1(C(c2c(N)cccn2)=O)CCC2(CCOC2)C(CNC(c2csc(Cl)n2)=O)C1 6176,C12(CNC(CCC)=O)CCCCC1N(C(=O)C(=O)Nc1cc(OC)nn1C)CC2 6177,C1(C(=O)NC(c2ccccc2)C(=O)N(CC(C(C)C)O)C)(CO)CCCCC1 6178,C(=O)(C(CC(C)(C)C)NC(c1ncccn1)=O)N1CCC(O)(CCC)CC1 6179,C(CCCCNC(=O)COCC(C)(C)C)N(C(CCC1CC(C)C1)=O)C 6180,c1(C(=O)NCC(CNC(C2C(c3ccn(CC)n3)C2)=O)F)ccc(C)c(C)c1N 6181,c1(C2C(NC(c3nocc3C(=O)NC(=O)C=C3CCC3)(C)C)C2)ccccc1F 6182,C1(CC)CC(O)CN1C(=O)C(COC)NC(=O)Cn1ncccc1=O 6183,N1(C(c2c(C)cc[nH]2)=O)CCC(C(C)(C)C)(CNC(C2(n3cccn3)CC2)=O)C1 6184,C=CCCC(=O)NC(CNC(C1CN(C2CCOC2)C1)=O)C1CCC1 6185,C(=O)(C(C)C(C)S(C)(=O)=O)NC1(c2cn(C(C(=O)OC)(C)C)nn2)CCN(C)C1 6186,C(=O)(C#CC1CCCO1)NCC1(C(C)NC(c2c(C)nn(C(C)C)c2C)=O)CC1 6187,C(=O)(C(F)(F)C1=CCOCC1)N1C(C)C(NC(c2cccc(Cl)c2N)=O)CCC1 6188,C1(CC(=O)NC(C2CCCC2)CNC(CCSCCC)=O)CCCC(C2CC2)O1 6189,c1(C(=O)NC(CNC(C2(CC=C)CCC2)=O)CC(C)C)cc2c(O)cccc2[nH]1 6190,C(=O)(C(CO)C(C)C)N1C(Cn2cc(-n3c(C)cc(C)n3)nn2)CCC1 6191,C(CC(C(C)C)NC(c1cscc1C(=O)OC)=O)N(C(C=C(CCC)C)=O)C 6192,N1(Cc2cc(CNCc3cccc(OC)c3)sc2)CCCC2(CCC2)C1 6193,c1(CC(=O)NC2CN(C(C3(COC)CCCO3)=O)C2)cc2n(n1)CCCC2 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6230,C(=O)(CC=C(Cl)Cl)NCCC(C)NC(c1ccccc1OCC1CC1)=O 6231,CSC1=C(C(=O)NCC(O)CNC(=O)CCCCCCCC2CC2)CCCC1 6232,N1(C(CC2CCN(OC)CC2)=O)CCCC(O)(CNC(c2ccncc2)=O)CC1 6233,N1(C(C(C)CN(C)C)=O)CC2CCC1C(CNC(C1(C3CCCCO3)CC1)=O)C2 6234,c1(C(N2CCC(C(C)O)C2)C(=O)NCC=C)cc2ccc(OC)cc2o1 6235,C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC2(OCC(NC(C(C)(C)CC#N)=O)C2)C1 6236,c1(NC)ccc(S(=O)(=O)NC(C2C(Cl)(Cl)C23CC3)=O)c(C)c1 6237,c12cc(ccn1)CNC2=O.C1(C(N2C(C=C)CCC2)=O)CC2(CCO1)CC2 6238,N1(C(CCCC)=O)CC2CN(C(c3cccc(C(C)=O)c3)=O)CC2C1 6239,C1(NC(C(CN(C)C)NC(C2CCCC2)=O)=O)CCCC(F)(F)C1 6240,C(C(C(=O)N(CCN(C(=O)C(C)(C)C1(C)CC1(F)F)C)C(C)C)N(C)C)OC 6241,c1(C2C(C(=O)NCCC3(O)CCOCC3)C2)cccc(Br)c1F 6242,c1(CC(C)C)cc(C(=O)NC(C2(CNC(c3ccnn3C)=O)CC2)C)cc(O)n1 6243,C12(C(=O)OC)CC(C(=O)NCC(CNC(N3CCC(C)C3)=O)CO)(C1)OC2(C)C 6244,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CCN(C(C=CS(C)=O)=O)CC1O 6245,c1(C(=O)NC(CC(=O)NC(C=C)(C)CC)CC)cc(Cl)ccc1O 6246,N1(C(C2C(CC)C2)=O)CCN(CC(N2CCC(C3(C)N=N3)C2)=O)CC1 6247,Fc1ccc(I)cc1CBr.C(CC(F)(F)C(=O)NCSc1c[nH]nn1)c1scc(N)n1 6248,C(=O)(C1=COCC1)NCC1(F)CC(CNC(C2C(C(=O)OC)C2)=O)C1 6249,CCCC(C(=O)N1CCCC1C(C)NC(c1cncc(F)c1)=O)OCC 6250,c1(C(=O)NC(C)C=C2CN(C(=O)CSC3CCCO3)C2)cnc(C(F)(F)F)cn1 6251,Cc1nnc2n1CC(C(=O)N(CC(O)CNC(=O)C(C)(C)c1cnn(C)c1)C)C2 6252,c1(CC)ccc(S(=O)(=O)N2CCN(C(c3c(C)ccc(OC)c3C)=O)C2CC)cc1 6253,CC(CN(C)C)C(=O)NCc1occc1C(=O)NC(C1CCCCO1)C 6254,C1(NC(C2(CC)CC2)=O)CCN(Cc2cccc(-n3cncn3)c2)C1(C)C 6255,C1(CNC(CC2(NC(C(CC)NC(N)=O)=O)CCC2)=O)CCCCN(C)C1 6256,C1(NC(c2c(CCCC)ocn2)=O)CC2CC(NC(c3scnc3CC)=O)CC12 6257,c1(NC(=O)NCC2CCCN(C(c3cc(C)no3)=O)C2)ccc(Cl)cc1Cl 6258,c1(C(N2CCC(CC(=O)NCCc3ccco3)C2)=O)ccc(F)c(F)c1 6259,CCC(CC)(CC(=O)NC1CCCN(C(=O)CC(=O)NC2CC2)CC1)C(=O)OC 6260,c1(C(N2C(CNC(c3ccc(CO)cn3)=O)CCC2)=O)cn2cccc(Br)c2n1 6261,c1(-c2c(CNCc3n(C)ncc3Br)scc2)nnc(S)nc1O 6262,CC1(NC(=O)CCc2ccc(F)cc2)CCN(C(=O)C(F)C2CC2)CC1 6263,c1(C(N2CCN(C(C3(CO)CCCO3)=O)CC2)=O)ncc(F)cc1F 6264,Cc1cc(Cl)c(C(=O)NC2CCC(CNC(C3CNC(=O)N3C)=O)C2)cc1N 6265,C(=O)(C(C)C(=O)N1CCC(C)(NC(C2(COC)CC(F)(F)C2)=O)C1)OC 6266,N1(C(CC(C)c2ccncc2)=O)CCC2(CC1)CC2CNC(=O)Cn1ccnn1 6267,C1(c2nnnn2CCNCCCC(=O)OC)(NCCC)CCN(C=O)CC1 6268,N1(C(C2CC(NC(CCN(C)CC)=O)C2)=O)CCC(N(C)C(C)=O)CC1 6269,CC(F)(F)CCC(=O)NC1CC2(C1)CC2C(=O)NC(C(=O)OC(C)(C)C)C1CC1 6270,C1(NC(C(CC)(C)OC)=O)C2CC3C1C3C2C(=O)OC.N12CC(C)(C1)CC2=O 6271,C(=O)(CCS(C)(=O)=O)NC(C(=O)NCCC=C=C)C1CCOC1 6272,N1(C(C(C)=C2CCC2)=O)CCN(C(=O)C(=O)NC2CC2)CC1c1ccccc1Cl 6273,c1(C2C(C(=O)NC(CC)CNC(c3cnn(C(F)(F)F)c3)=O)C2)cccc(Br)c1 6274,C(C1=NOC2CNCC12)C(N1CCC(c2c(C#N)cccc2)C1)=O 6275,Cc1cccc(C(=O)OCC(C)(C)O)c1F.C1(C)C(=O)O1 6276,C1(CC)(NC(c2csc(C(C)(C)C)n2)=O)CCN(C(=O)C(C)(C2CC2)OC)CC1 6277,N1(C(C(C)C)=O)CCC2(CC1)CC2CNC(C1CCn2cncc2C1)=O 6278,C1(C(=O)OC)CC2(CC(NC(C3CCCC(C(=O)O)N3)=O)CCS2(=O)=O)C1 6279,c1(C(=O)NC(c2ccc(C)cc2)C2C3CNCC23)cnc2n1CCS2 6280,C1(C(=O)NCC(C)(C2CC2)NC(=O)C(=Cc2cn(C)cn2)F)(OC)CCSCC1 6281,N1(C(c2n(C)nc(C3CC3)c2)=O)CC2CC(C1)C2N=c1[nH]nc(C(N)=O)s1 6282,Cc1cn(CCN2CC3C(C2)N3C(c2ccnc(F)c2)=O)nc1C(F)(F)F 6283,C1(CNC(Cc2ccc(C)cc2)=O)CN(C(c2ncnc(O)c2F)=O)C(C)(C)C1 6284,C(=O)(C(C)(C)C(=O)NCC1CCN(C(=O)C(C)(C2CC2)OC)C1)OC 6285,C1(CC#N)CN(C(=O)CCc2cccc(Br)c2)CCN1C(=O)Cc1ccncc1 6286,CC1CCN(C(C2CCCN2CC(F)(F)F)=O)C(CNC(=O)COCCCF)C1 6287,c1(C(N(CCCN(C)C)CCNC(C(C=C)O)=O)=O)cc(OC)cnn1 6288,C1(N(C(c2cc(CC)no2)=O)CC2CC2)CCCN(C(c2n[nH]c(C)c2F)=O)C1 6289,C(CCN(C(=O)COC1(C)CCC1)C)(C(C)C)NC(CC1(OC)CCCC1)=O 6290,N1(c2n(C)c(N3CCCC3=O)nn2)CCCN(S(C)(=O)=O)CC1 6291,Cc1ccc(C(N2CCC(C(C)NC(C3CC(=O)NC3(C)C)=O)C2)=O)cc1CO 6292,CCCCC(F)C(=O)N(C1CCCCC1NC(c1cc(C)c(Br)o1)=O)CC 6293,C1(F)(CNC(c2c(C)nc(CC)s2)=O)COCCN(C(c2nonc2N)=O)C1 6294,C1(CS(Cc2cn(C)nn2)(=O)=O)CCC(F)(F)CC1 6295,c1(OC)cc(N2CC(Oc3cncnc3)CC2CNC(=O)COC)nc(CO)n1 6296,C(=O)(CC(C)(C)CC(F)F)N1C2CC(N(C)C(C3CC(O)C3)=O)CC1CC2 6297,C(C(C)(C)CC(=O)NCC1=CCN(C(=O)C(F)OC(F)(F)F)CC1)OC(C)=O 6298,C1(C(=O)NCCC2CCCCC2O)(OC)CCN(C(=O)C#CC2CC2)C1 6299,Cc1c(C(=O)NCC2C3CN(C(c4nccn4C)=O)CC23)ccn1C 6300,c1(C(=O)NCCCN(C(c2c(COC)cc[nH]2)=O)C)ccc2c(c1)NC(=O)CS2 6301,N1(C(C(C)OC(C)=O)=O)CCC(C)(CC(=O)NCC(C)CC2CCC2)C1 6302,N1(C(C=CCC)=O)CC(O)C(O)C1CNC(=O)CCc1cccs1 6303,CC1(C)COc2cc(Br)ccc2C1NC(c1cc(F)cc([N+](=O)[O-])c1N)=O 6304,c1(N(C)CC2CN(C(Cn3c(C)cnc3)=O)C2)ncnc(Cl)c1[N+](=O)[O-] 6305,C(CC(C)(C)C(=O)N1CC(C2(NC(c3ccncc3N)=O)CC2)C1)OC 6306,N1(C(C(F)=CC)=O)CC(NC(=O)Cn2cnc(Br)n2)CC(O)C1 6307,C(=O)(C(C)(C)CCC#N)N(C1CN(C(c2cn3ccsc3n2)=O)CC1O)C 6308,N1(C(CCc2ccc(SC)cc2)=O)CCCC(CO)(NC(=O)C(C)CF)C1 6309,CCCCCC(F)C(=O)NCC1CN(C(=O)COC2CC(F)(F)C2)CC12CCC2 6310,N1(C(C(N2CCC(O)CC2)C)=O)CCN(C(c2ccncc2O)=O)CC1C1CC1CF 6311,C1(O)(CNC(Cc2cc(C)[nH]n2)=O)CCN(C(C2CC2c2ccccc2)=O)CC1 6312,C1(NC(CC(C)(C)SC)=O)CC2CCC(C1)N2C(=O)Cc1ccc(C(C)C)cc1 6313,C1(CNC(c2cn(-c3ccccc3)nn2)C)CCCN(CC#N)C1 6314,c1(C(=O)NCCN(C(c2c(OC)n[nH]c2)=O)CC)cn2cc(C)sc2n1 6315,c1(C(N(CCCN(C(=O)CCc2ccccn2)C)C)=O)cc(F)c(F)c(N)c1Cl 6316,N1(C(c2c(C(C)C)noc2)=O)CC2(CCN(C(=O)CNC(c3cccs3)=O)C2)C1 6317,N1(C(=O)Nc2ccc(OC(C)C)cn2)CC2(CC2)c2ccc(Br)cc21 6318,N1(C(=O)NC2C(OCC)CC2)CCC(F)(CNC(=O)C(F)(F)C(F)F)CC1 6319,c1(NC23C(CN(C(C(CCC)NC(N)=O)=O)C2)CCC3)nc2ccc(F)cc2o1 6320,C1(NC(=O)CN(C(=O)CCC2OCCO2)C2CCC2)CCC2CC12 6321,C1(NC(C2CCN2C(c2cnco2)=O)=O)CCNC(=O)CC1 6322,CN1CCc2ccc(C(N3CCOCC(CNC(=O)CCOCCO)C3)=O)cc21 6323,c1(C(N2CCN(C(CC)=O)CC2CC#N)=O)cn(CC)c2ccc(OC)cc2c1=O 6324,Cc1ncnc(C)c1C(=O)NC1C(C(=O)NCCc2cnn[nH]2)C1(C)C 6325,c1(CN2CC(C(=O)Nc3c(I)ccc(OC)c3)C2)ccc2cccc(Br)c2n1 6326,c1(C(N(CC(CN(C(CSCCCC)=O)C)O)C)=O)oc(C2CC2)nc1C 6327,CC1CCC=C1C(=O)NC1(C(=O)NC(C)(CO)C2CCC2)CCSC1 6328,CC1CN(C(c2ncc(F)cn2)=O)CC1NC(=O)Cc1cc(C2CC2)no1 6329,c1(NC(C)=O)ccc(C(=O)NCCC(C)(C)NC(=O)CC(C)(C)O)c(F)c1 6330,Cc1cc(-c2cn(CC(F)(F)CNC(=O)CCc3cn(C)nn3)nn2)ccc1F 6331,Cc1cc(OCC(O)CN(C)CCNC(c2csc(S)n2)=O)no1 6332,N1(C(C2(C=C)CCN(C(=O)CCc3cnn[nH]3)C2)=O)C2CCCC1CC(O)C2 6333,C1(C(C)NC(C(F)=C(C)C)=O)CCN(C(c2coc(CO)c2)=O)CC1 6334,C1(NC(C2CCC(=O)N2)=O)CCN(C(=O)CC2CC(=O)C2)C12CCCC2 6335,N1(c2cc(C(C)=O)ncn2)CC2(CCCC2NC(=O)Cc2ccc(C(F)F)cc2)C1 6336,CCCCC(C)CCC=O.C1(=O)CC(C)(N)C1.C(C)(C)(C)N 6337,C1(CNC(CCOCCCNC(COCC#C)=O)=O)(OC)CCOC1 6338,c1(CCOC)cc(C2CC2)no1.C1(=O)C(=O)NC(C)C(C)CN1C 6339,c1(C(N2CCC(C)(CNC(C3C(C)(C)CO3)=O)CC2)=O)ccccc1N=[N+]=[N-] 6340,N1(C(C2C(OCC)C2)=O)CCC(F)C(NC(c2sc(C(C)OCC)nc2C)=O)C1 6341,C=CC(O)(C(=O)NC1CCN(C(=O)Cc2csc(Cl)n2)CC1O)C(F)(F)F 6342,N1(C(CC2(C)N(C(Cc3c(C)ncs3)=O)CC2)=O)CCC2CCCC12 6343,N1(C(C(CC)(F)F)=O)CCCC(C)(CNC(c2ccc(Br)c(OC)c2)=O)C1 6344,c1(C(=O)NC2CN(C(C3C(C)CC(=O)CC3)=O)CC2C)ccc2cnccc2n1 6345,CC(CCCCNC(=O)C(N1CCCCCC1)C)NC(=O)CC1CCCC(=O)C1 6346,C1(OC)(CNC(C2COCCC2C)=O)CCN(C(c2cnc(=N)[nH]c2)=O)CC1 6347,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CCN(C(C=CC=CCOC)=O)CC1CO 6348,c1(OC)cc(-c2cn(CNC3CC4(C3)CC(F)C4)nn2)cc(F)c1Br 6349,C12(C(=O)NC(CC)(CNC(c3cc(C#N)c[nH]3)=O)CC)CC(C)(C1)OC2C 6350,N1(C(C2(CC=C)CCCC2)=O)CCC2(CC1)CC(NC(c1cc(O)ncn1)=O)C2 6351,Cn1ncc(NC(=O)COC2CCN(C(C3CCC(=O)CC3)=O)C2)c1Cl 6352,C(CCC(C)C)(C(=O)NCC12CC(CCO1)C2)NC(c1cccc(CC)n1)=O 6353,c1(C(=O)NC(C)CCN(C)C(c2scnc2C2CCCC2)=O)ccnc(O)c1 6354,c1(NC(C)=O)ccc(C(=O)NC2(CCCNC(=O)CCc3c[nH]c(=N)[nH]3)CC2)nc1 6355,CS(=O)(=O)C1(C(=O)NCCN2CCC(NC(=O)CC3C=CCCC3)CC2)CCC1 6356,CCCCC(CNC(=O)Cc1cncn1C)NC(=O)CC(C)N(C)C 6357,Cc1ncc(C(N2CC3CC(C2)C3NC(=O)CCC2CC2C)=O)c(=N)[nH]1 6358,C1(C(C)C)CC=C(C(C(=O)NC2(C)CC2)N2CCC(c3cnn[nH]3)C2)CC1 6359,N1(C(C(CC)OC)=O)CCC(NC(=O)CCc2cncc(F)c2)C(C(N)=O)C1 6360,N1(C(CC(CC)NC(=O)C(C)CCSC)=O)CCC(CO)(CC)CC1 6361,c1(C(N2C(CNC(C(C)NC(=O)C(C)(C)C)=O)CC2)=O)c(Br)ccc(F)c1C 6362,CC1SCCCC1C(N1CC(NC(=O)CCc2ccn(C)c2)CC1CO)=O 6363,C#CC1(F)CN(C(=O)CN(C(=O)C(C)OC2CC2)C)C1 6364,C1(CNC(=O)C2=CCCC2)CN(C(=O)C2=CSCCO2)CCCO1 6365,C(=O)(CCC(C)(C)C)N1C(C)CC(CNC(Cc2ccc(C)cc2)=O)C1 6366,Cc1cnoc1C(=O)NCC(C)(O)CNC(=O)Cc1[nH]cnc1C 6367,C1(C(=O)NC2CCCCN(C(C(C(CC)O)C)=O)C2)CCc2nccn2C1 6368,c1(C(C(=O)NCC)N(C2(C#N)CC(C)(C)C2)CC(=O)OC)cccc(OC)c1Cl 6369,C1(F)(CNC(CCC=CCC=C)=O)CCCN(C(=O)C(C)(C)CF)C1 6370,C1(NC(C=C(CC)CC)=O)CN(C(C2CC2c2ncc(C)[nH]2)=O)C2CCCC12 6371,C1(NC(CNC(CCCC=C)=O)=O)CCCCC1NC(=O)CCc1ccncc1 6372,C(=O)(C(C)(C)CC(F)F)NCC(C(C)C)NC(c1c(Br)cn(CC)n1)=O 6373,c1(CCNC(c2c(Br)cc(C)c(C)n2)=O)ccc2c(n1)OCCO2 6374,C1(C(=O)NCC(C)(C2CC2)NC(CCOc2cccc(C)c2)=O)CCCCN1N=O 6375,C1(CNC(C(Br)=C(C)C)=O)CN(C(C2CC2c2cncn2C)=O)CCCO1 6376,c1(CC(=O)NCC2N(C(C(C3CCCCC3)C)=O)CCC2)ccc2nc[nH]c2c1 6377,C(CCN=c1nc2c(ncn2C(C)C)c(NCc2cnco2)[nH]1)SC 6378,C(=O)(C(C)(C)Cc1ccc(O)cc1)NCCN(CC(C)O)C(c1n(CC)nnc1)=O 6379,Cc1cc(C(N2CCCCC2CCNC(c2cc(C(C)C)n(C)n2)=O)=O)sc1Cl 6380,O=C(N=c1[nH][nH]c2c1CN(C(c1cc(F)cc(Cl)c1Cl)=O)C2)c1cnnc(Cl)c1 6381,N#CC1=C(C(=O)N2CCCC(CCNC(C34CCC(CC3(F)F)C4)=O)C2)CCC1 6382,C(C(O)CCCCC)NC(CC1(NC(CCC=C=C)=O)CC1)=O 6383,N1(C(C2OCCN(CC)C2)=O)CC2CC3CC2C1C3NC(c1cc(Cl)cnn1)=O 6384,Cc1[nH]c(C#N)cc1C(=O)NCCCCCN(C(=O)COCc1nc[nH]n1)C 6385,C(=O)(C(C)C(C)NC(c1cc(C)no1)=O)N(C(C#C)C)C1CC1 6386,C1(C(N2CC(O)(C(C)NC(C3CCCC34CC4)=O)C2)=O)CCC2(CCCC2)CC1 6387,CC(CC(=O)NCCc1ocnc1CNC(=O)C#CC1CCOC1)C(C)(C)C 6388,S(=O)(=O)(c1cc2sc(=NCc3cc4n(n3)CCCO4)[nH]c2cc1Cl)NCCCC 6389,N1(C(c2cc(C)nnc2)=O)CCCCCCC1C(N1CCCC(O)(C(C)C)C1)=O 6390,C=CC1OCCCC1C(=O)NCCCN(C(C1CC=C(C)CC1)=O)CC 6391,C(=O)(CS(=O)(=O)CC(=O)N(C)CCNC(C1CCCC2(CCC2)C1)=O)OC 6392,N1(C(c2c(OC)ccs2)=O)CCCC(C2CCN(C(=O)Cc3nnc(C)o3)C2)C1 6393,C1(CNC(CCC(=C)Br)=O)C(C)CCCN1C(=O)Cc1ccc(F)cc1 6394,C1(NC(C(Cc2cn(C)nc2)O)=O)CCCN(C(=O)CC(F)(F)Cl)C1 6395,C1(C)(C(=O)NCC(c2ccc(O)cc2)OC)COCCO1 6396,C(CCS(C)(=O)=O)(C(=O)N(C)CC1CCCN(C(=O)COCCC(C)C)C1)OC 6397,CC(CN=c1cc[nH]cc1S(=O)(=O)NCC1CCCC12CCC2)S(N)(=O)=O 6398,c1(C(C2CCCCC2CCC(F)(F)F)Nc2n(C)nnn2)cc(CC)ccc1F 6399,CC1=CCN(C(=O)C(c2ccco2)NC(=O)C(C2CCCCC2)=O)CC1 6400,N1(c2ccnc(SC)n2)CCC=C(C(=O)NCc2ccc(C(=O)O)c(Cl)c2)C1 6401,C(CC(C(=O)NCCCCOC(C)=O)NC(=O)C(CC)N(C)C)=CC 6402,C1(NC(CCCC#C)=O)CN(C(=O)C(CC)CCC)CCC1F 6403,N1(OCC)CCC2(C1)C(=O)NC(=O)N2C.N1(C(C)C)CC2(CC(CC)C2)C1 6404,c1(OC)ccc(C(=O)NCC(C2(O)CN(C(C3CCC4CC34)=O)C2)(C)C)c(C)c1 6405,C(=O)(CC(C)(C)N(C)C(C1(CO)CCCC1)=O)NC(C)CC1CC1 6406,c1(C(=O)NC2C(N(C)C(=O)OC(C)(C)C)CCCC2)cc(Cl)c(F)cc1O 6407,c1(CN(C)C(=O)OC(C)(C)C)csc(I)c1.c12cn(nn1)C1COCC1N2 6408,Cc1ccc(F)c(C(=O)NCC2CN(C(=O)C#CC3CCC3)CC2C)c1F 6409,CC#CCCCC(=O)N1CCOCC1CN(C(=O)C(C)c1ncco1)C 6410,C(C(CC1CC1)C(=O)NCc1ccncn1)NC(C1(C)CC(=O)C1)=O 6411,N1(C(c2c(O)cc(C)nn2)=O)CC(NC(=O)CCc2ncc[nH]2)CC12CCCC2 6412,c1(C(=O)NCCCCCNC(CSc2n(C)cnn2)=O)cc(C#N)n(C)n1 6413,C(=O)(C(O)C(F)(F)F)NCC1(NC(C2CCN(C3CCN(C)CC3)CC2)=O)CC1 6414,N1(C(c2ccc(OC)cc2I)=O)CC2OCCN(C(=O)Cc3cc(C)on3)C2C1 6415,C(=O)(C(C)C(O)CC)OC(CC(=O)OCC)CC(F)(F)F 6416,n1(CC=C)cc(C(N2CCC(NC(C3(C)COC3)=O)C2)=O)cn1 6417,C(=O)(CC1COCc2ccccc21)NCCN(C(Cc1ccc(C)s1)=O)C1CC1 6418,C#Cc1ccc(F)c(C(=O)N(CC)CC2CCCN2C(C2CC(F)C2)=O)c1 6419,C1(NC(Cc2ccc(C)s2)=O)CC2(NC(=O)CCC3(C)CC3)COC1C2 6420,C1(C)(CNC(CCC=C=C)=O)CCN(C(=O)CCC2CCCC(O)C2)CC1 6421,c1(C(=O)Nc2nc(C)nc(O)c2)cnc2n1CCN(C(C1CCCS1)=O)C2 6422,c1(C(C)(C)C)cccc(CNC(C2CC(F)CN2C(C2CNC(=O)O2)=O)=O)c1 6423,N1(C(CC)=O)CCN(C(C2OCCOC2C)=O)C2CC12 6424,C1(C(=O)NCC2(C)N(C(C(C)=C(C)C)=O)CCC2)CC2(C1)CC(C)(C)C2 6425,CN1CCOc2c(C(N3CC(CNC(C4(C)COC4)=O)CC3(C)C)=O)cccc21 6426,c1(OCC(=O)NCC(CNC(CS(=O)(=O)NC)=O)C)cccc2c1OC(C)(C)C2 6427,c1(N(CCSC(C)(C)C)CCO)cc(N2CCOC(CCO)C2)ncn1 6428,c1(C(=O)NCCC=C)cn2cc(-c3c[nH]nc3C#N)ccc2n1 6429,CC1CC(C(=O)NCc2cc(C(=O)N(C)CC3(N(C)C)CCC3)ccn2)CN1C 6430,N1(C(CC2(NC(C3CC3)OC)CCOCC2)=O)CCC2CN(C(=O)CC)C2C1 6431,N1(C(CCCC=C)=O)CCC(C)C(NC(c2ccc(O)c(C(N)=O)c2)=O)C1 6432,C12(C(=O)NC3C(C)CN(C(=O)C=Cc4ncco4)C3)CCCN1S(=O)(=O)CC2 6433,c1(C(=O)N)cc2ccccn2c1.N1(C(C2(CO)CC2)=O)CCSCC1C1CC1 6434,C1(C(=O)NC2CC(C(C)NC(c3c(CC)nccn3)=O)C2)CC2(CCC2OC)C1 6435,c1(C(=O)NCC(=O)N(c2cccc(Cl)c2Cl)CCOC)cnn2cccc(Cl)c12 6436,Cc1cn2c(C(N3CC(N(C(=O)CC(C)C4CC4)C)C3)=O)c(Cl)nc2s1 6437,c1(C(C)C)noc(CNC(c2nnnn2C2CC2)C2(C)COC2)n1 6438,C1(OC)CN(C(=O)C(C)(C)N(C)C)CC1NC(=O)CC(C)Cc1cccc(F)c1 6439,C(=O)(CCCCCc1cccs1)NCCC(C)(C)NC(C1C(C)C1C)=O 6440,CCCCCC(O)CC(=O)NCCCC(CCC)NC(c1ccc(Cl)nc1N)=O 6441,C1(C(=O)NC(CCC)(C)C)CCN(C(=O)C(CCOC)OC)CC1OC 6442,C(CCC(C)C(=O)NC1(C(C)C)CCC1)OC.C12(CC1)CCCNC2=O 6443,N#Cc1cc(S(=O)(=O)N(C2CCCC23CCNCC3)c2cc[nH]n2)ccc1Br 6444,C(=O)(C1=CC2CCC1C2)N1CCCC(NC(C=Cc2cccc(C)c2)=O)(CO)C1 6445,C12(C(=O)NCC(CC)NC(=O)CCN3CCCS3(=O)=O)CCCC(CO1)C2 6446,Cc1cc(N)c(C(=O)N(C2CN(C(C3CCN3C)=O)CC23CC3)C)cc1C 6447,c1(C(=O)NC2C(NC(c3cncnc3)=O)CCC2)ccc(F)c2occc12 6448,c1(C(=O)Nc2ccc(SC)c(F)c2)nsc2ccc(C)cc12 6449,CC1CCCC(C)N(C(C23CC2CN(C(=O)CN2CC=CC2)C3)=O)C1 6450,C1(CNC(C(CSC)OC)=O)COCC(=O)NCC12CC(CO)C2 6451,C(=O)(C(O)C(C)(C)C)NC1(CNC(c2nccc(CC)c2)=O)CCCC1 6452,c1(C(C)C)nnc2cc(N3CCCC3C3(NC(=O)C(C)O)CCC3)ncn12 6453,N1(C(CN2C(C)CCC2)=O)CCOC2(CCN(C(=O)CC3CNC(=O)C3)CC2)C1 6454,N1(C(C2N(C(CC=CC=C)=O)CCCC2)=O)CCOC(C(=C)C)C1 6455,Clc1ccc2[nH]c(=NCc3cncnc3)[nH]c(=NCC3CC(=C4CC4)C3)c2c1 6456,CON(CCC(=O)N1C2CCC1CC(O)C2)C(=O)C(C)(C)CO 6457,Cc1cc(C#N)sc1C(=O)NCC1CC(NC(=O)CCc2csnn2)C(O)C1 6458,C1(NC(C(C2CC2)OC)=O)CCC(N(C(=O)C(CC#N)c2ccccc2)C)CC1 6459,C1(NC(CCNC(C)=O)=O)CCS(=O)(=O)C12CN(C(C1(C)CC=CCC1)=O)C2 6460,C(=O)(CCC(C)(F)F)NC(C(=O)NC1CC(=C)C1)CC1CC1 6461,C1(CNC(C(COC)C)=O)CC(N=c2[nH]c(C(=O)OC)nc3c2CCC3)C1 6462,c1(CNC2(c3nnnn3CC3(C)CCOC3)CCC(=C)CC2)c(Cl)cc(Cl)cc1Cl 6463,C1(CC=C)CCN(C(=O)C(CNC(=O)Cn2nccc2C)OC)C1 6464,C1(F)(C(N2C(C(=O)NCC3OCC(=O)NC3)CC3CC32)=O)CCCCC1(F)F 6465,C1(CC)CN(C(=O)C(C)n2cncn2)CC1NC(=O)CSC1CC1 6466,Cc1oc(C#N)cc1C(N1CCC(CNC(=O)C(F)(F)CO)CC1C1CC1)=O 6467,c1(OC)ccnc(C(N2CCC(NC(c3cccc(F)c3F)=O)C(C)C2)=O)c1N 6468,c1(C(N2CC(O)(CNC(c3c(CC)[nH]c(=N)s3)=O)C2)=O)cscc1S(C)(=O)=O 6469,C(CNC(=O)CN1CSCC1=O)(C(C)C(C)C)NC(C(C)=CC)=O 6470,C12(NC(c3c(C)nn(C(C)C)c3C)=O)CCCC1CN(C(=O)C(C)(C)CO)C2 6471,C1(C(N(CCCNC(=O)CCc2ncnn2C)CC)=O)CCc2ncccc2C1 6472,N1(C(c2c(C(C)C)occ2)=O)CCC(C)C1CNC(c1nccnc1Cl)=O 6473,c1(NCC)c(NC(=O)C(N)Cc2cc(OC)cc(C)n2)cc(Cl)cc1Br 6474,C=CCC(C)(C)C(=O)NCC(O)CN(C)C(c1nccnc1N)=O 6475,N1(C(c2cc(C)sc2C)=O)CC2CCC1(CNC(c1n[nH]cc1C)=O)CC2 6476,N1(C(c2cc(C)nn2C)=O)CCOC2CN(C(c3conc3C(C)(C)C)=O)CC12 6477,c1(CNC(C)CC2CN(C(=O)COc3cccnc3)C2)ccnc2ccnn12 6478,c1(CN2C(C(N3CCOC(CO)C3)=O)CCC2)cnc2ncccn12 6479,c1(SCC(=O)N(CCN(CC(C)O)C(C2CCC2C)=O)CC)nc2ccccc2[nH]1 6480,CCC(C)C(CC(=O)N(CC(C)(C)O)C)NC(c1cccc2ccnn12)=O 6481,c1(CC(=O)NC(CCOC)CNC(c2ncccc2F)=O)ccccc1[N+](=O)[O-] 6482,N1(C(C2=CC(C)(C)C2)=O)CC2CCCN(C(=O)Cc3cccc4c3CCC4)C2C1 6483,Cc1noc(C)c1CCNC(=O)CC1(C)CCN1C(C1CC1C(F)(F)F)=O 6484,c1(C(=O)NCC2N(C(C3CC(C)N(C)CC3)=O)CC3CC32)ccc2cccnn12 6485,C(C)(C)(C(=O)NCC(F)CNC(=O)Cc1coc(C(F)F)n1)OC(C)=O 6486,N1(C(C(C)C)C(=O)NCC2CCCO2)CCCCCC(N)C1 6487,c1(C(N(CC)CC2CCC2)=O)ccc(NC(CC)CC)cn1.C1(=O)CCCN1 6488,c1(N(CCCCc2cccnc2)C)nnc(C(=O)O)cc1N 6489,c1(C(=O)NCC2N(C(C(C=CCCC)O)=O)CCC2)cccc2ccc(O)nc12 6490,c1(C(=O)NCC(C)(O)CNC(=O)CSC2CC2)ccc2cc[nH]c2n1 6491,c1(C2N(C(Cn3c(C#C)cc(C4CC4)n3)=O)CCC2)sc2c(c1F)CCC2 6492,C(CCCCn1cc(CC2CCCOC2)nn1)NC(C1(C2CCCO2)CC1)=O 6493,C(=O)(C=C1SCC(=O)N1C)N1CC(OCC)C(NC(=O)C(C)CN(C)C)C1 6494,N1(C(COCCCCC)=O)CC(C)CN(C(=O)Cn2cnc(Br)c2)CC1C 6495,CCCC(CCC)=CC(=O)NC1CC(NC(=O)CCCn2cccn2)C(O)C1 6496,C12(C#N)CN(C1)C2=O.c1(CCC)ccc(C(N2CC(NC(=O)CC)C2)=O)[nH]1 6497,c12cc3c(cc(OC)cc3o1)C2.c1(CCCC)cnc(C(=O)NOCC)s1 6498,N1(C(CC(=O)OC)=O)CCC2(CCCC2CNC(=O)Cc2csc(C)c2)CC1 6499,c1(C(N2C(CNC(C3N(S(C)(=O)=O)CC3)=O)CC2)=O)coc2c(F)cc(F)cc12 6500,c1(C(N2CC(CCC(=O)NC(C3CC3CO)C)C2)=O)ccc(C2CC2)nc1 6501,C1(CNC(C(C)NC(c2ccoc2)=O)=O)C2CC1N(C(=O)C=CC1CC1)C2 6502,C1(C(N(CC(C)(C)CNC(=O)Cn2ncnn2)C)=O)CC12CCS(=O)(=O)CC2 6503,CC1CC(C(=O)NC2(CNC(=O)C(C)(C)c3cnc[nH]3)CCCC2)CC(=O)N1 6504,C1(C(C(C)NC(c2ocnc2C)=O)NC(CSC)=O)CCCCC1 6505,C12(NC(CCCCC)=O)CCCC1N(C(=O)COC1CCOC1)CCC2 6506,C(C(=O)NC1CN(C(c2cc(O)nn2C)=O)CC1C(F)(F)F)(C(C)C)SCC 6507,N1(C(CCc2ccc(C(=O)OC)o2)=O)CCC(NC(C2CCCO2)=O)CC1C 6508,C12(C(N3C(C)CCCC3)=O)CC(C3CCCCC3)(C1)C2 6509,N1(C(c2ccc(F)cc2Br)C(=O)NCCOC)CCOC2(CCSC2)CC1 6510,c1(C(=O)NCC2(CNC(C(CSC)OC)=O)CC2(F)F)ncccc1O 6511,Cc1cc(C(=O)N(C)CCN(C(=O)CC(C)N(C)C)C2CC2)ccc1N1CCOCC1 6512,c1(C(=O)NC(CC)CO)ccc(=NCc2cc(F)ccc2Br)[nH]c1 6513,Cc1cccc2c(C(=O)NC3CCC(N(C(=O)Cn4cnc(=N)[nH]4)C)C3)coc12 6514,N1(CC(N2CCC(OC(C)C)C2)=O)CC2(CCC(N(C)Cc3cc[nH]n3)CC2)C1 6515,Cc1cnc(C(=O)NC(C)CCN(C)C(C2CC2(C)C(C)C)=O)c(Br)c1 6516,Cc1ccc(C)c(C(N2CCCC(C)(NC(=O)C=Cc3cnn(C)c3)C2)=O)c1 6517,C1(O)(CNC(CN(C(C)=O)C)=O)CCCN(C(C2(n3nccn3)CC2)=O)C1 6518,N1(CCN(C(C2(OC)CCCC2)=O)C)CCN(C(=O)CCS(C)=O)CC1 6519,c1(C(=O)NC(C(C)NC(c2c(C)oc(C)c2C)=O)C)ccc2c(c1)COC2 6520,C1(CCC)CN(C(c2cc(C)n(CC)n2)=O)CCN1C(=O)Cc1nocc1C 6521,c1(C(=O)NC2C(CNC(c3cc(CC)oc3C)=O)CCCC2)ncc(Cl)cc1Cl 6522,c1(N2CCC(NC(c3ccc([N+](=O)[O-])cc3)=O)C2)ncnc2ccc(I)cc12 6523,C(=O)(C(CC(F)F)N(C)C(c1ccnc(C)n1)=O)NCc1nc(CC)on1 6524,O=C(C1=NOC2(CCC2)C1)NCC1(C(N2CCC(CCO)C2)=O)CCOC1 6525,C1(C(N2CC(C3(NC(c4c[nH]nc4C(F)F)=O)CC3)C2)=O)CCC2CCC(=O)N12 6526,C1(O)(C(=O)NCC2CC(CC3CC3)CO2)COCCC1O 6527,C12(COC)CC(CNC(=O)C(C)CC(N)=O)(CN1C(c1n[nH]c(C)c1O)=O)C2 6528,c1(C(=O)NC2CC(O)(CNC(C(C)(C)CC3CC3)=O)C2)cccc2c1OCC2 6529,N1(C(=O)CCN(C(C23CCCC2C3)=O)C2CC2)CCCC(CCCO)C1 6530,Cc1csc(CCCC(=O)NCCC2CCN(C(=O)CC34CCCC3C4)C2)n1 6531,C(CC(O)C(=O)N(CCCO)CCN1CCC1)NC(C(C)(F)F)=O 6532,C1(CNC(c2c(C)cn(C)c2)=O)CC2(CC2)CN1C(c1cc(F)n(C)n1)=O 6533,N1(C(C2N(C=O)CCC2)=O)CCC2(C1)CN(C(c1ccnn1CCF)=O)C2 6534,C12(C(N3CCC(C)(CCNC(c4nnc(C)s4)=O)CC3)=O)CCC(CC1)C(C)O2 6535,N1(C(c2[nH]c(=NCC)sc2)=O)CCC(NC(=O)C(C)Sc2nncn2C)C(F)C1 6536,c1(OC)cc(C(=O)NC2CN(C(=O)Cc3cc[nH]n3)CC2(C)C)c2ccccc2c1 6537,C1(CN)CN(C(C2(CCOC)CCCC2)=O)CC1C.C1(C(=O)N)CN(C2CCC2)C1 6538,CC1(NC(C2CC2(F)Cl)=O)CN(C(=O)CCCNC(=O)OC(C)(C)C)C1 6539,CC1(C)COc2c(NC(N3CC[Si](C)(C)C3)=O)cnn2C1 6540,C(=O)(C1=CCCCC1C)NC1C(C(=O)NC(C)Cc2ncn(C)n2)C1(C)C 6541,N1(C(c2c(CC)ccc(C)c2)=O)CCC2(COC(CNC(=O)C3=CCCC3)C2)C1 6542,CCCCC(F)C(=O)NC(c1ccccc1)C(=O)NC(C)C(=O)NCC 6543,C1(c2n(CCCC)nnn2)(NC(C)CCC2CC2)CCC(CCOC)CC1 6544,Cc1ccc(C(=O)NC(C)C(C2CCCCC2)NC(c2cc(CO)[nH]n2)=O)nc1 6545,c1(CNC(=O)NCC2CS(=N)(=O)C2)ccc(S(N)(=O)=O)cc1 6546,C1(C(N(C2CC2)CC2N(C(c3c(CC)non3)=O)CCC2)=O)CCS(=O)CC1 6547,CC1(C(F)F)CN(C(=O)C(c2ccc(F)cc2)=O)CCO1 6548,C(CC(C)(C)C)(C(=O)N1CCCCC1CCCNC(c1cc(C)oc1C)=O)OC 6549,C(=O)(CC(C)(C)CNC(C1(C(N)=O)CCCCCC1)c1nnnn1C)OC 6550,c1(CC)cccc(Cl)c1C(=O)NCC1CCC(CNC(C2CC2(C)CC)=O)CC1 6551,CCCC(C)(C)CC(=O)N1CC2OCC(NC(=O)C(C)(C)CN3CCOCC3)C2C1 6552,c1(C(N(C2C(N(C(C(C)=C(C)C)=O)C)CCCC2)C)=O)n[nH]c2ccc(O)cc12 6553,CCC(C(=O)N1CCCCC1CCCNC(=O)CNS(C)(=O)=O)C(F)(F)F 6554,Cc1cc(C(=O)NCC2CC(C)CN(C(=O)CCOCC3CCC3)C2)ccc1F 6555,CCCCCC(CC)C(=O)NC1CN(C(c2ccc(N)c(SC)c2)=O)CCC1C 6556,c1(OC)ccc(C(=O)NCC2(F)CN(C(=O)C(F)C3CCOC3)C2)c(F)c1 6557,c1(C(N2C(CN(C(=O)CCC3CCOC3)C)CCC2)=O)cc2cccn2cn1 6558,C(C)(C(F)(F)C(F)(F)F)=CC(=O)NC(CC=C)CNC(C1COCCN1C)=O 6559,C1(C)(CNC(c2cnc(OC)s2)=O)CCC(NC(=O)C(C)(CO)NC(C)=O)CC1 6560,CC1(C)OC(C)(C)C1C(=O)NCC1CN(C(C2CC=CCO2)=O)CC1(F)F 6561,c1(NC2(NC(=O)COc3cccnc3)CC2)ncc(Br)c(O)n1 6562,N1(C(=O)Cn2nccn2)CC2CCCC(Nc3ncncc3I)C2C1 6563,C#CCCCCCCCC(=O)NCC1C2CN(C(C3(CCC)CC3)=O)CC12 6564,c1(C(=O)NC23CC(C(N4CC(O)C(O)C4)=O)(C2)C3)nc(F)ccc1Br 6565,N1(C(=O)Nc2cc(C)cc(C)c2)CCC(C)(Nc2ccnc(CO)n2)C(O)C1 6566,C#CCCCCCC(=O)N1CCCC1(CC=C)C(=O)N(C1CC1)CC1CCOC1 6567,CC(CCC(C)(C)C)C(=O)N(C1CCCN(C(=O)CS(=O)(=O)C2CC2)C1)C 6568,c1(C(N2C(Cn3cc(C(C)N(C)C)nn3)CC2)=O)ccc(F)cc1C(F)F 6569,N1(C(C)=O)CCC(N)C1.C1(C(=O)N)CCS1(=O)=O.N12CC(C1)OCC2=O 6570,Cc1n[nH]cc1CC(=O)NC1CN(C(=O)CC2(CC(=O)NC3CC3)CCCC2)C1 6571,c1(CNC(c2n(C(C)(C)C)nnn2)c2ccns2)ccnc(SC2CCC=CO2)c1 6572,CCCC(C)(C)C(=O)NC(CNC(=O)C#CC(C)(C)C)CCCC 6573,N1(C(C=CCC(C)(C)NC(C(CCOC)OC)=O)=O)CC2(CC(OC)CO2)C1 6574,CC1CN(C(C2C=CC=CC=C2)=O)CCCN1C(c1cc(O)nc(Cl)c1)=O 6575,C1(CC(N2C(CNC(C3(F)CCOC3)=O)CCC2)=O)CCCOCC1 6576,N1(C(c2cccc(OC)n2)=O)CC(O)C(O)C1CNC(c1cnc(OC)s1)=O 6577,c1(-c2cn(CC(C)NC(CSCCC)=O)nn2)ccnc(C(F)(F)F)c1 6578,C(=O)(CCCCC(C)(C)C)N1CCC(NC(C(CCC(C)C)O)=O)C12CC2 6579,C1(CCOC)CN(C(=O)C(CO)OC)CCN1C(=O)CCN1CCCC1 6580,C1(C)(C(=O)NCC(CC)NC(c2cccc(COC)n2)=O)COc2ccccc2O1 6581,N1(C(CC2CC(OC)C2)=O)CCCN(C(C2C(C#N)C2(C)C)=O)C(C)C1 6582,Cc1nn(C(C)C)cc1C(N1CCC(O)(CN(C)C(C2COC(=O)N2C)=O)C1)=O 6583,c1(C(=O)NCCNC(C2(CC)CC2(F)F)=O)c(C(F)(F)F)nc2n1CCCC2 6584,c1(CCOC(c2c(C)occ2C(F)(F)F)=O)cccc(F)c1I 6585,C1(C(=O)NCC=CC(=O)NCCOCC)CCn2c(cnc2Br)C1 6586,c1(CCNC(C=C(COC)C)=O)cc(C(=O)NCCCS(C)=O)no1 6587,c1(CC)cc(OC)cc(OC)c1CN(C1CCC1)C=O.c1(CO)ccc(OC)c(O)c1 6588,c1(C(NOCC(C)C)=O)cc(CNC(C2C3CCCC23)=O)on1 6589,N1(C(C(C)N(C(C)=O)C)=O)CC(CNC(c2cn(C3COC3)nn2)=O)C(C)(C)C1 6590,N1(C(CSCCC)=O)CC(C2CN(C(c3sc(C(C)OC)nc3C)=O)C2)C1 6591,C(C(N=c1cc(CC2CCCCC2)n(C)[nH]1)c1nnnn1CCCC1CC1)OC 6592,c1(CN(CC(C)OC)C)cc(SC(c2nc(CO)no2)C)ccc1Br 6593,C1(CC(C)NC(c2ccc(Cl)cc2)=O)CC2CCC(C1)N2C(=O)C(O)C1CCC1 6594,c1(C(=O)NCCN(CC(C)O)C(C2CCC3(CC3)C2)=O)ccnnc1S 6595,N1(C(CC2(C(=C)F)CCC2)=O)CC2(CC2)CC1CC(=O)NCC(F)CO 6596,C12(C(=O)NCC(C)CNC(C3CC34CCCC4)=O)CC(CO)(C1)OC21COC1 6597,C1(NC(C2(C)COC2)=O)CCN(C(C23CCC(C2)OC3)=O)CC1F 6598,Cc1ccc(C(=O)NC(C)CNC(c2cc(C3CCC3)[nH]n2)=O)cc1S(N)(=O)=O 6599,C1(CC=C)(C(=O)NCC2NC(=O)NC2=O)CCCN1C(c1nscc1C)=O 6600,Cc1nc(-c2cnn(C)c2)oc1C(=O)N(C)CC1(NC(=O)CC2C=CCC2)CC1 6601,N1(C(=O)NCCC#N)CCN(C(=O)C(F)(F)F)CC1c1ccccc1Cl 6602,c1(N(CC(C)(C)CO)C)nc2cccnc2c(=NCCCSC(F)F)[nH]1 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6657,N1(C(C2(COCC)COC2)=O)CCN(C(=O)C(C)(O)C2CCC2)CC1C1CCC1 6658,C(C1CCN(C(=O)CC2CC(F)(F)C2)CC1)=CC(NCC=COCC)=O 6659,CCC(COC)C(=O)NCCCN(CCO)C(C1(c2cccs2)CC1)=O 6660,c1(CNC(C(C)NC=O)=O)cccc(-c2cn(Cc3cc(Br)c(Br)s3)nn2)c1 6661,c1(C(=O)NC(CC)CN(C)C(C2CCC(C)(C)O2)=O)cc2cnccc2o1 6662,C1(C)(C(N(C)CCNC(c2sccc2-c2ccccc2)=O)=O)CC2CC2C1 6663,C1(C(N2CC3C(CCNC(CC(C)F)=O)(CC3)C2)=O)CCC2(CC1)OCCO2 6664,N1(C(=O)NC)CCC(C(=O)NCCCCCNC(=O)C(C2CCCO2)OC)CC1 6665,Cc1cc(C(=O)NCCCCNC(=O)C(C(C)C)N(C)C)cc(C)c1N 6666,N1(C(CCCCOCC)=O)CCN(C(=O)CC2OCCOC2(C)C)C(C(C)C)C1 6667,c1(C(=O)NC2C(CCC)CN(C(=O)C(C)(C)C(N)=O)CC2)cc(C)c(F)cc1N 6668,C1(NC(C(C)=C2CCC2)=O)COC2(C1)CN(C(C1CC1c1ccnc(Cl)c1)=O)C2 6669,c1(C(N(CCN(C(=O)CC2CC2(Cl)Cl)C(C)C)C)=O)cc(Cl)ccn1 6670,c1(N2CCN(C(=O)NC(C3CC=CCC3)C(=O)O)CC2)cccc([N+](=O)[O-])c1 6671,Cc1c(C(N2CCC3(C2)CN(C(=O)C(CCO)N(C)C)C3)=O)nn2c1CCCC2 6672,C(=O)(C1Cc2ccccc21)N1CCC(N(C(=O)C(c2ccnn2C)O)CCC)C1 6673,C(C(C(=O)N1CCC1CC(=O)NCCCCCO)OC)OC 6674,c1(C(=O)NC2CC2)ccnn1CCO.N12CCC(C1)CC2=O 6675,C12(CNC(c3cc(C)no3)=O)CN(C(C3CCS(=O)CC3)=O)CC1CCO2 6676,c1(C(=O)NC(C)C(C)C(=O)NCCCC(O)CO)nccc2[nH]ccc12 6677,N1(C(C(C2CCCCC2)C)=O)CC=CCC1C(N1CCC=C(F)C1)=O 6678,C(=O)(CCC(C(=O)N1CC(C)N(C(=O)CS(N)(=O)=O)CC1C)N(C)C)OC 6679,CC(C)(C)CCCC(=O)NCC1(Cn2cc(-c3ccncc3C(=O)O)nn2)CC1 6680,N1(C(C(CC2CCC2)NC(c2c[nH]nc2Cl)=O)=O)CC2CCCC2C1 6681,CN1CC(NC(=O)NCc2cc(Cl)c(Br)cn2)C(C)(C)C1 6682,N1(C(C(C(C)C)N=[N+]=[N-])=O)CCC(O)(C2(NC(c3cnnc(O)c3)=O)CC2)CC1 6683,c1(C(N2CCC(C)C2)=O)ccc(=NCc2cccc(O)c2O)[nH]c1 6684,c1(CC)c(C(=O)N(CCCN(C)C(C2COC(C)C2)=O)C)cccc1F 6685,C(CCC(=O)NCC(C)C(=O)NC1CC1c1cncs1)OC(C)C 6686,C1(NC(C(CC(=O)OCC)C)=O)CCN(C(C2CCC3(CC3)C2)=O)CC1F 6687,C1(CN)(NC(C2CCC2C(F)(F)F)=O)CCCCC1O 6688,N1(C(C(CCCCCC)(C)C)=O)CCCCC(C2CN(C(=O)C(C)C#N)C2)C1 6689,C(CN=c1[nH]nc(O)s1)N(C(c1ccc(CC)c(CC)c1)=O)C 6690,c1(C(N2C(CNC(C(CC)(C)F)=O)CC2)=O)ccc2cc(F)ccc2n1 6691,c1(C2C(C(N3CC(C#C)(C(N4C5COCC4C5)=O)C3)=O)C2)ccc(C)c(C)c1 6692,CCCCC(O)CC(=O)NC1CCN(C(c2cnc(C3CCOCC3)s2)=O)CC1 6693,C12(C(=O)NC(C)CN(C)C(C3CCS(=O)(=O)C3)=O)CCCN1S(=O)(=O)CC2 6694,C1(C(N(C2CCN(C(=O)Cc3cc(C)no3)C2)CC#C)=O)CC(C)(F)C1 6695,C1(C(N(C2CCCC2)CC(C)C)=O)CCCC(NC(=O)C(O)C(C)C)CC1 6696,C1(NC(c2cncc(C)c2)=O)CCC2CCN(C(=O)Cn3nnc(=N)[nH]3)C1C2 6697,C(CNC(=O)C(c1ccc(Cl)cc1)N)(CCS(C)(=O)=O)OC 6698,N1(C(CC2(C)CCC2)=O)Cc2ccccc2C(NC(C2CC2C2CC2)=O)C1 6699,C1(C(N(CCOCCN(C)C(c2ccnn2CC#N)=O)C)=O)CCCCC1(C)C 6700,C=C1Cn2c(C(N3CCC(F)(CNC(=O)CC(C)C(C)C)CC3)=O)nnc2S1 6701,N1(C(c2c(CC)ccs2)=O)C2CCC1(CNC(=O)C=CS(C)=O)CC2 6702,c1(C(N(C)CC2COCCN2C(=O)CC2CCCOC2)=O)nnc(O)cc1O 6703,N1(C(CN(C)C)=O)CC2COCC2(C(=O)NCCc2ccco2)C1 6704,C1(C(C)C)CN(C(=O)CC2CSC2)CCN1C(=O)CCc1cnc(O)[nH]1 6705,Cc1cn2cc(CC(N3CCC(NC(=O)COC(C)C)CC3C3CC3)=O)nc2s1 6706,N1(C(Cc2c(C)cc(C)s2)=O)CCCCC(NC(=O)CCCF)C1 6707,C(C(=O)N1CC(C)(C)C1C(=O)O)(C(C)(C)C)N(C)C(c1ccccc1F)=O 6708,N1(C(C=CCCC)=O)CCN(C(=O)Cc2ccsn2)C2CS(=O)(=O)CC12 6709,c1(C(=O)OCC)cccc2nc(CNC(C)C(F)(F)F)sc12 6710,N1(C(C(CC)C(=O)NCC)=O)CC(C)(C)CC1NC(=O)C=Cc1ccco1 6711,N1(C(c2nc(OCC)sn2)=O)CC2CCC1C(NC(C1(C(F)(F)F)CC1)=O)C2 6712,c1(OCC(N2C(CNC(c3c[nH]ccc3=O)=O)C=CC2)=O)cccc(Cl)c1 6713,n1(C2C(C)C2)ccc(=NC(=O)C(=O)Nc2cc([N+](=O)[O-])c(F)c(F)c2F)[nH]1 6714,C(=O)(C1=NNC(=O)C1)NCC1CN(C(CCc2cnn(C)n2)=O)C1 6715,c1(C(C)C)cc(C(=O)NC(C)(CNC(=O)C(C)n2ccnc2)CO)on1 6716,c1(CCCNC(CC2CC(NC(C(C)OC)=O)C2)=O)nnnn1C 6717,c1(Nc2cc(N3C(c4cccc(Br)c4)CC(C)C3)ncn2)cc2c(ncn2C)[nH]1 6718,Cc1[nH]nc2ccc(C(=O)NCC(C)CNC(=O)CCOC3CCOC3)c(Cl)c12 6719,C1(C(=O)NC2CCCN(C(c3cnn(C4CC4)c3)=O)C2)Cc2nncn2C1 6720,N1(C(c2cccc(F)c2)=O)CCCC(N=c2cc(Cl)c(O)n[nH]2)C1 6721,C(=O)(C(C)(F)C(C)(C)F)N1C2(CNC(COCCC(C)C)=O)CCC(C1)C2 6722,CC(C)CC(C(=O)NC1CC(C)N(C(=O)C=CC2CCOC2)C1)C(N)=O 6723,Cc1ccccc1C1(C(=O)NC(C)C(C)NC(=O)C(F)C2CC2)CC1 6724,Cc1ccc(F)c(NC(=O)C(N2CCC(c3cc[nH]c(=N)n3)CC2)=O)c1F 6725,CC(C#N)C(=O)NCC(C1CCCCC1)NC(C1C(C)C1C)=O 6726,CN1CCN(C(c2ccnn2CC(F)F)=O)CC1CNC(C12CCC(C1)OC2)=O 6727,C(C)(CCC(=O)NC(C12CC(C(=O)OC(C)=O)(C1)C2)(C)C)OC 6728,C1(CC(=O)Nc2nc(C(F)(F)F)cs2)CCCCN1 6729,C(C(=O)N1CCC(CNC(c2cncnc2C(C)(C)C)=O)C1)(C(C)C)NC(C)=O 6730,c1(N(c2ncnc(OC)c2C)C(c2ccccn2)=O)ccc2c(c1)CCNC2 6731,Cc1ccc(C(F)F)c(C(=O)NC2(CNC(C3(C)CC4CC4C3)=O)CCC2)c1 6732,CC(CCC(C)(C)C)C(=O)N1CC2CC1C2NC(=O)CNC(=O)CC(F)(F)F 6733,C12(C(N(CCN(C(CCc3cnc(C)o3)=O)C)C)=O)CC(C3COC3)(C1)C2 6734,C1(C(N2CCC(O)(CN(C)C(c3cc(Cl)c[nH]3)=O)C2)=O)(OC)CCS(=O)(=O)C1 6735,C1(C(N2CCCC(CCNC(C(CC)(C)C)=O)C2)=O)CCOC(C)(C)C1 6736,c1(SCCCC2CCC2)ccc(NC(C(=O)NCC2CCN(C)C2)=O)cc1 6737,C1(C(N(CCNC(c2c(C)oc(Br)c2)=O)C(C)C)=O)Cc2ccccc2CO1 6738,C1(CNC(C(C)=C2CC2)=O)CC(NC(c2cnn(CCC(F)(F)F)c2)=O)CC1O 6739,N1(C(C=CCN(C)CC)=O)CCC2(CCCN2C(c2cc(N)cc(F)c2)=O)C1 6740,c1(C(=O)NC2C(NC(C(C(C)C)SC)=O)CCCC2)c[nH]c(=O)c2ccnn12 6741,c1(N(C(C(=O)NCC(C)N(CC(C)N(C(C)=O)C)C)=O)C)ccccc1 6742,CCC(C)C(C(=O)N1CC(C(C)C)=NO1)N(C(=O)CC1CCC(C)CO1)C 6743,C(=O)(C1=CC2C=CC(C1)C2)NC1CCCC(NC(c2n(C)cc(Br)c2)=O)C1 6744,C(CC(=O)N1CC=CC1CNC(C1(OC)CCCC1)=O)(C(N)=O)NC(CC)=O 6745,C=CCCCCC(C(=O)NC(CC(C)C)C(=O)OC)N1CCCCC1CN(C)C 6746,Cc1ccc(OCCCC(=O)NCC2CN(C(c3cocn3)=O)CC2C)cc1C 6747,c1(C(=O)NCC(CC)NC(c2cc(Cl)no2)=O)ccc(O)cc1F 6748,c1(C(=O)NC2(CCC)CCN(C(=O)C(C)CC(=O)OC)CC2)ccc(S(C)(=O)=O)o1 6749,C=CC(O)C(=O)N1CC(C(C)NC(c2cc(C(C)(C)C)c[nH]2)=O)C1 6750,c1(C(=O)OC)ccc(S(=O)(=O)N2CCC(N)C2)cc1.c12ccc(cc1)c(=O)[nH]2 6751,N1(C(CNC(CCC=C)=O)=O)CC(C(=O)N(CC(C)C)CCO)CC1(C)C 6752,C(CCN=c1[nH]ncs1)NC(=O)Cc1cccc(Cl)c1.C12(CCCCC1)C(=O)N2 6753,C(=O)(C(C)(C)CC(C)(C)C)NCCN(C(C1CCCCC1C1CC1)=O)CC 6754,C(c1c(F)ccc(Cl)c1F)=CC(N1CCC(O)(CNC(Cc2ccc(C)s2)=O)C1)=O 6755,N1(C(Cc2c(C)noc2)=O)CCC(N(C)C(=O)Nc2cnn(C)c2Cl)C(C)C1 6756,Cc1oc2ccccc2c1C(N1CCC(NC(c2nocc2C(C)C)=O)C(O)C1)=O 6757,C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CCCC(N(CC(N2CCC(C)C2)=O)C)C1 6758,C(=O)(NNc1ncnc2sc3c(c12)CCC3)C(N1CCC(C2CCOC2)CC1)=O 6759,n1(CCC(=O)NCCC(C(C)C)NC(c2cc(Cl)cn2C)=O)cc([N+](=O)[O-])cn1 6760,CC(C)(C(F)(F)F)OCC(=O)NCCCCNC(C1(C)CCCC1O)=O 6761,c1(OC)cc(C(=O)NCC2CCC2NC(c2ccnc(C)c2Cl)=O)ccc1Br 6762,N1(C(C(CCNC(CCC(=C)Cl)=O)OC)=O)CCC(O)C(F)(F)C1 6763,CC(C(=O)NC(C)(C)CCNC(C1CC2C=CC1O2)=O)S(N)(=O)=O 6764,CCCCCCC(=O)NC1CC(CCNC(c2cc(Br)n(C)c2)=O)C1 6765,C1(CNC(C(C2CCC(=O)N2)C)=O)CCCN(C(=O)Cn2cnnc2OC)C1 6766,N1(C(C2(OC)CN(C(=O)C(C)NC(=O)NC3CC3)C2)=O)CCC(O)C(F)(F)C1 6767,C(=O)(C1=NOC(C)C1C)NCSCC(=O)Nc1cn(CCCCC)nn1 6768,CCC(C)C(C(=O)NC1(C(C)O)CC1)N(C)C(C1CCCCN1C)=O 6769,c1(C(N2CC(C(=O)Nc3cc(S)ccc3Br)OCC2)=O)csc2ccccc12 6770,C=CCCC(C)NC(c1occc1CNC(C1(c2ccc[nH]2)CC1)=O)=O 6771,c1(OC)ccc(C(=O)NCC2(NC(=O)Cc3ccsc3)CCOC2)cc1OC 6772,C(CCCCC(=O)NC1(C(=O)NOCCOCCOC)CC(CO)C1)=CC 6773,C1(C(=O)OC)OCCC12CN(C(C1(C)CCN(Cc3ccccc3)C1)=O)C2 6774,C12N(CCCC1(C)C)C2=O.CC(CC(=O)N1CCCCC(C)C1)C(F)F 6775,c1(OC)ccccc1C1CC1C(N1CC(NC(C2COCCOC2)=O)C(C)C1)=O 6776,CC1(C)OC(=O)NC1C(N1CCC(CNC(c2cnccn2)=O)C1)=O 6777,C1(NC(CC2CC(=C)C2)=O)CCC2(CC1)CN(C(=O)CS(N)(=O)=O)C2 6778,C1(NC(C(CC=CC)C)=O)CC2(C1)CC(C(=O)N(C)CC1(CC3CC3)CCC1)C2 6779,Cc1cc2ccc(C(=O)NCC3(F)CC(NC(=O)CCCCN=[N+]=[N-])C3)cc2o1 6780,c1(CC(CO)NC(=O)NCCc2c(C)nn(C)c2)ccc(Cl)cc1F 6781,c1(C(=O)NCC2CCCCN2C(c2cnc(C3CC3)o2)=O)cc2cccc(Cl)c2o1 6782,C(=O)(C(C)CCC(C)(C)C)N1CC2CCC(C(N(CC(COC)(F)F)C)=O)(C1)C2 6783,CCC(CC(=O)N1CCC(N(C)C(C23CSCC2C3)=O)C1)C1CCC1 6784,c1(C(=O)NC2C3CN(C(c4cc(=N)[nH]cc4)=O)CC2C3)coc2c1C(=O)NCC2 6785,C1(N(C(C(C2CCC2)NC(CC)=O)=O)C)CCCCN(C(=O)CCC=CC(C)C)C1 6786,C1(C)(C(=O)NCC(C)N(C(=O)CC2C=CCCC2)C)CC(F)(F)C1 6787,C(=O)(C1=C(C)OCCC1)N(C1CCC(CNC(c2c(OC)scc2)=O)CC1)C 6788,c1(CC(=O)NCCCN(C(=O)CSCc2ccccc2Cl)C)ccc(O)nc1 6789,CC1CCN(C(=O)CCN(C(c2ccc(C3CC3)o2)=O)C2CC2)CCS1 6790,c1(OC)cc(C)ccc1C(=O)NC1CCN(C(C2(CCO)CC2)=O)CC1F 6791,c1(C(N2CCN(C(c3c(CC)ocn3)=O)CC2C(C)C)=O)ccc([N+](=O)[O-])nc1 6792,N1(C(C23CC(C)C2C3)=O)CCC(NC(c2ccn(CCF)n2)=O)C12CC2 6793,CCCCCCCCCC(O)C(O)C(=O)OCCC1CC2CC2C1 6794,C1(C(=O)NCC2(NC(C)=O)CCC2)CC2(CC2)CN1C(=O)C=Cc1ccn(C)c1 6795,C1(N(C(c2c(OC)noc2C)=O)C)CCCCN(C(=O)CCc2cncs2)C1 6796,C(C1C(C(=O)NCCCCN(C)C(c2ccn(C3CC3)c2C)=O)C1(C)C)=C(C)C 6797,C1(F)(C(=O)NC2CC=C(C)CC2)CCCN(C(=O)CCC2CCCO2)C1 6798,C1(C(N2CCC(N3CCN(C(=O)C(F)(F)C(F)F)CC3)C2)=O)CCCCC1(F)F 6799,C1(O)(C(=O)NCCNC(c2c(C)nc(-c3ccccc3)[nH]2)=O)CCCCCC1 6800,C1(N(C(c2cnc[nH]c2=N)=O)CC)(NC(=O)C2CC2)CCN(C(C)=O)C1 6801,c1(OCC(N2C(CC(=O)NCC34CCCC3C4)CCC2)=O)ccc(CO)nc1 6802,c1(SCCC)ccc(C(=O)N(C2CCC(NC(C3CC(CC(F)F)C3)=O)C2)C)cc1 6803,C(=O)(C1=CCCCC1C)N(C(CC)CC(=O)NC1CC1C(C)C)C 6804,CCC(CC(=O)N1CCCC(CNC(=O)CCCCC2CC2)C1)OC 6805,N1(C(c2cccc(SC)c2)=O)CC2CC1CC2NC(c1csc(C)n1)=O 6806,CC1COC(CO)CN1C(c1cc(CNC(C2(C3(O)CCC3)CC2)=O)cs1)=O 6807,c1(C(=O)NC2(C)CCN(C(c3cncc(C(=O)OC)c3)=O)C2)cccc2ccoc12 6808,n1(C2CN(C(c3cc(C4CC4)on3)=O)C2)ncc2c1CN(C(=O)Cc1cnoc1)C2 6809,c1(C(N(CC(=O)NCCSc2cccc(Cl)c2)CC)C2CC2)ccc(Cl)cc1 6810,C(=O)(CCCCC(C)(C)C)N(CC(CC)NC(c1cncc(OC)n1)=O)C 6811,n1(CCC(=O)NC(CNC(c2c(C)ocn2)=O)C(C)C)c(C)cc(O)cc1=O 6812,CCCCCC(C)(C)CNC(=O)C(C)NC(=O)C(F)CC1CCCCC1 6813,c1(N2CCCC(C(C)NC(CCC=C)=O)C2)cc(OC)nc(OC)n1 6814,C1(NC(c2nc(COCC)sc2)=O)C=CCN(c2nccc(CC#N)n2)C1 6815,N1(C(C2CC(N(C(C(C)OCCCC)=O)C3CC3)C2)=O)CCC2(CCCN2C)C1 6816,C1(CNC(c2ccc(Cl)o2)=O)CCCN(C(c2cc(O)ncn2)=O)CC1 6817,C1(COC)(NC(c2cc(Cl)c[nH]2)=O)CCN(C(=O)Cc2ccc(F)cn2)CC1 6818,c1(C(=O)NCCCCCNC(c2cc(COC)on2)=O)ccc2c(c1)CCC=C2 6819,N1(C(CN(CCC)C)=O)CC(NC(C2(O)CCSC2)=O)CC2(CC2)C1 6820,N1(C(c2cn(C(C)C(=O)N(C(C)(C)C)CCF)nn2)C)C(=O)c2cccnc2C1=O 6821,C(=O)(CS(=O)(=O)C(C)(C)C)NCC1C2CN(C(Cc3cccc(OC)n3)=O)CC21 6822,c1(NC(C)=O)ccc(S(=O)(=O)N2CCC(C(=O)Nc3nc(=N)[nH][nH]3)CC2)c(F)c1 6823,C(=O)(C1=CCOC1)Nc1cn(CCNC(C(C)NC(=O)NC)=O)nn1 6824,N1(C(C2C(CC)C2)=O)C2CCC1C1CC1(NC(c1c[nH]c3cc(F)ccc13)=O)C2 6825,N1(CCCc2nccn2C)CCC(CCNC(C(=O)NC)=O)CC1 6826,c1(NC(C2C(C(=O)OCC(=O)Nc3ccsc3)C2)=O)ccc2ccccc2c1 6827,C1(CCC)CN(C(=O)C(CC)SC)CC1C(=O)N(C)CCn1cnnc1 6828,c1(C(=O)NCC2(CNC(CCC(=C)Cl)=O)CCOCC2)ccc(Cl)c(CC)c1 6829,C1(CC(=O)N(C(C(=O)NCc2nc(CC)sc2)(C)C2CC2)C)C=NN(C)C1=O 6830,N1(C(CC2(C=C)CC2)=O)CC(N(C)C(c2ccc(O)c(C)c2)=O)C2(CC2)C1 6831,CCC(CCO)NC(=O)C(c1cnn(C)c1)=O.C12CC1C(=O)N2 6832,c1(N(C(=O)CN(C2CCCO2)CC2CCCOC2)C)cccc(C#N)c1 6833,N1(C(C23N(C(=O)OC(C)(C)C)CC2CCCCC3)=O)CCOCC2(CCCC2)C1 6834,C1(C(=O)NCC(=O)OCC=C)CC2CCC1N2C(C1CC(=O)C1)=O 6835,N1(C(CN2CCN(CC)CC2)=O)CCCN(C(=O)C2=CCC(C)CC2)CC1CO 6836,C(=O)(C1=CCN(C)C1)NCCC(N1CCCC1(C)C(=O)OCCCN(C)C)=O 6837,C(=O)(CC(C)CC(C)(C)C)N1CCC(F)(C(N2CCC(C#CC)C2)=O)C1 6838,c12nnc(o1)CC(=O)N1CC(C1)CC(C)NC(=O)CC2.c1(C(C)C)cnnn1C 6839,C1(C)(N(C)CC)COCCN1C(=O)C(CSC)NC(c1ccccc1)=O 6840,C(C(CNC(c1ccc([N+](=O)[O-])[nH]1)=O)C(F)(F)F)NC(C1N(CC)CC1)=O 6841,Cc1ccc(C(F)F)cc1NC(=O)Cc1cc(F)ncc1F 6842,C(=O)(C(C)C(C)S(C)(=O)=O)NC1(CCNC(c2ccn(CCC)n2)=O)CCCC1 6843,CCCC(C(=O)NC(C1CCCN(C(C2CC(C)(C)C2)=O)C1)C)c1ccccc1 6844,Cc1ccc(C(=O)N(C)CC2(NC(c3cnsn3)=O)CC2)c(CC2CCCC2)n1 6845,NS(=O)(=O)C1(C(=O)NC2CC(NC(=O)C=Cc3cocn3)C23CCC3)CCC1 6846,CN1C(=O)CCC1C(=O)NCC1CCCCC1NC(c1cccc(C2CC2)c1)=O 6847,CC(CCCCN=c1[nH]n(C)cc1[N+](=O)[O-])NC(=O)C=CC(=O)N(C)C 6848,N12CCC(C1)C2=O.N1(CC(=O)NC2CC(NC(=O)NC)C2)CC2CC2C1 6849,C1(c2cn(CC(c3c(N)ccc(F)n3)=O)c(C3CC3)n2)C2C3CC4C1C1C2CC3C41 6850,C(=O)(CCC(C)(F)F)N(CC(C)NC(=O)CC1(C)CC(F)(F)C1)C 6851,C1(C(=O)NC(C2CCOCC2)CC)CCN(C(=O)COC2CCCC2)O1 6852,c1(C(N2CCC(C(=O)Nc3c(C#N)ccs3)CC2)=O)cccn2c(O)nnc12 6853,N1(C(CC(C)F)=O)CCC2(CC(C(=O)Nc3ccccc3C3CC3)C2)C1 6854,C1(C(=O)NCC2(CC)CC2)(NC(=O)CC2(C)CC2)CCC(C)(C)C1 6855,c1(C(N(CC(C)O)CCNC(=O)C(C)C(F)F)=O)cccc2ncnn12 6856,C(C(=O)NCC1CCN(Cc2cccc(C)c2)CC1C)(C(C)(C)C)OC 6857,CC1(C)C(C(=O)NC2CCC(NC(C3COC(=O)N3)=O)C2)C1(C)C 6858,Cc1cc(=NC(=O)C(=O)NCC2C=CC(C(=O)NC(=O)Cc3cccs3)C2)[nH]o1 6859,C(C(CC(=O)NCC(C)C(=O)OC)C1CCC1)NC(CN(CCC)C)=O.CCCOC 6860,C1(N(C)C(c2cnsn2)=O)CN(C(=O)C=Cc2ccc(O)cc2)CC1(C)C 6861,C(CC(N)=O)(C(=O)NC(c1cnsc1)C)NC(Cc1nc(C)sc1)=O 6862,C1(C)(C(=O)NCC2CCC(F)(CNC(c3cc(OC)no3)=O)C2)CC2CCC1C2 6863,CC1COCC(C(=O)N(C)CC=CC(=O)N(C2CCCC(O)C2)C)O1 6864,N(C1CCC2(CC2)Oc2ccccc21)C(=O)NCCN(C)Cc1cccc(C)c1 6865,c1(CC(N2CC(CNC(=O)C(N3CCN(CC)CC3)=O)C2)=O)cc(Cl)ccc1Cl 6866,N1(C(C2(c3cccc(-c4cnn(C5CCC5)c4)c3)CC2)=O)CC(O)C(O)C1 6867,CC1(C)CC(C)(C(N2CCN(C(N)=O)CC2)=O)CN1C(=O)C(F)=CC(F)(F)F 6868,N1(C(C2C(CCC)CCC2)=O)CC(F)CC1CNC(=O)CNC(=O)NC 6869,C1(NC(c2c(C)nccn2)=O)CCCC12CCN(C(=O)C1=CCS(=O)(=O)C1)C2 6870,Cc1nc(S(=O)(=O)N(C(=O)C(F)CC(C)(C)C)C(C)C)ccc1Br 6871,C(=O)(C1=CCCCCC1)N(C)CC1(CNC(C2CCCNC2=O)=O)CCC1 6872,CCCC(C(=O)N1CCC(C2N(C(=O)C(C)=O)CC2(C)C)CC1)CC(=O)NC 6873,C1(NC(C2N(C)CC(C)(C)C2)=O)CCC2CC1CN2C(=O)C1=CCOCC1 6874,C(CCCCCNC(N)=O)NC=O.C1(CC=C)CCN(C(=O)CCO)C1 6875,N1(C(C2(C(=O)OCC)CCC2)=O)CC(=O)NCC1C(=O)NC1CN(CC(F)F)C1 6876,c1(OCC)ccc(Cl)c(C(N2CCN(C(c3sc(F)cc3C)=O)C3CC23)=O)n1 6877,CC(C)(CCC(=O)N1CCC(CO)(NC(C2OCCC2(C)C)=O)C1)[N+](=O)[O-] 6878,CC1(C)CCC(C(=O)N(CCNC(=O)C(c2cccc(F)c2)O)C2CC2)OC1 6879,N1(C(C=CCCC)=O)CCCC2(C1)CN(C(=O)Cc1nc(C)c(C)[nH]1)C2 6880,C1(NC(CN2CC(=O)N(C)C2=O)=O)CCCCCN(C(=O)Cc2cnns2)C1 6881,Cc1cc(=NC2CCC3(CC2)CSC3)[nH]c(=NCc2c(C)cnn2C)[nH]1 6882,c1(C(=O)NCCC2(O)CCN(C(c3[nH]c(=NC)sc3)=O)C2)c(C)cc(C)nc1S 6883,N1(C(C(Cc2cn[nH]c2)NC(COCC(=O)OC)=O)=O)Cc2c[nH]nc2C1 6884,C12(C(C)NCC3CCC(C4CC4)O3)CC(CCO1)C2 6885,c1(C(=O)NC2CCCN(C(c3c(C)con3)=O)C2C)cccc2nsnc12 6886,C1(C(=O)NC(CCN(C(COCC)=O)C)C(C)C)CC2(C1)C(F)(F)C21CC1 6887,N1(C(C(C2CCCC2)OC)=O)CCC(NC(=O)C(N)=O)C(C)(C)C1 6888,C1(C(=O)Nc2nnc(O)cc2O)CN(C(C2COCCC2(F)F)=O)CCC1O 6889,C1(C2CC2)(NC(NCC(C)(C)OC(F)F)=NCCCSC(F)(F)F)CCCCCC1 6890,C1(CNC(c2n(C=C)nnc2)=O)CCN(C(c2ccc(F)cc2C)=O)CC1C 6891,N1(C(C2C(C)SCCC2)=O)CCOC(C)C1C(N1CC2(CO)CC2(CO)C1)=O 6892,C(CC(=O)NOCCC(F)F)(C(F)(F)F)NC(C1(COC)CCCC1)=O 6893,c1(C(=O)NCc2c(C)cc(C(C)(C)C)o2)ccccc1S(=O)(=O)C(C)C 6894,N1(C(c2c(C)nn[nH]2)=O)CCN(C(c2ccc(Cl)s2)=O)C(C)C1C 6895,CC1CCN(C(=O)C(O)Cc2cn(C)cn2)C(CNC(c2cnccn2)=O)C1 6896,N1(CC(=O)O)CCN(C(c2ccc(SC3(CCl)CCOC3)cc2)=O)CC1 6897,CC1(C)CCC(NC(C2(CCNC(C3CC4CC4C3)=O)CCC2)=O)CC1 6898,C1(NC(C2OCCC(C)C2)=O)CN(C(C2CC3(CCO2)CC3)=O)C2(CCCC2)C1 6899,Cc1ccc(CC(C)C)cc1C(=O)NC(Cc1cnn(C)c1)C(=O)O 6900,C(=O)(C(C)(C)COC)NCC(CC)NC(c1cccc(F)n1)=O 6901,C(=O)(CN=c1cc[nH]cc1)NCCOCC(=O)NC(C)CCn1cncn1 6902,Cc1cnc(O)c(NC(C2(O)CCN(Cc3ccc(Br)c(O)c3)C2)=O)c1 6903,N1(C(CCCC(C)NCC=C(C)C)=O)CCC2COC(=O)NC2C1 6904,C(=O)(CC1CCOc2ccccc21)NC(CCNC(CCC(=O)N(C)CC)=O)C 6905,c1(OC)cc(C(=O)NC2CC2C(=O)NCCCc2cnccn2)n(C)n1 6906,CC1CN(C(C2CCCN(Cc3cn4ccc(C#N)cc4n3)C2)=O)CC(C)S1(=O)=O 6907,N1(C(CCCCOCCC=C)=O)CCN(C(=O)C(O)CCSC)CC1C1CC1 6908,C1(C(C)C)(C(=O)N(CC(=O)NC2(C)CCOC2)CC2CC2)CCCC1 6909,C(=O)(C(O)C(C(C)C)OC)NC(C(=O)NC(CCOC)C(N)=O)C(C)(C)C 6910,C(C)(C(=O)N1CC(C(C(=O)NCC)OC)C1)SCCCC.C(C)(CC)C1CC1 6911,C1(F)(C(=O)NCC2(CNC(c3c[nH]nc3Br)=O)CC2)CCOCC1 6912,Cn1cnc2c(O)nc(C(N3CCN(CC(O)COCC4CCC4)CC3)=O)nc12 6913,Cc1cccc(OCC(=O)NC2(CO)CCN(C(c3nc(Cl)sc3C)=O)C2)c1F 6914,CN(C1CCCc2ccc(Br)cc21)CC(N1CCC(CC2SCCS2)CC1)=O 6915,N(C(=Nc1ccccc1)N1CCC(OC)C1)C(C#C)CC1CC1 6916,S(=O)(=O)(c1cccc(F)c1)N1C(C(N2CCCN(C(=O)CO)CC2)=O)CC(O)C1 6917,CC1(C)CCN(C(C2CCC(F)CC2)=O)CC1CNC(c1c[nH]ccc1=O)=O 6918,C1(CN(C(=O)C(O)COC)CC)CCCN1C(c1cnn(C(F)F)c1)=O 6919,N1(C(CCOCCOC(C)(C)C)=O)CCC(NC(=O)C=CC(F)(F)F)C1 6920,c1(Cc2nc(C(c3ccccc3)C)oc2-c2ccccc2)ccnc(O)c1Br 6921,c1(OC)c(Cl)cc(NC(C2CC2NS(=O)(=O)c2cn[nH]c2)=O)cc1Cl 6922,Cc1cnc2n1CCCC2C(=O)N1CCN(C(C2C=CC=CC=C2)=O)C(CO)C1 6923,CC(C)C(N=[N+]=[N-])C(=O)N1CCC(C)(NC(c2ncn3ccccc23)=O)C1 6924,C(C)(CNC(c1ccc(C)nn1)=O)(CC(C)C)NC(CS(CC)=O)=O 6925,Cc1ccc(C(=O)NC2CC(CC(N3CCN4CCOCC4C3)=O)C2)c([N+](=O)[O-])c1 6926,c1(C(C(=O)NC(CCOC)CNC(=O)Cn2ncnn2)C)c(C)n[nH]c1C 6927,N1(C(C(C2CCN(C(c3ccnc(Br)c3)=O)CC2)C)=O)CCc2ncccc2C1 6928,C1(O)(C(C)NC(c2csc(-c3ccoc3)n2)=O)CCN(C(c2cncn2C)=O)C1 6929,C(=O)(CCC(C)(F)F)NC(CC(=O)NC1(C#C)CC1)COC 6930,CC(C)(C(=O)NCCCCNC(=O)C=CC(C1CC(C#N)C1)=O)C1CCOC1 6931,c1(NC(C)CNC(=O)C(F)(F)C2CCCO2)ncc(F)cn1 6932,Cc1[nH]nc(C(N2CCCN(C(=O)C(C)NC(C)(C)C)CCC2)=O)c1[N+](=O)[O-] 6933,n1(C2CN(C(COC)=O)C2)cc(C#CCNC(c2nccc3[nH]ccc23)=O)nn1 6934,N1(C(C(C)(C)c2cnsc2)=O)CCC(F)(CNC(C2CCC(F)CC2)=O)CC1 6935,C1(CC)C(NC(=O)CC2(NC(C)=O)CC2)CCN1C(c1cncc(O)c1)=O 6936,CC1CC(F)(F)CN1C(C1CC2CCC1N2C(=O)C(C)(C)C#N)=O 6937,CC(C)C(F)(CNC(=O)C(C)(C)CCN)C(=O)N1CCOC(CF)C1.C(N)=O 6938,c1(OC)cc(N2CCC(N(C)C(C3(C4CC4)CC=CC3)=O)C2)c(F)cc1[N+](=O)[O-] 6939,C1(C(N2CCC(C(C)NC(c3cn(CC)nc3)=O)C2)=O)C2CCC1CC2 6940,C1(CN(C)C(C2(C(=O)NC3(CO)CC3)CCC2)=O)CC(C)(CO)C1 6941,C1(NC(C#CC(=O)N(C)C)=O)CC(F)(F)CC1NC(C1COC(=O)N1)=O 6942,N1(C(c2ccc(C#C)cn2)=O)CC2(CCN(C(=O)C(F)CC(C)C)CC2)C1 6943,Cc1ccc(F)cc1CC(=O)NCC1C=CC(NC(c2cc(C#N)cs2)=O)C1 6944,O=C(CCC(=O)N1CCCC1)NC1CCOCC1NC(C1CC1c1ccns1)=O 6945,N1(C(c2c(C)nns2)=O)CC(NC(c2ocnc2C2CCC2)=O)CC(O)C1 6946,Cc1cc(C(=O)NC2COCCC2NC(=O)COCC2CCCOC2)n(C)n1 6947,c1(OC)c(C(=O)NC(C)(C)CCCNC(C2CCC(=O)O2)=O)cc(F)cc1F 6948,C1(CNC(CCSCc2cccc(C)c2)=O)CCCN(C(=O)C(C)(F)F)CC1 6949,C12(NC(Cc3n(C)cnn3)=O)CCC(F)(F)CC1CN(C(=O)CC1CC(=O)C1)C2 6950,N1(Cc2nn(CC)nc2C)CCC(CO)(NC(c2coc(C3CC3)n2)=O)CC1 6951,Cc1c(Cl)ccnc1-c1nc(-c2nncs2)no1 6952,n1(CCC)nc(C)cc1C(=O)NC1CCC(CCNC(=O)CCC=C(C)C)C1 6953,c1(CC)c(C(=O)NCC2CCN2C(c2cc(C(N)=O)ccn2)=O)nnn1CC 6954,C1(CNC(=O)NC2C3(CCN(CC(=O)N(C)C)CC3)C2)CCC2(CCCC2)CC1 6955,n1(CC(=O)N(CC)CC2(c3ccccc3)CCCO2)ccc(Br)n1 6956,c1(C(=O)NC(CCC)C(=O)NCC2(C(=O)OC)CC2)cccc(F)c1O 6957,N1(C(C(C)c2cc[nH]n2)=O)CCN(C)CC1NC(=O)CC(=O)N(C)C.C1(=O)CO1 6958,C1(C(=O)NC(C2CCCC2)CC)CN(C(c2[nH]ccc2C2CC2)=O)CCN1C 6959,c1(CC(=O)NCC(C)N(C(=O)CC2CC(=O)NC2=O)C)c[nH]c2c(F)cccc12 6960,Cn1ccc2sc(C(N3CCOC(CNC(=O)C#CC4(C)CC4)C3)=O)cc12 6961,C1(c2n(-c3c(SC)cccc3)nc(-c3ccc(F)cc3)n2)CC(=O)NC1(C)C 6962,c1(C2(NC(=O)NCC(F)C3CC3)CCC2)ccccc1 6963,C1(CNC(C(C)OCC)=O)CCN(C(C2CC2CC)=O)C1(C)C 6964,C(C(CC)CC)N(C(=O)CC1CCC(NC(=O)C=CC(C)(C)C)C1)CCC 6965,C1(N(C)C)CCC(C(=O)NC2CC(F)(CNC(c3csc(Cl)c3)=O)C2)CC1 6966,C1(C(N(C2CCCC2)CCOC)=O)COCC1C(=O)NC1CCCS1 6967,c1(OC)cc(CC=NO)ccc1C(=O)NCc1ccc(-c2cnc(F)nc2)nn1 6968,N1(C(CNC(C)=O)=O)CC2(COC(Cc3cn(Cc4c(C)noc4C)nn3)C2)C1 6969,C(=O)(C(O)CCCNC(C1CCC(O)CN1C)=O)NCc1cc(C)ns1 6970,CC(CCP(C)(C)=O)(c1nnnn1C1CCCC1)NCC(CO)SC(F)F 6971,N1(C(C(CC(C)C)N(C)C)=O)CCCC(NC(c2cn[nH]c2)=O)CCC1 6972,c1(C(=O)NC(Cc2cn[nH]c2)C(=O)NCCCCC2CC2)ccc(Cl)nc1 6973,N(C(=NCC1CCC1)N1CCN2C(=O)CCC2C1)Cc1cc(C)sc1C 6974,C(C)(CCCC(=O)NC(c1ncc[nH]1)CO)NC(Cc1c(C)cccc1)=O 6975,C1(C(=O)NC(C2CCCC2)C)CCCN1C(=O)CC1CCCSC1 6976,C=C1CC2CCC(C1)N2C(=O)C(C(C)CC)NC(c1cnn(CCC)c1)=O 6977,c1(C(N2C(C3(O)CN(C(c4c(C)ncnc4)=O)C3)CCC2)=O)cc(O)cc(O)n1 6978,CC1CC(NC(c2ccccc2C2CC2)=O)CN1C(=O)CC1CCOCC1 6979,Nc1cnccc1C(=O)NCC1CN(C(=O)CCN(c2cnccn2)C)CC1O 6980,C1(CNC(CC(CC)OC)=O)CCC2(CCC2)CN1C(C1SCCCS1)=O 6981,C1(NC(C2CCCC(=O)C2)=O)CCN(C(=O)CC=Cc2ccccc2)CC(O)C1 6982,N1(C(C2N(CC)CCC2)=O)CCN(C(c2c(Cl)cnn2C)=O)CC1CC(=O)NC 6983,c1(-c2c(C(=O)Nc3ncc(-c4ccccc4)cn3)csc2)ccc2sccc2c1 6984,c1(C(=O)OC)cc(NC2CCC(NC(N3C4CCC3CC4)=O)C2)n(C)n1 6985,CC1(C)CN(c2ccc(NC(=O)NC3C(O)CC3O)cc2)CCO1 6986,C(=O)(C(C1=NOC2CC12)N(C)Cc1ccc2c(c1)CCO2)NCCCOC 6987,N1(C(C(C(C)NC(c2cc(CC)ncc2)=O)C)=O)CC2(CCC2)CC1CO 6988,Cc1cnoc1C(=O)NC1(C)CN(C(C2(C3CCCO3)CCCC2)=O)C1 6989,N1(C(c2c(C)nns2)=O)CCC(CNC(c2cnc(O)c(F)c2)=O)C(O)C1 6990,C12(N)CCOC(CNc3ncccc3C3CC3)(C1)C2.CC(C)(C)OC(=O)OC 6991,c1(C(=O)NCCC2CCN(C(c3cnns3)=O)C2)csc(Cl)c1Cl 6992,c1(CCNC(=O)NCCc2ccc(N3CCN(C)CC3)cc2)c(F)cccc1F 6993,c1(CNC(c2c(NC(CC(=O)OC)=O)ccs2)=O)ccc2c(c1)COC2 6994,C(CS(=O)(=O)CC(=O)N(C1CCCN(C(c2ccc(C(C)(C)C)[nH]2)=O)C1)C)OC 6995,N1(C(CN2CCC(C)(O)C2)=O)CCN(C(c2ccnn2CCF)=O)CC12CCC2 6996,C1(NC(=O)NC(C)CCNC(=O)OC(C)(C)C)CC2(CCSCC2)C(=O)N1 6997,C(CNC(C12C=CC(CC1)C2)=O)(CC(F)(F)F)NC(c1c(SCC)nccn1)=O 6998,C(=O)(C(C)CS(C)(=O)=O)N1CCC(NC(c2sc(CC)c(C)c2)=O)C1 6999,CC(C)(C(=O)N1CC(NC(=O)Cc2cccs2)C(n2cccn2)C1)C(F)(F)F 7000,N1(C(CSCCCC)=O)CCOCC(F)(CNC(=O)C=Cc2cnc[nH]2)C1 7001,CCC(C)(C#N)C(=O)NCCOCCCN(C)C(c1ccc(-c2cccs2)o1)=O 7002,S(=O)(=O)(c1ccc(C2CC2(F)F)cc1)NC(c1cc(C)c(F)cc1)C 7003,C1(C)(C(=O)NCC(C(C)C)NC(=O)CCNc2cn(C)nc2O)CC=CCC1 7004,C1(CNC(c2cnc(C3CC3)s2)=O)CCCN(c2cc(-c3cccs3)ncn2)C1 7005,N1(C(CC(C)OC)=O)CCC2(CC1)CN(Cc1ccc(Cl)cc1C)CCO2 7006,c1(NCC(=O)OCc2ncccc2Cl)ccccc1Cl 7007,C1(C(=O)NC(c2nc3c(s2)CCCC3)C)CCSC12CN(Cc1ccc(F)o1)C2 7008,CC#CCCCC(=O)NCC1C=CCN1C(c1ccc(CC)c(N)c1)=O 7009,c1(N(C)Cc2cccc(CC)c2)nc(N2CCC(S(C)(=O)=O)C2)c2c(n1)COC2 7010,Cc1cc(=NCC2CCCO2)[nH]c(Nc2nnn(C(C)(C)C)n2)n1 7011,n1(CC#C)cc(CNC(C2CC(C)(NC(=O)CC3(N(C)C)CC3)C2)=O)cn1 7012,c1(C(=O)NC(C)CNC(c2cccnc2Oc2ccccc2)=O)cc(Br)ccc1F 7013,Cc1onc(CNC(C2CC2CNC(=O)Cc2ccccc2)=O)c1Br 7014,C1(CNC(C(COC)NC(=O)C(C)NC(C)=O)=O)CN(C(=O)N(C)C)CC1(C)C 7015,c1(-n2c(-c3ccc(F)[nH]3)nc(CC(N)=O)n2)ccnc2ncccc12 7016,C(=O)(CCCCCCC(=O)N1CC(CNC(C2(C(C)C)COC2)=O)CC1C)OC 7017,Cc1oc(C)c(C(=O)NC2CC2NC(=O)C(c2cccc(O)c2)C2CC2)c1C 7018,C1(C(=O)NC2CC(N(C(CSCCCC)=O)C)C2)CCc2nc(O)[nH]c2C1 7019,c1(CCC(=O)NCCC2(N(C(C3CC3C3CCCCO3)=O)CC)CC2)cccnc1 7020,Cc1nn(C(F)(F)F)c(C)c1CNC(C1NC(=O)CC1C)=O 7021,C1(CCC)(NC(c2cc(C(C)(C)C)no2)=O)CCCN(C(C2CC23CCC3)=O)C1 7022,C1(C(=O)Nc2ncc(C(=O)OC)cn2)CN(C(c2sccc2I)=O)CCC1(F)F 7023,c1(CN2C(C(N3CCC(F)(F)C3)=O)CSCC2)cnc(Cl)cc1Cl 7024,C1(NC(C(N2CCN(C(C)C)CC2)(C)C)=O)CCCC2NCCC12 7025,C1(CCNC(C(c2n(C)ncc2)(F)F)=O)CN(C(c2ccsn2)=O)CCO1 7026,Cc1cnncc1C(=O)NCC(C)(Cn1cccn1)NC(=O)C(C)OCCN(C)C 7027,N1(C(C(c2cccnc2)C)=O)CCOC(C2CN(C(=O)CCNC(=O)CO)C2)C1 7028,c1(C(C)NC(C(=O)NCCC(=O)NC)=O)nccc(C(F)(F)F)n1 7029,N1(C(C)C)CC(C(=O)NC(=O)C(C2CCN(c3nnco3)CC2)C)CC1=O 7030,C(=O)(CC(C(=O)NC1(C)CN(C(c2scnc2C(C)C)=O)C1)N(C)C)OC 7031,C1(C(N2CCC(NC(C=NOC)=O)C2(C)C)=O)CCc2nccn2C1 7032,N1(C(=O)CC2CC3(CC3)C2)CCC2C(C(=O)NC3CC3)C12.C12(C=CCC1)C(=O)NC2 7033,C#Cc1ccc(C(N2CCC(N(C(=O)C(O)C(C)c3ccccc3)C)C2)=O)nc1 7034,C(=O)(C1CCc2c[nH]nc21)NC1CC1.c1(C(=O)NC2CNC2=O)cnccc1Cl 7035,C1(CC)CCC(C(N2CCN(CC3CCCCN3C)CC2)=O)CC1 7036,CN1CCC(C(=O)N(C2CCC(NC(c3c[nH]nc3Br)=O)CC2)C)CC1 7037,C1(c2cn(Cc3onc(C)n3)nn2)CN(CC(=O)OC(C)C)CCN1.C1(C)C(=O)N1 7038,C1(C(=O)NCCOCC#C)CCN(C(=O)Cn2cccn2)CC1F 7039,Cc1cc(C)c(C(N2CC(CNC(c3ccon3)=O)C(C)C2)=O)cn1 7040,C1(C(=O)NC(C(=O)NC2COC3(CCC3)C2)Cc2cc[nH]n2)CC(=O)CC(=O)N1 7041,CC(C)CC(C)N(C)C.N1(CC(=O)NCCC(=O)N(CCN)CCOC)CCSCC1 7042,c1(OC)cc(CC(N2CCN(CCN(C)C(C3(O)CCCC3)=O)CC2)=O)ccc1C 7043,N1(C(c2c(C)nn[nH]2)=O)CC2CN(C(c3ccc(C(C)C)nc3)=O)CC12 7044,c1(C(=O)NC2CN(C(c3cc(C)cc(O)n3)=O)CC2C)[nH]cc2c1CCCC2 7045,C1(C(N2CCN(CCNC(C=C(C)C3CC3)=O)CC2)=O)CC2COCCN2C1 7046,c1(CN(C(C2CCN3CCCN2C3)=O)CC)cn2c(C)cc(C)nc2n1 7047,C(=O)(C(F)(F)C(O)C1CC1)N(C)CC1CCCN1C(=O)COc1ccsn1 7048,c1(CC)[nH]c(=N)sc1C(=O)NC1CC(CNC(c2cnsc2)=O)C1 7049,N1(C(C23CN(C(c4nc(C)oc4)=O)C(C2)CO3)=O)CCCCCCC1C 7050,N1(C(C(C)OCOC)=O)CC(C)(C)CC1C(=O)N(CC(CC)OC)C 7051,c1(CC)cnc(C(=O)NCC(O)CNC(C2C=CC2C(=O)OC)=O)cn1 7052,O(NC(=O)C(c1cccs1)NC(c1cc(C)n(C)c1)=O)CCCC#C 7053,N1(C(c2nc(NC)sc2)=O)CCC2(CCCN2C(C2(O)CCC(C)(C)CC2)=O)C1 7054,c1(OC)nccc(CNC(C2COCC2NC(c2csc(C)c2C)=O)=O)n1 7055,N1(C(CC(c2cccc(C#N)c2)C)=O)CCOC(CNC(c2csnn2)=O)C1 7056,c1(C(C(N2CCC(NC(C(C)OC(C)(C)C)=O)C2)=O)(C)C)cc(Cl)cc(Cl)c1 7057,C(CN=C(NCc1cn(C)nc1Br)NC(C)Cc1c(C)nn(C)c1C)SC 7058,c1(C(N(C)CCNC(C2CCC2C(C)(C)C)=O)=O)cc2sc(Cl)cc2s1 7059,N1(C(c2n(C)ncc2Cl)=O)CCC(NC(=O)Cc2c(O)ncnc2O)CC(O)C1 7060,C=CC(C)(C)C(=O)NC1CCCC(CC(=O)NCC(O)(COC)CO)C1 7061,N1(C(CCSCC)=O)CCCOC(CNC(=O)CCn2ccc(C)n2)C1 7062,Cc1c(CNCC2(c3ccccc3)CCOC2)cnn1-c1ccccc1 7063,C(=O)(C1=CS(=O)(=O)CCC1)N1CC(NC(CCC(=O)NCCC)=O)CC(C)(C)C1 7064,c1(OC)cc(NCC2CC(F)(SCc3cn4ccccc4n3)C2)ccc1[N+](=O)[O-] 7065,CCC(C)(C)CCCC(=O)NC1CCCC1NC(c1c(C)ccc(F)c1N)=O 7066,c1(-c2ccc(C(N3CC(C)(C(C)(C)C)OCC3)=O)cc2)noc2ccccc12 7067,N1(C(CCOCCC)=O)CCC2CCCC12C(=O)NC(CO)C(C)(C)CO 7068,C1(C(=O)NCC2N(C(C3N(C(CC)=O)CSC3)=O)CC2)CC(S(C)(=O)=O)C1 7069,S(=O)(=O)(c1ccn(CCF)n1)N(C)C(c1c(F)cc(F)cc1F)=O 7070,C12(CC(C)(C)C1)C(=O)NC2.C1(CN(C(C(C)c2ccsc2)=O)C)CCCC2CC12 7071,C1(NC(=O)NCC2CCN(C(COC)=O)C2)CC2CCC1O2 7072,n1(C(C)C)cnc(NC(=O)C(c2cnn(C)c2)NC(=O)OC(C)(C)C)n1 7073,C(=O)(C(CCC1CCC1)NC(=O)C(N1CCOCC1)=O)NC1CC(C)(C)C1 7074,c1(C(N(C(C(N2CCC(OC)(CO)C2)=O)C)C)=O)cnn2c1OCC2 7075,c1(C(=O)NCCC2CC(C(N3CCC(CC=C)C3)=O)C2)ccc([N+](=O)[O-])[nH]1 7076,c1(SCC)nccnc1C(N1CC(OC)C(NC(=O)CC(C)(C)O)C1)=O 7077,C1(C)(CC(=O)NCC2CCN(CCC)C2)CCN(C(C23CC(F)(C2)C3)=O)C1 7078,CC(C)CC(C)C(=O)N1CCC(N(C)C(C2CC3C=CC2CC3)=O)CC1 7079,C(=O)(CC(=O)NC(C)C(=O)NCC(c1cscn1)O)OC 7080,Cc1nn2c(C(=O)NC3CN(C(c4ccoc4Cl)=O)CC(C)(C)C3)c(C)nc2s1 7081,c1(C(=O)NCC(C2CCCCC2)NC(c2n[nH]c(=N)[nH]2)=O)cc2c(nn1)CCC2 7082,N1(C(CCC(C)NC(=O)C(F)(F)CO)=O)CC2C(C1)C2(F)F 7083,N1(C(C(=O)NC)=O)CCC2(CC(Nc3c(C)[nH]c(C(=O)NC4CC4)nc3=O)C2)C1 7084,C(C1=NOC(C)C1)NC(CCNC(CC(C)SC)=O)=O 7085,CCCCCC(O)CC(=O)NCC1(O)CN(C(=O)C(C#N)CC)C1 7086,c1(CC(=O)NC(C(=O)N(CCCSC)C)C2CCC2)cncn1C 7087,c1(C(N(CCCN(C(=O)CCc2cncn2C)C)CCO)=O)cc(N)cc(F)c1 7088,C1(NCC(c2ccncc2)CO)CC2CC2C1 7089,c12cccc(n1)NC2.C(C(F)(F)C(F)F)OCCOC(C)C 7090,C1(NC(CCNC(C(C)(C)C)=O)=O)CC2CC1N(C(C1CC3(CCOC3)C1)=O)C2 7091,C1(C(N(c2c(C)cccc2)C)=O)CCN(C(=O)C(CC(N)=O)NC(N)=O)O1 7092,c1(CCC)ncc(C(=O)NCCCN(C(c2ccc(OC)s2)=O)C(C)C)s1 7093,C1(C(N2CCN(C(CSCC)=O)CC2CC(F)(F)F)=O)Cc2cc(C)ccc2S1 7094,C1(CNC(C(C)Cc2ccco2)=O)CN(C(c2ccc(F)s2)=O)CCO1 7095,C(c1ccco1)=CC(N1CCC1C(N1CCCC1C(O)CO)=O)=O 7096,c1(C(=O)NCC(CNC(c2c(C(C)C)nns2)=O)F)cccn(C2CC2)c1=O 7097,C(=O)(CC(CNC(C1C(C)(C)C1(F)F)=O)C1CCC1)N1CC(C(C)OC)C1 7098,c1(CNC(C(C2CC(NC(C3(C)CC3(F)F)=O)C2)F)=O)ccccc1O 7099,N(C(=NCCC(=O)NCC)NC1C=CCCC1)Cc1c(C#C)cccc1 7100,Cc1nn(C)c(C(=O)O)c1CNCc1ccc(C(O)C(F)(F)F)cc1 7101,Cc1c(C(=O)NC2CCC2Cn2cc(C(C)(C)CC3CC3)nn2)cc(C)n1C 7102,C(c1c(Cl)cccc1Cl)=C(C)C(=O)NC1CC(F)(CNC(C2CCOC2)=O)C1 7103,N1(Cc2cc(C(N(CC(C)(C)NC(=O)CN(C)C3CC3)C)=O)no2)CCCS1(=O)=O 7104,C=CC(CC)CC(=O)NC1(C(=O)N(c2ccn(C3CC3)n2)C)CC1(C)C 7105,C1(CC=C)(C(=O)NCC2(CC)CCOCC2)CCCN1C(c1ccnc(C)c1)=O 7106,c1(C(N2CCCN(C(C(C)(C)OC)=O)CC2)=O)ccc2c(c1)C(=O)NCC2 7107,c1(OCC)ccc(Cl)nc1C(N1CC2C(C1)N2C(=O)CCCOC)=O 7108,N1(C(C(C)OC(C)(C)C)=O)CC2CC1CN(C(=O)Cc1cnoc1)C2 7109,c1(C(=O)NC2(C)CCN(C(CC(C)C3CC3)=O)C2)ccc2c(c1)CCCCC2=O 7110,c1(COc2ccnn2C)cccc2c1N(C1CCCc3sccc31)CC2 7111,C1(NC(Cn2c(C)ccc2C)=O)CCN(C(C2CCN(C3CC3)CC2)=O)C12CC2 7112,c1(CC(=O)NCc2csc(C(N3CC4CC4C3)=O)n2)cccnc1F 7113,c1(OC)cccc(O)c1C(N1CCCC(O)(CCNC(=O)CCC2CC2)C1)=O 7114,C(C(=O)NC1CCCN(C(=O)CSCSc2ccccn2)CC1)(C(C)(C)C)OC 7115,c1(C(N2CC(CN(c3nccc(OC)n3)C)C2)=O)ccc(F)nc1C 7116,CCCC(O)C(=O)N1CC(N(C)C(c2c[nH]nc2-c2ccc(Cl)cc2)=O)C(O)C1 7117,CCC(CC)(CO)C(=O)C(=O)CC1CCCCC1C.C(C(CC(F)(F)F)C(=O)N)N 7118,C1(NC(C2(OCC)CCOC2)=O)CCCCC1CNC(=O)CCC1CCOCC1 7119,c1(C(=O)OC2(C)CN(C(C(CCC)OC(C)(C)C)=O)C2)ccc([N+](=O)[O-])o1 7120,CC(C(CO)NC(c1sccc1CO)=O)NC(=O)CCC1CC1 7121,N12CC(=O)N(C1=O)CC(C)(C)S2.c1(SC(CC)(C)C)ccc(Br)cc1 7122,N1(C(C2CCCC(NC(Cn3c(C)ncc3)=O)CC2)=O)CCC2CCN(C)CC12 7123,CCCCC(CN=c1ccc(C(F)(F)F)n[nH]1)OCC(=O)NCC 7124,C12(C(=O)NCCCC(C)(C)C)CCC(CN(C(c3cc(=N)[nH][nH]3)=O)C1)C2 7125,N1(C(c2c(C)ncs2)=O)CCCC1(C)c1cn(CC2(CN3CCCC3)CC2)nn1 7126,N1(C(CCc2nc(C)sc2)=O)CCCCC12CC(NC(=O)Cc1ccccn1)C2 7127,c1(C(=O)NC2CN(C(=O)CC3=CCCC3)CC2F)cc(F)c(Cl)c([N+](=O)[O-])c1Cl 7128,C1(CC)CN(C(C2(COC)CCCC2)=O)CCC1NC(=O)COC(C)C 7129,c1(OCC(N2CC(CNC(C(COC)O)=O)C(F)(F)C2)=O)cc(C)c(Cl)c(C)c1 7130,c1(OCCC)cccnc1C(=O)N(CCCCN(C)C(c1cccs1)=O)C 7131,C#Cc1ccc(C2(C(=O)NC(CNC(=O)CC3(OC)CC3)(CC)CC)CC2)cc1 7132,C#Cc1cnc(C(=O)NCC(C2CCN(C(C3CC(F)C3)=O)CC2)C)c(C)c1 7133,N1(C(c2ccc(C)[nH]2)=O)CCCC(C)(CNC(C2(C)CCOC(C)C2)=O)C1 7134,Cn1ncc(C(=O)NCC2(C)CCCN2C(c2n[nH]cc2Cl)=O)c1C#N 7135,c1(C(c2ncccc2F)CNC(C(=O)N(CCOC)CO)=O)ccc(OC)cc1 7136,CC(C)(C)C(CNC(C1(C)CC1Br)=O)NC(=O)Cc1ccccc1C(F)(F)F 7137,c1(CC(=O)NCC2C3CN(C(C(C)CN(C)C)=O)CC32)cccc(Cl)c1Cl 7138,N1(C(C(=O)N(C)Cc2c(OC)cccc2)C)CCc2cc(Br)ccc21 7139,N1(C(C(OC)OC)=O)C2CCC1CC(CC(C)NC(c1c(F)cccc1Cl)=O)C2 7140,Cc1nn(CCO)c(C)c1CC(=O)NCCNC(c1cc(C(C)(C)C)no1)=O 7141,Nc1cc(C(=O)Nc2cc(C(F)(F)F)cc(CO)c2)cc(O)c1 7142,c1(C(=O)NC2(C)CCN(C(c3cncs3)=O)C2)cc([N+](=O)[O-])ccc1N 7143,N1(C(C(C(C)C)C2CCC2)=O)CCC(NC(=O)CCC2(C)CC2(F)F)C12CC2 7144,n1(CC(N2CC(C(=O)NCC(O)CF)(SCC)C2)=O)cccnc1=O 7145,C(=O)(C(C#N)C(C)(C)C)NC(CCC(=O)NC1C(OCC)CCC1)C 7146,C(C(C)N=c1[nH]c2c(c(=NCCCc3ccc(F)c(Cl)c3)[nH]1)CCC2)SC 7147,n1(CCC)c(N(CC(C)C)CC)nnc1CSc1ccc(F)cc1 7148,CCCCS(=O)(=O)N1CCCCC1CO.c12cn(nn1)CC(=O)NC2C 7149,CCC(C)(CO)C(=O)N1CCC(CN(C)C(c2cccc(C3CCCC3)c2)=O)C1 7150,C1(C(C)(C)C)(CN(C(=O)CCC2CCCC2)C(C)(C)C)CCN(C(=O)CCC2CC2)C1 7151,c1(NC(CC(CC)CN(C)C)=O)ccn2ncnc2c1.C12COCCN(C1)C2=O 7152,C1(C(N(C2C(C)C2)C)=O)CCCCN(C(C2(CCCF)CC2)=O)C1 7153,C1(C)(NC(C2C(C(C)C)C2)=O)CCC(NC(C2C3CC4C(C3=O)C24)=O)CC1 7154,CCCCC(C)(F)C(=O)NCC(CO)NC(C1CCC(CC)C1)=O 7155,C1(CN2CCC2)CC12CCCC2.O=C(C(O)C1CCCC1)NCC(O)CC1CCCC1 7156,C12(C(N(CCNC(=O)CCSC3CCCC3)C3CC3)=O)CC=CC(C1)OC2 7157,c1(C(=O)NCC2CC(C)N(C(c3ccc(Cl)c(CO)c3)=O)C2)nnc(Cl)cc1N 7158,C1(NC(C(c2cnccn2)C)=O)COCCC1NC(c1ccc(C(N)=O)[nH]1)=O 7159,c1(SC)ccc(C)c(C(=O)NCC2COCCN(C(=O)Cc3cc(C)ns3)C2)c1 7160,c1(C(=O)OC)ccnc(C(N2CC(OCCNC(=O)C(C)O)C2)=O)c1 7161,N1(C(C(C=CC)O)=O)CCCC(C2(NC(c3cc(=O)n(C)cn3)=O)CC2)C1 7162,N1(C(C2CCN2C(=O)Cn2nccn2)=O)CCC(CO)C(O)C1 7163,C(C(=O)N1CCC(O)(C(C)NC(=O)C2=NOCC2)C1)(C(C)C)NC(COC)=O 7164,C(C(C)(C(=O)NCC(c1ccsc1)O)NC(=O)CCC(C)N(C)C)SC 7165,c1(OCC)cc(NNC(=O)NCC(c2c(C)n[nH]c2C)C)ncn1 7166,C1(C(N2CCC(CCNC(c3n(C)cnn3)=O)CC2)=O)CCc2nc(O)[nH]c2C1 7167,C(=O)(C1=NNC(=O)CC1)N1CC(NC(C2(C(=O)NC)CC2)=O)C1(C)C 7168,c1(C(N(CCO)C(C2(C(C)C3CC3)CC2)=O)C)cn(CC2CCCOC2)nn1.CCO 7169,c1(C(N2CC(C(=O)Nc3cnc(C(F)F)cn3)SCC2)=O)c(Cl)ccnc1Br 7170,N1(C(C2CN(C(C(C=C=C)C)=O)CC23CC3)=O)CCc2ccccc2C1 7171,C1(C(=O)NCCC=C)CN(C)CCN1C(=O)C(C(C)O)N(C)C 7172,CC1(C)COC(CC(=O)NCC(C2CC2)NC(C2(C(F)(F)F)CC2)=O)CO1 7173,c1(CNC(C2CC(CNC(=O)CN3CC=CC3)C2)=O)ncc(F)cn1 7174,Cc1cc(CCC(=O)NCc2cc(C(=O)NCC(O)C(C)C)on2)on1 7175,c1(C(N(CC(C)NC(C2CCCN(CC)C2)=O)CC)=O)cc(C)nc(O)c1 7176,C1(c2n(CCC)nnn2)(Nc2ccc(F)c(F)c2C)CCCN2CCSCC12 7177,C1(C(=O)NCCCN(C(C2C(=C)C2)=O)C(C)C)CCc2nc[nH]c2C1 7178,C1(CNC(C(C)(C)O)=O)CN(C(C2CCN(C3COC3)C2)=O)CCCO1 7179,N1(C(COCCSC)=O)CCC(N(C)C(c2cccnc2S)=O)CC1 7180,c1(CC=C)ccccc1C(=O)NC12CC(C1)N(C(=O)C(F)C(C)C)C2 7181,N1(C(c2cc(C)oc2C)=O)CCOC(C(=O)NCC23CC(C(C)C)(CO2)C3)CC1 7182,C(=O)(CC(C)CCC=C(C)C)N1CC(CC=C)(NC(=O)C(=O)Nc2ncc[nH]2)C1 7183,C1(CNC(c2n(C)nc(C(F)(F)F)c2)=O)CC2CCC1N2C(=O)CN1CCC1C 7184,N1(C(CC2C(C)CCN(C(C3OCCC3C)=O)C2)=O)CCn2ncc(O)c2C1 7185,C1(C(N(CCC#C)CCO)=O)CC12CCN(C(=O)C(C)n1ccnn1)CC2 7186,N1(C(CC(C(F)F)c2cccc(OC)c2)=O)CCC2(C1)OCCO2 7187,Cc1ccc(C(=O)NC2CCCC(N(C(=O)CN3CC(C)C3)C)C2)cn1 7188,c1(C(=O)NC(CN(C(c2ccc(C)cc2C)=O)CC)C)csc2ccc(C)cc12 7189,C1(C(=O)NC(C#CC)(C)C)CN(C(C2(C)CCCCO2)=O)CC1C1CC1 7190,N1(C(=O)COC2CCCC2)CC(C2CCN(C(c3c(O)cccc3F)=O)CC2)C1 7191,c1(C(C)C)ccnc(NC2CCC(Cc3cccc(F)c3)C2)c1 7192,C1(NC(c2ccc(C)nn2)=O)CN(C(C2CCCCS2(=O)=O)=O)CC1(C)C 7193,N1(C(C(C)=C(CC)C)=O)CC(NC(c2c(C)noc2CC)=O)CC12CCCCC2 7194,C1(C)(C(=O)NCC(C(=O)NC(CN(C)C)CCO)N(C)C)CC(C#N)C1 7195,c1(C(N2C(CN(C)C(C3CC4CC3C4)=O)CCCC2)=O)cnc2cccnc2c1 7196,N1(C(C(CCOC)(C)C)=O)CCC2CCN(C(c3nccs3)=O)CC2C1 7197,CC1CCCCC1OCC(=O)NCC1CN(C(=O)Cc2ccncc2Cl)CC1C 7198,C(=O)(C1=CCN(C(=O)OC(C)(C)C)C1)N1CC(N(C)C)(Cc2c(C)noc2Cl)C1 7199,N1(C(C(CC#C)(C)NC(c2ccoc2C(C)C)=O)=O)CCCC(O)(C#C)C1 7200,c1(C(N2C(C(=O)NCc3cccc(OC)n3)CC3CC32)=O)cc2sccc2[nH]1 7201,Cc1ccc2ncccc2c1C(=O)NCc1cccc(Cn2cncn2)c1 7202,C1(NC(C2CN(CC(C)C)C(=O)C2)=O)CCN(c2ncccn2)C(C)C1 7203,C1(CNC(c2c(C)coc2C)=O)CCN(C(=O)CSCC(F)(F)F)CC1C 7204,N1(C(c2c(OC)cc(C)cc2C)=O)CC2OCCN(C(C3CCC(C)O3)=O)C2C1 7205,N1(C(CC(CC)C)=O)CCN(C(c2ccc(-c3ccccn3)cc2)=O)C(C#N)C1 7206,C1(C(=O)NCCN(C(c2c(N)ccc(CCC)c2)=O)C)CC2CC(O)CC(C1)C2 7207,CC#CCCCC(=O)N(C1CCCC(NC(c2nccc(F)c2Cl)=O)C1)C 7208,c1(OC)cccc2c(C(=O)Nc3cccc(NC(C4(O)CCOC4)=O)c3)n[nH]c12 7209,C1(NC(c2c(C)nc[nH]2)=O)CC(CNC(c2nc(Br)c[nH]2)=O)C1(C)C 7210,c1(SCC)cnc(O)c(C(=O)NCCC(C)N(C(=O)C(C)N(C)C)C)c1 7211,C=C(C)CC(C(=O)N1CC=C(C(=O)NC(C(=O)OC)C2CC2)C1)OC 7212,C1(C(=O)NCC2CCCCN2C(=O)Cc2cccs2)CCC=CCCC1 7213,C(=O)(C(C)(O)CC(F)(F)F)NCC(C)NC(c1ncccc1O)=O 7214,C12(C(N3CCC(CNC(Cc4nc(C)[nH]n4)=O)CC3C)=O)CC=CCN1CCC2 7215,O=C(NN1CCS(=O)(=O)CC1)c1ccn(CC(F)F)n1 7216,c1(OC)nc(N2CCCC(CNC(=O)C(C3CCCO3)C3CC3)CC2)cc(C)n1 7217,N1(C(c2c(C)c(C#N)[nH]c2)=O)CCOC2CN(C(=O)CC(C)C(C)(C)C)CC12 7218,CCC(C)C(C(=O)NCCC1CC(NC(C2(C)CC(F)C2)=O)C1)NC(C)=O 7219,c1(C(=O)NC(c2ccccc2)C(=O)NCC2CCCC3CC23)nc(C)c(CC)o1 7220,c1(C(N2CCCC(CNC(COC(C)=O)=O)C2)=O)oc2ccccc2c(=O)c1C 7221,c1(OC)ccc2c(=NCC3(CCO)CC3)[nH]c(N3CC4(C)CCC4(C)C3)nc2c1 7222,CC1CC(NC(c2ccnc(C3CC3)n2)=O)CN1C(c1cnn(C)c1Br)=O 7223,CC1(C)CCCOC1CNC(=O)CC12CCC1CN(C(=O)CC(F)(F)F)C2 7224,c1(C(C(=O)NCCC)N(C2CCN(CCOCCCO)C2)C)cnc(C2CC2)s1 7225,C1(CNC(CCCOC(C)C)=O)(CO)CCN(C(c2cc(F)cs2)=O)CC1 7226,c1(-n2cc(CN3C(C(CC)O)CCC3)nn2)cc(Br)ccc1Cl 7227,Cc1ccc(N)c(C(=O)NC2CC(NC(=O)CC3CCCC4(CC4)C3)C2)c1 7228,c1(C(=O)NCC2N(C(C(CC)(C)C)=O)CCCC2C)cccc2oc(C)nc12 7229,N1(C(Cc2ccc(NC(C3C=CCC3)=O)nc2)=O)CC2CC(NCC3CC3F)C1C2 7230,c1(C(=O)NC(C)(C)C)cnc(C(=O)NC(c2ccccc2F)CCO)nc1 7231,C(CO)(C(C)(C)CO)NC(C(C1CN(C(C2(C)CC2(F)F)=O)C1)O)=O 7232,C1(C(N2CCC(C)C2)=O)CCCN1C1CCC(C(=O)NC)C1.c1(SCCS)ccccc1.N 7233,c1(CCC)cc(C(=O)NCCN(C(=O)CC2CC3CCC2O3)C(C)C)sc1C 7234,C(=O)(C(CC(C)C)C(N)=O)NCc1cc(C(N2C(CC)C(C)(C)C2)=O)on1 7235,c1(CC(C)C)ccc2[nH]c(=NC(C)CCC3CC3)nc(N3CCCC(C)C3)c2c1 7236,C1(OC)CCC(OC2(C(F)(F)C(=O)NC3(c4ccccc4C)CC(O)C3)CC2)CC1 7237,C(C(=O)NC1CC2CCC1(C(N1CC3CC=CC1C3)=O)C2)(C(C)(C)C)OC 7238,C(=O)(C(CCO)N(C)C)NCCC(=C)CNC(c1sc(C)nc1CC(C)C)=O 7239,C=CC1(NC(C2CC2NC(=O)COCC(=C)C)=O)CCCCC1 7240,c1(C(N(CC(C)NC(=O)C=Cc2ccc(C)s2)CC)=O)cc2ccccc2[nH]1 7241,C(=O)(C1CCCc2scnc21)NC1CCN(C(C2(CN(C)C)CC2)=O)CC1F 7242,C(=O)(C1=C(C)OCCS1)NCCN(CCC)C(c1ccc(C)c(C(C)(C)C)c1)=O 7243,C1(NC(CCOC)=O)CN(C(=O)CC2CC(=O)C2)CCC1C 7244,C1(CNC(c2nocc2Cl)=O)CCN(C(=O)C=CCO)CC1O 7245,c1(OC)ccc2[nH]c(C(N3CC4CC4(NC(=O)C=C4CCOCC4)C3)=O)cc2n1 7246,NS(=O)(=O)c1cc(C(=O)NCC2CCC(NC(=O)Cc3ccco3)C2)co1 7247,C1(NC(c2cnc3c(c2)CCC3)=O)CCC2CCN(C(C3CCCOC3)=O)C1C2 7248,C=CC1(CC(=O)NCCC(C)NC(=O)C(O)Cc2ccccc2)CCCCC1 7249,CC(C)(C)C(CC(=O)N1CC(NC(c2ccc3c(c2)nnn3C)=O)C1)C(F)F 7250,c1(C(=O)NC(C)CC2CN(C(c3cnccc3Cl)=O)C2)cc2cncn2c(O)n1 7251,Nc1cc(C(=O)NC(C2CCOC2)CNC(=O)C=C2CCSCC2)ccc1F 7252,N(C(=NCCN1CCCC1)NCC1Cc2ccccc2C1)C(CC)CC 7253,C(=O)(C1=CCS(=O)(=O)C1)NCC1CCC(CNC(c2ccc(C)cc2N)=O)C1 7254,CC1(C2(C(N3CCCC(C(C)(C)CNC(C4CC4(F)F)=O)C3)=O)CC2)CC1 7255,C12(NC(C=CC(=O)NCCC(N)=O)=O)CCN(C1)C2=O.c1(NC)ccccn1 7256,C#CCC(C)(C)C(=O)NCCOC1CCN(C(=O)CC2CCOC(CC)C2)C1 7257,S(=O)(=O)(c1cc(C(F)(F)F)ccn1)N(CC(=O)Nc1ccccc1)C 7258,Cc1cccc2[nH]cc(C(N3CCC(C)(CNC(C4(C5CC5)CC4)=O)CC3)=O)c12 7259,N1(C(C2CC(C)N2C(c2cc(CO)[nH]n2)=O)=O)CCc2cnccc2C1 7260,C1(CC)CCC(C(N2CC(OCCNC(=O)C(F)CC3CCOCC3)C2)=O)CC1 7261,Cc1ccc(-c2ccc(Cn3cc(CC(C)C)nn3)cc2)cc1C 7262,C(=O)(C(=O)N=S(C)(C)=O)N1CC(C)C(N(C)C(C2(C(F)(F)F)CCCC2)=O)CC1 7263,c1(C(=O)OC(C)(C)C)cnn(CC2CC2)c1.CN1CCN(C)C1=O 7264,C(=O)(C(C)O)NC(C1CCCC1)CNC(CN(C(COC)=O)C)=O 7265,c1(C(=O)NCCN(C(c2c(COC)ncs2)=O)C2CC2)cnc2ncnn2c1C 7266,c1(CNC(CCN(CC#C)C(C2CC2(Cl)Cl)=O)=O)ccc(NC)nc1 7267,S(=O)(=O)(c1cnc(NCCc2nccnc2C)c(Cl)c1)NCC=C(CCC)C 7268,N1(C(c2c(C)ccnc2)=O)CC(C)C(C)(CNC(=O)C(C)S(N)(=O)=O)C1 7269,C(=O)(C(C)C(F)(F)F)NCCCCCNC(C(c1cccc(C)c1)F)=O 7270,C1(NC(C(c2cccnc2)OC)=O)COC2(C1)CN(C(c1csnn1)=O)C2 7271,n1(CC#N)c(C(N2CC(NC(c3ccnnc3O)=O)C2)=O)cc2ccccc12 7272,Cc1ccc(C)c(C(=O)NC2CCC(NC(=O)C(O)CC(C)C)C2)c1 7273,Cc1cc(C)c(C(=O)NCC2CCC(C)CN2C(C23CC(C2)C3)=O)c(C)c1 7274,Cc1cccc(Br)c1S(=O)(=O)NC(CC1CCCO1)CO 7275,C1(CNC(CN(CC)CC)=O)CC(F)(F)CN1C(c1cc(Cl)c[nH]1)=O 7276,N1(C(CSCC)=O)CCN(C(=O)CC2C(=O)NN=C2C)C(CS(C)(=O)=O)C1 7277,C1(C)(C(=O)NCCCOCCC(=O)NCCCOC(C)C)C=CCCC1 7278,C1(CNC(CCNC(C)=O)=O)CN(C(c2coc(Cl)n2)=O)C2CCN1C2 7279,Cc1cc(NC(C2CCN(C(=O)CCC3CC3)C2)=O)cc(O)c1 7280,C(=O)(C(O)CC(F)(F)F)N1CCC(C(=O)NCCC(C)N(C)C)C12CC2 7281,N1(C(c2c(C)nc(Br)o2)=O)CCN(C(C2(C)CCOC2)=O)C2(CC2)C1 7282,N1(C(C2(C)CCN(C)C2)=O)CCN(C(=O)C(C)(C)N(C)C)CC1c1ncc[nH]1 7283,C12(NC(C3CCC(C)(C)CC3)=O)CC1COC21CCC1 7284,C1(=CC)CN(C(=O)OC(C)(C)C)C1C(=O)N(C)CCNC(c1scnc1C)=O 7285,C=CC(C)(CC)C(=O)N(CCN(C)Cc1ccc(F)c(N2CCOCC2)c1)C(C)C 7286,c1(C(=O)NCC(C(C)(C)C)NC(CN(C)CCO)=O)ncc(Cl)cc1Cl 7287,c1(C(=O)NC2COCC2C(N2CCC(CCO)C2)=O)ccc2cc[nH]c2c1 7288,N1(C(C(C(C)C)NC(C)=O)=O)CC(CNC(=O)CCc2nc[nH]n2)C(C)(C)C1 7289,C(C)(C(C(=O)NCCSC)NC(=O)Cc1cccnc1C)OC.C1CO1 7290,CC1CCC(C)N(C(=O)CC2CN(C(c3ncn(C(C)C)n3)=O)CCO2)C1 7291,C12(NC(C3(CC(=O)OC)CC3)=O)CCCN(C(c3cc4nccnc4[nH]3)=O)CC1C2 7292,Cc1cc(N)c(C(N2CC3=C(C2)CN(C(c2ncoc2C(C)C)=O)C3)=O)cc1C 7293,C1(=CCC)CCN(C(=O)C(c2cccnc2)NC(C2CC2C(F)F)=O)C1 7294,N1(C(c2ccn(CCC)n2)=O)CC2CC(C(N3CCC(CC(C)C)C3)=O)(C2)C1 7295,C1(C(=O)NC(C(=O)NCCNC(C(C)(C)C)=O)Cc2cn[nH]c2)CC12CCCC2 7296,n1(CCC(=O)NCC2(O)CC(CNC(CCOC)=O)C2)nc(C)cc1C 7297,Cc1nccn1C(C)C(=O)NC1CC(CCNC(c2cnc(C3CC3)o2)=O)C1 7298,N1(C(C(CC)NC(c2ccco2)=O)=O)CCC(CNC(=O)C(C)OC)C(C)C1 7299,C(=O)(C1=Cc2ccccc2C1)N(CC(C)NC(=O)CCP(C)(C)=O)CC 7300,O=C(CCCOCl)NCC(c1ccccc1)NC(=O)CC1C=CCC1 7301,c12nccc(n1)N2.C1(CNC(COC)=O)C=CCN1C(=O)Cc1ccon1 7302,C1(NC(c2cnccn2)=O)CCN(C(c2c(F)cccc2I)=O)CC1F 7303,Cn1cc(S(N)(=O)=O)c(C(=O)NCC(C2CC2)NC(c2nncs2)=O)n1 7304,C1(C(=O)NCC(CC)NC(c2cc(C)sc2Br)=O)CC2(CCCO2)C1 7305,C(=O)(C1CCCn2cnnc21)NCn1cc(CCN(C)C)nn1.C1(C)CC1C(=O)O 7306,CC1CCCC=C1C(=O)N1CC(CNC(=O)CCC(=O)N(C)C)CC12CCC2 7307,C(CC#CC)(C(=O)NC1CCCSC1)NC(C1CC(CC=C)C1)=O 7308,c1(N2C(=O)CC(CC=CCNC(C=CCOCC)=O)C2)ccc2c(c1)SCCN2 7309,c1(Nc2ccc(-c3scc(C)c3)s2)ncnc2c1c(Br)cn2C 7310,N1(C(C2CC(C)OC2=O)=O)C2CCCC1CN(C(=O)C=CC1CCC1)C2 7311,c1(COC)cc(C(=O)N(C(C)CN(C(=O)CCCC2CCCO2)C)C)ccc1F 7312,O=S1(=O)CCC1c1ccc(CNC(=S)Nc2ccccc2)[nH]1 7313,C(=O)(C1=C(CN(C(C)(C)C)C(=O)OC(C)(C)C)NC(=O)NC1c1ccco1)OC 7314,c1(C(=O)NNC(c2cc(Br)cc(Cl)c2F)=O)ccc2ncnc(O)c2c1 7315,N(C1CCCc2cc(F)cc(Br)c21)Cc1ccc([N+](=O)[O-])c(Br)c1 7316,CC1(C)C2CC(C(=O)NCC(CO)NC(C3(F)CCCOC3)=O)CC12 7317,C1CCC(NC(c2cnc(C3CC3)o2)=O)CC1.C12(C(=O)OC)CC(NC=O)(C1)C2 7318,N1(C(C2C(CNC(Cn3c(=N)nc[nH]3)=O)CC2)=O)CC2CCCC2C12CC2 7319,N1(C(C(CC)OC)=O)CCN(C(C2(C#N)CC2(C)C)=O)CC1C 7320,c1(C(=O)NCCNC(C23C=CC(CC2)C3)=O)cccc2occc12 7321,C1(C(=O)NCC2C(NC(c3n(C=C)nnc3)=O)CCC2)SC2C=CC1CC2 7322,Cc1ccc2ncc(C#N)c(N3CCN(C4CCOC4)CC(C)C3)c2c1 7323,CCS(=O)c1ccccc1C(=O)NC1CN(C(c2cn[nH]c2)=O)CC1C1CC1 7324,C12CN(C(=O)C=CC(F)(F)F)CCN1C(=O)CONC2=O.CCC.OC 7325,CCCCC(C)CCC(=O)NOC(CC(C)C)C(=O)NC1CC2(CCCCCC2)C1 7326,c1(CN2CC(NC(C(CC)Cc3ccccc3)=O)C2)cc(OC)cc(C)c1 7327,N1(C(CC2C(C)CCO2)=O)CCC(CNC(=O)CCCC(N)=O)C(O)C1 7328,c1(C(C)N(C(C2(c3ccccc3)CC2C(=O)O)=O)C(C)C)cnc2ccccn12 7329,C=CC(C)(C)CC(=O)N(CC)CC1CCCN(C(C)=O)C1 7330,c1(C(=O)NCC2(COC)CN(C(C3(C)CCCN3C)=O)C2)c[nH]ccc1=N 7331,c1(CC(=O)NC2CCN(C(=O)CCC3CCCOC3)CC2)ccc(O)nc1 7332,N1(C(C2C(C(N)=O)C2)=O)CC2CN(C(c3ccc(O)nc3)=O)CC2C(F)(F)C1 7333,N1(C(=O)OCc2ccccc2)CCN2C(=O)OCCC2C1.c12cc(c[nH]1)C2=O 7334,S(=O)(=O)(c1ccc2[nH]c(=NCC3CCN(C)C3)ccc2c1)NC1(COC)CCC1 7335,C1(CC=C)(C(=O)NCC2COCC2NC(=O)C(N2CCOC2=O)C)CCCC1 7336,C(=O)(C1CCCc2cc(O)ccc21)N1C(C)(CNC(CNC(=O)OC)=O)CCC1 7337,C(=O)(N=c1ccc2nnc(-c3ccccc3)n2[nH]1)c1cccc(C2C(OC)CC2)c1 7338,N1(C(CN(CCC#C)C2CC2)=O)CCCC(C)C1CNC(=O)CCNC(=O)CO 7339,c1(CCNC(C2C(CC)CN(C(=O)C(=O)NC3CC3)C2)=O)cc(C)ccc1F 7340,C1(CNC(C2CN(S(N)(=O)=O)C2)=O)C2CCCC1N(C(c1csc(Cl)c1)=O)C2 7341,CC(C(O)C(=O)NC1C=CCC1)c1ccccc1F 7342,CCCCCCC(=O)NC(Cc1cn[nH]c1)C(=O)NC(C)CC1CCCO1 7343,c1(CN(CC(C)C)C)ccnc(NC(C(c2ccon2)N(C(C)=O)CC)=O)c1 7344,C(=O)(C(C)(C)S(C)(=O)=O)NC1CC(NC(C2(C)C(C)CCC2)=O)C1 7345,c1(C(=O)NC(c2cnoc2)CNC(CC2C(CC)C2)=O)cc(=O)c(OC)cn1C 7346,C1(CNC(c2c(CC)cc[nH]2)=O)CN(C(=O)Cc2ccc(Cl)cn2)CC12CCC2 7347,C1(CNC(C2(c3ccccc3)CCOC2)=O)CCN(C(=O)CC2(O)CC2)C1 7348,N1(C(CN(CCOC)C)=O)CC2CC(NC(c3c(C)nn(C)c3Cl)=O)C(C2)C1 7349,N1(CC)C(=S)NC(c2cc(OC)ccc2Br)C2=C1C(C)CN(C)C2=O 7350,Cn1ccnc1C(F)(F)C(=O)NCC1CC(CNC(=O)CSC(F)(F)F)CO1 7351,N1(C(c2c(CC)noc2)=O)CC(C)(C)CCC1CNC(C1CC(=C(F)F)C1)=O 7352,C(=O)(C1=CCCN(C(c2cc(O)nc(O)n2)=O)C1)NC(c1cncs1)C 7353,C1(C(=O)N)CCN(C(=O)C(C2CC2)C2CC2)CC1.CC1(N2CCC2)CCC1 7354,c1(C(=O)NCC(=O)NC(C)CC2CCCCO2)ccc2cc[nH]c2n1 7355,C(C(=O)N(C1CN(C(=O)CC2CC(=O)NC(=O)C2)CCC1O)C)(C(C)(C)C)OC 7356,C1(CCNC(c2ccsc2-n2cnnn2)=O)CCCCN1C(c1nocc1Cl)=O 7357,C12(C(N(C)CC3COCCO3)=O)CC(CO1)N(C(C1CC3CC(=O)C1O3)=O)C2 7358,C(CCCC(CO)NC(=O)CCc1cn(C)cn1)NC(C1OCCC(C)C1)=O 7359,C1CC2CC2N1C(=O)CC1NC(=O)NC1=O.C1CCC(=O)N1.NC(=O)NC 7360,C1(CNC(C(C2(O)CN(C(COCCCC#C)=O)C2)F)=O)CC=C(C)CC1 7361,N1(C(c2nc(COC)oc2)=O)CCC2(C1)CN(C(=O)CCC(C)C)C2 7362,C(C(F)C(=O)NC(C(C)C)C1CC1)N(CC)CC.C12(CC1)N(C)C2=O 7363,N1(C(=O)C(n2cccn2)C2CC2)CCCC1CC(F)(F)F.n1(CCN)ccnc1 7364,CC1(C)CC(CC(N2CCCC2(C)CNC(c2coc(Cl)n2)=O)=O)CO1 7365,O=C(C1CCc2ccccc21)NC1CCC1NC(C1C2(CCC2)C12CCC2)=O 7366,C(=O)(CC(CC)C(F)F)N1CCC(NC(CC(C=C)C)=O)C(O)C1 7367,c1(C(N2CCN(C(CC3CC(OCC)C3)=O)CC2C)=O)ccc2c(c1)CCCS2 7368,Cc1ccc(OCC(=O)NCC2CCCCC2NC(c2nnc(C)s2)=O)c(C)c1 7369,c1(C(N2C(C(C)NC(C(CSC)C)=O)CCC2)=O)nc2ncc(C)cn2n1 7370,Cc1c(-n2cc(C3CCN(C(=O)CC(C)C4CCCO4)C3)nn2)cccc1F 7371,c12cccc(c1)N2.C1(NC(=O)NCCC(N)=O)CCC(NC(=O)CSC(F)F)C1 7372,C1(C(=O)NC2CCOCC2)CCCCC1NC(C1CC=CC1)=O.c12ccccc1O2 7373,Cc1ccc(N)cc1C(N1CCCC(F)(CNC(=O)CNC(=O)CC(F)(F)F)C1)=O 7374,CCC(CC(C)C)C(=O)NC1(C)CC(C(=O)NC(C2CCCCC2)CO)C1 7375,CC1C(O)CC2CCC1N2C(=O)NCCC1C(CC(=O)NC(C)(C)C)CCCC1 7376,C1(NC(CC(C)c2ccncc2)=O)(CO)CCN(C(C2(CO)CCC2)=O)C1 7377,C(=O)(C(F)C(=O)N1CCC(NC(=O)CC=C(C)C)C1C(C)(C)C)OCC 7378,c1(NC(=O)CCCCN2CCOCC2)ccc(NCc2ccc(F)nc2F)cc1F 7379,c1(N(C(C2CC2c2ccc(Cl)cc2)=O)CC2CC2)ccccc1Cl 7380,C(=O)(CCC(F)(F)F)NCCC1C(C)CN(C(=O)C(C)(C)c2ccccn2)C1 7381,C(C(=O)N1CCN(C(c2cc(SC)c(C)o2)=O)CC1C)(C(C)(C)C)SC 7382,n1(CC(N2CC(NC(C(C)CC(F)(F)F)=O)C(C)(C)C2)=O)nc2n(c1=O)CCOC2 7383,C(=O)(C1CCCc2nc[nH]c21)N(CCCNC(c1cc(OC)nc(OC)c1)=O)C 7384,C1(C2CCCN(C(=O)C3=CCCS3)C2)(NC(C(C(C)C)OC)=O)CC1 7385,Cc1cc(C(=O)NCC(O)CNC(C2(S(N)(=O)=O)CCCC2)=O)ccc1[N+](=O)[O-] 7386,C1(CNC(c2c(CCC)nco2)=O)CC(NC(c2cnn(C)c2N)=O)C12CCC2 7387,N1(C(Cc2ccn(CC)n2)=O)CC2(COC(CNC(C3CC(C4CCC4)C3)=O)C2)C1 7388,C(CCC(C(=O)NC1CC1)N1CCN(SCC(=O)OC)CC1)OCC=C 7389,c1(C(=O)NCCC2(OC)CN(C(c3ccnn3CCF)=O)C2)cnnc(C)c1 7390,C(=O)(CCCCC(C)CC)NCC(CN(C(C1CC(CCC)OCC1)=O)C)C 7391,C1(SC)CN(C(c2oc(C)cc2C)=O)CC1NC(C1(c2cc[nH]n2)CCOCC1)=O 7392,N1(C(c2c(C)occ2)C(=O)NC(C)C)CC2OCCC2C1 7393,c1(C(=O)NC2C(CNC(C=COCC)=O)COC2)ccc(F)cc1Cl 7394,CC1CN(C(c2cn(CCC3CC3)nn2)=O)CCN1C(C1CC1CC1CCOC1)=O 7395,C(=O)(CC(C)C(=O)NCC1(CNC(c2ncc(Br)cn2)=O)CCCC1)OC 7396,CC1CN(C(=O)C=Cc2cn(C)cn2)CC(C)C1N=c1nc[nH]n2cccc12 7397,c1(C(=O)NC2C=CCN(C(c3c(CC)c[nH]c3)=O)C2)c(C)nc(O)nc1C 7398,C1(C)(C(=O)NC(CC)C(=O)N(C)C)CCCN1C(c1cc(C#N)c[nH]1)=O 7399,Cc1ccc(C2CC2C(N2CCC(C)(CNC(=O)C=C3CCC(C)C3)C2)=O)c(F)c1 7400,C(=O)(CCP(C)(C)=O)NC1CCC(NC(Cc2n[nH]c(=NC)s2)=O)C1 7401,C1(CNC(C2C(C)CCC2)=O)CCC2(CCN(C(=O)C#CC(C)(C)C)CC2)CO1 7402,C1(CNC(CC#N)=O)CC2(CC(NC(c3ccccc3C(F)(F)F)=O)C2)C1 7403,Cc1nn(C)c(=O)c(C(=O)N(C)CC2(NC(C3CCCS3(=O)=O)=O)CC2)c1C 7404,n1(CC)nnnc1C(c1cc(COC(C)(C)C)no1)NC1CCCC1C(=O)OC 7405,N1(C(C(c2ccc(OC)cc2)C)=O)CCOC2(C1)CN(S(=O)(=O)CCCCl)C2 7406,N1(C(CCCN(C(C(CCC)N(C)C)=O)C)=O)CCOCCC1C 7407,N1(C(CC=CCC)=O)C2CCC1CN(C(C1(CO)CCC(C)C1)=O)C2 7408,C(=O)(CCCCCCn1cc(C=CCC)nn1)N1C(CN2C(C#C)CC2)CCC1 7409,CCC(O)C(F)(F)C(=O)NCC1CC(F)(CNC(C2CCCN2C2CC2)=O)C1 7410,C1(C(=O)NC2CCCN(C(c3cncc(CC)c3)=O)CC2)CC(C2CCCC2)C1 7411,c1(CN(C(C2(CNC(c3cnc(C)cn3)=O)CC(=C)C2)=O)C)ccccc1C 7412,C(=O)(N1Cc2ccccc2CO1)C1(NC(c2cc(C(C)C)on2)=O)CC1 7413,c1(C(=O)NCC2N(C(COC(CC)C)=O)CC(O)C2)cc(F)cc(F)c1 7414,C1(CC(=O)O)CN(C(=O)CCn2cnc3c(N)ncnc23)Cc2ccnn2C1 7415,C1(NC(C=CC(C)NC(C(c2ccc(C)o2)C)=O)=O)CCOCC1C 7416,CCC(CNC(=O)CCCC1CC1C)(CC)C(=O)NC1(C)CCC(C)(C)C1 7417,N(C(=NCc1cn[nH]c1)N1CCCC(NC(=O)C2CC2)C1)CC(C)(C)C 7418,C1(CCC)(C(=O)NCC(C)CN(C(=O)Cn2cc(C(C)=O)nn2)C)CC(F)(F)C1 7419,C1(NC(C(CC)CC)=O)CCN(CC)CC1C.C12CC(CCO1)NC2=O 7420,C1(CN(C(c2ncc(C)cn2)=O)CC)CCCCN1C(C1CC(SC)C1)=O 7421,C1(CCC)(NC(=O)C#CC(=O)N(C)C)CCCN(C(C)=O)C1 7422,N1(C(CC2(NC(C)=O)CC2)=O)CCCCC(CC(=O)N(C2CCSCC2)C)C1 7423,C12(C(N3CC(NC(C(C)(C)SC)=O)(CO)C3)=O)C3C4C1C1C2C3C41C 7424,c1(CC)cc(O)ccc1C(=O)NCC1COCCN1C(=O)C(n1ccnc1C)C 7425,C1(NC(C2(NC(c3ncccn3)=O)CCN(C)C2)=O)CC2(CCCO2)C1 7426,n1(C2CCN(C(CC(CC)CC)=O)CC2)ncc2c1CN(C(c1csnn1)=O)C2 7427,N1(C(C(C)(C)CC#N)=O)CCC2(C(N3CCCOCC3)=O)CCCC12 7428,C(C(C(=O)N1CC2CC(NC(=O)C(C)(C)COC)CC2C1)C(F)(F)F)OC 7429,c1(C(=O)NC2CC(N(C(c3cc(C(C)=O)c(C)o3)=O)C)C2)cc2c(s1)CCCC2 7430,C12(C(N3CC(C(C)NC(=O)C=CC4CCC4)OCC3)=O)CCC(CO)(CC1)CC2 7431,CC1(C)CCC(CC(=O)NCCC(O)CNC(=O)CN2C(=O)CNC2=O)CC1 7432,c1(CNC(N(C(C)C)CCc2cccs2)=O)cnc2n1CCC2 7433,C#Cc1ccc(N(C(=O)CCOC(C)=O)C)cc1.C12CCC(CC1)CNC2=O 7434,N(C1CCCc2n[nH]cc21)C(C1C(CC(=O)N(C)Cc2cncn2C)CCC1)=O 7435,C1(F)(C(=O)NC(CC(C)NC(C(CC)(C)C#N)=O)C)CCC(F)(F)CC1 7436,C(=O)(C(C)CCC(C)(C)C)NCC(C)CNC(C1(c2cccnc2)CC1)=O 7437,c1(C(C(=O)NC(C)CCNC(=O)C(C)N2CCCC2)O)cccnc1 7438,c1(C(N)=O)ncc(C(=O)NC2CCCC2NC(C2COCCO2)=O)s1 7439,CCC1=NOC(C(N2CCOCC2C(=O)NC(c2nc[nH]n2)CC)=O)C1 7440,c1(C(N2CCOC(CNC(C34CCCC(C3)OC4)=O)C2)=O)ccc(F)c(O)c1 7441,CC1CCC(C(=O)N(C2CC3CC3C2)C)N(C(=O)Cc2ccon2)C1 7442,N1(C(C(C)(C)OCC)=O)CCC(C)(CNC(=O)CCc2cccc(F)c2F)CC1 7443,C1(F)(CNC(CC2C(C)C2)=O)CN(C(=O)C(C2CC(F)(F)C2)O)C1 7444,CC1(C)CN(C(C2CC(CCNC(c3coc(C4CC4)c3)=O)C2)=O)CCC1CO 7445,C1(C(=O)NCCCNC(c2c(C)c(Br)sc2)=O)CCCCC(C)(C)C1 7446,c1(SC)cccnc1C(=O)NC(C)(CNC(=O)CCC1C(=O)NN=C1C)C1CC1 7447,N1(CC)CC2CCCC2C1C.c12cncc(c1)C(C)NC(=O)N2 7448,CP(C)(=O)CC(=O)NCCCN(CCCNC(=O)CC1CCCCCC1)C 7449,CC(C)(C)CC(F)C(=O)N1CCC(Cn2cc(C3(CCO)CC3)nn2)C1 7450,c1(OCCC(N2C(C)CC(NC(CN(S(C)(=O)=O)C)=O)C2)=O)ccc(F)nc1 7451,CC1(C)CCC(C(=O)NC2CC(C(F)C(=O)NCCOCC3CC3)C2)C1 7452,N1(C(C2(O)CCN(C(C(C)NC(C)=O)=O)C2)=O)CC2CC1CC2(F)F 7453,C1(CNC(Cn2cc(CC(=O)NCCOC)nn2)CC(C)C)(CO)CCCCC1 7454,C12(NC(C3C(CC)C3(F)F)=O)COC(C1)C(NC(c1cnn(C)n1)=O)C2 7455,c1(C(C)(C)C)cnccc1NC(C1CS(=O)(=O)C1)=O 7456,CC1CN(C(=O)C(=O)NCc2cn(CC3CCCO3)nn2)CC1(C)CO 7457,N1(C(C2CC(=C)C2)=O)CCCC(C2CN(C(c3cc(O)n(C)n3)=O)C2)C1 7458,c1(CNC(C(SC)SC)=O)ccc(CCF)cc1.C12(CC1)CC(=O)N2 7459,Cc1n[nH]c(C)c1C(=O)N(C)CC1(O)CN(C(=O)C(C)(C)C2CCOC2)C1 7460,CCC(C)(C)CN(C(=O)Cc1cccs1)CC.c1(C(=O)NCC)cccnn1 7461,C1(NCC(CCC)CCC)CCc2nc(C(F)(F)F)cn2C1 7462,C(=O)(C1=CC2CCCC12)N(CC(CNC(c1cccc(SC)n1)=O)C)C 7463,Cc1nc(N2CCN(C(=O)COC3CC3(F)F)CC2)c2scc(C)c2n1 7464,CC1C2C(CCN2C(C2CC(=O)CC23CCC3)=O)CN1C(=O)CC1CCCN1C 7465,Cc1cc(C(=O)NCC(O)CN(C)C(C2OCC3CCCC23)=O)ccc1Cl 7466,N1(C(COCc2ncc(C)o2)=O)CCCC(C(C)NC(c2ncncc2Cl)=O)C1 7467,CC(C)C(C)(O)CN1CCC1CNC(=O)C(=O)NC(c1nc(Cl)cs1)C1CC1 7468,c1(CN2C(C(=O)Nc3cc(OC)cc(C)c3)CC(F)C2)c(C)cc(O)cc1O 7469,CCC(CC)C(C(=O)NCC1(CNC(c2cnn(CC)c2)=O)CCOCC1)OC 7470,c1(C(C)C)[nH]nc(C(=O)NC(CNC(=O)CCC2CCCO2)CO)c1[N+](=O)[O-] 7471,C1(CCC(=O)NCC(C)=CC(=O)NCc2cccc(Cl)c2)CCCN(C)C1 7472,c1(N(C)C)cc(F)ccc1NC(=O)C(C)(C)NC(C1C2CC(=O)CC12)=O 7473,C12(CNC(C(CCOC)C)=O)CN(C(c3c[nH]nc3C3CC3)=O)CC1CCO2 7474,N1(C(=O)CC2CCC3CC23)CCCCC1C1CCCN1C(=O)CC1CS(=O)(=O)C1 7475,C1(CNC(=O)CC2(CNC(C3CC3Cl)=O)CC2)CCC(O)C1 7476,c1(C(N(CCC(C)NC(=O)Cc2cnn(C)c2)C)=O)ccc2nccnc2c1 7477,c1(N(C2C3CCC2CNC3)C(CNC(=O)OCC)=O)cc2c(cn1)OCCC2 7478,CC1=C(C(=O)NC2CN(C(c3ccc(C)nc3)=O)CCC2C(F)(F)F)CCO1 7479,C(=O)(C1CCc2c[nH]nc21)N1CCC(C(C(=O)NCCC(C(=O)OC)(C)O)C)CC1 7480,C#CC1(C(=O)Nc2cnc(C3CC3)nc2)CCN(C(=O)CC=C(C)C)C1 7481,C1(C(N(C)Cc2cncnc2)=O)COC2(C1)CN(C(=O)CCC1CCOC1)C2 7482,N1(C(c2c(CC)nco2)=O)CCOCC(NC(c2cc(C(C)(C)C)n(C)n2)=O)C1 7483,c1(C(=O)NCC2(CCNC(=O)COCC3CC3)CCCC2)ccc2cccnn12 7484,C(=O)(CCCN(C)C)NCCCOCCC(=O)NCC(c1cncnc1)C 7485,N1(C(CCNS(CC)(=O)=O)=O)CCC(C2CC2NC(C2CC=CCC2)=O)CC1 7486,Cc1c(C(=O)N(CCC(C)NC(C2CCN(C(N)=O)C2)=O)C)ccn1C(C)C 7487,C12(C(=O)NC(CNC(c3ccc(N)c(Cl)n3)=O)CO)CCCCC(=O)N1CCC2 7488,CCC(C)(CCNC(=O)C(C)N1CCCC1)NC(=O)CC1CC=CCN1C 7489,C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)NCCCC(C)NC(C(C(=O)OCC)(C)C)=O 7490,N1(C(C(CCC)C)=O)CCC2CC(N(C(=O)OC(C)(C)C)CC)C2C1 7491,N1(C(c2c(Cl)sc(C)c2C)=O)CCC2(CC1)COC(CNC(c1cnsc1)=O)C2 7492,C(CNC(C1CC12CCCC2)=O)(CC(=O)N1CCOC(CO)C1)OC 7493,C1(NC(C2(C#C)CCCC2)=O)CCC(C)(NC(=O)C(N2CCSCC2)C)CC1 7494,N1(C(C(=O)NCCN(CC)Cc2ccc(CCC#N)nn2)C)C(C)CCC1C 7495,C1(CN(C(CCC=C(C)C)=O)C)C2CN(C(c3nocc3C3CC3)=O)CC12 7496,N1(C(C2ON=C(CC)C2)=O)CCCC12CCN(C(c1cccc(=S)n1O)=O)C2 7497,C1(NC(CCOCC#C)=O)CCN(C(=O)NC(C)(C)C)C(C2CC2)C1 7498,c1(C(CC)=O)cc(C(=O)N(C2CC(NC(c3ncc(F)cn3)=O)C2)C)ccc1F 7499,N1(C(C(C2CCCN(C(C(CC)(C)C)=O)C2)(C)C)=O)CCC12CCCSC2 7500,Cc1cc(Cl)cc([N+](=O)[O-])c1C(=O)NC(C)CCNC(c1c[nH]nc1[N+](=O)[O-])=O 7501,CCCC(C)(CCC)C(=O)NC1CN(c2ccc(C#N)c(OC)n2)CC(C)(C)C1 7502,C1(C(=O)NCCCN(C(=O)CC2=CCCCC2)C(C)C)CCCCC12CC2(F)F 7503,C1(NC(c2c(SC)csc2)=O)CC2(C1)CC(NC(=O)C=CCN1CCCCC1)C2 7504,O=C(CC1=CCCCC1)N1CC2CCCC1(CNC(C1(CF)CCOCC1)=O)C2 7505,Cc1ccc(NC(=O)CCC2CCC(NC(c3c[nH]c(C)c3)=O)C2)cc1CO 7506,C(CC1CCC1)(C(=O)N(C(C)C(=O)NCc1coc(C)n1)C)OC 7507,c1(OC)c(C(=O)NC2CC(O)CN(C(C3CCN(C)CC3)=O)C2)cc(F)cc1F 7508,c1(C(N(CC(C)NC(=O)C2=CC(C)(C)C2)CC)=O)c[nH]c2cc(C#N)ccc12 7509,C(=O)(CC(F)(F)C(F)F)NCC(C1CCC1)NC(c1cc(C)sc1C)=O 7510,C(=O)(C(CC(C)C)N(C)C)N(C1CCN(C(c2csc(CO)n2)=O)C1)CC 7511,N1(C(c2n(C(C)C)ncc2)=O)CC2CCCC2(NC(=O)C(=O)NCC(F)(F)F)C1 7512,N1(C(CNC(CNC(C)=O)=O)=O)CCCN(C(C2(F)CCCOC2)=O)CC1C 7513,C1(NC(c2cccc(C(=O)NC)n2)=O)CCCN(C(=O)Cc2occc2C)C1C 7514,N1(C(Cc2c(C)nc[nH]2)=O)CCN(C(=O)Cc2cnns2)C(C2CC2)C1 7515,C1(C(=O)NCCN(C(=O)CC(C)(F)F)CC)CCCC(F)C1 7516,c1(C(=O)NC(C2OCCN(C(C(CCCC)O)=O)C2)C)ccc2nnn(O)c2c1 7517,N1(C(=O)CCc2nncs2)CCC(NC(C2(Cc3cnn[nH]3)CCC2)=O)C12CCC2 7518,C12(C(=O)NC3(CNC(=O)C4=CSCCO4)CCC3)CCCC1CS(=O)(=O)C2 7519,C1(C(=O)N(CC(O)CSc2cc(C)[nH]n2)C)CCCN1C(=O)OC(C)(C)C 7520,C1(C(=O)NCCN(C(=O)Cn2nnc(=N)[nH]2)C)CCC2(CC2)C1 7521,N1(C(c2cc(C)on2)=O)CC(C)OC2(CCN(C(=O)CC(C)C(F)(F)F)CC2)C1 7522,c1(C(N2CCN(C(c3cccs3)=O)CC2)=O)cnc(O)n(-c2ccccc2)c1=O 7523,C(CC(C(C)(C)C)NC(=O)CC1CC=CCC1)N(C)C(c1sccc1CO)=O 7524,Cc1ccc(Cl)cc1C(N1CC(C)C(C)(CNC(=O)CC2CC3(CC3)CO2)C1)=O 7525,C1(C(N(CC(C)N(C(C)=O)C)C)=O)CCN(C(=O)C(C)Cn2ccnc2)C1 7526,N1(C(CC2CCC(NC(c3c(C)occ3)=O)CC2)=O)CC2C(C1)C2(F)F 7527,C1(C(N2CC(C)(CF)C2)=O)CC2CN(C(C3CC3c3ccco3)=O)CC2C1 7528,c1(C(C2CC2)NCc2n(CCC)c(C)nn2)ccc(Cl)cc1F 7529,N1(C(C(C)S)=O)CC(NC(=O)CNc2cccnc2)CC2(CCC2)C1 7530,c1(C(=O)NCC2CCCC(CNC(C(C)N3CCC3)=O)C2)noc2c1CCCC2 7531,N1(C(C(C2CC2)SC)=O)CCCC(C)(C)C1CNC(C1CC(CC(N)=O)C1)=O 7532,N1(C(C(n2cc(Cn3c(C)ccc3C)nn2)C)=O)CCOC(C2CC2)CC1 7533,C(=O)(C(C)(C)S(C)(=O)=O)N1CC(CC)C(NC(c2ccc(S(C)=O)cc2)=O)CC1 7534,C1(C(C)C)C(=O)N1.C1(SCC(=O)N(C)CC)CC1CNC(=O)OC(C)(C)C.NC 7535,N1(C(C(C(C)C)OCC)=O)CCC2(CCC(NC(=O)C3=C(Cl)CC3)CC2)CC1 7536,CCC(C(=O)N1CCCC(C)(CNC(c2cnn(C(F)F)c2)=O)C1)C(F)(F)F 7537,Cc1nn(C)c(NC2CC(C)CC(C)C2)c1C#N 7538,N1(C(COCC(C)C)=O)CC(CNC(=O)COCc2ccncc2)CC1(C)C 7539,N1(C(c2cc3sccc3s2)=O)CCN(C(c2cc(CO)[nH]n2)=O)C(C(F)F)C1 7540,CCC(C)(CN(C)N1CC(O)CC1c1ccccc1N1CCOCC1)OC 7541,c1(C(=O)NCC2CN(C(CS(CC)(=O)=O)=O)CC23CC3)cnc2c(C)cnn2c1 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7560,c1(C(=O)NCC2CN(C(C3CC4CC4C3)=O)C2)cc2c(Cl)cccn2n1 7561,C12(C(N3CC(C(=O)NC)C3)=O)COC(C1)C(OC)C2.C12CN(CCO1)C2=O 7562,C1(O)(CNC(=O)COC2CCOC2)CN(C(c2nccs2)=O)C1 7563,C1(CC(=O)NCCCN(C)C(c2csc(Cl)n2)=O)CCn2cncc2C1 7564,n1(COC(C)(C)C)ncc2c1CCCC2NC(=O)NOCCc1ccccc1 7565,C(=O)(C(C)S(C)(=O)=O)NC1CC(F)(CNC(c2cc(C)nn2C(C)(C)C)=O)C1 7566,C1(S(C)(=O)=O)(C(=O)NCC(C2CCCC2)NC(c2[nH]cc(CC)c2)=O)CCCC1 7567,C12(COC)CC(C(N3CCC(n4cc(NC(=O)C(F)(F)CO)nn4)C3)=O)(CO1)C2 7568,CC(C)CC(C(=O)N1CCCC1CS(N)(=O)=O)C(N)=O 7569,N1(CC)N=C(C(=O)N2CCCCC2CCNC(C2CCC(=O)O2)=O)CCC1=O 7570,C1(C(=O)Nc2ncc(CC)cn2)C2CCN(C(=O)CC3CCSCC3)CC12 7571,N(C(=NC1CCS(=O)(=O)C1)N1CCC2(CC1)CC(C)=NO2)C(C#C)C(C)C 7572,N1(C(c2cnc(C)nc2)=O)CC(NC(=O)C=Cc2cc[nH]c2)C2(CC2)C1 7573,N1(Cc2ncc(C)cc2Cl)CCCc2sccc2C1 7574,c1(C(N2CC(COC)(CNC(=O)C(C)C3CCC3)C2)=O)cccc(CC#N)c1 7575,c1(C(N2CC(NC(C(C3CC3)OCC)=O)(CF)C2)=O)cc2ccncc2[nH]1 7576,CCC(C(=O)NC1CCN(C(c2cc[nH]c2)=O)C12CCC2)C(F)(F)F 7577,N1(C(CC(C(C)(C)C)NC(CC=CCCCCC)=O)=O)CCC2CN(C)CC2C1 7578,C(=O)(C(CNC(=O)CC(O)C1CCCC1)C(C)(C)C)NC(C1(O)CCC1)C 7579,C(=O)(C1=CCCN(C(=O)CC(F)(F)F)C1)N(CC(F)(F)Cl)C 7580,Cc1ccc(C(N2CCC(CNc3ncnc(Cl)c3F)C2)=O)cc1C 7581,CCN=c1[nH]c(CNC(=O)NCC2CC(O)C2(C)C)cs1 7582,Cc1cccc(C(=O)NCC2(CN(C)C(C3CCCC34CC4)=O)CC2)n1 7583,N1(C(C2CCC(C)(CC)O2)=O)CC2CC(NC(c3ccc(C)c(F)c3)=O)C2C1 7584,C(=O)(C(CC)CC(C)C)NCCC1N(C(c2cc(COC)oc2C)=O)CCOC1 7585,Cc1cc(C(=O)NC2CC(NC(C3(Br)CC3)=O)C2)[nH]c1C 7586,C(Cn1cncn1)(C(=O)NOCC1CCCO1)NC(C(C(C)C)SC)=O 7587,C1(C(N2C(C(C)C)COCC2)C(=O)NC2CCOCC2)CCOC2(CCCC2)C1 7588,n1(CC(=O)NCCN(C(C)C)C(C2OCC2(C)C)=O)cnc(Br)n1 7589,CC1(C)CCC(NC2CN(C(=O)C(=O)NC(C)(C)C)C(C)(C)C2)OC1 7590,N1(C(C(n2cc(C)nc2)(C)C)=O)CCC2(CCC2)C(NC(C2CCCC2O)=O)C1 7591,c1(CNC(C(CC)O)=O)ncccc1NC(=O)Nc1cccc(Br)c1 7592,c1(C(=O)NCCn2cc(CNC(C)(C)CO)nn2)cc[nH]c(=N)n1 7593,CC1C(C)N(C(=O)Cn2cncn2)CCN1C(C12CC(C)(C1)C2)=O 7594,c1(C(N2CCCC(CCNC(c3ncn(CC)n3)=O)C2)=O)cnc2cc[nH]c2c1 7595,C1(C(N2CCC(C(=O)OC)C2)=O)CCC=CCC1C(F)(F)F 7596,C(=O)(C(C(C)(C)C)c1ccccc1)N1CC(NC(CCCSC)=O)C(C)C1 7597,Cc1nc(NC(C2COCC2c2ccccc2F)=O)c(Cl)cc1C#N 7598,c1(C(N(CCC)CCNC(c2ccc(C)o2)=O)=O)cn(C)nc1C(C)(F)F 7599,CC1C(NC(=O)CCn2ccnc2)CCN1C(c1cnc(C(C)(C)CF)o1)=O 7600,C(C1CCOCC1)=CC(N1CCCC1C1CCCCN1C(=O)Cn1cnnn1)=O 7601,CCCC(O)CCNC(=O)CCC1CC(OC)C1 7602,Cn1ccc(=O)c(C(N2CCC(O)(CNC(=O)C(C)(C)c3cnc[nH]3)CC2)=O)c1 7603,c1(SCC(=O)Nc2cn(CC(=O)NCCc3onc(C)n3)nn2)cccc(F)c1 7604,N1(C(C=CC(=O)N(c2nccs2)CC(N2CCCC2)=O)=O)CCc2cccc(F)c21 7605,C1(C(C)C(=O)NCCn2cncn2)CCCN(C(C2SCCS2)=O)C1 7606,C1(N(C(c2c(C)occ2)=O)C)CN(C(=O)C(c2ccc(F)cc2)=O)CC12CC2 7607,c1(C(=O)O)cc(Br)c(S(=O)(=O)NCc2cnccc2C(F)F)s1 7608,C=C(Cl)CC(C(=O)NCC(C)(C)C1CC1)NC(C1CC(=O)OC1(C)C)=O 7609,c1(CC)noc(C(N2CCSCC2CCNC(c2cnc(C)nc2)=O)=O)c1C 7610,CC1C(C(=O)N(CCC(=O)N(C)CCN2CCCC2=O)CCO)=NOC1C 7611,c1(C(N2CCCOC(CCS)C2)=O)cnc2c(Br)c[nH]c2c1 7612,c1(N2CCCC(CNC(CCC(=O)NC)=O)C2)cc(-c2ccco2)nc(C)n1 7613,Cn1cnc(I)c1N1CCC(CNC(N2CCCCC2c2ncccn2)=O)CC1 7614,C(=O)(CC(F)(F)C(F)(F)F)NC1CCCN(C(C(C)Cc2ccccc2)=O)C1C 7615,C1(NC(C(CC)Cc2ccccc2)=O)C(C)CCN(c2cncc(Cl)n2)C1C 7616,c1(NC(c2c(NC(C(C)OC(C)C)=O)ccc(Cl)n2)=O)cc(F)c(F)cc1Br 7617,N1(CC=CC(=O)NC(C(=O)NC2CC(n3ccnc3)C2)c2cccs2)CC(CF)C1 7618,C1(NC(=O)OC(C)(C)C)CCSC12CN(C(=O)C(O)CN1CCCC1)C2 7619,c1(NCc2cn(CC)nc2)ccc(F)c(C(F)(F)F)c1.N12CCOCC1C2=O 7620,n1(CCOC(C)C)nc(-c2cccc(F)c2)nc1-c1c[nH]c(=O)cn1 7621,c1(C(=O)NCC=CCNC(C2C(C=C(C)C)C2(C)C)=O)cc(N)c(Cl)c(O)c1 7622,c1(C(=O)NCC(C)NC(C2CCN(C)C2)=O)cn2cccnc2n1 7623,C(CC(=O)NC(C1CC(NC(C2C=CCC2)=O)C1)C)OCCOC 7624,CC1(C)CCC(C(=O)NCCC2CCCN2C(c2cc(O)cs2)=O)C1 7625,c1(OC)ccc(CO)c(NC(C2CC2NC(=O)C(CC2CCCC2)OC)=O)n1 7626,Cc1ccc(C(N2CC3(C2)CN(C(=O)C(=O)N(C)C)CC3CO)=O)c(N=[N+]=[N-])c1 7627,c1(OC)cncc(C(=O)NC(C)C(C)NC(=O)CC2CCC(=O)O2)c1C 7628,Cc1c(C(N2CCCN(C(=O)C(C)(C)C3CC3)C2C(C)C)=O)nn2ccccc12 7629,CCCCCC(F)C(=O)N1CCC(C)C1C(N1CCN(CC)CC1)=O 7630,c1(NC(C)C)ccc(C(N2CC(CC(C)NC(=O)C(F)C(C)C)C2)=O)cc1 7631,C1(NC(CC(=C)C)=O)CCC2(CC1)CN(C(=O)C1=COCCO1)CCO2 7632,c1(C(N2CCC(F)(CNC(C(C3CCC3)OC)=O)C2)=O)sc([N+](=O)[O-])cc1Cl 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7827,CC1CCCCC1Cc1nc(C2CC=CC2)nn1CC(C)(C)C 7828,C=CC(C)(CC)C(=O)NC1CC(CNC(c2cc(NC)ccn2)=O)C1 7829,Cc1c[nH]nc1C(=O)NCCCN(C(=O)C(F)C1CCC1)C1CC1 7830,N1(C(CCCc2n(C)cnn2)=O)CCCC(C(C)(O)CNC(=O)CSCC#N)C1 7831,C1(NC(C2(c3c(C)cccc3)CC2)=O)CC2CC(NC(c3ccncc3O)=O)C1C2 7832,Cc1cc(Cl)ncc1CNC1C2CN(C(=O)CC3CCN(C)CC3)CC12 7833,CCC1=NOC(CNC(=O)Nc2ccnc(OCCO)c2)C1 7834,Cc1nc(C)n(CC(=O)NC(CCN(C)C)C(=O)NCCCN=[N+]=[N-])n1 7835,c1(C(N2CCC(CC(C)NC(C3(C=C)CC3)=O)CC2)=O)ccc(F)c(Cl)c1N 7836,C1(NC(CC(CCC)C)=O)CN(C(c2nc(Cl)ccc2Cl)=O)C2CCCCC12 7837,C(c1ncc[nH]1)=CC(=O)NC(C)(CNC(=O)CCNC(=O)CO)C1CCC1 7838,C12(C(=O)OC)C(C)(C1)CNC(=O)NC1N(CCC1)C2.C(C)(C)(C)OC 7839,c1(C(=O)NC(CCC=C)C(=O)N2C(CC)CCC2C)cccn2nccc12 7840,N1(C(C(n2c(C)ncc2)C)=O)CC(NC(=O)CC(F)(F)C(C)C)CC12CCC2 7841,C1(CN(C(CC(=C)Br)=O)C)CCN(C(C2CCCC(OC)C2)=O)CC1 7842,c1(NC(=O)NCC2C(C)(C)COC2)cc(F)cc2ncoc12 7843,Cn1c(O)nc2cc(C(=O)N(C3(C)CCOC3)C(C3CCCO3)CC(N)=O)ccc12 7844,c1(C(=O)NC(C(=O)NCC(CCC)OC)COC(C)C)ccsc1C#N 7845,N1(C(CC2(OC)CCC2)=O)C2CCCC1CN(C(C1CC(O)C1)=O)C2 7846,n1(C(CC)CC)nccc1C(=O)NCC(C)(C1CC1)NC(=O)C(CO)N(C)C 7847,c1(C(=O)NCCCC2N(C(C3CCN(C)CC3)=O)CCC2)n[nH]c2c1CCC2 7848,C(CC(C)(C)C)(C(=O)N1CC=CC1C(=O)NCCC(C)(C)OC)OC 7849,C(C(C)(C)C#CC(=O)NCCOC1CCCCC1)NC(C1(CC)COC1)=O 7850,c1(OS(Cc2cnc(C=C(C)C(=O)O)s2)(=O)=O)sc2ccccc2c1Cl 7851,C=CCC(C)C(=O)NCC(CCCC)NC(=O)C(C)NC(C1CCCCC1)=O 7852,Cc1c(F)ccc(C(=O)NC23CC2CN(C(C2CCC(C(C)C)CC2)=O)C3)c1Cl 7853,N1(C(COC)=O)CCN(C(=O)CP(C)(C)=O)C(CO)C1 7854,Cc1cc2[nH]c(C(=O)NC3CC4CC3N(C(=O)CC3(O)CCC3)C4)cc2o1 7855,N1(C(C=CC(C)C)=O)C2CCC1C(N(C1CC3CNC1C3)C(=O)NC(C)(C)C)C2 7856,C1CCN=C2C=CC(=CN2)C(=O)O1.c1(CCO)cccc(Br)c1 7857,Cc1nc(F)ccc1NC(C1C=CC(NC(=O)CCCC#N)C1)=O 7858,N1(C(c2ccc(CC)cc2)C(=O)NC(C)(C)CC)CC(C)OC2(CCC2)C1 7859,c1(N(CCCNC(c2ccc(O)nc2)=O)C)ncnc2c1cnn2C 7860,C1(C(C)(CNC(=O)NC(C(=O)O)C2CC2)OC)CCOCC1 7861,CC(C)CCC(CO)NC(C1CC(NC(=O)CCc2cnoc2)C(O)C1)=O 7862,N1(C(C2C(C)CCN(C(CCC=CC(C)C)=O)C2)=O)CC(C)(CO)CC1(C)C 7863,C1(NC(c2ccc(OC3CCC3)cc2)=O)CN(C(c2ccccn2)=O)CC12CC2 7864,N1(Cc2c(C#C)cc(Br)cc2)CC2CCC1CN(C(c1cc(C)ccc1Cl)=O)C2 7865,C1(NC(c2cc(OCC)ncc2)=O)CCN(C(c2sc(C)cc2Cl)=O)CC1C 7866,C(=O)(C(C)CC(F)F)NCCC(C)NC(c1ccnc(OC(C)(C)C)c1)=O 7867,Cn1c(C(N2CC(O)(C(F)C(=O)NC3CC(=O)N(O)C3)C2)=O)ccc1C#N 7868,CC1CCCC1(O)CNC(C12CC(CN1C(c1coc(N(C)C)n1)=O)C2)=O 7869,c1(C(=O)NC2CCCN(C(C3CN(CC)C(=O)C3)=O)C2)ccc2c(c1)CCCN2 7870,C1(OC)CCC12CC(C(=O)NC13CC(NC(=O)CC4CCOC4)(C1)C3)C2 7871,C(c1cnn(C)c1C)=CC(N1C(CNC(C(CCC)F)=O)CC(O)C1)=O 7872,C(=O)(C(C)S(N)(=O)=O)NCC1CC(F)(CNC(C2(OCC)CCCC2)=O)C1 7873,N(C(=NCCC(=C)C)NC1CCN(C(c2cccnc2)=O)CC1)CCC(=O)N(C)C 7874,N1(C(CC(C(C)C)c2ccon2)=O)CC2CCC1C(CNC(C1(CO)CC1)=O)C2 7875,c1(C(=O)NCC2C(C)CN(C(C3(CO)CC3)=O)C2)ccc2c(O)ncnc2c1 7876,C(=O)(C1=CC2(CCOC2)C1)NCCN(C(=O)CCc1cnc[nH]1)C 7877,c1(CNC(C(CC)SC)=O)nc(CNC(C2CCC3CC2CO3)=O)cc(O)n1 7878,c1(CC)cnc(C(=O)NC2CCC(C(=O)N(C(C)CC(C)C)C)C2)nc1 7879,Cc1cc(=NC(=O)C(=O)NC2C(CNC(=O)CC3NC(=O)CNC3=O)CC2)[nH]o1 7880,C=CCS(=O)(=O)CCn1cc(C(C)NC(=O)C(=O)Cc2ccccc2)nn1 7881,C1(NC(C2(C)CC=CC2)=O)CC2CCCC(C1)N2C(c1cnc(Cl)s1)=O 7882,O=S(=O)(c1c[nH]c2cc(Cl)ccc12)N(C1CC2CCC(C1)O2)c1ccccc1 7883,N1(C2CCN(C(C3CN(C)C3)=O)CC2)Cc2cccnc2N2CCCC2C1 7884,C1(CCNC(C2C(CC(C)C)C2)=O)CN(C(c2c(Cl)cnn2C(C)C)=O)CCO1 7885,c1(NC(=O)CN2CCCC(CN3CCCNS3(=O)=O)C2)ccccc1[N+](=O)[O-] 7886,N1(C(c2cnc(CCCC)s2)=O)CCCC(C)(NC(=O)CC(C)(C)OC)C1 7887,c1(C(=O)NCC(CCCC)NC(C2(C)CCCS2)=O)cc(F)c2c(c1)CCC2 7888,c1(CCC(=O)NCC(C)(C)NC(C(CSC)OC)=O)nc2ccccc2o1 7889,N1(CC)CC(NC(=O)C(C(C)(C)C)NC(=O)C=Cc2nnn(C)n2)CCC1=O 7890,C1(n2cc(C(=O)NC3(C(=O)O)CC3)nn2)CCC(C(=O)NC2CC23CCC3)CC1 7891,C(=O)(C(CCNC(c1cccn1C1CC1)=O)OC)N(C)CC1CC(=C)C1 7892,N1(C(C(C2CC=CCC2)NC(C=CCOCCOC)=O)=O)CC(=O)NC(C)C1 7893,N1(C(COC(C)(C)C)=O)CCC2C(NC(=O)COC(F)(F)F)C2C1 7894,N1(C(C2C(C(=O)OC)C2)=O)CC(C(=O)NC2CCN(C(N)=O)C2)C2(CC2)C1 7895,C(=O)(C(CCSC)NC(=O)CC(C)O)N1CC(O)(CC)C1 7896,c1(COC)nc(C(=O)NCCN(C(=O)CN(C2CCSC2)C)C)cs1 7897,C1(O)(C(N2CCCC(CNC(C(CC)N3CCCC3=O)=O)C2)=O)CCCCCC1 7898,C1(NC(C2ON=C(C)C2)=O)CCCC2CN(C(c3csc(C(F)F)c3)=O)CC12 7899,CC1(CC(=O)NCC2CC=CC2)CCN(C(=O)CC2NC(=O)NC2=O)C1 7900,c1(C(C)C)ccc(F)cc1C(=O)N(CC(C)NC(c1cc(F)ccc1O)=O)C 7901,N1(C(CCOC(C)=O)=O)CCN(C(=O)CCN(CCC(C)(C)C)C)CC1CC(F)F 7902,C12(C(N3CC(CNC(C(C)OCCN(C)C)=O)C(C)C3)=O)CCC(C1)C(C)(C)O2 7903,c1(C(N2C(CNC(CCCN(C(C)=O)C)=O)CCC2)=O)ccc2nc(O)[nH]c2n1 7904,N1(C(Cc2cn(C(C)C)nc2)=O)CC=CC(NC(c2cnc(Cl)s2)=O)C1 7905,C(CC(C(C)(C)C)NC(C1CCCN1C1CCCCC1)=O)N(C(C)=O)C 7906,N1(C(CCOCC(C)C)=O)CC2(CCCC2)C1C(=O)NC(C1(O)CCC1)C 7907,N1(C(CNC(C(C)(C)C)=O)=O)CCC(N=[N+]=[N-])(C(=O)NCC2(O)CCCOC2)C1 7908,C1(OC)COCC1n1cc(CC2CN(C(C3CC(O)C3)=O)C2)nn1 7909,C1(N(C(COCc2c(C)occ2)=O)C)C2CN(C(c3cc[nH]c(=N)n3)=O)CC12 7910,c1(C(=O)NC(CNC(CC2C(C)=NOC2=O)=O)CC(C)C)nc(O)nc(O)c1N 7911,Cc1cc(CN2CCC(NC(C)C(F)(F)F)CC2)c(Br)cc1F 7912,CCC(C)C(O)CC(=O)NC(CNC(=O)CCCCN(C)C)CC(C)C 7913,C1(NC(C=C(C)C(F)F)=O)CCC(C(=O)NOCc2ccc(C)o2)C1 7914,c1(OC)ccc2cc(C(N3CCC(NC(c4cnc(=N)[nH]c4)=O)C3C)=O)[nH]c2c1 7915,C=CC(O)C(=O)N1CCC(C2CCCN2C(=O)CCc2cnccn2)C1 7916,N1(CC)CC(C(=O)NCC2CCCC2NC(=O)CC2CCCOCC2)CCC1=O 7917,N1(C(C(CC=CC)NC(=O)CC2(O)CCCC2)=O)CCC12CCCSC2 7918,C1(C)(CNC(c2nc(C(=O)OC)oc2)=O)CCCN1C(c1cnn(C)c1F)=O 7919,Nc1ccc([N+](=O)[O-])cc1C(N1CCC(C2(NC(=O)C3=NOCC3)CC2)C1)=O 7920,C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NCC1C(CNC(c2cc(C)c(Cl)cn2)=O)C1 7921,C(=O)(C1=CC(C)(C)C1)N(C)CC1CCN(C(c2cnc(C)nc2)=O)CC1 7922,C(=O)(C(C)(C)C(=O)NCC(C)CNC(c1cn(-c2ccccc2)nn1)=O)OC 7923,CC1(C)CCCN(C(c2ccc[nH]2)=O)C1CNC(C1CC(F)(CO)C1)=O 7924,c1(CNC(c2ccc(C)[nH]2)=O)ccc(C(=O)NCC2(F)CCOCC2)nc1 7925,C1(O)(CCCNC(CSc2n(C)nnn2)=O)CCN(C(=O)CC2CCCC2)C1 7926,C=C=CC(C)C(=O)N(C1CCCC1)CCNC(=O)C=Cc1c[nH]c(=N)c(C)c1 7927,C1(C(N(C)Cc2c(C)cco2)=O)C2CC3C(C2NC(C2CCC(F)C2)=O)C13 7928,C(=O)(C1=CC2CCCC12)N.O=C(CC(O)(Cl)c1ccccc1)N1CC(C)C1 7929,CC(CC(N)=O)C(=O)N(C)CCC1CCCCN1C(C1C=CCS1)=O 7930,c1(C(N2CC(NC(CN3CC(CC)C3)=O)CC2(C)CC)=O)ccn2nncc2c1 7931,N1(C(C2(CC=C)CN(C(=O)C(F)(F)C(C)(C)O)C2)=O)CC2OCC(CO)C2C1 7932,c1(C(N2C3CCC2CC(C(N2CCC(O)C(F)(F)C2)=O)C3)=O)c(F)cc(Cl)cc1Cl 7933,N(C1=NCc2cnc(s2)CN1)C(CC)C.C1(CSC)CCCSC1 7934,C=C(Br)CCC(=O)NCC(CC=C)NC(=O)C(COC)N(C)C 7935,C(N=c1ccnc(C2CC2)[nH]1)c1cccc(NC(C2(S(N)(=O)=O)CCC2)=O)n1 7936,c1(C(=O)NC2(C)CCN(C(=O)C3=CCCS3)C2)ccc2c(c1)C(=O)NCCO2 7937,c1(C(C(=O)NC(CCOCC)C(=O)OC)O)c(C)nn(C)c1C 7938,c1(-c2c(C(N(CCC(C)NC(C3CC3(C)C)=O)C)=O)c[nH]n2)ccccc1Br 7939,C(=O)(C(C)(O)CC(C)C)NC(C(=O)NC(CC)CCCO)CO 7940,c1(C(=O)NCC(CNC(=O)C(O)c2cnc[nH]2)OC)cnsc1C 7941,N#Cc1ccc(Cl)nc1NC(C1C2CN(C(c3ccc(O)nc3)=O)CC12)=O 7942,C=Cc1ccccc1-c1ccc(NC(N2CC3CC3C2C#N)=O)cn1 7943,S(=O)(=O)(c1cccnc1NC1CC(C)OC(C)C1)NCC(CC(C)C)OC 7944,c1(N(CC(C)O)CCNC(C2CNC(=O)N2C)=O)ncnc2c1ncn2C 7945,c1(C(=O)NC2CC3(CCN(C(C(CC)OC)=O)C3)C2)nc2ncc(Br)cc2[nH]1 7946,C(=O)(C1=C(Cl)CCCC1)NCCCCCN1CCN(C(=O)C2=CCCCC2)CC1 7947,N1(C(=O)CCC2CC2)CC2CCN(C(C3(C(F)F)CC3)=O)CCC2C1 7948,N1(C(C)=O)CCCC1CC(=O)NC(C1CCCN1C(=O)CC1(C(F)F)CC1)C 7949,Cc1ccc(Cl)cc1OC(c1ccc(N2CCOC(C)C2)cc1)=O 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8111,Cc1cc(C(=O)NC23CC(NC(C4CCC(C)(C)OC4)=O)(C2)C3)ccc1N 8112,c1(OC)ccc(C(=O)NCC(C2CCCN2C(c2n[nH]c(C)c2F)=O)(C)C)cn1 8113,C12(CNC(c3cc(C)on3)=O)CCC(CC1)N(C(c1cc3ccccn3c1)=O)C2 8114,c1(C(N(C(CNC(C2CC(S(C)(=O)=O)C2)=O)C2CC2)C)=O)ccc(N)c(Cl)n1 8115,Cc1ccnc(NC(C(=O)NCC2CC3CC3C2)C(C)C)n1 8116,C1(C(=O)OC)C2C=CC(CC2)C1C(=O)NCC1(CN(C)C(c2cscn2)=O)CC1 8117,c1(SC)c[nH]c2cccc(C)c12.c12ccc(cc1)NC(=O)COC(=O)C2 8118,n1(CC(=O)NCC=CCNC(=O)COc2ccc(F)cn2)ncc2cccnc12 8119,C1(NC(CC2(C)CCCCC2)=O)Cc2ccccc2N(C(=O)C=CC(N)=O)C1 8120,CC1CCSCCN1Cc1ccc(-c2cccnc2OC(F)F)cc1 8121,C1(C(=O)NC2CCCC2CNC(C2(O)CCSCC2)=O)CC2(CCC2)C1 8122,C(C)(C)(CC(=O)NC(c1ccc(F)cc1)CNC(=O)CC1CSC1)SC 8123,n1(CC)ccc(CNC(=O)C(C)N(C(=O)CCC2(C)CC2)C2CC2)n1 8124,N(C1CCC(N=c2cc(C)c(C#N)c[nH]2)c2ccccc21)Cc1cccc(C)c1 8125,c1(OC)ccccc1SCC(N1CC(CNC(c2cc(C)sn2)=O)CC1C)=O 8126,N1(CC(=O)NCC2C(NC(CCCc3nnc(C)n3C)=O)C2)CCc2sccc2C1 8127,c1(C(=O)NCC2CN(C(C(F)=CC)=O)C3(C2)CCC3)ccc2c(c1)ncn2C 8128,Cn1c(O)nc2cc(C(=O)Nc3cc(Cl)cc(Br)c3F)ccc2c1=O 8129,CCCC(C)N(CCC(=O)NCCN(C(=O)C(O)C1CCCC1)C1CC1)C 8130,C12(NC(c3cc(C)oc3)=O)CCCCCC1N(C(c1cc(N)ccc1O)=O)CC2 8131,c1(C(=O)NC(CC)(C)CNC(=O)Cc2cncnc2O)ccnc(Cl)c1Cl 8132,N1(C(c2ccc(=N)[nH]c2Cl)=O)CCC2(CCN(C(c3cc([N+](=O)[O-])c[nH]3)=O)C2)C1 8133,c1(-c2cn(CC(=O)NCC3CC3Cl)nn2)ccc(C(F)(F)F)cc1 8134,C(=O)(C(CC)C(=O)N1CCC2(CC2C(=O)NCc2c(O)cccc2Cl)C1)OCC 8135,N1(C(CCc2nnc(C)o2)=O)CCN(C(C)CNC(c2cnsn2)=O)CC1 8136,c1(C(=O)NC23CN(C(C(CCCC)F)=O)C(CC2)CC3)c[nH]c2c(F)cccc12 8137,C1(C(N(CCCNC(C2(COC)CCOC2)=O)CC)=O)C2CCCCC12 8138,N1(C(C(C(C)C)NC=O)=O)CC2(C1)CN(C(C1CC1C(C)O)=O)CC2CO 8139,Cc1c[nH]nc1C(=O)N(CCCOCCN(C)C(c1cnc(C(C)(C)C)o1)=O)C 8140,C=CC(C)(C)C(=O)N(CC(=O)NCC1(CO)CCOC1)C 8141,C12(NC(C=NOC)=O)CCCC1CN(C(c1ccc(-n3cccn3)nc1)=O)C2 8142,c12cccnc1NC2=O.C1(OC(C)C)CCC(NC(C2(CC3CC3)CC2)=O)C1 8143,c1(OC(C)C)ncccc1NC(c1csc(CNC(=O)C(C)C2CCOC2)n1)=O 8144,c1(OC)ncc(C(=O)NC2CC2NC(c2c(C)nn(C3CC3)c2Cl)=O)cc1C 8145,C1(C)(C(=O)NC2C(NC(C(C(C)C)SCC)=O)CCCC2)CCC(=O)N(C)C1 8146,CC1CN(C(=O)CN(S(C)(=O)=O)C)CCCN1C(C1C2COCC12)=O 8147,C1(NC(Cn2nnc(=N)[nH]2)=O)CCN(C(=O)CCOC2CCCCC2)CC1 8148,c1(COC)nc(N(CCCCN(C)C(C2CCC(F)(F)CC2)=O)C)cc(C)n1 8149,C1(NC(c2coc(Cl)n2)=O)CCC2(CC1)CN(C(c1ccc(I)c(O)c1)=O)C2 8150,C(C)(N=c1[nH]c(=N)[nH]c(=NCC(C)C)[nH]1)c1c(OC)cc(F)cc1.C=O 8151,c1(C(N(C(CNC(Cc2c(C)nsc2)=O)C)C)=O)cccc(-n2ccnn2)c1 8152,C1(C(C)C)CC1N=c1nc2sccc2c(NCc2ccccc2Cl)[nH]1.[nH]1cnnc1 8153,N1(C(c2cnc(CCC)s2)=O)CC(NC(=O)C(C)(CC)CO)C(C2CC2)C1 8154,CC1(C)COc2ccc(C(=O)NC3CN(C(c4cc(Cl)no4)=O)CC3O)cc21 8155,Cc1nnc2n1C(C(=O)N1CC(O)(CNC(C3CCc4ccnn4C3)=O)C1)CC2 8156,C1(C(=O)NC(C(=O)NCC)CC)CN(C(=O)CC2(C)CCCC2)CC12CC2 8157,C1(NC(C=C(C)Cl)=O)CCC2(CCN(C(C3(C)CC=CCO3)=O)C2)C1 8158,C1(O)(CNC(C2CCCOCC2)=O)CCN(C(c2coc(C(F)F)n2)=O)CC1 8159,Cc1cnn(C)c1C(=O)NCC1CCCN(c2nccc(OC(C)C)n2)C1 8160,C1(C(=O)OC)CCC(F)(CNC(=O)C(=O)Nc2ccccc2I)CC1 8161,C(C(C(=O)NCC1CC1C(C)(C)C)C(C)(C)C)NC(C(C)SC)=O 8162,c1(C(=O)OC)nc(C)cc(C)c1CN1CCCC(C(C)(O)C(F)(F)F)C1 8163,C(C)(C)(CCCC(=O)Nc1cnn(C)c1C)NC(Cn1ccc(C)n1)=O 8164,C12(C(=O)NC3CCN(C(CC(C=C)C)=O)C3C)CCC(CC1)C(C)O2 8165,C1(NC(Cc2c(C)con2)=O)CC2CC1N(C(c1nccc(F)c1Cl)=O)C2 8166,c1(C(=O)NCC2CC(NC(c3cn(C)nc3C3CC3)=O)C2)ccc2c(c1)CCC2 8167,N1(C(C=COCC)=O)CCC2(CC1)C(NC(C1CC(O)C1)=O)CS(=O)(=O)N2C 8168,N1(C(=O)NC2CN(C3CCCCC3)C2)CCC(C2CCCC23OCCO3)C1 8169,c12c(cccc1C)C2C(c1nnnn1C)CC.C(=O)(COC)OCC=C 8170,N1(C(c2occ(C(=O)OC)n2)C(=O)NCCSC)CC2CC1CS2=O 8171,N1(C(C(Cn2cccn2)NC(C=CCN(C)CC)=O)=O)CCCN(C(C)C)CC1 8172,Cc1ccnc(C(N2CCCC(C)(CNC(C3CCCCN3C)=O)C2)=O)c1O 8173,CC(C)(C#CC(=O)N1CCCC1CC1CCC1)CNC(c1ccc(F)c(C)c1)=O 8174,Cc1cc(C(=O)NC(C2CCN(C(c3ccccc3Br)=O)C2)C)ccn1 8175,c1(C(=O)NCC2N(C(C3CNC(=O)N3)=O)CCC(C)C2)c[nH]c2cccc(F)c12 8176,N1(C(C2C(C(C)(C)C)C2)=O)CCN(CCNC(=O)CCc2nncs2)CC1 8177,c1(COC)cc(C(N2CC=CC2C(=O)NCC(n2ccnn2)C)=O)n[nH]1 8178,C1(CCCC)(C(N2CCC(CNC3CCC3COC)C2)=O)CN(C(=O)OC)C1 8179,c1(C(=O)NCC2CCC(CC(=O)OC)CC2)cc2cccc(Br)n2c1 8180,C1(C(=O)NC(C)CC(=O)N(C)CCOCCCO)CC2CC(=O)C1O2 8181,C1(C(N(C(C(=O)OC)C)C)=O)CCN(C(=O)CC2CCN(C)CC2)C1C 8182,c1(C(N2C(C(=O)O)CC(CO)C(O)C2)=O)ccc(Cl)c2cc[nH]c12 8183,C1(CC(=O)N(CCCNC(C2CCC3(CCC3)O2)=O)C2CC2)CCC2(CCC2)O1 8184,C(=O)(CCC(=O)Nc1nnc(C)s1)NC(CNC(C1COCCN1S(C)(=O)=O)=O)C 8185,Cn1cccc(C(=O)N(C2(C(=O)NC3CC3CC(C)(C)C)CC2)C2CC2)c1=O 8186,C12(C(=O)NC3CC4(COCCO4)C3)CCCC1CN(C(C1(CO)CCCO1)=O)C2 8187,N1(C(c2c(N)nccc2)=O)CCC2(CNC(C3(C(F)F)CCCO3)=O)CCCC12 8188,c1(C(=O)OC)cc(C)cnc1NC1CC(C)N(C(c2cnn(C3CCC3)c2)=O)C1 8189,C(CC(C)C)(C(=O)N1CCC(C(C)CO)CC1)NC(CSCCC(C)C)=O 8190,N1(CC2C(C)(C)C(O)CC2)CCC2(CC1)COC2.C1(=O)CCC[SH](c2ccccc2)(=O)N1 8191,C1(C(N(CCCC(=O)NCC(COCC)O)C)=O)CC(=O)OC1(C)C 8192,C(=O)(C1=C(F)CN(C(C2CC23CCCCC3)=O)CC1)NC(C#C)C(C)C 8193,c1(C(N2C(CCNC(CCOCC#C)=O)COCC2)=O)cc(N(C)C)ccc1F 8194,c1(C(N2CC(OC(C)(C)C)CC(C)C2)C(=O)NC)cc(CC)ccc1F 8195,C1(N(C(C2CCN(CC(C)C)C2)=O)C)CN(C(=O)CCCC2CC2)CC1O 8196,C1(CNC(c2c(C)nc(C)s2)=O)CCC12CCN(C(C1CCCOC1)=O)CC2 8197,N1(C(c2cc(I)cn2C)C(=O)NCCCC)CCOc2cccc(F)c2C1 8198,N1(C(C2CC(C)(F)C2)=O)CC=CC1(C)C(=O)NCCC(=O)NC(C)(C)C 8199,c1(C(=O)NCCN(C(c2sc(C)cc2Br)=O)CC)cnc(OC(C)C)cn1 8200,Cc1ccc(-n2cc(CN(C(CC)=O)CC(=O)O)nn2)cc1Cl.C1CC1 8201,c1(C(=O)NC2CCC(CNC(COCCC)=O)C2)cc(-c2cccnc2)n(C)n1 8202,Cc1c[nH]nc1C(=O)NC(C)CC(C)NC(=O)C(c1cncnc1)C 8203,C(=O)(C1=CCCCO1)NCCCCNC(C1(O)CCN(C(=O)OC(C)(C)C)C1)=O 8204,c1(OC)ccccc1CN1CCC(CNC(c2cc(CCC(C)C)nn2C)=O)C1 8205,C1(CCC(=O)NC2CCCC2CNC(C2CC(F)C2)=O)CCCCO1 8206,C(=O)(CC(C)CNC(C1C=CCCN1C(=O)CN(C1CCCC1)C)=O)NC 8207,c1(C(N2CC(OC)(CNC(=O)C(C(C)(C)C)NC(C)=O)C2)=O)cnc2nccn2c1 8208,Cc1cn(C)nc1C(N1CCC(CNC(=O)CC2CCC(C(F)(F)F)O2)CC1)=O 8209,C(=O)(C(C)(C)c1cccnc1)NC(c1nocc1C(=O)NCC(F)F)C 8210,C1(NC(c2c(OC)csc2)=O)C2CC(O)C1N(C(=O)C=CC1C(C)C1(Cl)Cl)C2 8211,c1(CN(C2CCCO2)CCOC)[nH]c(=NCC2(F)CCC2)nc2c1ncn2CC 8212,CN1CCCN(C(=O)NCC2CC23CCOC3)CC1 8213,C1(C(N2CC(NC(C(c3cncnc3)C)=O)C3(C2)CC3)=O)CC2CC1CC2(F)F 8214,N1(C(CCc2cncc(C)c2)=O)CCCC1C1CCCN1C(c1nc(O)sc1C)=O 8215,c1(CCC(=O)NCC2CCN(C(C(CC#C)C)=O)C2)ccc(Cl)c(F)c1 8216,c1(CC(N2CC(C3N(C(C4C(C)CC4)=O)CCC3)(O)C2)=O)ncc(Cl)cc1Cl 8217,CC1COCC(CC(=O)NC(C)(C(=O)N(C2CCCC2)CCO)C2CCC2)O1 8218,C1(C(=O)NC2(C3C(=O)NC(=O)N3)CC2)C2CCC(C2)C1NC(C12CSCC1C2)=O 8219,c1(C(C(=O)Nc2c(C(=O)OCC)c[nH]n2)(C)C)ccc(Cl)cc1Cl 8220,C(=O)(C(CC1CCCC1)CC(F)(F)F)N(C(C)C(=O)N1CC(CN=[N+]=[N-])C1)C 8221,C(=O)(CCCC(C)(C)NC(=O)C(C#N)C(C)C)NC(CC)CO 8222,c1(NCC)ccc(Cl)cc1C(=O)NCC(C)NC(C1CCCC(F)(F)C1)=O 8223,C=CCC(CC=C)C(=O)N1CCCC(C)(NC(=O)CCOCCC)C1 8224,Cc1ccc(COCCC(=O)NC(C)CN(C)C(C2CCCO2)=O)nc1 8225,CC1CCC(CNC(=O)CCCC2CC2)CN1C(=O)CCOC1CC1 8226,CC(C(C)C(=O)NC1CCC(O)C1)NC(=O)Cc1ccncc1 8227,C1(CNC(C2(CCCC)CCCC2)=O)CC(NC(c2cc(Cl)ccn2)=O)C1(C)C 8228,C(CC(C)(C)C(=O)NC(c1cccc(C)c1)CNC(=O)CC1CC1)SC 8229,NC(=O)CCCC(=O)N.c1(C2(C(N3CCC3)=O)CCC2)cccc(F)c1Cl 8230,C(CCCNC(C1(Br)CC1)=O)N(C(=O)CNC(c1cscn1)=O)C 8231,C(CS(=O)(=O)CC(=O)NC1(CCCNC(=O)CN2CSCCSC2)CC1)OC 8232,N1(C(C2(C)CC(C)C2)=O)CCN(C)C(CNC(C2(C)CCCS2)=O)C1 8233,C(C(=O)NOC1CC2CCC1C2)(c1ccco1)NC(C1CC1(F)F)=O 8234,C1(NC(C(C=CCCC)O)=O)CC2CCCC(C1)N2c1cc(CC)ncn1 8235,C1(NC(CC2CC(SC)C2)=O)C=CCN(C(=O)Cc2ccc(C)cn2)C1 8236,CCCCC(C(=O)NCC1CCCN(C(c2ncccc2CO)=O)CC1)C(C)C 8237,C(CCCCCCCO)=CC(=O)NC1CN(C(C(C(C)(C)C)SC)=O)CC12CC2 8238,C1(NC(C2C(=C)C2)=O)CN(C(c2c(C3(CC)CC3)cnn2C)=O)CC1C 8239,c1(C(N2CCCC(C)(CNC(C(C(C)C)C#N)=O)C2)=O)sc2cccnc2c1Cl 8240,N1(C(C(=O)NC(c2cscn2)CO)=O)CCCC(C2CCCC2)C1 8241,C1(C(=O)NCC=CCNC(C2(CC)CCOC2)=O)CC2(C1)CC(C)C2 8242,C1(CC=C)(C(=O)OCC(=O)NC(C)(C)C)CCCC1.C12CN(C1)C2=O 8243,c1(NC(=O)OC(C)(C)C)cccnc1CO.C1(NC(=O)CN2CCCC2)(C)CC(CO)C1 8244,c1(OCC)cc(OC)cc(C(=O)NCC2CCN(CC(C)O)CC2)c1 8245,C1(NC(CNC(CCNC=O)=O)=O)CC(F)CN(C(=O)C(F)(F)CO)C1 8246,c1(CC=C)cccc(C(N2CCC(C(C)C(=O)NCCCN3CCC3)CC2)=O)c1 8247,C1(C(=O)NCCCN(C(C2(CCC=C)CC2)=O)C2CC2)CC2C=CC1CCC2 8248,c1(C(N2CC3CC(NC(C4CC(F)(F)C4)=O)CC3C2)=O)cc2cccc(F)c2s1 8249,CN1CCC(=CC(=O)NCCC2CCN(C(=O)CC3CCC(=O)N3)C2)CC1 8250,C(=O)(C(C)(C)C(F)F)NC(CN(C)C(c1cc(C2CCC2)on1)=O)(C)CO 8251,c1(CN2C(C)CN(C(C3CCCO3)=O)CC2)ccc2ccccc2n1 8252,N1(C(C2CN(C(c3c(C)nsc3C)=O)CC2C)=O)CCCc2occc2C1 8253,C1(c2ccccc2)C=CCN1C(c1cnsc1)=O.C1(C(=O)N)C2CCCC12 8254,C12(COC)CC(C(=O)N(C)CCNC(=O)C(C)OCC3CCCCO3)(C1)C2 8255,C1(CCNC(CCCSC)=O)CC2CCC(C1)N2C(c1cccc2c1COC2)=O 8256,Cc1ccsc1C1CCCN1CC(N1CCC(Nc2ccccn2)C1)=O 8257,c1(OC)ccc(-c2ncc(CN(S(C)(=O)=O)C)s2)cn1.c1cn(CCO)nn1 8258,C(C(CC(F)(F)F)NC(C1(O)CC1)=O)NC(c1nc(CC(C)C)sc1)=O 8259,N1(C(C2C(NC(=O)NCCCl)C2)=O)CCC(CC2CCCCC2O)CC1 8260,N1(C(CCOCCC)=O)CC2CCC2(CC(=O)N(c2ccsc2)CC)C1 8261,c1(C(=O)O)cncc(-n2cc(CNC(c3ccnnc3O)=O)nn2)c1 8262,N(C(=NCCC(C)NC(=O)OC)NC1CCC1)C1CC(OCC)C1 8263,Cc1ccc(CC(=O)NCC23CC(CO2)N(C(C2CCC(C)C2)=O)C3)cc1C 8264,C1(C#N)(C(N(C)CC2N(C(CN(CC)CC)=O)CCCC2)=O)CCCOC1 8265,C1(CC(=O)NC(C)C(C)n2cccn2)C(NC(=O)Cc2cncs2)CC1O 8266,N1(C(C(C)(C)OC)=O)CCC(C)C1C(=O)NCCc1cnc(C)[nH]1 8267,c1(CC)ccc(C)c(C(N2CCC(C(C)NC(C3SCC=C3C)=O)CC2)=O)c1 8268,c1(C(=O)NC2C(CNC(c3ccc(O)cc3)=O)C2)cccc(Cl)c1[N+](=O)[O-] 8269,C1(C(=O)NCC(C)NS(CCC)(=O)=O)CCC(Oc2ccccc2)CC1 8270,c1(OC)ncc(C(C)Nc2cc(N3CCCC3)ncn2)cc1F 8271,N1(C(CC=C)=O)CCC(C)C1CNC(c1snnc1C1CC1)=O 8272,Cc1cnc(-c2cn(CCNC(C3C4CC5C(C4=O)C35)=O)nn2)c(C)c1 8273,c1(C(=O)NC2C3CN(C(CCC)=O)C(C3)C2)ccc2nnn(C(C)(C)C)c2c1 8274,N1(C(C2(OC)CCC2)=O)CCC(C(C)CNC(C2CC(OC)C2)=O)CC1 8275,N1(C(CCCOCC=C)=O)CCC(O)C1C(=O)N(CCS(=O)(=O)O)CC 8276,C(CC(CC)(CC)NC(=O)C(C)n1cnnn1)NC(C(C)OCCOC)=O 8277,N1(C(c2ccc(CNC(C(CCCC)F)=O)o2)=O)CCC2(CCCOC2)C1 8278,c1(C(=O)OCC)cnc2c(=NC(=O)Nc3cccn3C)nc[nH]n12 8279,C1(CC(=O)N(CC(CN(C(C(C)c2cccs2)=O)C)O)C)CC(C)(C)CO1 8280,C12(CNC(=O)CC(F)(F)F)CCCCC1N(C(=O)CN1CC=CC1)CC2 8281,C(=O)(C(CNC(=O)C(N)=O)CC(C)C)N1CCC2(C(OC)C2)CC1 8282,c1(C(N(C2CCCC(NC(=O)CCc3cn(C)cn3)C2)C)=O)ccnc(CO)c1 8283,c1(C(=O)NCC2C3CN(C(CCC(=O)NCC)=O)C(C3)C2)csc2c1CCCC2 8284,N1(C(C2(OC)CCC2)=O)CCN(C(=O)CCn2nc(C)cc2C)CC12CCC2 8285,C(=O)(C(C)(O)C1CCCC1)N(C(C)C)CCN(C)C(c1csnn1)=O 8286,C1(CNC(C(C)N(C(C)=O)C)=O)C2CN(C(c3c[nH]nc3C(C)(C)C)=O)CC12 8287,N1(C(C2N(C(CC(C)O)=O)CCOC2C)=O)CCC2(CC1)CN(C)C2 8288,c1(OC)c(C(N2CC(CC(C)NC(=O)C(Cl)=CCl)C2)=O)cccc1Cl 8289,C1(C(N2CC(C(C)O)C2)=O)CC(NC(=O)CC2CNC(=O)O2)C(O)C1 8290,c1(C(=O)NC(CCCCNC(CN(C(C)=O)C)=O)C)ccc(N)cc1C(F)(F)F 8291,C1(COC)C=CCCN1C(C1CCCCC1NC(=O)C(C1CCC1)OC)=O 8292,C(=O)(CC(C)(C)CNC(C1CC12CC2)=O)NC(CCC)C(N)=O 8293,N1(C(C(C(C)C)OC)=O)CC2(CCCN(C(=O)CCc3nc(C)no3)C2)C1 8294,N1(C(CC(C)c2ccco2)=O)CCCC(CC(=O)NCc2ccc(Cl)cn2)C1 8295,C1(NC(C(C)N(C(=O)CC2CCOC2)CCC)=O)CCc2c[nH]nc2C1 8296,C(=O)(CC(C)(C)CCOC)NC1(CC=C)CCN(C(=O)C(C)(C)C(C)(C)O)C1 8297,N1(C(c2c(OC)ccs2)C(=O)Nc2ccccc2)CCC(c2nc(C)cs2)CC1 8298,CC(C)C(O)CC(=O)NCC1CN(C(=O)CCNC(N)=O)CC1C(F)(F)F 8299,CC(C)CC(O)C(C)C(=O)N1CCCCC1CN(C(=O)COCCCN(C)C)C 8300,C(=O)(C#CC(C)(C)CNC(c1c[nH]cc1C(C)C)=O)NCc1n(CCC)ncn1 8301,N1(C(C=C(C)c2ccsc2)=O)CCCC(CCO)(CO)C1 8302,C1(NC(CNC(N)=O)=O)CN(C(=O)CSCc2ncc[nH]2)C2(CCOC2)C1 8303,CC(C(=O)NCC1OCCC1C(N1CCN(C)CC1C1CC1)=O)C(C)(C)C 8304,C(=O)(CN=c1cc[nH]cc1)NCc1nnn(C)c1C(N1CC[Si](C)(C)C1)=O 8305,c1(C(N2CC(NC(=O)NC(C(=O)OC)C)C(F)(F)C2)=O)cc2ccc(Br)cc2s1 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8359,CC(C)(C)C(C(=O)N1CC(CNC(=O)CC2(O)CC2)C(C(F)(F)F)C1)NC(N)=O 8360,c1(OC)ccc(NC(=O)C(C2CN(C(=O)CC3CNC(=O)O3)C2)SC)cc1C 8361,c1(CC2CN(C(c3c(OC)c(Cl)ncc3)=O)CC2O)ccc(Br)c2cccnc12 8362,Cc1cc(C(=O)NC(CNC(=O)C=CC(C)C)C2CCC2)cn(C)c1=O 8363,N1(C(C2(CC)CCC2)=O)CCC2CN(Cc3ccc(OC)cc3)CC12 8364,C1(C(N2CC(C)(CC=CC)C2)=O)CCCCCN1C(=O)C(C1CCCCC1)F 8365,CCCCCCCCCCCC(=O)N(CCCNC(C1CC(CC)(CC)C1)=O)C 8366,c1(CC)cc(C(=O)N(CC(=O)NC(Cc2ccccc2)C(=O)OC)C)n[nH]1 8367,C1(C(=O)NCCN(C(=O)CC(C)F)CC)CCC2CC1CO2 8368,c1(OC)cnc(C(N2CC(F)(C(=O)NCc3ccc(C)cc3OC)C2)=O)c(F)c1 8369,C(=O)(C(C)(C)C(F)F)N(C(C)CNC(=O)CC(O)CSC)C.C(C)(C)(C)OC(=O)C1CC1 8370,C=CCC(CC(C)C)C(=O)NCC1COCC1NC(C12CCC(CC1)CO2)=O 8371,c1(OCC)cncc(C(N2CCC(Cn3cc(C4(O)CCC4)nn3)(CO)C2)=O)c1 8372,c1(C(=O)NC2CCC(C(=O)NCC(C)N(CC)CC)C2)ccc(I)cc1 8373,C1(C(=O)OCC)C2COC(C(=O)NCCCN(C(=O)C(C)SCC(C)C)C)CC12 8374,C(=O)(C1CS(=O)(=O)c2ccccc21)NCC1N(C(C(CC)C#N)=O)CCCC1 8375,C1(=CCNC(C2CC=CCC2)=O)CCN(C(c2cccnc2C(F)(F)F)=O)CC1 8376,C(=O)(C1=C(Cl)CCOC1)NCC1C(C)CN(C(=O)C=Cc2cccn2C)C1 8377,C12(C(N3CCC(CC(C)NC(C(C4CC4)OC)=O)CC3)=O)CCC(CC1)CO2 8378,c1(NCCCNC(=O)NC2CCC2O)csc(C2CCCO2)n1 8379,C(C(O)C(=O)NCC1CCC1C(=O)NCCCC1CCCCO1)=CCCC 8380,CC(C)CC(C)(O)c1cn(C2CC(C(=O)NCCCC3CCCC3(F)F)C2)nn1 8381,N#CC1(C(N2CCC(CO)CC2)=O)CCCOC1.N1(C2CC(C(=O)N)C2)CCCCC1 8382,C(=O)(C1=CC2C=CC(C1)C2)NC(CC(C)C)C(=O)NC1(c2cncs2)CC1 8383,c1(C(N2C3CCN(C(CSCCOC)=O)CC2CC3)=O)cnc2c(c1)CCCO2 8384,CCCC(C(O)C(=O)NCC1CC(O)C1(C)C)NC(C1(c2cccnc2)CC1)=O 8385,Cc1noc(N)c1C(=O)NCC(C)C(=O)NCc1cncc(F)c1 8386,c1(C(N2CCCC(CNC(C(C)OCC)=O)C2)=O)c(OC(F)(F)F)cccc1Cl 8387,c1(CCCNC(N2CCOCC(CC3(CO)CC3)C2)=O)nc2ccccc2s1 8388,c1(C(=O)N(C(C(C(=O)Nc2ccc(SC)cc2)C)C)C2CC2)cc(C)cc(O)c1 8389,N1(C(=O)Cc2nc(C3CC3)cs2)CC(NC(c2n(CC)ccc2)=O)C2(CC2)C1 8390,c1(OC)ccccc1C(C)C(=O)N(CC(C)CNC(c1nocc1C)=O)C 8391,N1(CCNC(C(C)C2CC2)=O)CCC(NC(=O)C(C)(C)N2CCCC2)CC1 8392,C(=O)(CS(=O)(=O)CCOC)NCC(C1(O)CN(C(COCCCCOC)=O)C1)OC 8393,N1(C(COCCCCC)=O)CC(NC(=O)C(c2ccccc2)C)C(O)C1 8394,C1(c2cn(CC3(Cl)C(C)(C)C3)nn2)CCN(C(=O)CSc2ccccn2)CC1 8395,C12(NC(Cc3cn(CC)nc3)=O)CCCC1CN(C(c1cnn(CCO)c1)=O)C2 8396,C1(C(=O)OC(C)(C)C)CCCN(C(c2cnsn2)=O)C1 8397,C1(CNC(c2ccc(C(F)F)nc2)=O)CC2(CC2)CN1C(C1CCCOC1)=O 8398,Cc1cc(S(=O)(=O)C(=O)C(N2C(=O)CN3CCC23)C)sc1C 8399,CCCCCC(F)C(=O)NC(COCC)C(=O)N(C(C)COC)C 8400,C(=O)(CC(C)P(C)(C)=O)N1C(CN(C)C(C2(N3CCCCC3=O)CC2)=O)CCC1 8401,O=S(=O)(CCNC1CCC(CO)CC1)c1ccc(Br)cc1 8402,N1(C(C2(CCOC)CCCC2)=O)CC(NC(=O)CCC2CCCN(C)C2)C(C)C1 8403,n1(CC(N2C(C)(CNC(c3nc(Cl)c(N)s3)=O)CCC2)=O)cc([N+](=O)[O-])cn1 8404,c1(C(=O)NCC2ON=C(C)C2)cncc(CNC(C2C=CCS2)=O)c1 8405,N1(C(c2c(OC)n[nH]c2)=O)CC2CN(C(=O)C(=Cc3ccccn3)C)CC2C1 8406,c1(CCN(CC(=O)NC(C)C(C)NC(=O)C(=O)Nn2cnnn2)C)ccccc1 8407,N1(C(c2cc(C#N)[nH]c2)=O)CCCC2CN(C(c3ccc(N=[N+]=[N-])cc3)=O)CC12 8408,c1(C(=O)NCC23CC(NC(c4cc(Cl)c[nH]4)=O)(C2)C3)ccc2ccsc2c1 8409,C1(CC)C(C(N2CC(CNC(c3ccc(SC)o3)=O)C2)=O)CCN1C 8410,Cc1ccc(C)c(C(=O)NC2CN(C(c3nnn(C)c3C)=O)CCC2F)n1 8411,C1(C(CNC(C2(CC3CC3)CCC2)=O)NC(C2C(=C)CC2)=O)CCCCC1 8412,CC#CCCCC(=O)N(C1CCN(C(=O)C(C)C2(O)CCC2)C1)CC 8413,C(CCCCN=c1[nH]c(=N)[nH]c(=NC2CCCN(CC)C2)[nH]1)OC 8414,C(=O)(C#CC1CCOC1)N1CCC(CNC(C2CCCN2C2CC2)=O)CC1 8415,C1(CC=C)(NC(C2(F)CC=CC2)=O)CN(C(c2cncc(OC(F)F)c2)=O)C1 8416,c1(C(=O)NCC(C)N(C)C(c2cncs2)=O)cc(Cl)ccc1OCC(=N)N 8417,N1(C(CCCOC(C)(C)C)=O)CC2(CCC2)CC1C(=O)NC1CCCCC1N=[N+]=[N-] 8418,N1(C(c2ccc(N)c(Cl)c2)=O)C2CCC1CN(C(C1CC1(F)Br)=O)C2 8419,c1(OC2(CC(=O)NCC(CC)NC(=O)COC(C)=O)COC2)ccc(OC)cc1 8420,C1(C(N(CC(C)NC(=O)CCSC(F)(F)F)C)=O)CCC2(CCCC2)C1 8421,Cc1cc(C(=O)NC2(CNC(=O)C(C3CCCCCC3)O)CC2)oc1C 8422,N1(C(c2cc(C(=O)NC(c3ccc(C)cc3)C)on2)=O)CCc2ccncc2C1 8423,C1(O)(C(=O)NC2(CN(C(=O)C(O)CN3CCCC3)C)CC2)CCOC1(C)C 8424,C1(NC(c2c(C)ocn2)=O)C2CCC1CN(C(c1ccc3nccn3n1)=O)C2 8425,N1(CC)CC2CN(C(=O)C(=O)N(c3ncc(Cl)n3C)CCOC)CC2C1 8426,C1(C(=O)NCC(C)CNC(=O)C(c2ccccc2)N(C)C)(CC)CC1(F)F 8427,Nc1cnc(Cl)cc1C(=O)NCCC1(NC(=O)COC2CCCC2)CCC1 8428,c1(CN(C2CCN(C(=O)C(F)(F)Cl)CC2)CC(F)(F)F)c(O)cccc1Cl 8429,c1(CC(N2CCC(NC(CC=C=C)=O)C2(C)C)=O)ccc2oc(O)nc2c1 8430,C1(C)(NC(Cc2ccn(C)n2)=O)CCCN(C(c2cc(C(F)F)ccc2F)=O)C1 8431,C1(=CC(=O)NCCC(CCNC(C(C)OCC=C)=O)C)CC2CCC(C1)N2C 8432,N1(C(=O)OC)CCc2cc(NC(N3C(C)COCC3C)=O)ccc21 8433,C1(CC)(CO)CCN(C(=O)C(=O)NC(C)Cc2cn[nH]c2)C1 8434,N1(CCOCC(=O)NCC(C)(C)OCCNC(C2CCCO2)=O)CC2CC2C1 8435,Cc1ccc2c(c1)CCC2C(=O)N(CC(C)CNC(=O)CC1CNC(=O)C1)C 8436,N1(C(C(CCSC)O)=O)CC2CC(N(C)C(c3cccc(SCC#N)c3)=O)C1C2 8437,C(CCCCC(=O)NC12COC(C1)C(NC(c1cnc(O)c(F)c1)=O)C2)N(C)C 8438,CC(C)CC(CNC(=O)CCSC(F)(F)F)NC(=O)CNC(=O)C1CC1 8439,C1(CNC(c2cn(CC)nn2)=O)CC2COCC2N1C(C1CC(=O)NC(=O)C1)=O 8440,C(=O)(CC(CC(C)C)NC(=O)CC1CC(=O)C1)NCCc1cc(C(=O)OC)no1 8441,Cc1c(C(N2CCCC2CN(C)C(c2cc(C(F)(F)F)on2)=O)=O)c(Cl)nn1C 8442,N1(C(C(C)CC(N)=O)=O)CC(C)(C)OCC1CNC(=O)Nc1cccc(Cl)c1 8443,C(=O)(CP(C)(C)=O)N1C(CC(=O)NC(CC)CNC(C)=O)CCC1 8444,N1(C(C2CC(OC)C2)=O)CCOCC1CNC(C1(C(F)F)CCOCC1)=O 8445,N1(C(CCC#CC)=O)CCC2C(CCCN2C(c2ccc(NC)cc2Cl)=O)C1 8446,c1(C2C(CC(=O)OC)C2)coc(NC(c2csc(Nc3cc[nH]n3)n2)=O)n1 8447,c1(C2(CNC(C(=O)NC3CCC(C(C)(C)C)C3)=O)CC2)cc(Br)ccn1 8448,C=CC(CC(=O)NC(CSC1CCCC1)CO)c1ccccc1 8449,c1(C(=O)Nc2cccc3nscc23)cccc2c1CN(C(c1nc[nH]n1)=O)CC2 8450,Cc1cc([N+](=O)[O-])ccc1OC(=O)C(N)CSc1ccccc1 8451,C(=O)(CCCS(C)(=O)=O)NC1(C)CC(NC(C2(O)CC(C)(C)C2)=O)C1 8452,N1(C(C2N(C(c3cc(OC)n[nH]3)=O)CC(F)C2)=O)CCC2(CCN(C)C2)C1 8453,c1(CNC(CCOCC)C2CC2)ccc(OC)c(C)c1Cl.c12nnnn1C2C1CC1 8454,Cc1cc(NC(c2cn(Cc3ccn(C)n3)nn2)=O)ncc1Br 8455,C1(C(=O)NC(C(=O)NC(C#C)C(C)(C)C)(C)C)CN(C)CCN1C 8456,N1(CCC)CCCC1CNC(=O)C(Cc1ccccc1)OC 8457,N1(C(c2c(C)csc2C)=O)CC(C(N2CCOC(C)(C(C)C)C2)=O)C2(CC2)C1 8458,C1(C(=O)NC(CC=C)C2CC2)(NC(c2ccccc2)=O)CCN(C)C1 8459,C(=O)(C(C(C)C)N1CCCCC1)NCCC(C)N(C(C(C)NC(=O)NC)=O)C 8460,c1(NC2CC(F)(CNC(=O)CS(=O)(=O)NCCCC)C2)nc(Cl)nc2[nH]c(O)nc12 8461,C1(C(=O)NCC2C(CC(=O)NC(C#C)C3CC3)C2)CC2(CCC2)C1 8462,C1(C(=O)NCCCNC(C(C(C)C)n2ccc(C)c2)=O)CC2OC1C1CC21 8463,Cc1ccc(Cl)c(OCC(N2CCC(NC(c3nc(C)sc3C)=O)C(O)C2)=O)c1 8464,C(=O)(CCC(C)(C)C#N)N(C1CC1)CC1(O)CN(C(CC2CC(SC)C2)=O)C1 8465,C1(CNC(C(=O)NCC)=O)CN(C(c2ccn3cncc3c2)=O)C2(CCC2)C1 8466,c1(CC2N(C(C)C)CCC2)cccc(C2(CN)CCC2)c1 8467,c1(NCCCC)ccccc1C1(C(=O)N(C)C(c2cccc(Cl)c2)C)CC1 8468,N1(C(C(C)OCCC(C)C)=O)CCC(C)(C)C1CNC(C1CC2(C1)CC(O)C2)=O 8469,N1(C(C(C)OC)=O)CCCN(C(c2ccc(SC(F)F)cc2)=O)C(COC)C1 8470,c1(COCCOCC)cccc(SC)c1C.C1CN=C(NCC(c2ccco2)O)N1 8471,N1(CC2(C#C)CC2)CCCCC(C(=O)N(CCCCc2ccccc2)C)C1 8472,CC(C)(C)C(C)(O)C(=O)NCC1CCCN1C(c1cnc2n1CCS2)=O 8473,C(=O)(CC1=NN(C)C(=O)C1)NC1CN(C(C=C(CCC)C)=O)CC1C 8474,C(C)(C)(CCCF)NC(c1c(CNC(C(C)SCC)=O)cno1)=O 8475,c1(N(C)C)ncc(C(=O)NC2(c3ccccc3)CC(F)C2)cc1Cl 8476,CCC(CNC(C1CCN1S(C)(=O)=O)=O)(CC)NC(=O)Cc1cncc(O)c1 8477,CC(C)(F)CCC(=O)NCc1cccc(CNC(C2CCC(=O)O2)=O)c1 8478,N1(C(C(C)NC(C)(C)C)=O)CCOC2(C1)CN(C(=O)C(c1cccc(Cl)c1)O)C2 8479,S(=O)(=O)(c1ccc(=NCCCCCSC)[nH]c1)NCCN(CCO)CC 8480,CCCC(CNC(C1CNC(=O)N1)=O)C(=O)N1CC(=O)NC(CC)C1 8481,C(C)(C(=O)NCc1ocnc1CC)(C1CCC1)NC(C(C)OCCC=C)=O 8482,C1(NC(CC(CC)OC)=O)CCC2CN(c3nnc(-c4ccon4)s3)CC12 8483,Cc1c(C(=O)NCC2(F)CC(CO)C2)cc(C(F)(F)F)cc1N 8484,C#Cc1cnc(C(=O)NCc2ccc(C(=O)N(C)Cc3cocn3)s2)c(C)c1 8485,c1(OC)ccc2cc(C(=O)NCC(C)(C(C)C)NC(=O)COC(F)F)[nH]c2c1 8486,C1(NC(C2(C(CC)(F)F)CC2)=O)C2CC(NC(=O)CCC3CCN(C)C3)CC12 8487,CCCCCC(O)CC(=O)N1CC2CC1CN2C(C1CCc2nccn2CC1)=O 8488,C(C)(C(C(C)C)Nc1cc(C2CC2)ncn1)NC(c1n(CC=C)ccn1)=O 8489,Cc1cc(C2CC2)ccc1C(=O)NCC1CN(C(=O)CC2COCC2O)CC1C 8490,C1(NC(C(c2ccnn2C)C)=O)CC(CC(=O)NCc2n[nH]cc2)C12CCC2 8491,N1(C(=O)NC)CCC(NC(=O)C(n2nnnc2C(C)C)C)CC1 8492,N1(C(c2n(CC)cnn2)=O)CCC2(CCN(C(C3CN4CCCN3CC4)=O)C2)C1 8493,c1(C(N2CC3CN(C(CCc4scc(C)c4)=O)C3C2)=O)ccc2ccoc2c1 8494,c1(C(N2CC(NC(C(C)(C)OC)=O)C(F)CC2)=O)ccnc2c1ncn2C 8495,c1(C(=O)NCC(CNC(C(C(C)C)O)=O)F)nnc2n1CCCCC2 8496,C1(CC(=O)OCC)Cc2ccccc2CN1CCCS(=O)(=O)NC1CC1 8497,Cc1c(C(N2C3CCC2C(NC(=O)C(C)CO)C3)=O)c(O)nc2ccc(F)cc12 8498,C12(C(=O)NC(C3CCN3C(C3CC(C)(O)C3)=O)C)CC3CC1C2C3 8499,C(=O)(C(O)(CN(C)C)C(F)(F)F)NC1CCN(C(c2cc(C)nc(C)c2)=O)C1 8500,C1(NC(c2c(OC)ccs2)=O)(CNC(c2ccc(C)nc2C)=O)CCCCC1C 8501,C1(C(C)C)CCN(C(C2CC3(C2)CC32CC2)=O)C(CNC(c2ccsc2Cl)=O)C1 8502,C(=O)(C1=CCCCCC1)NCC(N1CCCC12CC2C(N(C)C)=O)=O.C1C(=O)N1 8503,N1(CC)CCC(CN(c2ccc(C(F)(F)F)n2C)C(c2cn(C)nn2)=O)CC1C 8504,N1(CCN(CCCNC(=O)NC(CC)COC(C)(C)C)C)CCC(C)CC1 8505,c1(C(N(C2CCCN(C(=O)CCOCC(F)F)C2)CC)=O)cnc2nccn2c1 8506,N1(C(C(C)O)=O)CCN(C)C(CNC(c2cc(C3CCC3)nn2C)=O)C1 8507,C1(C(=O)NCC(C)OC)CCN(C(=O)C(F)(F)C=Cc2ccccc2)CC1 8508,N1(C(c2c(CC)cc[nH]2)=O)CC(CNC(=O)C(C)CC(C)(F)F)CC(C)(C)C1 8509,c1(C(N2CCC3(CC2)CC3C(=O)NCC)C(=O)NCC)cc2cc(C)ccc2s1 8510,N1(C(CN2CCN(C)CC2)=O)CCN(C(c2nc(=O)n(C)[nH]2)=O)CC1CC1CC1 8511,C(CC(=O)N1CCCC1CCCC)(C(F)(F)F)C(c1ccc(C#C)cn1)=O 8512,c1(C(C(N2CCN(CC(=O)C(F)F)CC2)=O)(F)F)cc2ccccc2o1 8513,C=CCCCC(C)(C)C(=O)NC1CC(N(C)C(c2ccc(C(=O)OC)n2C)=O)C1 8514,c1(OC)ccc(C(N2CC(NC(=O)CCNC(N)=O)C(F)C2)=O)c(F)c1F 8515,c1(C(=O)NCCOCC#C)cc(-c2ccc3ccoc3c2)cc2[nH]ccc12 8516,C1(C)(n2cc(SCC(C(C)C)O)nn2)CCCN(C(=O)C(C)CC(F)F)C1 8517,c1(C(=O)NCC(C(=O)N(C2C(C)C2)C)O)ccc(CO)cn1 8518,CC1CCCC=C1C(=O)N1CC(N=[N+]=[N-])CC1C(=O)NOCC1CC1 8519,c1(C(=O)NC2(C)CCN(C(c3ccc(C(C)=O)[nH]3)=O)C2)csc2ccccc12 8520,CC1(C)CC(CC(N2CCCC2C(C)(C)CNC(=O)CC2=CCCC2)=O)C(=O)O1 8521,C1(CNC(c2cc(COC)no2)=O)CN(C(=O)C(C)Cc2ccsc2)CCC1(C)C 8522,C1(C(=O)NCC2(CO)CC2)(CNC(c2cnc(C)s2)=O)CC12CCC2 8523,CC1CC(C(=O)NC2CN(C(=O)C=Cc3cc[nH]n3)CC2n2ccnn2)CN1C 8524,N1(C(C=CSC)=O)CCC2(CCC2)C(CNC(c2nc(C(F)(F)F)oc2C)=O)C1 8525,C1(C#N)(C(N(C(C)C)CCNC(=O)Cc2nccn2C(C)(C)C)=O)CC2CC2C1 8526,Cc1cc(C(=O)NCC(C)(O)CNC(=O)C(C)C(C)(F)F)cc(C)c1F 8527,S(=O)(=O)(c1[nH]c(=NC(C)c2cnsc2)ccc1Br)NCc1c(C#N)ccs1 8528,C(C(C(C)(C)C)NC(c1cccc(CC)c1)=O)NC(C(C=C)c1ccccc1)=O 8529,c1(C(N(C)CC2(NC(C3CC3c3cnc[nH]3)=O)CC2)=O)ccc2nccn2c1 8530,CCC(C)(CC)C(=O)NCC1(NC(c2cn(C)c(=O)n2C)=O)CC2CCC1C2 8531,N1(C(c2ccc(C(N)=O)[nH]2)=O)CCCC1C1CCCN1C(C1CC2(CC2)C1)=O 8532,Cc1cc(C)c(C(=O)NCCC2CN(C(C3(CF)CC3)=O)CC(C)O2)cc1C 8533,c1(CNC(c2c(CNC(C(CO)OC)=O)n[nH]c2)=O)cccc(C)n1 8534,c1(C(=O)N)cccc(C(=O)N)n1.CC(C(=O)NCCN(CC(C1CC1)C(N)=O)C)N(C)C 8535,CC1CCCN(C(=O)CCCCCF)C1CNC(C1CCCCS1)=O 8536,C(=O)(CC(=O)NC1CCCC1CNC(c1coc(Br)n1)=O)OCC 8537,CCCCCCCCC(=O)NC1CCCCC1NC(=O)CNc1nccs1 8538,c1(C(N2CCCC(NC(c3c(C)ocn3)=O)CCC2)=O)cc2c(=O)[nH]ccn2c1 8539,C1(C(=O)NCC(C)NC(C(C)NC(=O)OC(C)(C)C)=O)COCC1N(C)C 8540,C1(C(=O)NC2CN(C(CNC(C)=O)=O)CC2C)CCn2ncnc2C1 8541,C1(CNC(C(=Cc2cnc[nH]2)C)=O)CN(C(C23CC4CC2C3C4)=O)CC1C 8542,C(c1cn(C)cn1)=CC(=O)NCC(CC=C)NC(c1cc(C)c(C)o1)=O 8543,Cc1ccc(CC(N2CC(N(C(=O)Cc3cc(C4CC4)nn3C)C)C2)=O)c(Cl)n1 8544,C1(C(N(CC(C)(C)CNC(c2cn(CCO)nn2)=O)CC)=O)C2CS(=O)(=O)CC12 8545,c1(C(N2CCC(C)C2CNC(=O)CC2CCNC2=O)=O)ccc2cc[nH]c2c1 8546,C(=O)(C(C)CCOC)NCC1(OCC)CN(C(=O)CC2CN(C3CC3)C(=O)O2)C1 8547,c1(C(N2CC3CN(C(CCC(=C)C)=O)C3CC2)=O)cc(C)nc2c(Br)cnn12 8548,c1(CC(=O)NC(N2CCN(C(C34COCC3C4)=O)CC2)C)ccnc(O)c1 8549,c1(OC)cc(P(C)(C)=O)ccn1.C12(C(F)(F)F)CC(C(F)(F)F)(C1)C(=O)N2 8550,c1(-c2cccc(CNCC(C)C(C)(C)C)c2)c[nH]c2ccc(F)cc12 8551,Cc1ccc(C2CCN2C(=O)Nc2ccc(-c3ccccc3)o2)o1 8552,CCCCCC(CC)C(=O)NCCSCc1nc(C)no1 8553,C#CC12CCN(C1)C(=O)C(CC)OCC1CCN(CC1)C2=O.C1(CO)CC1 8554,C1(CNC(CCC=CC)=O)CN(C(C23CC(C)(CCO2)C3)=O)C2(CCC2)C1 8555,Nc1cnc(Cl)c(C(=O)NC2CCC(NC(=O)C(F)C3CCCC3)C2)c1 8556,Cc1ccc(OC(F)F)cc1C(N1CCC(NC(=O)C=CCO)C1C(C)C)=O 8557,CC(C)CC(C(=O)N(S(C)(=O)=O)CC1CCC1)N(C)C(c1cnn2c1OCC2)=O 8558,CC1CC1S(=O)(=O)NCC1(C2CCCO2)CCC1 8559,CC(=O)CCCC(=O)NCC(O)CNC(=O)CCc1ccnc(Cl)c1 8560,C(=O)(C(O)(C(F)(F)F)C1CC1)N1CCC(CNC(C2CCC3(CC2)CC3)=O)CC1 8561,C1(NC(C(C(C)C)C)=O)CCN(C(=O)C(C)n2cnnn2)CC1C(N)=O 8562,C1(CNC(CC=C=C)=O)CCCCN1C(c1ccc(N(C)C)cc1)=O 8563,c1(COC(C(n2ccnc2-c2ccccc2)C)=O)nccn1CCc1ccco1 8564,Cc1nnc(N2CC(O)(CCNC(c3ccnn3C(C)C)=O)C2)c(C#N)c1C 8565,C123C4C5C1C1C2C4C51NC3=O.CC(C(=O)NC1(CC(O)O)CC1)OC1CCCC1 8566,c1(OC)ccc2c(c1)C(C)CN(C(C1CCCC1C1CCNC1)=O)CC2 8567,Cc1cc(C(=O)NC2CCOCC2C(=O)NCCC2CC(C)(C)C2)nnc1C 8568,c1(N2CCN(C(=O)CC3C=CS(=O)(=O)C3)CC(O)C2)ncc([N+](=O)[O-])cc1F 8569,CC1CN(C(C2(C)CCCO2)=O)CCC1CNC(=O)CC(C1CC1)C1CC1 8570,C1(CC)CN(C(C2(C(C)=O)CC2)=O)CCC1NC(c1cc(Cl)ccn1)=O 8571,C1(NC(C(C)SC)=O)CN(C(=O)C(C)CC2CCC2)CC(F)(F)C1 8572,CC(CS(C)(=O)=O)C(=O)N1CCOCC(NC(c2cnoc2)=O)C1 8573,CCC(CNC(=O)CN(CC(C)C)C(=O)C=CC1CCCC1)C(C)C 8574,C(=O)(C1CSc2ccccc21)N1CCOCC1.C1(=O)CCC(=O)NC(CC)(C)CN1 8575,N1(C(C(=O)Nc2ccccc2)=O)CCCC12CCC(C(=O)NCC1(F)CC1)CC2 8576,N1(C(CN(c2ncccn2)CCC)=O)CCC2CC2C1 8577,CCCCCCN=c1cc(NCc2ccc(-c3ccncc3)cc2)nc(C)[nH]1 8578,c1(C(=O)NC2(C)CN(C(C3CCOC34CCC4)=O)C2)ccc(S(=O)(=O)N(C)C)o1 8579,C1(C(=O)NC2CCC(CNC(C3CC4(CC(C)C4)C3)=O)C2)CC2(CCO1)CC2 8580,CCCCCC(CC)C(=O)N(CC(O)CNC(=O)C=Cc1ccc(Cl)cc1)C 8581,C1(NC(CCC(=O)OC)=O)CN(C(=O)Cc2cc(Cl)ccc2Cl)CC1C#N 8582,Cc1cn2cc(C(=O)NC3CCC(NC(C4CSCC(=O)N4)=O)CC3)ccc2n1 8583,c1(C(N2CC3C(CNC(c4c(COC)cco4)=O)C3C2)=O)nc(C)ncc1Br 8584,N1(C(C=Cc2c(C)ccnc2)=O)CCCC(O)(CNC(=O)C(F)=CC(C)(C)C)CC1 8585,c1(-c2sc(-c3n(-c4nc(C)c(Br)cn4)ccn3)c(C)n2)ccc2nn(C)cc2c1 8586,C(C)(CC(=O)NC1(C)CC(NC(=O)CSCC2CCCCO2)C1)OC 8587,c1(C(=O)NCCCOCCNC(C(C)O)=O)cncc2c(O)nccc12 8588,C1(C(N2CC(O)C2)=O)(NC(C=CCN(C)CC)=O)CCSC1 8589,C(C(C)(C)C(=O)NCCNC(=O)Cc1coc(-c2cccs2)n1)N(C)C 8590,C#CC(CNC(=O)CSCCNC(=O)Cc1ccccc1)CC1CC1 8591,c1(CC)[nH]nc(NC(C2(CNCc3c(Br)cnn3C)CC2)=O)c1F 8592,C(=O)(CCCCCC(C)(C)C)NCC1N(C(C(c2ccccc2)C)=O)CCOC1 8593,N1(C(C2C3CC(=O)CC32)=O)CCC(O)(c2cn(CCN3CCCCC3)nn2)CC1.CO 8594,C(=O)(C(Cc1cn[nH]c1)NC(C1CCCO1)=O)N(C)Cc1cccs1 8595,N1(C(C2N(C)C(=O)C(F)C2)=O)CC2CC1CN(C(c1cncc(C(F)F)c1)=O)C2 8596,c1(C(N2CCOCC(NC(=O)CCc3cncnc3)C2)=O)cc(F)c(Cl)cc1O 8597,c1(C(N2CC3CCCC(C2)N3C(c2cccs2)=O)=O)cc2c(cn1)OCCO2 8598,c1(CCNC(CNC(CNC(C2CC(=O)NC2)=O)=O)=O)nccc(O)n1 8599,CCCC(C(=O)OC)C(=O)N1CCC(C)(CC(NC[Si](C)(C)C)=O)C1 8600,CC12CCC1(C)CN(C(=O)C(C1CCCCC1)Nc1nc3ccccc3s1)C2 8601,CC(C)CC(C(=O)N1CC(CNC(=O)CNS(N)(=O)=O)CC(C)C1)NC(N)=O 8602,C1(NC(CC(CC)(F)F)=O)CCN(C(c2[nH]c(=N)sc2C)=O)CCC1CO 8603,C(=O)(C1=CS(=O)(=O)CCC1)N1C(C)CC(NC(c2ccccc2C(C)(F)F)=O)C1 8604,C(C)(CCC(=O)NCCC(N1CCC(F)(CF)C1)=O)OC 8605,c1(CSC)noc2ccccc12.C1(C2c3n(nnn3)CCCN2)CCCC12CC2 8606,C1(CNC(C(C)OCCOC)=O)CCCCN(C(c2ccc(O)nc2Cl)=O)C1 8607,C(=O)(C(F)(F)C1CCCC1)NCCCN(CCC)C(C)C.C12C(C)CN1C2=O 8608,CCC(CC)(CO)C(=O)N1CCCCC(CNC(c2cc(C(F)(F)F)no2)=O)C1 8609,C(=O)(C(C)(C)C1=CCN(C(=O)C2=CCN(C)C2)C1)NC1CCN(C(C)C)CC1C 8610,C12CC(C)(C)CCN1C(C)(C)C1(CC1)CNC2=O.C1(C(=O)OC)CCCN1C=O 8611,C#CCCCCCC(=O)NC1CCC(C)N(C(c2ccc(F)cc2)=O)C1 8612,C1(C(=O)NCCCO)CCCCCCN1C(c1ccc(C(F)F)o1)=O 8613,C#CC(C)(C)C(=O)N1CCCCC1CNC(c1cnc(OC)cn1)=O 8614,CCC(C)C(C(=O)N1CCC(CNC(c2ccc(NN(C)C)cc2)=O)C1)OC 8615,N1(C(c2cc(CC)on2)=O)CCN(C(=O)CC2(C#N)CCC2)CC1COC 8616,N1(C(C(C2CCC2)OC)=O)CCN(C(=O)CCc2nccn2C)C(C(C)C)C1 8617,c1(C(C(=O)N(CC(C)NC(C2CC3CC3C2)=O)C)(C)C)ccc(C#N)cc1 8618,C1(OCCN(C2CCN(C(=O)C(N)=O)C2)C)CCc2nnc(O)cc2C1 8619,C(N=c1[nH]c(N2CC3CC2CO3)nc2c1CSC2)c1nnc(C(C)(C)C)s1 8620,n1(CC)cc(Cl)c(C(N2CC(NC(c3cccnc3O)=O)C(CC)C2)=O)n1 8621,CC1CCCC1(c1nnnn1C)NCC(c1ccccc1)(C)C 8622,O=S(=O)(c1cc2ccccc2s1)NCC1CCN(Cc2nccs2)C1 8623,C1(CNC(c2nc(CC)sc2)=O)CN(C(c2cnccc2Cl)=O)C2CCCC2O1 8624,C=CC1(C(=O)NCC(C2CC2)N(C)C(c2cc(C)c[nH]2)=O)CCCCC1 8625,CC(C)(CC(=O)N1CCCC(NC(c2ccc(OCC(N)=O)cc2)=O)C1)C(F)F 8626,CCCC(C)CC(=O)NCCCCC(C)NC(c1ccn(C(C)C)n1)=O 8627,C1(CCC(=O)NCC(CSC)OC)CCCCN1C(=O)CCCC1CC1 8628,Cc1cnc(N(C)CC2CC2)c(S(=O)(=O)NC2CCOC3(CCOCC3)C2)c1 8629,n1(CC(=O)NC2C(C)CCN(C(C34CCC(C3)C4)=O)C2)ccc(=O)c([N+](=O)[O-])c1 8630,C1(CC(=O)NC(C)CCO)CN(Cc2ccc(Cl)nc2)CCO1 8631,S(=O)(=O)(c1ccc2nc(O)oc2c1)N1CCCN(C(C(C)n2cncn2)=O)CC1 8632,C(CCC(C)C(=O)NCC1CN(C(c2cccc(C)c2N)=O)CCO1)OC 8633,Cc1ccc(C(=O)NC2CC3CC2N(C(=O)CN2CCC(C)CC2)C3)c(O)n1 8634,N1(C(C(CC)C(C)C)=O)CCCC2(NC(=O)Cc3cc[nH]n3)CC2C1 8635,c1(C(C)=O)c(C)[nH]c(C(=O)NCC2(O)CC(NC(=O)CCC3CC3)C2)c1C 8636,N1(C(c2cc(Cl)ncc2F)C(=O)NCC2CC(CC)C2)CCc2c(O)noc2C1 8637,c1(C(N2CC3(C(NC(C=CC=CC)=O)CCS3)C2)=O)cc(F)cc2ccncc12 8638,N1(C(C(C(COC)C)C)=O)CCc2sc(CNC(=O)COCC(=O)NC)nc2C1 8639,CN1CCOCC1CC(=O)NC1CC(NC(=O)CCc2cnn(C)c2)CC1O 8640,C1(C=O)CCC(F)(F)CC1.C12CCCN1N(C)CC(=O)NC2C 8641,C#CCCCC(C)C(=O)NC1CC2CC1CN(C(=O)CCc1cncc(C)c1)C2 8642,CCCS(=O)(=O)CC(=O)NCCCC(C)NC(C1(CC)CCOCC1)=O 8643,c1(CN2CCC(CC(=O)Nc3c(OC)ccnc3)C2)ccnc(Cl)c1Cl 8644,C(CCN=c1[nH]cnc2ccc(O)cc12)NC(=O)CSCC1CCCCO1 8645,C1(OC)CC(CC(N2CCN(C(=O)C(F)=C3CCC3)CC2)=O)C1(C)C 8646,C1(C(=O)NCc2ccccc2C(=O)O)CCC2(CN(C(C3C4CNCC34)=O)C2)O1 8647,CC(C)(CC(F)(F)F)C(=O)NCC(C(F)(F)F)N1CCN(C(C2CSC2)=O)CC1 8648,C12CC3(C1)CC(C3)C(=O)N2C(=O)CN(CC(C)C)CC.C1(CC)CCS(=O)(=O)C1.C=O 8649,CCCCCS(=O)(=O)CC(=O)NC(C)(C)C(C)NC(C1CC2(CCCCC2)C1)=O 8650,C12(CNC(CC(=O)N(C)C)=O)CC1CN(C(c1cncc(-c3cc[nH]n3)c1)=O)C2 8651,C(=O)(CS(=O)C(F)(F)F)N(CC(C)N(C(CNC(C)=O)=O)C)C 8652,C(N=c1[nH]c(=NC)[nH]c(=NCc2cccc(F)c2F)[nH]1)C1(CC)CCOC1 8653,n1(CC(=O)NCC(CNC(C2(C)CCOCC2)=O)O)cnc([N+](=O)[O-])c1 8654,C1(C(=O)NC(C(C)NC(C2(CF)CC(F)(F)C2)=O)C)CC(=O)NC(=O)C1 8655,C1(Nc2cnc(NC(C(N3CCC(C)(C(=O)OC)C3)=O)=O)s2)CC(C)CC(C)C1 8656,N1(C(COCCCC(C)C)=O)Cc2nccn2CC(NC(=O)C2CC2)C1 8657,C12(CNC(C(C)SC)=O)CC(NC(=O)C(c3ccc(Cl)cc3)=O)(C1)C(C)O2 8658,C(=O)(C1CCc2c[nH]nc21)NC1CC2CN(C(c3cc(C)c(O)cc3)=O)CC1C2 8659,N1(C(C=CC)=O)CC2COCCC2(NC(c2ccnc3c2CCC3)=O)C1 8660,C1(NC(C2=C(C)CC2)=O)CC12CCN(C(c1ccc([N+](=O)[O-])[nH]1)=O)CC2 8661,Cc1cc(C(N2C3CCC2CC(CNC(=O)Cc2cnc[nH]2)C3)=O)c(F)cc1F 8662,N1(C(CS(=O)(=O)NCC)=O)CCN(C(C2COC2)=O)C(CC(F)F)C1 8663,C(C(=O)N=c1ccn(CC2CC2)[nH]1)C1CN(C(CC=CC=C)=O)C1 8664,N1(C(c2c(CC)cccn2)=O)CCN(C(c2cccc(N)c2C(F)F)=O)CC1C 8665,C1(C(N(C2CCC2)CC#C)=O)CC2CCC(C1)N2C(=O)Cc1ccon1 8666,c1(C(=O)NCC2N(C(C(=O)NCC)=O)CCC2)nc(C)ccc1Br 8667,c1(C(=O)NC2C(C(=O)NC(c3cnc[nH]3)C)COC2)cnn(C)c1Cl 8668,CC1=C(C(=O)NCC2CCCCN2C(c2cccc3nonc23)=O)CCCC1 8669,c1(CC(=O)NCC2(NC(=O)Cc3ccc[nH]3)CC(OCC)C2)nnc(S)n1C 8670,C1(NC(Nc2cc(C)nc(C)c2)=N)(CC(=O)O)CCCS(=O)(=O)C1 8671,C#CCCC(O)C(=O)NCCC1CCCN(C(c2cc(C(F)F)on2)=O)CC1 8672,C12(C(N3CCC(CCNC(C4COC(=O)N4)=O)CC3)=O)CCC(CO)(CC1)CC2 8673,c1(C(N2CCC(NC(=O)CC3CCCOCC3)C(O)C2)=O)cnc2n1CCCC2 8674,O=S(=O)(c1ccc2c(c1)CC2)NC1CCc2ccccc21.C1COCC1 8675,N1(C(c2c(C(C)C)cnn2C)=O)CC(NC(C2CC(Cl)(Cl)C2)=O)C(C)(C)C1 8676,c1(CN2CCN(CCC)CC2)cc(OC)c(O)c(Br)c1.C12CC3(CC3)CN1C2=O 8677,c1(OC)ccc(C(=O)NC(C)CC(C)NC(c2cncnc2)=O)cc1C(F)F 8678,N1(C(c2c(C)scn2)=O)CCC2(NC(c3cnco3)=O)CCCCCC12 8679,N1C(=NCCO)NC(C)c2ccc(cc2)C1.c1(OCC)cccs1.C(CN(C)C)O 8680,C1(NC(C2(CC#C)CCCO2)=O)CCCCC1NC(c1ccccc1NCC)=O 8681,N1(C(=O)NCCC(=O)OCC)CCC2CN(C(=O)Nc3ccc(F)c(Cl)c3)CC12 8682,C12(NC(C=C(CCN(C)C)Cl)=O)CC(C1)N(C(=O)Cn1cnc(Br)n1)C2 8683,C1(NC(c2ccc(SC)s2)=O)CC2CC(NC(=O)C=Cc3cc[nH]n3)CC2C1 8684,c1(-n2cc(C(=O)NC(C)CCN(C)C(C3CC(C#N)C3)=O)nn2)ccccc1Cl 8685,c1(OC)cnc(C(N2CCCCC2CCCNC(=O)Cc2c[nH]nc2C)=O)cn1 8686,C1(NC(CN(C)CCO)=O)CN(C(C2CCN(C)C2=O)=O)CCC12CCC2 8687,C1(C2CCCN(C(C3CC(F)C3)=O)C2)(NC(C(C)NC(=O)CC(C)(C)C)=O)CC1 8688,c1(-c2ccc(OCC)cc2)ccc(=NCc2ccc(C3CCCN3)cc2)[nH]c1C 8689,c1(OCCN(C)C)ccccc1NC(C1C2CC1N(C(=O)CN1CCCC1)C2)=O 8690,c1(OC)ccc(C(N2CCC(C(C)NC(=O)Cc3cc[nH]c3)C2)=O)c(O)c1 8691,C=CC1CN(C(=O)C(C)(O)C(=C)C)CC1NC(c1cc(=O)cc(Cl)[nH]1)=O 8692,C1(NC(CCOC)=O)CC(C(=O)N(C)Cc2ccsc2)C1.C(C(=O)NC)N 8693,C1(C(=O)NCCN(C2CCCCCC2)C(=O)CN2CC=CC2)CC2CCC(C1)O2 8694,N1(C(C23C(CN(C(c4ccc(SC)s4)=O)C2)C3)=O)CCC2(CC1)CSC2 8695,c1(OCCC(N2CC(CCNC(C3CC3Br)=O)C2)=O)ccc2ccccc2c1 8696,N1(C(c2ncn(C)n2)=O)Cc2ccccc2C(CNC(c2ccc(Cl)nn2)=O)C1 8697,c1(OC)cc(C(=O)NCCC(O)CNC(=O)C(C)(C)C)ccc1[N+](=O)[O-] 8698,C(=O)(C1=CS(=O)CCC1)NCC1(C(=O)NC(c2cocn2)C)CC1 8699,CC(N=c1cccc(S(=O)(=O)NCC23CCCC2C3)[nH]1)c1cccnc1 8700,C1(O)(CN(C(CC=C(C)C)=O)C)CCN(C(=O)C(C(C)(C)C)c2cc[nH]n2)CC1 8701,N1(Cc2c(C)ccc(Cl)c2)CCCC12CCN(C(c1cnn3ccccc13)=O)CC2 8702,N1(C(C(n2ccc(C)n2)(C)C)=O)CCN(C(C2CCN(C)C2)=O)CC2(CC2)C1 8703,C(CN=c1[nH]c2c(c(=NC(C)c3cn(C)cn3)[nH]1)CCC2)(C1CCCC1)OC 8704,c1(C(=O)NC2C(OC)CN(C(c3cnns3)=O)C2)c([N+](=O)[O-])cnn1C 8705,N1(Cc2cn(CC3CN(C(=O)CC4(C)CCCCC4)C3)nn2)CCS(=O)(=O)CC1 8706,c1(CCC)noc(CCC(=O)NC2CCCC2NC(C2CC2C)=O)n1 8707,N1(C(C(F)=CCC)=O)CC2CC(C1)CN(C(C1CC(=O)N(c3cn[nH]c3)C1)=O)C2 8708,C(N=c1nc2ncn(C)c2c(NCC2(C)CCCC2O)[nH]1)c1nn(CC)nc1C 8709,c1(C(=O)NCC(CNC(=O)C2=CCS(=O)(=O)C2)O)cnc2c(c1)COCC2 8710,c1(C(N2CC3CCN(C(C(CC)C#N)=O)CC3C2)=O)cc2c(nn1)c(C)nn2C 8711,c1(C(N2CCC(NC(=O)CC3(CO)CC3)C2)=O)cc(-n2ccnc2)ccn1 8712,c1(C(N2CCN(C(COCC)=O)C(CO)C2)=O)cc2cc(Br)ccc2c(=O)o1 8713,C1(C(=O)NC2(CCC)CCC2)CCCN(C(=O)Cn2cc(C#N)cn2)C1CC 8714,C(=O)(C1=CCCCC1)N1CC2C(CC(=O)NOCCc3ccccc3)C2C1 8715,C1(C(=O)NC2CC(F)(CNC(=O)Cc3ccc(F)cc3)C2)COC2(CCC2)CO1 8716,Cc1ccc(F)c(C(=O)N(CC(C)CNC(C23CCC(C2)OC3C)=O)C)c1 8717,c1(C(=O)NC2CCC(N(C(c3ccc(OC)nn3)=O)C)C2)cc(F)c(F)cc1Cl 8718,c1(OC)ccc(COCC(N2CCN(CC(O)COC3CC3)CC2)=O)cc1 8719,Cc1ccc(C(N2CCCC(N(C)C(C3CC(O)C3)=O)CC2)=O)c(Br)c1 8720,C1(=O)C(F)(CC)C(=O)c2coc(c2CCCCOC)C(=O)NCCN1CC 8721,c1(SC)ccc(C(=O)NCC(C(C)(C)C)NC(c2cn(C)nc2O)=O)c(Cl)c1 8722,N1(C(c2ccn(-c3ccccc3)n2)C(=O)NCCSC)CCOC(C2(C)N=N2)C1 8723,CCCCC(CNC(=O)C(C1CCOC1)OC)NC(=O)CSCC(N)=O 8724,N1(C(CCCOC)=O)CC=C(CNC(=O)CCC2(C)CC2)CC1 8725,c1(C2C(C(=O)NNC(c3ccccc3C3CCCC3O)=O)C2)c(Cl)cccc1Cl 8726,C12=NC(=N)NC(=NCC(=O)N1)N2.C1(NCC)CCN(CC2CCCC2)C1 8727,Cc1sncc1C(=O)NC1(CNC(C2(c3cncnc3)CCCC2)=O)CCCC1 8728,N1(C(c2nc(CNC(C3CN(CC)C(=O)C3)=O)oc2)=O)CC2(C1)NC(=O)NC2=O 8729,c1(C(N2C(C(=O)Nc3c(C#C)nccn3)CC3CC32)=O)ccc2c(c1)CCCO2 8730,c1(N2CC(CC)SCC2)nc(=NCC(C)C(F)(F)F)[nH]c2c1CSC2 8731,Cc1nnccc1C(N1CC2CC1C2C(=O)NCCc1ccncc1)=O 8732,c1(C(=O)NC(CNC(c2cc(C)c(N)cc2)=O)CC(C)C)nsc2c(Cl)cccc12 8733,C1(C(=O)NC2C(C)(COC)C2)COCCN1C(C1(n2cncn2)CC1)=O 8734,c1(C(C(=O)NCC(C(C)C)NC(c2cn(CCF)nn2)=O)(C)C)ccc(Cl)nc1 8735,c1(NC(C(COC)Oc2ccccc2Cl)=O)cc(Cl)nn(C)c1=O 8736,Cc1ccnc(C(=O)NC(C2CCOC2)CNC(=O)C(F)(F)c2ccccn2)c1 8737,C(=O)(C1=NNC(=O)CC1)N(CCCCn1c(C)ncc1)CCC1CCCCO1 8738,N1(C(c2ncc(I)s2)C(=O)NC(C)C2CC2)CCC(C(C2CCCO2)C2CC2)CC1 8739,CCC(C)(C)C(O)C(=O)NC1(CC(=O)NCCC2CC(C)(C)CO2)CCC1 8740,CC(O)CCCCCC(=O)N1CCC(CN=c2[nH]nc(C3CC3)s2)C(C)C1 8741,CC(C)CCC(N)C(=O)NCC(c1ccco1)N1CCCC1 8742,C#CCCC(O)C(=O)N1CCCC1C(C)NC(=O)CCc1cncn1C 8743,C1(NC(C#CC(C)C)=O)CN(C(=O)C(C)(C)Cc2ccc(Cl)cc2)CC12CCC2 8744,C1(C(N(CC(C)(C)NC(c2c(CC)nco2)=O)C)=O)CCCCC1(F)F 8745,C1(C2CN(C(CNC(C)=O)=O)C2)CN(C(=O)COCC(F)F)CCO1 8746,C(=O)(CC1=CCCC1)NCCCOCCN(C)C(c1ccc(SCC#N)cc1)=O 8747,C1(CC)(CNC(C2OCCC2NC(=O)C(C)(C)C)=O)CCCO1.C1(=O)CN1 8748,CC(C)(C)C(O)CCNC(=O)C(C)(O)Cc1ccccc1 8749,C(=O)(C1Cc2ccccc21)NC1CCCN(Cc2nnc(C(C)C)o2)CC1 8750,C1(N(C)C(C2CC(C)(F)C2)=O)CCCN(C(=O)CCc2ccc(Cl)cc2)CC1 8751,CN1CCCCC1CC(N1CCCC1(C)CNC(c1cc(C2CC2)ncn1)=O)=O 8752,C1(NC(NCc2cc(C)on2)=NCc2ccccc2C(C)(C)C)CC(C)OC(C)C1 8753,c1(C(N2CC(OC)C(NC(C3(C)CCN(C)C3=O)=O)C2)=O)c(Cl)ccc(O)c1N 8754,Cc1cc(F)cc2c1N(C(=O)Cc1cnc(C)n1-c1ccccc1)CC2 8755,Cc1ccn(C(C)(C)C(=O)NC(C)CCNC(C2CC(OC(F)(F)F)C2)=O)n1 8756,c1(C(=O)NCCN(C(=O)CC2CC3CCC(C2)C3)CC)nc(C)ccc1OC 8757,c1(C(N(C(C2OCCC2C(=O)OC)=O)CC)=O)cccc(F)c1O 8758,Cc1cnc(NCc2c(C)cccc2C)c(S(=O)(=O)N2CCC(C3CCC3)C2)c1 8759,C(=O)(CC(C)CC(F)(F)F)N1CC(N(C(c2c(CC)c[nH]n2)=O)C)C2(C1)CC2 8760,c1(CC(=O)NC2(C)CN(C(C3(CC=C)CCOC3)=O)C2)cn2ccccc2n1 8761,C1(C(=O)NC2C(C(N3CCCC(OCCC)C3)=O)CC2)CCC2(CCC2)C1 8762,N1(C(c2c(C)ccs2)=O)CC(CNC(c2ccccc2CC2CCC2)=O)C(C)C1 8763,C(=O)(C1SCCc2ccccc21)N1CC(NC(=O)CSc2cn[nH]c2)C(F)CC1 8764,C1(N(C(=O)CCCc2ccsc2)C)CCCN(C(c2cccc(F)c2N)=O)CC1 8765,c1(C(N2CC3C(CNC(C(C)c4cccs4)=O)C3C2)=O)coc2cccc(O)c12 8766,c1(C(N2CC(C(N3CCC(C(C)C)C3)=O)C(C)C2)=O)cccc2[nH]ccc12 8767,CC(C)C(O)C(C)C(=O)N(CCCNC(=O)CC12COCC(C1)C2)C 8768,CN(CCNNS(=O)(=O)c1cc2c(cc1Cl)OC(C)(C)C2)N1C=CN=CC1CC 8769,c1(C(N(CC(=O)N(C(C(N)=O)C2CC2)C)CCC)=O)ccc(N)cn1 8770,C(=O)(CC1OCCc2ccsc21)NC(CCN(C(C=C(C)c1ccco1)=O)C)C 8771,N1(CCC)CCN(C(=O)NCC2(C)CCCC2O)CC1 8772,c1(C(=O)NCc2c(CC(C)NC(=O)CC(C)(C)O)cccc2)cc(N)cc(F)c1 8773,Cc1ncc(C(=O)NCC2CCCCN(C(=O)C(F)OC(F)(F)F)C2)cc1N 8774,c1(C(=O)NC2C(C)CN(C(=O)C3=CCSC3)C2)cccc2cnccc12 8775,c1(C(=O)NCCOCCOCCNC(C2(O)CCOC2)=O)ccc2c(c1)CCO2 8776,C1(CNC(c2n(CC)c(O)nc2)=O)CN(C(C2CCCCC2)=O)CC2(CCC2)O1 8777,c1(C(=O)NCCC(CNC(C2(CN(C)C)CC2)=O)O)cccc2ccn(C)c12 8778,N1(C(CSCCC)=O)CCCCC(NC(c2cn(C)nc2C2CC2)=O)C1 8779,c1(NC(c2c(C(=O)Nc3c(C)cnc(Cl)c3)cccn2)=O)ccc2ncccc2c1 8780,C(=O)(C(O)CCC(F)(F)F)NCC1CC(NC(CC(=O)OC(C)(C)C)=O)C1(C)C 8781,C1(C(=O)NC(c2c(C)cccn2)C)CC2(CC(NC(=O)Cn3nccn3)C2)C1 8782,C(CCF)(C(=O)NCCOCCC1CC1)NC(CCC=C(C)C)=O 8783,Cc1nc(C2CCN(CC3COC(c4ccccc4)C3)CC2)nc2c1CCCC2 8784,C1(C(=O)NCc2n(CC#C)cnn2)CCCN(C(=O)CCNC(C)=O)C1 8785,Cc1onc(C2CC2)c1C(=O)NCC1CCN1C(C1CC(C)(CN(C)C)C1)=O 8786,C1(C(=O)OC)CCC2(CCCCC2)N(C(=O)OC)C1.c12ccc(cc1)C1CC1N2 8787,C1(CNC(COCCCC)=O)CCCCN1C(c1cc(C(C)C)nn1CC)=O 8788,C(=O)(C1Cc2c(Cl)cccc21)NCC1(c2ncc(C(N)=O)s2)CCCC1 8789,c1(C(=O)NC(CCSC)C(=O)NCC(O)CN(C)C)ccnc2[nH]ncc12 8790,c1(C(=O)NC(CCC)CNC(C2CC3CCC2O3)=O)nc(C)c(C)nc1C 8791,N1(C(C(C)(C)C2CCOCC2)=O)CCC(O)(CNC(=O)C(C2CCCCC2)O)C1 8792,CC(C)CC(C)(CO)NC(=O)C(C)C(C)NC(c1c[nH]nc1C(C)C)=O 8793,N1(C(CSc2n(C)nnn2)=O)CCN(C(C2(Cl)CC2(F)F)=O)CC1C1CCC1 8794,N1(C(c2n(CC)nnc2)=O)CCC(C)C1CNC(=O)CS(=O)(=O)NC 8795,c1(C(N(CCCC(=O)NCC2CSCCS2)C)=O)ccc2[nH]nc(Cl)c2c1 8796,N1(C(C)=O)CCC(C(N2CCCCC2c2nnc(CS(C)(=O)=O)o2)=O)CC1 8797,c1(CNc2c(CC(=O)N(C)CCC3(C)CC3)cccc2)cc(I)cc(I)c1O 8798,c1(C(C(=O)NC2CCOC2)N(CCC#N)C2CC2)cnc(C)nc1 8799,C12(C(N)=O)CCCC1(C(=O)NCC1(O)CCN(C(=O)COc3ccccc3)C1)C2 8800,N1(Cc2cccc(C(=O)NCC(C)C#N)c2)C(=O)CN(C)C1=O 8801,c1(NC(=O)NC(CC(=O)NC)Cc2ccccc2C(F)(F)F)cccc(C)c1F 8802,c1(C(N2CCC(NC(c3cnc(C)nc3)=O)C2C)=O)cc2c(Cl)cccc2[nH]1 8803,C1(C(N2CCC(NC(CC(C)C3CCCCC3)=O)CC2)=O)CC2CCC(C1)C2F 8804,C(C(=O)NOCCCCC)C1C(NC(CN(CCC#C)C)=O)CCC1 8805,C(C1C(C(=O)NCCCCn2cc(-c3ccncc3Cl)nn2)C1(C)C)=C(C)C 8806,C(=O)(CC(C)(C)O)N(C)CC1CCN(C(CC2C(C(=O)OCC)C2)=O)C1 8807,n1(CCC)ccnc1C(F)(F)C(=O)N(C(=O)C(F)CN(CC)CC)Cc1ccccc1 8808,c1(C(=O)NCC(C)NC(c2nncc(OC)c2)=O)cc(O)nc2c1c(C)nn2C 8809,C(C(=O)N1OC2CCC1CC2)(c1ccoc1)NC(c1n[nH]cc1[N+](=O)[O-])=O 8810,Cc1cccc(F)c1C(=O)NC(C1CC1CNC(=O)C(C)(C)N(S(C)(=O)=O)C)C 8811,C1(O)(C(C(=O)OCC)(F)F)CCN(CC(C)C(C)(F)F)CC1 8812,c1(N(C)C(=O)Nc2scc(C(=O)OC(C)(C)C)c2)ccc(C(F)(F)F)cc1 8813,C(=O)(C(F)CC(C)(C)NC(c1ncccc1O)=O)NC(CC)C(C)C 8814,C1(C(N2CCN(C(C)=O)CC2c2cnn(C)c2)=O)CCc2cnc(C)n2C1 8815,C(=O)(C1=Cc2ccccc2C1)NCC1(C)CN(C(c2cnc(O)s2)=O)CCO1 8816,C1(NC(C2(OC(C)(C)C)CC2)=O)C=CCC(C(=O)NCCOCCF)C1 8817,c1(C(=O)NC2CN(C(c3c(OC)noc3C)=O)CC(O)C2)[nH]c2c(c1C)CCC2 8818,C=CC(C)(C)CC(=O)N1CCN(C(c2[nH]ccc2C2CC2)=O)CC1CF 8819,c1(C(=O)NCCCN)cscc1C1CC1.C(=O)(CO)OC.C1C(=O)N1C1CC1 8820,C1(CN(C)C(c2cnn(CC(F)F)n2)=O)COCCN1C(=O)CC(Cl)Cl 8821,Cc1cc(C(=O)NC2CCCCC2NC(C2CCN(C)C(=O)C2)=O)nc(O)n1 8822,c1(N(CCN(C(C)C)C(c2ccncc2Cl)=O)C)ncc2scc(Br)c2n1 8823,C(=O)(C1=CC2C=CC(C1)C2)N(C1CN(C(C(CO)OC)=O)CC12CC2)C 8824,C(=O)(C(CCSC)SC)NC1(C(=O)NCC(=O)OCC#C)CC1 8825,c1(C(=O)NCC23CC(CCO2)C3)coc2c1CN(C(=O)CCC1CC1(F)F)C2 8826,n1(CC)ccc(C(=O)NCC2(F)CCN(C(=O)C(c3ccnn3C)O)C2)cc1=O 8827,Cc1cc(C(N2CCCCC2CNC(=O)CCC2CC2C)=O)cc([N+](=O)[O-])c1Cl 8828,c1(OC)ccc2cc(C(=O)NC3CCCC3CNC(=O)C(C)(C)OC)[nH]c2n1 8829,C1(CNC(c2coc(C3CCC3)c2)=O)CCN(C(C23CCC(C2)C3)=O)C1 8830,C(=O)(C1=NOC2COCC12)NCCN(C(c1cccc(CC=C)c1)=O)C(C)C 8831,c1(C2C(C(=O)NCCCN(C(c3cnc(C(C)O)s3)=O)C)C2)ccc(F)cc1F 8832,n1(CCOC)ccc(=NC(=O)C2CN(C(c3[nH]ccc3COC)=O)C(C)(C)C2)[nH]1 8833,Nc1ccc([N+](=O)[O-])c(C(N2CCCCC(NC(=O)CC3CCCOC3)C2)=O)c1 8834,N1(C(CC2CC(CSC)C2)=O)CCN(C(c2n[nH]c(CO)n2)=O)CC1C 8835,C1(C(=O)NC(CNC(CCOCC#C)=O)CC)CNC(=O)CC1C 8836,n1(CC)nnc(C(N2CCC2CNC(=O)CNc2nccs2)=O)c1C 8837,c1(C(N(C)Cc2cccc(Oc3ccc(CC)cc3)c2)=O)c(C)cccc1C#N 8838,C(=O)(C(CC)C(=O)N1CC(C(=O)NCC2CC3(CC(OC)C3)C2)(OC)C1)OCC 8839,CC1CN(C(=O)CC2CC3(CCC3)C2)CC(C)N(C(c2cc3scnc3[nH]2)=O)C1 8840,C1(O)(C(C(=O)OCC)C)CCCN(C(=O)C(C)COCC(F)F)C1 8841,CN1CCN(C(C2C3COCC23)=O)CC1C(N1CC(c2ncccn2)C1)=O 8842,C(=O)(CCCCC(N)=O)NCC=CCC(N1C(C)(COC)C=CC1)=O 8843,C1(NC(CCC(CC)OC)=O)(CNC(C2CCC2)=O)CCC(F)(F)CC1 8844,c1(C(N2CCN(C(c3ccc(C#N)[nH]3)=O)CC2CCO)=O)nccc2nn[nH]c12 8845,c1(CNC(C2N(C(C#CC(=O)N(C)C)=O)CC(F)C2)=O)ccc(F)c(F)c1 8846,C1(NC(C=CCCC)=O)CCCN(C(C2CC3(CSC3)C2)=O)C1 8847,C1(NC(C(C)Cc2ccc(F)cc2)=O)CC2CC(NC(c3ccsc3)=O)C2C1 8848,C1(CNC(c2cc(C)cc(C)n2)=O)CN(C(=O)C(C)CO)C2COCC2O1 8849,C1(NC(CC(C)C)=O)CCCC(NC(=O)CC2CCC(=O)C2C)C1 8850,c1(-c2scc(CN3CCN(CCCCC)CC3)n2)ccc(F)c(OC)c1 8851,c1(C(N2CC(N(C(=O)Cc3ccccc3)C)C(F)C2)=O)ccc2sccc2c1O 8852,C1(CNC(CN(C(c2cc(OCC)n[nH]2)=O)C2CC2)=O)COC(C)(C)C1 8853,C1(CNC(C(C)NC(=O)NC)=O)N(C(=O)CCCC(C)(F)F)CCCC1(C)C 8854,C1(C(N(CC(=O)N(C2(CC#C)CC2)C(C)C)C2CCC2)=O)CCCC1 8855,C1(C(N(CCCCCCC)C)=O)CCN(C(C2(O)CCSC2)=O)C(C)(C)C1 8856,c1(C(=O)NC2(CC=C)CN(C(=O)CSC3CCOC3=O)C2)c[nH]nc1[N+](=O)[O-] 8857,c12nc(n(-c3cncc(Br)c3)n1)C1CCN1C2=O.C1(CC)CCCC1 8858,N1(C(C(C)=C(CC)C)=O)CC(C(=O)NCCC2(C)CC2(F)F)C(C(C)C)C1 8859,C1(NC(CCC=C)=O)CCCC12CCCN(C(=O)CC1CCC(F)(F)CO1)C2 8860,C(C(C)(C)C#CC(=O)NC(C)CN(C)C(C)C)NC(Cc1ccc(OC)cc1)=O 8861,O=C1OC(C(=O)NCC2CCN2C(=O)Cc2cn[nH]c2)Cc2ccc(Cl)cc21 8862,Cc1ccc(C)c(CC(=O)NC(CNC(c2cncc(C)c2C)=O)C2CC2)c1 8863,c1(COC)c(COC(C2CC(C)(C)CN2C)=O)oc2ccccc12 8864,N1(C(CSCCCC)=O)CC(S(=O)(=O)N2CCN(C(C3CCCSC3)=O)CC2)C1 8865,C1(C(N(CCC(=O)NCCCc2ccsc2)CC)=O)CCCC(=O)N1 8866,S(=O)(=O)(c1ccc([N+](=O)[O-])c(Br)c1)N(C)Cc1ccco1 8867,[N-]=[N+]=NCCCC(=O)NCCC12CCC1CN(C(c1nnnn1C1CCC1)=O)C2 8868,c1(CCC(=O)NCCN(C)C(C2CC2(Br)Br)=O)cncnc1 8869,c1(CC(=O)NCC2CNCCOC2)ccc(Br)c(O)c1 8870,N1(C(C=CCN(CC)CC)=O)CCC(NC(=O)C(CN(C)C)CCO)C(C)(C)C1 8871,C(=O)(C(CO)C(C)(C)C)N(CC(C(N1C2(CC(COC)C2)CC1)=O)C)C 8872,N12CCC(C1C(=O)N)CCN(CC)CC2=O.C(=O)(CCOCC)OC 8873,CCCC(C(=O)NCCn1cc(C(N2CCC(N3CCC3)CC2)=O)cn1)OC 8874,N1(C(c2c(OCC)cccc2)=O)CCC2(CCCCN(C(C3CCCO3)=O)C2)C1 8875,N1(C(c2cc(C(C)C)nc(O)c2)=O)CC2CN(C(=O)CSS(C)(=O)=O)CC2C1 8876,C1(NC(C2C(C)(C)CCC2)=O)COC2(C1)CN(C(=O)CCOc1ccccc1)C2 8877,C1(C(N2CCC(NC(C)=O)CC2)=O)CCN(C(=O)C23CCC(C)(C2)OC3)O1 8878,Cc1nnc2c(C(N3CCC(CNC(C4CCC4)=O)C34CCC4)=O)cccn12 8879,CC(C)(CCC(=O)N1CC(NC(c2ccc(Cl)c(Cl)c2O)=O)C1)[N+](=O)[O-] 8880,C=CCCCC(C)(c1nnnn1C)CCc1ccccc1.C(CC(C)C(F)F)N 8881,C1(O)(COC(C(CCC2(C)CC2)Oc2nc(CCOC)oc2)=O)CCCN(C)C1 8882,C(c1c(F)ccc(Cl)c1F)=CC(=O)NCC1(F)CN(C(CC(C)P(C)(C)=O)=O)C1 8883,c1(C(=O)NC(CNC(C=CC(CC)C)=O)(C)CO)cc(S(N)(=O)=O)c(C)cn1 8884,N1(C(CCCC(CC)CC)=O)CCOC2(CCN(C(=O)CSC(F)F)CC2)C1 8885,C(=O)(CC(=O)N(C)Cc1nc[nH]n1)NC(C1(CNCC(F)F)CC1)C 8886,Cc1cncc(C(N2CC(NC(C3CNC(=O)N3C)=O)C(C)C2)=O)c1 8887,N1(C(C(CCC)C)=O)CCN(C(c2n[nH]c(C)n2)=O)C(C2CCCC2)C1 8888,C(=O)(C1CCCn2ncnc21)N1CC(CNC(=O)NC2CC3CCCCN3C2)C1 8889,N1(C(C2CC(C)=C(C)CC2)=O)CCC(C)N(C(=O)C(c2cnn(C)c2)C)CC1 8890,C1(CC(=O)NCCC2(OC)CN(C(c3c(C)nsc3C)=O)C2)CCC(F)(F)CO1 8891,C1(N(CC#C)C(C2(CC)CC2)=O)CCN(C(c2ncn(C)c2C)=O)CC1 8892,c1(CC(=O)N(CC(C)CNC(=O)CC2CCCN2C)C)cnccc1Cl 8893,C1(O)(CC(=O)NC2C(CNC(c3n(C=C)nnc3)=O)CCC2)CCCN(C)C1 8894,C1(C(=O)NC2CC(OCC)C2)CN(C(c2sc(C)nc2CC)=O)CC1(F)F 8895,C(C1CCOCC1)=CC(=O)NC(CNC(c1cnn(CC(F)F)n1)=O)CO 8896,C1(C)(C(=O)NCC2CN(C(c3c(CC)onc3)=O)CC2O)CCCCC1(F)F 8897,C1(CC(N2CC(C)(NC(CN(CCOC)C)=O)C2)=O)COc2ccccc2O1 8898,CC(C)(C)C(C)(C)C(=O)N1CCC(CF)(NC(=O)CC2CCC(=O)NC2)C1 8899,CC(C)CC(CNC(=O)CC1CCC(C(F)(F)F)O1)NC(C1(C)CCOCC1)=O 8900,c1(CC(=O)NCC2(F)CC(NC(CCC#C)=O)C2)cccc(P(C)(C)=O)c1 8901,N1(C(CCC#C)=O)CC2COCC(C1)C2NC(=O)CN1CCS(=O)(=O)CC1 8902,c1(C(=O)NC2COCC2NC(C2CCCOC2)=O)ccnnc1S 8903,N1(C(C2CC(CCC)C2)=O)CC2CCC1C(CNC(c1nc(Cl)sc1C)=O)C2 8904,C1(C(N(CCN(C(=O)CCOCC2CCCC2)C)C)=O)OCCC1N(C)C.C1CCC1 8905,C1(C(=O)NCC(NOC(C)C)=O)C2CCC(C2)C1C 8906,c1(C(N(CC(C)CNC(c2ccc(C#N)cc2)=O)C)=O)ccc([N+](=O)[O-])cc1F 8907,C1(CC(=O)NCCCCCN(C)CC)CN(C(=O)CCOC(C)C)CC1C 8908,N1(S(=O)(=O)c2ccc(N3CCC3)nc2)CCn2cccc2C1CC 8909,N1(C(C(C)NC(c2cccs2)=O)=O)CCC(CCNC(=O)CCn2cc(Cl)cn2)C1 8910,c1(C(N2C(C3CCN(C(CCc4cnc(C)s4)=O)C3)CCC2)=O)ccccc1F 8911,C1(C(=O)NCC(C2(c3ccccc3)CC2)NC(CSCC)=O)CCC(C2CC2)CC1 8912,N1(C(=O)Cc2cnco2)CCCC(NC(=O)CSCc2ccc(F)cc2)C1 8913,c1(C(N(CCNC(C(c2c(Cl)cccc2Cl)C)=O)C)=O)coc2c1C(O)CCC2 8914,c1(C(=O)NC2CC3(CN(C(C(=O)NC(C)C)=O)C3)C2)cc(Cl)cc2c1CCC2 8915,c1(C(C)N)c(Cl)cnn1C.C(=O)(CCCNC(=O)CCN(C)C(C)C)NC 8916,CCC(CC(F)F)C(=O)N1CCC(O)(C(C)NC(c2cc3sccc3s2)=O)C1 8917,c1(C(=O)NC(C(C)NC(C(C)SCCCC)=O)CO)cnncc1O 8918,N1(C(c2c(C)cc(Cl)cc2C)=O)CCC2(CC1)CN(C(=O)CC(C)N(C)C)C2 8919,C(CC)(C(C)(F)F)NC(CC=CCC)=O.C1(C)CC(=O)N1C 8920,C(CC(O)C(F)(F)F)N(C(C(CCN(C)C)NC(C(Br)=C(C)C)=O)=O)CCO 8921,c1(N2CCC(OC)C2)ccc(S(=O)(=O)NCC(O)Cc2cccs2)c(Cl)c1 8922,C1(C(=O)NCC2CC(NC(C(C)c3cccs3)=O)C2)CC(=O)c2ccccc2O1 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8941,c1(C(=O)NCCN(c2ccc(Cl)nc2C)CC)cccc(S(N)(=O)=O)c1 8942,C1(NC(c2ncn(CC)n2)=O)COCCC1C(=O)N(CCF)C(C)C 8943,c1(C(=O)NCC2(F)CC(NC(c3c[nH]nc3Br)=O)C2)ccc([N+](=O)[O-])cn1 8944,c1(C(=O)NC2CN(C(C=CCC)=O)C(CC)(CC)C2)cc(Cl)cc(Cl)c1OC 8945,CC1CCN(C(C2CC23CCCC3)=O)C1CNC(=O)CSc1cccc(F)c1 8946,CC(F)(F)CC(=O)NCC1CC1CNC(c1cnc(Cl)s1)=O 8947,C1(NC(c2cc(C)no2)=O)CC(C)CN(C(C2CC(C)(C)CN2C)=O)C1 8948,CC(CO)CCCNC(c1cc(CCNC(C2(n3nccn3)CC2)=O)on1)=O 8949,c1(C(=O)Nc2ccc(-c3ccc(C(F)(F)F)cc3)cc2)cccc(F)c1Br 8950,C(=O)(C(C)CC(=O)N(CCC(N1CC(N=[N+]=[N-])C1)=O)C)OC 8951,C1(CC(N2CCC(NC(c3cc4occc4s3)=O)(CO)C2)=O)CCS(=O)(=O)CC1 8952,C1(NC(=O)NC(CC(=C)Cl)CO)CCOC2(CCCC2)C1 8953,c1(CC)ccc(C(C)NCc2cnc(-c3ccccc3)[nH]2)cc1F 8954,c1(CC(=O)OC)c[nH]cc1C(=O)NCC(C)(O)CNC(=O)C1=CCC1 8955,CC1(C(=O)NC2CN(C(=O)C(F)(F)C3CC3)CC2CC2CC2)CCCS1(=O)=O 8956,C1(CCCC)CN(C(c2nnc(S)n2C)=O)CCN1C(=O)CCCCCOC 8957,C1(NC(C(C)[SH](C)(F)(F)F)=O)CN2CCN1CCC2=O.C(COCCO)O 8958,C=CC(C)(CC)C(=O)N(C)CCOCCN(C)C(c1cc(O)cc(F)c1)=O 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8977,Cc1coc(C(=O)NCC2CC(NC(=O)Cc3ccco3)C2)c1 8978,C=C(C)C(O)CC(=O)N1CC=C(CNC(=O)C(CO)NC(N)=O)CC1 8979,c1(CN(C)C(C2(CF)CC2)=O)c(Cl)nn(C)c1Cl 8980,C(=O)(CCCS(C)(=O)=O)NC1C(CC)CN(C(=O)CC2NC(=O)NC2=O)C1 8981,c1(C(N2CC(C)C(NC(c3cccc(Cl)c3)=O)C2)=O)ccc2c(c1)CCCCS2 8982,C#CCCCCC(=O)N1CC2CC1CC2NC(c1cc(CSC)c(CC)o1)=O 8983,C1(C(N2C(CNC(c3c(C)cccc3Cl)=O)C=CC2)=O)CC2CCCN2C(=O)N1 8984,N1(C(C(=O)NCC(CC(C)C)(C)C)=O)CCC2CCC(C(=O)OC(C)(C)C)C12 8985,c1(C(N(CC(CNC(c2ncc(C)cc2C)=O)O)C)=O)ccnc2ncccc12 8986,C1(CC(=O)NC(C(C)C)(C)CNC(=O)C(C)(C)c2ccsc2)NC(=O)CNC1=O 8987,C(C)(CN=C(NCC1CCCC(F)(F)C1)NC1CCCCC1)SCC 8988,c1(C(=O)NCC(CCNC(CN2CC(C)C2)=O)O)cnc2cc(Br)ccn12 8989,c1(C(=O)NC2CN(C(Cc3ccc(OCC)nc3)=O)C2)oc(S(N)(=O)=O)cc1C 8990,C1(C(N(CC(O)C(F)(F)F)C)=O)CCN(C(=O)CC2CC=CC(O)C2)O1 8991,c1(OCC=C)ccc(Cl)c(C(=O)NCCNC(C2(O)CC=CC2)=O)n1 8992,c1(C(N2CC(SCC)C(NC(c3cnn(C)c3OC)=O)C2)=O)nc(C)ccc1F 8993,C1(CC(=O)NC(CN(C(C2CC(C)(C(C)(C)C)C2)=O)CC)C)CCCSC1 8994,c1(C(N2C(C)C2)=O)ccc(OC)c(OC)c1.C#CC(C(=O)NCC(=O)NC)SC 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9013,c1(C(=O)NC(C2CN(C(Cc3c(SC)cccc3)=O)C2)C)cc2cccnn2n1 9014,C12(O)CCN(CC1)C2=O.N1(CC)CCN(C2CCN(c3ccccc3)C2=O)CC1 9015,c1(C(N(C(CCNC(Cc2c(C)ccc(C)c2)=O)C)C)=O)ncc(Cl)c(N)c1Cl 9016,c1(CN2C(CC(=O)Nc3ccc(F)c(O)c3)CCC2)cnc2ncccn12 9017,c1(C(C)C)ccc(CSCc2cnn(C)c2)cc1OCC(F)F 9018,N1(C(C(C(=C)C)(C)C)=O)CC2CC(NC(C3(CC)CNC(=O)C3)=O)CC1C2 9019,C1(C(=O)NCC2(CNC(C(C)n3cccc3)=O)CCCC2)C2CCN1CC2 9020,C1(NC(C2CCC(C)(O)CC2)=O)CN(C(C2(C#N)CCOC2)=O)CCC12CCC2 9021,c1(CC)ccc(OC)c(C(=O)NCCN(C(=O)CC(=O)OC)C(C)C)c1 9022,Cc1cc(NC(=O)CN2C(=O)CNC2=O)ccc1NC(=O)CP(C)(C)=O 9023,CC1CN(C(c2ccc(C#N)c(O)c2)=O)CCCN1C(=O)C(F)C(C)(F)F 9024,C1(CC)CCN(C(=O)C=Cc2cc(C)no2)C1C(=O)N(C)CCn1ccnc1 9025,C1(C(N(C2CCN(C3CCCCC3)C2)C)=O)CC2CC2N1C(=O)Nc1ccccc1 9026,c1(N2CCCC(CC)C2)nc(=NCc2ncc(CO)s2)[nH]c2c1COC2 9027,c1(C(=O)NC(CC=C)CNC(C2CC(CCC)C2)=O)ncc(Cl)cc1Cl 9028,C#Cc1ccc(F)c(C(N2CCCC2CN(C)C(C2CCCCC2(C)C)=O)=O)c1 9029,n1(CC(=O)NCC2COCCN(C(C3C4CCCC34)=O)C2)cc2ccccc2n1 9030,C(C(CNC(=O)C1=CCSC1)S(C)(=O)=O)NC(C#CC(=O)N(C)C)=O 9031,C1(C(C)C)CCCC1NC(=O)NC.n12cc(nn1)CC(C)C2.C(C)(C)(C)OC(=O)N 9032,c1(C(=O)NS(C(C)C)(=O)=O)ccnc(CNC(=O)N(C)C(C2CCOCC2)C)c1 9033,C1(C(N(CC(N2CCN(C(c3cncnc3)=O)CC2)=O)C)=O)CC2C=CC1CC2 9034,C1(NC(c2c(CC)scn2)=O)C2CC3CN(C(c4c[nH]c(=N)s4)=O)C1C3C2 9035,N1(CC)CCCC(C(=O)N(C(CNC(c2cccn2C)=O)C2CC2)C)C1 9036,CN1C(=O)CCCC1C(=O)NCCNC(=O)COc1cccc(F)c1Cl 9037,C1(OC)CC2(C1)CC(C(=O)NCC(C)(CC(C)C)NC(c1nc(C)nn1C)=O)C2 9038,n1(CCC)ccnc1CN(C(=O)C(C)n1cncn1)C1CC1 9039,CC1(CNC(=O)CCCCc2cnn[nH]2)CN(C(C2NC(=O)OC2=O)=O)CCO1 9040,c1(NCc2c(Br)cc(C(=O)OC)c(F)c2)c(C(F)(F)F)[nH]c2c(C)cccc12 9041,N1(C(C(c2cccs2)NC(c2cccc(OC)n2)=O)=O)Cc2cnn(C)c2C1 9042,C(C(C(=O)N(CCCNC(C1CN(C(C)C)C1)=O)CCO)OC)OC 9043,C(=O)(CC(C)C(C)C)NCC(CNC(C1N(CCCC)CCCC1)=O)C 9044,N1(C(C2CN(C)C2)=O)CCC(NC(c2cnc(C(F)F)nc2)=O)C(F)C1 9045,c1(NC(C(=O)NC(C)CCCNS(C)(=O)=O)C)nc2cccnc2s1 9046,C1(NC(CCC=CCC=C)=O)CN(C(C2CC(O)CN2C(=O)NC)=O)CC1C(F)F 9047,c1(OC)ccc(C(=O)NC2(CNC(=O)C(F)C3CCC3)CCCCC2)cc1 9048,c1(C(c2n(CCSC)nnn2)NC(c2ccnc(F)c2F)C)c(C)oc(C)c1C 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9104,C1(NC(C2CC3(CC(=C)C3)C2)=O)CCC2CC1CN2C(=O)C(c1cnn(C)c1)=O 9105,c1(COC)cc(C(N2CC(CNC(C3(NC(C)C)CC3)=O)C(C)C2)=O)ccc1F 9106,C(CNC(C1(C#N)CC1(C)C)=O)(CC(C)C)NC(Cc1n(C(C)C)ncc1)=O 9107,CC(C(C)C(=O)NCc1cccnc1)NC(c1ncccn1)=O 9108,N1(C(c2c[nH]c(=NC)o2)=O)CCN(C(=O)CSc2nncn2C(C)C)CCC1C 9109,C1(C(=O)NCc2cccc(COC)n2)CC(F)CN(Cc2ccc(O)c(O)c2)C1 9110,c1(C(=O)NC23CC(C(=O)O)C(C2)C3)ccc2c(c1)nc(O)n2CC(F)(F)F 9111,Cn1ccc(C(=O)NCCC2CCN(C(c3ccnn3C(F)F)=O)C2)c1 9112,c1(C(NC(=O)NCC2(O)C(C)C2)C2CC2)cc(F)c2ncccc2c1 9113,CC(C)(O)C(F)C(=O)N1CCCCC1C(=O)NCC1CCC2(CCC2)O1 9114,C1(S)CC2CCC1C2.O(NC(=O)C1CC(C(N)=O)C1)CC(=O)NC 9115,Cc1nc(C(C)C)[nH]c(=NC2CN(C(c3n[nH]c4c3CCCC4)=O)CC2C)c1Br 9116,C1(OC)CN(C(=O)CC2CCN(C)C2=O)CC1C(=O)NCC1CCC1(F)F 9117,N1(C(c2c(CC)nns2)=O)CC(CNC(=O)C(C)Oc2ccccn2)C(C)(C)C1 9118,N(C1CCc2ccc(F)cc21)C(=O)C(F)(F)c1csc(Cl)c1 9119,N1(C(C2(C)C(C)CCC2)=O)CCC2(CCCC2Nc2ccnc(C#N)n2)CC1 9120,CC(CNC(c1ccnn1C1CC1)=O)(CO)NC(=O)CC1CC1c1ccccc1 9121,N1(C(CC(CC)C(C)C)=O)CCC2CCN(C(C3CCOC3C(C)C)=O)CC12 9122,c1(N(C)C)nc(C(N2CCC2CNC(C2CC2(C)C(F)F)=O)=O)co1 9123,C=C(C)CC(C(=O)NCC=Cc1ccccc1)NC(C1CCOC(=O)CC1)=O 9124,c1(NCc2c(OC)cccc2F)ncccc1S(=O)(=O)NC(C1CSCCO1)C 9125,c1(C(=O)NCCC(C)NC(C2CC2C2CCC2)=O)ccnn(C)c1=O 9126,N1(C(C2CCN(C(CN(C3CCC3)C)=O)C2)=O)CC(O)CC(O)C1 9127,N1(C(c2ccccc2CC#N)=O)CCN(C(c2ncn(CC(=C)C)n2)=O)C(C)C1 9128,c1(C(=O)NCC2N(C(c3c(C)cc(F)cn3)=O)CC2)cc2n(n1)CCOC2 9129,C1(CCNC(=O)Cc2cc[nH]n2)CC(F)(F)CN1C(c1cc(Cl)c(Cl)s1)=O 9130,C12(C(=O)OC)CCC(NC(c3ccnc(-n4ccc(O)nc4=O)c3)=O)(CC1)C2 9131,C(=O)(CN=c1[nH]c(N2CCCC=C(CNC)C2)nc2c(F)cccc12)NCC=C 9132,C12(CNC(C=CCOC)=O)CCC(CC1)CN2C(C1CCCC(OC)C1)=O 9133,c1(C(C)=O)ccc(C(N2CCN(C(=O)CCCF)C(C)C2)=O)cc1C 9134,C#CCC(CC#C)C(=O)NCC(F)CNC(C1(O)CCCCC1)=O 9135,c1(N(C)C)ccccc1C(c1nnnn1C1CCOC1)NCC1C=CCC1 9136,Cn1cnnc1CCCNC(C1CCN(C(c2cccn2C(F)F)=O)C1)=O 9137,c1(-c2cn(CC)nn2)[nH]ncc1C#N.Cn1cc(C2CC2C(=O)NC2CCC2C)cn1 9138,c1(CNC(C2C(NC(c3c(OCC)cccc3)=O)CCC2)=O)ccc(C)cc1O 9139,C1(C(=O)NC(C#C)C2CC2)(NC(=O)CNC=O)CC(CO)C1 9140,N1(C(C(CC)OC)=O)CCC(O)(C(C)NC(=O)CN2CCC(O)CC2)CC1 9141,c1(CN2C(C(N3CC(CC)OCC3)=O)CC(F)C2)cnc(OC)c(Br)c1 9142,c1(C(=O)NCCN(C(C2(CC=C)CC2)=O)C)nsc2ccc(C)cc12 9143,c1(C(=O)NCC(C(C)C)NC(C2CCCC2(C)C)=O)ncc(F)cn1 9144,Cc1cc(C(=O)NCC2CC(C)CN(C(C3(C)SCCCS3)=O)C2)c(O)nn1 9145,c1(C(N2CC(NC(C3N(C)CCCC3)=O)(CO)C2)=O)cc[nH]c(=N)c1[N+](=O)[O-] 9146,N1(C(CCC2(C)N(C(C(CC)SC)=O)CCC2)=O)CC2CC1CN2CC 9147,c1(C(=O)NC(CNC(c2nc(C)oc2C)=O)C)ccc(F)c2cccnc12 9148,c1(C(=O)NCC(CCNC(C2(CN(C)C)CCC2)=O)OC)cc(SC)nn1C 9149,c1(C(CN(C(C)C)Cc2cc(F)ccc2F)=O)ccc(C(F)(F)F)c(Cl)c1 9150,c1(CNC(=O)CN2CCN(CC3CCCCS3(=O)=O)CC2)c(F)ccnc1F 9151,N1(C(c2c(Cl)cc(C)s2)=O)CCC2(CCCC2NC(=O)Cc2coc(C)n2)C1 9152,N(C1CCc2cccc(F)c21)CC1C(C)(C(F)(F)F)C1 9153,Cc1ccn(C)c1C(=O)N(CC(C)CNC(c1nn(C(C)C)cc1Br)=O)C 9154,C(=O)(CCC(=O)NCC1(OC)CN(C(c2cnoc2CC)=O)C1)OCCC 9155,C1(C(=O)NCC(CCNC(C(C(C)(C)C)O)=O)O)CC(=O)c2cc(Cl)ccc2O1 9156,C1(C(=O)NC2C(N(C(=O)CCC(C)(C)C)C)CCC2)COCC1(C)C 9157,C(CC(CC)C(=O)N1CCN(C(=O)Cc2csc(COC)n2)C(C2CC2)C1)=CC 9158,c1(C(=O)NCCC2(NC(COCCCCC)=O)CC2)ccnn1CC 9159,c1(C(N2CCCC(NC(C(CC)F)=O)(CC)C2)=O)nnn2ccccc12 9160,c1(C(C)NC(C2CCN(C(=O)CC3CCC3=O)CC2)=O)cccc2ccccc12 9161,C1(NC(C=C(C)C)=O)CC2CN(C(C3CCS(=O)CC3)=O)CCN2C1=O 9162,CC(C)CC(C(=O)N1CCC(CO)C(NC(c2nnn(C)c2N)=O)C1)C(C)C 9163,C12(CN3CCC(c4cc(C)no4)CC3)CCCC1NCC2 9164,c1(C(N2C(CNC(CCN(C(CCC)C)C)=O)CCCC2)=O)ccn2nnnc2c1 9165,CC(F)(F)CCC(=O)NCCC1(CNC(C2(O)CCOC2(C)C)=O)CC1 9166,C1(CC)C2CCC1CN(C(C1(n3cc(CC4CCCO4)nn3)CCOCC1)=O)C2 9167,C1(SC)CN(C(=O)C(C)Cn2ccnc2)CC1C(F)F.C12(CCC1)C(=O)NCC2 9168,c1(C(C)C)nn(C)c(Cl)c1C(N1CC(NC(=O)CN2C(=O)CCC2=O)C1)=O 9169,c1(C(=O)NC(CC)CN(C)C(c2cn(CCCF)nn2)=O)nn(C)c(N)c1C 9170,Cc1cc(C(N2CCC(O)(CNC(C3(O)CCOCC3)=O)CC2)=O)cc(C)n1 9171,C1(F)(CNC(CCc2ccc(C(C)C)cc2)=O)COCCN(C(=O)CCC#N)C1 9172,C1(C(=O)NCC(C(C)C)NC(C2(OC)CCSCC2)=O)CC2(C)CC1CO2 9173,C1(CNC(=O)CSC(F)F)CN(C(C2CC2Br)=O)CC1O 9174,c1(OC)cc(N)c(C(=O)NC2CCCC(N)CC2)cc1Cl 9175,C1(C(N2C(CN(C(C(C)(C)n3ccnn3)=O)C)CCC2)=O)CC1C1CCCCC1 9176,N1(C(c2cc(CCC)on2)=O)CC2CC1CN2C(C1CCCCO1)=O 9177,c1(CN(C(=O)C(COCC(F)(F)F)NC(C)=O)CC)ccccc1C 9178,Cn1ncc2c(=O)n(CC(=O)NC(c3csc(Br)c3)C3CCC3)cnc12 9179,CC1CN(C(c2ccn(C(C)(C)C)n2)=O)CC2(CCN(C(C3CCCS3)=O)C2)O1 9180,N1(C(C2N(C(C)=O)CSC2)=O)CCC2(CC1)CCN2C(=O)COCCOC(F)F 9181,C1(CC(N2CC(OC)C(NC(c3ccn(C4CC4)n3)=O)C2)=O)CCC(=O)NC1=O 9182,N12CCCC1C1C(CC1)C2.C(=O)(C(C)(C)c1cnsc1)N(C(C(C)C)=O)C 9183,CN1C(=O)CN(CC(N2CC(CCCCNC(c3ccns3)=O)C2)=O)C1=O 9184,c1(C(=O)NCC(C)CNC(C2CCCO2)=O)[nH]cc2c1CCS2(=O)=O 9185,C1(N(C(=O)OC(C)(C)C)CC)CCN(C(=NCCC(C)(C)F)NCC2CC2)C1 9186,c1(C(N)=O)cc2cc(C(N3CCC(OC4CCNC4)CC3)=O)ccc2[nH]1 9187,c1(OC)c(CN2CCC(NCc3cccccccnn3)C2)cc(F)cc1F 9188,CCCCCCN(C(=O)C=CC(C)C)CCc1cnc(C)[nH]1 9189,Cc1ccc(CC(N2CC3C(N(C(=O)Cc4ccnnc4)C)C3C2)=O)cc1C 9190,C1(CCC(=O)NCc2cnc(CC)[nH]2)CCCN(C(=O)CCc2nccn2C)C1 9191,C1(O)(CN(C(C(=O)NCCOC)=O)C)CCN(C(C2CCCCC(=O)N2)=O)CC1 9192,C(=O)(CC(C)(F)F)NC1CCC(N(C(c2c(C(C)C)occ2)=O)C)C1 9193,C1(C(=O)OCC(=O)NCC(C)(C)COCCF)CCCCN1S(C)(=O)=O.CCC#N 9194,CC1(C)C2CN(C(CSC(C)=O)=O)C(C(=O)NC3C4C5CCC(C5)C34)C12 9195,C1(CNC(C=CC(C)(C)NC(=O)C(C2CCCCC2)F)=O)CCn2ccnc2C1 9196,C1(C(C)C)(C(=O)N(C(C)CCO)C)CCN(C(C2CCC2C)=O)C1 9197,C1(CCC)(NC(c2n[nH]c(C(C)C)n2)=O)CCN(C(c2ccc(F)s2)=O)CC1 9198,N1(C(=O)Cc2cc[nH]n2)CCCC(C2CCCCN2C(c2ccc(F)cc2)=O)C1 9199,c1(OCC)nc(C(=O)N(C(CC(=O)O)C(C)C)CCCC(C)(F)F)ncc1F 9200,C1(C(=O)NC2CC(O)C2)CNC(=O)CC1C(F)(F)F.CN1CCCC1CCC=O 9201,N1(C(C23N(C(=O)C(C4CCOCC4)O)CC(C)(C2)C3)=O)CC2CC3CC2C1C3 9202,C(C)(C(=O)N(CC(C)(N(C)CC=CC(=O)NC)C1CC1)C)OCC 9203,C1(CNC(Cc2cc(OC)c(C)cc2)=O)CN(C(C2(O)COC2)=O)CC12CCC2 9204,c1(C(N2CCC3(C(C(=O)Nc4ccnc(CO)c4)C3)C2)=O)ccc2occc2c1 9205,N1(S(C)(=O)=O)CCC(C(N2CCC3C(NC(=O)COc4ccccn4)C23)=O)CC1 9206,Cc1cc(C(=O)N(CCCNC(=O)CC2C=CCC2)C(C)C)nn1C(C)C 9207,C(C(=O)NCC1(C)CCCN1C(=O)CNC(C1CCCCC1)=O)(C(C)C)OCC 9208,N1(C(Cc2nc(C)on2)=O)CCC2(CC1)CC2C(N1CCCC(C)C1)=O 9209,Cc1nccc(CCC(=O)NCC2COC(CNC(c3cc(C(F)F)cs3)=O)C2)n1 9210,N1(C(C(CC)CO)=O)CC23CCCC2(C1)CN(C(c1c(C)cc[nH]c1=N)=O)C3 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9407,C=C(C)C1OCCC1CNC(=O)C(O)CNC(C1(C(C)C)CCC1)=O 9408,N(C(=NCCCCl)NC(c1cccc(C)c1)C)CC1(OC)CCCSC1 9409,c1(C(=O)NC2(CCC)CCCN(C(=O)CC(C)CC)C2)ccn2ncccc12 9410,c1(C(N2CCC(NC(C(C(CC)CC)C)=O)CC2)=O)cc(Cl)c2ccncc2n1 9411,C1(NC(C2(CC)CCCCC2)=O)CC2CC1N(C(c1cncc(COC)c1)=O)C2 9412,Oc1ccc(SC(F)(F)F)cn1.c1(S)nc(-c2ccccc2)ns1 9413,c1(C(C(=O)NCC(C)(C2CC2)NC(C2CC(SC)C2)=O)N(C)C)ccccc1 9414,CCCC(CCNC(C1(F)CCN(C(=O)CCC2(C)CC2)C1)=O)C1CC1 9415,C1(NC(Cc2c(C)con2)=O)CCN(C(=O)C(C)N2CCCC2)CC(C)(C)C1 9416,C1(C(=O)NCC=CCNC(CS(CC)=O)=O)CC(=O)N(C)C1c1nccn1C 9417,C(CC)(C(=O)NC(C)(CNC(=O)C(C)(C)N(C)C)Cc1ccccc1)OCC 9418,C#Cc1cccc(C(N2CC(NC(C3CCN3S(C)(=O)=O)=O)C(C)(C)C2)=O)c1C 9419,Cc1sc(C(=O)NC2(C)CC(NC(=O)C(C3CCOCC3)N(C)C)C2)nc1O 9420,n1(CC)nnc2c1CCC(C(=O)NCC1CCCCN1C(=O)C(C)NC(N)=O)C2 9421,c1(C(=O)NCC2(C)N(C(c3ccc(C)o3)=O)CCC2)nc2ncccn2n1 9422,c1(SC)cncc(C(F)(F)F)c1.N12CC3CC3C1c1noc(n1)C2(C)C 9423,C(=O)(CC(CC)CC(F)(F)F)N(CCNC(C(C)NS(CCCC)(=O)=O)=O)C 9424,N12CCC(O)CC1C2=O.c1(NC(C2N(CC)C3C(C2)C3)=O)c(SC)cccc1F 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9444,Cc1cccc2c(=O)c(C(=O)NC3CC(CN=c4[nH]nc(C5CC5)o4)C3)c[nH]c12 9445,C(CCC(=O)N1CCCC1C(C)(C)CNC(=O)CC1(C)CCCO1)N(C)C 9446,O=C(C1=CS(=O)(=O)CCC1)NC1CCCC1CNC(c1cnn2c1NCCC2)=O 9447,C#CCC(CC(=O)Nc1ccc(CC)c(F)c1)NC(c1cnn(CC)n1)=O 9448,C1(C(=O)NCCN(C(=O)C(C#N)C2CC2)CC)Cc2nnc(C)n2C1 9449,N1(C(C(=Cc2ccccc2)C)=O)CCC(F)(C(=O)NC2COC(=O)C2)CC1 9450,CC(C)C(C(=O)NC1CC1)N(C(=O)Cn1cc(Cn2cccc2C(=O)O)nn1)C 9451,Cc1cncc(CCC(=O)NC(C)CN(C(=O)CC2CCN(C)CC2)C)c1 9452,O=C1CCC(C(=O)N2CCC(NC(=O)Cc3c(F)cncc3Cl)C2)=NN1 9453,N1(C(C(C)SCCCC)=O)CCCN(C(C2(C(=O)NC)CCC2)=O)CC1C 9454,c1(N(CC)Cc2cccc(CSc3ccc(Cl)c(Cl)c3)c2)nc2ccccc2o1 9455,C12(CNC(=O)NCC(O)CO)CCC(CC1)OC2 9456,N1(C(c2c(C#N)cncn2)=O)CCC2(CCCN2C(=O)CC2CSCCS2)C1 9457,C12(C(N(CCCOCCNC(C(C=CCCC)O)=O)C)=O)CCCN(CCC1)C2 9458,N1(C(c2cnc(C)[nH]2)=O)CC2(C1)OC1(CO)CC2(NC(=O)COC2CCCC2)C1 9459,c1(CC(=O)NC2CCCN(C(CCC(C)(F)F)=O)C2)csc2cccc(F)c12 9460,C1(NC(=O)Cn2ccc(C(F)(F)F)n2)CC(O)CN(C(=O)C2=CCCCO2)C1 9461,C#CCC(C)(C(=O)NC(CC(=O)OC)SC)NC(=O)C(CC)CCOC 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9479,N1(CC(=O)NC2CCC(NC(=O)CCC3OCCO3)C2)CCCNC1=O 9480,NCCS(=O)(=O)c1ccc2c(c1)CCN2Cc1cc[nH]n1 9481,C(=O)(CCC(N)=O)N1C(C(N(CC(O)C2CC2)C)=O)CC1 9482,C1(NC(C2CN(Cc3c(OC)cc(F)cc3)C2)=O)CCCOC12CCC2 9483,C(C(F)(F)C(=O)N(C)CC1CN(C(=O)COCC(C)C)CCO1)OC 9484,C(C(CC(C)C)NC(C1(Cl)CC1(F)F)=O)NC(C(OC)OC)=O 9485,c1(NC(C)=O)cc(Br)ccc1C(=O)NCCN(C(=O)CCc1nc(=N)[nH][nH]1)C1CC1 9486,c1(NC(N2CCCC(N(CCC)C(=O)C3CC3)C2)=O)cc2c(s1)CCCCC2 9487,Cc1cnn(C)c1C(N1CC(O)(CCNC(c2cnn(C)c2CC(C)C)=O)C1)=O 9488,CC1C(C)N(C(c2cc(C3CCCC3)[nH]n2)=O)CCN1C(=O)CCc1cnc[nH]1 9489,c1(-c2cn(C3C(C(=O)OC)COC3)nn2)cnc(NC(=O)C(C)C)c(N)c1 9490,N1(C(C2CC3(CC(NC(CSCCCC)=O)C3)C2)=O)CCc2cccnc2C1 9491,C1(F)(C(=O)NCC(C)N(C(=O)CO)C)CS(=O)(=O)CC12CCC2 9492,C1(N(C(=O)C=CC2(C)COC2)C)(C(=O)NCCCC(F)F)CCC(C)(C)C1 9493,CCCC(C)CC(C)(c1nnnn1CCOC)NCc1nc(OC)cc(Cl)c1Br 9494,Cc1nnc2cc(N(C)CC3CCCN(C(c4cccc(Cl)c4Cl)=O)C3)ncn12 9495,c1(SCC)cnc(O)c(C(N2CC(NC(C3CC(=O)N(C(C)(C)C)C3)=O)C2)=O)c1 9496,CC(C)CC(F)C(=O)N1C2CCC1(CNC(=O)Cn1ncn(C)c1=O)CC2 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9515,N1(C(CNC(=O)OCCC)=O)CCCCC1CN(C)C(C1(C#N)CC=CC1)=O 9516,n1(CC(=O)NC(CC(C)NC(C2(C)CC(C)C2)=O)C)cccc(C(F)(F)F)c1=O 9517,N1(C(C=CCN(C)C(C2COCCO2)=O)=O)CCC(CO)C(O)C1 9518,CC(=NO)C1CC(C(=O)N(CCCCNC(c2ncoc2C2CC2)=O)C)C1(C)C 9519,C1(OC)CCCN(CC(N2CCCC2CCNC(c2cocn2)=O)=O)C1 9520,CC1CCC=C1C(=O)NC1(CCNC(c2cn(C)c(=O)n2C)=O)CCC1 9521,c1(CCCCC)nc(C(=O)NCCNC(=O)C(C2CCCCC2)C2CC2)cs1 9522,C12(CNC(c3cn(CC=C)nn3)=O)CC1CN(C(C1(OC)CCOC1)=O)C2 9523,CC1CN(C(C2CN(C(=O)CCc3ccncc3)CCO2)=O)CC1N(C)C 9524,CC1CN(C(c2ccncc2)=O)CC(C)N(C(c2ccncc2Cl)=O)C1 9525,c1(C(=O)NCC2(C)N(C(CC3CC(=C)C3)=O)CCC2)cc2n(n1)CC(C)NC2=O 9526,c1(C(N2C(CNC(CCCOCC)=O)C=CC2)=O)noc(C2CC2)c1C 9527,C(=O)(C1=NOC2COCC12)NC(C(=O)N(CC(=O)OCC)CC)Cn1cncn1 9528,C1(C(N(C2CCCN(C(C=NOC)=O)CC2)C)=O)CC2(CCC(F)(F)CC2)CO1 9529,N1(C(c2cc(C)n(C)c2C)=O)CC(C(=O)NCC2CCC(C)C2)CC(C)(C)C1 9530,c1(C(N2C3CN(C(c4n(C)nnc4)=O)C(C3)CC2)=O)c[nH]c2cccc(Br)c12 9531,c1(C(N(CC(=O)OC)Cc2ccc(Br)cc2)=O)ccc(O)c([N+](=O)[O-])c1 9532,CC(C)CC(O)CC(=O)NCC1CCN(C(=O)CC(C)C)CC1C 9533,c1(N(CCN(C(=O)CC2CNC(=O)C2)C)C)nc(C(F)(F)F)n2c1CCCC2 9534,C(=O)(C1=CC(O)C(NC(=O)C(C)C2CNC2)C1)NCC(C=C)O 9535,c12c[nH]c(c1)C(=O)NCCOCCCN(C)C(=O)C21CC1.C1CCCC1.COC 9536,c1(C(N(C2CCCC(N(C(C=C(C)C)=O)C)C2)C)=O)csc2c(F)cccc12 9537,C1(CNC(N2CCC(c3ccc(I)cc3)C2)=O)(CO)CC2(CCC2)C1 9538,c1(C(=O)NCCC2CC(NC(C(CCC)C#N)=O)C2)cnc2cccnn12 9539,C(=O)(CCS(N)(=O)=O)N1CC(C)(NC(C(C)(C)Sc2ccccc2)=O)C1 9540,C1(NC(CCC#C)=O)CN(C(=O)NC2CCCN(C(C)(C)C)C2=O)CC1(C)C 9541,C(=O)(C#CC(C)(C)CNC(C1(C)CCC(=O)C1)=O)NCCCNC(=O)NC 9542,N1(C(C(C(=O)OC)C)=O)CC2OCCN(C(c3cc(-c4ccco4)no3)=O)C2C1 9543,C12(C(=O)NC3(CC=C)CCOC3)CC(C)(CN1C(c1nnsc1N)=O)C2 9544,n1(CC)ncc(Cl)c1C(=O)NCC(O)CNC(c1cnn(CCC(C)C)c1C)=O 9545,C1(CC(=O)NCCN(C(=O)C(F)(F)c2cscn2)CCC)CCN(C)C1=O 9546,C1(Cc2ccc(C(N(C)CF)=O)cn2)CCCCN1C(=O)COCc1nc[nH]n1 9547,C(C(C)(C)C(=O)NC1CC1C(=O)Nc1cccc(C)c1)NC(CNC(C)=O)=O 9548,C(C(C(=O)NC1CC(NC(C2CC(=O)N(OC)C2)=O)C1)C(C)(C)C)OCC=C 9549,N1(C(CC=CC)=O)CCOCC(CNC(=O)CCCOc2ccccc2)C1 9550,C(=O)(CS(=O)(=O)C(C)C)N1CCC(NC(C2CN(C(=O)NC)C2)=O)C(F)C1 9551,n1(CC)cnc2c(NCCCCOCCOC(C)=O)[nH]c(=NC(C)C(F)F)nc12 9552,c1(-c2c(C)ncc(Cl)c2)cn2c(n1)CN(C(=O)NC1CC1C)CC2 9553,C1(C(=O)N(C)OC(C(C)(C)OC)=O)CN(c2nccc(CC#N)n2)CCO1 9554,N1(C(C2(Cl)C(C)(C)C2)=O)CCN(C(=O)C(F)F)C(c2ccccc2)C1 9555,Cc1cncc(C(N2CCCC(CNC(=O)C(C)(C)CC3CC3)C2)C)n1 9556,C(=O)(N1CC(O)C(O)CO1)C1CCCC(NC(c2ccc(S(N)(=O)=O)s2)=O)CC1 9557,C1(NC(c2ccc(CC)cc2)=O)CCCCN(C(=O)CCCC(C)C)C1.C(=O)CS 9558,c1(Cc2cccc(C3CC3)c2)cccnc1S.CC1CNC(=O)C=CC(=O)N1 9559,Cc1ccn(CC(=O)NCC(C2CCOC2)NC(=O)C(C)Cn2cccn2)c(=O)c1 9560,C1(CC(C)NC(C(=Cc2cnc[nH]2)C)=O)CCN(C(=O)Cc2sccc2C)CC1 9561,N1(C(CCOC)=O)CC2CC1CN2C(=O)CC1(c2ccccc2)CCCO1 9562,C1(CC(=O)NCCSCC=C)CN(C(c2cnc(C)cn2)=O)CCC1C 9563,Cc1ccccc1SCC(N1CCC(C(C)Nc2ncccn2)C1)=O 9564,C=C(Cl)CC(C(=O)NC1(CN(C)C)CC1)NC(=O)CCC1CC1 9565,Cc1ccc(C(=O)OCCc2nnn(C(C)(C)C)n2)c2cccnc12 9566,C1(CC(=O)NCC2(CNC(C(c3ccc(Cl)cc3)CC)=O)CC2)CC2(CC2)CO1 9567,c1(NCC(CN(C(C2CN(C)C(=O)CC2)=O)C)O)c(C#N)c(=O)n(C)c(=O)n1C 9568,c1(NCCN(c2cnccn2)C)ncnc(Cl)c1F.CC1CC2CN1C(=O)N2 9569,CC(C)(C)CC(O)CC(=O)NCC1CC(C)(C)CN1C(c1cnn(CCF)c1)=O 9570,c1(C(N2CC(NC(C=CC)=O)C(c3ccccc3)CC2)=O)cc(F)c(F)cc1Cl 9571,CC(C)CC(F)C(=O)NCCC(O)CNC(=O)CCC(=O)c1cccc(Cl)c1 9572,c1(CNC(c2cccnc2)CC)cc(F)c(C(F)(F)F)cc1F 9573,c1(CC)ncnc(Nc2cccc(F)c2C(N2CC(F)(F)C2)=O)c1F 9574,Cc1cccc2c(C(N3CC4CC4(NC(=O)CC4=CCN(C)CC4)C3)=O)cnn12 9575,Cc1ccc(CC(=O)C(C)=O)cn1.C1(C(=O)NC2CC(N)C2)CCOC(C(C)C)C1 9576,C(=O)(C(C)(C)C(C)(C)C)NCC(CC1CCCCC1)NC(CCCCC=CC)=O 9577,N1(C(C2ON=C(C(C)C)C2)=O)CC2(CCC(CNC(=O)CCCC#N)O2)C1 9578,c1(NC)ccc(C(=O)NC(c2ccccc2)C(C)NC(=O)Cn2nccn2)cn1 9579,N1(C(C(CC#C)C)=O)CCC2(CCC(CNC(C3(C(F)(F)F)CCC3)=O)O2)CC1 9580,CCCC(C)(O)CC(=O)N1C2CCC1CC(NC(=O)Cc1cc(OC)no1)C2 9581,C1(C)(C(N2CC(O)(CN(C)C(C3C(C4CC4)C3(F)F)=O)C2)=O)CCC(C)(C)CC1 9582,S(=O)(=O)(c1ccc(NCC2C3COCC23)c(Cl)c1)NC(CC(C)C)(C)C 9583,N1(C(C(CCC=C)(C)C)=O)CCC2CN(C(C3(OC)CCCCC3)=O)CC2C1 9584,c1(NCC(CC)CO)ccc(S(=O)(=O)N2CCC(C3CCCCC3)C2)cc1Br 9585,CC(C)C(C(=O)N1CC2CCC(CO)(C2)C1)C(C)NC(=O)CNS(C)(=O)=O 9586,N1(C(c2ccc(CSC)o2)=O)C2CCC1CC(NC(=O)C(O)C(F)(F)F)C2 9587,CC1COCCN1C(c1n[nH]cc1CNC(C1CCCOC1)=O)=O 9588,c1(C(=O)NC2C3CN(C(CC)=O)CC2COC3)ccc2cc(OC)c(F)cc2n1 9589,Cc1cc(C(=O)NCCOCCNC(c2cnn(C)c2Cl)=O)c2sc(=N)[nH]c2n1 9590,c1(OC)cccc(C(=O)N(CC(C)(C)NC(C2CN(C)CC(C)O2)=O)C)c1OC 9591,CC(C)C(O)C(C)C(=O)N1CCC(CNC(c2coc(CO)c2)=O)C(O)C1 9592,C1(CC)(NC(=O)C(C)CC2CC2)CCCN(C(c2ccc(C)c(C)n2)=O)C1 9593,C=C(Cl)CCC(=O)N1CCCC(C(C)NC(=O)COc2ccc(Br)cc2)C1 9594,N#Cc1cc(CNC(C2(F)CCCN(C(=O)CC3CCSC3)C2)=O)ccn1 9595,C1(C(=O)NC2C(CO)CCN(C(c3cc(C)sc3)=O)C2)CN(C)CCN(C)C1 9596,C(=O)(CCN=[N+]=[N-])N1CCC(C(C)NC(=O)CC2CCCC2)C1 9597,CCC(C(=O)OC)C(=O)NC1CC(NC(C2(CO)CCC2)=O)C1 9598,C=CCCC(CC(C)C)C(=O)NCC(C(F)(F)F)n1cncn1 9599,C1(CCN(CC(c2cccc(Cl)c2)N)C)CCCC2CC12 9600,C1(CC#C)(C(=O)Nc2nncn2C)CCN(CCOCCOC)C1 9601,C1(NC(C2(CC)CCCC2)=O)CCC(C)N(C(C2(c3cnccc3C)CC2)=O)C1 9602,Cc1ncc(Cl)cc1CC(=O)NC1CC(F)(F)CC1NC(c1ccon1)=O 9603,C=C1CC2(C1)CC(C(=O)NC1CC3(NC(C45CC6CC4C5C6O)=O)COC1C3)C2 9604,N1(C(C(CCSC)NC(=O)Cn2cnc(C#N)n2)=O)CC2CCCC2C1 9605,C1(CN(C(c2cn(CC)nn2)=O)C)COCCN1C(c1[nH]nnc1COCC)=O 9606,c1(C(=O)NC(=O)NC)cc2c(s1)CCC(C)C2.c12cn(nn1)CCCC2 9607,c1(C(C)C)nnc2cc(N3CCC(NC(C4(F)CCOC4)=O)C3)ncn12 9608,C(=O)(C(CC(C)CC)NC(C1CCC(=O)O1)=O)N(CC(=O)NCC)C 9609,C1(CC(c2nccs2)C)COC2(C1)CN(C(=O)CCC=O)C2.N1CCCCC1 9610,c1(N(CC(CN(C)C(c2ccon2)=O)O)C)cc2nncn2cn1 9611,CC(C)CC(O)C(C)C(=O)NC1CC(C(=O)N(C)C(C2CCC2)C)C1(C)C 9612,O=C(Nn1cnc2scc(-c3ccccc3)c2c1=O)NC1(CF)CC12CCOCC2 9613,C1(C(NOCC(=O)NC(COCC)CO)=O)C2CCCCC12.OC.O 9614,c1(C(=O)NC(C)CN(C(=O)COC2CCOC2)C)[nH]cc2c1CCC2 9615,CN=c1[nH]cc(C(=O)NOC(C(C2CCCN(C(C)=O)C2)(C)C)=O)s1 9616,c1(CC(=O)NC(C2CN(C(C3CC3C)=O)CCO2)C)nc2ncccn2n1 9617,c1(C(=O)NC2(C)CN(C(Cc3cc(C(C)C)no3)=O)C2)ccc2[nH]ccc2n1 9618,N1(C(c2cc(OC)no2)=O)CC(C)CC1C(=O)NCC(O)CN(C)C(C)=O 9619,CCC(CC)(CCNC(c1c[nH]c(=N)s1)=O)NC(=O)CC1(C(F)F)CC1 9620,Cc1cc(C(=O)NCCN2CCC(CC(=O)N(C)C)C2)ccc1F 9621,c1(OC(C)C)cccc(C(=O)NCC(C)CNC(=O)C=C(Cl)Cl)c1Cl 9622,c1(CC(N2C(CNC(C(CC(=C)C)C)=O)CCC2)=O)ccc(N)c([N+](=O)[O-])c1 9623,CC1(CC(=O)NCCOCCN(CCN=[N+]=[N-])C)CCS(=O)(=O)N1 9624,C(=O)(C(C)(C)CC(F)(F)F)NCC(N(C(C(C)OCC#C)=O)C)C1CC1 9625,N1(C(C2CC(C)(C)C2)=O)CCC(C(N2C3CCC2CC(CO)C3)=O)CC1(C)C 9626,Cc1ccc(N(C)C)cc1C(=O)N(C)CCNC(=O)CCc1ccc(Cl)s1 9627,Cc1ccc(=O)n(CC(N2CCN(C(C3COCCOC3)=O)CC2C2CC2)=O)c1 9628,c1(C(N2CC(CNC(C3(CC=C)CC3)=O)OCCC2)=O)c(C)nc2ccccn12 9629,C(CN=c1cccc(S(=O)(=O)NCCC2SCCS2)[nH]1)c1cccc(OC)c1 9630,Cc1cc(C(=O)NC2(CCC(=O)NC3(C)CCS(=O)(=O)C3)CCC2)nc(C)n1 9631,c1(C(=O)NC(CCCCNC(c2cccc(C)c2)=O)C)cc(O)ncc1Br 9632,N1(C(C(CC#C)C)=O)CC2CCCC2(NC(=O)CSc2ccc(C)cc2)C1 9633,c1(C(=O)NC(CCOC)C(=O)NC2(CCF)CC2)cc(C)nnc1C 9634,C1(C(=O)NCC2CCN(C(c3nnn(C)n3)=O)CC2)CCC2(CCCC2)CC1 9635,n1(C(C)C)nc(C2Cc3ccccc32)nc1-c1cc([N+](=O)[O-])ccc1F 9636,CC(=O)CCC(=O)N1CCCCC1C(=O)NCC(C)(O)C1CCCC1 9637,N1(CC(=O)NC2CC2NC(c2occc2Cl)=O)CCN(C2CCC2)CC1 9638,N1(C(CNC(CC)=O)=O)CCCC1C(=O)NC(c1ncc(C)[nH]1)C 9639,O=C(C1CCCc2scnc21)NC(CC1CCCC1)CO 9640,c1(C(=O)NCC2(C)CCC(NC(C3COC3)=O)C2)cc(Cl)c(F)c(Cl)c1 9641,C1(n2cc(CC(C3CCC(C)O3)=O)nn2)CCN(C(=O)Nc2cnn(C)c2N)CC1 9642,c1(C(=O)NCC2(F)CC(NC(C3(N(C)C)CCCC3)=O)C2)cccc(C2CC2)n1 9643,C(=O)(C(CC=C)C(C)C)NCC1(CNC(C(CC)OCC#C)=O)CCOCC1 9644,C1(CCNC(C2C(C)C2)=O)CCN(C(=O)Cc2cc(-c3ccco3)cs2)C(C)C1 9645,N1(C(CC(C)CNC(C2CCC3(CC2)CC3)=O)=O)CCC(F)(C#N)C1 9646,c1(C(C)NC(=O)NC2(c3cccs3)CCCCC2)cc(Cl)ccc1Cl 9647,c1(C(=O)NC2CC(CCNC(=O)Cc3csc(Cl)c3)C2)ccc(F)c2occc12 9648,n1(CC(=O)N(C2CN(C(C3CCOC(=O)CC3)=O)C2)C)[nH]cc2c(=O)ncnc1-2 9649,CC1CC(C(N2CCCC(C)(NC(c3ccc(C(C)(C)C)[nH]3)=O)C2)=O)CCC1=O 9650,c1(-n2ccc(SCC(=O)NC3CC(C)(NC(C(C)CO)=O)C3)n2)cccc(Cl)c1 9651,N#Cc1ccc(C(=O)NC2CCCN(C(c3cscn3)=O)C2)c(F)c1 9652,N1(C(C=CC(=O)OCC)=O)CC(CNC(=O)C2=C(C)OCC2)CC1(C)C 9653,Cc1oc(C)c(C(=O)NCC2CN(C(=O)CC34COC(C)(C3)C4)CCN2C)c1C 9654,C12(NC(c3c(NC)ccc(F)c3)=O)CCOCC1CN(C(c1cnc(S)[nH]1)=O)C2 9655,C12(C(N3CCC(COC)(NC(=O)CCC(N)=O)C3)=O)CC3CC(C1)C(=O)C(C3)C2 9656,C12(C(N(C)Cc3cn[nH]c3)=O)CC1CCN2C(C1CCSC1)=O 9657,N1(C(C(CCC)OC)=O)CC2CCC(C1)N2C(=O)COc1ccsc1Cl 9658,C1(C(=O)NCC2C(C(=O)NCc3cncnc3)CCO2)CC12CCCC2 9659,C1(N(C(COCCCC#C)=O)CC)CCCN(C(c2[nH]c(C)nc2CC)=O)C1 9660,C1(C(=O)NCc2scc(C(=O)NCC3=CCCCC3)c2)CC2CCC1CC2 9661,C(=O)(C1=NNC(=O)C1)NC(C)C=CC(=O)NC(C)(C)CCCO 9662,C=CCC(CC(=O)NCCC(O)C(C)CC)NC(=O)CC(C)(C)COC 9663,C#CCCC(C(=O)NCc1nc(COC)no1)NC(=O)C(COC)COC 9664,C1(C)(C(=O)NCC(CCCC)NC(c2ccc(C)c(Cl)c2)=O)CCCN(C)C1 9665,c1(C(=O)NC2CCN(C(C(C=C=C)C)=O)CC2)cc(=O)c2cc(F)ccc2o1 9666,C=CCN=c1[nH]cc(C(=O)NC2CCCC(NC(=O)CC3(OC)CCCC3)C2)s1 9667,c1(C(C)(C)OC)ccc(C(=O)NCCC(C)N(C)C(c2nocc2C)=O)cc1 9668,C12(NC(C(C)OC(C)(C)C)=O)COCC1CN(C(=O)CCCC1CCC1)C2 9669,c1(OC)cc(F)c(C(c2nnnn2C2CC2)NC2(C)CCSCC2)c(F)c1 9670,C1(C(NOCC(C(C)C)O)=O)CN(C(=O)CC2CC=CC2)CC1(F)F 9671,C1(NC(CN(C(=O)OC)C)=O)CC2CCC(C1)N2C(=O)Cc1sccc1Cl 9672,C(=O)(C(CCOC)OC)N(CC(C)NC(c1ccc(Cl)s1)=O)CC 9673,N1(C(CC(C(F)F)NC(C2(C)C(C)(C)C2(C)C)=O)=O)CCC(O)(C2CC2)CC1 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9692,CC1(C)CN(C(=O)C=CC(F)(F)F)CC1C(N1CC(CO)C(CO)C1)=O 9693,c1(C(=O)NC(CC=C)CNC2CC3C=CC2O3)cnn(C)c1-c1ccccc1 9694,N1(C(CC(C)F)=O)CCC(NC(=O)Cn2cc(Br)ccc2=O)C(F)C1 9695,CC(CCC(C)(C)C)C(=O)N1CCCCC1CNC(=O)CN1CCCC1=O 9696,N1(C(C=CC=CCC)=O)CCC(C(N2CCC(n3cnnn3)C2)=O)C1 9697,N1(C(c2sc(C)c(Br)c2)=O)C2CCC1(CNC(=O)C(C)CS(C)=O)CC2 9698,C1(C)(C(=O)NCc2ccnc(C)n2)CCCN(Cc2c(C)noc2C)C1 9699,Cc1ccc(I)cc1C(N1CC2C(NC(c3cccc(Br)c3O)=O)C2C1)=O 9700,c1(C(N2CCCC(N(C(C3CC3C(F)(F)F)=O)CC)C2)=O)cc(Cl)c(N)cc1F 9701,N1(C(C(CC#C)C)=O)CC2(CC(CNC(=O)CCC3CCCC(=O)N3)C2)C1 9702,n1(CC)cc(CC(=O)NC(C)C(N2CCCC2CCC(C)(C)CO)=O)cn1 9703,N1(C(c2nc(CC)oc2C)=O)CCC(CNC(c2ccccc2NC)=O)C1(C)C 9704,c1(C(=O)NC2C3(CC(NC(C4(CC)CCC4)=O)C3)C2)ccnc(O)c1Br 9705,N1(C(c2occ(OC)c(=O)c2)=O)CCC(NC(c2coc(C(C)=O)c2)=O)C12CC2 9706,C(C(C)C)(C(O)C(=O)NCCC(N1CC(O)(C(F)(F)F)C1)=O)OC.C(C(=O)O)S 9707,c1(CNC(c2ccc[nH]2)=O)nc2c(s1)CN(C(C1CCCCC(F)(F)C1)=O)CC2 9708,Cc1cnc(S(C)(=O)=O)nc1N(C(C1(F)CCNCC1)=O)CC1CCCN1C 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9885,N1(C(C2(S(N)(=O)=O)CC2)=O)CC2(C1)CN(C(C1(C3CCC3)CC1)=O)C2 9886,N1(c2cc(NC3C(C=C)OCC3)nc(C(C)C)n2)CCCC2(C1)OC(=O)NC2=O 9887,C1(NC(C)Cc2ccc(CO)cc2)CCCCC1C1CCN(CCCCC(N)=O)C1 9888,C#CC1(C)CCCN(C(=O)C(CCNC(=O)C(CC)N(CC)CC)OC)C1 9889,Cc1ncn(C)c(=O)c1C(=O)NCC1(NC(=O)C(N2CCCC2)C2CC2)CCC1 9890,CN=c1[nH]cc(C(=O)NCC2(NC(=O)CCCc3cc(C)no3)CCOC2)o1 9891,C1(NC(=O)Cc2cn[nH]c2)CC12CCN(C(c1ccc(O)cc1Cl)=O)CC2 9892,N1(CC)CCN(C(=O)C(C)CN(C(=O)C(C)C(F)(F)F)C)CC1C 9893,CC1=C(C(=O)NC2COCCC2NC(=O)C=Cc2cnc[nH]2)CCC1 9894,C(=O)(CCCCCC(=O)N1CC2CC2(NC(c2ccc(Cl)cc2C)=O)C1)OCC 9895,c1(C(=O)NC2CCC(NC(COCCOC)=O)CC2)c(C)ccc(Cl)c1O 9896,N1(C(c2cc(C)nn2C(C)(C)C)=O)CCC(F)C(NC(C2CCCC(C)C2)=O)C1 9897,Cc1c(C(N2CC(CCNC(=O)C(C)(C)C)OC(C)C2)=O)[nH]c2c1C(=O)CCC2 9898,N1(C(c2ccc(OC)s2)=O)CCC2CCN(C(c3ccc(OC)cc3CF)=O)C2C1 9899,C1(CNC(c2ncc[nH]2)=O)CC(F)CN1C(=O)CCC1OCCO1 9900,N1(C(c2c(OC)cccn2)=O)CCN(C(=O)C(Cl)=CCl)C(c2cccc(F)c2)C1 9901,CCCCC(C(=O)N1CCC(N(C(=O)CC23CC(C2)C3)C2CC2)CC1)NC(N)=O 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9955,c1(CC)c(N2CC(NC(C3CC(=O)N(CC(C)C)C3)=O)CCC2C)ncnc1Cl 9956,c1(C(N2CCCC(N(C)C(c3c[nH]ccc3=N)=O)C2)=O)ccnn2ccnc12 9957,N1(C(COC2(C#C)COC2)=O)CC(C(N2CCCCCC2)=O)C(C2CC2)C1 9958,c1(N(C)Cc2ccncc2F)cccc(S(=O)(=O)NC2CSC2)n1 9959,C1(CC(=O)NC2C(NC(=O)CC3(O)CCOCC3)CCCC2)CC(F)(F)C1(F)F 9960,c1(CCNC(=O)C(O)C2CCC2)ccccc1SC(F)(F)F 9961,C(=O)(CS(=O)(=O)C(C)(C)C)NC1C(C)CN(C(c2scnc2C(C)(C)C)=O)CC1 9962,c1(C(N2CCOCC(NC(c3cccc(SC)c3)=O)C2)=O)ccc2c(c1)CCC2 9963,N1(C(c2ccc3nc(C)oc3c2)=O)CCc2ccccc2C1CNC(=O)C1CC1 9964,C1(NC(c2c(OCC)nccc2)=O)CC(O)CN(C(C23CCCC(CO2)C3)=O)C1 9965,N1(C(C2CN(S(C)(=O)=O)C2)=O)CCCCC1C1(NC(C2CC2(Cl)Cl)=O)CC1 9966,c1(C(=O)NC2CC(NC(c3ccccc3O)=O)C2)cc2ccc(Br)cn2c1 9967,N1(C(CCOCCC)=O)CCCC1C1(NC(=O)C(C)NC(=O)Cn2cnnn2)CC1 9968,C1(C)(C(=O)NCC(n2cc(-c3cccc(NC)c3)nn2)C)CCC(=O)NC1 9969,Cc1cnccc1C(=O)NC1CCOC(CNC(=O)COC2CCCOC2)C1 9970,c1(C(N2CCC(OCC3CCC3)C2)C(=O)NCCCOC)ccc(C2CC2C)o1 9971,C(CCCCCC(=O)N1CCCC(O)CC1)OC.c12ccoc1C(=O)NC2 9972,c1(C(C(=O)NCC=C(C)C)NC(=O)C2=COCC2)ccc(C(C)(C)C)cc1 9973,C(=O)(C1=NOC(CNC(C2CCN2C(C)(C)C)=O)C1)N(C)CC1CCN(CC)C1 9974,C(CC(=O)N1CC(N(C)C(c2ccc(C)nn2)=O)C(C)(C)C1)(C(N)=O)NC(C)=O 9975,C(=O)(CC(C)(C)C(=O)NC1COCCC1C(=O)NCCC(C)(C)F)OC 9976,c1(C(N2CCC(CCCC)CC2)C(=O)NC2CCOC2)ccc(Cl)c(OC)c1 9977,N1(C(C(C=CC)O)=O)CCC(c2ccccc2CNC(C2(C(N)=O)CC2)=O)CC1 9978,N1(C(CCC2CCN(C(C3(CC)CCOC3)=O)CC2)=O)CC2C(C1)C2(F)F 9979,C1(CNC(c2cn(C3CC3)cn2)=O)C2CN(C(c3c[nH]cc3Br)=O)CC12 9980,C1(NC(CC2C(NC(c3nncc(OC)c3)=O)CCC2)=O)C2C=CC(C2)C1CO 9981,c1(C(=O)NC2C(CNC(CC(C)c3ccncc3)=O)C2)nnc2n1CCCCC2 9982,n1(CC(=O)NC2CCC(CC(=O)NCCOC3CCCCC3)C2)cccnc1=O 9983,CCC(CC1CCCC1)C(=O)NCC(=O)NCCNC(=O)Nc1ccc(Cl)cc1 9984,Cn1c(C(N2CCC(C)(CNC(=O)CC(F)(F)Cl)C2)=O)cc2sccc12 9985,C1(CC(=O)NCCc2cc(C(=O)NC(C3CSC3)C)no2)CCCCC1C 9986,C1(CNC(c2cc(C)c(Cl)cn2)=O)CN(C(=O)CCCOC(C)C)CC(C)(C)O1 9987,N1(C(C23CC(CC)(C2)C3)=O)CCN(C(c2c(C)nn(C)c2Cl)=O)CC1C.C1CC1 9988,C1(CCC)(CNC(=O)NCC(C2C(NC)C2)C)CCCC1 9989,N1(C(C2(C)CCC2)=O)CCC2(CCCN2C(=O)CS(=O)C(F)(F)F)C1 9990,c1(NC(=O)C(=O)NCc2ccccc2)nc(CCNC(C)CC2CCC2)cs1 9991,c1(CC)cccc(CC)c1CC(=O)N(C)CC1CCCN1C(C1CCOC1C)=O 9992,N1(C(c2c(CC)nco2)=O)CC2OCCN(C(=O)C(C)C(O)C(C)C)C2C1 9993,CC1(c2cn(CCCCCC#N)nn2)CCN(C(C2CCCCC2O)=O)CC1 9994,Cc1cc(NC(c2ocnc2C2CC2)=O)n(C2CCOC2)n1 9995,N12CCCC(C1)N(C(=O)C(C)C)C1(CC1)C2=O.C(C(C)C)NC(C)=O 9996,CC1(CNC(c2ccnc(S)c2)=O)CN(C(c2cccc(Cl)c2Cl)=O)CCO1 9997,C1(C)(CC)C=C(C(=O)NC2CC2NC(C2CC2C(=O)OC)=O)C1 9998,C1(CC(=O)NC(C2C(OCC)C2)=O)CCCCN1C(c1cc(C(C)=O)on1)=O 9999,c1(C(c2cnn(C(F)F)c2)NC(C2CCOC2)C)ccc(F)cc1 10000,C1(NC(N(C(C)C)CCc2ccsc2C)=O)CC=CCN1C(=O)OC(C)(C)C 10001,C(=O)(CCCCCCCC1CC1)NC(C)CNC(c1c(Cl)cnn1C)=O 10002,c1(-c2cc(CN(CCCNC(C3C(C)C3)=O)C)on2)cccc(F)c1 10003,C1(C)(NC(C(C(C)C)OCC)=O)CCN(C(=O)C(C2CCCCC2)N(C)C)CC1 10004,O=C(C1=CCC(NC(c2ccc(O)nn2)=O)C1)NCC1CCC(F)(F)C1 10005,N1(C(CCCC(C)=O)=O)CCC2(CC1)CCN(c1nc(O)c3c(ncn3C)n1)C2 10006,C1C#CC(=O)N1.C1(N(C)CC)CC(NC(C2CCCO2)=O)C1 10007,CC1(C)CN(C(=O)CC2(CO)CC2)CC1NC(C1(C)CCCS1(=O)=O)=O 10008,C1(NC(c2c(CC)onc2C)=O)CCCN(CCOc2ccc(Cl)cc2Cl)CC1 10009,C(CO)(C(C)(C)C)NC(CC1CC(C(=O)Nc2c(OC)ccs2)C1)=O 10010,C(C(C)C(=O)NCC1(C(C)(C)O)CN(C(=O)CCSC2CCCC2)C1)OCC 10011,CCCCC(C)CCC(=O)NCCCN(C(=O)C(c1ccccc1)F)C(C)C 10012,C1(CNC(COCC=C)=O)CCC2CN(C(c3ccncc3CC)=O)CCC2C1 10013,C1(=CC(N2CC(NC(=O)C=C3CCC3)CC(C)C2)=O)CCOc2ccccc21 10014,c1(CC)ccc(C(C)C(=O)NCC(O)CN(C(=O)CCOC(C)=O)C)cc1 10015,c1(CC(=O)N(C(CNC(c2c(CC)n[nH]c2)=O)C2CC2)C)cc(C)ccc1Br 10016,c1(C(=O)NC2CN(C(c3cc[nH]n3)=O)C3CC23)ccc2c[nH]nc2c1 10017,N1(C(c2c(C)cc(CNC(CC3ON=C(CC)C3)=O)o2)=O)C2CCC1CC(F)C2 10018,C#CCCCC(C(=O)NCCSC)N1CCC(Cn2cc(C)cn2)C1.OC 10019,C(CCCCC(=O)NC1(c2ccc(C)cc2F)CC1)NC(C(COCC)C)=O 10020,c1(NC(C)=O)cccc2c1CCCN2C(C1OCCC1C(=O)O)=O 10021,C1(NC(C)=O)CCC12CN(C(C1CCC(C(N)=O)CC1)=O)C2 10022,Cc1nc2ccc(C(=O)NCCC(C)NC(=O)C(C)O)cc2n(C)c1=O 10023,C1(C)(NC(C(c2ccc(Cl)s2)OC)=O)CCCN(C(c2coc(C(C)=O)c2)=O)C1 10024,c1(-n2cc(CCCC)nn2)cccc(C(=O)NCC(=O)N(CCSC)CC)c1 10025,C(=O)(C(C)(C)NC(=O)C(F)(F)F)N(C1CC(CNC(=O)CC(C)C)C1)CC 10026,N1(C(C(=C)C(C)C)=O)CC(F)(F)CC1C(N1C2CCC1COC2)=O 10027,N1(C(c2nc(C(C)=O)sc2)=O)CC(CNC(C2CS(=O)C2)=O)N2CCC1C2 10028,CC1(C)CC(NCc2ccc(C(F)F)o2)CC(O)C1 10029,c1(NC(C2CCC(CNCC3(SCC)CCC3)CC2)=O)ccc(F)c(Cl)c1 10030,c1(C(N2CC3C(NC(C4CCC(C)O4)=O)(C3)C2)=O)cc2c(Cl)nccc2s1 10031,CS(=O)c1ccc(C(=O)NCC2CC2NC(c2coc(Cl)n2)=O)cc1 10032,C1(NC(CCC2CCCN(C(c3c(C(C)C)occ3)=O)C2)=O)CNC(=O)C12CC2 10033,CCCC(O)CC(=O)NC(CN(C)C(c1nc(C)ccc1F)=O)CC 10034,C1(COC)(NC(=O)CC2CCCN2C)CCN(C(=O)C=CC(C)C)C1 10035,c1(NC(C23CC(NC(C4COCCC4O)=O)C(OC2)C3)=O)cn2ccccc2n1 10036,CC(CCCc1ccccc1)C(=O)NCC1CCN1C(=O)Cc1ccc(Cl)cn1 10037,C(c1ccc(F)c(OC)c1)=CC(N1C2CC(NC(C(CCOC)C)=O)C2CC1)=O 10038,N1(C(C(C)NC(CC)=O)=O)CC2CC1C2NC(=O)C(C)=CC1CC1 10039,c1(CC(=O)Nc2cnc(OC)c(C(N)=O)c2)nc2nc(C)cc(C)n2n1 10040,C#CCC(CC(=O)NC1CCCCCC1)NC(c1cccc(C)c1C)=O 10041,C(C(C)(C)C(=O)NCC1(CNC(=O)C(C2CCCCC2)F)CCCC1)SC 10042,c1(CN(C)C(=O)NCC2(c3cc[nH]n3)CC2)ccc(F)c(C(=O)O)c1 10043,N1(C(c2ccc(=NC)[nH]c2)=O)CCC(C)C(NC(=O)C(C)n2cccn2)C1C 10044,N1(C(C(C(=O)OC)C)=O)CCN(C(=O)C(F)F)CC1c1cn[nH]c1 10045,N1(C(Cc2ncc(C)[nH]2)=O)CCCC(CN(C)C(c2c(C)noc2C2CC2)=O)C1 10046,c1(C(N2CC(F)(COC)C2)=O)cccc(-n2cnnn2)c1.C12CC(C1)CNC2=O 10047,C1(C(=O)NC(CC)CNC(C2(OC(C)C)CCCC2)=O)CCC(F)(F)C1 10048,c1(CN2C(C(N3CCC(C(F)(F)F)C3)=O)CC(O)C2)cc([N+](=O)[O-])cc(Br)c1O 10049,Cc1ccc2nnc(CCNC(=O)CC3CC4CCCC4C3)n2c1 10050,N1(C(CC2CN(C(c3ccc(CC)s3)=O)CC23CC3)=O)CCn2ncc(C)c2C1 10051,C(=O)(C(CC(C)C)Sc1ccccc1)N(CCN(C(=O)C(O)C1CC1)CC)CC 10052,C1(F)(c2cn(CCC(=O)CC=C)nn2)CCCC1.C(CCC(=O)NC1CC1)NS(=O)(=O)CC 10053,c1(C2N3CCCC3CNC2=O)ccnc(Br)c1.c1(CSC(C)(C)C)ccccc1 10054,N#CC1CN(C(c2cc(Cl)ccc2Cl)=O)CCN1C(c1cnnc(Cl)c1)=O 10055,CCCCC(O)CC(=O)NCC1CC1CNC(C1CCC(CC)O1)=O 10056,C1(CS(C)(=O)=O)C2CCC1CN(CC(=O)NCCC1CCC(=O)N1)C2 10057,C(C(F)(F)C(=O)NC(C)COC1CCN(C(=O)CCc2ccsc2)CC1)OC 10058,N1(C(CCC2C(C)(C)C2)=O)CCN(CC2CC2NC(C2CC(=C3CC3)C2)=O)CC1 10059,N1(C(C=COCC)=O)CCCC(NC(=O)CCOCC2CCCO2)C1 10060,N1(C(Cn2ccc(C)n2)=O)CC2(C1)CN(C(=O)Cc1ccnc(F)c1)CC2CO 10061,c1(OC)ccc(-c2nc(C)c(C(=O)NCCC3(SC4CC4)CC3)s2)cc1 10062,c1(N(C(=O)CC2(C)CCCC2)CCC)cc(C)nnc1C 10063,N#Cc1c(F)cc(C(=O)NC2CC(CNC(=O)C3=CS(=O)CCC3)C2)cc1F 10064,C12(CNC(C(C)=CC)=O)CC(CO1)N(C(=O)C(c1ccccc1F)O)C2 10065,C(C(C)(C)CCCc1ccccc1)NC(CSC(C)CCO)=O 10066,Cc1ccc(C(C)CC(=O)NCC(O)CNC(c2ccnc(C3CC3)n2)=O)cc1 10067,N1(C(CC(CC)SC)=O)CCC2(CC(NC(c3csc(O)n3)=O)C2)C1 10068,C(=O)(C1=C(CCl)N(C2CC2)C(=O)NC1c1ccc(C)c2ccccc12)OCC 10069,C(=O)(C#CC1CCOC1)NC1C(C)(C)CN(C(=O)CSCc2csc(=N)[nH]2)C1 10070,C(=O)(C1=CN(C)S(=O)(=O)N=C1C)NCC(C(C)C)NC(C(C(CC)O)(C)C)=O 10071,C(=O)(C(CN=[N+]=[N-])NC(=O)CN1CCN(C)CC1)NCC(C)CCO 10072,CCCC(C(=O)NCCCN(C(C)C)Cc1csc(C(C)C)n1)OC 10073,N1(C(CC(=C)Br)=O)CC2CCCC2(NC(=O)CCc2ccccc2Cl)C1 10074,Cc1cc(P(C)(C)=O)oc1C(=O)NC(C)CNC(c1cc(C2CC2)cs1)=O 10075,N1(CC2(C)CC2C(=O)OC)CCC2(C1)CN(CCCc1n[nH]c(C)n1)C2 10076,N1(C(C=C(COC)C)=O)CC2ON=C(CNC(c3csnc3Br)=O)C2C1 10077,C1(NC(CCC#CC)=O)CC2(NC(c3scnc3COC)=O)COC1C2 10078,C1(C)(CCNC(C(CC)O)=O)CCN(C(c2ccc(-c3cc[nH]n3)cc2)=O)C1 10079,c1(OC)cccc(C(N2CCC(Br)C2)=O)c1.N12CCC(C1)OCC2=O 10080,Cc1ccc2c(CCCCCCC3(C(=O)CCCS(C)(=O)=O)N=N3)coc2c1 10081,C1(NC(C2(OCC)CCC2)=O)CCN(C(=O)C=C(C)C(C)(C)C)CC1CC 10082,C=C(C)CCC(=O)NC1CC(NC(=O)C(CCC)c2cccc(Cl)c2)C1 10083,C1(N=[N+]=[N-])(C(N(CC(C)(C)C)CC#C)=O)CCN(C(=O)CC2COCC2O)C1 10084,N12CCCC(C1)CC(=O)NC1(CC1)CC2=O.N1(CC)CC(N(C)CC)C1 10085,C1(NC(C2CC=C(C)C2)=O)(CF)CCN(C(=O)CCc2cncnc2)C1 10086,CC(C(O)C(F)F)NC(C1CC2CC2N1C(c1cccc(C2CC2)c1)=O)=O 10087,c1(C(N2CCCCC2C2CCCC2O)C(=O)NCCC)cc(Br)ccc1F 10088,CC1(C)C(c2cccc(Cl)c2)CCN1C(c1nn(CC(F)(F)F)cc1Cl)=O 10089,c1(C(=O)NC2CC(NC(c3c(CC)nccn3)=O)C2)nc(C2CC2)ncc1Cl 10090,CN1CCCC1C1CCCN1S(C)(=O)=O 10091,C(=O)(C#CC1CCCO1)NCC=CCNC(=O)COCC1(F)CC1 10092,C1(C(=O)NCC(CO)NC(C(C)CN2CCOCC2)=O)Cc2ccc(F)cc2O1 10093,C1(c2ccccc2)(NC(C(C)C2CCC2)=O)CCN(C(=O)COCCF)C1 10094,c1(C(=O)NCCCCCN(C(c2ccc(CC)nc2)=O)C)ccc(C)c(N)c1 10095,c1(C(=O)NC2C(CNC(CC3(COC)CC3)=O)C2)cn[nH]c1 10096,C1(NC(c2c(C)nns2)=O)CCCN(C(=O)CCc2cnccn2)C1C 10097,c1(C(=O)NC(C(=O)OC)C2CCCC2)csc(Cl)c1OC.C1C2CNCC12 10098,c1(NC(CCNC(C2CCCO2)=O)=O)ccc(O)cc1 10099,c1(C(=O)NC(C(C)NC(c2c(C)nsc2)=O)(C)C)cc(C2CC2)nnc1O 10100,c1(C(C)NC(CC2CCN(C(c3c(COC)cco3)=O)C2)=O)cncnc1O 10101,n1(C(CC)C)nc(CSC2CC2)nc1-c1ccc(OC(F)F)cc1 10102,CC(CCN(C(=O)CCc1nncs1)C)NC(C1CC1CN(C)C)=O 10103,Cc1cccc(N2CCC(NC3CC4CC4C3)C2=O)c1 10104,N1(C(C(Cn2ccc(C)n2)C)=O)CCC2CN(C(c3cn(C)ccc3=O)=O)C2C1 10105,C1(n2cccn2)(NC(C2C3CC(=O)CC32)=O)CCN(C(=O)CC(F)(F)F)CC1 10106,c1(C(=O)NCC(CN(C(c2ncc(C)c(C)c2)=O)C)C)ccc2ccnn2c1 10107,C1(C(N2CC(OC)(CNC(=O)C(C)C3CCCC3)C2)=O)COC(=O)N1C 10108,N1(C(C2CC(SC)C2)=O)CC(NC(c2csnc2C)=O)CC12CCCC2 10109,CC(=O)CCCC(=O)N(CC(=O)NCC1CC(O)C1(C)C)C(C)C 10110,C1(NC(c2c(CC)nns2)=O)CN(C(=O)C2=CSCCO2)CCC1CO 10111,N1(C(c2cn(C)c(=O)cc2)=O)CC(NC(=O)CC2CC(=O)C2)CC12CCCCC2 10112,CCC(C(=O)NCC1(CCNC(=O)Cc2ccncc2Cl)CC1)C(F)(F)F 10113,C12(NC(=O)COc3ccon3)CCCN(C(C3(CO)COC3)=O)CC1C2 10114,N1(C(c2n(CC)ccn2)=O)CC2CC1C2NC(=O)CN1C(=O)CCC1=O 10115,C1(CCC(=O)OC)CCCN(Cc2ncc(F)cn2)C1 10116,c1(C(=O)O)cnn2cc(CNc3cccc4cc[nH]c34)cnc12 10117,c1(C(N(CC(CN(C(=O)CC2CCCC2)C)O)C)=O)cc(P(C)(C)=O)cs1 10118,CC1CC(C2CN(C(C3CC=CCC3NC(C3OCCCC3(C)C)=O)=O)C2)=NO1 10119,c1(OC(N(CCC(=O)NCCC)CC(=O)NC)=O)cc(Br)c[nH]1 10120,c1(C(=O)NCC(CNC(CCCOCC=C)=O)O)ccc(S(=O)(=O)C(F)F)cc1 10121,Cc1cccc2c(=O)c(C(=O)NC(CNC(=O)COc3ccon3)C(C)C)c[nH]c12 10122,c1(C(N2CC(F)CC(NC(=O)CSc3ncccn3)C2)=O)cc2cn[nH]c2cn1 10123,c1(C(=O)NCCC2(NC(C3C(C)(C)C(F)(F)C3)=O)CCC2)ccccc1[N+](=O)[O-] 10124,CC1C(=O)CC2CCCC1N2C(=O)NNc1ccc(C(F)(F)F)cc1 10125,Cn1cc(CC(=O)NC2(CNC(=O)C(C)(c3cccs3)SC3CC3)CCOC2)cn1 10126,c1(C(=O)NCC2CC(COC)CN2C(=O)C(F)F)cccc(Br)c1C 10127,c1(C(=O)Nc2c(C)onc2-c2ccccc2F)cc(=O)c2ccccc2[nH]1 10128,c1(NC2CCCCN(C(C3C(C(=O)OC)C3)=O)C2)ncnc(OC)c1F 10129,C(=O)(C(N=[N+]=[N-])C(C)C)NC1CC(C(C(N2CCCC(C(=O)OC)CC2)=O)F)C1 10130,CCC(C)(CS(C)(=O)=O)C(=O)NCC(O)CNC(=O)CNC(=O)NC 10131,c1(C(=O)NC2(CN(C(C(CC)OC)=O)C)CC2)cc2c(C#N)cccc2[nH]1 10132,N1(C(CSCC#C)=O)CC(C2CCCN(C(C3(CO)CCCO3)=O)C2)C1 10133,N1(C(Cc2c(C)nc[nH]2)=O)CCC(C(F)(F)F)C(NC(C2(C(C)C)CCC2)=O)C1 10134,CN1CCC(C(=O)OCC(=O)Nc2cccn2C(Cc2ccccn2)CO)CC1=O 10135,c1(C(N(CCC(C)NC(=O)C(C)(C)C)C)=O)ccc2c(c1)OC(C)(C)OC2 10136,CC(C1OCCc2ccccc21)NCc1csc(Br)n1 10137,O=C(C(O)CNC(=O)Cc1cccnc1)NC(C1CCCC1)CO 10138,N1(C(c2c(C)scc2)=O)CCC(C(=O)NCC(F)Br)C1(C)C 10139,C1(NC(C2(CCC)CCC2)=O)COCCN(C(=O)COc2cccnc2)C1 10140,N1(C(c2ccc(SCC)c(C)c2)=O)CC=CCC12CCOCC2 10141,C1(CNC(CNS(N)(=O)=O)=O)CC2(CCC2)CN1C(c1cccc(C2CC2)n1)=O 10142,n1(CC)nccc1S(=O)(=O)NC(=O)N(CCCNC(=O)OC(C)(C)C)C 10143,N(C)(S(=O)(=O)N1CC(C(N)=O)CCO1)C(C)C 10144,c1(C(C(=O)NCC=CCl)NC(CN(C)CC)=O)cnn(C)c1 10145,C1(Nc2c(C)ccc(C)c2)CCN(N2CCCC(OC(F)(F)F)CC2)CC1 10146,N1(C(C(c2cccs2)NC(CC2C(C)(C)C(O)C2)=O)=O)CCOCC2(CC2)C1 10147,C1(C(=O)NC(COC)CO)CN(C(=O)CCOCC(F)F)C2(CCC2)C1.C1CN1 10148,C(N=c1[nH]c(N(CCC#CCO)C)nc2c1CCCCC2)c1ccc(SC)cc1 10149,C(=O)(CS(=O)(=O)CCO)NC1CCCC(NC(c2cncc(SCC)n2)=O)C1 10150,N1(C(C(COC)CC(C)C)=O)CC(C)OC2(CCN(C(=O)CCC(C)C)CC2)C1 10151,C1(C(=O)NC2CC(CNC(c3c(C(C)C)noc3)=O)C2)CCCCC12OCCO2 10152,C(CCC(N)=O)(C(=O)N(CC(C)C)Cc1cncn1C)NC(C)=O 10153,c1(CN(C(C(C(C)C)O)=O)C2CCCC2)ncnc2ccc(C(F)(F)F)cc12 10154,C(CCCCC(=O)NC1CCOC(CNC(c2ccnn2CC(F)F)=O)C1)OC 10155,Cc1nsc(CN(C)C(c2cn(CCNC(=O)CC(C)F)nn2)=O)n1 10156,C(CC(C)C(F)(F)F)NC(CC1(O)CCN(C(Cc2cccc(C)c2)=O)C1)=O 10157,C1(CNC(COCCOCC#C)=O)CC(C)N(C(=O)C(F)(F)C2CCOCC2)C1 10158,N1(C(C(C2CCC2)OC)=O)CC(N(C(=O)CC2CN(C)C2)C)C(C)(C)C1 10159,C1(NC(C2C(C(C)(C)C)C2)=O)CC2(CCN(C(C3(C)CCOC3)=O)C2)C1 10160,C1(NC2CCC(CC(=O)OC)C2)CCN(Cc2cccc(OC)c2C)CC1(C)C 10161,c1(C(N2CCC(O)(CNC(C3C(CCOC)C3)=O)C2)=O)ccc([N+](=O)[O-])o1 10162,C(=O)(C(C)(O)C(C)C)N1C(CCNC(C(c2nc(C)sc2)=O)=O)CCCC1 10163,C=C(C)CCCC(=O)NCCC1(O)CCCN(C(c2cc(COC)on2)=O)C1 10164,C1(NC(C(C)OC)=O)CCN(C(c2ccc(NC(C)=O)s2)=O)CC1(C)C 10165,CC(C)C(C(=O)N(C(CN(C)C)CCO)C)CCC(=O)OC(C)(C)C 10166,C=CCCCCC(=O)NCCCNC(=O)CO.C12(CC1)C(=O)NC2 10167,N1(C(=O)NC(C)(C)N)CCCC(Cn2cc(COC)nn2)C1 10168,N1(C(=O)NCc2ncc(CC)s2)CCCCC1CCNC(C)=O 10169,c1(CCCC(=O)Nc2ncnc(OC)c2OC)cccc([N+](=O)[O-])c1.C12CCN1C2 10170,CC(C(=O)NC1(CNC(C2(C(F)F)CCC2)=O)CCC1)F 10171,Cc1ncc(CNc2ccc(-c3cnc(N4CCC4)nc3)nc2)cc1Br 10172,C(=O)(C1CCc2ccccc21)NC1(C(N(C)CC2CCCOC2)=O)CC(CO)C1 10173,C1(CC=C)(NC(c2cnn(CCOC)c2)=O)CCCN(C(=O)Cc2ccns2)C1 10174,C#CCCCCCC(=O)N1CC(C2CN(C(C3CCCOCC3)=O)C2)C1 10175,Cc1cc(C(=O)Nc2ccc(NC(=O)CCn3ccnn3)c(C)c2)ncc1N 10176,c1(C(=O)O)ccc(S(=O)(=O)N2CCC3C(F)(F)C3(c3ccccc3)C2)nc1 10177,c1(C(=O)NCCC2CCCN(C(C3CC(F)C3)=O)C2)nccc2n[nH]cc12 10178,c1(C(N(C2CC(N(C(C3(n4ccnc4)CC3)=O)C3CC3)C2)C)=O)cnc(Br)s1 10179,N1(C(CC(C)OC)=O)CC2(CCN(C(=O)C(C)Sc3ccc(N)cc3)C2)C1 10180,c1(C(N2CCC(CC(=O)NC(C)C)CC2)C(=O)NC)sc(C)c(Br)c1C 10181,C1(C#N)(NC(Cc2ccc(OC)cn2)=O)CCN(C(C2(CN(C)C)CC2)=O)C1 10182,C(=O)(C(CC)(CC)NC(C)=O)N(CCNC(C(CC=CCC)C)=O)C 10183,c1(C(=O)NC2(CO)CN(C(Cc3cccc(OC)n3)=O)C2)ccc2snnc2c1 10184,c1(C(N2C(CNC(CNS(N)(=O)=O)=O)CC(O)C2)=O)cnn2c1CCC2 10185,O=C1CC2(CCCN(CC3CCCOC3C(F)(F)F)CC2)N1 10186,CC(CSC(F)(F)F)C(=O)N1CCCC1CN(C)C(c1ccco1)=O 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10310,C(=O)(C(C)C(C)S(C)(=O)=O)N1CC2C(NC(C(CC(C)C)N(C)C)=O)C(C2)C1 10311,C(=O)(CCCCCCN=[N+]=[N-])NCC1N(C(CCC2OCC(C)(C)C2)=O)CCC1 10312,C(=O)(NN=Cc1cccnc1)c1sc2cc(C)sc2c1 10313,N1(C(C(F)=CC)=O)CCC2(CC1)C(NC(=O)CSc1ccncc1)CS2(=O)=O 10314,C(=O)(N1CCCc2ccnn21)NC(=O)CC1CCC1.C12(CCOCC1)C(=O)N2 10315,c1(CC(=O)NCCN(CCC)C(C2CC(=C3CCC3)C2)=O)cc(CC)no1 10316,N1(C(C(CC(=C)C)OC)=O)CC2(NC(C3C4CCCCCC34)=O)CCC1CC2 10317,c1(OC)cc(OC)cc(C(=O)NC2CCCC2CNC(C2CN(C(N)=O)C2)=O)c1 10318,C1(C(=O)NC(c2onc(C)n2)C)CCC(C)N(C(=O)C(O)CC(N)=O)C1 10319,CC(C(C)(C)CN(C)C)NC(=O)CC1C=CC(NC(=O)COCCCN(C)C)C1 10320,Nc1cc(C(N2CC(CNC(C3(CO)CCOC3)=O)C2)=O)cc(F)c1 10321,c1(OC)cccc(C2(N)CCC2)c1.c1(CC2CC2)nnnn1C1(C)CC1 10322,CC1(C2CCCN(C(=O)CSc3cn(C4CCCC(NC(N)=O)C4)nn3)C2)CC1 10323,c1(CC)cc(N)ccc1C(=O)NCCC(O)CNC(=O)CCC1CCCOC1 10324,N1(C(c2c(C)nn(C3CCC3)c2)=O)CCC2(CCC2)C(NC(C2CC(O)C2)=O)C1 10325,n1(CC(=O)NCCC(C)NC(=O)CCOC2CC2)cnccc1=O 10326,c1(OC)ccnc(O)c1C(=O)NC1CCCCN(C(C2C3CC(=O)CC23)=O)C1 10327,N1(Cc2onc(C(C)(C)C)n2)CC(C)(C)OC2(CCCOC2)C1 10328,N1(C(COCC(C)C)=O)CCC(N(C)C(C2CC3(CC(=O)C3)C2)=O)C(C)C1 10329,CC(CC1CCC1)C(=O)NCC1(NC(c2cnnn2C)=O)CCCC1 10330,C1(C(C(C)C)NC(Cc2nnc(C)o2)=O)CCN(C(C2(O)COC2)=O)CC1 10331,C(=O)(C1=CC2CCC1C2)N1CC2C(CNC(c3cn(CCOC)nc3C)=O)C2C1 10332,S(=O)(=O)(c1cccs1)NC1(CC)CN(C(c2nccc(Cl)c2OC)=O)C1 10333,c1(N2CCC(=CCNC(C(CSC)(C)C)=O)CC2)nc(O)c2ccc(Cl)cc2n1 10334,c1(C2(C(N(C(C)CNC(C3CC3[N+](=O)[O-])=O)CC)=O)CCC2)ccccc1 10335,C1(NC(CCNC(=O)OCC)=O)CCC2CN(C(C3CCSC(C)C3)=O)CCC2C1 10336,N1(C(CC(=O)NC(CNC(C(C)P(C)(C)=O)=O)(C)C)C)CCCc2ccccc21 10337,c1(OC)c(C(N2CC(=C(F)CNC(=O)CC(O)C3CC3)C2)=O)c(C)nn1C 10338,C1(NC(C23CC(C)C2C3)=O)CN(C(c2ccc(C(F)F)o2)=O)C(C)(C)C1 10339,N1(C(C(=O)NCC(CC)NC(c2ccnn2CCF)=O)C)C(=O)CCC1=O 10340,c1(NC(C(C2(C)CC2)NC(c2cnc(OC)s2)=O)=O)ccc2c[nH]nc2c1 10341,C(=O)(C(C)(C)C(CC)NC(c1nnnn1-c1ccc(OC)c(C)c1)C(C)C)NC 10342,Cn1cnc2cc(C(N3CC4(CC(NC(c5c[nH]ccc5=N)=O)C4)C3)=O)ccc12 10343,CC(C)(C)C(O)CCC(=O)NCCC1CN(C(C2CC2CF)=O)C1 10344,c1(C(C)C)ccccc1OCC(=O)N(C1CN(C(c2[nH]nnc2C2CC2)=O)C1)C 10345,Cn1ccc2nc(N3CC4(CC4)CC3C(=O)NCC(O)CN3CCCC3)ncc12 10346,c1(CN(C)CCC2CCCCCC2)ccc2c(c1)CCCN2 10347,c1(CC(N2CC3(C2)SCCC3NC(c2ccno2)=O)=O)ccc2nsnc2c1 10348,CCC(C)(C)CCCC(=O)N1CCC(N(C)C(C2CC3CCC3C2)=O)C1 10349,C#CCC(C(=O)N1CC(OC)C(F)C1)NC(=O)CCN=[N+]=[N-] 10350,c1(OC)cnc(C(=O)N(C(C)CNC(c2n[nH]cc2C(F)(F)F)=O)C)c(OC)n1 10351,C(C#Cc1cn(-c2nccc(Cl)c2F)nn1)NC(C1CN2CCN1CC2)=O 10352,C1(CC)CN(C(C2CC(O)CN2C(c2nnsc2N(C)C)=O)=O)CCC1OC 10353,c1(CC(=O)NCC(C)(CO)NC(CCC(C)OCC)=O)cccc2c1OCCO2 10354,CC(C)CC(=O)C(=O)N(CCCCC(=O)NC(C)CCCCO)C 10355,N1(C(CCNC(=O)C2CC2)=O)CCC2(CC1)OCCCC2NC(=O)Cc1cc[nH]n1 10356,C1(C(=O)NCC(C)NC(c2cc(C)on2)=O)C2CN(CC(F)(F)F)CC12 10357,C1(OC)CCC12CC(C(=O)NCC(C1CCN(C(c3n[nH]c(=N)s3)=O)CC1)F)C2 10358,C(CCF)(C(=O)NCC(c1ccccn1)O)NC(c1c(C)csn1)=O 10359,C#Cc1cc(C(=O)NCC(C(C)C)NC(C2CCC(=O)NC2)=O)cc(Cl)c1 10360,C(=O)(CC(C)C(F)(F)F)NCC(C)NC(c1onc(CC)c1C)=O 10361,N1(C(C2(OC)CC2)=O)CC(NC(c2ccc(Cc3nccs3)cc2)=O)C(O)C1 10362,N1(C(C2N(C(CN(C)C(=O)C3CC3)=O)C(C3CC3)CC2)=O)CCOC(C2(C)N=N2)C1 10363,C1(CNC(C(C)N(CCOCC)C(C2CCCC2)=O)=O)CCNC(=O)C1 10364,C(c1ccc(CN(C)Cc2cc(Br)ccc2Cl)cc1)=CC(=O)OC 10365,CC(C(=O)NCCOCCOCCNC(=O)C=Cc1ncc[nH]1)C(C)O 10366,CCCCS(=O)(=O)CC(=O)NCC1(C2CC2)CCN(C(C2CCS(=O)(=O)C2)=O)C1 10367,c1(CN2CCC(C#N)(N(C)C)C2)cc(Br)cc(F)c1O 10368,S(=O)(=O)(c1c[nH]c(C(N2CC(NC(=O)C(C)N(C)C)C(C3CC3)C2)=O)c1)NC 10369,CC1CCCC=C(C(=O)NC(CC2CCCC2)C(=O)NCC2SCCS2)C1 10370,N1(Cc2cc(OC)cc(Br)c2)CCC2(CC1)CC2NC(c1ccn(C(C)C)n1)=O 10371,C1(NC(COC(CC)C)=O)CC2CN(C(=O)CC3CCCCC3(C)C)CC2C1 10372,C1(C(N2CCN(C3CN(C(c4ccc(=N)[nH]c4)=O)C3)CC2)=O)CC(C2CC2)=NO1 10373,C1(O)(CNC(c2csc(-c3ncc[nH]3)n2)=O)CCN(C(=O)Cc2cnns2)CC1 10374,c1(C(=O)NCC(C)(CC)NC(CC(CC)C(F)F)=O)c(F)ccc2occc12 10375,c1(CC(=O)Nc2cn(CC(=O)OC)nn2)ccc2c(c1)CN(CCn1cncn1)C2 10376,C(=O)(C1CCCc2sc(=N)[nH]c21)N1C(CNC(CNC(CC)=O)=O)CC(F)C1 10377,C(=O)(C(CCS(C)(=O)=O)OC)NC1CCN(C(CSCC#C)=O)CC(O)C1 10378,C1(n2c(C(CO)NCCSC(F)F)nnn2)CCC(F)(F)CC1 10379,C(CN=c1cc[nH]c(=NCCCCCCS(N)(=O)=O)[nH]1)NC1CCCC(C)CC1 10380,C12(NC(CNC(C3CCC3)=O)=O)CC1CN(C(=O)CC(F)(F)Cl)C2 10381,c1(NC(C2CNCC2NC2(n3ccnn3)CC2)=O)ccc(Cl)cc1 10382,N1(C(C(=O)NCC2CCSCC2)=O)CCN(c2ccc(F)cc2F)C(=O)C1 10383,C1(C2(O)CCN(C(=O)C(C)C(C)(C)C)CC2)(NC(CCc2scc(C)n2)=O)CC1 10384,N1(C(C(CNC(C2CCC(=O)N2)=O)CC2CC2)=O)CCSC2(CCC2)C1 10385,CC1COC(C)CN1CCCNC(c1cc(Cl)sc1Cl)=O 10386,C=Cc1ccc(C(=O)NC(CCCOC)C(=O)Nc2ccn(C(C)C)n2)cc1 10387,C1(C(N(CCCC)CCCC)=O)CCCC1CNC(c1c[nH]cc1C)=O 10388,C#CCC(CC(=O)Nc1cncnc1C)NC(C1OCCC1C(C)C)=O 10389,C(C(COC)C(=O)NCCC(N1CCOC(C2CC2)C1)=O)OC 10390,c1(C(=O)NC2CC2CNC(C2CC3COCC3C2)=O)ccc([N+](=O)[O-])cc1Cl 10391,C1(C(=O)NCC2CN(C(CCC#C)=O)CC2O)CNC(=O)CC12CCC2 10392,Cc1cc(CNC(N2CC3(OC(C)(C)C)CC2CO3)=O)c2[nH]cnc2c1 10393,N1(CC)C(=O)CCC1CC(=O)N(C)CCOCCN(C(=O)Cn1nnc(=N)[nH]1)C 10394,c1(C(N2C(CNC(C(c3nccc(C)c3)(C)C)=O)CCC2)=O)cc(Cl)ccc1N 10395,C(C(=O)NCCC1(OC)CN(C(=O)C(C)(C)C)C1)(C(C)C)OCC(C)C 10396,N1(CCNC(C2CCCN2S(C)(=O)=O)=O)CCC(O)C1.C1(=O)C=CCCCN1C 10397,c1(C(N(CCCn2cc(CCC(=O)O)nn2)C2CC2)=O)ccc2c(c1)CCSC2 10398,c1(CC)cnn2ccc(C(N3CCN(C(c4cscc4C)=O)C(C)C3)=O)nc12 10399,c1(C(N2CCC3C(NC(c4ccc5c(c4)CC5)=O)C32)=O)cnc2sccn12 10400,N1(C(C=CC)=O)CC2CN(C(C3C4C=CC(C4)C3CO)=O)CC(C1)O2 10401,Cc1cnc(C(=O)NCc2cccc(NC(=O)C(CC#N)c3ccccc3)c2)nc1 10402,C#Cc1ccc(CN=c2[nH]c(CC(N3CCC(CO)C(O)C3)=O)cs2)cc1 10403,c1(NC(c2ccccc2)NCCC(=O)NC)ccc([N+](=O)[O-])c(F)c1 10404,N1(C(C2CCC(=C)CC2)=O)CCCCC(NC(c2cc(C)[nH]n2)=O)CC1 10405,N1(C(C(CCC)CCC)=O)CC2(C1)CN(C(=O)C=Cc1cc[nH]n1)CCO2 10406,CC1(CNC(=O)NC2CC(N3CCC3)C2)CCC(CO)CC1 10407,C(CCCCCNn1cc(C2C3CN(C(=O)C(F)OC(F)(F)F)CC23)nn1)SC 10408,C1CN=C2N=C(C=CN2)N(C)C2CCC1C2.c1(OC)cc(C2(C)CC2)on1 10409,Cc1nc(C(=O)NC(C2(O)CN(C(=O)CC3CCC(=O)N3)C2)C)c(Br)s1 10410,c1(NC(C)CN=[N+]=[N-])cc(F)cc(F)c1Cl 10411,c1(C(N(CC(CC)NC(C2C3CCCC23)=O)CC)=O)csc(-c2ccccc2)n1 10412,C(=O)(CCC(C)(C)F)NC1CCN(C(C(C)NC(CC)(C)C)=O)C1 10413,C(=O)(C(O)CC(C)C)N1C(COC)(CNC(=O)CN(C(=O)C(C)C)C)CCC1 10414,C1(CCC(C)C)CCN(C(=NCCCCC(F)(F)F)NC(C)CCF)C1 10415,C1(C(=O)NCC(C(=O)N(CC(O)CF)C)N(C)C)C2CC(=O)CC12 10416,C(=O)(C(CC(C)C)C(N)=O)NC(CC=C)CNC(c1sc(F)cc1Cl)=O 10417,C=CCC(CNC(c1cn2c(n1)CCC2)=O)C(=O)NC(CN(C)C)CO 10418,C(=O)(C(C)C1=CCCC1)NC(CCCC)Cc1ccccc1.N1(CCN)CCCNS1(=O)=O 10419,C1(OCC=C)CCN(C(=O)C(CN(C)C)NC(=O)CCc2cc(C)on2)C1 10420,C1(CNC(C(C)=CC)=O)CCN(C(C2CCn3cc(C)nc3C2)=O)CCC1(F)F 10421,Cc1cccc(C(=O)NCC2(C)CCCN2C(=O)CC2C=CCC2)c1Br 10422,c1(CNCCCF)cc(OC)c(OC)c(Br)c1.C#CC1CCCC1CCO 10423,Cc1ncc2n1CCC(C(=O)NC1CCC(CNC(C3(C(C)C)CC3)=O)C1)C2 10424,c1(N(S(=O)(=O)CC2(O)CCCC2)CCNCc2ccc(F)nc2)cncc(Cl)n1 10425,N1(C(CC(C)NC(N)=O)=O)C2CC1CN(C(C1(Oc3ccccc3F)CC1)=O)C2 10426,c1(C(=O)NCCN(C(c2cccnc2O)=O)CC)cccc2c1OCC2(C)C 10427,N1(C(=O)NC2(C(C)C)COC2)CCC(N=c2nc(C3CCCC3)[nH]s2)CC1 10428,C1(CNC(c2c(OC)n[nH]c2)=O)CN(C(C2(F)CC=CCC2)=O)CCN1C 10429,C(c1ccncn1)=CC(=O)NC(CNC(CNS(NC)(=O)=O)=O)CO 10430,c1(CN(C(CC2CN(C(CC3(COC)CC3)=O)C2)=O)C)cn(C(C)C)nn1 10431,C(=O)(C1(C)CCn2ccnc21)NCC(C)CNC(=O)Cc1csc(C(F)(F)F)n1 10432,C1(CC)CCOCCN1C(=O)CC1CCCCC1NC(c1cc(C)no1)=O 10433,C(C1c2ccccc2CN1C(C1CC1c1ccc(C)s1)=O)NC(C(C=C=C)C)=O 10434,C=CC1(O)CCN(C(=O)CCN(CCCO)C(c2cc(O)n(CC)n2)=O)C1 10435,c1(C(=O)NCC2(O)CCN(C(Cc3n(C)nnc3)=O)C2)c2c(nn1C)CCSC2 10436,c1(C(=O)NC2CCN(C(=O)CCCc3nccs3)C2)ccc([N+](=O)[O-])o1 10437,Cc1cc(C(=O)NC2CC(F)CN(C(C3CC(=O)OC3(C)C)=O)C2)cc(Cl)c1 10438,C1(C(=O)NCCC2(C(=O)NCC(COC)CO)CCC2)CCC(C)(C)C1 10439,C1(CC)CCc2nnnn2CC1.C12C(C)CN(CCN1C(=O)OC(C)(C)C)C(=O)N2 10440,Cc1cc(=NCC(C)CNC(=O)C=C2CCSCC2)[nH]c(C(C)C)n1 10441,C(=O)(C(C)S(=O)(=O)CCC)NCC(CC=C)NC(c1nc2cc(F)ccc2s1)=O 10442,N1(C(C2C(C)C2)=O)CC=CC(NC(C2CCCN2C(c2ccc(Br)o2)=O)=O)C1 10443,C1(C(=O)NCC2(C)CCCN2C(C2(C(=O)NC)CC2)=O)(C2CC2)CC2(CCC2)C1 10444,Cc1cccc(C(=O)NCC2(CNC(C3(C(F)F)CCCO3)=O)CC23CCC3)n1 10445,C#Cc1cnc(C(N2CCOCCC2C(=O)NCC(C2CCC2)OC)=O)c(C)c1 10446,C1(C(=O)NC2CC(C(F)C(=O)NCCc3cncs3)C2)COC(=O)C1 10447,C(c1ccc(C2CC2C)o1)=CC(=O)NCC(N(C(C=CC)=O)C)C1CC1 10448,C(=O)(C1=CCC(C)CC1)N1CCC(C(C)NC(=O)Cn2cnnc2O)C1 10449,c1(C(N2C3CC(CNC(c4cc(C)nc(C)c4)=O)(OC3)C2)=O)nc2cccnc2s1 10450,c1(COC)cncc(C(=O)NCC(F)CNC(C2(C(=O)N(C)C)CCC2)=O)c1 10451,C(=O)(CC(O)CNC(=O)Cc1cccnc1O)N1C(CCC#C)CCC1 10452,c1(CC)cccc(F)c1C(N1CCN(C(C2COC(C(C)C)C2)=O)CC1)=O 10453,c1(C(N(CCN(C)C(c2csc(C3CC3)n2)=O)C)=O)c(N)ccc(F)c1F 10454,c1(C(=O)NC(CC2CCC2)C(=O)NCc2cscn2)cc(F)c(F)cc1 10455,C(CCC(C)(C)NC(=O)CCCC#N)NC(C(c1cccc(O)c1)C)=O 10456,Cc1ccc(C#N)c(-c2cn(-c3cc(F)cc(Br)c3)nn2)c1 10457,N1(C(C2N(CC)CC2)=O)CC2(CC2)CC1CNC(c1ccccc1COC)=O 10458,Cc1cc(C(=O)NCCCCNC(c2sc(C)cc2Br)=O)ncc1F 10459,C1(NC(CC(C)(C)NC(CCN(C)CC)=O)=O)CCCCC1(C)O 10460,N1(C(C2CCC(C)(C)O2)=O)CCCC2CN(C(c3c[nH]nc3F)=O)CCC12 10461,c1(C(N(CCOC)CCNC(C2CCC(OC)CC2)=O)=O)cc(C)nc(C)n1 10462,N1(C(c2cccc(NC(C)=O)c2)=O)CC2CC(NC(C3CCS(=O)(=O)N3)=O)C1C2 10463,CCCCC(C(=O)N1CCC(CCO)CC1)NC(c1cn(C)nc1OC)=O 10464,C1(C(N2CC3C(NC(c4ccc[n+]([O-])c4)=O)C3C2)=O)COc2ccc(O)cc2O1 10465,Cn1cnc2[nH]c(=NCC3CCC4(CCC4)C3NC(C3CC3F)=O)nc(O)c12 10466,C(=O)(CCC(O)C(C)(C)C)N1CCC(CCNC(CNC(CN(C)C)=O)=O)CC1 10467,N1(C(c2c(CC)ccs2)C(=O)NC2CC(C(N)=O)C2)CC2CCC(C(=O)OC)(C2)C1 10468,c1(OC)ccc(C(=O)OCC(O)CNC(C2(c3ccccc3)CC(C)C2)=O)cc1 10469,c1(C(=O)NCC(CO)NC(c2ccc(C(C)(C)C)nc2)=O)ccc(Cl)c(F)c1 10470,Cn1cc(C(N2CCC(OCCNC(=O)C3=CCCC3)CC2)=O)c(Br)n1 10471,CCCC(CN=c1cccc(S(=O)(=O)NC2CC(=C3CC3)C2)[nH]1)OC 10472,C1(CC(=O)N(CCOCCNC(c2c(C)csc2)=O)C)CCCC(=O)N1 10473,CCC(CC(F)(F)F)N=c1[nH]c(=NCc2cccc(C)n2)[nH]c2c1COC2 10474,C1(C(=O)NCCOCCCNC(C(C)C2=CCCC2)=O)CCC2(CC1)CC2(F)F 10475,C1(N(C(=O)C(c2ccc(F)cc2)F)CCOC)CCCC12CCOCC2 10476,CC(C)CN=C(NCc1cncc(Br)c1)NCC1CCN(C2CC2)C1 10477,CC(CO)C(=O)NCCOCCCN(C)C(c1cnn(C)c1)=O 10478,C=Cc1ccc(C(=O)NCC(C)(O)CNC(=O)COCc2ccccc2)cc1 10479,C(CCCC(=O)N(C)CCOCCN(C(=O)CCS(C)=O)C)OC.C(CSC)O 10480,n1(CC(N2CCCC(NC(C(CC)O)=O)CC2)=O)c(=O)nc(O)c2ccccc12 10481,c1(OC)c(F)cc(F)c(C(=O)NC2COCC2C(N2CCNC(=O)C2)=O)c1F 10482,c1(C(N2CCC(OCc3ccnn3C)C2)C(=O)NCC=C)cc(Cl)nn1C 10483,c1(C(C)NC(c2cn[nH]c2)=O)nocc1C(=O)NCC1(F)CC1 10484,c1(C(N(CC=C)CCC)=O)ccc(Sc2ccc(C(F)(F)F)cc2)cc1 10485,c1(C(N2CC(NC(C3C(CC(C)C)C3)=O)C(C)C2)=O)ccc(=O)n2c1CCC2 10486,CN(N)C(=O)C(O)CC1CCN(C(=O)OC(C)(C)C)C1 10487,C1(NC(CSCCC)=O)CN(C(=O)C(C)ONC(=O)OC(C)(C)C)CC1(C)C 10488,Cc1cccc(CSC(C)C(N2CCCCC2CN(C(=O)CC(C)CF)C)=O)c1 10489,c1(CNC(NCC2CC(CC)C2)=NCCF)nnc2c(=O)[nH]ccn12 10490,c1(C(N2CCCCC2CF)C(=O)NCCC)ccc(C)c(OCC)n1 10491,CC1CN(C(C2CC23CC(C)(C)C3)=O)CCC1NC(C1CC2(CCOC2)C1)=O 10492,CC1CC=C(C(=O)NCC(C)(C(C)C)NC(=O)CCCN2C(=O)CNC2=O)CC1 10493,c1(NC2C(CC)COC2)nc(=NC2CN(C)CCN(C)C2)[nH]c2c1CCC2 10494,N1(C(c2nc(C)n(C)c2C)=O)CC2CCCC2(NC(C2CCCC(=O)N2)=O)C1 10495,N1(C(Cc2c(C)non2)=O)CC(C(=O)NCCCCCCO)CC12CCC2 10496,c1(OC)ncc(NC(C2(F)CCN(C(c3ccnc(C)c3)=O)CC2)=O)cc1F 10497,C1(CNC(Cc2cnc(C)s2)=O)(NC(c2coc(C)c2)=O)CCCCC1 10498,CC(=NO)C1CC(C(=O)NC(C2CCN(C(=O)CC(C)N(C)C)CC2)C)C1(C)C 10499,c1(CC(N2CCN(C(c3n(C=C)ncc3)=O)CC2)=O)ccc(Br)c(O)c1 10500,N1(C(c2c(C)cc[nH]2)=O)CCC2(CC1)CC2CNC(c1cnc(S)[nH]1)=O 10501,c1(C(=O)NCCc2c(C(NOCC(C(C)(C)C)O)=O)c[nH]n2)cncc(C#N)c1 10502,N1(C(C(c2ccccc2)NC(C)=O)=O)CCOCCC1C(=O)NCc1cnns1 10503,N1(C(C2CCCC(OC)C2)=O)CCCC(NC(c2cc(Cl)cnn2)=O)C1C 10504,C(C)(CN=c1[nH]cncc1C)NC(C(c1ccc(C)cc1)C)=O 10505,c1(C(=O)NCCC(C)NC(c2c(C3CC3)cccc2F)=O)cn2cccnc2n1 10506,C(=O)(C(O)CCS(C)=O)N(CCC)CCNC(c1ncc(F)cc1N)=O 10507,C(C(=O)NCCN(C(C1CCC12CCC2)=O)C(C)C)(C(F)(F)F)OC(C)=O 10508,C#CCC(O)C(=O)N1CC(C(=O)NCCCCn2ccnc2)C(F)C1 10509,N1(S(CCCC)(=O)=O)CCC(C(=O)NCCc2nccs2)(CO)CC1 10510,c1(C(N2CC(C(C(=O)N(C(C)C(C)C)CC)OC)C2)=O)ncc(F)cn1 10511,C1(C(=O)NC2CCCC(CNC(=O)C3=CCCSC3)C2)CCc2ccccc2O1 10512,C1(C(=O)OC)CC(C(=O)NC(C)CCNC(C23COCC(C2)C3)=O)C1(C)C 10513,C1(C(=O)NC2CCN(C(=O)C(C)C(=O)N3CCOCC3)C2)(COCC)CCCCO1 10514,C(c1cccnc1)=C(C(=O)NCC(C)(CO)NC(CC(=O)OC)=O)F 10515,c1(C(N2C(C(C)NC(c3c(C)nc(C)o3)=O)CCC2)=O)ccc(C)c(Cl)c1 10516,N1(C(c2cccc(C(CC)=O)c2)=O)CCN(Cc2cc(F)cc(Cl)c2)C2CC12 10517,N1(C(c2ccc(CC)o2)=O)CCC(O)(CN(C(=O)Cc2ccsc2)C)CC1 10518,C1(C(=O)NC(CCCNC(CCSCC)=O)(C)C)COCCC1(F)F 10519,Cn1cc2cccc(CN3CCN(CC(=O)Nc4cccc(Br)c4O)CC3)c2n1 10520,CN1CCC(N(C(c2cnn(C3CC3(F)F)c2)C(=O)NCC(F)F)C)CC1 10521,CC(C)CC(CNC(=O)CCOC1CC1)NC(c1ccc(Cl)o1)=O 10522,CCC(C)(C)C(O)C(=O)N1CC(C(=O)NCc2nocc2C)C(C2CC2)C1 10523,C1(C)(CNC(COCC(=O)NC)=O)CC(OC)CN1C.c12sccc1NC2=O 10524,c1(OC)ccc(F)cc1C(=O)Nc1ncc(CCSC)s1 10525,N1(Cc2cn(C(COCC)C(=O)NCCc3csc(Br)c3)nn2)CCCNC1=O 10526,N1(C(C2(OC)CCOCC2)=O)CC(=O)NCC1C(=O)NC12CCC(CC1)C2 10527,N1(C(Cc2nc(CC)sc2)=O)CCCC(CO)(Nc2nc(C(C)C)ncc2Br)C1 10528,C1(NC(C2C=CCN(C(c3n(C)c(=O)ccc3)=O)C2)=O)CC2(CCCCC2)C1 10529,c1(C(N2CCN(C(=O)Cc3ccc(O)cn3)C3C2C3)=O)cc(Cl)c(Cl)cc1Cl 10530,C(CC(C)C)(C(=O)N)ONC(=O)C(C(CCO)C(F)(F)F)(C(C)=O)CC 10531,N1(C(c2ccc(C(F)(F)F)c(I)c2)=O)CC2(CCCN2C(=O)NC2CCOCC2)C1 10532,c1(CNC2CCN(C(=O)CCCn3ccnc3)CC2O)c(Cl)cc(F)cc1Cl 10533,N1(C(C=Cc2ccc(OC)cc2)=O)C2CCC1CN(C(c1cnncc1C)=O)C2 10534,N1(C(c2c[nH]c(=N)s2)=O)CCCC2C(NC(c3ccc(C4CCC4)cc3)=O)C12 10535,C=CCCCC(C(=O)N1CC(F)C(F)C1)NC(C1CC2CCC2C1)=O 10536,N1(C(C(F)=C(C)C)=O)CCCC2(CCC(NC(=O)CC3(C4CC4)CC3)C2)C1 10537,N1(CCCCNC(C=C(COC)C)=O)CCCN(C(=O)CC2CCOC2C)CC1 10538,C(=O)(C(C)(CC)CO)NCC12CC(CC(=O)Nc3ccc(CC)nc3)(C1)C2 10539,C1(CC)CN(C(=O)CC2CCCC(C)(C)O2)CCN1C(c1cncc(Cl)c1C)=O 10540,c1(C(N2C(CCNC(C3(N(C)C)CC3)=O)CSCC2)=O)cccc2cnccc12 10541,Cn1cnc2ncnc(NCC3CC4CCC(C3)N4C(c3ccc(CO)o3)=O)c12 10542,Cc1cc(S(C)(=O)=O)cc(C(=O)NC(C)C(C)(C)NC(=O)CC(O)C(C)C)c1C 10543,C1(C(=O)NC2(C)CC(=C)C2)CCCN(C(=O)C(F)(F)C2CC2)C1 10544,C(=O)(CC(C)COCC)N(CC=CC(=O)N(CC#C)CC1CCCO1)C 10545,C1(C(=O)Nc2cc(Cl)cn2C)(OC)CCN(C(c2cc(C)n(C)c2)=O)C1 10546,N1(C(CC)=O)CCOCC(NC(C2C(C)CCN2C(=O)OC(C)(C)C)=O)C1 10547,CN1CCN(C(c2ccc(-c3ncc[nH]3)nc2)=O)C(CNC(=O)C2=CCCCC2)C1 10548,C1(NC(c2ccccc2OC(F)F)=O)CC12CCN(C(=O)Cn1cnnc1)CC2 10549,c1(C(N2CCC(O)(CN(C(=O)C(C)(C)F)C)C2)=O)[nH]cc2c1CCS2(=O)=O 10550,CCCCCC(C)CC(=O)N1C(c2ccc(COC)o2)CN(C)C(=O)C1 10551,CC1CCCC(CC(=O)N(C2(O)CCOC2)C2CC2)C1.N12CC(C1)CCC2=O 10552,c1(C(C(=O)NC(C(=O)OC)C)N(CCCO)CC(C)C)c(Br)nc2n1CCOC2 10553,N1(C(CCCc2scc(C)n2)=O)CC2(CCN(C(c3cccc4sccc34)=O)C2)C1 10554,c1(C(=O)NCC2CCC(NC(C(CCOC)OC)=O)C2)ncc(N)nc1C 10555,C1(C(=O)NC(CNC(c2n(CC)nc(C(C)C)c2)=O)C)Cc2ccc(F)cc2O1 10556,C#CC1(C(=O)N(C)CC2CC2(F)F)CCN(C(=O)CS(=O)(=O)CC)CC1 10557,c1(C(=O)NC2(CCNC(c3coc(C(F)(F)F)n3)=O)CC2)ccc2ncnn2c1 10558,CC1C(C)N(C(=O)C#CCNC(=O)C(C)n2ccnc2)CCN1C 10559,N#Cc1ccccc1OCC(N1CCC(CCNC(c2ccncc2)=O)CC1)=O 10560,N1(C(C=CCCC)=O)CC(NCc2cc(F)cc(I)c2)C(F)(F)C1 10561,CC(C)CC(CNC(C12CC(F)(C1)C2)=O)C(=O)NC(C)CS(C)(=O)=O 10562,Cc1cc(C2(C3CCC(C)C3)CC2)on1.C1([NH2+][O-])CN(C(=O)CN(C2CCC2)C=S)C1 10563,CC1CN(C(=O)CC2(O)CCOCC2)CC(C)N(C(=O)CSc2nncs2)C1 10564,N1(C(Cc2cc(C)on2)=O)CC(NC(c2csc(C3CCCO3)n2)=O)CC1CO 10565,N1(C(C(COCC)C)=O)CCCCC(NC(c2cscc2Cl)=O)C1 10566,n1(CC(=O)NC2(COC)CCN(C(C3OCCN(CC)C3)=O)C2)nc(C)c(Cl)c1C 10567,c1(OC)cc(CCNC(=O)C(C)Oc2ccc(F)cc2)cc(OC)c1O 10568,C1(C(N2C(C(C(N3CCC(=CCC)C3)=O)(C)C)CCC2)=O)CC12CCCCC2 10569,Cc1ccc(S(=O)(=O)CCNC2(C)CCC(O)CC2)cc1 10570,N1(C2(C)CC(C(=O)OC(C)(C)C)C2)CC(NC(=O)OC(C)(C)C)CC(O)C1 10571,c1(C(N2C(CCCNC(C(C)SC(C)C)=O)CCC2)=O)cc2n(c1)CCSC2 10572,Cc1cc(C)c(C(=O)NC(CNC(c2nc(-c3ccco3)sc2C)=O)C2CC2)o1 10573,c1(NC(C)C)nnccc1C(=O)N(CCCCCCNC(=O)C(C)(C)N(C)C)C 10574,c1(C(=O)NCC(CCNC(C2CC2(C)C(F)F)=O)OC)cc2ccncc2[nH]1 10575,C1(C(=O)NCC2(C)N(C(CCCn3ncc(C)c3)=O)CCC2)CC12CC(F)(F)C2 10576,N1(C(CC(C)OC)=O)CC(NC(c2cccc(C3CCC3)c2)=O)C(C)C1 10577,CC(C)(C)C#CC(=O)N1CCN(C(=O)C=C2CCCCC2)C(c2ccncc2)C1 10578,C1(C(=O)NCCCC2CCCN2C(=O)CC2CC3C=CC2O3)NC(=O)C2CC12 10579,Cc1nc(C2CC2)[nH]c1C(N1CCC(NC(C2SCCC2C)=O)CC1)=O 10580,C1(CC(=O)NC2CC(NC(C3N(CCC)CCCC3)=O)C2)CCC(=O)NC1=O 10581,CCCCC(CNC(=O)CC1COCC1O)NC(C1CC(=O)N(C)C1)=O 10582,CC1(C)CCC(C(=O)NCCC2(C)CC2(F)F)CN1C(C1SCCS1)=O 10583,C1(NC(=O)COc2cccc(F)c2)CN(C(C2(CO)CCCO2)=O)CCC1F 10584,Cc1ccc(CCNC(C2(NC(=O)C(C)CCN(C)C)CC2(C)C)=O)cn1 10585,c1(CC(=O)N(c2cccnc2)CC(N2CCCCC2)=O)c[nH]nc1C1CCOCC1 10586,N1(Cc2n(CCC)nnn2)CC(NC(C)(C)CC)C(C(N)=O)C1 10587,C1(C(=O)NC(C2CCN(C(C(C=C=C)C)=O)C2)(C)C)CCC(=O)N(CC2CC2)C1 10588,C(=O)(CCCCC(N)=O)N1CCC(NC(c2n(C)nnc2)=O)CC1C1CC1 10589,c1(CC(=O)NC(C(CO)NC(C(F)=CCC)=O)C)cccc(C)c1 10590,C1(C2CCN(C(C3CCC4(CC4)C3)=O)C2)(NC(c2cn(C)c(=O)cc2)=O)CC1 10591,c1(OC)cc(OC)c(Br)c(C(C(=O)NCCF)N(C)CC2CC2)c1 10592,c1(C(=O)NC2CC(CNC(=O)CC3COCC3O)C2)cc2c(s1)CCCCCC2 10593,c1(C(=O)NC2(CNC(C34CCCC3C4)=O)CCCC2)ccc(Cl)cc1O 10594,C1(C2CN(C(C34COCC3C4)=O)C2)(NC(CCCn2c(C)ncc2)=O)CC1 10595,C(=O)(C(CC)CC(C)C)NCc1cncc(C(=O)NC(CCC(=C)C)C)c1 10596,c1(N2CCCC(C(C)NC(c3cc(SC)nn3C)=O)C2)nn2cc(C)nc2s1 10597,C(=O)(CCN(C(c1cocn1)=O)CC1CC1)NCCN(C)C 10598,C1(NC(CC=CCC)=O)COC2CN(C(C3CCCCC3)=O)CC12 10599,CCCCC(C)C(=O)N1CC(C(C)NC(=O)C(c2cnn(C)c2)O)C1 10600,Cc1ncnc(C(=O)NC(C)(C)CC=CC(N2CCOC(C(C)C)C2)=O)c1C 10601,c1(C(=O)NC(C)CN(C)C(c2cnn(C(F)(F)F)c2)=O)cnn2c1CN(C)CC2 10602,C1(C(N(CCNC(C2CCC23CCC3)=O)CC)=O)CC=CC(O)C1 10603,c1(C(N(C(CC)CNC(C2CCC2)=O)C)=O)oc(-c2cnn(C)c2)nc1C 10604,Cc1nc(C)c(CC(=O)NCC2CCCCN2C(=O)COc2ccon2)c(O)n1 10605,C(=O)(CCC1=NNC(=O)CC1)NC(C)CNC(=O)CC(C(F)F)n1cccn1 10606,N(C(=NCCSC(F)(F)F)NCC1CC(CF)C1)CC1CN(C(C)(C)C)C(=O)C1 10607,c1(C(C(=O)NCCC(=C)CNC(c2ocnc2C)=O)C)ccc(Cl)c(Cl)c1 10608,Cc1ccc(O)c(CNC(=O)CC2CCCN(C(=O)CC#N)C2)c1 10609,c1(C(=O)NC(C)CC(C)NC(c2c(C3CC3)cccc2F)=O)cc(C#N)ccc1Cl 10610,C1(C(=O)NCC2CCC(NC(c3cnc(CC)[nH]3)=O)C2)CCCCN1N=O 10611,c1(-c2nc(CNC(=O)NCCc3ccnc(C)n3)on2)c(Cl)cccc1Cl 10612,CC1CN(C(C2OCC2(C)C)=O)CCN1C(c1cnc(N2CCOCC2)cn1)=O 10613,C1(C(=O)Nc2cnc(OC)c(C)c2)CC2(CCN1C(c1cc(Cl)cs1)=O)CC2 10614,S(=O)(=O)(c1ccc(N(CC(C)O)C2CC2)cc1Br)N(C(CC)C)CC(F)F 10615,N1(C(c2c(CCC)n[nH]c2)=O)C2CCC1CC(N(C)C(C1CC3(CCC3)C1)=O)C2 10616,n1(CC(=O)N(CCNC(=O)C(c2ccc(C)cc2)C)CC)cnc2ccccc12 10617,c1(C(=O)NCC2CCN(C(c3ccc(C)cc3F)=O)C2)ccc(Br)c2cc[nH]c12 10618,Cc1nc2cccc(C(=O)NC3CCC3NC(=O)C(F)C(C)C)c2o1 10619,C(=O)(C(C)S(N)(=O)=O)NCCOCC(=O)Nc1c(CC)n(C)nc1 10620,c1(Cn2cc(C3CCN(C(C4C(C(C)C)C4)=O)C3)nn2)ccc2ccccc2c1 10621,C1(NC(C2CCN(C(C3CC(O)C3)=O)CC2O)=O)CCOC2(CCC2)C1 10622,c12nnn3c1CCCC3C=CC=C1N(C(=O)COCCF)CCN(C1CC)C2=O 10623,c1(C(N2C(CC)CN(C(=O)C(C)OCC3CC3)CC2)=O)cccc2sccc12 10624,c1(C(N2CCC(C(C)NC(=O)CC3(N(C)C)CCC3)C2)=O)cc(Cl)ccn1 10625,N1(C(CCCOCCOC)=O)C(CO)CSCC1CO 10626,c1(C(=O)NCC2N(C(C(C(=C)C)(C)O)=O)CC2)c(OC)cnc2ccccc12 10627,c1(SCC)ccc(C(N2CCCC2CC(C)(C)C)=O)nc1.c1(C=O)cccnc1S 10628,C(=O)(CCCCC(=O)NC(C1CCN(C(=O)CC2CCOC2(C)C)CC1)CO)NC 10629,c1(C(=O)NCC2CCC(NC(C3(OC)CCC3)=O)C2)cccc(C2(SC)CC2)c1 10630,C1(C(=O)NC(CCC)C2CCC2)CCC(C)(C)N(C(=O)C(F)C2CCC2)C1 10631,C12(NC(c3cc(C)c(C)o3)=O)COCCC1CN(C(=O)Cc1[nH]cnc1C)C2 10632,c1(C(N2CCC(Cc3ccccc3Br)C2)=O)ccnc2ncnn12 10633,C=CCC(C)(C)C(=O)N1CCN(C(=O)C(C2CC2)SC)C(C2CC2)C1 10634,N1(C(CSCC)=O)CCC(CC)(NC(=O)CCCCCSC)CC1 10635,CCC(C)(C#N)C(=O)N1CC2(NC(c3cc(-c4ccccc4)c[nH]3)=O)CC1C2 10636,c1(C(=O)NC(C)CC(C)NC(=O)CCCCCO)ccc2c(c1)COC2 10637,Cc1oc(C(=O)NC2C3CC2N(C(=O)CCCN(C)C)C3)cc1S(C)(=O)=O 10638,C1(O)(CNC(CN(CCOC)C)=O)CCN(C(c2ccn(CC(C)C)n2)=O)C1 10639,C1(C(=O)N(C2CC(SC)C2)C2CC2)CCCN1C(=O)Cc1csc(C)n1 10640,N1(C(Cc2c(C)ccs2)=O)CCCC2CN(C(=O)C=Cc3ccccc3)CCC12 10641,C12(NC(C3N(C(C)=O)CCC3)=O)CCN(C(C3(CF)CCC3)=O)CC1C2 10642,c1(C(N(CCCNC(C(OC)OC)=O)C(C)C)=O)cc(C#N)c(N)cc1O 10643,c1(CNC(C2CCCCS2)=O)ccccc1-n1cc(CN2CCCC2=O)nn1 10644,C1(n2cc(C(C)SC3CCCCC3)nn2)CON(C(=O)C(C)C(F)F)C1 10645,C1(C(N(C(C)C)C(C)C)=O)CCN(C(c2ccc(Cl)cc2)C)CC1O.C(=O)C(C)(C)C 10646,c1(C(N(C2CCN(Cc3scnc3Cl)C2)CC)=O)cc(-c2cccnc2)no1 10647,Cc1oc([N+](=O)[O-])cc1C(=O)N(C1CCN(C(C2CC(F)C(=O)N2)=O)C1)CCO 10648,N1(C(=O)C2=CCCCC2)C2CCC1C(F)C(NC(C1CCCN1C(=O)C1CC1)=O)C2 10649,N1(C(CC)C)CC(Cn2cc(Cc3c[nH]c(=O)cn3)nn2)CC1=O 10650,C(=O)(N=c1[nH]c(Cl)ncc1O)C1N(C(C(C)O)=O)CC2(CC2)C1.c1ccccc1 10651,C(=O)(C(O)C(F)F)NCCCN(C(c1ccc(NC(C)=O)s1)=O)CC 10652,c1(OC)cnc(NC(C2CC3C(OCc4cn(-c5ccsc5C)nn4)CC23)=O)cn1 10653,C(=O)NN(C(=O)C1CCCCN1)C(=O)CC(F)(F)F.CCC 10654,CCCCCC(O)C(=O)NCC=CCNC(C1CCN(c2cnn(C)c2)C1=O)=O 10655,c1(C(N(CC(C)NC(C2(F)CCC2)=O)C)=O)cc2ccc(Cl)cc2o1 10656,C1(NC(c2cc(CO)ccn2)=O)CCN(C(C2C(Cl)(Cl)C23CC3)=O)CC1F 10657,c1(CC)nc(NC(C2C(C(=O)Sc3ccncc3)C2)=O)c(NC(C)=O)c(Cl)n1 10658,N1(C(=O)NCc2c(F)cc(Br)cc2F)CCC2CCCC2CC1 10659,Cc1onc(C(=O)NCC2CCCC(NC(C3CC(=O)C3C)=O)C2)c1[N+](=O)[O-] 10660,Cc1ccc(C)c(C(c2nnnn2CCC2CC2)NCCOC2CC2(F)F)n1 10661,CN1CCCC(C)(C(=O)NCC=CCC(=O)NCC2(O)CCCOC2)C1 10662,C(=O)(CCN=C(NCCC(=O)N1CCCC1)NC1CCC(C)C1)NC 10663,OCC(Cc1cccc(F)c1)CN=c1[nH]c2c(F)c(F)c(F)cc2s1 10664,c1(C(=O)NC2CC3CN(C(c4c(C(C)C)ocn4)=O)C2C3)nccn2ccnc12 10665,N1(C(C(Cn2cccn2)NC(CC2(C)CC2)=O)=O)CCCC(F)(F)CC1 10666,N(C(=NCCCCl)NCCN1CCCC1)CC(C1CCOCC1)C 10667,c1(OC)cc([N+](=O)[O-])ccc1C(C)NC(=O)C(=Cc1ccc(Cl)cc1F)C 10668,C(=O)(C(C)(C)CC#N)N1C(CN(C(=O)CCc2cnc(O)[nH]2)C)COCC1 10669,C1(OC)(CNC(=O)CC2CCC2)CCN(C(=O)CC(N2CCCS2(=O)=O)C)C1 10670,CS(=O)c1ccccc1-c1cccc(C(N2CCCC(CC3CC3)C2)=O)c1 10671,c1(OC)ncnc(OC)c1C(N1CCCC(NC(=O)C=C2CCC(C)CC2)C1)=O 10672,C1(NC(N(C)CCc2ccncc2)=O)CCN2CCCCC12 10673,c1(OC)cccc2ccc(C(=O)NCc3cnn(-c4ccccc4)c3Cl)cc12 10674,C=C1CC2(C1)CC(C(=O)NC1CCN(C(=O)C=Cc3cncs3)CC1C)C2 10675,C(=O)(C(C)(C)NC(=O)C(C1CCN(C(=O)COc2cnn(C)c2)C1)C)NC 10676,C1(OC)CCN(CC(O)COc2ccc(C(C)C(=O)OC)c(C)c2)C(C)C1 10677,C1(C(NOCCCC(=O)OC)=O)CN(C)CCN1C(C1CCN1C)=O 10678,C1(O)(CCNC(C(CC)OCC)=O)CCN(C(c2cnccc2Br)=O)C1 10679,c1(C(N2C3CC(CC(NC(c4n(C)ccc4)=O)C3)C2)=O)coc2cc(O)ccc12 10680,c1(C(C(=O)N(CCNC(=O)C(F)(F)Cc2ccccc2)C2CC2)=O)ccc(F)cc1 10681,C(=O)(C1CCCc2ccnn21)N1CC(C2CN(C(CS(C)(=O)=O)=O)C2)C1 10682,Cc1nnc(CCC(N2CCCC(CNC(C3CCCN3C3CC3)=O)C2)=O)n1C 10683,C(=O)(C1=C(F)CN(C(C2CCCC(=O)C2)=O)CC1)N(C)Cc1cscn1 10684,C1(NC(CCN(CCC)C)=O)CC2CC1CN(C(c1ccnn1C1CC1)=O)C2 10685,C(=O)(CCCC(C)(C)C)NCC(CC=C)NC(=O)C=CCCC=C(C)C 10686,C#Cc1cn(C)nc1C(=O)NC1CCC(CC(N2CCCC2C2CCOC2)=O)C1 10687,CC1(F)CCCCN(C(c2ccc([N+](=O)[O-])s2)C(=O)Nc2ccccc2Cl)C1 10688,C#CCCCCC(=O)NCC1(CNC(c2ccncc2C)=O)CC1(F)F 10689,c1(C(C)NC(c2n(CC=C)nnn2)c2cc(C3CC3)[nH]n2)cc(F)cc(F)c1 10690,N1(C(CCn2c(C)cc(C)n2)=O)CCCC2(C1)CN(C(C1CCCC(O)C1)=O)C2 10691,c1(N(CC(=O)NC2CC(NC(=O)C(F)(F)F)C2)C)ccnc(Cl)n1.C(=O)(NC1CC1)CC 10692,Cc1cnn(CCCNC(=O)C=CCNC(=O)CCCC2CC2C)c1 10693,CCC(C)CC(=O)N(C1CC1)Cc1ccc(C(F)C(F)(F)F)cc1 10694,C(=O)(C(O)CCC(F)(F)F)N1CC(CC)N(C(c2nc(C3CC3)cs2)=O)CC1 10695,CCC(CC)(C(=O)OC(C)(C)C)C(=O)NCC(O)CNC(C1C(OC)C1(C)C)=O 10696,C1(C)(COC)CC(NC(=O)CC2CC2)CN1C(=O)Cn1cnc([N+](=O)[O-])n1 10697,CC1OC2(CO)CC1(C(=O)NC(C)CN(C)C(c1cc(C3CCCC3)no1)=O)C2 10698,C(CCN=c1[nH]c(=NCCC(C)S(C)=O)[nH]c2c1CCCCCC2)N(C(C)=O)C 10699,CCCC(CC)C(=O)N1CC(OC)CC(NC(=O)CSc2cccc(C)c2)C1 10700,c1(C(=O)OCc2cn(C)c(=O)cc2)ccc2ccnc(Cl)c2n1 10701,c1(C(=O)NCCc2cc(C(=O)NC3COCC3C(N)=O)no2)n[nH]c2c1COC2 10702,N1(C(C(C(C)C)F)=O)CCCN(C(=O)COC(C)(C)C)C(c2ccccc2)C1 10703,C(CC(C)C)(C(=O)N1CC2CC(C1)C2NC(c1snnc1C)=O)NC(C)=O 10704,CCC(O)C(C)C(=O)N(CCCNC(=O)CN1CCCC(N(C)C)C1)CC1CC1 10705,C(=O)(C1=COCCO1)N1C(CN(C(c2c(Cl)c(C)nn2C)=O)CC)CCCC1 10706,C1(CN(C(CCC=C)=O)C)CCN(C(=O)C(c2ccc(F)cc2)CO)CC1 10707,N1(C(C2(NC(=O)C(F)C3CCCC3)C(C)(C)C2)=O)C2CCC1COC2 10708,N1(C(c2c(C(C)(C)C)ocn2)=O)CC2CC(NC(c3cscn3)=O)C(C2)C1 10709,C12(C(N3CC(C)(C)SCC3)=O)CCC(CC1)N(C(=O)COc1ccccc1)C2 10710,Cc1ccc(C(=O)NC2CN(CCn3ccc(C(=O)NN(C)C)n3)CC2C)cc1F 10711,C1(CC(=O)OC(C)(C)C)(NC2CC3CC3C2)CCOCC1 10712,N1(C(C(C)NC(CC)=O)=O)CC2COCC(C1)C2NC(c1ccc(F)cc1)=O 10713,C1(C(F)F)CC(=O)N1.C(C)(C)(CO)O.CCC(=O)N(CCCO)CC1CC1 10714,c1(SCC(N2CCC(CN(C(CC(=C=C)C)=O)C)C2)=O)nc2ccccc2[nH]1 10715,C1(n2cc(CC(C(=O)NCC(COC)C(=O)OC)(C)C)nn2)CCc2nn[nH]c2C1 10716,C1(C(=O)NCCNC(Cc2c(C)occ2)=O)CCCC1P(C)(C)=O 10717,c1(NCCC(C(C)C)NC(C2C(CCC)CCC2)=O)ncnc(Cl)c1OC 10718,C1(NC(C=C(CC)C)=O)CC2CCC1C1CN(C(=O)C(=CC3CCCC3)C)CC21 10719,N1(C(C2N(C(c3nn(C)c(Cl)c3)=O)CCC(C)(C)C2)=O)CCCC(O)(C2CC2)C1 10720,C(c1ccc(C)cc1C)=CC(=O)Nc1c(C(=O)OC)cccc1 10721,N1(C(c2c(C#C)c[nH]n2)=O)CCCN(C(=O)C(O)CC(N)=O)C(C)C1 10722,c1(C(N2CCC(C)C2CNC(c2nnsc2CN)=O)=O)ccc(OC(F)F)cc1F 10723,C#Cc1ccc(C(N2CCN(C3CN(C(C4CC4c4cccs4)=O)C3)CC2)=O)cn1 10724,Cc1cc(=O)n(CCC(N2CCCC(CNC(=O)CC=C(Cl)Cl)C2)=O)cn1 10725,C1(NC(C2CC(CCC)C2)=O)CC(O)CN(C(c2ccc(SC)cc2)=O)C1 10726,N1(C(CN(C)CC)=O)C2CC=C(C(=O)Nc3cc(C)nnc3C)C1CC2 10727,c1(C(C(=O)N(C2CCCC2)CCCNC(CCC#CC)=O)C)c(F)cccc1F 10728,C(C(CC(C)C)C(=O)NC1(C(=O)NCC2COCCN2C2CCCC2)CC1)OC 10729,S(=O)(=O)(c1ccc(N2CCCC(C)(CO)C2)c(Cl)c1)NCCCC=C(C)C 10730,C1(CC)COCCN(C(=O)C(=O)N(CCCO)CCn2cc(CO)nn2)C1 10731,c1(C(N2CC(NC(C3(SC)CC3)=O)C(F)C2)=O)ccc2nc(O)[nH]c2n1 10732,C(CCN=c1[nH]c2c(c(=NCCN3CCOCC3C)[nH]1)COC2)OCC(C)C 10733,c1(CC)noc(C)c1C(=O)NC1(C2CCCCN2C(=O)Cc2c[nH]ccc2=N)CC1 10734,Cc1nc(N2CC3CN(C(c4cccc(F)c4N(C)C)=O)C3C2)c2c(n1)CCC2 10735,N1(C(CCCOCC=C)=O)CCN(C(=O)C(O)CC)C(CC(=O)NCC)C1 10736,C1(N(C)C(c2cccc(Cl)n2)=O)CN(C(=O)CC(F)(F)Cl)CC12CC2 10737,N1(C(C=C(CCC)C)=O)CCCC(C)(C(=O)NCCSc2cc(O)ccc2C)C1 10738,c1(CN=C(NCC23CC(CF)(OC2)C3)NC2CCC2)ncc2ccccn12 10739,C1(CC(=O)N(C2CN(C(c3ncc(Br)cc3O)=O)C2)C)CCCC2(CCC2)O1 10740,CCCCC(O)C(=O)NC1CCN(CCO)CC1.c12cn(nn1)CCOC2 10741,N1(C(C(C)(C)NC(=O)NCC)=O)CCCC(N(C(=O)C(O)CF)CC)CC1.CC 10742,c1(SC)c(C(=O)NCCC(C)NC(c2ccc(C)[nH]2)=O)cccc1F 10743,c1(C(N(C(CCNC(CC(CC)OC)=O)C)C)=O)ncnc2cc[nH]c12 10744,S(=O)(=O)(c1ccc(C(=O)NC2CCCC2NC(=O)CO)cc1)NC(COC)C 10745,Cc1cnc(C(N2CCC(C)(NC(=O)CCSc3ccccc3F)C2)=O)c(C)c1 10746,CC1=NNC(=O)C1CCC(=O)NC(CNC(=O)C(C)Cc1ccco1)CC(C)C 10747,c1(C(=O)NCc2cc(C(=O)OC)[nH]c2)cccc2ncccc12.c12n[nH]cc1N2 10748,c1(C(=O)OCC)ccc(NC(=O)NCC(CCSC2CCCO2)OCC)cc1F 10749,c1(C(C)OCC)noc(CCC(=O)NC(C)(C)CNC(=O)CC23CC(C2)C3)n1 10750,C=CCN=C(NCCC1CCN(C(=O)OC)C1)N1CCCC2(CCSC2)C1 10751,C=CC(C)(C)CC(=O)NCCOC1CCN(C(=O)CCS(C)=O)C1 10752,C1(C(=O)NCC(C)N(C(C(=O)NCCC)=O)C)CCS(=O)(=O)C1(C)C 10753,c1(C(=O)NCCC(C)N(C(CN2C(C)CC2)=O)C)nn(C)cc1N 10754,C1(CC)CCN(C(=O)CC(C)(C)O)C1C(=O)N(C)CCOC(F)F 10755,C1(CC(=O)NCCCCN(C(=O)CCN2CCOC2=O)C)CC(F)CN1 10756,c1(C(C(=O)N)N(c2ccc(OC)cc2)C)cc2c(s1)CCOC2.CCCOC 10757,C1(OC)CN(C(=NCC2CCCCO2)NCc2c(F)ccc(C)c2F)CCO1 10758,Cc1c(C(F)(F)F)n[nH]c1C(N1CC(CNC(c2cccc(N)n2)=O)CC1C)=O 10759,c1(CC(=O)NCC2(OC)CN(C(=O)CC3CCC(O)C3)C2)nc(F)ccc1Cl 10760,FC(F)C(F)(F)CCN=c1[nH]c(N2CC=C(Br)CC2)nc(Cl)c1F 10761,c1(C(=O)NC(CNC(C(COC)(C)C)=O)(C)CO)ccc(Cl)c(C#N)c1 10762,C1(CNC(=O)CCCn2cccn2)CC2(CC2)CN1C(=O)CN1CCCC1C(=O)O 10763,C1(C(C)C)C(NC(c2cnn[nH]2)=O)CCN1C(c1cnc(CN(C)C)s1)=O 10764,C(=O)(C1=CCCC1C)N1C(CO)CC(NC(c2n(CC)c(O)nc2)=O)C1 10765,C1(C(N2CC(C(C)NC(=O)CCSc3cccc(Cl)c3)C2)=O)CCCC2(CC2)C1 10766,C(=O)(CC(C)CC(C)(C)C)N1C(CN(c2ncc(C(=O)OC)[nH]2)C(C)=O)CCC1 10767,c1(C(C(=O)N(CCCCCNC(C(CC)C)=O)C)(C)C)c(F)cccc1F 10768,c1(N2CC3(C(C(=O)Nc4c(C)ccc(I)c4)C3)C2)ncnc2c(C)csc12 10769,S(=O)(=O)(c1ccc(Cl)cc1)COC(C(=O)NCCC(C)NC(=O)CC1(O)CC1)C 10770,C(=O)(CCN(OC)C(=O)c1coc2c1CN(C(C1OC3CCC1C3)=O)C2)OC 10771,c1(CCC)nc(C(N2CCOC3CC23)=O)nn1-c1cccc(Cl)c1 10772,c1(CC(=O)NCC(C)CNC(C2C(C)C2C)=O)csc(C(C)(C)C)n1 10773,C1(C(=O)NCCCC#C)CC(NC(c2cn(C)nc2OC)=O)CCO1 10774,c1(C(N2CCCC(C)(C(=O)NC3CNC(=O)C3)C2)=O)ccc(F)c2ccoc12 10775,Cc1cccc(OCC(=O)NCCCN(C(=O)CC(C)C2CC2)C2CC2)c1C 10776,c1(OC)c(Cl)ccc(C(=O)NCCC2CCC(NC(=O)C(O)CN(C)C)C2)c1F 10777,c1(C(N(CC(C)NC(=O)Cc2cnoc2)C)=O)cc(F)cc2nn[nH]c12 10778,c1(C(=O)NCCC(C)NC(=O)C(F)(F)c2csc(Cl)c2)cn(C)nc1Cl 10779,Cc1c(C(=O)NCC2(O)CN(C(=O)C(F)C3CCC3)C2)cnn1C1CCCCC1 10780,C1(C)(C(N(C2CC(NC(=O)C(O)Cn3cncn3)C2)C)=O)CCCO1 10781,CC(C)(C)C(=O)N1CCCC1C(=O)N(CCC=CBr)CC1CC1 10782,C(CC(C(=O)NCc1cc(C)c(C)s1)NC(C1CC(F)C1)=O)=CC 10783,N1(C(C2NCC(OC)C2)=O)CCC(C2(O)COC2)CC1 10784,C1(n2ncc(C)c2)CN(C(C2CCNCC2)=O)CCN1.c12nn(C)cc1C(=O)N2 10785,C1(CNC(C=CCOC)=O)CC(C)(C)CN1C(=O)CC1(O)CCCOC1 10786,C1(C(C)C)CN(C(C2CC2(C)C(F)F)=O)CC1C(=O)N(C)Cc1cnn[nH]1 10787,N1(C(c2csc(Br)n2)C(=O)NCC=C)CCC(CO)(COC)C1 10788,C1(NC(CC=CCC)=O)CC(O)CN(C(=O)C(=O)Nc2ccccc2)C1 10789,N(C1CCSc2ccc(Br)cc21)C(=O)NC1C(OCC)COC1 10790,c1(CC)ccc(C(=O)NCC2(CC)CC2)c(O)c1.C12CCC(CC)(CC1)NC2=O 10791,CCCCC(C)CCC(=O)NCC(CC)N(C)C(C1CC(F)(F)C1)=O 10792,c1(C(N2CCC(O)(C(=O)NC3CCNCC3)CC2)=O)cc([N+](=O)[O-])sn1 10793,CC1CC2(CC(C(=O)N(C(C)(C)CC(=O)N3CC(c4ncccn4)C3)C)C2)C1 10794,CC1CCN(C(c2cc(Cl)cs2)=O)CCN1C(=O)CC1OCCCC1(C)C 10795,C1(CNC(CN(CC)CC)=O)CN(C)CCN1c1ncnc(Cl)c1Br 10796,CC(C)(CCCNC(=O)C(F)=CC1CC1)C(=O)NCCC1CC=CCC1 10797,Cc1ccc(C2(C(=O)NCC34CC3CN(C(=O)Cn3ccnc3)C4)CC2)cc1 10798,N#Cc1ccc(C(O)C(N2CCN(C(=O)Nc3cccc(Cl)c3Cl)CC2)=O)cc1 10799,C1(NC(C=CS(CC)(=O)=O)=O)CCC2CCN(C(C3CC3(Cl)Cl)=O)C1C2 10800,C1(N(C(COCCCSC)=O)C)CCN(C(=O)Cc2cc(C)sc2C)CC1 10801,C1(C(=O)OC)CC(C)(C)CCN1C(c1cccc(C)n1)C(=O)NC1CCC1 10802,Nc1c(C(N2CCC2CNC(C2CC(NS(C)(=O)=O)C2)=O)=O)cc(F)cc1Cl 10803,c1(CC(C(=O)NCOC(CNC(C(N2CCSCC2)C)=O)(C)C)O)ccc(F)cc1 10804,c1(NC(=O)Cc2cc(F)cc(Br)c2)ccc(OCC(F)F)cc1F 10805,c1(OC)cc(C)cc(C(=O)NCC=CCNC(c2cnc(C)nc2CO)=O)c1N 10806,C(=O)(C(C)(C)C(F)(F)F)NC1CN(C(c2nc(CCC)oc2)=O)C(C)C1 10807,Cc1cc(C(=O)NC(C)(CNC(C2CC2C(N)=O)=O)C(C)C)cc(C)c1C 10808,Cc1cc(C(=O)NC(C2(CCS(C)(=O)=O)CC2)C)n(C(F)F)n1.C12(O)CN(C1)C2 10809,N1(C(C(CC)=CC)=O)CCC(C)C(NC(c2cc(Cl)cc(Cl)n2)=O)C1 10810,C1(Cn2cnnn2)CC(C)(C)CN1C(C1(n2cc(SCC)nn2)CC1)=O 10811,C1(N(C(CCCOCC)=O)C)CCCCC1NC(C1(C(F)(F)F)CC(F)(F)C1)=O 10812,C(=O)(C(=O)N=S(C)(C)=O)NC(C1CC2CCC(C1)N2C(=O)CN=S(C)(C)=O)C 10813,C1(N(C)C(c2ncoc2C(C)(C)C)=O)CCCC(NC(=O)C=Cc2cncn2C)C1 10814,c1(C(=O)NC2CCN(C(c3csc(C(F)(F)F)c3)=O)C2)nncc2c1CCCC2 10815,C1(NC(Cn2c(C)cc(C)n2)=O)CC2CC1CN(C(c1cnsn1)=O)C2 10816,C1(C(=O)OC)CCC2(CCC2)N(C(=O)CCC2CCOC2=O)C1 10817,C1(OC)CCC2(CCN(C(C3CCC(C)N3C(=O)OC(C)(C)C)=O)C2)C1 10818,C1(C(=O)NCC(C)C)CC(C)CN(C(C2CC2c2ccccc2)=O)C1 10819,c1(CC)nc(N2CC(NC(C3(C(F)(F)F)CCC3)=O)CC2C)c2ccsc2n1 10820,C(=O)(CS(=O)C(F)(F)F)N1CCC(CNC(CCOC)=O)C1(C)C 10821,Cc1cc(OCC(=O)NC2CC(CNC(C3CCOC(=O)CC3)=O)C2)ccc1Cl 10822,C(=O)(CCC[N+](=O)[O-])NC(CCN(C(c1c(C)noc1C)=O)C)C(C)C 10823,C1(CC)CC2CC1CN(C(c1cc(C(N)=O)c[nH]1)=O)C2.N1(CC(=O)N)CCCC1CO 10824,Cc1nn(C)c2c(NC3CCCCC3C)nc(=NCC3(C)NC(=O)NC3=O)[nH]c12 10825,C(N=c1[nH]c(N(C)CC2(C3CC3)CC2)nc2ccccc12)c1[nH]c2ncn(C)c2c1 10826,c1(NC(C(CN(C(C(CC)(C)CO)=O)C)C)=O)ccc2c(c1)CCO2 10827,C1CC2(CCN(C(=O)COCC(=O)NC3CC3)C2)C1.C(C(F)(F)F)OCCOC 10828,C1(n2cc(CNC(C(C)=C(C)C)=O)nn2)CCN(C(=O)CCc2cccs2)CC1 10829,C1(NC(=O)Cc2ccc(O)cn2)CCCCCCC1NC(=O)CCc1ncc[nH]1 10830,c1(CC(=O)NC2CCN(C(C(C(C)C)F)=O)C2)cccc2c1OCCO2 10831,N1(C(=O)OC(C)(C)C)CCC(C2OCCC2OC(C2CC2(C)C)=O)CC1 10832,N1(C(C(c2c(C)n[nH]c2C)C)=O)CCCN(C(c2cnns2)=O)C(C)C1 10833,C1(CC#C)(C(N2CC(C(F)(F)F)C(CNC(=O)CN(C)C(C)=O)C2)=O)CC=CCC1 10834,c1(OC)cc(CC(=O)N(CCCCCNC(C2(CF)CC(=O)C2)=O)C)on1 10835,Cc1ccsc1C=CC(N1CCC(OCCNC(=O)CCC2CCCN2C)C1)=O 10836,C12(C(N3CCC(C)(CCNC(c4ccccc4)=O)C3)=O)CC(C)(CCO1)C2 10837,CCC(C)CCC(O)CC(=O)NCCNC(=O)Cc1ccc(C)nc1 10838,C1(C)(CNC(C(=O)NC(C)C)=O)CCC(NC(=O)C(c2ccccc2)=O)C1 10839,c1(CC(N2CC(NC(Cc3cc(C(C)C)no3)=O)C(O)C2)=O)cc(Cl)ccc1O 10840,C1(C(C)(C)NC(C(C)OCCOC)=O)CCN(C(C2(C(F)F)CC2)=O)C1 10841,Cc1cccc(CN(CCCNC(c2ccc(C3CC(=O)C3)cc2)=O)C)c1 10842,Cn1c(=O)c2c(ncn2CC(=O)OCC(O)CCS(C)(=O)=O)n(C)c1=O 10843,N1(C(C(C(C)C)F)=O)CC2CCCC(Nc3ncccc3CCCCCF)C2C1 10844,CC(C)CCC(F)C(=O)NCC(C(C)C(C)C)NC(C1(N(C)C)CC1)=O 10845,c1(CC2CCN(N(C(C3CCCN(C(C)C)C3)=O)C)CC2)cnc(Cl)c(Cl)c1 10846,CCC(F)(F)CC(=O)N1C2CCC1C(CNC(=O)CN1C(=O)NC(C)(C)C1=O)C2 10847,C1(C(N2CCC(CNC(CC=C=C)=O)(OC)C2)=O)CCc2nccn2CC1 10848,c1(C(N(C2CCN(C(=O)Cc3ccn(C)n3)C2)C)=O)ccc(F)c(F)c1O 10849,c1(CNC(=O)NC2CC(NC(C(c3cnccn3)C)=O)C2)ccccn1 10850,C1(O)(CCCO)CCOCC1.N1(C(C)C=O)CC(C)(C(N)=O)C1 10851,c12ncccc1CC(=O)N1CCC1C(=O)N2C1CC1.C1(COC)CC(C(N)=O)C1 10852,Cc1ccc(CNC(C2(F)CCN(C(C3CC(N(C)C)C3)=O)CC2)=O)c(O)n1 10853,c1(C(=O)NCCCN(CCO)C(C2CCCSC2)=O)ccc2nn[nH]c2n1 10854,N1(C(C(COC)C)=O)CCC(C)(C)CC1NC(c1cncc(C#N)c1)=O 10855,C(c1ccccc1Cl)=C(C)C(=O)NC1CC(C)N(C(=O)C(n2cc(Cl)cn2)C)C1 10856,c1(CNC(C2C=CC(NC(C3(C(C)(F)F)CC3)=O)C2)=O)cc(F)cc(Cl)c1 10857,S(=O)(=O)(c1cccc(F)c1)N1C(C(=O)NC2C(SC)CCC2)CCC1 10858,C1(C)(CC)CC(NC(=O)NCC2(CC(=O)OC)CCOCC2)CCO1 10859,C1(NC(COCc2nnc(C)s2)=O)CCN(C(C2CC23CC(O)C3)=O)CC1 10860,c1(-c2cc(CC)no2)cnc(N(C)Cc2cc(OC)ccc2OC)c(Cl)c1 10861,CCC(C)C(CC(=O)N(C1CCC1C)C1CC1)NC(=O)C(C)(C)C1CCOC1 10862,C(=O)(CCCCC(=O)N1CC(CNC(=O)CN2CCCCC2)CC1C)OC 10863,c1(C(=O)NCC(CCC)NC(=O)CCN(C)CC)c(C)coc1CC 10864,c1(CNC(=O)NCC(=O)NCc2cncs2)ccc(F)cc1Br 10865,CC(C)C(C(=O)NCCC(C)NC(C1CCC(=O)C1)=O)NC=O 10866,N(C1COc2ccc(Cl)cc21)C(Cc1nc(CN2C(COC)COCC2)on1)=O 10867,c1(N(CCOC)C)nc(C)nc2sccc12.c12ccc(o1)C(=O)NC2 10868,c1(C(N2C(CC)CN(C(c3cc(Cl)n(C)n3)=O)CC2)=O)cccc2ccncc12 10869,c1(CN(C(=O)NC(c2nc(CO)n[nH]2)C)C)cccc(I)c1 10870,CC1(C)C(CNC(=O)CC2COC3CC2C3)CCN1C(=O)C=Cc1ccsc1 10871,N1(C(c2cn(C)nn2)=O)CCCC(CCNC(=O)CCC2CC2)CC1 10872,c1(OC)ccc(C(N2CCC(O)C2)C(=O)NCCC2CC2)cc1SC 10873,C12(CNC(c3n(CC)nnc3)=O)CC1CN(C(=O)Cn1cc(C#N)cn1)C2 10874,c1(C(=O)Nc2cc(F)c(F)cc2I)cc(Br)cc2[nH]ccc12.O=C1CCN1 10875,Cc1nc2ccc(CNC(=O)CCN3CC(C(N)=O)C(c4ccnn4C)C3)cc2o1 10876,CCC(C)(CNC(=O)CCC1CCCN1C)C(=O)N1CC(OC(F)F)C1 10877,C1(CC)(CC)CC(NC(c2cncc(CO)c2)=O)CN1C(C1CC=CC1)=O 10878,C1(C(C)(C)C)(CNC(c2nnsc2N)=O)CCN(C(C2CC(F)C2)=O)C1 10879,c1(C(C)(C)C)ncc(C(=O)NCC2CCCC2NC(c2cc(C3CC3)on2)=O)o1 10880,N1(C(Cn2c(C)nnn2)=O)CCCC(NC(=O)C(C)(C)c2ccn(C)n2)C(F)C1 10881,N1(C(C(C)C2CCCC2)=O)CCC2CCC(C1)N2C(c1cc(=O)cc[nH]1)=O 10882,c1(C(=O)NC2C(CNC(c3[nH]c(=N)sc3)=O)CCC2)cnn2cccc(Cl)c12 10883,N1(C(C(C)N(C(C)=O)C)=O)CCC(C(=O)NCCCC(C)(C)O)C12CCC2 10884,N1(C(CC(C=C)C)=O)CC(C)N(C(=O)CCc2cn[nH]c2)CC1C 10885,N1(C(CC2CCCC(C)(C)O2)=O)CCC2(CNC(=O)CC3CSC3)CCCCC12 10886,c1(OC)ccc(CC(=O)NC(C)CN(C)C(c2ocnc2C)=O)cc1 10887,C1(NC(CN(C(=O)OC)C)=O)C(C)CN(C(c2nccn2C(C)C)=O)CC1C 10888,CCCCC(F)C(=O)NC1CCCCC1C(N1CCC(CC(N)=O)C1)=O 10889,c1(CC(=O)NC2CC3(C2)CN(C(C2CC2F)=O)C3)noc2ccc(Br)cc12 10890,c12ccnn1S2.C(C(=O)NCC(=O)N(CC(C)C)C1CC1)OCCOCC 10891,Cc1cc(C(=O)NC2CC3CN(C(=O)C(F)(F)CO)CC23)cc2nn[nH]c12 10892,CCCC(C(=O)N(C(C)CC(=O)Nc1nnn(C)c1C)C1CC1)NC(N)=O 10893,CN(C)S(=O)(=O)N1CCCC1C(=O)NCC1(F)CC(NC(=O)CC(C)(C)C#N)C1 10894,C(=O)(C(O)C1=CCCCC1)N1C(CNC(c2c(C)cnn2C(C)C)=O)CCC1 10895,c1(C(=O)NCC2C(NC(c3cccc(O)n3)=O)C2)cc(Br)ccc1[N+](=O)[O-] 10896,c1(NC)ccc(C(=O)NC(C2(O)CCN(C(=O)CCc3cnc[nH]3)C2)C)c(Cl)c1 10897,c1(C(=O)NCC(C(C(C)C)C)NC(=O)CC2(C)CC2)cc2ccc(O)cc2[nH]1 10898,C1(CCNC(C2CN(C)C(=O)C2)=O)CN(C(c2cccc(Cl)c2F)=O)CCCO1 10899,c1(C(N(C)CC2CCN(C(C(C3CCCCC3)C)=O)C2)=O)cccc(=O)n1C 10900,n1(CCC)c(C(N2CCC(CF)(NC(=O)C3=CCOC3)C2)=O)cc2ccccc12 10901,C1(=O)CCCn2cc(nn2)NCC(O)CN1.C#CCOCCC 10902,C1(C(OCCOC)NC(C=O)=O)CCN(C(=O)C(O)Cc2ccc(Cl)cc2)CC1 10903,C(=O)(CC=CC=C)N(CC(=O)N(CC#C)CC1CC1)C1CC1 10904,c1(C(N2C(C3(O)CN(C(c4ccn(CCC)n4)=O)C3)CCC2)=O)ccc(=N)[nH]n1 10905,C(N=c1[nH]c(=NCc2cnn[nH]2)[nH]c2c1CC(C)CC2)C1CN(C)C(=O)C1 10906,C1(c2c(C(=O)NCc3cnc[nH]3)c[nH]n2)CCCCN1C(=O)CC1(O)CCCCC1 10907,N1(C(CCOCC#C)=O)CC2CCC1CN2C(C1CCCC(C)CC1)=O 10908,S(=O)(=O)(c1ccc(NCC(=O)Nc2cccc(Cl)c2)cc1Cl)NC(CCSCC)C 10909,C(=O)(CCCCC(N)=O)NC(c1ccc(OC)cc1)CNC(C1(CO)CCC1)=O 10910,C(=O)(CCCC(C)(F)F)N1CC(NC(C(=Cc2ccncc2)C)=O)C(C)(C)C1 10911,c1(C(=O)NCCC(C)NC(=O)CCC2CCC2)c[nH]c2cccc(Br)c12 10912,c1(C(=O)NC(C)CCNC(=O)C(C)(C)C2CC2)c(F)c(F)c(F)c(F)c1F 10913,C(=O)(CP(C)(C)=O)N1C(C(C)(C)NC(Cc2n(C)ncc2)=O)CCC1 10914,c1(C(=O)NCCC(C)NC(c2cn(C)nc2O)=O)nnc(Cl)cc1N 10915,c1(C(=O)Nc2cccc(C)c2O)cc2c(s1)CCN(C(c1ccnc(F)c1)=O)C2 10916,N1(C(C2(COC)CC(=C)C2)=O)CC=C(C(=O)N2CCC(CC)C2)C1 10917,c1(C(=O)NCc2nc(C)[nH]n2)c(NC(=O)Cc2ccccc2C)cccc1F 10918,C1(NC(C(CCCC)O)=O)Cc2ccccc2C1NC(C1(CC)CC1)=O 10919,C1(O)(CN(C(C(C)=CCNC(=O)OC(C)(C)C)=O)C)CCCN(C(C)=O)C1 10920,C1(CC(=O)NCC(CC)NC(C2CCC(C)CC2)=O)OCCCC1(C)C 10921,N1(C(C(C)OCC)=O)CCC2(CC1)COC(CNC(C1(CC)CC=CCC1)=O)C2 10922,c1(C2OCCN(CC3N(C)CC(C(=O)O)C3)C2)ccc(F)c(F)c1 10923,N1(C(C(CO)NC(C2OCCC(C)(C)C2)=O)=O)CCC2(COC(=O)N2)C1 10924,c1(CN2CC(NC(c3cccc(O)c3O)=O)C(O)CC2)cccc2nsnc12 10925,C(=O)(C1Cc2ccccc21)NC(CCC=C)C(=O)NC1CCC2(CC2)C1 10926,Cc1ccc(SCCCC(=O)NC2C=CCN(C(C3CCC(=O)NC3)=O)C2)cc1 10927,N1(C(C2(C(=O)NC)CC2)=O)CCc2sccc2C(CNC(=O)C(C)(C)C2CC2)C1 10928,c1(CC)nc(C)c(C(=O)N(CCC(C(C)C)NC(c2n[nH]cc2COC)=O)C)s1 10929,C1(NC(c2cnc(CC)[nH]2)=O)C2CCC1N(C(=O)Cn1ccc(Br)cc1=O)C2 10930,c1(NC)c(F)cc(C(=O)NC(C2CN(Cc3nn(C)cc3Br)CCO2)C)cc1F 10931,n1(CC)cc(C2CCC(NC(=O)N(C3(C)CC3)CCO)C2)cn1 10932,C1(C(N2CC(CCCCNC(C3CCCC(C)(C)O3)=O)C2)=O)CCC2(CCC2)OC1 10933,c1(C(=O)NC(CC)CNC(=O)CSCc2ccoc2C)nccc(OC)c1O 10934,S(=O)(=O)(c1ccc(OCCC)c(N)c1)NCCC(=O)NCC.C(C(=O)OC)OCC 10935,N1(C(C(C)NC(=O)NCC2C(C)C2)=O)CCC(C(=O)NCC2CC2Cl)C1 10936,c1(C(=O)NC(CCNC(CCNC(=O)OC)=O)C(C)C)ccc(F)c(C(C)C)c1 10937,O=C(C#CC1CCCO1)N1CC2(CCN(C(C3(C(F)(F)F)CC=CCO3)=O)C2)C1 10938,Cc1noc(C)c1S(=O)(=O)NCC1CCN(C(c2ccc(Cl)s2)=O)CC1 10939,c1(OC)cc2c(cc1C(=O)N(CCNC(=O)C(c1cccn1C)=O)C1CC1)OCO2 10940,c1(C(=O)OCCCCCN(C(CC)CC)Cc2ccccc2)c[nH]nc1C1CC1 10941,c1(CC(N2CC3N(C(C(CC)=O)=O)C3C2)=O)c(F)ccc(Cl)c1F 10942,C#CC1CN(C(=O)C(CNC(=O)CCC2CCC(=O)C2)CC(C)C)CCN1C 10943,C(c1ccccc1Cl)=C(C)C(=O)N(C)CCN(C(=O)CCCC(F)F)C(C)C 10944,c1(C(CC(N2CC(CNC(CN(C)CC)=O)OCC2)=O)C)ccc(C)c(OC)c1 10945,C(C)(C)(CCC(=O)NC1CC2CC1CC2(C)O)NC(CC1COCC(C)O1)=O 10946,c1(C(N2C3C(NC(c4occ5c4CCC5)=O)CC(C3)C2)=O)cccc2occc12 10947,C(=O)(CCCCCN=[N+]=[N-])n1cc(C(C(=O)NCC)N(CCSC)CCOCC)nn1 10948,C1(CNC(=O)CC2CC(NC(=O)Cn3ccnn3)C2)CNC(=O)CO1 10949,c1(C(N2CC(C)C(CNC(=O)CC3CC4(CC4)C3)C2)=O)ccc(Cl)c(Br)c1 10950,C1(C(=O)NCCOCCNC(c2cnc(CC)s2)=O)C(C2CC2)C1(F)F 10951,c1(C(=O)NC(C(C)NC(C=CCC)=O)C(C)C)c(C)nc(C(C)(C)C)nc1S 10952,N1(C(CC=CCCCCC)=O)CCC2CCC(C1)N2C(=O)CSCCC 10953,C1(O)(CCC)CCN(C(C2CCCN(C(C3OCCCC3(C)C)=O)CC2)=O)CC1 10954,Cc1ncc(C(=O)NCC23CC2CN(C(=O)Cc2ccc(Cl)nn2)C3)c(O)n1 10955,Cc1nnc2n1CCC(C(=O)NCCN(CCCN(C)C)C(c1cocn1)=O)C2 10956,N1(C(c2ccc(CC)[nH]2)=O)CC(COC)CC1CNC(=O)CNC=O 10957,C(=O)(C(C)C(C)(C)C)NC(C1CCCC1)CNC(c1c(CC)nn(C)c1)=O 10958,N1(C(c2cn(CCN(C)C)nc2)=O)CCC2(CC1)CC2NC(c1cscc1F)=O 10959,c1(C(=O)NCC2CC2CNC(c2cnc[nH]2)=O)cccc(Cl)c1 10960,C(C)(C(=O)NCC1C2CCCC1N(C(=O)CC(=O)N(C)C)C2)(C(C)C)NC(C)=O 10961,c1(C(N(CCCCCNC(=O)C2=COCC2)C)=O)cnn2c1N(C)CC2 10962,c1(CC(=O)O)c(C)cccc1Br.C1(C(N(CCC)CCC)=O)CCN(C(C)(C)C)CC1 10963,C1(C(N2CCC(O)(CCNC(CCc3nc(C)sc3)=O)C2)=O)CC12CC(C)(C)C2 10964,c1(C(N(CCCCCC)CCNC(=O)C(C2CCC2)C2CCC2)=O)n[nH]c(C)c1Cl 10965,N1(C(CSCC#C)=O)CCC(CNC(C2CC2C2CC2C)=O)C12CC2 10966,C=CC(C)(C)CC(=O)N(C(CC(F)F)C(=O)N1CCC(OC2CCC2)C1)C 10967,c1(C(N2CC(C)(C(=O)NC3CN(CC)C3)C2)=O)cc2ccccn2n1 10968,N1(C(c2nc(OC)sc2)=O)CCC(C2CCN(C(=O)C(=O)NC(C)C)C2)CC1 10969,c1(CCC(N2C(C)CCC(NC(C=C(C)Cl)=O)C2)=O)ccc2ocnc2c1 10970,c1(CC)ccc(C(=O)NC2CC23CC(NC(C2CC2C(N)=O)=O)C3)cc1C(F)(F)F 10971,N#Cc1cc2c(nc1N1CC3CN(C(C4CC4(F)F)=O)CC3C1)CCCC2=O 10972,C1(NC(CC(=O)OC)=O)C2CCCC1CC(NC(C1CN3CCN1CC3C)=O)C2 10973,N1(C(CC(=O)N(CC#C)CC)=O)CCN(C(C2CN3CCC2(C)C3)=O)C2CCC12 10974,C1(c2cn(CCCC(=O)OC)nn2)CCCN(C(=O)C(C2CCC(F)(F)C2)=O)C1 10975,c1(C(=O)NC(Cc2c(C)noc2C)C)cc(Br)ncc1F 10976,C1(c2nnnn2C2CC2)CCN(C2CCCC2)CC1.C1(SCC=C)CCCC(C)O1 10977,c1(C(SC(F)F)=O)ccc(NC2CC(NC(C3(C(=O)OC)C=CCC3)=O)C2)nc1 10978,C1(C(=O)NCCCN(C(=O)CCc2nncn2C)C)Cc2cccc(F)c2O1 10979,C1(N(C)C(c2coc(O)n2)=O)CC2(CCCCN2C(c2nnn(C(C)(C)C)n2)=O)C1 10980,Cc1c[nH]cc(C(N2CC(NC(=O)CSc3cn[nH]c3)CC(O)C2)=O)c1=O 10981,C1(CC=C)(C(=O)NCCC2CC2)CCN(C(C2CCCCN2C)=O)C1 10982,CC1(NC(=O)CCc2nccs2)CCN(C(=O)C(F)CC2CCC2)C1 10983,C#CC1(NC(=O)C(CCC=C)NC(c2cnn3c2OCC3)=O)CCCCCC1 10984,c1(CC)cnoc1C(=O)NCCN(C(c1cc(C(C)(F)F)n[nH]1)=O)CC 10985,c1(C(=O)NCCN(C(c2csc(CCC(F)(F)F)n2)=O)C2CC2)ccc(F)cc1 10986,CC1(O)CCC(CC(=O)NCCNC(c2n[nH]c(C3CC3)c2Cl)=O)CC1 10987,c1(OC)cccc(S(=O)(=O)N2CC3CC2C3C(N2CCN(C)C(=O)C2C)=O)c1 10988,N(C1CCc2c(CO)ccnc21)C(COc1nc2ccc(C)cc2s1)=O 10989,c1(CN(C)C)cc(C(=O)NC2CCC(CNC(=O)C(F)CC3CC3)CC2)ccn1 10990,C(CCCC(=O)NCC(N1CCCNCC1)=O)CCc1cn(CCCCC)nn1 10991,C1(CNC(c2ccc(CSC)cc2)=O)CC(F)(F)CN1C(=O)C(C)S(N)(=O)=O 10992,C1(C(=O)NCC2CC3CCC(C2)S3)C2CCCCCCC12 10993,Cc1cccc(Cl)c1C(=O)NC1CC(NC(=O)C(C2CCCCC2)C)C(O)C1 10994,C1(CNC(CN2CCC(C)(O)CC2)=O)CC2(CCC2)CN1C(=O)C1=CCSC1 10995,c1(C(=O)NC2(CC)CCCN(C(C(CCC)(C)C)=O)C2)nc2cc(C)ccc2o1 10996,C1(C(=O)NCC2CCC2(F)F)CCCN(C(c2ccc(O)nc2)=O)CC1 10997,C1(C(=O)NC2(C)CCC(NC(c3ccoc3Cl)=O)CC2)CCC(C2CC2)CC1 10998,c1(OCCCC(=O)NC2(CNC(C3CCC(F)C3)=O)CC2)ccc(Cl)c(Cl)c1 10999,CN1CC=C(CC(=O)N2C3CCC2CN(C(c2coc4c2CSC4)=O)CC3)CC1 11000,C12(C(=O)Nc3cccc(O)c3)CCC(CC1)N2Cc1ccccc1 11001,c1(C(N2CC(NC(C3C(CCC)C3)=O)C2)=O)cnc(CC2CC2)s1 11002,c1(NC(C2(F)CCCN(Cc3cn(CCC)nc3)C2)=O)cnc2[nH]c(C)nc2c1 11003,C1(CNC(C=CC=CC)=O)COCCN(C(C2CC3CC3C2)=O)C1 11004,c1(C(N2C(C(C)N)CCCC2)=O)ccc2c(c1)C(=O)OC2(C)C 11005,O=C1CCCC2CN(c3nccc(N4CCc5c4ccc(Br)c5F)n3)CC2N1 11006,c1(C(=O)NC(C2CCN(C(c3cccnc3)=O)C2)C)nc2ccccc2s1 11007,c1(CC)ncccc1C(=O)N(C1(CC(N2CC(SC)C2)=O)CC1)C 11008,C1(C(N(CC(=C)C)CC)=O)CC=CCN1C(=O)Cc1csc(C)c1 11009,C12(NC(CCc3n(C)c(S)nn3)=O)CCC(CN(C(c3ccc(F)s3)=O)C1)C2 11010,c1(OC)nc(C)ncc1C(=O)NCC1CC2(CC2)CN1C(C1CCC(=O)C1)=O 11011,Cc1cc(C(=O)NCC(C2CCCC2)NC(c2ccccc2F)=O)c(O)nn1 11012,CC(C)C(C)(CNC(C1CCCC(C)O1)=O)NC(=O)CO 11013,C1(C)(CNC(c2[nH]cc(CC)c2)=O)CCCN1C(=O)C(O)Cc1cccc(Cl)c1 11014,C1(NCCC(=O)N(c2ccccc2C)C)CC2CCCCC2O1.CCO 11015,C1(CNC(=O)OC)CC(C)(C)CN1C(=O)Cn1cc(NC(C(C=CC)O)=O)nn1 11016,c1(C(=O)OC(C#C)CC2CCOC2)ccc(-c2ccc(Br)cc2)n1C 11017,C(=O)(C1=NOC2(CCC2)C1)NCC(CN(C(c1ccc(CN(C)C)[nH]1)=O)C)(C)C 11018,C(c1ccc(Cl)cc1)=CC(=O)NCC1CC(OC)CN1C(=O)CCc1cnoc1 11019,Cc1nc(-c2c[nH]cc2C(N2CCC2CNC(C2CC2C(C)(F)F)=O)=O)cs1 11020,Cc1cc(Cl)c(Cl)cc1C(=O)NC1CCCCC1NC(=O)CC1(C)CC1 11021,c1(NCCCCN(C(C(C)Oc2ccccc2)=O)C)cc(C(F)(F)F)nc(Cl)n1 11022,N1(CC=C(C)Cl)CC=CC1CBr 11023,c1(OC)cc(COC(c2ccc(SC(F)(F)F)nc2)=O)c(C)o1 11024,c1(C(=O)CNC=O)cc(Cl)ccc1OCC1CCCO1.c1cccs1 11025,C1(C)(C(=O)NCC(C)(C)CNC(=O)C2=CCCSC2)CC2CCC1O2 11026,c1(OC)ncc(C)c(C(N2CCC(NC(c3ccncc3Cl)=O)C(O)C2)=O)c1Cl 11027,C12(CNC(C(CC3CCC3)NC(C3CN(C(C)=O)C3)=O)=O)CC(C)(CCO1)C2 11028,N1(C(C(=Cc2ccccc2)C)=O)CCC(N=[N+]=[N-])(C(N2CCCC3CC23)=O)C1 11029,N(C1CCOc2cc(CNc3ccccc3)ccc21)C(N1CCCC12CCNC2=O)=O 11030,N1(C(C(c2c(C)nn(C)c2)O)=O)CCOC2(CCN(C(=O)CN(C)CCO)C2)C1 11031,N1(C(CCCC#N)=O)CCN(C(C2CCCS2(=O)=O)=O)CC1CC1CC1 11032,C#CCC(C)(C(=O)N1CCN(C(C)C)C(=O)C1)NC(=O)CCCCCF 11033,C1(C(N(C2CCCC2)CC=C)=O)CC2C=CC1N(C(=O)CC(=O)OC)C2 11034,CC1(C)C(NC(=O)CNC(C2CCOCC2)=O)CC1CNC(=O)CC1OCCO1 11035,c1(C(=O)NC2C(CNC(C(COC)N(C)C)=O)CC2)cnn2ccn(C)c12 11036,N1(C(C(C)(C)OCC)=O)C2CCCC1CN(C(c1ccc(C)c(C)c1)=O)C2 11037,CCC(C(=O)NCC1(COC(F)F)CN(C(=O)CNS(N)(=O)=O)C1)OC 11038,N1(C(C(OC)OC)=O)CCC(CC2CCCN2C(c2nccs2)=O)CC1 11039,n1(CC)nc(C(N2CCCC2CC(=O)NC2CCC(O)CC2)=O)c(C)n1 11040,C(=O)(C1=CCCSC1)NC1C(CNC(c2ccc(CNC(C)=O)cc2)=O)CCCC1 11041,C(=O)(CCC(=O)NCCOC)N1CC(CC=C)(NC(=O)C(C)OC2CCCCC2)C1 11042,N1(C(CC(CNC(=O)CN(CCCN=[N+]=[N-])C)OC)=O)CCN(C)CC1C 11043,C(=O)(C#CC(C)(C)O)N(c1ccccc1)CCC1(NC(C(CC)(C)C)=O)CCCC1 11044,C12(C(N3C(CC)CC(C)C3)=O)COCC1CN(C(C1CC1(C)C)=O)C2 11045,C(=O)(C(O)CC(C)C)N1CC(O)(CC(N2CC(C#CC)C2)=O)C1 11046,c1(C(=O)NC(CC)(C)CNC(c2cscc2Br)=O)ccc2scnc2c1 11047,N1(C(CCCSC)=O)C2CCC1C(CNC(c1cc(Br)c[nH]1)=O)C2 11048,C1(CNC(c2c(C)c(F)ccc2)=O)CCCCN(C(c2ccccc2O)=O)CC1 11049,C1(C(=O)NC(C23CC(CF)(C2)C3)=O)C2CC3C(C2NC(C2(F)CCCC2)=O)C13 11050,C1(NC(C2CC2CF)=O)CCN(C(=O)COc2ccccc2)C1C1CC1 11051,N1(C(c2cc(CC)no2)=O)CCC(CN(C(=O)CC(C)C2CCCCC2)C)CC1 11052,C(=O)(CN=S(C)(C)=O)N1C(CN(C)C(C2CC2c2ccncc2)=O)COCC1 11053,N1(C(CC(=O)OC)=O)CC=CC(NC(c2cncc(N(C)C)c2)=O)C1 11054,CCC(C)(C)C(=O)C(=O)N1C(CNC(c2cc3occc3s2)=O)CC2CC12 11055,N1(C(c2ccccn2)=O)CCCC(C(N2CCN(S(=O)(=O)CBr)CC2)=O)C1 11056,C1(CNC(c2nccnc2N)=O)C(C2CC2)CCN1C(C12CC(CO1)C2)=O 11057,c1(CC)nnc(CN2C(C3COC3)C2=O)s1.OC.CC 11058,C=CCCCC(C(=O)NC(C=C)C(F)(F)F)NC(=O)CCNC(C)=O 11059,c1(C(N2CC(c3n(C)cnc3)OCC2)=O)cccc(N2CCCC2)c1F 11060,C1(CC(=O)N(C(C)C(=O)NC2C3CCCC23)CC)CCCC(C)O1 11061,c1(C(=O)NCC2CCC(NC(C3C(CCC)C3)=O)CC2)nccc2cccnc12 11062,C1(NC(C(CC)CC)=O)CCN(C(c2ccc(CC#N)cc2)=O)C(C2CC2)C1 11063,CC(C)CC(C)(c1nnnn1C1CCOC1)NCCCc1cccc(Cl)c1 11064,Cc1cc(CC(N2CCCCC2CNC(C2C=CCS2)=O)=O)cc(C)n1 11065,C1(NC(=O)Nc2c(C)cc(C)c(Br)c2)CCCCC12CCCC2 11066,c1(C(=O)NC2C(C)N(C(=O)Cc3cncnc3)CCC2)cn2ccccc2n1 11067,c1(C(N2CC(CC(C)NC(=O)COCC3CC3)C2)=O)nc2c(s1)COCC2 11068,N1(C(C2CC(NC(c3c(=N)[nH]cnc3)=O)C2)=O)CC2(CC=CC2)C1 11069,c1(C(c2ccncc2OCC(=O)OC)=O)ccc(F)cc1.C1(C=O)CCCCC1 11070,N#CC1CCN(C(C2CCCCN2C(C2CC(N(C)C)C2)=O)=O)CC1 11071,c1(CNC=O)cnc(F)c(C)c1.CCCC(C(=O)N1CC(CC(C)(C)COC)C1)OC 11072,N1(C(C(CC=C)C)=O)CC(NC(c2ccnnc2)=O)CC(C)C1 11073,CC(Cc1nn[nH]c1C(=O)O)CCC(=O)N1CCN(C)C(C2CCOCC2)C1 11074,C(=O)(CCC(=O)NN(C)C)N(C)CC1(O)CCN(C(C(CC#C)C)=O)CC1 11075,c1(C(=O)NC23CC(C(=O)Nc4cc(C)nc(F)c4)(C2)C3)nc2c(s1)CN(C)CC2 11076,C1(CNC(c2c(C)nco2)=O)CC2(CO1)CN(c1ccnc(-c3nccs3)n1)C2 11077,C1(C(N2C(C)CC(NC(c3cc(C(=O)OC)n(C)c3)=O)C2)=O)CCC2(CCC2)CO1 11078,c1(C(C)OC)cn(CC(F)CCNC(=O)OC(C)(C)C)nn1 11079,C1(NC(CN(C(=O)CCn2cnnn2)CC)=O)CCCCC1C(C)(C)C 11080,c1(C(C(C)NC(c2nc(SCc3ccccc3)no2)=O)O)cccc(Br)c1 11081,N1(C(COCCCOC)=O)CCC(C(=O)Nc2cnc(SC)[nH]c2=N)C(C)C1 11082,c1(N(C)C)ccc(Br)cc1C(F)(F)F.N12C(CC3CC13)C2=O.N12CCCC1C2=O 11083,N1(C(CC(C)NC(CC(C(=O)OC)(C)C)=O)=O)CC2(C1)NC(=O)NC2=O 11084,c1(CCN(C(=O)COC(c2ccccn2)=O)C)cccc(F)c1 11085,N1(C(C=Cc2ncn(C)c2)=O)C2CCC1CN(C(c1cc(C3CC3)sn1)=O)CC2 11086,c1(C(CNC(=O)OC)=O)ccc(Br)c(Cl)c1 11087,CCC(C)CC(=O)NC1CC(CNC(=O)CSCc2ccc(Cl)s2)C1 11088,c1(C(=O)OCC2CN(CCC)C(=O)C2)nccc(-c2nnc(C(F)F)o2)c1CN.OC 11089,CC1C(C(=O)N(C)CC2(N(C)C)CCCC2)CCN1C(c1coc(CO)c1)=O 11090,c1(C(=O)NC(CSC)C(=O)NC2CCC(F)(F)C2)cc(C#N)ccc1F 11091,c1(OC)ccc(CC(=O)NCC2C=CCN2C(c2conc2C)=O)cn1 11092,c1(C(=O)NCC2(NC(C3C(C(=O)OC)CC3)=O)CCOCC2)occ2c1CCC2 11093,C1(=O)C(C)(C)C(=O)N2CCCC(C2)CN1.Cc1ccc(CNC(C)(C)C)nn1 11094,Cc1ccc(C(=O)O)c(-n2cc(-c3ccns3)nn2)c1.C12CCCN(C1)C2 11095,N1(C(c2c(C)n[nH]c2C)=O)CCN2C(=O)C(NC(=O)CC(C)(C)C)CC2C1 11096,c1(CN2C(c3c(C)cccc3)CCC2)cccc2cnccc12 11097,C(CC(C)C(=O)NCC(C)(C)CC1CN(C(c2cc(C)n(C)n2)=O)C1)OC 11098,C1(O)(C(C(=O)NOCCF)NC(CN(C)C2CC2)=O)CCCCC1.C1(CO)(O)CC1 11099,Cn1c(CN2CCOC3c4ccccc4OC23)nc2cccc(F)c12 11100,c1(OCC(=O)NCC2(OC)CN(C(C3(O)COC3)=O)C2)cc(Cl)ccc1Cl 11101,c1(C(NNC(C(=O)N(C(C)C2CC2)CC)=O)=O)cn2c(n1)C(C)CCC2 11102,N1(C(c2ccccc2-n2cc(C(C)OC)nn2)=O)CCCCCCCCC1 11103,Cc1ccc(C(C(=O)NCCCCCNC(C2(F)CC2(F)F)=O)C2CC2)cc1 11104,C1(C(=O)NC2CCN(c3ccccc3)C2)CN(C(C2CCNC2)=O)CCS1 11105,C1(CNC(c2cncc(OC)n2)=O)CCCN(C(=O)CN2CC=CC2)CC1 11106,c1(C(=O)NC23COC(CNC(C4(O)CCC4)=O)(C2)C3)cc([N+](=O)[O-])cnc1O 11107,C1(CC(=O)NC(C(C)(C)NC(c2cnc(C(C)C)s2)=O)C)CC(=O)NC1=O 11108,N1(C(CCC(C)(C)NC(=O)Cn2cnnc2O)=O)CC2CC(C1)C2(C)C 11109,c1(OC)ccc(C)c(C(=O)NCC(C2CCC2)NC(=O)CC2(O)CCCC2)n1 11110,O=S(=O)(c1cccc(F)c1)NC1CN(C(C2(CC(F)(F)F)CC2)C2CC2)CC1O 11111,c1(OC)cc(C(=O)NC(C)C(C)NC(c2cc(Br)n(C)n2)=O)ccc1C 11112,c1(C(N2CCC(N(C(=O)CC3CCC(=O)N3C)C)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 11113,c1(C(=O)NC(C(N2CCC(CN(C)C)CC2)=O)CO)ccc2n[nH]cc2c1 11114,c1(C(C)OC(C2CCCCN2C)=O)cccc(Cl)c1Cl 11115,c1(N2CC3CCN(C)C3C2)nc(=NCc2nccc(O)n2)[nH]c2c1COC2 11116,c1(C(=O)NC2C(O)CCN(C(CSc3nc(C)[nH]n3)=O)C2)cccc2c1OCC2 11117,C(=O)(C(CC(N)=O)NC(C1CC2CCC1CC2)=O)NCCc1nccc(C)n1 11118,Cn1cnn(CCCC(=O)NC2CCCC(NC(=O)CS(C)(=O)=O)C2)c1=O 11119,C1(n2c(C)ncn2)COCCN1N1CCC(OC(C)C)CC1 11120,c1(C(N(CC(C)(C)NC(C2CN(C(N)=O)C2)=O)C)=O)coc(COC(C)(C)C)n1 11121,c1(CC(C(=O)NCC(F)F)NC(C(CC)OC)=O)cnn(C)c1O 11122,c1(N2CC3CC(CNC(C4(CC)CC4)=O)C3C2)cc(OC)nc(CC)n1 11123,C1(C(=O)NC(C)CN2CCCC2)C2CCCC2CN1C(=O)Cn1ccc(Cl)n1 11124,N1(CCCOC)CC(C(=O)N(C(C)CNC(c2sccc2C)=O)C)CC1=O 11125,n1(CC(=O)NC2CCCN(C(C3OCCCO3)=O)C2)nc(O)ccc1=O 11126,CCC(CNC(=O)C(=O)NC1CC(=O)N(C(C)C)C1)(CC)c1ccccc1 11127,Cc1c(C(=O)N(CCC(=O)NC(CO)CCF)C2CC2)ccn1C 11128,c1(CCC)cc(C(N2CCC(N(C(=O)CCC3CCCC3)CCC)C2)=O)ccn1 11129,CCC(C(=O)N(C1(C(=O)NCC(F)Cl)CC1)C)C(C)C 11130,c1(CC(=O)NCC(C)NC(c2c(CC)ocn2)=O)ccc(F)c(Cl)c1F 11131,CC1(C)C(C)(C)C1(F)C(=O)NCCCCC1CCCN(C(c2csc(O)n2)=O)C1 11132,c1(CC(=O)NCC=CCNC(=O)CC2CC3CCC2CC3)nc2ccccc2s1 11133,C(CCNC(c1ccncc1OC)=O)(C(C)(C)C)NC(c1cccc(CC)n1)=O 11134,Cn1nnc2c1CCN(C(=O)C(CCC1CCC1)NC(=O)CC1CC(F)(F)C1)C2 11135,C1(CNC(c2n(CCOC)nnn2)c2nnn(C(C)C)n2)COC(C)(C)O1 11136,C1(COC)CC(CN)N(C(=O)OC(C)(C)C)C1.C1(=O)C(c2ccccc2)CN1C 11137,C(C)(CCC(C)(C)C)NC(c1nnnn1CCC(=O)OC)CC 11138,CC(C)P(=O)(CC(=O)NCC1(C(N)=O)CN(C(=O)C=CBr)C1)C(C)C 11139,C1(O)(CNC(C2(C(N3CC(C(N)=O)(SC)C3)=O)CC2)C2CCC2)CCCC1C 11140,CCCCC(CNC(=O)CCOC(C)=O)NC(C1(Oc2cccc(F)c2)CC1)=O 11141,CC(=O)C(C)CC(C)C(=O)N(C)CCNC(c1n[nH]c2c1CCC2)=O 11142,c1(C(=O)NCC(CC)NC(c2ccncc2F)=O)cccc(F)c1SC 11143,c1(C(N(C)CC2CC(F)CN2C(=O)C=CCF)=O)cccn2nnnc12 11144,c1(C(C)N(C)C(=O)N(C)CC2CCCO2)cnn(C)c1 11145,Cn1nnc2ccc(C(N3CC(NC(c4ccc(=O)oc4)=O)C4(CC4)C3)=O)cc12 11146,N1(C(C2(SC)CCC2)=O)CCN(C(C2CCCCS2)=O)C(c2nccn2C)C1 11147,c1(C(=O)NC2C(CN(C(CN(C(C)=O)C)=O)C3CC3)C2)nnc2ccccc2n1 11148,c1(OCC)cccc(C(=O)NC(c2occc2C2CC2)=O)c1.C12(C)CCN(C1)C2 11149,c1(C(C(=O)NCCCN(C(C(C)C2CCCC2)=O)C)C)ccc(Cl)c(Cl)c1 11150,N1(C(Cn2c(C)ncc2)=O)CC2CCC(NC(c3ccnc4nccn34)=O)C2C1 11151,N1(C(C(C)SC)=O)CCC(CNC(C2(COC)CCC2)=O)C(C)(C)C1 11152,C(CC(C)(C)C(=O)NCC(C1CCCC1)NC(c1cnc(Cl)cc1Cl)=O)OC 11153,C(C(CCC(=O)O)CC(F)(F)F)NC(C(CC(=C)Cl)(C)C)=O 11154,N1(C(CC(COC)C)=O)CCCC(C)(NC(=O)CCCc2ccc(Cl)cc2)C1 11155,N1(C(CCCN(C(C)=O)C)=O)CC2CC(C)N(C(c3cc4n(n3)CCO4)=O)C2C1 11156,c1(CCC)cc(C(=O)NCCC(C)NC(C2(C(F)F)CC(O)C2)=O)c(C)o1 11157,C1(C(=O)NCC2(F)CC(CNC(C3CCCO3)=O)C2)Cc2ccccc2S1 11158,CCC(C#N)C(=O)NC(CNC(c1cnn(CC)c1C1CC1)=O)CC(C)C 11159,C(=O)(CCCCC(C)C)N(CC)CC1CCCN(C(=O)C(c2ccccc2)O)C1 11160,CC1COCCC1N(C(=O)CCC1CC(NC(=O)CCn2cccn2)C1)C 11161,C1(NC(CCOCC)=O)CN(C(c2ocnc2-c2ccccc2)=O)CCC1CO 11162,CC(C)CC(C(=O)N1CC(C(=O)NC2CC2c2ccsc2)CC(C)C1)C(N)=O 11163,CC(C)(C)C(CNC(=O)C(O)Cc1ccccc1)NC(c1cn(CCF)nn1)=O 11164,C(=O)(C(O)CCCNC(c1cccc(O)n1)=O)NCC(CC(C)C)OC 11165,N1(CC(CC)CC)CCC2(CCN(C(=O)C(O)(C(F)(F)F)c3ccccc3)C2)C1 11166,N1(C(C2C(=C)CC2)=O)CCC(C(C)(C)C)(CNC(=O)CCn2cccnc2=O)C1 11167,c1(NC(C2C3(CN(C(CC(CC)C)=O)C3)C2)=O)cc(F)c([N+](=O)[O-])cc1F 11168,c1(C(N(CC(CC)NC(C2(O)CCOC2)=O)C)=O)ccsc1SC 11169,c1(NC(=O)C(N2C3CCCC2CC(O)C3)=O)ccc(S(=O)(=O)C(F)(F)F)cc1 11170,N1(C(Cc2c(C)ccnc2)=O)CC2CCC1C(NC(c1nc(C)n(C)n1)=O)C2 11171,C1(CNC(c2cncc(OC)c2)=O)CC2CCC1N2C(C1(C)CCC(C)CC1)=O 11172,C(=O)(C1CCCc2ncccc21)NCC(CNC(c1c(C)onc1Cl)=O)C 11173,c1(CN2C(C(=O)Nc3nccc(CO)n3)CC(F)C2)ccc(Br)cc1F 11174,CC1(NC(c2cscc2Cl)=O)CC(NC(C2(C)CCOC2)=O)C1 11175,C(N=c1cc[nH]cc1S(=O)(=O)NC(C)(C)C1CC1)c1cnc(CC)s1 11176,N1(C(CC2(NC(C3C(C)CC(=O)NC3)=O)CCC2)=O)CCC2CCC(C1)N2C 11177,C1(C(=O)NCCC(C)N(C(C(C)OCC#C)=O)C)CC12CCOCC2 11178,CC(CN(C)C)CCC(=O)N1CCCC1C1CCN(C(c2ncc(F)cc2F)=O)C1 11179,N1(C(C(CNC(C2CCCC[SH]2C)=O)OC)=O)CC2(COC(=O)C2)C1 11180,c1(C(=O)NC(CNC(C2CC3(OC)CC2C3)=O)C)ccc(C(C)C)c(C)c1 11181,c1(C(=O)NCCCN(C(C2OCCN(C(C)=O)C2)=O)CCO)cnc(CO)nc1C 11182,C1(C)(CNC(C(c2cccnc2)C)=O)CCCN1C(c1cccc[n+]1[O-])=O 11183,c1(C(=O)NCC(C)NC(=O)C(c2ccc(Cl)cc2Cl)O)nccc2[nH]ccc12 11184,c1(C(=O)NC2(C)CCN(Cc3cc4ccccc4s3)C2)ccc2c(c1)CCO2 11185,C(=O)(CC(CNC(c1csc(F)c1)=O)OC)NC(c1nccs1)CC 11186,Cc1nc(NCC2(C)CCOC2)cc(=NC(C)c2nc3c(s2)CCCCCC3)[nH]1 11187,N1(C(C2(C)COC2)=O)CC(C(N2CCCCC2CCCO)=O)C(C)(C)C1 11188,C(=O)(CC1OCc2ccccc21)N1CCN(CCNC(C(CCOC)C)=O)CC1 11189,Cn1c(=N)[nH]c2ccc(C(=O)NCC3CCN3C(c3ccnn3C(F)F)=O)cc12 11190,C1(CC(=O)C(=O)NC2CC2)CCCN1C(c1csc(NC)n1)=O.CCC(CS)N 11191,c1(N(N2C(CNC(C=CC)=O)CC(F)C2)C)cnc2c(c1)COCC2.C=O 11192,c1(C(N(CCCCNC(C2CC2C2CCCO2)=O)C)=O)ccncc1Br 11193,C1(NC(C(CSC)C)=O)CC2CN(C(c3cc(-c4ccncc4)on3)=O)CC12 11194,N1(C(CC2(C)N(C(Cc3cc(OC)no3)=O)CC2)=O)CCOCC1C1CCC1 11195,CC1(C2(C(N3CCC(CCC(=O)N4CC=CC4)C3)=O)CC2)CC1 11196,N1(C(C(C)(C)c2cnco2)=O)CC2CN(C(=O)CC3(C4CC4)CCCO3)CC2C1 11197,C1(N=[N+]=[N-])(C(N(C2CCCC2C#N)C)=O)CCN(C(=O)CN2CSCC2=O)C1 11198,N1(C(c2nc(C)nc(O)c2)=O)CC2CCN(C(c3cc(CO)[nH]n3)=O)CC12 11199,c1(C(=O)NCCC(C)NC(=O)CCC(=O)c2cccs2)nc2ccccn2c1F 11200,C1(NC(c2cnc(C3CCC3)o2)=O)CC2CCC1CN2C(c1cn[nH]c1)=O 11201,c1(N(C(=O)C(C)(F)F)C)nccn1CC1CN(C(=O)OC(C)(C)C)C1 11202,N1(C(=O)CCC2OCCO2)CCCC2C1CCN2C(=O)CC1CCC1 11203,C(CC(F)(F)Cn1cc(CCN(C)C)nn1)NC(COCCCC)=O 11204,N1(C(CC2(C)CCN2C(=O)COCCF)=O)CCC2(CCCCC2)C1 11205,N1(C(c2[nH]c3ccc(C)cc3c2)=O)CCC2CN(C(c3cc(C)on3)=O)CC2C1 11206,C1(C(N(CC)CC)=O)(NC(C2CCCCS2)=O)CCOCC1 11207,c1(CC(=O)NC(C2CCN(C(=O)C(O)Cn3cncn3)CC2)C)ccccc1C 11208,S(=O)(=O)(c1cccs1)NCC(=O)NC1(C2N(C(c3c(C)nsc3)=O)CCC2)CC1 11209,N1(C(CC(=C)C)=O)CC(NC(=O)CCc2cc(Cl)no2)CC(C)C1 11210,c1(C(N2C3CN(C(C4C(CCC)C4)=O)C(C3)C2)=O)ccc(Br)c2cn[nH]c12 11211,c1(C(N(C2CCCN(C(=O)C(C)CCOC)C2)CC)=O)c[nH]nc1[N+](=O)[O-] 11212,N1(C(C(C)=C(C)C)=O)CCC(NC(c2cc(C)cnc2Cl)=O)CC1C 11213,C1(CCC)CCC(C(=O)NC2(C)CCN(C(=O)C(COC(C)C)NC(C)=O)C2)CC1 11214,c1(NCc2c(N)nccn2)ccc(S(=O)(=O)NC2CCS(=O)(=O)C2)c(Br)c1 11215,Cc1cc(C)cc(C=CC(N2CC(CC(C)(C)CNC(=O)CCC(C)(C)F)C2)=O)c1 11216,CC(C)(CCCF)C(=O)NCc1ncc(C(=O)NOCC(F)(F)F)cn1 11217,N1(C(C2N(C(c3c(C)cno3)=O)CCC2)=O)CCN2CCCCC1C2 11218,N1(C(C(C)N(C(=O)CCCN(C)C(C)C)CC)=O)CC(CO)CC1CO 11219,N1(C(c2cnc(C)o2)=O)CC(NC(c2ccc(CC(C)(C)C)cc2)=O)CC1C 11220,C(=O)(CC(C)(O)COC)N1CCC(CCC)C1CC(F)(F)F 11221,C1(C(=O)NC(C)CCF)CN(C(=O)Cn2ccnn2)C2(CCC2)C1 11222,c1(OC)ncc(C=CC(N2CC(NC(C3CCCS3(=O)=O)=O)C3(CC3)C2)=O)cn1 11223,C=CC1(CC(=O)N(C)Cc2ccnn2C)CN(C(=O)CCC2CCCO2)C1 11224,Cc1onc(Cl)c1C(=O)NCC(C)CN(C)C(c1ccc(SC(F)(F)F)o1)=O 11225,C1(C(N2CCC(CNC(CCNS(CC)(=O)=O)=O)CC2)=O)CCCCC1(F)F 11226,N1(C(c2c(Cl)cn(C)n2)C(=O)NC2CCOC2)CCCC2(CCCNC2=O)C1 11227,CC1CC=C(C(=O)N2CCC(CN(C)C(c3cccc(O)c3C)=O)C2)CC1 11228,Cc1cc2nc[nH]c(=NCCOCCN(C)C(c3n[nH]cc3[N+](=O)[O-])=O)c2[nH]1 11229,C1(C(N2CCN(C(c3c(Cl)ccc(C)c3)=O)C(C)C2)=O)CCCC2CCCN12 11230,Cc1cc(C(C)C)nc(=NCC2CN(C(=O)Cn3c(C)csc3=O)CC2C)[nH]1 11231,C1(CN(C(C(C)O)=O)C)CCCN(C(=O)C=CCN2CCC2)C1 11232,c1(C(=O)NC2CC2NC(C2CCN(CCO)C(=O)C2)=O)ccc(O)c(Br)c1 11233,c1(NC(C(CNC(=O)CCNC(N)=O)OC)=O)cccc(C(C)F)c1 11234,c1(NC2C(C(=O)Nc3c(OC)cc(F)c(C)c3)C2)ncnc2c(C)cccc12 11235,CC1=C(C(=O)N(CCCCCNC(=O)C(F)C2CCOC2)C)SCCO1 11236,N1(C(C2(O)CCCN(C(C)=O)C2)=O)CC2CN(C(c3c[nH]c(=O)cn3)=O)CC2C1 11237,c1(C(N2CC3=C(CN(C(C4C(C=C)C4)=O)C3)C2)=O)cc(OC)nc2ccccc12 11238,Cc1cc(O)ccc1CNC(C12CC(NC(=O)OC(C)(C)C)C1C2)=O 11239,c1(C(=O)NCC23C(CN(C(C(CC)COC)=O)C2)CC3)cnc2[nH]cnc2c1 11240,C1(NC(C(C)NC(=O)NC)=O)CCCC(CNC(C2CC3CC3N2C)=O)C1 11241,CC(C)C(O)C(C)C(=O)N1CC(C(=O)NC2CC(C3CC3)C2)CC12CCC2 11242,N1(C(COCCC)=O)CC(N(C(=O)CNc2cccnc2)C)C(C)(C)C1 11243,C1(C)(CNC(C2(CC=C)CC=CC2)=O)CCCN(C(=O)CCN2CCCCCC2)C1 11244,C#CCC(C)(CNC(=O)COCCNC(c1cc(NC)c(C)o1)=O)CO 11245,CC(CC(C)(C)C)C(=O)NCC12CCC(C1)N(C(c1cc(Br)n[nH]1)=O)C2 11246,N1(C(C(C)C2CC2)=O)CCCC(CN2CCN(C(C3(F)CC=CC3)=O)CC2)C1 11247,N1(C(Cc2nc(C)oc2)=O)CC2ON=C(CNC(c3nsnc3O)=O)C2C1 11248,C1(C(N)=O)CC2CC(NC(=O)C(=O)NCC3CCN3c3ccccc3)C2C1 11249,C1(=O)C(C(C)(C)C)N(CC)CCCN1.C12(C(=O)NCC)CCCC1(CO)C2 11250,N1(N(C(CCC2CCN(C(C3CN(C)C3)=O)C2)=O)C)CCC(F)CC1 11251,c1(N2CC(CCC)OCC2)nc(NC2CC2CC(C)C)c2cnn(C)c2n1 11252,c1(CN2CCCC(NC(c3cnc(C)s3)=O)C2)ccc(C(F)(F)F)cc1O 11253,Cc1cc(CC(=O)NC2CC2NC(=O)C=Cc2ccc(C3CC3)cc2)ccc1O 11254,Cc1nccc(C(=O)NC2CCCC2NC(=O)CC(C)(C)O)c1N 11255,CC1OC(C)C(C(=O)NC2(CCCCNC(=O)CC3CC(F)(F)C3)CC2)C1C 11256,c1(C(=O)NCCN(C(c2nncs2)=O)CC)cc(N)ccn1 11257,N1(C(C2CC(OC)C2)=O)CCCC(C(=O)OCCN(C(=O)CSC(C)(C)C)C)C1 11258,CC(C)C(CNC(=O)CC1CSC1)C(=O)NC1(c2ccon2)CC1 11259,N1(C(N2CCn3nncc3C2)=O)CC(C)(CNC(=O)OC(C)(C)C)CC1(C)C 11260,O=C(C#CC1CCCCO1)NC1CCC2CCN(C(=O)CN3CCCNC3=O)C12 11261,Cc1cn2c(n1)CCC(C(N1CC3(NC(c4sccc4F)=O)CC1C3)=O)C2 11262,C1(NC(=O)Cc2cc(OC)ccn2)CCCCCC1.CCC1CCC(=O)N1 11263,N1(C(C2(C(=O)OC)C(=C)CC2)=O)CCC(NC(=O)C(C)(C)C(N)=O)C(CC)C1 11264,Cc1ccnc(C(=O)NC2COCCN(C(C3(n4nccn4)CC3)=O)C2)c1F 11265,CC(C)CC(C)C(=O)N(CCC(C(C)(C)C)NC(C1CN(C)C(=O)N1)=O)C 11266,N1(CC(=O)NC2C(NC(=O)CC3CC(n4cccn4)C3)C2)CCS(=O)(=O)CC1 11267,Cn1nc(CNC(=O)N=c2ccn(CCCC(F)(F)F)[nH]2)c2c1CCC2 11268,C#CC1(C(=O)NOCC(C)=CCC)CCN(C(C2OC3CCC2C3)=O)CC1 11269,CC1(C)CCN(C(=O)C2=CCCCO2)CC1NC(c1ccc(Cl)s1)=O 11270,C(=O)(CCCCCCCSC)NC1(C)CCCN(C(c2c(CC)cccn2)=O)C1 11271,C12(NC(c3cc(C(F)F)[nH]n3)=O)CCCC1CN(C(=O)Cc1ccsn1)C2 11272,n1(CNC(NCc2nn(CC)nc2C)=NCCCCl)cnc2ccccc2c1=O 11273,c1(C(N2C(C3(NC(CCC=C(C)C)=O)CC3)CCC2)=O)ncc(Cl)cc1O 11274,Cc1cc(C(=O)NCC2CCN2C(=O)CCC2CCCOC2)c(C)n1CC1CC1 11275,C=CC(C)(O)CC(=O)NCc1cc(C(=O)NC(C)COCCOC)no1 11276,C(=O)(C1=CN(C(=O)OC)CC1)NCC(C)N(C(CCCOCCCOC)=O)C 11277,C(=O)(C(CNC(c1cc(O)cc(=O)o1)=O)C(C)(C)C)NCC1CC(CC)C1 11278,C1(NC(C23CC(C)C2C3)=O)CCC2CC1CN2C(=O)Cc1ncncc1Cl 11279,C(C)(C)(CC(=O)NCCCc1ccccn1)N(C(C1C(C)C1C)=O)C 11280,c1(CC)nc2n(n1)CC(NC1CCCC1C(=O)Nc1cc(O)ncn1)CC2 11281,N1(C(CN2CCCC(CC)C2)=O)CCC(NC(=O)Cc2ccsc2Cl)C12CC2 11282,N1(C(C2CN(CC)C(=O)C2)C(=O)NCCC2CC2)CCOC2(CCCSC2)C1 11283,c1(NC2(C)CC(NC(C3CC3C3CCOCC3)=O)C2)ccc([N+](=O)[O-])cc1 11284,CC(C)CC(CNC(=O)CCC(=O)c1cccc(F)c1)NC(=O)C(C)CC#N 11285,C(=O)(C1=CC2C=CC(C1)C2)NC(C(=O)NC(C=C)C1CC1)CO 11286,C1(NC(C=NOC)=O)C2CC3CN(C(=O)CCCCC(F)(F)F)C1C3C2 11287,CCC(CNC(c1cscc1C)=O)(CC)NC(c1ccc(C2COC2)cc1)=O 11288,N1(C(CC=C(C)C)=O)CCC2(NC(c3cccc(O)c3C(F)(F)F)=O)CC2C1 11289,Cc1ccc2n1C(=O)N1CC(C(C)C1)CC1(CC1)NC2=O.C1(C(C)C)CCCO1 11290,CCCC(C(=O)NC1(C)CN(C(c2nc(C)sc2C)=O)C1)N(C)C 11291,N1(C(CCC=CC(C)C)=O)CC2(CCCC2)C1 11292,CCC(COC)C(=O)NC(C)CC(C)NC(c1ccn(C(C)C)n1)=O 11293,C1(C(=O)NCCNC(=O)C(F)(F)F)CCCCN1C(=O)CCc1cncc(O)c1 11294,C(CCS(=O)(=O)NCC(N1CCC(c2ccc(CC)s2)C1)=O)OCC 11295,CCC(CC)C(=O)NCC(=O)NCCCC1(NC(=O)C(C)C(C)O)CC1 11296,CC1=C(C)CC(C)(C(=O)NCC2CC3CCC(C2)N3C(C2CCCO2)=O)CC1 11297,n1(C(C(=O)NCC(CCOC)NC(=O)Cn2ccc(C3CC3)n2)C)c(C)ccc1C 11298,Cc1ncc(F)c(N(C2CNCC2C#N)C(c2cccc(O)c2O)=O)n1 11299,C1(NC(c2n[nH]cc2-c2ccncc2)=O)CC2(C1)CN(C(C1CCCCO1)=O)C2 11300,c1(C(=O)NC2CN(C(=O)C(F)(F)c3nccs3)CCC2O)cccc2nccn12 11301,N1(C(c2c(C)n[nH]c2)=O)CCCCC1C1CCCN1C(=O)CCc1cnccn1 11302,c1(CC(=O)N(CCCNC(C(CCC)N(C)C)=O)CC)ccc2ocnc2c1 11303,CCC1c2ccsc2CCN1C(c1cc(F)ncc1F)C(=O)NC(C)(C)C 11304,C(C(C)(C)C(=O)NC(C)CCCNC(=O)C(O)CCSC)OCC 11305,Cc1cc(NCc2c(Cl)cncc2Cl)cc(C(F)(F)F)c1 11306,Cc1cc([N+](=O)[O-])cnc1C(=O)NC1(CCNC(=O)CC2C=CCC2)CCCC1 11307,CN1CCCC1C=CC(=O)NCCN(C(=O)C=Cc1cscn1)C1CC1 11308,c1(CCC(=O)NCC(CC)NC(=O)C(C)=CC(C)(C)C)ccc(OC)c(OC)c1 11309,C1(C(N2C(C(C)(C)NC(c3ccc(CC)cn3)=O)CCC2)=O)C(C)OC(C)C1C 11310,C(C(=O)OC(C)(C)C)(C(=O)N1CC(C)(NC(=O)CCCC2CCC2)C1)OC 11311,c1(C(N(CC(CC)NC(CC(=C)I)=O)C)=O)n[nH]c(C)c1O 11312,Cc1cc(Cl)cnc1C(N1CC(C(N2CC(O)(SC(F)F)C2)=O)C1)=O 11313,Cc1cc(F)c(CC(N2CCCC2C=Cc2ccccc2)=O)cc1F 11314,c1(NC(C2(O)CCC(CC)CC2)=O)cc(F)ccc1C(F)(F)F 11315,CCC(CC(=O)Nc1ccoc1)NC(=O)Cc1cnsc1 11316,c1(CNC(Cc2cn(CC)nn2)=O)ncccc1CNC(C1CCC(=O)C1)=O 11317,C(C(C(C)C(C)C)NC(=O)CCc1cccc(Cl)n1)NC(c1cnc(CC)[nH]1)=O 11318,C=CC1OCCC1C(=O)NCCOC1CN(C(=O)CC(O)CN(C)C)C1 11319,C=CC(C)(C)CC(=O)N(CC(C)O)CCN(C(=O)CC1(OC)CCC1)C(C)C 11320,c1(NC(=O)NC(c2ccn(C)c2)C)cc(C(N)=O)c2n1CCOC2 11321,NS(=O)(=O)c1cc(C(=O)NC2CC(F)CN(C(C3CCCOC3)=O)C2)ccc1F 11322,Cc1ccc(C(=O)N(CC(C)O)CCNC(c2coc(Br)c2)=O)o1 11323,c1(Cc2scc(C(=O)NCC3CC(F)(CNCC4CC4)C3)n2)cccc(Cl)c1 11324,C1(CCNC(c2ccc(C)o2)=O)COCCN1C(=O)CCc1ccccn1 11325,c1(OC)cc2[nH]ncc2cc1NC(=O)CC1CCN(C(c2cncnc2)=O)C1 11326,c1(OCC2CCCC2C(=O)OC(=O)OCC)ccc2c(c1)OCCO2 11327,Cc1cnc2n1CCCC2C(=O)NCC1CC1C1CCCC1 11328,c1(C(N2CC(O)(SC(F)F)C2)=O)ccc(CNC(C2CC(O)C2)=O)nc1 11329,N1(C(=O)CCc2cnc[nH]2)CC(O)C(O)C1CNC(=O)C(=O)NCC(F)F 11330,C1(C(N(C(C(=O)NC2CCC(C)C2)(C)C2CC2)C)=O)CC(=O)CC(=O)N1 11331,N1(C(C2CCC(=C)CC2)=O)CCC2CCN(C(=O)C(C)OCCN(C)C)CC2C1 11332,c1(C(=O)NC2CC(C)N(C(C3CSCC(=O)N3)=O)C2)cc2c(cn1)OCCO2 11333,c1(C(=O)NC2C(NC(c3c(CC)noc3)=O)C2)nc(C)n(C)n1 11334,C(C#CC(F)(F)F)NC(C(C1CCN(C(=O)OC)C1)F)=O 11335,c1(NC2CCC(CS(N)(=O)=O)C2)ccc(S(=O)(=O)NC2C=CCC2)cc1Cl 11336,c1(C(N2CCCC(N(C)C(C3CC(O)C3)=O)C2)=O)ccc2c(c1)C=CS2(=O)=O 11337,c1(CO)cccc(NC(c2cc(CC3CC3)on2)=O)c1.O=C1CC2(CC2)CN1 11338,Cn1c(C(N2CCOC(C3CN(C(=O)C=CCO)C3)C2)=O)cnc1O 11339,C(N=c1cc(C)nc[nH]1)C1CN(C(C(C)NC(COC)=O)=O)CC1(C)C 11340,C(CCO)(C(C)(C)O)NC(C(Cc1cn[nH]c1)NC(C(C)OCC1CC1)=O)=O 11341,c1(NC(C2CC(C)CN2C(=O)CCc2cncnc2)=O)ccc(CO)c(F)c1 11342,C1(NC(C=CCCC)=O)CC2COCC(C1)N2C(C1CN(C(C)=O)CCO1)=O 11343,c1(C(=O)NCC(CO)NC(c2ccc(COC)cc2)=O)cccc([N+](=O)[O-])c1 11344,Cc1c(Cl)ccnc1C(N1CCC(CF)(NC(=O)CCc2ncc[nH]2)C1)=O 11345,c1(C(=O)NCC2CCN2C(c2ccnnc2)=O)nc(O)c2ccccc2n1 11346,n1(CCC)nnnc1C(c1nc(Cl)cs1)NCCC(=O)OC(C)(C)C 11347,Cn1nccc1C(N1CCC(c2ccccn2)C1)C(=O)NC1(C)CC1 11348,N1(c2nnc(-c3n(C)c(=O)on3)n2C)CCN2C(=O)COCC2C1 11349,C(N=c1[nH]cnc2cc(C)[nH]c12)C1C(NC(Cn2ccc(C)cc2=O)=O)CCCC1 11350,N1(C(C(C(CC)C)C#N)=O)C2CCC1C(c1cn(CC(OC(F)(F)F)C)nn1)C2 11351,c1(C(C(=O)NC2CCC2)N(C2CCN(C)C(=O)C2)C)cccc2[nH]ncc12 11352,C12(C(N3CC(O)(CC(=O)NCC4(CO)CCN(C)C4)C3)=O)CCC(CC1)CO2 11353,C1(CC(=O)N(CCCOC)C)CN(C(c2snnc2C)=O)CC12CC2 11354,Cc1cc(C)c(C(N2CC3CCC2C(NC(c2cccs2)=O)C3)=O)c(C)c1 11355,C1(C(=O)NC2CCCC(N(C(=O)C3=CCOCC3)C)C2)C(C)(C)CCCC1(C)C 11356,N1(C(c2c(CC)c(C)sc2)=O)CCCC2(C1)CN(C(C1CN3CCN1CC3)=O)C2 11357,Fc1cccc2cccc(CNCc3cc(F)cnc3Cl)c12 11358,Cc1ccc(NC(=O)C=CC2CCN(C(C34CCCC(CO3)C4)=O)CC2)cc1F 11359,C(C(C)(C)C#CC(=O)N1CCCC(C(=O)NC)C1)NC(C(C)SCCCC)=O 11360,C(C(C)(O)C(C)CC)NC(c1cc(CNC(c2c(C(C)C)onc2)=O)sc1)=O 11361,N1(C(C(C(C)O)NC(c2c(NC)scn2)=O)=O)Cc2ccnn2CC1C 11362,C1(CNC(C2(COC)CCCC2)=O)CC(C)(C)CN1C(=O)C1CC1 11363,c1(C(N2CCCC(CC)(NC(=O)C3=CCCC3(C)C)C2)=O)ccc(Cl)c(C)c1N 11364,C(=O)(CCC(=O)NCC(C1CCCC1)NC(C1(C(C)OC)CCCC1)=O)OCC 11365,S(=O)(=O)(c1cccc(F)c1C)N1CCC(O)(C(C)NC(C2(CC)CCC2)=O)C1 11366,C(CCCCCC(=O)N(c1csnc1C)C)COC(C(OC)OC)=O 11367,C1(NC(=O)NC2CCCN(C3CCC3)C2)CCNC2(CC2)C1 11368,CN1CCCC1CCCNC(=O)Cc1cc(C(=O)O)cs1 11369,c1(C2(C(N(C3CN(Cc4cn(C)cn4)C3)C)=O)CC2)ncccc1F 11370,C1(C(C)C(=O)N(C2(C(=O)NC(C)C(=O)NC3CC3)CC2)C)CCC(=O)N1 11371,c1(OC)ncc(Cl)cc1C(=O)NC1CCN(C(=O)C(C)C(F)F)C1 11372,C#Cc1cccc(CC(=O)NC2CCN(C(=O)CC=C=C)C(C)C2)c1 11373,N1(C(C(C=CCCC)O)=O)CCN(C(=O)C=C(C)c2ccccc2C)CC(CO)C1 11374,C#Cc1cc(NC(=O)Cc2ccc(C=O)[nH]2)cc(COC)c1 11375,c1(NC(c2ccoc2)=O)ccsc1C(=O)NCC1CC1 11376,c1(C(=O)NC(c2ccc(C)cc2)c2c(C)noc2C)cc(Cl)ccc1C 11377,C=C(C)C1OCCC1C(N1CCC2(CC2NC(c2ccc(CO)o2)=O)C1)=O 11378,N1(C(c2cc(OC)no2)=O)CCC(C2CC2)(NC(C2(SC3CCC3)CC2)=O)C1 11379,c1(C(N2CCC(N(CC(F)(F)F)C)C2)C(=O)NCC(=C)C)ccccc1I 11380,N1(C(C(c2ccccc2F)C)=O)CC2(CCCC2)c2cc(Br)ccc21 11381,c1(N2CCCC(C)(OC)C2)ccc(S(=O)(=O)N2CCCC(N(C)C(C)=O)C2)cc1F 11382,C(=O)(C(CC)C(=O)OC)NCC(CCOC)NC(c1nccc(CC)c1)=O 11383,CC1=C(C(=O)NCC2CCC2NC(=O)CN2CCCC2=O)Cc2ccccc2O1 11384,C1(C)(N(C(=O)CCSC(C)(C)C)C)CN(C(c2cnc(C3CC3)o2)=O)C1 11385,N1(C(C(C)OC)=O)CC2(CNC(=O)C(C)CCc3ccc(F)cc3)CC1CCO2 11386,c1(C(C(=O)NCC2(NC(C3CC34CCC4)=O)CC2)(F)F)ccccc1F 11387,c1(C(N2C(CNC(c3cccc(OCCOCC)c3)=O)CC2)=O)c(I)ccnc1Cl 11388,C1(C(=O)NCC(C)(C)OC)CN(C(=O)C(O)CSC)CCC1(C)C 11389,N1(C(COCCCOC)=O)CCOCC1CNC(c1conc1C(C)C)=O 11390,C12(C(=O)NCC(CC(=O)OC)C)CCC(CN(C(=O)CCCNC(C)=O)C1)C2 11391,N1(C(C(C)NS(CC)(=O)=O)=O)CCOC(CNC(=O)C(C)(C)c2csc(C)c2)C1 11392,n1(CC=C)cc(C(=O)NCCN(C(c2cn(CC)nn2)=O)CC)nn1 11393,C12(C(=O)NC(COC)C(C)(F)F)CCC1(C(=O)O)CN(C(=O)OC(C)(C)C)C2 11394,c1(CC)ccc(C(=O)NC(CO)C(C)NC(C2CCCC2(F)F)=O)cc1 11395,CCC(C)CC(C(=O)NCc1cccnc1)NC(c1cc(C(C)=O)[nH]n1)=O 11396,N1(C(C2(C)CC(=C)C2)=O)CCC(CCCNC(C23CCCC2C3)=O)CC1 11397,N1(C(C2(CC)CC2)=O)CCCC2(C1)CN(C(c1ccnc(OCCN(C)C)c1)=O)C2 11398,C(C)(C)(CCCC(=O)NCc1cc(C)cc(C)c1O)NC(CC(=O)NCC#C)=O 11399,CCC(C(F)(F)F)CC(N)C(=O)N.c1(C)nc(CO)cs1 11400,N#CC1CCCCC(CC(N2CCC(CNC(=O)CC3CC=CCC3)CC2)=O)C1 11401,n1(CC)ccc(C(N2CCCC2C(C)(C)CNC(C2COCC2OC)=O)=O)n1 11402,CC1CN(C(=O)COc2cc(Cl)ccn2)CCCN1C(=O)CCCC1CCC1 11403,C1(C(=O)NC2C(CCC)C2)(COC)CCN(C(c2cc[n+]([O-])cc2)=O)C1 11404,C(=O)(C(C)(CC)C(=O)N1CCC1CNC(c1c(SC)cccc1F)=O)OCC 11405,C1(C(=O)NC(COC)CNC(=O)CN2CCCC2C)CC2CC(=O)C1O2 11406,Cc1cc(C(=O)NC2CCCC(NC(c3cc(C)sn3)=O)C2)ncc1S(N)(=O)=O 11407,C1(NC(c2c(C)onc2Cl)=O)CC(C)CN(C(c2ccc3c(c2)CC3)=O)C1 11408,N1(C(Cn2nnc(C)n2)=O)CCC2(CC1)CCN(C(=O)C(C)SC(C)C)C2 11409,CC1(C)CCc2c1n[nH]c2C(=O)NC1CCSC12CN(C(=O)C1CC1)C2 11410,N1(C(Cn2cc(C(N(C)C)=O)nn2)=O)C2CCCC1CC(NC(=O)CCCF)C2 11411,N1(CC(=O)NC2(C)CCCC2)CC2CCC1C(Nc1ncccc1C#N)C2.CO 11412,c1(C(=O)NC2C(NC(C(C)=C3CCCC3)=O)CC2)cc2c(C)cccc2[nH]1 11413,Cc1nc(C#N)c(N(CCC(=O)NC(C)C(C)NC(C2CCCCCC2)=O)C)o1 11414,N1(C(C(CO)NC(N)=O)=O)CCC(F)(C(=O)NCc2ccccc2F)C1 11415,C1(OC)CC(CO)(NC(=O)NCC2C=CCC2)C1(C)C 11416,c1(CCC)cc(C(=O)NCCCC(C)NC(c2c[nH]nc2F)=O)c(C)o1 11417,CCC(CC)(CC(=O)OC)NC(c1ccc(Cl)cc1NC)C 11418,N1(C(CC(=O)OCC)=O)CCC(NC(=O)C2=COCC2)C(F)C1 11419,c1(C(=O)OC)cc(Br)c2[nH]c(=NC3CC4C=CC3C4)[nH]c(=N)c2c1 11420,N1(C(C(C)SCC)=O)CCCCCC1CNC(=O)C1=CCOC1 11421,C1(C(N(C2CCCN(C(c3ccc(C(N)=O)o3)=O)C2)CC)=O)CC(=O)N(O)C1 11422,C1(CC(=O)NC(CCC)CNC(=O)C(C)=CC2CC2)(CC)CCOCC1 11423,C(=O)(C1Cc2ccccc21)N(C)CCOCCCNC(=O)CC1C=CCC1 11424,C1(C(=O)NC(C)CF)CN(C(c2cncc(N(C)C)c2)=O)CCC1(F)F 11425,N1(C(C2N(C(CCC3CC(C)C3)=O)C3(CC2)CC3)=O)CCC2CN(C)CC12 11426,C1(OC)CN(C(=O)C=CC2CCCC2)CC1NC(C1CCN1S(C)(=O)=O)=O 11427,c1(CN(C(C)C)C(C2CC(CNC(=O)CCCc3ncco3)C2)=O)cccnc1 11428,c1(C(N2CC3C(CNC(C=C(C)C(C)C)=O)(C3)C2)=O)ccc(Br)c(F)c1C 11429,C#Cc1ccc(C(=O)NC2(C(=O)NCc3ncn(C)n3)CCSC2)cc1 11430,C1(COC)(CNC(c2nocc2C)=O)CCN(C(C2CCC(C)(C)C2)=O)C1 11431,C#Cc1cc(C(=O)NCC2(C)CCC(NC(c3cnsc3)=O)C2)ccc1C 11432,n1(CC(C)O)nc(-c2ccc(Cl)cc2)nc1-c1ccn(Cc2cccc(F)c2)n1 11433,C(=O)(C(F)C(C)(F)F)NC(C(=O)N(CCOCC)C)(C)CO 11434,C12(CNC(COC)=O)CCCC(CN1C(=O)CCc1nc(C)c(C)o1)C2 11435,c1(C(=O)OC)sc(C(N2CC=CC(NC(C3(N(C)C)CCCC3)=O)C2)=O)cc1N 11436,Cc1cc(Br)cc(C)c1NNC(=O)CSc1cccc(F)c1C#N 11437,c1(C(=O)NC2CCCN(C(C3C(C=C)C3)=O)C2)cncc(C)c1O 11438,Cc1cccc(F)c1C(N1CCC(C)(CNC(=O)CC(F)(F)Cl)CC1)=O 11439,N1(C(CC(C)(C)O)=O)CCC(NC(=O)CCNC(=O)C=CCl)C(F)C1 11440,C1(C(=O)NCCCNC(c2occ(C(=O)OCC)n2)=O)CC2OC(C)(C)OC2C1 11441,N(C1CCc2cccnc21)C(CN(C(C(=O)NC1CCC1)c1ccoc1)C)=O 11442,c1(CC)cc(C(=O)N(CCCNC(=O)CC2CCC(C)C2)C)no1 11443,S(=O)(=O)(c1ccc(N(C)CCC2CC2)cc1Br)N(C(C)CN)C 11444,C1(C(=O)N(C)Cc2ccns2)(NC(C2N(C)CCC2)=O)CCCC1 11445,C1(CN(C(CC)=O)C)CCCC(NC(=O)CS(=O)(=O)NC(C)(C)C)C1 11446,c1(C(N(CC(CN(C(c2c(CC)nc(C)o2)=O)C)O)C)=O)cccc(F)c1C 11447,c1(OC)cc(C(=O)N(CCC(C)NC(=O)C(O)Cc2cn(C)cn2)C)[nH]n1 11448,c1(C(N2C(C(=O)Nc3ccc(F)c(I)c3)CCC2)=O)cc(O)c(Br)c(O)c1 11449,CCCCC(CNC(c1n[nH]c(C)c1C(F)(F)F)=O)NC(C1(CO)CC1)=O 11450,c1(CN(C2CCN(C(=O)CCn3ccnc3)C2)C)c(F)cc(C(=O)O)cc1F 11451,C1(CC)CN(C(=O)CCCOC(C)=O)CCC1NC(c1cc(C#N)cs1)=O 11452,N1(C(CC(=O)NCC)=O)CCC2(C=C(C(=O)N3CCOC(C)CC3)C2)C1 11453,C1(N=[N+]=[N-])(C(=O)NCCC(C)(C)SC)CCN(C(c2oc(C)nc2C)=O)C1 11454,C1(NC(CC(CNC(c2ccnn2CCF)=O)O)=O)CCCCCCC1O 11455,c1(CC)nc(C)c(C(=O)NCCN(C(=O)C(C)C2CCC2)Cc2ccccc2)s1 11456,C1(CC)CC(C(=O)NC(CNC(=O)CC2CCOC2(C)C)C(C)(C)C)CCO1 11457,Cc1cnc(N(C)CCN(C(=O)Cc2cnccn2)C(C)C)nc1C 11458,N1(C(c2ccnc(OC)n2)=O)CCCC2C1CCCN2C(=O)Cc1cc(C)ns1 11459,CCCC(CCC)C(C)NS(=O)(=O)Cc1ccc(F)cc1Cl 11460,N1(C(CN(C)C2CC2)=O)CCCC(O)(CNC(c2ccnnc2O)=O)C1 11461,c1(C(=O)NC(C=CC(=O)N(CCCCSC)C)(C)C)occc1C(C)C 11462,C1(C)(CNC(CS(=O)(=O)NC(C)(C)C)=O)CCCN(C(C2(C)COC2)=O)C1 11463,N1(CCC)CC(C(=O)NCCCCCCNC(c2ccsc2C)=O)CC1=O 11464,CC1CN(C(C23CC(C2)C3)=O)CC1N(C(C1CCC(N2CCCC2=O)CC1)=O)C1CC1 11465,C(=O)(CC1=CCCC1)NCC(c1ccccc1)CNC(C1CCN(CC)CC1)=O 11466,C(C)(CCCCNC(C1CCCC1(F)F)=O)NC(Cn1ccc(C(=O)OC)n1)=O 11467,N1(Cc2c(OC)cccn2)CC(C(=O)Nc2ncc(C(F)(F)F)cc2C)CC(F)C1 11468,CN1N=C(CC(=O)N2CCCCC(N(C)C(C3CC4(CCCO4)C3)=O)C2)CC1=O 11469,N1(C(c2c(CC)cco2)=O)CCCC(F)(C(=O)NCCOCC2CCCC2)C1 11470,CC(C(C)(C)NC(c1cc(CO)[nH]n1)=O)NC(c1cnn(CC(F)(F)F)c1)=O 11471,C(CC1=CCN(C(=O)C(N2CCCCCC2)C)CC1)NC(C=CC=CCC)=O 11472,C1(CNC(CC2CCC(=O)NC2)=O)(NC(c2csnn2)=O)CC2CCC1CC2 11473,c1(C(=O)NC2C(C)N(C(=O)CSC(F)F)CC2)c[nH]c2cnccc12 11474,N1(C(Cc2c(C)scc2)=O)CC2CC2(NC(=O)CCc2cncc(O)c2)C1 11475,C1(CNC(CCOC2CN(C(c3ccc(CC)[nH]3)=O)C2)=O)CCC(CO)CC1 11476,C12(NC(CC3CC(=C)C3)=O)CCCC(NC(c3ccc(=N)[nH]n3)=O)(C1)C2 11477,C1(O)(C(=O)NC2CCN(C(c3nccc(SC)n3)=O)C2C)CCCC(C)(C)CC1 11478,O(NC(=O)CC1(CNC(=O)C=CCNC(N)=O)CC1)CC(C)C 11479,Cc1cn2c(CC(=O)NC(C)C(C)(C)NC(C3CCCCC(=O)N3)=O)csc2n1 11480,C1(NC(c2ccc(Cl)[nH]2)=O)CN(C(C2C=CC=CC=C2)=O)CC12CC2 11481,c1(C(=O)NCC(C)(CC)NC(CC(C=C)(C)O)=O)cnc2ncnn2c1O 11482,Cc1ccc2ccccc2c1NCC1C2CCCC1NC2 11483,C1(NC(C2(CC(C)C)CCC2)=O)CN(C(C2(N3CCCC3)CCC2)=O)CC1F 11484,c1(OC)cccc(CCC(N2CC(NC(=O)CCC3CCC3)CC(C)C2)=O)c1F 11485,c1(C(=O)Nc2cc(C#N)nc(C)n2)n[nH]c2cc(-c3cc4sccc4s3)ccc12 11486,Cc1ccnc(C)c1C(N1CCCN(CCNC(C2CC(=C3CC3)C2)=O)CC1)=O 11487,C(C(C)CC(=O)NC1CC(NC(c2coc(-c3ccccc3C)n2)=O)C1)OC 11488,c1(C(=O)NCC23CCCC2CC3)cccc(N2CCCCC2)n1 11489,N1(C(C=CC=CC)=O)CCC(C(F)CNC(C2CC2[N+](=O)[O-])=O)CC1 11490,c1(C(N2CCC(F)(CNC(CC(CCC)C)=O)C2)=O)cnc2c(C)cccn12 11491,N1(C(Cc2nc(C)[nH]n2)=O)CCC2CCCC12CNC(c1ccc(F)s1)=O 11492,CC(C(=O)NCCCCN(C)C(C1OCCO1)=O)OC1COC1 11493,C1(F)(CNC(C=CC)=O)CCN(C(=O)CC2(O)CCCC2)C1 11494,C(=O)(CCCCCC(C)C)N(CCC(C(C)(C)C)NC(C1C(C=C)CC1)=O)C 11495,C1(NC(c2nnn(C)c2N)=O)CC2(C1)CC(NC(c1cc(Cl)c(Cl)n1C)=O)C2 11496,N1(C(=O)C(C#N)C(C)C)CC2(C)CN(C)CC2(C)C1.Cc1cccc(C)c1 11497,C1(CN(C)C(c2cnc(O)n2C)=O)CCC(NC(c2ncoc2C2CCC2)=O)CC1 11498,C1(C(N(CCCCC)C)=O)CCN(C(C23C=CC(CC2)C3)=O)CC1 11499,C1(C(=O)NCCOCCC(=O)OC)COCCC1NC(=O)Cc1ccccc1C 11500,N1(C(COCC=C)=O)C(CNC(=O)C(c2ccc(Br)cc2)C)CC2CCCC12 11501,C#Cc1cc(F)c(C(=O)NC(CNC(C2CC2C)=O)C(C)(C)C)cc1F 11502,C(=O)(C1CCCc2ncccc21)NC(CCCCOC)C 11503,Cc1cncc(C(=O)NCC2CC(C)N(C(c3csc(F)c3)=O)C2)c1 11504,C(C(C(=O)NC(C)Cn1ccnc1)NC(=O)C(N1CCCC1C)C)OC(C)C 11505,C(CCCC(=O)NC1(c2cc(C#N)cn2C)CC1)(c1cccs1)OC 11506,C1(NC(C(C(=C)C)(C)O)=O)(CNC(=O)Cc2ccc(Cl)nc2)CC2CCC1CC2 11507,c1(OC)cc(CNCCCNC(=O)CN(C)C(C)C)c(F)cn1 11508,N1(CC(C)OC)CCCC(NC(c2cc3n(n2)CCO3)=O)C1C 11509,C(C)(C(CC(=O)NCC1CC(CF)C1)NC(=O)C(C)NC=O)OC 11510,C12(CNC(c3c(OC)noc3C)=O)CCCC1N(C(=O)C(C)NC(C)=O)CC2 11511,c1(N2CC3CCN(C)CC3C2)nc(=NCC2(CC#N)CCC2)[nH]c2cccnc12 11512,CC1(C2(C)CC2C(N2CCCC(n3cc(CCS(N)(=O)=O)nn3)C2)=O)CC1 11513,C12(NC(=O)CC=CCNC(=O)C(O)c3ccsc3)CC(CO)(C1)C2 11514,CC(C)(CCNC(=O)CSS(C)(=O)=O)NC(=O)CN.C(C(N)=O)S(C)(=O)=O 11515,c1(C(N2C(C)(C(=O)Nc3cnnc(O)c3Cl)CCC2)=O)cc2ccc(Cl)cc2s1 11516,C1(CNC(=O)COCC2CCCCC2)CC2(CCC2)CN1C(=O)C1=COCCC1 11517,C(=O)(CCCCCNC(C1CC2CC2C1)=O)NC(c1cnc[nH]1)C 11518,c1(NCC(CCC=C)(C)C)[nH]c(=NC(C)c2ccncc2)nc2c1ncn2CC 11519,Cc1nn(C)c(C(=O)NCC(C)CN(C)C(C2CC3(F)CC2C3)=O)c1Cl 11520,N1(C(C(COC(C)C)N(C)C)=O)CCC(CC(C)NC(=O)C(CO)N(C)C)CC1 11521,c1(OC)cnc(C(=O)NC2CC2CNC(=O)CC(C)N(C)C)c(OC)n1 11522,c1(C(N2CC(NC(CN(CC)CC)=O)C(CC(C)(C)C)C2)=O)cc(=O)cc(Cl)[nH]1 11523,c1(NC(=O)Cn2ccnc2)nccc(N2CCCCC2)n1.n1(CC2CC2)cccn1 11524,CC(C)CC(C(=O)N1CCCC1C(C)(C)C)ONC(c1cnoc1)=O 11525,c1(CC)c(C(=O)NC2CCC(C)C2)cnn1CC(C)(C)O.C1(=O)CN(C2CC2)N1 11526,N1(C(C(C)OCC#C)=O)CCC2CN(C(c3cnc(C)nc3C(C)C)=O)CC2C1 11527,Cn1nc(Cl)cc1C(=O)NCCC1CCCN(C(C2(n3cccn3)CC2)=O)C1 11528,C1(C)(CC)CCCN(c2nnc(Cc3ccccc3C)n2CC2CCC2)C1 11529,c1(C(=O)NCCC(C)NC(C2CCCC(=O)CC2)=O)c[nH]cc(Cl)c1=O 11530,Cc1ccc(C(C)(F)F)cc1C(N1CC(CNC(=O)CC=C(Cl)Cl)C2(CC2)C1)=O 11531,CC1(C)CC(=O)OC1CNC(C1C=CCN(C(=O)C=CC2CCOC2)C1)=O 11532,C(CC(O)CC(=O)NC1CCN(C(=O)CCC(=O)N(C)C)C1C1CC1)SC 11533,c1(C(=O)NC2CC3CN(C(C4CC(C)(C)O4)=O)C2C3)ccc(Cl)c2ncccc12 11534,C1(C(=O)NC2C(O)CCN(C(CCNC(=O)NC)=O)C2)CC2CCCCCC12 11535,CCC(C(=O)NCC1(OC)CN(C(=O)CCc2cnc(O)[nH]2)C1)OC 11536,Cc1[nH]c(C(=O)NCc2ccc(F)cc2F)c(C)c1C(=O)NCC1CCCN1C 11537,N1(C(c2c(CC)scc2)=O)CC(C)N(C(c2csnc2OC)=O)CC1C 11538,N1(C(C2(CO)CC2)=O)CCC2CN(C=O)CC2C1.C1(C2CCCO2)(C2CC2)CCC1 11539,c1(CC)ncc(C(=O)NC2CC(F)CN(C(c3ccn(C4CC4)n3)=O)C2)c(O)n1 11540,N1(C(CSC2C(NC(C3C(C#N)C3)=O)CCO2)=O)CCCC2CCCCC12 11541,N1(CC(=O)OCC)CCC2(C1)NC(=O)N(C)C2=O 11542,c1(SC)ccc(C(=O)NCCC(C)NC(C2CCN2C2CCCC2)=O)cc1 11543,C1(CC(=O)NCC2(OC)CN(C(c3[nH]c(C)c(C)c3C)=O)C2)CCCNC(=O)C1 11544,Nc1cc(Cl)nc(Cl)c1C(N1CC2CCN(C(C3CC3(F)F)=O)C2C1)=O 11545,Cc1ccc(C=CC(=O)NCC2(O)CN(C(C3(Br)CC3(C)C)=O)C2)cc1Cl 11546,C1(O)(CNC(CC(CC)c2ccccc2)=O)CCN(C(c2ccc(=N)[nH]c2)=O)CC1 11547,C(=O)(C1CCc2ccccc21)N1CC2C(NC(C(C)OC)=O)(CCC2)C1 11548,C(=O)(CCCCN(C)C(C)C)NC1(CN(C(C(CC)n2cccn2)=O)C)CC1 11549,c1(CNCCCc2nnnn2C)cc(Cl)nc(Cl)c1.C1(CC=C)(OC)CC1 11550,C1(CNCC(c2cccc(F)c2)O)CCc2nncn2C1 11551,C1(CC=C)(C(=O)NC(C)CCC(=O)OC)CCN(C(=O)C(C)=C(C)CC)C1 11552,C1(C(=O)OC)CCc2nc(N(C)C)ncc2C1.C1CC(C)N1C(=O)OC(C)(C)C 11553,N1(C(c2ccc(=NC)[nH]c2)=O)CCC2CC2(NC(c2c(CO)noc2C)=O)CC1 11554,CCC(CC)C(=O)N(CC(C)NC(c1cnn(C(C)(C)C)c1CC)=O)C 11555,C(CC)(CC(C)CC)(c1n(CC(=C)C)nnn1)Nc1cc(CO)ccc1C 11556,c1(C(N(CCNC(c2c[nH]c(=NC)s2)=O)CC)=O)cccc(S(=O)(=O)C(F)F)c1 11557,C1(C)(NC(C=CC(C)NC(COC)=O)=O)CCC(C)=C(C)C1 11558,O=C(CCC(=O)c1cccs1)NCC1CC(F)(CNC(C2CC2(F)F)=O)C1 11559,c1(SC(CCN(C(c2nncn2C)C)C(C2CC(C(N)=O)C2)=O)=O)ccc(F)cc1 11560,C(CCCCCCCCCO)N(c1c(C)nsc1N)C(=O)C(N1CCNCC1)=O 11561,C=CC1CN(C(c2n[nH]c(C)c2C)=O)CC1NC(c1ncoc1C1CC1)=O 11562,c1(C(=O)NC2(CCCNC(C(C)n3cnnn3)=O)CC2)ccc(Br)nc1N 11563,N1(S(CC)(=O)=O)CCC(C(=O)NC(C)CCN(C(=O)CN(C)C(C)=O)C)CC1 11564,N#CC1(C(N2CCCCCC2C(=O)NC2CCC(C(N)=O)C2)=O)CCOCC1 11565,CC1(C)CN(C(C2(C)CCN(C(=O)CC3(O)CCC3)C2)=O)C12CCC2 11566,C(CN(C)N1CCC(COC)CC1)SC.C12=CC=C(c3ccccc31)C2 11567,c1(CN2CCC(C)(C(N3CCC(C4CC4)CC3)=O)C2)ccc(Br)cc1S(C)(=O)=O 11568,N1(C(c2cc(C(C)C)no2)=O)C2CCC1C(NC(c1ccc[nH]1)=O)C2 11569,c1(CC(=O)NCC(C)CNC(C2CCN2S(C)(=O)=O)=O)ccncc1Cl 11570,c1(C(C(=O)NC(CN(C(CNNC(CCC)=O)=O)C)CC)C)ccc(Cl)s1 11571,O=C1Nc2ccccc2CC1CC(N1CC2CC(CO)CC(C2)C1)=O 11572,C(=O)(C(F)C1=CCCCC1)N1CC(C)N(C(=O)C=Cc2cncnc2O)CCC1 11573,CC(C)N=c1[nH]c(=NCc2ccnc(C(N)=O)c2)c2cccc(F)c2[nH]1 11574,C(=O)(CCCCCn1cnnn1)NC(C)(C)CCCNC(=O)CCC1CC1(C)C 11575,c1(C(=O)NCC(CNC(Cc2cn(CC)nn2)=O)F)cc(Cl)ccc1OC 11576,C(=O)(CC1=CCOCC1)NCc1c(CNC(c2ncc(OC)cn2)=O)cccc1 11577,CCCCC(O)CC(=O)NCC1CN(C(=O)CNC(N)=O)CCCO1 11578,c1(C(=O)NC23CCN(C(c4c(OC)n[nH]c4)=O)CC2C3)cnc2cc(C)nn2c1 11579,C1(C(C)C)CN(C(=O)Cc2cnco2)CCN1C(c1cccc(C2CC2)c1)=O 11580,CC12CC(C(=O)NC3CN(C(c4ccc5cnnn5c4)=O)CC3F)(C1)C(C)(C)O2 11581,CCC(O)C(F)(F)C(=O)N(CC(C)(C)Nc1ncnc2[nH]cnc12)C 11582,C(=O)(C1CCc2c(Cl)cccc21)NC1CC2(C(NC(c3cc(=N)[nH]cc3)=O)C2)C1 11583,c1(C(=O)Nc2cncc(Oc3cnc(OC)s3)c2)cc2c(Cl)cccc2s1 11584,CCC(C(=O)Nc1nccc(N2CCC(C)C3(CCC3)C2)n1)C(C)(C)CC 11585,c1(OC)cccc(F)c1C(N1CCC(O)(CNC(=O)CCCCCNC(N)=O)C1)=O 11586,N1(S(=O)(=O)c2c(Cl)cccc2I)CCC(C2CCC3(CC2)OCCO3)CC1 11587,C1(C(=O)NC(C(=O)OCC)C)CCC(C)N1C(=O)C(C)NC(C)=O 11588,N1(C(c2c(C)coc2)=O)CC(NC(=O)C(C)(C)c2cscc2Cl)C(O)C1 11589,N1(C(C2(CNC(c3cccc(F)c3F)=O)CCOC2)=O)CCC2(CC1)N=N2 11590,C(=O)(CC(C)C(F)(F)F)N1CCC(NC(C(COC)(C)C)=O)C(O)C1 11591,c1(C(=O)NC2CN(C(C(C)C)=O)CC2C)cc2ccoc2cc1F 11592,C(N=c1cc[nH]c(=NCCCc2nccs2)[nH]1)C1(C)CC1.c1(C)ccsc1 11593,c1(OC)cc(C)cc(C(=O)NC2CCCC2NC(C2(OC(C)C)CCSC2)=O)c1O 11594,C(=O)(CC(=O)NCCCN(C(=O)Cc1cnn(C)n1)C)OCC 11595,Cc1nc(C)c(C(N2CCN(C3CCCN(C(=O)C=CC(N)=O)C3)CC2)=O)[nH]1 11596,C1(N(C)C)CCOC(C(=O)NC(C)(CNC(c2ccc(C(F)F)s2)=O)C2CC2)C1 11597,C(CC1=CCN(C(=O)CC2CCCCC23CC3)CC1)NC(=O)CCc1cscn1 11598,N1(C(c2ccoc2C2CCC2)=O)CC2(CCN(C(C3(c4cc[nH]n4)CC3)=O)C2)C1 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11669,C1(CC)(CNC(C2C(C(=O)O)C2)=O)CN(C(C2(c3ccccc3)CC2)=O)C1 11670,c1(OC)ccccc1C(CNC(c1c(OC)noc1C)=O)NC(=O)C(O)C(F)F 11671,N1(C(Cn2c(C)cc(C)n2)=O)CCC2C(C1)CN2C(C12CC(C)C1C2)=O 11672,N1(C(CC(CNC(COCCC#C)=O)OC)=O)CCCC2OCCC2C1 11673,c1(C(=O)OCC)ccc2[nH]c(C(=O)Nc3cc(C)nc4nc(C)nn34)cc2n1 11674,N1(CC2N(S(c3c(Cl)cc(Cl)c(C)c3Cl)(=O)=O)CCC2)c2ccc(Cl)cc2CCC1C 11675,N1(C(C2CC(O)(CNC(C3CC4(CCC4O)C3)=O)C2)=O)CCOCC2(CC2)C1 11676,c1(SC)c(C(N2CCC(NC(C3CCC(C)(C)O3)=O)C2C)=O)cnn1C 11677,c1(CNC(C(C2(O)CCC2)NC(c2ccc(CO)s2)=O)=O)ccc(O)nc1 11678,CC1CC(O)CCN(C(=O)CCOCCN(C)C(C2(C)CC2(F)F)=O)C1 11679,C12(C(N(CC(C)NC(C3(CCC=C)CC3)=O)C)=O)C3CCC(CC13)C2(F)F 11680,C1(NC(Cc2nc(C)sc2)=O)C2CC1N(C(C1(Sc3ccccc3)CC1)=O)C2C 11681,C1(C(=O)NCC(CC=C)NC(=O)C(F)(F)c2nccs2)CC2(C1)CC1(CC1)C2 11682,C1(C(=O)NCc2nc(CNC(=O)C(=O)NC3CC3)nc(O)c2)CCC(C2CC2)C1 11683,c1(NC(c2n(CC)nnn2)C23CCCC2C3)ccc(OC(C)C)cc1 11684,CC1(C)CC(NC(c2cccc(CC(F)(F)F)c2)=O)CN1C(=O)CCN1CCC1 11685,C(=O)(C(C)CC(C)(F)F)NC(CC(C)C)(C)CNC(=O)C(F)(F)c1cscn1 11686,CC1CCOC1CC(=O)N(C)CC1CN(C(c2sccc2SC(F)F)=O)C1 11687,c1(C(=O)NC23CCC(NC(c4c(CC)ncs4)=O)(CC2)C3)ccc2sccc2c1 11688,C(=O)(CCCCCO)NCC1C2CN(C(Cc3n(C)cnc3)=O)C1C2 11689,c1(C(N(C2CCN(C(c3cccnc3O)=O)C2)C)=O)ccc2nn[nH]c2c1O 11690,C1(C(=O)Nc2c(C(=O)OC)scc2)CCCC(NC(=O)NC(C)(C)C)C1 11691,c1(OC)cc(C(N2CCN(C(=O)Cc3cncnc3)CC2C(F)F)=O)c(F)cn1 11692,c1(-c2cn(CCCNC(C3CC(C)OC3=O)=O)nn2)ccc(N)c(Cl)c1 11693,CN1CCN(CC(=O)Oc2ccc(NC(C3CCC3)C3CCC3)cc2)CC1 11694,c12cc(co1)C2.N1(CC(=O)NCC(C)NC(C=CCN(C)CC)=O)CCOCC1 11695,C1(C2CCC2)(C(N(CC(O)CNC(c2ccn(C3CCCC3)n2)=O)C)=O)CCC1 11696,C(=O)(CCCCN(C)C)NC(C)C(CO)NC(c1cnc(C(F)(F)F)s1)=O 11697,N1(C(C(c2ccc(F)cc2)CC)=O)CC2C(CNC(c3cnn(CC)c3)=O)C2C1 11698,N1(C(C=C(C)C)=O)CCCC1C(C)(C)C(=O)NCCC(F)(F)F 11699,C(=O)(C(C(C)C)OCCN(C)C)NC(CN(C(=O)C=Cc1csnc1C)CC)C 11700,C=C=CC(C)C(=O)N1CCC(C)(C(=O)N(C)Cc2cnn(CC)c2)C1 11701,c1(C(N2C(CNC(C(CCN(C)C)O)=O)CCC2)=O)c[nH]c2cccnc2c1=O 11702,N1(C(c2cc(C)c(C)[nH]2)=O)CC(C2CCCCN(C(=O)Cc3ccccc3)C2)C1 11703,Cc1ccc2occ(C(C(=O)NCCSC3CCC3)N(CC(F)(F)F)CC#N)c2c1 11704,CC(C)(C)COC(CNC(C1(CC)CC1)=O)C1CCC1.C1(C(=O)N)CC=CC1 11705,C(=O)(CCC(O)C(C)(C)C)N1CCC(CN(C(=O)CN2CCSCC2)CC)CC1 11706,N1(C(COCCC#C)=O)CCN(C(c2nnc(C)cc2O)=O)C2CCCCC2C1 11707,c1(CC)nc(=N)[nH]cc1C(N1CCCCCC1CNC(C1CNC(=O)N1C)=O)=O 11708,N1(C(C2(C)CCOCC2)=O)CCCC(F)(C(=O)NCC(CO)CCO)C1 11709,c1(C(=O)NCCN(C(C2CCOC2C)=O)CC)cc2ccccc2cc1O 11710,CC(C)CCCC(C)C(=O)N1CCC(CC(=O)NCCC2(CO)CC2)C1 11711,N1(C(CCSCC)=O)CCC(NC(C23CCC(CC2)CO3)=O)C(F)C1 11712,C1(CNC(C=C(C)C)=O)CCN(C(c2n[nH]c(C)c2C)=O)C1(C)C 11713,C(c1ccncc1)=C(C)C(=O)N(C1CCCN(C(C2C(C)C2(F)F)=O)C1)C 11714,c1(C(=O)Nc2nsnc2C(=O)NC2CC2)cccc(S(=O)(=O)N2CCOCC2)c1 11715,c1(C(=O)NC(CNC(=O)Cc2ccc(Cl)s2)CO)cc(F)cc2nc[nH]c12 11716,c1(C(=O)NCC(CC)N(C(=O)C(F)C(C)C)C)ncnc(C)c1C 11717,C12(C(=O)NC3COCCN(C(=O)Cc4ccccc4Cl)C3)CC=CCN1CCC2 11718,C1(C(=O)NC2CC(NC(CCOCC)=O)CC2O)CCN(C(=O)OC)CC1 11719,c1(C(=O)NCC=CCNC(=O)C=CC=C(Cl)Cl)cccc(CF)c1 11720,C1(C(=O)N(C)CC2(CNC(c3ccc[n+]([O-])c3)=O)CC2)(OC)CCC(C)C1 11721,C1(NC(CC(OCC)OCC)=O)CC12CCS(=O)(=O)CC2.C12CC(O)CCN1C2=O 11722,CC(C)CC(CO)N(C)C(C1COCC1NC(=O)CC1(O)CCCC1)=O 11723,O(NC(=O)C(COCC)NC(=O)CCC1(C#N)CCC1)CCC=C 11724,c1(C(=O)NCCCCNC(C2(C(=O)OC)C3CCC23)=O)ccc(=O)n2c1CCCC2 11725,N1(C(CCNC(C)=O)=O)CC(C(=O)N(C(C)CO)C)C(F)(F)C1 11726,Cc1ccc(C(=O)NCC(C)CC(=O)NC(c2ncccc2F)C)cc1O 11727,C(CC(=O)NC1(C)CCN(C(=O)C(C)(F)F)C1)(C(N)=O)NC(C)=O 11728,CC(C(O)C(F)F)NC(C1(NC(=O)CC(=O)NC2CC2)CCCC1)=O 11729,c1(OC)ccc(S(=O)(=O)N2CCC(CNC(=O)CC3CCCC3)C2)c(F)c1 11730,N1(C(Cn2ncc(C)c2)=O)CCN(C)C(C(=O)NCC2CC(C)(O)C2)C1 11731,C1(NC(C=C(C)Cl)=O)CN(C(c2c(C)ccn2C)=O)CC1O 11732,N1(C(C2C(C(=O)OC)CCCC2)=O)CC2(CCN2C(c2cnn(C3CC3)c2)=O)C1 11733,N1(C(C(CC)C(=O)OC)=O)CC2(CCC(CNC3CCCO3)CC2)C1 11734,C1(NC(C(CO)OC)=O)CCCN(C(C)C)C1.C12(CC1)C(=O)N2 11735,CC1CN(CC(O)C(Cl)(Cl)Cl)CCC1NC(c1ccccc1)=O 11736,c1(NC(=O)OC)cnc(O)c(C(=O)NCCC2CC2(F)F)c1 11737,C1(C(=O)OC)CCN(CC(=O)NC2CCC(NC(N3CCCCCC3)=O)C2)CC1 11738,C(=O)(C1=CCN(C(c2ccc(O)cc2)=O)C1)NC(C)C(C)(C)c1ccccc1 11739,C(=O)(CC(C)(C)NC(C1(C(C)(F)F)CC1)=O)N(CC(COC)O)C 11740,C1(O)(CNC(c2cc(O)nnc2O)=O)CCCN(C)C1.CCCCCCc1cccs1 11741,c1(C(C)OC(c2ccc(C=CC(=O)OCC)o2)=O)cc2cnccc2o1 11742,c1(CC)nn(C)c(C(N2CCSCC2C(N2CC3CC2CO3)=O)=O)c1Cl 11743,C(=O)(CCC(=O)OC(C)(C)C)NC1CCC1C(NC)=O.CC(C)Cn1cccn1 11744,C(=O)(C1=CCN(C(C2(F)CCCC2)=O)C1)N(c1cnc(F)nc1)C 11745,N1(C(C(C)N2CCC2)=O)CC(CCO)(NC(c2cn(C3CCC3O)nn2)=O)C1 11746,N1(C(C(C)OC)=O)CC(CNC(=O)C(c2ccc(C)cc2)C)C2(CCC2)C1 11747,Cc1cc(C(N2CC(NC(=O)C(F)F)C(F)C2)=O)c(C)n1-c1ccc(Br)cc1 11748,C1(NC(C(C=C)O)=O)CCC(NC(=O)C(C)NC(=O)C(=O)NC)CC1 11749,C(CCCC1CC1)(c1cccnc1)NC(C(n1cc(-c2ccccc2)nn1)C)=O 11750,CCC(O)CC(=O)NC(C)(C(=O)N(C)CC1CCCC2CC12)C1CCC1 11751,CCC(C)(O)C(=O)NCC1(F)CCC(CNC(=O)C=C(C)C)C1 11752,c1(CC(N2CC(NC(CSCCCCCC)=O)(CO)C2)=O)ncn2c1CCC2 11753,CC1Cn2nccc2CN1C(=O)C1=CCCCO1.C12CCCN1C2=O 11754,CCC(CC(=O)NC1CCCCC1NC(=O)CSC1CC1)OC 11755,C1(NC(c2cnc(O)s2)=O)CCN(C(C2CC2C2CC2)=O)C1C(C)(C)C 11756,c1(OCC)cnccc1CNC(=O)CC1CCCN1C(C1C2CCOCC12)=O 11757,c1(C(=O)OC)cnc(C)nc1N1CCC(C)C(NC(c2cnn(C)n2)=O)C1 11758,N1(C(C(C)(C)OC)=O)CC2(CCCN(C(=O)CC3CCCC(=O)C3)C2)C1 11759,c1(C(=O)NCC(CNC(c2c(C)cc(C)nc2)=O)(C)C)ccc2nc(S)[nH]c2c1 11760,c1(C(N2CCOCC2COCC)C(=O)NCCCC)cccc(C(C)(F)F)c1 11761,c1(CC)cc(F)ccc1C(=O)NC(C)C(C)NC(C1(C2CC2)CC1)=O 11762,c1(C(=O)NCC(CNC(C2(CC=C)CCCC2)=O)O)cnc(C(C)C)nc1C 11763,CC1CCN(C(c2n[nH]cc2Cl)=O)C(CNC(c2cc(-c3ccco3)on2)=O)C1 11764,N1(C(c2c(C)nco2)=O)CCc2sc(C(=O)N)cc2C1.N1(CCC2CC2)CCOCC1 11765,N1(CC)CCC(C(=O)NC2CCCCC2CNC(c2cnsc2C)=O)CC1 11766,C(CN=C(NC1CC1)NC1CC2(CC2)C1)N(S(CC)(=O)=O)C.C1CCCO1 11767,C1(C(N(CC2=CCSC2)C)=O)C2CCC(C2)N1C(C1(C)CCC1)=O 11768,N1(C(c2cnn(CCC)c2C)=O)CCC2C(CCCN2C(=O)CC23CC(C2)C3)C1 11769,C(CNC(=O)C(n1ccc(Br)n1)C)(C(C)C)NC(C1(CCC)CC1)=O 11770,c1(C(N(CCN(C(=O)Cc2noc3ccccc23)C)C)=O)nc2c(s1)COCC2 11771,C1(NC(C(C)(C)N2CCC2)=O)CC2(C1)CC2C(N1CCC(O)(C(F)(F)F)C1)=O 11772,c1(C(N2CC(n3cc(C(=O)NCC(C)C)nn3)C2)=O)cc(Cl)cn1C 11773,C(C(=O)NC(C)(C)CC)(C(C)CC1CC(F)(F)C1)N(C(C)(C)C)CCC 11774,c1(C(=O)NC2CCCCC2CNC(C2CC=CCC2)=O)ccc2c(O)n[nH]c2c1 11775,CC1CCC(NC(c2cnc(Cl)[nH]2)=O)CN1C(c1ccc(-c2cn[nH]c2)cc1)=O 11776,C#Cc1cncc(C(=O)NCCC(C)(C)NC(c2cncn(C)c2=O)=O)c1 11777,Cc1cnc(NC(C2CC(C)CN2C(C2CCC(C3CC3)C2)=O)=O)c(C)c1 11778,Cc1ncsc1CN(C(=O)CCn1cc(-c2ccccc2)nn1)C1CC1 11779,c1(C(=O)NC2(CNc3ncc(C)c(NC(C)C)n3)CC2)cc([N+](=O)[O-])ccc1Cl 11780,n1(CC(=O)N(C(C(=O)N2CCCC2)C2CC2)CC)nc(C)nc1C 11781,C(=O)(CCCCCC(C)(C)C)NC(CN(C(C1CC12CCOCC2)=O)CC)C 11782,c1(CC)cnc(C(C)NC(=O)CCSc2cncnc2)s1 11783,C1(C(=O)NCCOCC(C)C)CN(C(=O)CCOC2CCC2)CCC1C 11784,N1(C(c2c(C)nc[nH]2)=O)CC2CC(NC(c3cc(N)ccn3)=O)C(C2)C1 11785,C1(C(=O)NCC2OCCN(C(C(CC)NC(N)=O)=O)C2)Cc2ccccc2N1C 11786,c1(C(N(CC(CC)NC(=O)C(C)S(N)(=O)=O)C)=O)cc(Cl)c(OC)c(Cl)c1 11787,N1(C(C(=O)N(C)Cc2ncc(I)s2)=O)CCSc2ccccc2C1 11788,N1(C(c2cc(C)nc(O)c2)=O)CC(CNC(c2nccnc2Cl)=O)OC(C)(C)C1 11789,N1(C(c2cc(CC)on2)=O)CCCC2(C1)CN(C(c1c(C)noc1C1CC1)=O)C2 11790,Cc1nc(CNC(=O)CC2C=CC(NC(=O)C(O)CC3CCOCC3)C2)sc1C 11791,N1(CCC(C)C)CCOC2(CCN(C(=O)C(=O)NC3CCC4CC4C3)CC2)C1 11792,Cc1ccccc1NC(=O)C(N1CCOCC1CNC(=O)C(C)n1ccnn1)=O 11793,C1(C(=O)NCCC(=O)OCCC)C2CC1N(C(=O)CC1(OCC)CCC1)C2 11794,c1(CC(C)C)cccc(C(N2CCCC2CNC(C2(C)CC2)=O)=O)c1 11795,CCCC(C)CCNC(c1nnnn1CCCF)c1cn[nH]c1 11796,N1(C(C(C)NS(CC)(=O)=O)=O)CC(Cc2cccnc2)C(C)C1 11797,Cc1c(F)cc(C(N2CC(NC(c3ccc(CO)cc3)=O)C(C#N)C2)=O)cc1Br 11798,N1(C(Cc2cn(CC)nn2)=O)CCC(C2(NC(=O)CCC(C)C)CC2)C1 11799,Cc1ccc(=O)n(CC(N2CC(NC(c3cc(C(C)(C)C)n[nH]3)=O)CC2C)=O)n1 11800,N1(C(C(CC=CC)CC)=O)CC(C2CCN(C(=O)CCNC(C)=O)CC2)C1 11801,CCCCCCC(C)C(=O)NCC1CC2CN(C(=O)C(F)(F)C(F)F)CC12 11802,c1(CN2C(CCOC)CCC2)ncc(Br)cc1Br 11803,N1(C(c2c(C)nc(C)[nH]2)=O)CC2CCCC2(CNC(C2(NC(C)C)CC2)=O)C1 11804,C#Cc1cc(C(N2CCCC2(C)CNC(=O)CCCC)=O)cc(C(F)(F)F)c1 11805,C(=O)(C1=CC2CC=CCC12)NCc1scc(CNC(c2cc(C)cc(C)n2)=O)n1 11806,CC(C)CC(=O)C(=O)NC(C(N1CC(CO)CC(C)C1)=O)C1(C)CC1 11807,C(=O)(CS(=O)(=O)C(C)(C)C)N1CC(C(N)=O)(CNC(Cc2c(C)nc(C)s2)=O)C1 11808,Cc1c(C(=O)NCCn2cc(C(=O)NC(c3ncnn3C)C)nn2)ccn1C 11809,C1(C(=O)NCCN(C(CC2C(C)=NOC2=O)=O)C)SC2C=CC1CC2 11810,n1(CC)nc(C(N2CC3CC3(NC(C3CCC(C(F)(F)F)CC3)=O)C2)=O)cc1O 11811,CCC(c1cccc(Cl)c1)=CC(=O)NC1CCC(CNC(C2CNC(=O)N2)=O)C1 11812,C(=O)(C(CC(C)(C)C)NC(c1ccnc(CO)c1)=O)NC1CCC(C)(OC)CC1 11813,C(CN=c1nc2scnc2c(NC2CCC3(CCC3)CO2)[nH]1)Oc1c(Cl)cccc1 11814,C1(NC(COCCCOC)=O)CCCC2CN(C(=O)C=CS(C)(=O)=O)CC12 11815,N1(C(CSCC)=O)CCCC2(CCCN(C(c3[nH]ccc3C)=O)C2)C1 11816,C1(NC(c2c(CC)nn[nH]2)=O)CC=CCC1C(=O)NCC(F)(F)CC 11817,C1(CC(N2C(Cn3cc(CSC)nn3)CC(F)C2)=O)CCCCC1(C)C 11818,c1(C(CN(C2CC(CO)C2)C)O)ccc(Cl)cc1 11819,C#CC(C)(C)C(=O)NC(C1CN(C(=O)C=CCN(CC(F)(F)F)C)C1)C 11820,c1(C(C)(C)C)c[nH]c(C(=O)NC(CNC(C2CCCCO2)=O)CO)c1 11821,c1(C(=O)NCC2CC2CNC(c2ccco2)=O)cc(=O)n(-c2ccccc2F)[nH]1 11822,N1(C(C(C)(C)NS(C)(=O)=O)=O)CC2ON=C(CNC(=O)CC3(CO)CC3)C2C1 11823,Cc1cc(CN2CCC(C)(NC(=O)Cc3cc(C)n(C)n3)C2)c(C)s1 11824,N1(C(c2c(C)nc(C)o2)=O)C2CCC1C(CNC(C1(O)CCSCC1)=O)C2 11825,Cn1cc(Br)cc1C(=O)NC1CC1CNC(c1cncnc1-c1ccccc1)=O 11826,c1(C(=O)NC2CC(CNC(C(C)O)=O)C2)ncoc1C1CC1 11827,c1(C(N2CCC(OC)(CNC(=O)C(N)=O)C2)=O)cc2n(n1)CCCC2O 11828,C1(CC(=O)NC(C(=O)OCCC)C)CC(C)N(C(=O)CC2CCCC(=O)C2)C1 11829,Cc1cc(F)cnc1C(N1CCCC1CCNC(C1(C(F)(F)F)CCC1)=O)=O 11830,N12CCCN(CC1)CC2.c1(CC(=O)NC(C2C=CCC2)C)csc(C2CC2)n1 11831,C(C(COC)CC(=O)N1CCC(C(=O)NCC2(C)CCCCO2)C1(C)C)OC 11832,N1(C(c2c(C)sc(O)n2)=O)CCCC(NC(c2ccnn2C2CCC2)=O)C(F)C1 11833,c1(OCC(N2CCCC(c3cn(CCCCCO)nn3)C2)=O)ncc(Br)cn1 11834,C(=O)(C1=CCCC1C)NCc1cc(C(=O)NCC(C)OCC=C)on1 11835,N1(C(C(CCCC)(C)F)=O)CCC2(CCN(C(c3ccc(CF)cc3)=O)CC2)C1 11836,c1(C(N(C)CC2N(C(C(C)C#N)=O)CCOC2)=O)cccc(Br)c1N 11837,C1(N(C(CC2(COC)CC2)=O)C)CCCN(C(c2c(C)ccn2C)=O)C1 11838,N1(C(CC2=NN(C)C(=O)C2)=O)CCC2CCN(C(c3ccc(F)nc3)=O)CC2C1 11839,CCC(C)(CNC(=O)C(C)CN(C)C)NC(=O)C1=CCC1 11840,C(=O)(C(F)(F)C(O)c1ccccc1)NCC(C)NC(=O)CSC1CC1 11841,C(=O)(C1CCCc2nccn21)N1CC(CC(=O)O)CC12CCC2 11842,C(=O)(C1=C(F)CN(C(C2CCC(C)(C)CC2)=O)CC1)N1CC2(CC(OC)C2)C1 11843,c1(CC(CC)C)nc(-c2cc(C(C)C)ncn2)n(CSc2ccccc2C)n1 11844,CC(Cc1ccc(Cl)cc1)CC(=O)NCC(C)CNC(=O)C(c1cnccn1)C 11845,Cc1ccc(C(N2CCC3CN(C(C4CCCO4)=O)CC3C2)=O)c2ccccc12 11846,N1(C(CN(C)CCO)=O)CCCCC(C2CN(C(=O)CCc3cncnc3)C2)C1 11847,c1(C(N2CC(C)(CC(=O)NC3CC3(C)C(=O)O)C2)=O)ccc(Cl)cc1 11848,N1(C(c2nsnc2O)=O)CC2CCCC2(Nc2cc(O)ncn2)C1 11849,C1(F)(C(=O)OC(C)(C)C)CN(CC(=O)N(CC(F)F)C(=O)O)CC1C1CC1 11850,CC1CCCC(C)N(N(C2CCNCCC2C)c2ccnc(-n3ccnc3)c2)C1 11851,C1(CC(=O)NC(C)(C)CC2CC2)CC(NC(c2ccc(CSC)cc2)=O)C1(C)C 11852,C12(NC(COC(CC)(C)C)=O)CCCCC1N(C(c1ccncc1NC)=O)CC2 11853,N1(C(C(CC)C(F)(F)F)=O)CCC(C2CCN(C(=O)CCn3cnnn3)CC2)C1 11854,c1(C(N2CCN(CC(C)NC(=O)CC34CC(C3)C4)CC2)=O)ccc(F)cc1Cl 11855,CC1(C)CC(CNC(c2cnc(N)cn2)=O)CN(C(=O)CN2CC3CCC2C3)C1 11856,Cc1ccncc1CC(=O)NCC#CCNC(C1(c2cncc(Br)c2)CC1)=O 11857,C(CC)(C(=O)NCC1CC1NC(c1n[nH]c(C)n1)=O)=CC 11858,N(C(=NCCc1cccs1)NCC1CC1)CCC(C)=O 11859,c1(C(N2CC(c3cn(CC(=O)O)nn3)C2)=O)cc(Br)cc(I)c1F 11860,C1(CNC(CC2(C)OCCO2)=O)CCCN(C(c2ncc(Cl)s2)=O)CC1 11861,c1(C(=O)NC2C(NC(CN(C)C)=O)COCC2)ccc(F)c(NS(C)(=O)=O)c1 11862,C=CCC(CC)C(=O)NC1(C(=O)NC2(CCCCO)CC2)CCN(C)C1 11863,Cc1cncc(CN2CC(C(=O)Nc3ncncc3F)C(F)C2)n1 11864,c1(C(N(C2CN(C(c3cccn(C)c3=O)=O)CC2O)C)=O)cccc2c1CCCC2 11865,c1(C(N2CCCC(CCNC(C(CC)CO)=O)C2)=O)ccc2nonc2c1 11866,C1(CNC(CNC(c2c(C)cno2)=O)=O)CCN(C(c2ccnc(Cl)c2)=O)CC1 11867,c1(CNC(C2CC2F)=O)ccc(CNC(=O)Cn2cc(CO)nn2)cc1 11868,N1(C(CCNC(C(=O)N(C2CCCCC2)CC(C)C)=O)=O)CCS(=O)(=O)CC1 11869,C1(C(=O)NCC2CCN(C(C3CCO3)=O)CC2(F)F)CCC2(CCCC2)CC1 11870,N1(C(CCCC#CC)=O)CCC2(CCC2NC(=O)Cc2ccc(C)nc2)CC1 11871,n1(CCC)c(N(Cc2cccc(C(C)C)c2)CC2CCC2)nnc1-c1cc[nH]n1 11872,C1(CCNC(C(C)N(C(=O)CCC2(C#N)CCC2)C)=O)CCN(c2ncco2)C1 11873,N1(C(COCCCC#C)=O)CCC(C2N(C(=O)C=C(C)C)CC2(C)C)CC1 11874,C(=O)(C1=C(C)CCCC1)NCC12N(C(C(CCCC)O)=O)C(CC1)CC2 11875,C(=O)(C=CS(F)(F)(F)(F)F)N1CCN(C)CC(C(N)=O)C1 11876,c1(CC)oc2ccccc2c1C(=O)NC(C)CCCNC(C1CCCCS1)=O 11877,N1(C(c2c(C)c[nH]c2)=O)CCc2cc(CNC(=O)C(F)OC(F)(F)F)ccc2C1 11878,C1(NC(c2c(CC)cno2)=O)CCN(C(c2cc(F)ccc2F)=O)C1(C)C 11879,CCCC(C(=O)N1CCC(NC(c2ccc(O)c(F)c2F)=O)CC1C)S(N)(=O)=O 11880,CC1OC2CCC1(C(N1CC(=C(F)CNC(c3cc(Cl)cs3)=O)C1)=O)C2 11881,c1(OC)ccc(C(=O)NCC(C(C)(C)C)NC(=O)CCC2CC2C)cc1C(N)=O 11882,C1(C#N)(C(=O)NC(C2CCCC2)CNC(C(C2CCOCC2)C)=O)CC=CC1 11883,C(=O)(CCCCCC(C)(C)C)NCC(CNC(CN1CC(CC)C1)=O)O 11884,C#CCCCC(=O)N1CC(NC(C2(CC#C)CC=CCC2)=O)C(C)C1 11885,C1(CC)CC(S(C)(=O)=O)C1.C1(CC(N2C(C(C)(C)N)CCC2)=O)CCCC(O)C1 11886,C12(C(=O)NCC3C(C(N4CC(CO)(CF)C4)=O)CCC3)CCCN(CC1)C2 11887,N1(C(=O)CC2CCCO2)CCN(C(c2cnc(O)o2)=O)C(c2ccccn2)C1 11888,C1(CNC(C2N(CC)CC2)=O)CN(C(=O)Cn2cc(C3CCC3)nn2)CCCO1 11889,c1(OC)ccc(CC(N)C(=O)NCC2CC(=O)N(c3ccccc3Cl)C2)cc1 11890,C1(NC(C2(CCOC(C)C)CC2)=O)CC(C(=O)NCCF)C1(C)C 11891,C#CC(CNc1cc(NC2CCC(CC#N)CC2)nc(C)n1)CC(C)(C)C 11892,C1(CCNC(c2cn(CC=C)nn2)=O)CCCN(C(=O)CCc2nc[nH]n2)CC1 11893,C1(O)(C(C)NC(COCC)=O)CCN(C(=O)C=C2CCCCC2)C1 11894,c1(OCC)cc(C(=O)NC(C)C=CC(=O)N(CCCOC(C)C)C)[nH]n1 11895,c1(OCC(=O)NCC2(CNC(C3N(N=O)CCC3)=O)CC2)ccccc1[N+](=O)[O-] 11896,c1(N2CCC(C(C)NC(C=COCC)=O)C2)ncc2cccnc2n1 11897,N1(C(CC2OCCN(C(c3c(C(C)C)ocn3)=O)C2)=O)CC2C(=O)NC(=O)C2C1 11898,C1(NC(C2ON=C(CC)C2)=O)CC2CCCC(C1)N2C(c1nonc1N)=O 11899,c1(C(=O)NC2C(NC(=O)CSC3CCCC3)CCOC2)cc([N+](=O)[O-])cnc1O 11900,N1(C(CC(C=C)(C)O)=O)CCC2(CC1)CN(C(c1scc(C)c1C)=O)CC(C)O2 11901,N1(C(C2N(CCC)C(=O)CC2)=O)CCCC(CNC(=O)C(F)(F)CC2CC2)CC1 11902,C1(C(N2CC(OC)(CNC(C3CCCC3SC)=O)C2)=O)C2(CCC2)C12CCC2 11903,c1(CC)ccccc1CN(C(c1cc(CO)on1)C(=O)Nc1ccc(F)cc1)C 11904,N1(C(COCCC)=O)CCCC(C)C1.C(=O)(CCCCc1ccc(F)cc1)NCC 11905,c1(-c2cn(CC(=O)N(CCC)CCN(C)C)nn2)ccc(COC)nc1 11906,c1(COC(c2sc(OC)c(Br)c2)=O)c(F)cc(F)c(F)c1F 11907,c1(C(=O)NC(C2CCN(C(C3(CN(C)C)CCCC3)=O)C2)C)ccc2c(c1)NCC2 11908,N1(C(CCCCC=C)=O)Cc2ccnn2CC(NC(c2nc(CC)sc2N)=O)C1 11909,N(C1CCc2cc(Br)cnc21)C(CNS(c1c(C)cccc1)(=O)=O)=O 11910,Cc1ccc(C)c(CNC(C2CCN(C(=O)Cc3cccc(C#N)c3)CC2F)=O)c1 11911,c1(C(=O)NC2C(C)CN(c3nc(C#N)ncc3Cl)CC2)ccc2ncccc2c1 11912,c1(OC)ccc2c(C(=O)NC(C3CCCCN3C(c3ccns3)=O)C)n[nH]c2c1 11913,C#CCCCCCC(=O)N1CCN(C(c2sccc2C(C)C)=O)C2(CC2)C1 11914,C1(NC(C2CC(CCC)OCC2)=O)CC2CCC(C1)N2C(C1CCOC(C)C1)=O 11915,O(N1CCC(c2ccc(F)c(NC(=O)Nc3cnc(Br)nc3)c2)CC1)CCOC 11916,c1(C(c2cccc(F)c2)NCC(CCCC)CO)ccc(S(=O)(=O)NC)cc1 11917,CC1(C)CC(C(=O)NC(C2CCC(F)(F)C2)=O)(CNC(=O)Cc2cc[nH]c2)C1 11918,c1(C(N2C(CNC(c3n(CC)ncc3)=O)C(C)CC2)=O)ncc(Cl)cc1Cl 11919,CC1(CNC(NCc2ccccc2Br)=NCC2CCCO2)C2COCC12 11920,CC1(C)CC(NC(=O)CC2CCC3CC3C2)N(C(c2csc(Cl)c2)=O)C1 11921,C(CCC(=O)NCC1(C(N2CC(CCO)C2)=O)CC=CC1)=CCC=C 11922,C1(CN(C)C(C2CC(C(=O)N(C)C)C2)=O)CCn2nnnc2C1.C1C(=O)O1 11923,CC(C)CC(F)C(=O)N1CC2CC1(CNC(c1csc3nnsc13)=O)C2 11924,c1(C(N(CC)CC2CCN(C(=O)C(=O)NC)CC2)=O)cc2n(n1)C(C)CCC2 11925,C(=O)(C(F)CCC(C)(C)C)N1C(CNC(C2CN(C)C(=O)C2)=O)C(C)(C)CC1 11926,CCCCC(C(=O)NCCC1(O)CCN(C(=O)C2=CCCC2)CC1)C(C)C 11927,C(=O)(C(C)(C)C1=CCN(C(=O)CC2CCOC2=O)C1)NC(CC=CC)CO 11928,n1(CC(=O)NCC(C)(CNC(=O)COCCC(C)C)OC)nc(C)nc1C 11929,O=C(C1=CC2(CCOC2)C1)NCC1CCN(C(c2cc(=O)cc[nH]2)=O)C12CC2 11930,c1(N2CC(C(C)C)OCC2)nc(N2CCC(C(C)C)CC2)nc2c1SCC2 11931,O=S(=O)(c1cc(Br)cc(Br)c1)N1CCCC12CCCNC2=O 11932,c1(C(=O)NCCC2(O)CN(C(C(CC#C)C)=O)C2)cc(NC(C)=O)cc(Cl)c1 11933,C1(NC(=NCC=C)N)Cc2cccc(C)c2C1.c1(NC(C)C)ccc(OC)c(Cl)c1 11934,C1(C(=O)NCCOCC#C)CCC(CNC(C2(C)CC3CC3C2)=O)CC1 11935,c1(NC(C2CC2C(=O)Nc2cncc(Cl)c2C)=O)cc(CCOC)ccc1O 11936,c1(C(=O)NC(CNC(C2(C#C)CC2)=O)CC(C)C)ccc(Cl)c(C(F)F)c1 11937,CC1(C)CC2(CC(C(=O)NCC(O)CNC(=O)CP(C)(C)=O)C2)C1 11938,S(=O)(=O)(c1ccc2c(c1)OCCO2)N1CC(c2nccc(C)c2)CC2(C1)CCC2 11939,C(=O)(C(CC(C)C)OC)NCC1(NC(C2(CC)CC(C)(C)C2)=O)CCOCC1 11940,N1(C(N2CCC(CCN(C)C)CC2)=O)Cc2ccccc2C(C(=O)O)C1 11941,Cc1cc2sc(C(=O)NCC(C(C)C)NC(=O)C(C#N)C(C)C)cc2s1 11942,CC1(C)CN(C)C(=O)CC(c2ncnn2C)C2=NNC(=N1)S2.c1cccs1.C1CC1 11943,c1(OC)ccc(O)cc1NC(=O)CCC(C)NC(=O)C(C)(C)C(C)O 11944,CCC(O)(CC)CCNC(C1CC(NC(c2c(C)n[nH]c2C)=O)C(O)C1)=O 11945,c1(C(=O)NC(CC=C)CNC(=O)C(C)CC)cccn2c(CC)nnc12 11946,C1(N(C(C2CCC(C(=O)OCC)O2)=O)C)CCCCC1N(C(=O)C1=NOCC1)C 11947,c1(C(N2CC(CNC(c3nc(C)nn3C)=O)C(C)C2)=O)cc(Cl)cc2c1CCC2 11948,C1(NC(C2CC3CCC3C2)=O)CCCC(CC(N2CCC(F)CC2)=O)C1 11949,CC(C)C(Br)C(=O)NCC1CCCC(C2CC2)O1 11950,C1(c2n(CCCSC)nnn2)(Nc2ccc(Br)cc2C)CSC(C)(C)C1 11951,N1(C(c2c(N)cncc2)=O)CC2(CCCC2NC(=O)COCC(F)F)C1 11952,C(=O)(C(C)(C)CCC#N)NCC1CN(C(c2scc(OC)c2)=O)C(C)C1 11953,C12(NC(C(CC#CC)NC(=O)C(COC)OC)=O)CCC(CC1)C2(C)C 11954,c1(C(=O)NC(CN(C(c2ccc(OC)c(F)c2)=O)C)C)csc2c1CCC(C)C2 11955,c1(C(N(C(CC)CNC(c2ccnn2C(C)C)=O)C)=O)cccc(C(C)C)c1 11956,C(CC(C(=O)NC1CC1NC(=O)CC1CC(CC2CC2)C1)c1ccccc1)=C(C)C 11957,c1(N2CCC(NC(c3cccc(Cl)c3)=O)C(O)C2)ncnc2ccc(O)cc12 11958,N1(C(c2cccc(NC)n2)=O)CCC(C)(C)C1C(=O)NOCCC(F)F 11959,c1(C(N2CCC(NC(c3nn(C)c(Cl)c3)=O)C2)=O)c(F)cncc1Cl 11960,C(=O)(C(O)CC(F)(F)F)N1CC(CCCCNC(c2ccc([N+](=O)[O-])o2)=O)C1 11961,c1(C(=O)OC)ccccc1C(N1CCCC(CNC(C2(CCF)CCC2)=O)C1)=O 11962,C(=O)(CCCCCC(C)C)N1CC(CC(N2C(CC)CCC(C)C2)=O)OCC1 11963,c1(OC)nc(N2CCCC(C(C)NC(C34CCCC(CO3)C4)=O)C2)ncc1Cl 11964,C1(C(=O)NC2CN(C(c3c(C(C)C)ocn3)=O)CC2C)CCC2(C1)CC2(F)F 11965,CC1(C)CN(C(=O)CC(F)(F)Cl)CCC1NC(c1ccc(C(F)(F)F)s1)=O 11966,N1(C(C(C)(C)N(C)C)=O)CCC(C2CCN(C(c3cn(C)nc3C(F)F)=O)CC2)C1 11967,CC1(C)COCC1CC(=O)NC1CCC=CC1C(=O)NCCc1nccc(O)n1 11968,c1(C(=O)NC2CC3CN(C(c4ccc(F)s4)=O)CC23)cccn2cncc12 11969,C(=O)(C1=CCC(C)CC1)N1CCN(C(c2ccc(C)cc2F)=O)C(C2CCC2)C1 11970,Cc1cc(C)n(CC(=O)NCc2cc(C(=O)NCC(c3ccnn3C)O)co2)n1 11971,c1(CC2N(C(COC(C(C)OCCC(C)C)=O)=O)CCC2)ccc(Cl)c(Br)c1 11972,C(=O)(C(C(C)(C)C)NC(C1CCN(C(C)=O)C1)=O)N1CC(C(CC)CC)C1 11973,C1(NC(c2c(SC)cccn2)=O)COC2(CCN(C(C3OCCO3)=O)C2)C1 11974,C(=O)(C1=CSCCO1)N(CCCNC(=O)Cc1sccc1Cl)CCC 11975,C(C(=O)N1CC(C(=O)NCC2CCC(C)(C)O2)C2(CC2)C1)(C(C)(C)C)OC 11976,C12(C(N3CC(CN=[N+]=[N-])C3)=O)C(NC(=O)C=C(C3CC3)C3CC3)C3CC1C2C3 11977,CC1C(NC(C2CCN(c3nccs3)CC2)=O)CCCN1C(=O)CNC=O 11978,C(C(C(=O)N(C1(C2CC2)CC1)C)NC(C1CCC(=O)O1)=O)N(C)C 11979,C1(C#N)(C(N2CCN(C(C(Cn3c(C)cc(C)n3)C)=O)CC2)=O)CCCC(=O)C1 11980,C1(NC(c2ccccc2OCF)=O)CCN(C(=O)Cc2cnc[nH]2)C2CC12 11981,Cc1[nH]nc2c(C(N3CCCCC(NC(C4(C)CCCOC4)=O)C3)=O)cccc12 11982,C1(C(=O)NCC2(C)CCN(Cc3ccc(C(=O)OC)s3)CC2)CCC2(CCC2)O1 11983,c1(C(=O)NC2CC(NC(CCOCC)=O)C2)cc(NC(=O)OC)ccc1N 11984,Cc1ccc(F)c(OCC(N2CC(NC(C3CCCS3)=O)C3(CC3)C2)=O)c1 11985,C(=O)(C#CC1CCOCC1)N1CCC(C(N2CCCC(CCCC)C2)=O)C1 11986,c1(C(=O)NC(CCCCNC(C(C)=C2CCC2)=O)CO)cc([N+](=O)[O-])cnc1O 11987,N#Cc1ccc(N2CCN(C(=O)C(=O)NC=O)CC2)cc1.C12(CN)CCCCC1C2 11988,N1(C(CCCCC)=O)CCCN(C(c2cc(O)n(C)n2)=O)C(CCC)C1 11989,c1(CC)cccc(C(=O)NCC2CC(NC(c3cc(C4CCC4)on3)=O)C2)c1F 11990,Cc1cc(C(N2CC(C(C)(C)CNC(=O)Cn3cc(C(N)=O)nn3)C2)=O)ccn1 11991,C1(C(=O)NCCS(=O)(=O)N2CCOCC2)CN(C(C2CCCC2)=O)CC1O 11992,C(C(=O)CCC(=O)NNC(=O)N=c1cc(C)n(C)[nH]1)OC(=O)OC 11993,Cc1cc(Cl)c(Br)cc1C(=O)NC1CC(NC(c2c(F)ccnc2Cl)=O)C1 11994,CCC(C)CCCC(=O)N(C(C(=O)NCC1CN(C)CCO1)C1CC1)C 11995,c1(OC)ccc(CCC(=O)N(C(C)CCNC(=O)C=CC(=O)NC2CC2)C)cc1C 11996,C1(O)(C(C)NC(=O)CCCOC2CCCC2)CCN(C(C2CC(=O)N2)=O)C1 11997,C1(C(N2C(CNC(C(Cc3c(C)nc[nH]3)O)=O)CC(O)C2)=O)CC2CCC(C1)S2 11998,Cc1cc(=O)n(CCC(=O)N(C)CCNC(=O)CNC(=O)OCc2n[nH]c(=N)s2)cn1 11999,N1(C(Cn2c(C)ncc2)=O)CCOC(CCNC(C2CC(F)C(=O)N2)=O)C1 12000,c1(C(=O)NC(C)CNC(c2nscc2Br)=O)ccnc(OCCO)c1 12001,c1(C(C)C)c(C(N2CCC(C)(NC(=O)COCC(=O)NC3CC3)C2)=O)cccc1F 12002,C1(C(=O)NCCN(CC(F)F)C)(NC(c2cc(F)c[nH]2)=O)CCN(C)C1 12003,c1(OC)c(N2CCC(NC(=O)Cn3nc(C)oc3=O)C2)ncnc1Cl 12004,Cn1cc(C(=O)NCCC2(NC(C3(C)CCNC3=O)=O)CCC2)c(=O)n(C)c1=O 12005,N1(C(c2c(CC)cns2)=O)CC(O)CC1C(=O)NC(COC)CC 12006,C1(CNC(CCCC)=O)CC2(CCN(C(=O)C(C(C)C)OCC)CC2)C1 12007,c1(N(C(C(=O)NC2(CCC)CCNC2=O)=O)CC)ccc(Cl)c(Cl)c1 12008,CCCCCCCCC(=O)NCC(CO)C1CN(C(=O)C(CC)C(=O)OCC)C1 12009,N(C(=NCc1ccc(C)cc1)NCC(F)(F)C1CC1)C(COC)C 12010,C1(OC)C(OC)CN(C(=O)CC2CC(F)(F)C2)C1CNC(c1c[nH]c(C)c1)=O 12011,C1(NC(Cc2c(C)scc2)=O)COC2(C1)CN(C(c1occc1F)=O)C2 12012,C1(OC)CC2(CCC(CNC(=O)C(=O)NCC3(C#N)CC4CCC3C4)CC2)C1 12013,Cc1cncc(CNc2cncc(NC(=O)C3CC3)c2)c1 12014,C1(OC)CC(CNC(=O)C=Cc2ccnn2C)N(C(c2cc(C)on2)=O)C1 12015,c1(C(=O)NC(C2CN(C(CC(C)SC)=O)C2)C)ncnc(C)c1C 12016,C(=O)(C(=O)CC(C)C)N1CCC(C(N(CCNC(C(C)SC)=O)C(C)C)=O)CC1 12017,C1(C(=O)NC2CC(CCNC(c3cc(F)c[nH]3)=O)C2)CC12CCOC2 12018,C12(C(N3CCCC(N(C(c4cncs4)=O)CC)C3)=O)CCC(CC1)CC2 12019,N1(C(c2cc(C)c(C)o2)=O)CCC(CCNC(c2csnc2C)=O)C(F)(F)C1 12020,CC(C)(C)C(C(=O)NCC(O)CF)NC(c1ccc(CC#N)cc1)=O 12021,C1(c2cn(CC3CCC(C(N)=O)O3)nn2)CCCCN1C(=O)CSc1cccnc1 12022,c1(C(C(F)(F)F)NC(C(=O)NC2C(CC=C)CCC2)=O)ccc(OCC#N)cc1 12023,c1(C(=O)NCC(C)(C2CC2)NC(C2N=C(C)SC2)=O)cc(-n2ccnc2)ccn1 12024,C(=O)(C#CC1CCCCC1)N1CCCCC(NC(c2c(SC)cn(C)n2)=O)C1 12025,N1(C(CSCC=C)=O)CC2(CNC(C3(C)C=CCC3)=O)CCC1CC2 12026,c1(C(F)(F)F)nc2n(n1)CC(N=c1ccnc(NCCN3CCCCCC3)[nH]1)CC2 12027,c1(C(N2CCC(CC=C)(NC(C3CSCCS3)=O)C2)=O)c(F)cc(F)c(O)c1F 12028,CC(CC(C)(C)C)C(F)C(=O)N(CCCN(C)C(C1CNC(=O)N1C)=O)C 12029,C1(NC(c2ccc(Cl)c(F)c2F)=O)CCC2(CC1)CN(C(=O)CC1CSC1)C2 12030,c1(NC(CCOC)=O)ccc(S(=O)(=O)N2CCCC(C(=O)O)C2)cc1 12031,CC(CC(=O)NCC1CC1[N+](=O)[O-])S(=O)(=O)c1ccc(F)cc1 12032,C(=O)(C1CCc2nccn21)NCCN(C(c1cccc(CC)c1)=O)C 12033,Cc1cc(C(=O)NC(CNC(c2ccc(CC(N)=O)cc2)=O)C2CC2)ncn1 12034,c1(C(=O)NC(C=CC(=O)NC2(C)CN(C(C)=O)C2)C)ccc(F)c(Cl)c1 12035,c1(C(N2CC3(C(NC(C4CCC(C)CC4)=O)CC3)C2)=O)cnc2ncc(Cl)cn12 12036,Cc1nncc(C(=O)NC(c2ncsc2C)C)c1C 12037,N1(C(C2=CCCN(C(C3CCC(C)O3)=O)C2)=O)CCCC(C2(C)CC2)C1 12038,c1(CNC(=NCCCN(C)C)NC2CCC2)ccc2o[nH]c(=N)c2c1 12039,C1(CNC(=O)OC)CCCN(C(=O)Oc2ccc(-n3cnnc3)cc2)CC1 12040,c1(C(N2CC3C(C2)N3C(c2cc(Cl)ncc2Cl)=O)=O)cc(Cl)c(Cl)cc1F 12041,N1(C(CC2(OCC)CCC2)=O)CCSCC1CCNC(C1(C)CCCC1)=O 12042,c1(C(=O)NCCCOCCNC(c2c(C)ccnc2O)=O)cc2c[nH]cnc-2n1 12043,C1(C(=O)NCC(C)CC(=O)N2CCC(CC(N)=O)CC2)CCC(=O)N(C)C1 12044,C(=O)(C(C(C)(C)C)OC)NCC(CC)(C)NC(=O)CSC(F)F 12045,N1(C(c2nncc(OC)c2)=O)CC2ON=C(CNC(=O)COCP(C)(C)=O)C2C1 12046,N1(C(Cc2scc(C)c2)=O)CC(CNC(C2CC(=O)N(O)C2)=O)CC(C)C1 12047,C(C(F)(F)CNC(=O)C(c1cc[nH]n1)N(C1CCC1)C)OCC 12048,n1(C(=O)NC2CC2NC(C2CC2F)=O)c(=O)c(F)cn(C2CCC2)c1=O 12049,c1ccc2cc(CN3CC4CN(CC56CCCCC5OCC6)C4C3)ccc2c1 12050,C1(CC(=O)NC)CN(C(C2(SC)CC2)=O)CCN1C(c1nccc(OC)c1F)=O 12051,c1(C(=O)NC2C(NC(COC(c3nccn3C)C)=O)CCC2)cccc[n+]1[O-] 12052,N1(C(CCCC)=O)CCC(CNC(=O)CC(C2CC2)NC(=O)NC)(OC)C1 12053,c1(C(N2CC(CNC(C3C(C)OCC3)=O)OCC2)=O)ccc(O)c(Cl)c1 12054,N1(C(CC=C)=O)CC(C(=O)N(CC2=CCSC2)C)C2(CCC2)C1 12055,C1(NC(C(C(C)C)NC=O)=O)C2CC3C1C3C2C(N1CC(C(N)=O)(CF)C1)=O 12056,c1(C(N2C(C(C)NC(C(C)=CC)=O)CCC2)=O)ccc(CO)cn1 12057,c1(C(=O)NC2CC(CCC(=O)OCCC3CC(F)(CF)C3)C2)c[nH]cc(Cl)c1=O 12058,c1(OC)cccc(CCC(=O)N(CCCCCNC(=O)C(C)(C)OC)C(C)C)c1 12059,N1(C(C2(c3nc(C)on3)CC2)=O)CCCC(CNC(c2scc(C)c2C)=O)C1 12060,CC1(C)C2CC(C(=O)NC3CCN(C(c4ncccc4Cl)=O)CC3CO)CC12 12061,N1(C(C2CC(NC(C=C(C)C3CC3)=O)C2(C)C)=O)CCN2CCCC2C1 12062,n1(CC(=O)N(CCCSC)CCn2cc(C3(O)CC3)nn2)cc2ncccc2n1.CO 12063,c1(C(C2CNCCO2)CN(CC(=O)O)C(C)C)ccc(C2CC2)cc1Cl 12064,C1(O)(C(C(=O)NCc2ccccc2)NC(C2CS(=O)C2)=O)CCCCC1 12065,C1(C(=O)NC2CC(CC)C2)C(OC)CCCN1C(c1ccc(C)c(C2CC2)c1)=O 12066,CC1CCc2c(COC(C3CC3c3ccccc3Cl)=O)n[nH]c21 12067,CC(C)C(CNC(C1(C2CCCO2)CCC1)=O)C(c1ncoc1C(C)(C)C)=O 12068,CCCS(=O)(=O)C(C)C(=O)NC1CC(CNC(C2CN(C)CCN(C)C2)=O)C1 12069,c1(C(N2CCC3(NC(=O)CNS(=O)(=O)C4CC4)C(C2)C3)=O)n[nH]c2c1CCCC2 12070,C1(CNC(CCc2cc(C)no2)=O)CCN(C(c2cc(Cl)c(Cl)n2C)=O)CC1C 12071,N1(C(Cc2c(C)n[nH]c2C)=O)CC(NC(C2CC2c2ccccn2)=O)CC(C)C1 12072,c1(C(=O)C)cccc([N+](=O)[O-])c1.N1(C(C(=O)NC)C2CCC2)CCOCC1C1CCC1 12073,CCC(CNC(C1C(C)CN1C(c1cscc1C)=O)=O)CCO 12074,C1(C(=O)NC(C2CN(C(=O)C=Cc3cocn3)C2)C)(CO)CCCO1 12075,C1(C(=O)NCC(=C)F)COC2(C1)CN(C(=O)C(C)OC)C2 12076,c1(C(N2CCCC(CCNC(CCC(C)OC)=O)C2)=O)ccnc(C)c1C 12077,C1(NC(C2CCCSC2)=O)CC2(CCN(C(C3(F)CC=CCC3)=O)CC2)C1 12078,C(=O)(C1=NN(CCO)C(=O)CC1)NC(C(C)C)CNC(c1ccc(CO)cn1)=O 12079,n1(CCC)cc(C(=O)NCCN(C(=O)CC2OCCC2C)C(C)C)nn1 12080,c1(C(=O)NC(CC)CN(C(=O)C(C)SC2CCCC2)C)ccc([N+](=O)[O-])s1 12081,N1(C(C(C)(CO)OC)=O)CC23CCCCC2(C1)CN(C(=O)C(O)CC(N)=O)C3 12082,C(=O)(C1CCCc2sccc21)N1CC(CNC(c2ccc(C(C)(C)C)cc2)=O)C1 12083,c1(C(N(C2CN(C(CCCN(C(C)=O)C)=O)C2)C)=O)ccc([N+](=O)[O-])s1 12084,C1(NC(C2(C)CC(=C)C2)=O)CC(OC)CN(C(=O)CCC(=O)c2ccc[nH]2)C1 12085,Cc1nc2cc(C(=O)NC(C)(C)CN(C(=O)CC3CCCC3C)C)ccc2o1 12086,C=CCC(C(=O)NCC1C=CCCC1)NC(=O)C(c1ccnn1C)C 12087,Cc1cc(C(=O)NC2CC(C(C)NC(C3CC3C#N)=O)C2)c(F)cc1Cl 12088,c1(CC)cc(C(=O)N(CC(CC)NC(c2cc(N)c(F)cn2)=O)C)cc(O)n1 12089,C1(C)CC(F)CN1C(c1c[nH]nc1C)=O.C1(N(C)OCC)CC(CNC=O)C1 12090,C1(CC(C)C)CCC(N=c2ccc(Br)c(S(=O)(=O)NCc3cccnn3)[nH]2)CC1 12091,N#CC1(CC(N2CC=CC2CNC(C2CCCCS2)=O)=O)CCCCC1 12092,CC1CCC(CC(N2CC=CC2C(=O)N(C)CC2CCC(=O)N2)=O)OC1 12093,C1(NC(C23N(C(CSCCOC)=O)CCC2C3)=O)CN2CCC1(C)CC2 12094,C(=O)(C(C)(C)CO)NCC(CCNC(Cc1n(C)ncc1)=O)O 12095,N1(C(c2c(CCC)nco2)=O)CCCCC(CNC(C2CCCC(CF)C2)=O)C1 12096,N1(C(CCn2c(C)cc(C)n2)=O)CCC2CC1CN2C(C1CCCS(=O)(=O)C1)=O 12097,Cc1cc(C)n(CC(=O)NCC(O)CNC(=O)CCc2c(C)n[nH]c2C)c(=O)n1 12098,C(CO)(CC(C)CC)NC(CN(C(C(C=C)C)=O)CCOC)=O 12099,c1(CCC(N2CCCC(N(C(C#CC(=O)NC)=O)C)C2)=O)c(C)ncnc1O 12100,N1(C(CN(C(CO)C(C)(C)CO)C2CC2)=O)CC2C=CC1C(NCC)C2 12101,N1(C(=O)CCOc2ccc(F)cc2)CCN(C(=O)Cn2ncnn2)C2CCCC12 12102,c1(C(N2C(C(C)(C)NC(C3CSCCS3)=O)CCC2)=O)ccc(O)nn1 12103,CN1CCC(C(=O)NCC=CCC(=O)NC2(C3CC3)CCCC2)CC1=O 12104,C1(CNC(C)=O)CCCC1NC(c1csc(-c2cnn(C)c2)n1)=O 12105,Cc1ccc(F)c(N)c1C(N1CC(NC(C2CC3(CC3)CO2)=O)C(C)C1)=O 12106,Cc1sc(C)c(C(N2CCC(C)C(NC(c3cnc[nH]3)=O)C2)=O)c1C#N 12107,c1(C(C)C)nc(-n2cccc2)sc1C(=O)NCC1COCC1NC(=O)CC(F)F 12108,CN(C)S(=O)(=O)N(C)CC(=O)NC1CC(O)CN(C(c2ccc(Cl)cc2Cl)=O)C1 12109,c1(C(N(CCCN(C(C2(C(=O)OC)CC2C)=O)C)C)=O)ccc2nccn2c1 12110,N1(C(c2[nH]cc(CC)c2)=O)C2CCC1CC(c1cn(CCN3CCCC3)nn1)C2 12111,Cc1occc1C(=O)NCc1cn(C(c2ccccn2)C)nn1 12112,Cc1[nH][nH]c2ncnc(=NC(=O)c3ccn4c(-c5ccc(C#N)s5)cnc4c3)c1-2 12113,c1(CCC)nc(C(=O)NC(CN(C)C(c2ccn(CCF)n2)=O)CC)cs1 12114,CS(=O)(=O)c1ccccc1CNCC1CC2CC1CC2(F)F 12115,N1(C(c2ccc(Cl)cc2F)C(=O)NCC2CC2)CC=C(c2ccccc2F)CC1 12116,C(=O)(CC1COc2ccccc21)NCC1C(NC(CC2(C=C)CCOCC2)=O)C1 12117,c1(C(=O)N(C2CC(CCNC(c3cnn[nH]3)=O)C2)C2CC2)cnc(C2CCC2)s1 12118,c1(N2CCC(CNC(=O)C(=O)NC3CCCC3O)C2)cccc2n[nH]cc12 12119,C(C(=O)N1CCC(C(=O)O)C(O)C1)(C(C)(C)C)n1cc(CC(=O)OC)nn1 12120,C(=O)(C(CC)n1cccn1)NCC1(CNC(CSCCC)=O)CCC1 12121,N1(C(C(CCSC)O)=O)CCC(CNC(=O)Cc2cnccn2)CC1C 12122,c1(C(=O)NCCCOCCNC(c2ccccc2C(F)F)=O)ccc(F)cc1Cl 12123,CC1CN(c2cc(-c3ccccc3)ncn2)CCC1NCC1CCC2CC2CC1 12124,C1(C(N2CC(NC(C3CC(=C)C3)=O)C(CC3CC3)C2)=O)CCn2c(O)nnc2C1 12125,C1(CC(=O)OC)CS(=O)(=O)CCN1C(=O)C(=O)N=S(C)(C)=O 12126,c1(CC)ccc(C(=O)N(CCCNC(=O)CN2CCNC(=O)C2)CCO)c(Cl)c1 12127,C1(NC(c2cccc(F)c2)=O)C2CN(C(c3cccc(OC(F)F)n3)=O)CC12 12128,CC1(C(N2CCC(CCNC(=O)CCSc3ccccc3)C2)=O)CCC(O)CC1 12129,Cc1noc(C)c1CNC(C1CCN(C(C2CCC(O)C2)=O)CC1)=O 12130,C1(NC(=O)COc2cccc(I)c2)CCCC12CN(C(c1cc[nH]c1)=O)C2 12131,C12(NC(CCN(C(=O)CN3CCC(C)C3)CC=C)=O)CC=CC(C1)OC2 12132,C1(CNC(CCC(=O)NC2CC2)=O)CCC2CN(C(C3(C4CC4)CCC3)=O)CC12 12133,C(c1ccc(NC(=O)OC(C)(C)C)o1)=NC(N(C(CO)CO)C)=O 12134,N1(C(CCCC)C(=O)NCCCCCn2ccnc2)CCN(C)C(C2CC2)C1 12135,CCC(C(=O)OC)C(=O)NC1CC(C(N2CC=CCC2)=O)C12CCC2 12136,N1(C(c2cn(C3CC3)cn2)=O)CCC2(C1)CN(C(C1CC=CC(O)C1)=O)C2 12137,N1(C(C23N(C(c4cn(C)c(=O)cn4)=O)CCC2C3)=O)CC2CC1C(F)(F)C2 12138,CC1CCC(NC(=O)C(N(C)C)S)CN1C(=O)CCC1CCCO1.C(C(F)(F)F)N 12139,c1(NC(N2CC(NC(N3CCCCC3)=O)C(F)C2)=O)ccc(F)c(C(F)(F)F)c1Br 12140,C12(CCNC(C3OCCN(C(C)=O)C3)=O)CCC(CC1)N(C(c1cnoc1)=O)C2 12141,C1(CC(=O)NCC(=O)N(c2nncn2C)C)C2CN(C(c3ccccc3O)=O)CC12 12142,c1(-n2c(C(C)CC3CC3)nc(C3CSC3)n2)ccc(F)c(Cl)c1 12143,C=C(C)C(C)(C)C(=O)N1CC(O)(CNC(C2CC2c2ccc(Cl)c(Cl)c2)=O)C1 12144,N1(C(=O)NC(Cc2cc(OC)cc(F)c2)C)CCC2(CCC(C#N)CC2)C1 12145,N1(C(C(CCC)C#N)=O)CC2CCC1C1CN(C(c3ccc(SC)s3)=O)CC21 12146,C(=O)(C1=CC2(CCOC2)C1)NC1C(C)CCN(C(C2(C#N)CCC2)=O)C1 12147,c1(C(c2n(CCOCC)nnn2)NCC2(C(C)C)CC2)cccc(OC)n1 12148,N1(C(CC2N(C(c3cnc(C)s3)=O)CCC2)=O)CC(C)CC(C)(C)C1 12149,N1(C(c2c(CNC(c3cnc(CC)s3)=O)ocn2)=O)CCCN(C)CC1 12150,c1(C(=O)NCC(N(C(Cn2ncc(CC)c2)=O)C)C2CC2)cnc[nH]c1=N 12151,c1(NC(c2cc(C)cc(Cl)n2)=O)ccc(C(N)=O)cc1C#N 12152,N1(C(c2c(CCC)[nH]cc2)=O)CC2CC(C1)N(C(=O)Cc1cc(O)nnc1O)C2 12153,c1(CC)nc(Cl)cc(=NCC(C)NC(=O)C(C2CC(F)(F)C2)O)[nH]1 12154,N1(CC(=O)CS(=O)(=O)CC2CC2)CC23COCC2(COC3)C1 12155,c1(C(C(=O)NCC(F)F)N(C)Cc2c(CC)ocn2)ccc2cc(OC)ccc2c1 12156,c1(C(C(=O)N(C2(COC)CCN(C(=O)C=CC(N)=O)C2)CC)=O)ccc(F)c(C)c1 12157,CS(=O)(=O)c1ccc(NCCCC2CN(C(C3CC34CC4)=O)CCO2)nc1 12158,C1(C(=O)NC(CCC)CCC)CCCCN(C(=O)CCc2cc(C)no2)C1 12159,c1(C(=O)NCCCOCCNC(c2cc(CCC)[nH]n2)=O)nccn2nccc12 12160,c1(C=O)ccccc1NC.C(=O)(C(C)(C)OCC)NCCN(C(CS)=O)CC#C 12161,N1(C(c2c(CC)noc2)=O)CCC2(NC(c3occ(C)c3C)=O)CCCCCC12 12162,C1(C(=O)NC2C(C(=O)NCC3(OCC)CN(C)C3)CCOC2)C2CCC(C2)C1C 12163,C12(C(=O)NC3CCC(NC(CCc4cncc(C)c4)=O)C3)CCC(CO)(CC1)C2 12164,C1(OC(C)=O)(CNC(C2CCN(c3ccccn3)CC2)=O)CCCCC1 12165,C1(N(C(=O)C(C2CCCC2)SC)CCOC)CCN(C(C2CS(=O)(=O)C2)=O)CC1 12166,C1(NC(CCNS(C)(=O)=O)=O)CCN(C2CCN(C(C3CC=CCO3)=O)C2)CC1 12167,Cc1cccc(Br)c1C(=O)Nc1ccsc1C(=O)Nc1c[nH]nc1C#N 12168,c1(NC(C2CN(c3ncnc4ccsc34)CCC2O)=O)ncc2c(n1)CCC2 12169,CC(C(=O)NCCCCNC(C1(CC(F)F)CC1)=O)NC(=O)C1CC1 12170,C(=O)(C(F)CCC)NC(c1ccccc1)CNC(CCOCC#C)=O 12171,N1(C(C(CC)OC)=O)CCC(CC(N2CC(C(C)C)C2)=O)C1(C)C 12172,CC(C)(C)C(=O)N1CCC1CNC(C1CCCCS1)=O.n12cnc(n1)C(=O)NCC2 12173,c1(OC)ccc(C(=O)NC2CCN(C(=O)CO)CC2C)c(CC2CC2)c1 12174,c1(C(=O)NCCN(C(c2c(C)cns2)=O)C)cnc2c(cnn2CC(F)(F)F)c1 12175,CC1(C)CC(NC(C2CCN2C(C2(NC(N)=O)CCCCC2)=O)=O)CO1 12176,C(C(C)C(F)F)NC(CCN(C(C(C)=C(C)C)=O)CCCO)=O 12177,N1(C(CCC(C)C)=O)CC(O)(C2(CNC(c3cccc4ccnn34)=O)CC2)C1 12178,Cc1c(C(=O)N(CC(C)(C)NC(=O)C=CCO)C)[nH]c2c1CCCC2 12179,C(=O)(CC1=NNC(=O)C1)N1CCN(C(c2c(C)oc(CC(C)C)c2)=O)CC1CO 12180,c1(C(=O)OCC(=O)N2CCC2)cc2n(n1)CCCNC2=O.C1(O)CCC1.CCCOC 12181,CC(CF)CC(=O)NCCCC1(NC(c2nccnc2N)=O)CC1 12182,Cc1nscc1C(=O)NC(C1CCN(C(=O)CC2CCCN2C(C)C)C1)(C)C 12183,CC1CC2CN(C(c3c[nH]nc3CNC(C3CCC(C4CC4)C3)=O)=O)CCN2C1 12184,Cc1nc(=NCCOCc2cccc(NC(C34CC(C3)C(C)ON4)=O)c2)[nH]cc1Br 12185,c1(OCC)nc(NC(C(C)NC(c2cc(C3CC3)cs2)=O)C(C)C)ncc1Cl 12186,C1(C(=O)NC2(CO)CN(C(c3ccc(C)c(Br)c3)=O)C2)CCn2ccnc2C1 12187,Cc1cn2cc(C(N3CCN(C(=O)CC(O)C(Cl)(Cl)Cl)CC3)=O)nc2s1 12188,CC(CC(=O)NCC1(C(N)=O)CN(C(=O)CC2CC(F)C2)C1)P(C)(C)=O 12189,[N-]=[N+]=NC1CCN(C(=O)C(C2CCCO2)NC(C2CCC2)=O)CC1 12190,c12ccc(cc1OC)CO2.c1(N(C)CC)ccc(C(=O)N(C)C)c(C)c1 12191,C(=O)(CCN(OC)C(=O)CS(N)(=O)=O)N(CCS(CC)=O)C1CC1 12192,N1(C(c2ccc(C)c(C)n2)=O)CCC2(CCCN(C(c3cn[nH]c3)=O)C2)C1 12193,C12(NC(C(c3cccc(Cl)c3)CC)=O)COC(C)(C1)C2 12194,C(=O)(C1=Cc2cc(Cl)ccc2OC1)N1CC(C)C(NC(=O)C2=CCOC2)CC1 12195,C1(CC)CCC(C(N2CCCC(CNC(=O)C(F)CC3CC3)C2)=O)CC1 12196,C1(NC(c2c(C)n(C3CC3)cc2)=O)(CO)CCCN(C(C2C3COCC23)=O)C1 12197,C1(NC(N)=O)CCCCCC1NC(CCNC(C(C)C)=O)=O 12198,C=C(C)C1CC=C(CNC(=O)C(C2CC3CCC2C3)(F)F)CC1 12199,C1(NC(c2nc(CCC)oc2)=O)CCC(C(=O)NC2C(C)CCC2C)CC1 12200,C1(C(=O)NCC2C3CN(C(C4CCN(C(C)=O)CC4)=O)CC32)CCC2(CC1)CC2 12201,N1(C(C(CCC)OC)=O)CC(C(=O)NCC2=C(C)CCC2)C(C2CC2)C1 12202,c1(CC)cnc(C)c(NC(=O)C(CCNC(=O)CP(C)(C)=O)OC)c1 12203,c1(OC)nscc1C(=O)NC(CO)C(=O)NCc1ccon1 12204,c1(CC)cc2cc(F)ccc2[nH]c1=NCC1(OC)CC1 12205,C(=O)(N=c1cc2ccccn2[nH]1)C1N(Cc2c(C)n[nH]c2)CCSC1 12206,C(CCN=C(NCC(Br)=C(C)C)N1CC(C)S(=O)(=O)C(C)C1)NC(=O)OC 12207,C1(CC(=O)N(CCCCNC(C2CCC(OC(F)F)CC2)=O)C)CC(C)(C)C(=O)N1 12208,c1(NCC(CCCC)NC(=O)OC(C)(C)C)cc(Cl)c(Br)cc1O 12209,N1(C(CC#N)=O)CCC2CCN(C(=O)CCn3ccnc3)CC2C1 12210,C1(C(N2C(C)C(NC(c3cc(C#N)c[nH]3)=O)CCC2)=O)CCc2cnn(C)c2C1 12211,N1(C(C(C2CC2)OCC)=O)CCOCC1CNC(C1CCN1C1CCCC1)=O 12212,C(CC(F)F)(C(=O)NC(c1cccs1)CO)N(C(Cc1cc(C)nn1C)=O)C 12213,c1(SC)ncc(N)c(C(=O)NC2CCC(NC(C3CC3C)=O)C2)n1 12214,N1(C(c2cc(COC)[nH]n2)=O)CCC(C)(NC(c2ccc(C(O)CF)cc2)=O)C1 12215,Cc1oc(Cl)nc1CC(C(=O)NC(=O)CN(C)C)Nc1ccccc1O 12216,C12(C3(C4CCCCO4)CC3)C(C(=O)OC)C3CC1C2C3 12217,C1(C)(CC)CCC(C(=O)N(C(C)(C(=O)NC(C)CCS(C)=O)C2CC2)C)O1 12218,C1(CC)COCC1(c1nnnn1C1CC1)Nc1cnn(CC(C)(C)O)c1 12219,CN1CC(C(N2CCCC(NC(=O)CCCc3ccsc3)C2)=O)CC1=O 12220,C(=O)(C1=C(C)CCCC1(C)C)N1CC(CNC(C(CCCC)(C)F)=O)OCCC1 12221,c1(OC)ccc(C(=O)Nc2sc(SC)nc2-c2ccccc2)cc1 12222,C1(NC(C2C(=C)CC2)=O)C2CC3CN(C(=O)Cc4nn(C)c5ccccc45)C1C3C2 12223,c1(CC(=O)NCC(CCOC)NC(=O)CC2CCNC2=O)cccc(C2CC2)c1 12224,N1(C(C2C(C)(C)OCC2)=O)CCOC(C(N2CC(c3ncccn3)C2)=O)CC1 12225,C(C(=O)N(CCC(=O)N1CCCC1CC1CCC1)OC)(C1CCCC1)OC 12226,Cc1cc(C(=O)NC(C(N2CCCC2CO)=O)C2CC2)sc1C 12227,C1(NC(C=CC=CCC)=O)CCCN(CCCc2cc(C(=O)NC)ccn2)CC1 12228,C1(NC(C(c2ccccc2F)(C)C)=O)CCN(c2nnc(CCO)s2)CC(O)C1 12229,N1(C(C2(C#N)CC=CC2)=O)CCCC(NC(=O)CCCc2ccsc2)C(F)C1 12230,Cc1ccc(OCC(N2CCC2CNC(=O)Cn2nnc(=O)[nH]2)=O)c(C)c1 12231,c1(C(=O)NC2(CC#C)CC2)n[nH]c2c1CN(C(C1CCCCS1)=O)C2 12232,C1(NC(=O)C(=O)N(CCCN(C)C(CC(F)F)=O)C)CCOCC1 12233,C1(CNC(COC)=O)CC2CCC1N2C(c1cc(C)cc(C)n1)=O 12234,N1(C(C2(CC)CCCC2)=O)CCOC(C)(CNC(=O)CC2CC(=O)NC2=O)C1 12235,Cn1c(C2CC2)nnc1C1CCCN(Cc2nc(C3CCC(N)C3)no2)C1 12236,N1(C(C(=O)NCCNC(=O)CCOCCOC2CC2)=O)CCC(O)C(F)(F)C1 12237,CCCCC(C(=O)N1CCCC(F)C1)NC(=O)CSCC(F)F 12238,S(=O)(=O)(c1cnc(Cl)cc1C)NC(c1ccc(OC)nc1)C 12239,CCCC(CC)C(=O)NCC1(F)CC(NC(c2cc(O)ncc2Br)=O)C1 12240,c1(C(=O)NC(CCCCNC(c2cccc(CC)n2)=O)C)cccc2occc12 12241,Cc1cc(C(=O)NC2CC(CCC(=O)NC(C(F)(F)F)C3CC3)C2)n[nH]1 12242,N1(C(CN2CCC(OC)C2)=O)CC2(CCN2C(c2ccc([N+](=O)[O-])[nH]2)=O)C1 12243,CC1(CNC(c2cnccn2)=O)CCN(C(c2c(Br)cnn2C2CCC2)=O)C1 12244,S(=O)(=O)(c1ccc2c(c1)CCCC2)N(C1CC2(CCC2)C1C(=O)O)C 12245,C1(NCCN(C(=O)CCS(=O)(=O)NC)CC)CCC2CN(C(C)=O)CC2C1 12246,C1(NC(CC(CC)C)=O)CC12CCC(NC(c1cccnc1C(F)F)=O)CC2 12247,c1(C(=O)NCC(CC)N(C(C(CCC)N(C)C)=O)C)cccc2ccc(C)nc12 12248,c1(C(NNC(c2c(C)cc(=N)[nH]c2)=O)=O)cc2c(F)c(Cl)c(Br)cc2[nH]1 12249,c1(NC(=O)NOCC2(c3cc(Br)no3)CC2)ccccc1 12250,N1(C(c2ccc(CCC)[nH]2)=O)CCCC(CN(C)C(c2ccc(C#N)s2)=O)C1 12251,N1(C(CCC)=O)CCN2C(=O)C(NC(=O)Cc3cnccn3)CC2C1 12252,c1(CC)nc(C)n(C)c1C(=O)NCCOCCNC(=O)CC1CCC2(CCC2)O1 12253,C1(CCC)CN(C(C2CC2OC)=O)CCN1C(c1cnn(CCN(C)C)c1)=O 12254,Cc1ccc2nc(SCC(N3CC4CCN(C(=O)C(C)CO)CC4C3)=O)[nH]c2c1 12255,c1(SC)nc(N2CC3CC2(CNC(C24CCC(CC2)CC4)=O)C3)cc(C(F)F)n1 12256,C(CCC(O)C(=O)NC(CC(CC)C)=O)NC(=O)OC(C)(C)C 12257,N1(C(C2CCC(C)C2)=O)C2CCC1C(CNC(c1sccc1-n1cnnn1)=O)C2 12258,C1(C(=O)NC2(CCCC)CCC2)(CCNC(=O)CCCn2ccnn2)CCCC1 12259,N1(CC(=O)NC(C(=O)NC(C(CC)C)C)CN(C)C)CCCCC1C 12260,N#Cc1ccccc1CCC(=O)NC1CCCN(C(c2ccc(Br)cc2F)=O)C1 12261,C(=O)(C1=C(Cl)CCCC1)N(C(C(=O)NCC1(C)N=C(C)SC1)C)C1CC1 12262,N1(C(C2(CC)CCC2)=O)CCC(O)(CNC(=O)COC2CC(F)(F)C2)CC1 12263,C(c1cncn1C)=CC(N1CC(C(=O)NC(C)C)(NC(C=C(C)CC(N)=O)=O)C1)=O 12264,c1(-c2cn(C3(C(N(C(C(=O)OCC)F)C)=O)CC3)nn2)ccc(F)c(F)c1 12265,CC1CCOCC1C(=O)O.C12(CCCCC1)CCC(=O)N2Cc1ccccc1 12266,c1(N(CCNC(C(c2ccc(N)cc2)N(CCC)CC)=O)CC)ccccc1Cl 12267,c1(C(=O)NCc2ccc(CN(C(c3c(C)[nH]cc3)=O)C)cc2)cc(N)c(Cl)cn1 12268,CCC(C(=O)NCCOCCNC(c1ccc(N)c(Br)n1)=O)C(C)(F)F 12269,C(=O)(CC(C)C(C)C)N1CCC(C(=O)NC(C(=O)OC)(C)CO)C1 12270,c1(C(=O)NC2CCN(C(=O)C3=COCCC3)CC2O)cnc2ccc(F)cc2c1 12271,c1(C(=O)NCC2(CNC(=O)Cc3nc[nH]n3)CCC2)nc2cnccc2s1 12272,CCC(C)(C)C(O)C(=O)NC1(C(=O)NCC2CCC(C)(C)CO2)CC(O)C1 12273,CCC(C)C(O)C(=O)N1CCCC(CNC(=O)C(CC2CCC2)OC)CC1 12274,c1(C(=O)NCC(C(C)C)NC(C2(C)C=CCC2)=O)cc2cc(F)c(F)cc2[nH]1 12275,C1(NC(COCc2onc(C)n2)=O)CN(C(=O)Cn2cncn2)CC1F 12276,CCC(CC(=O)NC1CC(CCNC(c2cc(Cl)ns2)=O)C1)C(C)(C)C 12277,C(=O)(C(CC)(CC)C(=O)O)N1CCC(Oc2cc(C(=O)OCC)c(OC)cc2)C1 12278,c1(C(=O)NC(CNC(c2cc(C)nnc2)=O)C2CC2)cc([N+](=O)[O-])ccc1N 12279,CCC(CC(F)F)C(=O)N1CC(C(C)(C)C)CC(CNC(=O)CC(C)(C)SC)C1 12280,N1(C(CN(CCCCCC)C)=O)CC(CNC(C2(CO)CC2(F)F)=O)C(O)C1 12281,N1(C(CCc2c(C)ncs2)=O)CCN2C(=O)C(NC(C34CSCC3C4)=O)CC2C1 12282,c1(C(=O)NC2CCN(C(c3c(C)ccnc3C)=O)CC2O)cccc2c1COC2 12283,c1(C(=O)NC2C(CNC(C(CCC)CC)=O)CC2)cc(C)c(Br)c(C)c1 12284,C(=O)(C(F)C(F)(F)F)NC1(CC(=O)NC2CCC(C(=O)O)CC2)CCOCC1 12285,C1(N(C(CCc2c(C)ncs2)=O)C)CC2CC1N(C(c1csc3nnsc13)=O)C2 12286,c1(C(N2CC(C(=O)NC(C=C)CO)C(F)(F)C2)=O)ccc2[nH]ccc2c1 12287,C1(C2CCN(C(C3CCCCS3)=O)CC2)(NC(C(C)c2cccs2)=O)CCC1 12288,N#CC1CCCN(C(=O)C(=O)NCc2cc(O)ncc2Br)C1 12289,N1(C(c2cc(OC)n[nH]2)=O)CC2COCCC2(NC(=O)Cn2ccc(C3CC3)n2)C1 12290,c1(C(N(CC(CC)NC(=O)C(C2CC2)OC)C)=O)cc([N+](=O)[O-])n[nH]1 12291,N1(C(C(C)CC2CC2)=O)Cc2ccccc2CC1CNC(=O)C(C)C(C)(F)F 12292,N1(C(C(F)=CCC)=O)CC2(CCC2)CC1CNC(c1c(C)nn(C(C)C)c1C)=O 12293,C1(C(N(C)CC2CCCN(C(C(C)(C3CC3)OC)=O)C2)=O)CC2CCC(C1)S2 12294,C1(CC(N2CC(COC)(NC(=O)CSS(C)(=O)=O)C2)=O)CCCCC1O 12295,C1(OC)CC2CC(NC(=O)C(CCNC(C3C4(CC4)C34CC4)=O)OC)CC12 12296,C1(OC)CCC(C(=O)N(C(C)(C(=O)NC(C)CCC2CC2)C2CC2)C)CC1 12297,N1(C(C(CC)C)=O)CCC(C)C(NC(c2cc(C(N)=O)ccc2F)=O)C1 12298,C#Cc1ccc(CN2CCN(CC)C(C(C)C)C2)c(F)c1 12299,C=CC1(C(=O)NC(C)CN2CCCC2)CCN(C(C2OCCC2(C)C)=O)CC1 12300,N1(C(CCC#CC)=O)CC(NC(=O)C=CC(c2ccc(F)cc2)=O)CC12CCCC2 12301,N1(C(COCCCC)=O)CCC2(CC1)OCCC2NC(=O)CSc1n[nH]c(O)n1 12302,C1(C(N(C(CC(F)F)C(=O)NCC(F)CO)C)=O)CC2(CC(=O)C2)C1 12303,c1(C(N(C2CCN(C(c3ccc(C4CC4)nc3)=O)CC2)C)=O)cc(N)nc(Cl)c1 12304,N1(C(CCC=C=C)=O)CCCC(O)(CCNC(=O)CCN2CCC(C)CC2)C1 12305,C1(NC(c2ccn(CC(C)C)n2)=O)CCC12CN(C(=O)CCOC1CCC1)C2 12306,CCCC(C(O)C(=O)Nc1cccnc1C)NC(c1c[nH]ccc1=O)=O 12307,C(=O)(C1=CCCC1C)NC1C(CNC(C2CCCN(C(C)=O)C2)=O)COC1 12308,C12(NC(c3cc(C)c(Cl)cn3)=O)CCCC1CN(C(C1CN(C(C)C)C1)=O)C2 12309,CCC(CC)C(C)C(=O)N1CCC(NC(c2cc(O)ccc2F)=O)CC1C 12310,N1(C(C(C)=C2CCC2)=O)CCN(CCCNC(=O)CCNS(C)(=O)=O)CC1 12311,N1(C(COC(C2(CC(C)C)COC2)=O)=O)CC(C)(OC(C(N)=O)C2CCC2)C1 12312,N1(C(CNC(C2C(CCC)C2)=O)C)CCN(C(=O)Cc2ccn(C)n2)CC1 12313,N1(C(C2N(C(c3cc(C)c(O)cc3)=O)CC2)=O)CCc2cc(C#N)ccc2C1 12314,c1(SC(c2cnc(C)s2)c2nccn2C)ccc(C(=O)O)cc1 12315,Cc1nc(Br)ccc1NC(=O)CC1CN(C(=O)CN2CCCC2=O)C1 12316,N1(C(C(C(=O)OCC)F)=O)CCC(C2(NC(c3c(Cl)cnn3C)=O)CC2)C1 12317,c1(OC)cc(CC(N2CCC(NC(=O)C(Cl)=CCl)CC2C)=O)ccc1[N+](=O)[O-] 12318,N1(C(CC=CCC)=O)CCN(C(=O)CN(CC)Cc2ccc(C)cc2)C(C2CC2)C1 12319,C=C(C)CN=C(NCCC1CCCCCC1)NCC1CCC(COC)O1 12320,n1(CC)ncc2cc(C(=O)NC(c3ccccc3)C3CC3)cnc12 12321,C(=O)(C(CC(C)(C)C)OC)NCCN(C(=O)CC1CCC(F)(F)CO1)CC 12322,N1(CC(N2C(C(C)NC(C(CC#C)C)=O)CCC2)=O)CCCCCCC1=O 12323,C1(NC(C2C(=C)C2)=O)CCCCCCC1NC(=O)CCc1cnc[nH]1 12324,c1(C(=O)NCCCCNC(CNS(N)(=O)=O)=O)coc(C(F)(F)F)c1 12325,C(=O)(C(O)C(C(C)C)OC)NC(CN(C(C(CC)N(CC)CC)=O)CC)C 12326,C(N=c1[nH]c(N2CCCC(OCC3CC3)C2)nc(=N)[nH]1)c1n(C)nc(CC2CC2)c1 12327,C1(F)(C(N2C(C)(c3ccc(F)cc3)CCC2)=O)CC2CC1(C(=O)O)C2 12328,C1(N(C(c2c(C)nccc2)=O)C)CN(C(C2CC3C=CC2C3)=O)CC1(C)C 12329,c1(C(N2CC(CN(C3CCS(=O)(=O)C3)C(C)=O)C(C)C2)=O)nc(C)cc(C)n1 12330,Cc1ccsc1CCCC(=O)NCC(CO)NC(=O)CN1CCCC1 12331,C12(CNC(CS(=O)(=O)NC)=O)CCCC1CN(C(c1cc(C)co1)=O)C2 12332,Cc1csc(=O)n1CC(=O)NC1C2CC1N(C(c1scnc1C1CC1)=O)C2 12333,c1(C(N(c2ccc(C)c(C)c2)CCC)=O)ccc2cnccc2c1O 12334,Cc1cnn(C)c1C(=O)NC(C)C(C1CCCCC1)NC(c1ccsc1)=O 12335,C1(CNC(C2N(NCc3cc(CC)nn3C)CC2)=O)CC12CCc1ccccc12 12336,N1(C(C=CC=CC)=O)CC(C(=O)Nc2ccc(C3CCCCC3)s2)CC12CCCC2 12337,N1(C(C2N(C(c3cccc(CC)c3)=O)C3C(C2)C3)=O)CCCC(C)(O)CC1 12338,c1(CCC(=O)NCC2CN(C(COC)=O)C(C)(C)C2)c[nH]c2ccccc12 12339,C(=O)(C1=NNC(=O)C1)N(CCCCCCNC(C(N1CCOC1=O)C)=O)C1CC1 12340,O=C(C1=CC2(CCN(C(=O)CSC3CC3)C2)C1)NCCc1ccc2c(c1)CCO2 12341,CC1CC(NC(c2cn(CCF)nn2)=O)CN1C(=O)CCC(F)F 12342,N#CCCCCCC(=O)NC1CC2CCC1CC2NC(C1CCS(=O)(=O)CC1)=O 12343,C=CC1CCCC(NC(C2CC(C)(NC(=O)C=CC(F)(F)F)C2)=O)C1 12344,N1(C(C)C)CCN(C(c2ccnnc2)C(=O)Nc2ccc(Cl)cc2F)CC1(C)C 12345,C(=O)(CCCC(=O)N1CCC(C(C)NC(=O)CC2CCC(C)(C)CC2)C1)OCC 12346,c1(CCC)ccccc1C(N1CCC(C)C1CN(C(=O)OC(C)(C)C)CC)=O 12347,N1(C(C(C(CC)C)O)=O)C2CCCC1CN(C(C13CCC(C#N)(CC1)CC3)=O)C2 12348,C1(CNC(C(CC(C)C)F)=O)CC2(CC2)S(=O)(=O)N1 12349,Cc1ccc(C=CC(N2CCC3C(NC(C4CCCN4C=O)=O)CC23)=O)cc1 12350,C(=O)(C1=NOC(C)C1)N(C1CN(C(=O)COC2CCC2)CC1O)C 12351,CN1CCC2CN(C(C3CN(C(=O)CCC4CC4)CC3(F)F)=O)CC12 12352,Cc1cccc2c1c(CNC1CC(C(=O)NC(=O)C(O)C(C)C)C1)cn2C 12353,N1(C(CNC(c2cnn(C(C)C)n2)=O)=O)CCN(c2ccc(Cl)nn2)CC1 12354,c1(CC(C)C(=O)Nc2cccc(C(N)=O)n2)c(N)cnn1C.C12CCN(CC1)C2=O 12355,c1(C(=O)NC(CC(C)NC(c2ccc([N+](=O)[O-])cc2)=O)C)cc2c(ccn2C)[nH]1 12356,C(=O)(CCCCCC(N)=O)N1C(C)CC(CC(N2CCCC2C(=O)NC)=O)C1 12357,C(N=c1nc2sccc2c(NCC2CC3CCC3C2)[nH]1)c1c(C)c(Br)cnc1O 12358,c1(CNC(C2N(C(CCC(N)=O)=O)CCOC2)=O)cccc(Cl)c1F 12359,Cn1cc(C(O)C(N2CCC(OCCNC(=O)C(c3cccnc3)O)C2)=O)cn1 12360,c1(OC)cc(C)ccc1OCC(=O)NCCC(C)NC(=O)C(C)S(N)(=O)=O 12361,CC(C)C(C(C)NC(c1c[nH]nc1-c1ccncc1)=O)NC(=O)CSCC(N)=O 12362,N1(c2nnc(C)s2)CC2(C1)SCCC2NC(C1CCc2c[nH]nc2C1)=O 12363,CC1NC(=O)CCC1CNC(=O)CN(C(=O)C1=NOC(C)C1)C 12364,C1(C(=O)NCC(=C)CCNC(=O)C=CCCC)CCC(=O)N(C(C)C)C1 12365,C12(C(=O)NCC3=CCN(C(CSCC(N)=O)=O)CC3)CCCN1S(=O)(=O)CC2 12366,c1(CC(=O)N(CCNC(C(C)OC)=O)Cc2ccccc2)cc(F)cc(Cl)c1 12367,N1(CC)N=C(C(=O)Oc2cc(C)ccc2-c2ccccc2)CCC1=O 12368,N#CC1(C(=O)NC2CC(CNC(=O)C=C(Cl)Cl)C2)CC2(CC2)C1 12369,Cc1c(C(=O)NC(C)(C)CNC(C2(F)CCOC2)=O)[nH]c2ccc(C(C)C)cc12 12370,Cc1cnc(C=CC(=O)NC2CCC(CNC(c3ccnc(C)c3)=O)CC2)[nH]1 12371,N1(C(c2c[nH]ccc2=O)=O)CCC(F)(F)C(CNC(C23CCCC2C3(F)F)=O)C1 12372,Cn1nc(C(N2CC(O)CC2(C)C(=O)NOC2CCOCC2)=O)ccc1=O 12373,C1(CNC(C2CC(C)NC(=O)C2)=O)CC12CCN(C(=O)OC(C)(C)C)CC2 12374,c1(-n2c(C3CCCN(Cc4cccs4)C3)nc(C(C)C)n2)cccc2n[nH]cc12 12375,c1(OC)cccc(N2CC3CCC2C(NC(C2CC(=O)N(C)C2)=O)C3)c1[N+](=O)[O-] 12376,CP(C)(=O)c1cc(C(=O)NCCC2CCCN(C(=O)COC(F)F)CC2)ccn1 12377,c1(C(N2C(CNC(c3cnc(C)[nH]3)=O)CC(O)C2)=O)cccc(C(C)C)c1C 12378,C1(NC(COCCSC)=O)CCCC1CNC(=O)CCC1CCN(C)C1 12379,Cn1cc(C(N2CC3CC3(C(=O)NCC(=C3CCCCC3)F)C2)=O)n(C)c1=O 12380,CCC(C)C(C)(O)CNC(C1CCC(C2CC2)N1C(c1cccc(O)c1F)=O)=O 12381,c1(C(N2C(NC(C3CC34CCCC4)=O)CCC(C)C2)=O)c[nH]c2ncccc12 12382,N1(C(COc2ccc(C)cc2)=O)CC2(CCC2NC2CNC(=O)C2)C1 12383,CC(=O)CCCC(=O)N(C)CC1CCN(C(=O)COCc2ccnc(O)c2)C1 12384,N1(C(=O)COC2CCCCC2)CCC(CNC(C2(F)CC2)=O)C12CCC2 12385,C12(C(=O)NCC(CN(C)C)OC)CC(C(=O)NC)(C1)C2.CCO 12386,C1(O)(CCNC(C)=O)CCN(C(=O)C(Cc2ccccc2)n2cnnc2)C1 12387,c1(CNC(C2CCN(CC(C)C)C2)=O)cccc(NC(C2COC2)=O)c1 12388,C1(CC(=O)NC(CC2CC2)C(=O)N(C2CC2)C2CC2)CNC(=O)O1 12389,CC#CCC(C(=O)NC(c1nc[nH]n1)CO)NC(=O)C(CC1CCC1)OC 12390,C(=O)(C(C)(C)C(C)(C)C)NCC1CCCC(NC(C(C)SC(C)C)=O)C1 12391,C(=O)(N=c1[nH]onc1-c1cccnc1F)N1CCCC(C)C1.CCOC 12392,N1(C(C2(CSC)CCOCC2)=O)CCN(C(=O)C#CC(=O)N(C)C)C(C)C1 12393,C1(CCOC)(NC(c2cc(C(C)C)sn2)=O)CCN(C(C2CSCCS2)=O)C1 12394,C1(CC)C(NC(=O)C=Cc2cncc(OC)c2)CCCN1C(c1cnc[nH]1)=O 12395,c1(OC)ccc(-c2ncc(C(=O)NCC(O)CNC(C)=O)s2)cc1 12396,C1(NC(CSc2n(C)ccn2)=O)CCC2(CC1)CCN(C(=O)CC1CC1(C)C)C2 12397,N1(C(C(CN=[N+]=[N-])NC(=O)COC2CCCOC2)=O)CCn2nncc2C1 12398,CC1OC2(C(=O)NC3C=CCN(C(c4c(F)cccc4F)=O)C3)CCC1CC2 12399,c1(C(N2CC(C)C(CNC(C3(O)CC(F)(F)C3)=O)CC2)=O)ccc2ncccn12 12400,C1(NC(C2CC(C)(C)C2)=O)CC1C1CCCN(C(C2CCC3CC3C2)=O)C1 12401,c1(NC(CCOC)C)ncccc1S(=O)(=O)N1CCCCC2(CCCC2)C1 12402,c1(NC(C(=O)NC2CC(CCC(=O)OCC)C2)=O)c(OC)cccc1Cl 12403,N1(CCNC(C(CC2CCC2)NC(N)=O)=O)CCN(C(C2(F)CC2)=O)CC1 12404,C=CC1(CC(=O)N(C)Cc2nnc(C)o2)CN(C(C2CC(C)(C)CO2)=O)C1 12405,C1(CSC)CC2CC2N1N1CC(NC(=O)OC(C)(C)C)C(C)C1 12406,C(CCOCCCN(C(=O)C1=CCCC1)C(C)C)(C(=O)N(C)CCOC)OCC 12407,C=CC1(C(=O)NC(c2nn[nH]n2)C2CC2)CCN(C(=O)C=CCC)C1 12408,c1(CNC(C2N(C(C(C3CCOCC3)C)=O)CCC2)=O)ncccc1Br 12409,CC1CCC(C)(C(=O)N(CC(C)CNC(=O)C(O)Cc2ccccc2)C)C1 12410,c1(C(N(CCNC(CCC(=O)NCC)=O)CC)=O)ccc(N)cc1Cl 12411,CC1C(NC(c2cccc(CN(C)C)c2)=O)CCCN1C(c1csnc1Cl)=O 12412,c1(NCc2c(C)nns2)cc(Br)ccc1S(=O)(=O)N1CCOCC2COCC12 12413,C1(NC(Cn2c(C)ncc2)=O)CC2CCC(C1C)N2C(c1ccon1)=O 12414,c1(C(N2CC3C(CNC(=O)CSC(F)(F)F)(CC3)C2)=O)cnc2cc[nH]c2c1 12415,N1(C(c2c(CC)nccc2)=O)CCCC(C)(C(=O)Nc2cc(Br)cnc2Br)C1 12416,CON(C)C(=O)CN(C)N1CCOC(C=O)C1.O(C(F)F)CCO 12417,c1(OC)cccc(C(C)NC(=O)NC(C(O)CO)c2ccccc2)n1 12418,CC1CSCCN(C(c2cnn(CCNC(=O)CC3CC(F)C3)c2)=O)C1 12419,CC1CC(CNC(C2(F)CCCOC2)=O)CN1C(=O)CN1CCCNC1=O 12420,C(CC(O)C(=O)N1CCCC(NC(c2cncn2-c2cccc(F)c2)=O)C1)SC 12421,c1(CNC(c2sccc2Cl)=O)ccnc(CO)c1 12422,C1(C(N2C(C(C)NC(c3ccc(Cl)cn3)=O)CCC2)=O)OCC2COCCC12 12423,C1(C(N2CC(c3cn(CCC=C=C)nn3)(C(=O)OC)C2)=O)CC2C=CC1C2 12424,C1(N(C(C(CCC)F)=O)C)CC2CCC(C1)N2C(=O)C(C(CC)CC)OC 12425,CC(C)C(CN(C)C)C(=O)NC(Cc1ccco1)C(=O)NCc1ccncc1F 12426,C(CNC(C1C=CCOC1)=O)(CC(=O)NC1CC1CCOCCO)OC 12427,C(CC(C)(C)C(=O)N1CCC(NC(=O)CC2CCC(C(F)(F)F)O2)CC1)SC 12428,N1(C(C(C(C)C)SC)=O)CCC(C)C(NC(c2cc(C(F)(F)F)n[nH]2)=O)C1 12429,N1(C(c2c(Cl)cn(C)n2)=O)CCC2(CC1)CN(C(C1CCC(C)(C)CO1)=O)C2 12430,C1(NC(c2ccc(C)nc2O)=O)CC(NC(c2ccoc2Cl)=O)C12CCOCC2 12431,CC1COC2(CCC2)CN1C(C1CC2CC1CC2NC(c1cccn1C)=O)=O 12432,C1(CC(=O)NC(C(=O)OC)(C)CO)C2CCCC2N1C(=O)C(C1CCCC1)OC 12433,N1(C(C=CC)=O)CCC2(CC1)CN(C(C1C3CCC13c1ccccc1)=O)CCO2 12434,C(CC(C)C)(C(=O)N1CCCC(NC(=O)C=Cc2cccs2)C1C)NC(=O)OC 12435,C(C(C)(C)CNC(C1(OC)CCC1)=O)N(CCOC)C(c1conc1C)=O 12436,c1(-c2cc(OC)ncc2)nc(C(N2CCC(C(F)(F)F)C2)=O)ccc1F 12437,Cc1nc(NC(C2CC(O)CN2C(c2cc3cn[nH]c3cn2)=O)=O)cnc1C#N 12438,O=C1CN(CC(N2CCC3CC23C(=O)Nc2cnccc2CO)=O)CCN1 12439,CC(C)C(O)C(C)C(=O)N1CC(=C(F)CNC(=O)CN2CCC2)C1 12440,Cn1nc(C(=O)NC2CC(CC(=O)NC(c3ccccc3)(C)C)C2)ccc1=O 12441,c1(C(=O)OCCOC)n[nH]cc1.C1(CN2CCNCC2)CCNC1=O 12442,Cc1cccc(N)c1C(=O)NC1CCC(N(C(=O)CCC2CNC(=O)N2)C)CC1 12443,c1(C(CNC(C2(CCC=C)CC2)=O)NC(=O)C2=CC(C)(C)C2)cc(C)ccc1OC 12444,C=CCC(C(=O)NCCCCNC(=O)C(C(C)(C)C)c1ccccc1)C(C)C 12445,CC1CC(NC(c2cscc2Cl)=O)CCN1C(C1CN2CCC1CC2)=O 12446,C1(C)(CNC(C(C=CC)O)=O)CC(F)(F)CN1C(c1cc(CSCC)on1)=O 12447,c1(C(=O)NCC2(O)CCN(C(CC3C(C)(C)C(O)C3)=O)C2)ccnc2ccnn12 12448,c1(CN(C)CC2CCCN2C(C2CCC(=O)N2C)=O)cccc2cc[nH]c12 12449,c1(C(=O)NCCCC2N(C(c3c(C)ccs3)=O)CCC2)ccccc1OC1CC1 12450,CC1=C(C(N)C(=O)NC(COC(C)(C)C)CN)SC1 12451,C1(C2CC2)(C(=O)NCC(C(C)O)C)CN(C(=O)C(C)n2cnnn2)C1 12452,CC(C)CC(CNC(=O)CNC(c1cn[nH]c1)=O)C(=O)OC(c1ccccc1)C 12453,C1(NC(c2cc(CC)on2)=O)CCCN(C(=O)CC2C=CCC2)C1 12454,c1(C(=O)NCC2N(C(c3c(Cl)cnc(C)n3)=O)CC2)cc(F)c(C)cc1O 12455,C1(C)(C(N(CC(N2CC(N(C)C)C2)=O)C2CCC2)=O)CCCCO1 12456,N1(C(C(C)SCC)=O)CCC2(CC(NC(=O)CSCc3ccc(F)cc3)C2)C1 12457,N1(C(C2C(C)CC2)=O)CCC(C(C)(C)CNC(c2nn(C)cc2Br)=O)CC1 12458,c1(OC)c(C)cc(C(=O)NCC2CCC(NC(=O)C(O)P(C)(C)=O)CC2)cc1C 12459,CC1CCc2nc(Cl)nc(N3CCCCC(NC(=O)C(C)(O)CN(C)C)C3)c2C1 12460,N1(C(C2N(C(C)=O)CSC2)=O)CCC12CN(C(=O)CSC(C)(C)C)C2 12461,C1(CC)CN(C)CCCN1C(C1COCC1NC(=O)C(F)C(C)(F)F)=O 12462,CC(C)CC(=O)NC(c1nocc1C(=O)NCCCC1CCN1C(C)(C)C)C 12463,Cc1cc(C(N2CC(OCC(=O)NC3CCSC(C)C3)C2)=O)n2ncnc2n1 12464,C1(C(N(C)CC2CC(F)C2)=O)CC2C=CC1N(C(C1CC=CC1)=O)C2 12465,C1(CN(CCNC(=O)CSC)CC)CCn2ncnc2C1 12466,N1(C(C2NC(C)C2)=O)CCCC2(CCC2)C1.CC1=C(C=O)CCC1 12467,c1(CC)c(C(=O)NC2CCC(NC(=O)C(N3CCCCCC3)C)C2)cccc1F 12468,c1(SC2CCN(C(C(=O)NCCCCc3ccccc3)=O)C2)ccccc1Cl 12469,C(=O)(C1CCc2snnc21)NCC1CCN(C(C(CCC)NC(N)=O)=O)C12CC2 12470,N1(C(C=CC(C)NCC=Cc2cn(C)nn2)=O)CCCC(C)(N(C)C)C1 12471,N1(C(CCS(=O)(=O)NC)=O)CC2(C1)CN(C(C1CCC3(CC1)CC3)=O)CCO2 12472,C1(NC(C2C3COCC23)=O)CN(C(=O)C(O)C2CC2)C2(CCC2)C1 12473,c1(CCNC(C=C(CNC(CCCOC)=O)C)=O)cccc(C)n1 12474,C1(NC(C2(CC)COC2)=O)CN(C(=O)CN2C(=O)CCC2=O)CC1SC 12475,c1(OC)c(Cl)cc(CN2CC(N(C(=O)Cc3cc(C)ccc3F)C)C2)cc1Cl 12476,N1(C(C=C(CC)CC)=O)CC(NC(=O)C(c2ccc(OC)cc2)C)CC(C)C1 12477,C(=O)(C(C)(C)C)NCC(C)(C)OCCNC(=O)C=Cc1ncco1 12478,c1(-c2n(-c3nc(C)nn3C)nc(CC3CCCC3)n2)ccc(S(C)=O)cc1 12479,CC1CC(NC(=O)C=Cc2ncc[nH]2)CCN1C(c1cc(N)ccc1Cl)=O 12480,C(c1ccc(C)c(Cl)c1)=CC(N1CCC(NC(C2C(C=C)CC2)=O)C(F)C1)=O 12481,N1(CC(=O)N)CCCNC1=O.C1(C(=O)NC(C(=O)OC)C2CCC2)(C)CCCO1 12482,c1(OCC=C)ccc([N+](=O)[O-])c(C(N2CC3CC3(NC(=O)CCCOC)C2)=O)c1 12483,CC(CCc1ccncc1)N=c1[nH]c2c(c(=NCCCCN(C)C)[nH]1)CSC2 12484,N1(C(C=CCOC)=O)CCC(C)C(NC(c2cc(OC)n(C)n2)=O)C1C 12485,CCCCCCCCC(=O)NCC1CCN1C(=O)Cc1ccc(CC)s1 12486,C(=O)(C1=C(Cl)CCOC1)NCCC1CC(NC(C=Cc2c(C)nccc2)=O)C1 12487,N1(C(CC(C)O)=O)CC(CNC(=O)CC2C=CCC2)C(F)(CO)C1 12488,C1(C(N(C(C(=O)NC(c2ccccc2)C#C)C)C)=O)C2CCC(F)C12 12489,N1(C(C=CS(C)=O)=O)CCC2OCCN(C(c3cnc4cccnn34)=O)C2C1 12490,n1(CCCOC)nnnc1C(c1cc(OC)ns1)NC(C)COC 12491,N1(C(CN(C)CC)=O)CC(NC(c2cc(F)n[nH]2)=O)CC1(C)C.C1CS1 12492,c1(NC(C(C2CCN(CC3CCCC3)CC2)C)=O)cc(Cl)ccn1 12493,N1(C(CN(CCC#C)C)=O)CCC(CNC(c2cc(F)cc(F)c2)=O)C(F)(F)C1 12494,N1(C(CCC2(C)CC2)=O)CC2C3CCC(C2C1)N(C(C1CCC(=O)O1)=O)C3 12495,c1(OCC(N2CCC(N(C)C(C3CSCN3C(=O)CCF)=O)C2)=O)ccc(F)nc1 12496,N1(C(c2cc(C)oc2C)=O)CCC(NC(=O)Cc2cc[nH]n2)C(CO)CC1 12497,c1(C(=O)NCC2CC(NC(=O)CSc3ccccn3)C2)cc2ccccc2o1 12498,C1(C(=O)Nc2c(C(N(CC(C)O)CCOC)=O)cccc2)CCOCC1(C)C 12499,C1(NC(c2cc(C)[nH]c2C)=O)CC2CN(C(C34CC(CO)(C3)C4)=O)CC2C1 12500,c1(NC2C3CN(C(CC4CC=C(C)CC4)=O)CC32)nc2cc(C)ccc2o1 12501,CC(C)(CCNC(c1c[nH]nc1Cl)=O)C(=O)NC1C2CCC1CC2 12502,C1(OC)CC(NC(C2CC(C(C)C)=NO2)=O)CN(C(c2scnc2C(C)C)=O)C1 12503,C(=O)(CCCC(=O)NCC1CCCC1NC(C1CC=CCC1)=O)N(C)C 12504,Cc1cc(F)sc1C(=O)N(CC(C)(C)CNC(C1CNC(=O)C1)=O)C 12505,CC1(C(=O)NCC2CCN(C(c3cccc(-c4cscn4)c3)=O)C2)CC2CC2C1 12506,Cc1ccc(CC(=O)NC(C)CCNC(=O)C(C)(C)c2nccs2)s1 12507,N1(C(Cc2c(C)cccn2)=O)CCC(C(=O)NCCCOC2CC2)C(C)C1 12508,C=CCC(CC(C)C)C(=O)N(CC(O)CNC(=O)COc1ccc(F)c(F)c1)C 12509,C#Cc1ccc(C(=O)NC2CC(NC(C3(C)CC=C(C)CC3)=O)C2)nc1 12510,N1(C(C(COC)N(C)C)=O)CCCC(CC(=O)NCCC2CC(C)(C)CO2)CC1 12511,C(C1=NOC2CN(C(=O)Cc3cccc4c3CCC4)CC12)NC(CC(=C)C)=O 12512,CC1CN(C(=O)Cn2ccccc2=O)CC(CCNC(C2CC(F)(F)C2)=O)O1 12513,C(=O)(C(C)(C)C(C)(F)F)NCC1N(C(CC(CC)SC)=O)CCOC1 12514,c1(C(=O)NCC#CCNC(c2cc(CC)nnc2C)=O)cnc2ccnn2c1C 12515,N1(C(c2ccc(C)nc2C(C)C)=O)CCOC2(CCN(C(C3CC3(C)Br)=O)CC2)C1 12516,C1(C(=O)NC2CC(CNC(C3CC4(CCC4)C3)=O)C2)CC12CCCOC2 12517,C1(NC(=O)C=C2CCOCC2)CC2CC1CN(C(C1CCCCC1)=O)C2 12518,CC1(C#N)CCN(C(=O)C(C2(O)CN(C(c3c[nH]nc3Cl)=O)C2)F)C1 12519,N1(C(c2cn(C(C)C)nc2)=O)CCCCCC1N=c1ccc(C#N)n[nH]1 12520,C1(CNC(C(C=C)O)=O)CN(C(=O)CNc2cccc(Cl)c2Cl)CC12CCC2 12521,C(c1ccc(Cl)cc1F)=CC(N1C2CC(CNC(C3(C)C(C)C3)=O)(OC2)C1)=O 12522,C1(NC(COCCSC)=O)COC2C(NC(c3ccc(F)c(N)c3)=O)COC12 12523,C(=O)(C(C)(C)C(C)O)NCCn1cc(C(N(CCCC)CC(C)OC)=O)nn1 12524,c1(COC)ccc(C(=O)NCC2(C)CCC(NC(=O)Cc3cnoc3)CC2)cc1 12525,N1(C(C(CC2CCC2)NC(CCCSC)=O)=O)CC2CCC(C1)C2C#N 12526,C#CCC(C(=O)NCCCSC)NC(=O)C(=Cc1cn[nH]c1)C 12527,C1(CC(C)C)CCN(C(=O)CCOCCN(C(=O)C(C)Cn2ccnc2)C)C1 12528,CN1CCN(C(c2sccc2C(=O)NC)=O)C(CO)C1.C1(C=O)CCCCS1 12529,C(=O)(C(C)S(=O)(=O)C(C)C)NCC(CNC(C(CC)(CC)CC)=O)C 12530,C1(c2nnnn2CCc2ccccc2)(NCC2(CSC)CC2)CCCSC1 12531,c1(C(N(CCNC(C2N(C(C)C)CCC2)=O)C)=O)c(Br)nc2n1CCC2 12532,C1(C)(N(C)C)CCCN(C(=O)C(c2ccnn2C)NC(=O)COC(C)(C)C)C1 12533,N1(C(c2cn(CCC)nc2)=O)C2CCC1CC(CNC(=O)C(C#N)C1CC1)C2 12534,CC1CCCC(N(C)C(c2cc(CNC(=O)CNC(C3CC3C)=O)cs2)=O)C1C 12535,c1(CN(C(c2ccccc2)C(=O)Nc2ccccc2)CC(C)C)ccncc1 12536,c1(C(=O)NC(C(=O)NCc2c(C)scn2)c2ccoc2)cnc(C)n1C 12537,CCCCC(S(=O)(=O)NC(=O)C(c1ccc(Br)nc1)(C)C)c1ccccc1 12538,CC(C)CC(C)(CNC(c1cc(Br)n[nH]1)=O)NC(=O)Cc1cccn1C 12539,Cn1cc(C(F)=CC(=O)NCC2C=CCN2C(=O)CC2CCCC2)cn1 12540,c1(C(=O)NCC2N(C(c3c(C)cncc3)=O)CCOC2)nc(C2CC2)ncc1Cl 12541,N#Cc1ccc(C(N2CCC(O)C(O)C2)C(=O)NCC2CCCO2)cc1F 12542,c1(C(N2CCN(C(C34OC(C)C(C3)C4)=O)C3C2C3)=O)nncc2c1CCCC2 12543,N1(C(c2c(C)cno2)=O)C2CCC1CC(Cc1ncsc1S(N)(=O)=O)C2 12544,c1(CNC(C(C=C)O)=O)nc2c(s1)CCN(C(=O)CS(=O)(=O)N1CCCCC1)C2 12545,C1(F)(C(=O)NC(C2CC(NC(Cc3cnc(C)o3)=O)C2)C)CCCOC1 12546,C(CCC(=O)NC1CCC(NC(=O)C(C)(O)C2CCCCC2)C1)NC(CC)=O 12547,c1(OC)nc(Cl)ccc1C(N1CCC(CO)(NC(C2CC2C#N)=O)C1)=O 12548,N1(C(C2(n3cc(CC(C)(C)CO)nn3)CC2)C2CC2)CC2CC2(C(F)F)C1 12549,CCCCCC(CC)C(=O)NCCCOCCNC(c1c[nH]c2cccc(C)c12)=O 12550,N1(C(c2cc(OCC)n[nH]2)=O)CCC2(C(=O)NCCC3CCOC3)CC2C1 12551,N1(CC(=O)NC2C3CC2N(C(c2snc(O)c2Cl)=O)C3)CCCCCCC1=O 12552,c1(C2(CNCC(=O)NC)CC=CC2)ccc(Cl)cc1 12553,C=C(C)C(C)(C)C(=O)NC1COCC1NC(=O)CCC(=O)c1ccncc1 12554,N1(C(C(CC)N(CC)CC)=O)C2CCC1CC(NC(=O)CC1CC(F)C1)C2 12555,C(=O)(N1CCC(C(=O)N(C2CC3CCC2O3)C)O1)C1CC(OC)C1 12556,CC(C)CC(C)(CNC(c1c[nH]ccc1=O)=O)NC(C1CN(C)CC(C)O1)=O 12557,C(N=c1nc2c(cnn2C(C)C)c(NCc2csc(Cl)c2)[nH]1)C1(CC)CCOC1 12558,C1(NC(c2nc(C)nc(O)c2)=O)CN(C(=O)CC2CCOCC2)C2CCCCC12 12559,C(CCS(=O)(=O)c1ccc(F)cc1)NC(=O)NC1CCC(C#C)C1 12560,c1(C(=O)NC2CC(O)C2C(=O)NC2CCCS2)cccc(N2CCCCC2)c1 12561,C(CC(C)(C)C(=O)NC(C1CCOC1)CNC(=O)C=CCCC(C)C)OC 12562,C1(C(=O)NCC(CCCC)NC(=O)C(C)(C)C2CC2)CCS(=O)(=O)C(C)C1 12563,Cc1nn(CCC(=O)NC2CCCC2CNC(c2cncc(N)n2)=O)cc1Br 12564,C1(C(N(CCOCCN(C(C(C2CCOCC2)C)=O)C)C)=O)COCC(C)O1 12565,c1(NCC2C(C)CCN(C(=O)C(C)Cn3ccnc3)C2)ncnc2cnccc12 12566,C1(CC(CC)NC(=O)Nc2ccc3c(n2)CCC3)C2C3CC4C1C1C2CC3C41 12567,N1(C(c2c(C)cnnc2)=O)CCC2(CC2)CC1C(=O)NCc1cccc(CO)n1 12568,C1(C)(CNC(CC=C)=O)CN(C(c2coc(COC)n2)=O)CC1C 12569,N1(C(c2ccn(CC)c2C)=O)CCCC(C2CCN(C(c3c[nH]c(=N)o3)=O)C2)C1 12570,C(=O)(C(F)(F)CCCn1cc(CCOC)nn1)N1C(c2cncc(Cl)c2)CCC1 12571,CC(CC(F)(F)F)C(=O)N1CC2(CC2)CC1C(=O)N(C1CC1(C)C)C 12572,C1(NC(c2ccccc2CO)=O)CN(C(c2cc(C(F)(F)F)ccn2)=O)CC1O 12573,c1(C(=O)NCC2C(NC(C(C(C)C)CO)=O)CCC2)cccc2c1nc(O)n2C 12574,Cc1csc(C(=O)N(C)CCOCCN(C(=O)C(N2CCN(C)CC2)C)C)c1Cl 12575,c1(OC)cc(Br)c(C(=O)NCC2CC3CC2CN3C(=O)C2CC2)cc1F 12576,N1(C(C)=O)CCCC2(NC(=O)NCc3ccc(C(F)(F)F)cc3)CC12 12577,N1(C(CCc2cccc(C)c2)=O)CCC(C)N(C2(c3ccn(C)n3)CC2)CC1.CO 12578,C1(c2nc(CC(=O)OCC)on2)CCCN(C(=O)CCc2c[nH]c(=N)o2)C1 12579,c1(NC(C2(C)CCCN(C(C(CO)N(C)C)=O)C2)=O)cc2ccccc2cc1O 12580,C12(CNC(C(=O)N(C)C)=O)CCC(CC1)N(C(C1CNC(=O)N1)=O)C2 12581,C1(C(N2C(CNC(C3(CC)CCC3)=O)CCCC2)=O)CCOC(=O)CC1 12582,Cc1ccn2ncc(C(N3CCCN(C(=O)C(C)SC(F)(F)F)CC3)=O)c2n1 12583,N=c1[nH]c2c(s1)CCCC2C(=O)NCCC1(O)CCCN(C(=O)C2=C(Cl)CCC2)C1 12584,CC(C)(CCCO)NC(C1CSCCN1C(C1CCCCC1)=O)=O 12585,c1(NC(Cn2cc(-c3ccc(OC)c(Cl)c3)nn2)=O)cc2[nH]ccc2cc1Cl 12586,C1(C(N(C(C)CNC(N)=O)CC)=O)CCCC(F)C1.C1(=O)CN1 12587,c1(C(=O)NC2CC(N(C)C)C2)ccnc(C(=O)NC2(N3CCCC3)CCC2)c1 12588,c1(C(N(CCC(C(C)C)NC(=O)C=C2CCCC2)C)=O)cn2cccc(Cl)c2n1 12589,CN1CC(NC(=O)CCOCCCNC(C2CCC(C#N)C2)=O)CC1=O 12590,C12(NC(C3N(CC)CC3)=O)CC(CNC(=O)Cc3ccno3)(C1)OC2C 12591,N1(C(C=C(CCN(C)C)Cl)=O)CC2C(CNC(=O)CNS(=O)(=O)N(C)C)C2C1 12592,C1(NC(c2ccc(C)cc2)=O)COC2(C1)CN(C(=O)CC1CC1C1CC1)C2 12593,C(=O)(CC1=CCOCC1)NC(COC)CC(=O)N1CC(OCCO)C1 12594,C(C(=O)NCC1(C)CCOC1)(C(C)(C)O)NC(C1CCC(CC)O1)=O 12595,c1(CC)cc(CC(=O)NCCN(C(=O)CCCc2cnn[nH]2)CC)on1 12596,CCCCCCCN(C)C(C1C2CCC12)=O.C(=O)(CCCC1CC1)N1CC(C=O)C1 12597,C1(C(N(C(CC)CC)C2CCC2)=O)CCN(CC(=O)NCC2CC(N(C)C)C2)C1 12598,N1(C(c2ccc(CC)s2)=O)CC(N(C(=O)COCC2CCOCC2)C)C2(CC2)C1 12599,C1(C(=O)NCC(C)(C)NC(=O)CC2(C)CCCC2)CCN(CCO)C(=O)C1 12600,C(CN=c1ccnc(NCC23CCCC2CC(=O)N3)[nH]1)c1c(C)n[nH]c1 12601,O=C1CCC(CC(=O)NCC2CC(NC(=O)COc3ccccc3C(F)F)C2)CN1 12602,c1(CC(=O)NC2(CC=C)CCN(C(=O)Cn3ncc(Cl)c3C)C2)cccc(C)c1Cl 12603,Cc1cc(F)sc1C(=O)N(C)CC1CCN(C(C2CC2(C)C)=O)C1 12604,N1(Cc2cccc(OC)c2)CCN(C(=O)C(F)(F)F)CC(C)(C)C1 12605,c1(C(N(C2CN(C(c3cnc(C(C)O)s3)=O)CC2O)C)=O)nccc2ccsc12 12606,Cc1cc(Cl)c(NC(C2CSCCS2)=O)cc1O 12607,CC(C)(C#CC(=O)NCC(C)(O)C1CC1)CNC(=O)CN1CCOC1=O 12608,C1(C(=O)NCC2(NC(c3cn(CC(=O)OCC)nn3)=O)CCC2)CCCCC1F 12609,CC1C(C)C1N=c1[nH]c2c(c(=NCc3ccc(C(C)(F)F)cc3)[nH]1)CCCCC2 12610,Nc1c(F)cc(-c2nc(C34CC(F)C3C4)n(C3CCC3)n2)cc1F 12611,C(=O)(CCCCCC(C)O)N(CC(CN(C(C(C)NC(CC)=O)=O)C)O)C 12612,Cc1cc(Cl)c(Cl)cc1C(=O)OCc1ncoc1C(C)C 12613,C(N=c1[nH]c(N2CCC(C3CCCC3)C2)nc2c1CSC2)c1ccc(N)cn1 12614,S1(=O)(=O)c2cnccc2N(C)N1CCOC.c1(CC)cccc(CNC)c1.CC 12615,c1(C2C(CNC(=O)Nc3sncc3Br)CC2)ccccc1 12616,N1(C(CCCCCOC)=O)CC2CCC1C(NC(c1cncnc1)=O)C2 12617,c1(C(=O)NC2(CC=C)CCN(C(=O)CC(C)OC)C2)cc(C)cc(Br)c1 12618,C1(C(N(C)CC2(O)CN(C(=O)C=Cc3cc[nH]n3)C2)=O)COCCN1C 12619,c1(C(N(CC(CC)NC(=O)CCC2CC=C(C)CC2)CC)=O)cccc(C)c1F 12620,N1(C(C(c2ccn(C)c2)C)=O)CC2CCCC(NC(=O)CSC(C)(C)C)C2C1 12621,c1(C(N(CCNC(=O)CC2CSCCS2)CC)=O)c[nH]c(C)c1Cl 12622,CN1CCCC2CCN(C(N3CC4CCCC(NC(C)(C)C)C4C3)=O)CC12 12623,CCN=c1[nH]cc(C(N2CCC(CNC(=O)Cc3cccs3)C23CC3)=O)s1 12624,N1(C(CCn2ccc(C)n2)=O)CCC(C)N(C(=O)CC2COCC2O)CC1 12625,C(=O)(C1=C(Cl)CCOC1)NC1(CCC)CCN(C(C2CN(C)C2)=O)CC1 12626,N1(C(C(C)(C)SC)=O)CCN(C(c2n[nH]c3c2CCC3)=O)C(C2CCC2)C1 12627,c1(C(N(CCCC(=O)NCCC(C)N(C)C)C)=O)c(O)cccc1F 12628,c1(C(=O)NC(C)CN(C)C(c2ccc(N)cc2)=O)cc2ccc(O)nc2s1 12629,N1(C(C2(C#N)CC2)=O)CCOCC(F)(CNC(c2n[nH]cc2F)=O)CN1 12630,CCC(CN=c1cc(NCCCN2CCCCC2C)nc[nH]1)OC 12631,CC#CCCC(C)(c1nnnn1C1CCC(F)(F)CC1)NC(C)CSC 12632,C1(C(=O)NC2COCCC2O)COC2(C1)CN(C(C1CC1(Cl)Cl)=O)C2 12633,c1(C(N2CC(OC)C(CNC(=O)C(C)CC3CCCC3)C2)=O)cc2n(n1)CCO2 12634,CC(C)CCC(C(=O)NCC(C)(O)CO)NC(=O)Cc1cn(C)cn1 12635,c1(NC(CC)=O)ccc(C)c(C(=O)NCc2ncc(Br)cc2N)c1 12636,C1(NC(C2(CC=C)CC=CC2)=O)CCCC12CCN(C(=O)CCC(C)(F)F)CC2 12637,c1(CCC(=O)NCC(C)(CO)NC(C2(OC(C)=O)CC2)=O)nnc(S)n1C 12638,N1(C(c2ccc(OC)c(O)c2)=O)CCC2(C1)CN(C(c1ncsc1C1CC1)=O)C2 12639,c1(C(N2CCN(C(C3CCC(=C)CC3)=O)C(C)C2)=O)cc2ccccc2nc1O 12640,c1(NC(=O)CCC(=O)N(CCNC(C)=O)C(C)C)ncn(C)c(=O)c1Br 12641,Cc1cnn2ccc(C(N3CC(F)(CNC(=O)CP(C)(C)=O)C3)=O)nc12 12642,C1(NC(c2cnsc2)=O)CN(C(=O)CC2(C3CCCC3)CCC2)C2(CCOC2)C1 12643,N1(C(C(CC)O)=O)CCC(C2(NC(=O)Cn3cccn3)CCC2)CC1 12644,C(=O)(C(O)P(C)(C)=O)NCC(CN(C)C(c1cncc(C(F)(F)F)c1)=O)(C)C 12645,N1(C(C(CCOC)OC)=O)CC(CO)C2(C1)CN(C(=O)CN1CC(=O)NC1=O)C2 12646,C(=O)(C(CNC(=O)CC(F)(F)F)C(C)(C)C)N(C)Cc1n(CC)ccn1 12647,CC(C)S(=O)(=O)c1cccc(C(=O)NC2COCC2CNC(=O)CNC=O)c1 12648,c1(C(=O)NC23CC(NC(CC4CCCN(C)C4)=O)(C2)C3)ccc(F)cc1Cl 12649,C(=O)(C(F)(CNC(C1CC12CCCCC2)=O)C(C)C)Nc1c(OCC)ncc(C)c1 12650,Cn1cc(-c2n[nH]cc2NC(c2nc(C3CC3)cs2)=O)cn1 12651,C(CCCCC(C(=O)NCC(F)F)N(C)C(c1cccc(C)c1)C)OC(C)=O 12652,O=S(=O)(c1ccccc1C(=O)O)N1C2CN(Cc3cncnc3)CC12 12653,C(=O)(CCCC(F)(F)F)NCCOCCN(C)Cc1nccnc1-n1ccnc1 12654,C1(COC)CN(C(=O)CC2(CO)CC2)CCN1C(C1CC1n1ccnc1)=O 12655,c1(C(=O)NCC(C)CNC(=O)C(F)C2CCC2)cccc(S(=O)(=O)CF)c1 12656,C12(C(N3CC(=C(CNC(c4n(CC)ccc4)=O)F)C3)=O)CC1CCC2(F)F 12657,C(N=c1[nH]c(=NCC2CC2)[nH]c2ccc(Cl)cc12)c1cccc(OCCOC)c1 12658,c1(N(C)CCOC(F)F)nc(=NCc2cc(Br)ccc2C)[nH]c2c1CSC2 12659,Cn1cc(C=CC(=O)NCC2CC(C(=O)NCCC3CC3C3CC3)C2)cn1 12660,C1(C(C)NC(C(CC)NC(N)=O)=O)CCN(C(=O)CCCC2CC2)CC1 12661,C1(COC)(CNC(=O)CCC2CCOCC2)CCN(C(C2CC(=O)N(C)C2)=O)C1 12662,C#CCC(C)(C)C(=O)NC(CNC(=O)C(C)n1ccnc1)CCOC 12663,C1(C(C)=O)CC(CC(=O)NC2CN(C(=O)CCC(=O)c3csc(C)n3)C2)C1(C)C 12664,C=Cc1cncc(C(=O)NCC2OCCC2C(N2CCC(CO)C(C)C2)=O)c1 12665,N1(C(C2N(C(C)=O)CC2)C(=O)OC)CC(N)CC1C.c1(C(=O)NC(C)(C)C)csnn1 12666,c1(C(=O)OCC)c(NC(=O)CCCc2ccsc2)sc2c1CCC(C)C2 12667,C(=O)(C(CC1CC1)C(=O)OC(C)(C)C)NCCN(C(=O)C=Cc1cncn1C)C 12668,C(=O)(C(C)(C)C(O)C(C)C)N1CCCC(C)(C(=O)NCc2cncc(OC)n2)C1 12669,S(=O)(=O)(c1ccncc1)N(c1ccccc1C(=O)OCc1ccco1)C 12670,C1(NC(c2ccc(CO)o2)=O)COCCC1NC(c1cnoc1-c1ccoc1)=O 12671,CCC(C(=O)NC(CNC(c1cc(C2CC2)ns1)=O)Cc1ccccc1)NC(N)=O 12672,C1(C2CN(C(=O)C=C(C)Cl)C2)(NC(C2ON=C(CC)C2)=O)CC1 12673,c1(C(N2CCC(C)C2CNC(=O)CCn2ncn(C)c2=O)=O)ncc(N)cc1Cl 12674,c1(OC(N2C(C(=O)NCc3c(CC)non3)CCC2)=O)cccnc1O 12675,c1(C(=O)OCC)nc(C(=O)OC(C)(C)C)n(C)n1.C12(C)CC1COC2=O 12676,C1(OC)CCC12CC(C(=O)NCCC1(NC(c3coc(C#N)c3)=O)CCC1)C2 12677,C(CC(=O)N=c1cc[nH]c(-c2ccc(C)s2)c1)Nc1c(C#N)cc(OC)c(Br)c1 12678,C1(CCNC(COCCSC)=O)CCN(C(=O)CCn2nc(C)cc2C)C(C)C1 12679,C1(C(=O)NCC2CCN(C(C3C(C)CC(=O)N3)=O)CC2)CCCCC1N=[N+]=[N-] 12680,CCCC(C)(C)CC(=O)N1CC2CCC2(CC(=O)NCc2cc(C)ncn2)C1 12681,c1(C(N2CCC(C)C2CNC(C2CCOC(C)C2)=O)=O)cc(C#N)ccc1F 12682,CN=c1ncc(-c2cnc(F)c(C(=O)Nc3cc(C)cc(Cl)c3)c2)c[nH]1 12683,C1(NC(c2cnn(-c3nccs3)c2)=O)CN(C(c2ccsc2Cl)=O)CCC1CO 12684,N1(C(Cc2scc(C)c2)=O)CCC(C)(NC(c2sccc2C)=O)C1 12685,C1(C(N(C)CC2(NC(CCCOCCC)=O)CC(CO)C2)=O)CCC(CC)CC1 12686,N1(C(C2OCC(CN)C2)=O)CCc2cc(C(C)=O)ccc2C1 12687,C(=O)(CCS(C)(=O)=O)NC(CCC)C(O)Cc1ccccc1.C1(=O)CN1 12688,C(=O)(C1c2c[nH]nc2CN1C(=O)CCCn1ccnc1)NCC(N1CCCC1)C 12689,c1(C(=O)NCCOCCC(=O)N(C(C)CC)C)ccc(C(F)F)o1 12690,c1(NC(C)=O)ccc(Cl)c(C(=O)NCC(C)NC(=O)C(c2ccccc2Cl)O)c1 12691,c1(C(=O)NC2CC(C)(NC(c3ccnc(C)n3)=O)C2)cc(N)c2ncccc2c1 12692,c1(C(N2CCCCC2C(=O)Nc2ccc(I)cc2)=O)cc(F)cc(Br)c1Cl 12693,C(=O)(C1=CCC(NC(C2(C#N)CCC2)=O)C1)N(CCC(=O)OCC)C 12694,C1(C(=O)NCCNCC2CCC(C(=O)OC)C2)CCCC(C)(C)CC1 12695,N1(C(C(CCC)O)=O)CCC(C(C)C)CC1CNC(=O)Cn1nnnc1C 12696,Cn1ccn2ncc(C(N3CC4C(NC(=O)C=Cc5cc[nH]c5)C4C3)=O)c12 12697,C1(NC(C(CSC)O)=O)CC2CC1CC2C(=O)NC(CCO)C(C)(C)C 12698,C=CC(CC)CC(=O)Nc1c[nH]ccc1=O.C12CN(CC1C=C)C2=O 12699,c1(C(N(C2CCN(C(C3(C#N)CC3(C)C)=O)C2)C)=O)cn2c(Br)cnc2s1 12700,Cc1nn(C)c(=O)c(C(=O)NCCCC(C)NC(=O)CC23COCC(C2)C3)c1C 12701,C(=O)(C1Cc2ccc(Cl)cc21)NC(CCCC)CNC(c1cc(C2CC2)[nH]n1)=O 12702,C(=O)(C(C)(C)N(C)C)NCCC(C)N(C)C(c1ccc(Br)o1)=O 12703,c1(C(N2C(C)(CNC(c3ccsc3Cl)=O)CCC2)=O)ccc2nonc2c1 12704,c1(CCC(=O)NC(C)CNC(C2(CC3CCC3)CC2)=O)ccc(Br)s1 12705,C(=O)(C1=CCCC1)N(CC(=O)NC(CC)(C)C1CCOC1)CC1CC1 12706,c1(C(=O)NCC2(F)CN(C(c3ccn(C)c3)=O)C2)ccc([N+](=O)[O-])cc1 12707,C(=O)(C(CNC(C1C2CCCC12)=O)N(C)C)NC(C1CCOC1)C#C 12708,N1(C(CC2(OC)CCC2)=O)CCC2(CC1)CC2NC(=O)CC1CC=CC1 12709,c1(C(=O)NCC2CCC(NC(c3c(CC)non3)=O)C2)nccc2c1NCCC2 12710,N1(C(c2cc(Br)c[nH]2)=O)CCOC(C(F)(F)F)C1.S(=O)(=O)(CCc1ccccc1)N 12711,C(=O)(C1=Cc2ccccc2C1O)N1CCC(CNC(c2cncc(SC)c2)=O)C1 12712,CC1(C(=O)NCCN(C(=O)CSc2ccccc2Cl)CCO)COCCO1 12713,C(=O)(C(C)C(F)(F)F)N(CC=CC(=O)N(C)Cc1c(CC)noc1)C 12714,CC1(C)NC(=O)CC1C(=O)NCC1(CNC(C2(C)CC3C=CC2C3)=O)CC1(F)F 12715,CCC(CC)CC(=O)N1CCCC1CNC(c1nccc(-n2ccnc2)n1)=O 12716,C#Cc1ccc(C(=O)NC(CCN(C)C)C(=O)NCc2nnc(C)n2C)cc1 12717,C=C(Br)CC(=O)NC(C(CC1CCCCC1)NC(=O)C=CCF)C1CC1 12718,c1(OC)cscc1C(=O)NC(CNC(=O)C(C)Sc1ccccc1)C(C)C 12719,CCCC(CCCNC(=O)C(c1ccccc1)SC)NC(=O)CCCCC1CC1 12720,c1(C(=O)NCC2(NC(CN(CCC)C)=O)CCC2)nccnc1O 12721,C1(F)(C(=O)NCC2(O)CC(CNC(CC3(C)OCCO3)=O)C2)CCCCC1 12722,CCCC(CC)CCC(=O)NC(C)CNC(C1CCCCC1OC)=O 12723,CC1=CCC(C)(C(=O)NCCC23CCC(C2)N(C(c2csc(C)c2N)=O)C3)CC1 12724,N1(C(C2(COC)CC(=C)C2)=O)CCC(CNC(=O)C=CCCC)(OC)C1 12725,C1(NC(c2nc(CC)oc2C)=O)COC2CN(C(=O)C=CC(=O)NC(C)C)CC12 12726,C1(CCN(C(=O)C(O)Cn2cncn2)C)CCCCN1C(=O)CCC#N 12727,c1(C(=O)NCCN2CCCN(C(C3C(OC)C3)=O)CC2)cccc2c1ncn2C 12728,Cc1cccnc1CCN1CCC(C(C)NC(c2ccc(C(F)(F)F)s2)=O)C1 12729,c1(NCC(C)(CO)C2CC2)ccc(C2CC2)c2cnn(-c3ccccc3)c12 12730,C1(O)(CNC(c2cc(OCC)n[nH]2)=O)CCN(C(=O)CCC2CC(F)(F)C2)C1 12731,C1(C(=O)NCc2ncc(C)nc2)CC12CCN(C(=O)CCc1cncn1C)CC2 12732,C1(NC(c2ccc(Cl)cc2)=O)CN(C(=O)C(O)Cc2cnc[nH]2)CC1CC1CC1 12733,CCC(CC(=O)NC1CCN(C(c2cnn(C3CC3)c2)=O)C1(C)C)CC(C)C 12734,c1(C(=O)NCC(CN(C(C(c2ccn(C)n2)C)=O)C)O)cc(F)cc2cc[nH]c12 12735,C1(NC(CCN(C(CC)CC)C)=O)C2CN(C(C3(C(C)C)CNC(=O)C3)=O)CC12 12736,N1(CC)CCN(CC(=O)NCC(CO)NC(=O)Cc2ccco2)CC1 12737,N1(C(Cc2c(C)cccc2C)=O)CCC2CCCN(C(C3(C#N)CCC3)=O)C2C1 12738,c1(C(=O)NCC(CC(=O)NCc2c(C)non2)C)cnc(C)c(C)c1 12739,C(=O)(C(C)CCC(C)(C)C)NC1(C(=O)Nc2ccc(C)cc2)CC1(C)C 12740,c1(N(C)Cc2c(C)ccnc2)nc(N(C)CC2CC(F)C2)nc2ncn(C)c12 12741,c1(C(=O)NC2(C)CC2)cn2c(n1)CCN(C(=O)Cn1cc(S(C)(=O)=O)cn1)CC2 12742,C(=O)(CCCC(C(=O)NCCS(=O)(=O)CC)N(C)CC1CCOC1)OCC 12743,C1(C2(NC(=O)C=Cc3ccco3)CC2)CCCCN1C(=O)CSC(F)F 12744,C(=O)(CCC(=O)NC1CC1)N(C1CC(c2ccccc2)(NC(=O)C=CS(C)=O)C1)C 12745,Cc1cnc(C)c(C(=O)NCC(C)CN(C)C(c2sc(F)cc2Cl)=O)c1 12746,C(=O)(C1=CC2CCC1C2)N1CCCC(N(C(=O)CCc2cccc(Cl)c2)C)C1 12747,c1(C(N2C(CC(N3CC(CC)OCC3)=O)CC(O)C2)=O)c(C)ccc(I)c1C 12748,c1(C(N2CC(F)(CC)C2)=O)nccnc1Cn1cc(C2CCCNC2=O)nn1 12749,C1(NC(C=CCC)=O)CCCC(NC(c2cccc(C(=O)NC)c2)=O)CC1 12750,c1(C(=O)OC)c[nH]cc(Br)c1=NCC1CCN(C(=O)CCc2cncc(F)c2)C1 12751,C(CC(C)(C)CC(=O)NCC1C=CCN1C(=O)Cn1c(C)csc1=O)OC 12752,C(C)(CCCC(=O)N1CCCC(C)(C(C)C)C1)NC(C=C(C)C1CC1)=O 12753,C1(NC(Cc2c(C)noc2Cl)=O)CC1C1CCN(C(c2cncc(O)c2)=O)CC1 12754,C1(O)(CNC(C2(N(C)C)CC2)=O)CCN(C(c2cc(Cl)ccc2F)=O)CC1 12755,c1(C(N2C(CNC(C3(COC)CCCC3)=O)CCC2)=O)cccc2oc(C)cc12 12756,CCC(C)(O)C(=O)NCC(O)CNC(=O)Cn1[nH]cnc1=N 12757,CC(CNC(=O)CC(C)CNC(c1cncn1C)=O)C(F)(F)F 12758,C(=O)(C(C)(C)C(F)(F)F)N1CC(CNC(Cc2cccc(SCC)c2)=O)OCC1 12759,CCS(=O)(=O)CCNC(C1(CNC(C2CC2(F)Cl)=O)CC(=C)C1)=O 12760,c1(C(=O)NCC2CN(C(CS(=O)(=O)NC)=O)C(C)C2)nn(C)c(Cl)c1Cl 12761,c1(CNC(C(CCOC)NC(=O)CSC(F)F)=O)cccc(F)c1F 12762,C1(C(=O)NCCN(CC(C)O)C(c2[nH]nnc2C(F)F)=O)CC(F)C(=O)N1 12763,c1(CC2(F)CCNCC2)ncnc2ccccc12.c12ccc(cc1)CNC(=O)C2 12764,N1(C(C(C)SC(F)(F)F)=O)CC2CC(NC(=O)C=Cc3cccnc3)CC1C2 12765,c1(C(=O)NCC(=O)NCCCN(C(=O)Cn2nnc(=O)[nH]2)CC)ccc(SC)o1 12766,C1(C(N(C)Cc2snc(C)n2)=O)CN(C)CCN1C(c1cccc(O)c1)=O 12767,C1(O)(CNC(c2nc(C)n(C)n2)=O)CCCC(C)(C)CC1 12768,c1(C(N(CCCNC(=O)CCNS(C)(=O)=O)CC)C)cc(Cl)cc2c1OCC2 12769,C1(C(=O)NC)CCN(C(=O)NCCNC(=O)CC2COCCOC2)C1C 12770,C1(NC(CCCCC=C)=O)CN(C(=O)C(F)(Cl)c2ccccc2)CC(F)(F)C1 12771,N1(C(C(C)(C)C#N)=O)CCC2CCCN(C(c3ccc(CCF)cc3)=O)C2C1 12772,c1(C(N2CCC(CNC(CC(CC)C3CCC3)=O)CC2)=O)nnc2ccccn12 12773,C(C(C)N=c1nc(N(C)Cc2cc(F)ccc2F)c2sccc2[nH]1)c1ccc(C)s1 12774,N1(C(C(C(C)NC(C(CC2CC2)OC)=O)C(C)C)=O)CCCC12CCOC2=O 12775,N1(C(C(C)OCC=C)=O)CC(C(=O)N(c2ncccn2)CC)CC(F)C1 12776,CC1CCCCC1(CO)NC(=O)C(=O)NCCCNC(c1ccc(=O)n(C)n1)=O 12777,C(CN=C(NCC(F)F)N1CCCC(OC2CCCCO2)C1)SCCOC 12778,N1(C(CC(CC)C)=O)CC2CCC1(CNC(=O)C#CC(C)(C)C)CC2 12779,N1(C(c2cc(CCOC)on2)=O)CC(C)CN(C(=O)CC2CCSCC2)CC1C 12780,C1(OC)(CO)CCN(C(=O)C(CN)OC(c2nc(C)cs2)=O)C1 12781,C(=O)(C#CC1(C)CCCO1)N(CCCCN(C)C(C1(C)CC1Br)=O)C 12782,c1(C(N(C)CC2CCN(C(Cc3c(C)ccs3)=O)CC2)=O)csc2ccncc12 12783,N1(C(c2cc(CC)oc2C)=O)CC2CCC1CN2C(=O)CC1CCN(C)C1=O 12784,Cc1nnc2n1C(C(=O)NCCCC(C)NC(=O)Cc1sccc1Cl)CC2 12785,Cn1cc(Cl)c(C(=O)NCCCOCCCNC(c2cnccn2)=O)n1 12786,CC1(C)OCCC1(O)C(N1CC(NC(c2coc(C3CC3)n2)=O)C(O)C1)=O 12787,C1(CC(=O)Nc2c(C)noc2)CC(NC(C2CC3CC3C2)=O)C1(C)C 12788,N1(C(C(CCSC)NC(C2CN(C)CC(C)O2)=O)=O)CCn2nccc2C1 12789,C(=O)(C(F)CCC(C)(C)C)NCc1c(C(=O)Nc2c(C)csc2)nco1 12790,CC1ON=C(C(=O)NC(C2CCCN2C(c2csnn2)=O)C)C1C 12791,CCCCCC(O)CC(=O)NC1CCCC1NC(C1(CO)CC1)=O 12792,C1(C)(C(=O)NC(CC)C(=O)NC)CCN(C(c2c[nH]nc2OC)=O)C1 12793,CCC(CC)CC(F)C(=O)NCCC1(O)CCN(C(C2OCCC2CC)=O)CC1 12794,c1(C(=O)NCC2C(NC(CCn3ncc(C)c3)=O)C2)ccc(C)c2c1CCC2 12795,N1(C(c2c(OC)scc2)=O)CCN(C(C2CCCN2C(C)=O)=O)C(COC)C1 12796,c1(OC)ccc(C(CNC(=O)Cc2nnc(C)n2C)NC(=O)C(O)C(C)C)cc1 12797,C1(O)(COC)CN(C(C2CCC2CNC(=O)C(C)c2ccco2)=O)C1 12798,CCC(C(=O)Nc1cc(C(=O)Nc2nn[nH]n2)cs1)c1cccs1 12799,Cn1nc(CCNc2cc(-c3ccccc3Br)n[nH]2)c2ccccc2c1=O 12800,C1(CN(C(C(C)OC)=O)C)CCCCN1C(c1sccc1OC)=O 12801,C(C1CCCCCC1)=CC(=O)NCC1(F)CN(C(CCC(=C)Cl)=O)C1 12802,C=CC1CN(C(c2cnc(C)c(CC(C)C)c2)=O)CC1NC(=O)C#CC1(C)CC1 12803,CC(C)CC(O)C(C)C(=O)NCC1CN(C(=O)CN(S(=O)(=O)c2cccs2)C)C1 12804,CC1CCCC=C1C(=O)NCC1CCC1NC(c1ccn(C(C)(C)C)c1)=O 12805,c1(C(N2CCC(C(C)(C)NC(Cc3c(C)con3)=O)C2)=O)c(C)coc1C 12806,C(=O)(C1=NOC(CNC(=O)CC(=O)N(C)C)C1)N(CCCCO)C(C)C 12807,N1(C(C)C(=O)NCCC2CC(NC(C3(C4CC4)CC3)=O)C2)CCCCC1=O 12808,c1(CC)ccoc1C(=O)NCCCCCNC(c1ccn(-c2ccncc2)n1)=O 12809,c1(-c2cc(C(C3(C)CN(C(c4nn(C)c(O)c4)=O)C3)=O)no2)cc(Br)ccc1F 12810,c1(CC)nc(Cl)c(F)c(=NCCCCNC(=O)C(Cc2ccccc2)CC)[nH]1 12811,c1(C(N2C(CNC(C3C(C=C)C3)=O)CC(C)(C)C2)=O)ccc2oc(=N)[nH]c2c1 12812,N1(C(C(C2CC(C)(C)C2)OC)=O)CCC2(CCC(NC(=O)CC(F)(F)F)C2)C1 12813,C(C)(c1ccccc1C)=CC(=O)NCC(CNC(C1(COC)CC=CC1)=O)OC 12814,c1(C(=O)NC(CCCC=C)c2ccccc2)[nH]cc2c1CCCC2 12815,N1(C(CN(C(COC)=O)C)=O)Cc2[nH]nc(C(=O)N(C3CCC3)C(C)C)c2C1 12816,c1(C(N2C(CN(C(CN(C)CCO)=O)C)COCC2)=O)cc(O)c2ccoc2c1 12817,C(=O)(C#CC1(C)CC1)N(CC(=O)N(CC(O)CN(C(=O)C(C)(C)C)C)C)C 12818,c1(C(=O)NC23C(NC(c4ccon4)=O)CC(CC2)C3)cc2ccccn2c1 12819,c1(C(N(CCC)CCNC(=O)CSCC(C)C)=O)ccc2c[nH]nc2n1 12820,C1(S(C)(=O)=O)(OC)CC1C(=O)NCc1c(CC)nccc1 12821,CC(C)(C)CCCC(=O)C(=O)N1CCCC(Cn2cc(C3CCCOC3)nn2)C1 12822,C1(CC(=O)NCC(C2CCC2)NC(c2ccc(C3CC3)o2)=O)CC2CC2C1 12823,N1(CCOC)CCC(N=c2[nH]c(N3CCSC(C(F)(F)F)C3)nc3c2COC3)C1 12824,c1(CC)nn[nH]c1C(=O)NC(C)C(C)NC(=O)CN(C)C(=O)C1CC1 12825,c1(SC)cccnc1C(=O)NCC1CC2CC2N1C(=O)CCc1cscn1 12826,C1(NC(C#CC(C)(C)C)=O)CC(N=c2ccnc(Cl)[nH]2)C1(C)C 12827,c1(C(=O)NCC(CNC(CNC(=O)NC)=O)O)c(Br)nc2n1CCCC2 12828,N1(C(C)=O)CCN(C(C2COC(CNC(=O)C(Cl)Cl)C2)=O)C(C)C1 12829,N1(C(C(C)OCC(C)C)=O)CCC(C2CCN(C(C3CCCCN3C)=O)CC2)C1 12830,C1(N(CCCC(=O)NC)C)CCCN(C(=O)CCC(C)OC(C)=O)C1 12831,N1(C(c2n(CC)nnc2)=O)C2CCC1CC(N(C)C(c1ccc(OC)s1)=O)C2 12832,c1(C(CF)NC(C2CCCO2)=O)ccc(F)cc1.c12cc([nH]n1)COC2=O 12833,c1(C(N2C(C)C(NC(=O)C(N3CCSCC3)C)CCC2)=O)cncc2nc[nH]c12 12834,c1(OC)ccc(Cl)cc1C=CC(N1CC(NC(C2CC2(Cl)Cl)=O)CC(C)C1)=O 12835,N1(C(C(C)OCCCC)=O)CCCC2(CCCCC2NC(=O)C=C(C)C(F)F)C1 12836,C1(C(=O)NC2CC(CNC(c3ncsc3C(F)(F)F)=O)C2)CCCC2(CCC2)C1 12837,C1(NC(c2cc(OC)n(C)n2)=O)CCCN(C(C2CN(C(C)C)C2)=O)CC1F 12838,CC1C2CCCN1n1cc2nn1.N1(C(C2CC23CC3)=O)CCC(c2ccn(C)n2)C1 12839,C(C(C(C)(C)C)NC(=O)CCCN1CCCC1)NC(CC1CC(OC)C1)=O 12840,N1(C(C2(C)COCCO2)=O)C2CCC1CN(C(c1ccc(C(F)F)nc1)=O)C2 12841,Cc1cc2[nH]c(C(=O)NCC3(C(=O)NCC(C)CN(C)C)CC3)cc2o1 12842,C1(CN(C(=O)CSCCC#N)C)CCCN1C(c1ccc(-c2cccnc2)s1)=O 12843,C1(NC(C(C)(CSC)NC(C(C)N(CC)CC)=O)=O)CCOC12CCCC2 12844,N1(C(CSCCNC(c2cccc(CO)c2)=O)=O)CCC12CCSCC2 12845,C(=O)(C(CC)CCOC)N1CC(c2c(CNC(CCCOC)=O)nco2)C1 12846,N1(Cc2n(C)cnn2)CCOC(CNC(c2cc(C(F)(F)F)cs2)=O)C1 12847,Cc1cc(CNC(N2CCCCC2C(O)C(F)(F)F)=O)cc(N)c1 12848,Cc1cc2ccccc2nc1C(=O)NC1CC(C)(NC(=O)C2=CCS(=O)(=O)C2)C1 12849,c1(CC(=O)NC2CCC(CC=C)C2)cccc(C#N)c1OC 12850,C1(CC(=O)NCC2(C)CCN(C(c3c(CC)ccs3)=O)C2)CCCC2(CCC2)O1 12851,N1(C(Cc2c(C)nsc2)=O)CCC(F)C(NC(c2ccnc(C(F)(F)F)n2)=O)C1 12852,C#CC1CN(C(C2COCCN2C)=O)CCN1C(=O)C(C1CCOCC1)C 12853,N1(C(C(Br)=C(C)C)=O)CC2CN(C(c3cccc4cncn34)=O)CC2C1 12854,C1(NC(CCC(=O)NC)=O)CC(O)CN(C(c2cc(Br)cn2C(C)C)=O)C1 12855,N1(C(C(CC)NC(C)=O)=O)CC(C(=O)NCC)C(CCC)C1.C(=O)(CCCF)N 12856,c1(C(N2CCCC(CCNC(CC3C(C)(C)CC3)=O)C2)=O)cccc(Cl)c1 12857,C1(C(C(=O)NCCCCCC)CC)CCN(c2n[nH]c(=N)s2)CC1 12858,Cn1nc(C(N2CC3CC2(C(N2CCC(C)(F)C2)=O)C3)=O)cc1O 12859,N1(C(c2cncc(C#C)c2)=O)CCC2CCCC12CNC(=O)C(C)(C(C)C)OC 12860,CCCC(C)(CC)C(=O)NCC1CC(C(=O)Nc2cccc(C(C)=O)c2)=NO1 12861,C1(CC)CN(C(=O)CCc2ccncn2)CC1C(=O)NCC(c1cccnc1)O 12862,CCC(CC(=O)NCC(C)CC(=O)N1CC(CO)C(C)C1)C1CCC1 12863,c1(C(=O)NC2CN(C(C(C(C)C)N3CCC3)=O)C2)cc2c([nH]1)CCC2 12864,C1(NC(C)C(C)(C)C2CCC2)CCCC12CCC2 12865,CC12CN(C(=O)C(=O)NCCCC(F)F)CC1(CO)C2 12866,c1(NC(=O)N(C)CCC2CCN(C(=O)C(=O)C3CC3)CC2)ccc(COC)cc1 12867,CC(CCCCNC(=O)C(C)Cc1cnc[nH]1)NC(c1cc(Cl)cnn1)=O 12868,c1(NC(CCC)CC(F)F)ncccc1S(=O)(=O)NCCCCCCF 12869,C(CC(C(C)(C)C)NC(C1CC2CC2C1)=O)N(C(c1c(C)cncn1)=O)C 12870,O=C(C1=CCCN(Cc2cc(Br)c[nH]2)C1)NCCn1ccc2ccccc12 12871,C1(NC(C(CN(C)C)O)=O)CCC2(CC1)CCN(C(=O)C1=NOC3(CCC3)C1)C2 12872,C(=O)(C(O)CC(N)=O)N1CCC(O)(C(=O)NCC2(OC(C)C)CCC2)C1 12873,C#Cc1ccc(CC(N2CC3(CNC(=O)C(COC)CC)CC2CO3)=O)cc1 12874,CC(C)CC(O)C(=O)N1CC(O)CC1CNC(C1C2(CC2)C12CC2)=O 12875,C(=O)(C(CO)C(C)(C)C)N1CC(C(=O)N(C2CCCCC2)C2CC2)(COC)C1 12876,CC(C)CC(CNC(c1cccc(=O)o1)=O)C(=O)N(C)CC1CC1 12877,C1(NC(CSc2ccc(OC)cc2)=O)CCC(C)N(C(=O)CSS(C)(=O)=O)C1 12878,C(C(=O)N1CCCC1CC)(C(C)(C)C)NC(c1c(CC)cno1)=O 12879,CC1=C(C(=O)NC2CN(C(c3nn(C)c(Cl)c3Cl)=O)CC2F)SCCO1 12880,C(=O)(CC(F)(F)F)NCC(=O)NC1(CN(C(=O)CC2CCC3CC23)C)CC1 12881,C1(CCC(=O)OC)CCN(C(=O)CC2CCCO2)C1.C12(CCC1)CC(=O)N2 12882,CCC(O)C(F)(F)C(=O)N1CCOCC(F)(CNC(=O)C#CC(=O)N(C)CC)C1 12883,N1(C(C=C(CC)CC)=O)CCC2CCC12CNC(c1ccc(O)c(Br)c1)=O 12884,CCC1=C(C(=O)NC2CC2CNC(c2ccc(OC)o2)=O)CCCO1 12885,C1(NC(CC2N(C(C=C(C)C3CC3)=O)C3C2CCC3)=O)CCc2n[nH]cc2C1 12886,c1(C(=O)NS(=O)(=O)c2cncc(Br)c2)cc(Cl)cc2nc(O)[nH]c12 12887,C1(S(N)(=O)=O)(C(=O)NC(C)(C)CN(C)C(C(C(C)CC2CCC2)=O)=O)CCCC1 12888,C(O)(C(=O)NCC(C)N(C(=O)COC)C)SCC 12889,C1(NC(c2ccccc2Br)=O)CCN(C(C2CN3CCC2CC3)=O)CC1O 12890,Cn1nc2c(c1C(N1CC(NC(=O)CSC(C)(C)C)C3(CC3)C1)=O)COCC2 12891,C(=O)(CC(C)(C)C(F)F)N(C1CN(C(C2C(OC)CCC2)=O)CC1O)C 12892,c1(C(=O)NCC(CNC(C2C(CC)C2)=O)(C)O)cc2cc(C)ccc2nc1C 12893,C1(CNC(C(=Cc2cccs2)C)=O)C2CCC(C2)N1C(=O)CNS(N)(=O)=O 12894,C12(NC(c3c(C)coc3C)=O)CCC(c3nn[nH]n3)(CC1)CC2 12895,N1(C(C(C)NC(CC)=O)=O)CCC(COC)(NC(=O)CN2CCCC2)CC1 12896,n1(CCC(=O)NCCOCCN(C)C(c2cc(C(F)(F)F)no2)=O)cc(Cl)cn1 12897,Cc1[nH]c(C)c(C(=O)NCC2CC(C(=O)NC3C(C)C3(C)C)C2)c1C 12898,C#CCC(C(=O)NCC(O)COC)NC(=O)C=CCOC 12899,c1(C(=O)NCC(C)(CO)NC(=O)CSC2CC2)cccc(OC(F)F)c1 12900,N1(C(C2(NC(c3ccc(C)n3C)=O)CCCC2)=O)CCOC(C)(C)CC1 12901,Cc1cc(=NCc2cnc(C)c(Br)c2)[nH]cc1S(=O)(=O)N(C(C)CN(C)C)C 12902,c1(C(N2CCN(C(c3ccccc3)=O)C(CC3CC3)C2)=O)cc([N+](=O)[O-])n[nH]1 12903,c1(NC(=O)NC2C(C)(C)C2)cccc(CN2CCOCC2)c1 12904,C(C)(CCC(=O)N1CCCC(NC(c2cncc(O)c2)=O)C1)OC 12905,c1(C(N2C(C)(C)CC(CNC(c3ncc(Cl)s3)=O)C2)=O)ccc2cc[nH]c2n1 12906,C1(NC(C(=O)OC)c2nccs2)CCCC1(C)C 12907,C1(C(=O)NC2CCN(CCC3CC3)CC2)CC2CCCC2C1 12908,c1(C(N2C(C(=O)NC3CCCC3)CC(=C)C2)=O)cc(C)ccc1Br 12909,C1(C(=O)NC2(C(=O)NC)CCC2)CNC(=O)CN1C(C1CC(C)(C)CN1C)=O 12910,Cc1cc(NCCCNC(C2(O)CCCC(C)(C)C2)=O)n2ncc(C)c2n1 12911,C#Cc1c[nH]nc1C(=O)NCCN(C)C(C1CCC(NC(C)=O)CC1)=O 12912,C(CCC#N)(C(=O)NCc1cccs1)NC(CCCC#C)C 12913,C1(C(N2CCCC(CN(C)C(c3cc(CO)ncn3)=O)C2)=O)CC2(CCCC2)CO1 12914,C1(NC(=O)OC(C)(C)C)CC(C(=O)OCCCc2ccno2)C12CCC2 12915,c1(CNC(C(C)O)=O)cn(CC2CCCN2C(c2cc(C(F)F)on2)=O)nn1 12916,N1(C(C(CCCC)C)=O)CCCC2CN(C(=O)COC)CC12 12917,c1(NC2C(CCC)CN(C(=O)CNC=O)C2)ncnc2sc(C)nc12 12918,C=CC1(C(N2CCC(CF)(NC(c3nccnc3N)=O)C2)=O)CCOCC1 12919,c1(C(N2CCC(C(C)NC(c3c(C)nn[nH]3)=O)C2)=O)cncc(N)c1C 12920,CCCCC(F)(F)C(=O)NC(CN(C(=O)C1=NOC(C)C1C)C)CC 12921,c1(CC(C(=O)O)N(C(CC2CC(C)(C)OC2=O)=O)CCO)cccc([N+](=O)[O-])c1 12922,c1(NC(C(C2CCN(C(c3sccc3Cl)=O)C2)C)=O)ccc2c(c1)OCC2 12923,N1(C(C(CCCNC(C2CCC3CC23)=O)O)=O)CC=CC12CCCCC2 12924,N1(C(C(c2ccc(C)cc2)(C)C)=O)CCN(CCO)CC1(C)C 12925,N1(C(C(C)SCC)=O)CC2CCCC2(NC(=O)CC2(OC)CC2)C1 12926,C(C(CC(C)C)NC(=O)C(c1cccc(Br)n1)(F)F)NC(COCC=C)=O 12927,N1(C(C2C(C)(CC)C2)=O)CC(C)CN(C(C2CCSC(C)C2)=O)CC1C 12928,C(=O)(C1CC(NCc2c[nH]c3ncc(Br)c-3c2)c2ccccc21)OC 12929,c1(C(=O)NC2CCCN(C(c3ccc(C)s3)=O)C2)cccc2c1NCC(C)C2 12930,c1(C(=O)NCC2N(C(C(C)C3CCCC3)=O)CCCC2C)nccc2occc12 12931,c1(C(N(CCCNC(C2CCC(C(F)(F)F)CC2)=O)C)=O)ncn2c1COCC2 12932,C12(C(=O)N(C3CC3)Cc3c(Cn4cc(C(C)O)nn4)nco3)CCN(CC1)C2 12933,c1(C(=O)NCC2CCCN2C(c2ccnc(Br)c2)=O)cc(O)nc(Cl)c1 12934,c1(CN2C(C(=O)Nc3ccc(C)nc3Br)CSCC2)ccc(C)c2cccnc12 12935,N1(C(C2CCN(C(=O)CCc3cncs3)C2)=O)CCC(COC2(C)CCC2)CC1 12936,Cc1cnc(NC(C)CC(C)C)c(S(=O)(=O)N2CC(CO)C3(CC3)C2)c1 12937,c1(CC)cc(N2CC(CN(C(=O)CC3SC(=N)NC3=O)C)C2)nc(CC)n1 12938,N(C)(C1CCCc2c1cnn2C)C(=O)Nc1ccc(OCCOC)cc1 12939,C1(CNC2C(CO)N(OC)C2)(OC(=O)OC(C)(C)C)CC2CCC1C2 12940,C1(C(=O)NCCCn2ncc(C)c2)CCCCC1(C)NC(c1ccc(C)c(C)c1)=O 12941,c1(C(N2CCC(OCCNC(CC(C)C(F)F)=O)C2)=O)cc(C#N)ccc1N 12942,N1(C(C2CC(SC)C2)=O)CC(NC(c2ccc(-c3cccs3)s2)=O)CC(C)C1 12943,N1(C(CNC(Cc2nc(=N)[nH][nH]2)=O)=O)CCCN(CC(N)=O)CC1.C(CN)=CCO 12944,c1(C2(C(N(C3CCN(C(CCCOCC)=O)C3)C)=O)CC2)cc(Cl)ccc1OC 12945,c1(C(C)C)nnc2n1CC(C(N1CC(O)CC1CNC(=O)C(C)(C)O)=O)CC2 12946,Cc1cc(C)c(C(=O)NC2CC3CC(C2)N(C(=O)Cn2nccc2C)C3)c(S)n1 12947,C#Cc1ccc(OCC(=O)NCC2(F)CCCN(C(=O)CCC(=O)NC)C2)cc1 12948,c1(C(=O)NC(C)CCNC(C2(c3ccno3)CCOCC2)=O)nc(Cl)ccc1Cl 12949,N1(C(C2(OC)CCCCC2)=O)CCC(C)C(NC(c2cc(F)ccc2Cl)=O)C1 12950,N=c1[nH]c2ccc(C(N3CC(NC(c4nc(Cl)sc4Cl)=O)CC(F)C3)=O)cc2o1 12951,N1(C(C2CC(NC(C(COC)(C)OC)=O)C2)=O)CC2CCCCC2C1C 12952,C(=O)(C(F)C(=O)NC1(C)CC(NC(C2(C)CC=CC2)=O)C1)OCC 12953,c1(C(C(=O)NCCCC2CC2)N(C(C)C(F)(F)F)CC)sc2ccccc2c1Cl 12954,CC1CCCCC1(C)C(N1CCC(CCCCCn2cc(C3CCC3)nn2)C1)=O 12955,N1(C(C2CC3(C2)CC3(F)F)=O)CCC2CCN(C(c3cc(CO)on3)=O)CC2C1 12956,Nc1ncc(C(N2CCCCC(CNC(c3ccc(CC4CC4)s3)=O)C2)=O)cc1Cl 12957,C1(C(=O)NC(CCC)C(=O)OC)CN(Cc2ccn(C)n2)CC(F)(F)C1 12958,c1(C(N2CCC(N(CCO)C(C3CC4CCCC34)=O)CC2)=O)cnc(O)c(F)c1 12959,Cc1ccc2nc(N3CCC(F)(CNC(c4c[nH]c(C(N)=O)c4)=O)CC3)sc2n1 12960,c1(C(N(C2CC(NC(C(C)(C(C)C)OC)=O)C2)C)=O)cc(C)c(=O)n(C)c1 12961,N1(C(c2c(OCC)scc2)=O)CC2(C)CN(C(=O)CNC(C)=O)CC2(C)C1 12962,Cc1csc(=O)n1CC(N1CCN(CC(C)(C)F)CC1)=O 12963,C1(CC=C)(C(N2CC(NC(C)C(=O)NCCOC)C2)=O)CCOC1.OC 12964,C1(NC(C2(SCC)CC2)=O)COC2(CCN(C(C3(c4ccccc4)CC3)=O)C2)C1 12965,c1(CC2CC2)ccccc1.C1(C(C(=O)NCC2CC2)N2CCC2)(CN)CC=CC1 12966,Cc1ncc(C=CC(N2CCC(C)(CNC(=O)CC3CC4CCC3C4)C2)=O)s1 12967,C(c1cccnc1)=C(C)C(=O)NC1CN(C(c2ccc(C(=O)OC)nc2)=O)C2CC12 12968,c1(C(=O)NC2CC(F)(CNC(C3C(C)OC(=O)N3)=O)C2)cc(NS(C)=O)ccc1F 12969,CCC(O)C(F)(F)C(=O)N1CCCC(CNC(C2COCC2(C)C)=O)C1 12970,CCCCC(O)C(C)C(=O)N1CC(O)(C(C)(C)CNC(=O)Cc2cnoc2)C1 12971,C1(CNC(C2(CC#C)CCOC2)=O)CN(C(c2cnc(=N)[nH]c2)=O)CCC1(F)F 12972,c1(OC)cc(C(N2CC(NC(=O)CSCC3CCCCO3)CC2CO)=O)ccn1 12973,c1(C2(C)CCN(C(C(=O)NCCCC)CC3(C)CCOC3)C2)cc(Cl)ccc1Cl 12974,c1(OC)ccc(Br)c(CN2CCCCC2CCC2CCC2)c1OC 12975,Cc1nc(C(C)C)ncc1C(=O)NCCNC(C1CCCC(=O)N1C)=O 12976,c1(NC2CC(CNC(CNC(CC)=O)=O)C2)snc(Cl)c1C#N 12977,C(C(=O)N1CC2C(C(=O)NC(C)(C(N)=O)C3CC3)C2C1)(C(C)(C)C)OC 12978,Cc1cnc(C(=O)NC2CCCC(NC(C3(NC(N)=O)CC3)=O)C2)nc1 12979,c1(C(C)(C)C)n[nH]c(=NC2CC23CC(NC(=O)CCc2ncc(F)cn2)C3)o1 12980,N(C1CCOc2ccc(F)cc21)Cc1ccc(-c2ccc(N)c([N+](=O)[O-])c2)s1 12981,C(=O)(CC(C)CC(C)C)N1CCC(C(C)(C)C)(CNC(C(CC)N(CC)CC)=O)C1 12982,C1(NC(c2c(Cl)cn(C(C)(C)C)n2)=O)CCC12CN(C(=O)CC1CC(F)(F)C1)C2 12983,C(C(O)CCNC(=O)C(Cc1ccoc1)C(=O)NC(C)C)OC 12984,N1(C(CC2CC(=C)C2)=O)CCN(CC(C)NC(=O)CNc2cn[nH]c2)CC1 12985,N1(C(=O)CCN2CCC(O)CC2)CCC2(C1)CN(C(c1cc(Cl)n[nH]1)=O)CCO2 12986,C(=O)(C1=CC2C=CC(C1)C2)N1C(C)(C(=O)NC2CCNC2=O)CCC1 12987,N(C1CCc2cccnc21)C(c1n(C)cc(NC(c2ncc(Br)cc2Cl)=O)n1)=O 12988,c1(C(=O)NCC(C2CC2)NC(Cn2ccc(C)n2)=O)cnn2cc(C#N)cnc12 12989,C1(CC)CCC(C(N2CCCCC2CC(=O)NCc2ncco2)=O)CC1 12990,C12(CNC(C(C)NC(COC)=O)=O)CC1CN(C(C1(F)CCCCC1)=O)C2 12991,N1(C(c2nc(CCC)sc2)=O)CC(F)CC1CN(C)C(C1CCCC(OC)C1)=O 12992,c1(CNC(c2[nH]cc(COC)c2)=O)cccc(C(N2CCC2C(C)O)=O)n1 12993,N1(C(C2CCCN(C)C2)=O)CCC(CNC(=O)C=C2CCCC2)C12CC2 12994,C1(CN(C(CN(C)CC)=O)C)COCCN1C(=O)CCCc1csc(C)n1 12995,c1(NCCc2c(C)cc(C)s2)ncccc1S(=O)(=O)N1CCn2ncc(Cl)c2C1 12996,c1(CC(C)NC(=O)C(=O)Nc2nc(Br)cs2)cn(C)nc1-c1ccco1 12997,N1(C(C(C)N(C(=O)CC2CCCSC2)C)=O)CC2(CCNC(=O)O2)C1 12998,c1(C(=O)NC2C(C)CCN(C(C(C=C)(C)O)=O)C2)cc(O)nc2ccc(F)cc12 12999,C(CNC(=O)CCOCC(F)F)(C(=O)NC(C)Cn1cccn1)OC 13000,C#Cc1ccc(C(=O)NCCOCCC(N2CC3CC(CO)C(C3)C2)=O)c(C)c1 13001,c1(NC(C=CCNC(c2c(CC)nn(C)c2)=O)=O)ccc2occc2c1 13002,c1(CCC=C)ccccc1CC(=O)NCC1(CNC(C2CNC(=O)C2)=O)CC1.SC 13003,C(=O)(C(C)(C)CC(F)F)N1CC2C(NC(Cc3c(C)n[nH]c3)=O)(CC2)C1 13004,C(=O)(C1COc2ccc(F)cc21)NCC(C1(CNC(=O)OC(C)(C)C)CCCC1)C 13005,CC(N=c1[nH]c(=NC2CC=CCC2)[nH]c2cccc(F)c12)c1nc(=N)[nH][nH]1 13006,c1(C(=O)NCC(CNC(c2nc(CC)oc2)=O)OC)cccc2c(C#N)c[nH]c12 13007,c1(OC)nnc(Cl)cc1NC(c1n[nH]cc1NC(c1cccc(I)c1)=O)=O 13008,CCC(C)CCC(O)CC(=O)N1CC(NC(=O)CS(=O)(=O)C2CCCC2)C(C)C1 13009,C=C(C)C(C)(C)C(=O)NC1CC1NC(C1CCN(C(c2cccnc2)=O)CC1)=O 13010,N(C(=NCCc1nccs1)NCC(N1CCOCC1)=O)C1C(c2ccc(C)o2)C1 13011,N1(C(=O)CSC(F)F)CCCC2CN(c3nc4ccccc4oc3=O)CCC12 13012,c1(C(N(CCCCN(C(CCN(C)CC)=O)C)C)=O)cc2cc(C)ccc2[nH]1 13013,C(C)(CCC(=O)N1CC(Cn2cc(CCC3CCCC3)nn2)C1)OCC 13014,c1(CN2CCC(NC(C3CCc4nc[nH]c4C3)=O)CC2)n[nH]c2ccc(F)cc12 13015,N1(C(c2cnc(C)[nH]2)=O)CCC(C2CCCN(C(c3nc(C)c(C)s3)=O)C2)C1 13016,N1(C(c2c(C(F)(F)F)cc(OC)nc2)=O)CCN(Cc2nc(C)sc2C)CC12CC2 13017,C(=O)(C(C)(C)CC)NCCCC(C)NC(C1C(C#C)C1)=O 13018,C1(O)(CCOC)CCN(C(=O)C(C)(C)CNC(=O)C(C)OC(C)(C)C)CC1 13019,c1(CN(C(C23CCNCC2C3)=O)Cc2cccc(Cl)c2)cccc(Br)c1 13020,N1(C(COCCC=C)=O)CCC(O)(NCCOCCn2cc(COC)nn2)C1 13021,Cc1cc(=NCC2CCOC2c2ccc(Cl)cc2)[nH]c(N2CC(=O)NC(=O)C2)n1 13022,C=C(F)C1(CC(=O)NC(C)(C)C(C)NC(C2CC2(F)C(=O)O)=O)CCC1 13023,C1(N(C(CC)=O)C)CCCCN(C(C23CC(c4ccc(OC)cc4)(C2)C3)=O)C1 13024,c1(NC(C2CN(C(C(C)NC(=O)NC)=O)C2)=O)ccc2ccccc2c1 13025,c1(OC)ccc(C(N2CC3CC(NC(C4CCC(=O)CC4C)=O)C3C2)=O)c(C)c1 13026,c1(CC(C)C)ccc(OC(C)C(N2CC(NC(C3CC3CF)=O)C(O)C2)=O)cc1 13027,c1(C2C(C(=O)NC)CC2)ccccc1.O=C(C=CBr)NN1C(C)CC1 13028,C1(CC(N2CCC(N(C(=O)C=CCOC(C)(C)C)CC)C2)=O)CC(C2CC2)C1 13029,N1(C(C(N2CC=CC(C(=O)OC)C2)=O)=O)CCC2(CCC2)C1 13030,C(=O)(C1=NOC2COCC12)N1CC(OC)C(CNC(=O)C2=CCCS2)C1 13031,C12(OC)CCC(C(N3CCC(CCNC(=O)CC4C=CCC4)C3)=O)(CC1)C(=O)C2 13032,C1(NC(Cc2n(C)ccc2)=O)CCCC(NC(c2cc(C(F)(F)F)ns2)=O)C1 13033,N1(C(C(C)C2CCC2)=O)CCN(C(=O)CC2CN(C(C3CCC3)=O)C2)CC1 13034,C1(C(N(CCCCN(C(CC(CC)C)=O)C)C)=O)CCc2nn(C)cc2C1 13035,C=CC(CC)CC(=O)Nc1ccccc1F.C1C(O)CCC2CN(C2)C(=O)N1CC 13036,c1(OC)ccc(NC(=O)CN(C)C2CC2)cc1.C1C(=O)N1 13037,c12ccccc1O2.c1(NC(CNC(C)C2CC2)=O)nnc(C2CC2)s1.C(C(=O)N)N(C)C 13038,C1(C(=O)NC23CC(NC(C(CC=CCC)C)=O)(C2)C3)CN2CCN1CC2 13039,CC(C)CC(C(=O)N1CCC1C1CCC1)ONC(c1cc([N+](=O)[O-])c[nH]1)=O 13040,c1(C(=O)NCC(CNC(CC(=C)Br)=O)(C)O)cc(C(N)=O)cn1C 13041,N1(C(c2n(CC)ncc2)=O)CCC(C)N(C(C2C(Cl)(Cl)C23CC3)=O)CC1 13042,c1(OC)ccc2c(C(=O)NCC3CC3NC(=O)CCn3ccnc3)cnn2c1 13043,n1(CC)c(=N)[nH]c2cc(C(N3CCC(CNC(C4CCN(C)C4)=O)C3)=O)ccc12 13044,c1(CC)cc(NC(=O)CN(C)C2CC2)ccc1O.C1C(CC(C)C)NC(=O)CO1 13045,C(=O)(C(CC(C)C)Nc1cccc(C(C2CC(C)CC2)C#N)n1)NC(CC)(C)C 13046,C(=O)(C1CCc2ccccc21)NC(CO)CO.N12CCCC1C2=O 13047,c1(NCC2N(C(=O)COc3cccc(Cl)c3)CCC2)ncnc2[nH]c(Cl)cc12 13048,C(=O)(C(F)CC1CCCC1)N(CCC)CCNC(c1cc(CC2CC2)on1)=O 13049,c1(-c2c(OC)cncn2)ccc(C(=O)O)n2nccc12 13050,C1(C#N)(C(N2CCC(CNC(C(C3CC3)OCC)=O)C23CC3)=O)CC12CCCC2 13051,c1(OC)ccc(C(=O)NC(C)C(C)NC(=O)CCOC(C)C)c2[nH]ncc12 13052,N1(C(c2cc(CNC(C(C)(C)c3ccsc3)=O)sc2)=O)CCCCC1CCO 13053,c1(C(N2C3CC(CC(NC(C(C)CF)=O)C3)C2)=O)cc(F)cc2ccncc12 13054,c1(C(N2CCCC(CNC(c3c(C)ncnc3)=O)C2)=O)ccc(F)c(C(F)F)n1 13055,C1(CC(=O)NCC(CCCNC(=O)OC(C)(C)C)O)CC2(CCO1)CC2 13056,c1(C(=O)N(C(C(C)(C)NC(CSCC=C)=O)C)CCCC)c[nH]c2ccc(Cl)cc2c1=O 13057,O=C(C1=CCC2(COC2)OC1)NCC1CCCN(C(c2ccccc2Cl)=O)CC1 13058,C1(CC(=O)NCC2(C)CC(NC(Cc3c(C)n(C)nc3)=O)C2)CCCCC(=O)N1 13059,C(=O)(CC1=NN(C)C(=O)C1)N(CCCNC(c1cccc2ncsc12)=O)C(C)C 13060,C1(C#CC(=O)N2CC=CC(NC(=O)C(c3cccc(Cl)c3)O)C2)(CC)COC1 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13130,N1(C(C(=Cc2ccccc2)C)=O)CCCC(C)(NC(=O)CN(C)S(N)(=O)=O)C1 13131,C=CC(CC)C(=O)NC1COCCC1C(=O)N(C1CCOC1)CC 13132,C1(C(N2CC(N3CCN(CC4C(C#N)C4)CC3)C2)=O)Cc2ccccc2S1 13133,C1(CC)CN(C(C2(COC(C)C)CC2)=O)CCN1C(C1CC(C(C)C)=NO1)=O 13134,C(C(C(=O)N1CCCC1CNC(c1cnn(C(C)(C)C)n1)=O)OC)OC 13135,C1(C(=O)Nc2ccc(C3CN(Cc4cccs4)CCO3)cc2)CCC(F)(F)CC1 13136,N1(C(COC(C)=O)=O)CCC2CCN(C(=O)C3CCCc4n[nH]cc43)CC2C1 13137,c1(C(N2CCC(C(N(C3CCNCC3)CC=C)=O)C(O)C2)=O)cc2cccnn2c1 13138,c1(C(=O)NC2CN(C(C(C3CCC(=O)N3C)C)=O)C2)cc2c(nn1)CCOC2 13139,Brc1nsc(I)c1C(c1nnnn1C1CC1)NCc1cnn(C2CCCCC2)c1 13140,C(CN=c1[nH]cnc2c1SCCC2)(C1CCCC1)NC(c1cccnc1S)=O 13141,CCC(C)(CO)C(=O)N1CC(CNC(c2ccnnc2)=O)C(F)(F)C1 13142,CC1CC(C)(C(N2CC(F)(CNC(=O)CCOc3ccccc3F)C2)=O)CCO1 13143,c1(CC)cc(C(=O)NC(C)(CNC(C2CCCCC2O)=O)CC)ccc1Cl 13144,CC(CC1CC1)CC(=O)N1CCSCC1C(N1CCOC(C(N)=O)C1)=O 13145,C(=O)(C(C)CS(C)(=O)=O)NC1CC(C)(NC(CC2N(C(C)=O)CCC2)=O)C1 13146,c1(NC(COC(=N)O)=O)cccc(Sc2ncccc2Br)c1 13147,CC1CN(C(c2ccc(C(F)(F)F)cc2Br)=O)CCN1C(c1ccoc1)=O 13148,c1(CCC(=O)N(CCC(=O)NC(C(C)SC)C)C2CC2)ccnc(C)n1 13149,N1(C(CN(C)C(N)=O)=O)CC2(C1)C(NC(C1CCC3CCC1O3)=O)CCS2(=O)=O 13150,Cc1cc(C(=O)NCCCNC(C23COCC2C3)=O)n2ncnc2n1 13151,c1(C(=O)NCC(c2ccc(OC)cc2)NC(CC=CCC)=O)cc(C)c(F)cn1 13152,c1(C(=O)NCC(C)CNC(C2CC2C(C)(C)O)=O)cc(F)c(C(F)F)cc1F 13153,c1(C(N2C(CC)CC(C)CC2)C(=O)NC2CC(F)(F)C2)ccc([N+](=O)[O-])cc1OC 13154,C12CN(CCN1C(=O)CC1CCCCC1O)C(=O)C2.N1(C(C)(C)C)CCNC(=O)C1 13155,c1(C(N(C2CCN(C(C3(C)CCCS3)=O)CC2)CC)=O)n[nH]c2c(C)cccc12 13156,c1(C(=O)NCC(C(C(C)C)C)NC(c2ncccn2)=O)cc(F)c(F)c(F)c1F 13157,c1(CCC(=O)NC2CC(CNC(C(C)(F)F)=O)C2)cccc2cnccc12 13158,C(=O)(C1=NOC2(CCC2)C1)NCC(C)(C1CC1)NC(C1(C)CCC(=O)N1)=O 13159,C1(C(N2CCC(N(CC)CC)C2)=O)C2CCCC1N(Cc1ccc(F)c(F)c1)C2 13160,C(=O)(C(C)CS(C)(=O)=O)NCC1CCCN(C(c2cc(C)nc(C)c2)=O)C1 13161,C=CCC(C)(C)CC(=O)NC1CC(NC(c2ncccc2Cl)=O)C1 13162,c1(C(N2CC(C(C(=O)OC)NC(=O)C3CC3)C2)=O)c[nH]nc1-n1cnnn1 13163,C1(C(=O)NCc2cn(C3CN(Cc4cnsn4)C3)nn2)CCCCC1O 13164,C1(NC(C2C=CCC2)=O)C=CCN(C(=O)CC(c2ccccc2)c2ncc[nH]2)C1 13165,CC1(C)CCC(O)(CNC(=O)CCN(C(=O)CCCC2CC2)CCCO)C1 13166,C(=O)(CCCCCC(C)C)NC(CC)(CNC(=O)C(O)C(F)(F)F)CC 13167,c1(C(N2C(Nc3cc(C(=O)OCC)c(F)cn3)CC2)=O)cccn2ccnc12 13168,CC1CN(C(c2ncn3c2CCCC3)=O)CC(C)C1NC(c1ccc(CO)o1)=O 13169,CS(=O)(=O)CC(=O)NCC1(C(=O)Nc2ccc(F)nc2)CC12CCC2 13170,C1(F)(CNC(C(c2c(C)cccc2)C)=O)COCCN(C(=O)CSC(F)F)C1 13171,c1(CN2CCC(N(C)C(c3ccsc3)=O)C2)cccc(C=O)c1Br 13172,C(CC(=O)NC1CCN(C2CCN(C)C2=O)CC1)(C(F)(F)F)OC 13173,C(=O)(C(F)C(F)(F)F)NC1C(CNC(C2CCC(Cn3ccnc3)O2)=O)CCC1 13174,c1(COC)noc(C(=O)NC2CCC(NC(C3CCC3)=O)C2)n1 13175,c1(NC)ccnc(C(N2CCC(CNC(=O)CCC(C)c3ccccc3)C2)=O)c1 13176,C(=O)(CCCC(=O)NCCCC(C)(C)NC(C1CC2CCC1C2)=O)NCC 13177,N1(C(c2ncc(C)nc2)=O)CCC(N=c2cc(C)nc(S(C)(=O)=O)[nH]2)C(C)C1 13178,N1(CCN(C(c2c(C)ccs2)=O)C)CCC(N(C)CC2CCOCC2)CC1 13179,c1(CNC(C2CCN(C(=O)NCCCOC)C2)=O)c(C(C)C)cccc1F 13180,c1(C(N(CC(O)CN(C)C(c2ncn(C)n2)=O)C)=O)ccnc(C#N)c1 13181,Cc1cccc(C(=O)NCC(C)N(C)C(c2ccc(CCF)cc2)=O)c1C 13182,N1(C(Cc2cc(C)c(F)cc2)=O)CC=C(CC(=O)NCc2cc[nH]c2)CC1 13183,N1(c2cc(N(C3CCN4CCCC3C4)C)ncn2)CCCC(C)(C)CC1 13184,C1(CNC(c2nn(CC)nc2C)=O)(NC(C2CC(O)C2)=O)CCCCC1C 13185,c1(-c2nc(CCCCCC)nn2Cc2ccccn2)cc2nc(OC)ccc2[nH]1 13186,c1(C(=O)NC(C2CCN(C(C=CCC)=O)C2)C)c(C)cnn1C 13187,c1(CNC(C2CCCN2C(c2ccno2)=O)=O)ccc2ncsc2c1 13188,C(CC(C)C)(C(=O)NC1(CNC(C2CCOC2)=O)CC1)OC 13189,C1(C(=O)NCC(CNC(=O)CSS(C)(=O)=O)OC)CC2CCC(C1)N2C(C)C 13190,C(C(C)C(=O)NC1CCC1)NC(CCNC(C)=O)=O 13191,C1(NC(C(CC=CCC)C)=O)C2CCC(C2)C1C(=O)NCC1CCC(C)C1 13192,c1(NC(C2CC(=C)CN2C(C)C(=O)NOCC)=O)ccc(C(C)CC)c(Br)c1 13193,C1(C(=O)NCC(C)(C)C(F)F)CN(C(=O)CC2CC(C3CC3)C2)C2(CCC2)C1 13194,N1(C(CNC(=O)CN2CCCC2)=O)CCCC1CCNC(N)=O.C12(CC1)CC2 13195,C(=O)(C1CCc2c[nH]nc21)N1CCCN(C(C(CCC)(C)O)=O)CC1 13196,c1(C(C(=O)NCCC2(C)CC2)N(C(c2cccc(F)c2)CC)C)ccc(F)cc1Cl 13197,C1(CN(C(=O)C(C)C2CCCC2)CC)CCN(C(=O)CN2CCC2)CC1 13198,N1(C(C=CCC)=O)C2CCC1C(NC(c1cccn1C1CCCC1)=O)C2 13199,C1(CCC)CN(C(=O)C(C)(C)n2cccn2)CC1NC(C1C=CCC1)=O 13200,N1(C(c2cc(C)nn2C)=O)C2CCC1C(C)C(NC(C1CCC(F)(F)CC1)=O)C2 13201,N(C1c2ccccc2CC1NC(c1cccc(SC)c1)=O)C(C(CC=C)C)=O 13202,Cc1cnc2n1CCC(C(=O)OC(C)(C)C)C2.C1C(c2ccccc2)C(=O)N1 13203,CN1CCN(C(=O)Cc2ccnc(O)c2)C(CNC(C2CC3(CC3)CO2)=O)C1 13204,c1(CC)cc(C(=O)NC(C)CCCCNC(=O)CCF)ccc1Cl 13205,C(=O)(CC(C)(C)C1CC1)N1CCC(SCc2ccc(C(N(C)CC)=O)o2)C1 13206,N1(C(c2cc(C(C)=O)no2)=O)C(CNC(=O)C(C)CO)CC2COCC12 13207,C(N=c1[nH]c(=NCc2[nH]nnc2C)c2ccccc2[nH]1)c1ncc(C)o1 13208,C1CCCC(=O)N2CCC(O2)C(=O)N1.N1(CC)CC(N(C)C)C(C)C1 13209,CC(C(CO)NC(c1csnc1-c1ccccc1)=O)NC(c1ncccn1)=O 13210,C(CS(=O)(=O)C1=C(F)CCC1)NC(c1ccc(F)c(C(=O)O)c1O)C 13211,C12(CNC(COC)=O)CN(C(c3cccc4c3CCO4)=O)CC1CCO2 13212,CC(C)CC(O)CC(=O)N1CCCCC(NC(=O)C(F)(F)C2(O)CCC2)C1 13213,C#Cc1c[nH]nc1C(=O)NC1CC1NC(c1ccccc1COC(C)(C)C)=O 13214,N1(C(CCCC)=O)CCC(NC(c2csc(-c3ccsc3)n2)=O)C(CO)C1 13215,c1(C(=O)NCC(N(C(C(C)SCC)=O)C)C2CC2)nnc(O)c2ccccc12 13216,N1(C(CC(N2C(C(N)=O)CC=CC2)=O)=O)CC2C=CCC(C2)C1 13217,c1(C(=O)NC2(C3CCCN3C(=O)Cn3ccnn3)CC2)cn2ccnc2cn1 13218,N1(Cc2n(CC)nnc2)CCc2c(OCC)cccc2C1 13219,Nc1ccc(C(N2CCCC2CCCNC(=O)C#CC2CCC2)=O)nc1C(F)(F)F 13220,C(C(O)CNC(C1CCCO1)=O)NC(CSCC#N)=O 13221,C1(C(N)=O)(NC(C2(C)CN(C(c3c(CC)[nH]cc3)=O)C2)=O)CCCCC1C 13222,C1(C(=O)NCCNC(c2cc(CCCCC)[nH]n2)=O)CCc2nc(C)[nH]c2C1 13223,CC1CC(=O)NC1C(N1CCC(CCCNC(=O)Cc2cccc(O)c2)CC1)=O 13224,c1(OCCOC)ccc(NC2COC3CC2C3)cc1 13225,c1(NC2(CNC(c3cncc(NC)c3)=O)COC2)ncnc2cc(Br)ccc12 13226,C(=O)(C1CCCc2sccc21)NCC1(NC(C2CCN(C)C2)=O)CC1 13227,Cc1cccc(CN(C(=O)C(CCC2CCC2)NC(=O)C(C)(F)c2ccon2)C)n1 13228,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC1CC1CNC(C1CCC2(CCC2)C1)=O 13229,c1(OC)cc2nn[nH]c2cc1C(=O)NCCCCNC(c1cnn(C)n1)=O 13230,C1(C(N(CCNC(C)=O)C2CC2)=O)CCN(C)S1(=O)=O.N12CCCC(C1)C2=O 13231,c1(CC(=O)NC(C2CC2C(=O)NCCC2(C)N=N2)C)ccnn1C 13232,c1(CC(=O)NCC2CC2F)ccc2nonc2c1.C12CCCC1CNC2=O 13233,C1(CC(=O)NCC23CCC(CC2)C3)(NC(C2CCO2)=O)CCCCC1 13234,c1(C(N2CC3CC3(C(=O)NCc3ccncc3Cl)C2)=O)cc(Cl)c(O)cc1F 13235,C#Cc1ccc(C(=O)NC(C2CCCCN2C(=O)CSCCC(C)C)C)c(F)c1 13236,CC(C)C(F)(CNC(C1CCCN1C(C)C)=O)C(=O)NCC(C)(C)CN=[N+]=[N-] 13237,n1(CC(=O)NC2C(NC(=O)C3=CCCC3)C2)ccc2cc(C(=O)NC3CC3)ccc12 13238,C1(NC(CCC2(NC(CC(=O)OC(C)(C)C)=O)CCC2)=O)CC(C2CCCC2)C1 13239,C(CC1=CCN(C(c2ccc(F)c(F)c2N)=O)CC1)NC(C(=Cc1cnc[nH]1)C)=O 13240,c1(CC(N2CC(NC(C)=O)C(C3CC3)C2)=O)nc2c([nH]1)CCCC2 13241,c1(C(=O)NC(C)CC2CN(C(c3cscc3Cl)=O)C2)nnn(C)c1C(F)F 13242,C1(C(=O)NC(CC=C)C(=O)OC)CNC(=O)CN1C(C1CC1CCOC)=O 13243,n1(CC)ccc(CC(=O)NCc2csc(CC(c3cncnc3)=O)n2)n1 13244,C1(C(N2CCN(c3nc(C)cc(C)n3)C3C2C3)=O)CCCC2CCCCC12 13245,Cc1ncccc1C(N1CCCC(CNC(=O)Cn2cnc(C(N)=O)n2)C1)=O 13246,c1(C(=O)NC(CC(C)NC(C2NC(=O)CC2C)=O)C)ccc(N)cc1O 13247,C1(C(=O)NCCOCCC(=O)NC(CC)C2CC2)CCC1C#N 13248,c1(OC)cc(F)c(F)cc1C(=O)Nc1nc(Cl)c(Cl)nc1NC(C)=O 13249,N1(C(=O)OC(C)(C)C)CC2(CCC2)CC1NCCCC1CCOC1 13250,C1(CC#C)(C(=O)NC(CC(N)=O)C2CC2)CCN(C(c2ccnn2C)=O)C1 13251,c1(C(N2C(C(=O)NCc3cc(C)ncc3)COCC2)=O)cc(C)c(Br)c(C)c1 13252,O=C1CN(CC2CC(=O)N(C3CC3)C2)CCN1Cc1nc(C2CC2)no1 13253,N1(c2snc(COCC)n2)CCS(=O)(=O)C(CCNC(=O)C(C)(C)CF)C1 13254,N1(C(C(CC#C)C)=O)CCOC2CN(C(=O)Cc3cccc(OC)c3Cl)CC12 13255,C1(NC(C(C)=C(C)C)=O)CCC(NC(=O)C(C2CCOCC2)C)C1 13256,Cc1ncc([N+](=O)[O-])cc1NC(=O)CC1CCN(C(c2cc(F)c(F)c(F)c2)=O)C1 13257,O=CN1CCCN(C(=O)CC(CC2CC2)NC(C2(CO)CCCO2)=O)CC1 13258,c1(C(N(C2CCCN(C(C3CCC(=O)NC3)=O)C2)CCO)=O)coc2c1COC2 13259,C(CC)(CCCO)OC.c1(OC)sccc1CO.C1(N)C(=O)N2CC1C2 13260,c1(OC)ccc2[nH]ccc2c1C(=O)NCCC1(OC)CN(C(=O)C2=CCCS2)C1 13261,C(=O)(C(C)(C(C)C)OC)NC(CC=C)CNC(c1n[nH]c(C)n1)=O 13262,c1(CC(=O)NC2C(NC(C=C)=O)C2)ccc(C)cc1Cl 13263,C=CCC(C)(C)C(=O)NC1(CCCC(C)NC(=O)Cn2cccc2)CC1 13264,Cc1ccc(O)cc1C(N1CC(C)CC1C(=O)NC1CC2C=CC1C2)=O 13265,c1(CC)nn(C)cc1C(=O)NC1CC(CNC(=O)OC(C)=O)C1(C)C 13266,CC1(C)C(C(=O)NCC(F)(F)C(F)F)C2CCCN(C(=O)CC3CCOC3=O)C12 13267,Cc1ccc2ccc(C(=O)NCC(C3CC3)NC(C3C(F)(F)C34CC4)=O)nc2c1 13268,CC1CCN(C(=O)COc2ccn(C)n2)CCN1C(=O)CCOCC1CCCO1 13269,C(CN=c1[nH]c(=NCC2CCOC(C)C2)[nH]c2c1CCC2)NS(CC)(=O)=O 13270,CC(CO)(C(=O)NCC1CCCC1F)NC(C1CCOCC1)=O 13271,N1(C(CC=C)=O)CCOC(Cn2cc(CC(c3ccccc3)C)nn2)C1 13272,c1(COC)cnc(NC(=O)NCC(c2ccccn2)C)nc1 13273,CC1CN(C(=O)C(=O)C(F)(F)F)CCC1NC(=O)CCC1CC1(F)F 13274,C1(C(N(CC(CC)NC(=O)CCCCCSC)C)=O)CCS(=O)(=O)CC1 13275,CCC(CC)C(=O)NCC1CC(O)CN1C(=O)CCCOc1ccccc1Cl 13276,CC1CC2CN(C(C3CC3(F)Cl)=O)CC2N1C(=O)C(O)CC(N)=O 13277,C1(COC2CN(C(=O)Cc3cc[nH]n3)C2)CCN(C(C23C=CC(CC2)C3)=O)CC1 13278,C1(C(=O)NC(c2ccnc(F)c2)C)CCCCCN1C(c1ccc(C(N)=O)o1)=O 13279,CCC(C(=O)NCCOC1CN(C(c2occc2Cl)=O)C1)OC 13280,C1(C(=O)NC(CC2(O)CN(C(C=CC(C)=O)=O)C2)(C)C)CCN(CCO)C(=O)C1 13281,C1(N(C(C(C)OCC#C)=O)C)CN(C(c2c(Cl)csc2Cl)=O)CC1(C)C 13282,N1(CCF)CCC(CNS(=O)(=O)CC2CCOC2)CC1 13283,CC(=O)C(C)CC(C)C(=O)N1C(C(N2CCC(C)(C)C2)=O)C2CC(O)C1C2 13284,C1(C(=O)NC2CCC(CNC(=O)CCN3CCCC3)C2)CC2(CCOC2)C1 13285,C(=O)(CC(C)C(F)F)NCC(CC=C)NC(=O)CSCC(C)C 13286,CN(C)S(=O)(=O)N(C)CC(=O)NCCC1CCCN(C(c2cc[nH]c2)=O)C1 13287,c1(OC)cc(C2(CCC(=O)OC)CCC2)c(NC(=O)CCN2CCCCC2)cn1 13288,c1(C(=O)NCC2(F)CC(NC(C3C(OC)CCC3)=O)C2)oc(CO)nc1C 13289,C1(NC(CC(n2c(C)cc(C)n2)C)=O)C2CC1CN(C(=O)CNS(N)(=O)=O)C2 13290,CC1CCC(NC(c2ccn(C3CCCC3)n2)=O)CN1Cc1cscc1Cl 13291,CC(C#N)CCC(=O)N1CC(CNC(c2ccc(C3CC3)nc2)=O)C2(CC2)C1 13292,C1(N(CC#C)C)CCN(C(C2CC2C(=O)OC(C2CC(=O)N(C3CC3)C2)=O)=O)CC1 13293,c12cnc(s1)N1CCC(C1)C2.C(C1CCCC1)=C(C(=O)N(CC)C1CC1)C.C(=O)OC 13294,C1(C(=O)NCC(C(C)C)O)CN(C(=O)CC2CCCC2)CC1(C)C 13295,c1(CCC)c(C(=O)N(C)CC2CCCN(C(=O)C(C)n3ccnc3)C2)cnn1C 13296,C(=O)(C(CO)C(C)C)NC1CCN(Cc2cccc(CC)c2)CC1 13297,c1(OC)ccc(C(=O)NCCN(C(=O)CC2CCCC(C)C2)C)nc1Br 13298,N1(C(C(CCC)OC)=O)CCCC2(CCN(C(=O)C(CC)SC)CC2)C1 13299,C1(NC(c2c(C)cns2)=O)CCC(CNC(=O)Cc2csc(Br)n2)CC1 13300,C1(OC)CC(N=c2[nH]c(C(F)(F)C(F)(F)F)nc(C)c2C)C1 13301,CC(C)C(CNC(=O)C=C(C1CC1)C1CC1)C(=O)N1CCC(CCN(C)C)C1 13302,Cc1c(CC(=O)NC(C(=O)N(C)Cc2ccnn2C)C2CC2)ncn1C 13303,N1(C(CSCC(C)C)=O)CC2(C1)SCCC2NC(=O)CCCC(N)=O 13304,CC1CN(C(c2cccc(F)c2)=O)CCC1C(=O)NCc1ccc(O)nc1 13305,C1(C(N(C)CC)=O)(CNC(c2nc(O)sc2C)=O)CC12CCC2 13306,C1(Cn2c3cn(nn3)c2=O)CC2(C1)CC21CCC1.C1(C(=O)OCC)(CSC)CC1 13307,c12cc(c([N+](=O)[O-])cn1)SC2.C(C(=O)N(CCOC)CCOCCO)OCC#C 13308,N1(C(C(CC)NC(C)=O)=O)CC2CCC1C(C(N1CCC(Br)C1)=O)C2 13309,C12(C(=O)NCCCC(=O)OCC)CC1CN(C(c1c[nH]c(C)c1)=O)C2 13310,C1(C(N(CCN(C(=O)C(O)CC(N)=O)C)C)=O)CSc2ccccc2O1 13311,c1(NC(c2cnc(C3CC3)s2)=O)ccc(F)c(-c2nn[nH]n2)c1 13312,C(C)CCC(=O)NCCCOCCOCCNC(c1cc(CSC)on1)=O.CO 13313,c1(CC(=O)NCCCC(C)NC(c2ccoc2)=O)cccc(OC(F)(F)F)c1 13314,N1(CC(=O)NC2CCC2NC(=O)CC2(CO)CC2)Cc2ccccc2C1 13315,Cc1nc(O)nc(O)c1CC(=O)NC12CCCC1N(C(=O)C(=O)C(F)(F)F)CC2 13316,N1(C(CC(CC)(C)C)=O)CCCN(C(c2ccc(OC3CCC3)cc2)=O)CC1C 13317,CC1CCC(c2nc(C3CCCS3)nn2CCCNC(=O)OC(C)(C)C)OC1 13318,C1(C(=O)NCC(c2ccccc2)CNC(COCCC(C)C)=O)CCCCCC1 13319,c1(C(=O)NCC(CC)NC(c2ccn(-c3cccc(F)c3)n2)=O)cccnc1C 13320,C12(C(=O)NCCCN(C(=O)CN3CCCS3(=O)=O)CC)CCCCC1C2(F)F 13321,c1(COC)nc(NCCC(O)C2CC2)cc(=NCC2(C(N)=O)CC2)[nH]1 13322,N1(C(C)=O)CCC(CC(=O)NC(C2NC(=O)NC2=O)COC(C)C)CC1 13323,CC1CC(NCCN2CCCCC2=O)CCN1CC1CCC2(CC2)C1 13324,CC(C)CC(C)(CNC(C1CC(=O)NC(=O)C1)=O)NC(C1CC(F)(F)C1)=O 13325,C1(C(=O)NCCN(C(=O)CCc2cnoc2)CC)CCC(=O)N1CCC(F)(F)F 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13344,C1(F)(C(N(C)CC2COCCN2C(=O)C=CC(F)(F)F)=O)C(C)(C)C1(C)C 13345,C(C(CC(C)C)NC(C1CC(=O)N(CC)C1)=O)NC(c1c(CC)noc1)=O 13346,c1(C(C)C)onc(C2CCCCC2)c1C(=O)N(C)CCNC(=O)C=C(Cl)Cl 13347,c1(C(=O)NCC(C)(CO)NC(C2CC(OC)C2)=O)c(OC)ccc(Cl)c1C 13348,C1(CNC(C(C)CC2CC2)c2nnnn2C2CCOCC2)CCCCS1(=O)=O 13349,c1(C(N(CCCCCC)C(C)C2CC2)=O)cccc(-n2cc(-c3ccncc3)nn2)c1 13350,N1(C(c2c(C)oc(Cl)n2)=O)CC(NC(C2CN3CCN2CC3)=O)CC(F)(F)C1 13351,N1(C(CNC(C)=O)C)CCCC(C2(Cc3c[nH]nc3C3CC3)CC2)C1 13352,N1(C(C=CC(C)(C)C)=O)CC(CNC(=O)CCc2ccc(F)nc2)CC1(C)C 13353,C1(Br)(C(=O)NCC(C)N(C(c2cc(CC)on2)=O)C)CC12CCC2 13354,c1(C(=O)NCC(CCNC(c2cscn2)=O)OC)cn(C)ccc1=O 13355,Cc1ncnc(C)c1C(=O)NCC(C)N(C)C(c1coc(C(F)(F)F)c1)=O 13356,C1(C(=O)NC2C(NC(C(OCC)OCC)=O)C2)CCCC2(CC2)C1 13357,c1(N2CC(NC(CC3CC(=C)C3)=O)C3C(C2)CCC3)nc2ccc(F)cc2o1 13358,c1(NC(=O)Nc2cccc(C(=O)NCCC)c2)ccc(P(C)(C)=O)nc1 13359,C#CCC(C)(C)C(=O)N1CCOC(CCNC(=O)Cn2ccc(C)c2)C1 13360,CC(O)C(C(=O)NCC1CCCCN1C(c1coc(C(F)F)c1)=O)N(C)C 13361,c1(C(N2CCC(C(C)(C)NC(CCC=C(C)C)=O)CC2)=O)cc(S(C)(=O)=O)cs1 13362,N1(C(CCCCSC)=O)C2CC1CN(C(=O)CCP(C)(C)=O)C2 13363,c1(CN2CC(NC(C3(F)CCCCC3(F)F)=O)C2)nc2ccccc2[nH]1 13364,N1(C(c2cnc(CC)[nH]2)=O)CC2CC2(CNC(=O)CC2CCC(=O)N2C)C1 13365,c12ccc(OC)nc1NC(=O)C2NC(c1cc(Br)cs1)=O.C(COC)OC 13366,Cc1ccc2[nH]c(C(=O)NCCC3(NC(C4CCCCN4C)=O)CC3)cc2c1F 13367,Cc1cccc2c(C(=O)NC(C)C(C)NC(=O)COc3ccc(Cl)cc3)c[nH]c12 13368,C(=O)(CCCCC(F)(F)F)NC1CC(NC(c2ccnc(C3CC3)c2)=O)CC1O 13369,c1(-c2onc(-c3c(C)noc3C)n2)ccc2c(c1)C(=O)CC2 13370,C(=O)(CC(C1CC1)NC(C1C=CCS1)=O)N(C1CCOC1)CC#C 13371,N1(Cc2nnc(CC)s2)CCCOC(CNC(c2occ3c2CCC3)=O)C1 13372,CC1CCN(C(C23CC(C)(C2)C3)=O)CCN1C(=O)C(C)N1CCC1 13373,C1(C(=O)NC2CC2)CC(CO)N(C(c2cn(C)cn2)=O)C1.c1(CC)ccnc(O)c1 13374,Cc1cc(C(=O)OCC2(O)CCCOC2)cc(Br)c1C 13375,C=CCCCCCC(=O)NCC(CCCC)NC(=O)C(N1CCCCC1=O)C 13376,N1(C(=O)Cn2ccc(O)nc2=O)CCCC(n2cc(Cn3cncn3)nn2)CC1 13377,C1(NC(C(C)(F)CC2CCC2)=O)CCCC2CN(C(=O)CCOC(=N)O)CC12 13378,C#CC1(C(=O)NCc2ccn(C)n2)CCN(C(C2C(C(F)F)C2(C)C)=O)C1 13379,Cc1noc(C(C(C)C)NC(=O)C(C2CCN(C(=O)C(C)CN(C)C)C2)F)n1 13380,c1(CC(=O)NCC2(O)CC(NC(C(C(C)(C)C)O)=O)C2)c[nH]c(=N)nc1O 13381,C1(N(C(C(CCC)=CCC)=O)C)CCN(C(=O)CCCCOCC)CC1C 13382,C(=O)(C(CCNC(=O)CCCCSC)OC)N1CCC(N(C)CC)C1 13383,C(=O)(C(C)OC(C)=O)N(CC(C)NC(=O)NCC)C.C1(=O)CN1 13384,C(=O)(CCCCCO)N(C(C)C)CCN(C)C(c1coc(C2(C)CC2)n1)=O 13385,c1(CNC(=O)NC23CCC(NC(CCC(C)C)=O)(CC2)C3)ccc([N+](=O)[O-])cc1 13386,NS(=O)(=O)CCCC(=O)NCC1CCCCN1C(=O)CCN1CCCCC1 13387,N1(C(C=CCN(C)C(c2cccc(C(C)C)c2O)=O)=O)CCC12CC(O)C2 13388,C1(NC(C(CO)OC)=O)C2CCC(C2)C1C(=O)N(C)CC1CC1(F)F 13389,C(=O)(C1=CS(=O)CCC1)NCC1CC(NC(CCNS(CC)(=O)=O)=O)C1 13390,c1(C(=O)NCC2(F)CCN(C(CN3C(C)CCC3)=O)C2)nc2ncccn2n1 13391,c1(CNCc2cc(=O)n(O)c(O)n2)nc2c(s1)CN(C(F)(F)F)CC2 13392,C1(SC)CN(C(=O)CCc2cncs2)CC1NC(=O)CN1CCCCCC1 13393,C(C)(C)(CC(=O)NCCC1CC(NC(=O)CCN2CCCCC2)C1)SC 13394,c1(C(=O)NC(C)CN(C(=O)CCCCc2cnc[nH]2)C)cnc2ncccn12 13395,c1(C(N2CCC(N(C3CCCCC3)Cc3ccc(Cl)cc3)C2)=O)cccc(O)c1 13396,C#Cc1cccc(C(N2CCC(NC(c3ccc(S(C)(=O)=O)[nH]3)=O)C2)=O)c1C 13397,C#CCC(C)(C)C(=O)NC1CCC(CCNC(C2CCCOC2)=O)C1 13398,c1(C(N2CC3(CO)CCC2CC3)C(=O)NCC2CCCO2)ccc2ncnn2c1 13399,c1(C(=O)OC)nn(C)cc1C(=O)N(C)CCNC(C1CC(C)OC1=O)=O 13400,C1(NC(C2N(CC)CC2)=O)CCN(N2CCC(c3cccc(Cl)c3)C2)CC1 13401,CC(C(C(=O)N1CC(C)(S(CN)(=O)=O)C(C)C1)N1CCCC(O)C1)C(C)(C)C 13402,C1(F)(C(=O)NC2CN(C(c3ccco3)=O)C2)CCN(C(=O)C2CC2)C1 13403,c1(N2CC3CC(NC(CN4CCN(C)CC4)=O)C3C2)nc(Cl)nc2ccccc12 13404,C=CCCCC(=O)NCC(C)(C)Cn1cc(-c2ncccn2)nn1 13405,c1(CN2CCCC(CS(=O)(=O)NC)C2)cc2ccncc2s1 13406,c1(CC(=O)NCC2CN(C(c3ccc(OC)s3)=O)C3C2C3)cc(C)ccc1OC 13407,C(N=c1[nH]c(=NCc2ccc(C#N)o2)c2[nH]ccc2[nH]1)c1c(SC)cc(F)cc1 13408,n1(CC)nnc2c(N3CCCC3CCCNC(=O)C(C)(C)C(N)=O)ncnc12 13409,C(=O)(CC(C(F)F)n1ccnc1)N1CC(O)(CC(=O)NCCc2cc[nH]n2)C1 13410,c12cccc(c1)CCNC2.c1(-n2cc(-c3c(I)c[nH]n3)nn2)ccccc1N.C1CC1 13411,c1(C(N(C(C)CN(C)C(C2(CF)CC2)=O)C)=O)nccc(Br)c1O 13412,c1(C(N(CCCCN(C(=O)CCc2ccn(C)c2)C)C)=O)csc(C(C)(F)F)n1 13413,C1(NC(C2C3CNC(=O)C32)=O)CCN(C(=O)CC2(O)CCC2)C12CC2 13414,C(C(CC(C)C)C(=O)N1CC(n2cc(C(C)(C)CO)nn2)C(O)C1)SC 13415,C1(C)(C(=O)NCc2c(C(=O)NCc3ncc(CC)s3)[nH]cc2)CCC2CC2C1 13416,N(C(=NCC1CCCO1)NC1CC(c2ccc(F)cc2)C1)CC1(C)CCC1 13417,c1(OC)ccc(C(=O)Nc2cccc(CNC(=O)C(F)(F)C(F)F)c2)c(C)n1 13418,CC(C)C(C#N)C(=O)N1CCC(NC(c2cnc(-c3cnccn3)s2)=O)C12CC2 13419,c1(CNC23CC(C(=O)NCC4(F)COC4)(C2)C3)cccc(O)c1 13420,CC#CC1CN(C(C2CC(NC(=O)CCc3cscn3)CCO2)=O)C1 13421,C(CC1=CCCCC1)N(C(c1cc(Cl)cs1)C(=O)NCCCC)C 13422,N1(C(c2cnc(C)c(Cl)c2)=O)CC2CC1CCN2C(C1CC(=O)N(C2CC2)C1)=O 13423,c1(C(N2CCC(N(C)C(c3ccccn3)=O)C2)=O)ccc(CO)nc1 13424,N1(C(CCOCC#C)=O)CCC(C)N(C(=O)CCCCC(N)=O)CC1 13425,O=C(C1=CCCSC1)NCCCCCCNC(C1COCCO1)=O 13426,C1(CNC(COC2(C)CCCC2)=O)CCCCN1C(=O)CC1(C2CCC2)CC1 13427,c1(C(N(C)CCOCCNC(C2CCC23CCC3)=O)=O)cc2cccnc2cn1 13428,C1(C(=O)NCCC2(C)CCOC2)C=CCN(C(C2CCCC(=O)C2)=O)C1 13429,N1(C(CC2(C)CCNC2)=O)CCN(c2ccccc2F)CC1.C(C(=O)O)N 13430,C(=O)(CC(C)(C)C(F)F)N1CC2C(C(N(CC(CC)(C)OC)C)=O)(C2)C1 13431,C1(CCNC(Cc2c(C)noc2C)=O)CN(C(=O)CN2CCCC2)CC(C)O1 13432,C1(CC)CCC(C(=O)NCC=CCNC(c2ccoc2C(C)C)=O)O1 13433,c1(C(=O)NC2CCN(C(CC=CCC)=O)C2C(C)(C)C)ncnc2c1CCC2 13434,c1(C(=O)NC(C2CCN(C(=O)C(C)CC(C)(F)F)CC2)C)ccc2nncn2c1 13435,c1(NC(C(C(C)(C)C)O)=O)ccc2c(c1)CN(C(=O)CCN1CCOCC1)C2 13436,N1(C(C(C=C)C)=O)CCC=CC1C(N1CCOC(CO)C1)=O 13437,c1(C(=O)NC(C2CCCC2)CNC(C2C(C)=C2)=O)c(C)cc(C#N)cc1C 13438,CN1CC=C(C(=O)NCCC(c2ccccc2)N(C)C(C2CC3(CSC3)C2)=O)C1 13439,c1(C(N2CC(C(N)=O)(CNC(C(C)n3cncn3)=O)C2)=O)ccnc2[nH]ncc12 13440,c1(OC)ccc(CCNC(C2CN(C(=O)CN(c3ccccc3)C)C2)=O)c(C)c1 13441,Cc1[nH]nc(Cl)c1C(=O)NCC1CC(NC(=O)CCc2cn(C)nn2)CCO1 13442,N1(C(C(CC)(CC)CO)=O)CCOC2(CCCN(C(=O)CCCC3(C)N=N3)C2)C1 13443,c1(OC)ccc(C2CCN(C(=O)C(N3CCCCC3C3CCOCC3)=O)CC2)cc1 13444,c1(C(=O)NCCCNC(CCC=C)=O)ccc(NC=O)cc1.C12CC1N2 13445,Cc1cc([N+](=O)[O-])ccc1C(=O)NC(C)C(C(C)C)NC(c1sc(C)cc1Cl)=O 13446,c1(C(=O)NC2CC(CNC(C3=CCCC3C)=O)C2)n[nH]c2c1CCSC2 13447,C1(C(=O)NCC2(C)CC(NC(CC3(OC)CC3)=O)C2)CC(c2ccccc2)=NO1 13448,c1(C(N2C(C(C)NC(CN(CC)CC)=O)COCC2)=O)cc2ccccc2s1 13449,N1(CC(=O)NCC(C2CCSCC2)OC)C2CCC1CC(C(C)(C)C)C2 13450,C1(NC(C(N2CCC(C)(CCO)C2)c2ccc(CF)cc2)=O)CCC(F)(F)CC1 13451,CC(C)(O)C(C)(C)C(=O)N1CCCC1CNC(C1OCC2CCCC12)=O 13452,C1(C)(N(C)C(C2(CCNC(=O)CCCC3CCCC3)CC2)=O)CCCC1 13453,C(=O)(CC(CC(C)C)NC(c1cc[nH]c1C)=O)NCCC(CC)O 13454,c1(C(=O)NC(C)CN(C)C(C2CCCC23CC3)=O)cc2nc(=O)ccn2[nH]1 13455,C(=O)(C#Cc1ccccc1)N1C2CN(C(c3cc(NC(C)=O)ncn3)=O)CC21 13456,C1(C(=O)NC2CC(C(F)F)(NC(CC3(OC)CCC3)=O)C2)CC(C)CC(C)C1 13457,CC#CCC(C)NC(C1(CCNC(=O)CC(Cl)Cl)CC1)=O 13458,c1(C(=O)NC2CC(CNC(C3C(C)CC(=O)N3)=O)C2)cc(N)cnc1Cl 13459,c1(C(=O)NC2(CO)CN(CC)C2)cncc([N+](=O)[O-])c1.c1(CC=O)cnsc1 13460,C1(NC(COC2CCCC(C)C2)=O)(CNC(=O)C=CS(C)=O)CC2CCC1CC2 13461,C1(C(=O)NC2CC(NC(c3c(C)n[nH]c3)=O)CC2O)C(F)(F)C12CCC2 13462,c1(C(N(CCCNC(C(C)OCC#C)=O)C2CC2)=O)ccc2nccnc2c1 13463,C(C1=CCCOC1)NC(C1CCC(NCCCc2c[nH]ccc2=N)C1)=O 13464,N1(C(C=C(C)C)=O)C2CCC1C(CNC(=O)C(F)F)C2 13465,Cn1ccc(C(=O)NC(C2CCOC2)CNC(c2ccsc2)=O)c1C1CCC1 13466,C(C)(C)(CCN(C)C(c1cnc(C(C)(C)CF)o1)=O)NC(C1CC(OC)C1)=O 13467,c1(C(=O)NC2CC(F)(CNC(C(C)C3CCOC3)=O)C2)[nH]nc([N+](=O)[O-])c1Cl 13468,CC1C(NC(=O)CN2C(=O)CCC2=O)CCN1C(=O)Cc1ccccc1Cl 13469,N12CCSCC1C2.CC(CC1CC1)CON 13470,C#CC1(NC(C2CN(C3CCC3)C2)=O)CC2CCCC12.C12(CC1)C(=O)NC2 13471,C12(CNC(CCN(C(C)=O)C)=O)CC1CN(C(c1cc(-n3cccc3)ccn1)=O)C2 13472,C(=O)(C(CC(C)C)N(C)C)NCC(=O)NCc1cncc(C)c1 13473,N1(C(c2c(CC)n[nH]c2)=O)CC2CC2(CNC(=O)C(O)CC2CC2)C1 13474,n1(C(C)(C)C)cc([N+](=O)[O-])cn1.c12cn(nn1)CC1CCN1C(=O)CC2 13475,N1(C(c2c(C)nc(O)cc2)=O)CC2CCCC1C2CNC(C1(CO)CCCC1)=O 13476,N1(C(C(n2c(C)ccn2)C)=O)CCCC(N(C)C(c2ccnc(N(C)C)c2)=O)C1 13477,CCCCCC(C)CC(=O)N(C1CC(NC(C2C=CCS2)=O)C1)C 13478,C(=O)(CC(C)(C)O)N1CC(C(C(N2CC(OCC(C)C)C2)=O)O)C1 13479,Cc1cc(CNC(=O)C(CC2CCOCC2)NC(c2scnc2Cl)=O)n[nH]1 13480,C(=O)(C(CC(C)C)n1cc(CO)nn1)NC.C1(O)(C(C(=O)N)(F)F)CCCCC1 13481,C1(C(N(C)CC2CCN(C(=O)CN3CCCCC3=O)C2)=O)CCc2cnnn2C1 13482,C(=O)(CCCCC(=O)N1CC(NC(=O)CC2C(C)(C)C2(C)C)CC(C)(C)C1)OC 13483,c1(C(N(CCC)CC2CCOCC2)=O)ccc(Cl)nc1NC(C1CCCO1)=O 13484,C(=O)(CCC(=O)N1CCC(C(C)(O)CNC(=O)C(C)SC2CC2)CC1)NC 13485,C1(CCNC(C2CSCCS2)=O)CCCN(c2nc(C3CCCC3)ns2)C1 13486,C1(C)(CNC(C(N2CCCCC2)C)=O)CN(C(c2cnsc2)=O)C(C)(C)C1 13487,C1(N)(CNC(c2cc(COC)oc2C)=O)CCC(C)(C)CC1 13488,CC1CCC(NC(c2nnsc2C(F)F)=O)CN1C(=O)CCCCc1cnc[nH]1 13489,c1(OC)ccc(C(=O)NCCC2CCCN(C(=O)CCC(C)N(C)C)C2)c(N)c1 13490,Cn1nc(Cl)c(C(N2CC(CNC(=O)CSc3nncs3)C(F)(F)C2)=O)c1Cl 13491,N1(C(CCS(C)=O)=O)C2CCC1CC(NC(C1(CO)CCC1)=O)C2 13492,c1(C(CNC(c2cnc(O)s2)=O)NC(C(=O)NCC)=O)ccc(Cl)cc1 13493,c1(C(=O)NCC2CC(NC(CC=C=C)=O)C(O)C2)cc(Br)cc([N+](=O)[O-])c1Cl 13494,CCC(CC(=O)NCCC1CC(NC(C2CCCSC2C)=O)C1)c1ccccc1 13495,c1(C(N2CCC(N(C(=O)C=Cc3cnc[nH]3)C)CC2)=O)ccc(Br)cc1[N+](=O)[O-] 13496,C1(C(=O)NC2(CO)CCN(C(Cc3c(C)nc(C)s3)=O)C2)CCCCC12CCC2 13497,C(=O)(C1CCCc2ncccc21)N(C)CC1CCCN1C(c1cc(Cl)ns1)=O 13498,c1(NC(C2(O)CCN(Cc3cccc(-c4cnoc4)c3)C2)=O)cc(Br)ccc1Br 13499,C1(NC(c2cc(Cl)cnn2)=O)C2CCC1N(C(=O)Cc1cccc(F)c1O)C2 13500,N1(C(CSCC)=O)CCN(C(c2cnn(C)c2C(C)C)=O)CC1CC(F)F 13501,N1(C(C2CN(CCC)C(=O)C2)=O)CC(NC(=O)CC2(OC)CC2)CC12CCCC2 13502,C1(C(N2C(CNS(C)(=O)=O)CCC2)=O)Cc2ccccc2N1 13503,C1(NC(CCCCSC)=O)COC2(C1)CN(Cc1c(C)noc1C)C2 13504,N1(C(CSCC(=O)OC)=O)CCCC(F)(C(=O)NCCCCNC)C1 13505,C1(NC(C(CC)(C)OC)=O)CCCCN(C(c2ccc(C)nc2N)=O)C1 13506,CON1CCC(=O)NON2C(C3CC3C)=C(C1=O)C2.C1(C)CCCCO1 13507,N1(C(C2C(CC)OCC2)=O)CC2CC(NC(=O)C(c3ccc(F)cc3)(F)F)C1C2 13508,N1(C(CC2(C)CC2)=O)CCC(CNC(c2ccn3cnnc3c2)=O)C12CCC2 13509,N1(C(C(=O)NCC)=O)CC(F)(CNC(C2(CC)CC2(F)F)=O)C1 13510,N1(C(C(CC=C)C)=O)CCC(CNC(=O)CCSc2nccn2C)C(F)(F)C1 13511,CC(CF)CC(=O)NCC1CC1CNC(c1cc(-n2ccnc2)ccn1)=O 13512,N1(C(Cc2c(C)ncs2)=O)CC2(CCC2NC(C2COC(C)(C)CO2)=O)C1 13513,C(=O)(C(N=[N+]=[N-])C(C)C)N1CCN(C(C2C(C(=O)OC)COC2)=O)CC1CF 13514,c1(C(N(C2CCCC2)CCCNC(C2C(C)(C)CC2)=O)=O)cc[n+]([O-])cc1 13515,c1(OCCC(=O)NCC2(NC(=O)C=CCF)CCCC2)ccc(F)cc1Br 13516,C(N=c1[nH]cnc2ccc(O)cc12)C12CC(NC(CC)=O)(C1)C(C)O2 13517,n1(C(C)C)ccc(C(=O)NC(C)(C)C(=O)NC(C2CCC2)C)n1 13518,CC12COCC1CN(C(c1cc(Cl)cc(I)c1)C(=O)Nc1ccccc1)C2 13519,c1(C(C(=O)NC(C2N(C(CC(=O)OCC)=O)CCC2)C)O)cccc(C)c1Br 13520,N1(CC)CCN(c2ncc(Cl)s2)C(C)(C)CC1 13521,C1(CC)CCCC(N=c2nc3scnc3c(NCc3c[nH]nc3C)[nH]2)CC1 13522,c1(C(=O)NC(CC)CN(C(=O)Cc2cccnc2)CC)cn(C)nc1CSC 13523,C1(NC(C(C)CC2CCC2)=O)CN(C(=O)CCC=Cc2ccccc2)CCC1C 13524,Cc1nn(C)c(F)c1C(=O)NCC(C)NC(=O)C(n1ccc(C(F)(F)F)n1)C 13525,Cn1nc(C(F)(F)F)cc1NC(=O)NCCC(O)C(=O)NC1CC=CC1 13526,C1(C(CNC(C2(OC)CC2)=O)NC(C2CCOCC2)=O)CCCCC1 13527,N1(C(c2n(COC)ncc2)=O)CCC(C)C(CNC(c2nc(Cl)cs2)=O)C1 13528,N1(C(C(C2CCOCC2)C)=O)CC2(CC(NC(=O)CC34CC3COC4(C)C)C2)C1 13529,c1(C(N2CC(NC(c3cc(OC)c(C(F)F)cc3)=O)C2)=O)cc2n(n1)CCO2 13530,Cc1cccc(C(N2CC(O)(C(C)NC(c3ncccc3N)=O)C2)=O)c1C 13531,c1(OC)[nH]c(=NC2CCCCCN(C(=O)C(=O)NC(C)C)C2)sc1C 13532,C1(CNC(C2N(CC)CCCC2)=O)CN(C(C2(CC3CC3)CC2)=O)CC12CCC2 13533,c1(N2CCC3(CC(OCC)C3)C2)nc(N2CCN(CCF)CC2)nc2sccc12 13534,CC(CCCC(=O)NCc1cccc(CO)c1)NC(c1cccc(CO)c1)=O 13535,C1(C)(C(=O)NCCCN(C(C2CC(C(=O)OC)C2)=O)C2CC2)CCCNS1(=O)=O 13536,c1(N(C(=O)OC(C)(C)C)C2CC2)cnn(C)c1.C1(=O)CCN(C)CC1=O 13537,c1(CC)[nH]ccc1C(=O)N(CC(=O)N(C)C(C1CCC1)C)C1CC1 13538,c1(C(C(=O)N(Cc2cc(I)cs2)CC2CC2)F)ccc(C(F)(F)F)cc1 13539,Cc1csc(=O)n1CCC(N1CC2CC2(NC(=O)COCCF)C1)=O 13540,C1(C(=O)NC2C3CN(C(C4(C(=O)OC)CC4)=O)C2C3)Cc2ccc(F)cc2O1 13541,N1(C(c2c(CC)scc2)=O)CCCC(CO)(NC(=O)CNc2nccs2)C1 13542,C1(N(C(C2C(OC)CC2)=O)C2CC2)CCCN(C(c2ccc(O)c(Cl)n2)=O)CC1 13543,c1(CC)ncc(C(=O)NC(CNC(C2CC3C=CC2O3)=O)CCOC)c(O)n1 13544,C1(C(N2CCCCC2)=O)CCCN(C(=O)COC(C2CCC2)C2CC2)C1 13545,C1(OCC(C(F)(F)F)NC(C)=O)CCCN(C(=O)Nc2ccc(Cl)cc2)C1 13546,Cc1cc(C(=O)NCC2CN(C(c3cn(C)nc3C(C)C)=O)CC2C)ccn1 13547,C1(NC(C(c2ccc(C)cc2)=O)=O)CCCN(C(=O)CC(O)C(C)C)CC1 13548,C1(NC(=O)NCCC(CSC)(C)C)OCCCCCC1c1ccccc1 13549,c1(C(N2CCC(C(C)C(=O)NCC(C)(C)O)CC2)=O)ccc(C#N)cn1 13550,c1(C(=O)NC(C(C)NC(C2C(OCC)C2C)=O)C)cnc2c(c1)nnn2C 13551,n1(CC(=O)C2(C(=O)O)CC2)nc(C)cc1C.C(CCNC(=O)NC)NCCN 13552,Cc1coc(C)c1CNC(=O)C(C)N(C(=O)C(c1ccccc1)=O)C1CCCC1 13553,N1(CC(=O)NCCCN(C2CCCC2)C(C=C(COC)C)=O)CC2CC2C1 13554,c1(OC)cnc(Br)cc1C(N1CCN(Cc2cnn(C)c2)CC1CC#N)=O 13555,C1(C(N2CC(O)(CNC(c3c(C)cc[nH]3)=O)C2)=O)C2C(=O)OCC12Br 13556,c1(CC(=O)NC2CC(NC(=O)C(F)=CC3CC3)C2)noc2ccccc12 13557,Cc1cc(C(=O)NC2CCCC(NC(C3C4CCCOC34)=O)C2)cc2ccsc12 13558,C(c1ccccc1)=C(C)C(N1CC2CC2(C(=O)NC(C)(C)C(F)(F)F)C1)=O 13559,C1(CC(N2C(CNC(c3cn(CCO)nn3)=O)CC2)=O)CC(=O)c2ccccc2C1 13560,C#Cc1ccc(NC(C2CC(F)(F)CN2c2nccc(C)n2)=O)cc1Cl 13561,C1(CNC(C(N2CCC(O)CC2)C)=O)CCN(C(=O)CNC(N)=O)C12CC2 13562,CN1CCC(CCC(=O)NCCC2CCCN2C(c2cc(C3CC3)on2)=O)CC1 13563,N1(C(c2c(CC(=O)OC)cccc2)=O)CC2CC(Nc3nnco3)CC2C1 13564,C1(Nc2ccn(C3CN(C(=O)OC(C)(C)C)C3)n2)CCCC12CC2 13565,C1(NC(Cn2ncn(C)c2=O)=O)CCN(c2cc(C(F)F)ncn2)CC1O 13566,C(=O)(C(C)(CC)C(N)=O)N1CCCC(N(C(=O)COc2cc(F)ccc2F)CC)C1 13567,n1(CCOC)cc(C(=O)NC2CC2CNC(c2ccc(O)cn2)=O)c(C)n1 13568,C(=O)(CCC(C)(C)F)NC1C(C)CN(C(c2ccc(N3CCCC3)nc2)=O)C1 13569,C=CC1CN(C(=O)C=CCC2(NC(=O)CNC(N)=O)CCC2)CCO1 13570,C1(C(=O)NC2(CC(N)=O)CCC2)CCC2(CC2)N1C(c1cnc(O)o1)=O 13571,N1(C(C(C)CC2CC2)=O)CCCC(C(=O)NC(C)(C)C(F)(F)F)CC1 13572,C1(C)(CC)NC(=O)N(CC(=O)OCCCOc2ccc(Cl)cc2C(F)(F)F)C1=O 13573,c1(C(C)N(C)C)cn(CC(=O)NOCC2CCN(C)C2)nn1 13574,CCC(CC(C)C)C(=O)NCC1CN(C(c2ccc(C#N)nc2O)=O)CCO1 13575,CC1CCC(C(=O)N(C)Cc2nnnn2C)N1C(c1ccn(C)n1)=O 13576,N1(C(c2[nH]c(=NC)sc2)=O)CC(N(C(=O)CCNC(C)=O)C)C(C)(C)C1 13577,C=CCCCC(C(=O)NC(C)CCCNC(=O)C1=NOC(C)C1)NC(C)=O 13578,Cc1cc(C(=O)N(C2CC(NC(C3(SC(C)(C)C)CC3)=O)C2)C)n(C2CCC2)n1 13579,CCCC(C(=O)N1CC(NC(C2(C3CCCCO3)CCOCC2)=O)C1)OCC 13580,c1(C(=O)NCC(C)CNC(c2cnn(C)c2)=O)c(F)ccc(C(F)(F)F)c1F 13581,N1(C(c2cnc(OCC)s2)=O)CCCC(O)(CNC(=O)C2=C(Cl)CCOC2)CC1 13582,Cc1cc(NC(c2ccc(CNC(c3cnns3)=O)s2)=O)c(O)cc1F 13583,c1(CNC(C2CC(OCC)C2)=O)ccnc(C(=O)Nc2cccnc2C)c1 13584,C12(CNC(C3(CO)CCC3)=O)CC1CN(C(=O)COC1CCC1)C2 13585,N1(C(CCC(C)C)=O)CCCC2C1CCCCN2C(c1cscc1F)=O 13586,C(=O)(C(F)C(F)(F)F)NC1CC(N(C(c2cc(N3CCCCC3)ncn2)=O)CO)C1 13587,N1(Cc2c(CC)cc(Cl)cc2)CCCC2C1CCN2C(=O)CN1C(=O)C=CC1=O 13588,C12(CNC(C=CC(C)(C)C)=O)CCC(CC1)CN2C(C1CC12CCC2)=O 13589,N1(C(CC(=O)OC)=O)CC(C(=O)Nc2c(CO)noc2C)CC12CCC2 13590,C1(C(C)C)C(C(=O)O)CCN1C(c1ccccc1Cl)=O.C12CCN(C1)C2 13591,CC1=C(C(=O)N2CC(CNC(=O)CN3CCSCC3)CC(C)C2)CCCO1 13592,CCC(CC(=O)N1CC2CN(C(c3c[nH]c(=NC)o3)=O)CC2C1)C(C)C 13593,N1(C(=O)CC2CCC3CC3C2)CC23CCCC2(C1)CN(C(C1CCC=CO1)=O)C3 13594,C1(CCNC(CC2(CC)CCC2)=O)C(C)CCCN1C(c1ccc(C)nn1)=O 13595,C(C(C)(C(C)C)C(C)C)NC(CC1C(C)CN(C(=O)C=Cc2nccs2)C1)=O 13596,c1(C(=O)NC2CN(C(c3cnc(SC)nc3)=O)CC23CC3)ccc2cc[nH]c2n1 13597,c1(OC)cc(C(=O)NC2CCC(NC(=O)Cn3cc(Cl)cn3)CC2)ccc1[N+](=O)[O-] 13598,c1(-n2cc(CC(C(N)=O)NC(C3CCOC3)=O)nn2)cc2c(O)ncnc2cn1 13599,c1(CC)nccnc1C(N1CCCCC1CCCNC(C1(C)CCC(=O)N1)=O)=O 13600,C(C(C)(C)C(=O)N1CCC(OCC2(C)CCCN2C(C)=O)C1)SC 13601,c1(C(=O)NN(CC(C)NC(C2CN(C(C)=O)C2)=O)C2CC2)ccc(C)c(Br)c1 13602,Cc1ccc(C#N)cc1C(N1CC2CC1CCC2NC(=O)C(F)(F)C(F)F)=O 13603,C1(NC(CC2C(C)CCO2)=O)CCN(C(c2cccc(C(C)(F)F)c2)=O)C(C)C1 13604,Cc1conc1C(=O)NCC1CC1CNC(c1ccc(-c2ccccn2)s1)=O 13605,N1(C(C(CC2CCC2)OC)=O)CC(CC(N2CCCC(CC3CC3)C2)=O)CC1C 13606,c1(C(N(C(C)CCNC(C2SC3C=CC2CC3)=O)C)=O)cc2ccc(Cl)cc2o1 13607,c1(CCC)cc(C(=O)N(CCC(C)NC(=O)CC2COC(C)(C)C2)C)cc(O)n1 13608,c1(CC)ccccc1NC(C1N2C(CCCC2)CN(C)C2CCCC21)=O.SC.SC 13609,c1(SC)cccc(C(=O)NCCN(C(c2cnc(S)[nH]2)=O)C2CC2)c1 13610,c1(C(CNC(=O)CCn2cccn2)NC(CNS(NC)(=O)=O)=O)ccccc1Cl 13611,Fc1cc([N+](=O)[O-])ccc1-c1ccc(NCC2COCC2N)cc1 13612,C(=O)(C(C)(C)C(N)=O)NC1CCC(C)(CNC(C2(c3cccnc3)CC2)=O)C1 13613,c1(OC)ccc(C(=O)NC2CC(C(=O)Nc3cnc(O)c(F)c3)C2)cc1C 13614,Cc1cc(C(=O)NC2CCCN(C(C3CCN(C)C3)=O)C2)cc([N+](=O)[O-])c1O 13615,c1(OC)ccc(CC(=O)NC2CC(C)(NC(=O)CCc3ccccn3)C2)cn1 13616,C(=O)(C1=CCCOCC1)N(CCNC(c1c(C)oc(Br)c1)=O)C 13617,C1(CCNC(=O)NC(c2ncc(C)s2)C)CCCN(S(C)(=O)=O)C1 13618,C(=O)(C(C)(C)CNC(=O)COC(=O)CO)N(CCCC)CC 13619,n1(CC)cnc2c(N3CCCC3c3ccc(F)cn3)nc(N3CC(F)C(F)C3)nc12 13620,N1(C(C(C2CCC2)OCC)=O)CCC2C(NC(=O)Cc3c[nH]nc3C)C2C1 13621,CN1C(C)(COCNc2ccccc2)CCS1(=O)=O.C1C(C)(O)CNC(=O)N1 13622,CCCCCCCC(CC(=O)N1CC(C(=O)NOC)Oc2ccccc21)SC 13623,C(=O)(C(C)CCCC)N1CC(CC(=O)NCC=CC)OCC1 13624,CCCC(O)(CCC)CC(=O)NC(C)(CNC(c1ccc(C)o1)=O)C1CC1 13625,N1(C(Cc2c(C)non2)=O)CC(NC(=O)CCC2CCCC2)CCC1C 13626,C=CC(F)(F)C(=O)NCC(O)CC(=O)N(C)CC1CCOC1C 13627,c1(C(=O)NCc2cn(CC(C)NC(=O)CO)nn2)ccc2[nH]c(=N)sc2c1.C1(C)CC1 13628,C1(CNC(c2cn(C)cc2C(F)(F)F)=O)COCCN(C(C2(O)CC2(C)C)=O)C1 13629,c1(C(=O)NC(CC(C)NC(c2c(OC)ccs2)=O)C)ccc(-c2cccs2)cn1 13630,C1(NC(C2(CNC(CSCCC)=O)CC(C)(C)C2)=O)CC2(CCC2)C1O 13631,N1(C(C2(COC)CCCCC2)=O)CCOCC(NC(c2cncnc2)=O)C1 13632,Cc1nc(-c2ccccc2)c(CNC2CCCN(C(=O)C=Cc3cnc[nH]3)C2)o1 13633,C1(C(C)(C)C)(C(=O)NCCc2cc(C(F)F)no2)NC1=O 13634,N1(C(C(C)n2cccc2)=O)CC(C(=O)NCc2ccnc(F)c2F)C2(CCC2)C1 13635,N1(C(c2ccc(C)s2)=O)CCc2nc(CNC(=O)C(C)(C)C3CC3)sc2C1 13636,c1(C(=O)NCC(CCOC)NC(C2(C(=O)OC)C(=C)CC2)=O)cnc(C)n1C 13637,Cc1cc(C)c(C(N2CCN(C(c3cnc(S)[nH]3)=O)CC2CC(F)F)=O)cc1N 13638,Cc1cc(CC(=O)NC(CNC(=O)Cc2[nH]cnc2C)C(C)C)n(C)n1 13639,C1(C2CCC2)(C(=O)NCC(C)NC(=O)COc2cccnc2)CC1(F)F 13640,C1(CN(C(C(C=C)C)=O)C)CN(C(=O)Cc2cc(C)cs2)CC12CC2 13641,O=C1CCC(S(=O)(=O)NC2CCC(CC(=O)NC(C3CCC(F)C3)=O)CC2)CC1 13642,Cc1nccc(CCNC(C2(CNC(C3CCCN3C=O)=O)CC23CCC3)=O)n1 13643,C1(CC)CC(C(N2CCCC2(CNC(C2CCOCC2)=O)COC)=O)CC(=O)N1 13644,Cc1cc(C(=O)NCC2N(C(C3CC(O)C3)=O)CCC2(C)C)cnc1O 13645,C12(CNC(CC3C(CC)C3)=O)CC(NC(c3scnc3Br)=O)(C1)C2 13646,C(c1nc(C)co1)=CC(=O)NCCC(=C)CNC(C1CC(CC)C1)=O 13647,c1(C(CNC(C2(C=C)CC2)=O)NC(=O)C(C)(C)c2cncnc2)cccc(Cl)c1 13648,c1(OC)sccc1C(=O)N(C)CC=CC(=O)NC(C)C(C)F 13649,C1(CNC(Cc2c(C)cco2)=O)CC(NC(=O)COc2ccccc2)CC1O 13650,N1(C(c2cc(=NCC)[nH]cc2)=O)CCN(C(c2csnn2)=O)C2CCCC2(C)C1 13651,C1(CNC(C2(C#C)CCCC2)=O)CN(C)CCN1C(c1cc(C(C)C)on1)=O 13652,C(C(CC(=O)NC1CCN(C(=O)Cc2ccn(C(F)F)n2)C1)C(F)(F)F)N(C)C 13653,Cc1cc(Cl)cnc1S(=O)(=O)N1CCSC(Cn2ccnc2)C1 13654,c1(OC)ccnc(C2CCCN2CC(=O)NC2CCC(C)CC2)n1 13655,CCC(C)(O)C(=O)N1CC2CC2(C(N2CCC(C(C)CO)CC2)=O)C1 13656,N1(C(C(CC)C#N)=O)CC(C(=O)NCC(=O)N(C)C)C2(CC2)C1 13657,Cc1cc(C(=O)NCC2CCCN2C(=O)C2CC2)cc(C)c1F 13658,N1(C(c2ncc(C)s2)C(=O)NCC=C)CCC(C(CC)NC)CC1.OC 13659,N1(C(COCC(C)C)=O)CC2OCC(NC(=O)CC3CCCCC3(F)F)C2C1 13660,N1(C(CSCCOC)=O)CCC2(C1)CN(C(=O)Cc1ccnn1C(C)C)CC(C)O2 13661,O=C(CC1CCN1C(c1c[nH]c2ccccc12)=O)N=c1cc(C(F)(F)F)[nH][nH]1 13662,c1(C(=O)NCCCN(C(=O)CCCc2cn(C)nn2)CC)coc(SC)c1 13663,c12cc(cc(Cl)c1)N2.N12CCC(C1)C(=O)NCC2=O.CCSCC 13664,C1(NC(C2C(C(N)=O)C2)=O)CC2CCCC(C1)C2NC(C1CN2CCC1CC2)=O 13665,Cc1cc(=NC(=O)C(=O)N2CCN(C(=O)Cc3occc3C)CC3(CC3)C2)[nH]o1 13666,CC1(C(N2CCC3(CCC3)C2)=O)CCN(S(=O)(=O)CCCC#N)CC1 13667,C(C(C(C)C(C)C)NC(=O)C(O)C1CCC1)NC(C(c1cccc(C)c1)(F)F)=O 13668,CN1CC(C)(C)CC1C(N1CCCCC1C(N1CCC(O)C(O)C1)=O)=O 13669,C1(C(N2CCC(CCC(=O)NC(C#C)(CC)CC)C2)=O)CCC(C#N)CC1 13670,CC(F)(F)C(F)C(=O)N1CCC(CN(C)CC2CCCCC2)C1 13671,C1(CNC(CCCOCC=C)=O)CC2CCC1N2C(=O)CC1CC1CC 13672,CN1CCn2cc(C(N3CCCC4CN(C(C5(C)CC5)=O)CCC34)=O)nc2C1=O 13673,C(=O)(C(C)S(=O)(=O)C(C)C)NC(CCCNC(c1c(C)onc1Br)=O)C 13674,N1(C(c2c(CC)c(C(=O)OC)c(C)[nH]2)=O)CC2CC(NC(=O)CC3(C)CC3)CC2C1 13675,CC1CC(NC(=O)Cc2sc(O)nc2O)CN(C(=O)C(C2CCOCC2)O)C1 13676,C1(CCN(CC(C)(C)C)C(=O)CNC)COC(C)C1.C1(C(C)=O)(C(=O)OC)CCC1 13677,N1(C(c2ncn(C)c2)=O)CCCCC(NC(C2OCC3CCCC23)=O)C1 13678,CCCCCCCCOCC(N1CCCC1CCCNC(=O)CC1CCC(C)C1)=O 13679,c1(C(N(c2cc(C)cc(OC)c2OC)C)=O)ccc2c(c1)N(C)C(=O)C2 13680,C1(C(C)C)(NC(c2ncc(-c3ccc(Br)cc3)o2)=O)CNC(=O)C1 13681,C(=O)(CCCC(OC)OC)NCCC(CNC(c1nc(CCC)oc1)=O)O 13682,C1(NC(c2ncc[nH]c2=O)=O)CC12CCN(C(c1ccc3ncccn13)=O)CC2 13683,c1(Cc2nc(C)sc2)ccnc(Nc2cc(N(C)CC3CCCCC3O)ncn2)c1 13684,C(=O)(C(Cc1cnc[nH]1)NC(C1CCOCC1)=O)NCCC=C 13685,c1(C(=O)Nc2c(F)ccc(OCCC)c2)c2c(nn1C)CCNC2 13686,c1(C(=O)NCC2CCN(C(COCCC#C)=O)CC2)ccnc2ncnn12 13687,c1(C(N2CC(CNC(C3CC3F)=O)CC(C)(C)C2)=O)ccc2c(c1)NS(=O)(=O)C2 13688,C(=O)(C#CC1CCCCO1)N(CCNC(CNC(N)=O)=O)Cc1ccccc1 13689,C1(C(N(C(CN(C(C=C(C)C2CC2)=O)C)C)C)=O)(CO)CCOC1 13690,c1(COC(C2(CC#C)CCCN2C(C)=O)=O)sccc1S(C)(=O)=O 13691,c1(-c2cc(C(=O)OCC)cc(F)c2F)n[nH]c2c1CN(C(=O)CC(F)(F)F)CC2 13692,N1(S(=O)(=O)Cc2cccnn2)CC(C(F)(F)F)C2(CCC2)C1 13693,c1(CO)cc(F)ccc1Oc1ccccc1CN(C=O)Cc1cc(Br)cs1 13694,c1(N(CC(CC)O)C)ccc(Br)c(S(=O)(=O)N(CC)Cc2ccsc2)n1 13695,C(=O)(C#CC1(C)CCCO1)OC(C)(C)C.C12CC(C)(C1)C1(CCC1)N(C)C(=O)N2 13696,C1(NC(CCC(C)OC)=O)CCCN(C(C2CCC(C)C(C)C2)=O)C1C 13697,C1(C(=O)NCC2(C(=O)NCC(COCC)O)CC=CC2)CC2CCCC2C1 13698,C=CCCCCC(=O)NCC(CCC)C(=O)NC1CC1c1cncn1C 13699,Cn1nc(C(F)F)cc1NC(=O)NC(CNC(=O)C(F)(F)CCl)C(C)(C)C 13700,CCCCCC(C(=O)NC1CC2CC1N(C(=O)CCCCC1CC1)C2)C(C)C 13701,N1(C(c2c(C)cccc2Cl)C(=O)NCCC2(C)CC2)CCOCC12CCOC2 13702,C12(C(N3CCN(C(c4c(C)occ4)=O)C(C)C3)=O)CCC(C)(CC1)OC2 13703,C(=O)(CC1NC(=O)c2ccccc21)NC1C(C)CN(C(C2CCC(F)CC2)=O)C1 13704,c1(N2C(C3(NC(c4cc(C)n(C)n4)=O)CC3)CCC2)ncnc2c1SCCC2 13705,C1(CN(C(=O)COc2ccsn2)C)CCCN(CC2CN(S(CC)(=O)=O)C2)C1 13706,c1(-c2cc(NC(N3CCC3C(c3ccccc3)=O)=O)sn2)cccc(Cl)c1 13707,N1(C(C(CC)CC)=O)CCN(C(c2cnn(-c3ccccc3)c2F)=O)C2CC12 13708,C1(NC(C(C)OC2CCOC2)=O)CCCC(NC(c2c(Cl)cnn2C)=O)C1 13709,C1(NC(C2=C(C)OCC2)=O)CCN(C(c2nc(C)n(C)n2)=O)CC12CCC2 13710,Cc1ncccc1C(=O)NC1CCC(CC(N2CCCC(CCO)C2)=O)C1 13711,C1(C(=O)OC)CCN(N2CC3C=CCOC3C2)C1 13712,Cc1cc(C(N2CCC(O)C(NC(c3ccc(C)n3C)=O)C2)=O)c(S(N)(=O)=O)s1 13713,N1(C(CC2CN(C(C#C)=O)C2)=O)CC(C#C)(CCC(=O)N(CCC(O)CO)C)C1 13714,C1(C(N2CCC(C(N)=O)C2)=O)(CC)CCCN1C(=O)C=CCO.C1CO1 13715,c1(N2CCCC(CN(C)C)C2)nc2ccccc2nc1NCC1CCC1(F)F 13716,c1(NC(C=Cc2c(Nc3cc(OC)cc(F)c3)cccc2)=O)ncc2cn[nH]c2n1 13717,c1(N2CCCC(C)C2)nc(=NCCc2nncs2)[nH]c2c1CCCCCC2 13718,C=C=CCC(=O)NCC1CCC1NC(=O)Cc1cnn(C(C)C)c1 13719,c1(OCC(C)Cc2ccccn2)cc(C(F)(F)F)nc(C(F)(F)F)c1 13720,C1(C(=O)NCC2CCC(NC(C3CC4(CSC4)C3)=O)C2)CCCNC1=O 13721,Cc1c(Cl)ccnc1C(=O)NC1CCC(F)(CNC(=O)C=C2CCSCC2)C1 13722,c1(C(=O)NC2C(C)CN(C(=O)Cc3cnoc3)CC2)c(F)ccc2occc12 13723,N1(CC(C)NC2C3CCCC2CC3)C(=O)NC2(CCCCC2)C1=O 13724,N1(C(=O)COC(F)(F)F)C2CCC1C(CNC(C1(c3ccccc3)CC1)=O)C2 13725,C1(CNC(Cc2ccc(OC)c(Br)c2)=O)CCc2nccn2C1 13726,N1(C(c2ccc(N(CCCC)C)cc2)=O)CC2CC1CCN2C(=O)CCS(C)=O 13727,C1N=C2N=c3sccc3=C(N2)NCC2CC12.c1(CCCC(F)(F)F)cccs1 13728,Cc1noc2nc(C(N3CC(NC(=O)Cc4cccn4C)CC3C)=O)ccc12 13729,C=Cc1cc(C(N2CCC(NC(=O)CCSCCCC)C2CC)=O)cc(F)c1 13730,C(=O)(CCC(=O)NN(C)C)NCCC1(O)CCN(C(C(=O)NCC)=O)C1 13731,c1(CC(=O)N(CC(C)(C)CNC(C2CCCCC2O)=O)CC)cccc(SC)c1 13732,C#CCC(CC(=O)Nn1cnn(C)c1=S)NC(c1cnc(O)o1)=O 13733,c1(NC(CC2N(C(C(CC)OCC)=O)CCC2)=O)ccc2nonc2c1 13734,C1(C(=O)NCC=C(C)C(F)F)(NC(=O)CCOCC(C)(C)C)CC1(C)C 13735,C1(NC(CCC=CC(C)C)=O)CCCC(N(C)C(c2csc(C(N)=O)n2)=O)C1 13736,c1(NC(=O)NCC(CNC(=O)Cc2nnc(O)s2)OC)ccccc1C 13737,c1(NC(=O)C(=O)NCCOC(C)CC(C)(C)O)ccc(I)cc1Br 13738,Cn1c(C(=O)NC2CC2CNC(c2cc3ncccc3[nH]2)=O)cc2sccc12 13739,C1(CC(=O)NC(C(=O)NC(CC)C2CCC2)Cc2cc[nH]n2)CCCC12CC2 13740,C1(NC(C2(C)CC(=C)C2)=O)CCCC(NC(c2cccc(C(=O)NC)n2)=O)CC1 13741,CC1(CNC(C2CCC(=O)N2)=O)CCN(C(C2CCCN2N=O)=O)C1 13742,C1(C)(NC(C(C)SCC)=O)CCN(C(C2CCCC2(C)C)=O)CC1 13743,CC1CN(C(=O)Cc2cnns2)CCC1CNC(=O)C(C)SCc1ccccc1 13744,c1(CC(=O)N(C(COC(C(C2CCCCC2)NC)=O)=O)C)ccc(Br)cc1 13745,N1(C(C(C)SC(F)(F)F)=O)CCC(C(C)CNC(c2scnc2C(F)(F)F)=O)C1 13746,C1(CNC(COCc2n(C)ccn2)=O)CN(C(=O)CC2CCOC2)CCC1(C)C 13747,Cc1nnc2n1CCC2(C)C(=O)NCC1C=CCN1C(c1ccsc1)=O 13748,C(CCC1CC1)(C(=O)c1scc(C)c1C(=O)OC)NCC1(SCC)CC1CO 13749,CCC(C)C(O)C(C)C(=O)N1CC(NC(c2cnc(COC)s2)=O)C2(CC2)C1 13750,CC1CCC(F)(C(=O)NCC(C)(C)OCC(=O)NCCCCCCC2CC2)CC1 13751,c1(C(N2C(C(C)(C)NC(c3cncc(O)c3)=O)CCC2)=O)cc(F)c(N)c(F)c1 13752,C(=O)(C(CO)C(C)C)NC12CC(CNC(C=C(C)C(C)(C)C)=O)(C1)C2 13753,C(=O)(CCCCc1cnc[nH]1)NCCCC1N(C(C(C)n2ccnn2)=O)CCC1 13754,C(C(CN=c1[nH]c(N2CCC(C)(C)CCCC2)nc2c1CCCCC2)OC)OC 13755,CC1C2CC(C2NC(c2cnc(-c3ccc(Cl)cc3)s2)=O)N1C(C1(F)CC1)=O 13756,N1(C(C23C(C(N)=O)(CCC2)C3)=O)CCC2C(NC(c3ccn(CCF)n3)=O)CC12 13757,N1(C(Cc2ccn(C)n2)=O)CC2CC(C(=O)Nc3ccccc3C(C)(F)F)C1C2 13758,N(C1CCCn2ncnc21)C(C(C)NC(C1CN(C2COC2)C1)=O)=O 13759,N1(C(CCN(C(C2C(C)C3CCC2C3)=O)C2CC2)=O)CCCC2CCCCC12 13760,C(CC1=CCN(C(c2nc3cnccc3s2)=O)CC1)NC(CCN(C)CC)=O 13761,Cc1nc(NC(c2ccc(-c3ccccc3[N+](=O)[O-])nn2)=O)ccc1[N+](=O)[O-] 13762,C1(C(=O)NCC2C(NC(=O)CC34CC(C3)C4)CCC2)CCCN1c1ncccn1 13763,c1(NC2(OC)CCN(c3ncc(Br)cn3)CC2)nc2ccc(I)cc2s1 13764,CN(CCCC(=O)N1CCOC(CCCNC(C2(C)COCCO2)=O)C1)N=O 13765,n1(CC)ncc(C(=O)NC2CN(C(C3CC3Br)=O)CC2F)c1C 13766,C1(CNC(CCNC(=O)OCC)=O)CCN(C(C23CCC(C2)C3)=O)C(C)C1 13767,CC(O)C(C)(C)C(=O)N1C2CCC1C(CNC(=O)C(C)(C)Oc1ccccc1)C2 13768,c1(NC(C(C)OCC=C)=O)[nH]nnc1C 13769,C(C)(CCC(=O)NC(COC)C(=O)N(CC(F)(F)Cl)C)OCC 13770,c1(C(N(C2CC(C(N3CC4CCC3CC4)=O)C2)C)=O)cc(I)c(O)c(I)c1 13771,N1(C(C2(CC)COC2)=O)CCC(C)(NC(=O)CCc2cccc(NC(N)=O)c2)C1 13772,N1(C(c2ccc(N(CCCC)CC)nc2)=O)CCC(NC(=O)CCC(C)O)C1(C)C 13773,CCC(O)CC(=O)N(CC(=O)NC(c1cnc(C)s1)C)C1CCC1 13774,C(=O)(CCCCC(=O)NCCC1CCCN(C(=O)COc2cccnc2)C1)OC 13775,Cc1cccc2cc(C(N3CCCCC3CNC(=O)C(F)C3CCC3)=O)oc12 13776,C(C(O)CC(=O)N1CCC1C1CCC1)NC(=O)CC1CC2(CC2)C1 13777,Cc1[nH]c2ccc(Cl)cc2c1C(=O)NC1CC1NC(=O)C(C(C)(C)C)N(C)C 13778,C1(CNC(c2c(C)cc(C)nc2)=O)CC(C(C)(C)C)=NO1 13779,N1(CCC)CCCCC1C(=O)NCCC(C(C)C)NC(=O)Cc1cc(C)[nH]n1 13780,C1(C)(C(=O)NCC(CNC(c2c(C)cc(CC)o2)=O)(C)C)CCC(C)=C(C)C1 13781,c1(C(N(CC(C)O)CCNC(c2cc(CC)ncc2)=O)=O)ncnc2ccsc12 13782,c1(OC)cc(C(=O)Nc2cccc(C(C)(C)C)c2)cnc1-c1ccccc1COC 13783,c1(C(=O)NCC(CO)NC(c2ccn(C)c2)=O)cccc(S(C)(=O)=O)c1 13784,C1(CNC(C(C(C)C)OC)=O)(NC(=O)C(c2cccnc2)C)CCC(F)(F)CC1 13785,C(=O)(C(C)(F)CC1CCCC1)NC(C1CCN(C(=O)CC23CCCC2C3)CC1)C 13786,CC12CC(C(=O)NCC3CC3NC(c3cc(C(F)F)[nH]n3)=O)(CCO1)C2 13787,N1(C(CS(CC)=O)=O)CCC2(CCCC2NC(=O)CSc2n[nH]c(C)n2)CC1 13788,c1(N2CCC(N(C(=O)Cc3c[nH]ccc3=O)C)C2)cc(Cl)nc(C(F)(F)F)n1 13789,N1(C(COCC(=C)C)=O)CCC(CNC(C2CCS(=O)(=O)C2)=O)C12CC2 13790,N1(C(C2(OC)CCC2)=O)CCC(C2(NC(=O)COc3ccc(Cl)c(F)c3)CC2)C1 13791,c1(CC)nc(C)c(CC(=O)NCC(C(C)C)NC(C2CCCC23CC3)=O)c(C)n1 13792,N1(C(CC(CN(C)C)O)=O)CC(N(C(=O)Cc2cncc(O)c2)C)C(C)(C)C1 13793,N1(C(c2cc(C)sn2)=O)CCC(O)(C(C)NC(C2(C(F)F)CCC2)=O)C1 13794,N(C(=NCCCOC1CCSCC1)Nc1ccc(OC)cc1)C(CC)C 13795,C1(CNC(C(=O)NC2CC(C)N(S(C)(=O)=O)C2)=O)CCC2CC(C)CN2C1 13796,c1(CC(=O)NCCN(C(=O)CC2CCNC2=O)C)cc(Cl)sc1Cl 13797,N1(C(CC2CC(CC)C2)=O)CCCC(CC(=O)N(C2CC(OC)C2)CC)CC1 13798,C(=O)(C(C)CS(C)(=O)=O)NCC=CCNC(C(C1CCC(C)CC1)CC)=O 13799,C1(NC(=O)NC2CC3CC2CN3Cc2ccccc2)CCCC12CCOCC2 13800,C#Cc1cc(NC(C2CC(=O)C2C2CCC2)=O)ccc1C 13801,N1(C(C)=O)CCC(C)(C(=O)N(C)CC2CCCCN2C(c2cncn2C)=O)C1 13802,C1(NC(c2cccc(OCCOC)c2)=O)CC(F)CN(C(=O)COC2CC2)C1 13803,CCCCC(C(=O)N(C1CCCCC1)CCNC(=O)C(C)(C)NC(C)=O)C(C)C 13804,N1(C(C(=O)C(C)=O)=O)CCCC(C)C1.CC(C(C)C)=CC(=O)N(C(C)CCN)C 13805,N1(CC(=O)NC2CCC(C(CC)=O)CC2)CCP(C)(=O)CC1.c12cccc(c1)S2 13806,c1(CC)nc(C(C)NC(C2CCN(C(C)(C)C)C2)c2nnnn2C2CC2)cs1 13807,N1(C(C)=O)CCC(c2ncc(C(C)C)[nH]2)C1.C(C(=O)O)S 13808,C1(C2(O)CCN(C)CC2)(C(N(CCCCN(C)C(c2ccoc2)=O)C)=O)CC1 13809,C(C)(C)(C(O)C(F)F)N(Cc1c(C)nn(-c2ccccc2)c1)CC1CC1 13810,Cc1nc2[nH]c(C(=O)NC3CC(O)(CNC(C4CCCC(C)(C)C4)=O)C3)cc2s1 13811,c1(C(N2CCCC(N(C(c3c(C)cncc3)=O)C)C2)=O)noc2c1COCC2 13812,C12(CNC(C3C(CC)CCC3)=O)CCC(CNC(c3sccc3C)=O)(CC1)CO2 13813,Cn1ccc2cc(C(N3CCC(C4CC4)(CNC(=O)C4=CCCC4)C3)=O)cnc12 13814,N1(C(=O)NCC=CCC)CCC(F)(Nc2nc(-c3ccco3)cs2)C1 13815,c1(C(C)C)noc(CNC2CC2C(=O)NC(c2nc(C)no2)CO)n1 13816,c1(-c2nc(CCCN(C)C)nn2CC(C)(C)C)cncc2c(Cl)cccc12 13817,c1(C(=O)NCC=CCNC(CCc2cc(C)cc(C)c2)=O)cc(Cl)cc(C)c1C 13818,N#CC12CCC(C(=O)Nc3nc(-c4cccs4)cs3)(CC1)CC2 13819,c1(C(C(=O)NCCCNC(C(n2ccc(C)n2)C)=O)C)cccc(O)c1 13820,C1(C(C)C)CN(C(C(=O)NC2COC2)C2CCC2C(F)(F)F)CC=N1 13821,N1(C(c2nncc(C)c2)=O)CCC(C)C(NC(c2ccoc2)=O)C1 13822,CC1C(C)N(C(c2ccn(CCC(F)(F)F)n2)=O)CCN1C(c1csc(=N)[nH]1)=O 13823,N1(C(CC(C)F)=O)CCCC2C(NC(c3nn(C)c(Cl)c3Cl)=O)C(C)(C)C12 13824,Cc1nn(-c2cccc(Cl)c2)c(C)c1CNCCS(=O)CCc1ccccc1 13825,c1(CC)ccc(C(=O)NCC2(NC(c3cncc(OC)c3)=O)CC2)c(F)c1 13826,N1(C(c2c(C)ccnn2)=O)CC(N(C)C(c2cnc(CO)nc2C)=O)C2(CC2)C1 13827,N1(C(C(C)NC(N)=O)=O)CCC(C(=O)NCC=CC(C)(C)C)=C(F)C1 13828,c1(OC)cc(C(=O)NCCN(C(=O)C(F)=C2CCC2)C)[nH]n1 13829,c1(C(N2CC3C(NC(CN(C4CC4)CC)=O)(C3)C2)=O)cc2cn[nH]c2cn1 13830,C(=O)(CC1=NN(C)C(=O)C1)NC(C1(O)CCN(C(=O)CCCCCNC(N)=O)C1)C 13831,C(=O)(CC(F)(F)C(C)C)N1CCCC(NC(C(CCCOC)C)=O)C1C 13832,N1(C(C(C2CCOC2)NC(C(CSC)OC)=O)=O)CC(C2CCCCC2)C1 13833,Cc1noc(C2CC2)c1C(=O)N(C1CCC(NC(C2(C(C)(C)O)CC2)=O)C1)C 13834,C(=O)(C(F)CCC(C)C)N1CC(CNC(C(CC)C(C)C)=O)OCC1 13835,c1(C(N(CC(C)O)CCNC(=O)CC(C)CF)=O)ccc(C(F)F)c(F)c1 13836,c1(C(N(CC(CN(C(c2[nH]cc(C)c2)=O)C)O)C)=O)ccc2c(c1)CCCCS2 13837,N1(c2nccc(OC)n2)CCN(C(C2(c3ncccc3F)CC2)=O)CC1C 13838,C1(NC(CC2CC(CC)C2)=O)CN(C(c2cn(C)c(C)n2)=O)CC1C 13839,C1(C(=O)OC)CC2(CC(NC(=O)C(N3CCN(CCCN(C)C)CC3)C)C2)C1 13840,c1(CCCC)ccc(S(=O)(=O)N2CC3CC2CCN3C(=O)CCS(C)(=O)=O)cc1 13841,C1(C(=O)NC2C(CNC(CC(C)(C)OC)=O)CCCC2)CCC2(CC1)CC2(F)F 13842,C(=O)(NNC(=O)C(C)(C)CCCCNC(=O)C(C)=CCC)C1(CC=C)CCOCC1 13843,C(CC1=CCCCC1)NC(c1c(CNC(C2(Cl)C(C(C)=O)C2)=O)ccs1)=O 13844,c1(C(=O)NCCC(C)NC(=O)CC(C)C(F)F)cc(Cl)c(F)cc1Cl 13845,C1(NC(c2c(C)nn(CC(F)F)c2)=O)CCN(C(C2(C)SCCCS2)=O)CC1C 13846,C1(C)(C(N2CC3(C(NC(C=COCC)=O)CC3)C2)=O)Oc2ccccc2NC1=O 13847,CC1CCc2[nH]c3ccc(C(N4CCN(C(=O)CCN(C)C)CC4)=O)cc3c2C1 13848,Cc1ccc(C(=O)NCC2(C(=O)NC(Cc3cnc[nH]3)CO)CCC2)c(O)c1 13849,Cc1cc2ncn(CC(=O)NC(C)(CNC(C3CCCO3)=O)C(C)C)c2cc1C 13850,c1(C(=O)NCC(CNC(CCc2cc(C)on2)=O)C)cn(C)nc1-c1cccs1 13851,C1(C)(Nc2cnc(CC)s2)CCN(C(c2nccc(C#N)n2)=O)CC1 13852,C1(C)(C(=O)NCC2C(NC(=O)COC3CC=CC3)CC2)CCC(=O)NC1 13853,N1(C(CC2C(=O)NC(=N)S2)=O)CC2CCN(C(=O)C(O)CF)CC12 13854,N1(C(C(C)Oc2cccnc2)=O)CC=CC(C(=O)NCC2(C)CC2(C)C)C1 13855,N1(C(C2(COC)N(C(c3ccc(CC)[nH]3)=O)CCC2)=O)CCC(C)C(CO)C1 13856,C(=O)(CCCCCCCCCO)N1C(CCNC(c2cc(C)no2)=O)CCC1 13857,c1(C(=O)NC2C(C)CCN(C(=O)Cn3nccn3)C2)cc(C#N)ccc1Cl 13858,c1(C(N2CC(C)(CNC(C3CC=CC3)=O)OCC2)=O)ccc(S(N)(=O)=O)cc1 13859,c1(COC)cnc(OC)c(C(=O)NCC(C)CNC(c2coc(Cl)n2)=O)c1 13860,C1(c2n(CC=C)nnn2)(NCC2CCN(S(C)(=O)=O)CC2)CC(C)SC(C)C1 13861,C1(CNC(C2CC(SC)C2)=O)C=CCN1C(c1ncn(C)n1)=O 13862,N1(C(C23C(CN(C(c4cc(C5CC5)no4)=O)C2)CC3)=O)CCCC12CCOC2 13863,c1(CN2C(CCC(N3CCCC3c3ccccc3)=O)CCC2)cc(Br)cc(Cl)c1O 13864,N(C(=NCC(C)N1CCCC1)NC(C1CCCCC1)C)Cc1ccc(C(C)C)cc1 13865,c1(C(=O)NC(CNC(c2ccc(COC)o2)=O)CO)cc(Cl)c(C)cn1 13866,CC1(C)CC(CC(=O)NCC(C)(CO)NC(c2cccnn2)=O)C1 13867,c1(C(=O)OC)cc(F)cc2c1CCN(C(C1CCC(COC(C)(C)C)O1)=O)C2 13868,C1(C(=O)NC(CCC)C)CCN(C(=O)c2ccc(CSC)o2)O1 13869,Cc1cnc(C=CC(=O)NCCC2COCCN2C(=O)Cc2cc(Cl)cs2)[nH]1 13870,N1(C(C=CC(=O)NC2CC2)=O)CCCCCC(NC(C2(C3CCC3)CC2)=O)C1 13871,C#CCCCC(C)C(=O)N(C)CCOCCNC(=O)CCc1cocn1 13872,C(c1ccccn1)=C(C)C(=O)NCCOC1CN(C(C2OCCC2C)=O)C1 13873,Cc1cc(C(=O)NCC(C)NC(=O)C(C)(C)C(C)C)cc(F)c1C 13874,O=C1CC2C(C(=O)NCc3cccc(C(N4C(CO)CCC4C4CC4)=O)n3)C2C1 13875,C(=O)(C(C)C(C)(C)C)NC(C(C)C)CNC(C1CN(S(C)(=O)=O)C1)=O 13876,N1(CC(N2CCC(C(C)CI)C2)=O)CC2(CC2)CC1C.c1(C)ccccc1.N1CCO1 13877,CC1CC(C)(C(=O)N(C)CCN(C(=O)C(N2CCN(C)CC2)(C)C)C)CCO1 13878,n1(CC(=O)NCC2N(C(c3cc(C(=O)OC)sc3)=O)CC2)nc(C)cc1C(N)=O 13879,Cc1cc(=NC2CCCCC2N(C)Cc2cnc[nH]2)[nH]c(N(C)C)n1 13880,c1(OCC)cncc(C(=O)N(CCCCCNC(c2cncc(OC)n2)=O)C)c1 13881,CCC(CNC(C1CCCN1C)=O)(CC)C(=O)NCCCn1ccnn1 13882,N1(C(CCC#C)=O)CC(NC(c2cccnc2C)=O)CC12CCCCC2 13883,C(CC(CC)C(=O)NC1CCCCC1C(=O)N(C(C)CC)CCO)=CC 13884,c1(C(=O)NC(C(C)NC(c2cc(OC)c(Br)s2)=O)C)cc([N+](=O)[O-])nn1C 13885,C1(C(=O)NCc2n(C)cnc2)CCN(C(c2ocnc2C2CC2)=O)C1(C)C 13886,c1(C(=O)NCCN(C(c2ccc(CC)cn2)=O)C(C)C)nc(C)c(N)cc1C 13887,CN1CCC(C(N2CC3(CCN3C(c3ccccc3C3(C)CC3)=O)C2)=O)CC1=O 13888,CCC(C)C(O)C(C)C(=O)N(CCC(=O)NCC1CC1)CCCO 13889,c1(C(=O)NCC2CCCCCN2C(=O)COC2CCCC2)cc2c(nn1)CCC2 13890,N1(N2CCCC(N=[N+]=[N-])C2)CCC2(CC1)CN(C(=O)CC(F)(F)F)CCO2 13891,Nc1ncc(C(N2CCN(C(=O)C(F)C3CCC3)CC2)=O)cc1Cl 13892,C1(C(N2CC(CCNC(C(C)(F)F)=O)C2)=O)CCCCN1O 13893,CC1(C)CC(C)(C)C1C(N1CCC(N(C(c2cnc(Cl)s2)=O)CC2CC2)CC1)=O 13894,CC1CCCCC1C(=O)NCC1(CNC(=O)C(F)(F)c2ccncc2)CC1 13895,c1(C(=O)NC2CCC2NC(=O)C(O)c2cnc[nH]2)ccc2c(c1)CCCS2(=O)=O 13896,C1(CNC(c2csc(C)c2C)=O)CN(C(=O)CCC#N)CCC1C 13897,C1(C(=O)N(Cc2ccc(CCNC(CCCC)=O)cc2)CCC)C2CC2C2CC12 13898,C1(CNC(c2ccn(CCOC)n2)=O)COC(C)(C)CN1C(c1cn[nH]c1)=O 13899,c1(Cc2ccccn2)nc(CCSCCF)nn1Cn1cc(-c2nc[nH]n2)nn1 13900,C(=O)(C1=C(C(C)F)N(C(C)CC)C(=O)NC1c1cc(Cl)c(F)cc1F)OCC 13901,N1(C(Cc2c(C)ccs2)=O)CCC(C)(NC(=O)Cc2nnn(C(C)(C)C)n2)C1 13902,c1(C(=O)NCC(C2CCN(C(CCCC3C(C)C3)=O)CC2)O)cn2ccnc2s1 13903,c1(C(=O)NCC2CN(C(C3(OC)CCC(C)C3)=O)C2)ccc2cc[nH]c2c1 13904,C#Cc1ccc(CCCC(=O)NC2CCN(Cc3c[nH]c(=N)o3)CC2C)cc1 13905,CC#CCCCC(=O)NC(C(=O)NCC1CCCC1CF)c1cccs1 13906,c1(C(N(CC)Cc2ncc[nH]2)=O)occc1CNC(=O)CC1CCSC1 13907,C(=O)(C(COC)N(C)C)N(CCN(C(c1cn(C(C)(C)C)cn1)=O)CC)C(C)C 13908,C(=O)(C1CCCc2nn[nH]c21)NCC(C)CNC(c1ncn2c1CCCC2)=O 13909,c1(C(=O)NCC2CCC(NC(=O)CSCc3ccccc3)C2)ccc(O)nc1Cl 13910,Cn1c(C(=O)NCc2cncc(C(=O)NCC3CCOC3(C)C)c2)cccc1=O 13911,CCCCC(C)CCC(=O)N1CCC(F)C(NC(c2nc(Br)c[nH]2)=O)C1 13912,c1(C(N2CC(O)(CN(C)C(c3cnn(C)c3C3CC3)=O)C2)=O)n[nH]c2c1COC2 13913,C1(CNC(C=Cc2n(CC)ncc2)=O)CCN(C(=O)C=C(C)I)CC1C 13914,Cc1cc(C(N2CC(O)(CNC(=O)CSc3cccnc3Cl)C2)=O)cc(F)c1C 13915,C(=O)(C(F)(CNC(C1CC(N=[N+]=[N-])C1)=O)C(C)C)N1C(CC(C)C)CCCC1 13916,CC(C(=O)NCC(C)(C)CNC(C1(c2ncco2)CC1)=O)C(C)(C)C 13917,c1(C(C)C(=O)OCCNC(=O)Cc2csc(NC=O)n2)ccc(OC(F)F)cc1 13918,c1(N(C)C)ccc(Br)cc1C(N1CCC(C)(CNC(C2(O)CCC2)=O)C1)=O 13919,C1(CC(=O)NC(c2ccc(C)cc2)CNC(C2CC(=C)C2)=O)CCC2(CC1)CC2 13920,Cc1cnc(C)c(C(N2CC(NC(c3c[nH]nc3C3CC3)=O)CCC2C)=O)c1 13921,N1(C(C)Oc2ccnnc2S)CCCC(C)(c2cn(-c3cncc(Cl)c3)nn2)C1 13922,CCCC(O)C(=O)NC(C(=O)N1CCC(C(N)=O)CC1)C(C)C 13923,c1(NC(C(CCC)C)C)[nH]c(=NCCCOc2ccncc2)nc2scnc12 13924,CCCCCCC(C)C(=O)NCC1CC(C(=O)N2CCC(F)(CF)CC2)=NO1 13925,Cc1c[nH]nc1CC(=O)NCC1CN(C(C2CCCN2C2CCCC2)=O)C1 13926,N1(C(c2cncc(C)c2)=O)CC2CCCC2(NC(=O)Cn2nc(C)ccc2=O)C1 13927,CC1(C)C(c2ccc(Br)cc2)CCN1C(C1CCN(C(=O)C(F)(F)F)CC1)=O 13928,c1(C(N2C(COC)CN(C(=O)CSC3CC3)CC2)=O)cc([N+](=O)[O-])cc([N+](=O)[O-])c1 13929,C1(C(N(C2CCC2)CC)=O)C=CCN(C(=O)COC2CCC2)C1 13930,N1(C(C(C)C(C)(C)C)=O)CCC2(CCCCN(C(c3ccsc3)=O)C2)C1 13931,C1(C(N2C(CC)CC(O)C2)=O)CN(C(=O)C(F)CC(C)(C)C)CCC1(C)C 13932,c1(CCNC(C2C(O)CCN(C(CCCCC#C)=O)C2)=O)cc(Cl)cc(Cl)c1O 13933,n1(CC)nc(CC(N2CC(c3ccc(OC)nc3)(O)C2)=O)cc1C(F)(F)F 13934,c1(C(=O)NC2CC(F)(CNC(C(CC)C(C)C)=O)C2)c(F)cc(Cl)cc1F 13935,C1(C(N(C)CC2CCN(C)C2)=O)CC2(CCC2)CN1C(c1ccc(C#N)s1)=O 13936,CCC(C)CCC(=O)NCc1nc(C)c(C(=O)NCC2(CC)CCCC2)o1 13937,C(=O)(C1=NOC2(CCN(c3nccc(C#N)n3)C2)C1)Nc1cc(C)c(C)c(C)c1 13938,C1(C(=O)NC(C(C)C)CNC(c2csc(CC(C)(C)C)n2)=O)CC(=O)N(C)C1 13939,c1(NC(=O)C(N2CCC23CCOC3)=O)ccc2sccc2c1 13940,N1(C(c2ccc(CC)s2)=O)CCC(F)CC1C(N1CCN(C)CC1C1CC1)=O 13941,C(CC1=CCCCC1)N(C)C(C1C=CCN(C(c2c[nH]nc2Cl)=O)C1)=O 13942,C(=O)(C(C)(C)CF)N(C1CCN(C(C2CCN(C)C2=O)=O)CC1)C 13943,C1(C(=O)NCC2C3CN(C(CCn4c(C)ncc4)=O)CC32)CN2CCN1C(C)C2 13944,c1(C(=O)NCC2C(CNC(C(OC)OC)=O)C2)cc(C)c[nH]1 13945,Cn1c(CCNC(=O)C(=O)NCc2ccc[n+]([O-])c2)nnc1-c1cccnc1 13946,c1(NC2CN(C(C)C)C2)[nH]c(=NC(C)c2cnc[nH]2)nc2sccc12 13947,N1(C(C=CC=CC)=O)CC2CC(N=c3cc(Cl)nc(C(C)C)[nH]3)C2C1 13948,C(=O)(CCNC(=O)CCc1cnco1)NCC1(C)CC1 13949,c1(OC)cc(C)ccc1CN(C(=S)NCC(C)(C)F)C1CC1 13950,C(c1ccc(Cl)s1)=CC(N1CCCC(NC(=O)C(O)CC2CCCCC2)C1)=O 13951,C(=O)(C(CCNC(=O)C(CC1CCC1)OC)OC)NCCCC#C 13952,C1(C2(NC(=O)CCCCN(C(=O)CCCNC(=O)OC)C)CC2)(OC)CCC1 13953,C1(C(N2CC(O)(CNC(C(CC)NC(N)=O)=O)C2)=O)CC2(CCC2O)C1 13954,C12(C(=O)NC3CCN(C(C(C)OCC=C)=O)C(C)C3)CCC(N(C)C)(CC1)CC2 13955,S(=O)(=O)(CCC(=O)NCC1COCCN1C(c1ncnn1C(C)C)=O)NC 13956,N1(C(C(CC)C)=O)CCC(NC(c2ccc(OCC3CC3)nc2)=O)C2(CCC2)C1 13957,C=Cc1ccc(C(N2CCCC(CC(=O)NCC3CC(CC)=NO3)CC2)=O)cc1 13958,c1(C(=O)NC2CCC(CNC(c3ccc(Cl)o3)=O)C2)cccc2cc[nH]c12 13959,Cc1c(Cl)cc(Cc2cn(C3CN(C(C4CCCCC4F)=O)C3)nn2)cc1Cl 13960,c1(C(N2CCN(C(CNC(C)=O)=O)CC2C(C)C)=O)c(C)cc(Br)cc1C 13961,c1(CC)cc(C(=O)NC2CC(C(=O)NC3C=CCC3)C2)ccn1 13962,c1(C(=O)NCC23CC(NC(COCCC)=O)(C2)C3)ccc2cccnc2c1 13963,C1(CCC)(C(=O)NCCCN2CCN(C(=O)CCC(F)F)CC2)CCNC1=O 13964,N1(C(c2[nH]c(=NC)sc2)=O)CCCC12CCCN(C(c1nccnc1C)=O)C2 13965,c1(C(=O)NC2CCN(C(c3nn(C)c(CO)c3)=O)CC2)cccc(Cl)c1[N+](=O)[O-] 13966,C(CCCCN(C(=O)CC(C)n1cc(Br)cn1)C)NC(C=C(C)C1CC1)=O 13967,n1(CCC)cc(Cl)c(C(=O)NC(C)CN(C(c2cccc(F)c2)=O)CC)n1 13968,c1(OC)cc(C)c(C(=O)NCC2CCC3(CN(C(=O)CCCSC)C3)O2)c(C)c1 13969,C1(NC(C(CC=C)NC(=O)C(C)OCOC)=O)CC(C)(C)OC1(C)C 13970,C1(N(C(c2cc(CC)on2)=O)C)CCCC(NC(=O)CCCN2CCCC2)C1 13971,CCC(CCCO)N=c1[nH]c(=NCCCN(C)C(C)C)[nH]c2c1CCC2 13972,N1(C(CC(C(C)CC)NC(C(CCC)N(C)C)=O)=O)CC=C(C(C)(C)C)CC1 13973,C(c1ccc(NC(N2CCC(C(=O)OC)CC2)=O)n1C)=CC(=O)OCC 13974,C12(NC(CC3CC(OC)C3)=O)CC3CC(C1)CC(NC(C1CCC(C)O1)=O)(C3)C2 13975,C1(C(=O)NCCOCC(=C)C)CCCC(NC(c2ccc(CC)nc2)=O)C1 13976,N1(C(COC(CNC(c2c(NC)cccc2)=O)(C)C)=O)CC(O)CCC1C 13977,c1(OC)ccccc1CC1CCCN1C(=O)C(=O)NCCc1ccc(C)cn1 13978,N1(C(C(CC=CCC)C)=O)C(C(N2CCCC2C(O)CC)=O)CCC12CC2 13979,C1(NC(Cc2nc(C)sc2)=O)CC(F)CN(C(c2ccccc2CNC(N)=O)=O)C1 13980,Cc1cccc(C(=O)NCC23CCC2CN(C(c2nocc2Br)=O)C3)c1O 13981,c1(C(=O)O)coc2cc(N)c(CNC3COC4(C3)CN(CC3(O)CCC3)C4)cc12 13982,CC1=C(C(=O)N2CCC(O)(CNC(=O)CC(C)(O)C(F)(F)F)C2)C(=O)OC1(C)C 13983,c1(CNC(=O)C2CC2)ccc(F)c(O)c1F.C12CC(C1)C(=O)N(C1CC1)C2=O 13984,C(=O)(CCN=c1cc(NCC2CC(C3CC3)=NO2)nc[nH]1)CCF 13985,c1(CO)cccc[n+]1[O-].C12CN(C1)C(=O)COCC1(CC1)C(=O)NC(C)C2 13986,N1(C(=O)C=Cc2cc[nH]n2)CCC2CC12C(=O)NCC1(Cl)CCC1 13987,N1(C(=O)CSc2n[nH]c(O)n2)CCN2CCNCC2C1 13988,C1(COC)(CNC(=O)C(C)(O)COC)CCCN1C(C1CC2(C1)CC2F)=O 13989,N1(CCSCC)C(=O)NC(c2cn(CC3CCOC3)nn2)C(C(=O)OCC)=C1CC 13990,c1(C(C(=O)NCC(CNC(Cc2cnc(C)[nH]2)=O)CO)C)ccc(Br)cc1 13991,c1(C(N2C(C)CCC(NC(=O)C=Cc3cn[nH]c3)C2)=O)cc2c[nH]cnc-2n1 13992,c1(OC)ccc(S(=O)(=O)N2CCCC(C)(C(=O)Nc3c[nH]nc3C#N)C2)cc1Br 13993,C(=O)(CCCCN(C)C)NCCOCCNC(C=NOC)=O.C1(O)CC1(F)F 13994,C1(NC(CN(C(=O)OC)C)=O)(CNC(c2cnc[nH]2)=O)CCCCCC1 13995,c1(OC)ccc(CN2CCCC(C(=O)N(C)CC3CCCCC3)CC2)c(Cl)n1 13996,C(CN=C(NCC1CCOC1)NCC1(C)CCC1)(c1ccc(Cl)cc1)OCC 13997,CCCC(C)(CC)C(=O)NC1CC(CCNC(=O)C(C)(CC)CC)C1 13998,C1(NC(C(CC)N(C)C)=O)C2CN(C(=O)CSCc3cccnc3)CC12 13999,N1(Cc2n(C)ncc2)CCCC=C1C(=O)N=c1ccn(C2CCCCC23CCC3)[nH]1 14000,CC1(NC(c2cccc(C3CC3)n2)=O)CCN(C(C2(C(F)F)CC(O)C2)=O)C1 14001,Cc1cc(CCC(=O)NCCCN(CCO)C(C23CC(CO)(C2)C3)=O)n(C)n1 14002,CCCCC(O)C(C)C(=O)NC1(CC(=O)NCCn2ccccc2=O)CCC1 14003,c1(C(=O)NCC(CC=C)NC(C2CCCC2OC)=O)cccc(C(F)(F)F)c1F 14004,c1(NC(=O)C(c2ccccc2Cl)O)ccc2c(c1)CCC2 14005,c1(CN(CCOC)CCN(C)C)ccc(NC(=O)Cn2cnnc2O)cc1 14006,c1(CCC(=O)NCC2N(C(Cc3cn(CC)nc3)=O)CC=C2)cc(C)nn1C 14007,c1(C(N2CC(C(C)NC(C3C(OC)CCC3)=O)C2)=O)ccc2nc(O)[nH]c2c1 14008,N1(C(CSCC=C)=O)CC(NC(c2cnoc2-c2ccc(Cl)s2)=O)CC1(C)CC 14009,Cc1cccc(C)c1C.C(=O)N(C)CCOC(F)F.C1CO1 14010,C1(=CC(=O)NCC(c2ccccc2)NC(=O)C=C2CCSCC2)CCCC(=O)N1 14011,c1(OC)c(F)ccc(C(N2CCC(O)(C(C)C)C2)C(=O)NC2(C)CC2)c1F 14012,c1(-c2nc(C(C)OC)nn2-c2cccc(OC)c2)onc2cc(C)ccc12 14013,c1(C(N2C(CNC(=O)CCCn3cccc3)CC2)=O)ccc2c(c1)CCCS2 14014,c1(CC)ccc(C(=O)NC(C2CC(F)(F)C2)C(=O)OC)c(C(F)(F)F)c1 14015,c1(CNC(c2c(CCC)n(C)nc2)=O)n[nH]c2c1CN(C(C1CC1F)=O)CC2 14016,C1(CNC(C(=O)NCC2CC2)=O)C2CCCC1N(C(C1(c3ccncc3)CC1)=O)C2 14017,Cc1nn(CC(F)F)c(C)c1C(=O)NCC(C)(C)CN(C(=O)Cc1cccs1)C 14018,c1(C(N(CCCNC(C(C)c2cc[nH]n2)=O)C)=O)cccc(NS(C)(=O)=O)c1 14019,C(C(C(=O)NC(CNC(=O)CO)C1CC1)C(F)(F)F)OC 14020,c1(N(C)C)ncc(C(=O)NC(CC(N)=O)c2cn(Cc3cccs3)nn2)cn1 14021,C(c1cccc(O)c1)=CC(=O)NCC(C)(F)CNC(C1CCCN1C1CC1)=O 14022,N1(C(C23C(C)OC(CON)(C2)C3)=O)c2c[nH]nc2CCC1C(c1ccccc1)=O 14023,CCCCC(C(=O)NC1CC2(C1)CN(C(c1cc(C(=O)OC)[nH]n1)=O)C2)NC=O 14024,C(=O)(CCCCCCC=C)NC(CC#C)C(=O)NCCCc1ccccc1 14025,C1(NC(c2ccc(C#C)o2)=O)(CO)CCCN(C(=O)CCCc2ccccn2)C1 14026,c1(C(=O)NCC2(F)CCCN(C(C3C(C)C3C)=O)C2)ccc2c(c1)C(=O)NC2=O 14027,c1(SC)ncc(C#N)c(N(C2CNC2)Cc2cc(Br)cnc2Cl)n1 14028,C1(CNC(c2cncc(C)c2)=O)CCC(F)(CNC(c2cc(C#N)cs2)=O)CC1 14029,N1(C(C(C)CN(C)C)=O)CCCC(C)(C(=O)NCCc2cccc(O)n2)C1 14030,C(=O)(C(C)(C)C(N)=O)NCCCCC(C)NC(=O)C(C)c1ccco1 14031,C1(CC)(NC(c2ccc(Cl)c(OC)c2)=O)CCCN(C(=O)CCc2cn[nH]c2)C1 14032,CC1CN(C(=O)CC(C)(C)O)CC2(CCN(C(c3ccc(=O)n(C)n3)=O)C2)O1 14033,c1(CC)cccc(C(=O)N(CCC(C)(C)NC(C2C3CN(C)CC23)=O)C)c1 14034,c1(N(C(=O)C(F)CC)CCNC(CCC)=O)ncc2c(F)cccn12 14035,CC(C)C(C(=O)NC1CCC1NC(c1cccnc1C1CC1)=O)c1ccn(C)n1 14036,C1(CNC(C(C)=CC2CC2)=O)C(C)CCN1C(c1n[nH]c(C)c1C)=O 14037,C12(NC(C34CC=CC(C3)OC4)=O)CCC(C(=O)NC3(CCCCO)CC3)(CC1)C2 14038,C1(NC(c2c(CC)noc2)=O)CN(C(c2cccc(N)n2)=O)CC(C)(C)C1 14039,C1(C2(O)CN(C(c3cccc(OC)c3)=O)C2)(CNC(C(COCC)C)=O)CC1 14040,C(=O)(CCCCNC(=O)Cc1cncc(C)c1)NCC#CC 14041,CCCCC(C)(F)C(=O)N1CC2(CCN(C(c3cocc3Br)=O)C2)C1 14042,c1(CC)ccccc1-c1ccc(N2CCN(C(=O)CCC3CCCC3)CC2)nc1 14043,C1(CCCC)CN(C(c2csc(C)n2)=O)CCN1C(c1cn(CC2CC2)nn1)=O 14044,c1(C(=O)NCCC(CNC(c2ccc(CO)s2)=O)OC)cccc(C)n1 14045,N1(N2C(c3nc(C)[nH]n3)CCC2)CCc2c(C(F)(F)F)ccc(Cl)c2C1C 14046,C1(CNc2cc(OC(C)C)ncn2)CN(C(=O)C(F)=C2CCCC2)CCC1(F)F 14047,C12(C(=O)NCCCCNC(c3cn(C)nc3Cl)=O)CCC(CC1)C(C)(C)O2 14048,c1(CC)ccc(C=CC(N2CC(CCNC(c3cn(CC)nn3)=O)C(C)C2)=O)o1 14049,CC1CC(NC(=O)C(c2ccccc2)N(C)C)CN(C(C2(F)CCC2)=O)C1 14050,Cc1c(NCc2csc(O)n2)nc[nH]c1=NCCc1nc(-c2ccccc2)cs1 14051,N1(C(C2CC(C)OC2=O)=O)CCC(C)(NC(=O)Cc2nncn2C)CC1 14052,CN1CCC(C(=O)NOCC(O)CO)(NC(C2CCCC2F)=O)C1 14053,c1(C(N2CCC(N)(CC(=O)OC)C2)=O)cc(Br)c(O)nc1C 14054,N1(C(c2cc(CC)[nH]n2)=O)CC(CC)CC1CNC(=O)COC(F)(F)F 14055,c1(OCC(CC)OC)ccc(C(=O)NCCNC(=O)C(C2CCC2)OC)cn1 14056,N1(C(c2n[nH]c(C)c2N)=O)CCCCC(NC(=O)C=Cc2ccc(C(F)F)o2)C1 14057,c1(CNC(c2c(C)ccnc2)=O)n[nH]c2c1CN(C(=O)CCNS(C)(=O)=O)CC2 14058,c1(CN(C2CCCO2)C(C)=O)ccc(C(N2C(Cc3ccc(C)s3)CC2)=O)s1 14059,N1(C(C(C(C)O)(F)F)=O)CC2(C1)CN(C(C1(c3ccno3)CC1)=O)CCO2 14060,c1(C(C(=O)NCC(C)N(C)C(c2cnccn2)=O)(C)F)ccccc1F 14061,CS(=O)CCC(O)C(=O)NC1CC(C)(NC(c2cncc(F)c2Cl)=O)C1 14062,C1(C2(O)CN(C(C3CCCC(C(N)=O)C3)=O)C2)(CNC(C(C)(C)CO)=O)CC1 14063,C(=O)(C(C)(C)C(F)F)NCCCCNC(C1C(OC)CC1)=O 14064,CC1CN(C(c2c(N)cc(F)cc2F)=O)CC(C)N1C(C1CC(N(C)C)C1)=O 14065,c12ncnc(c1C)N2.c1(C(=O)NSC)cccc(CC2CC3CCC2C3)n1 14066,CCCCC(C(=O)NCC1C(C)(C)C1(F)F)NC(c1cc(C2CC2)[nH]n1)=O 14067,Cc1nn(C2CC2)cc1C(=O)NCC1CCC(NC(=O)CCOCC(F)(F)F)C1 14068,C(=O)(C(CC(=C)C)NC(c1c[nH]nc1OC)=O)NCCCCCC=C 14069,C1(C(=O)Nc2cn(CC)nc2)CN(C(C2(NC(N)=O)CC2)=O)CCO1 14070,C1(O)(CCNC(C(C)(F)F)=O)CCN(C(=O)COCC2CCCOC2)C1 14071,C=CCC(C)(CC)C(=O)N1CCCCC(NC(=O)CC2CNC(=O)C2)C1 14072,C12CCN(CC1)C2.C1(C(N)=O)CCC(C(=O)NC(=O)Cc2coc(C(F)F)n2)C1 14073,C1(C(=O)OC)CC12CCC(NC(=O)Nc1ccc(F)cc1Cl)CC2 14074,CC(C)(C)C#CC(=O)NCC1CN(C(=O)C=Cc2ccsc2)CC1(F)F 14075,N1(C(C2N(C(Cc3cc(C)[nH]n3)=O)CC2C)=O)CCC2(COC(=O)N2)C1 14076,N1(C(C(C)c2ccsc2)=O)CC(O)(CN(C(=O)C2CC2)C)C1 14077,C1(C(=O)NCC)CCCN(C(C2(C)COC(=O)C2)=O)C1 14078,C(=O)(C(C)(CC=C(Cl)Cl)c1ccccc1)NCCCNC(C=CC(=O)N(C)C)=O 14079,C1(C)(C(=O)NC(CC)(C)CNC(=O)CC2(CSC)CC2)CC(C)(C)C1 14080,N1(C(C(C=CC)O)=O)CCC(CC(=O)NCCCOC(=N)O)CC1 14081,N1(C(C2(CC=C)CCCC2)=O)CCC2CC2(C(=O)Nc2cccnc2C)CC1 14082,Cc1nsc(-c2noc(C3CCN(c4ccccc4)C3C)n2)c1N 14083,N1(CC(c2cn(N(C(=O)CSc3ccccc3)C)nn2)(C)C)CCCC(=O)C1 14084,c1(C(N(CC(Cc2ccccc2)NC(=O)CO)C)=O)c[nH]cc(F)c1=O 14085,c1(C(=O)NC(CC)CNC(C2CCN2C2CCCC2)=O)ccc2ncccc2c1 14086,c1(NC(C2C(CNC(c3c[nH]ccc3=O)=O)CCC2)=O)cc(C2CC2)ccn1 14087,c1(C(N(C)CCN(C)C(C2(C(F)(F)F)CCCC2)=O)=O)ccnc(OCCO)c1 14088,N1(C(C=CC)=O)CCC(N(CCCn2ccc(NC(=O)CC)n2)CCO)C1 14089,N1(C(C2(OC)CC2)=O)CC2CC(NC(=O)C(C(F)(F)F)=Cc3ccccc3)C1C2 14090,C1(S(=O)(=O)C(N2CCSCC2CCO)=O)(C(C)C)CC1 14091,N1(C(c2ccc(C)nc2)=O)CC2CC(NC(C34CCC(N(C)C)C3C4)=O)CC1C2 14092,C#Cc1ccc(C(C2NC(=O)N(c3cccc(C)c3)C2=O)=O)cc1C 14093,CC(C)C(O)C(=O)NC1CN(C(=O)CN(C)Cc2cccc(Cl)c2)CC1F 14094,c1(CCc2ccn(CC)n2)cccc(S(C)(=O)=O)c1.c12nc(n[nH]1)-c1cnn-2c1 14095,C1(NC(c2c(OC)oc(C)n2)=O)CN(C(=O)CC2CCC(=O)NC2)CC1C1CC1 14096,C1(NC(c2c(O)ncc(NC(C)=O)c2)=O)CN(C(=O)C=CC(C)C)CC2(CCC2)C1 14097,c1(NC(C)=O)ncc(S(=O)(=O)NC2CCN(C(c3cc(Br)ncc3F)=O)CC2)s1 14098,c1(OC(CC)C(=O)N(C(C)CNC(=O)C(C)N2CCC2)C)cccc(C)c1 14099,N1(NC(c2ccn(C3CC3)n2)=O)CCCN(CCNC(C(C)(O)C2CC2)=O)CC1 14100,CC1CCCC(C)N(C(=O)C=CCC2(NC(=O)Cc3cn[nH]c3)CCC2)C1 14101,CC(O)C(C(=O)N(C1CC1)CC1CCN(C(c2ncoc2C(C)C)=O)CC1)N(C)C 14102,C1(CC(=O)NC2CCCC(CNC(c3cccc[n+]3[O-])=O)C2)CCS(=O)(=O)CC1 14103,N1(CCCCC(C)Nc2cc(OC(F)F)ncn2)C(=O)c2ccccc2C1=O 14104,N1(C(CCN(CCC)C)=O)CCC(N(C(=O)CCC2CC3C=CC2C3)C)CC1 14105,N#CC1(C(N2CCC(NC(c3cnccn3)=O)C(F)C2)=O)CC12CCC2 14106,Cc1cccnc1CCNC(=O)Nc1ccc(-n2ccnc2)nc1 14107,c1(C(N2CC(C)(C(N3CCCC(C)(O)C3)=O)C2)=O)ccc2[nH]ccc2n1 14108,Cc1ccc2c(NC(C3(C)CCN3Cc3cnc4ccc(F)cn34)=O)cccc2n1 14109,C1(CNC(COCc2onc(C)n2)=O)CN(C(=O)CCCc2ncco2)CCO1 14110,N1(C(C2(C)CCC2)=O)CCC(CNC(=O)Cn2nnc(=N)[nH]2)C1 14111,c1(CC)cc(CC(N2CCCC2C(C)NC(c2cnoc2C(C)(C)C)=O)=O)on1 14112,n1(CC(=O)NCC(CNC(CC)=O)F)cnc(-c2ccccc2)n1 14113,N1(C(COCCSC)=O)CCC(CNC(c2ccc(O)nn2)=O)C(C(F)(F)F)C1 14114,Cn1cc(C#N)cc1C(=O)NC1CN(C(c2coc(-c3cccnc3)n2)=O)C1 14115,C(CCCC#N)(c1nnnn1C1CCOCC1)NCC(=O)N(CC(F)F)C 14116,C1(C(=O)OC)CCN(C(=O)C(CNC(=O)Cc2cnn(C(C)C)c2)N(C)C)C1 14117,C(=O)(C1=CCSC1)N1C(C(C)NC(C2C(C)(C)C2(C)C)=O)CCC1 14118,C=CCC(F)(F)C(=O)NCC(C1(O)CCN(C(c2coc(C(N)=O)c2)=O)C1)C 14119,CC(CCNC(N1CC(C(=O)O)CC(CO)C1)=O)CC(C)(C)C 14120,CCCN(Cc1cnn(C)c1)N1Cc2ccccc2C1CC 14121,N1(C(C(C(C)O)C)=O)CC(NC(=O)CN(C)Cc2ccccc2)CC2(CC2)C1 14122,N1(C(=O)Cc2cc3occc3[nH]2)C2CCC(CO)C1CC2 14123,CCCC(C)(O)C(=O)N1CCCC1C1(NC(c2ccc(=O)n(O)c2)=O)CC1 14124,c1(C(=O)NCC2(O)CN(C(C=COCC)=O)C2)cc(C)c(C)nc1C 14125,C1(NC(=O)COCC(F)F)CC1C1CCN(C(C2CCc3nn[nH]c3C2)=O)CC1 14126,N1(C(C2(CC=C)CC=CC2)=O)CCC(CNC(C2CCCC(=O)N2)=O)(OC)C1 14127,c1(C(N2CCC(O)(NC(c3c(SCC)cccn3)=O)C2)=O)coc2ccccc12 14128,N1(C(Cc2ccc(C)nc2)=O)CCN(C(c2ccc(C)cc2Cl)=O)C(CCO)C1 14129,N1(C(C2N(C(c3ccc(C#N)cc3)=O)CCCCC2)=O)CCC2(COC(=O)N2)C1 14130,C1(O)(C(C)CNC(c2cc(C(N)=O)oc2)=O)CCN(C(=O)CCC#N)C1 14131,c1(C(C(=O)NC)N(C)CC2CCC3(CNC3)O2)c(F)ccc(Br)c1F 14132,c1(NC(C23CCCCC2C3)=O)ccc(NC(c2nccs2)=O)c(F)c1 14133,c1(NC(C2(SC)CN(C(CC3CCC(OC)C3)=O)C2)=O)cc(C)ncc1C 14134,N1(C(c2nc(C(=O)NC3(c4ncc(Cl)cn4)CC3)sc2)=O)CC2C(CO)C2C1 14135,c1(C(N(CC(C2CCCC2)C)C)=O)cc(C(F)F)nc2ccc(Cl)cc12 14136,c1(C(=O)NC2CN(C(CC3CC(OC)C3)=O)C2)ccc(Cl)c(N)c1 14137,N1(C(C2C(N(C)C)CNC2)=O)C=Cc2ccccc2C(C(F)(F)F)C1 14138,c1(SC)ccc(C(=O)NC(C)CNC(=O)CS(=O)(=O)C2CC2)cc1[N+](=O)[O-] 14139,C1(C)(N(C)C)CCN(C(c2csc(Cl)n2)C(=O)NC2CC(F)(F)C2)C1 14140,CCCC(O)(CCC)CC(=O)NC(C)C(CO)NC(C1CCn2nccc2C1)=O 14141,N1(C(C2C3CCC2(c2ccccn2)C3)=O)C2CCC1C(CNC(C1CCCS1)=O)C2 14142,CC1CCC(C(=O)NCCOCCNC(c2cnn3c2CCC3)=O)C(=O)N1 14143,C(CN(C)C)(CC(C)C)NC(C1C(NC(c2cnc(C)s2)=O)C1)=O 14144,C1(F)(C(=O)OC)CN(C(C)C(c2ccnn2C)=O)CC1c1ccc(Cl)cc1 14145,c1(C(=O)NC(CC(C)C)CNC(=O)C=CS(C)=O)coc2cccc(O)c12 14146,c1(OC)ccc(C(N2CCCCC2CN(C(=O)CCC2CC2(F)F)C)=O)nc1 14147,C1(C(N(CC=CC(=O)NCCN(CCCC)C)C)=O)CCCCC1F 14148,Cc1ccc2sc(NC(=O)C(=O)NC(c3cc(O)ccc3C)C)cc2c1 14149,C1(NC(C(C)C)=O)CN(C(c2n[nH]c3c2COCC3)=O)C2(CCCCC2)C1 14150,N1(C(c2ccc(SCC)cc2)=O)CC2CC(C)N(C(C3COCC3COC)=O)C2C1 14151,N1(C(c2ccc(OC)c(Br)c2)=O)CCC2(CCN(Cc3nc(Cl)cs3)C2)C1 14152,O=C(C1CCc2cccnc21)NC1CN(C(c2cccc(CO)c2)=O)CC1O 14153,C1(NC(C)C)CCN(C(=O)C(c2ccoc2)NC(=O)C(F)C2CCCC2)CC1 14154,C(=O)(C1=CC2CC=CCC12)NCC1(CNC(C2CCN(OC)CC2)=O)CC1 14155,c1(C(=O)NCC(C)NC(CN(C2CC2)CC)=O)cnn(C2COC2)c1 14156,C(=O)(C(C(C)NC(C1CCC(C)=C(C)C1)=O)C(C)C)N1CC=C(C)C1 14157,C(C(C)(C)CNC(c1cc(C)ns1)=O)NC(CCOCC)=O 14158,C#CCC(C(=O)NC)NC(=O)CC1(CNC(C2CCCN(CC)C2)=O)CC1 14159,Cc1cc(C(N2CCC(NC(C3CCC4(CC3)OCCO4)=O)C2)=O)ccc1[N+](=O)[O-] 14160,CON1CCC(CC(=O)NCC2CC(F)(F)CN2C(C2C(C)(C)C2(F)F)=O)CC1 14161,c1(OCCC)ccc(C(=O)NCC2CC2NC(C2(CF)CCOCC2)=O)cc1 14162,N1(C(C(CC)(C)C)=O)CCC2CC2(C(=O)Nc2cc(C)cc(C)c2)CC1 14163,c1(C2(C)COC2)nocc1C(=O)NCC1(NC(c2cc[nH]c2)=O)CCC1 14164,C#CCCCCCC(=O)N(CC(CC)NC(=O)Cc1cncn1C)C 14165,N1(C(c2ccc(Br)s2)C(N2CCC(C(=O)NCCC)CC2)=O)CC2CCCC2C1 14166,CC(C)CC(O)C(=O)NCC1CCCN1C(=O)C1=CCCCC1 14167,C1(C)(COC)CN(C(c2conc2C(C)NC(=O)C(C)O)=O)C1 14168,c1(N(C(=O)NCC(C)CC2CC(F)(F)C2)C)cccc(C(F)(F)F)c1F 14169,c1(SCC(=O)NCC(C)NC(=O)C=CCN2CCCC2=O)nccn1C 14170,C1(C(=O)NC2C(NC(COCCOCC)=O)COC2)CC2CCCC2C1 14171,CC1CC=CCC1C(N1CC(NC(c2ccccc2C(C)(F)F)=O)C(F)C1)=O 14172,c1(C(=O)NCC2(CN)C(C)(C)C2)ccc(-c2ccccc2)n1C 14173,c1(C(N2c3ccc(cc3)C(N)C2=O)=O)cc(OC)ccc1N.CNC 14174,c1(OC)cscc1C(N1CCC(CCNC(c2ccn(C(F)(F)F)n2)=O)C1)=O 14175,C1(CC(=O)NCC2(CN(C)C(C3CC=CC3)=O)CC2)C=CCCC1 14176,c1(C(C)(C)C)conc1C(=O)NCC1CCC1NC(=O)CCC1CCCO1 14177,c1(OC)cccc(NC(c2c(C(F)(F)F)ccc(Cl)c2Cl)=O)c1[N+](=O)[O-] 14178,C=CCCCCCCCC(=O)NC1CC(O)C1CC(=O)NC1CC(O)C1(C)C 14179,C1(CNC(C(C)N(C(C)=O)C)=O)(NC(c2nnn(C)c2N)=O)CCOCC1 14180,N1(C(C2(C(C)=O)CC2)=O)CC(C(=O)NC(c2ccc(O)cc2)C)C(F)C1 14181,c1(OCC)ccc(C(=O)NCCN(C)C(c2ccccc2C2CC2)=O)cc1N 14182,N1(C(COCCOCC)=O)CCC(NC(=O)CSCc2cccc(C)c2)CC1 14183,c1(-c2onc(CCCSC)n2)cc2ccc(O)cc2[nH]1 14184,C=CCC(C)C(=O)NC1(CCOC)CCN(C(c2ccc(SCC)nc2)=O)C1 14185,C(=O)(CC(C(F)(F)F)P(C)(C)=O)NCCC1CC(NC(c2c(C)[nH][nH]c2=N)=O)C1 14186,CCCCCCC(CC)NC(=O)C(C1CCCN(C(=O)CC(C)(F)F)C1)C 14187,CC1(C)CN(c2ccc(F)cn2)CCN1C(c1cc(Cl)ccn1)=O 14188,c1(NC(CC2CCN(C(c3nc(CC)oc3)=O)C2)=O)cc([N+](=O)[O-])ccc1SC 14189,c1(OC)c(Cl)ccc(C(=O)NCCCCNC(=O)CN2C(=O)CN(C)C2=O)c1F 14190,C(c1nc2ccccc2o1)=CC(=O)NCC1(F)CCN(C(C(C)OCC)=O)CC1 14191,N1(C(C=CC)=O)CC2(CC(NC(Cn3c(NCC4CC4)c(C)nc3)=O)CO2)C1 14192,Cc1[nH]c(=N)sc1C(=O)OC1CCOC(C)C1 14193,CC1CN(C(=O)CC2(C)CCCO2)CC1CNC(c1cncc(Cl)c1)=O 14194,C1(C(c2n(CC(=C)C)nnn2)NCCc2cnoc2)CCCC(C)C1 14195,C(=O)(C1=NNC(=O)CC1)N(CCCNC(c1cc(C)cc(C)c1)=O)CC 14196,c1(C(=O)NC2C=CCN(C(c3c(C(=O)OC)cco3)=O)C2)cc(F)ccc1Cl 14197,N1(C(c2c(COC)noc2)=O)CCC2(CCCN(C(=O)C(C)CC(N)=O)C2)C1 14198,c1(CC(N2CCC(N(C(=O)CS(=O)(=O)CC)CC)CC2)=O)nc2ncccn2n1 14199,c1(N2CCCC3(NC(c4nccs4)=O)C(C2)C3)ncnc2sc3ccccc3c12 14200,N1(CC(=C)Br)CCN(C2(C(F)(F)F)CCCC2)CC1 14201,C(C(F)(C(=O)NCc1cnccc1Cl)C(C)C)NC(c1c(CC)nccc1)=O 14202,C1(C(=O)OCC)CCC(NCC(F)(F)CCn2cc(C(C)(C)C)nn2)(COC)C1 14203,N1(C(CC2CC2(F)F)=O)CCOC(C)(CNC(=O)C(=O)NC2CC2)C1.C(=O)OC 14204,Cc1cc(=NC(=O)NCC2CN3CCC2C3)c(CO)c[nH]1 14205,c1(N(C(C2CC2NC(c2cc(Br)co2)=O)=O)CC)ccccc1O 14206,N1(C(C(CC=C)NC(c2cccc(F)c2O)=O)=O)CCC(F)C(F)C1 14207,c1(OC(C)C)cccc(CC(=O)Nc2coc(-c3ccccc3Cl)n2)c1 14208,c1(OCC)nc(N2CC3C(CNC(C4OCCN4C=O)=O)C3C2)ncc1C 14209,c1(C(C)=O)ccc(C(N2CCCCC2CCNC(=O)CC2CC2C)=O)c(O)c1 14210,N1(C(c2c(CC)nn(C)c2)=O)CCCC(F)(C(N2CCCC2(C)CC)=O)C1 14211,c1(C(=O)NC2CC(N(C(C(C(C)C)N(CC)CC)=O)C)C2)cc(F)cnc1O 14212,C1(NC(C2CCN(C)C2)=O)C2CN(Cc3ncc(Br)s3)CC12 14213,c1(CCC(=O)NC(CN(C(c2c(C)oc(CO)c2)=O)C)C)cccc([N+](=O)[O-])c1 14214,c1(N(C)CC2CCN(C(=O)Cc3ccn(C)n3)C2)ncc([N+](=O)[O-])c(=N)[nH]1 14215,N1(C(=O)OCC)CCCC(NC(c2ccc(Br)c(F)c2)C2CC2)C1=O 14216,O=C(C1CCCc2c[nH]nc21)NC1CN(C(c2cc(F)c(F)cc2N)=O)CC1F 14217,Cc1cnc(Cl)c(C(=O)NC(C2CCN(C(c3ccco3)=O)C2)C)c1 14218,c1(C(=O)NCC2(CNC(CC(COC)C)=O)CCCCC2)cnn2ncccc12 14219,C1(C(=O)NCC2CN(C(=O)CC3CSC3)C2)CCC(CC(F)(F)F)CC1 14220,C1(CNC(c2nn(CC)c(=O)cc2)=O)CC2(CCN(C(=O)C3=CCCC3)C2)CO1 14221,c1(NC(C)CN(C)C(c2cc(C3CCC3)on2)=O)ncc(C#N)cc1F 14222,C1(CCNC(c2csc(Br)n2)=O)CCCCN1C(C1(C2CC2)CC1)=O 14223,n1(CC(=O)N(C)C)cc(C(N2CC(C)(NC(C3CC4CC4C3)=O)C2)=O)cn1 14224,C1(CN(C)Cc2cccc(F)c2)CC(F)(F)C12CC2 14225,N1(C(CCN(C(CC(CC)C(C)C)=O)C(C)C)=O)CC2CCCC(O)C2C1 14226,C(=O)(CC(C)CC(C)(C)C)NC(C(C(=O)NCCC(CC)(F)F)C(C)C)C 14227,N1(C(c2ccnc(C)c2N)=O)CCCC(C)(C)C1C(=O)NCCC(C)C(F)F 14228,O(S(=O)(=O)c1cccc2c1OC(C)C2)c1n(C)nc(CC)c1C(=O)O 14229,CC1(C)OC2CC(C(=O)NCC3CN(C(=O)Cc4nnc(O)s4)CC3O)CC2O1 14230,Cc1n[nH]c(C)c1CC(=O)NC1CCC(CNC(c2cnsc2)=O)C1 14231,CCCC(=O)NCC(F)CNC(=O)COCCc1cccs1 14232,C1(C(=O)Nc2cccc(CCC)c2)CN(C(=O)COc2ccon2)CCC1CO 14233,N1(C(CCCC)=O)CCC2(CCC(N(C(C3CC3CC(C)(C)C)=O)CC)C2)C1 14234,N1(C(COc2cccc(C)c2)=O)CCC2CN(Cc3ccc(C)[nH]3)CC12 14235,c1(C(=O)NC(CC)C)cccc(C(=O)NC(C)(C)Cc2cccnc2)c1 14236,C#Cc1cncc(C(N2CC(F)CC2C(=O)Nc2ccc(O)cc2F)=O)c1 14237,C1(CC)CN2CCC1CC2=O.C(=O)(C(C)(C)C1CCC1)N(C(COC)C)C 14238,N1(C(CSc2n(C)cnn2)=O)CCC(C)(C)C(NC(=O)CSC(F)(F)F)C1 14239,C1(NC(C2CCCC2)=O)COCCN(C(=O)CC(O)Cc2ccccc2)C1 14240,C1(C(=O)NC(CC)CNC(=O)CN2CCCCC2)CCC2(CCC2)OC1 14241,c1(C(=O)NCCCN(C(C2CC3CC2C3)=O)CC)cc(S(=O)(=O)CC)cnc1O 14242,CC1CC(C(=O)NC2CS(=O)(=O)C2(C)C)CCN1C(c1cnnn1C(C)C)=O 14243,C=CC(C)CC(=O)N1CC(C(O)C(=O)NCc2cnoc2)C1 14244,Cc1n[nH]c(C)c1CCC(=O)NCC1CC1NC(c1coc(N(C)C(C)C)n1)=O 14245,c1(C(N(C)CC2COCCN2C(=O)CC2(C)CCCC2)=O)cccc(S(C)=O)c1 14246,N(C1c2ccccc2CC1NC(=O)C(O)P(C)(C)=O)C(C(CCSC)OC)=O 14247,c12c(cccc1C)C(=O)N1CC=CC1C(=O)N2.C1(CCCN(C)C)CCCC1 14248,C1(CNC(CC(CC)N(C(c2c(C)nc(CC)o2)=O)C)=O)CC12CCCCC2 14249,N1(C(CCC=CCC=C)=O)CCN(C(C2CCCN2C2CCCC2)=O)CC1C 14250,N1(C(C(C)=C2CC2)=O)CCC2C(CCN2C(=O)Cn2cnnn2)C1 14251,C(S(=O)CC(=O)N1CCC(Cc2nnc(OCC)o2)CC1)Cc1ncccc1C 14252,C1(NC(C(CC)COC)=O)CN(C(=O)CN2CCNC(=O)C2)CC(C)C1 14253,Cc1c(C(=O)NC2CC(C)CN(C(C3CCC(C)CC3)=O)C2)cccc1F 14254,C1(NC(c2occ(C(=O)OC)c2)=O)C2CC(CN(C(C3CCC3)=O)C2)C1CO 14255,CCCC(C(=O)NCC(C(C)C)NC(c1cn(CCCOC)nn1)=O)N(C)C 14256,N1(C(=O)NC(C)(C)C)CC2=C(C1)CN(CC1OCC(C)(C)C1)C2.C1(=O)CCN1 14257,N1(C(c2cc(CCC)[nH]n2)=O)CCCC(N(C)C(c2c[nH]c(=N)o2)=O)CC1 14258,Cc1ncc(C#N)cc1NC(=O)C(O)CCNC(C1C2CCCCCC12)=O 14259,N1(C(C2=CCN(C(c3c(C)n(C)cc3)=O)C2)=O)CCC(O)C(C)(C)C1 14260,CC1(C)CC(CNC2CNCC23CCCC3)CC(C)(C)O1 14261,C1(C(=O)NCCCN(C(=O)Cc2nn(C)cc2Br)CC)CC2CC(=O)C1C2 14262,C#CCCCCCC(=O)NCC1(O)CCN(C(=O)CC2CC(C)(C)CCO2)CC1 14263,Cc1cc(F)c(C(=O)NCCN(C(C2CCCC3CC23)=O)C2CC2)cc1F 14264,C1(C#N)(CC(=O)N(CCNC(C(C)OCC)=O)CCOC)CCCCC1 14265,c1(C(N2CCC(C(C)NC(C3CCN(C(C)(C)C)C3)=O)C2)=O)ccncc1I 14266,C1(C2CCC2)(NC(c2ccn(CCNC(CCSC(C)C)=O)n2)=O)CC1 14267,c1(CN2C3C(C(=O)Nc4c(OC)ccc(F)c4)C(C3)C2)cccc(F)c1C#N 14268,C1(CNC(CCOCCC)=O)CC(F)(F)CN1C(=O)Cc1ccn(C)n1 14269,c1(OC)cccc(CC(N2CC(N(C)C(C34CC(C)C3C4)=O)C3(CC3)C2)=O)c1F 14270,N1(C(C(C)=C(C)C)=O)CC2CC3CC2C1C3NC(=O)Cc1ccoc1 14271,Cc1ccccc1CC1CCN(C(C2(CN(C)C(c3cn(C)cn3)=O)CC2)=O)C1 14272,C1(N(C)CC)CCN(C(c2ccc(NC(C)=O)o2)=O)CC1 14273,C1(CNC(=O)C2=CCOCC2)CC2(CO1)CN(C(C1CC(=O)N(C3CC3)C1)=O)C2 14274,c1(C(N2CC(C=C)(CC(=O)NCCC3CCCC(C)C3)C2)=O)cc(C)n(C)c1C 14275,c1(C(=O)NC(C)C(C)NC(c2cnc3[nH]cncc2-3)=O)ccc2ncnn2n1 14276,Cc1nnc2n1CC(C(=O)NC(CNC(c1nccn3cnnc13)=O)C(C)C)C2 14277,C1(C(N(C2CN(C(C=C(CC)CC)=O)CC23CC3)C)=O)CC(=O)N(C)C(=O)N1 14278,C#Cc1cccc(C(N2CCOC(C)(CC)C2)C(=O)NC2CCCCC2)c1F 14279,c1(C(=O)NCC(C)CN(C(=O)C2=CCCC2C)C)cc2c([N+](=O)[O-])cccc2[nH]1 14280,C=C(C)C(C)(O)C(=O)NCC1(C)CCN(C(c2ccc(C)c(C(C)=O)c2)=O)C1 14281,C1(NC(c2cccs2)=O)CC(N=c2[nH]nc(-c3ccon3)s2)C1.O=C1CCCN1 14282,C12(CNC(C34CC(CC(C)O3)C4)=O)CN(C(=O)C=C3CCC3)CC1CCO2 14283,C1(OC)CCC(CC(=O)NCC2CC(C)N(C(=O)Cc3c(C)n[nH]c3C)C2)CC1 14284,C(=O)(C1=CC2(CCOC2)C1)N1C(C(N(C(C)C)CCOC2CCCCC2)=O)CCC1 14285,C1(C(N2CC(COC)(CNC(=O)Cc3cnoc3)C2)=O)CCC(C)(C)O1 14286,C12(N(c3ncnc(C)c3F)C3CCC3)CCCC1CN(C(=O)Cc1ccc(Cl)cn1)C2 14287,c1(CNc2c(OCC)ccc(C)c2)nc2cc(Cl)c(Cl)cc2[nH]1 14288,C1(CNC(c2c(CC)cncc2)=O)CN(C(c2nc(C)ccc2F)=O)CCC1C 14289,C(c1c(C)cc(C)cc1C)=CC(=O)N(CC(C)NC(c1snnc1C)=O)CC 14290,c1(C(N2CCCC(CN(C(CNC(CC)=O)=O)C)C2)=O)csc2ncnc(O)c12 14291,c1(C(=O)NC2CC2F)cc(F)cc(Cl)c1.C12CC(O)(C1)CNC2=O 14292,CCCC(C(=O)NCCN(c1ncnc(=N)[nH]1)CC)S(N)(=O)=O 14293,c1(C(=O)NC2CC3CC(NC(c4c(C)cns4)=O)C2C3)nc2ccccc2[nH]1 14294,c1(C(N2CC(N(C)C)C(C)(C)C2)=O)coc2c1CN(C(C1CCCC(O)C1)=O)C2 14295,C1(C)(C(N2CC(CNC(c3c(CC)occ3)=O)C(O)C2)=O)Cc2ccccc2C1 14296,C1(NC(CCCC(C)=O)=O)CCN(C)C12CCCN(C(C1CCC(=O)N1)=O)C2 14297,Cc1cc(NCC2CN(C(=O)C(F)(F)C(O)C3CC3)CC2C)ncc1C#N 14298,CCC(O)C(F)(F)C(=O)N1CCN(C(=O)CN2CCNC(=O)C2)C(CC(F)F)C1 14299,C1(NC(c2c(OC)c(F)ncc2)=O)CC2(CCN(C(c3scnc3Cl)=O)C2)C1 14300,N1(C(C(CCC)C)=O)C2CCC1CN(C(C1CCN(CC(C)C)CC1C)=O)CC2 14301,N1(C(c2c(OC)csc2)=O)CC2CCCC(NC(c3cc(N)nc(Cl)c3)=O)C2C1 14302,C(C(=O)NC1C=CC(C(=O)NCc2c[nH]nc2C2CC2)C1)(C(C)C)OCC 14303,C1(NC(CC(C(=C)C)OCC)=O)C2CCCN(C(C3CCCC3F)=O)C2C1(C)C 14304,c1(C(N2CCCN(C(c3ccco3)=O)CC2)=O)ccc(Br)c(O)n1 14305,Cn1nnc2cc(CN3CCN(c4ccc(Cl)cc4Cl)CC3)cnc12 14306,Cc1cc(N)n2ncc(C(N3CCC3CNC(C3(C(=O)N(C)C)CC3)=O)=O)c2n1 14307,CC(C)CC(C)(O)C(=O)NC1CCC1C(=O)NC1CCCC(CO)C1 14308,c1(C(=O)NCC2(CNC(c3cnc(CC(C)C)nc3)=O)CC2)cc(F)cc(N)c1F 14309,C1(OCCCC)CC(C(=O)Oc2cnccc2N2CCCCC2)C1(C)C 14310,O=C(C(O)C(F)(F)F)N1CCOCCC1C(=O)N(C1CCC1)C1CCC1 14311,CCC(C#N)C(=O)NCC(C)CN(C(=O)Cc1ncc(Br)s1)C 14312,c1(C(N2C(CCNC(CCC(N)=O)=O)CCCC2)=O)cc(S(N)(=O)=O)c(Cl)o1 14313,c1(C(C)C)c(F)ccc(C(N2CCC3(CC3C(N3C4COCC3C4)=O)C2)=O)c1F 14314,C=C(CNC(C1CC12CCN(CC(CO)C(F)(F)F)CC2)=O)C1CCOCC1 14315,C1(N(C(C(CCC)N(C)C)=O)C)CCCN(C(c2cnc(O)o2)=O)CC1 14316,c1(CNC(C2C(c3ccc(C)o3)C2)=O)cccc(N=c2cc[nH]cc2)c1 14317,N1(C(c2c(C)cc(SC)o2)=O)CC2CC(NC(C3CCCC3(C)C)=O)C2C1 14318,C1(CCNC(CSC)=O)CCN(C(c2noc3cc(Cl)ccc23)=O)CCC1(F)F 14319,C1(OCC)CCN(C(=O)N(C(C)C)CC2CC2c2ccccc2)CC1 14320,N1(C(CC(C)OC(C(CCCC)O)=O)=O)CC2(CCCCCC2)C1 14321,O=C(C(O)C1CN(C(=O)CC2CC2)C1)NC(CC(O)CO)C1CC1 14322,C1(C(=O)NCCC2N(C(CSCCCC)=O)CCOC2)CCC(C)=C(C)C1 14323,N1(C(C(CN(C)C)NC(=O)C(C2CCOCC2)F)=O)CCCC2(CC1)CC2 14324,C(=O)(C1=NOC2(CCC2)C1)N(CCNC(c1n(C)c(S)nn1)=O)C1CC1 14325,CC1=CCC(N=c2ccc(Br)c(S(=O)(=O)NC3CCC4(CC3)OCCO4)[nH]2)CC1 14326,C(c1cc(Cl)c2c(c1)OCO2)=CC(=O)NC1CC(NC(C2(C)CC(F)(F)C2)=O)C1 14327,S(=O)(=O)(c1ccc(Cl)cc1)N1CC(n2ncc(N(C(CCC)C)C)c2)C1 14328,c1(C(=O)OC)cc(-n2cc(SCc3nocc3Br)nn2)nn1C 14329,c1(C(=O)NCC2C3CN(C(C(C(C)C)OC)=O)C2C3)cc(Cl)cc2cccnc12 14330,C12(NC(C(C)(C)F)=O)CC(CNC(c3cccc(F)c3O)=O)(C1)OC21CCC1 14331,C(=O)(CC(C(F)(F)F)NC(=O)Cn1ccc(C)n1)NCCC1ON=C(C)C1 14332,Cn1ncc2cccc(CNC(N3CCC4CNCC4C3)=O)c12 14333,CC1(C#CC(=O)NCCc2ocnc2C(=O)NC2C3COCC23)COC1 14334,S(=O)(=O)(c1cc(C(=O)O)cc(C(=O)O)c1)N1CCCC(N(C)C)(C(N)=O)C1 14335,c1(C(N2CCC(C)(NC(c3cc(CC)oc3C)=O)C2)=O)oc2ccccc2c1Cl 14336,c1(C(C)C)cccc(F)c1C(=O)NC1CC(NC(C2C3CC4C(C3)C24)=O)C1 14337,C#CCCCCC(=O)NC(Cn1cccn1)C(=O)N(C1CCC1(C)C)C 14338,c1(C(=O)NCC(C2CC2)NC(C(CSC)C)=O)cnc(O)c(C(F)(F)F)c1 14339,Cc1cc(=O)n(CCC(N2CCC(NC(c3cnns3)=O)C2C(C)(C)C)=O)cn1 14340,C=CCC(CO)NC(c1ccc(CNC(C2CCC(O)C2)=O)o1)=O 14341,C1(CN(C)C(C23CC(C)(C2)C3)=O)CCN(C(C2CC23CCC3)=O)CC1 14342,C1(N(C(C(=O)NS(=O)(=O)CC)=O)CCCNC)CCCN(C(C2CC2(F)F)=O)C1 14343,C1(CNC(CCCC#C)=O)COC(C)(C)CN1C(C1(C)CCC(=O)C1)=O 14344,C=CC(CCC)CC(=O)NCCC1CCCN(C(C2(C(C)C)CCC2)=O)C1 14345,c1(C(=O)NCCNC(c2c(C)n3c(s2)ncc3)=O)cc2c(s1)CC(C)CC2C 14346,c1(N2CCCC(C(C)NC(CC=CC=C)=O)C2)nc2ccccc2s1 14347,n1(CC(=O)NC(C)CNC(C2(C)CC2(C)C)=O)c(-c2cccs2)nnc1S 14348,c1(CC)nn(C2CC2)cc1C(=O)NC(CNC(C1C2COCC12)=O)CC(C)C 14349,c1(C(N2CC(NC(CCSCC)=O)C(C)CC2)=O)nn2c(c1C)OCCC2 14350,CCC(CC)(CC)C(=O)N1CCC(N(C)C(c2csc(C3CCCC3)n2)=O)C1 14351,C#Cc1ccc(C(=O)N(C2CCCN(C(c3ccn(C4CCC4)n3)=O)C2)C)nc1 14352,C(CNC(c1cccn(C)c1=O)=O)(CC(F)(F)F)NC(CCC=CCC=C)=O 14353,c1(CNC(=O)C#CC2CCCO2)nc2c(s1)CN(C(c1ncc(F)cn1)=O)CC2 14354,c1(OC)ccc(S(=O)(=O)Nc2cccc(OC)c2OC(F)F)c2ncccc12 14355,C(CCC(N)=O)(C(=O)NCc1cc(C2CC2)n[nH]1)n1cc(COC(C)(C)C)nn1 14356,N(C1CCCn2ncnc21)C(CC(C(F)(F)F)NC(c1ccc(O)nn1)=O)=O 14357,CN1N=CCCC1C(N1CC(NC(=O)CCc2cccc(F)c2)C(O)C1)=O 14358,CC1=C(C(=O)NC2C(C)(C)C(NC(C3C4(CC4)C34CC4)=O)C2(C)C)CCCO1 14359,c1(CC)nc(NC2CC(F)(CNC(C3CN(C)CC(C)O3)=O)C2)c(C#N)cc1C 14360,N1(C(CCC(=C)C)=O)CCC(NC(c2ccc(OC(F)F)cn2)=O)CC1C1CC1 14361,C(c1ccc(Br)cc1)=CCC(=O)N(CC(C(=O)NC)C)C1CC1 14362,N1(C(COCc2cc(C)no2)=O)CCCC1(C)CNC(c1nccs1)=O 14363,c1(C(F)(F)F)nc(NC(CC2CC2)C2CC2)cc(N2CCC3(CC3)C2)n1 14364,C(=O)(C(CC1CCCCC1)C(C)C)NCC1CN(C(CCC(=C)Cl)=O)CC1O 14365,CC1CCCC=C1C(=O)NCC1CC(O)CN1C(c1coc(C(N)=O)c1)=O 14366,C#CC1CCC(C(=O)NCCN(C(=O)C(C)N2CC(C)C2)CCOC)CC1 14367,C12(C(N3CC(CN(C(=O)Cc4ccc(O)cc4)C)C3)=O)CCCC1OCC2 14368,C1(O)(C(C)NC(CSCCC)=O)CCN(C(C2C=CC=CC=C2)=O)CC1 14369,C(CC(C(=O)N1CC(c2csc(O)n2)C1)NC(=O)Cc1ncoc1C)OC 14370,C1(C(=O)NC2C(CCC)C2)CCCN(C(c2ccccc2N(C)CC)=O)CCC1 14371,Cn1[nH]nnc1=NCCCC(C)(C)NC(C1(c2cccc(F)c2)CC1)=O 14372,c1(OC)ccc2c(c1)c(C(N1CC3CCN(C(c4cncs4)=O)C3C1)=O)c(C)n2C 14373,c1(CC)ncc(NC(C)CN(C(=O)C(C)OCC2CC2)C)s1.C1(C)C(=O)N1 14374,N1(C(c2ccc(Cl)cc2)C(=O)NCCC#N)CCCN2CCCCC12 14375,C(=O)(C1=CN2CCS(=O)(=O)N=C2C=C1)NC(C)CN(C)C(C1CC(F)(F)C1)=O 14376,Cc1nn(C)c(C(N2CC3C(NC(C4CC4CF)=O)C3C2)=O)c1I 14377,c1(C(N2CC(SC)C(NC(=O)CCC(N)=O)C2)=O)cc(C)cc(O)n1 14378,C(=O)(C(C)(CC)CCCCCC)NC1C(NC(CCCC=C)=O)CCC1 14379,Cc1ccc(C(N2CC(N(C)C(C3CC(CN(C)C)C3)=O)C3(CC3)C2)=O)c(CO)c1 14380,N1(C(CNC(C(C)C)=O)=O)CCN(C(=O)CNC(=O)Cc2cc(C)nn2C)CC1 14381,C1(C)(CC)CCC(C(=O)NC2CC(CCNc3ncncc3Br)C2)O1 14382,c1(C(=O)NC(CC#C)COCC(F)(F)F)cc(C)ccc1N 14383,c1(OC)cc(C(=O)NCCC2CC(NC(c3c(C)nn(C)c3N)=O)C2)nc(C)c1 14384,N1(C(CCn2cc(C(CCC)=O)nn2)=O)CCCCC(C(=O)NC2CC2)C1 14385,O=S(=O)(c1ccc2nc(N3CCC(CF)C3)sc2c1)Nc1cccnn1 14386,c1(CC(=O)NC(C2CCN(C(c3cncnc3)=O)CC2)C)ccccc1S(C)=O 14387,C1(n2c(CCOC)nc(-c3ccc(OCC)cc3)n2)C(C)CCCC1C 14388,N1(C(c2c(OC)nc(C)nc2)=O)CCCN(C(c2ccc(F)cc2C)=O)CC1C 14389,c1(CNC(CCC)C)cc(=NCCc2cnc3ncccn23)[nH]c(C(F)(F)F)n1 14390,CCCC(CCC)CC(=O)N1CCOCC1CNC(=O)C(C)(CC)CO 14391,CONC(=O)COC1(C(=O)NC)CC1.c12coc(n1)CNC2=O 14392,C1(CC(=O)NCC(C)=O)C(CCC(C)C)NC1=O 14393,C1(NC(c2cc(C3CC3)cs2)=O)CCN(C(C2CCCCS2(=O)=O)=O)CC(O)C1 14394,N1(C(CSCC#C)=O)CCN(C(=O)CCCc2cc[nH]n2)C2CC12 14395,C1(Cc2c(F)cccc2)CCN(N2CCN(C3CCOC3)CC2)C1.C1C(=O)O1 14396,CC(CC#N)N=c1[nH]c(=NCCNC(c2cccc(Cl)c2)=O)c2ncccc2[nH]1 14397,N1(C(C(CC=CCC)C)=O)C(CC(N2CC3CC(OC)C3C2)=O)C2CCCC12 14398,c1(C(=O)NCC2CC(NC(C3(CC)COC3)=O)C2)cc(C)c(O)c(C)c1 14399,c1(CC)cccnc1C(=O)NCCC(C)CCNC(C1CNC(=O)N1)=O 14400,c1(C(=O)NC2CN(C(c3c(C)onc3Br)=O)C2)cnn2c1OCC(C)C2 14401,C(=O)(C(C)CC(C)C)N1CCC(N(C(C(C(=O)OCC)F)=O)C)CC1 14402,c1(C(=O)NCC23CC(C(N(C(CC)CO)CC)=O)(C2)C3)cc(Br)cc(F)c1F 14403,N1(C(Cn2c(C)ncc2)=O)CC2C(C(=O)NC(C)C(C)CO)C2C1 14404,c1(C(=O)NC2(CC(=O)NC3CCCC(C(=O)OC)C3)CCC2)ccc(Cl)c(C)c1F 14405,N(C(=S)N1CCC1C(=O)Nc1ccccc1OC1CC1)C(C)(C)C 14406,Cn1cc(CC(=O)NCC2(C)CCCN2C(=O)CCC2(C)CC2)c(Cl)n1 14407,CCC(C)(C)CCNC(=O)CC(CNC(=O)CNc1ncccn1)C1CCC1 14408,C(C)(C)(CC(=O)NCCC(O)CNC(=O)CCCCC1CCCCC1)OC 14409,C1(C(N2CC(NC(C(CC)(C)O)=O)C(C)C2)=O)CC(c2cccnc2)=NO1 14410,C1(N(C(c2ccc(CC)o2)=O)C)CN(C(c2ccnn2CC(C)C)=O)CC1O 14411,c1(C(=O)NC2(CF)CCN(C(C(COC)O)=O)C2)cc(F)c(SC)cc1N 14412,C1(CC)C(C(=O)N(C)Cc2cccc(OC)c2)CCN1C(c1cnn(C)c1Cl)=O 14413,N1(C(C(F)(F)C2(OC)CCC2)=O)CCC(NC(=O)C2=CCCCC2)CC(C)(C)C1 14414,N1(C(C2C(OCC)C2)=O)CCC(C)C(NC(=O)C(C)(C)CO)C1 14415,CCC(CC)C(C(=O)N1CCCOC(CCSc2ccc(C)cc2)C1)OC 14416,c1(CNC(CSCC=C)=O)cnn2c1CN(C(c1cc(CC)no1)=O)CC2 14417,N1(C(CC(=C)C)=O)CCC2CCN(C(C3CC(C)(C)CN3C)=O)CC2C1 14418,C1(C(=O)NCC(C)OCC)CN(C(c2cc(Br)cs2)=O)CCS1 14419,C#Cc1cccc(C(=O)NC2CCN(C(C3C=CC=CC=C3)=O)C(C3CC3)C2)c1Cl 14420,c1(N2CCC(C(CC)CC)CC2)nc2c(c(=NC3CCSC3)[nH]1)CCCCC2 14421,C(C(CO)(CO)NC(c1cncnc1)=O)N(C(C1C(OC)CC1)=O)C 14422,c1(C(=O)Nc2ccc(OCC(=O)NCC)cc2)c(C#N)cnn1C 14423,C1(C(C(=O)NC(CC(=O)OC)C)N)CC2CCC(C1)N2 14424,c1(C(=O)NC23C(CN(C(C(C)CF)=O)C2)C3)cccc2c1OCCO2 14425,C1(C(N2CC(C(=O)OC)(COCc3cc(OC)no3)C2)=O)CCCCN1C(C)C 14426,C(CC(C)(C)C(=O)N1CCCC(NC(c2csc(Br)c2Cl)=O)C1)OC 14427,C1(NC(C(CCCOC)NC(c2cc[nH]n2)=O)=O)CCCCCC1(C)C 14428,N1(C(=O)OC)CCCC(CSC2CCN(C(=O)NCCC#N)C2)C1 14429,N1(C(C(CC=CC)CC)=O)CCCN(C(=O)C(C#N)C(C)C)C(C)C1 14430,N=c1cc[nH]cc1C(=O)NCC(O)CCNC(c1ccnc(OCCO)c1)=O 14431,C1(O)(CNC(Cc2ccc(C)cc2)=O)CCCN(C(c2nn(C)c(C)c2Cl)=O)C1 14432,c1(C(=O)NCCCN2CCN(C(COC(CC)C)=O)CC2)c(C)nc(O)nc1C 14433,Cc1nc(CN)sc1C(=O)NCC1CC1c1ccco1 14434,Cc1c[nH]cc1C(=O)N(C)CCOCCNC(C1CC1CF)=O 14435,C12(CNC(C3C(OC)C3)=O)CC(NC(=O)CC(C)F)(C1)C(C)(C)O2 14436,C1(N)(C(=O)NC(c2nc(CC)on2)C)CCCN(C(=O)N(C)C)C1 14437,CCCC(CC)CCC(=O)NC12CC(C(N3CC(O)(CO)C3)=O)(C1)C2 14438,CCCCS(=O)(=O)NCC(=O)NC1CC1NC(c1ccc(CSC)cn1)=O 14439,C(=O)(C(CC(N)=O)NC(c1cc(C)n(C)c1)=O)NCCCOCCCC 14440,c1(COCC)nc(CSC)n(C(C2CC2OC)=O)n1.c1(C(F)CO)ccccn1 14441,N1(C(CSCC=C)=O)CCCN(C(C2(C3CC3)CC2)=O)CC1c1ccccc1 14442,N1(C(CN2C(C)CCC2)=O)CC=CC(NC(C2CC2C)=O)C1 14443,N1(C(c2n(CC)cnn2)=O)CCOC2(C1)CN(C(c1cnn(C)c1F)=O)C2 14444,C1(NC(c2c(C(C)O)cccc2)=O)CCN(C(C2CC(O)C2)=O)C(C)C1 14445,C1(C2(O)CCC2)(C(=O)NCC(CCNC(CCCC=C)=O)O)CC1 14446,CCC(C)(C)CCCC(=O)NC1CCN(C(c2cc(C)cc(F)c2)=O)C12CC2 14447,c1(NC(N(C)CC2CCNC2)=O)cccnc1Oc1ccccc1 14448,C1(C(N2CCC(NC(=O)COC)C2)C(=O)NCCCC)CCCC1S(C)(=O)=O 14449,c1(C(=O)NC2CN(C(=O)C(C3CC=CCC3)F)C2)cncc2nc[nH]c12 14450,C=Cc1ccccc1NC(C)(CCC=C)C1OCCO1 14451,Cc1c(C(=O)NCC(C2CCCC2)NC(=O)CCF)cc(-c2ccccc2)n1C 14452,N1(C(CC2(OC)CCC2)=O)CCN(C(c2cccc(F)c2O)=O)C2(CC2)C1 14453,N1(C(C2(C)C=CCCC2)=O)CCC2CCN(C(c3nc[nH]c4ncnc3-4)=O)CC12 14454,C1(O)(CNC(COCCNC(c2c(C)scc2)=O)=O)CCCCC1 14455,C1(C(=O)NCCN(C(=O)CC2(C(F)F)CC2)C(C)C)CCC(C(F)(F)F)O1 14456,CC1CN(C(C2CC3C(C2)C3(F)F)=O)CCC1CNC(c1c[nH]c(C(N)=O)c1)=O 14457,c1(CC(N2CC3(CC(CNC(C(C)(C)C4CC4)=O)C3)C2)=O)csc2ccccc12 14458,N1(C(C2CCCO2)=O)CC2(C(=O)NCC3=CCSC3)CC1CO2 14459,N(C1CC2(CN(C(=O)C=CCF)C2)n2ccnc21)C(C1C2C(=O)C3C(C2)C31)=O 14460,C1(C(=O)NCc2nc(CNC(=O)OC(C)(C)C)oc2)CCc2nnc(O)n2C1 14461,Cc1cccc(NC(=O)C(Cc2cc[nH]n2)NC(=O)CCN=[N+]=[N-])c1 14462,CCCCC(C(=O)N1CCN(C(c2cc(CO)on2)=O)CC1CC)N(C)C 14463,c1(-c2onc(-c3c(O)ccc(C#C)c3)n2)ccc2ccccc2c1 14464,C(=O)(C(C)S(N)(=O)=O)NCCC1(O)CN(C(c2c(C)n(C)c(C(C)(C)C)c2)=O)C1 14465,C(=O)(CC1C(=O)Nc2ccccc21)NCC(CO)NC(CC(C)(C)CC(F)F)=O 14466,C1(C2CCNCC2)(C(=O)NC(C)CCc2ccccc2)CCC1 14467,C(=O)(C(C)CC(C)(F)F)NCC(c1cccc(C)c1)NC(=O)C(CO)N(C)C 14468,C1(NC(C(=O)N(C)Cc2cccnc2Br)=O)CCCN2CCCCC12 14469,C(=O)(CCCCC(N)=O)N(C1CCCN(C(C2CC23CC(O)C3)=O)C1)CC 14470,CC1OC2(C(=O)NC3CC(O)(CNC(=O)CNC=O)C3)CCC1CC2 14471,c1(CC)nc(N2CC=CC(NC(c3ccc(C)s3)=O)C2)[nH]c(=N)n1 14472,CCC(C)(C)C(C)CC(=O)NC1CC2CCC1(NC(=O)CN(CC(C)(C)C)C)C2 14473,c1(C(=O)NCC2(C(=O)NCC3CCC(CC)O3)CCCC2)cc[n+]([O-])cc1 14474,c1(C(C(F)(F)F)N(C(c2ccc(C)o2)C)C(N2CC(F)(F)C2)=O)ccc(O)cc1 14475,C1(NC(=O)CN2CCCOC2=O)CC2(CCN(C(C3(F)CCOC3)=O)CC2)C1 14476,C1(C(N)=O)CCC(CCC(=O)NCC2CCN2C(c2ccsc2Cl)=O)O1 14477,c1(OC)ccncc1C(=O)N(C)CCN(C(c1ccn(C)n1)=O)C(C)C 14478,c1(C(N2CC3(CCN3C(=O)CCc3cc(Cl)cs3)C2)=O)cc2n(c1)CCOC2 14479,N1(C(CC=CCC)=O)CCCC(C(N2CCC2C)=O)C1.C(C)(=O)O 14480,c1(C(=O)NCC(C)N(C(=O)CC2C=NN(C)C2=O)C)coc2c(Cl)cccc12 14481,C1(NC(C2(C(=O)NC)CCC2)=O)CCC(Nc2ncncc2I)CC1 14482,c1(CNC(c2c(C)n[nH]c2)=O)ccc(CNC(c2c[nH]c(C(F)(F)F)c2)=O)cc1 14483,C1(C(=O)NC2CCC(NC(c3cc(C)ncc3)=O)C2)CC12CCCCC2 14484,C(=O)(C(CCC=C)NC(=O)C(c1cnn(C)c1)=O)NC(C#C)CC1CCCC1 14485,C1(CNC(=O)C=Cc2cn[nH]c2)(NC(C2CC3CC3C2)=O)CC2CCC1C2 14486,c1(C(=O)NCC(c2cccs2)N)ccc(NCC(F)(F)F)nc1 14487,C(CC(F)=C(F)F)NC(COCCNC(C1CCC(C)O1)=O)=O 14488,CCC(CC(=O)NCC1(O)CC(NC(c2cccc(F)c2)=O)C1)OC 14489,c1(C(N(C2CCN(C(CSCC=C)=O)C2)C)=O)cc(C)nc(N2CCCC2)n1 14490,C1(NC(CC2C(C)C2)=O)CCN(C(=O)Cc2ccc(Cl)nc2)C12CCC2 14491,N1(C(C(CC(N)=O)O)=O)CCN(C(=O)Cc2noc3ccccc23)CC(CO)C1 14492,C1(C(CNCc2nnnn2-c2cnccc2C(F)(F)F)OC)C=CCCC1CO 14493,N(C1CC2(CN(C(=O)CC(C)SC)C2)n2ccnc21)C(C(CC)(C)CC)=O 14494,C1(CNC(c2ccno2)=O)CN(C(=O)COC2CC2(F)F)C2(CCC2)C1 14495,C(=O)(C(C)(C)CC(C)C)NC1CCN(C(CC(CSC)(C)C)=O)C1 14496,N1(C(CCOC)=O)CCCC1C(C)(C)CNC(C1C(C)C1(F)F)=O 14497,C(=O)(C(C)(C)C(F)F)NC1CC2(C(NC(c3cc(COC)cn3C)=O)C2)C1 14498,c1(CC)ccccc1NC(=O)C#CCNC(=O)C(C)O 14499,C1(NC(C2CC(OCC)C2)=O)CCCC(NC(=O)CCc2cncc(F)c2)CC1 14500,C12(C(N3CCC(CNC(C4(CC5CC5)CC4)=O)C3)=O)CCCCC1OCC2 14501,C1(CC(=O)NCCC(C(C)C)NC(C23CC=CC(C2)OC3)=O)CN2CCC1CC2 14502,c1(NC(CC(C(C)(C)OC(C)C)C)=O)cccn2nccc12.C1CC(=O)N1 14503,C=C(Cl)C(C)(C)C(=O)NCC=CCNC(c1cc(NC)nnc1C(=O)NC)=O 14504,Cc1c(C(=O)NCc2ccsc2C(=O)NCC2CCN2C(C)(C)C)cccc1F 14505,c1(C(=O)NCCN(C)C(c2ccc(N)c(Cl)c2)=O)nsc2ccccc12 14506,C(=O)(C1=CC2(CN(C(=O)NC3CCO3)C2)OC1)NCCOC 14507,O=C(CCCN1CCCC1)NCC1C=CC(NC(C2(n3ccnn3)CC2)=O)C1 14508,C(CNC(=O)CC1CCC1(C)C)(C(C)(C)C)NC(C(C)OC(C)(C)C)=O 14509,N1(C(c2c(O)ccc(C)n2)=O)CCCC2C1CCCN2C(=O)CN1CC(C)C1 14510,c1(C(=O)NCC(C)CN(C(=O)CC(C)CN(C)C)C)cnn2ccncc12 14511,c12cccc(n1)S2.CC1(C(N2CC(NC(=O)COC(F)(F)F)C2)=O)COC1 14512,C1(NC(c2ccc(C)o2)=O)CC(O)CN(C(=O)COCC2CCCC2)C1 14513,Cc1ccc(C)c(C(N2CCN(CCCNC(C3CC4(CC4)CO3)=O)CC2)=O)n1 14514,c1(CCC(N2CCC(Cc3c(C)ncs3)C2)=O)ccc(NC(=O)OCC(C)C)cc1 14515,c1(OCC(N2CCC(CNC(=O)C(CO)c3ccccc3)C2)=O)cccc(Cl)c1 14516,CCCN=C(NCCCCN1CC(C)CC(C)C1)N1CCC(Cc2ccsc2)C1 14517,c1(C(=O)NC2(CNC(CCc3c(C)ncs3)=O)CCCC2)cc(C)n(C)n1 14518,C1(C)(CC)CC(C(N2CC(N(C(=O)CCc3cc[nH]n3)C)C2)=O)C1 14519,c1(C(N2CCCC(N(C(C34CC(C)C3C4)=O)C)C2)=O)cccc(C#CC2CC2)c1 14520,C1(O)(CCNC(C2CCCN(C(C)C)C2)=O)CCCN(C(=O)COCCF)C1 14521,c1(C(=O)NCC(CNC(CCCCC#C)=O)(C)F)ccc2cccnc2n1 14522,CCCCN=C(NCC(C)CC(F)(F)F)N1CCCC(O)(CO)C1 14523,C1(C(=O)NCCC(C)(C)N(C)C)(CNC(CCCSC)=O)CC2(CC2)C1 14524,N1(C(CCCCC)=O)CC2CCC(C1)N2C(=O)CC1(O)CCOCC1 14525,C(=O)(C1SCc2cccnc21)N1C(CNC(c2c(Cl)cnc(CC)n2)=O)CCC1 14526,N1(C(CCCOC)=O)CCN(C(C2(NC(C)=O)CCCC2)=O)CC1CCOC 14527,c1(C(=O)NC2CN(C(C3CCCCO3)=O)C2)cc([N+](=O)[O-])c2nsnc2c1 14528,c1(C(=O)OC)cc(CN(C(C)CS(C)=O)C)c(Br)cn1 14529,CC(C)CCCCCC(=O)N1CCC(O)(CNC(=O)C2=CC3C=CC2C3)C1 14530,c1(C(N(C2C(C)CN(C(C3C4COCC34)=O)CC2)C)=O)c[nH]c2cc(O)ccc12 14531,Cc1cc(Br)cnc1C(N1CCCC1CCC(=O)Nc1cn(C)nn1)=O 14532,C(=O)(C(C)C(=O)NCc1ccc(C(=O)NC2CC(=O)N(C)C2)nc1)OC 14533,c1(CCC)ccc(C=CC(=O)N(CCC(C(C)C)NC(=O)C(O)CCC)C)cc1 14534,Cc1ccc(F)c(C(=O)N(CCCOCCN(C)C(c2cnc(Cl)[nH]2)=O)C)c1F 14535,C(=O)(C(F)C(F)(F)F)NC(C1N(C(c2cc(SC)ncc2)=O)CCC1)C 14536,CCC(CC)(CCNC(c1cc(C)ccn1)=O)NC(=O)C(c1cccc(C)c1)=O 14537,N1(C(COC)=O)CC(C)(C)CCC1CNC(=O)CS(=O)(=O)CC1CCCO1 14538,Cc1cnccc1C(C(=O)NCC(C)C)N(CC(N1CCCCC1)C)C 14539,N1(C(C2CC(SC)C2)=O)CC(NC(c2cc(C)c(N)cc2Cl)=O)CCC(O)C1 14540,c1(OC(C)C(=O)NC2(C)CCN(C(=O)CC(C)(C)C3CC3)C2)ccc(F)cc1 14541,N1(C(C(C)NC(C)=O)=O)C(C(=O)N(C2CCN(C)C2=O)C)C2CC(O)C1C2 14542,C1(NC(C(F)=CCC)=O)CCC(NC(=O)CCCC2CCCC2)C1 14543,n1(CC)nc(C(N2CCN(C(C3ON=C(C)C3C)=O)CC2COC)=O)ccc1=O 14544,N1(C(c2cncc(C(=O)OC)n2)=O)CCCN(C(=O)C2=COCC2)CC1CO 14545,N1(C(c2c(OC)cncn2)=O)CC2(CC(NC(=O)CSC(C)(C)C)c3nccn32)C1 14546,C(=O)(CCC(F)(F)F)N1CC(NC(C(C)NC(CC)=O)=O)C(N(C)C)C1 14547,C1(CC(=O)NCC2C(C(=O)NCC3(C(C)(F)F)CC3)COC2)CCCCCC1 14548,CC1CCC2(CN1S(=O)(=O)c1ccc(F)cc1Br)OCCC2 14549,C=CCCN=C(NCCOc1ccc(F)cc1)NCCNC1(C)CC1(F)Cl 14550,C1(N(C)C(c2coc(C(F)F)n2)=O)CCN(C(c2cc(Br)n(C)c2)=O)CC1 14551,N1(C(c2c(OC)scc2)=O)CCN(C(=O)C=CC2CC2)CC1 14552,CC(C)(C(=O)NC(C1CCOC1)CNC(c1csc(O)n1)=O)c1cnsc1 14553,C12(CCCC1C)C(=O)N2.c1(OCC(N2CCC(OC(C)C)C2)=O)cccc(O)c1 14554,c1(C(=O)OC)c[nH]c2cc(NC(=O)C(=O)NCCC3CCC(C)(C)C3)ccc12 14555,c1(C(=O)NCC2CN(Cc3ccc(-c4cccs4)s3)C2)n[nH]cc1I 14556,C=C1CC2CC1CN2C(=O)CC1CC(C)N(C(c2cnn(C)c2C=C)=O)C1 14557,n1(CCCC)nc(C)c(C=CC(N2CC(C(C(=O)O)C(C)C)C2)=O)c1Cl 14558,c1(CN2CCC(O)C(O)C2)ccc2nn[nH]c2c1 14559,C=C(C)C1CCC(C)(O)C(NC(=O)N(CCNc2ccc3c(c2)CCO3)CC)C1 14560,N(C(=NCC(C)C)N1CCCCC(C)(F)C1)CC1(OCC)CC1 14561,C1(NC(C2C(N)CCC2)=O)CCCC(F)(F)C1 14562,c1(CNC2C(C(N(CCCC)C)=O)C2)sc2ccccc2c1Br 14563,CC(C)CC(C)(C(N)=O)NC(c1ccc(CNC(c2cncn2C)=O)nc1)=O 14564,Cc1cc(=O)oc(C)c1C(=O)N(CCCCCNC(c1c(C)cnnc1O)=O)C 14565,C1(NC(C2(OC)CC2)=O)CCC2CCN(C(c3c(C(F)F)cccc3N)=O)C1C2 14566,C12(CNC(C=COCC)=O)CCCCC1CN(C(c1ccc(SC)o1)=O)C2 14567,CC1CCCN1CCSc1cn(C2CCC(C(=O)Nc3cnc(C4CC4)s3)C2)nn1 14568,C1(C#N)(C(=O)NC(C2CN(C(c3cc(CO)ncn3)=O)CCO2)C)CCOCC1 14569,Cc1ccnc(C(N2CCC2C2CC2c2cccs2)=O)c1.C1(C=O)CC(F)(F)C1 14570,Cc1cnc2cc(C(=O)N(C)CCNC(=O)CCn3cncn3)ccn12 14571,C(=O)(C1=CC2CCCC12)NC12CN(C(CSCC=C)=O)C(CO)(C1)C2 14572,C(=O)(C1=C(Cl)CCOC1)N1CCN(C2CCCN(C(C3C(C)C3C)=O)C2)CC1 14573,C(c1cncc(OC)c1)=CC(=O)NCC(C1CCC1)NC(c1n(CC)ncc1)=O 14574,CCC(CC(=O)NC1CCCC(CC(=O)NCCC(C)(C)OC)C1)OC 14575,CC(C)C(F)(F)CC(=O)NC(C)(CNC(c1ccc2[nH]ccc2c1)=O)C1CC1 14576,CC1(C)C(NC(=O)CC2CCC(O)C2)C1C(=O)NCCN1CCCC1=O 14577,Cn1nccc1C(O)C(=O)NCC1CCCN1C(C1CC(CC(F)F)C1)=O 14578,CC1CC2(CC(C(N3CCCC3CCC(N3CCC(CC(F)F)C3)=O)=O)C2)C1 14579,C=CCCC(C)(C)C(=O)N(C)CCOCCNC(c1nn[nH]c1C(C)C)=O 14580,N1(C(c2nc(C(C)C)oc2)=O)CCCC(C2(NC(C3CC3(C)C)=O)CC2)C1 14581,c1(C(=O)NCCCCCNC(C(C)SCCOC)=O)cc(Cl)cnc1NC(C)=O 14582,c1(C(=O)NC(C2CCCN2C(c2cc(Br)n(C)n2)=O)C)ccc[n+]([O-])c1 14583,N1(C(C(CC)n2cncn2)=O)CC(NC(=O)CC2CCN(CCF)CC2)C(O)C1 14584,C1(=O)CCC(=O)NCC2C(C2)N1.C(O)(C(C)C)C1(NC(C=C(C)Cl)=O)CC1 14585,C(C)(C(=O)NCC1(CNC(CC2(N(CCC)C(C)C)CC2)=O)CC1)C(=O)N.C 14586,c1(CCC(=O)NC2CC(NC(=O)Cc3cnn(C(F)F)c3)C2)ccc([N+](=O)[O-])cc1 14587,C1(C(N2CC3C(CN(C(Cc4ccc(C)o4)=O)C)C3C2)=O)CC2OC(=O)OC2C1 14588,C12(C(N3C(CC(NOCC(N)=O)=O)CCC3)=O)CCCC1C2(F)F 14589,Cc1ccc2nc(C(N3CCOCC3CNC(C3(C)CC=CCC3)=O)=O)cn2c1 14590,C(=O)(CC(CC)C(C)(C)C)N(CC(=O)N(C(C=C)C)CC)CC(C)C 14591,N1(C(c2cn(CCCC)nn2)=O)CC2=C(C1)CN(C(C1(C3CCCO3)CCC1)=O)C2 14592,C(CNC(C1CC2(CSC2)C1)=O)(CC(F)(F)F)NC(C=NOC)=O 14593,CC(C)(C)C(CO)C(=O)N1CCCC1CCNC(=O)CC1C=CCC1 14594,C12(C(N(CCCN(C)C)CCNC(=O)C=CC3CC3)=O)CCC(F)(CC1)C2 14595,n1(CC(=O)NC2C3CC(NC(c4cccnc4O)=O)CC23)ncccc1=O 14596,C(C)(C(=O)NCc1cn(C(C)C(=O)Nc2ccc(Cl)cc2)nn1)(C(C)C)OC 14597,C1(C2(C(=O)NC)CC2)CCCCN1C(C1C(NC(=O)CC(F)F)COC1)=O 14598,N1(C(c2ccc(C#C)cn2)=O)C2CCC1CN(C(c1ncc(C)cc1OC)=O)C2 14599,C12(COC)CC(CNC(C3C=CCC3)=O)(CN1C(c1ccccc1O)=O)C2 14600,C1(NC(Cc2cc(C(C)C)no2)=O)CN(C(C2CC2CN(C)C)=O)C2(CCCC2)C1 14601,C1(CCC)CCCCC1CNC(=O)C(C)OCOC 14602,c1(C(=O)NCCNC(CN(C2CCCCC2)C(C)=O)=O)cn2c(n1)CCCC2C.N 14603,CN1CCCC(C)(C(NOCC(=O)NCCN2CC3CC3C2)=O)C1 14604,N1(C(C2(CC#C)CCCC2)=O)CC(CNC(=O)Cc2cnnn2C)C(C)C1 14605,N1(CC(=O)NCCOCCNC(C2C(C)CCO2)=O)CCC(O)CC1 14606,c1(C(N2CCN(C(c3c(C)nc(CO)s3)=O)CC2C)=O)cc2cc(Cl)ccc2[nH]1 14607,C12(C(=O)NC(CNC(c3c(OC)n[nH]c3)=O)C)CC(CC3CC3)(CO1)C2 14608,C#Cc1cc(C(N2CCCCC2CCN(C(=O)C(O)CC2CC2)C)=O)ccc1Cl 14609,C1(CNC(C(CSC)OC)=O)CN(C(c2cn3ccsc3n2)=O)CCC1C 14610,C1(C(N2CCCC2c2cccc(F)c2)=O)CCCN(Cc2cccnc2)C1 14611,c1(CS(N2CCC(CN3CCC(N(C)C)C3)CC2)(=O)=O)ccc([N+](=O)[O-])cn1 14612,c1(C(=O)NC2C(C(=O)NCc3cc(C)no3)COC2)c(F)cncc1F 14613,c1(C(=O)NCC(CC)(C)NC(C2CCOCC2)=O)cc(C(F)(F)F)cnc1O 14614,C#Cc1cccc(C(=O)NC2CC3CCC2N3C(c2ccc(F)cc2OC)=O)c1 14615,c1(CC)ccc(C(N2CC(NC(c3nscc3C)=O)C(CC3CC3)C2)=O)c(Cl)c1 14616,CCC(C)(CC)C(=O)N1CC(NC(c2cnc(OCC(F)F)cn2)=O)C(O)C1 14617,S(=O)(=O)(c1cccc(=NCc2c[nH]nc2-c2ccco2)[nH]1)NC1C(CC)CCC1 14618,c1(OC)ccncc1C(=O)NCC1(C(C)NC(c2cc(F)cs2)=O)CC1 14619,C1(OC)CC(C)CN(C(=O)CC(C)CNC(C2CCOC2(C)C)=O)C1 14620,c1(OC)cc2c(cc1S(=O)(=O)NC1(C(F)(F)F)CCC1)C(=O)NCCC2 14621,CC1N(C(=O)C(C)(C)CCNC(c2csnn2)=O)CCOC1(C)C 14622,C#Cc1cnn(C)c1C(N1CC=CC(NC(=O)CCC2CC2CC2CC2)C1)=O 14623,C1(C(=O)NCC2(CNC(C(CCC)OC)=O)CCCC2)CCc2nnn(C)c2C1 14624,N1(C(C(C)(C)CO)=O)CC2CC(NC(=O)CCc3cccc([N+](=O)[O-])c3)CC1C2 14625,c12cc(ccc1Cl)C(=O)N2.C(C(=O)N1CCC(C)(O)C1)(C(C)C)OC 14626,c1(C(N(C2CCCN(C(=O)CN(C)C(=O)OC)C2)CC)=O)ccc(OC)c(N)c1 14627,C1(C(=O)NCCCCN(C)C(c2coc(-c3ccccn3)n2)=O)C2COCC12 14628,N1(C(C=CC(CC)C)=O)CCC(N(C(=O)CCOCC(F)(F)C(F)F)C)C(C)C1 14629,C1(C(=O)NCC2C(C(=O)Nc3cn(CC(C)C)nc3)CCC2)CC1C1CC1C 14630,c1(C(=O)NCC(C2CC2)NC(=O)C=CBr)cc(Cl)ccc1F 14631,CC(C(=O)N1CCN(C(=O)CCC2(C)CC2)CC1Cc1ccoc1)C(F)(F)F 14632,C1(CNC(C(C)n2cnnn2)=O)CCCCC1NC(=O)C(c1cccc(F)c1)O 14633,c1(CC)cccc(C(=O)N(CCNC(c2ccc(C(C)C)o2)=O)CC)c1O 14634,c1(C(=O)NCC2N(C(c3c(CC)cc[nH]3)=O)CC2)cc(F)ncc1OC 14635,c1(C(=O)NCc2scc(CNC(C3(CC(C)=O)CC3)=O)n2)cc(C)ncc1C 14636,C12(CNC(C(CC)N(C)C)=O)CCC(CC1)N2C(c1nncn1CC)=O 14637,Cc1sc2ncnc(NCCC(=O)NCC3CCCCN3C(C3CC3C)=O)c2c1C 14638,N1(C(CCNC(C)=O)=O)CCC2CCC(NC(C3(C)CCCCC3)=O)C12 14639,c1(C(N(C(CC)CC(=O)NCCc2ncon2)C)=O)ccc([N+](=O)[O-])[nH]1 14640,S(=O)(=O)(c1cnc(N2CCC(n3nccn3)CC2)c(Cl)c1)NC(CCSC)C 14641,C(=O)(C(CC(C)(C)C)NC(c1cscc1C)=O)NCC(CC(=O)OC)O 14642,N1(C(C2CC(C)(CNC(CCOCC#C)=O)C2)=O)CCN(C)C(C)C1C 14643,CCC(C)CCC(O)CC(=O)NCCC(C)N(C(=O)C(C)(C#N)CC)C 14644,C(C1CCCN1C(=O)CC1CCC1)=CC(=O)NCCCc1cccs1 14645,N1(Cc2ccc(F)c(I)c2)CC=C(CC(=O)N2CCCC3CCOCC23)CC1 14646,N1(C(c2ccc(F)c(C)c2N)=O)CCCN(C(c2ccc(CO)cc2)=O)CC1C 14647,c1(C(N(CCC(C)NC(C2CC(N(C)C)C2)=O)C)=O)cc(CO)[nH]n1 14648,CC1(CNC(=O)CP(C)(C)=O)COCCN(C(c2cc(C#N)ccn2)=O)C1 14649,c1(C(N2C3CC(NC(=O)CC4CCCCO4)(C3)C2)=O)cnc2occc2c1 14650,C#CCC(C)(C(=O)N1CC(C)(CO)C1)NC(C1(C#N)CC(F)(F)C1)=O 14651,c1(CC(=O)NCCCCCNC(C2CC2CF)=O)cc(O)cc(Br)c1 14652,Cc1nn(C)c(C)c1CC(N1CCC(O)(CCNC(c2c(Cl)nsc2Cl)=O)C1)=O 14653,C(C1CCCN1C)=CC(N1CC(c2ccccc2)(NC(c2cnc(SC)s2)=O)C1)=O 14654,C(C(C(F)(F)F)OC)NC(c1scc(CNC(C(C)OCCCC)=O)c1)=O 14655,C1(C(=O)NC(C)CNC(C2CC2c2cncn2C)=O)C2C3CCC(C3)C12 14656,C(=O)(C1=CCC(C)CC1)NC1CCCN(C(Cc2cccc(C)c2F)=O)C1CC 14657,C(=O)(C(C)C(C)COC)NC1CC(CNC(C(c2ccccc2)OC)=O)C1 14658,c1(OC)cc(C(=O)NCCC(C(C)C)NC(C2CCCC2)=O)c2c(c1)CCCC2 14659,c1(CCC(=O)NCCN(C(=O)CSCc2ncccn2)CC)ccc(Cl)cc1 14660,C(C)(C)(CC(=O)NCCC1CN(c2cc(OC)ncn2)C1)OCC.c1(CN)ccccc1 14661,Cc1c(C(=O)NC2CC2CNC(=O)Cc2ccc(O)cc2)c(C(F)F)nn1C 14662,C1(C)(C(=O)NC(C)CC2CN(C(=O)Cn3cnc(=N)[nH]3)C2)CCC(C)(C)CC1 14663,N1(C(c2cccc(F)c2)=O)CCC2(CCN(C(=O)OCc3ccccc3)CC2)C1 14664,C#CC1(C(=O)NC(CCO)C(C)(C)O)CCN(C(c2cc(C)ncc2Cl)=O)C1 14665,CC1=C(C(=O)NCC(C2CCCC2)NC(C2CCC(C)NC2=O)=O)CCO1 14666,C1(NC(C2(C)CC(=C)C2)=O)CC(NC(=O)CC2CCOC(CC)C2)C(O)C1 14667,C(c1ccc(C(C)(C)C)cc1)=CC(=O)NCC1CCC(NC(C(C)(C)OC)=O)C1 14668,c1(CC(=O)NC2CN(C(CC)=O)CC2NC(C)(C)CCS)ccn2cncc2c1 14669,CC1=C(CC(=O)NC(=O)NNc2ccccn2)c2ccccc2C1 14670,C(=O)(CCCC(C)(C)C)N1C(C)CC1C(=O)NCC1CCNC(=O)C1 14671,CC1(C)CC(NC(c2cccc(C(N)=O)n2)=O)CN1C(c1ccc(Cl)cn1)=O 14672,C(=O)(CC(C)(C)C(=O)NCC1C2CN(C(=O)C(CSC)OC)CC12)OC 14673,N1(C(COC(CC)C)=O)CCOC(C)(CNC(=O)CN2CC(C)(C)C2)C1 14674,C1(NC(Cc2c(C)noc2C)=O)CC2(C1)CN(C(c1occc1F)=O)C2 14675,CC(C)(C)CC(O)C(=O)NC1CCCCC1C(=O)NCCCCCN1CCCC1 14676,c1(OC)nccc(C(=O)N(C)CCNC(C2CC(F)CN2C)=O)c1Br 14677,C(=O)(CCCC(CC)NC(C1CCCO1)=O)NC(CC=C)CC(F)F 14678,N1(C(C(CC)OCC)=O)CC(NC(C2(N3CCCC3)CC2)=O)CC1(CC)CC 14679,Cc1cc(C(=O)NC2(C)CCCN(C(=O)CCCc3ccncc3)C2)nc(O)c1 14680,C(=O)(C(F)(F)C(C)(C)O)N(C1CCN(C(=O)CSC(F)(F)F)CC1)C 14681,N1(C(C(CC(C)(C)C)(C)C)=O)CCc2sccc2C1CNC(C1CC=CCC1)=O 14682,c1(C(=O)NC2(C)CCN(C(Cc3ncc(C)s3)=O)C2)ccc2c(c1)C(C)CO2 14683,C(CCN=c1[nH]ccc(=NC2CC3(C2)CC3(F)F)[nH]1)c1cnn(C)n1 14684,C(c1ccccc1)=CC(=O)NC12CC(C(N3CCC(CNC(N)=O)C3)=O)(C1)C2 14685,N1(C(C(C(C)C)NC(C)=O)=O)CCC(C)C(NC(c2snc(Cl)c2Cl)=O)C1 14686,CCC(CCCO)(N=c1cc(F)nc(C(=O)O)[nH]1)Oc1ccccc1 14687,CC(O)(CC(=O)N1CCCCC1CCNC(c1cc(Br)c[nH]1)=O)C(F)(F)F 14688,C1(NC(c2c(C)ccc(C)c2)=O)CCSC12CN(c1nc(N(C)C)ncc1Cl)C2 14689,c1(C(N2CCC(N(c3ncc(Br)cn3)C)C2)=O)cc(F)ccc1Br 14690,S(=O)(=O)(c1ccc(C)c(C)c1)NCCNC(=O)NCc1c(SC)cnn1C 14691,c1(OC(N2CCOC(C(F)F)C2)=O)ccc(-c2cnco2)cc1 14692,N1(C(CCNC(C(C)C)(C)C)=O)CC2CN(C(=O)COCCF)CC(F)(F)C2C1 14693,c1(C(N(C2CCN(C(=O)CC3CC34CC4)CC2)CCC)=O)cn2ccnc2cn1 14694,Cc1cc(NCC(C)(C)C(C)C)ncc1S(=O)(=O)N1CCOCCC1C1CC1 14695,c1(OCC)cncc(CCC(=O)NCC(CO)NC(c2ncoc2C(C)C)=O)c1 14696,N1(C(c2c(N)nccc2)=O)CCC2(NC(=O)C3=CCCCC3)CC2C1 14697,C1(CNCC(CO)OC(C2CCCCO2)CC)(CC)CCNC1=O 14698,C#CC1CC2CCC1N(C(c1ccc(SCC3CC3)cc1)C(=O)NCCC)C2 14699,CC(C)(C)C(C(=O)N1CCC(NC(=O)C=CCNC=O)CC1)c1ccccc1 14700,C(=O)(C(O)CCCN(C(=O)CCc1ccc(OC(C)(C)C)nc1)c1cscn1)OC 14701,C(CC(=O)NCCC1CCCO1)(C(F)F)NC(C1(Cl)C(C(C)=O)C1)=O 14702,C1(CCC(=O)NC23C(CN(C(C(C=C)(F)F)=O)C2)C3)CCc2ccccc2C1 14703,C1(S(N)(=O)=O)(C(=O)NC(C)C(CO)NC(=O)CCOCCCCO)CCCC1 14704,N1(C(C2C(C)OCCC2)=O)CCOC2(CCN(C(=O)Cc3cnccc3Cl)C2)C1 14705,N1(C(c2c(C)nc(CNC(=O)CC3(C)CCC3)o2)=O)CCN(C)CC1CCO 14706,N1(C(C2C=CC(NC(C(CN(C)C)O)=O)C2)=O)CCC(O)CC1C1CC1 14707,C#CCC(C)(C(=O)Nc1cc(CO)ccc1C)NC(c1ccc(OC)nc1)=O 14708,c1(C(=O)NC(CC=C)CNC(=O)CNC(c2cccs2)=O)cc([N+](=O)[O-])oc1C 14709,c1(OC)ccc2c(C)c(C(N3CCC(C)C(N(C)C(C)=O)C3)=O)[nH]c2c1 14710,O=C(C1CCCc2scnc21)NC1CC2(C1)CN(C(C13CCCCN1CCC3)=O)C2 14711,CC(C)(C)C(CNC(c1ccc2nccn2c1)=O)C(=O)NC1(C(N)=O)CC1 14712,CC(CCCCNC(C1(CO)CCCO1)=O)NC(c1ncc(C(F)F)s1)=O 14713,Cc1nccc(C(=O)NCC(O)CNC(c2ccc(CN(C)C)o2)=O)n1 14714,C=CCCCC(=O)NC1(CNC(=O)CCN2CCCC(C(N)=O)C2)CCOC1 14715,Cc1ccc(C)c(C(=O)NCCCCCNC(c2nccc(Cl)c2F)=O)c1 14716,N1(c2nnc(CCOC)n2CCOc2ccccc2)CCCC(C2CC2)C1 14717,Cc1ccc(CN2CCC(O)(C(=O)NCCC(C)CO)CC2)c(F)c1F 14718,Cc1ccc(NC(=O)CN(C)C)cc1C.C1(O)(C(F)(F)F)CNC(=O)NNC1=O 14719,C=CCC(C)(CC)C(=O)NCCC1(O)CCCN(C(c2ccc(OC)nc2)=O)C1 14720,c1(NC(C#C)C)nc(N2CCc3nocc3C2)nc2c1ncn2C(C)C 14721,c1(C(=O)NC2CN(C(C(C)CC3CCCOC3)=O)C2)cccc([N+](=O)[O-])c1 14722,CC(C(=O)NCC1CC(NC(c2cc(CCCO)on2)=O)C1)C(C)(C)C 14723,C1(C(=O)NCC(C(C)C)NC(=O)Cc2csc(NC=O)n2)COC(=O)N1C 14724,CSC1=C(C(=O)NC2(C)CCN(C(C3CC3(C)C)=O)C2)CCCC1 14725,c1(CC(=O)NC2CCCCC2NC(C2(n3nccn3)CC2)=O)c(O)ncnc1O 14726,c1(CC(N2CCC(N(C)C(C3CC3C(F)(F)F)=O)C2)=O)cccc2nsnc12 14727,N1(C(C(CC2CCCC2)OC)=O)CCN(C(c2cnc(C)o2)=O)C(C(C)C)C1 14728,N1(C(COC)=O)CCOC2CCN(C(c3cccc(C4(F)CC4(F)F)c3)=O)CC12 14729,C(=O)(CCC(=O)NCC1(NC(C2SCCC2C)=O)CCCCC1)NC 14730,c1(N(C)C)ccc(C(=O)NCC2CCCN2C(C2CC(C)(F)C2)=O)cc1 14731,CCCCN=C(NCCNS(C)(=O)=O)NCC1(S(C)(=O)=O)CCC1 14732,c1(C(=O)NC(C)CCCCNC(C2CCN(C3COC3)C2)=O)cc2n(c1)CCC2 14733,C(N=c1[nH]c2ccccc2s1)C1C(C)CN(C(=O)Cc2ccc3c(c2)COC3)C1 14734,n1(CC(=O)NC2CC(CC)(CC)N(C(=O)CCS(C)(=O)=O)C2)nc(O)ccc1=O 14735,c1(C(N2C(C(C)NC(=O)C(N3C(=O)CCC3=O)C)CC2)=O)cn(C)c(C)cc1=O 14736,N1(C(c2c(CC)c(C)sc2)=O)CCN(C(=O)C(C)(C)CC)CC1CS(C)(=O)=O 14737,C1(C(=O)NCC2CCN(C(=O)C(c3cccc(C)c3)C)C2)(CC)CCCCC1 14738,N1(C(CSCCOC)=O)CCCC(C)(C(N2CCC(n3ccnc3)C2)=O)C1 14739,C1(C(=O)NCCCCCNC(C(c2ccccc2)OC)=O)C2CCC1(C(N)=O)C2 14740,c1(C(=O)NCCC(C)N(C(CCCC(=O)OC)=O)C)cccc2c1CCO2 14741,CC1=C(C(=O)NCC(CNC(=O)C(C)(C)C2CCOCC2)OC)C(=O)OC1(C)C 14742,C1(CC=C)CCCCN1N(C)CC1CCCc2cc(C)ccc21 14743,C1(C(N(CCOCc2cc(NC(COC)=O)ncc2)C)=O)C2C3CCC(C3)C12 14744,N1(C(C(c2cccnc2)OC)=O)CC(NC(=O)CC(C)CF)C2(CCOCC2)C1 14745,C1(F)(CNC(CC2CCCC(C(C)C)C2)=O)CCCN(C(C2CCCO2)=O)CC1 14746,C(c1cc[nH]c1)=CC(=O)N(CCC(=O)NCC1(C(C)(F)F)CC1)C 14747,CON(CCC(=O)NCc1ncc(CO)o1)C(=O)C(C)(C)c1ccno1 14748,CCCCCC(=O)NC1CC1CNC(=O)CN(c1ccc(Br)cn1)C 14749,O=C1CC(=O)NC(C(=O)NCc2cc(C(=O)NCC3CC3(Cl)Cl)n[nH]2)C1 14750,C1(NC(CC2CC(=C)C2)=O)CCN(C(=O)CCc2cccnc2F)CC1C(N)=O 14751,Cc1ccc(F)cc1C(=O)NC1C2CC3C(C2)C13C(=O)NC1C(O)CC1O 14752,C1(CC(=O)NC2CCN(C(CCCc3onc(C)n3)=O)C2)C(C)(C)C1(F)F 14753,N1(C(c2cc(C)n(C(C)C)c2)=O)CCC2CN(C(C3CC4(C3)CC4F)=O)CC12 14754,N1(C(C2OCCN(CC)C2)=O)CCC2(CCN(c3cc(C)ncc3C#N)C2)C1 14755,C1(NC(CN(C(COCCCC)=O)CC2CC2)=O)CCCC(C)(C)C1 14756,C(CCN=c1[nH]c(=NCC2CCCS2)[nH]c2cccc(F)c12)(C(C)C)OCC 14757,c1(C(=O)NC2CN(C(Cn3c(C)csc3=O)=O)CC2C)cnc2ccc(F)cn12 14758,N1(C(c2ccc(OCCO)cc2)C(=O)NC(CC)(C)C)CCOC2(CCCCC2)C1 14759,N1(C(c2c(C)ocn2)=O)CCC(NC(c2cc(C)c(C)nc2C)=O)C12CCCC2 14760,C1(C(N(CC(CC)OCC)C)=O)(CC)C=CCN1C(=O)CNC(=O)CN(C)C 14761,C1(OC)CN(C(=O)COc2cccnc2)CC1NC(C1CC12CC(O)C2)=O 14762,C1(C(=O)NC2(CC)CC(C)(C)C2)CN(C(=O)C=Cc2cc[nH]n2)CC1C1CC1 14763,c1(C(c2cscn2)NC(C2CNCCC2(F)F)=O)cc(F)c(F)c(F)c1 14764,C1([Si](C)(C)C)(NC(C(CN(C(C)=O)C)C)=O)CC1 14765,C12(NC(=O)C(O)C3CCC3)CCN(C(C3CC(F)(CO)C3)=O)CC1C2 14766,c1(OC)nccc(C(=O)NC2COCC2CNC(c2ccn(C3CC3)n2)=O)n1 14767,C1(N(C)C)CCCC(C(=O)NCC2CC2NC(=O)C(F)CC2CCC2)C1 14768,CC1CCN(S(=O)(=O)CC(=O)NCC(C2CC2)NC(C2NC(=O)NC2=O)=O)CC1 14769,C(C)(CNC(c1nc[nH]c1C(C)(C)C)=O)(CNC(=O)C(C)=C(C)C)OC 14770,c1(NC(CC(C)OCCC)=O)cccc(CNC(=O)C(F)CC2CCCCC2)c1 14771,Cc1cccc(C(CNC(=O)C#CC(=O)N(C)C)NC(=O)C=CC(F)(F)F)c1 14772,C(=O)(C(C)CNC(C1CCC1C(C)(C)C)=O)N1CC(CSC)C1 14773,c1(C(=O)OCC2(CC(=O)OC)CC2(F)F)nc(C)c([N+](=O)[O-])cc1Br 14774,N1(C(C2CC(C)(F)C2)=O)CC2CCC(C(=O)NCCCCCO)(C2)C1 14775,C1(CNC(CC=C)=O)CC2(CCOCC2)CN1C(c1cc2cc(Br)sc2[nH]1)=O 14776,C(CC(=O)N(C1CN(C)C1)C)(C(F)(F)F)NC(C(CC(C)C)O)=O 14777,C1(CCOC)(NC(c2ccsc2Cl)=O)CCN(C(C2OCCC2C)=O)C1 14778,N1(C(C(CC)NC(C)=O)=O)CCC2(CC1)CN(Cc1ccc(Cl)cc1F)CCO2 14779,C1(CNC(CCOCCC)=O)CN(C(c2c(N)cc(C)cc2F)=O)CC(C)(C)O1 14780,N1(C(CCCN(CCC)CCC)=O)CC(CNC(=O)CCC(C)(C)F)CCC1C 14781,C1(C(=O)NCc2cscn2)C2CN(Cc3nc(-c4ccccc4)cs3)CC12 14782,C(=O)(C1=NOC(CC2(O)COC2)C1)N(CC(C)O)CCNC(=O)CC(F)(F)F 14783,c1(C(=O)NC2(C)CCN(C(CC(C)(C)C#N)=O)CC2)cc(Cl)ccc1[N+](=O)[O-] 14784,C(=O)(C(CCC(N)=O)N(C)C)NCC1OCCN(C(C(CCCOC)C)=O)C1 14785,c1(CC)nn(C)c(CC)c1C(=O)NC1CCCCC1NC(C1CC(O)C1)=O 14786,C1(NC(CCCC=C)=O)CN(C(=O)CC23CCCN2CCC3)CCC1F 14787,c1(OC)ccc(C(N2CC(CNC(C3CCSC3)=O)C2)=O)c(OC)c1 14788,c1(C(N2CCC(CC#C)(C(=O)NC(C)CF)C2)=O)cccc2c1CCC2 14789,Cc1cc(C(N2CC(=C(F)CNC(=O)C(F)CCCO)C2)=O)sn1 14790,Cc1c(C(N2CC(NC(C3CCCO3)=O)CC2C)=O)sc2ccccc12 14791,c1(OC)ccc(Br)c(C(N2C3CCC2C(C(=O)NC24CC(F)(C2)C4)C3)=O)c1 14792,c1(NC)cnncc1C(=O)NCC(c1ccc(Cl)cc1)NC(c1cncs1)=O 14793,C1(CC(=O)NC23CC2CN(C(=O)CCCN2CCCC2)C3)(OC)CCCCC1 14794,C(c1cccc(F)c1)=CC(=O)NC1C(CNC(C2(C(C)C)CCCO2)=O)CCC1 14795,c1(C(=O)NC(C(C)C)CNC(=O)C=CCF)cc2cc(Cl)cnc2[nH]1 14796,CC1CCC(C)(C)CC1(c1nnnn1C1CC1)NCCC=CCC1CC1 14797,N1(C(CNC(CCCCC)=O)=O)CC(NC(=O)Cc2ccc(C)s2)C2CC2C1 14798,Cc1ncn(C)c1NC(C1CCN1C(C1CC(F)(F)C1)=O)=O 14799,N1(C(CCCC#C)=O)CC(NC(c2cnc(N(C)C)c(Cl)c2)=O)CC2(CCC2)C1 14800,CC1(C)CC=C(c2ccncc2C(=O)NNC(=O)C(F)F)CC1 14801,CCC(CC)C(C)C(=O)NCC(=O)N(C1CCCCC1C)C 14802,c1(CC2CNCCC(=O)N2)ccccc1C.N1(CC)CCC(C)C1C 14803,c1(C(=O)NC(C)CCN(C(=O)CCC2CCCCO2)C)ccnc2ccsc12 14804,C=C(C)C1OCCC1C(=O)NCCCN(C(=O)COCCCF)C(C)C 14805,c1(C(=O)N)cnn(C(C)C)c1C.C1(C(=O)NC(COC)COC)CCCN1C(C)C 14806,CC(C)(CCC(=O)N1CC(NC(C2CCC(CN(C)C)O2)=O)C2(CC2)C1)[N+](=O)[O-] 14807,Cc1ccnc(O)c1C(=O)N(C)CC1CCN(C(=O)CC2(O)CCC2)CC1 14808,c1(C(=O)NCC2CC(NC(CCC(C)(F)F)=O)C(O)C2)ccc2c(c1)CCCS2 14809,C(=O)(CC1OCCc2sccc21)NC1CCC(CC(=O)Nc2ccccc2)C1 14810,CC1OCCC1CNC(=O)CCC1CCC(NC(=O)C=Cc2ccsc2)C1 14811,C1(OC)CCCC(CNC(C2C3CC3CN2C(=O)CC2(C)CCOC2)=O)C1 14812,c1(C2(O)CN(C(c3cc(C(F)F)no3)C(=O)NC3(C)CC3)C2)cccc(Cl)c1 14813,c1(CC(N2CCC(C(C)NC(C3(CC4CCC4)CC3)=O)C2)=O)ccncc1Cl 14814,Cc1cnc(NCCCCC2CC2C)c(S(=O)(=O)NCCCCS(C)=O)c1 14815,c1(OC)ccncc1C(N1CC(O)(C(F)C(=O)NCc2nccnc2C)C1)=O 14816,c1(OC)ccc(C(N2CCN(C(=O)C=CC(C)(C)C)C(CCOC)C2)=O)nc1Cl 14817,C1(C(N(CCC(N2CCC(C(C)(C)O)C2)=O)C)=O)CC2(CC2)CN1C 14818,c1(OC(C2CC3CCC2C3)=O)cncc2cc(Cl)ccc12 14819,CC1(CNC(C2(CF)CC(F)(F)C2)=O)CCCN(C(=O)CN2CCCNC2=O)C1 14820,c1(C(=O)NCC2(C)CCCCO2)ccc(I)c(F)c1 14821,O1C2CCCc3ccc(cc32)C1=O.c1(-c2nc(COC)on2)cccc(OC)c1 14822,C1(C(N2CC(O)(CCNC(C3CC(SC)C3)=O)C2)=O)CCOC(=O)CC1 14823,CC#CCC(C(=O)Nn1cnn(C)c1=S)NC(c1cscc1C)=O 14824,CCC(C)C(O)C(=O)NCCCCCN(C(=O)C(C)SC(C)C)C 14825,CCC(C)C(=O)C(=O)NC1CC1CNC(=O)CN1CC(C)(OC)C1 14826,C1(NC(C2(CC=C)CC=CC2)=O)CC2CC1CN(C(=O)C(C)(C)CF)C2 14827,c1(C(N2CCCC(NC(C3C(=C)CC3)=O)C2)=O)ncnc2c1c(Br)cn2C1CC1 14828,C1(NC(c2c(Cl)cc(C)s2)=O)CCOC12CCN(C(=O)C=Cc1ccsc1)CC2 14829,C1(SC)CCCCN(C(=O)CC(C(C)C)NC(c2cnc(Cl)s2)=O)C1 14830,C(=O)(CCCCCC#N)N1CCC(NC(C(C)(O)c2ccccc2)=O)C(O)C1 14831,C1(C(=O)NC2C3CN(C(c4c(C)n(C)nn4)=O)C2C3)CC12CCS(=O)(=O)CC2 14832,Cc1cccc(CNC(c2c[nH]nc2CCNC(=O)Cn2cc(C)cn2)=O)n1 14833,c1(C(=O)NCCC(=O)NC(C#C)CC)c[nH]nc1[N+](=O)[O-] 14834,Cc1ccc(C(N2CCC(C)C2C(N2CC(C(=O)OC)C2)=O)=O)cc1C#N 14835,c1(C(c2n(CCC)nnn2)NCC(C)Cn2ccnc2C)cc(Br)ncc1F 14836,c1(CC)nc(N2CCCC(NC(c3cc(C)ccc3C)=O)C2)cc(C)n1 14837,C(N=c1[nH]c(N(C)Cc2nccs2)nc2c1SCC2)c1ccc(C)c(C)n1 14838,C1(NC(CCC(C)O)=O)CC2CCCC(C1)N2C(=O)Cn1cnc(=N)[nH]1 14839,c1(NC(CC2(C)CN(C(CCCCN(C(C)=O)C)=O)C2)=O)ccc2nncn2c1 14840,C1(n2cc(-c3nccc(OC)n3)nn2)CCC(C)(C)N(C(C2CCC(=O)C2)=O)C1 14841,c1(C2(C(=O)NC(C)CNC(=O)CCC3CCCO3)CC2)cccnc1Cl 14842,C(=O)(CCCC#Cc1ccccc1)NC1C(C)N(C(=O)C2=COCCC2)CCC1 14843,C(=O)(CCC(=O)N1CCCC1)N1CCC(NC(c2cccs2)=O)C1 14844,CC(CC(N)=O)C(=O)NCC1=CCN(C(=O)C(C(C)(C)C)C2CCC2)CC1 14845,C#CC1(NC(=O)C(C)(C)CCNC(c2n[nH]c(=N)[nH]2)=O)CCC(C)CC1 14846,c1(CC)cc(C(=O)NC(C)(C)CN(C(=O)C(C)(Cl)Cl)C)on1 14847,C(=O)(C(C(C)C)CNC(C1CC1)=O)NCCCNC(c1scc(C(=O)OC)n1)=O 14848,C1(C(=O)NCc2n(C(C)C)ncn2)CCN(C(c2ccc(=N)[nH]c2)=O)C1C 14849,Cc1ccc(C(=O)N(C)CCOCCC(=O)NCCN2CCCC(C)C2)cn1 14850,C(=O)(C(COCC1CC1)CC(C)C)N1CC2CN(C(CCN(CCC)C)=O)C2C1 14851,C1(NC(c2ncc(C)c(Cl)c2)=O)CN(C(c2cc[n+]([O-])cc2)=O)CC1N=[N+]=[N-] 14852,Cc1ccc(C(=O)N(CC(O)CNC(=O)CC(C)c2ccco2)C)c(SC2CC2)c1 14853,N1(C(C(C)=C(C)C)=O)CC=C(CNC(c2cc(C)cnc2C(F)(F)F)=O)CC1 14854,C1(NC(CNC(CNC(C2C(C)OCCO2)=O)=O)=O)CC2(C1)CC(O)C2 14855,N1(C(CC2CC(N(C)C)C2)=O)CCC(C(=O)NC2CCOC(C)(C)C2)CC1(C)C 14856,O=C(C1CCCc2cncn21)NCC1CN(C(C2(F)CCC(=O)CC2)=O)C1 14857,S(=O)(=O)(c1ccc(F)c(C(=O)N(C)C)c1)NC(C)C(CO)NC(=O)C=C1CCC1 14858,C(=O)(CC1OCc2ncccc21)NCC1C(C)(C)CCCN1C(=O)C1=CCCC1 14859,C1(C)(CNC(C(Cc2cc[nH]n2)NC(CCc2ncn(C)c2)=O)=O)C=CCCC1 14860,N1(C(CNC(c2c[nH]c(=N)o2)=O)=O)CC=C(CNC(c2ccnc(Cl)c2)=O)CC1 14861,C1(OCC)CC(c2ccccc2)(NC(=O)C(n2cc(CCCC(C)=O)nn2)C)C1 14862,CC1CC2CN1C2.c1(CC(=O)NC)cccc(Br)c1.S(C(F)(F)F)CC(=O)NCCO 14863,N1(C(c2cc(C)c(N)cc2Cl)=O)C2CCC1C(C)C(NC(=O)C(C)C1CCC1)C2 14864,c1(C(N(CC(CC)NC(=O)Cn2cc(CO)nn2)C)=O)cccc2nn(C)nc12 14865,c1(CC(=O)N(C)CC2OCCN(C(C(C=C)(C)O)=O)C2)cc(F)c(C)cc1F 14866,Cc1c(NC(c2cc(I)cs2)c2nnnn2C2(C)CC2)cccc1Cl 14867,C1(C(=O)NCC2N(C(C(C(CC)C)O)=O)CC(C)(C)C2)CCOC2(CCC2)C1 14868,C1(NC(c2cccc(O)c2Cl)=O)CN(C(c2ccoc2)=O)CCC1C(F)(F)F 14869,CC#CCC(C(=O)Nc1cnc(C(C)C)nc1)NC(=O)C=CC(C)C 14870,C(=O)(C1=C(Cl)CCOC1)Nc1cc(C)c(NC(=O)CC2CC(CN(C)C)C2)cc1 14871,N1(CC)CCOc2cc(CNc3nccc(=NCCCSC)[nH]3)ccc2C1 14872,c1(C(=O)NC2CC(CCNC(C(CCC)(C)C)=O)C2)ccc2nccc(C)c2c1 14873,c1(C(=O)NCC(C)N(C(C23COCC2C3)=O)CC)cc(F)cnc1O 14874,C(C(C)(C)CC(=O)N1CC(CNC(C2CC(O)(NC(C)=O)C2)=O)C1)NC(=O)OCC 14875,C1(C2(O)CN(C(C3CCC(F)C3)=O)C2)(CNC(c2ccc(N)c(F)c2)=O)CC1 14876,CCC(C)CC(C(=O)OC)NC(c1ccnc(O)c1F)=O 14877,c1(OC)ccc2[nH]nc(C(N3CCN(C(C4CC5(CC5)C4)=O)C(CO)C3)=O)c2n1 14878,Cc1ccc(=N)[nH]c1C(N1CCCC(NC(c2nc(Br)c[nH]2)=O)CC1)=O 14879,CC(CS(C)(=O)=O)C(=O)N1CC2(CC(NC(=O)Cn3ccc([N+](=O)[O-])n3)CO2)C1 14880,N1(C(c2n(CCC)ncc2)=O)CCC(CNC(=O)C(C)C#N)CC1 14881,N1(C(C(C)Br)=O)CCCn2nc(C(N3CCC(O)C(F)C3)=O)cc2C1 14882,CC(CC(=O)NC1C=CCN(C(c2sccc2CN(C)C)=O)C1)CC(C)(C)C 14883,C1(N(C(CN(C)C2CC2)=O)C(c2ccc(C(N)=O)s2)=O)CCC(NCCO)CC1 14884,C1(C(=O)N(C(C)C(N2CC(C)(C(F)(F)F)C2)=O)C2CC2)(OC)CCOC1 14885,CC1CC(CCNC(c2cncnc2)=O)CCN1C(=O)CSCC(F)F 14886,c1(CCC)cc(C(=O)N(C2CCCN(C(C3(F)CCCC3)=O)C2)CC)c(C)o1 14887,c1(OC)cc(C(=O)NCC2(F)CC(NC(=O)C3=C(C)OCC3)C2)c(Cl)cn1 14888,c1(C(=O)OC)cc(C#N)cnc1NCC1CC(C)N(C(=O)CCc2cncn2C)C1 14889,N1(C(C(CC)C)=O)CCCC2C1CCN2C(=O)Cc1scnc1C 14890,CC(C)(F)CCC(=O)N1CCC(CCCCCNC(=O)Cc2csc(=N)[nH]2)CC1 14891,Cc1ccc(C(N2CC(NC(c3csc(C4CCCN4C)n3)=O)C2)=O)nc1 14892,S(=O)(=O)(c1cccc(OC(C)C)c1)NC(c1cc(CC)oc1C)=O 14893,NC(=O)CS(=O)(=O)CC(=O)N1CCC1c1ccc(F)c(F)c1 14894,C(=O)(C#CC(C)(C)CNC(=O)C(O)C(F)(F)F)NCC1CCN(CC)C1 14895,C1(SC)CN(C(=O)C(=O)NCCc2ccc(P(C)(C)=O)o2)CC12CCC2 14896,N1(C(CCn2nc(C)c(Br)c2)=O)CCCC2C(NC(C3CC3F)=O)C(C)(C)C12 14897,c1(CC(C)(C)C)ccc(C(=O)NCC2CN(C(c3ncccn3)=O)C3CC23)cc1 14898,N1(C(C(C)C2CC2)=O)CCCCC(CNC(C2(C(N)=O)CCC2)=O)C1 14899,C(C(CNC(C1(C(F)F)CC(=O)C1)=O)C(F)(F)F)NC(C(n1c(C)ncc1)C)=O 14900,N1(C(CCOCC#C)=O)CCCC1(C)CNC(c1ccc(Cl)cn1)=O 14901,c1(CC(=O)N(C(CN(C(C2CCN(CC)C2)=O)C)CC)C2CC2)ccc(O)c(F)c1 14902,C(=O)(C1=CC2CCCC12)N1CC(C(C)NC(=O)CC2CC2)C1 14903,C1(NC(c2cncc(N(C)C)c2)=O)CN(C(c2sccc2F)=O)C(C)(C)C1 14904,Cc1ccc([N+](=O)[O-])c(C(N2CC3CCC2CN3c2ncnc(Cl)c2F)=O)c1 14905,c1(C(=O)OC)nc(=NC2CC(NC(C3(C)CCC(=O)N3)=O)C2)cc[nH]1 14906,C(=O)(C1=CCC1)NCCOC1CN(C(C=CCN(C)C)=O)C1 14907,C1(Cn2cc(CCSCC)nn2)CC2(CCC2)CN1C(C1COCCO1)=O 14908,Cn1ncc2c1C(=O)O2.C(=O)(CCC(=O)c1cccnc1)NC(C)(C)C 14909,CN1CC2CCN(C(c3cccc4c3COC4)=O)C2C1 14910,c1(C(C)NC(CCc2c[nH]c(=N)[nH]2)=O)ccc(CNC(=O)CCC2CC2)cc1 14911,c1(C(=O)NC)cccc(C(=O)N(C)CCN(C(C2CCO2)=O)C(C)C)c1 14912,C1(N(C)C)CCC(c2nc(-c3cccnc3)nn2Cc2ccsc2)CC1 14913,c1(C(=O)NCC(CC)NC(C2CC(C3CCC3)C2)=O)c(F)ccc(OC)c1N 14914,c1(CCC(N2C(CCNC(CC(CC)C)=O)CCCC2)=O)ccc(C#N)cc1F 14915,C1(C(=O)NCC(=O)OCC=C)CC2(CCC2)CN1C(=O)CNC(=O)CC 14916,Cc1ccc2ncc(C(=O)NC3CC(NC(=O)Cc4scnc4C)C3)c(=O)n2c1 14917,c1(CC)n[nH]c(CC)c1CC(=O)N(CCCNC(=O)C(c1cccc(Cl)c1)C)C 14918,CCCCCC(O)C(=O)NCCC(C)(C)NC(C1(n2cncn2)CC1)=O 14919,C#Cc1ccc(C2CC2C(=O)N(CCCNC(C)=O)C2CC2)cc1 14920,C1(C)(OC)CCCN(C(=O)C(C)(C)CCNC(C2CC(C)(C)CCO2)=O)CC1 14921,C(=O)(CCc1ccco1)N(CC(=O)NCCSC)C 14922,c1(C(=O)NC(CNC(CC(C)(C)C(F)F)=O)CC(F)(F)F)nccc2c1NCCC2 14923,c1(C(=O)NC2C(NC(C(C)OCCCC)=O)CC2)cnc2c(ccn2C)c1 14924,C1(CNC(c2ccc(CC)c(CC)c2)=O)CC2(CCC2)CN1C(=O)CC(C)F 14925,CCCC(O)CC(=O)NCC1C2CCC(C2)N1C(c1cnn(CC(F)(F)F)n1)=O 14926,c1(CC(CN2CC(N(C)C)(C(N)=O)C2)O)ccccc1C(F)(F)F 14927,c1(C(N(CC(O)CNC(C2(C)CC=CC2)=O)C)=O)cccc2c1nc(O)n2C 14928,N1(Cc2ccc(OC)c(Br)c2)CC2CCC1CN2C(c1cocn1)=O 14929,O=C1C=C(c2cnn3c2CN(C(C2(c4cnccn4)CC2)=O)CC3)CCC1 14930,C1(NC(c2c(CC)ncnc2)=O)CCN(Cc2nc(-c3ccccc3)cs2)CC1C 14931,C=CCCCC(=O)N1CC(O)(C2CCCN2C(=O)C=CCCC=C(C)C)C1 14932,c1(OC)ccc(Cl)c(CN2CCNCC2C(=O)NCc2cc(C)on2)c1F 14933,Cc1nc(C)c(C(N2CC(O)(C(C)NC(c3scnc3C3CC3)=O)C2)=O)s1 14934,N1(C(C(C(C)C)=O)=O)CCC2(CCCN2C(C2CCC=CCC2)=O)C1 14935,c1(C(=O)NCC(CCOC)NC(=O)CC2(COC)CC2)cccc2c1CCCN2 14936,N1(CC)CCOCC1CC(=O)NCC1(F)CC(NC(c2cccc(CO)n2)=O)C1 14937,CN1CCN(C(=O)CCC2CCC(=O)NC2)CC1CNC(=O)C1=COCCC1 14938,C1(CCN(C)C)CCN(C(=O)C(=O)Nc2ccc(C(F)(F)C(F)(F)F)n2C)CC1 14939,CC1CCCN(C(c2ccc(F)c(F)c2)=O)C1CCO.C12C=CC(C1)C(=O)N2 14940,N1(C(CC2C(CNC(C=CC)=O)C2)=O)CC(C2=NOC(C)C2)C1 14941,N1(C(C2(C(C)C)CCN(C(c3cccc(NC)n3)=O)C2)=O)CCC2(CC1)N=N2 14942,C1(C(N(CCC(C)NC(=O)CNC=O)C)=O)OCCC1C(N)=O 14943,c1(O)cc(C)nc(N2CCOCC(CNC3(COC)CC3)C2)n1.c1(C)ccccc1.O 14944,c1(COC)cccc(CNC(C2CC(C)N2C(=O)CC2CC(F)(F)C2)=O)n1 14945,C1(C(=O)NC(C)CNC(=O)CCCN2CCOCC2)CCc2nncn2C1 14946,C(CCC(N)=O)(C(=O)NC1CCN(C(=O)COCC(C)(C)C)CC1O)NC(C)=O 14947,N1(C(Cc2ccn(C)n2)=O)CCOC(C)(CNC(=O)CC2CCS(=O)(=O)CC2)C1 14948,C1(NC(C2C(OCC)C2)=O)CN(C(=O)CCn2cc(Br)cn2)CC2(CC2)C1 14949,N1(C(c2ccc(C#C)cc2)=O)CC(NC(=O)CCN2CCOCC2)CC2(CC2)C1 14950,C1(C)(C(N(CC(C)O)CCNC(=O)C(=O)NCC2CC2)=O)CCN(C)C1=O 14951,c1(C(=O)Nc2nc(C3CC3)[nH]c3ncnc2-3)scc2c1OCCO2 14952,N1(C(C(C(CC)C)O)=O)CC2CCCC1C2CNC(=O)C1=CCOCC1 14953,C1(C(C)C)CCNC(c2nnnn2Cc2ccccc2)CO1.C(C)(C)(C)OC 14954,N1(C(c2cccc(OC)n2)=O)CC(C(=O)Nc2sncc2C(N)=O)CC(F)C1 14955,C1(CN(C(=O)C=Cc2cc[nH]n2)C)CCCN(C(C2CCOC(=O)N2)=O)C1 14956,c1(CNC(C(CC)N(C)C(c2ccnnc2O)=O)=O)cc(O)ccc1F 14957,C12(CNC(CC3C(C)(C)C3)=O)CC(CN1C(c1nocc1-c1ccccc1)=O)C2 14958,c1(C(=O)OC)ccc(F)c(CN)c1F.c1(-c2cn(C)nn2)cccc(C#N)c1 14959,C(c1cnc[nH]1)=CC(=O)N(CCOCCNC(=O)CCOCC1CCCO1)C 14960,C(=O)(CC(C)CC(C)(C)C)NCCC1N(C(COCc2onc(C)n2)=O)CCC1 14961,Cn1cnnc1CCC(=O)NCC=CCNC(c1ccsc1Br)=O 14962,Cc1cnc(-c2noc(C(C3(C)CC3)F)n2)nc1 14963,c1(OC)ccc(NC(=O)Nc2cc(N3OCCNC3=O)ccc2F)cc1F 14964,Cc1nn(C(C)(C)C)c(C)c1C(N1CC=CC(NC(C2(F)CC=CCC2)=O)C1)=O 14965,Cc1cc(F)ccc1NC(=O)C(c1cccc(F)c1F)N(C1CCOC1)CCF 14966,C1(Cc2cn(CCCC(=O)NC(CC(C)=O)C)nn2)CN(C)CC(C)O1 14967,C(=O)(N=c1ccc(Oc2ccccc2)n[nH]1)Nc1cccc(OCC(N)=O)c1 14968,Cc1cccc2cc(C(N3CCC4(C3)CN(C(=O)Cc3nc[nH]n3)C4)=O)nn12 14969,C1(NC(CC(=O)NCC#C)=O)CN(C(=O)C(C)(C)c2ccccc2)CC12CC2 14970,C1(C(=O)NC2(CC)CC2)(CNC(=O)CC2(C)CCOC2)CC(F)(F)C1 14971,C1(NC(C2(F)C(C)OCC2)=O)CC2(CCN(C(=O)C=Cc3ccccc3)C2)C1 14972,C1(NC(C=C(C)C(F)F)=O)CCC(N(C(=O)C(c2cnn(C)c2)C)C)CC1 14973,C(=O)(C1=NNC(C(F)(F)F)C1)NC(C1CN(C(=O)CCC(C)(C)F)C1)C 14974,c1(OC)ccc(NCC(=O)NC(c2nncs2)C)nc1 14975,C1(C)(C(N(C)CC2(NC(C(COC(C)C)NC(C)=O)=O)CC2)=O)CCC12CCC2 14976,C=CC1CN(C(=O)CC(C)COC)CC1NC(=O)Cc1cc(C)ns1 14977,N(C(=NCC1CCCCCC1)N1CCC2(C1)Oc1ccccc1O2)C(C)C 14978,N1(C(c2n(C)c(Cl)c(Cl)c2)=O)CC(NC(C2CC(O)CN2C)=O)C2(CCC2)C1 14979,c1(C(=O)NCCCCCN(C(C2(C=C)CCOCC2)=O)C)cc(C)cc(C#N)c1 14980,C1(C(=O)N)CC2(CCN(C(=O)CN3CCOCC3=O)C2)C1.N#CC1CC(C)C1 14981,N1(C(C(C)CC(F)F)=O)CCC(C2CC2NC(C2(O)CCC(C)(C)CC2)=O)CC1 14982,C1(C)(C(=O)NC(C)CNC(=O)CSC(=N)N)CC(c2ccccc2)=NO1 14983,N1(c2nc(N(C)Cc3ncc(CC)s3)nc(C)c2)CCCc2ccccc2CC1 14984,C1(CC)(NC(C2CCC(=O)C(C)C2)=O)CCN(C(C2CCC(=O)N2C(C)C)=O)CC1 14985,c1(C(C)C)ccccc1OCC(=O)NC1CC1NC(c1cc(CF)on1)=O 14986,c1(C(N2C(CNC(c3cc(C)[nH]n3)=O)CC(OC)C2)=O)csc2cccnc12 14987,c1(C(N2CCC3(NC(C=CC)=O)C(CC2)C3)=O)c[nH]ccc1=Nc1ccccc1 14988,N1(C(Cc2n(C(C)C)cnn2)=O)CCC2CC12C(=O)NCCC1(C)CCCO1 14989,c1(C(=O)NC(c2ccccc2)CNC(CCC(=C)C)=O)cc2c[nH]nc2s1 14990,C1(CNC(c2cc(Cl)cnc2O)=O)CC(F)(F)CN1C(=O)C=Cc1cnc[nH]1 14991,c1(COC)noc(CNC(=O)CC2CCN(C(=O)C(F)C3CCOC3)C2)n1 14992,Cc1nn(CC(N2CCC(CO)C(NC(=O)CCSCC(C)C)C2)=O)c(C)c1Cl 14993,N1(C2CCN(C(C(CSC)OC)=O)C2)CCN(C(=O)CC2CCOCC2)CC1 14994,n1(CC(=O)NC(C2(O)CN(C(=O)C=Cc3cncs3)C2)C)cc(N)cn1 14995,c1(C(N(C(CNC(C(C)NS(C)(=O)=O)=O)C2CC2)C)=O)sc(F)cc1Cl 14996,S(=O)(=O)(CCC(=O)NCC(C1CCOC1)NC(=O)C(F)(F)c1cscn1)NC 14997,CC1(C)CCCC2(CN(C(C3COCCO3)=O)C2)O1 14998,C(=O)(C(C)CC(F)(F)F)N(CC(CN(C(C=CC=C1CC1)=O)C)O)C 14999,C(C(C)CN=c1c(C#N)c[nH]c2cccc(C)c12)NC(c1cc(C)nn1C)=O 15000,c1(CC(=O)NCC23CC(NC(CC4CCC(C)CO4)=O)(C2)C3)coc2ccccc12 15001,CN1CCCC(C(=O)Nc2cccs2)C1=O.c12csc(n1)NC2=O 15002,c1(OC)cc(N)c(C(N2CCCCC(NC(=O)C(C)NC(N)=O)C2)=O)c(F)c1 15003,C(CO)(C(=O)N(CCNC(C1CC12CCC2)=O)C(C)C)NC(C(C)C)=O 15004,c1(NC)ccc(C(=O)OCCN2CCOCC2CC(=O)NC(=O)C(Cl)(Cl)Cl)cc1 15005,C1(CC(N2CC(C)(NC(=O)CCC(=O)N3CCC3)C2)=O)CCOC(C)(C)C1 15006,C(=O)(C1CCCn2cnnc21)N(CC(=O)NC1CC1)CC1CN2CCC1C2 15007,c1(C(N2C(CC)C(C(=O)NCc3cc(=O)cc[nH]3)CC2)=O)cnc2cc[nH]c2c1 15008,C1(CNC(c2ccc3ncccn23)=O)CCCC(F)(F)CC1 15009,CC#CCCC(=O)NC1CN(C(c2cnc(-c3ccc(Cl)s3)s2)=O)CC1OC 15010,C1(CC)=NC(C)(C(=O)NCCCC(C)(C)NC(C2CCC2C)=O)C(C)=N1 15011,c1(C(=O)NC(C)C(C)(C)NC(c2ccc(CO)c(F)c2)=O)ccc(N)c(Cl)n1 15012,C12CN(CCN1C)C2=O.CC(C)C(O)Cc1cn(C(C)C(=O)O)nn1 15013,C1(C(N2CCN(C(C(C)CO)=O)C(CO)C2)=O)CC2CCC(C1)S2(=O)=O 15014,c1(C(N2CCC(OC)CC2)C(=O)NCC=C)cnc2sc(Br)cn12 15015,c1(C(=O)NC(CNC(c2cncc(C)c2)=O)(C)C2CC2)ccc2c(c1)SCC(=O)N2 15016,c1(N(CC(O)CN2CCOCC2)C(CC2CC(N)C2)=O)ccccc1 15017,C1(C(N(CCC)CCNC(=O)C(CC)(CC)CO)=O)Cc2cccc(F)c2O1 15018,C(N=c1[nH]cnc(Cl)c1CC)C1OCCCN(C(CC2(C=C)CCOCC2)=O)C1 15019,CCCC(C)(C)C(=O)N1CC(OCC(=O)NC2CC2COC)C1 15020,N1(C(c2nn(C)nc2Br)=O)CCN(C(c2cc(Cl)ccn2)=O)CC12CC2 15021,C(C)(C)(C(C)(C)CO)NC(CC1CCCN(C(=O)Nc2cnn(C)n2)C1)=O 15022,c1(OC)nc2c(C)csc2cc1C(=O)NC1CC(C(N2CC3CC3C2C#N)=O)C1 15023,CC(C(=O)NC(C)(CNC(=O)CCc1cnoc1)C1CCC1)C1CC1 15024,N1(C(N2CCCC(N3CCN(C)CC3)C2)=O)CCCCCC1C(C)(C)C 15025,C1(N(C)C(c2cc[nH]n2)=O)CCCCN(C(C2CC(C)(C)O2)=O)C1 15026,C1(C(=O)NCC(C(C)(C)C)NC(=O)CNC(c2ccco2)=O)C(Cl)(Cl)C12CC2 15027,N1(C(COC2CCN(C(C3(C#C)CCC3)=O)C2)=O)CC(F)CC1COC 15028,c1(CNC(CC2CC(OCCCC)C2)=O)c[nH]nn1.c1(CO)cc(C(N)=O)co1 15029,CC(CS(C)(=O)=O)C(=O)NCC1(F)CCN(C(c2ccc3ncnn3n2)=O)CC1 15030,C1(NC)COC2(CCCN(C(c3ccc(NCC(=O)NCC=C)cc3)=O)C2)C1 15031,C1(C(N(C)CC2CCN(CC)C2)=O)CCN(C(c2csc(Cl)c2)=O)C1(C)C 15032,S(=O)(=O)(c1c(Cl)cc(Br)cc1Cl)N1CC2C(C(=O)Nc3c(F)cncc3F)(C2)C1 15033,N=c1[nH]nc(Cl)cc1CNc1cccc(Cc2ccccc2)c1 15034,C1(CN(C(CCCOCC)=O)C)CN(C(=O)CC2(O)CCCOC2)CCO1 15035,N1(C(C(C)SCCC)=O)CCN(CC(C)(C)NC(=O)C(C)C(F)F)CC1 15036,c1(C(=O)NC2C(NC(C(CSc3ccccc3)OC)=O)C2)ccc(N)c(Cl)c1 15037,N1(C(c2nc(CNC(c3nn(C)c(Cl)c3)=O)oc2)=O)CCN2CCC1C2 15038,C(=O)(C1=C(Cl)CCOC1)N1CCC2(C(C(N(C(C(C)C)C)C3CC3)=O)C2)C1 15039,C1(CNC(c2cc(C(C)=O)on2)=O)(NC(c2cc(O)ncn2)=O)CCCC1C 15040,CC1CCC(NC(=O)CCOCC(F)F)CN1C(=O)Cc1ccc(O)c(O)c1 15041,c1(C(=O)NC2COCC2NC(C2CCCCC2O)=O)cnc2nccn2c1 15042,C12(OC)CCC(C(=O)NC3CCN(C(=O)C(F)(F)C(F)(F)F)CC3F)(CC1)CC2 15043,N1(C(CC=CCC)=O)CC2(CC2)CC1CNC(=O)C(C#N)CCC 15044,c1(CNC(C(=O)NCC=CC)=O)cncc(Br)c1 15045,N1(C(c2ccc(C#C)o2)=O)CC2CC(NC(=O)C(C)C3CCCO3)CC1C2 15046,N1(C(CCCC(=C)C)=O)CCOC2(C1)CN(C(C1CC(=O)N(CCOC)C1)=O)C2 15047,C1(N(C(C(c2ccc(F)cc2)C)=O)C)CCCN(C(=O)Cc2cccc(F)c2)C1 15048,N1(C(Cc2c(CC)noc2CC)=O)CC2(CNC(C3CSC3)=O)CC(F)(C1)C2 15049,C1(C(N(C(CC)C)C)=O)(N(C(=O)C=C(C)COC)C2CC2)CCC1 15050,C1(C(N(C(C)C)Cc2ccccc2)=O)CN(C(C2CCC=CO2)=O)CCO1 15051,N1(C(C(CC)C)=O)C2CCC1CC(F)(CNC(=O)C=C(C)C(F)F)C2 15052,N1(C(C2COCCN(C(C3CN(C(C)C)C3)=O)C2)=O)CCC12CCCOCC2 15053,C=CCCCCCNC(C1(CF)CCN(C(c2ccnc(NC)n2)=O)C1)=O 15054,N1(Cc2ccc(C(=O)OC)cc2)CCSC(C)CC1.C12CCN(CC1)C2=O 15055,C1(CC=C)(C(=O)N(C)Cc2csc(C)n2)CCCN1C(=O)CCc1cn[nH]c1 15056,c1(C(N(CC(=O)OC)CCO)=O)cc(NC(=O)OC(C)(C)C)cn1C 15057,N1(C(CC2C(C)C(=O)CC2)=O)C2CC1CN(C(c1ccc(CO)cn1)=O)C2 15058,c1(C(=O)OCc2nn(C)c(Cl)c2)nc(Cl)c(=O)[nH]c1N 15059,C=Cc1ccc(C(=O)NCC(C)N(C(C(=O)OC)C)C2CC=CC2)cc1 15060,CS(=O)(=O)c1ccccc1-c1ccc2c(N3CCOC(CC(N)=O)C3)[nH]nc2c1 15061,N1(C(CSCC)=O)CC(F)(F)CC1CCNC(=O)Cc1ccccc1OC(F)F 15062,C1(CNC(CC2(CC=C)CCCC2)=O)CC12CCN(C(=O)Cn1ccnn1)CC2 15063,N1(C(C2C(C(C)C)CCC2)=O)C2CCC1C(F)C(NC(c1cc(Cl)cs1)=O)C2 15064,c1(C(CNC(=O)C(C)(C)CO)NC(C=CC)=O)ccccc1CC 15065,C1(NC(c2cn[nH]c2)=O)CCN(C(c2ccncn2)=O)CC1CO 15066,c1(C(C)C(=O)NC2CC(O)(CNC(c3ccccn3)=O)C2)cc2ccccc2o1 15067,C(=O)(C(C)(C)CC(C)(C)C)NC1(COC)CN(C(c2ccnnc2C)=O)C1 15068,C1(CNC(c2cc(OC)no2)=O)CC2CC2N1C(c1cc(C)n(C(C)(C)C)n1)=O 15069,c1(C(=O)NCCOCCCN(C)C(c2cnc(O)o2)=O)cc(Cl)ns1 15070,c12ccccc1CNC(=O)COC2.CCS(=O)CCNCc1ccccc1 15071,Cc1cc(C(=O)NCC(C)(C)NC(=O)Cc2sc(C)nc2C)c(O)cc1F 15072,C1(NC(c2ccc(NC(C)(C)C)nc2)=O)CCC2(CC1)CN(C(=O)CCl)CCO2 15073,c1(CC(=O)N(C2CCC(NC(=O)C(F)(F)C3CC3)C2)C)cncc(C#N)c1 15074,c1(N2CC(C)CS(=O)CC2)nc2cc[nH]c2c(=NCC(C)(C)c2ccccc2)[nH]1 15075,C1(C(=O)OCC)CCC(C(F)(F)F)(NC(C2(N=[N+]=[N-])CC(C)C2)=O)CC1 15076,c1(N2CC3C(C)C3C2)nc2ccccc2nc1N(C)Cc1ccc(S(C)=O)cc1 15077,C1(CNC(=O)CC(C)(C)C)CCN(CC2(O)CC(NC(C3CC(=C)C3)=O)C2)CC1 15078,C#Cc1cnn(C)c1C(=O)NC1CCCCC1C(N1CC(C)C(O)C1)=O 15079,CCC(C(=O)NC1(CC=CC(N2CCC(CCC)C2)=O)CCC1)C1CCC1 15080,CC(O)C(C(=O)NC(C(N)=O)C1CC1)NC(c1ccc(O)cc1)=O 15081,c1(CN(C2CC3(CN(C(C)C)C3)C2)C)cc(Cl)c2cnn(C)c2n1 15082,c1(CN(C(CC)C)C(C2(c3ccccc3)CC2C#N)=O)cnn(C)c1C 15083,C1(CC(=O)NCCC2(CNC(C(C)C)=O)CC2)CC(C(C)=O)C1(C)C 15084,N1(C(C2(C)C(C(=O)OC)CC2)=O)CCC(CNC(=O)C(C)(C)C2CC2)CC1 15085,C12C3CN(CC13)C2.C1(C(=O)OC)(CN)CC1(F)F 15086,C1(CC)(CNC(=O)C)CN(CC2(CS)CC2)C1.C1(=O)CN1.C1(OC)CC1 15087,CC1(C)CN(C(=O)Cc2ccc(F)cn2)CCC1NC(=O)C1=CSCCO1 15088,c1(SCC(=O)NC2CC(NC(C3COCCC3(F)F)=O)C2)ccc(F)c(F)c1 15089,S(=O)(=O)(c1cccnc1NC(C1CCCS(=O)(=O)C1)=O)NCCNC(C)=O 15090,Cc1ncccc1CC(N1CCC(C)C1CNC(=O)CN1C(=O)CCC1=O)=O 15091,C(=O)(C(c1ccccc1Cl)=CCO)N1CCC(CN(C)C(C2(O)CC2(C)C)=O)C1 15092,N1(CCCCC2CCCN(CC)C2)CCN(CC(=O)NCc2ccccn2)CC1 15093,CC(CCNC(=O)CN1CCC(CO)CC1)CCNC(c1ccc(O)nn1)=O 15094,N1(C(C(CCC)(C)O)=O)CC(C2CCCN(C(c3cnc4cccnn34)=O)C2)C1 15095,C1(NC(C(C2CC2)OCC)=O)CCC(F)(CNC(c2cc(CC3CC3)[nH]n2)=O)C1 15096,C1(F)(CNC(c2c(C)snc2)=O)CCCN(C(c2cnnn2C2CC2)=O)C1 15097,CCCCC(F)C(=O)NC(C(N1CCCC1C)=O)c1ccco1 15098,CC1CN(C(C2CN(C(c3ccc(C#N)o3)=O)CC2(C)C)=O)CCS1=O 15099,C1(NC(C(C)C2CCCC2)=O)CCN(C(=O)CP(C)(C)=O)CC1C(N)=O 15100,c1(C(=O)NC(C)CC(C)NC(=O)C(C)CSC(F)(F)F)csc(=NC2CC2)[nH]1 15101,Cc1ccccc1Oc1ccc(CNC(=O)C(c2c(C)noc2C)(C)C)cc1 15102,c1(CC)onc(C)c1C(=O)NC1CCC(CNC(C2CCOC2=O)=O)CC1 15103,CC1CN(C(=O)C=Cc2ccco2)CC(CCNC(=O)CCC2CC2)O1 15104,C=CCCCC(=O)NCCC1(OC)CN(C(c2csnc2Cl)=O)C1 15105,c1(CC)cccc(C(=O)NCC2CN(C(c3n[nH]cc3F)=O)CC2C)c1N 15106,c1(C(=O)NC2(COC)CCN(C(=O)C#CC(C)(C)O)C2)cc(S(N)(=O)=O)c[nH]1 15107,Cc1nnnn1CC(=O)NCC(C1CC1)NC(=O)CCN(C1CCCCC1)C 15108,Cc1ncc(C(C)NC(=O)C(CC2CCCC2)NC(c2cnsc2C)=O)s1 15109,C(C)(C)(C(CO)CO)NC(C1N(C(CCCOCC=C)=O)CCC=C1)=O 15110,C1(NC(C(CCCOC)C)=O)CCCCN(C(=O)Cc2cccc(C)c2)CC1 15111,Cc1cccc(C(N2CCCC(C)C2CNC(c2c[nH]ccc2=O)=O)=O)c1O 15112,c1(NC(c2nc(C(=O)Nc3ccc(I)c(Cl)n3)cs2)=O)cccc2[nH]ncc12 15113,N1(C(c2cc(C)ncc2C)=O)CCCC(O)(CNC(=O)CCNS(C)(=O)=O)CC1 15114,N1(C(Cn2c(=O)sc(C)c2C)=O)CC2ON=C(CNC(c3ccn(C)n3)=O)C2C1 15115,N1(C(c2c(C)nco2)=O)CCC2(CC1)CC2C(=O)NC1CC1(C)C 15116,N1(C(c2c(C)cns2)C(=O)NC2CCOC2)CCCC(c2ccc(CO)o2)C1 15117,N1(C(C2C(SC)CCC2)=O)CCC(=CCNC(c2sccc2C2CC2)=O)CC1 15118,C1(OC)CN(C(=O)C(C)=CC2CC2)CC1NC(c1ccc(F)s1)=O 15119,Cc1cc(COCC(=O)NC2(C)CN(C(C3CCCN3C)=O)C2)on1 15120,N1(C(CN(C(C)=O)C)=O)CC2CC(C1)N2C(C1CC(C)(C)CO1)=O 15121,Cc1cc(C(=O)NC2CCN(C(c3nocc3Cl)=O)CC2O)c(C)n1NC(N)=O 15122,C1(C(N2CC(N(C(=O)COC3CCCC3)C)C2)=O)CCCCS1(=O)=O 15123,C12(NC(C(C)CC3CCC3)=O)CC(C1)N(C(C1C(C)C1C)=O)C2 15124,C1(CNC(c2nc(C)oc2)=O)CCN(C(c2cc(C)n(C)n2)=O)C1(C)C 15125,C(C)(C(=O)NNC(=O)C1CC1)Nc1ccsc1CS(=O)(=O)CCn1c(C)cc(C)n1 15126,C(CCC(CO)NC(c1coc(C2CCC2)n1)=O)NC(=O)CCCF 15127,c1(OC)cc(OC)[nH]c(=NCC2(C)CCN(C(=O)C=C3CCSCC3)C2)n1 15128,Cc1cccc(O)c1C(=O)NC1CC(CCC(=O)NCc2cn(C3CC3)cn2)C1 15129,N1(C(C(CC)OC2CCCC2)=O)CCCC(CC#N)C1 15130,c1(OCC)cnc(C(=O)NCc2cccnc2NCc2cscn2)cn1 15131,C1(C(=O)NC(CSC)(C)C(=O)N2CCOC(C(C)C)C2)CC2(CC(=O)C2)C1 15132,C(C(CC(C)C)C(=O)NCC(O)C(C)C)NC(CC(CC)(F)F)=O 15133,C1(C(=O)NCC2(CCOC)CC2)CC12CC(NC(=O)CN1CCNC(=O)C1)C2 15134,CCCCCS(=O)(=O)NC(C1(C(F)F)CCNC1)=O 15135,Cc1c(C(C(=O)NCC(F)F)N(CC(=O)N(C)C)C)cnn1CC(F)F 15136,C1(CNC(C2CN(CC(C)C)C2)=O)COC(CNC(=O)CCc2nccn2C)C1 15137,N1(C(CNC(CCCC)=O)=O)CC2CC2C1CNC(c1cnccc1C)=O 15138,c1(C(=O)NC2CCN(C(C(C=C=C)C)=O)C2)ccc(Cl)c(C(=O)OC)c1 15139,N1(CC)C(C)C2CCCCC2C1.C12CC13CC(C3)C(=O)OC2=O 15140,CC1(CNC(=O)CC2CCSCC2)CC(NC(c2cn(C3CC3)cn2)=O)C1 15141,c1(CCC(=O)NC2C(OC)CN(C(C(CC=C)C)=O)C2)ccc(Cl)c(C)c1 15142,CCCC(O)CC(=O)NC(C)(C)CN(C(=O)C(c1ccc(Br)cc1)CC)C 15143,c1(C(N2CCC(NC(CC(CC)SC)=O)(CF)C2)=O)ncc(F)c(OC)n1 15144,c1(C(N(CC(CC)NC(C2CCCSS2)=O)CC)=O)ccc2ccccc2c1 15145,c1(C(=O)NCC2CC(NC(=O)CC3COCCO3)C2)c(Br)ccc2cccnc12 15146,Cc1ccc(SC(C)C(=O)N(CCCN(C)C(c2cc(C(C)C)no2)=O)C)cc1 15147,c1(C(C(N2CCC(N(CCO)CC3(C=C)CCC3)C2)=O)C)ccc(C#N)cc1 15148,C(=O)(C=CS(C)=O)NC(C)C(c1ccccc1F)NC(C1CC2(CSC2)C1)=O 15149,CC1(C)CCC(C(=O)NCC#CC(=O)NCc2c[nH]nc2C2CC2)CO1 15150,c1(C(=O)NCC(=O)NC2(C)CC(C(=O)NCC(=O)NC)C2)cccc(F)c1 15151,N1(C(C(C)CC2CCC2)=O)CCC(CO)(CNC(c2c[nH]cc2C2CC2)=O)CC1 15152,C1(NCC(C)(C)Cc2nnnn2C2(C)CCOCC2)CC2CCC(C1)S2 15153,Nc1cc(C(N2CCCCC(NC(C3CC4OC3C3CC43)=O)C2)=O)cc(F)c1O 15154,C1(NC(C2(CC#C)CCCC2)=O)CCC(C)N(C(c2ccc(Cl)cc2N)=O)C1 15155,c1(CNC(C2CSCCN2C(c2cnc(O)o2)=O)=O)ccccc1F 15156,c1(C(N2CC(C(C)(C)O)(CNC(C3C(C)(CC)C3)=O)C2)=O)ccc2cc[nH]c2c1 15157,C12(NC(C#CC(C)C)=O)CCN(C(c3cccnc3C(F)(F)F)=O)CCC1C2 15158,C1(CC(=O)NC(C)CCCNC(c2cnn(C(C)C)n2)=O)CCCCCO1 15159,CC(c1cnn(C)c1)=CC(=O)NC1CCC(NC(C2CCN(C)C2C)=O)C1 15160,C#CCCC(O)C(=O)N1CCN(C(=O)CSCCCC)CC1C(F)F 15161,c1(C(=O)NCCCC2(NC(C(CC)NC(C)=O)=O)CC2)cnn(C)c1Br 15162,C1(CC(=O)NCc2nc(C)on2)CCCN(C(C2CCN(C)CC2)=O)C1 15163,C1(CNC(C(C=CC)O)=O)CC2CCC1N2C(=O)C(c1cccc(F)c1)O 15164,N1(C(CCSCC(C)C)=O)CC(C(=O)NCC2CC23CCC3)CC1(C)C 15165,N12C(CC1C)C2=O.C1(COC)C=CC1C(=O)NCCS(C)(=N)=O 15166,N1(C(C)=O)CCN(C(C(=O)NCCCF)C2CC2)C(CC(F)F)C1 15167,CC1(CNC(C2OCCC2C(F)F)=O)CCN(C(c2csnn2)=O)C1 15168,C(=O)(NNC(=O)C(C)(C)CCCCNC(C1(SC)CC1)=O)C1(OC)CCCCC1C 15169,C(=O)(C(Cc1cnc[nH]1)NC(C1CC(O)C1)=O)NCC(=O)NCC(C)C 15170,Cn1cccc1CC(N1CC(C(=O)NCCNC(=O)CCC2CCN(C)C2)C1)=O 15171,C(C)(CC(C)NC(C1CC1OC(C)(C)C)=O)NC(C1C(CCC)C1)=O 15172,N1(C(CCCC2CN(C(C=CCCC)=O)C2)=O)CCC(n2ccnn2)C1 15173,C1(C)(CNC(C(C(C)(F)F)F)=O)CC(F)(F)CN1C(c1cccn2cnnc12)=O 15174,C=CC(C)(C)C(=O)NCC1CCN(C(=O)C(F)C2CC(NC(C)=O)C2)CC1 15175,N1(CC(=O)OC(C)(C)C)CCC(CC(=O)NC(CNC(=O)CC2CCCC2)CO)C1 15176,C1(CC)CCOC1C(=O)N(CCCNC(c1nnn(C)n1)=O)CC1CCCC1 15177,C1(NC(C(CC)(C)C)=O)CCC2CCN(C(=O)CCc3ccccc3[N+](=O)[O-])C12 15178,c1(CCN(C(C(CCC)c2ccc(Cl)cc2)=O)C)ccc(Cl)cc1Cl 15179,C12CCN(C1)C(=O)c1sccc1NC(=O)C2.c1(C2C(C(=O)O)C2)ccncc1 15180,C(=O)(C(CCCC)C(C)C)NCCCOCCC(=O)Nc1cc(C#C)c(C)cc1 15181,C1(CCNC(=O)C=CCF)(OC)CCN(C(=O)C(c2cccnc2)C)CC1 15182,c1(C(=O)NC2CC(CNC(C3N(CC)CC3)=O)C2)c(N)cc(F)cc1Cl 15183,C1(CCC(=O)NC(C)CNC(=O)C(CO)NC(N)=O)Cc2ccccc2NC1=O 15184,C(=O)(C#CC1CCOCC1)NC(C(C)(C)NC(C(F)OC)=O)C 15185,CC(C)(CCC(=O)N1CC(O)CC1Cn1cc(C2(CO)CC2)nn1)c1ccon1 15186,c1(SC(C(N2CCN(C(c3c(C)csn3)=O)CC2)=O)C)nc2ccccc2[nH]1 15187,c1(C(=O)NCC2N(C(C(CC(C)C)O)=O)CC=C2)ccc(Br)c2cn[nH]c12 15188,c1(SCC2N(C(C3CCCC3NC3CCNC3)=O)CCCC2)ccc(F)nc1C 15189,N1(C(CC=C=C)=O)CCC2(CCCCN(C(c3cnn(C)c3F)=O)C2)C1 15190,c1(C(=O)NC2CCC(CNC(CC(=C)Br)=O)C2)nnc(O)cc1O 15191,c1(C(N2CCCC(N(C(c3ccns3)=O)CC)C2)=O)c(OC)cccc1O 15192,c1(C2(C(=O)OC)CCC2)cccc(C(C)Nc2cccc(-c3ccncc3)c2)c1 15193,c1(C(=O)NC2CCCC(NC(Cn3c(C)ccn3)=O)CC2)cnn2c1CC(F)(F)C2 15194,c1(COC)nc(-c2cnc(S)n2C)n(-c2ccc(Cl)nc2)n1 15195,C1(OC)=CC=NC=CC=C1S(=O)(=O)NCC(=O)NCc1cnc(Br)s1 15196,C1(C(=O)NCC(C)NC(C(C)CO)=O)CCC2(CC1)NC(=O)NC2=O 15197,CCCC(C)(C)C(=O)NCCC1CN(C(=O)CCN(C)CCC)CC(C)O1 15198,Cc1cc(C(=O)N(C(C)CCNC(c2cc(C(C)C)no2)=O)C)n(C2CC2)n1 15199,C(=O)(C(O)CC(C)(C)C)NCC1ON=C(C(=O)NCC(C(C)C)(C)C)C1 15200,c1(-n2cc(CCCNC(C(C)N(C)C)=O)nn2)cccnc1C(=O)O 15201,N1(C(C2OCC(C)C2)=O)CCC2(CCCN(Cc3ccccc3)C2)C1 15202,C1(O)(C(C(=O)N(CC(F)F)CCO)F)CN(C(=O)CC2OCCO2)C1 15203,C(=O)(C1=NOC2(CCC2)C1)NCC(CO)(CO)NC(C(c1ccc(F)cc1)C)=O 15204,N1(C(C=CC)=O)CC2(CCN(Cc3ccc(OC)c(Oc4ccccc4)c3)CC2)C1 15205,Cc1cnc(CN(C)C(=NCC2CCS(=O)(=O)N2C)NC2CCC2)c(C)c1 15206,Cc1cc(C)c(C=CC(=O)NC(C2CCCN2C(c2cccnn2)=O)C)c(C)c1 15207,Nc1nc(C(N2CCC(NC(=O)CC3(CO)CC3)C(O)C2)=O)ccc1[N+](=O)[O-] 15208,C(=O)(CC(C)CC(C)C)N1CCC(C(N2CC(O)(CC)C2)=O)(CCOC)CC1 15209,C(=O)(C#CC1(C)CCCO1)N1CC(C(=O)NCCc2c(C)n[nH]c2)C(CO)C1 15210,c1(OC(C)C(=O)NCC2(O)CC(NC(C3OCCO3)=O)C2)ccc(F)nc1 15211,c1(C(=O)NCC2C(CNC(c3c(C)cc(C)s3)=O)C2)cccc2c1nc(O)n2C 15212,C(=O)(C(C(C)C)NC(=O)CC1(OC)CCC1)NCC(C)(CSC)OC 15213,C12(C(=O)NCCn3ncc(C(=O)NCC4(n5nccn5)CC4)c3)CCC(CC1)C2 15214,c1(CC(=O)NCC(C(C)(C)C)NC(C2(O)CCCCC2)=O)cnc2[nH]ccc2c1 15215,Cc1ccc2oc(C(=O)NC3CC4CCC(C3)N4C(c3ccc(C#N)[nH]3)=O)cc2n1 15216,c1(OC)ccc(CN2CC(F)(C(=O)NCCC3CCCN(C)C3)C2)c(OC)c1 15217,C1(NC(C(C)OC)=O)CC2CCCC(C1)N2C(=O)CCc1nnc(C2CCC2)o1 15218,CC1(C)CN(C(c2cnc(Br)s2)C(=O)NC2CC(F)(F)C2)CCS1=O 15219,C(=O)(C1=NOC(C(=O)NC2CCCN(C(=O)CC(C)(C)O)C2)C1)OC(C)(C)C 15220,C1(O)(OC(C)(C)C)CN(N2CCC(COC3CC3)CC2)C1 15221,N1(C(C(CCCC)O)=O)CCC(C2CC2)(NC(c2ccccc2NCCO)=O)C1 15222,C1(O)(C(C)NC(C=C(COC)C)=O)CCN(C(c2cnn(C)c2)=O)C1 15223,CCC(C(=O)N1CCCC(C)(NC(c2ccncn2)=O)C1)C(C)C 15224,N1(C(CN(C(C2CCCN(C)C2)=O)CC2CC2)=O)CC23CCC2(COC3)C1 15225,C1(C(N2C(CN(C(c3cn(CC(C)C)nc3)=O)C)CCC2)=O)CCCCC1(F)F 15226,CC1(C)CC(NC(C2CC(C)(C)OC2(C)C)=O)CN(C(c2c[nH]ccc2=O)=O)C1 15227,c1(C(=O)NCC(CO)NC(c2csc(CO)n2)=O)cc(C(F)F)ccc1Cl 15228,CCCC(CNC(C1CCC(C)(C)OC1)=O)C(=O)NC1(CO)CC(F)C1 15229,c1(C(N2CCC(C(CNC(C3C4CCCC34)=O)F)CC2)=O)cccc2cncn12 15230,C1(CC)(NC(=O)CNC(c2csc3nccn23)=O)CCCN(CCCC(F)(F)F)C1 15231,C1(NC(CS(CC)=O)=O)CC2CC1CN(C(c1c(C)ccc(Cl)c1F)=O)C2 15232,CC1CC2CC(C(=O)NC3CN(C(=O)C=Cc4ccccc4Br)C3)(C2)O1 15233,C1(C(CC(=O)OC)NC(=O)CSc2n[nH]c(C)n2)CCC(F)(F)CC1 15234,c1(C(N(CCCNC(C2(C)CC(C)C2)=O)C2CC2)=O)n[nH]c2cc(Cl)ccc12 15235,C(=O)(CC(C)(O)C(F)(F)F)NCC(C)CNC(=O)C=Cc1cccc(O)c1 15236,C(=O)(C(S(C)(=O)=O)C1CC1)NC1C(OC)CN(C(=O)COC2CC2)C1 15237,C1(C2CC2)(C(=O)NC2(CN(C(C3CN(S(CC)(=O)=O)C3)=O)C)CC2)CCC1 15238,Cc1noc2nc(C(=O)NC(C)CCCCNC(c3cnc(Cl)s3)=O)ccc12 15239,C1(CC(=O)NCC(CC)(C)NC(=O)CC(C)COC)CCC=CCC1 15240,CC1CN(C(=O)CCC(=O)c2cccc(F)c2)CCC1NC(=O)C(C)(C)C1CC1 15241,N(C(=NCc1ccc(C#N)c(C)c1)N1CCC2=C(CCCC2)C1)C(CC)C 15242,C(CC(=O)NCc1cc(C2CC2)no1)(C(C)(C)C)NC(c1cc(OC)no1)=O 15243,C1(CC)C(NC(=O)C=CC=C(Cl)Cl)CCCN1C(c1cn(CC(F)F)nc1C)=O 15244,O=C1CC2(CCCN(C(c3ccc(C(F)Cl)cc3)=O)C2)CN1 15245,N1(C(CN2CCN(C)CC2)=O)CC2(CC(NC(=O)C(O)C(F)F)CO2)C1 15246,C12(C(=O)NCc3cc(C)c(C)[nH]3)CCC(CC1NC(c1ccc(C3CC3)o1)=O)C2 15247,C1(C(N2CC(C)C=C(C)C2)=O)CN(C(c2ncn(C)n2)=O)CCN1C 15248,c1(CCC(=O)N(c2cccc(I)c2)C)ccc(C#N)nn1 15249,c1(C(=O)N(CC(N)=O)CCC#N)ccc2nc(-c3cnn(CCF)c3)cn2c1 15250,c1(C(=O)NCCC(C(C)C)NC(c2c(CC)nn[nH]2)=O)cncc(Cl)c1C 15251,c1(C(N2CCCC(C)(C(N3C(COC)CCC3)=O)C2)=O)cnc2cc(Cl)ccn12 15252,CCC(C(=O)N1CC(O)CC1CNC(C1(c2ccccc2)CCC1)=O)C(C)C 15253,c1(OC)c(Br)ccc(CN2CC(NC(=O)CCc3cccc(O)c3)C(F)C2)c1F 15254,C(=O)(C(C(C)CC(C)(C)C)N1CC2OCCN(C)C2C1)NCC=C 15255,N1(C(C(C=CC)O)=O)CC23CCCC2(C1)CN(c1cc(Cl)nc(C2CCCO2)n1)C3 15256,c1(CC)c(C(N2CCOC(CC(=O)NC3CCC=CCC3)C2)=O)cnn1C 15257,c1(CC(=O)N(C(C)CNC(=O)CC2OCCOC2(C)C)C)coc2ccccc12 15258,C1(C(=O)NCC2(C(N)=O)CN(C(c3c(C)onc3)=O)C2)CC2CCC1C2 15259,CC(CNC(=O)COCCN(C)C)(CO)NC(c1cnoc1C1CCC1)=O 15260,c1(CCC(=O)NC2CCCC2CNC(=O)COCCF)ccc(SC(F)(F)F)cc1 15261,C(C1=NOC2CN(C(c3csc(C4CCC4)n3)=O)CC12)NC(c1cnsn1)=O 15262,c1(OC)ccc(Cl)cc1CC(=O)NC1CN(C(C2CC(C(C)C)C2)=O)CC1(C)C 15263,S(=O)(=O)(c1nc(N2CCNC(=O)C2)ccc1Br)N1CC2CN(C)CC2C1 15264,C1(CNC(c2c(C)nn(C)n2)=O)CN(C(=O)Cc2ccc(O)nc2)C2CCN1C2 15265,c1(C(N(CC(C)NC(c2ccc(C(C)C)cc2F)=O)C)=O)n[nH]c2c1CC1CC21 15266,N1(C(C2(C3CC3)CN(C(CCCOCCC)=O)C2)=O)CCCC12CCOC2=O 15267,CC1(NC(=O)CC2CCC3CC23)CCCN(C(c2ccccc2C(F)F)=O)C1 15268,c1(C(N(CCCNC(CCOC)=O)C2CC2)=O)c[nH]cc(C)c1=O 15269,C(=O)(CS(=O)(=O)C1CC1)N1CCC(C(=O)Nc2c(N(C)C)cccc2)C1 15270,c1(CC)cccc(CNC(C2CCCCN2C(C2(C)CC=CC2)=O)=O)c1 15271,C1(OC)C(OC)CN(C(c2ccon2)=O)C1CNC(C1(C)CC2CC2C1)=O 15272,c1(N(C(CCNC(c2cc(CCC)[nH]n2)=O)C)C)ccc(S(C)(=O)=O)cn1 15273,c1(C(=O)NCC2C3N(C(c4ncn(C)n4)=O)C(CC3)C2)cn2cccc(Cl)c2n1 15274,c1(C(=O)NC(CC)CN(C)C(C2(C)CCC(O)CC2)=O)ccnc2c1cnn2C 15275,C1(N(CCC)C(c2cc(C(C)(F)F)on2)=O)CCN(C(=O)COC2CCC2)CC1 15276,C(=O)(C1(Cl)C(=O)N(C)c2ccccc21)NCC1CCC(C)CN1C(=O)CNC=O 15277,C1(NC(c2cncc(CO)c2)=O)CN(C(C2CC3CC3C2)=O)CC1n1ccnn1 15278,c1(Cn2cc(CNCCC(F)(F)F)nn2)cc[nH]c2nccc1-2 15279,CN1CCN(C(C2CC(C)(C)CCO2)=O)C(CNC(c2ccc(O)cn2)=O)C1 15280,C1(NC(C2C(C)CCO2)=O)CCSC12CN(C(C1CCCCC1N=[N+]=[N-])=O)C2 15281,C1(C(C)NC(=O)OC(C)(C)C)CCN(C(C2CCC(C(=O)O)C2)=O)C1 15282,c1(OC)cc(O)ncc1C(N1CCC(CN(C)C(C2CCN(C)C2=O)=O)C1)=O 15283,CC(CCCC(F)(F)F)N=c1[nH]c(=NCc2ccc(F)cc2N)[nH]c2ccsc12 15284,C1(CC)CN(C(c2cn(C)nc2C(F)F)=O)CCN1C(=O)CC(C1CC1)C1CC1 15285,c1(SC)ncc(C(=O)NCC2CC2NC(c2cnn(C)c2S(N)(=O)=O)=O)c(O)n1 15286,Cc1cc(O)nc(C)c1C(N1CC2(CO)CC1(CNC(=O)C#CC(C)(C)C)C2)=O 15287,C1(NC(C(C2CCCC2)NC(C(CC(=C)C)OC)=O)=O)CCn2ncnc2C1 15288,c1(CC)cc(C)ccc1C(=O)NCC1CC(NC(=O)C(C)(C)CC#N)CC1O 15289,C1(C(=O)NCCC(C)(C)NC(C(C2CCCC2)OC)=O)Cc2ccccc2S1 15290,N1(C(C=COCC)=O)CC2C3CCC(C2C1)N(C(c1coc(C(F)(F)F)c1)=O)C3 15291,N1(C(C)=O)CCCCC1c1cccnc1C(=O)NCCn1cnc(C)c1 15292,C1(CC(N2C(CNC(c3cnc(OCC)s3)=O)CCCC2)=O)CN2CCN1CC2 15293,S(=O)(=O)(C1CCCN(C(c2c[nH]nc2-c2ccc(C#N)cc2)=O)C1)N(C)C 15294,c1(N(CC(=O)OCC)CC)ncnc2c1ncn2CC(O)C(C)(C)C 15295,N(C(=NCCC(C)(C)O)NC1CC1C1CCCC1)C(C=C)C 15296,Cc1ccc(NC(C23CCC(CC2NC(=O)CC(O)CN(C)C)C3)=O)c(C)n1 15297,C(=O)(CS(=O)(=O)CC)NCC1CN(C(c2cn(CCCC)nc2C)=O)CC1C 15298,N1(C(CCSCCCC)=O)C(CNC(c2cnn(C)c2OC)=O)CC2COCC12 15299,c1(C(=O)NCC2C(NC(c3cn(CC=C)nn3)=O)C2)cc(OC)cc(Br)c1 15300,c1(N(CC(=C)C)C)nc(=Nc2cccnc2C)nc(-c2ccccn2)[nH]1 15301,C=C1C(=O)ON2CCC1CC2.c1(C(=O)OC(C)(C)C)ccc2c(c1)CCCC2 15302,N1(C(Cc2c(C)cccn2)=O)CCN(C(C2CC23CC(O)C3)=O)C2CCC12 15303,N1(C(C(CSC)OC)=O)CCCCCC1CNC(=O)Cc1ccc(F)c(F)c1 15304,c1(C(=O)NC(CNC(C(C(C)C)C)=O)CO)cc(N)cc2ccccc12 15305,c1(C(=O)NCC(C)CNC(C2CC23CC(O)C3)=O)cnc(-c2ccccn2)nc1 15306,C#CCCN=C(NCC1CC1C1CCOCC1)N1CCC2NC(=O)OCC2C1 15307,C#Cc1ccc(C(=O)NC2CCC(C)(NC(=O)CSC)CC2)nc1 15308,N1(C(C=C2CCC(C)C2)=O)CCCC(CNC(=O)CCc2cncs2)CC1 15309,N1(C(C)=O)CCC(NC(c2ccc(C(=O)O)s2)=O)CC1.N12CCCC1CCNC2=O.O 15310,c1(C(N2CC(O)(CNC(CC3(C)CC3)=O)C2)=O)ccncc1Br 15311,C(C)(CN(C(Cc1cn(NC(c2coc(C)c2)=O)nn1)=O)C)(C(C)C)NC(CC)=O 15312,c1(OC)ccc(NC(=O)Cc2sccc2Cl)c(OC)c1C 15313,Cc1cccn2c(C(N3CCCC(CO)(NC(=O)Cc4cnsc4)C3)=O)cnc12 15314,C(=O)(CC(C)(C)CN(C)C)NC(C(C)NC(c1csc(C)c1C)=O)C(C)C 15315,N1(C(c2c(C)cc(C(F)(F)F)s2)=O)CCN(C)C(CNC(=O)CCOC2CC2)C1 15316,C1(CNC(C(C(C)C)SC)=O)CN(C(=O)CC(C)(C)C)CC1(C)C 15317,c1(C(N2CCC(OCCNC(c3ncc(C)nc3)=O)C2)=O)cn2nc(C)sc2n1 15318,c1(OC)ccc(N2CCC(C(=O)Nc3ccccc3Cl)CC2)nn1 15319,C1(C(=O)NCC(CCNC(C2CNC(=O)C2)=O)OC)CN(C)C(=O)CCO1 15320,C1(NC(C2C(C)(C)C2NC(C2CC(O)(C#N)C2)=O)=O)C=CCCCC1 15321,C#CCC(C)(C(=O)N1CC(CO)CC1CO)NC(c1ccc(C)o1)=O 15322,C1(C)(C(=O)NC(CCNC(C(CC)C2CCOCC2)=O)C)CC(C)(C)C1 15323,C(CCC(C)(C)C(=O)N1CCCC1C(N1CC(O)(CCO)C1)=O)OC 15324,N1(C(c2n(C(C)C)cnc2)=O)CC2C(CNC(=O)Cc3ccncc3Cl)C2C1 15325,c1(COC)ccccc1N(CC(=O)NC)C(=O)NC1CCC1C 15326,c1(CN(C)CC2CCC(NC(CN3CCCC3C)=O)CC2)ccc(Cl)c(Cl)c1 15327,C1(CNC(COCC#C)=O)CN(C(=O)CC(C)(O)CCC)CCC1(F)F 15328,c1(C(=O)NCC2C(C)CN(C(c3cc(C(C)(C)C)on3)=O)C2)nc(Cl)ccc1F 15329,c1(C(N(C2CCN(C(=O)C(CCOC)OCC)C2)CC)=O)cccc2ncsc12 15330,c1(C(N2CCC(NC(c3c(CC)nccn3)=O)C2)=O)c(Br)sc(C)c1C 15331,n1(CCCC)ccc(C(N2CC(CC)(NC(=O)CSc3nc[nH]n3)C2)=O)n1 15332,c1(N2CC(NC(C3CC4(CCC4)CO3)=O)CC(C)(C)C2)nc2cccc(F)c2s1 15333,C1(CNC(C(CNC(c2ccnc(O)c2)=O)OC)=O)CC2(CC2)C(=O)O1 15334,Cc1ccc2c(CC(=O)N(C)CCOCCNC(C3(C)CCCC3)=O)c[nH]c2c1 15335,N1(C(C2(C)CC=C(C)CC2)=O)CC2CC1CCC2NC(=O)C(C)C1CCCC1 15336,Cc1ccc(C(=O)NC23CCN(C(C4(C)CCCC4)=O)CCC2C3)cc1C#N 15337,n1(CCOCC)nnnc1C(C(C)SC1CC1)NCC1CCCC1 15338,C1(C(N(CCN(C)C)CCO)=O)CCC2(CN(Cc3ccc(C#N)cc3Cl)C2)O1 15339,N1(C(CCOCCC)=O)CCN(C(C2COCCC2(F)F)=O)C(C)C1 15340,N1(CS(=O)(=O)CC)CCCC2CN(C(=O)CCCNC(CCC)=O)CCC12 15341,c1(CNC(C(=Cc2cn[nH]c2)C)=O)nnn(C)c1C(N1CCC(C)(CO)C1)=O 15342,C=CCC(C)(C)CC(=O)N1CCC(N(C(=O)C(C)(C)C(N)=O)CCC)CC1 15343,N1(C(=O)CN(S(CC)(=O)=O)C)CCC(COC2CCN(C(C3(Cl)CC3)=O)C2)CC1 15344,C1(NC(C2CS(=O)(=O)C2)=O)C2CC3CN(C(=O)COc4ccc(O)cc4)C1C3C2 15345,CC1(C(N2CCC(NC(c3cccn4ccnc34)=O)C2)=O)CCCC(F)(F)C1 15346,C12(NC(=O)CCC3CCCC3O)CCC(CN(C(=O)CNc3cccnc3)C1)C2 15347,C12(NC(C(c3ccnn3C)C)=O)CC(C1)N(C(C1CCN(C(=O)N(C)C)CC1)=O)C2 15348,c1(C(=O)Nc2ccnc(C(C)(C)C)n2)cn(CCO)c(=O)nc1O 15349,C1(C)(OC)CCN(C(C2CC3C=CC2CC3)=O)CC1 15350,C1(C#N)(C(=O)NC(C2CCN(C(CC(C)OC)=O)C2)C)CC1(C)C 15351,C#CCC(C)(CC)C(=O)NCc1csc(C(=O)NC(COC)CO)c1 15352,N1(C(COCC=C)=O)CCC(C)C(CNC(c2cccc(NC(=O)OC)c2)=O)C1 15353,N1(C(CCC=CC(C)C)=O)CCC(C)C1C(=O)NC(C1CCCC1)C 15354,C(C(=O)NC1CC(C)(NC(c2ccon2)=O)C1)(C(C)C)n1ncc(C)c1 15355,C1(C(=O)NCCOCCOC)CCOC1CNC(=O)CCNC(C)=O 15356,O=C(CC(CNC(C1CCC2CC12)=O)C1CCC1)NCC1(Cl)CCC1 15357,C1(CNC(=O)COCC2CCC2)CC(F)(F)CN1C(=O)CC12COCC(C1)C2 15358,c1(-c2cn(Cc3c(C(=O)NC(C)C(N)=O)cccc3)nn2)cnc2n1CCC2 15359,C1(=O)C(C(C)C)N1.C(CCC(=O)NCCN(C(=O)CC(C)C)CC)OCC 15360,c1(OCC)ccnc(N(C2CC2)Cc2ccnc(Oc3ccccc3F)c2)n1 15361,Nc1c(C(=O)NCC(=O)NC2CC2CNC(=O)Cc2cnns2)cccc1Cl 15362,Cc1cn2c(n1)C(C)CC(C(=O)N(CCCCNC(=O)C1=CCCC1C)C)C2 15363,c1(CN(C(CC2(N(C(C(C3CC3)SC)=O)C)CC2)=O)C)ccc(Cl)o1 15364,Cn1nc(C(=O)NC2CCOCC2C(=O)NCc2ncnn2C)cc1F 15365,N1(C(C=CCCCCC)=O)CCOC2(CCN(C(c3cccc(Br)c3Br)=O)C2)C1 15366,N1(ONC(c2nc(C(=O)OC)oc2)=O)CCn2c(cnc2-c2ccccc2)C1 15367,C(CC(C)C)(C(=O)N1CCCC(N(C)C(c2[nH]ccc2C)=O)CC1)NC(=O)OC 15368,c1(CC(=O)NCC(C2CCCC2)NC(c2cnccc2C(F)F)=O)c[nH]ccc1=O 15369,c1(CN(CCNC(c2n[nH]cc2Br)=O)C(C2CC2C(F)F)=O)ccccc1 15370,c1(NC(c2c(-c3c(C)csc3)cncn2)c2ccccc2)ccc2cc[nH]c2n1 15371,CC(C)(C)C(CCO)NC(C1(CCNC(=O)C2=COCCC2)CC1)=O 15372,Cc1ccc(CCCCC(=O)NCC(=O)NCC2CCSC2(C)C)cc1 15373,C1(CNC(c2c(C)nc(C)o2)=O)CC2CCC1N(C(c1ccnc(O)c1)=O)C2 15374,C1(NC(c2c(C)ocn2)=O)CN(C(c2cc(Cl)cn2C)=O)CC1C 15375,c1(C(=O)NC2CN(C(C3N(C)CCOC3)=O)CC2F)cccc2nn[nH]c12 15376,C1(=O)CCNCCN1CCC.C1(CC(C)C)(NCCOCC)CCC1.C(=O)N 15377,c1(OC)cccc(OC)c1NC(C1CSCCN1Cc1cccc(O)n1)=O 15378,c1(C(=O)NC2C3CCN(C(CCCCCC)=O)C32)cn(CCC)c2ccccc12 15379,C1(NC(C(CC)OC)=O)CCCCN(C(=O)C(O)CC2CCCC2)C1 15380,CC(C)(CNC(=O)CC1COCC1O)CC1CN(C(N)=O)C1.C1(=O)COCCN1 15381,c1(CNC(=O)CSc2n[nH]c(O)n2)ccc2c(c1)CN(C(=O)C1=CCSC1)C2 15382,C12(C(=O)NC34CC(NC(c5c(OC)cncn5)=O)(C3)C4)CC=CCN1CCC2 15383,N1(C(c2nc(CC)oc2C)=O)CCC(C)(C)C(NC(c2cc(C)nc(O)n2)=O)C1 15384,C1(NC(c2n[nH]cc2I)=O)C2CN(C(=O)Cc3cccc(O)c3)CC12 15385,c1(C(=O)NC(CC)CNC(C2CCCC2(C)C)=O)cccc2c[nH]nc12 15386,c1(C(=O)NCC=CC(=O)NC(CN(CCCC)C)C)cccc(C)c1N 15387,N1(C(c2c(C)cc(Br)o2)=O)CC(NC(C2CCNC2=O)=O)CC(C)(C)C1 15388,Cc1cccnc1-c1cn(CCCCNC(=O)C(O)C(C)C)nn1 15389,N1(C(CSCC)=O)CCC(CNC(C2CCC23CCC3)=O)C12CCC2 15390,C1(CC)(CC)SCCNC1C(=O)NCc1ccc(C(=O)OC)o1 15391,Cc1csc(C(=O)NC2CCC(NC(C3CSC3)=O)C2)c1Cl 15392,C12(NC(CCC3CC(NC(CC4C(C)(C)C4(C)C)=O)C3)=O)CC=CC(C1)OC2 15393,O=C1CC(C(=O)NCCOCCOCCNC(c2cncc(Br)c2)=O)C2(CCC2)C1 15394,CCCCC(CN(C)C(c1cc(CNC(C2(C#N)CC2(C)C)=O)ccn1)=O)CC 15395,n1(C(C(C)C)NC(c2n(C3(C)CC3)nnn2)c2ccco2)nc2ccccc2n1 15396,c1(C(CC)O)nc(C2CC3CC2C3)n(-c2cccc(F)c2)n1 15397,Cc1cc(S(=O)(=O)NCc2nc(C3CCCC3)no2)ccc1-c1cc2ccccc2s1 15398,C1(NC(C(C)(F)c2ccccc2)=O)CN(C(c2cnc(C(F)F)nc2)=O)CCC1F 15399,c1(CC)nc(C)ccc1NC(c1nnnn1CCOC)C1(CF)CC1 15400,CC1(C)CN(N2CCN(S(=O)(=O)NCCO)C2)CC1C1OCCO1 15401,C(c1ccncn1)=CC(=O)NC1(C)CC(NC(=O)CCC2CC2(F)F)C1 15402,C(=O)(CCCC(=O)NC(CN(C)C)C(N1CCCC(C#N)C1)=O)OC 15403,C1(C(=O)NCC(C2CCCCC2)NC(c2occ(C)c2)=O)CC2CCCC(C1)C2 15404,N1(C(=O)C(Cl)(Cl)Cl)CCC2(CC1)CN(S(=O)(=O)Cc1ccccc1Br)C2 15405,C1(F)(CNC(CC2N(CC)CCOC2)=O)CCN(C(=O)CN(C)S(N)(=O)=O)CC1 15406,c1(C(C(=O)NC(C(C)C)CNC(=O)Cc2ccc(Cl)s2)(C)C)ccnc(O)c1 15407,C(=O)(C(C)(C)C(C)(C)O)N(CC(C)C(=O)N1CCC(C(F)(F)F)C1)C 15408,Cc1ccc(C(=O)NC2CN(C(C3C4CCC(F)(F)C34)=O)C(C)(C)C2)c(N)c1F 15409,c1(C(N(C(C)CCNC(c2cccc(F)c2)=O)C)=O)ccc2[nH]ccc2n1 15410,C(=O)(C1CCC(=O)c2cccn21)N1CC(COC)(CNC(=O)C2=CC(C)(C)C2)C1 15411,c1(C(=O)NCc2c(CNC(C(C)n3cnnn3)=O)cccc2)ccc(Cl)nc1 15412,c1(OC)ccc(C(=O)Nc2ccc(C(N3CCCCC3C(N)=O)=O)cn2)cc1Cl 15413,N1(C(c2cn(CCC=C)nn2)=O)CC(NC(=O)C=Cc2cc[nH]n2)C(CCC)C1 15414,c1(OCC(C)C)ccccc1C(=O)N(C)CC1(NC(C2CCOCC2)=O)CC1 15415,C1(CNC(C2C(C(N)=O)C2)=O)CCC2(CCC2)CN1C(C1(C(F)(F)F)CC1)=O 15416,c1(C(=O)NC(C2CN(C(=O)C(C)(F)C(F)(F)F)CCO2)C)cc2n(c1)CCCC2 15417,C12(NC(=O)Cc3ncsc3Cl)CC1CN(C(c1cnn(CCNS)c1)=O)C2 15418,N1(C(C(CCC)O)=O)C(CNC(=O)CCCC(C)C)CC12CCC2 15419,C1(O)(CCC)CN(C(C2(CNC(=O)C(C)CC3CC3)CCC2)=O)C1 15420,c1(NCC2(OCC)CCOC2)ccnc(O)c1 15421,C1(C(N(CC(CC)NC(=O)CCSC)CC)=O)CCc2nc(C)ncc2C1 15422,Cc1nnc(N2CC3CC(NC(c4n[nH]cc4C(C)C)=O)C3C2)nc1C 15423,c1(CNC(CC2CCN(C(C3(CC=C)CC=CC3)=O)C2)=O)ccc(O)c([N+](=O)[O-])c1 15424,C(CCN=C(NCC1CCSC1)N1CCN(c2cccs2)CC1)OC 15425,N1(C(=O)NC2CCN(CC(C)(C)C)C2=O)CCC(F)(F)C2(CCOC2)C1 15426,CN=c1[nH]cc(C(=O)NCc2ccnc(N3CCN(C(=O)CNC=O)CC3)c2)o1 15427,CCCCCCCCCCCCC(=O)NC1CCC(NC(=O)CC(C)(C)CC)C1 15428,CN1CCC(C)(C(N2CC3(CNC(c4cc(N)nc(Cl)c4)=O)CC2CO3)=O)CC1 15429,Cc1cc(C(F)F)n2nc(C(N3CC4CC(C3)C4O)=O)cc2n1 15430,c1(-n2c(C3CCN(C(C)C4CC4)C3)nc(-c3ccco3)n2)ccccc1S(C)(=O)=O 15431,CCCC(C(=O)NCCCN(C(c1ccn2cccc2c1)=O)CC)C(C)C 15432,c1(C(=O)OCC)cc(CNC2CCN(c3cnn(C)c3)C2=O)oc1C 15433,CC1CN(C(C23CC4CC2C3C4)=O)CC(C)N(C(=O)COCC2CCCO2)C1 15434,Cc1cnc(C)c(C(=O)NCC2CCCN2C(=O)C(C2CCCCCC2)C)c1 15435,c1(C(=O)NCCn2cc(C(N(CC(C)O)CC)=O)nn2)cc(C)n(C)c1 15436,C(=O)(C(CN=[N+]=[N-])NC(=O)C(O)C1CCC1)N(c1ccccc1)CC(N)=O 15437,C(CCOCCO)(C(=O)NCC1(Cl)CC1(F)F)NC(C(N1CCNC1=O)C)=O 15438,N1(C(c2cc(OC)no2)=O)CC(C2CN(C(c3ccc(CC(C)C)cc3)=O)C2)C1 15439,N1(C(c2ccc(CCC)[nH]2)=O)CCC(C(F)CNC(c2ccccc2C)=O)CC1 15440,Cc1c(F)ccc(C(=O)NC(=O)CC2CCN(C(=O)CN3CCCCC3)C2)c1F 15441,C(=O)(C(O)CC(F)(F)F)NC1CN(C(c2cc3n(n2)CCO3)=O)CC12CC2 15442,c1(C(=O)NCC2(COC)CN(C(=O)C(O)C(F)(F)F)C2)ccc2oc(C)nc2c1 15443,N1(C(C(CNC(c2cn(CCC)nn2)=O)OC)=O)CCC(O)C(F)C1 15444,c1(C(N(CC(C)N(C(Cn2cccc(C)c2=O)=O)C)C)=O)cc(O)cc(C#N)c1 15445,C#CC1CCC(NC(C2(CNC(=O)C(OC)OC)CC(=C)C2)=O)C1 15446,c1(OCC)ccc(C)cc1C(=O)NCCC(C)NC(c1nncn1C1CC1)=O 15447,C1(NC(CCNC(c2c(C(C)C)cccc2)=O)=O)CC(F)CN(C(=O)CCF)C1 15448,S(=O)(=O)(c1cc(NC(=O)C(F)(F)F)ccc1O)NC(CC)C(N)=O 15449,c1(CC)sc(C(=O)NCC#CCNC(=O)C(c2ccc(Cl)cc2)C)cc1C 15450,N1(C(=O)NC(C)Cn2cnc(Br)n2)CC2CC3CC2C1C3 15451,c1(C(N(CCCCNC(C2(Cl)CC2(C)C)=O)C)=O)ccn2c1CCCC2 15452,C(CC(CNC(=O)CC1(CSC)CC1)NC(c1cc(Br)no1)=O)OC 15453,c1(N2C3CN(C4CCN(C)CC4)C(C3)C2)ncnc2c1ncn2CCCOC(F)F 15454,Cn1nc(C(N2CC=CC(NC(C3CN4CCC3CC4)=O)C2)=O)c2c1CCOC2 15455,c1(OCC)ccccc1C(=O)NC1CCN(C(=O)CCNC(C2CC2Cl)=O)CC1 15456,C1(C(=O)NCCn2nnnc2C2CC2)(NC(C2CCC(C)O2)=O)CCOCC1 15457,C1(CC)CCN(C(c2cccc(O)n2)=O)C1C(=O)NCC(F)(CC)CC 15458,C(=O)(C1=NOC2(CCOC2)C1)NC1C2CCN(C(c3c(N)non3)=O)C21 15459,c1(C(N2C(CC)(CC)CC(OC)C2)=O)cc2scc(Cl)c2[nH]1 15460,N1(C(C(C)C2CCCO2)=O)CC2(CCN2C(c2ccc(C(N)=O)c(Cl)c2)=O)C1 15461,CC(CNC(=O)CC(C)(C)O)C(F)C(=O)N(C)Cc1cccnc1O 15462,C1(C(=O)NCC(CCNC(c2ccc(CO)o2)=O)O)CN2CCCN1CC2 15463,C1(C(N2CCC(CNC(C3CC(O)(c4cccnc4)C3)=O)C2)=O)CC2CC1C2 15464,c1(N(C(=O)Cn2cc(C3CCCC3)nn2)C)ccccc1CNC(=O)CC#N 15465,N1(C(=O)Nc2ccc(OC(C)=O)nc2)CCOc2ccc(N(C)C)cc21 15466,c1(C(=O)NC(C2(O)CCCCC2)C(=O)NC2CC(F)(F)C2)ccc(Cl)cc1O 15467,C12(CCNC(C3N(C(=O)OC)CC3)=O)CCC1CN(C(c1cnccc1Cl)=O)C2 15468,Cc1oc(C)c(C(=O)NCCCOCCN(C)C(C2(c3cc[nH]n3)CC2)=O)c1C 15469,C(=O)(C1CCc2cccc(Cl)c21)N1CCC(NC(c2cc(Cl)cc(Cl)c2)=O)C(F)C1 15470,C1(C(=O)NCC2CCC2NC(c2cnc(C)cn2)=O)(CC)CCC(O)CC1 15471,N1(C(CC2CCCCN(CCC(=O)OCC)C2=O)=O)CC2COCC(C1)C(=O)N2 15472,C1(C)(C(=O)NCCCNC(CC(C)Cc2cccc(F)c2)=O)CCC(=O)NC1 15473,N1(C(CN(C(C(C)C)=O)C)=O)CC=CC(NC(=O)CC2CCC(C)(C)O2)C1 15474,C1(NC(c2cc(C(F)F)cs2)=O)CC(F)(CNC(C2C=CCC2)=O)C1 15475,C(=O)(C1=CCC2(COC2)OC1)NC(CC)CN(C)C(c1nc(Cl)cs1)=O 15476,C(=O)(CCS(C)(=O)=O)N(C(C)C)CCN(C)C(C1CCCCC1O)=O 15477,CC(C)(C(=O)N1C2CCC1COC2)C(F)c1ccccc1OC(F)(F)F 15478,C(c1ccccc1Cl)=CC(=O)NC1CN(C(C(C)(C)OCC)=O)CC1SC 15479,c1(CCC(=O)NC2OCCN(C(CNC(CC)=O)=O)C2)ccc2ncccc2c1 15480,CC1(C)CCC(C)(NC(=O)CC(CNC(c2cccnc2O)=O)C2CCC2)C1 15481,C1(NC(C(CC=CC)NC(=O)CC2CCC(=O)C2)=O)CC2CCC(C1)N2C 15482,CC1CCC=C1C(=O)NCC=CCC(=O)NOC(c1ccccn1)C 15483,C(=O)(CCC(=O)N(C)C(C)C)N1C(C(C)NC(=O)CCCc2cnn[nH]2)CCC1 15484,C(c1ccncn1)=CC(=O)NC(C)C(C)NC(c1cc(C2CCC2)no1)=O 15485,C(C(=O)NC1CCN(C(C2(F)CC=CC2)=O)C1)(C(C)C)OC 15486,c1(C(=O)NC(C)CCNS(C)(=O)=O)ccc2oc(O)nc2c1 15487,C(=O)(C(C)(O)C(C)(O)C(=O)NCC)N(CCOCCCNC(CSCCCC)=O)C 15488,c1(C(=O)NCC2CN(C(CC)=O)C3C(O2)COC3)cc2cccnc2cc1F 15489,Cc1ccc(C(=O)NC2(C(=O)NC3(C)CCSCC3)CCSC2)nc1O 15490,n1(C(C)C)cnc(C(N2CC(O)(C(F)C(=O)NCC3CCCCO3)C2)=O)n1 15491,C#Cc1cc(C(N2CCC(C3(NC(c4ncccn4)=O)CC3)C2)=O)ccc1Cl 15492,C(CCN(C(=O)C(C)n1ccnc1)C)(C(C)(C)C)NC(CCOCC(C)C)=O 15493,C(=O)(C(F)(F)CNC(C1CC(CNC(=O)CCN(C)CCO)C1)=O)OC 15494,N1(C(C(=O)Nc2c(O)ccc(C(C)=O)c2)=O)CCCN(C)CC1(C)C 15495,c1(COC)cc(CNC(c2ccoc2CNC(C2(C(C)C)CC2)=O)=O)no1 15496,c1(C(=O)NC2C(NC(CSc3nc(C)[nH]n3)=O)CCCC2)ccc2nccn2n1 15497,CC1(C(=O)NCc2ccc(C#N)s2)CCCN(C(=O)CCc2ccc(O)cc2)C1 15498,C1(CC)C(NC(=O)C(C)(C)n2cc(Cl)cn2)CCCN1C(=O)C(C)COC 15499,N1(C(c2cnc(C)s2)C(=O)NCCC)CCCC(c2ccc(Cl)nc2)C1 15500,CC1(O)CCCN(C(C2(NC(=O)CSc3cn[nH]c3)CCOCC2)=O)C1 15501,C#Cc1ccc(C(=O)NC2C3CC2N(C(=O)Cn2nnc(=N)[nH]2)C3)nc1 15502,c1(C(=O)NC2CC(CCNC(COC)=O)C2)cc(Br)c(OC)cc1C 15503,c1(N2CCC(c3cccc(C)c3)CC2)ccncc1S(=O)(=O)N1CCC=C(Br)C1 15504,N1(C(C(C=CCCC)O)=O)CCN(CCNC(=O)C(C#N)CC)CC1 15505,c1(C(=O)NC2(CNC(=O)COCCF)CC2)ccc(C(F)F)cc1Cl 15506,C1(NC(c2ccnc(C(C)C)n2)c2nnnn2CCCF)CCC2(CCC2)CC1 15507,CC1(C)CCN(C(=O)C2=CCCSC2)C1CC(N1CCC(CCCO)CC1)=O 15508,C12(CC)COC(C(=O)NC(CNC(=O)CCCc3cccc(Cl)c3)C(C)C)(C1)C2 15509,C1(NC(C2CC(=C)C2)=O)CN(C(=O)C(C)(C)Oc2cccc(F)c2)C2CC12 15510,CCCC(C(O)C(=O)N1CCCC(CCO)C1)NC(C1CCCCO1)=O 15511,N1(C(C2CC(NC(=O)Cn3cc(Cl)cn3)C23CCC3)=O)CCC(F)(F)C(F)C1 15512,c1(N2CC(N(C(C)C)CC)C2)ccc(S(=O)(=O)NC(C)C(CO)N(C)C)cc1Br 15513,O=C(C1=NOC2(CCN(Cc3c(Cl)cccc3Cl)C2)C1)NCc1nc(C2CC2)no1 15514,CCC(C)CC(CO)NC(c1nnc(CSc2cccc(C#N)c2)s1)=O 15515,C(=O)(C(Cc1ccccc1)C(F)(F)F)N1C(N(C(=O)CS(N)(=O)=O)CC)CCCC1 15516,CC(N)CCCC(=O)N1CCC(c2ccc(F)cc2F)C1C.c12cn(nn1)CC2 15517,Cc1cc(CN2CCC(=O)N(C(=O)NC3CC4(CNC(=O)N4)C3)C2=O)c(C)cc1Cl 15518,c1(-n2c(C(CCOC)NC(CCC)C(C)C)nnn2)c(C)cccc1C 15519,N1(C(C(C)NC(C)=O)=O)CC2CN(C(=O)Cc3ccnc(C)c3)CC12 15520,CC(C)C(C#N)C(=O)N(C1CCN(C(=O)C(C)(C)c2ccncc2)C1)C 15521,C1(O)(C(N2CCN(C(=O)CSc3ccc(Cl)c(F)c3)CC2)=O)CN2CCC1CC2 15522,c1(C(=O)NCCCCNC(CSCCOC)=O)ccc(F)c(Cl)c1 15523,N1(C(CSCC(N)=O)=O)CCC2C(C1)CN2C(=O)C(=Cc1c[nH]cn1)F 15524,Cn1nc(C(=O)NCC2C(C(=O)NCC3(F)CC3)C2(C)C)cc1CO 15525,Cc1cnc(C(=O)NCC(C)(C)CN(C(=O)CC2COCC(C)O2)C)cc1C 15526,C1(C(=O)N(C)Cc2cccc(C)n2)(COC)C=CCN1C(c1scc(C)c1C)=O 15527,c1(N2CCC(CNC(=O)C(c3ccc(F)cc3)F)C2)ncnc(O)c1Br 15528,C1(NC(c2n(C(CC)(C)C)nnn2)c2cnns2)(OC)CCCCCCC1 15529,CC1OC(=O)NC1C(=O)NCC(C)(C)CCNC(=O)Cn1cnc(C(F)(F)F)n1 15530,C=CC(C)C(C)C(=O)NCC(C)(C)CNC(=O)CC1(CC(=O)OC)CCCC1 15531,C=C(F)C1(CC(=O)NC2CCCC(NC(C3(C(C)C)CCCO3)=O)C2)CCC1 15532,Cc1noc(C(F)F)c1C(=O)NCCC1CCCN(c2ncc(F)cn2)C1 15533,C1(CC)CN(CCc2cc(-c3ccco3)on2)CCO1 15534,c1(N(C)C)ccc(CCC(=O)NCC2(C(=O)NCc3ccns3)CCC2)cc1 15535,O(N1CCC(NC(=O)N(C)CCO)CC1)CC 15536,N1(C(COC)=O)CC(F)(F)CC1CCNC(=O)CN1CCCCC1 15537,c1(C(=O)NCC(CC)NC(c2ccc(=N)[nH]c2Cl)=O)cccc2c1C(=O)NC2 15538,C#Cc1cncc(NC(C2CNC(=O)CN2C(=O)C2=COCC2)=O)c1 15539,C1(CNC(CCN(CCC)C)=O)CCC2(CN(C(c3cc(N)cnc3C)=O)C2)O1 15540,S(=O)(=O)(c1ccc(N2CCSCC2)c(C#N)c1)N(C1CC(F)C1)C 15541,c1(C(N2CCC(C(C)(C)NC(CC3CC(C)C3)=O)C2)=O)c(O)cccc1Cl 15542,C1(C)(C(=O)NCC(C)N(C(c2c[nH]nc2C2CC2)=O)CC)CCC(C)C1 15543,C1(CC(=O)NCC23CC(NC(C(c4cscn4)N(C)C)=O)(C2)C3)CC(O)C12CCC2 15544,c1(C(=O)NCCNC(C(N(C)C)C2CC2)=O)scc2c1OCCO2.C(C)(C)(C)O 15545,c1(OC)ccc(-n2nc(Cc3nc[nH]n3)nc2COC(F)F)cc1 15546,c1(Nc2ncnc(NCC(CC(CC)C)C)c2C)noc2c1CCCC2 15547,N1(C(c2cc(C(F)(F)F)cs2)=O)CCCC(C2CC2NC(C2(CC3CC3)CC2)=O)C1 15548,CCC(C)(C)C(O)C(=O)NC1CC(C)CN(C(=O)C(C)(CO)OC)C1 15549,c1(CC)ccc2nc(C)[nH]c2c1.C12CC3C(C3C1)NC(=O)C1CC1C(=O)N2 15550,c1(CNC(C2(CC#N)CC2)=O)ccc(CNC(=O)CC2CNC(=O)N2)cc1 15551,N1(C(CC(C=C)C)=O)CCCC(NC(c2ccc(C(F)(F)F)cc2N)=O)CC1 15552,C1(C(=O)NCc2cc(C(=O)N(C(C)C(C)C)C)on2)(COC)CCCO1 15553,CCCC(C)(CO)NC(c1cc(CNC(C2CN(C(C)C)C2)=O)ccn1)=O 15554,C#CCCCC(=O)NCC1C=CC(NC(c2ncsc2-c2ccccn2)=O)C1 15555,CCCC(F)C(=O)NCc1cccc(CNC(=O)C(F)CC)c1 15556,c1(C(=O)NC2CN(C(C#CC(=O)N(C)C)=O)CC2F)noc2c1CC(C)CC2 15557,CC1CCCC(O)(C(=O)NCCCCN(C(=O)COc2cnc(Cl)cn2)C)CC1 15558,Cc1nccnc1C(N1CCC2CC12C(=O)Nc1cnc(C#N)s1)=O 15559,C(=O)(CCCCC(C)(C)OC)N1C(C(C)(C)NC(CCC=CCC=C)=O)CCC1 15560,Cc1cc(C(=O)NCCCN(C(=O)CC2CC2)C)nn1C(C)C1CC1 15561,CC1CCCCC1(CNC(=O)CCC1(C)CCC(=O)N1)NC(c1cnco1)=O 15562,c1(N2CCN(CC(=O)NC(COC)C)C(=O)C2)ccnc2cc(Br)nn12 15563,CCCC(CCCNC(=O)CCCOC)NC(c1cc(F)ccc1N)=O 15564,c1(C(N2CCN(C)CC2CNC(C2CN(C)CCO2)=O)=O)n[nH]c2cccnc12 15565,C1(CC(=O)NCCCC(C)NC(c2c(C)nsc2C)=O)CCCNC(=O)C1 15566,C1(C(=O)NCC2CCCCN2C(c2ccc(F)c(Cl)c2)=O)CC2(CCC2)CCO1 15567,O=S(=O)(c1c[nH]c2cc(Cl)ccc12)N1CC(O)(c2cccnc2)C1 15568,C=C(C)CCC(C)(c1nnnn1Cc1ccccc1)NC(c1ccc(Br)cc1)C 15569,N1(C(C=CSC)=O)CC2CCC1C(CNC(C1CCN(C3CCCCC3)C1)=O)C2 15570,Cn1ccnc1SCCC(=O)NC1CC1NC(=O)CSCC1CC1c1cccs1 15571,C1(NC(C(CO)NC(C(CC#C)O)=O)=O)CCC(N=[N+]=[N-])CC1 15572,N1(C(CCc2ccc(OC)nc2)=O)CC(CNC(=O)Cc2nc[nH]n2)CC1(C)C 15573,C1(C(=O)NCC(CC)(C)O)CNCC(F)C1 15574,CC1CCCC=C1C(=O)NC1CC12CC(NC(=O)COC1CCOC1(C)C)C2 15575,c1(C(C(=O)N(CC(C)NC(=O)Cc2ccc(Cl)s2)C)CO)ccc(F)cc1 15576,C1(CC=C)(NC(=O)CN2CCCCC2C)CCN(C(c2cnn(CC)c2C)=O)C1 15577,C=C1CCN(C(=O)C(C)OCCC(C)C)C(C(=O)NCCC2CCN(C)C2)C1 15578,N1(C(COCCOC)=O)CCC2(C)CN(C(=O)CNC(=O)C(C)C)CC12 15579,CCCCC(C(=O)NCC(C)(C)C#CC(=O)NC1CC(CCF)C1)C(C)C 15580,C1(NC(=O)C(F)=C2CCC2)COC2CN(C(=O)CC3=CCCCC3)CC12 15581,C1(C(=O)NC2(C)CN(CCOC)C2)CCCCC1NC(=O)Cc1cccnc1O 15582,C(=O)(C(O)CCC)NC(c1ccnn1C)C(N1CCC(=C)C1)=O 15583,CC(C)C(C(=O)NCC1(C(=O)NC2CCOC2(C)C)CCCO1)NC=O 15584,c1(OC)cc(C(=O)NC(C)CCCCNC(C2CCC3(CC3)C2)=O)cc(OC)n1 15585,C#CCC(C(=O)N(C(CO)CC(C)C)C)NC(c1cnc(CC)nc1)=O 15586,c1(N(CCCNC(c2[nH]nnc2C2CC2)=O)C)nccc(CO)n1 15587,C#Cc1ccc(C(=O)NC2(CC(N3CCC(O)(CN(C)C)C3)=O)CC2)o1 15588,C=C(F)C1(CC(=O)NCC(C)NC(=O)CCCC(=O)OC(C)(C)C)CCOCC1 15589,n1(CC)cc(CC(N2CC(O)(CC(=O)NOC(C)CC(=O)OCC)C2)=O)nn1 15590,C=CCC(CC(=O)OC)NC(=O)Cn1nc(C)oc1=O.N12CCC(C1)C2=O 15591,C1(CNC(C(CO)NC(N)=O)=O)CN(C(=O)CN2CCS(=O)(=O)CC2)CCCO1 15592,c1(C(=O)NCCNC(c2c(C)nsc2)=O)c(Cl)cc(F)cc1Br 15593,c1(C(=O)NC2CC2C(=O)Nc2ncc(Cl)cc2Br)c(F)cc(Br)cc1Br 15594,C1(C)(C(=O)NCCN(C(c2cc(CC)c(C)s2)=O)C2CC2)CCC(=O)N(C)C1 15595,CC(C)C(CCO)N=c1ccnc(NC2CNC(=O)C2)[nH]1 15596,C1(CC(=O)NCC2(C(=O)OC)CCC2)CCN(C(=O)C(C)O)CC1 15597,C(CCCCC(=O)N1CCC(C(=O)Nc2cccc(F)c2O)C(O)C1)OCC 15598,C1(C(=O)NCC(C)(C)OCCNC(CCC(=O)OCC)=O)CC12CCCOC2 15599,N1(C(c2c(C(C)(C)C)nns2)=O)CC(NCc2cc(=O)cc[nH]2)C(O)C1 15600,c1(OC)cc(=NC(=O)CC2CN(C(C3(C(N)=O)CCC3)=O)CCC2C)[nH]n1C 15601,N1(C(CC(CC)CN(C)C)=O)CCCC12CCN(C(c1cnc(O)n(C)c1=O)=O)C2 15602,c1(C(CC)=O)ccc(NCC2CCN(C(C3CCOCC3(C)C)=O)C2)c([N+](=O)[O-])c1 15603,CC(CNC(=O)C(C(C)O)N(C)C)C(F)C(=O)NCCCC1CC1C 15604,C(=O)(C(CCCCCN)C(F)(F)F)NC1CC2(CC(C(=O)OC)C2)C1 15605,C1(CNC(C(CC)F)=O)CC(OC)CN1C(=O)C(C1(O)CCCC1)F 15606,N1(C2CCN(CC(C3C4(CCC4)C34CCC4)=O)C2=O)CCC(F)(F)C(O)C1 15607,c1(C(=O)NC(CNC(Cc2c(C)scc2)=O)C2CCC2)cc2cnccc2[nH]1 15608,C(=O)(CCC1=NNC(=O)CC1)NCC(CNC(C1(C)C=CCCC1)=O)C(F)(F)F 15609,C(CC(F)F)(C(=O)NC1C(O)CC1O)N(C)C(C1CCC1)=O 15610,CCC(CNC(C1CC(C)CCN1C(=O)CSCC(N)=O)=O)(CC)CO 15611,C1(C)(C(=O)NC2C(CC(=O)NCCC(C=C)(C)C)CCCC2)CCC2CC2C1 15612,C12(CC(=O)NCC(F)CO)CCC1CN(C(c1cc(CO)on1)=O)C2 15613,Cc1cc(=NCc2csc(Br)n2)[nH]c(=NCc2cc(C)on2)[nH]1 15614,Cc1ccc(C(=O)NC2COCC2NC(c2snnc2C(C)C)=O)c(Cl)c1 15615,c1(C(=O)NCC(CNC(c2cc(C(C)C)on2)=O)O)cccc2c[nH]nc12 15616,Cc1ncsc1C=CC(=O)NCC1(NC(=O)CS(=O)(=O)NC(C)(C)C)CC=CC1 15617,C1(CC(=O)NC2C3CC(NC(=O)CCc4cscn4)CC32)CN2CCC1CC2 15618,c1(C(=O)NC2C(OC)CN(C(c3cnn(C(F)F)c3)=O)C2)ccc2cc[nH]c2n1 15619,C1(C(N2CC=CC(NC(=O)CC3CC(=O)NC3=O)C2)=O)(COC)CCC(=O)N1 15620,C1(CCNC(C2C3CCC23)=O)COCCN1C(=O)CNc1cccnn1 15621,c1(CN2CCC(O)(CNC(c3c(OC)nccc3)=O)C2)c(F)ccc(F)c1O 15622,C1(NC(C2(OC)CC2)=O)C2CN(C(C3CCCN3Cc3cccnc3)=O)CC12 15623,c1(OC)c[nH]c(C(=O)NC(C)CCCCNC(=O)C(F)n2cccn2)cc1=O 15624,N1(C(CN(CC)CC2CCCC3CCCC23)=O)CCOc2ccccc21 15625,N1(C(Cc2nc(C)sc2)=O)CC(NC(c2ccsc2)=O)C2CC2C1 15626,C1(C(N2CC3C(C)(C)C3C2)=O)CC2C=CC1N(C(c1cccc[n+]1[O-])=O)C2 15627,C1(NC(=O)CCc2ccc[nH]2)CCC(NC(C2(C(F)(F)F)CCC2)=O)C1 15628,N1(C(C2(CC)CCOCC2)=O)CC2CC(NC(c3cn(C)cn3)=O)CC2C1 15629,Cc1ccc2ncc(C(N3CCC4CCN(C(C5CCC5)=O)C4C3)=O)cc2c1 15630,c1(C(=O)NC2(CC(=O)Nc3cncc(C(C)=O)c3)CCC2)c(C)cc(F)cc1Br 15631,CC1CN(Cc2ccncc2Cl)CCC1OC(C1CCCN(C(C)(C)C)C1)=O 15632,N1(C(C(C2(O)CN(C(c3cccnc3O)=O)C2)F)=O)CC2C(C1)C2(F)F 15633,N1(C(CC2(C=C)CC2)=O)CC(C)CN(C(c2cc3c(nn2)CCC3)=O)C(C)C1 15634,N1(C(C2CC(CCCC#N)OC2)=O)C(C(=O)NOCCCCF)CCC1C1CC1 15635,C#CC1(C(=O)NC(CNC(=O)CC2CCOC2)CCC)CCCCC1 15636,C1(NC(C(F)=CC)=O)CC2CCC1CN(C(c1cc(C(F)(F)F)ccc1C)=O)C2 15637,c1(C(=O)N)c(S(C)(=O)=O)cnn1C.C1(C)(C(C)(C)C)CCCC1NC(C1CC1F)=O 15638,CS(=O)(=O)CC(=O)NC(C(=O)N1CC(CC(F)F)C1)C1CC1 15639,CC(CCCCCO)NC(c1nnnn1C(C)(C)C)C1(C#N)CCC1 15640,c1(C(=O)NC2C(OCC)CC2)cnn(CCNC(C2COCO2)=O)c1 15641,Cc1cnccc1CNC(C1(NC(=O)C(C(C)C)NC(N)=O)CCCC1)=O 15642,Cc1cnccc1C(C)C(=O)NCC(C)(C)CN(C)C(c1[nH]nnc1C1CC1)=O 15643,C1(NC(C2COCCO2)=O)CN(C(c2ccc(-n3ccnn3)cc2)=O)CC1(F)F 15644,N1(C(C(CO)NC(C)=O)=O)CC(N(C(=O)Cc2cccc(Cl)c2)C)C(C)(C)C1 15645,CN1CC=C(CC(=O)NCC2(O)CCN(C(c3cccc4ccnn34)=O)C2)CC1 15646,C(=O)(CCCCC(=O)OC)NCC1CCC(NC(C(CCOC)OC)=O)C1 15647,CCCCC(COC)OC(=O)CNC1(CC2CCCC2)CCOC1 15648,C1(NC(c2nc(C(C)C)sc2)=O)COCCN(C(=O)CC2CCC3(CC2)CC3)C1 15649,c1(C(=O)NCC2N(C(=O)C3=CCCSC3)CCC(C)C2)cnc2ccoc2c1 15650,C1(C(=O)NCC2CCOC2Cc2ccccc2)CCCC1CCCl.C12(CC1)C(=O)N2 15651,N1(C(C(C)CO)=O)CCOC2(CCCN(C(C3(C#N)CCC3)=O)C2)C1 15652,N1(C(c2c(COC)scc2)=O)CCC=C(CNC(C2CCCCC2OC)=O)C1 15653,C1(CNC(c2cc(CNC(CCCC)=O)on2)=O)CCCCCC1 15654,C1(CC)CN(C(c2cc(C(C)(C)C)c[nH]2)=O)CCN1C(C1COCC1C)=O 15655,Cc1nnc2n1CCCC2C(=O)N(CCNC(=O)Cc1cnccn1)C(C)C 15656,c1(C(=O)NC2C3CN(C(c4cnc(C)nc4)=O)C(C3)C2)ccc2c(c1)CCC=C2 15657,c1(C(=O)NCC(CNC(=O)CO)OC)cnn(-c2ccccc2Cl)c1C(F)(F)F 15658,C(=O)(C(C)(C)C)N(CCn1cc(C2CC(C)CO2)nn1)CCSC 15659,Cc1cc(C(=O)NCc2ncc(C(=O)NC3CC4CCC3C4)cn2)cnn1 15660,Cc1cn(C)c(C(=O)N(c2ccccc2C)CC=CCN2C(C)CCC2C)n1 15661,C(=O)(CCC(CF)CF)N1CC2C(CCNC(c3cc(COC)sc3)=O)(CC2)C1 15662,c1(CCC)nc(C)c(C(=O)N(CCNc2ncc(N(C)C)cn2)CC)s1 15663,c1(CC(=O)NC2C(CC(C)(C)C)CN(C(C3CCCS3)=O)C2)ccc(Cl)cc1F 15664,c1(C(=O)NCCN)cnc2[nH]c(C)nc2c1.Cc1ccc(CO)cc1.C12(CC1)C(=O)N2 15665,C(CCN=c1[nH]c(=NCC(C)C2CCC2)[nH]c2c1CSC2)SCc1ccccc1 15666,C1CCC(C(=O)N)N(C)CCOC(CC)C(=O)N1.CCCOCC1CC1.C(CC)OC 15667,CC1CC(NC(C2CN(S(C)(=O)=O)C2)=O)CN(C(=O)C(N2CCCC(C)C2)=O)C1 15668,c1(C(=O)NCC2(F)CCC(NC(CCC(C)OCC)=O)C2)cnc(C)nc1CC 15669,N1(C(CCC2C(C)(C)C2)=O)CC2CCCC2(CNC(=O)CCOC(C)=O)C1 15670,c1(CC(N2CC(NC(=O)C=Cc3cnc[nH]3)C2)=O)ccc([N+](=O)[O-])cc1 15671,C12(SCCNC(=O)C(C3CCCCC3)O)COC(CF)(C1)C2 15672,C1(NC(COCP(C)(C)=O)=O)CCCN(C(=O)Cn2nc(C3CC3)cc2C(F)F)C1 15673,c1(C(=O)NCc2c(CNC(C(C)CC3CCC3)=O)cccc2)ccc([N+](=O)[O-])s1 15674,C(=O)(C(O)C(F)F)N1CCC(CN(C(COCCOCC#C)=O)C)C1 15675,c1(C(=O)NC(C(C)NC(C2N(CC)CCC2)=O)CO)cc(Cl)cc2c1NCCC2 15676,N1(Cc2ccc(-c3cc(C#N)c(O)nc3N)s2)CC(F)(F)Oc2cccc(F)c21 15677,C1(C(=O)NC(C2CCCC2)CC)CSCCN1C(=O)CCC1CCCC1 15678,N1(C(c2c(C)cco2)=O)CC2(CC(NC(=O)C(F)C3CCC3)CO2)C1 15679,C1(C(N2C(C)(CNC(CSCCC)=O)CCC2)=O)COCC(C)(C)O1 15680,c1(C(=O)NC(C(CC)CC)C)n[nH]c2c1CN(C(C1(F)CC=CCC1)=O)C2 15681,N1(C(c2cnc(CNC(C3(C)CCCC3)=O)nc2)=O)CC2CCCC(O)C2C1 15682,Cc1cnc(Br)cc1NC(C1C2CC1N(C(c1cccc(I)c1C)=O)C2)=O 15683,N1(C(C2(SCC)CC2)=O)CC(NC(=O)C=C(C)c2ccsc2)C(O)C1 15684,C12(CNCCCC3C(Cl)(Cl)C3)CCCN(CC1)C2 15685,C1(CC(=O)N(CCCNC(C(CCC)O)=O)C2CC2)OCCCC1(C)C 15686,C1(O)(CCNC(c2nn(C)c(F)c2)=O)CCN(C(c2cnsn2)=O)CC1 15687,N1(C(CCC(=C)Cl)=O)CC(NC(c2cnn(C3CCC3)c2C)=O)CCC1C 15688,c1(NCS(C(COC)C)(=O)=O)[nH]c(=NCC2OCCc3ccccc32)nc2c1cnn2C 15689,c1(CNCCC(c2cccnc2)C)cccnc1-c1cccnc1 15690,N1(N2CC(N)CC(OC)C2)c2ccccc2C(C)(C)C1C 15691,C(C(C)(C)NC(=O)CCn1ccnn1)N(C(=O)COCCN(C)C)C 15692,N1(C(c2n(C)nnc2)=O)CCOC(C(=O)NC2COC3(CCC3)C2)CC1 15693,N1(C(C2C(CCC)C2)=O)CCC2(C(=O)NCC(N3CCOCC3)C)CCCC12 15694,c1(C(N2CCCC(C(C)NC(=O)C(SC)NC(N)=O)C2)=O)cncc2c1CCC2 15695,c1(NC(C2N(C(=O)NCC(=O)OCC)C3CC2C3)=O)cccc(Cl)c1C.OCC 15696,CC1CCCC1(C(=O)Nc1ccccc1)NC(=O)Cc1cncnc1 15697,CCC(CC)(CCNC(C1(SC)CCC1)=O)NC(C1CCCN1C(C)C)=O 15698,C1(CN(C(C)=O)C)COCCN1C(=O)CC1CC1C(F)(F)F 15699,Cc1[nH]nc2c1CCC(C(N1CCC(C)(CNC(c3c(Cl)n[nH]c3C)=O)C1)=O)C2 15700,Cc1cc(F)c(F)cc1C(=O)NC1CN(Cc2ccc(F)c(O)c2)CC1F 15701,Cc1cc(=N)[nH]cc1C(=O)NCC1(CNC(=O)C(O)CC(N)=O)CCC1 15702,C1(NC(CN2CCCC(OC)C2)=O)CCN(C(=O)CC2CCC(C)CC2)C(C)C1 15703,CCCCCCCCC(=O)NCC(C)(CC(C)C)NC(=O)CSCc1ccncc1 15704,c1(C(=O)NCC(CNC(=O)C(C2CCC2)C2CCC2)O)ccc2c[nH]nc2c1 15705,C1(C(N)=O)CCN(NC(=O)c2ccc3nnc(-c4cccc(Br)c4)n3c2)CC1 15706,c1(CNCC2CC(NC(C#C)=O)C2)ccc(Br)cc1C#N 15707,c1(OC)ccc(C)c(CNC(C2CC(NC(c3cnc(Br)n3C)=O)C2)=O)c1 15708,c1(C(=O)NCC2(NC(c3c(C#C)c[nH]n3)=O)CCCCC2)cc(C)ccc1O 15709,CCC(CC(=O)NCC(C)N(C(=O)CCCc1cncs1)CC)C(C)(C)C 15710,Nc1cnc(C(=O)NCc2nocc2C(=O)NCCCOC2CCC2)cn1 15711,S(=O)(=O)(c1cncc(Br)c1)N(CC)Cc1cccc(C2CC2)c1F 15712,C1(O)(C(C)NC(c2cn(C3CCC3)nn2)=O)CCN(C(C2(F)CCC2)=O)C1 15713,C1(C(=O)NCC(C)CC2CC2)CC(N=[N+]=[N-])CN1C(=O)CC(C)(C)C#N 15714,c1(CC)cnn2c1CN(C(=O)CCc1c[nH]c3c(C)cccc13)CC2 15715,c1(OC)cc(CCC(=O)NC23CC(NC(c4ccc[nH]4)=O)(C2)C3)ccc1O 15716,c1(OC)cccc(C(=O)NC2CCC(CNC(C3(OC)CN(C(C)=O)C3)=O)C2)c1 15717,CC(C)C(C)CN(C(C(=O)NCCNC(=O)OC(C)(C)C)C1CC1(C)C)C 15718,C12(C(N3CCC(CCC(c4ccccc4)O)C3)=O)CC1CN(C(C)C(=O)OC)C2.CO 15719,C1(c2cn(C3CC(NCCNC(c4nsnc4O)=O)C3)nn2)CCCCCC1 15720,C1(C(C(=O)NC2CCC2)N(C2CCCOC2)C)CCC2CC2C1 15721,C(=O)(C1CCCc2ncnn21)NCC1(OC)N(C(c2c[nH]c(=NCC)s2)=O)CCC1 15722,N1(CC)CC(C(=O)NCC2(C)CCCN2C(C2CC3C=CC2C3)=O)CC1=O 15723,CC(C)CC(C)(O)C(=O)NCC12CCC(CC1)N2C(C1CC1F)=O 15724,C(CC(F)=C(F)F)NC(C1(COCC)CN(C(CCC=CC)=O)C1)=O 15725,c1(OC)cccc2c1C(C(=O)NCC(C)NC(c1coc(CO)c1)=O)CC2 15726,c1(OC)nsc(Sc2nnc(C(C)C)n2CC(C)C)c1Br 15727,C1(CC=C)(NC(C2CC(OC)C2)=O)CCCN(C(c2cnccc2C)=O)C1 15728,N1(C(c2cccc(CC)n2)=O)CC2CN(C(=O)Cc3cc(O)nnc3O)CCC12 15729,N1(C(CC(=O)OC)=O)CCCCC1C1CCCN1C(c1cnn(C)c1)=O 15730,c1(CN=C(NC(C=C)C)NC2CCc3ncsc3C2)cc2c(cc1Br)CCO2 15731,Cc1ccc(C(C)CC(=O)NC23CC(NC(c4cncc(N)n4)=O)(C2)C3)cc1 15732,C1(C(=O)NC2C(NC(c3c(C)nn[nH]3)=O)CC2)CCCC2(CC2)C1 15733,C1(C(=O)NCC2(NC(CC3CC(OC)C3)=O)CCOC2)CC2CC1CC2O 15734,c1(C(=O)NCC23C(CN(C(C4C(=C)CC4)=O)C2)C3)c[nH]c2cc(F)c(F)cc12 15735,c1(CO)ccc(C(=O)NCCC(CNC(Cc2cn(CC)nc2)=O)O)nc1 15736,c1(NC(C2C(C)CCN(C(=O)COCC(F)F)C2)=O)ccc([N+](=O)[O-])cc1I 15737,c1(C(N2CC3(C2)CN(C(=O)C(c2ccccc2)C2CC2)C3)=O)cc(Cl)nnc1Cl 15738,C1(C(=O)NC(C(C)C)(C)CNC(c2ccn(C3CCC3)n2)=O)CCCCCCC1 15739,C(=O)(C1=CNS(=O)(=O)N=C1C)NCC(CC)N(C(CNC(=O)OCC)=O)C 15740,c1(C(=O)OCc2cncnc2)ccc(OS(=O)(=O)Cc2ccc(Br)cc2)cc1 15741,N1(C(C2OCC(C)C2)=O)CCOCC(CNC(=O)CC2NC(=O)NC2=O)C1 15742,C(=O)(C1=CNC2=NCCC2=C1)N1CC(O)(CCNC(=O)CC2CCCCCO2)C1 15743,C1(NC(C(C)Oc2ccc(C#N)cc2)=O)CC2CN(C(=O)C(Cl)=CCl)CC2C1 15744,CC(c1cccs1)=CC(=O)NC(C)CC(C)NC(=O)Cc1nc(C2CC2)cs1 15745,c1(CC)cnc(CC(=O)N(C(C)CN(C)C(c2cc(C)c[nH]2)=O)C)[nH]1 15746,CC(C)CC(C(=O)NCC(C)(C)CCNC(C1(C#N)CCCO1)=O)C(C)C 15747,C1(CC(=O)NCC=CCNC(C2CC3OC(=O)OC3C2)=O)CCc2sccc2C1=O 15748,C(=O)(CC=C(Cl)Cl)NCC(CCC)NC(=O)CCc1cnn(C)c1C 15749,c1(C(=O)OC)cnn2c(NCCC(C)NC(=O)CNc3nccs3)cc(C)nc12 15750,N1(C(C(C)=CC)=O)CCC(NC(=O)CC(O)c2ccccc2)C1(C)C 15751,c1(CN2CCC(O)(C(=O)Nc3cnsc3)C2)cc([N+](=O)[O-])c(O)cc1F 15752,N1(C(c2c(F)ccc(C#C)c2)=O)CC2ON=C(CNC(=O)C=CCF)C2C1 15753,c1(OCC)ncnc(OC)c1C(=O)NC1CCC(NC(=O)C(O)P(C)(C)=O)C1 15754,n1(CC)nc(C2CC2)cc1C(=O)NC1CN(C(=O)COC(C)=O)CC1CC 15755,C1(S(N)(=O)=O)(C(=O)NCC2N(c3ccnc(C(C)C)n3)CC3(CC3)C2)CCCC1 15756,C1(C(=O)NC2CN(C(c3n[nH]c(C)c3Cl)=O)CC23CC3)CCc2cnnn2C1 15757,CC1(Nc2ccncc2Oc2ccccc2)CCCN1C(C1CC(=O)N1)=O 15758,C=CCC(C(=O)NC(C)CN(C)CCOC1CCCCCC1)C(C)C 15759,c1(CC(=O)NC2(C)CC(NC(c3coc(C(N)=O)c3)=O)C2)ccc(CC(N)=O)cc1 15760,C(=O)(C1COc2ccc(F)cc21)N1CC(CNC(C2(C(F)(F)F)CC(=C)C2)=O)C1 15761,c1(CC(N2C(CNC(C3C4CCCCCC34)=O)CC2)=O)cnn2c1OCCC2 15762,c12ccc3nc(sc3c1)c1cn2nn1.C1(C)(NC(C2(SC)CC2)=O)CCOC1=O 15763,c1(CSCC)ccc(C(=O)NC(C2CN(C(=O)C(F)CC)C2)(C)C)cc1 15764,c1(C(N2CC3CC2CO3)=O)cc2n(n1)CCCN(Cc1cc(F)c(Cl)c(F)c1)C2 15765,N1(C(C2(C=C)CC2)=O)CCC(C2(CNC(C3CCC(=O)N3)=O)CCOCC2)CC1 15766,c1(C(N2C(C(N(CC)Cc3ccncc3)=O)CC(O)C2)=O)cc(F)c(O)cc1F 15767,C=C(C)C1OCCC1C(=O)NCCN(C1CCCC1)C(=O)Cc1ccc[nH]1 15768,c1(OC)ccc(OC)c(C=CC(=O)NCC2CCC2NC(c2ccn(C)c2)=O)c1 15769,c1(OCC)cccc(C(=O)NCC2(O)CC(Cc3cn(C(C)C)nn3)C2)c1 15770,CC(C)C(CNC(c1cn(CC2CC(CF)C2)nn1)=O)NC(C1CC12CCC2)=O 15771,c1(C(=O)NC(C2CCCCN2C(C2CCC(C)(C)O2)=O)C)ccc2ncsc2c1 15772,C1(C(N2C(CNC(c3c(C)cn(C)c3)=O)CCCC2)=O)CCc2nnc(O)n2C1 15773,N(C(=NCCSC(F)(F)F)NCC12CCC(C3CC3)(CO1)C2)CCOC(C)(C)C 15774,N1(CCNC(c2c(OC)nsc2)=O)CCC(NC(=O)C#CC(=O)N(C)C)CC1 15775,C1(NC(C=CC)=O)CCN(C(=O)CCOc2ccccc2C(N)=O)C(C)C1 15776,c1(C(N2CCC(C(CNC(C(CC)NC(C)=O)=O)O)CC2)=O)c[nH]c(=N)cc1C 15777,C(c1nc(C)co1)=CC(=O)NC(c1ccccc1F)CNC(CC1CC(=C)C1)=O 15778,C12(CNC(c3n(C)ccc3)=O)CCCC1CCN2C(c1csc(C2CC2)n1)=O 15779,CC(C(=O)N(C)CC1CCCO1)OC(C1(CN)CC1)=O 15780,c1(OC)cc(C)cnc1C(N1CC(CNC(c2cc(C)co2)=O)C(C)(C)C1)=O 15781,C1(NC(C(COC)O)=O)C2CCN(C(=O)CCSc3nnnn3C)C12 15782,CCC(C(=O)N1CCCC1CC(=O)NC(C)(C)C#CC)NC(N)=O 15783,C(c1ccoc1)=CC(N1C(CC(=O)N(C)C)CC1)=O.C1(COCC=O)CCOC1 15784,N1(C(CN2C(C)CC2)=O)CC2CC1CCC2NC(c1ccc(F)c(C(F)F)c1)=O 15785,Cc1cccc(OCCC(N2CC=CC(NC(=O)C(C)CC3CCC3)C2)=O)c1C 15786,c1(C(=O)NC2C(NC(C(CC)N(C)C)=O)CCOC2)cccc2[nH]cc(C#N)c12 15787,C1(C(N(CCNC(C)=O)C)=O)CC2CC1CC2NC(c1cncc(C#N)c1)=O 15788,Cc1nc2c(C(=O)NCC3CC3NC(=O)CCc3c(C)noc3Cl)ccnc2[nH]1 15789,N1(C(C2CCC(=O)O2)=O)CCCCC1CNC(C1CCC(O)CC1)=O 15790,c1(C(=O)NC(c2cnn(C)c2)C(=O)NC(C)CS(C)(=O)=O)ccn2ccccc12 15791,C#CCCCC(C)C(=O)N1C(CNC(=O)Cn2ccccc2=O)CC2CCCC12 15792,C(=O)(C(C)(C)CNC(C1CC(F)CN1C(=O)Cc1cccc(Cl)c1)=O)NC 15793,C1(C#N)(C(=O)NCC(C(C)C)NC(=O)Cc2ccon2)CCCO1 15794,C=CCC(C)(C)C(=O)NC(c1nocc1C(=O)NCCn1ccnc1)C 15795,N1(C(c2cnc(CCC)s2)=O)CC(C)(CNC(=O)CCCC(C)(C)C)CC1(C)C 15796,N1(C(CC2(CC(=O)OC)CCCC2)=O)CCC2CN(C(C3SCCS3)=O)CC12 15797,C=C(C)CCC(=O)NCC(C1CC1)N(C(=O)CN(C1CC1)CS(=O)(=O)CCCC)C 15798,N1(c2nccc(C)n2)CCC2(CCC(NC(c3cc4c([nH]3)CCC4)=O)CC2)C1 15799,CC1CC2CCC(C(=O)NC(C3CCN(C(c4ccccc4F)=O)C3)C)CN2C1 15800,C=C(C)CN=c1[nH]c(=NCC2(CCF)CCC2)c2ccccc2[nH]1 15801,N1(Cc2n(CCCC)nnn2)CCCC2CN(C)CCC12 15802,c1(CC(N2CCN(C(c3cc(N)c(F)cc3)=O)C3C2C3)=O)cnc2c(=O)[nH]ccn12 15803,CCCCCCC(=O)N1CCCC(CCCNC(C2CCCNC2=O)=O)C1 15804,Cc1ccc(C)c(C(=O)NC2C=CC(CC(N3CCC4CC34C)=O)C2)n1 15805,N1(C(CC(CC)OC)=O)CCc2nc[nH]c2C12CCN(Cc1cn(CC)nn1)C2 15806,c1(C(=O)NC2C(CNC(COC)=O)C2)cc2ccccc2nc1C(F)(F)F 15807,N1(c2nnc(-c3c(C)nn(C(C)C)c3)n2CC2CCSC2)CCC2(CCCC2)CC1 15808,c1(C(N2CC3C(C(=O)NC(C)CC(N)=O)(C3)C2)=O)c(O)cccc1F 15809,C1(NC(C2C(CC)OCC2)=O)(CNC(=O)Cc2nonc2C)CCOCC1 15810,C1(C(=O)NCC2OCCC(C)(C)C2)CCC(C)(C)N(C(=O)CSC2CC2)C1 15811,C1(CCCNC(CN(c2ccccc2)C)=O)CCN(C(C2(C)C=CCCC2)=O)CC1 15812,C1(OCC)CC2CCCCN2C1.N1(C(C2(CCN=[N+]=[N-])CC2)=O)CC2C(C1)C(=O)N2 15813,C1(NC(Cc2cc(C(C)C)no2)=O)CN(C(=O)Cc2nc[nH]n2)CC2CC12 15814,c1(C(N2CC(CC(C)NC(C=CC=CC)=O)C2)=O)cc(CC(C)(C)C)[nH]n1 15815,C(=O)(CC(O)CCCCC)N1C(C#C)CN(C(=O)CSC(C)(C)C)CC1 15816,N1(C(CN(C(C(COC(C)=O)C)=O)CCO)=O)CC2(C1)CN(C)C2 15817,c1(OCC)ccccc1C1(C(=O)OCCCCn2c(O)nnc2O)CCCC1 15818,C1(C(=O)NCc2cc(C(N3CCC(CCC)C3)=O)sc2)CCC2(CC2)C1 15819,CCCCC(=O)C(=O)NCCCOCC(C)(C)NC(=O)CC1CCCO1 15820,C(C1CC1)(C1CC1)=CC(=O)NCC1(CNC(C2C(CCC)CCC2)=O)CC1(F)F 15821,C(=O)(CS(=O)(=O)C(C)(C)C)NC(CNC(CC1(C=C)CCOCC1)=O)C1CCC1 15822,N1(C(C2(CC#C)CCOCC2)=O)CC2CCC1CC2NC(=O)CCC1CCOC1 15823,c1(C(=O)O)c[nH]cc(-c2ccc(CN3CCN(C(=O)C(F)(F)F)CC3)cc2)c1=O 15824,C(=O)(C(C)C(F)(F)F)N(C(C)C)CCN(C(=O)C(O)Cc1ccc(Cl)cc1)C 15825,C(=O)(C(F)(CNC(=O)CCc1cnco1)C(C)C)NC(c1cccs1)CC 15826,c1(C(=O)NCCC2CCN(C(C(C)OCCOC)=O)CC2)nccc2n[nH]cc12 15827,C(CCCC(=O)N(C)CC1CCC(NC(=O)C(N2CCOC2=O)C)CC1)OCC 15828,C1(CC)(CNC(=O)C(CNC(=O)Cc2ccnc(F)c2)CC2CC2)CCC(=O)N1 15829,C(c1cccc(O)c1)=CC(=O)NC(CC1CN(C(c2cccc(C)n2)=O)C1)C 15830,C1(NC(c2c(C)[nH]cc2)=O)CCC12CN(C(C1CCCN1c1ccccc1)=O)C2 15831,O=C1CCC(CC(N2CCC(O)(C(F)F)C2)=O)CN1 15832,N1(C(Cc2c(C)nc(C)s2)=O)CC(C)CN(C(c2cn(CCO)nc2C)=O)C(C)C1 15833,C1(C(=O)NCC2(NC(=O)Cc3ccccc3Cl)CCC2)CCC(F)(F)CC1 15834,c1(C(N2CCC(CNC(c3n(C)ccn3)=O)C23CC3)=O)cc2cc(O)ccc2[nH]1 15835,N1(C(CCOC)=O)CC(=O)NCC1C(=O)NC1(CN(C)C)CC1 15836,C1(C(N2C(CNC(=O)C=C3CCSCC3)CC2)=O)CC2(CCCCC2)C1 15837,C#Cc1ccccc1-c1ccc(F)c(C(=O)NC(c2ccc(Cl)cc2)CO)c1 15838,C(CCCCC(=O)N1CC(C2CCCCN2C(=O)C(CC)SC(C)C)C1)OCC 15839,Cc1cnccc1C=CC(=O)NC(C)C(C)(C)NC(c1cncc(C#N)c1)=O 15840,C1(NC(c2c(C(C)C)ocn2)=O)CC2CC1N(C(C1CCCC13CCC3)=O)C2 15841,C1(CN(C(=O)Cc2conc2C)CC)CCCN1C(c1coc(Cl)c1)=O 15842,N1(C(c2n(CC)nc(Br)c2)=O)CCCc2ccccc2C1 15843,C1(C2(O)CN(C(C3(Cl)CC3(F)F)=O)C2)(CNC(C(C)=C(C)C)=O)CC1 15844,c1(C(=O)NC2(C)CCN(C(C(CC)OC)=O)C2)cccc(O)c1C 15845,C(C)(CCCCN=c1nc2c(cnn2C)c(NCC(C(C)C)C(C)C)[nH]1)OC 15846,Cc1csc(CC(=O)NCC2(C(N)=O)CN(C(=O)CN3CCNC3=O)C2)n1 15847,c1(CCOC)n[nH]c(=NCCCN(C)C(C2CCCC2OCc2cccc(F)c2)=O)s1 15848,c1(-c2c(OCCN(C)C)nccc2)ccc2c(c1)CCN(Cc1cccc(Br)n1)C2 15849,c1(NC2C(C(=O)OC)C23CC3C(=O)OC)ncnc(Cl)c1C#N 15850,O=C(C1=NOC(CNC(C2CC3CCCC3C2)=O)C1)NC1CCN(CCCO)C1 15851,c1(CC(N2CC(NC(C(=C(C)C3CC3)F)=O)C(C)CC2)=O)c(N)nc(C)nc1O 15852,C(C(C)(C(=O)N1CCC(F)(CF)C1)NC(c1nocc1C)=O)SC 15853,Cc1csc(C(N2CCCC2C(C)NC(=O)CSc2nc[nH]n2)=O)n1 15854,N1(C(c2cscn2)=O)CC2CC(C1)N(C(C1CC(F)(F)C1)=O)C2 15855,C1(n2cc(C(C)NC(=O)CSC(F)(F)F)nn2)CCCC=C1Br 15856,C1(NC(c2ccoc2)=O)CCN(C2(C(=O)Nc3ccccc3)CC2)C(C2CC2)C1 15857,c1(C(=O)NCCN(C(C=Cc2cc(C)no2)=O)C(C)C)ccccc1S(C)(=O)=O 15858,C1(NC(c2n(CC)ncc2)=O)CC2CCC(C1)N2C(c1nonc1N)=O 15859,Cc1cc(=NC(=O)C=CCC2CC(NC(c3cnncc3C)=O)C2)[nH]n1C1CC1 15860,N1(C(c2n(CC)ccc2)=O)CCC(CC(C)NC(=O)COCC2CCOC2)CC1 15861,Cc1cc(NC(C2CN(Cc3cccc(C#N)c3)CCO2)=O)cnc1F 15862,Cc1cc(C(=O)N(C(C(=O)NCC2(C)NC(=O)NC2=O)C2CC2)C)nc(O)n1 15863,C1(C2CCN(C(=O)CCC3CCC3)C2)CCCCN1C(=O)CCC1CCCOC1 15864,CC1CC(C)N(C(=O)CC(C)(C)C)CCN1C(=O)Cc1nc2cc(Cl)ccc2s1 15865,c1(CNCc2cc(C)cc(F)c2)ccc2c(c1)CCC2NC(=O)OC(C)(C)C 15866,c1(C(N2CC3CCN(C(COCCC#C)=O)C3C2)=O)cnc2c(c1)CCOC2 15867,C1(NC(c2c(CC)cno2)=O)CN(C(=O)Cc2cscn2)CCC1O 15868,C12(CC(=O)NCCC3CCC(NC(c4cnnc(O)c4)=O)C3)CCC(CC1)OC2 15869,C1(N(C)C(c2ccn(C)n2)=O)CC2CC1N(C(=O)C(CC1CC1)CC1CC1)C2 15870,n1(CC2C(C)C2)nc(CC(F)(F)F)nc1-c1nc(-c2cc[nH]n2)nn1C 15871,C1(CC)CCN(C(=O)C(C)S(C)(=O)=O)CC1(C)C.c1(C)nc(=NCC2CCCN2)s[nH]1 15872,Cc1csnc1C(=O)NC(Cc1ccoc1)C(=O)NC(C)CCC1CC1 15873,c1(NC(C2N(C(CCc3cccc(OC)n3)=O)CCOC2)=O)ccc2cnoc2c1 15874,C(=O)(C(F)CCCC)NC(C1CCN(C(CCC=CC)=O)CC1)CO 15875,C1(NC(c2cc(CC)n(CCO)n2)=O)CN(C(c2cccc(N)n2)=O)CCC1O 15876,c1(OC)ccc(C(=O)OCc2csc(C)n2)c(Cl)c1 15877,Cn1ncc2c1CC(CC(N1CCC(CCNC(c3cn[nH]c3)=O)CC1)=O)CC2 15878,c1(C(=O)NCC2C(NC(C3(CCOC)CCC3)=O)COC2)cc(C)c[nH]1 15879,C1(CNC(=O)NCc2cnc(Br)s2)CC(O)CN1C(=O)C(Cl)(Cl)Cl 15880,C(N=c1[nH]c(N(CCCN2C(=O)CCC2=O)C)nc2c1SCC2)C1OCC(C)C1 15881,c1(C(C(=O)NCCC2(C)CC2)N(C(CCC)C#N)C)nc(Cl)ccc1Cl 15882,N1(C(CCC#N)=O)CCC(CO)(CNC(C2CC23CCOCC3)=O)CC1 15883,N1(C(CCc2c(OC)cccc2)=O)CC(NC(=O)C(C)C2(O)CCC2)C2(CC2)C1 15884,c1(NC2C3CCCN(C(c4c(C)occ4)=O)C32)ccc([N+](=O)[O-])cc1 15885,Cn1cnc(CCC(=O)NC2CCC2CNC(C2CCN2C2CCCC2)=O)c1 15886,Cc1ccc(SC2CCC(C(=O)NC(C)CNC(C3CCC(=O)N3)=O)CC2)cc1 15887,C12(NC(C(C)NC(c3c[nH]c4ccccc34)=O)=O)CC1COC21CCC1 15888,N1(C(c2c(CC)occ2)=O)CCC(C2CCN(C(=O)CCCCO)C2)C1 15889,C(=O)(C(C)CCCCCC)N1CCC(O)(CCNC(CSCC=C)=O)C1 15890,C1(F)(C(=O)NCC(CN(C)C(c2cn(CC3CCCO3)cn2)=O)(C)C)CCCOC1 15891,Cc1csc(=NCC(=O)NCC2CC(F)(CNC(C3(C)COC(C)(C)CO3)=O)C2)[nH]1 15892,Cc1nc(C(F)(F)F)c(C(N2CCC2CNC(c2cccc(CO)n2)=O)=O)s1 15893,C=CCC(C)(C(=O)N(CC(C)NC(c1cc2n(c1)CCC2)=O)C)N(C)C 15894,N12CCC3(CC1)CN(CCO3)CC(CC)C2=O.c1(OC2CNC2)cccc(C)c1 15895,C1(CCCC)CN(C(=O)CC2CCOC2)CCN1C(=O)C=Cc1cccc(F)c1 15896,c1(NC(C2CCC(CC)O2)=O)ccc(NC(=O)CCCC(C)=O)c(C)c1 15897,N1(C(c2cc(OC)c(C)cc2C)C(=O)NCC=C)CCC2(CCCN(C)C2)C1 15898,c1(C(N2CCCC(CNc3nc(COC)nc(O)c3)C2)=O)ccc(F)c(C#N)c1 15899,Cc1cc(C(=O)NC2CC(NC(C3CCCN(CC(C)C)C3)=O)C2)ncc1C#N 15900,C1(C(C)C)(NC=O)CCN(C(c2nscc2C)=O)C1.C(C)(C)(C)OCCNC=O 15901,c1(C(=O)NC(CC)CNC(C2(CF)CC2)=O)ccc2c(n1)NC(=O)CO2 15902,c1(C(=O)NC2CN(C(C3CCC(F)(F)C3)=O)C2)cnc2cccnc2c1 15903,c1(CNC(N(C(Cc2nncn2C)C2CC2)C)=O)ncnn1CCF 15904,C#CCC(C)(C(=O)NCc1c(C)cccc1F)NC(c1nc(C)ccc1C)=O 15905,N1(C(c2cn(CC)nn2)=O)CCC(C)C(CNC(c2cn(CC3CC3)nn2)=O)C1 15906,C1(NC(CCCCN(C)C)=O)CCCC12CN(C(C1CN3CCCC1C3)=O)C2 15907,CON1CCC(C(=O)NC(C2(O)CCN(C(C3CCCCN3C)=O)C2)C)CC1 15908,c1(NS(Cc2nc(C(=O)OC)sc2)(=O)=O)cccc(Oc2ccc(F)cc2)c1 15909,C1(CC)C(NC(=O)Cc2ccco2)CCN1C(C1CCS(=O)(=O)N1)=O 15910,C1(N(C)C(c2ccc(-n3cnnc3)cc2)=O)CN(C(=O)C(C)(F)F)CCC1O 15911,c1(C(=O)NC(C)CNC(C2CCC(C)C2)=O)csc2cncn12 15912,CCCCCCC(C(=O)N1CC(OC)CCC1C)c1ccccc1 15913,CC(CC(=O)NC1(C2CCN(c3nc(Cl)ncc3C3CC3)C2)CC1)C(F)(F)F 15914,CC1CCOC1C(=O)NCCCCNC(c1csc(C(C)(C)C)n1)=O 15915,CN1CCCCC1CN1CCC(C(=O)NCc2ccnc(N3CCCC3)c2)C1 15916,C1(C(=O)NCCC2(OC)CN(C(C3C4CC4C4CC34)=O)C2)CC2(CC(OC)C2)C1 15917,N1(C(C=CCCC)=O)CC(NC(=O)C(=O)N(C)C)C2(CCOCC2)C1 15918,Cc1cc2c(C(N3CC4CC(NC(C5CCC(C)CC5)=O)C3C4)=O)nccn2n1 15919,C(CC1(CO)COc2ccccc21)N(C=O)CC1CC12CCCC2 15920,O=C1C=C(c2cc(-c3c[nH]nc3C(N3CCC4(CCCO4)C3)=O)ccn2)CCC1 15921,C1(C)(NC(C(C(C)(C)O)NC(c2ncc(F)cc2F)=O)=O)CCCC(C)(C)C1 15922,C1(C)C2CCC(C2)N1C=O.c1(C(NOCCOC(C)C)=O)ccnn1CCF 15923,C12(C(=O)NC(C)(C)CNC(=O)C(CO)C(C)(C)C)CCCC(C1)C(=O)NC2 15924,C1(C(=O)NC(C2CN(C(=O)CN3CC(=O)NC3=O)C2)C)CCOCC1(C)C 15925,Cc1nc2cc(F)ccc2cc1C(=O)NCC=CCNC(c1ccn(C2CC2)n1)=O 15926,S(=O)(=O)(c1ccc(NCC2CC2(Cl)Cl)cc1Br)NCc1cncc(OC)n1 15927,c1(-c2cccc(NC(N3C(C(=O)O)CCOCC3)=O)c2)c[nH]c2ccc(Cl)cc12 15928,C1(C(N(CC(=O)N(CC(F)Cl)C2CCC2)C)=O)CCC(=O)O1 15929,CC1(C#CC(=O)NCCC2(O)CCN(C(=O)CCOc3ccccc3F)C2)CC1 15930,C1(NC(CCOCCOC)=O)C(C)(C)C(NC(c2cc(F)n[nH]2)=O)C1(C)C 15931,N1(C(C2N(C)C(=O)NC2)=O)CC2(CC2)CC1CNC(=O)CCC(F)(F)F 15932,C(C#CC(F)(F)F)NC(C1C(NC(C2(COC)CC=CC2)=O)CCO1)=O 15933,N1(C(C2(C)CC2(F)F)=O)CCC2(CCN(C(=O)C(C3(O)CCOCC3)O)CC2)C1 15934,C1(C(=O)OCC)CC(NC(=O)NCc2ccnn2CC(F)F)CCO1 15935,Cn1c(C(=O)NC2CCOC(NC(=O)COC3CCOCC3)C2)cnc1S 15936,Cc1cc(F)cc2[nH]c(C(=O)N(C)CCNC(c3ccc(F)c(Cl)c3)=O)cc12 15937,C(=O)(C1=CCN(C(C2CC(=O)N(OC)C2)=O)C1)NC(CC)CCCO 15938,c1(C(=O)NC(C(=O)NC(C#C)Cc2ccco2)C2CC2)cc([N+](=O)[O-])c[nH]1 15939,C1(C(=O)NCC(C)CN(C(=O)C(F)CC2CCCCC2)C)CCC2(CC1)CC2 15940,c1(C2N(C(CN(C)C(=O)Nc3ccc(F)cc3)=O)CCC2)n[nH]c2ccccc12 15941,c1(C(=O)NCCC2CC(NC(CC=C)=O)C2)cn(-c2ncccn2)cn1 15942,S(=O)(=O)(c1ccccc1)N(CC(N1C(CNC(C(C)SC)=O)CCC1)=O)C 15943,C1(C(N2CCCC(NC(c3c(C)nc(C(F)(F)F)o3)=O)C2)=O)C2CCC3C(C2)CC13 15944,C(=O)(C(CC(C)C)N(C)C(C1CNC(=O)O1)=O)N(C(CC)C1CC1)C 15945,N1(C(CC(C=C)(C)O)=O)CC2CCC(C1)C(NC(c1cnc(OC)c(C)n1)=O)C2 15946,C1(O)(CNC(c2n(CCC)nnn2)C2COC2)CCCN(C(=O)OC(C)(C)C)C1 15947,N=c1nc2c(c[nH]1)CCC(C(=O)NCCNC(=O)C(C1CCCCC1)O)C2 15948,N1(C(C=CC(CC)C)=O)CCCCCC(NC(=O)C(c2ccc(F)cc2F)=O)C1 15949,C1(C(=O)NC2CCCC2CCCNC(C2(C3CCCO3)CC2)=O)CC12CCOC2 15950,CC(O)C(C)C(=O)N1CCCC1C(=O)NC1CCCN(S(C)(=O)=O)C1 15951,C1(C(C)S(=O)(=O)c2ccc3c(c2)COC3)CCN(C(=O)C(C)CC(F)F)O1 15952,C(=O)(CC(C)(O)C(F)(F)F)NCC(C)NC(CCC(=C)Cl)=O 15953,C1(NC(CSCC=C)=O)CC(C)(CNC(=O)C(C)CC2CC2)C1 15954,C1(NC(C(C=C)(C)CC)=O)CCN(C(c2ccc(OCOC)cc2)=O)CC1(C)C 15955,N1(C(c2cc(C)nc(C)n2)C(=O)NC(CC)C)CCc2ccc(F)c(Br)c2C1 15956,N1(C(C2CCc3ccccc3O2)=O)CCC(C2CCOCC2)C1 15957,N1(C(c2cnc(C(C)=O)s2)=O)CCCC(C)(NC(C2C(F)(F)C23CCC3)=O)C1 15958,c1(COC(C(c2c(C)cccc2)(F)F)=O)ccc(S(=O)(=O)C(F)(F)F)cc1 15959,c1(C(N(C(CCSC)C)C)=O)cc(CNC(=O)CCc2cnn[nH]2)no1 15960,N1(C(C2N(CCC)CCC2)=O)CCCCC(NC(=O)CCC(=O)c2ccncc2)C1 15961,c1(C(N2CCC(C)(NC(c3cnn(C)c3F)=O)C2)=O)ccc2ncncc2c1 15962,n1(C(CC)C)ccc(=NC(=O)C2=CCCN(C(=O)Cc3ccc4c(c3)CCC4)C2)[nH]1 15963,N=c1cc[nH]cc1COc1cncc(Nc2cccc(C(F)(F)F)c2)c1 15964,c1(C(C(=O)N2C(CNC(C(CCCC)O)=O)CC2)=O)ccc2c(c1)CCCC2 15965,C(CC(C(=O)NCC1CCCC1(C)C)NC(c1cncc(C)n1)=O)=CC 15966,CCCC(C)(O)C(=O)NCC1CCCC1C(=O)NC1CN(C)CCC1O 15967,c1(C(=O)NCC2(COC)CCN(C(C3CCC3C)=O)C2)cc2ccccn2n1 15968,S(=O)(=O)(c1cccc(CN2CC(F)(c3ccccn3)C2)c1)N1CC(C)NC(=O)C1 15969,C(=O)(CS(N)(=O)=O)NCC1(F)CC(CNC(C(CC2CCCC2)OC)=O)C1 15970,c1(C(N(CCCNC(C2CC(C)CO2)=O)CC)=O)cc2n(n1)CCCO2 15971,C1(OC)CCC(C(F)(F)F)(NC2CCCN(Cc3nccn3C)C2)C1 15972,C1(C(=O)N(C)CCNC(c2ccn(C(C)C)n2)=O)(CC)CCOC1 15973,CN1CC(C(=O)NC2CC(F)(CNC(=O)Cn3cnnc3)C2)C(C(F)(F)F)C1 15974,C12(C(=O)NC3CC(NC(C4CCCS4)=O)C3)CCC(O)C1CC2 15975,C1(CCOC)CN(C(=O)Nc2ncc(I)cn2)C12CCC2 15976,CC1CCC(c2nnnn2C)(NCc2cc(C(F)F)on2)C1 15977,C(c1cccc(F)c1)=CC(=O)NCC(C)(F)CNC(C1CC(F)(CF)C1)=O 15978,C1(c2c(OC)cccc2)CCN(C(c2ncc(Cl)n2C)C(=O)NC2CC2)C1(C)C 15979,CC(C)(C)C(C(=O)NCC1CCCN1C(N)=O)NC(c1ccccc1Cl)=O 15980,N1(C(CC(CC)OC)=O)CC(C)(C)C(NC(c2cnc(Cl)s2)=O)C(C)(C)C1 15981,Cc1cccc(C(=O)NCCCCCNC(C2(C3CCCCO3)CC2)=O)c1O 15982,N(C(=NCC1CCC(=O)NC1)NCc1ncccc1C(F)F)C(C)C 15983,C1(C(=O)Nc2c[nH]c(-c3ccncc3)n2)CCCN(C2CC2)C1=O 15984,C1(C(=O)NCC#C)CCCN1C(=O)CNC(C1(NC(C)=O)CCCC1)=O 15985,C(=O)(C(C)CC(F)F)N(C1CCN(C(c2ccc(C(C)C)s2)=O)CC1)CC#C 15986,N1(C(c2ccc(CCC)cc2)=O)CCC2(CC1)CC(NC(C1CC=CCO1)=O)C2 15987,Cc1cc(NC(C23CC(CNC(=O)CC4C5CCC(F)C45)(C2)C3)=O)sc1C 15988,CC1CC(NC(=O)C(C)C(=O)OC(C)(C)C)CCN1C(=O)CN1CC(C)(CO)C1 15989,c1(C(=O)NC(CC(C)NC(C(CN(CC)CC)F)=O)C)cc(S(N)(=O)=O)sc1C 15990,C(CCC(=O)NCCC(C)NC(=O)C(C)OCCC(C)C)=CCC=C 15991,C1(NC(NCC=CC)=NCC2CCCCC2)CC2CCCN2C1 15992,CC(CCCNC(C1CCN1C(C)(C)C)=O)NC(C1CC(=O)N1)=O 15993,CC1C(NC(c2c[nH]cc2C(N)=O)=O)CCCN1C(=O)Cc1cnccc1Cl 15994,c1(C(=O)NCC2CCN(C(C(C)C3CC3)=O)C23CC3)cccc2ncnc(O)c12 15995,C1(CNC(c2cnn(-c3ccncc3)c2)=O)C2CN(C(=O)C)CC12.C1(N)CC1 15996,[N-]=[N+]=NC1CN(C(=O)CN2CCSCC2)CC1NC(c1cc(C#N)ccc1O)=O 15997,N1(C(c2cnc(C(=O)OC)cc2C)C(=O)NC)CCC(S(=O)(=O)NC)C1 15998,C1(CNC(CC(C)F)=O)CN(C(=O)CSC(F)(F)F)C2COCC2O1 15999,Cn1c(CCN=C(NC2CCC2)NC2CC23CC3(F)F)nc2cc(F)ccc12 16000,c1(OC)ccc(CC(N2CC3CC2C3NC(=O)CC(C)c2cccnc2)=O)c(Cl)c1 16001,N1(C(CCS(C)(=O)=O)=O)CCC2(CC1)CC(NC(C1(CO)CCOCC1)=O)CO2 16002,c1(C(C)=O)nc(C(=O)N(CC(C)(C)NC(=O)Cc2csc(C(F)(F)F)n2)C)cs1 16003,CN1CCN(C(=O)C(CNC(C2C3CN(C)CC23)=O)CC2CCCC2)CCC1=O 16004,C(=O)(C1=NOC(C)(C)C1)NC(C)C(C)(C)C(=O)NCCCN1CCC1 16005,CN1CC(O)CC1C(=O)NCC(C1CC1)NC(=O)CCCc1ccsc1 16006,CC1(C)CCC(CN(C(=O)Nc2ccc(F)cn2)CC23CCC(CC2)C3)CC1 16007,C=C=CC(C)C(=O)NCc1c[nH]nc1C(=O)NCCOC1CCCC1 16008,Cc1cc(C(=O)N(C)CC2(O)CN(C(C3(C(=O)N(C)C)CC3)=O)C2)cc(C)c1F 16009,c1(C2(C(=O)NCC(CNC(c3ccc(OC)nc3)=O)O)CC2)cc(C)cc(C)c1 16010,c1(C(=O)NCC(CNC(c2c(C)n(C3CC3)nc2)=O)C)cc(S(N)(=O)=O)cn1C 16011,c1(C(N(C2CCCC(NC(C=CC=CCC)=O)C2)C)=O)c(F)cc(OC)cc1Cl 16012,C1(NC(CCN(CCC)C)=O)CC(O)CN(C(c2cnc(SC)s2)=O)C1 16013,C(=O)(C1CCc2c(Cl)cccc21)NCCNC(c1cnc(C2(C)OCCO2)s1)=O 16014,C(=O)(CC(=O)NC(C)C=CC(N1CCC1CF)=O)OC 16015,c1(C(N2CCC(NC(C(CC)SC)=O)CC2C)=O)ncn2ccccc12 16016,C1(NC(CC(=O)N(C)C)=O)CC2CCC(C1)N2C(=O)Cc1cccc(F)c1Cl 16017,C1(NC(CNC(=O)OCC=C)=O)CN(C(=O)C(C(C)C)n2ccnc2)CC1F 16018,C12(C(=O)NC(CCO)C3CCCC3)CC(CCO1)N(C(C13CC(C1)C3)=O)C2 16019,CC(CC(N)=O)C(=O)N1CC(CNC(c2ccnn2C(C)(C)C)=O)C2(CC2)C1 16020,c1(CNC(C2(CC)CCCC2)=O)cccc(NC(=O)CC2CC(C)OC2C)c1 16021,c1(C(=O)N(CC(=O)NCC(O)CC2CCCC2)C2CCC2)ncoc1C1CC1 16022,Cc1cccc(F)c1CC(=O)NC1CC(NC(C2C3CCC(F)(F)C23)=O)CC1O 16023,Cn1cc(C(=O)NC2COCC2NC(=O)CC(=O)NCC2CC2)c(C2CCC2)n1 16024,CC1=C(C(=O)NC2CCN(C(=O)C=C(C3CC3)C3CC3)C(C3CC3)C2)CCC1 16025,C1(F)(CNC(C2C(=O)NCC2)=O)CCN(C(c2cccc(OC(F)(F)F)c2)=O)C1 16026,C1(NC(C(C(C)C)N(C)C)=O)CCN(C(c2cc3occc3s2)=O)CC1C 16027,c1(CC)cccc(-n2nc(C(CC)OC)nc2-c2coc(C3CC3)n2)c1 16028,CCCCS(=O)(=O)NC(C)C(=O)NC1CC(CNC(=O)C(C)(C)NC(C)=O)C1 16029,CC1=C(C(=O)N2CCCCC2C2CCCN(S(C)(=O)=O)C2)CCC1 16030,N1(C(C(C)=CC(C)(C)C)=O)C2CCC1CC(CC(=O)Nc1cnc(C)nc1C)C2 16031,CC1(NC(C2(C(=O)OCc3ccc(F)cc3)CC2)=O)CCC(=O)NC1=O 16032,C(CNC(C1(O)COC1)=O)(CC(C)C)NC(C1C(CC)C1)=O 16033,Cc1cc(N2CC3CC3(C(=O)NC(C#N)C(N)=O)C2)ncn1 16034,c1(C(=O)NCC2CCN(C(C3CCC(C)O3)=O)C2)csc2ccccc12 16035,C1(NC(C2CCC(C)C2)=O)CCOC2(CCN(C(C3(O)COC3)=O)CC2)C1 16036,c1(C(N2C3CC(CNC(C4CC(=O)NC4)=O)C2CC3)=O)cccc2sncc12 16037,C1(NC(CCC#C)=O)CN(C(c2cc(F)c(Br)cc2F)=O)C2CCCCC12 16038,C12(C(=O)NCC(=O)NCC3CC3NC(=O)Cc3cccs3)CC1COC21CCC1 16039,Cc1cc(NC(CNC(c2nc3ccccc3[nH]2)=O)C(C)C)n2nc(C)cc2n1 16040,C(=O)(C(F)(F)C(C)O)N(C1CCCCC1)CCNC(C(CCC)O)=O 16041,C1(NC(c2cc(C)cc(C)c2)=O)CN(C(c2ccc(O)cc2F)=O)C2CCCC12 16042,CS(=O)(=O)CCCC(=O)NC1(CF)CCN(C(C2(Oc3ccccc3)CC2)=O)C1 16043,CCCCCC(O)CC(=O)NC(c1cn(C)nn1)CNC(c1cc(Cl)c[nH]1)=O 16044,c1(CC(=O)NCC2C(C)CN(C(=O)C(C3CC3)C3CC3)CC2)ccc2c(c1)CCC2 16045,C1(NC(c2c(C)[nH]cc2)=O)CCOC(C(=O)NC2CC(CCO)C2)C1 16046,C(Cc1ccoc1)(C(=O)NOCC1CC1)NC(C1CC2CCC1CC2)=O 16047,C(=O)(C(CCOC)OC)N1CC(CCO)(NC(c2nc(CCCCC)sc2)=O)C1 16048,N1(C(CCNC(=O)NC)=O)CCC(O)(C(=O)NCCNC(=O)CC(C)(C)C)C1 16049,N1(C(CSCCN(C)C)=O)CC2CC(O)C1C2NC(C1CCCCNC1=O)=O 16050,C(=O)(C1=NNC(=O)C1)N(C)CC1(O)CCN(C(C(C(C)C)OC)=O)CC1 16051,c1(C(=O)NCC2(C(=O)NCc3ncc(C)nc3)CC2)cccc(O)c1C 16052,CC(C)CCC(=O)C(=O)N1CCC(C(c2cc(C(C)(F)F)[nH]n2)=O)CC1 16053,c1(C(N2CC(NC(COCCC#C)=O)C(C)(C)CC2)=O)cc(S(C)(=O)=O)c(C)o1 16054,C1(NC(c2nc(OC)c(C)s2)=O)CCN(C(C2CCC3CC2CO3)=O)C(C)C1 16055,Cc1ccc(CC(C)C(=O)NC(C2CCCN(C(=O)CSCC(C)C)C2)C)cc1 16056,c1(C(=O)NC(CNC(CSCCN(C)C)=O)CO)cc(N)c(Cl)c(O)n1 16057,CCC(CC)CCC(=O)NC(C1CCCC1)CC1CCN(C(=O)Cn2cccn2)C1 16058,C1(C(=O)NC2CN(C(C=CCOC)=O)C2)(OC)CCCC(C)C1 16059,Cc1ccnc(C(N2CCC(C)(CC(N3CC(n4cnnn4)C3)=O)C2)=O)c1F 16060,C1(C(NOCC(C)O)=O)CCN(C(c2cc[nH]n2)=O)CC1O 16061,CCCCCCCCNC(=O)C(=O)NCCCN(CCO)C(C1CC1(C)CC)=O 16062,c1(CCNC(c2n(C)cnc2Br)=O)nc2c(o1)CCSC2 16063,C1(C(=O)NCC=CCNC(=O)CC2CCCC2(F)F)CCn2ccnc2C1 16064,c1(CC(C)N(C(=O)C(c2ccnn2C)O)CC#C)ccccc1F 16065,C1(NC(C(C(C)C)SCC)=O)CC2CCC(C1)N2C(c1ccc(C(C)=O)[nH]1)=O 16066,N1(C(C(C2CCC2)OC)=O)CCC(C)CC1C(=O)NC(COC)C(C)C 16067,C(C1c2ccccc2CN1C(C1CC2(CC2)C1)=O)NC(C(C)CS(C)(=O)=O)=O 16068,C12(NC(=O)NC3CC(=C)C3)CCOC(Cc3nn(CC)cc3Br)(C1)C2 16069,Cc1ccc(C(=O)NC(C)C(CO)NC(C2CC(S(C)(=O)=O)C2)=O)cc1C 16070,C1(CCC#C)CCCN1C(=O)C(c1cccs1)NC(c1ccon1)=O 16071,c1(C2c3nnnn3CCN2)ccc(C)cn1.C1(OC)(CN2CCCC2)CCSC1 16072,Cn1ccc2c(C(N3CCN(C(=O)C(F)=C4CCCC4)C(CF)C3)=O)cccc12 16073,C1(CCCC)CN(C(c2ccnc(C)c2N)=O)CCN1C(=O)CCC(C)CC 16074,n1(CC(=O)NCC23CC(CO)(C2)C3)cc(C(F)F)cn1.N12CCC(C1)CC2=O 16075,C(=O)(C1CCc2ccccc21)NCC(=C)CCNC(C1CC(=O)N(O)C1)=O 16076,C12(C(=O)NC(CNC(c3ccco3)=O)CO)CC(=O)C1C2 16077,N1(C(Cc2c(C)ccs2)=O)CCN(C(c2cc(CO)[nH]n2)=O)C(C2CCC2)C1 16078,C=CC(CC)C(=O)N(CCC)CCNC(c1cccc(-c2n[nH]c(C)n2)c1)=O 16079,C(=O)(C(C)(C)C(F)F)N(C(CC(=O)NCc1c(C)occ1)C)C 16080,C(C1CCN(C(C2CCCC(=O)C2)=O)CC1)=CC(=O)NCC1N(CC)CCC1 16081,C12(CCNC(=O)C(=O)NS(C)(=O)=O)CCCN1CCC2.C1CCCC(=O)N1C 16082,C=CC(C)(CCOC)C(=O)NC(CN(C(=O)C(O)C1CCCC1)C)CC 16083,c1(C(=O)NC2CCN(C(Cc3ncc(CC)[nH]3)=O)C2)cc(F)cc(F)c1N 16084,CS(=O)CCC(=O)NCCN(C(=O)CN(C)CCOCc1ccc(Cl)nc1)C1CC1 16085,CC(C)CCCC(C)C(=O)N1CC2(CC(C(=O)N(C3(C)CC3)C)CO2)C1 16086,C(=O)(CCS(N)(=O)=O)NCC1N(C(c2cccc(C(C)C)c2)=O)CC=C1 16087,c1(NC(C(C2CN(C(c3cc(CCC)[nH]n3)=O)C2)O)=O)ccc(C)c(C)c1 16088,c1(C(N(CCCNC(c2cnsn2)=O)C)=O)cccc(-c2nc(=O)o[nH]2)c1 16089,C1(C(=O)NCCCn2ncc(C)c2)(CNC(c2scc(C)c2C)=O)CCCCC1 16090,CC1CC(C(=O)N2CCC2CNC(c2cncc(-c3cccc(F)c3)c2)=O)=NO1 16091,CC(C)(C)C(C(=O)NCCc1nc[nH]n1)NC(c1ccnnc1)=O 16092,c1(CC(N2C(CN(C(c3cnc(C)s3)=O)C)CCC2)=O)ccc2[nH]ccc2c1 16093,CC1CCCN1CC(=O)NCC(N1CCC(N(C)CC2(O)CC(O)C2)C1)=O 16094,n1(CC)cc(Cl)c(C(=O)NC2CCCCC2Cn2cc(CNC(C)=O)nn2)n1 16095,C#CCCC(O)C(=O)Nc1cccc(NC(=O)C(c2ccc(F)cc2)OC)c1 16096,n1(CCC)nc(C)cc1C(=O)N(CCCN(C(=O)C(C)CC)C)C 16097,N1(C(CSCC)=O)CCC2(CCN(C(c3ccc(OC)nc3)=O)C2)C1 16098,C(=O)(C1=NN2CCCN=C2N1)N1C(C)(C)CC(CNC(=O)COC2(C)CCC2)C1 16099,c1(COC)ccc(N(C)C(C2(CNC(=O)CC3COC(=O)N3)CC2)=O)cc1 16100,c1(C(=O)NC(CC)(CNC(=O)C(C)CCO)CC)ccc2nc(N(C)C)oc2c1 16101,CC1(C)CN(C(c2csc(=N)[nH]2)=O)CC1C(=O)NCCC1OCCC1(C)C 16102,C1(NC(c2ccc(C)cn2)=O)CCCC12CN(C(C1CCCC1C(F)F)=O)C2 16103,C#CCC(C(=O)N1CCCC1C(=O)NOCc1nc[nH]n1)C1CC1 16104,c1(C(N2CCOC(CCO)C2)C(=O)NC(C(=O)OC)C)ccncc1Cl 16105,C1(C(=O)NCCN(C(c2c(C)cc(F)cn2)=O)C2CC2)CCC2(CCC2)CO1 16106,CC(C)CC(C(=O)NC1(F)CN(C(c2ccc(F)cc2F)=O)C1)N(C)C 16107,c1(N2CCCC(CNC(C3(C)CC3Br)=O)CC2)ncnc2cccc([N+](=O)[O-])c12 16108,CC(C(=O)N1CCN(C(c2nccc(N)c2Cl)=O)CC1CF)C(C)(C)C 16109,C(CC(F)(F)CO)NC(C1CC=CCN1C(=O)Cc1cncnc1O)=O 16110,C1(CCCc2cn(Cc3scc(C(=O)NC(CCCC)C)n3)nn2)CCCCCC1 16111,c1(CCN(C(=O)CC2(O)CCOC2)CC(O)C2CCC2)cccn2ccnc12 16112,N1(CC)CCCCC1C(N1CC(C(=O)NC(C2CSC2)C)C(CC)C1)=O 16113,CC(O)C(=O)N1CC(C(=O)NCC2CC2CO)C1 16114,c1(C(N2CCCC(C(C)NC(Cc3c(C)scc3)=O)C2)=O)cc2ncccc2[nH]1 16115,n1(CC=C)nnnc1C1c2nncn2CCN1.C1CC(=O)O1.C1(COC)CC1 16116,C(=O)(CC(C)C(=O)N(CC(=O)NCC1CC(C)C1)C(C)C)OC 16117,c1(CC(N2CC(O)(CCNC(C(C)N3CCC3)=O)C2)=O)ccc(Cl)cc1Cl 16118,N(C(=NCCC(C)C)N1CCc2ocnc2C1)CCc1c(C)noc1C 16119,C1(C)(C(=O)NCCCC(C)NC(c2c(CC)n(C)nn2)=O)CC2(C1)CC2(F)F 16120,c1(C(C(=O)NC2(CNC(C3C(CC)C3)=O)CC2)(C)C(=O)OC)ccc(F)cc1 16121,c1(C(=O)NC2CC(CNC(CC3(OC)CC3)=O)C2(C)C)cc([N+](=O)[O-])cc(C)c1Cl 16122,C(=O)(CC1OCCc2ccccc21)NC1CC1C.N1(CCNC(=O)CO)CC=CC1 16123,N1(C(C(C2CCCN(C(c3coc(C4CC4)c3)=O)C2)C)=O)CCCCCCCC1 16124,C1(C(=O)NCCCN(C(C(C)NC(COC)=O)=O)C)COCC(C)(C)O1 16125,C1(CC)COCC1N=c1[nH]c(N2CCC=C(C)C2)nc2cc(OC)ccc12 16126,C(=O)(C#CC1CCCOC1)N1CC(OC)(CNC(C2(C)COC(=O)OC2)=O)C1 16127,N1(C(c2nnc(C)s2)=O)CC2C3CCC(C2C1)N(C(c1conc1C(C)C)=O)C3 16128,N1(C(C(C(CC)C)NC(C)=O)=O)CCC2(CCC2)C(NC(C2CCC(=O)NC2)=O)C1 16129,C1(NC(C2(OCC)CCC2)=O)COCCC1NC(c1scc(C)c1C(C)=O)=O 16130,n1(CC#C)cccc1C(=O)N(C(C)CNC(C1(COCC)CC1(F)F)=O)C 16131,C(=O)(C1=NOC(C)(C)C1)N1C(CCOC)CN(C(=O)Cc2cccc(F)n2)CC1 16132,N1(C(=O)C=Cc2ccco2)CC2(CNC(=O)CC3(O)CCCCC3)CCC1C2 16133,C(=O)(C1=NNC(=O)CC1)N1CCN(C(c2c(C)nn(C)c2C)=O)C(C2CC2)C1 16134,N1(C(c2c(CC)ccs2)=O)CC2CCC2(CNC(=O)CCCc2csc(=N)[nH]2)C1 16135,c1(CN)cccc2nc(N3CCOc4ccc(F)cc43)sc12 16136,c1(C(CC(=O)NCC(C)N(C(CCOC(C)=O)=O)C)C)ccc(F)c(F)c1 16137,C1(C2CCCN(C(c3c(C4CCC4)cnn3C)=O)C2)(NC(CC(C)C)=O)CC1 16138,N1(C(C2(CCl)CN(C(c3c(C(=O)OC)nsc3N)=O)C2)=O)CCC(=O)N(C)CC1 16139,Cc1noc(CN2CC3CCC(N)(C(=O)O)C3C2)c1[N+](=O)[O-] 16140,N1(C(CCCC)=O)C2CCC1CN(C(=O)CCc1cn(C)nn1)C2 16141,O=c1nc(O)c(CN(C2CC2)Cc2nc3c(s2)CCCC3)cn1-c1ccccc1 16142,CC1CCN(C(c2cc(C3CC3)ccn2)=O)C1CNC(C1CC1CF)=O 16143,CCC(CC)CCC(=O)N1CCN(C(=O)CC(O)CC(C)C)CCC1C 16144,C1(NC(C2C(NC(CCC(C)SC)=O)CCO2)=O)CCN(C)C1(C)C 16145,C(=O)(C1CCc2nccn21)NC(C(=O)NC1(CC)CCCC1)CC1CC1 16146,C(C)(C(=O)NN1CCN(S(=O)(=O)c2cnc3c(ccn3C)c2)CC1)c1scc(C)n1 16147,N1(C(C(CCC)O)=O)CCN(C(c2ccc[nH]2)=O)CC1c1cccnc1 16148,Cc1cnc(C(=O)NC2CCC(C)(NC(=O)CS(=O)(=O)N(C)C)C2)c(C)c1 16149,C1(NC(Cc2cn(C)nn2)=O)CCN(C(=O)CC2CC(C(F)F)C2)C12CC2 16150,N1(C(CC2(C=C)CCC2)=O)CCCOC(CNC(=O)CCS(C)(=O)=O)C1 16151,C1(C(N(C)CC2CC(=C)C2)=O)CCN(C(=O)CCCCOCC)C1CC 16152,C=CCC(C)(C)C(=O)N1CCCC(COC)(NC(c2cc(C)n(C)c2)=O)C1 16153,N1(C(c2c[nH]nc2C2CC2)=O)CC2C(NC(C3(c4cccc(Cl)c4)CC3)=O)C2C1 16154,C1(CN(C(C(c2ccc(CC)s2)=O)=O)C)CCCCN1C(=O)CCN1CCCC1 16155,C1(C(N2C(CC)CC(C)C2)=O)CCC2(CC2)N1C(c1c[nH]c(C)c1)=O 16156,c1(C(=O)NC2CCC(C)(CNC(c3c(CC)scn3)=O)C2)ccc(OC)c(O)c1 16157,C12(C(N(CCC)CCNC(=O)C(N)=O)=O)CCC(CO)(C1)NC2 16158,C1(CC(=O)NC2C(CNC(Cc3c(C)n[nH]c3)=O)C2)NC(=O)NC1=O 16159,N1(C(C(C=C)O)=O)CC(NC(=O)CC2CCCCCC2)CC2(CCC2)C1 16160,c1(C(CC)=O)cccc(NCc2cscc2C)c1C 16161,N1(C(C(CN(C)C)O)=O)CCC2C(CCCN2C(C2CCCCN2C)=O)C1 16162,C1(CCC(=O)N(CC(C)O)CC(C)O)CCC(NC(C2CCCN2C2CC2)=O)C1 16163,N1(C(CC2(C)CCOCC2)=O)CCC2(CC1)CC2C(N1CC2CC2C2CC12)=O 16164,C12(CNC(C3C(C)(C)C3)=O)CCC(C1)N(C(=O)CCCN1CCCC1)C2 16165,Cc1ncc(C(N2CC=C(CNC(C3CCC4C3C4(F)F)=O)CC2)=O)cc1C#N 16166,c1(NC(=O)C(CCC)N(C)C)cccc(NCCCC)c1F 16167,N1(CCN)CCN(CCO)CC1.c1(CC(=O)N(C(=O)C(F)F)C(C)C)cccs1 16168,c1(COC(C(=O)NCC(C)CN(C)C)C)ccccc1 16169,C1(NC(C#CC(C)C)=O)CN(C(C2COC(C)C2)=O)CC12CCOCC2 16170,C(CC(C)C(=O)N1CC(C)(NC(=O)C(C)NC(C2CCCC2)=O)C1)OC.C1C(=O)S1 16171,C=CC1(C(=O)N(C)Cc2ccccc2F)CCN(C(c2nocc2C)=O)C1 16172,N(C1CCCc2occc21)C(C(CC(C)C)NC(C1C(C)(C)C1(F)F)=O)=O 16173,c1(OC(F)(F)F)cc(C(=O)NCCNC(=O)CC(C)OC)ccc1F.CO 16174,Cc1cc(C)n(C(C)C(=O)N2CC(N3CCN(N4CCOC(C(N)=O)C4)CC3)C2)n1 16175,c1(C(=O)NCC2CCCN(CCC3CC3(Cl)Cl)C2)cc(F)ccc1-n1ccnc1 16176,N1(C(CNC(CC)=O)=O)CCN(C(=O)CN2CCNC2=O)C(CCC(C)(C)C)C1 16177,Cc1ccc(-c2oncc2C(=O)NC2CN(C(c3ccnn3C3CCC3)=O)C2)o1 16178,Cc1cc(NC(c2cc(C)n(C)n2)c2nnnn2C2CCOC2)ccc1C(C)C 16179,c1(C(=O)NC2C(C)CN(C(c3ccnc(F)c3)=O)CC2)cc2c(F)cccc2[nH]1 16180,c1(C(=O)NCCCN(C(COC)(C)C)C)cc(O)c(OC)cc1Br 16181,N1(C(COC2CCN(C(C=C(C)C)=O)C2)=O)CCC(C)(C)C(C(=O)O)C1 16182,c1(C(N(CCCNC(=O)C(C)=C2CCCC2)CC)=O)ccc(F)nc1 16183,C12(NC(c3cc(C)ns3)=O)CCCC1N(C(c1cn(C)nc1O)=O)CCC2 16184,c1(SC)cccc(C(N2CC(C(C)NC(c3cn(C4CC4)nn3)=O)C2)=O)c1 16185,C1(CC)CCC(C(N2CCC(CC(=O)NC3(CCF)CC(O)C3)C2)=O)O1 16186,CC1CCN(C(c2cn(C)nc2C(C)(C)C)=O)CCN1C(C1CNC(=O)C1)=O 16187,C(=O)(N1OC2C=CC1CC2)C1(C(C)C)CCN(C(C(CCC)OC)=O)C1 16188,Cc1nn(C)cc1C(=O)NC1CCCCC1CNC(c1ccnn1CC#N)=O 16189,N1(C(CCOC(C)=O)=O)CCC(F)(C(=O)NC(c2nc(C)cs2)C)CC1 16190,c1(C(=O)NCC2CC(NC(C3N(C(=O)OC)CSC3)=O)C2)c[nH]nc1[N+](=O)[O-] 16191,c1(C2C(C(=O)NC3C(NC(C4CC(OC)C4)=O)C3)C2)c(F)cc(F)cc1F 16192,C1(NC(C(C)n2cccn2)=O)CN(Cc2ccccc2C(F)(F)F)CC1C#N 16193,c1(C(N2CC(C)C(C(N3CCC(C)(O)C3)=O)C2)=O)cnc2cc[nH]c2c1 16194,N1(C(C(=O)NCC2CCCO2)Cc2ccccc2)CCc2cc[nH]c(=O)c2C1 16195,C1(NC(CSC)=O)CCN(C(=O)COC(F)(F)C(F)F)C1C.c1(S)ccc(OC)cc1 16196,C#Cc1ccc(C(=O)NCC2CCN2C(c2nocc2C2CC2)=O)o1 16197,c1(C(=O)NCC2(NC(c3cnc(CC(C)C)[nH]3)=O)CCCC2)cc(O)cc(=O)o1 16198,C1(C(=O)NCCN(C(=O)CC(C)(C)c2ccccc2)CCC)CC(O)C1(C)C 16199,CC1(C)CCN(C(=O)CCNS(C)(=O)=O)CC1C(N1CCCCC1C1CC1)=O 16200,CCCC(F)C(=O)NC(C)CC1CN(C(c2n[nH]c(C)n2)=O)C1 16201,N1(C(C2C=CCN(C(CC(C)O)=O)C2)=O)CCC(=O)N(C)CC1 16202,C(C(CC(C)C)C(=O)N1CC2=C(C1)CN(C(=O)OC)C2)NC(C(C)SCC)=O 16203,c1(C(=O)OCC)cc(=NC(=O)C2(c3nccc(=N)[nH]3)CCC2)[nH][nH]1 16204,c1(C(=O)NC23CC(CNC(C(CSC)C)=O)(C2)C3)snc2ccccc12 16205,C1(NC(=O)Cc2cccs2)CC2CC1N(C(C1(Cl)CC1)=O)C2 16206,c1(CNC(C(C)N(CCC)C(C2CC2(C)C(F)F)=O)=O)cccc(F)c1C 16207,C=Cc1cccc(-c2ccc(C(=O)Nc3ccccc3N(CCCO)C)s2)c1 16208,C1(CCC)CN(C(c2ncccc2Br)=O)CC1NC(C1COC(=O)C1)=O 16209,c1(N2CCC(N(CCC)C(c3ccc(F)cn3)=O)C2)nc(CC)nc(Cl)c1C 16210,C1(C(=O)NC2(CCNC(CCOC(C)C)=O)CCC2)CCCC1O 16211,C(=O)(C(C)CC(F)(F)F)NC1CN(C(c2cc(C)cc(N)c2)=O)C1 16212,CCS(=O)CC(=O)N1CC(CC(N2CCC(C)(C(N(C)C)CNC(C)=O)C2)=O)C(C)C1 16213,N(C)(C1CCCCCc2ccccc21)c1cc(NCC(C)F)nc(C(C)C)n1 16214,N1(C(CCSCCC)=O)CCC2CCN(C(=O)CCNS(C)(=O)=O)CC12 16215,c1(N2C(N3CCC(C(C)C(N4C(C(C)C)CC5CCCC45)=O)CC3)CCC2)ccc(Cl)cc1C 16216,c1(C(=O)NCCC2N(C(CCCCOC)=O)CCCC2)cnc(N)c(Cl)c1 16217,C1(C(=O)NC2CCC(CNC(CC(=O)NCC3CC3)=O)C2)CCC=CCCC1 16218,C(=O)(C(CCCC)NC(C1CCOC(C)(C)C1)=O)NC(CCC=C)C 16219,c1(NC2CC(NCC(C3CC3)OC)C2)cnc(OCC)nc1 16220,c1(N2C(C)CC(NC(C3CC(C)(F)C3)=O)C2)ncnc2sc3c(c12)CCC(C)C3 16221,Cn1nncc1CC(=O)NC1(C)CC(NC(=O)C=CCSC(C)(C)C)C1 16222,N1(C(C(CSC)O)=O)CC=CC(C(=O)N(C)CCOCCO)C1 16223,c1(OC)cccc2[nH]cc(CC(N3CC(CNC(C4CCC(=O)CC4C)=O)C3)=O)c12 16224,C1(C(=O)NC2(CF)CCN(C(c3c(C)nsc3N)=O)C2)CCc2ncncc2C1 16225,C1(OC)CN(C(c2ccnn2C2CC2(F)F)=O)CC1NC(=O)CSc1cnn(C)c1 16226,C1(c2nc(NC(N(C)C)=O)on2)CCC(c2ccccc2)=NO1 16227,C1(C2CN(C(=O)CC3CCC3OC)C2)(OC)CC1.c1(CC(=O)OCC)ccc(C=O)cc1 16228,c1(C(=O)NC(CNC(=O)Cc2cnccc2Cl)CO)cc(Cl)c([N+](=O)[O-])[nH]1 16229,N1(C(C(C)(C)OC(C)C)=O)CCN(C(=O)CC(C)Sc2ccccc2)C(CO)C1 16230,C1(C(=O)NC(CNC(C(C)OCC=C)=O)C2CC2)CCC(C)(C)O1 16231,CC(=Cn1ccnn1)C(=O)NC(c1ccccc1)CNC(C1(CO)CCC1)=O 16232,N1(CC(=O)NC(C(=O)N(CCF)CC)C2(C)CC2)CCNC(=O)C1 16233,C1(C(N2C(CNC(c3cc[nH]c3)=O)CC(O)C2)=O)CC12CCOc1ccccc12 16234,N1(C(C=Cc2ncn(C)c2)=O)CCC2(CC1)CC2NC(c1csc([N+](=O)[O-])c1)=O 16235,c1(C(N2C(C(C)NC(CCCN(CCC)CCC)=O)CCC2)=O)nc(C)sc1C 16236,C(C(C)CN=c1ccnc(NCCS(=O)C(C)(C)C)[nH]1)OCC 16237,c1(CC(CCC)CC)cc(N)ccc1C(=O)N(CC(C)CNC(=O)C=C(C)Cl)C 16238,Cc1cnc(C(N2CCC(NC(c3cnc(N)c(Cl)c3)=O)C2C)=O)cc1Cl 16239,C1(C2CC2)(NC(CCCC)=O)CCN(C(c2ccc(-n3ccnc3C)cc2)=O)C1 16240,c1(OCC)cnc2[nH]cc(-c3ccnc(C4(C(=O)NC(C)COC)CC4)c3)c2c1 16241,N1(C(=O)CCC2CCOCC2)CC2=C(C1)CN(C(c1cnc3ccnn3c1)=O)C2 16242,O=C(CC(C(F)(F)F)NC(C1CCC2(CC2)C1)=O)NCc1ccco1 16243,C1(C(=O)NCc2csnn2)CC(F)CN1C(=O)CC1CC=CC1 16244,C(=O)(CCC(=O)NC1CC(SCC)C1)OCC.C12CCCCC1CNC2=O 16245,c1(C(N2C(CCC(=O)NCC(CNC(N)=O)O)CCC2)=O)ccc2c(c1)CC2 16246,C1(NC2(C)CN(C(C(=O)OC)=O)C2)CCCN(Cc2ccccc2)C1C 16247,C1(CNC(Cc2cnc(C)s2)=O)CC(C)CN(C(=O)CS(=O)(=O)N(C)C)C1 16248,CC1=C(C(=O)NC2CCCC(NC(c3c(N)cnn3C)=O)CC2)CCCC1 16249,C1(C(=O)NC2C(C)N(C(=O)CC3CC4CC4C3)CC2)Cc2ccccc2NC1=O 16250,C1(C(=O)NCCOC2CN(C(=O)C3CC3)C2)CC2(CCCCC2)C1 16251,C1(C(=O)NC2CCN(C(C(C)(C)OC(C)=O)=O)C2)CCc2[nH]nc(O)c2C1 16252,c1(C(=O)NCC23CC2CN(C(=O)C=C2CCOCC2)C3)cccc2scnc12 16253,c1(C(CNC(C(CC)CC2CC2)=O)(C)C)ccc(F)cc1F 16254,C(=O)(CCC(=O)NCc1n[nH]cc1C(=O)NC1CCC(C)(C)C1)NCC 16255,C1(C)(CNC(C2C(C)CCO2)=O)CN(C(c2ccc(CO)cn2)=O)C(C)(C)C1 16256,C1(C(N(C(CC)CC)C)=O)CC2(CCN(C(=O)CCC3CCCCO3)C2)C1 16257,C(C)(CNC(=O)C(C)(C)CF)(C(C)C)NC(CC(n1ccc(C)n1)C)=O 16258,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CC2N(C(CC3(C)CCCO3)=O)C(CC2)C1 16259,c1(OC)ccc(C)c(C(N2CCCCC2c2cn(CCC(F)(F)Cl)nn2)=O)n1 16260,Cc1[nH]nc(Br)c1C(=O)NC(C)CC(C)NC(=O)CSC1CC1 16261,CC(=O)CCCCC(=O)N1CCC(NC(=O)CC(=O)OC(C)(C)C)CC(O)C1 16262,C1(C(N2C(C)COCC2)=O)CC12CCN(C(c1cc(Br)cs1)=O)CC2 16263,S(=O)(=O)(c1cccc(C2CC2)c1)NC(c1cccc(Cl)c1)c1n(CC)nnn1 16264,c1(C(=O)NC2CN(C(C3CC34CC4)=O)CCC2F)cc2ccnc(Cl)c2s1 16265,c1(C=O)ccc(C2=CCN(N(C)C)CC2)cc1.C1CC1 16266,c1(OC(C)(C)C)ccccc1C=CC(N1CC(COC(=O)Cc2cnsc2)C1)=O 16267,C1(CNC(C(C)(C)C)=O)Cc2ccccc2CN1C(C1CC(S(C)(=O)=O)C1)=O 16268,C1(C(=O)NCC(CNC(COC(CC)(C)C)=O)(C)OC)OC(C)(C)OC1(C)C 16269,N1(c2nccc(C)n2)CCC(C(=O)Nc2cnn(-c3ccccc3Br)c2)C(O)C1 16270,Cc1cc2ccc(C(N3CCC(F)(F)C(CNC(=O)COC4CC4)C3)=O)cc2o1 16271,C=C=C(C)CC(=O)NC1(CN(C)C(C2CCN2C2CCCC2)=O)CC1 16272,N1(C(CC(C=C)CC)=O)CCN(C(=O)CNC(=O)CNC(C)=O)C2COCC12 16273,C(=O)(C(F)(F)C(O)C(C)C)N1CC2(C(NC(c3cccc(C)c3F)=O)CCC2)C1 16274,C1(C(=O)NCCOC(CNC(C2C(COC)C2)=O)(C)C)CC(=O)N(CCO)C1=O 16275,c1(C(N2CCN(C(C)C(=O)NCC(F)(F)F)CC2)=O)nccn2nccc12 16276,c1(C(N(C)CCn2ccnc2)=O)cccc(CNC(C2OC3CCC2C3)=O)n1 16277,Cc1c(Cl)ccc(C(N2CCOC(C)(CNC(=O)C(C)OC(C)(C)C)C2)=O)c1O 16278,c1(C(=O)NC2CC3(C2)CN(C(=O)C#CC2CCCO2)C3)cccc2c1OCCC2 16279,N1(C(C(F)=CCC)=O)CCC2CCCN(C(=O)Cc3cnnn3C)C2C1 16280,C1(OC)CCCCC1(c1nnnn1C1CCCCC1)NCc1ccc(C)cc1F 16281,C1(NC(CC(C)SC)=O)CC2(CCN(C(c3cc(N)nc(Cl)c3)=O)CC2)C1 16282,C1(O)(CNC(Cc2ccc(OC)cc2)=O)CCN(C(=O)Cc2cnns2)CC1 16283,c1(OCCCOCC)ccnc(N2C3CCC2CC3)n1.C1(=O)C(C)(CO)N1 16284,N1(CC(=O)NCC2N(C(Cc3nc(C)[nH]n3)=O)CC=C2)CCCCS1(=O)=O 16285,N1(C(c2nccc(SC)n2)=O)CC2CCC(C1)C(NC(=O)C(C)C(C)COC)C2 16286,C(=O)(NN1CCCC(C(=O)CNC(=O)Nc2ccccc2)C1)c1cnc(C)[nH]1 16287,n1(CC)cc(Cl)c(C(N2CC(CNC(=O)CC(C)(F)F)CC2C)=O)n1 16288,C1(C(=O)NCC23CC(CNC(c4n(C)ccn4)=O)(OC2)C3)CC12CCC(=O)CC2 16289,C1(C(C)C(=O)N(C2(C)CC2)C)CCN(C(C2CC(=O)C2)=O)C1 16290,C(CCCCNC(=O)Cn1ncnn1)NC(C=CC(C)(C)SC)=O 16291,N1(C(=O)C2=CCCC2)CC2(CO)CC1(C(=O)NCC1CC(O)C1)C2 16292,N1(C(c2cccc(C)n2)=O)CCC(NC(=O)Cn2ncc(C#N)c2N)C(C)C1 16293,N1(C(C2(CC)CCOCC2)=O)CCC2CCN(C(=O)CC3(CO)CCC3)CC2C1 16294,C1(C(=O)NC(CC(=O)OCC)C)CCN(C(c2c(C)cnn2C)=O)CC1(C)C 16295,Cc1cc(Cl)ncc1C(=O)NCC1CC(NC(c2nc(Cl)c(Cl)s2)=O)C1 16296,C=C(C)CC(C)C(=O)N1CC2CC2(CNC(=O)CCC=Cc2ccccc2)C1 16297,c1(C(N2C(CN(C(c3nc(Cl)oc3C)=O)CC)CCC2)=O)cnn2ccsc12 16298,N1(C(CCCC#C)=O)CCN(C(=O)CCCc2ccncc2)C(CCC)C1 16299,c1(OC)ccc2cc(C(=O)NC3CC3NC(=O)C(C)S(C)(=O)=O)n(C)c2c1 16300,N1(C(C2(F)C(C)C2)=O)CCC(C2CCCN2C(=O)CCc2ccc(F)cc2)CC1 16301,Clc1ccc2ccc(=NCCc3cnn(-c4ccccc4)n3)[nH]c2n1 16302,C1(NC(C2CC3CCCC23)=O)CCCNC12CC2 16303,c1(C(=O)NC2CCN(C(c3cc(Cl)sc3Cl)=O)CC2)cc(Cl)nc2ccccc12 16304,c1(NC2(COC)CC2)ccc(S(=O)(=O)NCC(CO)C(C)C)cc1Cl 16305,c1(C(N(C(C(=O)OCC)C)C(C2OCCC2n2cccn2)=O)=O)ccc(Cl)cc1Cl 16306,c1(C(=O)NCCOCCNC(C2(C)CNC(=O)C2)=O)cc(Cl)cc(F)c1F 16307,N1(C(CCSCCCC)=O)C(CNC(c2cc(CO)oc2C)=O)CC2COCC12 16308,c1(CCCC)ncc(C(=O)NC2CC(CNC(c3cn(CC)nn3)=O)C2)s1 16309,C1(NC(=O)NC2C(OC(C)(C)C)C2)CN(C(c2cn[nH]c2)=O)CC1O 16310,C1(NC(C2(SC)CC(O)C2)=O)CN(C(=O)CSc2cccc(Cl)c2)CC1(C)C 16311,C(N=c1[nH]cnc2c(Br)nn(C)c12)C1CN(CC=C)C(=O)C1 16312,c1(CC)cc(C(=O)NCC2CCC2NC(C2(C#N)CCC=CC2)=O)cc(F)c1 16313,N1(C(C2CC(OC)C2)=O)CC(CNC(c2cc(C(F)F)[nH]n2)=O)C(C)C1 16314,CCCCCCCCC(F)C(=O)Nc1nnc2c(=O)n(-c3ccccc3O)ccn12 16315,c1(C(=O)OC)ccc(NC2C3CN(c4ccccc4)CC23)c(F)c1 16316,C12(CNC(C=CSC)=O)CCC(CC1)N(C(C1(C)CC1c1ccccc1)=O)C2 16317,c1(C(=O)NC2(CF)CCN(C(C(CCC)OCC)=O)C2)cncc2ccsc12 16318,c1(C(N2C(CNC(C3=C(C)S(=O)(=O)CC3)=O)CC2)=O)n[nH]c2c1CC(C)OC2C 16319,c1(CC(=O)NC(CNC(CCCn2ncc(C)c2)=O)C(C)C)cccc(C)c1F 16320,C(=O)(CC(C)CNC(c1ccccc1CC#N)=O)NCC(=C)Cl 16321,c1(CCCC(=O)NCCCNC(CSCCC(C)C)=O)cc2ccccc2o1 16322,c1(NC(c2ccc(NC(C3N(C(C)=O)CC(O)C3)=O)o2)=O)c(C)ccnc1C#N 16323,c1(C(N2CC(CNC(C(CC)CO)=O)C(C)CC2)=O)cn2cnnc2cn1 16324,C1(NC(C=C(C)C(F)F)=O)CCCCN(C(=O)CN2C(=O)CN(C)C2=O)CC1 16325,C1(CNC(COCc2cc(C)on2)=O)C2CCC(C2)N1C(C1(C#N)CC2CC2C1)=O 16326,N1(C(CSCC#C)=O)CC(C(=O)NC23CCC(CC2)OC3)OC(C)C1 16327,c1(C(N2C(Cc3cccc(F)c3)CCC2)=O)cccc(Cc2n(C)nnn2)c1 16328,c1(C(C)=O)ccnc(C(=O)NCC(O)CCC2(O)CCC2)c1 16329,Cc1ccc(F)cc1C(=O)NCC1CN(C(C2CCCC23CC3)=O)CC1(C)C 16330,C1(N(C(=O)CC2CCCCC2)C)CC2CC1N(C(c1c[nH]cc1C(F)(F)F)=O)C2 16331,C1(CC#C)(C(=O)N(C(C)CNC(=O)Cc2ccnn2C(C)C)C)CCCCO1 16332,N1(C(CNC(CN(C)C)=O)=O)CC(NC(C23CCCC2C3(F)F)=O)C(C)(C)C1 16333,c1(C(N2CCC(NC(C3CC(c4cn[nH]c4)C3)=O)C2)=O)ccc(C2CC2)c(Cl)c1 16334,C(N=c1[nH]c(=NCCCOCC(F)F)c2sccc2[nH]1)C1C(C)(C)OCC1 16335,c1(C(C)C)ncc(C(=O)NCC2CCN2C(C2(CCF)CCC2)=O)cn1 16336,c1(C(N2CCC(NC(CC(CCC)O)=O)CC(O)C2)=O)cnc2c(cnn2C)c1 16337,C#CCCCCCCCC(=O)N(CCCCCNC(=O)C(C)OCC1CC1)C 16338,N1(C(c2n(CC)nc(C)c2)=O)CCCCC(CCC(=O)NCC2CC(CF)C2)C1 16339,N1(C(c2cc(N3CCOCC3)ncn2)=O)CCC(C2CC2(F)F)C1 16340,CCC(F)(F)C(=O)NCC1CN(C(c2ccccc2OC(C)C)=O)C1 16341,c1(C(=O)NCC(O)CCNC(C2CCCCCCC2)=O)cncc2c1CCCC2 16342,C1(N(C(C=C(C)C(F)F)=O)C)CCC2CN(C(=O)Cc3ccsc3C)CC12 16343,N1(C(c2c(COC)ccs2)=O)CC(=O)NC2CN(C(=O)C(C)(C)CF)CCC12 16344,C1(CNC(C(CCOC)(C)C)=O)CC2COCC2N1C(=O)Cn1ncn(C)c1=O 16345,N#Cc1ncn(CC(=O)NC2(CC=CC(=O)NCC3C=CCOC3)CCC2)n1 16346,C(CNC(c1nscc1C)=O)(CC(=O)NCCN1CC2CCC1C2)OC 16347,c1(C(C(=O)N(C(C)C(=O)N2CCC2CC(C)C)C(C)C2CC2)C)ccnn1C 16348,N1(C(CNC(=O)OC)=O)CCCN(C(C2CCS(=O)(=O)N2)=O)C(CC2CC2)C1 16349,C=CCCCN=c1cc(Cl)nc(-c2cccnc2)[nH]1 16350,c1(C(=O)NC2CCCCC2CNC(C2CCCC2F)=O)ccc2cnncc2c1 16351,c1(C(=O)NC2CC(CCNC(c3cncc(C#C)c3)=O)C2)cc(S(C)(=O)=O)cs1 16352,N1(C(Cc2cn(CC)nn2)=O)CCC2(CCC2)C(CNC(c2cn[nH]c2)=O)C1 16353,C(=O)(C#CC(C)(C)CNC(c1c[nH]c(C)c1)=O)NC1CCCN(CC)C1 16354,C(=O)(C(C)CC(C)C(C)=O)N1C(C)(CC(=O)NCC=CCSC)CC1 16355,Cc1cc(C(=O)NCC2CCC(CNC(C34CCCCC3C4)=O)CC2)ccc1F 16356,C1(C(N2CCC(N(C(=O)CCSCC)CCC)C2)=O)CC(F)CN1C 16357,C(=O)(CCCC(OC)OC)NC(CC)CC(=O)N(C)Cc1ccccc1C1CC1 16358,C1(CNC(c2noc(C)c2C(F)(F)F)=O)CN(C(=O)CC(C)(F)F)CCC1(F)F 16359,C1(CCC(=O)NC(C)(CNC(c2ccc[nH]2)=O)C2CC2)CCCCO1 16360,c1(C(=O)NC(C)CCCCNC(=O)C(C)(O)C2CCC2)cn(C)c(=O)nc1O 16361,Cc1cc(F)c(C(N2CCN(C(=O)CC(C)(C)C)CC2c2cn[nH]c2)=O)cc1F 16362,N1(C(C2OCCC(C)(C)C2)=O)CCC2CN(C(C3CCC(=O)O3)=O)CC2C1 16363,n1(CC(=O)NC2CN(C(C(=O)OCC)=O)C3C2C3)nc(C)ccc1=O 16364,N1(C(C(C=C)O)=O)Cc2ccccc2C(C(=O)OC)C1.C12CCN(CC1)C2=O 16365,Cc1cc(CC(=O)NC2CC(=O)N(C3CN(C(c4ccco4)=O)C3)C2)cc(F)c1 16366,c1(CN(C(CC(OCC)OCC)=O)C)cc(NC(=O)C2CC2)cc(O)n1 16367,Cc1cc(C)c(CC(=O)N(C(C(=O)NCc2cncc(O)c2)C2CC2)C)s1 16368,C(C(c1nnnn1C)Nc1ccccc1Cn1ccnc1C)(C(C)C)OC 16369,CC(C(CO)NC(=O)CCN(C)C)NC(C1CC1C(=O)OCc1ccccc1)=O 16370,C1(C)(CNC(CC=CCC)=O)COCCN(C(=O)C(C)C(F)F)C1 16371,N1(C(=O)NC)CC2CCC2(OCCCSC)C1 16372,C1(CNC(c2cnn(CC)c2C)=O)CCCCCN1C(C1CC(C)(C)CO1)=O 16373,c12nc(cc(C(F)(F)F)n1)N(CCC)C1CCN2C1.C1(C=O)CCS(=O)(=O)C1 16374,Cc1ncc(C(N2CC3(CCN3C(c3ccoc3)=O)C2)=O)c(Br)c1Cl 16375,C(=O)(C#CC1(C)COC1)N(CCCCCNC(c1c(C)ccnn1)=O)C 16376,C12(NC(CCOC)=O)CCCC1(F)CN(C(c1nc(O)nc(O)c1OC)=O)C2 16377,c1(C(N2CC(CN(C(=O)C(N)=O)C)OCC2)=O)cn2ccsc2n1 16378,C1(NC(C(CC2CN(C(C3CCN(CCOC)C3)=O)C2)F)=O)C(C)CCC1C 16379,Cc1ccc2nc(C(N3CCOC(CNC(=O)CC4(O)CCC4)C3)=O)c(N)n2c1 16380,C1(OC)CCCC(C(=O)NCC23CC2CN(C(=O)C(CCSC)OC)C3)C1 16381,CC1CN(C(c2cc(Cl)ccc2Cl)=O)CC(C)N(C(c2nnc(O)nc2O)=O)C1 16382,c1(CC(=O)NCC2C(NC(C(C)OC)=O)C2)cc(C)nn1C 16383,C#CCC(O)C(=O)NCC1C=CC(NC(c2cc(Nc3ccccc3)cs2)=O)C1 16384,C1(=CCNC(C(C)n2cncn2)=O)CCN(C(c2c[nH]c(C(N)=O)c2)=O)CC1 16385,C(=O)(NNc1cc(F)ccc1-n1ccnc1)c1ccc(OCC)cc1Cl 16386,C1(NC(c2cc(C(N)=O)ncc2)=O)CN(C(=O)C(F)(F)Cl)CC1(F)F 16387,c1(OC(C)C)ccc(S(N)(=O)=O)cc1C(N1CCC1CNC(=O)C(O)C1CC1)=O 16388,c1(CN(CC(=O)NCCC(C)N(C(C(CSC)C)=O)C)CC)cccc(Cl)c1 16389,C(=O)(CC(C)(CN(C)C)C(F)(F)F)N(C)CC1CCCN(C(C(F)=CC)=O)C1 16390,c1(C(=O)NCC2N(C(CSC)=O)CCC2)ccc(-c2ccc(NC(C)=O)cc2)cc1 16391,Cc1ccc(C2C(C)CN2C(C2(Cc3ccccc3)CCC(=O)C2)=O)cc1 16392,C(Cc1ccccc1)(C(=O)N1CC(O)(CNC(=O)Cc2nc(=N)[nH][nH]2)C1)N(C)C 16393,c1(C(=O)NC(C2CCN(C(c3nn(C)nc3Br)=O)C2)C)ccc(Cl)c(N)c1 16394,C(CC(C(=O)N1CCN(CCOC)CC1)NC(=O)CC1CCCN1C)=CC 16395,C1(NC(c2ccc(COC)cc2)=O)CC2CN(C(C3(C)CCCCO3)=O)CC12 16396,C1(C(=O)NC(CC)CNC(=O)C(=O)NCc2sccc2CC)CCN(C)C1C 16397,N1(C(C)C)CCC(C(=O)NCC2CCCN2C(C2CCCC3CC23)=O)CC1 16398,Cc1ccc(O)c(C(=O)NC(Cn2cncn2)C(=O)NC2(CC3CCC3)CC2)c1 16399,N1(C(C(C)(O)C2CCC2)=O)CCCC2(C1)CN(C(C1C3(CC3)C13CC3)=O)CCO2 16400,c1(C(N(C(C)C(=O)NCc2cc(O)cc(F)c2)CCC)=O)cnn2cccc2c1 16401,Cn1c(C(N2CC3CC3(NC(=O)CC3=NNC(=O)C3)C2)=O)c2n(c1=O)CCCC2 16402,CCCC(C)CC(C)(c1nnnn1C(C)C)Nc1ccc(C(=O)N(C)C)c(C)c1 16403,C12(NC(CCCCC(N)=O)=O)CN(C(=O)CCN3CCCC3)CC1CS(=O)(=O)C2 16404,CC(CC(=O)NC1CCCN(C(c2ccc(C3CC3)cn2)=O)CC1)C(F)F 16405,CC1CCN(C(C2CCN(C(=O)O)CC2)=O)CC1N.C(C)(C)(C)NC(C1(C)CC1)=O 16406,CCCC(CC)CC(=O)N1CC(COC)(NC(c2ccn(CCN(C)C)n2)=O)C1 16407,N1(C(c2nc(OC)oc2)=O)CCC2(NC(c3cn(C)c(C)cc3=O)=O)CCCC12 16408,c1(C(N2C(C(=O)O)C=CC2)=O)cc2c(Cc3ccccc3)cccc2[nH]1 16409,C(=O)(C(C)(C)CC(C)C)NCC12C(CN(C(C3CCC(CC)O3)=O)C1)CC2 16410,Cc1cc(Cl)c(C(=O)N(CC(C)(C)NC(c2onc(C)c2C)=O)C)s1 16411,CCCC(CNC(=O)C(C)SC(C)(C)C)CCO 16412,S(=O)(=O)(c1ccc(NCC2CC(O)CN2C)c(Cl)c1)NC(COC)CCO 16413,c1(OC)ccc(CCC(N2CCCC(NC(C3(C(F)F)CCC3)=O)C2)=O)cc1Cl 16414,CC1CC(C(N2CCCC2CC(=O)NCCOC(F)F)=O)CC(C)C1 16415,c1(CNC(C2CC2Cl)=O)cccc2c1CN(C(c1ccn3nnnc3c1)=O)C2 16416,c1(C(=O)NC23CC(NC(C4CCC5(CC4)CC5)=O)(C2)C3)ccc2c(c1)CCC2=O 16417,N1(C(c2ccc(CSCC)cc2)=O)CCCC(C)(CNC(=O)C(F)C(=O)OC)C1 16418,c1(NC(=O)NCC#C)cc(C)on1.c12ccc(o1)CCCN(CC)C2=O.SC 16419,CC(CC(C)(C)C)NC(=O)C(c1cccs1)NC(=O)CC1NC(=O)NC1=O 16420,C(=O)(CCCCC(C)CC)N1CCC(C)(CCNC(c2c(CC)noc2C)=O)C1 16421,c1(OC)ccnc(CC(=O)NCC2CCCCC2NC(C23CCCCC2C3)=O)n1 16422,N1(C(C(C)(C)C#N)=O)CCN(C(c2ccc(F)nc2F)=O)C(c2ccccn2)C1 16423,C1(C(N2C(C(=O)NCC(O)CO)COCC2)=O)CCC(F)(F)CC1 16424,N1(C(C(C)OC(C)=O)=O)CC(C(=O)NCC2CCCS2)OC(C)C1 16425,N1(C(Cc2n(C)cnc2)=O)CC2CCC2(C(=O)Nc2cc(O)n[nH]2)C1 16426,C1(C(=O)NC(CCCOCCOCCOC)C)Cc2ccncc2C1.C1C(=O)S1 16427,c1(CC(=O)OC)cn(CCCC(=O)OC(F)F)nn1 16428,C1(CNC(c2c(C)scn2)=O)CC2CCC1N2C(C1(C)CC(F)C1)=O 16429,CC(CC1CC1)C(=O)N(CC(C)(C)NC(=O)C(C)n1ccnc1)C 16430,C1(C(=O)N2CCC(CO)C2)(NC(CC)=O)CCOc2ccccc21 16431,CS(C)(=O)=NC(=O)C(=O)NC1CC(c2ccccc2)(NC(=O)COC(F)F)C1 16432,C1(NC(C(COC)OC)=O)CN(C(C2CSCN2C(C)=O)=O)CCN1C 16433,O=C1NCC2(CCN(C(C3(NC(c4cnsc4)=O)CCC3)=O)C2)O1 16434,C(=O)(CC(C)NC(=O)CC1(C)OCCO1)NC(c1nc[nH]n1)CC 16435,N1(C(c2c(CC)[nH]cc2)=O)Cc2nccn2CC(NC(=O)C=Cc2cc[nH]n2)C1 16436,C(c1cccc(CO)c1)=CC(=O)NC1C(NC(C(c2nccc(C)c2)(F)F)=O)C1 16437,c1(OC)ccc(C(=O)N(C(C)CNC(c2ncc(N)nc2C)=O)C)c(Cl)c1 16438,Cc1cc(C(=O)NC(C)(C)CC=CC(=O)N(C(C)C(C)(C)O)C)n[nH]1 16439,CCC(CC(=O)N1CCC1C(OC)OC)c1ccccc1.c12ccc(s1)CNC2=O 16440,N1(C(c2c(C)noc2C)=O)CC2(C1)SCCC2NC(=O)C(O)C1CCCC1 16441,CC(CNC(=O)N(C(c1ccc(Cl)cc1)C1CC1)C1CC1)CC(F)(F)F 16442,c1(OC)cc(Br)cnc1C(=O)NCC1(NC(=O)C(c2cnn(C)c2)=O)COC1 16443,c1(C(c2n(CC(=C)C)nnn2)NCc2ncc(C)o2)cc2cc(Cl)cc(Cl)c2o1 16444,c1(C(C(=O)NC(C(C)NC(c2ccn(CC)c2C)=O)C)(F)F)ccc(C)cc1C 16445,C1(NC(c2occ(OC)c(=O)c2)=O)CCOC2(CCOCC2)C1 16446,N1(C(c2ccc(-n3ccnc3)nn2)=O)CC(NC(C2(F)CC2)=O)CC2(CC2)C1 16447,CC(=O)CCCC(=O)NC(C)(CNC(c1nccc(Cl)c1Cl)=O)C1CC1 16448,n1(CCNC(C(C)C2(O)CCC2)=O)ccc(C(=O)NC2(C(O)CO)CC2)c1 16449,CC1CN(C(C)CCc2ccccc2)CC1CCN1CCCNC1=O 16450,CCCCCC(C)(CC)C(=O)NCCN(C(=O)CCc1ncc(C(C)(C)C)o1)C 16451,C(=O)(CCCCCCn1cc(-c2csnn2)nn1)NC(c1cccnc1Br)C 16452,C(C)(C)(CCN=c1[nH]cnc(C)c1Br)NC(c1c(OC)ccc(C)c1)=O 16453,CC(C)(C(=O)NCC(C(=O)NCC1CCC(C)(C)O1)C(C)(C)C)C(F)(F)F 16454,C#CCN(OC)C(=O)C1C=CCCN1C(C1CCC2(CCC2)C1)=O 16455,C1(CCNC(C2N(C)CC2)=O)CN(C(C2CC(C(F)(F)F)C2)=O)CC1C(F)(F)F 16456,CC(CCC(F)(F)F)NC(=O)CC(C)(C)NC(=O)Cc1ccsn1 16457,C(=O)(C1=CCCCCC1)NCc1ocnc1CCNC(=O)CCC1NC(=O)NC1=O 16458,c1(COC(C)C(=O)NCC2(O)CN(C(=O)Cc3cc(Cl)no3)C2)ccc(F)cc1 16459,Cn1cc(CC(=O)N(CCCNC(c2ccc(F)s2)=O)CC2CCCC2)c(Cl)n1 16460,CCC(CC(F)F)C(=O)N1CCC(CN(C(=O)C(C)c2ccco2)C)C1 16461,c1(CC)nc(C)c(CCC(=O)NC23CCCC2CCN3C(=O)COC)c(O)n1 16462,C(C(=O)NNC(=O)c1ccc(Br)s1)C12CCCCC1C2.c12ccccc1SC2=O 16463,C1(NCC2N(C)CCC2)CC(NC(=O)Cn2cc(Cl)cn2)C12CCC2 16464,C(=O)(CC1=CCCCC1)N1C(CNC(c2ccc(C(C)=O)c(O)c2)=O)C(C)CC1 16465,c1(C(N2C3C(NC(=O)C=CC(F)(F)F)C(CC3)C2)=O)sc2ccccc2c1CO 16466,Nc1nc(C(N2CCC3(NC(=O)CCSC(F)(F)F)CC3C2)=O)ccc1O 16467,C1(CCCC)CCC(C(N2CC(NC(c3cncc(F)c3)=O)C(C)C2)=O)CC1 16468,c1(C(N2CCC(N(C(C=CC=CCC)=O)CCO)C2)=O)csc(=NC2CC2)[nH]1 16469,N1(C(c2cn(CC=C)nn2)=O)CCC(NC(=O)Cc2cccc(C)c2)C(CC)C1 16470,C(c1ccncc1)=C(C)C(=O)N(C1CCC(NC(C2CC2CF)=O)CC1)C 16471,CCC(C)(C)C(=O)NCC1(NC(C2CCC(C)(C)OC2)=O)CCOC1 16472,c1(C(C(=O)NCC2CC2)N(CCC)CC2CC(C)=NO2)cc(Cl)ccc1C 16473,C1(C)(CNC(COC(CC)C)=O)CCCC1NC(c1ccc(C(=O)CC)cc1)=O 16474,CN1CC(C)(C)CC1C(=O)NCC12CC1CN(C(=O)Cc1ncc(F)cc1F)C2 16475,N1(C(c2c(C)c[nH]n2)=O)CCN(C(=O)CC2CC(O)C2(C)C)C(CCO)C1 16476,N1(C(c2cc(Br)ccc2F)=O)CCn2ncc(CC)c2C1.CC(CN(C)C)N(C)C 16477,N1(C(C2CCC(=C)CC2)=O)CCC(C)C(CNC(=O)CCCC(=O)NC)C1 16478,c1(C(N(C2CN(C(C3CCCC3O)=O)C2)C)=O)cccc(O)c1Cl 16479,N1(C(COCCOC)=O)CCOC(CCNC(=O)CN2CCCCC2C)C1 16480,Cc1ccc(C(N2CCC(F)(C(=O)NCCCC(O)C(C)C)CC2)=O)nc1C 16481,C1(CC)CN(C(C2OCCC2C)=O)CC1C(=O)NCCc1ccn(CC)n1 16482,CCC(C)(COC)C(=O)N(CCCCCNC(c1nccc(Cl)c1C)=O)C 16483,C1(O)(C(=O)NCC2CC(NC(Cc3ccn(CC)n3)=O)C2)CCCC(C)(C)CC1 16484,Cc1ocnc1C(N1CCCC1CCC(=O)NCCn1ccnn1)=O 16485,N1(C(=O)OC(C)C)CCCC1C(N1CCCC1C(C)(C)C)=O 16486,C(=O)(C1=NOC(C)C1C)N(CCCNC(c1cc(Cl)cc(Cl)c1OC)=O)CC 16487,CN1CC(N=c2nc3c(cnn3C)c(NCCc3c[nH]c4ccc(F)cc34)[nH]2)C1 16488,c1(N2CCN(CC(C)F)CC2)nc2ccc(F)cc2c(=NCCCC(C)C)[nH]1 16489,C(=O)(C1=Cc2cc(Cl)ccc2OC1)NC1C2CN(C(Cc3cc(C)[nH]n3)=O)C1C2 16490,CC(C)(CC(F)C(=O)NCCC1CCCC2CC12)NC(C1CC2CC2C1)=O 16491,C(=O)(CC1OCc2ccccc21)NC1C2CN(c3ncnc(=N)[nH]3)CC21 16492,c1(C(N(C(C)CCNC(C2CCCC(F)C2)=O)C)=O)cn2c(n1)CCC2 16493,C(=O)(CCCN=[N+]=[N-])N1CC(CCNC(c2n(C(C)C)nnc2)=O)C(C)C1 16494,C1(CNC(c2coc3c2CSC3)=O)CN(C(=O)C=CBr)C2CCN1C2 16495,c1(C(N2CC(c3n(C)ccn3)OCC2)=O)ccc(OC(F)F)c(F)c1 16496,c1(C(C(=O)OC(C)(C)C)N(C)C)ccnc(O)c1.C1(C(=O)OCC)COCC1C=O 16497,C1(C(N(C(C)CNC(=O)CSCC(N)=O)CC)=O)CCC2C(C1)C2(F)F 16498,C1(N(C)Cc2cc(C)c(-c3ccc(O)cc3)s2)CN(CC(F)(F)F)CC1(C)C 16499,C1(NC(C2(C(=O)NC)CC2)=O)CC2CCC1CC2NCc1cc(Cl)ncc1OC 16500,N1(C(CCC#C)=O)CCC2CC(C(N3CCC(F)(CO)CC3)=O)C2C1 16501,C(C)(C)(C(C)CC(=O)NC1(C)CCCC1SC)OC 16502,N1(C(=O)Cc2cc[nH]n2)CC2(CCCCN2C(=O)C(C2CCCCCCC2)O)C1 16503,C1(N(C(C=CC(CC)=CC)=O)C)CN(C(=O)Cn2ncc(Cl)c2C)CC1(C)C 16504,Cc1nnccc1CNC(=O)C(O)C1CN(C(c2ccc(CO)cc2)=O)C1 16505,N1(C(c2c(CC)nco2)=O)CCC2CN(C(c3ccc(O)cn3)=O)CC2C1 16506,C1(C(N(CCOC)C)=O)(NC(=O)Cc2ccc(C)cc2)CCCCC1 16507,Cc1nn(CC(N2CC3C(CNC(=O)CC(=O)N(C)C(C)C)C3C2)=O)cc1Cl 16508,CC1(C)C(C(=O)NCCCNC(=O)C=CSCc2ccco2)C1C#N 16509,NC(CC(=O)N1CCOC(=O)C1)C(=O)NCc1ccco1 16510,c1(OC)c(Br)cc(CNC(C)CC(=O)N(C)C)cc1Br 16511,Cc1cnc2n1CCC(NC1CCS(=O)(=O)CC1)C2 16512,c1(OC)ccc(C(=O)NCCCCCC(=O)NC(c2ncccc2C)C)c(F)c1 16513,S(=O)(=O)(c1cc(C(=O)OC)c(Cl)cc1F)NCC.C1(=O)C(COC)N1 16514,N1(Cc2ncn(C)n2)CCC(C2CCCN(C(c3cc4ncccn4n3)=O)C2)C1 16515,C(C(C)(O)CC(=O)NC1CCC(CNC(c2nc(C)n(C)c2C)=O)C1)OC 16516,c1(CC)[nH]nc(C(=O)NC(CNC(c2ccnc(C(C)C)n2)=O)C(C)(C)C)c1C 16517,c1(C(=O)NCC2CN(C(c3cn(CC=C)nc3)=O)CC2C)cccc2c1NCC2 16518,O=C1CN(C(=O)Cn2ncnn2)C2CCN(C(C3CC=CCC3)=O)CC2N1 16519,C(=O)(CCC(C)NC(C1CC(O)C(F)C1)=O)NC1(C(=O)OC)CC(C)C1 16520,c1(C(=O)NC2CC(C)N(C(=O)C#CC3CCCO3)C2)cc2c(F)ccc(F)c2[nH]1 16521,c1(CC(=O)NCC(C(C)(C)C)NC(c2cnc(S)[nH]2)=O)cc(O)ccc1Br 16522,C1(C(N2C(CNC(C3(CCOC)CCCC3)=O)CC(O)C2)=O)CCCCN1N=O 16523,N1(C(=O)CC2(CO)CC2)CC2CN(C(C3(c4cccs4)COC3)=O)CC2C1 16524,C(=O)(C(F)(F)C1CC1)NC(C1CCCN1C(c1nnn(C)n1)=O)C 16525,N1(C(C2CC(=C)C2)=O)CC(N(C)C(c2cccc(F)c2C)=O)C(C)(C)C1 16526,C(=O)(C1=NOC(C)C1)N(CCCC(=O)NC(CCOC)COC)C 16527,NS(=O)(=O)c1cccc(C(=O)NCc2nc(CO)cs2)c1 16528,C(=O)(C1=CCC2CCC1N2C(=O)C(C#N)C(C)C)NCC(COC)C 16529,C1(NC(c2cncc(SC)c2)=O)CC2CCC(C1)N2C(=O)CC(C)F 16530,C1(C(=O)NCCC(C)(C)NC(COCc2ncc(C)o2)=O)CC2(CCC2O)C1 16531,N1(C(COC(CC)(C)C)=O)CC(C(N2CCOC(C3(C)CC3)C2)=O)C(F)C1 16532,CN=c1[nH]c(C(N2CC(CCNC(C3CCN(CC(F)(F)F)CC3)=O)C2)=O)cs1 16533,c1(OC)ccc(C(C)NC(C2CCCCC2(F)F)=O)cc1Cl 16534,C(=O)(C(CNC(c1cc(C(N)=O)[nH]n1)=O)OC)NCC(=C)Cl 16535,C1(O)(CCNC(CSS(C)(=O)=O)=O)CCN(C(=O)Cc2sccc2Cl)C1 16536,N1(C(C(C(C)C)(C)C)=O)CCCC(NC(C2CC=CCC2)=O)C(F)C1 16537,Cc1ncccc1CC(=O)NC1CC1CNC(=O)COCCCF 16538,C(=O)(C(C)CCCOC)N1CCC(C(CNC(C(C)OCCC=C)=O)F)CC1 16539,c1(SCC(=O)NC(C2CCN(C(C(CC)F)=O)C2)=O)ccc(Br)cc1C 16540,c1(CC)nccnc1C(=O)NCC=C1CCN(C(=O)CC2CCOC2=O)CC1 16541,C1(NC(=O)COCC2CCCO2)CC(F)CN(C(=O)CCc2cc(F)cc(F)c2)C1 16542,N1(C(C=C2CCC(C)C2)=O)CCC2CN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CC12 16543,S(=O)(=O)(c1ccc(C#N)c(N2Cc3ccc(C)cc3C2)c1)NCC(CC=C)(C)C 16544,Cc1c(NCC(C)N(C)C)nc[nH]c1=NCCS.N1(CC2(C(=O)N)CC2)CCOCC1 16545,N1(C(C(=C(C)C2CC2)F)=O)CCCCC(CNC(c2cc(SC)n(C)n2)=O)C1 16546,c1(C(N(c2ccc(CO)cc2F)C2CCCC(=O)CC2)=O)cc2n(n1)CCCO2 16547,N1(OCC)CCC(N(C2CCN(c3ncccn3)CC2)CCO)CC1 16548,C1(C(N2CCC(CC(=O)O)(C(=O)NCc3cccnc3)C2)=O)CCOC(=O)CC1 16549,C#CC1CCN(C(=O)C(CN(C)C)NC(=O)CCOCC(C)(C)C)CC1 16550,c1(C(=O)NC(C2COCCN2C(C2CC(=O)C2(C)C)=O)C)cc2nc[nH]c2cn1 16551,N1(C(C(C2CCN(C(=O)CCCC3CCCO3)C2)C)=O)CCCC2(CCC2)C1 16552,C12(CNC(C(C)(C3(C)CC3)OC)=O)CN(C(=O)CC3C=CCCC3)CC(F)(C1)C2 16553,CC1(C)CC(NC(c2ccc(-c3cccs3)o2)=O)CN(C(c2cccnc2)=O)C1 16554,N1(C(C(CC=C)CNC(C2C3(CC3)C23CC3)=O)=O)CCc2ccc(F)cc21 16555,N1(C(C)=O)CC(CC(c2ccc(Cl)cc2Br)=O)Oc2ccccc21 16556,c1(C(N2CC(COC)(CNC(C3CC3C)=O)C2)=O)noc2ccc(Cl)cc12 16557,N1(C(Cc2cc(C)cc(Br)c2)=O)CCCC2(NC(=O)CCC=CC(C)C)CC2C1 16558,S(=O)(=O)(c1cc(Cl)sc1Cl)NC(C(=O)OCC)Cc1cncs1 16559,c1(Oc2cncc(CN(C=O)CC3CC(C=C)C3)c2)cc(C)cc(C)c1 16560,CC1CN(C(c2ccoc2)=O)CCC1NC(c1cccc(C#N)n1)=O 16561,C1(C(N2CCCC(C)(C)C2)=O)CCC2CCC1N2C(c1cscc1F)=O 16562,C(C(C)(C(=O)N1CC(C)(CO)C1)NC(=O)Cc1ccc(C)nc1)SC 16563,c1(NC(C2(CNC(c3cc[nH]c3)=O)CCCC2)=O)cccc(-c2nccs2)c1 16564,C1(NC(CSCCC)=O)CCCN(C(c2c[nH]cc2C(C)(C)C)=O)CC1 16565,C1(C2(O)CCC2)(C(N2CC(CC(N3CCC4(CC4)C3)=O)OCC2)=O)CC1 16566,C1(C)(N(C(=O)Nc2cnc(COC)o2)C)CN(C(=O)OC(C)(C)C)C(C)(C)C1 16567,Cc1ccc(Cl)c(CN(C)CC2CCN(C(c3c(O)cccc3Cl)=O)CC2)c1F 16568,n1(CCC2c3nnnn3C2)cc(Cl)cn1.C1(C(C)CN)CCCC1.C1CC1 16569,N1(C(c2c(C)c[nH]n2)=O)CCOCC(CNC(=O)C(C)OC2CCCCCC2)C1 16570,Cc1c(C(N2CC(CNC(c3cc(C4CC4)no3)=O)C2)=O)nnn1C 16571,N1(CC)CC(C(=O)NC2CCC2NC(=O)C=C(Cl)Cl)CCC1=O 16572,c1(C(=O)OC)cccc2c1CCC2NC(C1CCC(C(F)(F)F)N1)=O 16573,C1(CC(=O)NCCCCNC(C2CCCC2)=O)(NC(C)=O)CCCCC1 16574,C1(NC(C2N(C)CCCC2)=O)C2CC3C(C2)C13C(=O)NC1(C2CC2)CC1 16575,c1(C(N2C3CC(C(=O)NC(CC#C)C(=O)NC)C2CC3)=O)ccn2ccccc12 16576,C1(NC(C2ON=C(C)C2)=O)CCOCC1NC(=O)CCCC1CCC1 16577,c1(CC(=O)NCC(N(C(C(C2CCC2)OCC)=O)C)C2CC2)sc(O)nc1O 16578,C1(OC2CN(C(C(C)OCC#C)=O)C2)CCN(C(=O)C=Cc2csc(C)n2)CC1 16579,N1(C(C2COCCN(C(C=CC(C)(C)C)=O)C2)=O)CCCc2ccccc21 16580,C1(N(C)C)CCCN(CC(=O)Nc2ccc(N(C(CN(S(C)(=O)=O)C)=O)C)cc2)C1 16581,CCCCN=C(NCCc1ncc(C)cn1)NC(C)CCC(C)C 16582,CC1OCCOC1C(=O)NC(C)(C)CC(=O)N1CCC(C(N)=O)C1 16583,c1(C(=O)NCC2CCN(C(=O)Cc3cn[nH]c3)C2)cc2n(n1)CCO2 16584,C1(N(C(=O)C(F)(F)c2nccs2)C)CCN(C(=O)CCc2ncco2)CC1 16585,C1(CC=CC)CCCN(C(=O)CC(C)(C)NC(=O)C=C(C)C(C)(C)C)C1 16586,CCCCCC(C(=O)N1CCC(NC(c2ccn(C(F)F)n2)=O)C1)C(C)C 16587,C1(C(=O)NCCC2(NC(C(CC)F)=O)CC2)CCCCN1C1CCCC1 16588,N1(C(C2(C#C)CN(C(c3cc(C)ccc3O)=O)C2)=O)CCC(C2CCC2)C1 16589,CC(C)(F)CC(=O)NCC1COC(CNC(c2ncsc2Br)=O)C1 16590,C(=O)(C1=NN(C(C)C)C(=O)CC1)N1C(CC)CN(C(c2ccnc(Cl)c2)=O)CC1 16591,CS(=O)CCC(O)C(=O)NC12CC(NC(=O)C=Cc3cccs3)(C1)C2 16592,CCCCCC(O)C(C)C(=O)NC(C)CC1CN(C(C2Cc3nccn3C2)=O)C1 16593,c1(C(=O)NCC2C(CC(=O)NCCSCC#C)C2)ccccn1 16594,C=CC1CN(C(C2(N(C)C)CCCC2)=O)CC1NC(=O)CC(C)C1CCCCC1 16595,N1(C(c2ccc(C(C)=O)o2)=O)CCCC(CC(=O)NC2CCCC2C)C1 16596,c1(NCCS(=O)(=O)NC)nccc(=NC2CC3CSCC(C3)C2)[nH]1 16597,C1(C(C)C(=O)NCCc2ccccc2)CCCN(C(C2CC(F)(F)C2)=O)C1 16598,C1(CNC(CC=C)=O)CCCCC1NC(c1cnn(CCOC)c1)=O 16599,Cc1oc(C)c(C(=O)NC2CCCC(N(C)C(C3CC(Cl)(Cl)C3)=O)C2)c1C 16600,C1(C(N2C(C)(CNC(=O)CC3C=CCC3)CCC2)=O)CCCC12CCC2 16601,C1(CCNC(CCC=C)=O)CN(C(=O)C(F)CC)CCCO1 16602,N1(C(C(C)C2CCOC2)=O)CCCCC1CNC(c1cnsc1)=O 16603,C1(CNC(C(CN(C)C(C2CCC=CCCC2)=O)(C)C)=O)CC2CCCC2C1 16604,Cc1cc(=NC(C)CCNC(C2(F)CCC2)=O)c([N+](=O)[O-])c(C)[nH]1 16605,c1(C(=O)N)ccccc1.c1(C(N2N(C)CC2)=O)c[nH]c(=N)s1.c1(C)ncc[nH]1 16606,CC(C)CC(C(=O)NC(CN1CCOCC1)CO)NC(=O)NC1CCC1 16607,N1(C(CC(C)OC)=O)CCCC(C)(C(=O)Nc2cccc(F)c2)C1 16608,c1(OCC)ncc(C(C(=O)NCC(F)F)N(C(c2ccc(Br)cn2)C)CC)cn1 16609,Cc1c(NC(C23CCC(C(N4CC(O)C(F)C4)=O)(CC2)C3)=O)nc2ccccn12 16610,C1(CNC(C2C(CC)CC2)=O)CN(C(C2(C3CCCO3)CCC2)=O)CCC1C 16611,C=CCC(C(=O)N1CCCC1CCNC(C1CN(C(N)=O)C1)=O)C(C)(C)C 16612,c1(C(=O)NC2CCCCN(C(C3CC(C)NC(=O)C3)=O)C2)cn2cccnc2n1 16613,CCCC(C(=O)N1CC(O)CC1CC(N1CC2(CC(OC)C2)C1)=O)C(C)C 16614,CC1CN(C(c2cc(=O)cc[nH]2)=O)CC1CNC(=O)CC1CC1C(F)(F)F 16615,C1(NC(C(=O)N(c2nccs2)CC)=O)C2CCC1(c1ccnn1C)C2 16616,S(=O)(=O)(c1ccc(Cl)cc1)N(CC(=O)NCC1CC(NC(CCC(=C)Cl)=O)C1)C 16617,CCCC(CCCNC(c1ccc(CO)nc1)=O)NC(=O)CN(C)C(C)=O 16618,C1(CNC(C(C(CC)C)O)=O)C(C2CC2)CCN1C(c1ccsc1C)=O 16619,c1(CN2CCC(NC(c3cncc(Br)n3)=O)C2)cc(O)cc(O)c1 16620,C1(C(N2CC(N(C)C(c3csc(=N)[nH]3)=O)C(F)C2)=O)CCC2(CCC2)CC1 16621,C1(C(N(C(C2CCCC2)CO)C)=O)CN(Cc2ccc(C#N)s2)CCN1 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16640,c1(C(N2C(C)CN(C(C3CC34CC(O)C4)=O)CC2)=O)cc(Cl)c2[nH]c(O)nc2c1 16641,N1(C(N=c2n(CC(C)C)[nH]cn2)=O)CCCC2CN(C)CC12 16642,Cc1cc(F)c(I)cc1C(=O)Nc1cc(C(=O)NC(C)C(C)C)[nH]n1 16643,CCCC(C(F)(F)F)c1nc(-c2cc(OC(C)C)ccn2)nn1CCN(C)C 16644,c1(OCCOC)ccc(C(=O)N(CC(C)NC(=O)Cc2ccccc2)C)cn1 16645,C1(Nc2cc(NCCCN(OC)C)nc(COC)n2)CCS(=O)(=O)C2(CCC2)C1 16646,C1(C(=O)Nc2cnc(C)nc2)C2CCC(C2)C1NC(C1CC1C)=O 16647,C1(C)(NC(CC(=O)OCC)=O)CCCN(C(C23CCC(CC2)C3)=O)C1 16648,c1(C(N2CC(CC(CNC(C(C)CC(F)F)=O)(C)C)C2)=O)c(O)cc(Cl)cc1F 16649,N1(C(C(CSC)C)=O)CCC(C(=O)NC2CCC23CCCC3)C12CCC2 16650,C12CC1C1CCCN(C1)C2.O=C1CCCCN1CCCC(=O)Nc1cc(O)ncn1 16651,c1(C(=O)NC2CC(N(C)C(c3[nH]nnc3C3CC3)=O)C2)cccc(F)c1C1CC1 16652,C(=O)(C1=CCCOCC1)C(c1n[nH]c2c1CCSC2)=O.C12CCN(C1)C(=O)CC2 16653,c1(OC)cc(Cl)c(CN2CCC3CN(C(=O)C=CCBr)CC23)cc1OC 16654,C1(NC(=O)OC(C)(C)C)(OC(C23CCCC2CCC3)=O)CCS(=O)(=O)C1 16655,c1(N(C2CCCCC2)C(COC)=O)cc(Cl)c2ccccc2n1 16656,c1(C(=O)NC2C(CN(C(C3OCCN(CC)C3)=O)C)CCC2)cc(=O)c(C)c[nH]1 16657,C(=O)(CCC(=O)NN(C)C)N1CCC(C(CO)NC(C(CCC)OC)=O)CC1 16658,S(=O)(=O)(c1cccc(C(=O)NCc2cc(C)cc(Br)n2)c1)Nc1ccc(C)s1 16659,C1(O)(C(N(C)CC2CCCN(C(c3ccnnc3O)=O)C2)=O)CCCC(C)CC1 16660,C(C(=O)NCCCF)(C1=CCSC1(C)C)N(C(C(C)OCCCC)=O)CC 16661,CCC(CC)(CC)C(=O)NCC1CN(C(=O)CN2CCC(CO)CC2)C(C)(C)C1 16662,c1(NC(C2C(NC(c3c[nH]c(Br)c3)=O)CCC2)=O)ccc(N2CCCC2=O)cc1 16663,C1(CCC)CN(C(C2CC3CCC2O3)=O)CCN1C(c1c[nH]nc1OCC)=O 16664,c1(C(=O)NC(CC)CNC(=O)CC(C2CC2)NC2CCC2)n[nH]c2c1CCC2 16665,C(=O)(C(CCF)NC(c1ncccc1C)=O)NCC=C=C 16666,C(CCC(=O)N(C)CCNC(C1CCCC1CC)=O)N(CCC)CCC 16667,Cc1nc(C)c(C(C)NC(C2(CO)CN(C(=O)C(C)n3ccnn3)C2)=O)s1 16668,N1(C(c2c(N)cccn2)=O)CCC(C2CCCN(C(C3CCCO3)=O)CC2)CC1 16669,c1(C(C)NCC2C(C)(C)C2(C)C)ccc(Cl)cc1F 16670,CC1(C)CCC(=CC(N2CCCCC2CNC(c2n[nH]cc2[N+](=O)[O-])=O)=O)CC1 16671,c1(CCC(=O)N(C2CCN(C(C3CN(C(C)C)C3)=O)C2)CC)n[nH]c(=N)s1 16672,C12(C(=O)NCCC(C)NC(Cc3cc(C)ns3)=O)CC(C)(C1)OC2(C)C 16673,c1(OC)cc(C(=O)NC(Cc2cnn(C)c2O)C(=O)N2CC(CCO)C2)n(C)n1 16674,C1(OC)C2CC3CN(C(c4scc(Cl)c4Cl)C(=O)NC4CC(F)(F)C4)C1C3C2 16675,C1(NC(Cc2c(C)ccs2)=O)C2CC3CN(C(=O)CC4(C)CCCO4)C1C3C2 16676,c1(NC(C(CNC(COCC(=O)NC)=O)C)=O)csc(C#N)c1 16677,C(=O)(C(CCC)NC(=O)C(n1cc(CC(C)O)nn1)C)OCC=C 16678,Cc1cc(F)cc(C(=O)N(CC(C)NC(c2nc(C)n(C)c2C)=O)C)c1N 16679,CC(C)C1=NOC(C)(C(=O)NCC(CNC(=O)CC(=O)N(C)C)S(C)(=O)=O)C1 16680,n1(CCC)nnnc1C(C1(C)CC(C)C1)NCC1CN(CC(F)(F)F)C1 16681,CCC(C)CCC(=O)N(CCC(C)NC(c1cnn(CCN(C)C)c1)=O)C 16682,c1(NC)ccc(C(N2CC3CC(NC(c4cc(C)c(C)o4)=O)C2C3)=O)cc1F 16683,N1(C(C(C)OCCC=C)=O)CCN(C(=O)CC)CC(COC)C1 16684,c1(C2CCCN(C(C3CCC4(CCC4)CC3)=O)C2)nc2cccnc2[nH]1 16685,C12(C(=O)NCCOCCNC(C3CCS(=O)(=O)N3)=O)CCN(CC1)CC2 16686,c1(C(=O)NCCN(CC(C)O)C(C23CC4CC2C3C4)=O)nccn2nccc12 16687,c1(C(=O)NCC(C)NC(C(CC(C)C)OC)=O)ccc(C(C)=O)cc1F 16688,C1(C(=O)NC2C(NC(C(C=CC)O)=O)COCC2)C2CCC1(C)C2(C)C 16689,c1(CN2CC3C(C(=O)NC4CCCCC4(F)F)C3C2)cc(F)cc(F)c1F 16690,Cc1cnc(CCC2(CSc3noc4c3CCC4)CCCO2)nc1O 16691,Cn1c(C(=O)NCC2(F)CC(NC(=O)C(C)(F)c3ccccc3)C2)nnc1S 16692,N1(C(C2=CCN(C(c3c(C(C)C)c[nH]c3)=O)C2)=O)CCC(=O)N(C)CC1 16693,N1(C(C(=O)NCc2cccc3cccnc23)=O)CCSC2(CCCCC2)C1 16694,c1(C(N2CCC(NC(C(COC)N(C)C)=O)C2(C)C)=O)cnc2n1CCCCC2 16695,CCCCC(O)CC(=O)OCc1nc(N2CCCCC2)cc(C(F)(F)F)n1 16696,C1(C(N2C(CNC(=O)C=Cc3cnccn3)CC(F)C2)=O)C2C3CCC(C3)C12 16697,c1(C(=O)NCC2C(NC(C3CC(C)(C)C3)=O)CCC2)c[nH]c(=O)cn1 16698,C1(NC(CCCCCSC)=O)CN(C(c2scnc2C(F)F)=O)CC2CCCC12 16699,c1(C(N2CC(C(=O)NC3CC4CCC3O4)(COC)C2)=O)ccc(C)nc1 16700,c1(CCC(=O)NC2CCC(NC(CN(CCOC)C)=O)C2)cc(F)cc(F)c1 16701,C1(NC(c2c(SCC)nccn2)=O)COC2CN(C(c3cc(OC)no3)=O)CC12 16702,C(=O)(C(CCOCCO)NC(=O)CCC1(C)N=N1)N(CC(COCC)O)C 16703,C=CCC(C(=O)NC(C)CNC(=O)Cc1ccsc1)NC(=O)OC(C)(C)C 16704,c1(C(=O)NC(CNC(C(CCC)C(C)C)=O)(C)C)cc(O)nc2cnccc12 16705,C(C1=NOC2CN(C(C3(C#N)CC=CC3)=O)CC12)NC(c1ccc(OC)s1)=O 16706,c1(C(=O)NCC2(F)CCCN(Cc3c(C)ccc(C)c3)C2)c(Br)ccc(C)c1F 16707,C1(NC(c2c(C)ccn2C)=O)COC2(CNC(=O)CSc3n[nH]c(=N)s3)CC1C2 16708,C1(C(=O)NCCCNC(=O)CC2C=CCCC2)C(Cl)(Cl)C12CC2 16709,c1(OC)cncc(NC(C2(O)CCN(C(=O)C(C)(C)N3CCCC3)C2)=O)c1 16710,N1(C(Cc2nnc(C)o2)=O)CCCC12CCN(C(c1cn(C(C)(C)C)cn1)=O)C2 16711,S(=O)(=O)(c1ccc(NC2CCCCCC2CO)c(F)c1)NC(CC)CSC 16712,C1(NC(C(C=C)(C)CC)=O)CC2(CCN(C(C3(C#N)CCCC3)=O)CC2)C1 16713,C(CC1=CCN(CCOc2cccc(Cl)c2)CC1)NC(c1n(C)cc(Cl)c1)=O 16714,CC1=C(c2ccccc2)CN(C(c2ncncc2Cl)=O)CC1 16715,CN1CCC(NC(=O)NCC2CCN(c3ccccc3Br)C2)CC1=O 16716,n1(C(C)C)cc(C(=O)NC2(C)CN(C(=O)CN3CCCC3C)C2)c(O)nc1=O 16717,c1(C(C)NC(c2ccc(OC)cc2)C(=O)O)cc(Cl)cc2c1OCC2 16718,CC1CC2(CC(C(=O)Nc3c(CN4CCN(C(=O)C(C)C)CC4)sc(=N)[nH]3)C2)C1 16719,C1(C(=O)NCCCn2cc(-c3cc(C(F)(F)F)ccn3)nn2)CN2CCC1C2 16720,Cc1nc2cccc(C(N3CC(CNC(c4ccc(=N)[nH]c4)=O)CC3C)=O)c2[nH]1 16721,N1(C(c2nc(Cl)cs2)=O)CCN(Cc2ccc(Br)c(F)c2)C2CC12 16722,N1(CCC(=O)OC)CCC(NC(=O)NC(c2snnc2C)C)CC1 16723,c1(C(=O)NCCC2(CNC(COCC=C)=O)CC2)ncn2c1CCC2 16724,C1(CNCCOCCOCCOCC(C2C(C(=O)SCC)CC2)=O)CCCCO1 16725,c1(C(N2CC3N(S(C(C)C)(=O)=O)C3C2)=O)cccc(Br)c1[N+](=O)[O-] 16726,C1(NC(C23CC(C(=O)Nc4cccc(CO)c4)(C2)C3)=O)CCC2CCC(=O)N2C1 16727,N1(C(C2(CNC(c3ccn(C)c3C)=O)CC(=C)C2)=O)CCCC(CC(C)C)CC1 16728,N1(C(C(C)(C)C(N)=O)=O)CCCCC(CNC(=O)CC2CCSCC2)CC1 16729,c1(C2(C(N(CC(O)CNC(C3C4CCCC34)=O)C)=O)CC2)ccc(F)cc1Cl 16730,N1(C(C(CNC(CC)=O)(C)C)=O)CCCC2(CC(NC(=O)C(C)C3CCC3)C2)C1 16731,N1(C(C(C)CN(C)C)=O)CC2CC(NC(=O)CCC3CCC3)CC1C2 16732,N12CCC3(CCN(C3)C1=O)C2.c1(NC(c2cccc(Br)c2)=O)c(F)cncc1F 16733,N1(C(CC2(NC(=O)Cc3nncs3)CCC2)=O)CCC(C2CC2)C1 16734,C(=O)(C(CO)C(C)(C)C)NC(C(=O)NCC(C(=O)OC)C)C 16735,N1(C(c2c(C)snn2)=O)CCCC(O)(CCNC(=O)C(O)C(F)(F)F)C1 16736,C=CC(C)CC(=O)N1CCC(O)(CN(C(=O)CNC(=O)CC(F)(F)F)C)C1 16737,C(CNC(c1[nH]nnc1C(F)F)=O)(C(C)C)NC(C1CN(S(CC)(=O)=O)C1)=O 16738,c1(CC(=O)NC2CC(CNC(c3cc(F)cs3)=O)C2)nnc(O)s1 16739,C1(C(=O)Nc2cc(OC)cc(C(=O)O)c2)CCc2nnc(C(F)(F)F)n2C1 16740,C1(C(=O)NCCc2c(C)n[nH]c2)CCCCC1NC(=O)CCCC1CC1 16741,C1(NC(C2C(OC)CCC2)=O)CCN(Cc2ncc(C)o2)CC(C)(C)C1 16742,N1(C(=O)COCCc2ccccc2)CC2CN(Cc3c(Br)ccnc3Br)C2C1 16743,C1(C(=O)NC2(CNC(c3c(C)[nH]cc3)=O)CCOCC2)CC12CCOCC2 16744,c1(OC)cc(C(=O)N(CCCNC(=O)COC2CC2)C2CC2)cc(Cl)n1 16745,c1(CC)ccc(C(=O)N(C)CCNC(c2ccccc2CS(C)(=O)=O)=O)cn1 16746,c1(C(c2n(CCC)nnn2)NC2CC(CNC(C)=O)C2)cc(Br)cc(F)c1O 16747,c1(C(=O)NC2CC(O)CN(C(c3ccnc(Cl)c3O)=O)C2)cnc2nccn2c1 16748,N(C(=NCCCC(C)(C)C)NC1CCCCC1)C1C(C)CCCC1 16749,C1(NC(C(=Cc2cccs2)C)=O)CC2(CCN(C(=O)CCc3n[nH]c(=N)s3)C2)C1 16750,C1(NC(c2n[nH]cc2Cl)=O)CCN(C(c2nnc(O)cc2O)=O)C(C2CC2)C1 16751,C1(N(C(CCOC(C)(C)C)=O)C)CCCCN(C)C1=O.C(C(O)C)N(C)CCO 16752,c1(C(N2CCN(C(c3c(SC)ccs3)=O)C(CO)C2)=O)cccn2nncc12 16753,C(CCCCC(=O)NC)NC(=O)CC.n12cc(cn1)-c1cn(nn1)CCN2CC 16754,C(=O)(C1=NOC2(CCNC2)C1)N1CC(C)N(C(=O)Cc2ccc(F)cc2)CC1 16755,C1(CNC(C=C(COC)C)=O)CC(C(C)C)CCN1C(=O)CCCc1ncco1 16756,N1(C(c2ccn(CC)n2)=O)CC2CN(Cc3ccc(C)cc3C)C2C1 16757,N1(C(=O)C=C(Cl)Cl)CCN(c2cc(Cl)ncn2)C(c2cc(F)ccc2F)C1 16758,C1(CC(NOCCCC)=O)CCN(C(c2ncoc2C)=O)CC1 16759,C(=O)(CC(F)(F)Cl)NCCOC1CCN(C(C2CC(CC(C)(C)C)C2)=O)C1 16760,CC1CC(CNc2nc(C3CCCCC3(F)F)no2)CC(C)C1 16761,CC(CC(=O)NC1C(C)(C)CN(C(c2c[nH]c(=N)s2)=O)CC1(C)C)CC(C)(C)C 16762,Cc1ccc(CNCC2(CO)CCCCO2)cc1C1CC1 16763,CN1CCOC(C(=O)NCC(C2CCCC2)NC(c2cnc(N(C)C)s2)=O)C1 16764,C#CC1(C(N2CC(CO)CC2CO)=O)CN(C(=O)C(COC)OC)C1 16765,C(=O)(CCC(=O)N1CCOC(CNC(=O)CN2CCCC2=O)C1)OC 16766,c1(Cn2c(N3CCC(C)(NC(=O)OC)C3)nnn2)c(C)sc(C)c1OC 16767,N1(C(c2ccc(OC)cn2)=O)CCC(N2CCC(CCCO)CC2)C2(CC2)C1 16768,N1(C(C2C(C)C2)=O)CCC(C2CCCN(C(c3cc(C(N)=O)ccn3)=O)C2)C1 16769,N1(C(c2cnn(C3CCC3)c2)=O)CC2CCCC2(Nc2cc(C(F)F)ncn2)C1 16770,c1(OCC(=O)OC)ccc(OCC(=O)NC(=O)C(C(C)C)NC(C)=O)cc1 16771,C=Cc1ccc(C(N2CC(NC(=O)CCc3ccsc3Cl)CC(O)C2)=O)cc1 16772,c1(C(N2CC(O)(C(C)NC(=O)C(C)C3CCOC3)C2)=O)cc2n(n1)CC(F)C2 16773,CC1CCN(C(=O)Cn2cncn2)CCN1C(=O)CC1CC2(CC2)CO1 16774,CC(C)(C(=O)N1CCC1CNC(c1cncnc1O)=O)C1=CCS(=O)(=O)CC1 16775,c1(C(=O)NC(CNC(C2(CN=[N+]=[N-])CC2(F)F)=O)C)ccc(C(N)=O)cn1.CC 16776,c1(C(N2C(CC(N3CCC(NC(C)=O)C3)=O)CCC2)=O)nccc(Cl)c1F 16777,C1(NC(c2nc(C)oc2)=O)CCN(CCNC(C2CCS(=O)(=O)C2)=O)CC1 16778,N(C1c2ccccc2CC1NC(=O)C(C)CS(C)(=O)=O)C(CC(CCC)(C)C)=O 16779,C(=O)(C1=CS(=O)CCC1)NCCN(C(c1cn(C(F)F)c(C)n1)=O)CC 16780,c1(C(=O)NCC(CN(C(c2c(C)[nH]oc2=N)=O)C)O)ccc(Cl)c(O)c1 16781,N1(C(c2nccc(C)n2)=O)CC(N(C)C(c2oc(C)cc2C)=O)C2(CC2)C1 16782,c1(OC)cc(C(=O)NCC(O)CN(C(=O)C=C2CCOCC2)C)c(OC)cc1Cl 16783,Cc1ccc(N)c(C(N2CCC(C(F)(F)F)C(NC(C3(CO)CC3)=O)C2)=O)c1 16784,c1(C(N2CCN(Cc3cccs3)CC2)=O)cn2ccc(Cl)cc2n1 16785,N1(C(c2cc(C)oc2C(F)(F)F)=O)CCc2cc(C(C)(C)C)ccc21 16786,C1(C)(CC)C=C(C(=O)NC2CN(NC(c3ncccc3SC)=O)CC2C)C1 16787,C1(C(N(CC(C)O)CCNC(C(CC(C)C)N(C)C)=O)=O)CCC2C(C1)C2(F)F 16788,c1(C(N2CCCCC2C2CCN(Cc3cscn3)C2)=O)cc(C(F)(F)F)ncn1 16789,Cc1cc(C(=O)NCC(C)(O)C(=O)O)ccc1S(=O)(=O)N1CCOCC1 16790,N1(C(CCC)=O)CCCC1(C)CNC(C1CC(C(=O)NC)C1)=O 16791,C1(NC(C)=O)(CO)CCN(C(=O)NC2CCN(C(c3ccccc3)C)C2)C1 16792,C(=O)(C1CCCc2nn[nH]c21)N(C)CCNC(c1cccn1-c1cnccn1)=O 16793,C1(CNS(C)(=O)=O)CC2CC2N1C(=O)NCCc1ccc(F)cc1.c1(C)cnc[nH]1 16794,c1(C(C(=O)NCC(F)F)N(C)Cc2nc(CC)sc2)cc2c(s1)CCOC2 16795,C(=O)(C(F)CC(C)(C)NC(=O)C(C)=C1CC1)N1CC(OC(=O)NC)C1 16796,c1(-c2cn(CC3CN(C(C(COC)O)=O)CC3SC)nn2)ccc2c(c1)CCO2 16797,N1(C(N)=O)CC2CCN(C(=O)COC(C)=O)C2C1C.N12CCCC(C1)C2=O 16798,O(NC(=O)C(C)(C1CC1)N(C)C(c1ccc(SC)o1)=O)CCCOC 16799,c1(C(C)C)nc(NCc2csc(Br)n2)cc(N2CCC(OCCF)C2)n1 16800,N1(C(C(C(=O)OCC)(C)C)=O)CCN(C(=O)CCCC(=O)N(C)C)CC(C)(F)C1 16801,CC1CC(O)CCN(C(C2CC(CNC(=O)C(O)CC(F)(F)F)C2)=O)C1 16802,c1(C(N2CC(C#C)(CC(=O)O)C2)=O)nn(C)c2c1CCC2 16803,C(=O)(CCCN(C)C)N(C(C)CNNC(=O)C(C)(c1ccccc1)N(C)C)CC 16804,S(=O)(=O)(c1ccc(Nc2scnc2C)c(C#N)c1)NC(CCC)(C)CO 16805,c1(OCC)ccc(C(N2CC(CO)(NC(c3ccc(F)o3)=O)C2)=O)c(F)c1F 16806,N1(C(c2n(CC)cnn2)=O)CC(NC(c2nc(Cl)cs2)=O)CC(C)C1 16807,C(=O)(CCCCCO)NC1C2CN(C(C(c3cccc(Cl)c3)NC(C)=O)=O)CC21 16808,C1(OC)CCCN(C(C2CC23CC(NC(c2ccc(Cl)cn2)=O)C3)=O)C1 16809,C(=O)(C(O)C(C)(C)C)N1C(CC(=O)N(C)CC2CC2(C)C)CCC1 16810,CC1CCC(O)C(C2CCCN2CCC2CC23CC3)C1 16811,CC1CCc2nc(C(=O)NC(CCN(C(=O)COC(F)F)C)C(C)(C)C)cn2C1 16812,CC1(C)C(CC(N2CCCC(NC(C3CCCCO3)=O)C2)=O)C1(C)C 16813,c1(OC)ccc(C(=O)NCCNC(c2cc(Br)cnc2O)=O)cc1N 16814,c1(C(C)=O)cncc(NC(=O)C(=O)NCCCc2cn(C)cn2)c1 16815,c1(SC(C)C(C)(C)C)cccc(F)c1.c1(C2C(=O)N2)ccc(Cl)cc1 16816,CCC(CCCC(=O)NC1CN(C)CC(F)(F)C1)NC(c1ncccc1N)=O 16817,c1(CC)ccc(OCCC(=O)NC(C)C(C)NC(C2CCCCC2)=O)cc1 16818,c1(C(N2CC(N(C(Cc3c(C)ncc(Cl)c3)=O)C)C2)=O)cccc2c1OCCN2 16819,C1(NC(CCNC(C)=O)=O)CCN(C(C2C3CCCC23)=O)C(C)C1 16820,c1(C(N2C(CNC(=O)Cc3cnc[nH]3)CCCC2)=O)cc(F)nc(F)c1 16821,c1(CNC(Cc2cnn(C)c2O)=O)c(Cl)ccnc1Br 16822,C1(C(=O)NCCC=C=C)CN(C(=O)CCc2ccccn2)CCN1C 16823,C(=O)(C(CC(C)C)OC)NC(C(N1C(CC)(CC)CC1)=O)CC1CC1 16824,N1(C(C(C)C2(O)CCC2)=O)CCc2[nH]nc(C(=O)Nc3cc(Cl)nc(Cl)c3)c2C1 16825,C1(C(N2C(C#C)CC2)=O)C2CC3C(C2NC(C2CCCC(CF)C2)=O)C13 16826,c1(C(=O)NC2CCC(NC(c3ccc(Cl)o3)=O)C2)cc2ccc(F)cc2o1 16827,Cc1[nH]nc2c(C(N3CC4(CNC(c5conc5C)=O)CCC3C4)=O)cccc12 16828,c1(C(C)NC(c2nn(C)nc2Br)c2nnnn2CCCF)cc(F)cc(F)c1 16829,n1(CC(=O)NC(C2CCCC2)CNC(=O)C2=CCC2)nc2n(c1=O)CCCCC2 16830,C(C)(C(C)(C)C(=O)NC1COC(C(C)C)C1)NC(c1cccc(CC)n1)=O 16831,N1(C(C(C)SC(F)(F)F)=O)CC2CC(C)N(C(=O)CCc3nccn3C)C2C1 16832,c1(OC)ccccc1C(=O)NCC(CNC(=O)Cc1sc(C)nc1C)OC 16833,C#CC1(OCC(=O)NCC(=O)NCCc2noc(CC)n2)COC1 16834,n1(CCCC)cc(C(=O)NC2C3CC2N(C(=O)CC(C)C2CCCO2)C3)c(C)n1 16835,C1(CNC(C2(OC)CN(C(c3cc4occc4[nH]3)=O)C2)=O)CCN(C)C(=O)C1 16836,N1(C(C2CCCN2C2CC2)=O)CCCCCC(NC(CCC(=O)OCC)=O)C1 16837,N1(C(C)=O)CCC2(CC1)CN(C(C1NC(=O)CC1c1ccc(Cl)cc1)=O)CCO2 16838,C#CCC(CC(F)F)C(=O)N(C(C)CCNCCC(N)=O)C.c1(=O)c(=O)[nH]1 16839,Cc1oc(C(=O)NC(c2cn(C3CCC4CC4C3)nn2)C)cc1S(N)(=O)=O 16840,C12(CC)COC(C(N3CCC(O)(C(C)NC(=O)CCNS(C)(=O)=O)C3)=O)(C1)C2 16841,C(=O)(C(C)C(O)CC(C)C)N1C2(C(=O)OCC)CC(C1)C2 16842,C1(C(C(=O)NCCCOCC(F)F)NC(C(=O)OCC)=O)CC=CCC1 16843,c1(NC(=O)CCC2COCCC2=O)ccc2nc(O)[nH]c2c1 16844,C1(NC(C(C)(C)c2ccccn2)=O)CCCC2CN(C(=O)COCCCF)CC12 16845,C1(=O)CCC(=O)N2CCN(CC2)CCN1.CCC(C(=O)NCC)C1CCOCC1 16846,N1(C(c2c(C)nn[nH]2)=O)CCC(C(=O)NC(C2CCCCO2)C)=C(F)C1 16847,c1(C(N(CC(C)OC)C(C)C)=O)conc1C(C)NC(=O)C(C)SC 16848,C=CCC(C)(N)C(=O)NC1CC(C)CCC1C 16849,c1(C(N(CCNC(CC2C(CC)C2)=O)CCOC)=O)cnn(C(C)C)n1 16850,CC1(C)CCC(n2cc(-c3cnc(Cl)s3)nn2)CN1CC(N)=O 16851,C1(n2c(C(CC)OC)nc(C3CCC3)n2)CCC(F)(F)CC1.N1CCCC1=O 16852,C1(OC)CCCC(C(=O)NCC2CC2NC(=O)C(C)=C2CCC2)C1 16853,N1(C(C=CC(C)(C)SC)=O)CCCC(CCNC(=O)Cc2ncoc2C)C1 16854,C1(NC(CC2CCCC(C)(C)CC2)=O)CCC2(CCN(C(=O)C3=CCC3)CC2)C1 16855,C1(OC)CN2CCCC2(C(=O)NCC(C(C)C)NC(c2ccc(O)cc2Cl)=O)C1 16856,C12(C(N(C(CC)CNC(C3CC(C)(C)C3)=O)C)=O)CC1COC2(C)C 16857,C1(NC(C(C)OCCCCCC)=O)CC2CC(C1)N(C(c1c(C)coc1C)=O)C2 16858,C1(F)(C(=O)NC2CN(C3CN(C(c4cn(C)nc4)=O)C3)C(=O)C2)CC2(CCC2)C1 16859,C1(CNC(C2(C)COC2)=O)CCC2(CCC2)C1NC(=O)C(C1CCOCC1)F 16860,c1(C(=O)NC2CC2)ccc(C(=O)NC(=O)Cc2nocc2CSC)c(Cl)c1.C(C)C 16861,c1(N(C)C)cccc(C2=NOC(CN3C(C(NC=CCl)=O)CCCC3)C2)c1 16862,c1(C(N2CC(CNC(C=C(C)C(F)F)=O)OCC2)=O)c[nH]c2c(Br)cccc12 16863,C(=O)(NNc1cc(Br)ccn1)n1cc(-c2cc(C)c(SCC(=O)O)nc2)nn1 16864,C1(COC)(CNC(=O)CSC2CC2)CCCN1C(=O)CN1CCC(C)C1 16865,CC1(CNC(=O)CCOC2CCCOC2)CCN(C(C2(C)CC=CCC2)=O)C1 16866,CC(C)(C)CC(=O)C(=O)NCC(C(C)(C)C)NC(=O)CN=S(C)(C)=O 16867,CC(C(=O)NCC1CCC(NC(C2C=CC=CC=C2)=O)CC1)C(F)F 16868,N1(C(c2c(CC)ocn2)=O)CC2CCCC(NC(C3CC(OC(F)F)C3)=O)(C2)C1 16869,C(=O)(CC=C(Cl)Cl)NCC1(NC(=O)C=Cc2cnc(C)s2)CC(OC)C1 16870,c1(N2C(CN(C(COC3CCCC(C)C3)=O)C)CCC2)c([N+](=O)[O-])cnn1C 16871,C12(NC(c3c(C)cn(C)c3)=O)CCOCC1CN(C(c1ccc(Cl)c(N)c1)=O)C2 16872,N1(C(c2ccc(C#C)o2)=O)CCN(C(C2CCN(C)C(=O)C2)=O)C(CCOC)C1 16873,N1(C(c2ccc(N)c(N)n2)=O)CCC2(NC(=O)C3=CCCCC3)CCCCCC12 16874,Cc1ccc(NCC(=O)N(CC(O)CN(C(=O)C=Cc2cocn2)C)C)cc1 16875,C1(CNC(=O)CCc2cncnc2)CC(F)CN1C(C1OCCCO1)=O 16876,c1(OC(c2n(CCOC)ncc2C)=O)ccc2c(c1)OC(C)(C)CC2=O 16877,c1(CC)onc(C)c1CNC(=O)CCN(CCO)C(C12CCCCC1C2)=O 16878,C1(N2CCC(CC)C2)CC(NC(c2scc(C)c2Cl)=O)C1(C)C 16879,N1(C(c2cc(CCC)on2)=O)CCCC(C2(NC(=O)C(F)n3ccnc3)CC2)C1 16880,C(c1cccc(C#N)c1)=CC(N1CCN(C(C(CC)N(CC)CC)=O)C2C1C2)=O 16881,C12=CC=C(C=C1)C2C.C1(=O)CN(CCCO)CCCN1.C(C(C)C)SC 16882,C(=O)(C1=NN2CCCN=C2N1)N1CC2(N(C(C(C=C)(C)C)=O)CC2)C1 16883,c1(C(=O)NCCCNC(CC2(OC)CC2)=O)cc(=O)n(-c2ccccc2)[nH]1 16884,c1(NC)ccccc1C(=O)NCCOCCNC(C1CCN(C)C1C)=O 16885,C(=O)(C(F)CCC(C)C)NC(C(C(=O)NCC1CC(CC)C1)(C)C)C 16886,C1(C(C)C(NCP(C)(C)=O)=O)CCCN(C(c2cc[nH]c2)=O)C1 16887,c1(OCC)cc(CN2CCCC(C)(C(=O)O)C2)ccc1OC 16888,O=C(CC(C(F)F)n1ccnc1)NCCCNC(=O)C=Cc1cccnc1C 16889,c1(CCC)cc(C(=O)NC(C)(C)CNC(=O)C=C(C)CCC)ccc1Cl 16890,c1(C(=O)NC2(CF)CCN(C(c3c(CC)nccc3)=O)C2)cc2nc[nH]c2cn1 16891,c1(C(=O)NC2CCN(C(C(COC)C)=O)CC2F)nc2cnccc2s1 16892,CS(=O)(=O)c1ccc(Cl)cc1NC(=O)C(=O)NCC(F)C1CCC1 16893,C1(NC(C2=C(C)CCC2)=O)CCC2CN(C(C3CC4(C3)CC(C)(C)C4)=O)CC2C1 16894,C1(C)(CNC(C2(NC(C=C(C)C3CC3)=O)CC2C)=O)CCN(C)CC1 16895,C(=O)(C1CCCc2nc[nH]c21)NCCCCN(C(=O)CNC(C1CCCC1)=O)C 16896,C1(C(=O)NCCC2COCCN2C(C2CCSCC2)=O)Cc2ccccc2O1 16897,Cc1c(C(=O)N(C2CCN(C(C34CC(C(C)C)(CO3)C4)=O)C2)C)cccc1Cl 16898,N1(C(c2n(CC)nc(C3CCCC3)c2)=O)CC2CCC(NC(=O)OC)CC2C1 16899,c1(C(=O)NC(CC)CN(C(=O)COCC(C)C)C)cc(C)nn1C1CC1 16900,c1(C(=O)NC2C(NC(C3(CCC)CC3)=O)CCC2)c(C)cc[nH]c1=N 16901,c1(CC)nccnc1C(N1C(C(N2CC(C)(C)C2)=O)CC2CC12)=O 16902,C1(C(=O)NC(CO)C2CCC2)(COC)CN(C(=O)CC(C)C2CC2C)C1 16903,c1(C(=O)NC2C(NC(CC(C)C3CCC3)=O)CCCC2)ncc2cc(Cl)ccn12 16904,Nc1c(C(=O)NCC(CO)NC(=O)CC2COC3CC2C3)cnc2ccnn12 16905,C1(=O)C#CC(C)(C)CNCc2cccc3c1c(CCCOCC)[nH]c23 16906,c1(C(=O)NC2CC(OCC(=O)N(C3CCSC3)C)C2)cnoc1C1CC1 16907,C1(=O)C(C)(C)C(C)N1.C(C)(C)(CNC(=O)COC1CC1)OCCOC 16908,c1(C(=O)NCCNC(N2CCCC2c2ccncc2)=O)ccccc1Cl 16909,N1(C(CN(C(C2C(C#N)C2)=O)CC2CC2)=O)CCn2cccc2C1 16910,C(N=c1[nH]c(-c2ccccc2)ccc1CO)c1scc(-c2c(C(N)=O)cccc2)c1 16911,C1(C(=O)NCC(CN(C)C(c2ccc(C#N)[nH]2)=O)(C)C)C2CCC(=O)C12 16912,N1(CC(=O)N(C)C)C(=O)CCC1=O.C12(C(=O)OC)CCC1(C(=O)C=O)C2.C12(CC1)NC2 16913,C1(NC(c2ccc(Cl)cc2Cl)=O)CC2CC(C1)N(C(=O)C(O)C1CCC1)C2 16914,[N-]=[N+]=NC1CC2(C(N3CCCC3CNC(=O)COC(F)(F)C(F)(F)F)=O)CC12 16915,c1(C(N2CCC(C(=O)Nc3cc(Cl)cnc3O)C2)=O)ccc(F)c([N+](=O)[O-])c1 16916,C#CCCCCC(=O)N1CCCC1C1CCN(C(CCCCCCC=C)=O)C1 16917,c1(NC)ccc(F)cc1C(N1CC(C(F)(F)F)OCC1CNC(=O)C(C)(C)C)=O 16918,c1(C(=O)NCC(N2CCCC2)C)cc(Cl)ncc1CNC(C(C=C)OC)=O 16919,N1(C(c2c(C)[nH]nc2CO)=O)CC2(C1)CN(C(C1COCCN1C=O)=O)C2 16920,C(=O)(CC1=NN(C)C(=O)C1)NC(C(C)NC(CCCNC(COC)=O)=O)(C)C 16921,C1(CC(=O)NCCN(C(C)C)C(c2n[nH]cc2Cl)=O)CCC2(CCC2)CO1 16922,c1(OC)ccc(C(=O)NCCNCC(C)=CC(=O)NC23CCCC2C3)cc1 16923,C1(C(=O)NC2CC3CNCC23)CC2(CCCCC2)CN1 16924,c1(NC2(CNC(C3(CF)CCC3)=O)C(C)CCCC2)ncc2c(n1)CCOC2 16925,c1(C(=O)NCC2CC(C)N(C(=O)CC34CCCC3C4)C2)sc2nccnc2c1N 16926,CC(C)(C)C(C)(C)C(=O)N1CCOC(C(N2Cc3c[nH]nc3C2)=O)CC1 16927,N1(C(Cc2cn(CC)nn2)=O)CC(C)CCC1CNC(c1[nH]cnc1C#N)=O 16928,C1(NC(c2ccc(C)c(C(F)(F)F)c2)=O)CC2CCC(C1)N2C(C1CC1(C)C)=O 16929,C(CC1CC1)(C(=O)NC1COCC1NC(=O)C=CSC)OC 16930,c1(C(N2C(CNC(c3c(C)sc(O)n3)=O)CC2)=O)cc2c(Br)cccc2cn1 16931,c1(N(C(=O)NC(C)CCCc2ccccc2)C)ccc(F)cc1 16932,C1(NC(=O)C=CCF)CCC1C(=O)NCCc1cnc[nH]1 16933,c1(OC)cccc(F)c1CC(=O)NC1CCN(C(c2cccc(F)c2)=O)C1C 16934,c1(NC(=O)CCC2CCCC2)ccc(OC(F)(F)F)cc1 16935,C1(CNC(=O)C=CC=C(Cl)Cl)CCCC2(CN(C(=O)CCC(F)(F)F)C2)O1 16936,C1(C(=O)NC(C2CN(C(CC3CC(C)C3)=O)C2)C)NC(=O)OC1C 16937,C(=O)(CC(C)CC(C)(C)C)NC1C(CC(=O)N(C(CCC(C)C)C)C)CCC1 16938,C(=O)(C(CCC1CCC1)NC(=O)NCCc1cnsc1)NC 16939,Cc1nnc(C(C)NC(=O)CC2CCN(C(=O)CC3OCCCO3)C2)o1 16940,c1(C(CNC(c2cncn2C)=O)NC(C2C(C)OCC2)=O)ccc(F)cc1 16941,C1(C)(NC(COC(CNC(CC2CC(=C)C2)=O)(C)C)=O)CCOCC1 16942,C12(C(=O)NCC)CCCC1(C(=O)CC1(C(F)F)C(CNC(=O)OC)C1)C2 16943,C12(CNC(c3ncn(CCOC)c3)=O)CC1CN(C(=O)C(C)(C)c1cnsc1)C2 16944,Cc1coc(C2CCCCC2)c1C(=O)NC1CC1NC(=O)COCCN(C)C 16945,c1(C(=O)NCC2N(C(CCS(C)=O)=O)CCCC2)c(Cl)ccc(F)c1F 16946,C1(CCNC(CSCC(C)C)=O)CC(NC(c2ccsc2)=O)C1 16947,c1(C(C)C=O)cn(CC)nc1-c1ccc(F)cc1.C1(C(=O)NC2COC2)CC12CC2 16948,C1(NC(COCCN(C)C)=O)CCCC12CCN(C(c1ccc([N+](=O)[O-])o1)=O)C2 16949,C1(CN(CC(=O)NC(c2ccccc2)CC)C)(CC)CCOCC1 16950,C1(CNC(C(C(C)(C)C)C#N)=O)CN(C(=O)C(N)=O)CCC12CCOCC2 16951,CC(C)C(N=[N+]=[N-])C(=O)N1C(C(N2CCC(OCCN(C)C)C2)=O)CCC1C 16952,C(=O)(C#CC1(C)COC1)NC1(COC)CCCN(C(CC(C=C)CC)=O)C1 16953,c1(C(N2CC(OC)C(C)C2)=O)cn2ccc(-c3cncs3)cc2n1 16954,C1(SC)CN(C(C2CCN2C(C)(C)C)=O)CC1NC(=O)CN1CCN(C)CC1 16955,CCCC(O)CC(=O)NC(C)(CNC(c1ccc(NC)cc1)=O)Cn1cccn1 16956,Cc1nc(=N)[nH]cc1C(=O)NCC12CC(NC(c3ccc(C)n3C)=O)(CCO1)C2 16957,C#CCC(C)(C(=O)Nc1ccc(CO)c(F)c1)NC(=O)C(CC1CC1)SC 16958,N1(C(C2C(C)C2)=O)CC2CN(c3cc(Cl)ncn3)CC2C1 16959,c1(OC)cccc(C)c1NC(=O)CCCCCNC(C1NC(=O)OC1C)=O 16960,N1(C(CCCn2ncc(C)c2)=O)CCN(C(c2cc(C)ccc2O)=O)C2CCC12 16961,N1(C(c2c(C)ocn2)=O)CCC2(CC1)COC(CNC(C1(C(N)=O)CCC1)=O)C2 16962,c1(C(=O)NC(C(C)NC(=O)Cn2cnnn2)C)cncc(Br)c1 16963,CC1N(C(C2CCCN(C(c3nc(=N)cc[nH]3)=O)CC2)=O)CCC1(C)C 16964,N1(C(=O)CN2CCOCC2)CCN(C(c2ccncc2Cl)=O)C2CC12 16965,C1(CC(=O)N(C(C)CCNC(C2CC(C#N)C2)=O)C)CCCC(O)C1 16966,N1(C(c2cccc(CC)c2)=O)CC(C)CCC1C(N1CCCC(CCO)CC1)=O 16967,C(=O)(CCC(=O)NC(C)(C)CC(=O)N(C)Cc1cscn1)NCC 16968,C12(C(N(CCCNC(CCC=C(C)C)=O)C)=O)CC3CC1C2C3(F)F 16969,N1(C(c2n(CCCC)ncc2)C(=O)NC(C)C)CCC2OC(=O)OC2C1 16970,c1(C(N(C2CCN(C(c3n[nH]c(C)c3C)=O)C2)CC)=O)cncc2ccccc12 16971,c1(OC)cc(C(=O)NCC2CC2NC(C2(C)CC=CC2)=O)on1 16972,C1(C(=O)NCCCOCCOC)CCN(C(C23CCC(CC2F)C3)=O)CCO1 16973,N1(C(c2c(CC)nsc2)=O)CCC(C)(NC(c2cnn(C3CCCCC3)c2)=O)C1 16974,c1(OC)cc(C)c(C(=O)NCC2CC(O)CN2C(=O)CCC(N)=O)cc1Br 16975,c12nc3nc(ccn3n1)C1(CC1)N2C(C1CCC1c1nc[nH]n1)=O.C(F)(F)F 16976,C(=O)(C(C)(C)C(=O)NCC1(F)CCCN(C(C2CC(C)(C)CCO2)=O)C1)NC 16977,c1(C(N2C(C)CC(CNC(c3cncc(F)c3)=O)CC2)=O)nn(C)c2c1CCC2 16978,C1(CN(C(=O)Cn2cnc(C(N)=O)n2)C)CCC(NC(=O)CCC2OCCO2)CC1 16979,N1(C(c2cc(CCC)oc2C)=O)CCN(C)CC1CNC(=O)CCC(C)O 16980,C(c1ccc(Cl)c(Cl)c1)=CC(=O)NC1CCN(C(=O)CC2CCCC2(F)F)C1 16981,C1(CNC(C(=O)NCC(CCOC)OC)=O)CC(C)CCO1 16982,C=CC(C)CC(=O)N(CC(C)O)CCNC(=O)Cn1cc(-c2ccccc2)cn1 16983,C1(C(=O)NC2CC(C(C)NC(c3cccc(C4CC4)c3)=O)C2)CC2CCCC2C1 16984,c1(C(=O)NCc2cnc(CC(C)C)s2)cc(Cl)cc2c1NCCC2 16985,N1(C(CCC#CC)=O)CCCC(C(=O)NCCC2CCCCCC2)C1C 16986,N1(C(c2ccc(C#C)cn2)=O)CC(N=c2nc(C(C)C)[nH]s2)CC2(CCC2)C1 16987,C1(NC(c2cncc(NC)c2)=O)CN(C(C2CC23CCC3)=O)CC(C)(C)C1 16988,CC(C(=O)NCCCCC(C)NC(c1sccc1CO)=O)C(=O)N1CCOCC1 16989,C12(C(N(C3CCCN(C(C4(CCF)CCC4)=O)C3)C)=O)CCC(CF)(CC1)CC2 16990,c1(C(N2CC3(CCN(C(Cc4ccc(C)s4)=O)C3)C2)=O)cc([N+](=O)[O-])c(C)cc1C 16991,C1(NC(C2N(CC)CC2)=O)CCCC(CC=CC(N2CC(CO)C2)=O)C1 16992,C(=O)(C(C(C)(C)C)N1CCCCC1=O)NC1C(NC(CS(=O)(=O)NC)=O)CC1 16993,C(=O)(C#CC(C)(C)CNC(C1CCC2(CC2)C1)=O)N(C1CCOC1)CC 16994,N1(C(C(CC)(F)F)=O)CCN(C(=O)CCC2CCCN2C)C(C(C)C)C1 16995,C1(SCc2n(C=C)ccn2)CCCSC1 16996,C(=O)(C(F)(F)CCc1ccccc1)NCC(C1CCCC1)NC(C(C(C)C)O)=O 16997,N1(C(C=C(CCC)CCC)=O)CCN(C(=O)CC2(C#N)CC2)C(CC)C1 16998,c1(C(=O)O)ccnc(C(F)(F)F)c1.CC1CCN(CCOC)C1 16999,C1(N)(C(=O)Nc2cccc(N(C)C)n2)CC2CCC1CC2 17000,c1(C(N(c2ccccc2)S(CC)(=O)=O)=O)ccc(C#N)n1C 17001,c1(C(=O)NCCC(CCNC(C2CC(=C)C2)=O)C)cc(Br)ccc1OCC 17002,N1(C(c2cc(CC)no2)=O)CCN(C(=O)CCC2CCCC2)CC1c1cn[nH]c1 17003,c1(C2C(CO)(CNc3ccc(N4CCC(O)C4)nc3)C2)c(F)cccc1Cl 17004,c1(CNC(=NC)NCC2COC(=O)N2)cc(Cl)ccc1Cl 17005,C#CCC(O)C(=O)NCC1(CNC(c2cnn(C(C)C)c2CCC)=O)CC1 17006,Cn1nc2c(c1C(N1CCC(NC(C3CCNC(=O)C3)=O)C(F)C1)=O)COCC2 17007,C1(NC(C2C(OCC)CC2)=O)CCC2(CCN(C(c3cc(C)oc3C)=O)C2)C1 17008,S(=O)(=O)(c1cnc(NC2CC3CCCC3C2)c(Cl)c1)NCCCCC 17009,C1(C(=O)NCC(C)NC(=O)C(C)(C)n2cc(Cl)cn2)(OC)CCCCC1 17010,N1(C(C(C)C(C)(C)C)=O)CC2CC(O)C1C2NC(=O)C=CC1(C)COC1 17011,C(=O)(N=c1cc(Cl)nc(C)[nH]1)C1N(c2nc(OC)c(C)cn2)CC(F)(F)C1 17012,N1(CC(=O)NC(Cc2cc[nH]n2)C(=O)N2CCC(OCCF)C2)CCC2(CC2)C1 17013,C1(CCNC(COCCCC#C)=O)(NC(CC(C)(F)F)=O)CCCC1 17014,C1(Cc2coc(C(F)(F)F)n2)CCCCN1C(=O)NC(=O)CCc1cnccn1 17015,N1(C(C(C)=CC2CC2)=O)CC(CNC(=O)C(C)SC(F)(F)F)C2(CC2)C1 17016,C1(NC(C2CCC2)=O)CC2CC1CN(C(c1cccn3nccc13)=O)C2 17017,Cc1nc(N2CCC(NC(C3(C(F)F)CCOCC3)=O)C(C)C2)c2cc[nH]c2n1 17018,c1(C(=O)NCC2N(C(CSCC#C)=O)CCC2(C)C)ccc2c(c1)COC2=O 17019,c1(C(=O)NC2CC(CCNC(c3scc(C)c3C)=O)C2)ccc(F)cc1F 17020,C(=O)(C1=C(Cl)CCC1)NC1C(NC(c2ccn(C(CC)CC)n2)=O)CC1 17021,CC(C)C(C(=O)N1CCCC1CN(C(=O)C(C)Cc1ccccc1)C)n1cnnn1 17022,c1(N2CCC(N(C(c3ccn(C4CC4)n3)=O)CCO)C2)ncnc2ncn(C3CC3)c12 17023,C(=O)(CC(F)(F)F)NCC1C(CC(=O)NC(c2c(OC)c[nH]n2)=O)CC1 17024,CC1=C(C(=O)N2CCC(F)C(NC(c3cnc(C)o3)=O)C2)S(=O)(=O)CCO1 17025,N1(C(C2C(CC)CCC2)=O)CCN(C(C)CNC(=O)Cn2cccn2)CC1 17026,C1(CC)CCN(C(C2CC(=O)N(C)C2)=O)C(C(=O)NCc2ccc(OC)cn2)C1 17027,Cc1cc(F)ccc1NC(=O)C(C)CN(C=O)Cc1cn(C)nc1I 17028,C=CCCCCC(=O)N(C1CN(C(C2CC2C)=O)C(CC)(CC)C1)C 17029,c1(C(=O)NC(CC)(C)CNC(=O)CSS(C)(=O)=O)cncc(OC)c1 17030,Cn1cnc(C=CC(N2CCCC2(C)CNC(=O)CCCc2cc[nH]n2)=O)c1 17031,N1(C(c2ccc(C)c(C#N)c2)=O)CC2(CCN(Cc3ccc(Cl)nn3)CC2)C1 17032,Cc1ccc(C(CC2CCCS2)NC(=O)NC2(Cc3csc(C)n3)CC2)cc1 17033,c1(C(N2CC(NC(C3(COC)C=CCC3)=O)(CC)C2)=O)nccc2ccncc12 17034,N1(C(c2scc(CC)c2)C(=O)NCC2CCCO2)CCN(C)C(=O)C1C 17035,C#Cc1cnc(C(=O)NCC(F)CNC(=O)C(C)CC(F)F)c(C)c1 17036,c1(CC(N2CC(CNC(C3C(C(=O)OCC)C3)=O)C2)=O)ncc(F)cc1F 17037,C1(CNC(C(C2CCOCC2)C)=O)CCN(C(C2CC3(CCC3)C2)=O)CC1O 17038,C(=O)(CC(CN(C)C)CC(C)C)NC(C1CCCN(c2cc(OCC)ncn2)C1)C 17039,C1(NC(=O)NC)CCNCC12CCCCC2.C1(=O)CN1CCNC(=O)OC(C)(C)C 17040,C1(CNC(=O)Cc2cccs2)CCC1C(N1CCC1C(N)=O)=O 17041,C1(CCOC)CN(C(=O)Cc2ccnc(O)c2)CCN1C(=O)CC1C=CCC1 17042,c1(C(N2CCCC(NC(C3C(C)(C)CO3)=O)C2)=O)cc(S(N)(=O)=O)cc(Cl)c1Cl 17043,C1(C(N2CCC(OC3CC3)C2)=O)COCCN(C(C2(O)CCCCCC2)=O)C1 17044,N1(C(C(C)CN(C)C(C2(CO)CCCC2)=O)=O)CCC(N=[N+]=[N-])C1 17045,C(=O)(CCO)N(CC(O)C1CC1)C.C1(C(=O)NCC(C2(O)CC2)O)CCCC1 17046,c1(C(=O)NCC2(OC)CN(C(C34CCCC3C4)=O)C2)ccc(C)c(F)c1F 17047,c1(C(=O)NC(CNC(C(C(C)C)N(C)C)=O)(C)CO)ccc(F)c(CO)c1 17048,CC(C)(C)CC(C(=O)NCc1cccnn1)NC(=O)CCCC#N 17049,CCCC(C(=O)NC(c1nc[nH]n1)C1CC1)NC(=O)C(CCC)NC(N)=O 17050,Cc1oc2ccccc2c1C(N1CCCC(CNC(C2(C)CCNC2=O)=O)C1)=O 17051,N1(C(C(C)C2CCCC2)=O)CCC(C)(C)C1C(=O)NCCCCCO 17052,c1(NC(CN2CC(CC)C2)=O)ccc(NC(=O)C=C(C)C)c(C)c1 17053,c1(OC)ccc(F)c(-c2cnc(C(=O)Nc3ncco3)cc2OC)c1 17054,C(c1cccc(F)c1F)=CC(N1CC(O)(C(C)NC(C2COCC(C)(C)O2)=O)C1)=O 17055,c1(OCC#C)ccc(Cl)c(C(N2CCC(N(c3ncccc3C#N)C)CC2)=O)c1 17056,N1(C(=O)OC(C)(C)C)CCS(=O)(=O)C(CCOC(C2CCC3CC3CC2)=O)C1 17057,C1(CC(=O)NCC2CN(C(c3nc(COC)sc3)=O)C2)CCCCC1C 17058,c1(COCC(=O)NCC2C=CCN2C(=O)CCC2CCCO2)ccccc1Cl 17059,c1(CN2CC3C(NC(=O)COC4CCCC4)(C3)C2)ccc(O)cc1F 17060,CCCCCCCCCC(=O)N1CCC(O)(CNC(c2csc3nccn23)=O)C1 17061,c1(N2CCC(C(=O)NC)C2)cc(N2CCCC2c2cccc(F)c2)ncn1 17062,c1(NC(C2C(C=C)C2)=O)cccc(NC(=O)C=CC=C(Cl)Cl)c1 17063,N1(C(C=C(COC)C)=O)CC=C(CC(=O)N(C(C)C(C)(C)C)CC2CC2)CC1 17064,C1(CNC(C2CN(C)C(=O)C2)=O)CN(C(c2cnn(C3CC3)c2)=O)CCCO1 17065,c1(C(=O)NC(CC)CN(C(=O)CCc2ncccn2)C)ccc2occc2c1 17066,N1(C(C(C)CC(F)(F)F)=O)CC(CNC(=O)CS(C)(=O)=O)CC12CCOCC2 17067,CC1(C)CC(NC(C2CCCN2c2ncccn2)=O)CN1C(=O)CC1(CO)CC1 17068,C1(C(N(C2CCN(C(=O)CCC(C)NC(N)=O)C2)CCC)=O)CCC=CCCC1 17069,C=C(C)CCCC(=O)NCCC(O)C(=O)N(CCCN(C)C)CCC 17070,Cc1ccc(CN2CC(C)(CC(=O)NC(CO)CC(C)C)C2)c(F)c1.C1C(=O)O1 17071,c1(CC(=O)NCC2C(NC(C3CC(F)(COC)C3)=O)C2)cccnc1OC 17072,CC(CCS(=O)(=O)c1ccc(Cl)cc1)C(N1CCC(c2cc(O)ncn2)C1)=O 17073,CC1CN(Cc2csc(Br)n2)CC1NC(=O)CCn1ccnn1 17074,Cc1cc(C(=O)NCC(C)N(C)C(C2CCN(C)C2=O)=O)cnc1C(F)F 17075,Cc1nn(C)c(NC(C2CC2C)=O)c1C(=O)O.c12cn(nn1)C2.C12C=CCN1C2 17076,C#Cc1ccc(C(=O)NC(CN(C)C(c2cnn(C(C)(C)C)n2)=O)CC)c(C)c1 17077,C1(C(CC)C)CCN(C(=O)CNS(=O)(=O)C2CC2)CC1 17078,CC1C2C(CCN2C(C2CCC(=O)C2)=O)CN1C(C1CCNC(=O)C1)=O 17079,C1(CNC(CS(CC)=O)=O)CCC2(CN(C(=O)Cc3ncc(C)o3)C2)O1 17080,C1(C(=O)NC2C(CNC(=O)Cc3ccsn3)CCC2)CCc2ccnn2C1 17081,Cc1sc(C(=O)NC2CC(CNC(C3CC4CCC4C3)=O)C2)cc1[N+](=O)[O-] 17082,C1(NC(C2CC(=C)CN2C(c2ccc(Cl)o2)=O)=O)CCOC12CCOC2 17083,c1(NC(CC)C(=O)Oc2ccccc2F)cc(O)nc(C)n1 17084,C1(C(N2CC(NC(C(C(CC)(C)C)O)=O)C(C)CC2)=O)COc2ccccc2O1 17085,c1(C(=O)NCCC(C)(C)NC(c2cc(C3CC3)ccn2)=O)cc(Cl)cnc1O 17086,c1(OC)cccc(Cl)c1C(N1CC(NC(C2CC23CCC3)=O)CC(F)C1)=O 17087,c1(N(C(CNC(C2CN(CC)C(=O)CC2)=O)C)C)nc(C(C)C)ncc1Br 17088,C1(NC(C2(C(=O)OCC)CC2)=O)CN(C(=O)C(C)(C)SCC)CCC1CO 17089,CCC(C(=O)N1CCC(CN(C)C(C2(CN(C)C)CCCCC2)=O)C1)C(C)(F)F 17090,CC1CC(NC(C23CC2C3)=O)CN1C(=O)CO 17091,CC(C)(C)C(CNC(=O)CC(=O)C(C)(C)C)C(=O)NCC(C)(O)CO 17092,C1(NC(=O)Cn2cc(Cl)cn2)CN(C(C2CC(CF)C2)=O)CC2(CC2)C1 17093,CC(C)CC(CNC(c1ccn(CCF)n1)=O)C(=O)NCCC(C)NC(N)=O 17094,C(c1c(C)noc1C)=CC(N1C(CN)CCC1)=O.CC(c1cccs1)=CC(=O)NC 17095,c1(NCCC2(OC)CN(C(=O)C3=C(C)CCC3)C2)cc(C(N)=O)ccc1[N+](=O)[O-] 17096,CCCCCC(O)CC(=O)N1CCN(C)C(CNC(=O)Cc2ncccc2C)C1 17097,CC(C)CC(C(=O)NCC(C)(CO)NC(=O)C=Cc1cocn1)N(C)C 17098,c1(C(N2CC(NC(CC=C)=O)C3(C2)CCC3)=O)nc2cccnn2c1Br 17099,N1(C(c2ccc(C(CC)=O)cc2)=O)C2CCC1C(NC(C1(CO)CC1(F)F)=O)C2 17100,c1(C(N2CCCC(O)(CC)C2)C(=O)NCc2ccco2)c(C)ccc(Br)c1C 17101,C1(NC(C(COC)NC)=O)CN(C(c2cc(OC(C)(C)C)ccn2)=O)CC1(C)C 17102,C1(NC(C2CC(C3CC3)=NO2)=O)CN(C(c2cnc(C3CC3)[nH]2)=O)C2CCCC12 17103,C12C3CCCC1N(C3)C2=O.C1(C(N(S(C)(=O)=O)C)=O)C2C3CCC(C3)C12 17104,C(=O)(CC(C)(O)C=C)C(=O)C=CC(C)N.C=CCC(C(=O)OC)N 17105,CCC(CC)CC(F)C(=O)NC1(C)CCC(C(N2CCCN(C)CC2)=O)C1 17106,c1(CN(C)C(C2C=CCN2C(=O)CC2CCCC2)=O)ccncc1F 17107,C1(NC(c2cn(CC(C)(C)CNC(C3CCSCC3)=O)nn2)=O)CC(F)C(=O)N1 17108,N1(CC(C)N(CC)CC)CCC(NC(c2sccc2C(C)C)=O)CC1 17109,C#CCCCCCCC(=O)NCc1ccc(C(=O)NC2(C3CC3)CCOC2)n1C 17110,N1(C(CCNS(C)(=O)=O)=O)CC2CCCC(NC(=O)C=CS(C)=O)(C2)C1 17111,c1(C(N(CC(CN(C(=O)CCC(N)=O)C)O)C)=O)cccc2occc12 17112,c1(C(C)(C)C)cccc2c1OCC2C(=O)NCCC1CCCCC1O 17113,C(C(C)(C)CCNC(c1ccnc(CNC(=O)C(C)(C)C2CCCC2)c1)=O)OC 17114,C(=O)(C(F)(F)C(F)(F)C(F)F)NCC(C1CC1)NC(C1OCC(C)(C)C1)=O 17115,C(c1cn(C(C)C(=O)OC(C)C)cn1)=CC(=O)N(c1ccccc1)S(CC)(=O)=O 17116,S(=O)(=O)(c1cccnc1N1CC2(CC(C)CO2)C1)NCc1c(COC)noc1 17117,C1(C(N2C(C)CN(C(=O)CC#N)C(C)C2)=O)=CC=CC=CC=C2N(C=C1)C2=O 17118,N1(C(CSC)=O)CC2CCCC(CNC(C3CC34CCCCC4)=O)C2C1 17119,CN1CCN(C(c2cc(CF)on2)=O)C(CNC(c2cnn(CC(F)F)c2)=O)C1 17120,c1(NC(C2C3CN(C(CCCN(C)C)=O)CC32)=O)ccc2ncnn2c1 17121,c1(CCNC(C2(O)CN(C(C(C)(C)C)=O)C2)=O)ccccc1O 17122,c1(C(=O)NCC(C)N(C)C(c2nn[nH]c2Cl)=O)cc(C#N)cs1 17123,N1(C(c2ccc(OC)nc2C)C(=O)NCCC2(C)CC2)CCC(C2CC2)CC1 17124,c1(OC)ccccc1C(O)C(=O)NC1CCC1CNC(=O)Cc1ccc(Cl)cn1 17125,C12(C(=O)NC34CC(NC(C(C)N(CC(F)(F)F)C)=O)(C3)C4)CC=CCN1CCC2 17126,c1(C(N2CC3(C(NC(CCc4ccc(C)cn4)=O)C3)C2)=O)cc2ccoc2cc1C 17127,N1(C(C2(COC)CCCO2)=O)CCCC(NC(=O)CCOC2COC2)C1 17128,N1(C(C(Cc2cnn(C)c2O)OC)=O)CC2=C(C1)CN(C(=O)C1=CCCCO1)C2 17129,C(C)(C)(CCC(=O)NCc1ncccc1C(N1CC(C)(CO)C1)=O)OC 17130,c1(C(=O)NC(C)CC(C)NC(=O)C=CS(C)=O)cccc2nc(C(F)(F)F)[nH]c12 17131,n1(C(C)C)cnc(C(=O)NCC2CCCN2C(c2csc(SC(F)(F)F)n2)=O)n1 17132,C(=O)(CCCC(F)(F)CO)NCCNC(C(CCCC)NC(N)=O)=O 17133,C1(NC(c2c(OC)scc2)=O)CCN(C(=O)CCn2cc(Cl)cn2)CC1F 17134,S(=O)(=O)(c1cccc(F)c1)N(C(C)C(=O)Nc1ccccc1)C1CC1 17135,N1(C(CN(C(C)=O)C)=O)CCCC(CN(C(=O)CCc2ccnc(OC)c2)C)C1 17136,n1(CCOC)ncc(C(=O)NCC(C2CCC2)NC(C2C3CCN2CC3)=O)c1C 17137,C1(COC)CN(C(=O)CC2(C)CC(F)(F)C2)CCN1C(c1ncccc1C)=O 17138,S(=O)(=O)(c1ccc(F)c(F)c1)N1C2CCN(C(c3cc(Cl)ncn3)=O)C2CC1 17139,N1(C(C=C(CC)C)=O)CCC2C(NC(=O)C(C)NC(=O)C=CCl)CC12 17140,c1(COC(C2C(=C)CN2C(=O)OC(C)(C)C)=O)cnc(F)c(C)c1 17141,c1(C(N2CCCC(NC(CC3(C=C)CC3)=O)C2)=O)cccc(C(=O)OC)c1C 17142,C1(C(N2CCCC2)=O)CCC(CNC(N(C)CC2CC2Cc2ncn(C)n2)=O)CC1 17143,c1(C(C)C)ccccc1C(=O)NC1CC(C(=O)N(C2CCC2C)C)C1 17144,Cn1nc(O)cc1C(N1CCCC1CCC(=O)NCC(c1ccccn1)O)=O 17145,C(N=c1nc(C(C)(C)C)[nH]s1)C12CC(CNC(C3CCCC3)=O)(C1)C2.CC1C(=O)N1 17146,c1(C(=O)NC(CCNC(CC2CCN(C(C)=O)C2)=O)C)c(N)cc(OC)cc1F 17147,CC(C)CC(O)C(C)C(=O)N1C(C(=O)NCC2(C)CCOCC2)CC2CC12 17148,N1(ONC(C2CCCC(C#N)C2)=O)CCC=C(C(=O)Nc2cnn3cccc3c2)C1 17149,Cc1c(Cl)c(C(F)(F)F)nn1CC(N1CCN(C(=O)C2=NOCC2)C(C2CC2)C1)=O 17150,C(C)(C)(CC(F)C(=O)NCC1(C)CSC1)NC(C(CCC)OC)=O 17151,CCCC(C)(C)CC(=O)N1CCCC(C)(C)C1C(=O)NC1CN2CCCC1C2 17152,N1(C(c2nc(C)c(C)[nH]2)=O)CCC(C2CCNC2)C1 17153,C1(C(N(C(C)CNC(=O)C2=CCCCC2)C)=O)CCCC2(CCC2)C1 17154,N1(C(CCCOCC=C)=O)CC=CC(C(=O)NC(c2scnc2C)C)C1 17155,CC1=C(C(=O)N2CCC3CN(C(=O)C(c4ccc(Cl)cc4)C)CC23)CCCC1 17156,c1(SC)ccc(CC(N2CCC(N(C)C(c3cc(C(F)F)no3)=O)C2)=O)cc1 17157,C1(C(=O)NC(CC)(C)CC)CN(C(=O)CSC(F)(F)F)CCC1(C)C 17158,C(=O)(Nn1c(C)nc2ccccc2c1=O)c1ccc(-c2cccc(OC)c2)cn1 17159,c1(N(CC(C)C)C)nc(N2CCOCC(F)(F)C2)c2c(n1)CCC2 17160,Cc1ncccc1CC(=O)N(C(C(=O)NOCCN1CCOC1=O)C1CC1)C 17161,N1(C(c2cnc(C)nn2)=O)CC2CCN(C(=O)COCc3ccncc3)CC2C1 17162,C(C(=O)NCC(C)(C)CCNC(c1ccc(C(C)(F)F)cc1)=O)(C(C)C)OC 17163,c1(OC)ccc(S(C)(=O)=O)cc1C(N1CCC(N(C)Cc2nc(Br)cs2)C1)=O 17164,CC(C(=O)N(CC(=O)N(C(C)Cc1cn[nH]c1)C1CC1)CC1CC1)NC=O 17165,CCCC(C)(CC)C(=O)NC1CCN(C(c2cnc[nH]2)=O)CC1(C)C 17166,c1(NC(=O)NC2CC(C(F)C(N3CC4C(C3)C4(F)F)=O)C2)ccc(C#N)cn1 17167,c1(C(C(=O)NCC2(F)CC(NC(COCCCC)=O)C2)C)ccc(F)cc1F 17168,CC(C)(O)C(C(=O)NCCCOCC(F)F)NC(c1ccsn1)=O 17169,C(C1=NOC2CCCCC12)NC(C1N(C(C)C)CCC1)=O 17170,c1(NC(C2C3CN(S(c4c(C)onc4)(=O)=O)CC32)=O)ccc2c(c1)C(=O)N(C)C2=O 17171,N1(CCOCC=C)CCN(C2CCN(C(C3CC34CC4)=O)C2)CC1 17172,N1(C(C(C)OCCC(C)C)=O)CC2CCN(C(c3cc4ncccc4s3)=O)C2C1 17173,c1(CC)ccc(F)c(C(N2CCC(NC(c3ccnc(S)c3)=O)C(C)C2)=O)c1F 17174,C1(CC=C)(NC(=O)C(O)COCc2ccccc2)CCN(C(=O)CC(C)OC)C1 17175,C(C)(C(C(=O)NCCC1CC(C)C1)C(C)C)NC(C(C)=CC)=O 17176,C(=O)(C(C(CC)CC)OC)N(C(C)C(=O)N(C)C(C)C)CCC 17177,c1(CN2CC(NC)C(C)(C)C2)ccc(C)c2c1CCC2 17178,N=c1cc(C(N2CCN(CC(N3CCC(O)(CO)C3)=O)CC2)=O)cc[nH]1 17179,Nc1cc(C(=O)NCC2(CNC(=O)CC3C=CCCC3)CC2)ccc1Cl 17180,C1(C)(CC)CCC(C(=O)N(CC(=O)N(C2CCCC2C)C)CCOC)O1 17181,c1(C(=O)NCC(CCCC)NC(c2cccs2)=O)n[nH]c2c1COCC2 17182,C(=O)(CCS(C)(=O)=O)N1CC(OCC)C(CNC(c2cc(N)ccn2)=O)C1 17183,c1(C(=O)NCC2CCC(CNC(C(CCC)OC)=O)CC2)nc(OC)ccc1C 17184,c1(C(=O)OCC(CC)F)cnc2sc(C)nc2c1 17185,C=CCCCC(C(=O)Nc1ccc(OC)cc1)N(C(c1ccc(C)o1)C)CC 17186,N1(C(CN(C(c2ccns2)=O)CC2CC2)=O)CCc2c(cccc2[N+](=O)[O-])C1 17187,c1(NC(c2cn(Cc3ccc(F)cc3)nn2)=O)[nH]nc(C(F)(F)F)c1Br 17188,C(CC(F)F)(C(=O)NCCCc1cccs1)NC(C1OCCN(C)C1)=O 17189,C1(c2nc(CNC(=O)CC3CCC3)[nH]n2)CCCN(C(=O)CC2CCOC2)C1 17190,C#Cc1ccnc(C(N2CCC(N(C)C(c3cccc(N)c3F)=O)C2)=O)c1 17191,N1(C(C2(NC(=O)CC3CCCSC3)CCSC2)=O)CCc2cncnc2C1 17192,C(=O)(C(C)(C)CC(C)(C)C)N(C)CC1CCCCN1C(c1cc(Cl)no1)=O 17193,CN1CC(=O)N(CC(=O)NC2CCCCC2CNC(c2nccc(Cl)c2F)=O)C1=O 17194,C(=O)(CC(CC(N)=O)CC(C)C)NC(CNC(c1c(C)nco1)=O)(C)Cn1cccn1 17195,C(=O)(CCC(C(C)C)NC(c1ncnc(O)c1F)=O)Nn1c(CC)nnc1 17196,N1(C(CCSC)=O)CC(CNC(c2c[nH]nc2-n2cnnn2)=O)CCC1C 17197,C(=O)(C1=C(c2ccccc2)SCCO1)NCC1(NC(CC(C)(C)C#N)=O)CC1 17198,c1(CC(N2CC(NC(C(C)OCC#C)=O)C(C)CC2)=O)cn2cccc(C)c2n1 17199,CC1CC(C(=O)N2CCN(C(=O)CNC(c3cccnc3)=O)CC2CCO)=NO1 17200,c1(CC)ccc(F)c(C(N2CCCC(CCCCNC(=O)C(F)(F)C(C)O)C2)=O)c1 17201,N(C(=NCC(C(C)C)C(C)C)NCC1CCCC1)CC1C(CC)CC1 17202,C12(O)CCN(CC1)C2.c1(-n2cc(C(N3CCOCC3)C)nn2)ccc(C)cc1 17203,Cc1ccc(C)c(C(=O)N(C(C)C(=O)NC2CCCCCC2CO)C2CC2)c1 17204,c1(OC)ccc(CSCCC(=O)NC2CC(C)N(C(c3ccc(F)s3)=O)C2)cc1 17205,C(=O)(C(C(C)C1CCCCC1)N1CCCCC1C(C)C(C)C)NCCCSC.C(C)=O 17206,Cc1nc(CC(=O)N(C2CC2)CC2CCCCN2C(C2CC3CC3C2)=O)c(C)s1 17207,CCCCCC(C)(CC)C(=O)NC1CCC(NC(c2ccn(C)c2)=O)CC1 17208,C12(C(N(C3CC(=O)CS3)CC(C)OCC)=O)CC3CC(CC1C3)C2 17209,C(C)(C)(CC(F)C(=O)Nc1ccc(Cl)c(O)c1)NC(c1cc(C)nnc1)=O 17210,Cn1c(O)nc2ccc(C(=O)NCCC3CCN(C(C4(C)CC4(C)C)=O)C3)cc12 17211,C=Cc1cnn(C)c1C(=O)N(CC(CO)(CO)NC(c1ccc(CC)cn1)=O)C 17212,c1(CC)cnn2ccc(C(=O)NC(C)CCCNC(=O)CN(C)CC)nc12 17213,C1(CC=C)(NC(C2CC(C)(NC(=O)C=CCO)C2)=O)CCCC1 17214,C1(COC)C(NC(C2CCCSC2)=O)CCCN1C(c1sccc1OC)=O 17215,C(CCN(C)C(C1CC2(C1)CC(F)C2)=O)(C(C)(C)C)NC(CC(=O)OCC)=O 17216,c1(Sc2ccc(C(N(c3cc(F)c(C)c(Br)c3)CC)=O)[nH]2)c[nH]c2ccccc12 17217,CC1=C(C)CC(C(=O)N(C)CC2CN(C(C3CN(C4CCCCC4)C3)=O)C2)CC1 17218,CC(C)(CCC(=O)N1CC2CC1CS2=O)c1ccc(OC(F)(F)F)cc1 17219,C1(=CC(=O)NCC(C2CCC2)NC(=O)Cc2cnc[nH]2)CN2CCC1CC2 17220,Cc1sc(N2CCCC2c2ncccn2)nc1I 17221,c1(C(N(CC)Cc2nncs2)=O)ccc(CNC(c2oc(C)cc2C)=O)nc1 17222,C1(NC(C(C)NC(=O)NC)=O)CCCC12CCN(C(c1occc1Br)=O)C2 17223,c1(CNC(c2nnc(SCCC)s2)=O)nc2cc(Cl)ncc2n1C 17224,CCC(CC)CC(F)C(=O)N1CCCC1C(C)(C)CNC(c1n[nH]cc1C)=O 17225,CC(C)C(C(=O)NC(C1CCCC1)CNC(=O)C(c1ccccc1)F)NC(N)=O 17226,c12nc(-c3nc[nH]n3)nn1C2.Cc1cc(CSc2csc(Cl)n2)no1 17227,CCC(C)C(C(=O)NCC1(CNC(=O)CC2CSC2)CC12CCC2)OC 17228,N1(C(C(CN(C(C(CCC)OCC)=O)C)C)=O)CC2CCC(C1)N2CC 17229,C1(CNC(CCCCSC)=O)N(C(=O)Cc2cc[nH]c2)CCCC1(C)C 17230,CC(F)(F)C(C)(C)CC(=O)N1CCCCCC(N)C1.n12cc(nn1)CCC2 17231,C=CCC(C)(C)CC(=O)NCC(=C1CN(C(=O)C(CCC)c2ccccc2)C1)F 17232,C1(C)(C(N(C)CC2CCCN(C(C3CC4CCC3C4)=O)C2)=O)CC(C)OC(C)C1 17233,CC(C)C(C)(O)C(=O)N1CC(F)(C(=O)NCC2CCC3(CC3)C2)C1 17234,C(=O)(C(C#N)C(C)C)NC1(CCNC(Cc2c(C)oc(-c3cccs3)n2)=O)CC1 17235,C12(CCNC(C(CC)(F)F)=O)CCC1CN(C(c1cncc(C)n1)=O)C2 17236,C1(C2CC2)(CNC(=O)CCc2cnoc2)CCN(C(c2cccnn2)=O)C1 17237,c1(C(N(CC(C)O)CC2CC2)=O)cn(CCNC(=O)CCOCC2CCCO2)nn1 17238,CC(C)(C)CCCC(=O)N1CCCC(CCNC(C2COC(=O)C2)=O)C1 17239,CCC(Cc1ccccc1)(CCn1cc(C2(C)CCCO2)nn1)C(=O)O 17240,c1(C(C)NC(c2c(CNC(CCCOCC=C)=O)noc2)=O)cccnc1F 17241,C(=O)(C(CCOCCO)NC(=O)C=C1CCCCC1)NCCC1(N(C)C)CCC1 17242,c1(N)ccc(OC)nc1Cl.C(=O)(CCC(=O)N1CCN1CCC)NCC 17243,C1(C(=O)NCC2(O)CCOCC2)CCC2(CN(C(=O)C(O)C3CCC3)C2)O1 17244,C1(CCCC)CCC(C(=O)NC(C)CCNC(c2cccc(CC3CC3)c2)=O)CC1 17245,N1(C(C=C2CCN(C)C2)=O)CCCC2C(NC(=O)C=CC(F)(F)F)C(C)(C)C12 17246,c1(C(C(=O)O)=O)ccc(F)c(F)c1F.c1(C2C(CCN(C=O)CC)C2)sccc1C 17247,C(=O)(C1=NN(CC)C(=O)CC1)N(CC(CC)NC(=O)Cc1c(C)cccc1Cl)C 17248,c1(N(CC(CN(C)C(C2(F)CCCCC2)=O)O)C)nc2c(cc1C#N)CCOC2 17249,Cc1ccc(CNC(=O)CCC2(NC(c3[nH]nnc3C)=O)CCC2)o1 17250,n1(C(C)C)ncc(C(=O)NC(C)CNC(=O)C=Cc2cccnc2)c1F 17251,C12(OC)CCN(C1)C2=O.C1(C2CC2)(CNC(=O)Cc2ccoc2C)CCC1 17252,C(=O)(C1=CC2CCC(C1)C2)N1CC2C(CN(c3ccccc3)C(C)C)(CC2)C1 17253,N1(C(C2CC(OC)CN2C(=O)CC2CCN(C)CC2)=O)CCC2(CNC(=O)O2)C1 17254,c1(C(=O)NCC(=C)CCNC(=O)C(C)(C)N(C)C)cnc(OC)cc1C 17255,C1(C(N2C(CC(=O)NC3CC(CSC)C3)C(C)(C)C2)=O)CCC=CCCC1 17256,C12(C(=O)NC3CC(O)(CNC(c4ccoc4Cl)=O)C3)C(=O)C3CC1C2C3 17257,c1(C(N(C)CC2CCN(C(C(CCC)O)=O)C2)=O)cc(S(=O)(=O)N(C)C)oc1C 17258,c1(C(N(CCCC)CC(N)=O)=O)ccc(CNC(C2CCCS2)=O)nc1 17259,N1(C(C(C)Cc2cccnc2)=O)CCCN(C(C2(CCN(C)C)CCCC2)=O)CC1 17260,C=Cc1cncc(C(N2CCC3CC23C(=O)NCCc2cc(C)no2)=O)c1 17261,C1(NC(=O)NCCOC)CCN(c2ccnc(NC3CCCCC3C)n2)CC1 17262,C(=O)(CC(C)(C)COC)NC1(CC=C)CCN(C(c2cc(Br)n[nH]2)=O)C1 17263,c1(C(N2CCCC(N(C(=O)CCN3CCOCC3)C)C2)=O)ccc2c(n1)COCC2 17264,C1(CC)CC(C(N2CCC(=O)NCC2)=O)CCN1C(c1cccc(Cl)c1)=O 17265,C1(NC(C2(C)CCN(C(C)=O)C2)=O)CCN(C(C2CCS(=O)(=O)CC2)=O)C(C)C1 17266,c1(C(=O)OC)cc2c(cc1Br)CN(C(c1ccc3ncncc3c1)=O)C2 17267,C1(NC(C(CSC)(C)C)=O)CN(C(c2cc(Cl)c(Br)[nH]2)=O)CCC1C 17268,C12CCN(CC1)C(=O)C(C(C)C)O2.CCC(F)C(=O)NCC(C)C 17269,N1(C(C2(OCC)CCC2)=O)CCC(CN(C(=O)CN(C)C(C)C)C)CC1 17270,C1(C(N2CC2)=O)C(OC)CCC12CCC2.C(C(F)(F)F)N(C(=O)COC(C)=O)CC 17271,N1(C(CCC)=O)CC(NC(c2ccc(Br)c(C)c2F)=O)C2(CCC2)C1 17272,c1(C(c2ccccc2OC(F)(F)F)OC)cc(C)c(Cl)s1.n12nnnc1NCC2 17273,N1(C(Cn2nc(C)oc2=O)=O)CCC(NC(C2(CC(F)F)CCC2)=O)C(O)C1 17274,c1(N(C)CC2CCN(C(=O)CC3CCC(C)(C)O3)CC2)ccc([N+](=O)[O-])cn1 17275,CC(C)(C)CC(C)(C)C(=O)NCC1CC1CNC(=O)CCn1cc[nH]c(=O)c1=O 17276,c1(C(=O)NC(CNC(c2nc(C)[nH]n2)=O)C)coc(=O)c2ccccc12 17277,c1(C(=O)NCC2CCC(NC(CC3CN(C)C3)=O)C2)sc(F)cc1Cl 17278,c1(CC)cc(C(N2CCC(CCNC(c3cc(COC)no3)=O)CC2)=O)c(C)o1 17279,c1(OC)cc(Br)ccc1C(=O)CNC1CCCCC1NC(=O)OC(C)(C)C 17280,C1(C(N2CCCC(c3ccccc3F)C2)=O)CC2CCCCCCC12 17281,n1(C(C)C)ncc(Cl)c1C(=O)NCC(C1CC1)N(C)C(C1CC1F)=O 17282,N1(C(c2cccc(-c3cn[nH]c3)c2)C(=O)NCC=C)CCC(C)C(C)(C)C1 17283,c12ccc-1cc2.CC(O)CCN(CCC#N)C1CC1 17284,C1(C(=O)NC2(CN(C)C)CCCCC2)CN(C(c2cnco2)=O)CC12CCC2 17285,C1(CNC(Cc2nc(COC)sc2)=O)(OC)CCN(C(C2CC2CF)=O)C1 17286,CCCCCCCC(=O)N1CC(NC(c2cc(F)ccc2C)=O)C(O)C1 17287,c1(CC)cccnc1C(=O)NC(CCN(C(=O)C(C)CSC(F)(F)F)C)C(C)C 17288,c1(C(=O)CC#N)cnn2c1CCC2.C1C(C)(C)CCN1C(C1CN(C(C)C)C1)=O 17289,Cc1sc(Cl)c(C(=O)NCCOCCCNC(=O)CCC2CCN(C)CC2)c1C 17290,CC#CCCCC(=O)N1CCCC1CCCNC(=O)COc1cccc(C)c1 17291,CCCCC(C(=O)NC1CC1)NC(=O)CONC(=O)C(C)SC(C)(C)CC 17292,C1(NC(C(COCC)n2cc(-c3ccsc3C)nn2)=O)COCCC1(F)F 17293,CC(C)CS(=O)(=O)CCC(=O)NC(CNC(C1CCN(C)C(=O)C1)=O)C1CCC1 17294,C1(C(N(C)Cc2c(C)cco2)=O)CC(NC(=O)Cc2cncn2C)C1(C)C 17295,N1(C(c2cc(C(C)C)on2)C(=O)NC2COC2)CCc2ccc(Cl)nc2C1 17296,c1(OC)ccc(C(=O)NCC2CN(C(=O)CC34CCCC3C4)CC2O)cc1OC 17297,N1(Cc2cc(OC)ncc2)CCN(C(=O)C(C)CC(C)=O)C2CC12 17298,C1(NC(Cn2ncn(C)c2=O)=O)CC(NC(=O)CC2COC(=O)N2)C12CCC2 17299,N1(C(=O)CCc2ccccn2)CCC2(NC(C34C(=O)C5CC3C4C5)=O)CC2C1 17300,C#CCCCCC(=O)N1CC(CNC(c2cc(C(N)=O)cc(C)c2)=O)CC1C 17301,c1(C(N2CCN(C3CCN(C(C4(CCCC)CC4)=O)C3)CC2)=O)ccc(O)nc1C 17302,C1(C(=O)NC(C(C)NC(c2cc3occc3s2)=O)(C)C)CCc2nncn2C1 17303,c1(C2C(C(=O)NCC3(CNC(C4CCCCC(F)C4)=O)CC3)C2)cc(O)ccc1F 17304,C=CCC(C)(C)CC(=O)NC1CN(C(c2cnc(CC)s2)=O)CCC1CO 17305,c1(C(N2CCC(NC(c3c(CC)ocn3)=O)C2C2CC2)=O)c(F)cc(F)cc1Cl 17306,N(C1CCc2c(Br)cccc21)C(c1cccnc1-c1cnn(CCF)c1)=O 17307,CCCC(CCC)C(=O)NCCC(C)NC(C1CCS1(=O)=O)=O 17308,C1(C(N2CCC(OCCNC(c3ccc(SC)cc3)=O)C2)=O)CCCCN1N=O 17309,c12cc(co1)CNC2=O.C(C(COC)OC)C1(C(=O)OCc2ccon2)CC1 17310,C=C(C)CCCNC(=O)CO.C1(C)(C)CNC(=O)C(=O)NCCCO1 17311,O=C(C1=CS(=O)(=O)c2ccccc21)N1CCC(NC(C2(Br)CC2)=O)CC1 17312,C1(NC(c2n(C)ncc2)=O)CCC2CCN(C(c3ncncc3Cl)=O)C1C2 17313,N1(C(CCCNS(C)(=O)=O)=O)CCOCC1CCNC(C1CCOC1C1CC1)=O 17314,O=C(C1=CC(O)C(O)C(O)C1)NC1CC(F)(CO)C1 17315,c1(C(N2C3CC(NC(c4cc(=O)cc[nH]4)=O)C(C3)C2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 17316,N1(C(CCS(C)=O)=O)CCC(NC(=O)Cc2ccc(F)c(Cl)c2)C12CC2 17317,c1(C(N(CC(CNC(Cc2scc(C)n2)=O)C)C)=O)cccc(C2CC2)n1 17318,CCCC(O)(CCC)CC(=O)N1CCCC(C2(NC(C3(N(C)C)CC3)=O)CC2)C1 17319,C(c1cnn(C)c1C)=CC(N1CC=CC(NC(c2ccc(NC)cc2)=O)C1)=O 17320,c1(C(=O)NC2C(NC(C3(CC)CC34CCC4)=O)CCC2)cnnc2ccccc12 17321,c1(-c2cnc(CCC(=O)NCCCNC(c3cnn(C)n3)=O)o2)cccc(F)c1 17322,C(=O)(C1CCCc2nncn21)N(CCN(C(=O)C=Cc1ccco1)C)C 17323,S(=O)(=O)(c1ccc(C(N2CCC(C)(CNC(c3ccoc3)=O)C2)=O)cc1)NCC 17324,c1(C(=O)NCC(CC=C)NC(c2nn(C)nc2Br)=O)cnc(C)n1C 17325,N1(C(c2cc(C(C)C)on2)=O)CCCC(CC(=O)NC2CC3CCC2O3)C1 17326,Cc1oc(S(C)(=O)=O)cc1C(=O)NCCOC1CCN(C(C2CC2Cl)=O)CC1 17327,c1(CSC)c(C(=O)NCC2CC2NC(c2csc(=N)[nH]2)=O)oc2ccccc12 17328,C1(C(C)(C)C)(CNC(=O)COCCF)CCN(C(=O)CCOC2CCSC2)CC1 17329,C1(C)(NC(c2ncn(C(C)C)n2)=O)CCN(C(c2cc3n(n2)CCO3)=O)CC1 17330,c1(C(N2CCCC3(NC(C(C)OC)=O)C(C2)C3)=O)cc2c(F)ccc(Br)c2[nH]1 17331,N1(C(c2c(C)csc2C)=O)CCCN(C(=O)C=CCCc2ccccc2)CC1 17332,S(=O)(=O)(c1csc(C(N2CC(N(C(=O)COC(F)(F)F)C)C3(CC3)C2)=O)c1)NC 17333,c1(C(=O)NC2(CF)CCN(C(=O)C=CC3CCC3)C2)cnc2ccc(F)cc2c1 17334,c1(C(N2CC3C(CNC(c4n(CC)cnn4)=O)(C3)C2)=O)ccc2c(n1)CCCC2 17335,CC(O)CC(=O)NC(Cc1cc[nH]n1)C(=O)N1CC(O)(c2cc[nH]n2)C1 17336,CN1C(=O)CCC1C(=O)NCCN1CCC([NH+](C(=O)C(F)n2ccnc2)[O-])CC1 17337,N#Cc1cc(N2CC3(CN(C(c4ns[nH]c4=O)=O)C3)C2)nc(C2CC2)n1 17338,C1(NC(c2c(CC)occ2C)=O)CN(C(c2ocnc2C2CC2)=O)CCC1F 17339,CC1CCCN(C(c2cnsc2)=O)C1CNC(C1OCCN(C)C1=O)=O 17340,C1(NC(C(CC2CCCC2)NC(C)=O)=O)C=CCN(C(C2(C)CCC(=O)N2)=O)C1 17341,c1(N(CCCNC(CC2C(OC)COCC2)=O)C2CC2)ncn(C)c(=O)c1Br 17342,c1(C(=O)NCCCCCN(C(C)C)C(C2C=CCC2)=O)ccc(O)c(F)c1F 17343,N(C(=NCCC(=O)N(C)C)N1CCC2(CCN(C)C2)C1)C1C(CC(C)C)C1 17344,c1(SCCNC(=O)NC(CC)CCCO)cc(Cl)ccc1Cl 17345,CC1(C)CC(NC(C2CC2c2ccc(Cl)cc2)=O)CN1C(=O)Cc1ccc(F)cn1 17346,C(CCCC(=O)NC(C)(C)C(=O)N1CCOCC1)C1C(C)C1 17347,C1(NC(C)(C)C)CC2CCC1C1C(=O)N(CC(=O)NC34CC(F)(C3)C4)C(=O)C21 17348,C1(C(=O)NCCCCNC(c2c(C)cc(C)nc2)=O)CCc2nnc(O)cc2C1 17349,c1(C(N2CCN(Cc3ccc(C(F)(F)F)nc3)C3CC23)=O)cn2ncccc2n1 17350,N(C1CC(F)(F)c2ccccc21)C(=O)C(N1CCc2ccc(F)cc21)=O 17351,Cc1nc2cc(C(=O)NCC3(F)CCN(C(c4cnc[nH]c4=N)=O)C3)[nH]c2s1 17352,C(C1CCOC1)=CC(=O)NC1(CC(=O)NCC2(CO)CCOC2)CC1 17353,C1(CC(N2CCC(COC)(NC(=O)C3=C(C)CC3)CC2)=O)CC(C)CC(C)(C)C1 17354,c1(C(=O)OCC)cc(C(N2CCOC(c3ccsc3)C2)=O)n(C)n1 17355,c1(C(=O)NC2CC(C(N(CCCC(C)O)C)=O)C23CCC3)cccc2[nH]ncc12 17356,Cc1c(NC(=O)C(=O)NCC2CCCN2C)cnn1-c1ccncc1 17357,CCC(CC)C(C)C(=O)N1CCN(C(=O)CC(F)(F)CC)C(c2ccccc2)C1 17358,c1(C(=O)NCC(C)CNC(=O)CCN(C)CCO)ncnc(O)c1Cl 17359,CC1CCC(CCC(=O)N(C(Cc2cccs2)CO)CC(F)F)O1 17360,c1(CN2CCCC(C(=O)Nc3cccnc3S)C2)cccc2ncccc12 17361,C(=O)(CCCC(C)(C)C(=O)OC)NC(CN(C(C(C(C)OC)N(C)C)=O)C)C 17362,Cc1ccc(CNC(C2C3CC3CN2C(=O)CCC2CC2C)=O)nn1 17363,N1(C(c2cn(CC)nn2)=O)CC2(CCCC2NC(c2cc(C)no2)=O)C1 17364,c1(C(N(C2CCCCCC2)CCNC(c2c(C)cns2)=O)=O)nnn2c1CCCC2 17365,c1(CN2CC(NC(CS(=O)(=O)N(C)C)=O)C(F)CC2)ccc2c(c1)OCCCO2 17366,N1(c2ncc(C#C)cn2)CCN(C(c2cc(F)c(Cl)cc2F)=O)C(C#N)C1 17367,Cc1cc(C(=O)N(CCCNC(=O)Cc2sc(C)nc2C)C)c([N+](=O)[O-])c(O)n1 17368,C1(NC(C2(CCCC)CC2)=O)CC2(C(=O)NCC3CC(=O)N(C)C3)COC1C2 17369,c1(C(N(C(CNC(C(CC=CC)C)=O)C2CC2)C)=O)cc2occc2s1 17370,C1(=O)C(C)C(C)N1C(=O)C(n1cc(-c2c(C)ncn2C)nn1)C.C(=O)(CO)OC 17371,N1(C(C(Br)=C(C)C)=O)CC2CCN(C(c3scc(C)c3Cl)=O)C2C1 17372,Cn1cnc2c(C(N3CCOC(CNC(=O)CC4(C)CCCO4)C3)=O)ccnc12 17373,Cc1cc(C(N2CC(C)C(C)(CNC(=O)C(C)OCC3CC3)C2)=O)nnc1C 17374,CCCCCC(O)CNC(C1CCC(NC(c2cc(C)oc2CC)=O)C1)=O 17375,CC#CCCCC(=O)NC1CCC(CCNC(=O)Cc2cnc(C(F)(F)F)s2)C1 17376,c1(C(=O)NCC2(CNC(C3C(C=C)OCC3)=O)CCCC2)cc(Cl)c(Cl)n1C 17377,Cc1cc(C)c(S(N)(=O)=O)cc1C(=O)NCC1C2CN(C(=O)C3CC3)CC12 17378,O=C1Cc2ccc(C(=O)NC3(c4ccc(Cl)c(Cl)c4)CCC3)cc2N1 17379,N1(C(CC2(OCC)CCC2)=O)CCCC(CF)C1.c12cc(no1)C(=O)NC2 17380,C1(C)(NC(C(CC)O)=O)CCN(C(c2sc(CCCC(F)(F)F)nc2C)=O)C1 17381,C1(C(N(CC(NOCC#C)=O)C(C)C)=O)CC12CCCC2 17382,C(=O)(C(C)(C)CC(F)F)NC(C)CC(C)NC(C1CCN1C(C)(C)C)=O 17383,CCC(C(=O)N1CCC(C(C)(C)NC(C2CCC(N(C)C)CC2)=O)C1)C(C)C 17384,Cc1sc(O)nc1C(N1CC(C=C)(CC(=O)NCC2(C)CC2(C)C)C1)=O 17385,CC1OC2(C(=O)OCc3cccs3)CCC1CC2.c12ccc(cc1)[nH]c2=O 17386,CC1C(C)CCN1C(c1c[nH]nc1CCNC(=O)CCC(=O)N(C)C)=O 17387,N1(C(C(CC2CCC2)NC(c2c(C)nc(C)o2)=O)=O)CCN(C)C(C2CC2)C1 17388,c1(CC)ccccc1C(c1nnnn1C1CCNC1=O)Nc1c(SC)csc1 17389,C(CCNCC(O)CC(=O)OCc1ccccc1Cl)(C(=O)OCC)OC 17390,CC1CN(C(C2CS(=O)C2)=O)CCC1NC(=O)CC(C)(O)C1CC1 17391,CC(C)(C)CCCCC(=O)NC1CN(c2c(Br)cccc2[N+](=O)[O-])CC(C)(C)C1 17392,C(C)(CCC(=O)NC(CNC(C1CCN(S(C)(=O)=O)CC1)=O)CO)OC 17393,c1(C(N2CC(O)C(F)C2CNc2ccc3c(n2)CCC3)=O)cc(Cl)c(Cl)cc1Cl 17394,C1(NC(c2sc(CC)c(C)c2)=O)CN(C(C2(CCOC)CCC2)=O)CC1(C)C 17395,CC1(C)CC(NC(C2(n3cccc3)CCCC2)=O)CN1C(C1CCOC1)=O 17396,c1(CCC)ccc(C(=O)NCC(Cc2ccco2)CC(=O)OC)cc1CO 17397,C1(C(=O)NCCC2N(C(CCC(=O)NC(N)=O)=O)CCSC2)CCCC(F)(F)CC1 17398,N1(C(C(c2cnn(C)c2)C)=O)CCC(NC(c2cc(C(N)=O)no2)=O)CC1 17399,C12(CNC(=O)NCc3[nH]cc(C)c3)CCCC(C)(C1)OC2 17400,c1(OC)cncc(C(C(=O)NCC2CCOC2)N(CC(F)(F)F)CC2CC2)c1 17401,C1(CNC(c2cc(CC)no2)=O)CC(F)(F)CN1C(c1ccc(N)c(Cl)n1)=O 17402,N1(C(c2occ(C(C)=O)c2)=O)CC(NC(=O)CCn2ccc(C)n2)C(C)C1 17403,CCCCN=C(NCCN1CCCS1(=O)=O)NCC1CC(CC(N)=O)C1 17404,N1(C(CSS(C)(=O)=O)=O)C2CCC1CC(NC(c1cc(Cl)no1)=O)C2 17405,C=CC(CC)CC(=O)N1CCC(C(=O)NCCn2cncc2C)C12CC2 17406,CC1(C)OC2(CC3CCCCC3)CC1(C(=O)NCC1(C(=O)NC3CC3)CCC1)C2 17407,CN=c1cc(C(=O)NCC(c2cn(C(C)C)nn2)(C)C)c(Br)c[nH]1 17408,C1(C(=O)NCCN(C2CC2)CC)CN(C(c2ccn(C)c2)=O)CCN1C 17409,C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NC1CN(C(c2c(OC)nsc2OC)=O)C1 17410,c1(CN2CCC(N(C(c3cccc(CC)n3)=O)C)C2)ccc2c(c1)OCCO2 17411,C1(CNC(C2(NC(=O)NC)CCCC2)=O)CCC(NC(C2CC2CF)=O)CC1 17412,C=CCCC(O)CN(C)C(C1CC(C)CN1C(=O)C=C1CCCCC1)=O 17413,C1(NC(c2c(C)[nH]cc2)=O)CC2CC1N(C(=O)CNC(c1cccnc1)=O)C2 17414,c1(CC)ncc(Br)cc1C(N1CC2CC2(NC(C2CCC(CC)O2)=O)C1)=O 17415,c1(C(=O)OC)c(NC(=O)NCc2ccc(N(C)C)cn2)cccc1C 17416,c1(SCC(=O)NC2(C3CN(C(C4(C)CCC(C)C4)=O)C3)CC2)cccc([N+](=O)[O-])c1 17417,N1(C(C2C(OC)CCC2)=O)CCC(C)C1C(=O)N(C)Cc1ccncn1 17418,CC1(NC(=O)NCC(CN2CCOCC2)CO)CS(=O)(=O)CCO1 17419,Cc1ccc(CC(=O)NC(C)(C)CCN(C)C(C2(C)CC2F)=O)o1 17420,C12(C(N3CC(N4CCN(C5CC5)CC4)C(O)C3)=O)COCC(c3cccs3)(C1)C2 17421,CC1CCC(CC(=O)NC(C)CCCNC(=O)C(C2(O)CCCC2)F)O1 17422,c1(C(=O)NCC2C3CCC(C3)N2C(C2CC23CCC3)=O)ccc2c(c1)COCC2 17423,N1(C(c2n[nH]c(C)c2C)=O)CCOC2CN(C(=O)C(C)(O)C(F)(F)F)CC12 17424,C12(NC(CC(C)C3CC3)=O)CCCN(C(=O)COc3ccccc3O)CC1C2 17425,N1(C(CNC=O)=O)CCCC(CCNC(C2CC3C=CC2CC3)=O)CC1 17426,C1(NC(CSC)=O)CCN(C(=O)C(C)C2CCOC2)CCC1CO 17427,C(=O)(C1=CSCCO1)N1CC(CCNC(C2CN3CCC2CC3)=O)OCC1 17428,c1(C(N2CC(NC(C#CC(=O)N(C)C)=O)C(O)C2)=O)cc(F)cc([N+](=O)[O-])c1 17429,c1(C(=O)NCC(CO)NC(C2(C)CC2(F)F)=O)cc2c(nn1)CCC2 17430,Cc1cc(F)c(C(=O)NCC(C)(C2CC2)NC(c2csc(CO)n2)=O)c(Cl)c1 17431,CC1=C(C(=O)NC(C2CCCN2c2ccnc3ncnn23)(C)C)CCS1(=O)=O 17432,c1(C(=O)OC)ccc(-c2cccc(C(F)F)n2)c(Cl)c1 17433,N1(C(C2C(=O)NCC2)=O)CCC2CC1CN(C(c1ccc3c[nH]nc3c1)=O)C2 17434,c1(C(=O)NCCC2N(C(C3(SC)CCC3)=O)CCCC2)noc2cc(Cl)ccc12 17435,Cn1cc(CC(c2cn(CCC3COC(=O)C3)nn2)(C)C(=O)O)cn1 17436,N1(C(CONC(C(C)N(C(C)=O)C)=O)=O)CC2CCCC(O)C2C1 17437,CC1(C(=O)N(CCNC(=O)C(CO)c2ccccc2)C2CC2)CC1(F)Cl 17438,N1(C(CCc2nnc(C(C)C)o2)=O)CCN(C(=O)C(C)N(C)C)CC12CCC2 17439,c1(C(=O)NC2CC3(CC(C(=O)NCc4ccc(C)cn4)C3)C2)ccnc([N+](=O)[O-])c1 17440,N1(C(C(C)C2(O)CCC2)=O)C(C(=O)NCCN(C)CCF)CCC1C 17441,C1(O)(CC(C)C)CCN(C(=O)CC2(NC(c3ccnnc3)=O)CC2)C1 17442,CC1(CCC(N2CC=CC(NC(c3cnoc3C3CCC3)=O)C2)=O)CCC(=O)N1 17443,c1(CCC(N2CCC(C)(CNC(C)=O)C2)=O)cccc(C#N)c1 17444,C#CCC(CC#C)C(=O)NCC(C)N(C(=O)CCc1cccc(OCC)c1)C 17445,c1(C(C)N(C)C(=O)NCC(C)C#N)cccc(C(F)(F)F)c1 17446,C1(NC(c2c(SC)n(C)nc2)=O)CN(C(=O)CN2CCCCC2)CC(C)(C)C1 17447,N1(C(=O)CSc2ccc(F)cc2)CCCN(C(C2CCC3(CCC3)O2)=O)CCC1 17448,N1(c2nccc(SC)n2)CC2CCCC(NC(c3ccc(CCO)cc3)=O)C2C1 17449,C12(OC)CCC1CN(C(=O)C(CNC(=O)C(C)Cn1ccnc1)N(C)C)C2 17450,c1(C2(C(=O)NCC(CNC(=O)CC34CCCC3C4)CO)CC2)ccccc1Cl 17451,C(=O)(C#CC1(C)CC1)NCC(CCC)NC(=O)CC1CC=CC1 17452,c1(OC)ccc(Cl)c(F)c1C(=O)N(CCCN(C)C(C1(C)CC=C(C)CC1)=O)C 17453,c1(CC)ccc(C(=O)O)cc1F.n12cc(nn1)-c1ccc(s1)NC(=O)C2C 17454,c12ncc(s1)C(=O)N(CC)CCNC(=O)C(=O)NC2C.C(C)SC.C(C)(=O)N 17455,c1(C(N2CC(C(=O)NC(CCCC)C)C2)=O)ccnc2cc[nH]c12 17456,c1(NC(=O)OC(C)C)ccc(NC(C)(C)CNC(=O)CCc2ccccc2)nc1 17457,C1(C(=O)Nc2c(C(C)C)ncs2)CCN(C2CCN(CC(N3CCCC3)=O)C2)CC1 17458,c1(C(=O)OC)ccnc(N(CCCNC(c2occc2Br)=O)CC2CCCC2)n1 17459,C(CCCCCNC(c1nocc1Br)=O)NC(C1CC(OC)C1)=O 17460,C12(NC(=O)CSCCC(F)(F)F)CCC(C1)N(C(c1cccc(C3CC3)c1)=O)C2 17461,N1(C(C(CC=CC)C)=O)CC(NC(CC(F)Cl)=O)CC12CCC2 17462,C1(C)(C(=O)NCC(C)CN(C)C(c2cnn(C(F)(F)F)c2)=O)CCNC1 17463,C1(C(N2CCCC(CCC(=O)NC3(C)CCC3)C2)=O)CC2CCCC2C1 17464,C1(NC(c2n(C)cc(Cl)c2)=O)CCN(C(C2CCCOC2)=O)CC12CCC2 17465,c1(CC)cc(C(N2CC(NC(c3csnn3)=O)C(n3ccnn3)C2)=O)c(C)nn1 17466,c1(C(=O)NC(C)C)ccc(N(C)C)cc1.N12CCCC1NC(=O)C2c1cnc[nH]1 17467,C(=O)(C(C)(C)C(=O)NC1CCCN(Cc2cc(Cl)ncc2NC)C1)N(CC)CC 17468,CC1(C)CCCC(CC(=O)NC2CN(c3nc(Cl)ncc3C(F)(F)F)CC2(C)C)C1 17469,N(C(=NCCc1ncccc1C)NCc1nn(C)cc1Br)C(COC)C 17470,N1(C(C(C)OCC(F)(F)F)=O)CCN2CCN(C(C3(C)CC3F)=O)CC2C1 17471,N1(C(C(C)=C2CCCC2)=O)C2CCCC1CN(C(C1CC3CCC1O3)=O)C2 17472,CCC(CC)C(C)C(=O)N(CC(=O)N(C1(COC)CC(C)(C)C1)C)CCOC 17473,c1(CC)occc1C(=O)NC1CC1CNC(=O)CCc1cn[nH]c1 17474,c1(C(N2CC(SC)C(NC(C3(C)CC=CCC3)=O)C2)=O)cc(C)cc(C)c1N 17475,C12(NC(C(C)(C)O)=O)CN(C(c3[nH]nnc3C3CC3)=O)CC1CS(=O)(=O)C2 17476,CC1CCCN(C(c2ccsc2)=O)C1CNC(c1cnn(CC(F)F)c1)=O 17477,c1(NC2(CCCC)CC2)ncccc1S(=O)(=O)NCCc1cccc(F)c1 17478,C1(CC(C)NC(C2C(COC)C2)=O)CC2CCC(C1)N2C(=O)C=Cc1cnc[nH]1 17479,c1(C(=O)NCC(C2CCN(C(CC(C)SC)=O)CC2)(C)O)c(O)cccc1F 17480,CCCCC(F)C(=O)NCCC1CC(C(N2CCC(CC(C)(C)C)C2)=O)C1 17481,c1(COCC#C)cccc(C(=O)NC2CCC(CCNC(=O)CC3CCC3)C2)n1 17482,CCC(CC(=O)NCC(C)(C)OCCN(C)C)CC(C)C.n12cc(nn1)C2 17483,C1(F)(CNC(C=CCCC)=O)CCN(C(=O)CSCCOC)C1 17484,C(=O)(C(O)CC(C)(C)C)NCC1(F)CCN(C(C(CC)C#N)=O)CC1 17485,C(=O)(C1=C(Cl)CCC(C)C1)NCCCC1CCN(C(CCC#CC)=O)CC1 17486,C1(C(=O)Nc2n(C)c(S)nn2)CC2(CCCCN2C(=O)COCP(C)(C)=O)C1 17487,N1(C(CCC)=O)CCCC(CCNC(=O)C(c2cc(Cl)cc(Cl)c2)(C)C)CC1 17488,Cc1ccc(C(C)NC(=O)NCC(c2ccc(C(=O)O)o2)C)cc1 17489,c1(CN(C(c2ccncc2)C)C)cc(Cc2ccccc2)on1 17490,CN1CCOCC1CC(=O)NC1CCC1NC(C1CC(n2ccnn2)C1)=O 17491,c1(NCCCSC)cc(C)c(S(=O)(=O)N2CCSC2c2ccco2)cn1 17492,C(C(=O)NOCc1cccnc1)(C1CC1)NC(C1CCS(=O)(=O)N1)=O.C(COC)S 17493,C=CCC(CNC(c1ccc(F)s1)=O)NC(=O)CC1CCCOC1 17494,N1(C(C2CN(C(C)=O)C2)=O)CC2C(C1)C(C)N2.c1(CC(=O)N)csc(C)n1.C(F)F 17495,N1(C(c2nn(CC)c(C)c2)=O)CCC2(CCCN2C(=O)C(O)C2CC2)CC1 17496,Cc1nn2cc[nH]c(=O)c2c1C(=O)NCCC(O)CNC(=O)C(C)C(C)(C)C 17497,C1(C)(C(=O)NC2C(O)CCN(C(C(C)OCC(C)C)=O)C2)CCS(=O)(=O)CC1 17498,CON(CCC(=O)Nc1ccsc1C)C(=O)C1(C#N)CCOC1 17499,N1(Cc2ccc(CC)cc2)CC(C(=O)NC2(C(N)=O)CCC2)CC(C(F)(F)F)C1 17500,CC(C)CC(C)(C)CNC(C1CCN(C(=O)C2C(C)(C)C2(F)F)O1)=O 17501,C1(C(N(C(CC(=O)NC)C)C)=O)COCCN(CC2CCCO2)C1 17502,C1(NC(CCOCC)=O)CN(C(C2Cc3nccnc3C2)=O)C2(CCOCC2)C1 17503,c1(NC(C2COCCN2C(C2CC(O)C2)=O)=O)c(F)c(F)nc(F)c1F 17504,c1(CC)cc(C)[nH]c(=NCC2CC(NC(=O)Cc3nn(C)cc3Cl)C2)n1 17505,C1(C)(CCNC(c2n(C(CC)(C)C)nnn2)c2c[nH]nc2C2CC2)CCC(=O)N1 17506,CC1(C)C(NC(c2ccnc(NC(N)=O)c2)=O)CCN1C(c1n[nH]c(=N)[nH]1)=O 17507,c1(CN=c2scc(C(=O)Nc3ccc(O)c(C)c3C)[nH]2)c(F)cccc1[N+](=O)[O-] 17508,CS(C)(=O)=NCC(=O)NC1CCOCC1NC(=O)C=Cc1ccccn1 17509,C#CCC(CC(F)F)C(=O)N1CCC(C(F)C(N2CCCC2CC(=O)OC)=O)C1 17510,C12(NC(C=CS(C)=O)=O)CCOCC1CN(C(c1ncnc3ccsc13)=O)C2 17511,C1(NC(C2N(C(c3c(CC)cc[nH]3)=O)CC=C2)=O)CC2(CCOC2)C1 17512,c1(C(=O)OC(=O)CCc2nnc(CCC(=O)OC)o2)ccc2[nH]cc(C#N)c2c1 17513,N1(C(CCN2C(=O)OCC2)=O)CCC(CCO)(CNC(C2(CO)CCC2)=O)C1 17514,C12(C(=O)NC3(CC=C)CN(C(c4csc(CC)n4)=O)C3)CCC(F)(CC1)CC2 17515,Cc1nc(SCC(=O)N(CCCNC(=O)C(C)CC2CCCC2)CCO)n[nH]1 17516,Cc1ccc(-n2ccnc2)cc1C(N1CCN(CC2CC2C)CC1)=O 17517,N1(C(C2CN(C(C)C)C(=O)C2)=O)CC2CCC2(CCNC(=O)C#CC2CC2)C1 17518,C1(NC(=O)NC2CCN(S(=O)(=O)C(F)F)CC2)CCCN(c2ncc[nH]c2=O)C1 17519,N1(C(c2cc(C)c(Br)s2)C(=O)NCCSC)CCC12CCN(C)C2 17520,c1(C(N(C(CNC(=O)C2=CCCC2(C)C)C2CC2)C)=O)cc(F)cc(N)c1F 17521,C(=O)(CCS(C)(=O)=O)NCC(CC)(CC)NC(C1CC2C=CC1O2)=O 17522,Cc1cc(Cl)ccc1C(N1CC(CN(C(=O)Cn2cnnn2)C2CC2)C1)=O.CO 17523,C1(C(N2C(C)C(CO)CCC2)=O)CC2CC1CN(C(=O)CCc1cscn1)C2 17524,C1(NC(Cn2c(C)nnn2)=O)CN(C(=O)C(C)(C)N(C)C)CCC1C(N)=O 17525,Cn1cc2c(n1)CCC(C(N1CCC(NC(=O)C=Cc3ccc(Cl)cc3)C1)=O)C2 17526,Nc1ncc(C(=O)NCC2CN(C(=O)Cc3cncs3)CC2(F)CO)cc1Cl 17527,C1(N(C)C)(C(=O)NCCCNC(C2CC2F)=O)CC1 17528,N1(C(c2c(C)c[nH]c2)=O)CCCCCC1C(=O)Nc1cnc(O)c(F)c1 17529,CC1CN(C(c2coc(C3CC3)n2)=O)CCN1C(=O)CCc1cc(Cl)no1 17530,c1(NC2CN(C(CCc3cc(C)cc(C)c3)=O)CC(F)C2)ncnc2occc12 17531,CC(C)C(C)CC(=O)NC(CC1CCC1)C(=O)N1CC(c2cnsc2)C1 17532,CC(C)(C)C(CNC(C1CC2CCC1C2)=O)C(=O)NCC1CCC(=O)NC1 17533,C1(C(N2CC(OC)C(NC(C34CC3C4)=O)C2)=O)CN2CCCN1CC2 17534,C(=O)(C1=C(CC)OCCC1)N(C1CCN(C(=O)CC(Cl)Cl)CC1)CC#C 17535,C1(C(=O)NC(c2ccc(F)cc2)C(=O)OC)Cc2cccc(C)c2O1 17536,N1(C(CCCCCC)=O)CC(C)CN(C(=O)CCC=CC(C)C)CC1C 17537,c1(C(=O)NC(CNC(C2N(C(C)C)CCCC2)=O)C)ccc(N)c(O)c1 17538,c1(C(N(CCC(C)NC(C2CC3(C2)CC(F)C3)=O)C)=O)coc2c(F)cccc12 17539,CC1CCOC(C(=O)NCCCCNC(c2cccc(C3(C#N)CC3)c2)=O)C1 17540,c1(C(=O)NC2C(CNC(C3C(CC)CCO3)=O)CCC2)ccc(C2CC2)cc1C 17541,CC1(C)C(C)(C(=O)NC2CN(C(c3cn(CCO)nn3)=O)CCC2CO)C1(C)C 17542,c1(NC(C2N(C(C(CC)SC)=O)CCCCC2)=O)ccc(OC)c(F)c1 17543,C1(C(=O)NCC23CC2CN(C(=O)Cc2cnncc2O)C3)CC12CCSCC2 17544,N1(C(CN(C(=O)OC)C)=O)CCCC(NC(=O)CCc2cncc(F)c2)C(F)C1 17545,C1(C(N2CCC(CCNC(c3ccccc3Cl)=O)C2)=O)CCC2(CC1)CC2(F)F 17546,C(=O)(CCCCC(N)=O)NC1C=CCN(C(c2nccc(C)n2)=O)C1 17547,N1(C(CCN2C(=N)NCC2)=O)CC2CC(C1)C2NC(=O)C(=O)NC1CC1 17548,CC1CCN(C(C23CC(CO)(CN2C(C2CC4(CCO2)CC4)=O)C3)=O)CC1CO 17549,N1(C(=O)CCC2CC2)CCC(N(CCO)C(C2(F)CCOC2)=O)C1 17550,C12(C(N3CCC3c3ncc(C)o3)=O)CCN(C1)C2=O.C1(CC)CC(F)(CF)C1 17551,C1(C(=O)NCC(C(C)C)NC(c2c(C(=O)OC)c(C)[nH]n2)=O)CC2(CCO1)CC2 17552,C1(N(C)C(C2CCC(O)CC2)=O)CCCN(C(=O)CN2CSCC2=O)CC1 17553,c1(CC)nc(C)oc1C(=O)NC(CO)C(=O)NCC1CCCSC1 17554,C(=O)(C1=CC2CCCC12)NCC=CCNC(c1cc(C)c(Cl)s1)=O 17555,N1(C(c2c(CC)nccc2)=O)CCC2C(C(=O)NC3CCCC(C)(C)C3)C2C1 17556,N1(C=O)CCc2c1ccc(F)c2Br.CC1(CN)CC1 17557,C1(NC(C2(COC)CCC2)=O)CN(C(c2ccccc2Cl)=O)C(C)(COC)C1 17558,c1(OC)cc(CNC2=NCCCS2)c(F)cn1 17559,C1(CNC(c2n(CC)ncc2Br)=O)CC2CCC1N(C(=O)C=CCOC)C2 17560,C=CCCCCCCCC(=O)N1CC2(C1)CN(C(=O)Cc1cnoc1)CCO2 17561,C(CS(=O)(=O)CC(=O)NCc1ccc(C(=O)NCC(CO)C2CC2)nc1)OC 17562,C(=O)(C#CC1CCCCO1)NC(C)(CNC(c1cc2n(n1)CC(F)C2)=O)CO 17563,C=CC(CC)CC(=O)NC1CCN(C(=O)CC2(CSC)CC2)C(C)C1 17564,C1(C2CCCN(C(=O)C3=C(Cl)CCC3)C2)(NC(C2(C)ON=C(C)C2)=O)CC1 17565,c1(CC)ccc(OCC(=O)NC2CCN(C(C3(C)COCCO3)=O)C2)cc1 17566,c1(C(=O)NCC(C2CCC2)NC(CC2C(C(C)=O)C2(C)C)=O)n[nH]cc1[N+](=O)[O-] 17567,C1(CNC(C(N2CCOCC2)C)=O)CCC(NC(c2ccnn2CC(F)F)=O)C1 17568,c1(C(=O)NCCCCNC(C2=CCCCC2C)=O)cc(=O)c2cc(F)ccc2o1 17569,c1(OC)cc(C(=O)NC(C)CCNC(c2ncc(F)cc2N)=O)cc(Cl)c1OC 17570,C(C)(CO)(C(=O)NCCCN(C(c1cnc(N)cn1)=O)C1CC1)OC 17571,C(C)(CCC(=O)NC(Cc1ccccc1)CCNC(C1(O)CC1)=O)SC 17572,N1(Cc2ccc(C(=O)OC)cc2)CCC(C#N)(Nc2ccc(CN(C)C)cc2)C1 17573,C(CC(=O)NC1CCCC1NC(c1c(C)nn(C)c1Cl)=O)(C1=CCCC1)OCC 17574,Cc1nc2ccc(C(N3CC(NC(C4CCC45CCC5)=O)C4(CC4)C3)=O)cc2o1 17575,c1(SC)cc(C(=O)NC2CCC(NC(=O)C(c3cncn3C)O)C2)n(C)n1 17576,C(=O)(C(C)C(O)C(C)C)NC(C1(CC=C)CCN(CC2C3C4CCC(C4)C23)C1)=O 17577,N1(C(c2c(N)nccc2)=O)CC2CCCN(C(c3cc4n(n3)CC(F)C4)=O)C2C1 17578,Cc1ccc(O)c(NC(c2cc(CNC(C3(COC)CCOC3)=O)cs2)=O)c1 17579,C1(CC)CCCC1C(=O)NC12CC(C(=O)NCCCc3ccncc3)(C1)C2 17580,N1(C(C=CC)=O)CCC2(CCCC2C(=O)Nc2cccc(Cl)c2F)C1 17581,CC1(C#CC(=O)NCC2CC(CNC(=O)Cn3cnnn3)CO2)COC1 17582,Cc1cc(NC(C2(NC(=O)COC3CCCC3)CCSC2)=O)nc(O)c1 17583,CC(C)P1(=O)CCN(C2CC(C)(C)S(=O)(=O)CC2)CC1 17584,c1(SCC(=O)NC(C2CCN(C(=O)Cn3ncn(C)c3=O)C2)C)cccc[n+]1[O-] 17585,c1(OC(C)C)ccnc(CO)n1.c12ocnc1C(=O)NCC1CC1CNC2=O 17586,c1(C(N2CC(C(C(=O)NCC(O)C=C)OC)C2)=O)ccc(O)cc1 17587,Cc1cc(C)n(CCC(N2CCC(CNC(=O)C=CS(C)=O)C2)=O)n1 17588,Cc1cc(=O)oc(C)c1C(=O)NC1CCN(C(=O)C(C)Cc2ccc(O)cc2)C1 17589,N1(C(c2cnn(CCCC)c2C)=O)CCCCC(CNC(C2(F)CCOC2)=O)C1 17590,c1(CC)ccccc1C(=O)NC1CCC1NC(c1cn(CCO)nc1C)=O 17591,CN=C(NCCCCSC)N1CCN(c2ncccc2[N+](=O)[O-])CC1 17592,n1(CC(=O)NCC(C(C)C)NC(c2cncc(OC)n2)=O)cc2ncccc2n1 17593,C=Cc1cc(C(=O)NCC2(O)CCN(C(=O)CC3CCCN(C)C3)C2)cc(F)c1 17594,C12(NC(CC3CC(OC)C3)=O)CCC(NC(=O)Cn3cc(C)ccc3=O)(CC1)C2 17595,CCC(CC(=O)N(CCCN(C)C)C1CC1)NC(=O)COCCCN=[N+]=[N-] 17596,C(CC)(CC)(CCNC(=O)Cn1cnc([N+](=O)[O-])n1)NC(C(C)SCC)=O 17597,N1(CCNC(=O)CNc2cncc(Cl)n2)CC2CN(Cc3ccc(O)cc3)C2C1 17598,N1(C(CCC(C)(C)OC)=O)CCCC2(NC(=O)CN3C(=O)CNC3=O)CCCC12 17599,c1(SCC(=O)NCC(=O)NCCNC(c2n[nH]cc2F)=O)cccc(F)c1 17600,CC12CC(NC(c3cncnc3)=O)(C1)C1(CN(C(=O)CC(O)C3CC3)C1)O2 17601,c1(CNc2c(Br)cc(C(=O)NC)nc2)ccc(F)c2[nH]ncc12 17602,O(C1CCCc2ccccc21)OCCNC(=O)NCc1cnon1 17603,C(c1ccc(C)c(Cl)c1)=CC(N1CCN(C(c2cccc(C)c2)=O)CC1C)=O 17604,c1(OC)cncc(C(N2CC(NC(=O)COC3(C)CCOCC3)CC2C)=O)n1 17605,N(C)(C1c2ccccc2CCC1N=c1nn[nH]n1C)C(C(c1ccccc1)C)=O 17606,N1(C(C(C=C)O)=O)CCC(C2CCOCC2)(CNC(c2cc(O)nn2C)=O)C1 17607,c1(C(=O)NC(c2nccn2C)C)cccnc1CNC(=O)C(O)CC1CCCC1 17608,c1(C(C2(O)CCN(C(=O)OC(C)(C)C)C2)OC(F)(F)F)cc2c(cn1)OCCO2 17609,Cc1ccc(O)c(CNCc2cc(C(=O)NOCc3c(C)noc3C)n[nH]2)c1 17610,C12(CO)CCC(C1)C(C)(C)O2.C12CCCCC1NC(=O)NCCO2 17611,N1(c2ccc(C)s2)CCCC(n2cc(-c3ccsc3)nn2)C1.C12CC(OC)CN1C2 17612,c1(C(=O)NCC2(F)CCC(NC(Cc3nc(C)sc3)=O)C2)c(Cl)ccc(O)c1N 17613,C=CC1(C(=O)N(C)CCC2CCCN2C)CCN(C(=O)COCCCOC)C1 17614,c1(C(N2CC(CC)(NC(=O)C(C)(C)Br)C2)=O)cc(C)c(OC(C)C)c(C)c1 17615,C1(C(N(C2CCN(C(C3(Oc4ccccc4)CC3)=O)C2)C)=O)CCC(=O)N(C)C1 17616,c1(C(=O)NCCCC(C)NC(=O)C(F)C2CC2)ccc(C(F)F)c(F)c1 17617,C1(NC(CC(CC)OC)=O)CCN(C(c2cc3nccnc3[nH]2)=O)CC(C)(C)C1 17618,N1(C(c2c(C(C)C)c[nH]n2)=O)CCC(F)(F)C(NC(=O)C2CC2)C1 17619,C1(OCC)CCC2(C(=O)NOc3ccnc(C)n3)CC12.N1(C=O)CC(OC)CC1 17620,C(=O)(C(C)(C)CC(=O)N1CCC(F)(C(=O)N(C)CC2C(C)(C)C2(C)C)CC1)OC 17621,c1(C(=O)NCC(C(C)C)NC(C2CC3CCC2O3)=O)ccc2ncnn2c1 17622,Cc1coc(C)c1C=CC(=O)NCC1CC1NC(=O)CCS(=O)(=O)N(C)C 17623,C1(CC(=O)NC2CCC2NC(C2CC(CF)C2)=O)CCCCC1(F)F 17624,C1(NC(CC2(C)CC2)=O)CC2COCC(C1)C2NC(c1cnn(CCO)c1)=O 17625,C(=O)(C1=CC2CCC=CCCC12)N(C1(CNC(C=CC(C)(C)C)=O)CCCC1)CC 17626,C(c1ccccc1F)=CCC(=O)NCC(CC)(C)NC(c1cnc(O)n1C)=O 17627,CC(C(=O)N1CC(O)CC1CC(N1CC(C(=O)N(C)C)C1)=O)S(C)(=O)=O 17628,C1(NC(CC(=O)NCC#C)=O)CC2CCC(C1)N2C(C12CCC(F)(CC1)CC2)=O 17629,c1(C(N2CCN(C(CC3CC(=C)C3)=O)C(C3CC3)C2)=O)c(C)[nH]c2ccccc12 17630,C(c1ccc(C(F)(F)F)cc1)=CC(=O)NC1(C)CCN(C(c2ccsn2)=O)C1 17631,C12(NC(c3ncn(C(C)(C)C)c3)=O)CC1CN(C(=O)Cc1csc(C(F)F)n1)C2 17632,c1(CC(=O)NC(C2(O)CN(C(C(C)OCCOCC)=O)C2)C)ccc(C)c(Cl)c1 17633,C12(NC(C3CCC(=C)CC3)=O)CCC1CN(C(c1csc(CC(F)F)n1)=O)C2 17634,CC1=C(C(=O)N(C2CCN(C(=O)CCCc3cc(C)no3)C2)CCO)CCO1 17635,C(=O)(C(C)(C)S(C)(=O)=O)NCC1N(C(c2c(C)cc(O)nc2)=O)C2CCC1C2 17636,C(c1ccc(O)cc1)=CC(=O)Nc1ccc(-c2cccnc2)cc1.C(F)(F)F 17637,CC1(C)CN(C(=O)C2=C(C#N)CCC2)CCC1C(=O)NCC1CN2CCC1CC2 17638,C1(CC)CN(C(C2(F)CCCCC2)=O)CCN1C(c1cnc(OC)c(Br)c1)=O 17639,C1(O)(C(C)NC(c2c(C)scn2)=O)CCN(C(c2ccnc(F)c2)=O)C1 17640,Cc1noc(C)c1C(C)C(N1CC(C(F)(F)F)(C(N)=O)C1)=O 17641,C(=O)(CCCC(C)(C)C#N)N1CC(NC(Cc2ccn(C(C)C)n2)=O)C(C)C1 17642,c1(C(C)OC)nc(C)c(C(N2CCCC(CCNC(C3CN(C(C)C)C3)=O)C2)=O)s1 17643,c1(C(=O)NCC)ccc(N)c(C)c1Cl.C1CC(=O)N2CC(C2)CC(C)N1CC 17644,c1(C(N2C#CCCCCC2)C(=O)NC2CC(C(=O)OC)C2)ccc2nc(C)oc2c1 17645,c1(OC)c[nH]nc1C(=O)NC(C(=O)NCCN1CCCC1C)C1(C)CC1 17646,Cc1cn(C)cc1C(=O)NCC1CC(CNC(=O)CN(C)C(=O)C2CC2)CO1 17647,C1(NC(COC(CC)CC)=O)CN(C(C2CC23CC(OC)C3)=O)CC1F 17648,CC(C)(C)CC(=O)NCC(=O)NC1CCC(CNC(=O)Nc2ccc(F)cc2)C1 17649,N1(C(C2C(C)(Br)C2)=O)CC2(CCC2)CC1CNC(=O)CCn1ccnc1 17650,c1(CC)c[nH]nc1C(=O)NCC1C(NC(=O)CC2(CC(=O)OC)CC2)CCC1 17651,CC(C(C)(C)NC(C1CSCCS1)=O)NC(=O)COc1ccon1 17652,Cc1nc(N2CC(CNC(C3(N(C)C)CCCOC3)=O)CC2C)c2cnn(C)c2n1 17653,Cc1nc(C2CCOC2C(N2CC(O)(CNC(=O)OC(C)(C)C)C2)=O)n[nH]1 17654,N1(C(c2[nH]nc(OC)c2Cl)=O)CCC2CN(C(C3(CF)CCOCC3)=O)CC12 17655,c1(COC)cc(=NC(=O)CC2CC(NC(=O)Cc3ccc(Br)nc3)C2)[nH][nH]1 17656,C1(C)(C(=O)NCC(CN(C(CC)=O)C)(C)C)Cc2ccccc2C(=O)O1 17657,N(C1COc2ccccc21)C(C1N(Cc2cc(OCC)c(O)c(Br)c2)CCC1)=O 17658,N1(C(C2CCN(C)C2)=O)CC2C(CNC(C3CC(c4ccc(F)cc4)O3)=O)C2C1 17659,C1(OCC(C(C)C)O)C2CN(CC(O)C(C)Nc3ccccc3)CC12 17660,C1(CC(=O)NCc2cc(C)ns2)CN(C(=O)CCc2cncs2)CCO1 17661,C(=O)(C(C)(C)C(=O)N(C)CC1CCCN1C(=O)CCc1csc(C)n1)NC 17662,C(=O)(C(F)(CNC(=O)C1=CCN(C)C1)C(C)C)N(C)Cc1cccc(C)n1 17663,N1(C(C2CC(=O)NCC2)=O)CC(NC(=O)CCc2cnco2)C(F)(F)C1 17664,CCCC(C)(C)C(=O)NC1CC=CCC1C(=O)NCC(=O)N1CCCO1 17665,c1(C(N2CCC(CNC(CN3CC(=O)NC3=O)=O)C2)=O)cc2c(s1)COCC2 17666,C(=O)(C1=C(Cl)CCCC1)NC1C(N2CCN(C(C(C(C)C)C)=O)CC2)COC1 17667,CC(CC1CCCCC1)CN=c1[nH]c2c(c(=NCc3ccncn3)[nH]1)SCC2 17668,C12(C(N(C3CCN(C(=O)C=C4CCC4)CC3)C)=O)CCCC1CC(=O)CC2 17669,C1(C(=O)NC2(CC(=O)OC)CC2)C2CCC(C2)C1CNC(=O)CCNC(C)=O 17670,N1(C(c2cc(C(C)C)n[nH]2)=O)CCN(C(=O)C(C)c2ccco2)CC(C)(C)C1 17671,CC1CC(C)C1C(=O)NCCCNC(=O)C(C)(C)F 17672,Cc1ccc(C(=O)NCCCCCN(C)C(c2coc(Cl)n2)=O)c2ncccc12 17673,N12CCCC(O)(C1)CNC(=O)C1(CC1)C2.c1(C(N(C)C)=O)cnsn1.CC 17674,N1(C(C2C(C(=O)OC)C2)=O)CC(CNC(C2CCCC2)=O)C2(CC2)C1 17675,CC1CN(C(C2CCCC(CF)C2)=O)C(C)CN1C(=O)CC1CSCCO1 17676,C1(NC(c2c(C(C)C)con2)=O)CC2CC(C1)N(C(=O)CC1CSCCO1)C2 17677,C(CCCCCC(=O)NCC1CCCC1O)NC(C1CN(C2CCC2)C1)=O 17678,CCCCC(C)C(=O)N1CC(C(C)(C)NC(=O)CCOCC(F)F)C(O)C1 17679,Cc1c[nH]c(C#N)nc1=NCCN(C)C(C1COc2ccc(F)cc2C1)=O 17680,C1(C(N2CCN(CCC#C)CC2)=O)CCN(C(C2CS(=O)C2)=O)C12CC2 17681,c1(OCC(F)(F)F)ccc(Cl)cc1-c1nnc(Cc2cc(F)ccc2Br)o1 17682,N#CC1CN(C(=O)CN2CCOC2=O)CCN1C(c1ccc(S)cc1)=O 17683,c1(C(=O)NCC(=O)N(CCCCCC)C(c2ccco2)C)ccc(OC)cc1C 17684,CC(C)C(O)CC(=O)N(C1CCN(C(C23CSCC2C3)=O)CC1)C 17685,C1(CNC(c2nc[nH]c3ncnc2-3)=O)CN(C(=O)C(F)(F)C2CC2)CC12CCC2 17686,c1(C(c2n(CC)nnn2)NC(C2CCC2)C2CC2)ccc(OC)cc1[N+](=O)[O-] 17687,C1(NC(C=C(C)C(C)C)=O)CCCCC1CNC(c1ccno1)=O 17688,C1(CC(=O)NC(CNC(=O)Cc2ccon2)C2CCC2)NC(=O)NC1=O 17689,n1(CC)nnc2c1CCC(C(=O)NCC1CCN(C(C3COC(=O)N3)=O)CC1)C2 17690,c1(C(=O)NC2(CCNC(C3C(C(=O)OC)C3)=O)CC2)cccc2c1NC(=O)CO2 17691,C(=O)(C(CC=C)CC(C)C)N(CC)CC1CN(C(=O)C=C2CN3CCC2CC3)C1 17692,c1(C(N2C(C(=O)NCC(C)CO)C=CC2)=O)cc(F)ccc1O 17693,C1(NC(CC(C=C)C)=O)CN(C(c2cccc(CS(N)(=O)=O)c2)=O)CC12CC2 17694,n1(CCOC)cc(-c2ccc(C(=O)NCc3cc(C#N)cs3)nc2C)ccc1=O 17695,c1(C(N2CCC(NC(C3(SC)CC3)=O)C(O)C2)=O)ccc(P(C)(C)=O)cn1 17696,c1(C(=O)NCCOCCC(=O)NCC2(SCC)CC2)ccc(C)cc1C 17697,C(=O)(CCS(=O)(=O)NCC1CC(F)CN1c1ncc(C2CC2C(C)O)cn1)NC 17698,O(NC(=O)C(C)(C)C1CCCN(C(=O)CN2C(=O)CNC2=O)C1)Cc1ccn(C)n1 17699,C1(NC(C(CC)(F)F)=O)CC(CNC(C2(CC3CC3)CC2)=O)C12CCC2 17700,c1(OC)cnc(C(N2CCCC2CCNC(=O)C=C(C)C(C)C)=O)nc1 17701,N1(C(c2cn(CCC)nn2)C(=O)NC2CCCC2)C2CCC1CN(C)CC2 17702,C1(C(=O)Nc2ccc(Br)nc2)COCCN1C(c1ccc(-c2ccccc2)s1)=O 17703,CCCCC(C)(F)C(=O)N1CC(NC(C23CC(C)(C2)OC3(C)C)=O)C(O)C1 17704,C(=O)(C(CNC(=O)C1=CC2(CCOC2)C1)CC(C)C)NC(c1ccccn1)C 17705,c1(C(COC(=O)C(O)CO)O)ccnc2ccccc12.n1(C(C)C)cc(CN)cn1 17706,C12(NC(c3c(NC(N)=O)c(F)ccc3)=O)CCCCC1CN(C(=O)C1=CCCS1)C2 17707,N1(C(C2C(C(=O)NCC#C)C2)=O)CC2(C1)CN(C(=O)C(N1C(=O)CCC1=O)C)C2 17708,N1(C(CSC)=O)Cc2ccccc2CC1CNC(c1cc(Cl)ccc1NC(C)C)=O 17709,NC(=O)CCCC(=O)N1CCC(NC(c2ccnc(OCCO)c2)=O)C(F)C1 17710,CC1(C)OC2CCN(C(c3ncoc3-c3cccs3)=O)CCC2O1 17711,CCC(C)CCCCC(=O)NC(C)CNC(c1ccc(S(C)=O)cc1)=O 17712,CN1CCN(c2ccc(C(N3CC(NS(=O)(=O)CC4CC4)C(O)C3)=O)cc2)CC1 17713,c1(C(N2CC(O)CC(NC(CCc3n[nH]c(=N)s3)=O)C2)=O)[nH]nc([N+](=O)[O-])c1Cl 17714,c1(C(N2C(CN(C(=O)CC3NC(=O)NC3=O)C)CCC2)=O)ccc(CO)cc1F 17715,N1(C(c2c(C)c[nH]n2)=O)CCCC(NC(=O)Cc2ccsc2Cl)C1C 17716,c1(C(N2CC(CO)(COC)C2)=O)cc([N+](=O)[O-])c[nH]1.C1CC(C)C(=O)N1.CC 17717,CN1CCC(C(=O)NC2CCC3(CC3)C2)(NC(C2C=CCCC2)=O)C1 17718,C1(C(N(CCCC#C)CCOC)=O)CCN(C(C2CC(C)CCO2)=O)C1(C)C 17719,C1(CNC(=O)C2CC2)CCN(Cc2c(F)cccc2F)CC1(F)F 17720,C1(C2CC2)(CNC(c2c(CCC)n[nH]c2)=O)CCN(C(=O)CC(C)(C)O)C1 17721,C(=O)(CCCC(=O)NCC)NC1(CC=C)CCN(C(C2CNC(=O)C2)=O)C1 17722,C1(F)(CNC(c2cccc(CCC)c2)=O)CCN(C(=O)C(F)=CC2CC2)CC1 17723,c1(CNC(c2c(C)ocn2)=O)cccc(NC(=O)CC2CC2(Cl)Cl)c1 17724,c1(NC(CN2CCCC(C)C2)=O)ccc2nn[nH]c2c1 17725,C(=O)(CCCNC(C)=O)N(C1CCN(C(=O)CC(=O)N2CCOCC2)C1)CCC 17726,C1(F)(NC(=O)CC2CS(=O)(=O)C2)CC2CCC(C1)N2C(=O)CNS(=O)(=O)C1CC1 17727,Cn1cnc(C(=O)NCC23CC(C(=O)NCc4ccnn4C)(C2)C3)c1 17728,c1(C(=O)NC2C(CNC(C(COC)(F)F)=O)CCCC2)cnc2c(n1)CCCC2 17729,c1(NC)cccnc1C(=O)NCCCC1CCCN1C(=O)C1=CCCC1.C1C(=O)N1 17730,C1(C)(CCC(=O)NC2CC(CCNC(c3c(Cl)cc(C)s3)=O)C2)NC(=O)NC1=O 17731,S(=O)(=O)(c1cnc(C(C)(C)C)[nH]1)N(C1C(CO)C1)C 17732,NS(=O)(=O)c1ccsc1C(N1CCC(CO)C(NC(c2cn[nH]c2)=O)C1)=O 17733,c1(CC(N2CCC(C(C)C(=O)NC3CC(F)C3)CC2)=O)ccc2c(c1)CCCO2 17734,c1(C(N2CCC(N3CCN(C(CCOC)=O)CC3)C2)=O)c(C)cc(O)nc1C 17735,N1(C(C(C2CCC2)OCC)=O)CCC=C(C(=O)N2CCC(C)(O)C2)C1 17736,Cc1ccc(C(=O)NC2(CCNC(C34CC(CN(C)C)(C3)C4)=O)CCC2)o1 17737,c1(OC)ccc(CC(N2CC(OCCNC(=O)CCc3cn(C)cn3)C2)=O)cc1 17738,C1(C(=O)NCc2cn(CCCOC3CCCCC3)nn2)(CCO)CCCS1(=O)=O 17739,c1(C(N2CC(COC)N(C(C3CCC(C)(C)O3)=O)CC2)=O)ccc2cc[nH]c2n1 17740,C1(NC(c2nc(-c3cn(C)nc3)oc2)=O)CCCCN(CC2CC(F)C(=O)N2)C1 17741,N1(C(CCCOC(C(C)C)=O)=O)CCCC(C(=O)Nc2cccc(O)c2)C1 17742,c1(CC(=O)NC2CN(c3ncnc(C)c3Br)C(C)C2)oc2ccccc2c1C 17743,C1(C(=O)NC(C2CCCCC2)C)CCCC1CNC(C1CS(=O)(=O)C1)=O 17744,C1(C)(C(=O)NC2(CC=C)CN(C(=O)CC(C)(O)c3cccs3)C2)CCCCNC1=O 17745,CC(C#N)C(=O)NCC(C)CC1CN(C(=O)N(CCO)Cc2ccccc2)C1 17746,C1(CC#C)(C(=O)N(CCCO)CCC)CCN(C(=O)CN(C)C2CC2)C1 17747,C#CCCCC(C)C(=O)NCc1ccc(C(N2CCCC(C)(C)C2C)=O)cn1 17748,N1(C(C(CC)(C)C)=O)CCN(C(C2CCCC23CCC3)=O)C(C)C1 17749,c1(C(=O)NC2(C)CC(NC(C3N(C(C)=O)CC(O)C3)=O)C2)cc(O)cc(C#N)c1 17750,Cn1cnc(C=CC(=O)NCC(=O)NC2CC(O)C(F)C2)c1 17751,n1(CC(=O)N(C2C3CN(C(CCCOCC)=O)CC32)C)cc2ncccc2n1 17752,c1(C(=O)NCC2(C(C)NC(=O)CC3CC3(Cl)Cl)CC2)c[nH]cc(F)c1=O 17753,c1(CCN(C)CC2(O)CCCNC2)nc2ccccc2n1C 17754,Clc1ccc(C(c2nnnn2CC2CC2)NC23CC(C2)C3)cc1Cl 17755,c1(CNC(C2CC(C)(C)C2)=O)cccc(NC(=O)CC2C=CCC2)c1 17756,C1(C)(CC(=O)NCC(n2ccnc2)C)CCN1C(=O)COC1CCCCC1 17757,C1(C(=O)NC2CN(C(=O)OC)C2)CN(C(c2cc(C)co2)=O)Cc2nccn2C1 17758,C1(c2cn(C(COCC)C)nn2)CN(C(=O)Cc2csc(C)c2C)CC1C 17759,c1(C(=O)NCCC(C)N(C(CCCOC)=O)C)cc(F)ccc1C 17760,N1(C(c2ccc(N(CCC)C)cc2)=O)CCN(C(C2CC(CF)C2)=O)C(CC)C1 17761,c1(C(C)=O)cc(C(C)(C)C)c(NCc2cc(Br)cn2C)s1 17762,C(=O)(C(C)n1cccn1)N(CC(=O)NC(C)(C)C)CC=C.C1CCOC(=O)N1 17763,C1(CCNC(c2[nH]cc(C)c2C)=O)CCN(C(=O)C(C)n2cncn2)CC1(F)F 17764,N1(C(C(CC=C)c2ccccc2)=O)CCC(F)(Cc2ncccc2C)CC1 17765,C(c1cccs1)=CC(=O)N(CC(CC)NC(=O)CC1CCOC1)C 17766,c1(C(=O)NCC(CC)NC(=O)Cc2ccccc2Cl)cc(C)c(C#N)c(C)c1 17767,C=CCC(C(=O)NC(C=C)CO)NC(=O)C=CC1CCCN1C 17768,C1(CNC(CSCC=C)=O)CN(C(C2COCOC2)=O)CCC1C 17769,CN1CC(C(N2CCC(c3ccc(Cl)cc3Cl)CC2)=O)C2(CC2)C1 17770,C=C(C)C(C)(C)C(=O)NCCN(C)C(C1CCC(C#N)C1)=O 17771,CC1CC(NC(=O)Nc2nccc(-n3cccn3)n2)CCN1C 17772,c1(C(C)=O)c(C)[nH]c(C(=O)NC(C2CCCN2C(=O)C(C)N=[N+]=[N-])C)c1C 17773,N1(C(COCCCCC)=O)CCC(CC)C1CNC(=O)Cn1cnc(C#N)n1 17774,C1(C(=O)NCC2(CNC(Cc3ncn(C)c3)=O)CC2)Cc2nccn2C1 17775,c1(OC)ccc(NC(=O)C(C)(CNC(=O)CSc2nc[nH]n2)CC)cc1O 17776,C1(NC(c2c(CC)c[nH]n2)=O)CN(C(=O)CC2CCCC2(F)F)C2CCCCC12 17777,c1(C(C(=O)NCC(=C)C)NC(=O)CCNc2ccccn2)ccc(Cl)cc1 17778,C(=O)(C1CCc2c[nH]nc21)C1(C2CCCN2C(c2cccc(O)n2)=O)CC1 17779,C1(C(=O)NCC2CCN2C(=O)C(F)(F)CC2CCCO2)CCC([N+](=O)[O-])CC1 17780,CCC(CCOC)NC(=O)C(CC1CCC1)NC(=O)CSCCOC 17781,Cc1nc(O)ccc1C(=O)NCCOc1ccc(C#N)cc1 17782,c1(CN(C(CNC(C(C)=C(C)C)=O)C2CC2)C(=O)CC2CSC2)ccccn1 17783,C1(C(=O)NCC(CN(C(c2c(OC)c(Cl)sc2)=O)C)C)OCCOC12CCC2 17784,N1(C(C2C(c3n(CC)ccn3)C2)=O)C2CCCC1CN(C(C1CCCSC1)=O)C2 17785,CC1C(NC(c2ccc(N(C)C)s2)=O)CCN1C(=O)CC(F)(F)F 17786,N1(C(CC(CC)OC)=O)CCC(C2(O)CN(C(C3(CC)CCC(=O)N3)=O)C2)CC1 17787,N1(C(c2c(Br)ccc(Cl)c2Cl)=O)CCC2C(CCN2C(c2cc(C3CC3)no2)=O)C1 17788,CCC(C)CC(=O)C(=O)N1CCOC(C(=O)NCC2(C)CSC2)C1 17789,N1(C(CC2(COC)CC2)=O)CCCCC(NC(c2cc(C)nn2CCO)=O)C1 17790,Cc1csc(C(=O)NCC(C2CCCC2)NC(=O)C(F)F)c1Cl 17791,c1(C(=O)NCC(CC=C)NC(c2csc(=N)[nH]2)=O)nn(C)c(Cl)c1Cl 17792,C1(NC(COC(CC)(C)C)=O)C=CCN(C(=O)C(CC)OC2COC2)C1 17793,C1(C)(CCNC(CC(C)OC)=O)CCN(C(c2ccc(SC)s2)=O)C1 17794,C1(NC(c2ccc(Cl)nc2Cl)=O)CCN(c2ncncc2I)CC1F 17795,O=C1NC2CCC1CN(S(=O)(=O)c1ccc(N3CCCC(C(F)F)C3)nc1)C2 17796,C1(O)(CC(=O)NCC(CC=C)NC(=O)CCc2cccnc2F)CCCCCC1 17797,N1(C(c2cccc(NC)c2)=O)CCC(CNC(=O)C(C2CC2)SC)C(C)(C)C1 17798,C1(COC)(NN(C)C)CN(C(=O)COc2cccnc2)C1.C1C(=O)N1.C(C)(C)C 17799,c1(C(N2CCCC(c3ncc[nH]3)C2)=O)cccc(-n2cnnn2)c1 17800,c1(C(=O)NC2C(N(C(=O)C(O)Cn3cncn3)C)CC2)cnc2[nH]ncc2c1 17801,c1(C(=O)NC2CN(C(C(CSC)(C)C)=O)CC23CC3)ccn2ccnc2n1 17802,c1(NC(CCC=C)(C)c2nnnn2Cc2ccco2)ccc2[nH]c(CO)nc2c1 17803,C#Cc1ccc(F)cc1C(N1CCC(CNC(c2cn(C(F)F)c(C)n2)=O)C1)=O 17804,N1(C(CC)=O)CCCC(C(=O)NC(CNC(c2ocnc2C(F)F)=O)C2CC2)C1 17805,N(C1CC2(CC2)Oc2c(F)cccc21)C(C1CC(F)C(=O)N1)=O 17806,C12(CNC(C3(C=C)CCC3)=O)CC1CN(C(=O)CCc1cc(C)on1)C2 17807,c1(CNC(CSCCC)=O)cccc(C(=O)Nc2ccc(C(N)=O)nc2)c1 17808,Cc1cc(C)c(C(N2CCC(N(C)C(c3cn(C(C)(C)C)nc3C)=O)C2)=O)cn1 17809,CCCCCC(=O)NC1CC1.N12CCC(CC1)N(C(C1CC1Cl)=O)CC2=O 17810,N1(c2ccnc(C(C)C)n2)CCCC(C(N2CCC(C)(O)CC2)=O)CC1 17811,C1(NC(C2(CC(C)C)CCC2)=O)CN(C(c2sc(CO)nc2C)=O)CC1C.CC 17812,CC#CCCCC(=O)NCC1CCC(NC(=O)Cc2noc(C)c2C#N)CC1 17813,N1(C(C2C(C(C)C)C2)=O)CCC(C)(CCNC(c2cc(Cl)n(C)n2)=O)C1 17814,C1(NC(C=CCOC)=O)CCC(C)(C)CC1CNC(c1cnc(C(C)(C)C)[nH]1)=O 17815,C1(CC(=O)NC)CN(C(C2CC(N(C)C)C2)=O)CCN1C(=O)C(C)C#N 17816,N1(C(CSC)=O)CC2(C1)SCCC2NC(=O)CC1CC(O)C12CCC2 17817,C1(CC)CCCN(C(=O)Cn2ccnc2)C1C(=O)NC1COCC(C)(C)C1 17818,C12(CNC(c3cc(C)oc3C)=O)CC(C(=O)O)(C1)C1(COC1)O2 17819,c1(NC(c2[nH]c(=NCc3ccc(C)cn3)sc2)=O)ncc([N+](=O)[O-])cc1I 17820,c1(C(=O)NC(C(C)NC(C2CCOCC2(C)C)=O)CO)cc2cc(Cl)cnc2[nH]1 17821,c1(Cn2cc(COC)nn2)cc2cc(C)cc(C)c2[nH]1 17822,CC1CN(C(=O)C=Cc2cn(C)cn2)CCN1C(c1ccc(C(C)(C)C)cc1)=O 17823,c1(C(=O)NCCC(CNC(C2N(C)CC(O)CC2)=O)O)cc2ccncc2o1 17824,Cc1ccc(NCC2(C(=O)Nc3ccc(-c4ccc(C)nc4)cc3)CC2)c(O)c1 17825,c1(CN2C(C(=O)NC(C3CCC(C)(CC)O3)=O)CC2)cc(C)nc2onc(C)c12 17826,c1(C(=O)NC2C(C(N3C(COC)C=CC3)=O)COCC2)ncnc(O)c1F 17827,C1(C(=O)NCC2CC(NC(C(Cn3ccc(C)n3)C)=O)C2)CCC(=O)NC1 17828,C1(CC(=O)NCC2C(NC(COCC(C)C)=O)C2)CC(OC(C)(C)C)C1 17829,c1(C(N2C(CC#C)CCC2)=O)ccc(OCC)cc1.C1(=O)C(=O)NCC(C)N1C 17830,c1(C(=O)NC2C3CN(C(c4cncc(C#C)c4)=O)C2C3)[nH]cc2c1CCCC2 17831,c1(C(N(C)CCC2CCCCN2C(=O)CC2CCNC2=O)=O)cc2sccc2[nH]1 17832,N1(C(C(=O)NC(c2ccc(F)cc2)C)C2COC2)CCC(C)(O)C(O)C1 17833,C1(C)(C(N(CCCCCCNC(=O)C(F)(F)CO)C)=O)CC2CCC1C2 17834,CCCC(C(=O)N1CC(N(C)CCO)C1)OC.N12CC3C(C3C1)C(=O)NCCC2=O 17835,CC(CNC(=O)CCCC#N)CC(=O)NC1(CCF)CCC1 17836,N1(C(C=C(CCC)CCC)=O)CCN(C(C2CC2CCOC)=O)CC1CCCC 17837,c1(OC)nc(Cl)ccc1C(=O)NC1(CO)CCN(C(c2cc(N)cnc2Cl)=O)C1 17838,c1(NC(CC)C2CCC2)[nH]c(=NCc2cc(N)ccc2Cl)nc2c1ncn2C(C)C 17839,C1(O)(C(C(=O)NCC=CC=C)N(C2CCCC2)CC)CCCCC1 17840,C#CCC(C(=O)NC(c1cccc(Cl)c1)CNC(=O)CSc1nncn1C)C1CC1 17841,c1(NCC(C)(C)NC(C(C(C)C)OC)=O)cc2nnc(-c3ccccc3)n2cn1 17842,C(=O)(C1Cc2c(Cl)cccc21)N1CC(C(C)NC(c2ccc([N+](=O)[O-])n2C)=O)C1 17843,c1(NC(C=CC2N(C(CN3CC(C)(OC)C3)=O)CCC2)=O)ccc(Cl)nc1C 17844,N1(C(C(CC)N(C)C)=O)CC(CC(=O)NCc2cc(=O)cc[nH]2)C2(CC2)C1 17845,N1(C(c2n(C(C)C)ncc2)=O)CCOC(C)(CNC(c2nn(C)nc2Br)=O)C1 17846,C1(CNC(=O)NC(C)COC(F)(F)F)Cc2ccc(F)cc2C1 17847,C12(C(N3CCC4(NC(C(=Cc5ccco5)C)=O)C(C3)C4)=O)CCC(F)(CC1)CC2 17848,Cc1ccc(-n2nnc(C(=O)NC3CCCC(CO)C3)c2C)cc1 17849,N1(CCC(=O)NCC2(NC(=O)COCCF)CCC2)C(=O)C2CCCCC2C1=O 17850,C1(C(N2CCC(C)C2)=O)C2C3CCC(C3)C12.C1(N2CCOCC2)(C(=O)NC)CCCC1 17851,Cc1ccc(Cl)c(C(=O)NCC2CCCCN2C(=O)Cc2cc(C)ccc2C)c1 17852,c1(CC)ccc(C(=O)NCC2C3CCC(C3)N2C(C2CC23CCOC3)=O)c(F)c1 17853,c1(C(N2CCC(NC(c3c(CC)c[nH]n3)=O)(CF)C2)=O)cc2ccccc2o1 17854,c1(C(N(CCCCCC)C2CCN(C(=O)CC(CC)OC)C2)=O)c[nH]c(=NCC)s1 17855,N1(C(C(CC)SC)=O)C(C(N2CCC(C(=O)OC)C2(C)C)=O)CCC12CC2 17856,Cc1ccncc1-c1cn(CC(N2CCCC(COC3CCOCC3)C2)=O)nn1 17857,Cn1c(CNS(=O)(=O)CC2(C)CCCCC2)cc2c1CCOC2 17858,N1(C(CC(=C)C)=O)CC2CC(CNC(=O)Cc3ccoc3)C(C2)C1 17859,N1(C(CCOCCOC)=O)CC(C)(NC(c2cc(Cl)n[nH]2)=O)C1 17860,c1(C(=O)NCCCCCNC(c2cncc(N)n2)=O)ccc(S(N)(=O)=O)cc1Cl 17861,c1(CC)cc(C(=O)NCCNC(=O)COCc2cccc(C)c2)nn1C 17862,C1(C(=O)NC(c2cnc(C)s2)C)CCC(C)(C)N(C(=O)CC2=CCCCC2)C1 17863,c1(C(=O)NC(C(=O)N(CCC#C)C)C2CC2)ncnn1CC 17864,N1(C(C=Cc2nc(C)sc2)=O)CCCCC1C1CCCN1C(=O)C(O)C1CCC1 17865,n1(C(C)C)cc(C(=O)NC(C)CN(C)C(C2CCCSC2)=O)c(Br)n1 17866,C(=O)(C(C)(C)C(=O)NCCC(O)C(=O)N1CCCCC1C)OC 17867,c1(C(=O)NCC(C)NC(c2n(C(C)C)ccc2)=O)cc(Cl)ccc1F 17868,C1(O)(C(C)NC(=O)CSC(C)(C)C)CCN(C(C2CCCN(C(N)=O)C2)=O)CC1 17869,c1(C(=O)NCCCNC(c2cn(C3CCC3O)nn2)=O)cc2ccsc2s1 17870,C1(C#N)(CC)CC2CCC1CC2NCc1cnnn1-c1ccccc1 17871,C1(NC(CN(C(COC)=O)C)=O)CC2CC1CN(C(=O)CCn1ccnc1C)C2 17872,CC(C(=O)NCCC1(NC(C2CCNC(=O)C2)=O)CC1)C(F)(F)C(F)F 17873,c1(C(=O)NCC(CO)NC(c2cnc(O)c(F)c2)=O)cc2cn[nH]c2cn1 17874,C1(NC(C2N(CC#C)CCC2)=O)CC2(CCCN(C(=O)C(F)C(C)(C)O)C2)C1 17875,C=C1CC(C(=O)NCCCCC2CC2C)(CNC(c2c[nH]cc2C)=O)C1 17876,c1(C(C(=O)N(C2CCN(C(C3CCOCC3)=O)C2)CC#C)(F)F)ccc(Cl)cc1 17877,CNS(=O)(=O)NCC(=O)NCC1(OC)CN(C(=O)Cc2cn(C)nn2)C1 17878,C1(C(N(C)C)=O)CCCN(c2nnc(C(O)CC(C)(C)C)n2Cc2ccco2)C1 17879,N1(C(CC2CN(C(C)=O)C2)=O)CC(O)CC1(C)C(=O)N(CCCC(C)(F)F)C 17880,Cn1cccc(Cc2ccc(C(F)(F)F)c(F)c2)c1=O.N12CCC(C1)C2=O 17881,C1(O)(CC(=O)NCC2(CO)CCCO2)CCN(C(C2CCCC(O)CC2)=O)CC1 17882,n1(CC(=O)Nc2nc(C3CCCC3)cs2)cc(Br)c(O)nc1=O 17883,C=CC1(CC(N2CC(O)CC2CNC(c2csnc2C)=O)=O)CCOCC1 17884,c1(-c2n(-c3n(C)nnc3)nc(N3CCOCC3)n2)ccc(C(F)(F)F)cc1Cl 17885,C(=O)(C(CNC(c1cc(F)c[nH]1)=O)CC1CCCC1)NC(C1CCC1)C 17886,N(C(=NCCCN1CCc2ccccc21)N1CCC(C)C2(CCC2)C1)C(CC)C 17887,c1(C(C(C)C)=O)ccc(C(=O)N(CCCc2cn(Cc3nc[nH]n3)nn2)CCO)o1 17888,C=CC(C)(C)CC(=O)NC(C1CCN(C(=O)C(Cc2cccc(Cl)c2)=NO)C1)C 17889,Cc1ccn(C)c1C(=O)NCC=CCNC(=O)CCc1ccnn1C 17890,C(=O)(C1=CCC2CCC1N2C(=O)C(F)C1CCCC1)NC(C)Cc1ccco1 17891,c1(CC)ccc(N)c(C(=O)NCC(C2CC2)N(C)C(C2(CF)CCCOC2)=O)c1 17892,c1(OC)cc(CC(=O)NCCCC(C)NC(c2cocn2)=O)cc(Cl)c1 17893,C1(NC(CCCC#C)=O)CCCC12CN(C(c1cccnc1OCCOC)=O)C2 17894,C1(NC(CCOCC#C)=O)CC2(C1)CC2NC(c1cnn(CCOC)c1)=O 17895,C1(CC(=O)NC2(C(=O)NC3C(C(=O)OCC)CC3)CC2)CCCC1C 17896,c1(C(=O)NCC2C(NC(CC(C=C)C)=O)CCCC2)ccc(C(F)(F)F)c(N)c1 17897,C1(C)(CNC(CCN(C(C)=O)C)=O)CCN(C(c2coc(C(F)(F)F)c2)=O)CC1 17898,c1(-c2scc(C)n2)ccc(C(=O)N(C2CN(C(C3(C)CCCN3C)=O)C2)C)cc1 17899,c1(CCC(=O)NC2(CNC(CCC(CC)C)=O)CCOC2)cnc2ccccn12 17900,N1(C(c2nc(COC)sc2)=O)CCC(C2CC(NC(=O)CC3CCCCC3)C2)C1 17901,c1(C(=O)NCC(c2ccc(C)cc2)NC(C2(C3CC3)CC2)=O)cnc2n1CCS2 17902,CC1CN(C(c2cn(C(C)(C)C)cn2)=O)CC1(C)CNC(=O)CCC1CC1(Cl)Cl 17903,C(=O)(CCCC(F)(F)CO)NC1C(SC)CN(C(c2c[nH]nc2[N+](=O)[O-])=O)C1 17904,N1(C(c2n(C(CC)C)ncc2)=O)CCC(F)C(NC(c2cc(=O)c(C)c[nH]2)=O)C1 17905,N1(C(C2C(C)CCO2)=O)CCC(F)(C(N2CC(C3CCCO3)C2)=O)C1 17906,N1(C(C(C)c2ccco2)=O)CCC(O)C(N(C)C(c2cc3n(n2)CCO3)=O)C1 17907,CC1CC(C(=O)N(C(C)CNC(=O)C=Cc2ccc(=O)oc2)C)CC(=O)N1 17908,N1(C(CC2CC(=C)C2)=O)CC(NC(c2cncc(C3CCCCC3)c2)=O)C(C)C1 17909,C1(C(C)NC(=O)Cc2cnc[nH]2)CCCCN1C(c1ccc(C2CCC2)cc1)=O 17910,c1(OCCC(=O)N(C2CCC2(C)C)CCOC)ccccc1F 17911,CC1(C)C(CNC(c2nc(Cl)sc2Cl)=O)CCN1C(=O)CC1CCC(O)C1 17912,C1(NC(CCCOCCC)=O)CCCN(C(=O)CC2(N3CCCC3)CC2)C1C 17913,C1(CC)CC(C(=O)NCC(C)(C)O)CCN1C(=O)C(C)CC#N 17914,c1(CCN(C)CC2(F)CCN(C(=O)OC(C)(C)C)C2)ccc(Cl)c([N+](=O)[O-])c1 17915,N1(C(CC2CC(CC)C2)=O)CC(C)N(C(=O)CN2CSCCSC2)CC1C 17916,c1(CC(=O)OC)ccc(C(=O)NC(CN(C(=O)CO)C)C)c(C)c1 17917,C(=O)(C1(C)CCn2c(C)nnc21)N1CC(NC(c2nc(CC)oc2)=O)CC1(C)C 17918,c1(C(=O)NC2CCCC3CN(C(C(C)OC)=O)CC32)cccc(S(N)(=O)=O)c1C 17919,N1(C(C2(C(C)C)CC2)=O)CC(NC(c2sncc2Br)=O)C2(CCC2)C1 17920,c1(NC(=O)NC(C)(C)CC2CCOC2)c(F)cccc1Cl 17921,Cc1cccc(CC(N2CC3CC3(NC(=O)CC3CC4C=CC3CC4)C2)=O)c1F 17922,C1(NC(c2ccc(N(C)C)cn2)=O)CC2CCC1C(NC(=O)C1=CCCOC1)C2 17923,C1(C(N2C(C(N(C3CCCC3(C)C)C)=O)COCC2)=O)CC(=O)NC(=O)C1 17924,c1(C(N2C(CN(C(C(C)N(C)C)=O)C3CC3)CCC2)=O)c[nH]c2cc(C#N)ccc12 17925,N1(C(C(Cc2ccccc2)OC)=O)CCC2(C1)CN(C(=O)C(O)C(C)C)C2 17926,N1(C(c2cc(SC)c(C)o2)=O)CC(C)N(C(c2cn(C)c(C)cc2=O)=O)CC1C 17927,CCC1=NOC(C(=O)NCCCN(C(c2cnc(CC(C)(C)C)s2)=O)C(C)C)C1 17928,c1(C(=O)NCC(C)N(C)C(C2CCCCCN2C)=O)cccc(C#N)n1 17929,C(=O)(CC1c2ccccc2CCN1S(C)(=O)=O)NCC1N(C(CC=C)=O)CC1 17930,N1(C(C2CCC(CC)CC2)=O)C(CNC(c2cncc(Cl)c2)=O)CC2COCC12 17931,N1(C(C2(N(C)C)CCN(C(C3CC4(CCC4)C3)=O)C2)=O)CC2(CCCC2)C1 17932,C1(CCNC(c2cccc(F)c2Cl)=O)CCN(C(=O)CO)CC1(F)F 17933,N1(C(C(CC#C)CC#C)=O)CCC2(CC1)CN(C(=O)CC1CC3(CC3)CO1)C2 17934,N1(C(CC2ON=C(C)C2)=O)CCOC2CC12.C1(Cn2ccnn2)C(=O)N1 17935,c1(C(=O)NCCOC)cccc(C(=O)Nc2cc(C(F)F)ncn2)c1 17936,CCCC(CCC)CC(=O)NCC1CN(C(c2cnn(CC)c2C)=O)CCC1C 17937,n1(CC(=O)NC2CC23CC(NC(C2(C(F)(F)F)CC2)=O)C3)cnc([N+](=O)[O-])n1 17938,N1(C(C=NOC)=O)CC(CNC(=O)Cc2cccc(F)c2F)CC2(CCC2)C1 17939,CC1CCCn2cc(C(=O)NC(C)(C)C(C)NC(C3CN(S(N)(=O)=O)C3)=O)nc21 17940,CCC(O)(C(=O)NCCCCC(C)NC(c1nc(C)cs1)=O)c1ccccc1 17941,N#CC1C2CCC1CN(C(C13CC(CCO1)N(C(=O)C=CC1CCOC1)C3)=O)C2 17942,CN1CC(NC(C2CC23CC(NC(C2CCOCC2)=O)C3)=O)C(C)(C)C1 17943,C1(C(=O)NCCN(C(=O)CC(C)(C)C)CC)CC12CCOCC2.C12CCCN(C1)C2 17944,Cc1cc(Cl)cc(NC(=O)CC2COCCN2Cc2ccc(C)c(C)c2)c1O 17945,N1(C(C(C)SCC2CCCO2)=O)CCCN(C(=O)C(C2CCCCC2)F)CC1 17946,c1(C(=O)NC(CCNC(Cn2ccc(C)n2)=O)C)c(C)nc(O)nc1S 17947,n1(CC(=O)NCC(=O)NC(C)(C)CNC(N2CCCC2)=O)cc(NC(N)=O)nn1 17948,c1(CC(=O)NCC2N(C(C3(C#N)CC3)=O)CC2)cc(F)ccc1Cl 17949,C(=O)(CCCCC(=O)NCC1CC(CNC(C23CCC(C)C2C3)=O)C1)NCC 17950,N1(S(CC)(=O)=O)CCN(C(c2c(C)noc2C)=O)C(=O)C1C 17951,N1(C(CC(C=C)CC)=O)CC2(C(=O)N(C)Cc3cncnc3)CC1CCO2 17952,c1(CC(=O)NCCC2(O)CN(C(c3c(C)coc3C)=O)C2)cccc(Cl)c1Cl 17953,C1(CCNC(C(C)SC)=O)CSCCN1C(c1ccccc1C(N)=O)=O 17954,C1(NC(C2CC=CCC2C(F)(F)F)=O)CCCN(C(=O)CCc2cncs2)C1 17955,c1(C(N2CCC(CNC(C3CC(CC)OCC3)=O)CC2)=O)cc2nc[nH]c2cn1 17956,C(c1ccc(C)c(C)c1)=CC(=O)NC(CCOC)CNC(=O)C(O)CC1CC1 17957,c1(C(=O)NCC(C)N(C(C(CCC)CC)=O)C)ccc2c(c1)CN(C)CC2 17958,C=CCC(C(=O)NCC1(CN(C)C(C2CCC3CC3CC2)=O)CC1)C(C)C 17959,C(=O)(C(C)(C)CCCNC(C1CCO1)=O)NCCC(C(C)C)CO 17960,Cc1cc(Cl)cc(-c2nc(C3CC4CCCCN4C3)no2)c1O 17961,C(C(CC(C)C)C(=O)NCC(C(C)C)NC(c1occ2c1CCCC2)=O)OC 17962,C1(NC(c2cccc(CC)c2)=O)CCCCN(C(=O)C(CO)NC(=O)C=COC)C1 17963,C=C(Cl)CC(C(=O)N1CCC1CO)NC(c1nnn(C)c1C)=O 17964,C(=O)(C(C)(C)C(=O)NC1CCCN(C(c2cc(Cl)sc2Cl)=O)CC1)NC 17965,C1(NC(c2c(CCC)onc2C)=O)CN(C(C2(C)COC2)=O)CC12CC2 17966,C(=O)(C1=CSCCO1)N(CCN(C(C=C(CC)c1cccs1)=O)C)C(C)C 17967,N1(C(CN(c2ccncc2)C)=O)CCC2CC1CN2C(c1csc(Cl)c1)=O 17968,CC1CC(C)N(C(c2c(Br)ccnc2F)=O)CCN1C(=O)CC1CC1 17969,N1(C(C2=CCCC2C)=O)CCC2CC(n3cc(C4(CCO)CC4)nn3)CCC2C1 17970,C1(CCC(=O)N(CCOC)CCOC)CCN(C(=O)CN2C(=O)CNC2=O)CC1 17971,C1(NC(CCC#CC)=O)CCSC12CN(C(=O)CCOc1cccc(C)c1)C2 17972,C(N=c1[nH]c2ccc(F)cc2o1)C1CCCN(C(CC(CC(C)C)C)=O)C1 17973,CC1(C)CC(NC(=O)CCN(C(=O)CCc2cnn[nH]2)C2CC2)C1 17974,C1(C(=O)NCC(C2CC2)NC(c2cn(C)nn2)=O)C2CCC(F)C12 17975,N1(CC(=O)NC2CN(C(C(C(C)C)F)=O)CC2C)CCc2ccccc21 17976,C12(NC(c3n(C)ccc3)=O)CN(C(C3CC(F)C3)=O)CC1CS(=O)(=O)C2 17977,C1(NC(C(C2CN(C(C3(CC)CCCO3)=O)C2)O)=O)CCCCCC1C 17978,Cn1ncc(C(=O)NCC(C)(C)OCCNC(=O)CSCc2csc(=N)[nH]2)n1 17979,CCCCCCCC(=O)NCC(C)(O)CNC(C1CNC(=O)CC1(C)C)=O 17980,c1(C(N2CCCC(CCCCNC(C(C)N=[N+]=[N-])=O)C2)=O)ccc(O)c(F)c1 17981,c1(C(=O)NCC2C(C)CCCN2C(C2(N(C)C)CCCC2)=O)cccc2ccnn12 17982,Cc1oc2ccccc2c1CC(N1CC(NC(C2CCCCN2C)=O)C(C)C1)=O 17983,C1(NC(Cc2c(C)nccn2)=O)CN(C(=O)CCC=CBr)CCC1CO 17984,c1(CCC(=O)NCC2C(NC(C(C)OC(C(C)C)=O)=O)C2)ccc(Br)nc1 17985,C1(C(=O)Nc2cccc(C(F)(F)F)n2)CC(O)CCN1C(c1cccc(Cl)c1Cl)=O 17986,Cc1ccc(C(=O)NCC2CN(C(C3CN(C)CC(C)O3)=O)CC2C)nc1F 17987,CC1CN(C(=O)C(C)(C)C2CC2)CC2(CCN(C(c3cc(O)nc(O)c3)=O)C2)O1 17988,C(=O)(CC(C)C(F)F)N1CCC(C(C)(CC(=O)OC)NC(c2c(C)cncc2)=O)C1 17989,Cc1ccc(Cc2nc(-c3cccs3)nn2CCN2CCCC2)c(C)c1 17990,C1(NC(CC(=C)I)=O)CC(C)CN(C(c2ccc(C)nc2)=O)C1 17991,c1(-c2cn(C3CCN(C(C(=O)O)C4CCCC4)C3)nn2)ccc(Cl)c(Cl)c1.O=CC 17992,CC(C)(C)CCC(F)C(=O)NC1CC(NC(c2cn3cnnc3cn2)=O)C1(C)C 17993,C1(NC(C(c2ccccc2)OC)=O)CCCCC1CNC(c1ncsc1C)=O 17994,C1(CC(=O)NCC2(C)CN(C(c3ccoc3)=O)CCO2)COC2(CCC2)CO1 17995,CCC(C)(CO)C(=O)NC(C)CCCNC(=O)CCN1CCCCC1=O 17996,C1(C)(CC(=O)N(CCN(C(CN(CCC)C)=O)C)CCOC)CC1(F)F 17997,C1(CNC(NCC(CC)CC(F)(F)F)=NCCF)CCC2(CCCC2)CC1 17998,C1(O)(CCNC(CN(CCC)C(C2CCC(C)C2)=O)=O)CCCC1 17999,Cc1cc(C)c(CCN2CCC(=CC(=O)NC(=O)NC(C)(C)C)CC2)c(C)c1 18000,C1(CNC(C2(CC#C)CC=CCC2)=O)N(C(=O)Cc2cnsc2)CCC1(C)C 18001,C1(N(c2nc(=N)cc[nH]2)C(CC2C(C)(C)C2)=O)CCCN(C(C2CCCC2)=O)C1 18002,c1(C(=O)NC2CC3(C(NC(CCc4n(C)cnc4)=O)C3)C2)cc2cn[nH]c2cn1 18003,c1(C(C)=O)csc(C(=O)NCC2(O)CN(C(C3CC3(C)C)=O)C2)c1 18004,N1(C(CCC(C)OC)=O)CC(C(=O)NCCNC(=O)C(C)C)C2CCCC12 18005,N1(C(C(=O)NC(C)C)=O)CC(NC(=O)Cc2ccccc2Cl)CC12CCC2 18006,C1(NC(C(C)C2CC2)=O)CC(F)(F)CC1NC(c1ccc(CN(C)C)o1)=O 18007,C(=O)(C(C)CC(=O)OC)N1CCC(CCOC)(NC(C(C)SCCCC)=O)C1 18008,c1(C(=O)NCC2CCCC2NC(C2(CF)COC2)=O)cc(Cl)cnn1 18009,C1(NC(C(C)=CC2CC2)=O)CN(C(C2CCN(CC(C)C)C2)=O)CC1C 18010,S(=O)(=O)(c1ccc(F)cc1)N(c1ccccc1)CCC(=O)OCC 18011,c1(NC(C2CC(=C)CN2C(c2cc(O)nc(Cl)c2)=O)=O)cc(C)cnc1C 18012,c1(C(=O)Nc2cccc(NC(CC(C=C)(C)O)=O)c2)cc2cccnc2o1 18013,C1(NC(=O)Cc2cnnc(O)c2)CC2CC1N(C(=O)COCCN1CCCC1)C2 18014,c1(NCC23CC(NC(c4ncc(C(C)C)cn4)=O)(C2)C3)cccc(Br)c1Cl 18015,C(=O)(C(C)(C)CNC(=O)CC1CC=CCC1)N(C)CC1CCN(C)C1 18016,C(=O)(CC(C(F)F)NC(C1CC(F)C1)=O)N(CCCCC)C 18017,C(=O)(C1=CCCCO1)N1CC(NC(Cc2c(C)oc(-c3cccs3)n2)=O)C(F)C1 18018,CC1(C)CC(CNC(=O)NC2CC2c2cccs2)C1 18019,C1(C(=O)NCCCC(C)NC(CCN(C(CCC)C)C)=O)CN(C(C)C)CCO1 18020,Cc1nc2c(Cl)cccc2cc1C(=O)NCCN(C)C(C1CNC(=O)N1)=O 18021,c1(C(N2CC(O)(CCNC(c3c(CC)ocn3)=O)C2)=O)c(C)cc(Cl)nc1N 18022,C1(NC(c2cnc(OCC)s2)=O)CCCCC1NC(c1cnn(C)c1SC)=O 18023,C1(NC(C2CCCC2)=O)CCOC12CCN(C(C1COC3COCC13)=O)CC2 18024,C1(CN(C(C2N(CC)CCC2)=O)C)CCCN(C(=O)CCC(C)(C)N(C)C)CC1 18025,N1(C(C2CC(=O)NC2)=O)CCOCC(F)(CNC(C2CC2c2ccsc2)=O)C1 18026,c1(C(=O)NC(C(C)NC(CCN(C(CCC)C)C)=O)C)cc(C)nc(O)n1 18027,c1(OCC)ccc(CCNC(=O)NCc2ccc(CN(C)C)cc2)cn1 18028,N1(C(CC(CNC(C(C(COC)C)C)=O)(C)C)=O)CCC2(CCOCC2)C1 18029,CCCCCCCCC(=O)NC(c1cccnc1)CNC(C1CC1C)=O 18030,N12CC(CC1c1ncc[nH]1)C(=O)NCC2.N1(CC)CCCC1CCO 18031,C(=O)(C1CCC(=O)c2ccccc21)N1CC(C2CCCN(C(C(C)(F)F)=O)C2)C1 18032,N12CCCCCC(C1)CNC(=O)C2=O.C1(C(=O)CC)CC12CC2.C1CO1 18033,N(C(=NCCCP(C)(C)=O)NCC(C)SC)CCc1cc(OC)cc(OC)c1 18034,C1(CNC(C2CCC(OC)CC2)=O)C2CCCC1N(C(C1CCOC(C)C1)=O)C2 18035,CN1CCC(C2(NC(=O)CC3(C#N)CCOCC3)CC2)CC1 18036,CC1CCC(C(=O)NCC(C)N(C)C(c2ccc(C(F)(F)F)cn2)=O)C(=O)N1 18037,N1(C(CC(CC2CC2)NC(C2CN(C)C(=O)C2)=O)=O)CCN(C)C2(CCC2)C1 18038,c1(C(=O)NC2(CO)CN(C(C3OCC(C)C3)=O)C2)ccc(C#N)c(O)c1 18039,CCC(C(C)CN(C)C)NC(=O)C(Cn1cncn1)NC(=O)CCCn1cccn1 18040,c1(N(C(=O)CC2CCN(c3ncncc3I)C2)C)ccc(Cl)c(F)c1 18041,C(=O)(C(O)P(C)(C)=O)N1CCCC(NC(CS(N2CCC(C)CC2)(=O)=O)=O)C1 18042,c1(OC)c(C(=O)NC(C)(CNC(c2nccn2C)=O)C(C)C)cc(F)cc1F 18043,CC1(C)CC(NC(=O)CN)CN1C(c1c(Br)cccc1Br)=O 18044,C1(CCN(C(CC)C(=O)NC)C(c2ccccc2)=O)CCCN(Cc2ccccc2)C1 18045,N1(C(c2cc(C(C)(C)C)n[nH]2)=O)CCCC(C)(CNC(C2(C)CCCCO2)=O)C1 18046,c1(C=O)cccc(Cl)c1C.c1(C(=O)OO)csc(C2CCCN2N(CCCC)CC)n1 18047,c1(C(=O)OC)ccc(C(=O)NC2CCN(c3ncnc(N(C)C)c3F)C2)cc1C 18048,N1(C(C23CCC(C2)C3)=O)CC2(C(=O)NC(c3nc(C)sc3)(C)C)CC1CO2 18049,O=C(C1=Cc2cc(Cl)ccc2OC1)NCC1C2CCC(C2)N1C(=O)Cc1cc[nH]n1 18050,CC(C)C(C(=O)NCC1(C)CN(C(=O)COC2CC=CC2)C(C)(C)C1)C(C)C 18051,C1(N(CC(=O)NCCOCCNC(C(C)CF)=O)C)CCS(=O)(=O)C1 18052,C(=O)(C(C)CC(F)F)NCCN(C(C1C(C=C)OCC1)=O)C 18053,C1(C(N(CCCNC(c2ccc(C3CC3)s2)=O)CC)=O)C2CCC(=O)C12 18054,N1(C(c2c(C)cco2)=O)CCC2(CCCN(C(c3scc(Cl)c3Cl)=O)C2)C1 18055,C(C(C)(O)C(C)CC)NC(C1(CC#C)CCN(C(=O)C(C)c2cccs2)C1)=O 18056,Cc1ncsc1C(=O)NCC(O)CNC(=O)C(C1CC1)Sc1ccccc1 18057,C1(C(C)N)CCN(C(=O)C(=O)N(CC2CCOCC2)Cc2ccccc2)C1 18058,c1(C(N(CCC(C)NC(CC2CC(=C)C2)=O)C)=O)nnn(C(C)C)c1N 18059,c1(C(=O)NC(CC(C)NC(CNC(=O)NC)=O)C)cc(C(C)C)ccc1F 18060,CN1C2CC(O)C(C2)C1C(N1CCCC(N2C(=O)NC(C)(C)C2=O)C1)=O 18061,N1(C(COCC(=C)C)=O)CC=CCC1C(=O)NC1CC(C)OC1=O 18062,C(=O)(CC(O)C(C)CC)NC1(CC=C)CCN(C(=O)CC2OCCO2)CC1 18063,C1(=O)CC(c2ccc(Cl)cc2)CO1.C(=O)(C(C(C)C)NC(C)=O)N(C)CC 18064,n1(C(C)C)nncc1C(=O)N(CC(N1CCC(N(C)C2CC2)C1)=O)C 18065,c1(NC)c(C(=O)NC2CC(CNC(=O)CN(C)C(C)C)C2)sc2nccnc12 18066,C1(S(C)(=O)=O)(C(=O)NCCNC(c2c(CC)cc(Br)cc2)=O)CCCC1 18067,OCCC#CCN=c1nc(N2CCCC(c3nc[nH]c3Br)C2)cc[nH]1 18068,N(C(=NCCC)NCCC(C)CC)CCc1cccc(OCCN(CC#C)C)c1 18069,c1(C(C(F)(F)F)NC(=O)Cn2cnc(Br)n2)ccc(NS(C)(=O)=O)nc1 18070,c1(COC)nc(C(N2C(C(N3CC(CO)(CO)C3)=O)CC2C)=O)co1.C(=O)OC 18071,N1(C(c2c(COC)cco2)=O)CC2CC1CN2C(c1cc(C(C)C)on1)=O 18072,CC1CN(C(=O)CC2CC(O)CN2C(=O)CCCn2cncn2)CCS1 18073,Cc1nc(Cl)ccc1CNC(C1CCN(S(=O)(=O)C2CC2)C1)=O.c12cn(nn1)C2 18074,c1(C(=O)NCC(CN(C(C2CN(C)C(=O)N2)=O)CC)(C)C)cc2[nH]ccc2s1 18075,C1(CNC(c2c(C)coc2C)=O)CC(C)(C)CCC1NC(=O)CC1CCOCC1 18076,c1(C(=O)NC2(CO)CCCN(Cc3ccncc3Br)C2)cccc([N+](=O)[O-])c1O 18077,C1(NC(C(C(C)C)OC)=O)CCN(C(C2CCCCC2C)=O)CC1F 18078,C1(NC(c2ccc(CC)[nH]2)=O)CCCC(CNC(c2cn(C3CC3)nn2)=O)C1 18079,N1(C(C2(CC)CCOC2)=O)CC=C(C(=O)NCC(C)(C)OCCO)C1 18080,C(C(C)(C)CN(C(c1ccc(C(F)(F)F)o1)=O)CC)NC(CCSCCC)=O 18081,C1(C(=O)NC2C(NC(c3cn(CCCOC)nc3C)=O)C2)CC(C(C)C)=NO1 18082,c1(NC(c2ccnc(OC(F)F)c2)=O)cc(F)c2c(c1)OCCO2 18083,O=S(=O)(c1[nH]c(=NCC(O)c2ccncc2)ccc1Br)NC1CCCC1C1CC1 18084,N1(C(C(C(C)C)(C)C)=O)CC2CCOCC2(NC(c2ccc(Cl)c(N)c2)=O)C1 18085,C(=O)(CCCC(C)(C)C)N(C1CCN(CC2CCCCO2)CC1)CCC 18086,C1(C(C)Sc2ccc(OCCCOC)cc2)CCCC(C)(C)C1 18087,c1(C(=O)NCC(CCC)NC(c2cnc(C3CCCO3)s2)=O)cncc(Cl)c1 18088,C1(OC)CCC(C)(C(N2CCC(NC(c3ccn(C4CC4)n3)=O)C2)=O)CC1 18089,N1(C(c2nccc(C(F)F)n2)=O)CCCCC2(CCN(C(C3CC3(Cl)Cl)=O)C2)C1 18090,c1(C(=O)NC2(CNC(C(=O)N(C)C)=O)CC3CCC2C3)nnn2c1CCCC2 18091,CCC(C)(CCC(C)C)C(=O)N1CC(NC(=O)CCc2cnn(C)n2)C2(CC2)C1 18092,c1(C(N(C2CCCN(C(=O)CC(=O)OC(C)=O)C2)CC)=O)ccccc1C 18093,C1(CNC(CCOC(C)=O)=O)CCC2(CCC2)C1NC(=O)C(CO)C(C)(C)C 18094,N1(C(CCCN(C(C(N2CCNC2=O)C)=O)C)=O)CCCC2CCCC12 18095,CC1(C)CC(C(=O)NC2CN(C(c3cnc(-c4cccnc4)s3)=O)C2)=NO1 18096,c1(CNC(CCCC#C)=O)c(C)nc(NC(=O)OC(C)(C)C)nc1O 18097,c1(OC)ccc(C(N2CC(CCNC(C3CCC(O)CC3)=O)C2)=O)c(N)c1F 18098,N1(C(c2cc(CC)ncn2)=O)CCCC(C)C1CCNC(=O)CN1CC2CC2C1 18099,O=C1NOC2C(C2)C(=O)NC(=O)N2CC(O)(C1F)C2.c1(N)ccccc1 18100,CCCC(CC)CCC(=O)NCCC1(O)CCN(C(c2cc(F)cc(Cl)c2)=O)C1 18101,CN1CC2CCC(C1)N2C(C1CC2(CC(NC(C3CC4(CSC4)C3)=O)C2)C1)=O 18102,C1(NCc2ccc(C)cc2)CCCN(Cc2ccc(C#N)s2)C1C 18103,c1(C(=O)OC)ccnc(S(=O)(=O)NNc2cc(Br)nc3c2CCCCC3)c1 18104,Cc1cc(C(=O)NC(c2cnccn2)C)nnc1C 18105,C1(c2ccccc2)(CNC(C(C)=C2CCCC2)=O)CCN(C(=O)CO)CC1 18106,C(=O)(C1=CC2CC=CCC12)N(CCCN(C)C(c1c(O)cc(Cl)cc1Cl)=O)C 18107,N1(C(c2c(OC)nccc2)=O)CCN(C(=O)C(C)c2cc[nH]n2)CC12CC2 18108,C1(C(N2C(CCCNC(C(C)Oc3ccccc3)=O)CCC2)=O)CCCCC1O 18109,N1(C(C(CC)(C)C)=O)CC(C(N2CC(c3nnc(C)n3C)C2)=O)CCC(O)C1 18110,CCC(CCCC(=O)NOCCC(C)O)NC(=O)CC1CC2(CC2)CO1 18111,Cc1csc2ncc(C(=O)NCC3CCCN(C(C4CNC(=O)C4)=O)C3)c(=O)n12 18112,C1(N(C(C)=O)C)CCCCC12CCCN(C(=O)C1CC1)C2 18113,c1(CC(N2CC3(CN(Cc4cncc(C)n4)C3)C2)=O)c[nH]c2ccc(F)cc12 18114,C(CC(=O)NC1(C)CCCC1(C)C)(C(C)OC)NC(CC=CCCCCC)=O 18115,c1(CC)oc(C)cc1C(=O)OCc1ccnn1C(C)(C)C 18116,N1(C(C(C)OCC2CC2)=O)CCC2(CC1)CC2CNC(=O)CC(C)CF 18117,CC1C(C(=O)N(C(C)(C)CC(=O)NC(c2cccnc2)C)C)CCN1C 18118,N1(C(CCN2C(C)CCCC2)=O)CCC(NC(C2CCC(=O)NC2)=O)C(C)(C)C1 18119,N#Cc1cc(N2CCCC2CNC(c2cccc3c2ncn3C)=O)ccc1[N+](=O)[O-] 18120,C=C(C)CCC(=O)N(CCCOCCNC(=O)CCCOC1CCCCC1)C 18121,c1(C(N2C(C)CN(C(C3CCC4CC4C3)=O)CC2)=O)cc2ncccc2[nH]1 18122,C1(C(=O)NCC(C)(C)NC(Cc2c(C)noc2)=O)CCS(=O)(=O)C1 18123,C1(C)(COC)CCC(CNC(C2(NC(c3cnc(Cl)n3C)=O)CCCC2)=O)O1 18124,N(C(=NCCCCF)N1CCC(NC(=O)NC2CC2)C1)C(C)C 18125,N1(C(CCSC)=O)CC2(CCC(NC(C34CCCCC3C4(F)F)=O)CC2)C1 18126,C1(OC)(CNC(=O)CN2CC3CC3C2)CCN(C(C2CC(=O)N(C)C2)=O)CC1 18127,c1(CC(N2CCC(CNC(=O)COC(F)F)C2)=O)cc(F)ccc1C(F)(F)F 18128,N1(C(CCN(C(=O)CN=[N+]=[N-])C)=O)CCC(C)(N(C)C)C1 18129,C(=O)(NNC(=O)C(C)(C)CCCCNC(=O)Cc1cccnc1)c1c(C)ccs1 18130,n1(CCNC(C(C)c2ccco2)=O)cc(C(=O)NCC(C)OC(F)F)cn1 18131,CC1(C)C(C)(C)C1(F)CNC(=O)CNc1cnc(Cl)c(Cl)c1 18132,C1(NC)CCN(C(c2ccnc(Cl)c2F)=O)CC12CC2 18133,N1(c2ccnc(C)n2)CCC(F)(F)C(C(=O)NC2CCCCC2C(F)(F)F)C1 18134,c1(OC)ccccc1C(=O)NC1CC(C)N(C(=O)C(C)C2CCCO2)C1 18135,C1(C(=O)NC(CC(=O)OCC)Cc2ccccc2)CCCC1S(C)(=O)=O 18136,c1(OCCCNC(=O)NCCNS(CC)(=O)=O)ccc(O)nc1.C1CN1 18137,c1(N(C(C2COCCO2)=O)CC)ncc(Br)c(C)c1[N+](=O)[O-] 18138,N1(C(C(=O)NCc2c(Cl)cccc2Cl)=O)CCC2(CC(=O)NC2=O)C1 18139,c1(C(=O)NC2C=CCN(C(C(C)Oc3cccc(O)c3)=O)C2)c(Cl)cccc1Cl 18140,N1(C(c2c(OC)c(Cl)ccc2)=O)CCN(C(c2cc[nH]n2)=O)C2CCCCC2C1 18141,C1(C(=O)NCC2C(CNC(Cc3c(C)ncs3)=O)C2)CC2CC(=O)C1C2 18142,C1(C(N(CC)CC2CCCN2C(=O)CC#N)=O)Cc2cccc(F)c2O1 18143,N1(C(c2ncn(CC)c2)=O)CCC(C(=O)NCC2(N(C)C)CC2)=C(F)C1 18144,C1(CC)CCN(C(=O)CC2CN(C(c3cc(C)[nH]n3)=O)C2)C1CNC(C)=O 18145,c1(C(=O)NCC(CC)NC(C2(C)C=CCC2)=O)ccc(OC(F)(F)F)cc1Br 18146,C(=O)(CC(C)C(=O)NCCOCC1CC1)OCC.C(C=O)OCC 18147,Cc1cc(Br)cnc1C(c1nnnn1C1COC1)NCCC1CCC(C)(C)C1 18148,CCC(C(O)C(F)(F)F)NC(C)C(=O)OCc1ccccc1 18149,S(=O)(=O)(CC(=O)NC1COCC1CNC(=O)CSCC1CCCC1)NCC 18150,Cc1ncc(C=CC(=O)NCC2CCN(C(C3(O)CCOC3)=O)C2)c(O)n1 18151,c1(C(N2C(CNC(CSc3nc(C)[nH]n3)=O)CCC2)=O)nc(O)c(C)s1 18152,N1(C(C2N(C)CSC2)=O)CCCC(N(C(=O)CN(C)C(=O)C2CC2)C)C1 18153,c1(C(=O)NC2C(OC)CN(C(CS(=O)(=O)NC)=O)C2)ncc(C)nc1OC 18154,Cc1cccc2c(C(N3CC(C)(C)OCC3CNC(=O)CC(C)O)=O)nccc12 18155,C=CC1(C(=O)NCC2CCCC3CC23)CCN(C(=O)CCc2cncnc2)CC1 18156,C=CCC(CO)NC(=O)COCCNC(C1CC12CC2)=O 18157,C1(CC(=O)NC(C)Cc2cccnc2)CC(C)N(C(=O)CCC2CC2(F)F)C1 18158,C(CC(C(=O)NCC1(COC)CCC1)NC(=O)CC1C=CCCC1)OC 18159,c1(C(N)=O)cccc(NCC(N2CC=CC(NC(c3ccc[n+]([O-])c3)=O)C2)=O)c1 18160,c1(OCC)cc(C(N2CCC(CNC(=O)C3=CCC(C)CC3)C2)=O)cc(Cl)c1O 18161,C1(N(C(c2cc(C)c(O)nc2)=O)C)CC2CCC(C1)N2C(C1(C)CCOC1C)=O 18162,CCCCCC(CC)C(=O)N1CCC(CNC(=O)CCc2ccoc2)(COC)CC1 18163,N1(C(CCC(=C)Cl)=O)CC2CN(C(c3c(C4CC4)noc3C)=O)CCC2(CO)C1 18164,C(=O)(CC(C(C)OC)NC(c1ccc(O)cn1)=O)NCC(C=C)(C)O 18165,c1(CN2CC3C(C(=O)NCCc4ccc(F)cn4)C3C2)cccc(O)c1F 18166,C1(C(=O)NC(C2N(C(c3c(C)cc(C)s3)=O)CCC2)C)CCC(=O)CC1(C)C 18167,N1(C(C2C(C)OCC2)=O)CCC(NC(=O)CSc2cnn(C)c2)C12CCC2 18168,c1(C(=O)NC2C(C(=O)NC(C)CCO)C2)cc2c(cc1O)OCCO2 18169,c1(OCC)ncc(C(=O)NC2CC(CNC(c3ncn(C)n3)=O)CC2O)cn1 18170,Cc1cc(C(N2CC3C(CNC(c4ccc[n+]([O-])c4)=O)C3C2)=O)cc(C)c1N 18171,C(=O)(C(C)P(C)(C)=O)N(CCOC)CCNC(=O)Cc1c[nH]ccc1=O 18172,CC1(C)CC(CC(=O)NC2CN(c3ncco3)C2)N(C(c2cnsn2)=O)C1 18173,C(CCC(C)(C)C(=O)O)N(CC(C1CCSC1)=O)C 18174,C(=O)(CCC(F)(F)C(F)F)OCC1C2N(C(=O)OC(C)(C)C)CC(CC2)C1 18175,Cc1ncc(C(N2CCC23CN(C(c2cn4ccnc4s2)=O)C3)=O)c(C)n1 18176,C1(NC(=O)NCC(=O)N(C2(CNC(=O)C(C)(C)C)CCC2)C)CCCCC1F 18177,N1(C(C(F)OC)=O)CCOC2CCN(C(C3(C)CCS(=O)(=O)CC3)=O)CC12 18178,c1(C(=O)NCCN(C(CC(C)OC)=O)CCCN(C)C)csc(C)c1C 18179,c1(C(=O)NCCCN(C(C(c2c(C)noc2C)OC)=O)C)cc(F)cc(Cl)c1N 18180,c1(C(CC)=O)cc(C(N2CCC(CCNC(C3CC4CC3C4)=O)C2)=O)ccc1F 18181,c1(OCC=C(C)C)ccccc1NC(C1CCCC(NC(=O)N(C)C)C1)=O 18182,C1(O)(CCNC(c2ccc(C(F)F)nc2)=O)CCCN(C(c2cncs2)=O)C1 18183,C1(CC(=O)NC(CC)CN(C(C2(CC(F)(F)F)CC2)=O)CC)CCN(C)CC1 18184,C1(NC(=O)CCN2CCOCC2=O)COC2(CCN(C(=O)COCC3CC3)C2)C1 18185,Cc1ccc(C(=O)NC2CC3CN(C(C4CC4(C)C)=O)CC23)c(C2CC2)n1 18186,C(=O)(CCCCCC#N)N1C(C(N2CCC3C(C(N)=O)C3C2)=O)CC(C)(C)C1 18187,c1(C(=O)NC(C2CCN(C(c3c(C)cnc(F)c3)=O)C2)C)cc(C)c(C)cc1Cl 18188,c1(C(N2C(CCNC(C3CCC(=C)CC3)=O)CCC2)=O)ccc2nc(S)oc2c1 18189,N1(C(C(C)SC)=O)CCN(C(c2ccccc2Oc2cccnc2)=O)C(CF)C1 18190,c1(C(=O)NC(C(C)NC(C2(C(C)C)COC2)=O)C)cccc(P(C)(C)=O)c1 18191,C1(C(=O)NC(CC=C)CO)CN(Cc2ccccc2C(=O)O)CCS1 18192,c1(C(=O)NCCSCC(=O)NCC2C(C)(C(F)F)C2)cc2ccncc2s1 18193,N1(C(CCNc2cn(C)nc2)=O)CCN(C(c2cnn(C)c2)=O)CC12CCC2 18194,N1(C(C2(CC)CC2(F)F)=O)CCC(C2(NC(C3CCCCCC3)=O)CC2)C1 18195,c1(CNC2CCC2)ccc2c(c1)C(=O)NCCO2.O=Cc1cc2cc(c1)N2 18196,N1(C(C(c2ccc(N(C)C)cc2)NC(CC(=C)C)=O)=O)CC2(CC2)CC1C 18197,C1(C(N2C(C(=O)OCC)CCC2)=O)CN(Cc2csc(Cl)n2)CCO1 18198,N12CC(CC1=O)C(=O)NC1CC2C1.c1(C(CC)CC)nnnn1CC(=O)NC 18199,c1(C(=O)NC(C2CCN(C(=O)C(CC)(CC)OC)CC2)CC)cncc(F)c1C 18200,C1(C(=O)NCc2c(OC)csc2)COCCN1C(C1(CN2CCOCC2)CC1)=O 18201,N1(C(CC(C)(C)NC(C2CN(C(C)=O)C2)=O)=O)CCCC(C)(C#N)C1 18202,S(=O)(=O)(c1cccc(Br)c1[N+](=O)[O-])N(C(C#C)C(C)C)CC 18203,c1(OC)cc(NC(=O)CCCC(C)NC(=O)C(C)NC(C)=O)cc(F)c1 18204,CCC(O)C(C)(C)C(=O)N(CCC(=O)NC(CC(=O)OC)C1CC1)OC 18205,C1(CC)CNC(C)CN1C(=O)Nc1ccccc1OCC(F)F 18206,N1(C(C2C(C)OC(=O)N2)=O)CC2CN(C(c3cnc(O)o3)=O)CC2(C(F)(F)F)C1 18207,c1(CC(=O)NC(C2C(C(=O)OCC)C2)C)ccnn1C1CCC1 18208,CCC(C)(C)C(O)C(=O)N(CC(C)O)CCNC(=O)Cc1ccoc1C 18209,c1(CC)nocc1C(=O)NC1CCN(C(c2nnnn2C)C)C1 18210,C(=O)(C(CCCC)NC(=O)C=CCN(C)C)N(C)Cc1cccnc1 18211,C1(O)(CN2C3CCN(C3)C(=O)C2=O)CCNCC1.Cc1nccs1 18212,C1(NC(c2c[nH]c(=N)s2)=O)CCC(NC(=O)CC2CC23CC3)CC1 18213,Cc1nn(C)c(Cl)c1C=CC(N1CCCC(OC(=O)C(C)(C)CF)C1)=O 18214,N1(C(C(C2(C)CC2)NC(=O)C2=C(C)CC2)=O)CC2(C1)NC(=O)NC2=O 18215,c1(OC)cccc(C2CC2C(=O)NCC2CCCN2C(C2CC(Cl)(Cl)C2)=O)c1 18216,C1(C(N(CCCN(C(=O)CCCC2CCCCC2)C)C)=O)CCCC(N(C)C)C1 18217,CC(CC(F)F)C(=O)NC1CN(C(c2ccsc2)=O)CC12CC2 18218,c1(C(C(=O)NCC(CNC(CCc2onc(CC)n2)=O)O)OC)ccccc1F 18219,c1(C(=O)NC(CC2CN(C(C3(COC)CCC3)=O)C2)C)ccc2nc(C)sc2c1 18220,C1(CC(=O)NCCCCNC(C2CC(CC(=O)OC)C2)=O)CCCC(=O)N1 18221,C1(NC(c2cccnn2)=O)CCC2CN(C(c3nccnc3Br)=O)CC2C1 18222,c1(NC(c2ccc(CCNC(C(C=C)(C)C)=O)cc2)=O)ccc2nnsc2c1 18223,CC(C)CC(C)CC(=O)NC1CCCC1NC(c1cscc1-c1ccccc1)=O 18224,N#Cc1cc(F)ccc1-c1cccc(C2CCN2C(=O)CC2CC2)c1.C=O 18225,CC1C(C)N(C)CCN1C(=O)CC1COCCN1C(c1c[nH]nc1Cl)=O 18226,Cc1c(C(N2CC(=O)CC2C(=O)NC(CC2CC2)C2CC2)=O)nnn1C 18227,N1(C(C2N(C)C(=O)NC2)=O)CCC(C2CC2)C1Cn1cc(CCO)nn1 18228,C(=O)(CC(O)CC(C)(C)C)N1CC(C(C)NC(c2nc(-c3nc[nH]n3)sc2C)=O)C1 18229,N1(C(C(CCSCC)NC(C)=O)=O)CCC(O)C(NC(=O)Nc2nnc(C)o2)C1 18230,c1(CC)csc(CNC(C)(COC)c2nnnn2C(C)(C)CC)c1 18231,Cc1nc(NCC2CCC(C)(C)OC2)cc(=NCC2CSCCS2)[nH]1 18232,c1(OC)nc(C)ccc1C(=O)NC1CCCN(C(=O)C(C)C2CCCC2)C1C(C)C 18233,C(CCC(C)(C)C(=O)NCC(C(=O)OC)OC)NC(c1ncc(CC)cn1)=O 18234,c1(C(N(C2CCCN(C(=O)Cc3cnns3)C2)C)=O)cnc2c(c1)NCC2 18235,C(C1CN(C(C2CC=CC2)=O)CC1C(=O)NC1CC(C)C1(C)C)=CC 18236,N1(C(CC)CC)CC(C(=O)NCCCN(C(c2cccs2)=O)CC)CC1=O 18237,N1(C(C2CC(C)C2)=O)CC(C)(C)OCC1CNC(C1(C(F)F)CCCC1)=O 18238,C(=O)(C1CCc2cccnc21)NCC(C)(C)NC(C(N1C(=O)CCC1=O)C)=O 18239,CC1CN(C(=O)C(C)(C)COCC(F)F)CC1NC(=O)CCC1CC1(Cl)Cl 18240,CC(CO)C(C)N=c1cc(NCCSc2ccccn2)nc(-c2cccnc2)[nH]1 18241,C1(N(C(CSS(C)(=O)=O)=O)CC2CCCC2)CCCN1C(=O)CC1CC=CC1 18242,C(=O)(CC(COC)COC)N1C(C(=O)NC(CCC)C(N)=O)CSC1 18243,c1(C(CNC(C2CCCSC2)=O)NC(C(C)(C)OC(C)=O)=O)cc(F)cc(Cl)c1 18244,C(=O)(C#CC1CCCC1)NN(CCCCCn1ncc(C)c1)CCC1CC1 18245,CC1(C(N2CCCC(CCNC(c3cc([N+](=O)[O-])n[nH]3)=O)C2)=O)CCC(=O)NC1 18246,N1(CC)CCCC(C(=O)OC)C1.C1(NC(C(c2cn(C)cn2)C)=O)C=CC(C=O)C1 18247,N1(C(C(CSC)O)=O)CCOC(CN(C(=O)CCc2cc(C)co2)C)C1 18248,C(=O)(CS(=O)(=O)C1CC1)NCC1N(C(c2cc(C)c(C)s2)=O)CCCC1C 18249,CC(C)(CC(=O)NC1CCCN(C(c2nccc3c[nH]nc23)=O)C1)CC(F)(F)F 18250,CCC(C(=O)N1CC2CC2(NC(c2cc(C(=O)OC)no2)=O)C1)C(F)(F)F 18251,CC(CCNC(=O)CC1CCCO1)NC(=O)C=C1CC1 18252,CCC(CC)(CO)C(=O)N1CC(O)C(O)C1CNC(=O)CC1CC2C=CC1C2 18253,CC(C)CC(O)C(C)C(=O)N1CC2=CC2C1.C1(CCNC=O)CC=CCC1 18254,N1(CCCCNC(CC(C=C)C)=O)CCN(C(c2ccncc2)=O)CC12CCC2 18255,Cc1ccc2oc(CC(=O)NCC3CCCCN3C(c3ccncc3Cl)=O)nc2c1 18256,CC(C)(C)CC(C)(C)C(=O)NC1CCN(C(=O)CC2CCCC3(CCC3)O2)C1 18257,CN1CCCC(C)(C(N2CCC(C(=O)NC3(c4ncccn4)CC3)C2)=O)C1 18258,c1(SCCC(=O)NCC2CN(C(C(C)=C3CC3)=O)C3C2C3)ccc(F)c(F)c1 18259,c1(N2CCN(CC(=O)NC(CCCOCC=C)C)CC2)ccccc1C#N 18260,c1(CNC(C2(F)CCN(C(C=Cc3cn(C)nc3)=O)C2)=O)nnc2n1CCC2 18261,C=CCC(C)(C)CC(=O)N1CCC(C)C(CNC(=O)C(C)n2cccn2)C1 18262,c1(C(N(CCNC(=O)C(C2(O)CCCCC2)(F)F)CC)=O)cnc2nccn2c1 18263,N1(C(C(C)NC(N)=O)=O)CCN(C(CNC(C2CCCSS2)=O)C2CC2)CC1 18264,C(CCN=C(NCc1ccc2c(c1)CCO2)N1CCC(CCO)(CO)C1)OC 18265,c1(C(=O)NCCCN(C(C(CC(C)C)(F)F)=O)C)cc(=O)c2ccccc2o1 18266,c1(CNCC2N(C(C3(O)CC3)=O)CC(F)C2)c(OC(F)(F)F)cccc1F 18267,c1(NCC)cc(C(=O)OCC23CN(C(=O)OC(C)(C)C)C(C)(CO2)C3)ccc1O 18268,c1(C(=O)NCC(C)NC(c2snc(O)c2Cl)=O)ccc(C2COC2)cc1 18269,C1(N(CC)CC)CCCC1(C)C(=O)NCC1=NOCC1 18270,n1(C(C)C)ccc(C(=O)NC(CNC(=O)C(C)C2(O)CCC2)CO)n1 18271,C1(NC(CCOCCOC)=O)CN(C(C2CC(C3CC3)=NO2)=O)C2(CCOCC2)C1 18272,c1(OC)cccc2cc(CCNC(=O)NCc3ccc(C#N)c(OC)c3)oc12 18273,c1(C(=O)NC(C(C)NC(=O)CCC2CC2)(C)C)cc2ccccc2n1C 18274,CCCCCC(C)CCC(=O)NCCN(C(=O)C(CC)CCC)C 18275,C(=O)(CC(C)CC(C)(C)C)NCC1(F)CCCN(C(CCOCCCOC)=O)C1 18276,Cc1cc(C(C(F)(F)F)NC(c2csc(Br)c2)=O)ccc1OCCN(C)C 18277,c1(CN(S(=O)(=O)CC2CCC2)Cc2ncc(CC)o2)cccc(C(F)(F)F)c1 18278,CCC(C)(C)C(O)C(=O)N1CC(F)CC1CNC(=O)C(C)(C)C1CCCCC1 18279,CC1CN(C(C2CC(Cl)C2)=O)CCC1NC(=O)Cc1cccs1 18280,CC1CCCN(C(=NCCN2CCOCC2)NCC2(COCCO)CCOCC2)C1 18281,N1(C(COc2c(OCC)cccc2)=O)CCC(C)(C(=O)N(C)CCN(C)C)C1 18282,c1(C(=O)NCC(C)NC(c2cc(F)c(C)cc2F)=O)ccc2[nH]ccc(=O)c2c1 18283,c1(C(N2C(CNC(c3c(C)c(Cl)ccc3)=O)CC(F)C2)=O)cccn2cncc12 18284,C(=O)(CCCCCN(C)Cn1nc(C)cc1C)NC1(COC)CN(C(C)=O)C1 18285,Cc1cncc(CC(=O)NCC2CC(CNC(c3conc3C3CC3)=O)CO2)c1 18286,Cn1c(C(=O)NCC(N2CCCC(c3ccco3)C2)=O)cc2sccc12 18287,C1(NC(C2(C)CNC(=O)C2)=O)CCCCN(C(C2CC2(F)F)=O)C1 18288,c1(C(N2CCC(OCCNC(C3CC(SC)C3)=O)C2)=O)cncc2[nH]ccc12 18289,C1(N(C)CCC2CC(F)C2)CCN(C(C2CCCC2O)=O)CC1 18290,N1(C(c2cn(CCC(C)C)nn2)=O)CC2CC1C2NC(c1sccc1CC#N)=O 18291,Cc1cc(CNC(=O)C(O)c2ccsc2)oc1C(=O)NOCc1ccccn1 18292,c1(C(=O)NC2CCCCC2NC(C2CCO2)=O)[nH]cc2c1CCS2(=O)=O 18293,Cc1cccc(C(=O)NCCC2(O)CN(C(=O)CCOc3cccnc3)C2)c1 18294,C1(NC(C2CCC(C)(C)O2)=O)CN(C(c2cnns2)=O)Cc2nccn2C1 18295,N(C1CCC(NC(c2ccnc(-n3cccn3)c2)=O)c2ccccc21)C(CC)=O 18296,c1(C(C)C)ccc(C(=O)NCC(C)CNC(c2coc(C(F)F)c2)=O)o1 18297,C(CC(=O)NCC(=O)N(C)OC)(C(F)(F)F)NC(C(CC#C)C1CC1)=O 18298,c1(SC(C(=O)CCOC(CC)=O)C)cccc(C#N)c1 18299,c1(C2(C(=O)O)CCCN2C(c2cccc(C3CCC3)c2)=O)c(F)cccc1F 18300,c1(C(N2CCC(C)C2CNC(c2ncn(C)n2)=O)=O)ccn2c1CS(=O)(=O)CC2 18301,CC1CC(c2nnnn2-c2ccc(F)cc2)(Nc2nnn(C)n2)CC(C)O1 18302,C(c1ccncc1C)=CC(=O)NCCc1c(CNC(C(C)=C(C)C)=O)nco1 18303,CC1(C)C=C(C(=O)NC2(C(=O)NCC3(C)CC3(C)C)CC(F)(F)C2)C1 18304,C1(C(=O)NCC2CC(C(=O)Nc3cn(CC#C)nc3)C2)C2CCCC(=O)C12 18305,C12(CNC(c3cnc(C4CCCCC4)s3)=O)CC(CO1)N(C(=O)C1CC1)C2 18306,C1(CNC(CNC(C2N(C)CCOC2)=O)=O)CC(C(N)=O)=NO1 18307,c1(C(N2C(CNC(C3C(C4C(C)C4)C3)=O)CC2)=O)cnn2cc(C#N)cnc12 18308,CC(C)(CNC(C1CC(F)CCN1C(C1CCOC1(C)C)=O)=O)CN=[N+]=[N-] 18309,c1(C(=O)NC2CC(F)CN(C(c3ccns3)=O)C2)cccc2sccc12 18310,CC(C)C(C(=O)NCCCN(C(c1cc(F)n[nH]1)=O)C(C)C)N1CCCC1=O 18311,c1(C(=O)NCC=CCNC(C(F)OC)=O)nc2ccccc2c(Cl)c1Br 18312,C1(C(=O)NCC2N(C(C)=O)CCC2)CN(C(=O)CN2CCCC2)C(C)(C)C1 18313,c1(C(=O)NCCN(C(CCCC(=O)NCC)=O)CC(C)O)ccnc2c1CCO2 18314,C(=O)(C(C)(C)C(F)F)N1CCCC(CCC)C1.C1C(O)(C(F)(F)F)c2cn1nn2 18315,C1(NC(=O)CC2CCC2)CCCC1NC(c1ccc(Cn2cccn2)o1)=O 18316,N(C1COc2ccc(F)cc21)C(CCCC=C)c1ccc(OC(C)C)cc1 18317,C1(C#N)(C(=O)NCC2CC(C(=O)NC(C(=O)NCC)C)C2)CC1(C)C 18318,N1(C(=O)OC(C)(C)C)CCOC2(C1)CN(N1CCc3cncnc3C1)C2 18319,C1(COC(C(C2CCN(C(=O)OC(C)(C)C)CC2)F)=O)CCc2nncn2C1 18320,CP(C)(=O)c1cccc(C(=O)NCCCNC(C2CC3CCC3C2)=O)c1 18321,c1(NC(=O)Cc2cccnc2O)cc(-n2ccnn2)ccc1F 18322,Cc1nc2cc(C(N3CCC(C#N)(NC(=O)C(C)(C)C)C3)=O)ccc2n1C 18323,C1(C(N(CC(CN(C)C(C2CCC2)=O)O)C)=O)CN2CCN1CC2C 18324,N1(C(C=C(CCC)C)=O)CC(C2CC2)(C(=O)NCCCCc2cnc[nH]2)C1 18325,c1(C(N2C(CNC(C(CC3CCCCC3)OC)=O)CCC2)=O)sc2cncn2c1C 18326,C=CC1(CC(=O)NC2(N3CCNC3=O)CC2)CN(C(=O)C(O)CCSC)C1.C(N)=O 18327,S(=O)(=O)(c1c2ccccc2nn1C)NC(c1c[nH]c(=NC)s1)C(N1CCCC1)=O 18328,C12(C(N3CC(C)(NC(CC(CC)C4CCC4)=O)C3)=O)CCCC(C1)OC2 18329,n1(CCC(=O)N(CCCCCNC(C2C(C)C2)=O)C)cc([N+](=O)[O-])cn1 18330,c1(C(N2CCC(NC(C)=O)C23CC3)=O)cc(C)cc2c1NCCC2C 18331,N1(C(C2(F)CN(C(C(C)OCCOC)=O)C2)=O)CCCCC(C)(F)C1 18332,N1(C(C(C)(C)CO)=O)CC(CNC(=O)C(O)CC[S+](C)C)OC2(CCC2)C1 18333,c1(CN(C(C(=O)N)=O)CCNC(C2(C(N)=O)CC2)=O)cccc(C2CC2)n1 18334,C1(C(N2CC(CCOC)C2)=O)(CNC(c2cscn2)=O)CC12CCC2 18335,N#Cc1cnc(Cl)c(C(=O)NCCC2(O)CN(C(=O)CC3C=CCCC3)C2)c1 18336,CC(O)C(C)C(=O)N1CCN(C(C2(C)CC(C)(C)C2)=O)CC1 18337,C(c1cncc(OC)c1)=CC(=O)NCC1C(NC(C2CC(C)(CC)C2)=O)CC1 18338,N1(C(CC(C)C(F)(F)F)=O)C(C)CC2CN(C(c3c(Cl)cncc3Br)=O)CC12 18339,c1(C(N(CCNC(C(C)CC2CC2)=O)C)=O)cc2ncccc2[nH]1 18340,C=C(C)C(CC(=O)N1C(C(=O)NC2CCCNC2=O)CC2CC12)OCC 18341,c1(C(N2CC(O)(CNC(c3c(SC)cccc3)=O)C2)=O)cc(Cl)ccc1Cl 18342,c1(C(=O)NC2CN(C(C3(Oc4ccc(F)cc4)CC3)=O)CC2O)cc2occc2s1 18343,C12(C(=O)NC(C)CCN(C)C(c3cncc(Cl)c3)=O)CCCN(CCC1)C2 18344,c1(C(=O)NC2CCC(NC(C(CC)(C)C#N)=O)C2)cnn2c(Br)cccc12 18345,C1(CC)C(C)CCN1C(=O)CSCCNC(c1cccc(NC)c1)=O 18346,c1(N2CCCC(=C)C2)nc(=NC(C)F)[nH]c2cc(C)ccc12.C(CO)OCC=C 18347,c1(N2CC(CNC(C(CCC)NC(N)=O)=O)OCC2)ncc2c(ncn2C)n1 18348,C(C1=NOC2CC12)(c1nnnn1C1CC(F)(F)C1)NCC(C(C)C)(C)C 18349,C(=O)(CCCCCCc1ccccc1)N1CCC(NC(C(C=C)(C)CC)=O)C1 18350,c1(C(=O)N(C2CC2)CC2(Br)CC2(F)F)cccc(C(=O)NC2(CCO)CCC2)n1 18351,C(c1nc2ccccc2o1)=CC(=O)N(C(C)CNC(=O)Cc1ccnc(O)c1)C 18352,CCC(CCCC(=O)N1CCCOC(C)C1)NC(=O)C1=CCCC1 18353,c1(CC(=O)NC2CC(F)(CNC(=O)Cc3ccccc3O)C2)cc(F)ccc1Cl 18354,N(C1CCc2ccccc21)C(CCNC(C(C)(C)SC)=O)=O 18355,N12CC1(C)C(=O)NCCN(C)CCOC2=O.C(C)(C)(C)NCC=CCO 18356,c1(C(C(=O)NCC2N(C(C3CN(C(C)C)C3)=O)CC2)O)cnccc1C.c1ccsc1C 18357,c1(C(N2C(C(C)NC(CC(=O)NCC)=O)CCCC2)=O)nc(C)c(N)cc1C 18358,N1(C(C(OCC)OCC)=O)CCCC(C)(C(N2CC=CC2N(C)C)=O)C1 18359,Cc1coc(C=CC(=O)NCC2CCCN2C(=O)CCc2cc[nH]n2)n1 18360,C(=O)(CC(=O)N(CC(O)CN(C)C(c1ccsc1SC)=O)C)NCC#C 18361,Cc1nccn1CCC(=O)NCC1CC(NC(c2ncoc2C(C)(C)C)=O)C1 18362,c1(Cn2cc(C3(C)N(C(CC(CC)C)=O)CCC3)nn2)cc(C)cc(O)c1 18363,CON1CC(C(=O)NCC2(CO)COC2)CC1=O.N12CCC(C1)OCC2=O 18364,C1(NC(C=CC(C)C)=O)CCCC(CN(C(c2cc(C(F)(F)F)c[nH]2)=O)C2CC2)C1 18365,C(=O)(C(COCC1CC1)C(F)(F)F)N1CCC(NC(C(C)OCC)=O)C1 18366,Cc1cc(Br)cc2c1CCN(S(=O)(=O)C1CC(S(C)(=O)=O)C1)C2 18367,CCC(C)CC(C)C(=O)NCCCOCCN(C(=O)CSc1ccc(C)nc1)C 18368,C(=O)(CCCC(O)c1ccccc1)OCC(=O)NC1CCC(OC(F)(F)F)CC1 18369,N1(C(C2C(C)(CC)C2)=O)CCCCC12CC(NC(=O)Cn1ccnc1C)C2 18370,N1(C(c2c(=O)ccn(C)c2)=O)CCN(C(C2(F)CC2)=O)CC12CCC2 18371,C1(NC(c2c(C)nn(C)c2)=O)CCCCC12CCN(C(=O)COC1CCOC1)C2 18372,C=C(C)CC(C(=O)NCc1ncc(C)s1)NC(C1CCCN1CC)=O 18373,C1(C(=O)NC2C(C#C)CCC2)CNC(=O)CN1C(=O)COC1CCC1 18374,C(=O)(CC(C)C(F)(F)F)N1CCCC(F)(C(N(CCCC(=O)NC)C)=O)C1 18375,N(C1CCCc2c(F)cccc21)C(C(C1(C=C)CCOCC1)C)=O 18376,C#CC1CN(C(C2CN(C(c3nscc3C)=O)CC2(C)C)=O)CCN1C 18377,C1(COC)CC(CNC(=O)CN2CCN(C)CC2)N(C(=O)CCCC2CC2)C1 18378,c1(C(=O)NCC(C)NC(=O)C(c2ccc(Cl)cc2)(C)O)nc(Cl)sc1Cl 18379,C1(NC(C=C2CCC(C)CC2)=O)CCN(C(c2cc(Cl)c(Br)[nH]2)=O)C12CC2 18380,c1(C(N(C2CC(NC(=O)CCc3cccs3)C2)C)=O)ccoc1I 18381,N1(C(C(C(C)(C)C)=O)=O)CC(CNC(C2COCCOC2)=O)CC12CCC2 18382,N1(C(CC2C(C)(C)C2)=O)C2CCC1CN(C(c1cc(C3CC3)ccn1)=O)C2 18383,C12=NC=CC(=NCCOCC1)N2.c1(CNC2(CC=C)CCOC2)cc(C)cc(C)n1 18384,CC(C)C(C(=O)NCCC1CN(C(c2cccn2C)=O)CCO1)c1ccn(C)n1 18385,N1(C(C(C)=C2CC2)=O)CCC2(C1)CN(C(c1ccc(F)c(O)c1)=O)C2 18386,C1(CNC(C2(O)CC2)=O)CCC2CN(C(c3ccc4ncnn4c3)=O)CCC2C1 18387,n1(CC)nc(CN2CC3CC2(C)C3)c2c1CCOC2 18388,C1(NC(C2(CCOC)CC2)=O)CN(C(c2cncn(C)c2=O)=O)C2CCCCC12 18389,C#CC(C)(C)C(=O)NC1CCC(C(=O)NCC2CC2C)CC1 18390,Cc1nnsc1C(=O)NC1(CCNC(c2cnn(Cc3ccccn3)c2)=O)CC1 18391,c1(C(N2CC(N(C(c3c(C)cn(C)c3)=O)C)C(F)C2)=O)ccc2nonc2c1 18392,c1(CC(=O)NCC2CN(C(C(C)NC(CC)(C)C)=O)C2)ccc2c(n1)NCCC2 18393,C1(C)(NC(C(C2CN(C(=O)COCCOCCO)C2)OC)=O)CC2(CCC2)C1 18394,C(=O)(C1=CC2CCC1C2)NCCN(C(c1cnn(-c2ccccn2)c1C)=O)CC 18395,C1(CNC(C(C)(C)SC(F)(F)F)=O)CN(C(c2cnns2)=O)CCO1 18396,C(CCC(C(=O)NC1C(O)CC1O)NC(c1ccc(C)c(C)n1)=O)OC 18397,N1(S(CC)(=O)=O)CCC(C(=O)NC(C)(CNC(C2(O)CCSC2)=O)C2CCC2)C1 18398,N1(C(c2c(C(C)C)onc2)=O)CC(C(=O)NCC2CCCC2O)C2(CC2)C1 18399,N(C1c2ccccc2CC1NC(=O)C1Cc2ccccc21)C(c1cc(Cl)no1)=O 18400,c1(C(=O)NC2(c3ccc(NC(C)=O)cc3)CCOCC2)cnc(F)cc1C 18401,C(CCN=C(NCc1cncc(O)c1)NC1CCOC(c2ccccn2)C1)OC 18402,C#Cc1ccc(C(N2CCCC2CCNC(=O)C(O)CN(C)C)=O)c(OC)c1 18403,C(=O)(CCC(=O)NCC(C)(C1CC1)NC(=O)C(n1ccnc1C)C)NC 18404,N1(C(C(C2CC2)OC)=O)CCCC2CCN(C(=O)C(F)(F)CC3CC3)CC12 18405,Cc1cnc(C)c(C(=O)NCCC2(CNC(c3n[nH]cc3C(C)C)=O)CC2)c1 18406,c1(C(N2C(CCNC(C(CCOC)C)=O)CCCC2)=O)ccc(C#N)c(Cl)c1 18407,C1(C(=O)NCC(C(C)C)NC(C2(CC#C)CC2)=O)CC2(C1)CC(C#N)C2 18408,c12ccc(cc1)C(N)CC(=O)NCC2C.c1(O)ccc(Cl)cn1.CCN 18409,c1(OC)cccc(C(N2CCC(N(C)C(C3C(C)(C)C3(F)F)=O)C2)=O)c1[N+](=O)[O-] 18410,C(=O)(N(OC)C(C)C)C1(C=C)CN(C(=O)CCOC(C)=O)C1 18411,N1(C(C2CC(OCC)C2)=O)CC(CNC(=O)C(C)OC2CCOC2)C(C(F)(F)F)C1 18412,C(C1CCCCCC1)=CC(=O)NC1(CO)CN(C(c2ccc(N(C)C)nc2)=O)C1 18413,C1(CC)CCN(C(=O)C(O)CC2CCCC2)C(C(N2CCC2(C)COC)=O)C1 18414,c1(NC(COC)Cc2ccco2)[nH]c(=NCCC2CC=CCC2)nc2c1ncn2C 18415,N1(CC)CCN(c2ccc(F)cc2Cl)CC1C.C1(=O)C(CC)N1 18416,C(=O)(C(C)C1=CCCC1)NC(CCCNC(C=CC=CC)=O)c1ccccc1 18417,C1(C(=O)OCC)CCC(C(=O)NCCSc2cn(C(C)CO)nn2)S1 18418,c1(CC)cc(C(=O)NC2CCCC(NC(C34CCC(C3)NC4)=O)C2)n(C)c1 18419,N1(C(C(CCCC)C)=O)Cc2n[nH]cc2C1C(=O)NC(c1nccc(O)n1)C 18420,CN1CCC(C)(C(=O)NCC(O)CCNC(=O)C(CO)Oc2ccccc2)CC1 18421,c1(CN2CC(C(=O)NC(CCC)CO)SCC2)ccc2c(c1)OCCO2 18422,N1(C(CC=C=C)=O)CCOC2CN(C(c3[nH]c(=N)ccc3C)=O)CC12 18423,N1(C(CCOCCCOC)=O)CCC(C)(C)C1CC(=O)NC(C)CCCCO 18424,C12(C(N(C3CN(C(=O)COC4(C(F)(F)F)COC4)C3)C)=O)CC(F)(C1)C2 18425,c1(CN(CC(C)NC(=O)C(C)CN2CCC2)CC)ccc(F)cc1C 18426,c1(OCC)cccc(C=CC(=O)NC2CCCN(C(C3(C)CNC(=O)C3)=O)C2)c1 18427,CC1(C)CCN(C(=O)C=Cc2cccs2)CC1CNC(=O)CCc1cc(Cl)cs1 18428,CC1CCCN(C(=O)CC(F)(F)c2ccccc2)C1CNC(=O)CC1OCCO1 18429,S(=O)(=O)(c1c[nH]ccc1=NCC1CC(C(F)(F)F)CO1)NCc1c(Cl)cn(C)n1 18430,N1(C(C2N(Cc3cc(OC)cc(F)c3)CCNC2)=O)Cc2ccc(Br)cc2C1 18431,c1(OCCC(=O)NCC2CC2NC(=O)C(C2CCCCCC2)O)ccc(F)cc1Cl 18432,C1(C(N2CCC(c3ccon3)C2)=O)COC2(C1)CN(C(c1cccnc1O)=O)C2 18433,C#Cc1ccnc(C(=O)N(CCNC(=O)C(C)(C)NS(C)(=O)=O)C2CC2)c1 18434,C(CC(=O)NC1CC(C)CCC1O)(C(C)NC(N)=O)NC(CN(C)CC)=O 18435,C1(NC(c2cc[nH]n2)=O)CN(C(c2cscn2)=O)C2(CCC2)C1 18436,C1(n2cc(C3C4CN(C(c5c(C(C)C)ocn5)=O)CC43)nn2)CCCCNC1=O 18437,c1(C(=O)OC)cc(CN2CCOC(c3ccc(C(F)(F)F)cc3)C2)cc(N)c1 18438,C(=O)(N=c1[nH]nc(-c2c(F)cccc2Cl)s1)NC(c1nc(C)[nH]n1)C 18439,N1(C(C2C(NC(C(C)NC(CC)=O)=O)CC=CC2)=O)CCOC(C)C1C 18440,C1(C(N(CCCCCC)CCNC(=O)CCF)=O)OCCCC1C(C)C 18441,S(=O)(=O)(c1ccc(S(=O)(=O)N2CCCC2)cc1)N(C(C)(C)C(=O)O)C1CC1 18442,C1(CCC)(NC(=O)C=C(C)C(C)C)CCCN(C(=O)C(C)CC(F)F)C1 18443,C=Cc1ccc(C(=O)NC(C2CCOC2)CNC(c2scnc2Cl)=O)cc1 18444,c1(C(=O)NCC(CNC(c2c(CC)nns2)=O)CO)cc(Cl)cc2c1OCC2 18445,Cc1cc2c(cc(C(N3CC4CCN(C(=O)CS(C)(=O)=O)C4C3)=O)n2CC)s1 18446,C1(C(=O)Nc2c(C#C)cccc2)CCN(C(=O)CN(C)CCOC)CC1(C)C 18447,C12(NC(C3CN(C(C(CC#C)O)=O)CC34CC4)=O)CCC(C1)C(O)C2O 18448,c1(C(N2CCC(NC(c3ccn4c3CCCC4)=O)C2)=O)cc2c(cc1Cl)NCC2 18449,C=C(C)C1OCCC1C(=O)N(C(C)C(=O)N(C1CCC1)CC(C)C)CC 18450,C1(O)(CNC(Cc2c(C)cccc2)=O)CCCN(C(c2cc(Cl)no2)=O)CC1 18451,c1(CC)cc(C(N2CCCC(C(C)NC(=O)C=CC(C)(C)C)C2)=O)nn1CCO 18452,C(=O)(C(F)CCC(C)(C)C)NC(C(C)C)CCNC(c1noc2c1COCC2)=O 18453,C1(NC(CC2(OC)CCOCC2)=O)(CNC(=O)C(C)C(F)F)CCOCC1 18454,C1(C(N2CCOCC2)=O)CN(Cc2ccnc(Br)c2)CC(F)(F)C1 18455,c1(C(=O)NC(C)CCNC(c2c[nH]c(Br)c2)=O)cccc2ncccc12 18456,Cc1cccc(C2(C(=O)N)CC2)c1N.C1(c2ccccn2)CCN(C)CC1 18457,Cc1ncn(C)c1C(N1CC(n2cc(CNC(c3csc(S)n3)=O)nn2)C1)=O 18458,c1(C(=O)NCCCCNC(C2(C)CC2)=O)cc2occc2[nH]1 18459,C1(NC(=O)CC2(O)CCOC2)CCCCCN(C(c2ccc3cnoc3c2)=O)C1 18460,N1(C(C(C=CC)O)=O)CCCCCCC1C(N1CC2CCC2(CO)C1)=O 18461,CC(C(=O)NCC1(O)CN(C(c2ccnn2CC2CCC2)=O)C1)C(C)(F)F 18462,Cc1oc(S(C)(=O)=O)cc1NC(C1CC(O)CN(C(=O)CNc2ncccn2)C1)=O 18463,N1(C(C2(C)CCN(C)C2)=O)CCC(NC(c2ccc3ccsc3c2)=O)C(C)(C)C1 18464,N1(c2nnc(CC)o2)CCC2(CC1)CN(C(=O)C(F)C1CCOC1)CC(C)O2 18465,c1(N2CCN(C(=O)NCCCc3ccc(F)cc3)CC2)ncc([N+](=O)[O-])cc1F 18466,N1(C(C2=CC(C)(CC)C2)=O)CC2CCCC2(NC(c2ccn(C)c2)=O)C1 18467,N1(C(C2CC(C)SCC2)=O)CCC2(C1)CN(C(=O)Cn1cccc1)CCO2 18468,n1(CC)cc(C(N2CC(C(O)C(=O)NC3CC(C(C)C)C3)C2)=O)nn1 18469,C1(NC(c2ccc(C)nn2)=O)CN(C(C2CC2C(C)O)=O)CCC12CCC2 18470,N1(C(COCCC(C)C)=O)CC2(CCC2)OCC1C 18471,N1(C(CN(C2CCC2)C(C2CC(C)N(C)CC2)=O)=O)CC(C2CC2(F)F)C1 18472,c1(C(N(CCCN(C(C(C)NC(C)=O)=O)C)C2CC2)=O)cnn(CCO)c1 18473,C1(NC(c2ccc(C)o2)=O)CCCCC12CCN(C(c1cncc(F)n1)=O)C2 18474,C1(C(N2CC(CC(C)NC(CCNS(CC)(=O)=O)=O)C2)=O)CCCN1C 18475,Nc1ccc(C(N2CC3(CC3)CC2CNC(=O)C(F)=CCCF)=O)c(Cl)c1 18476,c1(C(=O)NC2C(C(N(C3CC(F)(F)C3)CC)=O)CC2)ccc(C2CC2)cc1 18477,c1(C(=O)NCC2(NC(C(CC)C)=O)CCC2)cccnc1-n1ccnc1C 18478,c1(CNC(=O)C(N2CCC(F)(c3ccc(F)cc3)C2)=O)ccc2c(c1)OCCO2 18479,CONC(=O)C(C)(C)CCNC(=O)CC(C)C(=O)OC 18480,c1(C(=O)NCCC(C)CCNC(=O)CS(C)(=O)=O)cc(C(F)F)cc(F)c1 18481,C1(NC(CCC(C)OC)=O)C(C)CCN(C(=O)COCCN(C)C)C1C 18482,C1(NC(=O)Nc2cccnc2)CCCC(CN2CCN(c3ccncn3)CC2)C1 18483,C(=O)(C1=CCS(=O)(=O)C1)N(C)CC1CCCCN1C(c1cccc(C2CC2)c1)=O 18484,CS(=O)C=CC(=O)N1CCC(CCCNC(=O)C(N2CCCC2)C2CC2)CC1 18485,c1(CC(=O)N(CC(C)CNC(C2CC(C)OC2C)=O)C)coc2ccc(F)cc12 18486,Cn1c(C(N2CC(O)(CNC(=O)Cn3ccnn3)C2)=O)cc2c1CCOC2 18487,N1(C(C(C)OCOC)=O)CCC2(CCC(NC(c3ccc4n[nH]cc4c3)=O)C2)C1 18488,C1(C(N2CCC(C#C)(O)CC2)C(=O)NCC=C)CC2(CO1)CC(F)(F)C2 18489,c1(C(=O)OCC)cc(C)c(C(N2CCN(c3ccco3)CC2)C(=O)NCC)cn1 18490,c12cn(C)nc1C(=O)N1CCCC(C1)C(=O)NC2.C1(SC)(CC2CC2)CN(C)C1 18491,c1(CC=C)cccc(C(=O)NCC2CCC2NC(=O)CSCC(=O)NCC)c1 18492,CC1CC(C(=O)N(C2CCCC2O)C)N1C(=O)CCN(C)C 18493,c1(C(=O)NCC(C(N2CC(C)(CC)C2)=O)C)n[nH]c2c1COC2 18494,C1(CNC(NNC(=O)c2scc(N(C)C)n2)=O)CCn2ccnc2C1 18495,N1(C(c2cccc(-c3ncn(C)n3)c2)=O)CCN(C2CC2)CC12CCOCC2 18496,c1(C(=O)NCCN(C(C2CC(CCC)C2)=O)C)occ(C)c1C 18497,N1(C(CC2(OC)CCCC2)=O)CC(O)(CNC(c2cnn(CC3CC3)c2)=O)C1 18498,N1(C(=O)NC(CCCC)C)CCc2ccc(C#N)c(Cl)c2C1 18499,c1(C(=O)NCC2CCN(C(c3cn(CC)nc3)=O)CC2O)cccc2c1CCN2 18500,c1(C(N2CCC(C)(C(=O)NC(C(C)SC)C)C2)=O)cnc2cc[nH]c2c1 18501,c1(C(N2CCC(=CCNC(C3(C#N)CCCC3)=O)CC2)=O)ccc2c(c1)CCO2 18502,N1(C(c2c(C)cc(C)s2)=O)CCC(CNC(c2c[nH]nc2C2CCC2)=O)C(C)C1 18503,C(c1ccc(Cl)c([N+](=O)[O-])c1)=CC(=O)NCC1N(C(c2nc(C)sc2)=O)CC1 18504,c1(CC)cc(C(=O)NC2(C(=O)NC3CCN(C)C3C)CCCC2)n(C)n1 18505,C1(C(=O)NCc2snc(C)n2)CN(C(C2CNC(=O)N2)=O)CC1C(C)C 18506,C(=O)(C1=CCOCC1)NCC1(F)CCC(CNC(C2CN(C(C)=O)C2)=O)C1 18507,N1(C(=O)C(c2cnc(Cl)s2)Sc2cccc(Br)c2)CCCN(C2CCOCC2)CC1 18508,c1(C(=O)NC2CCN(C(C(COC)NC(C)=O)=O)C2)nn(C)c2ccccc12 18509,N1(CC(=O)Nc2ccc(C)nc2Cl)CCN(C(c2ccco2)=O)C(C)(C)C1 18510,N1(C(C=CC(=O)NCC2CCC(=O)NC2)=O)CCN(C(C2CCC2)=O)CC1 18511,c1(N2CC(NC(c3c(C)c(Cl)ccc3)=O)C(F)CC2)ccnc(S(C)(=O)=O)n1 18512,C1(NC(=O)CN(CCO)Cc2cccc(F)c2F)CC2CCC1CC2O 18513,C=C(C)C(C)(O)C(=O)N1CCCC(C)(NC(c2cnc(S)n2C)=O)C1 18514,Cc1ccc(Br)c(N)c1C(N1CCCC(NC(C2CC3CCC2C3)=O)C1)=O 18515,C1(NC(=O)Cc2ccns2)CN(C(C2(CC3CC3)CCC2)=O)CCC1C(F)(F)F 18516,N1(C(CN(CCOC)C)=O)C2CCC1CC(N(C)C(C1(C)CCC(O)CC1)=O)C2 18517,Cc1cc(CC(N2CCC(N(CCO)Cc3cnc(S)[nH]3)C2)=O)n(C)n1 18518,c1(C(=O)NC(CC=C)CNC(=O)CSC2CCCO2)ccc2nccnc2n1 18519,C1(C#CC(=O)NC2CC23CCN(C(c2csc(COC)n2)=O)CC3)(CC)COC1 18520,CC1CCC(NC(C2CCC(C)(C)CC2)=O)CN1C(C1CN2CCC1CC2)=O 18521,c1(CC)ccc(C)cc1C(N1CC(O)(C(C)NC(=O)CC(C)SC)C1)=O 18522,C1(C(=O)NCC2(C(=O)NCCN(C)CCO)CC(C)(C)C2)CC(=O)NC(=O)C1 18523,C1(NC(=O)C(O)CC2CC2)CN(C(c2ccc3nonc3c2)=O)C2(CCC2)C1 18524,C1(OCC#C)CCCN(C(c2ccc(CC(=O)Nc3cccn3CC)cc2)=O)C1 18525,c1(C(=O)NC2C(NC(c3ccc(C4OCCO4)cc3)=O)COC2)ncc(F)cn1 18526,Cc1cc(CN(CCNC(c2cnc(Cl)s2)=O)CC2CC2)c(C)n1CC(F)(F)F 18527,c1(CC2CN(C(=O)NCc3nn[nH]c3C(F)(F)F)C2)ccccc1F 18528,C1(C2N(C(C(=O)NC(c3ccc(C)cc3C)CC)=O)CCC2)CCC(F)(F)CC1 18529,c1(C2CNC(=O)N2)cc(F)ccc1F.O=C1CC(CNC(c2ncco2)(CC)C)CCN1 18530,C1(F)(C(=O)NCCC2(CNC(C3CC=CCC3)=O)CC2)CC1(Cl)Cl 18531,C(=O)(C1CCCc2ncnn21)N1CC2C(Nc3nc(C)nc4c3ccs4)C2C1 18532,C(=O)(CC(C)O)NCC(C)=CC(=O)N(CC(c1nn[nH]n1)C)C 18533,C1(NC(c2c(C)cnnc2)=O)CC(C)CN(C(C2CC2(F)F)=O)C1 18534,Cc1nccc(C(=O)NCC2(CNC(C3(C(C)C)CC3)=O)CC2)c1N 18535,c1(C(=O)NCC2C(NC(C(C)C#N)=O)CC2)c(F)ccc(F)c1Cl 18536,c1(CC(=O)N(C(C)CNC(C2CCC3CC23)=O)C)cccnc1F 18537,N1(C(C(C=C)(C)CC)=O)CC2CN(C(c3c(-c4ccsc4)noc3C)=O)CC2C1 18538,c1(C(N(C(C)CNC(c2ccoc2C)=O)CC)=O)cc(Cl)n(C)n1 18539,N1(C(c2c(OC)csc2)=O)CCOCC1C(=O)Nc1cncc(C(F)(F)F)c1 18540,C1(CC(N2C(CNC(C(C)n3cccc3)=O)CCC2)=O)SC(=N)NC1=O 18541,C(CCCNC(=O)C=CC(N)=O)N(C(C=C(C)C)=O)C 18542,C1(NC(Cc2c(C)cco2)=O)CCCN(C(=O)C(C)c2cccs2)C1 18543,c1(OC(c2cc(C(=O)O)[nH]c2)=O)ccc(F)c(F)c1.N12CCCC(C1)C2=O 18544,C(CC(F)(F)F)SCCNC(=O)C(=O)NCC1CCC2CC12 18545,c1(C(=O)NCC2(NC(C(c3ccccc3)N(C)CC)=O)CC2)cnn(C)c1F 18546,C1(C(Cn2ccc(=NC(=O)OC(C)(C)C)[nH]2)=O)CCCC12CCOCC2 18547,C1(CNC(c2c(CC)onc2)=O)CCCCC1NC(c1cnn(CC)c1Br)=O 18548,C1(CNC(c2cc(C)[nH]n2)=O)CC2CC2N1C(=O)CC(F)(F)Cl 18549,C(CC(=O)NOCCN1CCCC1=O)(C(F)(F)F)NC(C(CCC)=CCC)=O 18550,N1(C(C(C(C)C)CN(C)C)=O)CCC2CCCC12C(N1CC(O)(CC(N)=O)C1)=O 18551,c1(C(=O)NCCC2N(C(CCC=C(C)C)=O)CCC2)nc(O)sc1C 18552,C(=O)(C(C(C)C)NC(=O)C(=O)NCC(F)F)NC(CC)COC 18553,C1(C(C)NC(C(CC)SC)=O)CCN(C(c2c[nH]cc2OC)=O)CC1 18554,NS(=O)(=O)c1sccc1C(=O)N(CCNC(C1COCCO1)=O)C1CC1 18555,c1(C(=O)NCCCC(CCC)NC(=O)CNS(N)(=O)=O)cc(F)cc2nc[nH]c12 18556,C1(CCNC(c2c(CC)ocn2)=O)CSCCN1C(C1CCCC1C)=O 18557,c1(C(N2C(CNC(c3[nH]cc(C(C)=O)c3)=O)CCC2)=O)ccc2c(n1)NCCO2 18558,c1(C(c2n(CC=C)nnn2)NC(C(C)C)c2cccs2)ccc(CCCCO)cc1 18559,C1(C(=O)NC(CN(C(c2cnc(O)c(C)c2)=O)CC)C)CC(=O)N(OC)C1 18560,c1(CC(=O)NC(C(=O)NCCC(C=C)C)CN(C)C)ccccc1C 18561,N1(C(COCC(=O)OC)=O)CCOC2CCN(C(=O)C(C)Cn3ccc(C)n3)CC12 18562,C1(CNC(C(C=CC)O)=O)CN(C(=O)C=CCCC(C)C)CCO1 18563,c1(-c2cc(-c3nc(CCCOC)nn3CCS(C)(=O)=O)n[nH]2)ccc(C)c(C)c1 18564,CC1CCC(CNC(C2N(C(c3cc(CC(=O)OC(C)(C)C)cs3)=O)CC2)=O)N1C 18565,C1(CNC(C(C)(C)OC(C)C)=O)CCC(CNC(=O)CC(O)C2CCCC2)CC1 18566,c1(NC(c2c(CNC(C(CC)OCC)=O)occ2)=O)cc(C)cnc1O 18567,N1(C(C(C)=CC2CC2)=O)CCCCC1C(C)NC(=O)Cn1ccc(C)n1 18568,N1(C(Cc2cc(CC)nn2C)=O)CC(C)N(C(=O)CCc2ncc[nH]2)CC1C 18569,Cn1c(C(=O)NCCC2CC(NC(=O)CSCc3ccccn3)C2)cnc1Cl 18570,N1(C(c2c(C)nc(Br)s2)=O)CC2CCC(C1)N2C(c1ccc2c(c1)OCO2)=O 18571,c1(NC(c2nc(CN(C)C)[nH]n2)C)cc(Cc2cncc(Cl)c2)ncn1 18572,C12CC(C13CCC3)C(=O)N2.N1(CCC)CCCC1CN(C)C 18573,c1(C(=O)NC(C2CCCN(Cc3cc(Br)ccc3Cl)C2)=O)cnc2ccc(F)cn12 18574,c1(SCC(c2n(C(C)(C)C)nnn2)NCc2ccn(C3CC3)n2)cccc(Br)c1 18575,N1(C(C(CC2CC2)NC(c2c(CC)cccn2)=O)=O)CC2(CC=CC2)C1 18576,N1(CCN(CCC)C(=O)NCC2CC2(F)Cl)CCCCS1(=O)=O 18577,N1(C(c2scnc2C2CC2)=O)CC2CCC(C1)N2C(C1CCCC1O)=O 18578,C(=O)(C(F)(CNC(C1(CF)CCOCC1)=O)C(C)C)NC(C#C)CC(C)(C)C 18579,C1(C#N)(COCC)CCCN(C(=O)NCCC2CC2)C1 18580,C1(NC(C2CC(C#C)(O)C2)=O)CCN(c2ncncc2I)CC1F 18581,C(=O)(CCCC(=O)N1CCCN(C(=O)CNC(=O)CCCCO)CC1)OC 18582,c1(C(=O)OCC)cc2c(s1)CCN(C(=O)C(N1CCCCC1=O)C)C2 18583,CC(O)C(F)(F)C(=O)NCCSCC(=O)NCC1CC(O)C12CCC2 18584,C1(NC(C(CC)C2CC2)=O)CCN2CCC1OCc1c(nccc1)C2=O.O(CCC)OC.OC 18585,N1(C(c2ccc(C(C)=O)cn2)=O)CC(CNC(=O)Cc2ccccc2)CC(C)C1 18586,C1(C(N2CCN(C(c3c(C)nn(C)c3C)=O)C3C2C3)=O)Cc2cncn2C(=O)N1 18587,c1(OC)cccc(NC(C2(C)CCN2C(c2cccnc2O)=O)=O)c1 18588,C1(NC(C(CC#C)C)=O)COC2(CNC(c3cc(Cl)ccc3Cl)=O)CC1C2 18589,C1(NC(C2CN(S(CC)(=O)=O)C2)=O)CC(F)CN(C(c2csc(C(F)F)n2)=O)C1 18590,Cc1ccc(Cl)c(CCCN2CCC2C)c1.C12(CC1)C(=O)N2C 18591,C1(CN(C(=O)CC2(C)CC2(F)Cl)C)CCN(C(C2(O)CCCCC2)=O)CC1 18592,c1(OC)ccc(N)c(C(N2CCC(NC(C3CC3(C)C)=O)C2(C)C)=O)c1 18593,c1(NC2(c3n(CCCSC)nnn3)CCCSC2C)cc(Br)cc2cccnc12 18594,c1(C(=O)NCC(C)(C)NC(c2cnn[nH]2)=O)ccc(F)c(Cl)c1N 18595,CC1(C)OCCCC1C(=O)NCC1CN(c2nnc(CC(F)(F)F)s2)CCCO1 18596,N1(C(CSC)=O)CC(NC(=O)Cn2nc(C)c3cccnc23)C2CCCCC12 18597,c1(C(C(=O)N(C)CCN(C)C(C2CCCC(O)C2)=O)(C)C)cccc(C#N)c1 18598,C1(CNC(c2ccccc2)c2nc[nH]n2)CC(C2CC2)=NO1 18599,C12(CC(=O)NC3C(CNC(CCC#CC)=O)C3)CC3CC(C1)CC(O)(C3)C2 18600,c1(OC2CCC2)ccc(C(=O)NC2C(NC(C(C3CC3)OCC)=O)CC2)nc1 18601,CN1CC(C)(C(N2CC(N(C)C(c3cc(C4CC4)no3)=O)C3(CC3)C2)=O)CC1=O 18602,C(=O)(C(CC(C)(C)C)N(C)C)NC(CNC(c1ccc(SC)s1)=O)C(C)C 18603,C(C(C)C(=O)NC(C)CNC(c1cnc(-c2ccoc2)s1)=O)OC 18604,c1(C(N2CCCC2)=O)cccc(C)n1.C(C(=O)NC(C)CN)=CCN(CC)CC 18605,CC(CC(=O)NCC(C1CCCOC1)NC(C1(CO)CC=CC1)=O)n1ccnc1 18606,C1(CNC(C(c2cccc(C)n2)(F)F)=O)CN(C(=O)C(C)(C)CC#N)CC12CC2 18607,Cc1cc(C#N)nc(=NCC2CC(C)N(C(c3cc4cccc(C)n4n3)=O)C2)[nH]1 18608,c1(CN(C(C)Cc2cccc(OCC(=O)O)c2)CC)ccc2c(c1)CC(=O)N2 18609,c1(C(=O)NC2CC3CN(C(c4ccnc(OC)n4)=O)CC32)cccc(S(C)=O)c1 18610,c1(C(=O)Nc2cc(-c3c(O)ccc(C)c3)ncc2)c(O)cc(O)cc1O 18611,Cc1cc(-c2cn(CC(N3CC(Oc4c[nH]nc4C4CCC4)C3)=O)nn2)ccc1F 18612,N1(C(Cc2c(C)cccc2)=O)C2CCCC1CN(C(c1sccc1C)=O)C2 18613,n1(CC)cc(Cl)cc1C(N1CC(C(C)NC(c2ccc(C#N)[nH]2)=O)C1)=O 18614,N1(C(=O)CCc2nnc(C3CC3)s2)CC2(CCN(C(C34CCCC3C4)=O)C2)C1 18615,c1(C(=O)NCC(C)N(C(c2cc(OCC)n[nH]2)=O)C)cc(C)c(Br)cc1C 18616,C1(C)(C(=O)NCC2(NC(C3CCCN(C)C3)=O)CC2)Cc2ccccc2C(=O)O1 18617,c1(C(=O)NCC(CC)N(C(=O)C=Cc2ccc(C)s2)C)ccc(=N)[nH]c1 18618,C12=CC(=O)NCCCN(CC1)CC2.C1(OC)CCC(C(=O)OC)C1 18619,C(C1(C)C(=O)C(CCCNCCF)C(C(=O)NCC=CC(C)(C)C)O1)OC 18620,N12CCC(CC1)C2.C(C)(CC(=O)NCCNC(c1ccc(C(C)=O)[nH]1)=O)OC 18621,C1(NC(CSCC=C)=O)CC2(CCN(C(=O)C=Cc3cncc(C)c3)C2)C1 18622,CCC(C)(CCNC(=O)CCCn1ccnc1)NC(=O)C(C)n1ccnc1 18623,c1(C(=O)NCC(C)CNC(C2(C(F)F)CCCO2)=O)ncccc1Cl 18624,c1(OC)ccc(F)c(F)c1-c1cn(CC(N2CCC(NC(C)=O)C2)=O)nn1 18625,C1(CNC(C2CCS(=O)(=O)CC2)=O)CC2CCC(C1)N2C(C1CCOC1)=O 18626,C1(OC)CN(C)C(C)(C(N2CCCCC(CNC(C3(O)CCCCC3)=O)C2)=O)C1 18627,C1(CNC(c2c(C)n(C3CC3)cc2)=O)CN(C(=O)C(C)SC(F)(F)F)CCCO1 18628,N1(C(C(COC)OC)=O)CC(NC(c2ccc(OC)c(Br)c2)=O)CC1(C)C 18629,Cc1cncc(C=CC(=O)Nc2cccc(OC3CCCC3)c2)c1.C1(=O)CN1C 18630,C#CCC(C)(C)C(=O)N1CCC(C)C(NC(c2cncc(C(C)C)c2)=O)C1 18631,c1(CC(=O)NC2CCC(C)N(C(=O)CC3CCOC3)C2)cccc2c1OCCCO2 18632,c1(OC)ccnc(C(=O)NCC(CCOC)NC(C2CC2CC(C)C)=O)c1 18633,C12(C(N3CCC(CN(C)C(c4csc(=N)[nH]4)=O)C3)=O)CC(C)(C1)OC21CCC1 18634,OC1COc2c(NCc3cc(Cl)sc3Cl)ccnc21 18635,C#CCC(C(=O)N1CCC(O)C1C)NC(=O)CSCCCC 18636,c1(C(N(CCCNC(C2CCN(CC(C)C)C2)=O)C)=O)cc(Cl)cc2c1OCC2 18637,C#Cc1cccc(CC(=O)NC2CCOC2C(N2CCNC(=O)C2CC)=O)c1 18638,C1(CNC(C2N(C)CCCC2)=O)CC2(CCC2)CN1C(=O)CC1C=CCC1 18639,Cc1ccnc(C(=O)NCC2(NC(=O)C=CS(C)=O)CCC2)n1 18640,C=C(Br)CCC(=O)NCC(C)CN(C)C(C1CC(=O)N(C)C1)=O 18641,c1(SCC(=O)NCC(=O)NC2(CC(=O)OC)CC2)nnnn1C 18642,C=CCCCC(C)(C)C(=O)N1CCC(NC(c2ccc(C)c(Br)c2C)=O)CC1 18643,C=CCN=C(NCC)NCc1ccc(C(=O)NC)nc1.C1CCCCS1 18644,N1(CC2(NC(CCOC)=O)CC2)CCN(C(C2OCCOC2C)=O)CC1 18645,c1(N(C)Cc2ccc(F)cc2)nc(N2CCC3(CC2)CSC3)nc2c1SCC2 18646,C(=O)(C(C)(C)CC(=O)OC)NCC(CC=C)NC(=O)C1=CCCCC1 18647,n1(C(OC)C2CC2)cnc2c(N(CCN3CCCC3)C3CC3)ncnc12 18648,c1(C(N2C(CNC(C(C)NS(C)(=O)=O)=O)CC2)=O)ccc(C2CC2)cc1F 18649,CC#CC1CCN(C(=S)NCCC2(NC(=O)OC(C)(C)C)CCCCC2)C1 18650,C#Cc1ccc(C(=O)NCC(CNC(c2ccsc2COC)=O)OC)cc1Cl 18651,c1(C(=O)NCCOCCCN(C(C(C)SCC)=O)C)ccc2cn(C)nc2c1 18652,C(=O)(C1CCCn2cnnc21)NC1C(CNC(c2cccc(C(C)C)c2)=O)C1 18653,CC(C)CC(CNC(C1CCC1C(C)(C)C)=O)NC(=O)CCCCC1CC1 18654,C(=O)(N(CCC(=O)N(C1COCCO1)CC1CC1)OC)C1N(CC)CCOC1 18655,c1(C(=O)NCC(C2CCN(C(c3c(C)coc3)=O)CC2)F)cccc(O)c1F 18656,Cc1ccc2oc(C(=O)NC3CC(CNC(c4cc[n+]([O-])cc4)=O)C3)cc2n1 18657,c1(C(N2CCC(N(C(=O)C(C3CC3)SC)CC)CC2)=O)cnc([N+](=O)[O-])n1C 18658,C(C(CNC(=O)CCOCC(F)(F)C(F)F)C(F)(F)F)NC(c1c(CC)ncs1)=O 18659,C(=O)(C#CC1(C)CCCO1)NC(C)CNC(c1cnn(C)c1C1CC1)=O 18660,CC1=NOC(C)(C(=O)NCC2(C(N)=O)CN(C(=O)CSC(F)(F)F)C2)C1 18661,C1(O)(CN(C)C(c2occc2C2CC2)=O)CCN(C(=O)CCOCCOC)C1 18662,CCCCS(=O)(=O)CC(=O)NCCNC(c1c(C)cccc1Br)=O 18663,CC(C(=O)OC(C)(C)C)C(=O)N(C)CCC(=O)CCc1cncn1C.C1CO1 18664,N1(C(C2(CC)COC2)=O)CCCC(CO)(NC(=O)Cn2ccc([N+](=O)[O-])n2)C1 18665,C1(N(C(C(c2cnn(C)c2)NC(C(CSC)O)=O)=O)C)CC2CCC1CC2 18666,N1(C(C(CCCC)NC(C2CC(N(C)C)C2)=O)=O)CCCC2NC(=O)CC12 18667,N1(C(c2ncc(OC)cn2)=O)CCC(NC(c2cc(C)c[nH]2)=O)C(C)(C)C1 18668,c1(C2C(C(=O)NCCCCNC(C(C)(C)OC)=O)C2)cc(F)ccc1F 18669,C1(C(=O)OC)CNC(=O)CN1C(=O)COC1CCN(C(=O)C(O)Cn2cncn2)C1 18670,C1(NC(c2c(C)nsc2)=O)CC2(C1)CN(C(=O)C(Cc1ccccc1)C(C)C)C2 18671,C1(NC(NCc2ccnc(C(C)(C)C)c2)=NCCF)Cc2nccnc2C1 18672,C1(CNC(COCCC#C)=O)CC(NC(=O)C(C)C2CCCC2)C1 18673,N1(C(Cc2ncn(C)c2)=O)CC(C(=O)NC(c2nc[nH]n2)C2CC2)C2(CC2)C1 18674,O=C(C#CC1CCCC1)NCC1(N(C(c2cc(N3CCCC3)ncn2)=O)C2CC2)CC1 18675,C(=O)(C1=CCC(F)(F)CC1)N1CC(N2CCN(C(CC(C(C)C)O)=O)CC2)C1 18676,Nc1cccc(C(=O)NC(CNC(=O)CCc2ccc(O)nn2)C2CC2)n1 18677,C1(CC)(NC(=O)NCCc2ccc3nsnc3c2)CCCCCCC1 18678,Cc1ncc(NC(C2CC3CC3N2Cc2cccc3ccnn23)=O)c(C)c1Br 18679,N1(C(C(F)=C(C)C)=O)CCOCC(C(=O)NCc2cc(F)ccc2F)C1 18680,Nc1c(C(N2CC3CC2CN3C(=O)CC2CC2(Cl)Cl)=O)ccnc1F 18681,CC1=CCC(C)(C(=O)NCC23CC(NC(=O)CN4CCC(C)C4)(C2)C(C)O3)CC1 18682,c1(CNC(=O)COCCNC(C2C3CCCC23)=O)ccnnc1 18683,C(C(C)(C)C(=O)N1CCC(O)(Cn2cc(-c3cnn(C(C)(C)C)c3)nn2)C1)SC 18684,C1(CNC(C(CC=C)OC)=O)CN(C(c2sc(C3CC3)nc2C)=O)CCN1C 18685,Cc1cc(C#N)ccc1C(N1CCC2(CC2C(=O)NCC23CC(F)(C2)C3)C1)=O 18686,CCCCCCCCC(C)CC(=O)N1CC=CC1CNC(c1ncncc1F)=O 18687,C#CC1CCCC(NC(=O)C(CNC(C2CC(COC)C2)=O)N(C)C)C1 18688,C1(CC#C)(CNC(C2(CO)CCCO2)=O)CCN(C(c2snnc2C2CC2)=O)C1 18689,C(=O)(C(C)CCCC(C)=O)N1C(CN(C(c2ccn(CC)n2)=O)C)CCC1 18690,N1(C(c2ccn(CCC)n2)=O)CCC(N=[N+]=[N-])(C(=O)NC2CC3(C2)CC(C)C3)C1 18691,N#Cc1cc(C(=O)NCC23CC(CN2C(=O)Cc2cncnc2)C3)co1 18692,c1(OC)ncccc1C(c1nnnn1C)NC(C1CCC1)C 18693,c1(C(=O)NC2C=CCN(C(Cc3n(C)ccn3)=O)C2)cccc2scnc12 18694,N1(C(CCCCC(CC)C)=O)CCC2(CCCCC2NC(=O)CCC2CC2)CC1 18695,C1(CC(C)C)CC(C(=O)NCCCNC(c2cc(=O)cc[nH]2)=O)CC(=O)N1 18696,C1(CCC(=O)NC(C(C)CO)C)CCN(C(=O)CCN2CCCCC2)CC1 18697,N1(C(c2cc(CC)nn2C)=O)C2CCCC1CC(NC(C1CC1(C)Br)=O)C2 18698,c1(C(N2CCCN(C(c3n(C)ncc3)=O)CCC2)=O)cc2nccc(Cl)c2s1 18699,N1(C(=O)NC(Cc2cccc(C)c2)C2CC2)CCCC(O)(c2cnn[nH]2)C1 18700,C12(NC(=O)CC3CCOCC3)CCCC1N(C(C1CC1(Cl)Cl)=O)CC2 18701,c1(CC)nccnc1C(=O)NCC1CCN1C(=O)C(=CC1CCCC1)C 18702,C(=O)(NNc1cccc(F)c1)N(C(CC)CN1CCOCC1)C 18703,CC1(C)CCCCC1NC(=O)CCCC1CN(CC(C)(C)C(=O)OC(C)(C)C)C1 18704,N1(C(CCCNC(=O)OC)=O)CC2(COC(CNC(=O)C(C)C)C2)C1 18705,S(=O)(=O)(c1ccc(N2CC(CO)C3(CCC3)C2)c(C#N)c1)N(CCSC)C 18706,c1(NCC(C)(C)NC(Cc2ccc(OC)cc2)=O)ccc(C#N)cc1[N+](=O)[O-] 18707,C1(N(C(C(C)=C(CC)C)=O)C)CC2CC1N(C(C1CCC(NC(C)=O)CC1)=O)C2 18708,C12(CC(=O)N(c3c(C)nsc3)C)CCC1CN(C(=O)CCc1ccnn1C)C2 18709,Cc1cc(Cl)cc(C(=O)NCC2(NC(C3CC(O)C3)=O)CCCC2)c1C 18710,C=CC(CCC)CC(=O)N1CC(C(=O)NCC2CCOC(C)(C)C2)C(F)(F)C1 18711,c1(OCCCC)cc(C)ccc1NC(=O)N(C1(CC)CC1)C 18712,C1(C(N(CCOC)CC2CC2)=O)COCCC1NC(C1CCC(C2CC2)C1)=O 18713,c1(C(=O)NC(CNC(C2CCC=CO2)=O)CO)ccc2ccc(Br)cc2c1 18714,c1(C(=O)NCC(CCCC)NC(=O)C(C)CF)ccc2n[nH]c(C)c2c1 18715,N1(Cc2c(N(C)C)ccc(Br)c2)CCC2CCCC2C1 18716,C1(NC(C2(CO)CCN(C(CCC=C)=O)C2)=O)CCN(C)C12CCC2 18717,c1(NC)ccc(C(N2CCC2CNC(=O)CCCC(=O)NC(C)C)=O)c(Cl)c1 18718,C1(C(N(CC#CC)CC#C)=O)N(C(c2conc2C)=O)CC12CCCC2 18719,CCC(CC(=O)N(C1CN(C(C2CC=CCO2)=O)CCC1O)C)C(C)C 18720,C(C)(N=c1[nH]c(N2CCC3(CCN(C)C3)C2)nc2ncn(C)c12)c1c(OC)nccc1 18721,Cc1nn(C(C)C)c(C)c1CC(N1CCCC(N(C(=O)CC#N)C)CC1)=O 18722,c1(CC)cc(C(=O)NC(CC)CC(=O)NCC2COCC2(C)C)ccn1 18723,C1(F)(C(N2CCC(N(C(=O)CC(C)(C)O)C)C2)=O)CCC(F)(F)CC1 18724,C1(CNC(CCSC)=O)CC2(CCN(C(c3cc(N)ccn3)=O)CC2)CO1 18725,C(=O)(CCCS(C)(=O)=O)N1CCN(C(C(C)NC(=O)NC)=O)C(C)C1 18726,c1(C(=O)NC(C2CCN(C(=O)CCc3ncc[nH]3)CC2)C)cc(Cl)cnc1O 18727,CCC(CCCC(=O)NCc1cc(C)cc(C)c1)NC(C1(Cl)CC1(F)F)=O 18728,c1(NC2(c3ccc(F)cc3)CC(C(=O)NCCC)C2)cnc(NC)c(Cl)c1 18729,c1(C(N2CC(C(=O)NC3(CC=C)CC3)C(C)(C)C2)=O)ccc2occc2c1 18730,Cc1cc(CO)oc1C(=O)NC1CCC(C)(CNC(C2(C(N)=O)CCC2)=O)C1 18731,CCC(C)(C)C(=O)N1CCOC(CCNC(=O)CCn2cncn2)C1 18732,N1(C(C2C(CC)CN(C(=O)C(C)(C)CO)C2)=O)CCCC(O)(C(N)=O)C1 18733,N1(C(c2c(OC)nsc2)=O)CCC(NC(c2sccc2Cl)=O)CC1 18734,N1(C(c2cc(C)cc(C)n2)=O)CC(C)CN(C(C2CCCCN2C)=O)C(C)C1 18735,n1(CCOC)cc(C(=O)N(CC(C)O)CCNC(=O)CC2CCCN2C)cn1 18736,c1(C(N2CCN(c3ccnc(C(C)C)n3)CC2)=O)cccc2ncccc12 18737,N1(C(C(N)Cc2ccc(F)c(F)c2)=O)CC2CCCC(O)C2C1 18738,O=C(C1=CCCOC1)NCCCCNC(C1CCCCS1)=O 18739,CC1CCC(C)(C(=O)NCCN(C(c2ccnc(OC(C)C)c2)=O)C2CC2)C1 18740,N1(C(C#C)C)CCN(C(=O)C(CCF)NC(c2cnncc2C)=O)CC1 18741,C(=O)(NNc1ncc(Cl)c(O)n1)C1CCCN(C(C)C)C1 18742,c1(C(=O)NCCOCCN(C)C(=O)OC(C)(C)C)cc(C(C)(C)C)[nH]n1 18743,Cc1cccc(C(=O)NCCCCCC(=O)NC(c2cn(C)cn2)C)c1N 18744,N1(C(CC2ON=C(C)C2)=O)CCC2C(CCN2C(=O)CC2CCOCC2)C1 18745,N#CC1(CC(N2CC3CC(NC(=O)CSc4nncs4)C3C2)=O)CCOCC1 18746,C1(C(=O)NC(C2CCN(C(C3COC(=O)O3)=O)CC2)C)CCSC(C)C1 18747,C1(F)(CNC(c2ccnc(O)c2)=O)COCCN(C(=O)C(O)c2ccco2)C1 18748,Cc1cc(C)c(C(=O)NC(Cc2ccoc2)C(=O)NCc2ccc(C#N)s2)s1 18749,C1(C(=O)NCCOC2CCC2)N(C(=O)CCn2cccn2)CC12CCCC2 18750,N1(C(CC(CCC)NC(C2COCC(C)O2)=O)=O)Cc2cccc(F)c2C1 18751,CC(C(=O)OC(C)(C)C)C(=O)NC1CN(C(c2cc(=O)n(C)o2)=O)CC1F 18752,C1(CNC(C2CCC(NC(c3cnn(CO)c3)=O)C2)=O)CCCC1C1CC1.C1CC1 18753,c1(C(=O)OC)ccc(C=CC(=O)NC2CCN(C(=O)C=CCOC)C2C(C)C)o1 18754,C(=O)(C1=CCOCC1)NC1CCCN(C(c2c(CSCC)cccn2)=O)C1 18755,C(=O)(CC(C(F)F)C(C)(C)C)NCC(CCNC(CNC(=O)OCC)=O)O 18756,Cc1cc(Cl)cc(C(N2CCCC2CNC(c2ncnn2C)=O)=O)c1O 18757,Cc1cc(NC2CN(C(=O)C(C)C(C)C)CC2C)c(C#N)cc1[N+](=O)[O-] 18758,C1(C(=O)NCc2n(CC)ncn2)CC=CC(NC(=O)C(C(C)C)SC)C1 18759,C1(NC(CNS(CC)(=O)=O)=O)CCCCC12CCN(c1nc(Cl)nc(C)c1Cl)C2 18760,c1(CCC(=O)NC2CN(C(=O)Cc3ccsc3)C2)cccc(F)c1 18761,c1(C(=O)NCCN(C(c2onc(CC)c2C)=O)C2CC2)cnc2cc(C)ccn12 18762,c1(C(=O)OC)ccc(CC(C)C)nc1N1CC2CC(NC(=O)CSC(F)F)C2C1 18763,c1(C(=O)NCCCCC2CN(C(C3C(C)CC3)=O)C2)cc(Cl)ccn1 18764,N1(C(c2c(C(C)=O)cn(C)n2)=O)CC2CC(N(C(=O)CCC(C)C)C)C1C2 18765,c1(OC)ccc(-c2ccnc(C(N3CCC(F)(Cn4ccnn4)C3)=O)n2)cc1.OC 18766,c1(C(=O)NC(C(C)NC(CCC(C)OC)=O)C)c[nH]c2cccc(C)c12 18767,c1(C(N(C(C)CNC(c2cccc(SC(F)(F)F)c2)=O)CC)=O)cc(C)n(C)c1 18768,CC1(C)CC(=O)NCC1C(=O)NCC1CCN(C(=O)COC(F)F)C12CC2 18769,c1(C(=O)NC(C(C)C)CCNC(C2(CCN(C)C)CC2)=O)nn(C)c(C(F)F)c1Cl 18770,C1(NC(C(C2CCN(C(c3c(CC)c[nH]n3)=O)C2)(C)C)=O)C2CCCCC12 18771,c1(N(C)CC2CCC(O)C2)nccc(=NCCOc2ccccn2)[nH]1 18772,C(=O)(CCCCCCCSC)NCC1(NC(Cc2ncn(C)c2)=O)CC1 18773,c1(OC)ccnc(Cl)c1CCC(N1CC(c2ccccc2)OCC1C)=O 18774,c1(C(N2CCC(C3CCCN3CC3CC(=O)C3)CC2)=O)ccc2ccncc2c1 18775,N1(c2ncc(C(=O)OCC)nc2)CCCC2(CC(NC(=O)C(C)C3CC3)C2)C1 18776,C1(NC(c2ccc(C(C)(C)C)cn2)=O)CC2CC(NC(=O)C3=CCCS3)CC12 18777,C1(NC(CNC(CN(C)C)=O)=O)CCOC12CCN(C(=O)CC(F)(F)F)CC2 18778,C=CCCCC(=O)N(C1CCC(NC(C2(COC)C=CCC2)=O)CC1)C 18779,c1(C(=O)NC(CC)(CNC(=O)C(C)C(C)(F)F)CC)cc2c(s1)CCC(C)C2 18780,C(=O)(C(C)CC(F)F)NC(C(=O)N(C1CC1)CC1(OCC)CCC1)Cn1cncn1 18781,N1(C(C2C(OC)CCC2)=O)CCc2[nH]nc(CNC(=O)CC3(OC)CC3)c2C1 18782,C1(NC(=O)C=CC=C(Cl)Cl)CN(C(c2cnc3n2CCC3)=O)CC12CCC2 18783,Cc1csc2ncnc(N3CCC(NC(=O)C(c4ccc(F)cc4)O)C(F)C3)c12 18784,C(=O)(CC(N)OCC)NCc1ccccc1.C1(C(N(CC#C)CC)=O)CC1C(=O)N 18785,C1(C)(C(F)F)CC(=O)NNC(=O)N1.CC(C)(C)OC(=O)NCCOC1CC1 18786,N1(C(Cc2c(C)cnn2C)=O)C2CCC(C2)C1C(=O)NOC1CC1 18787,CCCC(C)CC(=O)N(CCNC(c1ccncc1C1CC1)=O)C(C)C 18788,CCN=c1[nH]cc(C(N2CCC(C)C(CNC(C3(C)CC3)=O)C2)=O)s1 18789,CC1C(NC(c2cncc(Br)c2)=O)CCN1C(c1cnc(C(N)=O)s1)=O 18790,Nc1nc2ncccc2cc1C(=O)NC1CC(F)(CNC(=O)Cc2nc[nH]n2)C1 18791,N1(c2nc(N3CCCC(c4cc[nH]n4)C3)cc(C)n2)CCc2occ(CO)c2C1 18792,Cc1nc2cccc(CN(C)Cc3cc(Cl)ccc3-n3ccnn3)n2n1 18793,c1(C(N)=O)cccc(C(N2CCOCC2CNCC(F)(F)F)=O)c1F 18794,C(=O)(C(F)(F)CCC1CC1)NC1C(CNC(C(=O)N(C)C)=O)C1 18795,S(=O)(=O)(c1ccc(NCc2ccco2)c(Br)c1)NC(C)CS(C)=O 18796,CC1CC(C(=O)OCCCCF)CCN1C 18797,S(=O)(=O)(c1ccc(Cl)c(C(=O)NCC(c2ccccc2Cl)O)c1)NCC 18798,N1(C(C2C(=C)CC2)=O)CCN(C2CCN(C(=O)Cc3ccc(C(C)=O)s3)C2)CC1 18799,c1(C(=O)NC2CN(C(c3scc(C)c3Cl)=O)C(C)C2)cc(N)cnc1C 18800,C(CC(C(=O)N1CCC(NC(=O)CC2CCCC23CC3)C1)OC)OC 18801,C1(NCc2cnc(C(F)(F)F)[nH]2)CCN(c2ccccn2)C1=O 18802,C(CC(=O)NC(C1(O)CN(C(=O)C(=O)NC(C)C)C1)C)(C(F)(F)F)OC 18803,Cc1nsc(N)c1C(C(=O)NC1CC1)=O.C1(C(=O)NCCN)CCCCC1(C)C 18804,C(=O)(C1=NNC(=O)CC1)N1CCCC(C(=O)NCc2nccc(C)c2)C1 18805,c1(N(CCOC)C)ccc(CNC(C2CCN2C(C2CC(O)CN2C)=O)=O)cc1Cl 18806,C1(O)(CN(C)C(c2cncnc2)=O)CCN(C(c2ccc(C3CC3C)o2)=O)C1 18807,C(=O)(C1=CC2(CN(C(=O)CC3CCCC(O)C3)C2)OC1)NC(c1ccnn1C)C 18808,c1(C(C(N2CCN(c3ncc[nH]3)CC2)=O)F)ccccc1I 18809,CC1(C)COc2ccc(C(=O)NCCC3(O)CN(C(=O)C4=CCCC4)C3)cc21 18810,N(C1CCCc2ccc(F)cc21)C(=O)NNC(=O)C(F)C1(O)CCC1 18811,C(=O)(C(C)CC(F)(F)F)NCc1c(C(=O)NCC2(CC)CCCO2)cco1 18812,C1(NC(C2CCC(C)C2)=O)CC2CC(C1)N(C(=O)CCCCCN(C)C)C2 18813,c1(OC)ccc(C(c2ccc(C)s2)NC(Cc2ccccc2)C2CC2)cc1Br 18814,c1(C(=O)NCC2(C(=O)NC3CC(C)OC3=O)CCCO2)cn(C)c(=O)cn1 18815,c1(C(N(C(CN(C(C(C)NC(C)(C)C)=O)C)C)C)=O)ncc(F)c2ccccc12 18816,C1(C(=O)NCc2ccn(C3CC3)n2)CCCN1CCCO 18817,c1(OC)cc(C(=O)NC(C)CC2CN(C(C)=O)C2)ccc1O.C1(C=O)CCNC1=O 18818,C(=O)(C#CC1(C)CC1)NCC1C(NC(CS(=O)(=O)NCC)=O)CCC1 18819,c1(C(=O)NC(C)(CNC(=O)C(F)CC2CC2)C2CC2)cc(CC2CC2)ccc1F 18820,N1(CC)CCOC(C(=O)NCCCCCN(C(=O)C(C2CC2)OC)C)C1 18821,c1(C(=O)NCC(C)C(=O)NCC2CC3C=CC2CC3)ccc2n[nH]cc2c1 18822,N1(C(c2c(OC)cccn2)=O)CCc2ccccc2C1CNC(c1ccc(C)s1)=O 18823,c1(C(=O)NCC2CC(NC(c3c(CC)ocn3)=O)C2)cc(C)c(C)o1 18824,Cc1ccc(F)c(O)c1C(N1CC2CC(NC(C3CCCCC3)=O)CC2C1)=O 18825,C1(NC(c2cnc(C(C)O)s2)=O)CC(C)N(C(=O)Cc2cnn(C)c2C)C1 18826,C1(C(=O)NCC(C)(C2CC2)NC(c2cc(F)cc(Cl)c2)=O)CCC(=O)NC1=O 18827,C1(F)(CNC(Cc2cc(CC)no2)=O)CCN(C(=O)CC2NC(=O)NC2=O)CC1 18828,C1(C(N2C(C=C)COCC2)=O)CC12CCN(C(C1(C#N)CCOC1)=O)CC2 18829,C12(CC(N3CC(C(=O)N(CCCO)C4CC4)OCC3)=O)CCCN1CCC2 18830,N1(C(C#CC2(CC)COC2)=O)CCCC(C2CCN(C(=O)C(F)=C(C)C)CC2)C1 18831,C1(NC(c2ncc(NC)nc2)=O)CCN(C(c2csc(C3CC3)n2)=O)CC1C 18832,C1(C(=O)NC(C(C)(C)C)CNC(=O)C(N)=O)CCn2c(O)nnc2C1 18833,c1(C(C(=O)NC(C)CC)N(C(C)COC)CC=C)ccc(OC)c(Br)c1F 18834,C1(NC(c2c(CC)con2)=O)CC2CC(NC(C3CC(C)C3)=O)C2C1 18835,CC1(C)CC(N=c2ccnc(C(F)(F)F)[nH]2)CN(C(c2cccnc2O)=O)C1 18836,N1(C(c2cc(C(C)=O)[nH]c2)=O)CCC2CCN(C(=O)CN3CCC3C)CC12 18837,C(C(C)(C(=O)N(C)Cc1cc(C)n(C)n1)NC(C1CCC(C)(C)C1)=O)SC 18838,C1(NC(CCOC)=O)CN(C(c2sc(Br)nc2C)=O)CCC1CO 18839,Cc1nc(-c2noc(Cc3c[nH]nc3C)n2)nc(O)c1F 18840,c1(OC)ccc(NC(c2nnnn2CC(F)F)(C)CC2CCOC2)c(OC)c1 18841,C12CC3CC(CC13)C(=O)N2.C1(NC(C(CN(CC)CC)F)=O)COCCOC1 18842,c1(C(N2C(C)CCC(NC(C(C)=C(CC)C)=O)C2)=O)cc[nH]c2nccc1-2 18843,C1(NC(C(=O)NCC#CC)=O)CCCN(c2ccccc2C)C1 18844,C1(NC(C(CSC)O)=O)CC2CCC1N2C(c1ccc(Cl)cc1N)=O 18845,Cc1cccc(COCC(=O)NC2CC(F)(NC(C3(C(=O)N(C)C)CC3)=O)C2)c1 18846,N1(C(C(C(C)C)(F)CNC(=O)CC2CCC(C)(C)O2)=O)CCn2ccnc2C1C 18847,C#Cc1ccccc1CC(N1CCC(N(C(=O)CC2CCC(C)O2)CC)CC1)=O 18848,C1(NC(CC(C)CF)=O)CC2CN(C(c3cc(Cl)n(C)n3)=O)CC2C1 18849,c1(C(N2CC(CC(C)NC(c3n(CC)cc(Cl)c3)=O)C2)=O)cc(C#N)cn1C 18850,c1(CC(C(=O)NC2CN(C(c3cc(COC)sc3)=O)C2)O)cc(Cl)cc(Cl)c1 18851,N1(C(c2c(CC)nc(C)o2)=O)CCC2(CC1)CCN(c1nnc(C#N)s1)CC2 18852,Cc1cnc(C(N2CCC(NC(C3CC3C(N)=O)=O)C(O)C2)=O)cc1Cl 18853,n1(CC)nncc1C(=O)NCc1cc[nH]c1C(=O)NCCOCC(F)(F)F 18854,c1(OC)cc(F)c(C(N2CC(NC(C3CC3C)=O)CC3(CC3)C2)=O)c(F)c1 18855,C1(C(N(C(C)C(N2CC[Si](C)(C)C2)=O)CC)=O)CCCC(C#N)C1 18856,Cc1ccc(C(N)=O)cc1OCC1CCCN(C)C1.n12cc(nn1)C(=O)NOCC2 18857,CCC(CC(C)C)C(=O)N1CC2CCC1C(CNC(=O)C(C)NS(=O)(=O)CC)C2 18858,N1(C(C(CCC)n2cc(-c3cccs3)nn2)=O)CCCN(C(=O)C=CBr)C(C)C1 18859,N1(C(c2ccc(OC)s2)=O)CC=C(C(=O)N2CCC2C(N)=O)C1 18860,c1(C(=O)NCC(C)(C(C)C)NC(C(CCSC)NC(C)=O)=O)ccc(O)nc1C 18861,C1(CC(=O)NCC(C(C)C)(C)NC(c2c[nH]c(=N)s2)=O)CCCC(C)(C)C1 18862,c1(OCCC)cccnc1C(=O)NCC1CCCCN1C(C12CCC(CO1)C2)=O 18863,N1(C(C(n2cc(Cl)cn2)C)=O)CCC2(C)CN(C(C3CCC4CC34)=O)CC12 18864,CC1(C(=O)NCc2cn(CC(=O)Nc3ncccc3Cl)nn2)CC2CC2C1 18865,C12(c3cn(CC4CCC(NC(C(CCC)O)=O)CC4)nn3)CCCN1CCC2 18866,c1(CNC(=O)NCC2OCCC2F)ccc(Cl)cn1 18867,C1(C(=O)NC2(CO)CC(F)(F)C2)CC12CCN(C(=O)CC1CCCSC1)C2 18868,c1(NC(C(C)C)=O)ccc([N+](=O)[O-])cc1C(N1CCN(c2ccncn2)C2CC12)=O 18869,C(=O)(C1=CC(C)(C)C1)N1C(CNC(c2ncc(N(CC)CC)nc2)=O)CCCC1 18870,Cc1ccc(=O)n(CC(N2CCN(C(c3ccc(C)c(C)n3)=O)C(CO)C2)=O)n1 18871,N1(C(C(C(CC)O)C)=O)CCC2(CCN(c3nnc(C(C)(C)C)s3)C2)C1 18872,N1(C(c2c(C)c[nH]c2)=O)CCN(C(C2(c3ccccc3F)CC2)=O)CC2(CC2)C1 18873,CCCS(=O)(=O)C(C)C(=O)N1CC(NC(c2nnc(O)nc2O)=O)C(C)(C)C1 18874,C1(C(N(CC(C)C#N)CC)=O)CC2(CC2)CN1C(=O)CSC 18875,C1(NCC(C)NC(CCNC(=O)NC)=O)CCCN1C(=O)C(C)(C)C 18876,N1(C(C2C(COC)CC2)=O)C2CCC1CC(N(C(=O)Cc1cn(C)nn1)C)C2 18877,C#Cc1ccc(Cl)c(C(=O)NC(C)(CNC(=O)CNC(=O)CC)C2CCC2)c1 18878,C(=O)(CC(C)CNCC(C(=O)C(c1ccnn1C)O)=O)N(C1CCNC1=O)CCC 18879,Cc1nc(N2CC3(CCC(NC(=O)Cn4cc(Cl)cn4)CC3)C2)c2ccsc2n1 18880,c1(-c2cn(-c3ccc(CC(=O)NCC=CBr)cc3)nn2)ccc(C2CC2)cc1F 18881,S(=O)(=O)(c1cccnc1N(C)Cc1ccc(F)cc1)N1CC(C)C(CO)CC1 18882,c1(C(=O)NC2C(NC(CCCC)=O)C2)cnn(CC)c1C(F)(F)F 18883,C(=O)(C1=NOC2(CCN(Cc3cccc(OC)c3Br)C2)C1)OC 18884,c1(CNC(CCC(=C)C)=O)nc2c(s1)CCN(C(=O)C(CCC)N(C)C)C2 18885,C12(C(=O)NCC(C)(CO)NC(c3c(OC)scc3)=O)CCCC1C2(F)F 18886,c1(C(=O)OC(C(=O)OC)c2cccs2)ccc(C=O)c(C)c1 18887,C(=O)(C(C)(C)CCNC(C1CC(C)(F)C1)=O)NC(C(=O)OC(C)C)C 18888,N1(C(CCCC(=O)c2cccs2)=O)CCCC2(CCCN2C(C2CC2F)=O)C1 18889,c1(C(=O)NC2C(CNC(CC3C(C)(C)CCCO3)=O)C2)scc2c1OCCO2 18890,C(=O)(C#CC1(CC)CC1)NC1CN(C(CN(S(CC)(=O)=O)C)=O)CC1O 18891,C1(S(N)(=O)=O)(C(=O)NCC2CC(CNC(CCOC)=O)OC2)CC1 18892,CCC(CC(=O)NCCC(C)(C)NC(=O)CS(=O)(=O)N1CCOCC1)SC 18893,c1(COC(C)C(=O)NCC2CC2NC(=O)CSS(C)(=O)=O)ccccn1 18894,C1(CS(Oc2ncnc3ncc(Br)n32)(=O)=O)CCC2(CCOCC2)CO1 18895,C1(C(N2CC(C3CN(C(C(C=C)O)=O)C3)C2)=O)CCc2c(C)nnn2C1 18896,C(CC(=O)NC(c1cnn[nH]1)(C)C)(CC(C)C)NC(c1c(CC)n(C)nn1)=O 18897,Cc1cnc(NC(CC2CC2)CO)c(S(=O)(=O)NCC2CCC(C)(C)O2)c1 18898,C1(C(=O)NC2(CF)CCN(C(C(C(C)C)NC(C)=O)=O)C2)CN(C)CCN(C)C1 18899,N1(C(c2cncc(C)n2)=O)CC(CNC(=O)Cc2ccc(F)cc2)CC(C)C1 18900,C#CCCCCCCC(=O)NCCN(C(C1(S(C)(=O)=O)CCOCC1)=O)C1CC1 18901,c1(CC(=O)N(C(C)CN(C(=O)C(F)CC2CCOC2)C2CC2)C)cncnc1O 18902,C(=O)(C1Cc2ccc(Cl)cc21)N1CC2CCN(C(c3cn(CC)nc3)=O)C2CC1 18903,c1(C(CNC(C2(C)CCCS2)=O)NC(=O)CN2CCOCC2)ccc(F)cc1F 18904,C#CCCN=C(NCCc1ccc(C(C)(C)O)cc1)N1CCC(SC)C1 18905,C1(NC(COCCC=C)=O)CCN(Cc2nnc(-c3ccco3)o2)CC1C 18906,N1(C(c2c(C)cc(=N)[nH]c2)=O)CC(C)N(C(=O)C(=O)Nc2ncc[nH]2)CC1C 18907,C1(C(=O)NCC23C(CN(C(c4ccc(C)o4)=O)C2)C3)CN2CCN1C(C)C2 18908,CC1CN(C(C2(F)CCCCC2)=O)CCN1C(c1ccc(-c2cn[nH]c2)nc1)=O 18909,Cc1ccncc1C(=O)NC1CCC(CNC(C2OCCC2C)=O)C1 18910,C1(C(=O)NC(C(C)NC(=O)CSCC(N)=O)C)(CF)CCOCC1 18911,c1(OC)cc(C#N)ccc1NC(c1cc(-c2cnc3[nH]ncc3c2)[nH]n1)=O 18912,CC(C)(O)CC(=O)NC1CCC(N2CCN(C(=O)C=Cc3cc[nH]n3)CC2)C1 18913,CN1CC2(CCN(C(C3CCN(C(C4CC4c4ccccc4)=O)CC3)=O)C2)C1 18914,C1(NC(C=C(C)C)=O)CC(CNC(c2cc(-c3cnn(C)c3)no2)=O)C12CCC2 18915,C1(C(F)(F)F)(C(N(C)CC2CCCN2C(=O)CN2CSCC2=O)=O)CCCCO1 18916,Cc1ccc(C)c(C2=NOC(C(=O)NC3CCC(NC(=O)CC4=CCC4)CC3)C2)c1 18917,c1(C(=O)Nc2ccc(-c3c(C)nn(C)c3)s2)cccc([N+](=O)[O-])c1N1CCCC1 18918,C1(=CC(=O)NC(C)CC(C)NC(=O)COC2CCCOC2)CCC(C)(C)CC1 18919,c1(-c2nnc(C(N(CC(=O)C(c3ccc[nH]3)C)C)C)o2)ccc(C)cc1 18920,C1(CC=C)(C(=O)NCCC2(C)CC2(F)F)CCCN1C(C1CCC1C)=O 18921,CC(C)CC(C(N)=O)NC(=O)CC(CNC(C1CC2CC(=O)C1O2)=O)C1CCC1 18922,C1(C(=O)NCC(C)(C)C)(NC(CCC2N(C)CCC2)=O)CCN(C)C1 18923,Cc1cc(C(=O)NCC(C)(C(C)C)NC(c2nn(C)cc2C)=O)n(C(C)(C)C)n1 18924,C1(C(N(CCC(=O)NCC(CC)C)C)=O)CCC2CC12 18925,C1(C(N(CC(C)C)CCCCl)=O)CN(C(=O)C(c2ccc(Cl)cc2)=O)CC(C)O1 18926,C(=O)(C(F)(F)C(F)F)N1C(CN(C)C(C2CC2c2ccc(F)cc2F)=O)CCC1 18927,c1(C2(C(=O)NCC(CNC(C(COC)C)=O)C)CCOCC2)ccc(Cl)cc1Cl 18928,C(CCCCCCC(=O)NC(C)C(C)NC(c1cnn(CCO)c1C(C)C)=O)SC 18929,CCC(CC(=O)N1CC(C(C)C)C1)NC(=O)Cc1ccc(C)cc1 18930,CCC(C)(C#N)C(=O)NC1CN(C(=O)CSC(F)F)CC1c1ccc(OC)cc1 18931,N1(C(C(C(C)C)C(C)NC(c2cncc(O)c2)=O)=O)Cc2cccc(F)c2C1 18932,C1(C(=O)NCc2cccc(CNC(C3(C)CC3)=O)c2)(OC)CCOCC1 18933,CCC(O)CC(=O)NCC(C)NC(C1(NC(C)=O)CCC1)=O 18934,c1(C(N2CCCCC(CNC(COC(C)=O)=O)C2)=O)n[nH]c2ccccc12 18935,N1(C(C(C)NC(CC)(C)C)=O)CC2(C1)CN(C(c1cc(O)cc(F)c1)=O)CCO2 18936,n1(CCCNC(c2cc(CNC3CCCC3)on2)=O)cc(C(=O)O)nn1 18937,c1(C(N2CC(OCC)(CNC(C3CC3Cl)=O)C2)=O)cccc2nsnc12 18938,C(C(O)C(=O)NCC1CC(NC(C2CCC(C(N)=O)O2)=O)C1)SC 18939,C1(OC)(CNC(=O)C(N2CCOCC2)C)CN(C(=O)C=C2CCOCC2)C1 18940,c1(-n2cc(C(C)N(C)C(C3(C)CC3F)=O)nn2)c(F)cccc1Cl 18941,c1(C(C)C)ccc(NC(=O)C(F)C2CC(NC(C3(F)CC=CCC3)=O)C2)cn1 18942,c1(C(N(CCN(C(C(F)=CCC)=O)C)C)=O)ccc(-c2nnnn2C2CC2)cc1 18943,N1(N2C(CC=O)CC(O)C2)CCC2(CCC(O)C2)C1.CC1(C)OCCC1C=O 18944,c1(C(=O)NC(CN(C(c2ccc(CCC)s2)=O)C)C)cnc(OCC)cn1 18945,C1(C(N2CC(CNC(C(CC)(C)O)=O)(COC)C2)=O)CC(C)CC(=O)N1 18946,c1(C(=O)NCCC2CSCCN2C(=O)CC2C=CCC2)cccn2ncnc12 18947,Cn1cc(I)c(C(N2CCCC(C3CCCC3)C2)C(=O)NC2CCOCC2)n1 18948,c1(C(=O)NC(C)CCNC(c2cc(O)n(C)n2)=O)cnn2cc[nH]c12 18949,CC1CN(C)CCC1N(C)C(C1(NC(C2CC3(CCC3)C2)=O)CCC1)=O 18950,c1(C(=O)NCCC2CCCN(C(=O)CC(F)(F)F)C2)ccn2ccsc12 18951,N1(C(c2cccc(-c3c(OC)nccc3)c2)=O)CC(C)(C)c2ccccc21 18952,C1(NC(CN(C(C)=O)C)=O)CCCN(C(c2cc(CC(C)C)[nH]n2)=O)CC1F 18953,C1(C(N2CC(CNC(CCCCOC)=O)(COC)C2)=O)CC2CCCN(C1)C2 18954,c1cc2occc2s1.c1(CN(C)C)ccc(F)cc1.C12CCN(C1)C(=O)NC2 18955,N1(C(c2ccc(C#N)s2)=O)CC(NC(=O)CC2COCCO2)C2(CCOCC2)C1 18956,CC(O)CCCC(=O)N1CCCC1C(C)(C)N(c1cnccc1Cl)CCO 18957,c1(CN(C(=O)C(c2ccccc2)C)C(C=C)C)ccc(F)cc1F 18958,C1(CNC(C(CCC)=CCC)=O)CCN(C(c2cn(C)c(=O)n2C)=O)CC1(F)F 18959,CCCCC(O)CCC(=O)N1CC(C)(C)CC1CNC(c1cnc(C)cc1C)=O 18960,C(=O)(C(C)CCOc1ccccc1)N(CC(C)NC(=O)CCCc1cccnc1)C 18961,N1(C(CCC(=O)NC)=O)CCOC2(C1)CN(C(c1onc(Br)c1C)=O)C2 18962,N1(C(c2c(C(=O)OC)cco2)=O)CCN(C(C2(C)CCCS2)=O)CC1c1cn[nH]c1 18963,N1(C(c2cccc(SCC)c2)=O)CC2CCN(C(C3CCC4CC34)=O)C2C1 18964,N1(C(Cc2c(C)n(C)nc2)=O)CCN(C)C(CNC(=O)COC2CCC2)C1 18965,C1(NC(C=Cc2nc(C)sc2)=O)CCC(O)CN(C(=O)CCc2nc[nH]n2)C1 18966,c1(CC)cc(C(=O)NCC2COCCN2C(C2CCC(=O)N2)=O)cn(C)c1=O 18967,Cn1c(C(=O)NC2C3CC2CN(C(=O)C(F)C2CCOC2)C3)cccc1=O 18968,C1(C(=O)NC2CON(CC)C2=O)CN(C(C2(C)CCCN2C)=O)C(C)(C)C1 18969,C1(CCCC)CCC(C(N2CC(F)(C(=O)N(C3CCCC(O)C3)C)C2)=O)CC1 18970,N1(C(c2cc(C(C)(F)F)ccn2)C(=O)NCC)CCOc2ccc(Br)cc2C1 18971,c1(C(C)C)ncsc1C(=O)NCC1CCN(C(=O)C(F)(F)Sc2cnn(C)c2)C1 18972,CCC1CC(=O)C(=O)C(C)(CNc2ccccc2)O1.NC 18973,N1(C(COC2CCN(C(C3(C)CCOCC3)=O)CC2)=O)CC=C(C(=O)O)C1 18974,C(CCCCC(=O)NCC1CC=CCO1)N(C(C(C1CC1)OCC)=O)C 18975,N1(C(C(CC=C)NC(=O)C(C)(C)N=[N+]=[N-])=O)CCCCCCC1C 18976,N1(C(CCOCC(C)C)=O)CCC(C)(NC(C2CCC2SC(F)F)=O)C1 18977,O=[N+]([O-])c1cc(CNS(=O)(=O)CC2CC3CC3C2)cc(N2CCOC2=O)c1 18978,C(c1ccccc1Cl)=CC(=O)NCCCC(C)(C)NC(c1nc(C(C)C)sc1)=O 18979,N1(Cc2nc(C(C)C)sc2)CCC(NC(c2cccnc2N)=O)CC1 18980,c1(C(N2CCC(N(C)C(C3CC(C)(C)CN3C)=O)CC2)=O)nccc2[nH]ccc12 18981,N1(C(c2c(C)cncc2)=O)CCN(C(=O)C(C)Oc2cccc(O)c2)CC1C 18982,c1(OCC(=O)N(CCC)CCNC(=O)C=Cc2ccsc2)ccccc1OC 18983,Cc1nc(C(N2CCC(C)(NC(C3CC4C=CC3C4)=O)C2)=O)c2ccccn12 18984,CC1C(=O)N(CC(=O)NC2CC(O)(CNC(c3cncs3)=O)C2)C(=O)C1C 18985,C(=O)(C(O)CCn1cncn1)N.C(C(=O)N(CCCOCCOCC)C)=CC=CC 18986,c1(C(=O)NC2CCN(C(C3C4COCC34)=O)CC2F)cc2ccccc2[nH]1 18987,C1(CNC(C(C)=C(C)C)=O)CCN(C(C2CNC(=O)N2)=O)C12CCC2 18988,c1(OC)ccc(CO)cc1C(=O)NC1CC(O)CN(C(=O)Cc2cnn(C)c2)C1 18989,c1(-c2cc(CC(=O)N(C(COC)O)C)ncc2)ccc(OC)c(F)c1 18990,CCC(C)C(C(=O)Nc1cn(C)nc1C#N)NC(c1ccc(COC)cc1)=O 18991,CC1CN(C(c2ccc(Cl)cc2)=O)CCC1CNC(C1OCCOC1C(F)(F)F)=O 18992,CC(C)C(CNC(c1ccnc(CO)c1)=O)C(=O)NCC(C)(O)C(C)(C)C 18993,C#CCCCCCCC(=O)NC(C1CCN(C(=O)CSC(C)(C)C)CC1)CO 18994,N1(S(CC(C)C)(=O)=O)CC2(CCN(C(c3ccn(C(F)F)n3)=O)C2)C1 18995,c1(C(=O)NCC2N(C(C(C)n3cccn3)=O)CC(O)C2)cncc2ccccc12 18996,C1(C(N2CCN(C(C(C(=O)OCC)(C)C)=O)CC2CC)=O)CCn2ncnc2C1 18997,N1(C(C(C)(F)F)=O)CCOC2(CCN(C(=O)C=Cc3c(F)ccc(Cl)c3F)C2)C1 18998,N1(C(c2cnccn2)C(=O)NCCCC)CCC(C(N)=O)C(CC)C1 18999,c1(N2CC3C(N(C)C)C3C2)nc(=NCC2(C3CCC3)CC2)[nH]c2c1SCC2 19000,N1(C(C=CC=CCC)=O)CCC(C)(CC(=O)NC(C)(C)CCOC)C1 19001,C(C(=O)NC1COCC1NC(c1cc(C)ns1)=O)(C(C)C)n1ncc(C)c1 19002,c1(C(N(CCC(N2CC(C(CC)CC)C2)=O)C)=O)cn(CC)cn1 19003,CN1CC(C)(C)CC1C(N1CC(C(=O)NCC2CCCCCCC2)CC1(C)C)=O 19004,N1(C(C(C)SC(C)C)=O)CC2(C(=O)NC3CC4(CCC4)C3)CCC1CC2 19005,c1(C(C(=O)OCC)=O)cccnc1C(=O)NCCCCCNc1cc(Cl)cn1C 19006,N1(C(C)=O)CCC(CNC(c2coc(CC3CCCC3(F)F)n2)=O)CC1 19007,c1(CC(=O)NCC(C)CNC(=O)C(F)CC2CCCC2)cnc2c(=O)[nH]ccn12 19008,c1(NCCCCCC(C)O)cc(=NCC(c2ccsc2)N(C)C)[nH]cn1 19009,c1cc(Br)cnc1Cl.c1(C(=O)O)c[nH][nH]c1=NC(=O)C1(CC(=O)OC)CCCC1 19010,C1(C(=O)NCC2(CCNC(C=C(COC)C)=O)CC2)CCNC1=O 19011,CCC(C)(C)C(O)C(=O)NCC#CCNC(C1CCC2(CC1)CC2)=O 19012,C1(OCC)CC2CN(C(=O)C(CNC(=O)CCCNC(C)=O)CC3CC3)CC12 19013,c1(C(=O)NC(c2ccccc2I)c2ccccc2)ccc2c(c1)COC2 19014,N1(C(C(C)n2cccc2)=O)CC2CC1(C(=O)NC1CCOC1(C)C)C2 19015,C(=O)(C(C)CS(C)(=O)=O)NC1C(NC(c2ccc(-c3nc(C)on3)cc2)=O)C1 19016,C1(NC(C2CN(C(CNC(C)=O)=O)CC23CCC3)=O)CCc2cnn(C)c2C1 19017,c1(C(N2CCC(N(S(C)(=O)=O)C)C2)=O)cc(F)c(F)c(F)c1 19018,C(=O)(C1=CCCN(Cc2ccc(Cl)c(I)c2)C1)Nc1cc(C(=O)OC)cc(F)c1 19019,c1(CN(C)Cc2cc[nH]c3nccc2-3)cccc2ccccc12 19020,C1(C(C)(C)NC(COCCC=C)=O)CCN(C(=O)C(C2CCCCCC2)C)CC1 19021,c1(C(N(CCCCNC(CCC=C=C)=O)C)=O)cc2c(C)c(F)ccc2[nH]1 19022,N1(C(C(C(C)C)C)=O)C2CCC1CN(C(=O)Cc1cnn(C)c1)CC2 19023,c1(C(=O)NC2CCN(C(C(F)=C(C)C)=O)CC2)ccc2nnc(C3CC3)n2c1 19024,N1(C(CC(CNC(=O)C#CC(C)(C)O)OC)=O)CC2(CCNC(=O)O2)C1 19025,C#Cc1ccc(C(=O)N(CCC(C)NC(C2CCC(NC(C)=O)CC2)=O)C)cc1 19026,c1(SC)ccccc1CC(=O)NC1(CNC(C2CC3CC3C2)=O)CCCCC1 19027,N1(CC(=O)N(CC(=O)NC(C2CCC2)C2CCC2)C)CCNC(=O)C1 19028,c1(C(=O)NC(CNC(c2cn(CCOC)nn2)=O)C(C)C)nccc(C#N)c1F 19029,Cn1c(C(=O)NCC2C(O)C(O)CN2C(C2CC2(C)C)=O)cc2ccsc12 19030,C1(C(=O)NCc2nnnn2C2CC2)N(C(c2cn(CCO)nn2)=O)CC12CCCC2 19031,C(=O)(CC(C)P(C)(C)=O)NCC(CNC(c1c(CC)c[nH]c1)=O)C(F)(F)F 19032,C(c1cc(Br)cs1)=CC(=O)NC1(CC=C)CN(C(C2CC2(C)C(F)F)=O)C1 19033,c1(N(CC(=O)N(C2CCC(NC(=O)C3CC3)C2)C)C)cccc(C#N)c1 19034,N(C1COc2ccc(Cl)cc21)C(C1C2CN(C(C(c3ncccn3)C)=O)CC21)=O 19035,Cc1ccc(F)c(C(=O)NCC(=O)NCC(=O)NCCCS(C)(=O)=O)c1 19036,C(C)(CCCCNC(=O)CCc1cccc(Br)c1)NC(c1cnc(C)o1)=O 19037,C(CCCCC(=O)Nc1nc[nH]n1)=CCCC.c1(CC2CCC2)ccccc1F 19038,C(=O)(CCS(=O)(=O)CC(C)C)N1C(CCNC(C(C)SCCCC)=O)CC(OC)C1 19039,c1(C(=O)NCc2cc(C(=O)OCC)[nH]c2)nc(C)nn1C.C1(C=O)(C)CC1 19040,c1(C(CC)NC(=O)NC2CCCN(C(=O)NC)C2)cc(C)ccc1Br 19041,C1(C)(NC(Cc2c(CC)con2)=O)CCN(C(=O)CCC(F)F)CC1 19042,c1(C(N(C)CC2CCCC(NC(c3csc(S)n3)=O)C2)=O)c[nH]nc1[N+](=O)[O-] 19043,c1(OC(C(=O)NC2CC(NC(C3N(CC)CCC3)=O)C2)C)cccc(F)c1 19044,CCCC(C)(O)CC(=O)N1CC2(C1)CN(c1ccc([N+](=O)[O-])cc1)C2 19045,N1(C(c2ccc(C)o2)=O)CCN(C(=O)C=CCN2CCCC2)C(CCO)C1 19046,N1(C(C=CC2CCN(C(C(COC)OC)=O)CC2)=O)CCCC(N=[N+]=[N-])C1 19047,c1(C(N2C(COC)CN(C(=O)C(F)C3CC3)CC2)=O)cc(C)c(C)cc1C 19048,c1(C(C(=O)NCCSC)N(c2cc(OC)ncc2)C)ccc2c(c1)OC(C)(C)O2 19049,N1(C(c2ccc(C(C)C)nc2O)=O)CC2CCCC2(Nc2ccnc3ncnn23)C1 19050,c1(OCC(CNc2nccc(C)c2I)O)nc2ccccc2o1 19051,c1(C(N2CCCC(CNC(C(F)=CCC)=O)C2)=O)cc(C)cc(OC)c1O 19052,C12CCCCC1(C(=O)C1CC1)C(=O)N2.C(CCCN(CCC(=O)OC)CC)OCC 19053,O=C(C1=NOC(CO)C1)N1CCC(CF)(NC(=O)C(F)(F)c2cccnc2)C1 19054,C12(C(N3CC(C(C)NC(C45CCN(CC4)CC5)=O)C3)=O)CCCCC1C2(F)F 19055,c1(C(=O)O)ccnc2c1CCN(CC1CCCNCC1)C2 19056,C(=O)(C1CCCn2nccc21)N1C(C)(CNC(CC2CCCN(C)C2)=O)CCC1 19057,CCC(CC(C)C)C(=O)NCC(C)(CNC(c1cc(CF)on1)=O)OC 19058,C12(CNC(c3cc(C)c(C)o3)=O)CCCCC1CN(C(c1cccn1C)=O)C2 19059,C#CCCCCCCC(=O)NCC1(O)CCN(C(=O)CCC2CCCCC2)CC1 19060,C(CCCCC(=O)NC(CNC(c1ccncc1C)=O)c1cccs1)OC 19061,N1(C(c2c(C)[nH]nc2C(F)(F)F)=O)CC2CCN(C(C3CC3F)=O)CC(C2)C1 19062,C1(CCC)CCCCN(C(C2CC3(CC(NC(=O)OC(C)(C)C)C3)C2)=O)C1 19063,c1(N(C2CN(C(=O)C(c3ccc(F)c(Cl)c3)O)C2)C)cccc(F)c1Cl 19064,N1(C(Cc2cnc(C)s2)=O)CC2(CCC2NC(=O)CC2CCCC(=O)N2)C1 19065,Cc1nc(C(=O)NC2CC2NC(c2ccnn2C(F)F)=O)cs1 19066,c1(C(C)C)ccc(C(N2CC(NC(C3(N(C)C)CC3)=O)C(n3ccnn3)C2)=O)nc1 19067,c1(C(N2CCC(C3N(C(CC(=O)OCC)=O)CCC3)C2)=O)cncc(N)c1C 19068,n1(CC)nc(C(=O)NCC2COC(CNC(c3sncc3C)=O)C2)cc1O 19069,c1(-c2cnc(CC(=O)Nc3c(Cl)ccc(C(C)=O)n3)nc2)cccc2[nH]ncc12 19070,N1(C(C2(OC)CCC(C)(C)C2)=O)CCC2(CC1)CC2NC(=O)C=Cc1ncc[nH]1 19071,CC1(C)CCC(C(=O)NCCc2ccncc2)(NC(C2CCCC(C#N)C2)=O)C1 19072,C1(N(CC#C)C(c2nncn2CC)=O)CCN(C(=O)C(C)Cn2cccn2)CC1 19073,N12CC3CCC1CN3C(=O)CC2=O.c1(C(=O)OCCC)cc(CCCO)on1 19074,C1(C2(O)CCOCC2)(C(N2CC(F)(CNC(c3c(CC)onc3)=O)C2)=O)CC1 19075,C1(C(=O)NC2C(CNC(CCC(=O)NC)=O)CCC2)CC(C)OC(C)C1 19076,CCC(C)CCC(=O)N1CC(O)CC1C(=O)NCC1(CCCO)CC1 19077,c1(C(=O)NCC(C(=O)NCC(COC(C)C)O)CC2CC2)cnn(C)c1C#N 19078,C1(CCC)CCCC1CNC1(COC)CC(C)C1 19079,c1(OCC)cc(C#N)ccc1NC(c1ccc(C)cc1C)C 19080,C1(NC(C2(NC(C)=O)CCCC2)=O)CCCN(C(C2CC(=O)NC(=O)C2)=O)C1C 19081,Cc1n[nH]c(C)c1C(=O)NC(Cc1ccc(F)cc1)CC(=O)NCC1CCOC1 19082,c1(C(N(C(CNC(=O)CC2CCSCC2)C2CC2)C)=O)cc(Cl)cnc1O 19083,c1(OC)ccc(CC(=O)NC2CC3(C2)CN(Cc2cc(Cl)ccc2O)C3)c(F)c1 19084,c1(CC)[nH]c(C(=O)NC2(C)CC(NC(=O)C(C)(O)CC)C2)nc1Cl 19085,Cc1ccc(F)c(C(N2CC3CC2C3NC(=O)CC(C)(C)c2ccccc2)=O)c1 19086,C1(C)(NC(CCOC)=O)CCCN(C(C2OCCO2)=O)C1 19087,N1(C(C2CSCCN2C(=O)COCC2CCCO2)=O)CCc2ccccc2C1 19088,c1(CC(=O)OC)cccnc1N1CCCC(NC(C2CC2C2CC2C)=O)C1 19089,N1(C(C(C)Oc2ccccc2Cl)=O)CC2OC(=O)N(C3CCN(C(N)=O)C3)C2C1 19090,Cc1c(-n2nc(C3CC34CC4)nc2C2CC(C(C)C)=NO2)cc(Cl)cc1Br 19091,c1(C(N2CC(O)CC(NC(C(=Cc3cccs3)C)=O)C2)=O)cn2cc(C)nc2s1 19092,C12CCC(CC1)C(=O)NCC2.C(C)(C(=O)NCC1(C(C)C)COC1)OCCOC 19093,c1(C(N(CCCNC(C2(C)CC(=C)C2)=O)C(C)C)=O)ccnc(C2CC2)c1 19094,N1(C(c2ccc(C)n2C)=O)CCN(C(c2n[nH]cc2F)=O)C(CS(C)(=O)=O)C1 19095,C(C#CCN=c1cc(C)c(S(=O)(=O)NC(C)Cc2ccccn2)c[nH]1)OC 19096,O=C(N=c1[nH]nc2[nH]ccnc1-2)C12CC1CN(Cc1nc(Cl)ccc1Cl)C2 19097,C1(OC(C2C(C)CN(C3CC4CC3C4)C2)=O)CCCCCCC1(C)C 19098,C(=O)(CCCC(F)F)NC(C1CCCCN1C(=O)Cc1cscn1)C 19099,c1(CC)ccnc(C(=O)NCC#CC(N2CC[Si](C)(C)C2)=O)c1 19100,N1(C(c2c(CC)scc2)=O)CC2CC(C1)CN(C(=O)C(C)(C)CC)C2 19101,N1(C(=O)OC(C)(C)C)CCC2(CCC(C(=O)NCCSC3C=CCC3)CC2)C1 19102,C1(C(N2CCOC(c3cccs3)C2)C(=O)NCC(C)C)CC2(CCCO2)C1 19103,NS(=O)(=O)N1CC(C(=O)NC(CNC(C2CCN(C3CC3)S2(=O)=O)=O)C2CC2)C1 19104,c1(CC)noc(C(=O)N(C2CN(C(c3cn(CC)nc3C)=O)C2)C)c1C 19105,C(=O)(C(C#N)N)Nc1ccccc1.C1(C(=O)NCCN(C(=O)CO)CC)CCCO1 19106,C1(CNC(CCCC=C)=O)CN(C(C2(NC(C)=O)CCCC2)=O)CCCO1 19107,c1(C(=O)NCC(C2(O)CN(C(C(C)OCC)=O)C2)(C)C)ccc(Cl)c(F)c1 19108,C12CCC(=O)N(C1=O)C2.c1(CN(CC(C)OC)C)cnccc1C 19109,N1(C(c2ccc(CO)o2)C(=O)NC(C(=O)OC)C)CCC(C)(C)C(CO)C1 19110,CC1CC(C)(C)N1C(=O)C=CC1CCCN1C(=O)Cc1cccc(O)c1 19111,c1(C(=O)NCC(C)N(C(Cc2cc(COC)on2)=O)C)ccn2c1CCCC2 19112,C1CCCCC(N2CC(OC)CC(O)C2)C1=O.C1(C)(CCNC(C)C)CC1.CO 19113,CC(c1ccccc1)=CC(=O)NCC1CC(NC(c2ncccc2F)=O)C1(C)C 19114,C1(NC(=O)C=Cc2ncc[nH]2)COC2(C1)CN(C(C1CCCCC1O)=O)C2 19115,C(=O)(C(C(C)C)NC(C)=O)N1CCC(OCCNC(C2(C)CC(=C)C2)=O)C1 19116,N1(C(c2c(CC)oc(C)c2)=O)CCN(C(=O)CC(C)(F)F)C2CCCCC2C1 19117,c1(SC)ccc(C(=O)NC2CCN(C(=O)CCS(C)=O)C2C)cc1[N+](=O)[O-] 19118,CCC(C)(CC)C(=O)N1CCN(C(c2sc(C)nc2C)=O)C(CC(F)(F)F)C1 19119,C1(CC)CN(C(=O)C(=O)NCC2(C)CCCOC2)CC(=O)N1 19120,c1(C(=O)NCC23N(C(C)=O)CC(COC)(C2)C3)cc(OC)c(O)c([N+](=O)[O-])c1.CN 19121,N1(C(C2C(C(N)=O)C2)=O)CCC(C(=O)NC2CC(C(N)=O)C23CCC3)=C(F)C1 19122,c1(C(N2C(CNC(CC(CC)CC)=O)C=CC2)=O)cn(CC#N)c2ccccc12 19123,N1(C(c2cccs2)=O)CCN(C(C2CCC3(CCC3)C2)=O)C(C(F)F)C1 19124,CC1CCC(CO)N1C(=O)C(O)CCNC(=O)Cc1cscn1 19125,C1(N(C)C(c2cnc(-c3ccoc3)s2)=O)CCN(C(c2ccncc2O)=O)CC1 19126,Cc1c(C(=O)NC2CCC(CNC(c3ncc[nH]3)=O)C2)cnn1CCO 19127,Cc1nc2c(C)cc(C(=O)NCC3C4CN(C(C5CC5F)=O)CC34)cn2n1 19128,c1(C(N2CC(C)C(NC(c3c(F)ccc(O)c3F)=O)C2)=O)cccc(S(C)=O)c1 19129,C1(C(=O)NC(CCCNC(Cc2ccc(COC)cc2)=O)C)CC(F)(F)C1(C)C 19130,N1(C(CC)=O)CCC2(CCC2)C(NC(=O)CC(C)(O)C2CC2)C1 19131,CCC(CC1CCCC1)C(=O)N1CC(COC)(NC(=O)Cc2nonc2C)C1 19132,c1(C(N2CC(CN(C(C(C(C)OC)O)=O)C)C2)=O)cn2ccccc2n1 19133,CC1COC(C(=O)NCc2ocnc2C(=O)NC2(c3ncc[nH]3)CC2)C1 19134,C(=O)(CCCCCC#N)NCCC1CCCN(C(c2c(C)noc2C(F)F)=O)C1 19135,C(=O)(C1CCCc2c(O)cccc21)NC1CC(NC(=O)CN2CCCS2(=O)=O)C1 19136,C1(CC(=O)NCCC(C)N(CCC)C)CCN(C(c2cscc2C)=O)C1 19137,c1(CNCc2ccc(F)nc2)c(F)cc(Cl)cc1Cl 19138,C1(C(C)(C)C)(CNC(C(C)Cc2ccncc2)=O)CCN(C(=O)CSC(C)(C)C)C1 19139,N1(CCC#C)CCN(C(=O)C(CCF)NC(=O)CC2CCCN2C)CC1 19140,C(=O)(CC(C)(C)C)NC(C1CCN(C(c2cnc(C(C)C)[nH]2)=O)CC1)C 19141,[N-]=[N+]=NCCCCCC(=O)OCC1CCCC(F)C1 19142,C1(NC(C2CC2CNC(C2C(C)(C(F)F)C2)=O)=O)CC2(CCC2)C1 19143,CCC(CC)(C(=O)NCc1cncc(C(=O)Nc2cccc(O)c2)c1)OC 19144,CCCC(O)(CCC)CC(=O)N1CC(C)N(C(c2ccccc2)=O)CC1C 19145,N1(C(CN(CCCOCCC(C)C)CC)=O)CC(C(N)=O)C2(CC2)C1.C(=O)(COC)NC 19146,C(=O)(C(CCC)c1ccc(Cl)cc1)NCC(C1CC1)NC(C=CCCC)=O 19147,C#CC1(C(=O)NCC(C)(F)C(C)C)CCN(C(=O)CNc2ncccn2)C1 19148,C1(N(c2ncc(Br)nn2)C(=O)C(O)O)CC2CCC(C1)N2 19149,C(=O)(C(F)C1=CCCCC1)N1CCC(CCN(C(=O)COCC2CCCC2)C)C1 19150,c1(NC(C(C)C)C2CC2)nc2ccccc2nc1NCC1CCC(C)(C)O1 19151,C(=O)(NNc1ccc([N+](=O)[O-])cc1Br)Nc1cn(C)nc1-c1cccc(Cl)c1 19152,C(c1ccoc1)=CC(=O)N(C(C)C(=O)NCc1[nH]nnc1C)CC 19153,C1(NC(C(c2ccccc2)NC(C2CCC(=C)CC2)=O)=O)CCCC(C)(C)C1 19154,c1(C(=O)NCC(CC)C(n2ncc(C(=O)N)c2)=O)coc(C2CC2)n1.C1CC1 19155,C(=O)(CC(Cc1ccccc1)NC(N1CCC(SCc2csc(C)n2)C1)=O)OC 19156,C(CC1CC1)(C(=O)NC(C)C)NC(CSCC=C)=O 19157,C(CCCCCNC(=O)C(n1cnnc1)NC(=O)CC1(C)CCOC1)OC 19158,C(C(C(C)C)NC(c1ocnc1CNC(=O)CCNC(N)=O)=O)OCC 19159,C(=O)(C(CC)N(C)C)NCC(CC)NC(=O)CC1(CNCC)CC1 19160,C=C(Br)CCC(=O)NC(CCN(C)C(C1(c2cc[nH]n2)CCC1)=O)C(C)C 19161,c1(C(C)=O)cc(C(=O)NC(CNC(c2cc[nH]c2C)=O)C2CCC2)cs1 19162,C(CCSC)(C(=O)NC(C)(C)C(C)NC(=O)COCc1cccnc1)OC 19163,c1(C(=O)NCC(C)(CO)NC(c2nc(Br)c[nH]2)=O)c(F)cc(F)cc1F 19164,Cc1cc(C(=O)NC2C3CN(C(c4cc(C)ccc4F)=O)CC23)cc([N+](=O)[O-])c1 19165,c1(C(C)C)nc(NCCCC2CC2)cc(=NC2CCC3CC2C3(C)C)[nH]1 19166,CN1CC(NC(C23CC(CN(C(C4(C)C=CCCC4)=O)C2)C3)=O)C2(CC2)C1=O 19167,CC1=C(C(=O)N2CC3=C(C2)CN(C(c2c(C)ncn2C)=O)C3)C(=O)OC1(C)C 19168,C(CC(C)C(=O)NCC1(CC(=O)NCC(C)(C)C(F)F)CC1)OC 19169,c1(C(=O)NC2CC(OC)C23CC3)cccc(CCCOC(C)C)c1F 19170,C1(CNC(c2ccn(CC)n2)=O)(NC(C2CCCCCC2C)=O)CCCCCC1 19171,CC(CC(=O)N1CCCCC(N(C(=O)CN2C(=O)CCC2=O)C)C1)C(F)(F)F 19172,C1(NC(C(C)S(C)(=O)=O)=O)CCN(C(=O)CC2C=CS(=O)(=O)C2)CCC1CO 19173,CC1CC(NC(c2cc(N)ccn2)=O)CCN1C(=O)CC1CCCN(C)C1 19174,CCC(C(=O)OC)C(=O)N1CCN(C(=O)CCOCC(F)(F)F)C(CO)C1 19175,c1(C(=O)NC2(c3ccccc3)CC2)csc(-c2cnn(CCNC3CCC3)c2)n1 19176,N1(C(c2cc(Cl)no2)=O)CCCC(C2CCN(C(=O)Cc3cscn3)CC2)C1 19177,c1(C(=O)NCC2C(COC)C2)ncccn1.C(=O)(C1CC1)N 19178,CCCC(C)CCNC(C1CCOCC1NC(C1CC1OC(C)=O)=O)=O 19179,Cn1c(C(=O)NCC(C2CCN(C(=O)CO)CC2)O)cccc1=O 19180,c1(C(N2CCCC2=O)C)ccc(OC(=O)Cn2cc(Cl)cn2)cc1 19181,C(=O)(C(C(C)(C)C)n1cc(C)nn1)N.CS(=O)C1CN(C(N2CCOC2=O)(C)C)C1 19182,CCC(C)(COC)C(=O)NC1CCCC(CNC(c2cccc(NC)n2)=O)C1 19183,c1(NC(Cc2nccc(C(C)C)c2)=O)ccc2c(c1)CCC2N(C)C 19184,C12(NC(=O)Cc3csnn3)CC(NC(=O)Cc3nnc(O)s3)(C1)C2 19185,C1(C(=O)NCC(CCOC)NC(=O)C(C)(C)C(N)=O)CC12CCCCC2 19186,Cc1ccc(C(=O)NC2CC(N(C(=O)CC(C)C3CC3)C)C2)c(O)c1C 19187,C(=O)(C1=NOC(c2ccccc2)C1)NCC(C)NC(c1csc(Cl)c1)=O 19188,c1(OC)c(C(=O)NC2CC3(NC(=O)C#CC4(C)CC4)COC2C3)cccc1F 19189,c1(OCCOC)ccc(CC(F)(F)F)cc1S(=O)(=O)N(C(C)C(N)=O)C 19190,Cc1nc(-c2cccs2)ccc1C(=O)NCC1CN(C(=O)C(C)(C)O)CC1C 19191,C(CCN(C)C)(CN=c1[nH]c(=NCc2csc(C#N)c2)[nH]c2cc[nH]c12)OCC 19192,N1(C(CSCC#N)=O)CC2CN(C(=O)Cn3nc(Cl)ccc3=O)CC2C1 19193,c1(C(=O)NCC(C)N(S(CC)(=O)=O)C)ccc(CCNC(=O)OC(C)C)cc1F 19194,C1(C(=O)NCCCOC=C)CCCN1NC(=O)C(CCC1CCC1)NC(C)=O 19195,C1(C(=O)NC2CN(C(c3ccc(C)cc3)=O)C(C)CC2)CC2(C1)CC1(CCC1)C2 19196,C(=O)(CCC(=O)NN(C)C)N1C(CNC(c2ncn(C(C)C)c2)=O)CC(O)C1 19197,N1(C(C2N(CC(C)C)CCC2)=O)CCOCC(NC(=O)C(C)N(C)C)C1 19198,CC(C)C(C(=O)NCC(C1CCCC1)NC(=O)CC1CC1)Oc1cccc(Cl)c1 19199,c1(C(=O)NC(C(C)C)CCN(C)C(c2coc(Cl)n2)=O)cc(F)ccc1N 19200,c1(C2C(C(=O)Nc3c(C)cnc(C(C)(C)C)c3)C2)cccc(Cl)c1[N+](=O)[O-] 19201,C1(CC)CN(C(C2C3CC4C(C3)C24)=O)CCN1C(c1cnn(CC2CC2)c1)=O 19202,N1(C(c2c(C)cc(C)nc2)=O)C2COCC1CC(NC(C1CCCC(C)C1)=O)C2 19203,c1(C(=O)NCC2N(C(C(C)CC3CC3)=O)CCC2)ccn(C(=O)OC(C)(C)C)n1 19204,C1(NC(c2cnc(F)c(Cl)c2)=O)CCC2CCN(C(c3nocc3Cl)=O)C1C2 19205,Cc1ccc(Cl)c(C(=O)NCC2CC2NC(=O)Cc2ccc3c(c2)CCO3)c1N 19206,C1(C(=O)N(C)CCN(C)C(C23CC(CC(F)F)(C2)C3)=O)(OC)CCS(=O)(=O)C1 19207,C12(C(=O)NCCC(C)N(C(=O)C(C)OCC3CCCO3)C)C=CC(CC1)C2 19208,N1(C(C=CC(C)(C)NC(c2c(C)n(C)nn2)=O)=O)CCC(C)C2(CCC2)C1 19209,C1(C(C)NC(C(C)OCCCC)=O)CCCN(C(c2cccs2)=O)C1 19210,c1(C(=O)NCCN(C2CCCCC2)C(C(C2CCOC2)OC)=O)c(C)ccn1C 19211,C1(NC(C2CCC=CCCC2)=O)CCC2CN(Cc3ccncc3Cl)CC2C1 19212,C(CN=c1nc(-c2cccs2)[nH]s1)NC(CCOCCCOC)=O 19213,c1(C(N(CCN(C(=O)Cc2ccc(F)cc2F)C)C)=O)ccc(F)c2[nH]ccc12 19214,N1C(=NCC#C)NCC1.C1(C2CN(C(CC)(O)CC)C2)CCN(c2nccs2)CC1 19215,C1(CCC)CCC(NCC2CCC2C(F)F)CC1 19216,c1(OC)ccc2cc(C(=O)NCC3CN(C(=O)C(C)S(C)(=O)=O)CCO3)[nH]c2n1 19217,C1(C(=O)NCCCN2CC=CC2)(NC(C(C)n2cccn2)=O)CCN(C)C1 19218,c1(NCC2CC(C)SC2)cc(N2CCOC(c3ccco3)C2)ncn1 19219,CC(C)C(C(C)NC(=O)CCc1ccc[nH]1)NC(c1sccc1C(C)(C)C)=O 19220,C=CC1COCC1NC(=O)C(c1ccoc1)NC(=O)C(C)(C)CC 19221,c1(N(CCNC(C(C2(O)CCC2)OC)=O)CC2CC2)n[nH]cc1C(C)C 19222,N1(C(C2CCC(CC)CC2)=O)CCCC2(CCC2NC(=O)Cc2cnn(C)c2)C1 19223,CCCCCCCCC(=O)N(CC(O)CNC(=O)C(C)OCc1ccoc1C)C 19224,c1(CS(=O)(=O)NC(C(C)N(c2scc(C)n2)C)=O)cccnc1Cl 19225,N1(C(COCCSC)=O)CC(O)CC1CNC(=O)CCc1ccc(C)s1 19226,c1(CC(=O)NCCCOCCCNC(C(CC(=C)C)C)=O)cccc([N+](=O)[O-])c1 19227,C1(C(=O)Nc2c(C)scc2)CCCC(CNC(=O)C(CO)N(C)C)C1 19228,c1(C(=O)NCC(CC)(CC)NC(CSCCCC)=O)cncc(S(C)(=O)=O)c1 19229,c1(COC)cc(C(=O)NC(C)(C(=O)NCCCCCN(C)C)C2CCC2)no1 19230,N1(C(C(CC)F)=O)CCC(C)C(NC(c2ccn(C3CCC3)n2)=O)C1 19231,C1(NC(c2cc(C)c(C)o2)=O)CCC2CC1CN2C(c1coc(CO)c1)=O 19232,C1(O)(CNC(C(C)OCCOC)=O)CCCN(C(c2ncccc2N)=O)CC1 19233,C(=O)(C(F)C(F)(F)F)NCCCCNC(CC(=O)Nc1c(C(C)O)cccc1)=O 19234,C(=O)(NNc1cc(F)cc(F)c1F)NCC(C(C1CC1)OC)(F)F 19235,CC1CCN(C(c2cc(CNC(=O)CC3=CCCC3)no2)=O)CC1(C)C 19236,C12(CNCC(O)Cc3ccccc3F)CCCC1CCC2 19237,N1(C(CCNC(COC)=O)=O)CCN(C(C2CCC3(CCC3)C2)=O)CC1CCO 19238,S(=O)(=O)(c1cccc(=NCC2(C3CCCO3)CCC2)[nH]1)NC(CC)CN(C)C 19239,CCC(CC)C(=O)N1CC(NC(C2(Cc3cccc(F)c3)CC2)=O)C(C)C1 19240,C(=O)(CCC(CC)CC)NC1CCC(CC(NOCCCC=C)=O)C1 19241,C(=O)(C(C)C(C)(F)F)N(CC(C)NC(c1n[nH]c(C2CC2)c1Br)=O)C 19242,Cc1cc(C)c(C(N2CCCC3(NC(C4CCC4)=O)CC3C2)=O)c(Cl)n1 19243,CN1CCN(C(c2cccnc2)=O)CC1C(=O)N(C1CCCC1)C1CC1 19244,N1(C(CC(C(C)C)C)=O)CC2CCC1C(CNC(c1c(C(N)=O)cnn1C)=O)C2 19245,Cc1ccccc1C(=O)NCC(=O)N(C(C)C)C(C)C.C12CCCN1C2=O 19246,c1(C(=O)NCC2(C(=O)NCc3ccc(C)[nH]3)CCCCC2)ncc2ccccn12 19247,Cc1noc(C2CC(NC(C3(C#N)CC3)=O)C2)n1 19248,C1(N2CCC(NC(c3c(C(C)C)ncs3)=O)C2)CCN(c2ccnc(Cl)n2)CC1 19249,CS(=O)(=O)CCC(=O)N1CCC(C2CCCN2C(c2ccoc2Cl)=O)CC1 19250,C1(NC(C2CSC(C(F)(F)F)C2)=O)CN(C(c2c(OCC)cccc2)=O)CCC1F 19251,C(=O)(C(C)CN(C(=O)C(Cc1cc[nH]n1)NC(=O)CCn1cc(C)cn1)C)NC 19252,C(=O)(C1=C(C)OCCS1)NC1CC2CN(C(c3nn(C(CC)C)c(C)c3)=O)C1C2 19253,C(=O)(C(F)CCC(C)C)NC12C(NC(C3OCCN(C(C)=O)C3)=O)CC(CC1)C2 19254,C12(C(N3CCC(C)(NC(=O)CCN4CCOCC4)C3)=O)CC1CCC2(F)F 19255,C1(C(=O)NCC2(NC(c3c(OC)scc3)=O)CC2)CCCC(C(N)=O)C1 19256,N1(C(C#CC(=O)N(C)C)=O)CC=C(CCNC(C2(F)CCS(=O)(=O)C2)=O)CC1 19257,C(=O)(C1=CCCCC1)N(CC(CC)NC(c1cccc(-c2cccs2)n1)=O)C 19258,CCCC(CCCNC(=O)C(C(C)O)NC(=O)OC(C)(C)C)OCC 19259,CS(=O)c1cccc(C(N2CCN(C(=O)CCn3cnnn3)C3CCC23)=O)c1 19260,C(CC(C)(C)C)(C(=O)NC(C)(CSC)C(=O)NC(C)COC(C)C)OC 19261,c1(C(=O)NCC(C)CNC(=O)Cc2cc[nH]n2)ccc2c(n1)NCC2 19262,C1(NC(=O)CSC(F)F)CCCN(C(c2ccc(Cc3cn[nH]c3)cc2)=O)CC1 19263,c1(CC)ncc(S(=O)(=O)NCc2c(C)[nH]c(C(N)=O)c2C)n1C1CC1 19264,c1(C(=O)NCCC2(C(=O)NC(C#C)C(C)OC)CCCC2)c(C)cccc1O 19265,C1(NC(c2c(CCC)nns2)=O)CN(C(=O)C(C)S(N)(=O)=O)CC12CCC2 19266,N1(C(C(CC)CC)=O)CCC2(CC(NC(=O)CCCN(C)C)CO2)C1 19267,C1(NC(CNC(CC2(NC(=O)CSc3nc[nH]n3)CC2)=O)=O)CCC2CC1CO2 19268,c1(CCC)nc(C)cc(=NC(=O)c2ccn3ncc(I)c3n2)[nH]1 19269,Cc1cc(C)c(CC(=O)NCC2(F)CC(NC(=O)CCn3cc[nH]c(=O)c3=O)C2)s1 19270,c1(C(C(=O)NCCCSC)N(CC2=CCSC2)C)ccc2nn[nH]c2c1 19271,C#CC(CNC(=O)C(C1CCOC1)NC(c1ccc(C2CC2)o1)=O)CC1CC1 19272,c1(OC)cccc(C)c1C1(NC(c2cc(OC(C)C)ccc2F)C)CC1.CO 19273,C#Cc1cn(C)nc1C(=O)NC(C)CC(=O)N(CC(N)=O)CC(N)=O 19274,c1(C(=O)NCC2C(NC(c3c(=O)cc(C)[nH]c3)=O)CCC2)ccc(F)c(Cl)c1F 19275,N1(C(C(C)NC(=O)NC)=O)CC2CC(NC(c3ccnc(C)c3Cl)=O)C1C2 19276,Cc1nc2ccc(C(=O)NCCNC(=O)CCC3CCCCC3)cc2n1C 19277,N1(C(C2C(C=C)C2)=O)CCCC(CN(C(=O)COCc2ncc(C)o2)C)C1 19278,N1(C(CC(C(C)C)OCC)=O)CCC2CCN(C(C3(SC)CC3)=O)CC2C1 19279,C1(C(=O)NC(COC)C)CC12CCN(c1ncccc1C)CC2 19280,CC(C)(C)CC(O)CC(=O)N1CC(CNC(=O)C=Cc2cscn2)C(C(F)(F)F)C1 19281,C(=O)(CCCCCCN=[N+]=[N-])NCC1CCCN(C(C(OC)OC)=O)C1 19282,C1(CC#C)(C(=O)NCCC2CC3C=CC2C3)CCCN1C(C1C2CC3C(C2)C13)=O 19283,N1(C(C(C)OC(C2CC(C(=O)OCC)C2)=O)=O)CC(O)CC1c1cccs1 19284,C1(NC(CC2ON=C(C)C2)=O)CCN(C(c2cnccn2)=O)CC1CO 19285,N(C(C)S(=O)(=O)c1ccc(F)cc1)(CC(=O)O)C(c1c2c([nH]n1)CC(C)CC2)=O 19286,c1(OC)ccc(C)c(C(N2CCSCC2C(=O)NCCN2CCNC2=O)=O)c1 19287,C1(NC(CCCNC(N)=O)=O)CC(C(=O)NCCCN2CC=CC2)C12CCC2 19288,Cc1cc(N)cnc1-c1noc(CC2CC2)n1.C12N(CC1(C)C)C2=O 19289,C(=O)(C1=NNC(C(F)(F)F)C1)NCC1CCC(NC(CC2(OC)CC2)=O)CC1 19290,Cc1cnc(C(N2CCC(NC(c3cc(F)c[nH]3)=O)C(CO)C2)=O)c(C)c1 19291,CC(C)(CNC(=O)NCCC1CC(O)C1)CCO 19292,CC1(C#CC(=O)NCC2(O)CN(C(=O)COc3cc(F)cc(F)c3)C2)CCCO1 19293,C(=O)(C(C)(C)C(C)C)NCC(CNC(Cc1ncc(C)s1)=O)O 19294,C(CCCCCNC(C1CCCN1C)=O)NC(C(F)=CCC)=O 19295,C(=O)(CCCCC(=O)N1CCC(C)N(C(C2CCCN(C(N)=O)C2)=O)CC1)NC 19296,CC1CC(=O)NC(C(=O)NCC2(CNC(c3nocc3C3CC3)=O)CC2)C1 19297,N1(C(c2cnc(O)c(F)c2)=O)CCC2CN(C(c3cc(Cl)ccn3)=O)CCC2C1 19298,N1(C(C(CCOC)C)=O)CC(CNC(c2cccc3scnc23)=O)CC12CCC2 19299,C12CCCN(CC1)C2.C1(NC(C(C)OC2CCCC2)=O)CC(=O)N(C2CN(C=O)C2)C1 19300,c1(C(=O)OCC(=O)N(CCCC(C)O)CC)nc(C)ncc1Cl.C(CCF)O 19301,N1(C(Cc2c(C)noc2Cl)=O)CCCC(N(C(=O)C(F)CC2CCCC2)C)CC1 19302,C12(C(=O)NC3CCN(CC)C3=O)CC(CCO1)N(C(=O)Cc1cc(C)cs1)C2 19303,C(=O)(CC(=O)NC(C)CNC(=O)C(C)C1CC1)NCC 19304,N1(C(C2(CCCC)CC2)=O)CC2CCCC(N(C(=O)C(CC)NC(N)=O)C)C2C1 19305,CC(C)CC(C)CC(=O)NC1C2CC1N(C(=O)C1=COCCO1)C2 19306,CC1CCCC(C(=O)NCC(N2CCOCC2CO)=O)C1C 19307,CC1CN(C(c2cnsc2)=O)CC(CCNC(c2ncc[nH]c2=O)=O)O1 19308,C(=O)(CC(F)(F)C(F)F)NCC(C1CCCCC1)NC(C(C)NC(CC)=O)=O 19309,C12(C(N(CCCNC(C3CC3C(C)C)=O)CC)=O)CC3CC1C2C3O 19310,N1(CC(=O)N(c2nnc(C)o2)C2CCCC2)CCCC(C(=O)Nc2ccn(C)n2)C1 19311,C(=O)(CCC(=O)NN(C)C)N1C(C(N2C(C(C)C)C(C)(C)C2)=O)CC1C 19312,Cc1cc(N2CCC3CCC(NC(=O)C(C)(C)C(N)=O)C2C3)ncc1[N+](=O)[O-] 19313,C1(CC(=O)NCCC(C)NC(C2(C(=O)OCC)CCC2)=O)(OC)CCCC1 19314,c1(C(N2CCCC(CCNC(C(C)OC(C)(C)C)=O)C2)=O)cccc2nonc12 19315,N1(Cc2ccc(CC)s2)CCS(=O)(=O)CC1c1cnn(C)c1 19316,N1(C(C(C)(N(C(Cc2onc(C)n2)=O)C)C2CC2)=O)CC=C(CO)CC1 19317,C(=O)(C(CC1CCCC1)NC(=O)C(CO)OC)NCC#CCC 19318,C(=O)(C#CC1CCCO1)N1CCC(NC(c2c[nH]c3nccc-3c2)=O)CC1 19319,c1(C(=O)NCC2CCCC(NC(C(C)c3cccs3)=O)C2)ccc2nccn2n1 19320,C=CCC(C(=O)NCC1CC2CCC(C1)N2C(=O)C=NOC)C(C)(C)C 19321,C12(C(N3CC4CC3C4C(N3CCC(CC45CC(C4)C5)C3)=O)=O)CCCC(CO1)C2 19322,C(C)(CNC(c1ccc(-c2nnc(S)o2)cc1)=O)(C(C)C)NC(C(C)=C1CC1)=O 19323,C#CCCC(O)C(=O)NCCC1(CNC(=O)CCCc2cccc(Cl)c2)CC1 19324,CC(C)(C(=O)NC(CNC(=O)C(C)(C)n1cnnn1)CC(F)(F)F)C(F)(F)F 19325,CC1(C(=O)NCc2n[nH]cc2C(=O)NCCC2C=CCC2)CCCC1O 19326,N1(C(c2c(F)ccc(C)c2)=O)CCC2(CCCN2C(C2CSCCS2)=O)C1 19327,C(=O)(C(C)C1=CCCC1)NC1C2(CN(C(c3cncc(C(=O)OC)c3)=O)C2)CC1 19328,CC(C)C(CC(=O)NCCCc1ccsc1)NC(c1c[nH]nc1C(F)F)=O 19329,C(C(C)(C)C(=O)NC1C2CN(C(C3CCCN3C(C)=O)=O)CC12)NC(C)=O 19330,c1(-c2cn(CCCN(C)C(C3CC(C)CO3)=O)nn2)cc(F)c(F)c(F)c1 19331,C(C(=O)N1CCCC1(C)CNC(=O)CCc1cnn(C)c1C)(C(C)(C)C)OC 19332,CCCC(C)C(=O)NC(C)(CNC(=O)Cc1nccc(OCC)n1)C1CC1 19333,C1(NC(C=C2CCC(C)C2)=O)COC2CN(C(=O)CC(F)(F)C(F)F)CC12 19334,N12CC(CC1(C)C)NC2=O.C(c1ccc(Br)cc1)=Cc1cccc(C(=O)NC)c1 19335,C(=O)(C(F)CC(C)(C)NC(=O)CC(C)(C)CC)N1CCCC(C=C)C1 19336,C1(C(N(CC(CC)C)Cc2[nH]cnc2C)=O)CCN(c2ncccn2)CC1 19337,c1(N)ncc(C#N)cc1I.Cc1cccc(O)c1NS(=O)(=O)Cc1nc(CO)cs1 19338,c1(C(=O)NC2C(NC(C(c3c(F)cccc3F)C)=O)C2)c(F)ccc2nc[nH]c12 19339,C1(CNC(CCn2c(C)ncc2)=O)CN(C(=O)CC2CC=CC2)CC12CC2 19340,c1(C(=O)NC(C)C(C)NC(c2sccc2-n2ccnn2)=O)cccc([N+](=O)[O-])c1 19341,C(CC(C)(C)NC(=O)CCOCC1CCC1)=CC(=O)NCCCC#C 19342,C1(C)(C(=O)NCc2occ(N(C)C(C3CC3F)=O)n2)CCCOC1 19343,Cc1cc(CC(N2CCC(F)C(NC(c3ccoc3Cl)=O)C2)=O)ccc1CO 19344,N1(C(C=CC(C)(C)C)=O)CC2CCC(NC(=O)Cc3ccc4c(c3)OCO4)(C2)C1 19345,C(=O)(CCCCC(F)F)N1CC(C)(C)C(C(=O)NCC2C3CCCC23)C1 19346,CC(C(=O)NCc1cn(C2CN(C(c3ncccc3Cl)=O)C2)nn1)C(C)(F)F 19347,C1(NC(=O)COC2CCC2)CCN(C(C2(C3CCCO3)CCCC2)=O)C1 19348,C(=O)(C(C#N)C(C)(C)C)N1C(CC)CN(C(c2c(C)c[nH]c2CC(N)=O)=O)CC1 19349,C12CCN(CC1C1CC1)C(=O)C(C)CO2.C(CCCO)OCCCC.C12CC1OC2 19350,CN1CC2CN(C(=O)CC3CC(NC(=O)C#CC4CC4)C3)CC2C1 19351,c1(C(N2C(C)CC(NC(c3ocnc3C3CC3)=O)C2)=O)ccc2c(c1)CCC2 19352,C(=O)(CS(=O)C(F)(F)F)NCC1C(N(C)C)CN(C(CC=CC=C)=O)C1 19353,CCCCCC(C(=O)NCC(CC)NC(=O)CC(F)(F)F)C(C)C 19354,N1(C(C2N(S(C)(=O)=O)CC2)=O)CCCC2CN(C(=O)Cc3cnsc3)CC12 19355,N1(C(c2c(CC)cccc2)=O)CCCCC(NC(C23CC(CO)(C2)C3)=O)C1 19356,C1(C(N2CCC(OCC#C)C2)=O)CCCN(C(=O)C=C(C)C2CC2)C1CC 19357,C1(C(N2CCN(C(=O)CNC(CC(=O)OC(C)C)=O)CC2)=O)COCCNC1=O 19358,c1(CCNC(=O)NC(CC)CC2CCCO2)cccc(F)c1Br 19359,c1(NC(C23CCC(CC2)CC3)=O)n[nH]c2c1CN(C(c1ccc([N+](=O)[O-])o1)=O)C2 19360,N1(C(CCC=C)=O)CC(C2CN(C(=O)Nc3ccccc3C)C2)C1 19361,CCC(CC(=O)NC1(C(=O)N(C2CC2)Cc2cnn(C)c2)CC(F)C1)C1CC1 19362,Cn1nc(C(N2CCCCC2CCC(=O)NCC(C)(F)C(C)(C)F)=O)ccc1=O 19363,C12(NC(C3C(C(C)(F)F)C3)=O)CC(NC(=O)C=CSC3CC3)(C1)C2 19364,C12(NC(c3cc4ncccc4s3)=O)CCCC1CN(C(=O)CN(CCO)CCO)C2 19365,c1(N(C)C)ncc(C(=O)NCC2CC(O)CN2C(c2ccc[n+]([O-])c2)=O)cc1Cl 19366,c1(CN(C(=O)NC2CCC(c3ccc(F)cc3)C2)CC)csc(C#N)c1 19367,N1(C(=O)CCc2ccccc2)CCN(C(=O)Cc2ccc(Br)cn2)C(CF)C1 19368,C(=O)(C1=COCCO1)NCC(C)(C1CCC1)NC(c1cc(CN(C)C)on1)=O 19369,C(=O)(C1=C(Cl)CCOC1)NCC1N(C(CCCCCOC)=O)CC(O)C1 19370,Cc1nc(C)n(O)c1C(=O)NC1CCCN(C(=O)C(C)(C)C(N)=O)C1 19371,N1(C(CC(C)n2ccnc2)=O)CCCC(CNC(C2(C3CCCO3)CC2)=O)C1 19372,C1(CC(N2CCC(C(C)CNC(=O)C(C)O)CC2)=O)CC2(CCO1)CC2 19373,c12cc(cnc1-c1ccco1)C(=O)N2.N1(C(=O)OC)CC(CC=C(C)C(=O)O)C1 19374,N1(C(C2CCCCN2C(c2ccc([N+](=O)[O-])o2)=O)=O)CCC2CCCCC2C1 19375,C1(NC(C2(OC)CCSC2)=O)CC(NC(c2[nH]nnc2C)=O)CC1O 19376,Cc1ccc(C)c(NC(=O)CCC(C)NC(=O)CCc2nncn2C)c1 19377,Cc1cc(C(N2CC(NC(C3CC34CCC4)=O)C(C)(C)C2)=O)cc(C(F)F)c1 19378,N1(C(C2(CCN=[N+]=[N-])CC2)=O)CCC2(CC1)CN(C(c1n[nH]cc1C1CC1)=O)C2 19379,C=CCC(C)(C)C(=O)NC1CCC1NC(c1cccc(C(C)=O)c1)=O 19380,O=S(=O)(c1ccc(NCC2CCOC3(CCOCC3)C2)c(Br)c1)Nc1cnsc1 19381,C=CCC(C)(CC)C(=O)N1CCC(C)C(CC(N2CC(CCOC)C2)=O)C1 19382,N1(C(c2nsnc2O)=O)CCC(F)(C(=O)NCCN2CCCC2=O)C1 19383,CC(O)(CNC(=O)C(C1CCC1)NC(c1cc(O)ccc1F)=O)C(F)(F)F 19384,N1(C(c2cn3cnnc3cn2)=O)CCC2CCCN(C(c3cnsn3)=O)C2C1 19385,C1(C(=O)Cc2cc(C(=O)NCCNC(C3(C)CSC3)=O)no2)CCC(O)CN1C 19386,c1(OC)ncc(Cl)c(N2CCCC(NC(c3sccc3Oc3ccccc3)=O)C2)n1 19387,N1(C(CCN(C)C(c2[nH]ccc2C2CC2)=O)=O)CC=CC(O)C1 19388,N1(C(c2c(C)nsc2)=O)CCC(CC(=O)N(C)CCC2CCCO2)CC1 19389,Cn1nc(C(N2CCC2CNC(C2C(C)(C)C2(F)F)=O)=O)c2c1CCCC2 19390,c1(NCc2nnn(C(C)(C)C)n2)ccc(S(=O)(=O)NCc2ccncc2)cc1Cl 19391,C1(C(=O)Cc2c(C(N(CCC(=O)NC)CCCO)=O)c[nH]n2)OCCOC1C 19392,O=C(CC1CCOC1)NOCCOCCNC(=O)CSc1nc[nH]n1 19393,C(C(C)(C)C(=O)NC1CNC(=O)C1)NC(C(c1cccnc1)C)=O 19394,O=S(=O)(c1ccc(Cl)c2cccnc12)N1CC(C(F)CO)C1 19395,C1(CC=C)(NC(=O)CC(C)F)CCCN(C(c2cc(C(F)F)ccc2Cl)=O)C1 19396,CC(C(=O)NCC1(O)CCCN(C(c2ccn3c2CSCC3)=O)C1)C1=CCCC1 19397,CC(C(=O)N1CCCC1C(C)NC(C1(C)CCC(O)CC1)=O)S(N)(=O)=O 19398,Cc1cccc(F)c1CC(=O)N(C1CC(NC(C2CC3COCC3C2)=O)C1)C 19399,N1(C(CSCC#C)=O)CCC(NC(=O)C(C(C)C)n2cnnn2)C1C1CC1 19400,C(=O)(CC(C)CNC(C1CCNC(=O)C1)=O)NCCC(COC)OC 19401,c1(C(N2CCC(C)(C(=O)NCc3ccn(CCC)n3)C2)=O)ccc(C)cc1C 19402,C1(C(N(C2C(C)C2)C)=O)CC2CC1CN(C(=O)CCC1CCCO1)C2 19403,N1(C(C=C(C)C(C)(C)C)=O)CC(N=[N+]=[N-])CC1C(=O)NCc1cscn1 19404,N1(C(=O)CCc2cccs2)CCCN(C(C2CC3CC2CC3O)=O)CC1 19405,c1(CC)c(C(=O)N(C)CCNC(c2cn(C(C)(C)C)nc2C)=O)nnn1C 19406,c1(OC)ccc(C(=O)NC(C)CC2CN(C(C3(n4ccnn4)CC3)=O)C2)cc1O 19407,C1(N(C(c2n(CC)ncn2)=O)C)CCCCN(C(=O)C=Cc2ccc(C)cn2)C1 19408,N1(C(C(C)Nc2ccnn2Cc2ccsc2)=O)CCNC(=O)C1C 19409,C(C)(CO)(C(=O)NCc1ncccc1C(=O)NCCN(C1CCCC1)C)OC 19410,CC1(NC(=O)CNC(=O)CC2CCCC(F)(F)C2)CCN(C(N)=O)CC1 19411,C1(C(=O)NC(C(=O)NCC(=O)OCC=C)CC2CCC2)CCCCCCC1 19412,N1(C(CC2CCC(NC(CN=[N+]=[N-])=O)C2)=O)CC=CC(O)C1 19413,c1(CC)onc(C(N2CC(C3CN(C(c4cc(C)no4)=O)CCO3)C2)=O)c1C 19414,C(C(O)C(=O)NCCNC(=O)C(CN(C)C)N(C)C)=CCCC 19415,c1(NC(C2CCC(N(C(=O)COCC3CCCO3)C)CC2)=O)nnc(O)cc1O 19416,c1(COC)nc(C)ncc1C(=O)N(C1CN(C(C23CCC(C2)S(=O)(=O)C3)=O)C1)C 19417,CCC(CC)(C(N)=O)NC(=O)C(C)N(C)C(C1CC(=O)CC(=O)C1)=O 19418,C(C)(CC(C)CC(C)C)(c1n(CC=C)nnn1)NCc1ccc(C2CC2C)o1 19419,c1(CN2CCCC(NC(C3(CC#C)CC=CCC3)=O)C2)cc(C(C)C)nc(C)n1 19420,C1(N(C(Cc2nc(C)sc2)=O)CCO)CCN(C(=O)CC2(O)CCOC2)CC1 19421,Cc1nc(N2CCSCC2CCNC(C23CCCC(CO2)C3)=O)c(Cl)cc1C#N 19422,C1(CNC(CSCCCC)=O)CC2(CCN(C(c3cc(C4CC4)ns3)=O)CC2)C1 19423,c1(Cc2cc(CC)on2)nc(C(N2CC(C(=O)O)CC2C)=O)c(N)s1 19424,c1(CC(=O)NCCCOCCNC(C=CC)=O)csc(S)n1 19425,c1(OC)ncc(OC)s1.C12CC1C(=O)NC2.c1(OCCCNC(=O)C2CC2)cccs1 19426,C1(C(=O)NCC(C)CNC(=O)CC2COC(=O)N2)CCC12CCC2 19427,N1(C(C(C)C2CCCO2)=O)CCC2CCN(C(c3ccc(O)nn3)=O)CC2C1 19428,c1(C(C)C)nnc(C=CC(=O)NC(C2CCCC2)CNC(C2CCN(C)C2)=O)o1 19429,Cc1cccc(C)c1CNC(=O)CN1CCOCC1(C)C 19430,C(c1cc(Cl)ccc1Cl)=CC(N1CC(CNC(C2(COC)CCC2)=O)C2C1C2)=O 19431,c1(C(N(C2CN(C(=O)Cn3ccnc3)C2)C)=O)cccc(C(F)(F)F)c1 19432,C(C)(CC(=O)N1C2CCC1CC(NC(C1(CF)CC1)=O)C2)(C(F)(F)F)N(C)C 19433,C(=O)(C(F)CC(C)C)NCC1N(C(c2n(CCC)ncc2)=O)CC1 19434,C(C(C(=O)NCC(C1CC1)NC(c1cncn1C1CC1)=O)c1ccccc1)OCC 19435,S(=O)(=O)(c1cnn(C)c1)N1CC(CC(N2CCC(C(N(C)C3CC3)=O)CC2)=O)C1 19436,S(=O)(=O)(c1ccc(Nc2csc(=N)[nH]2)c(F)c1)N(C)CC.C12CC(C1(C)C)N(C)N2.O 19437,c1(OCC)ncc(C)cc1-c1cccc(CC(=O)NCc2ccnc(C)n2)n1 19438,N1(C(c2cnc(C)n2C)=O)C2CCC1C(C)C(NC(C1CCCN1C(N)=O)=O)C2 19439,C1(C2N(C(c3conc3C(C)(C)C)=O)CCC2)CCCN(C(=O)CC2CSC2)C1 19440,C1(NC(N(CC)CC)=O)CC2(C1)CC(O)C2.C1(=O)CC(c2cccnc2)N1 19441,c1(NC(C(C(C)C)NC(=O)NCCCC)=O)ccnc(OCCOC)c1F 19442,N1(C(c2c(C)cco2)=O)CCN(CC(C)NC(=O)CC2CCC2)CC1 19443,c1(C(=O)NC(c2ccccc2)CNC(C=CSC)=O)cccc2c1OCCN2 19444,C1(C2CCCN(C(=O)C3=CCCC3)C2)(NC(c2cc3cnccc3o2)=O)CC1 19445,c1(CC)nn(C)c(Cl)c1C(N1CCC(O)(CN(C)C(C2CC23CCC3)=O)CC1)=O 19446,c1(C(N2CC(CNC(CC(CCC)CC)=O)C2)=O)ccn2ncc(CC)c2n1 19447,C(C(=O)NC(C1(O)CN(C(c2ccnc(O)c2)=O)C1)C)(C(C)C)NC(C)=O 19448,C12(Nc3cc(N(C)C)ncn3)CCC(CC(COCCCC)C)(CC1)C2 19449,CCC1CC(=O)N2CCC(C2)Cn2cc1nn2.c1(C(=O)NCC)ncc[nH]c1=O 19450,c1(C(=O)NCC2CCCCN(C(C(C=C)O)=O)CC2)c(C)nn2c(C)cccc12 19451,N1(CC(=O)OC)Cc2ccccc2C1C(=O)Nc1c(C#C)nccn1 19452,C(C)(C)(CCCC(=O)N1C2CCCC1COC2)NC(CC(CC)(C)OC)=O 19453,S(=O)(=O)(c1ccc2ccccc2c1)N1CC2N(C(=O)C(F)Cl)C(COC2)C1 19454,N1(C(c2ccc(C)o2)=O)CCCCC1C(=O)NC1CC(=O)N(CC2CC2)C1 19455,C12(CC(=O)NCCCCCNC(C3CC(SC)C3)=O)COCC(C1)C2 19456,C1(CNC(CC(CNC(=O)C(N2CCOC2=O)C)OC)=O)CCCCC1(C)C 19457,c1(C(N(CC(C)NC(C2CC2(C)CC)=O)CC)=O)cc(-c2ccncc2)on1 19458,C(=O)(C(C)CC(C)(F)F)NCC1(C(C)(C)O)CN(C(C=CSC)=O)C1 19459,C1(C(=O)NCCC(C)O)C=CCN1C(=O)CC1CCC(=O)C1 19460,Cc1cc(NC(=O)C(=O)N(C2(C(F)(F)F)CC(C(F)(F)F)C2)C2CC2)cc(Cl)c1Br 19461,c1(SC)ccc(C)c(C(=O)NCC2COCC2NC(C2(N(C)C)CC2)=O)c1 19462,C12(C(N3CC(CCNC(C4CCC(C)O4)=O)C3)=O)CC3CC1C2C3 19463,C1(C(=O)Nc2n[nH]c(-c3ccc(Cl)c(Cl)c3)n2)CCn2c(O)nnc2C1 19464,C1(C(=O)N)CCCCN(C)C1=O.C(CSC)(C(=O)NCC1(n2cccn2)CC1)OC 19465,C(=O)(C(CC(C)C)C(N)=O)N1CCCC(O)(CNC(c2c(C)sc(Br)n2)=O)C1 19466,C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NCC(CNC(C1(C)CC(O)C1)=O)F 19467,N1(C(C2CN(C(C3C(C#C)C3)=O)CC2C)=O)CCOC2C(O)CC12 19468,N1(C(c2cc(CC)ncc2)=O)CC(C)(C)CC1CNC(C1CCCSC1)=O 19469,c1(C(N2C(CNC(CCCOC(C)=O)=O)CC(O)C2)=O)ccc([N+](=O)[O-])s1 19470,N1(C(C2(C(CC)=O)CC2)=O)CC2CC1(C(=O)NCCC1CC(C)=NO1)C2 19471,C1(C(C(=O)OC)NC2CC(n3cncn3)C2)CC2CCC1C2 19472,C(=O)(C1SCCc2ccccc21)N1CC(CNC(C(=O)NCC)=O)C(C)C1 19473,c1(C(N2CCN(CCCNC(C3C(C)C3)=O)CC2)=O)cccc(F)c1Br 19474,Cc1ccoc1C(c1nnnn1C1CCCC1)NC(C1CCOCC1)C 19475,C1(C)(CNC(C=C(C)C(C)(C)C)=O)CCN(C(C2(C#N)CC(=O)C2)=O)CC1 19476,N1(C(C(CC)CO)=O)CCCCC2(CCN(C(=O)CCc3c(N)cnn3C)C2)C1 19477,c1(C(=O)NCC2CN(C(C3C(C=C)C3)=O)C(C)(C)C2)cc(Cl)cc(Cl)c1O 19478,Cc1ccc(C(=O)NOC(C2C(C(N3CC(SCC)C(O)C3)=O)CCC2)=O)cc1C.OC 19479,C1(NC(C2=NNC(=O)C2)=O)CCCC2CN(C(C3C=CC=CC=C3)=O)CC12 19480,CC(C)CC(O)C(=O)NC(Cc1ccco1)C(=O)NC(C)Cc1nc[nH]n1 19481,O=C(CCCCCCBr)N1CCC(O)C(NC(C2(C(F)(F)F)CC(O)C2)=O)C1 19482,C12(C(=O)NCCCCC)CCCC1CCN2C(c1ccc(CC)cn1)=O 19483,Cc1ccc(C(=O)NC(=O)C(C)SC(C)C)c(Br)c1.N12CC3(CCC3C1=O)C2 19484,C(=O)(CCC(CC)OC)NCC(C)N(C(C1CCN(S(CCC)(=O)=O)CC1)=O)C 19485,CCC(CC(F)F)C(=O)N1CCCC1(C)CNC(c1c(F)ccc(C)c1F)=O 19486,C1(CC)CN(c2ncc(C3CC3)cn2)CCN1C(c1ccccc1SC)=O 19487,Cc1cc(C(=O)N(CCNC(C2(NC(N)=O)CCC2)=O)C2CC2)c2ncccc2c1 19488,C=CCC(CC)N=c1[nH]c(N2CCC(OCCO)C2)nc2ncn(C)c12 19489,C1(CN(C(=O)CCC)CC)CCN(C(=O)C(O)C2CCC2)CC1 19490,C(=O)(C(F)(F)C(O)C(C)C)N1CCCCC(NC(c2c(C)nc(CCC)s2)=O)C1 19491,C1(CNC(COCCC#C)=O)CCOC1C(=O)N(C1CC(O)C1)C 19492,N1(C(=O)NC(c2nc(=O)[nH][nH]2)C)CCCC2(C=CCO2)CC1 19493,N1(C(CC(=C)C)=O)CCN(C(=O)C(C)Oc2ccc(Cl)c(Cl)c2)CC(O)C1 19494,c1(C(=O)OC)ccc(F)c(C(=O)NCC2CC(NC(=O)C(F)(F)C(C)O)C2)c1C 19495,C1(C(=O)NCC(C)(C)C(=O)N2CCC(C)(F)C2)CCCC(C#N)C1 19496,C1(NC(=O)CN(c2ccncc2)C)CCC2CN(C(=O)CC3CCC4CC34)CC12 19497,CC(C)C(Cc1ccccc1)C(=O)NCCC(C)N(C)C(c1cc(C#N)c[nH]1)=O 19498,c1(NC(C2(C)CCC(C(N(C)C)=O)C2(C)C)=O)cc(C#N)ccc1O 19499,C1(N(C)C(c2cnn(C(F)F)c2)=O)CN(C(=O)CC2C(C)(C)C2(C)C)CCC1O 19500,CC1(CNC(N2CCC(Oc3ccccc3)C2)=O)OCCc2sccc21 19501,N1(CC)CC(C(N2CC3CC2C3NC(c2nccnc2N)=O)=O)CCC1=O 19502,c1(C(N2CC(C#C)(F)C2)=O)ccc(C(F)(F)F)cc1I 19503,c1(C(C)C)ccc(C(=O)NCC(=C2CN(C(c3ocnc3Br)=O)C2)F)o1 19504,C1(C(N2CC(NC(CCc3cnc(C)s3)=O)C2)=O)CN2CCN1C(C)C2 19505,C(=O)(CN1C(=O)CSc2ccccc21)N1CCC(NC(C2C(C)CCC2)=O)C1 19506,c1(C(=O)NCCCNC(C2CC(OCC)C2)=O)cccc(OC)c1 19507,N1(C(C(c2cccnc2)NC(C)=O)=O)CCC(CO)C1.C12(CCCO1)C(=O)N2 19508,O=C1CCC(C(N2CCN(C(=O)Cc3cn(C4CC4)cn3)C(CO)C2)=O)CCO1 19509,c1(CC)cc(C#N)nc(N2CCC(NC(c3cnc(C)[nH]c3=N)=O)C2)n1 19510,C12(CCOCC1)C(=O)N(C)C2.c1(CCC)ccc(CC)cc1 19511,c1(C(=O)NCC2CCCN(C(=O)COC3CCOC3)C2)ccc(C2CCC2)nn1 19512,C#CC1CC2(CC2)CN1C(=O)CC1CC(C)(C)CN1C(=O)CC1CC1CC 19513,C1(N(C(=O)Cc2cc(C)[nH]n2)CC)CCCN(C(=O)C(C#N)NC(C)=O)C1 19514,c1(NC(C(C)NC(C(C)OC)=O)=O)cnc(F)nc1 19515,C1(CNC(CC(C)C)=O)C(O)C(O)CN1C(=O)CC#N 19516,C1(N(C(C)=O)C)CCC(C(N2CCCC(CC(C)C)C2)=O)CC1 19517,N#Cc1ccc(C=CC(=O)NCCNC(=O)Cc2cn3c(n2)CCCC3)cc1 19518,c1(CNCC2C(C)(O)CCC2)ccc(-n2cncn2)c(F)c1 19519,CC1(F)CCN(C(=O)CC2CCN2C(c2ccccc2F)=O)C1 19520,c1(C(=O)NCC(N(C(=O)C=CC2CCCC2)C)C2CC2)cc2cccn2c(O)n1 19521,N1(C(Cc2c(C)non2)=O)CCC(CNC(=O)CN(C)C2CC2)CC1C 19522,N1(C(c2scc(C)c2C)=O)CCC2(CC2NC(C2CC(C(C)C)=NO2)=O)C1 19523,C(=O)(C1=CC2CCCC12)NCC(C)N(C(Cn1c(C)ncc1)=O)C 19524,C1(CCNC(C23CC(C)(C2)C3)=O)CCCCN1C(=O)C(C1(O)CCCC1)F 19525,CN1C(=O)CC2C1NC2=O.c1(SCC#N)ccccc1 19526,Cc1c(Br)cc(C(N2CC3CC3(CNC(c3cnc(Cl)cn3)=O)C2)=O)cc1Br 19527,C(=O)(C(O)CC(N)=O)N1CC(C(N2CC(C(=O)OCC)OCC2)=O)C1 19528,c1(N(CCCNC(C(C)C2CCCC2)=O)C(C)C)ncnc2c(Br)csc12 19529,N#CC1(C(=O)NC2CC(NC(=O)CC=CC(C)(C)C)C2)CCCC(=O)C1 19530,C1(NC(c2ccc(Cl)cn2)=O)CC12CCC(NC(=O)CCn1cncn1)CC2 19531,N#Cc1ccccc1-n1ccc(C(N2CSCC2C(=O)N2CCC2)=O)n1 19532,N1(C(c2cnc(CC(C)C)s2)=O)CCN(C)C(CNC(=O)C(C)CN(C)C)C1 19533,CC1CN(C(C2(C)CCCN2C)=O)CCC1C(N1CCCC(C(N)=O)C1)=O 19534,CCCCC(CC)CC(=O)NCC1(F)CC2CCC(C1)N2C(C1CC2(CC2)C1)=O 19535,C1(OC)CCCC1NC(=O)CN(C1CC(C#N)C1)C(=O)Cn1cc(C)cn1 19536,c1(NC(C2C3CN(C(c4cc(SC)ncn4)=O)CC32)=O)cccc(F)c1O 19537,C1(CNC(c2cn(CC)nc2)=O)COCCN1C(C1CC(F)CN1C)=O 19538,C(=O)(C(CCNC=O)N(C)C)N(CCC)CCO.C1(=O)CN1 19539,c1(OC)cc(C(=O)NC2CC(C)N(C(c3cc(Cl)sc3Cl)=O)C2)ccn1 19540,N1(C(CC(=O)NCC2CC2)=O)CC2CCC1CN2C(c1cc(SC2CCC2)c[nH]1)=O 19541,C1(C)(CNC(c2n(C)ccc2)=O)CCCN1C(=O)CCc1ccc(CO)cc1 19542,Cc1ccnc(SCC(=O)NC2(C)CCN(c3nnnn3C)C2)n1 19543,c1(OC)sc(C(N2CCC2CNC(C2CCOC2C2CC2)=O)=O)cc1Br 19544,C1(C(=O)NC(CNC(C(C)=CC)=O)C(C)(C)C)CCCCC(F)(F)C1 19545,CC1C(NC(c2ccc(O)c(F)c2)=O)CCCN1C(c1coc(C(F)F)c1)=O 19546,c1(OC)cccc(F)c1C(=O)N(C1CCN(C(C2CCC(F)CC2)=O)C1)C 19547,N1(C(c2c(OC)cc(O)cc2)C(=O)Nc2ccccc2)CC=C(c2cncs2)CC1 19548,Cc1c(CNC(C2C3CN(Cc4cc(O)cc(Br)c4)CC23)=O)cncc1Br 19549,C(CC)(CCN(C)CCOc1ccccc1)(OC)NCC1CCC(C(=O)NC)O1 19550,c1(N2C(CNC(C3(C(=O)NC)CC3)=O)CC3COCC32)ncc2scc(Br)c2n1 19551,CC1CC(N(C(=O)C(C2CCOC2)NC(=O)Cn2cccc2)C)CCO1 19552,c1(CCC)ncc(C(=O)NCC2CCN(C(=O)C(C)c3ccsc3)C2)s1 19553,N1(c2cc(N(C)CCC3CCOCC3)nc(C)n2)CC(C)(C)CCC1CO 19554,C1(C(=O)NCC(CSC)OC)CC(O)CCN1C(c1ccns1)=O 19555,C#CCC(CC(=O)NC1CC(C)CC(=O)N1)NC(C1(COC)CCCC1)=O 19556,C1(C(N2C(C#C)CC2)=O)CCCCCN1C(C1CCCCN1C)=O 19557,c1(C(=O)NC2C3(CC(NC(C(CC=C)(F)F)=O)C3)C2)ccc2cnc(C)n2c1 19558,N12CCOC(C1)C2=O.C1(C(=O)NC2(CSC)CC2)(OC(C)C)CCSCC1 19559,c1(NC(c2c(C)cc(C)c(C)c2)C)nc(C)cc(=NCc2nc(C(C)C)cs2)[nH]1 19560,c1(C(N2CCC(OCc3ccccn3)CC2)=O)cnccc1Cl 19561,c1(C(=O)NC2C(OC)CC(NCC3=CCN(C(C)=O)CC3)C2)ccc2[nH]ccc2c1 19562,CC(C)(C)C(O)C(=O)NCc1nocc1C(=O)Nc1cnc(Cl)cn1 19563,C(CC(C(=O)N1CCCC(CN(C)C(C2(CCF)CC2)=O)C1)NC(C)=O)SC 19564,CCCCS(=O)(=O)CC(=O)N1CC2C(n3cc(-c4cc(C)nn4C)nn3)C2C1 19565,C1(NC(c2c[nH]c(C(F)(F)F)c2)=O)CC2C1CCN2C(=O)C(=C1CCCCC1)F 19566,N1(C(CC(C)F)=O)CCSCC1C(=O)NCc1cnnn1C 19567,c1(C2(C(N3CC(CNC(C4CC4C(F)(F)F)=O)C3)=O)CC2)ncccc1F 19568,C1(C(F)(F)F)(C(=O)NCCCN(C(=O)NCCCl)CCO)CC2C=CC1CC2 19569,Cc1cc(C(N2CC(O)(CNC(=O)CC3(O)CCCN(C)C3)C2)=O)cc(C)c1F 19570,c1(C(=O)NCC(C)N(C(c2ocnc2C)=O)CC)ccc(C)c(C)c1F 19571,CCC(CCCC(=O)NCC(O)CC(C)C)NC(=O)C=CCO 19572,c1(OC)ccc(CN(C(c2ccc(=N)[nH]n2)C(=O)NCC2CC2)C2CC2)cc1 19573,C1(CNC(C=C(CC)CC)=O)CCC(C(=O)N(CC)CC2CC2)O1 19574,C1(C(=O)NCC(C)(C)F)C2CC(O)C(C2)N1C(c1cccc2cc[nH]c12)=O 19575,C1(C)(C(N2CCCCC(CNC(CCC(C)(C)O)=O)C2)=O)CCCCC1(F)F 19576,CC1(CCNC(C2(C)C=CCC2)=O)CCN(C(c2csc(Br)n2)=O)C1 19577,C(=O)(C1=CCOCC1)N1CCC(N(C(C2C(C#C)C2(C)C)=O)CC)C1 19578,CN1CC(C(=O)NCC2(C(=O)NCc3cccs3)CC2)NC1=O 19579,N1(C(c2c(CCC)nco2)=O)CCN(C(=O)Cc2cnns2)C(CC(C)(C)C)C1 19580,C=CC(C)(C)CC(=O)NCC1(C)CCCN1C(=O)C=Cc1scnc1C 19581,CN(CCCC(=O)N1CCN(C)CC1CNC(=O)CC1CC(O)C1(C)C)N=O 19582,c1(C(=O)NC2(C)CCN(C(C3(CCO)CC3)=O)C2)ccc(Br)cc1[N+](=O)[O-] 19583,c1(CNC(C2(CNC(CCc3onc(C)n3)=O)CC2)=O)cc(O)ccc1F 19584,c1(C(=O)NCCCCCN(C(CNC(CC)=O)=O)C)ccc(N(C)C)cn1 19585,N1(C(CCCC#CC)=O)CC(CNC(=O)C(O)CC(C)C)CC(C)(C)C1 19586,N1(C(C=CCC)=O)CCC2CN(C(=O)C(O)C(C)(C)C)CC12 19587,N1(C(Cc2scc(C(=O)OC)c2)=O)CCC(NC(c2nn(C)cc2C)=O)C(C)C1 19588,c1(C(=O)NC2(C)CC(NC(c3n[nH]c(C)c3Br)=O)C2)csc2nccn12 19589,c1(C(=O)NCC(C)NC(c2n(CC)nc(C)c2)=O)ccc(F)c(C)c1C#N 19590,N1(C(c2c(C)coc2)=O)CC(C)N(C(c2cc(Cl)c[nH]2)=O)CC1C 19591,C(=O)(C1CCC(=O)c2ccccc21)N1CCCC(NC(=O)CSc2ccsc2)C1 19592,c1(CC(=O)NCC(CC)NC(c2n(CCC)ncc2)=O)noc(C)c1C#N 19593,C=CCC(C(=O)N(CC(C)O)CCNC(C12CCC(OC)(CC1)C2)=O)C(C)(C)C 19594,CCC(CC(=O)N1CCC(OCCNC(C2CCN2C2CCCC2)=O)CC1)C(C)C 19595,N1(C(C(C(C)C)SC)=O)CC2C(NC(=O)CC(C)(C)C(C)(F)F)CS(=O)(=O)C2C1 19596,C1(NC(C(C(C)CC2CC2)N(CCCN(C)C)CCOC)=O)CN2CCC1(F)CC2 19597,Cn1nc(CC(N2CCC(NC(=O)Cn3cnnc3)C2)=O)cc1F 19598,C(=O)(C(F)C1=CCCCC1)N(CCCNC(c1ccc(C(=O)OC)[nH]1)=O)CCC 19599,C(=O)(CCC(F)(F)F)N1CCC(N(CCC)C(c2nn(CCC)cc2Cl)=O)CC1 19600,c12ccc(o1)c(=O)[nH]2.N1(S(C)(=O)=O)CC(C(=O)NCCC2CN(OC(F)F)C2)C1 19601,c1(CS(N2CC(C(=O)OCC)C3(C2)CC3)(=O)=O)c[nH]c2nccc-2c1 19602,N1(C(C(C)(C)Br)=O)CC2(CCCN(C(c3cccc4nscc34)=O)C2)C1 19603,C(=O)(C1=CNC2=NCCCN12)N1C(CNC(Cc2c(C)non2)=O)C(C)CC1 19604,c1(C(N2C(C(C)NC(c3n(CC)c(O)nc3)=O)CCC2)=O)cc2ccccn2n1 19605,c1(C(N2CC(C(C)NC(=O)C(C)C(F)F)C2)=O)ccc(N)c(F)c1F 19606,c1(C(=O)NC2CCCCN(C(Cc3c(C)nc(S)s3)=O)C2)ccnc2c1CCC2 19607,c1(C(=O)NCC2C(C(=O)NC3C(C)CN(C)CC3)CCC2)nccc2[nH]ccc12 19608,C1(CCC)CN(C(=O)CCc2ccsc2)CCN1C(=O)CN(C)C(N)=O 19609,N1(C(c2c(C)scn2)=O)CCCC(N(C(=O)Cc2cc(Cl)cs2)C)CC1 19610,n1(C(C)C)ccc(C(=O)NCC(C)(C)NC(c2cnn(CC(F)F)n2)=O)cc1=O 19611,N1(C(c2scc(C)c2C)=O)CCN(C(C2CCN2S(C)(=O)=O)=O)C(C(C)(C)C)C1 19612,N1(C(=O)OC(C)(C)C)Cc2nccnc2CC1C(=O)NC(C1CCOC1)CO 19613,C1(CNC(Cc2cn(C(C)C)nc2)=O)CN(C(=O)COC2(C)CCC2)CC1C 19614,CC(N=c1ccc(C#N)n[nH]1)C1CCN(C(c2nccc3[nH]ccc23)=O)C1 19615,C1(NC(CCN(CCC)C)=O)CCCCC1NC(=O)C=Cc1nccs1 19616,Cc1cccc(SCC(=O)N(C2CCCC(NC(=O)CC(F)F)C2)C)c1 19617,c1(C(N(C2C(NC(C(C(C)C)SCC)=O)CCCC2)C)=O)nc(C)c(C)nc1C 19618,CCC(C)(CNC(c1c[n+]([O-])c(C)cn1)=O)C(=O)N1CCCCC1C 19619,c1(NC(=O)NCCCCC(C2CC3CCC2C3)CC)cc2ccccc2o1 19620,N1(C(c2ccc(C)nc2C)=O)CC(C(N2C(CO)CC2C)=O)C(C2CC2)C1 19621,C1(C)(C(=O)NCCOCCN(C)C(c2cc(Br)cn2C)=O)CCCNC1=O 19622,N1(C(=O)Cn2cc(CO)nn2)CC(C(=O)NCC2CC(F)(F)C2)CC(F)(F)C1 19623,C(CCCCC(=O)NC(C)CCN(C(=O)Cc1cc(C2CC2)no1)C)OCC 19624,N1(C(COCC=C)=O)CCC(N(C(=O)CCN2CCCS2(=O)=O)C)C(C)C1 19625,C#Cc1cc(NC(=O)CC2CC(NC(C3(C)CC3(C)C)=O)C2)cc(F)c1 19626,c1(C(=O)NCC2CC(OC)CN2C(C2CCNC(=O)C2)=O)ccncc1F 19627,N1(C(C(C)N(C(CSC(C)C)=O)C)=O)CCCC(C)(O)C1 19628,C12(CNC(CCN(CCC)C)=O)CN(C(=O)CC=C(C)C)CC1CCO2 19629,c1(C(=O)NC(CCNC(c2nc(C)nn2C)=O)(C)C)nccc(N)c1Cl 19630,CC1CC(NC(=O)C(=O)N(c2cccs2)CCNC(=O)OC(C)(C)C)CC(C)C1 19631,c1(OC)cc(Br)c(CCNC(=O)NCCC(O)Cn2cccn2)cc1OC 19632,N1(Cc2cc(C(=O)OC)oc2C)CCC(n2cc(CCO)nn2)C(O)C1 19633,c1(C(=O)NCC(CNC(c2nc(C(C)=O)sc2)=O)CO)nnc(C)cc1O 19634,Cc1noc(C)c1S(=O)(=O)N1CC2CN(S(=O)(=O)CCBr)C2C1 19635,c1(OC)cc(C(=O)NCC2CN(C(C3CC34CC4)=O)CCO2)cc2c1OCCO2 19636,c1(N2CC(C(=O)NCc3c(C)cccc3C)C2)c(C)ccc(F)c1[N+](=O)[O-] 19637,C(=O)(N=c1ccn(C2CC2)[nH]1)C1(O)CCC1.C12(CCC1)CC(=O)NC2.CN(C)C=O 19638,c1(C(=O)NCC2(O)CCCN(C(C3ON=C(CC)C3)=O)C2)cccn2nccc12 19639,N1(CC(=O)NC2CC2)CCS(=O)(=O)C(CCNC(C2CCCCC23CC3)=O)C1 19640,CCS(=O)(=O)CCCNC(N1CC(C(=O)OC)OCC1C)=O 19641,N1(C(C(CC)CC2CCCCC2)=O)CC(C)CN(C(C2(O)CCSC2)=O)CC1C 19642,N1(C(C(F)=CCC)=O)CC(O)(C2(CNC(C3CC3c3cccc(C)c3)=O)CC2)C1 19643,c1(CCC)nc(=NC(C)CN(C(=O)C(n2cc3ccccc3n2)C)C)s[nH]1 19644,N1(C(c2c(CC)cno2)=O)CCC2C(C(=O)NCCCCC3CC3)C2C1 19645,c1(CCNC(N2CC(C(C(=O)OC)OC)C2)=O)coc2ccc(C)cc12 19646,C1(OC)CN(C(c2cc(C)n(C)n2)=O)CC1CC(=O)NCCc1cc(C)ns1 19647,c1(C(=O)NC2CCN(C(=O)CC3CCOC3)C2)cnnc2ccccc12 19648,c1(C(=O)OC)ccccc1C(N1CC(NC(c2nc(C)c(C)s2)=O)CC1CO)=O 19649,N=c1[nH]c(=NCC2CCNC(=O)C2)[nH]c(=NC2CC(NC3CCC3)C2)[nH]1 19650,c1(C(=O)NC2(C(=O)NC)CCC(F)(F)CC2)ncn2c1CCNCC2 19651,CCC(Cc1ccccc1)CC(=O)N(C)CCN(C(=O)CCC(C)(C)C)C 19652,c1(OC)ccc(SCCCCCn2cc(C3CCCN3C)nn2)c(Br)c1 19653,N1(C(CC(CC)SC)=O)CCN(C)C(CNC(C2CN3CCC2CC3)=O)C1 19654,C12(C(N3C(CN(C(CCCC(C)C)=O)C)CCC3)=O)CC=CCN1CCC2 19655,C1(NC(c2c(C)csc2)=O)COCCN(C(c2cn(C(C)C)cc2C)=O)C1 19656,Cc1cc(CO)oc1C(=O)NCC1(F)CC(CNC(=O)CC2CC3CC3C2)C1 19657,C(C1CN(C(=O)COCC2CC2)CC1C(N1CCOCCC1C)=O)=CC 19658,C1(NC(C2CCN(C)C2)=O)CC2(C1)CC(NC(c1cc(C(F)F)no1)=O)C2 19659,C1(C(N2CCN(C(COCCCCCC)=O)CC2CF)=O)CCc2nn[nH]c2C1 19660,C(C)(C(=O)NOC1CCOC1)(N(C(c1cccc(CC)n1)=O)C)C1CC1 19661,c1(SC)nccnc1C(=O)NCC(C)N(C)C(C1CCC1(F)F)=O 19662,C1(CCNC2CCS(=O)(=O)N2CCOc2ccc(F)cc2F)CCOC2(CCC2)C1 19663,Cc1cc(F)cc(C(=O)NCC2CN(C(C3CC4(CC4)CO3)=O)CC2(C)C)c1N 19664,n1(CC)c(C)cc(C=CC(=O)N(CC(O)CNC(c2cn(C)nc2C)=O)C)c1C 19665,N1(C(C(CCC)CC)=O)CCCCCCC1C(=O)Nc1ccc(F)cc1C#N 19666,Cc1cn(C)nc1CNC(C1(C)C=CCN1C(=O)CC1CCC(=O)NC1)=O 19667,C(=O)(C1=CCN(C(=O)CC2C=CCC2)C1)NCC(CC)C#N 19668,N1(C(c2ccc(OC)o2)=O)CCn2cc(C(N3CCC(F)(F)C(O)C3)=O)nc2C1 19669,C1(CSC2(CC=C)CN(C(=O)OC(C)(C)C)C2)CNC(=O)CC12CCC2 19670,C#CCC(C)(CNC(=O)C(C)CNC(=O)CCc1ccsc1)CO 19671,C(=O)(C1CCCc2nncn21)NCCNC(c1c(C(F)F)ccc(C)c1)=O 19672,N1(C(CSc2ccc(COC)cc2)=O)CC2CC1CCC2N(C)C(C1(C)CC1)=O 19673,c1(C(=O)NC2CC(C)(NC(C(CC)COC)=O)C2)cc(O)cc(F)c1 19674,N1(C(C=CCCn2ncc(C)c2)=O)CCC(CF)(NC(=O)C(C)CF)C1 19675,C1(NC(c2c(OCC)n[nH]c2)=O)CN(C(=O)CCSCC(F)F)CCC12CCC2 19676,C1(OC)CCC2(C(N3CCC(C)C3CNC(C3COCCN3C)=O)=O)CC12 19677,N#CC1(C(=O)NCCNC(=O)CCN2CCCS2(=O)=O)CC2CCC1C2 19678,C(CC)(CCC(=O)N1CC(CNC(CC)=O)(CC)C1)OC 19679,CCC(CC1CCCCC1)C(=O)NCC1CC(F)CN1C(=O)Cc1[nH]cnc1C 19680,N1(C(C2CC(NC)C2)=O)CCCC(C)(CNC(=O)CS(=O)(=O)NC2CC2)C1 19681,CC(C)C(C)(C)C(=O)NCC(=C1CN(C(C2CNC(=O)C2)=O)C1)F 19682,C1(NC(CC=C)=O)Cc2ccccc2C1NC(=O)CC1C(=O)ON=C1C 19683,C1(F)(CNC(c2cc(C)nn2C)=O)CCN(C(=O)C(C)(Cl)Cl)CC1 19684,C12(C(OC(F)F)=O)CC(CC3C(CC(=O)NC(C4CC4)C)C3)(C1)C2 19685,Cc1cccc(C(=O)NCC(c2ccccc2)N(C(=O)CCN2CCC2)C)c1C 19686,C=CC1(CNC(C2CC(OCC)CN2C(=O)Cc2c[nH]nc2)=O)CCCC1 19687,Cn1c(CCc2ccco2)ccc1C=O.N1(CC=O)CCCC1 19688,c1(C(=O)NC2CCC(NC(c3coc(O)n3)=O)CC2)ccc2c(c1)CCCC2=O 19689,C1(CC)CN(C(C23CC(F)(C2)C3)=O)CCC1NC(c1conc1C)=O 19690,C1(COC(CC2CCC(C)O2)=O)OC(=O)NC1(C)C 19691,C(CCCCC(=O)N(C1CCN(C(c2cc(C)co2)=O)C1)C)OCC 19692,c1(C(N(C(C)C(=O)Nc2ccc(CC)nc2)CCC)=O)[nH]ccc(=O)c1C 19693,CC1(C)C=C(C(=O)NC(C)(CNC(C2(N3CCCC3)CC2)=O)C2CC2)C1 19694,C(=O)(CC(C)(C)C(F)F)NCCCCC(C)NC(C1CCS(=O)(=O)C1(C)C)=O 19695,c1(NC(=O)CN2C(=O)Nc3cccc(c3)C2)cccc(Br)c1F.C(C)(C)(C)OC 19696,c1(CN(c2nnc(C3CCCC3)n2CCC#N)C)cc(Cl)ccc1F 19697,C1(NC(C(C)=CC2CC2)=O)CCC(C)N(C(=O)CCCn2ccccc2=O)C1 19698,C(=O)(CC(C)(C)N(C(=O)C(C)n1cncn1)C1CC1)NC(C)C1CC1 19699,C1(C)(CNC(c2ccc(COC)cc2)=O)CN(C(C2(C)CCC2)=O)CC1C 19700,n1(CC(=O)NCC=CCC(=O)NC2CCN(CCC)C2)ncn(C)c1=O 19701,N1(C(C2(CCC)CCC2)=O)CC2(CCC(CNC(=O)C(C)CC(C)(F)F)O2)C1 19702,Cc1cc(-n2cc(C(C)(C)NC(=O)C(C)NC(=O)CC#N)nn2)cc(C)c1 19703,c1(NCC2C(c3cn(C)nc3)C2)nccc(=NC2COC3(CCC3)C2)[nH]1 19704,C1(CNC(c2nnc(CC)s2)=O)CC2COCC2N1C(c1sncc1C)=O 19705,N1(C(c2ccc(CC)s2)=O)CCC(NC(c2c(C(F)F)nn(C)c2C)=O)C(C)C1 19706,C1(NC(CN2CCC(C)C2)=O)CCCCN(C(c2cccc(OC(F)F)c2)=O)C1 19707,C(CNCc1c(C)cncc1)(CC(F)(F)F)NC(=O)COCC1CCCO1 19708,C1(C(N2CCC(C(F)F)C2)=O)CCCN(C(C2(Cl)CCC2)=O)C1 19709,Cc1ccc(F)cc1CC(N1CCCC1CN(C(C1CC1(F)Cl)=O)C1CC1)=O 19710,C1(NC(c2ccncc2Cl)=O)CC2CN(C(C3CCCSC3)=O)CC12 19711,C1(NC(c2coc3c2COC3)=O)CCCC2CN(C(=O)CC3CC34CC4)CC12 19712,c1(C(N2CCC(O)(C(C)NC(C3(C(=O)OCC)CC3)=O)C2)=O)cc(=O)cc(Cl)[nH]1 19713,N1(C(c2cc(Br)ncc2Br)=O)CCC2CN(C(c3cc(O)cc(Br)c3)=O)CC2C1 19714,c1(NC(=O)NCc2cnc3c(c2)CC(CSCC)CO3)cccc2ccn(C)c12 19715,C1(C(N2CC(C(C)NC(=O)CC3CC3C3CC3)OCC2)=O)CCOC2(CCC2)C1 19716,C1(N(C(=O)C(C)c2cc[nH]n2)CC(=O)NCCC)CCCC12CCNCC2 19717,c1(C(=O)NC(COC)CCS(C)(=O)=O)ccc2n1CCNC2 19718,N1(C(c2nc(CNC(C3N(C)CCOC3)=O)oc2)=O)CCC(O)C(O)C1 19719,C1(CC(=O)N(C2CCN(C(C34COCC(C3)C4)=O)C2)CC)CC2CCC1C2 19720,Cc1cccc(F)c1CC(=O)Nc1nc(CC(=O)NC(c2cncn2C)C)cs1 19721,c1(C(=O)NC2C(C(=O)NCCC(C)C)C2)ccc2ccc(O)nc2c1 19722,CC1CCCN(C(c2cccnn2)=O)C1CCNC(c1cc(F)ccc1Br)=O 19723,N1(C(C(C=CCCC)O)=O)CCCC(C)(CNC(=O)CN2CCCC2CO)C1 19724,NC(=NCC1CCCN1C1CC1)NCC1CC1(Cl)Cl.c1(C(C)C)conc1C 19725,c1(CC)nc(O)c(C(=O)NC2CCCCC2CNC(C2(C)CC=CC2)=O)cc1C 19726,N1(C(c2c(CC)ncnc2)=O)CCC(C(=O)NCCC(C(C)C)OC)C(O)C1 19727,C1(C(N(CCC)C(C)C)=O)CCCC(NC(C2CCC(=O)NC2)=O)C1 19728,N1(C(c2cc(I)ccc2Br)=O)CCC2C(CCN2C(=O)CC2CCCCO2)C1 19729,N1(C(Cn2c(CC)nnn2)=O)CCC2CCC(C1)N2C(=O)Cc1cc(C2CC2)on1 19730,C(C(C)C(F)C(=O)NCC(n1ccnn1)C)NC(c1scc(CC)c1)=O 19731,c1(OC)cc(Cl)ccc1C(F)(F)C(=O)NC1CCN(C(=O)C=CC=C(Cl)Cl)CC1O 19732,CCC1=C(C(=O)NC2(C)CCN(C(c3cnn4c3CCC4)=O)C2)SCCO1 19733,c1(C2CN(C(C(c3cccs3)SC)=O)C2)nccc(C)n1.C1=CC(=O)NC(C)(C)C1 19734,C1(C(=O)NC(C2(O)CN(C(C(c3ccccc3)OC)=O)C2)C)C2CC2C2CC12 19735,C1(CC(=O)NC2C(OC)CCCC2)C2CCCC2N1C(c1nscc1C)=O 19736,N1(C(C2CC3CCC(C2)N3C2CC2)=O)CCC2CCN(Cc3ccccc3)CC12 19737,N1(C(Cc2ncc(C)[nH]2)=O)CCC2C(CCCN2C(C2CC2Br)=O)C1 19738,C1(C(=O)NCC2C(NC(c3cc(C(C)=O)on3)=O)C2)CCCC1S(C)(=O)=O 19739,CCS(=O)CC(=O)N1CC(O)CC1CC(=O)NCC(O)CF 19740,Cn1nc(C2CCC2)cc1C(=O)NCCCCCCNC(C12CCC1C2)=O 19741,C(=O)(CC(C)NS(C)(=O)=O)NCC(CC)NC(c1sccc1Br)=O 19742,N1(C(C(C(CC)C)O)=O)CCCC2(C1)CN(C(=O)CN1CCP(C)(=O)CC1)C2 19743,CC1(C)CCOC(C(=O)NC2C=CC(C(=O)NC3CN4CCCC3C4)C2)C1 19744,c1(C(=O)NC(CC=C)CNC(=O)C(C)(C)c2cscc2Cl)cc(N(C)C)ccn1 19745,C1(C(=O)NOCC2CCC2)C(C2CC2)CCN1C(c1cccc2occc12)=O 19746,c1(OCCC(=O)NC2CC(F)(CNC(=O)NC3CC3Cl)C2)ccccc1F 19747,N#CC1(C(=O)NC2CN(C(=O)CCCCCNC(N)=O)C2)CC2CCC1CC2 19748,C(=O)(C(CC(N)=O)NC(=O)COC1CCCOC1)NCC(C=C)O 19749,C=CCCCC(=O)N(C1CN(C(C2(C3CCC3)CC2)=O)C1)C 19750,CC(C(C)(C)C(=O)NCCN(C)C)NC(=O)CCOC(C1(C)CC=CCC1)=O 19751,c1(C(=O)NC2C(NC(C3N(C)C(=O)CC3)=O)CCC2)cccc2c1CCCCC2 19752,N1(C(C2=C(C)OCC2)=O)CCC(NC(C2(c3cc[nH]n3)CC2)=O)CC(C)(C)C1 19753,c1(NC(C)CN2CCCC2)cc(S(=O)(=O)Nc2ccc(Cl)cc2)ccc1C#N 19754,C1(NC(C(C)OCc2ccncc2)=O)C2CC(O)C1N(C(C1(N(C)C)CC1)=O)C2 19755,C1(NC(C(=Cc2ccccc2)CC)=O)CCCCN(C(=O)C(C)C2CC2)CC1 19756,N1(C(C(C)OCCOC)=O)CCc2nc(CNC(=O)Cc3cn(C)nc3C)sc2C1 19757,C(N=c1[nH]cnc2c1COC2)C1CC2(CC(NC(=O)Cn3cc(Cl)cn3)C2)C1 19758,C(=O)(C(CC)n1cncn1)N(CCCNC(=O)CN(C)CC1CCC(=O)N1)CC 19759,C(CCCCCC(=O)NCCC1CCC(=O)N1)NC(C(=Cc1cn[nH]c1)C)=O 19760,C12(CNC(c3c(C)coc3N)=O)CCCC1CCN2C(=O)CN1CCCNC1=O 19761,N1(C(Cc2cc(C)sc2)=O)CC2(CO)CC1(C(=O)NC1CC(O)CC1O)C2 19762,C(=O)(C(C(C)CC)OC(C)(C)C)N(CCOC(CNCCCCCC)=O)CCC(C)C 19763,C1(NC(C(CC=C)C)=O)CN(C(c2nccc3[nH]ccc23)=O)CC1C1CC1 19764,c1(C(=O)OCC)ccc(COC(C2(C)N(C(C3(C)COC3)=O)CCC2)=O)cc1F 19765,N1(C(C2N(C)C(=O)CC2)=O)CCC(O)(C2CCN(C(=O)CCC3CC3)CC2)CC1 19766,N1(C(c2cc3nc(C)sc3[nH]2)=O)CCC2(CC1)CCN(C(C1OCC1(C)C)=O)C2 19767,N1(C(c2cc(CC)n(C)n2)=O)CC(NC(=O)CS(=O)(=O)CC)C(C2CC2)C1 19768,c1(C(=O)NCC2(NC(CSCC#C)=O)CC2)ccccc1SC(C)C 19769,c1(C(=O)NCCC(C)NC(c2nocc2Cl)=O)c[nH]c2ccc(Cl)cc2c1=O 19770,c1(C(=O)OCC)ccc(N2CC(C(=O)Nc3cnc(Br)cn3)CCC2)nc1 19771,c1(NC(C2C(CNC(c3cncs3)=O)CCC2)=O)c[nH]nc1Br 19772,c1(C(=O)NCc2conc2CNC(=O)C(O)C2CCC2)ccncc1C1CC1 19773,Cc1ccncc1C(C)NC(C1CCCC1CNC(=O)Cc1cccc(F)c1)=O 19774,c1(C(N2C(C(NOCCOCCOC)=O)C=CC2)=O)ccnc(C)c1C 19775,Cc1cccc(-c2cncc(C(=O)NCC(O)CCNC(C3CCCS3)=O)c2)c1 19776,CCCC(O)CC(=O)NCCCCC(CO)NC(=O)CN1CCOC1=O 19777,CC(C)(C)C1=NOC(C(N2CC3CC3(NC(c3ccns3)=O)C2)=O)C1 19778,C1(CNC(C#CC2(C)CCCO2)=O)C2CCCN(c3nnc(C4CC4)s3)C2C1(C)C 19779,c1(C(N2CC(O)(CCNC(C3C(CC(C)C)C3)=O)C2)=O)cccc([N+](=O)[O-])c1N 19780,Cc1cc(CC(=O)N(C(C)CCNC(c2[nH]nnc2C)=O)C(C)C)cs1 19781,C1(CC)CN(C(c2cncn2C)=O)CCC1CNC(c1ccnn1C)=O 19782,C1(C(=O)NCC(c2ccccc2)C)CC(F)CN(C(c2cc(O)n[nH]2)=O)C1 19783,N1(C(C(CC(C)C)(F)F)=O)CCCC2(C1)CN(C(c1ccnn(C)c1=O)=O)C2 19784,C(=O)(CS(=O)(=O)NCC(C)(C)CSC1CC1)NCC(C)C(=O)N(C)C 19785,c1(C(=O)NCC2C(C)CN(C(=O)C(O)C3CCC3)CC2)cccn2ccnc12 19786,N1(CCC)CC(C(=O)NC2CN(C(c3c[nH]nc3F)=O)CC2C)CC1=O 19787,c1(C(=O)NC2CC(NC(=O)C(F)(F)c3ncccn3)C2)cc2c(Cl)cncc2s1 19788,c1(C(N(CCCNC(C(CCC)NC(N)=O)=O)C2CC2)=O)c(Cl)ccc(Cl)c1O 19789,C12(CNC(C(C)(C)SC)=O)CCC(CN(C(C34CCC(C)(C3)OC4)=O)C1)C2 19790,CC1CC(O)CN(C(=O)CC2CCN(C(=O)Cc3ccsc3)C2)C1 19791,C1(C(=O)NCCOCC2CCC2)C(C2CC2)CCN1C(=O)C#CC1CCC1 19792,Cc1cccc(Cl)c1C(N1CC(CC(N2CCC(CF)CC2)=O)C1)=O 19793,c1(C(=O)NC2CCC(C)N(C(C3C4CC5C(C4)C35)=O)C2)ccc2nn[nH]c2c1O 19794,CC(C)CC(C(=O)NC1CC(F)(F)C1)ONC(=O)C1CC(C)C1 19795,N1(C(C2N(C(C(C(=O)OC)(C)C)=O)CC(O)C2)=O)CCc2ncncc2C1 19796,C1(C(=O)NCC2CCCN(C(c3cnc(C)[nH]3)=O)C2)COC2(CCC2)C1 19797,c1(OC)ccc(NC(C2CC3CC3N2C(=O)CCCCCBr)=O)cc1C 19798,c1(CC)ccc(CC(C)C)c(NC(=O)NC(c2nc(C3CC3)n[nH]2)C)c1 19799,C1(=O)C(CC(C)C)O1.c1(C(Cc2ccccc2)NC(=O)OCC)ccccc1C 19800,c1(C(N2C(C)CC(CNC(C(C)NC(C)=O)=O)C2)=O)ccc(C(F)(F)F)cc1Cl 19801,Cc1ncc([N+](=O)[O-])n1CC(=O)NC1CC(CCNC(C2CC(C)CCO2)=O)C1 19802,C12(CNC(C(CC(C)C)N(C)C)=O)CN(C(c3cc(Cl)no3)=O)CC1CCO2 19803,Cc1sc(O)nc1C(=O)N(C)CC1CCN(C(=O)COCC(F)F)C1 19804,c1(C(=O)NC2CN(C(CCC(=C)Cl)=O)C(C)C2)c(F)cc(OC)c(F)c1F 19805,C1(C(=O)NCCSCC)CCC(C(C)C)N1C(c1cc(C2CC2)on1)=O 19806,C1(OC)CCN(CCCNC(=O)NC(C)(C)CSC)C1 19807,c1(CC(N2CC(O)(C(C)NC(C=C(C)C3CC3)=O)C2)=O)cc(F)ccc1F 19808,C1(CNC(c2ccc(F)cc2)=O)CCC2(CN(C(C3(CO)CCC3)=O)C2)O1 19809,C1(SC)CN(C(=O)CC(F)(F)F)CC1C(=O)NC1CC(N(C)C)C1 19810,O=C(C1=CCCC1)NCc1ccc(C(=O)NCCN2CCCCCC2)nc1 19811,c1(C(=O)NC(CNC(C2N(CC)CCC2)=O)C(C)C)ccn(CC)c(=O)c1 19812,c1(C(=O)NC2(C3N(C(c4n(CCC)ccc4)=O)CCC3)CC2)cc2n(c1)CCC2 19813,c1(C(C)NCc2cn(-c3cccc(C(=O)O)c3)nn2)cc(-n2cccc2)ccn1 19814,N1(C(c2c(C)cc[nH]2)=O)CCCC(C(=O)NC(C)COc2ccc(F)cc2)CC1 19815,Cc1ccn(CC(=O)NC(C)C(C)NC(c2coc(COC(C)(C)C)n2)=O)c(=O)c1 19816,c1(C(C)C)n[nH]cc1C(N1CCC(C(=O)N(C(C)CC2CC2)C)C1)=O 19817,C1(CC)CC(O)CN1C(=O)C(CC1CCC1)NC(=O)C=CC(=O)OC(C)(C)C 19818,N1(C(C(C)OCC#C)=O)CCCC2(CC(NC(=O)CC(O)CN(C)C)C2)C1 19819,N1(C(C(COC)O)=O)CC(NC(c2nccc3[nH]ccc23)=O)C2(CCOCC2)C1 19820,c1(CNC(c2cccc([SH](c3ccc(Cl)c(F)c3)C)c2)C)cncc2c1CCC2 19821,S(=O)(=O)(CCCCCl)N1CC2C(C(N3CCC(CC#N)CC3)=O)(C2)C1 19822,C=CCCCCCCCC(=O)NC1CC2CN(C(=O)Cn3nnnc3C)CC2C1 19823,N1(C(=O)C=C2CCCC2)CC2C3CCC(C2C1)N(Cc1c(F)cccc1F)C3 19824,CON1CCC(CN(C=O)CCc2ccc(O)cc2)CC1 19825,N1(C(C2C(C(N)=O)COC2)=O)CCC(NC(C23CCC(CC2)OC3)=O)C(O)C1 19826,c1(C(N2CC(NC(=O)C=C(Cl)Cl)C(CO)CC2)=O)ccn2nccc2n1 19827,c1(NC(C2(C)CN(Cc3c(OC)ccc(I)c3)C2)=O)cccc2sc(C(C)C)nc12 19828,c1(C(=O)NCC2CCN(C(CC3(C)CC3(F)F)=O)C2)ccc2c(c1)NC(=O)CN2 19829,c1(C(=O)NCC(C(C)C)NC(C2CC(OC)C2)=O)ccc2ccsc2c1 19830,CC1(C)CC(NC(=O)C(=Cc2ccccc2)C#N)CN(C(c2coc(Br)c2)=O)C1 19831,c1(CC)ccoc1C(=O)N(CC(C)(C)N(C(c1ccc(C(F)(F)F)[nH]1)=O)C1CC1)C.CO 19832,S(=O)(=O)(C=Cc1ccccc1)N(CCC(N1CC2(CCS2)C1)=O)C 19833,N1(C(C(CSC)C)=O)CC(O)CC1CNC(c1nc(C2CC2)cs1)=O 19834,C12(C(=O)NCCN(C(C3CC(C(C)C)OCC3)=O)C3CC3)CCN(CC1)S(=O)(=O)C2 19835,C1(CNC(c2ccon2)=O)COCCN(C(C2(c3cc[nH]n3)CCC2)=O)C1 19836,N1(C(C(CCC)OCC)=O)CC2(CCC2)CC1CNC(C1(CC)CCCC1)=O 19837,c1(C(=O)NCC(CNC(CC2(OC)CCCCC2)=O)F)c(C)cc(F)cc1C 19838,N1(C(c2cccc(COC)n2)=O)CCC2CCN(C(c3ccoc3Cl)=O)CC12 19839,C1(NC(C2C(C(C)C)OCC2)=O)CC=C(C(=O)NCc2ccncn2)C1 19840,CC(C(=O)NCC1CC2(C1)CN(C(=O)Cc1cccc(C#N)c1)C2)C(C)(F)F 19841,C1(NC(C2CC2F)=O)(CO)CCN(C(=O)Cn2cc(-c3ccccc3)cn2)C1 19842,O=C(CCC(F)F)NCCCCNC(C1(c2cncs2)CCCC1)=O 19843,C1(C(=O)NC2CC(CNC(=O)CC3C=CCN3C)C2)(OC)CCSC1 19844,c1(OC)ccc(NC(=O)C(c2cc(Cl)ccc2C)N2CC(O)CC2C2CC2)c(Br)c1 19845,c1(OC2CCCC(C(=O)NCCNC(CC(=C=C)C)=O)C2)ccccc1C#N 19846,C(C1CCCC1)=CC(=O)N(CC(=O)NCCCC=C)C1CC1 19847,C(=O)(C1=CCCCCC1)NC(C(=O)NCC1CC[Si](C)(C)C1)c1ccoc1 19848,c1(C(=O)NCC2C3CCC(C3)N2C(c2ncccc2F)=O)ccc2c(c1)CCO2 19849,Cc1cc(C)n(CC(=O)NC(C2CCCC2)CNC(=O)CCCC2CCC2)n1 19850,C(=O)(C(C)CC(=O)c1cccc(F)c1)NCCNC(C(N1CCNC1=O)C)=O 19851,C1(O)(C(=O)NCC(C2CC2)NC(CC2(C=C)CCCCC2)=O)CN2CCC1CC2 19852,c1(OC)cc(C(=O)NCCCN(C(=O)C(C)C(F)F)Cc2ccccc2)ncn1 19853,CCC1=C(C(=O)NC2CCN(C(=O)C(c3cccc(F)c3)F)C(C)C2)CCCO1 19854,c1(C(N2CC(O)CC(NC(C3C(C)(C)C3(C)C)=O)C2)=O)cc2nc[nH]c2cn1 19855,Cc1sc(C(=O)NC(C(=O)OC(C)(C)C)C2CC2)c(C#N)c1C 19856,C1(NC(C(=Cc2ccccn2)C)=O)C2CCC1CN(C(c1ccc(O)cn1)=O)C2 19857,C(C)(C)(C(=O)OCC)NC(C(Cc1ccco1)NCC)=O 19858,N1(Cc2ncc(-c3c(F)ccc(F)c3)nc2)CC2CCCCC2C1 19859,N1(C(CC(CC)C2CC2)=O)CCN(c2ncnc(Cl)c2Br)C(C)C1 19860,O=C(CCCC(F)(F)F)N1CC(C2(NC(=O)C(F)n3cccn3)CC2)C1 19861,N1(C(=O)C(F)Cc2ccccc2)CCN(C(c2ccc(C(F)F)cn2)=O)C(CO)C1 19862,C(=O)(C(C)(C)C1=CCN(C(=O)C=C(C)C(C)C)C1)NC(CCC=C(C)C)C 19863,N1(C(C(C2CC2)OC)=O)CCCC(N(C)C(c2cccc(F)c2C(C)C)=O)CC1 19864,c1(C(=O)NCC(CC(C)C)NC(C(COC)(C)C)=O)cnn2cc(C)cnc12 19865,N1(C(c2scc(C(C)=O)c2)=O)CCCC(C)(NC(=O)CN2CSCC2=O)C1 19866,CC(CC(F)(F)F)C(=O)NCC(C)(C)CCNC(=O)CSCc1cccc(Cl)c1 19867,c1(C(N(CCCCCNC(=O)CNC=O)C)=O)ccc2ocnc2n1 19868,C1(Oc2c(NC(N3CC(OC)C3)=O)cccc2)CCc2c[nH]nc2C1 19869,N1(C(Cc2c(C)ncs2)=O)CC2CC(N(C(=O)COCCOCCO)C)C1C2 19870,N1(C(C(F)=C(C)C)=O)CCN(C(C2CC2(Cl)Cl)=O)C(C(C)C)C1 19871,N1(C(CC(n2c(SCC)ncc2)C)=O)CCCC2CN(C(C)=O)CC12 19872,Cc1nc(N2CC=CC2)cc(N2CCC(c3ncccn3)CC2)n1 19873,C1(N(C)C(c2cncnc2)=O)CCCC2CN(C(=O)CC3CC3(Cl)Cl)CC12 19874,c1(C(N2CC(CCOC)N(C(=O)CCNC(C)=O)CC2)=O)cc2oc(C)cc2[nH]1 19875,C(c1c(C)nn(C)c1Cl)=CC(=O)N(CCNC(c1cnc(=N)[nH]c1)=O)CC 19876,c1(C(=O)N)cccn2c(O)nnc12.CC(CCCC)NC(=O)C=CCN(C)CCOC 19877,N1(C(C(C)OC)=O)CC(c2cn(CCNS(C)(=O)=O)nn2)C(C2CC2)C1 19878,Cn1cc[nH]c(=NCC2(CC3CCCCC3)COC2)c1=O 19879,C12(C(=O)NC3CCN(C(=O)Cc4ccsc4)CC3)CCCCC1C2Br 19880,O=C1CCOCCN1Cc1cn(CC(N2CC(CCC34CC(CO3)C4)C2)=O)nn1 19881,C(CC(C)C(=O)NC1CCOCC1NC(=O)Cn1cccnc1=O)=CC 19882,C1(COC)(NC(c2ccc(CO)o2)=O)CCN(C(=O)Cc2cnoc2)C1 19883,c1ccc(C(=O)N(C2CCCC2)CCNC(C2CCCN2C)=O)cc1.CC(=O)OC 19884,n1(CC)cncc1C(N1CCC1CC(N1CCCC1CO)=O)=O 19885,CC1(C)CC(C(N2CCCC2CC2CC2)=O)CN(C(=O)Cc2ccsc2)C1 19886,Cc1noc(C)c1CNC(C1CCC(CNC(=O)C(C)(C)N2CCCC2)O1)=O 19887,N1(C(CS(=O)(=O)N(CC)CC)=O)CC(NC(c2cccc(C)c2)=O)C(C2CC2)C1 19888,C(=O)(CC1=CCN(C)CC1)NCC(CC=C)C(N1CCCC2(CO)CCCC12)=O 19889,c1(C(=O)NC2CCN(C3CC3)C2)cc(C)n(C)c1.C1(C(=O)NCC)(COC)CCCC1 19890,c1(C(=O)NC(CNC(C(COC)OC)=O)CO)ccc2ncccc2c1F 19891,O=C(CCC(F)(F)F)NCC(C1CC1)NC(c1cnn[nH]1)=O 19892,c1(CNC(CC(C)CF)=O)nc(CNC(=O)C(CO)c2ccccc2)cc(O)n1 19893,C1(N(C)C(C2CCO2)=O)CCC2CN(C(c3ccc4c(n3)OCCO4)=O)CC12 19894,C1(C(=O)OC(C)(C)C(=O)NCC(C)N(C)Cc2ccccc2)CC2(CCC2)C1 19895,N1(C(C2CC2Cl)=O)CCC(F)(CNC(=O)C=CC=C(Cl)Cl)CC1 19896,c1(C(N2CCC3(NC(c4ccsc4)=O)C(CC2)C3)=O)cc2c(O)ncnc2cn1 19897,C(=O)(C(F)CCC(C)(C)C)N1CCC(CC#C)(C(=O)NCC2CC2(Cl)Cl)C1 19898,C1(C(N2CC(O)(CCNC(c3n(C)c(Cl)nc3)=O)C2)=O)CC1C1CCCC1 19899,C#CCC(CC(F)F)C(=O)NCC(C1CC1)NC(C1(OC)CCOC1)=O 19900,C1(NC(c2ccn(CC)n2)=O)CCC12CN(C(c1nc[nH]c1C(F)(F)F)=O)C2 19901,C(=O)(CN1C(=O)CCc2ccccc21)N1CCC(CNC(c2cc(Br)c[nH]2)=O)C1 19902,C(c1cccc(F)c1)=C(C(N1C(CNC(C(N2CCCC(O)C2)C)=O)CC1)=O)F 19903,C1(C(NOCC(C)C)=O)CN(C(C2CC2(Cl)Cl)=O)CC1(C)C 19904,N1(C(C(C(C)C)C)=O)CCC2(CC2NC(c2ncccc2Cl)=O)C1 19905,C1(CC(=O)NC2(C(C)NC(=O)C(C3CCCCC3)O)CC2)C(=O)NN=C1C 19906,C1(CNC(C23CC(C)(C2)C3)=O)CN(C(C2CNC(=O)C2)=O)CCCO1 19907,C1(NC(c2cc(C)oc2C)=O)CC2(CCCN(C(C3(CC(F)F)CCC3)=O)C2)C1 19908,N1(C(C(C)(C)CCF)=O)CCC2CN(C(C3CC(=O)CCO3)=O)C2C1 19909,C1(NC(CCc2c(C(=O)OC)c(C)[nH]c2)=O)CCC2CN(Cc3ccsn3)CC12 19910,C(C(N=[N+]=[N-])C(=O)NCCCCNC(c1csc(C(C)=O)n1)=O)OCC 19911,CC1(C)C(C)(C)C1(F)C(=O)NCCC1CCN(C(c2cccc(N)n2)=O)C1 19912,C(=O)(CC(C)(C)CC(=O)Cc1nc(CO)cs1)N(CC(=O)NC(C)(C)C1CC1)C 19913,c1(N(CCCN=[N+]=[N-])C)ccccc1NC(=O)C(N1CCCCC1)=O 19914,c1(C(=O)NCC2N(C(C3C(=C)C3C(=O)OC)=O)CC(O)C2)cccc2c1CNC2=O 19915,C(=O)(C(C)(C)N=[N+]=[N-])NCC(C(=O)NC(C(=O)OC)(C)C1CC1)O 19916,CN=c1[nH]c(=NCC(C)F)[nH]c(=NCCc2ccc(OC)cc2OC)[nH]1 19917,CC1(NC(=O)CC2(O)CCC2)CCC(NC(C2C=CCC2)=O)CC1 19918,c1(NC(N2C(NC(=O)NC)CCCC2)=O)ccc(C#N)cc1C(F)(F)F 19919,C1(NC(C(N)=O)=O)CC(C2CCN(C(c3n[nH]c4c3CCOC4)=O)CC2)C1 19920,C1(n2cc(CN(CC)CC)nn2)CN(C(c2conc2C)=O)CC1C 19921,c1(C(=O)NC2C(CC)N(C(=O)CCS(C)(=O)=O)CC2)ccc2c(c1)OCO2 19922,N1(C(C2(CNC(C3CC3(Cl)Cl)=O)CCCCC2)=O)CCC(F)(F)C(O)C1 19923,c1(NC(C)=O)ccc(C(=O)NCCCN(C)C(c2ccc(CO)cn2)=O)cc1F 19924,C1(C(N2CCC(O)(C(F)(F)F)CC2)=O)CC12CCN(C(C1CCC1)C1CC1)CC2 19925,N1(C(=O)NC)CCC(NC(=O)NCC(C2CCCC2)N(C)C)C1 19926,O=C(C1=COCCO1)NCC(C1CCN(C(=O)CC2CC3C=CC2C3)CC1)F 19927,CC(=O)C(C)CC(C)C(=O)NC(C(=O)NCCN(C)C1CC1)c1ccco1 19928,c1(CC(=O)N(CCNC(c2c[nH]ccc2=N)=O)CC)cc(OC)cc(C)c1 19929,S(=O)(=O)(c1ccc(C)c(C(=O)O)c1)N(n1nccc1C(F)(F)F)C(CC)C 19930,C1(CC(=O)NCC(F)(F)F)CC2(C1)CN(C(=O)CN(C(=O)CC(F)(F)F)C1CC1)C2 19931,c1(OC)ccncc1CN1CC=CC1C(=O)Nc1cncc(C(F)(F)F)c1 19932,c1(C(N(C2CCN(C(C(C(C)C)OC)=O)C2)C)=O)cc2nccn2c(O)n1 19933,C1(N(CCc2nncn2C)C)CCN(C(=O)CNC(C2CC(C(F)(F)F)C2)=O)CC1 19934,N1(C(C)=O)CC2(CC(S(=O)(=O)N3CC(N4CCOCC4)C3)C2)C1 19935,c1(C(=O)NC2CC(NC(C)=O)C2)cc2nc(C)sc2[nH]1.C(=O)(C1(C)C(=O)N1)OC 19936,N1(C(C2(C#N)CCC2)=O)CCN(CCC2(Nc3ccc(F)cc3)CC2)CC1 19937,C(CCN=c1[nH]c(=NCC2CCCCC2O)c2cccc(F)c2[nH]1)=C(C)C 19938,C(O)(CCC(=O)NCC1CC1(C)C)(C(F)(F)F)c1ncc(C)o1 19939,N1(C(COC)=O)CC2CCC2(CNC(=O)C(C2CCCCCC2)O)C1 19940,C1(C)(C(=O)NCC2(OCC)CCC2)CN(C(=O)CCCCC(N)=O)C(C)(C)C1 19941,C(=O)(C1SCCc2ccccc21)NC1CCC(C)(NC(c2cc(F)c[nH]2)=O)CC1 19942,c1(C(N2CC(CNC(C(C)n3cncn3)=O)N(C)CC2)=O)cnc2occc2c1 19943,C1(NC(c2cc(CC)oc2C)=O)CN(C(C2(C)CCCCO2)=O)CCC1O 19944,N1(CC)CCCN(C(C2OCCC2NC(=O)C(C2CCCCC2)O)=O)CC1 19945,N1(C(c2cnc(OC)s2)=O)CCCC1C1CCCN1C(=O)C=Cc1nc(C)co1 19946,C(CCC(C)(C)NC(c1scc(C)c1Br)=O)NC(CC1(OC)CC1)=O 19947,C1(C=O)CCC(O)CN1C.C1C(=O)N1CCSC.C(C(C)O)NCCF 19948,n1(CC(c2cncn2C2CC2)=O)cnnc1O.c12cn(nn1)C1CN(C1)C2=O 19949,C(=O)(CC(C(F)(F)F)OC)NC(C(C)NC(c1nc(OC)c(C)s1)=O)CO 19950,CC1CN(C(c2ncccc2C(F)(F)F)=O)CC1(C)CNC(=O)Cn1cncn1 19951,CC1=C(C)CC(C(=O)NCCC(O)CNC(=O)CC2(n3cncn3)CC2)CC1 19952,c1(C(N2CCC3(C(CNC(CC=C=C)=O)C3)CC2)=O)coc2c(OC)cccc12 19953,CC(C)CC(C)(CNC(=O)COC1CCCC(C)C1)NC(C1CC(F)(CO)C1)=O 19954,CCCCC(C(=O)NCCC1CCCN(C(C2CCCC2C)=O)C1)NC(N)=O 19955,CC(C)CC(CC(=O)O)NC(c1cnc(CC2CCC2)s1)=O 19956,c1(CC)nnc2c(C(=O)NC3CCCC3NC(C3CCCN3CC)=O)cccn12 19957,C(CCCC(=O)NCC(C)(CO)NC(=O)COc1csc(C(F)(F)F)n1)N(C)C 19958,C1(NC(c2ccc(C)o2)=O)COCCC1NC(C1(F)CC=CCC1)=O 19959,N1(C(C2N(C(C)=O)CCCC2)=O)CCC(C)C(NC(c2cnc(C(N)=O)s2)=O)C1 19960,c1(C(N2CC(OC)(CNC(=O)COC3CCOCC3)C2)=O)cc2c(C)[nH]nc2s1 19961,N1(C(C(c2cccc(F)c2)C)=O)CCN(C(=O)C(O)C2CCC2)CC(C)(F)C1 19962,c1(C(N2CCN(C(C#CC(C)C)=O)CC2)=O)ccnc2cc[nH]c12 19963,c1(C(=O)NCC23C(CN(C(CC(C=C)C)=O)C2)C3)cc(Cl)ncc1O 19964,C1(C(=O)NCCCCC2(NC(C3CC4CC4C3)=O)CC2)CC2CC(C1)CS(=O)(=O)C2 19965,O=C(C1=C(Cl)CCC1)NC1CCCN(C(=O)CC2C=CS(=O)(=O)C2)C1 19966,c12onc(C)c1C(=O)NC(CNC(C1(COCCC)CCC1)=O)C1CC2C1.SC 19967,N1(C(CC(C)C2CCC2)=O)CCN(C(=O)CNC(C2CC3CC2C3)=O)CC1 19968,CC(=O)C(C)CC(C)C(=O)N1CCN(C(=O)C#CC2CCC2)C(C(C)C)C1 19969,C(C1c2ccsc2CCN1C(c1c[nH]c2nccc-2c1)=O)NC(=O)C1=C(Cl)CC1 19970,C1(C)(NC(C=Cc2nc(C)sc2)=O)CCN(C(c2cc(C)ccc2F)=O)CC1 19971,Cn1cc2c(n1)CC(C(N1CCCC(C(=O)NOC)C1)c1ccccc1)CC2 19972,N1(C(C2C(OC)CC2)=O)CCC(NC(=O)CC2CSCCS2)C1C1CC1 19973,C1(=O)CCC(=O)N1C(C)C.C(CCC(=O)N1CCC(CC2CCCC2)C1)SC 19974,Cn1cc(C(=O)NCCC2(NC(=O)C(O)C3CCC3)CC2)c(-c2cnccn2)n1 19975,C(=O)(CC(C(F)F)NC(=O)CC1CC(F)(F)C1)NCC1N(C)CCOC1 19976,C1(C(=O)Nc2cn(CC)nc2)CCC(NC(=O)CC2CC=CCC2)CC1 19977,C1(NC(c2nc(C)oc2)=O)CCCCC12CCN(C(C1CSC1)=O)C2 19978,C(=O)(C(CO)C(C)(C)C)NCC1CC(CNC(Cc2nn(C)c(Cl)c2)=O)C1 19979,c1(C(N2CCC(C(F)(F)F)(OC)C2)C(=O)NCC=C)ccc(OC)cc1Cl 19980,C1(N(C(c2nc(OCC)c(C)s2)C(=O)NC(C)(C)C)C)CCOC(C)(C)C1 19981,CC1CCCC(C(=O)NCCCOCCC(=O)NCc2ccn(CCF)n2)C1 19982,C(=O)(C1=CCCCCC1)NC(C)CCCCNC(=O)CCNC(C1CCCCC1)=O 19983,c1(CSCC(=O)N(C)CC2CN(C(=O)C(C3CCCCC3)O)C2)ccccc1 19984,c1(C(=O)NC2CC(O)(CNC(c3n(C)ncc3C#N)=O)C2)cc(F)cc(Cl)c1N 19985,C=C(C)CC(C(=O)NCC1CSCCO1)NC(=O)C=C1CCOCC1 19986,N1(C(C(=O)NCC(C2CN(C(=O)C#CC(=O)N(C)C)C2)C)C)CCP(C)(=O)CC1 19987,CCCCCS(=O)(=O)CC(=O)N(CCNC(C1CC12CC(F)(F)C2)=O)C(C)C 19988,C1(C(=O)NCC2CC(OC)C2)(NC(c2cnncc2C)=O)CCN(C)C1 19989,Cc1ccc(C(=O)NCC(CNC(c2cn(C)nc2C)=O)C(F)(F)F)cc1Br 19990,N1(C(CSCC(N)=O)=O)CC(CNC(=O)C(F)(F)C2(O)CCC2)C(C(F)(F)F)C1 19991,C(=O)(CCC(F)(F)C(F)F)NC1CCC(CCNC(c2c(C)cnnc2O)=O)C1 19992,N1(C(C(COC)(C)OC)=O)CCC2(CC1)CN(C(c1cocc1C)=O)C2 19993,c1(C(C)OC)cn(CC2C=CCN2C(c2cc(C(C)=O)on2)=O)nn1 19994,N1(C(CC(C(C)C)O)=O)CCC(C2(O)CCN(C(C3(O)CCCC3)=O)C2)CC1 19995,c1(OC)c(C(=O)NC(CNC(=O)Cc2ccc(C)nc2)CO)ccnc1Cl 19996,c1(C(=O)NCC2CC(CNC(CSS(C)(=O)=O)=O)OC2)cc2ccnc(Cl)c2s1 19997,c1(C=O)cnc(C)c(CC)c1.CCC(C(=O)N1CCC(NCCO)C1)NC(N)=O 19998,c1(-c2cccc(C3(C(=O)Nc4cccc(I)c4F)CC3)c2)cccc2ccncc12 19999,C(c1c(C)noc1C)=CC(N1C(C2CCCN(C(CS(CC)=O)=O)C2)CCC1)=O 20000,C1(CNC(C2C=CCCC2)=O)CN(C(=O)C2=CCCSC2)CC12CCC2 20001,c1(C(N(C2CCCN(C(=O)C(C)(F)C(C)(C)F)C2)C)=O)ccn2nncc2c1 20002,Cc1nnc2ccc(C(=O)NCCNC(C34CCCC3CC4)=O)cc2c1C 20003,Cc1cc(C(=O)NCC2CN(C(c3cnnc(Cl)c3)=O)CCCO2)cc(C)c1N 20004,CCCC(C)(O)CC(=O)NCc1cccnc1C(N1CCNC(=O)C1C)=O 20005,C1(C(N(CCCCNC(c2c[nH]nc2-c2cccnc2)=O)C)=O)CCNC(=O)C1 20006,C#Cc1c(Br)ccc(NC2CCCC(C(C)C)CC2)c1Br 20007,CCC(C)(C)CC(=O)N(C(CC(F)F)C(=O)N1CC(CC)C(F)C1)C 20008,C(CC(=O)N(C(CNC(=O)CC1(C)CCC1)C1CC1)C1CC1)OCC 20009,CCC(COCC)C(=O)NCC(C)(C)C(=O)N(CC(C)C(=O)OC)C 20010,N1(C(C=CC)=O)CC(C)(C)CC1C(=O)NCC1COCCO1 20011,C1(NC(c2c(C)nsc2C)=O)CC(NC(C2CC(n3cnnc3)C2)=O)C12CCC2 20012,C(CCC(C)(C)C)(C(=O)NC1CCC1)N1CC(O)CC(c2cccc(C)c2)C1 20013,C(=O)(C1CCCc2nc[nH]c21)N(CC(C)N(C)C(C1(C)CC2(CCC2)C1)=O)C 20014,CC1CCC(C(=O)NC2CC3(CC3)C2)N(C(C23CCC(C2)C3)=O)C1 20015,N1(CC(=O)NC2CCCC(NC(c3ccnc(S)c3)=O)C2)CCNC(=O)C1 20016,c1(C(=O)NC(C)C(=O)NC2C(C(N(CC)CC)=O)CC2)cccc(C)c1O 20017,C1(CN(C(C(C2CCC2)OC)=O)C)CCN(C(c2cnnn2C(C)C)=O)C1 20018,c1(C(=O)NC(CC)CNC(=O)CCCOC2CCOCC2)c(C(C)=O)cnn1C 20019,C1(F)(CNC(C(CC)=CCCC)=O)CCC(NC(=O)CC2(COC)CCCC2)C1 20020,Cc1ccc(-c2ccccc2)cc1-c1nc(C(C)O)nn1C(C1CCCC1)C 20021,c1(CC(N2C(COC)(CNC(c3n[nH]cc3SC)=O)CCC2)=O)c(C)cccc1C 20022,c1(C(=O)NCC2(CNC(C3C4CC4C4CC34)=O)CC2)c[nH]nc1[N+](=O)[O-] 20023,C12(CCN(C)C1)C(CC(=O)OC)N2.c1(SC)ccc(I)cc1 20024,c1(SC)cc(C(=O)NC(C)CCCNC(C2OC3CCC2CC3)=O)ccc1N 20025,CC(=O)CCCC(C)C(=O)N1CCCCC1CCC(=O)NC1CCN(C)C1 20026,C1(C(=O)NCC23OCC(NC(c4ccnc(C)n4)=O)(C2)C3)COCC(C)(C)O1 20027,c1(CCC)ccc(-c2nc(C(=O)NC3CCC3CNC(=O)CSCC)cs2)cc1 20028,N1(C(C(c2cc(Cl)sc2Cl)C)=O)CCN(C(=O)C(C)(C)O)CC1C 20029,Cc1ccc(C(N2CCC(CC(N)=O)(NC(=O)CCn3ccnn3)CC2)=O)cc1F 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20237,Cc1cc(C(=O)NCC2CN(C(=O)CN3CCCS3(=O)=O)C2)ccc1Cl 20238,N1(CCN2CC(NC(=O)CNC(C)=O)CCC2=O)CC2(CCCC(COC)O2)C1 20239,N(S(=O)(=O)N=S(C)(=O)c1ccccc1)c1nc(C(C)(C)C)c(C=O)[nH]cccc1 20240,c1(CC)ccc(C(=O)NC2(CNC(=O)CC3CC34CC4)CCCC2)cn1 20241,CS(C)(=O)=NC(=O)C(=O)NC12CC(NC(=O)C=CC(N3CCOCC3)=O)(C1)C2 20242,C1(CNC(=O)Nc2cnn(CC(F)F)c2)CC(F)(F)CN1C(=O)Cc1ccno1 20243,N1(C(c2c(N)ccc(C)c2)=O)CC(NC(=O)CC2OCCCO2)C2CCCCC12 20244,CCCCC(C(=O)N(C)CC1CCC(CNC(=O)Cn2ccnn2)CC1)N(C)C 20245,c1(C(=O)NCCC(C)NC(C2CC(C(C)C)C2)=O)ccc2cc(O)ccc2c1 20246,CC(C)C(O)(C(=O)OC(C)(C)C)C(F)(F)F.C12C(C1(F)F)CNC(=O)OC2 20247,C(C(C(C)(C)C)NC(C1(C#N)CC(=O)C1)=O)NC(c1nnc(C)s1)=O 20248,CC1(CNC(=O)Cn2cc(CS(C)(=O)=O)nn2)CCCCC1(F)F 20249,C#Cc1ccc(C(N2CCC(C(=O)NCC(O)C(C)C)(COC)C2)=O)o1 20250,N1(C(=O)Nc2cc(F)cc(Br)c2)CCC2CCCCC12 20251,c1(C(N2CCCCC(NC(c3ccc(C)s3)=O)C2)=O)cc(Cl)c(N)cc1F 20252,c1(-c2n(CC=C)c(N(CC(C)C)CC)nn2)ccc(S(C)(=O)=O)cc1 20253,C(=O)(C#Cc1ccccc1)NC1CCCC(C)C1.N12CC(CC1=O)C(=O)N1CC2C1 20254,c1(C(C)C)ccccc1C(=O)NC1CC1CNC(=O)C=C1CC1 20255,C1(NC(C2(C)CC2)=O)CCN(C(=O)C=Cc2cc(Cl)ccc2Cl)CCC1CO 20256,N1(C(CC(C)SC)=O)CCCC(C(=O)NCC2(n3ccnn3)CC2)C1 20257,N1(C(CN(C2CC2)CC)=O)CC2CC(C(=O)NCc3cnc(C)cc3C)(C2)C1 20258,CN=C(NCC(=O)NC(C)C)N(C)CC(C(C)C)OCCOC 20259,c1(C(N2C(C)C(NC(=O)C=Cc3nccs3)CCC2)=O)cc(F)c(F)c(C#N)c1 20260,c1(C(C(C)C)NCC(Cc2ccc(OC)cc2)C)cc(Cl)cc(Cl)c1 20261,C1(CNC(COCC(=O)OC)=O)CC2CCC1N(C(=O)C(C)C1CCOC1)C2 20262,C(=O)(CCCC(F)(F)C(F)(F)F)NC1C2CN(C(C(C)(C)CC#N)=O)CC1C2 20263,n1(CC)cnc2c(N3CCC(CC(C)C)C3)nc(NC(C)(C)CF)nc12 20264,C1(NC(c2cc(COC)[nH]n2)=O)CCCCC1CNC(=O)Cc1ccns1 20265,CN1CC(CNC(=O)CC(O)CNC(C2CCCC(=O)N2)=O)C(O)C1 20266,c1(C(N2CCC(N(C)C(C3(C)CCCC3)=O)C2)=O)cc(F)c2cn[nH]c2c1 20267,N1(C(Cc2cc(C)nn2C)=O)CCCC(C)(C(=O)Nc2cccnc2C(C)C)C1 20268,C1(CCCC)CCCN1C(=O)C(C1CC1)N(C(=O)CC1CCCC1)C(C)C 20269,c1(C(=O)NC(C(C)NC(=O)Cc2ccccc2)C)cc(OCC(C)C)ccc1O 20270,CCC(CC)CC(=O)N1CCN(C(=O)CCCC2CC2)C(C(C)C)C1 20271,C1(NC(C(C)OCC)=O)CCCCN(C(C2(C)CCN(C)CC2)=O)CC1 20272,C(=O)(C1CCC(=O)Nc2ccccc21)NC(CC)CNC(=O)C(C)CNC(N)=O 20273,Cc1nc(CO)ncc1NC(=O)C(C)N(C(C1CCN(C)C1)=O)C1CC1 20274,CCCCCCCCCCCC(=O)N(CC(C)NC(C1(OC)CCSC1)=O)C 20275,C1(NC(c2c(C)nc(C)[nH]2)=O)C2CC(CN(C(=O)CN3CCCC3C)C2)C1CO 20276,Cc1cccc2c(CC(=O)NC3COCC3NC(C3CC4(CCC4)C3)=O)c[nH]c12 20277,C1(C(=O)NCC2(C)N(C)C(=O)CC2)CCCN1NC(=O)C(O)CN(C)C 20278,C1(C(=O)O)(CNC(C(=O)NCC2CCCC(C#C)C2)=O)CC2(CC(F)C2)C1 20279,C(CC1=CCN(C(C2CC(=O)OC2(C)C)=O)CC1)NC(CC(C)CN(C)C)=O 20280,C1(C(=O)Nc2ccc(CC)s2)CN(Cc2nc(C)cs2)CCO1 20281,Cc1cc(C(F)F)oc1NC(C12CC1CN(C(=O)CSc1cnn(C)c1)C2)=O 20282,C1(C(N(C)C)=O)CCN(C(=NCc2cc(Cl)ccc2F)NCC2CCOC2)CC1 20283,CC1CCCN(C(c2c[nH]c(=O)cn2)=O)C1CNC(=O)C(O)CC1CCCC1 20284,Cc1ccc(C(F)(F)C(=O)NC2CCC(NC(C3CC(=O)N(O)C3)=O)CC2)cc1 20285,c1(C(=O)NCC2CN(C(=O)C(O)C3CCCC3)C2)cc(Br)c2occc2c1 20286,C=CCCCC(C(=O)N1CC(=O)N(C)C(=O)C1)NC(c1nc(C)ccc1C)=O 20287,O=C1NCCCCC1NC(c1ccc(I)cc1)c1nnnn1CCCF 20288,N1(C(CC(CC)OC)=O)CCC(N=[N+]=[N-])(C(=O)NCc2ccnc(C)c2)C1 20289,Cc1cc(NC2CCCNC2=O)ncc1S(=O)(=O)NCC1CC(=O)NC(C)C1 20290,O=C(CC1=CSC2=NCCN12)N1CCC(CCNC(=O)C(F)OC(F)(F)F)CC1 20291,c1(OC)ccc(C(N2CC(O)(CCCNC(=O)C(O)Cc3[nH]cnc3C)C2)=O)o1 20292,CCC(C(=O)N1CC2CC1(C(=O)NCCC1(COC)CCC1)C2)C(F)(F)F 20293,c1(CC)occ(C)c1C(=O)NCC1CCCC(NC(C2(CC)CCC2)=O)C1 20294,c1(C(=O)NCC(CN(C)C(C2CC2c2cnccn2)=O)O)cn2cnnc2cn1 20295,CN1CCC2(CCCN(C(c3ccc(S(C)=O)cc3)C(=O)NC(C)(C)C)C2)C1 20296,C(CCCN=[N+]=[N-])NC(C1(CNC(=O)COC(C)CC)CC(=C)C1)=O 20297,C1(C(=O)NCCc2c(C)n[nH]c2)C2CCN(C(=O)C(C)(C)C3CCOC3)CC12 20298,Cc1ccnc(-c2cn(CC(C3CN(C(C45CCCC4C5)=O)C3)F)nn2)c1 20299,Cc1c(C=CC(=O)NC2CC(C)N(C(=O)C3=CCCSC3)C2)cnn1C 20300,c1(N(C(c2ccc(C)cc2)c2ccccn2)CCO)ccc(F)c(C)c1Cl 20301,N1(C(C=COCC)=O)CCC2(C(=O)Nc3cccc(N4CCCCC4)c3)CC2C1 20302,CC1CN(C(=O)C(F)(F)F)CC(C)C1NC(c1nnn2c1CCC2)=O 20303,N1(C(C(CC)F)=O)CC2CCC(NC(=O)C3=CCOCC3)CC2C1 20304,c1(C(=O)NC2CCN(C(=O)Cn3cc(Cl)cn3)C(C3CC3)C2)noc2c1CCCC2 20305,C1(C#C)(C(=O)NC(C#C)C)CCN(C(c2cccc(=O)n2C)=O)CC1 20306,c1(CCCNC(C(COCC)N(CCCOC)C)=O)ncc(Br)cn1 20307,c1(C(N2CC3(OCC(NC(c4ccco4)=O)C3)C2)=O)c(F)ccc2occc12 20308,O=C(C#Cc1c(F)cc(F)cc1F)Oc1nnc(CC2CC2)s1 20309,S(=O)(=O)(C1CCCCC1)N1CCN(C(C2(C)CCN(C(=O)OC(C)(C)C)C2)=O)CC1 20310,C1(C(=O)NC2CCCC(C(N(CCCC(C)C)CC(C)C)=O)C2)CC2(C1)CC(O)C2 20311,C1(CNC(CCC(=O)N(C)C)=O)C(C2CC2)CCN1C(=O)CC1(O)CC1 20312,C1(CNC(CS(C)(=O)=O)=O)CC2(CCN(C(c3cccc(C#N)c3F)=O)CC2)C1 20313,C1(C(=O)NC2CCN(C(N)=O)C2)CC(N=[N+]=[N-])CN1C(c1cn[nH]c1)=O 20314,C1(NC(C(C)(C)C)=O)CN(C(c2n[nH]c3ccc(Cl)cc23)=O)C2(CCOC2)C1 20315,c1(C2CCN(C(c3cc(Cl)ccn3)C(=O)NC(C)C3CC3)C2)ccc(F)c(F)c1 20316,N1(C(c2c(CC)nc[nH]2)=O)CCC2(C1)CN(C(=O)Cc1cncnc1)C2 20317,N#Cc1ccc(C(=O)NC2CC2CNC(C2CCS(=O)(=O)C2)=O)o1 20318,CC(CN(C)C)CCC(=O)NCC(O)CNC(C12CCC(CC1O)C2)=O 20319,c1(C(=O)NCCCN(C(c2nccc(OC)c2F)=O)CC)cnn2c1CCC2 20320,C#CCCCC(C)C(=O)NCC1CC1NC(c1ccc(C(F)(F)F)nc1NC)=O 20321,c1(C(N2CC(NC(=O)CCOC(CCC)CC)C2)=O)cc2occc2[nH]1 20322,N1(C(C2CN(C)CC(C)O2)=O)CCOC2(CCN(C(=O)C3=CCCCCC3)C2)C1 20323,c1(OCC)cnc(C(=O)NC2CCC2NC(c2ccon2)=O)cn1 20324,C#Cc1ccc(C(=O)NCC(CO)NC(=O)C(C)OCC(C)C)cn1 20325,c1(C(N2CCCCC2)=O)cc2cc[nH]c(=O)c2s1.c1ccccc1-c1cn(C2CCOC2)nn1 20326,CC1C(NC(=O)C(C)NC(N)=O)CCCN1C(C1CC12CCCC2)=O 20327,C1(NC(c2scc(CNC(C(C(CC)C)N(C)C)=O)c2)=O)CCN(C)CC1(C)C 20328,c1(CCC(=O)NCCOC(CNC(C(C)CC2CCCC2)=O)(C)C)cccnc1Cl 20329,N(C1CCCc2cccc(C)c21)Cc1cc(C)cc(Cl)c1 20330,N1(c2nnc(C)n2CCCc2cccc(Cl)c2)CC(N2CCCC2)CC(C)C1 20331,N1(C(C(=O)NCCOC)=O)CCCC(C(=O)NCC23CC(C2)C(C)O3)C1 20332,c1(CN(C)C(C2CCCN(C(c3ccc(F)cc3Cl)=O)C2)=O)ccc(C#N)cc1 20333,C=CCC(C)(C)CC(=O)NCc1ccccc1CNC(C1NC(=O)CC1C)=O 20334,N1(C(C2C(=C)C2C(=O)OC)=O)CCC(C(=O)NCC(C)(C)O)C(O)C1 20335,O=C(N=c1nc(-c2ccsc2)[nH]s1)c1cncc(OC2CCOCC2)c1 20336,C1(NC(c2ccsc2)=O)CCCC1(C)NC(C1CCN(CC2CC2)CC1)=O 20337,C12(NC(c3cccc4nonc34)=O)CCCN(C(C3CC(F)(F)C3)=O)CC1C2 20338,Cc1cc(C(N2CCC(O)(CN(C(=O)CCc3nccs3)C)CC2)=O)nc(C)n1 20339,N1(C=O)CC2(CC=CC2)C1.C1(N2C(=O)C=CC2)CC(C)(C(C)(C)C)C1.C(CO)OC 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20604,C1(N(C(CCc2ncc(C)[nH]2)=O)CC2CC2)CCN(C(C2COC(C)C2)=O)CC1 20605,c1(C(N2C(Cn3cc(C=CC)nn3)CCCC2)=O)ccc2oc(N(C)C)nc2c1 20606,N1(C(C)C)CCCC(NC(=O)C(Cc2ccoc2)NC(=O)C(C)(C)CF)C1 20607,Cn1nc2n(c(=O)c1=O)CCN(C(=O)C(c1cc(Cl)ccc1F)(C)C)C2 20608,N1(C(=O)OCC2CCCCC2(F)F)CC2(CCC(C(=O)OC(C)(C)C)O2)C1 20609,CC(C)CC(O)C(=O)NCC=C1CCN(C(C2(C#N)CCC2)=O)CC1 20610,N1(C(C(c2ccccc2F)OC)=O)CCC(CNC(=O)CCCC(N)=O)C1(C)C 20611,c1(CCCC)ncc(C(=O)NC2CC2NC(c2nc(C(C)(F)F)cs2)=O)s1 20612,N1(C(c2c(C)nc[nH]2)=O)CCCC2(NC(=O)CCn3c(C)c(C)sc3=O)CC2C1 20613,c1(CNC(C2(C(C)C3CC3)CCC2)=O)nc(CNC(=O)CSC(F)F)cs1 20614,CC1CN(C(=O)OC(C)(C)C)CCC12CCN(C(c1cnc(N3COC3)s1)=O)CC2 20615,N1(C(C(C)=C(C)C)=O)CCC(O)(CNC(c2ccnc(-c3ccccn3)n2)=O)C1 20616,C(=O)(CCC(C)(C)C)N1C(CNC(C2N(C)C(=O)CC2)=O)CCC1 20617,Cc1ccc(N(C(=O)CSCCCCl)Cc2cccnc2)cc1F 20618,c1(C(=O)NCCCNC(CC(C)(C)SC)=O)noc2ccc(Br)cc12 20619,C1(NC(c2ccn(C)n2)=O)CCCCC12CCN(c1ncnc3[nH]cnc13)CC2 20620,Cn1cccc(CNc2ncnc(Cl)c2C#N)c1=O 20621,CC(Cc1cnn(C)c1)C(=O)N(CCCCNC(=O)C(C)Cc1ccncc1)C 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20640,CCC(C)CCCC(=O)NCCC1(NC(c2cn(C3CCC3)nc2C)=O)CCC1 20641,c1(CCC(=O)NCC(C)NC(C(F)CCOC)=O)ccc(OCC(F)(F)F)cc1 20642,C1(C(N(CCC(=O)OC(C)(C)C)CCO)=O)CCN(C(C2CC(Cl)(Cl)C2)=O)C1 20643,N1(C(C2N(C)CCN(C(c3scc(C)c3)=O)C2)=O)CCN2C(=O)OCC2C1 20644,CCC(CC(=O)NC1CC(NC(c2cccc(O)c2C)=O)CC1O)C(C)C 20645,C1(C)(C(=O)NCc2cc(COC)on2)CCN(C(C2CC(=O)CS2)=O)C1 20646,C1(C(=O)NC2C(OC)CCC2)(CO)CCCN(C(=O)CC2NC(=O)NC2=O)C1 20647,C1(C(=O)NC(CNC(C2(SC)CC2)=O)C(C)C)CCN(c2ccccc2)C1=O 20648,N1(C(c2c(NC(C(OCC)OCC)=O)occ2)=O)CCCC12CCNC2 20649,Cc1cc(F)ccc1C(=O)N(C)CC1CCCCN1C(C12CCC(F)(CC1)C2)=O 20650,c12cc3ccccc3cc1C(=O)N2.c1(C(N(CCOC)C2CC2)=O)ncnn1CC 20651,C1(C(=O)OC)CCC2CCC1N2C(=O)NC(=O)C(C)C.C12CCN(CC1C)C2 20652,Cc1n[nH]c(C)c1CCCNc1cccc(C(N)=O)c1 20653,N1(C(c2ccc(C)nc2)=O)CCC2CN(C(=O)CN3CCCC3C)C2C1 20654,Cc1ccc(C=CC(=O)N(CCC(C)NC(=O)CCc2cccnc2C)C)nc1 20655,Cc1cc(C#N)cc(C)c1O.C1(CN(C2CC2)C)CCCCN1C(c1n[nH]cc1Cl)=O 20656,c1(OC)cc(C(=O)NC2CCN(C(c3noc(C(C)C)c3C)=O)C2)ccc1O 20657,C(=O)(C(C)CCC(C)(C)C)NC(CC)CC(=O)NCC1(C(=O)OC)CC1 20658,c1(OC)cccc(Cl)c1NC(=O)CN1CC(CC2CCOC2)C2(CC2)C1 20659,CCC(C)(F)C(=O)N1CC2CC2(NC(=O)CCCc2ccc(F)cc2)C1 20660,C1(C(=O)NCCC2(O)CCN(C(C=CCCC)=O)CC2)C2CCC(C2)C1(C)C 20661,N1(C(C(C(C)C)N(C)C)=O)CCC(C)C(NC(C23CC4CC2C3C4)=O)C1 20662,c1(C(N2CCC(n3ccc(C(F)(F)F)n3)CC2)C(=O)NC)cc(C)nn1C 20663,C1(n2cc(C3N(C(C(C)CCN(C)C)=O)CCOC3)nn2)CCOC(C)(C)C1 20664,CCCCCC(=O)NCC(C)N(C(=O)CCNC(=O)NCC1CCOCC1)C 20665,c1(C(N(C)CC=CC(=O)NC2CCN(C)CC2)=O)cccc(O)c1F 20666,C(CCC(C)CNC(c1scnc1Br)c1nnnn1C1CC(F)(F)C1)OC 20667,C1(C(=O)NCc2ncoc2CCNC2CCC3CC3C2)C2CC3C(C2=O)C13 20668,c1(OC)nccc(C(=O)NCC(O)CN(C(=O)CC2CC3CCC2C3)C)n1 20669,CCCC(O)(CCC)CC(=O)NC(c1ccccc1)CNC(C1CC(OC)C1)=O 20670,c1(C(=O)NCC2C(C)CCN(C(c3cccc(C)c3)=O)C2)cnn2c1NCCC2 20671,c1(CNC(C=Cc2n(C)cnc2)=O)nc2c(s1)CN(C(C1CC13CCC3)=O)CC2 20672,c1(C(=O)NCC2C3CN(C(C(CC=CC)C)=O)CC32)ccc2c(c1)CC(C)(C)C2 20673,CP(C)(=O)c1ccc(O)c(NC(=O)NC2CCOCC2)c1 20674,c1(CN2CCC(N(C(c3c(OC)cccc3O)=O)C)C2)c[nH]c2ncccc12 20675,C1(C(=O)N(C2(CCC(N3CC(C)(OCC)C3)=O)CCCC2)CC)CCN(C)C1C 20676,C12(C(N(CC(C3CCC3)OC)C)=O)CCC(CC1)N(C(c1cn[nH]c1)=O)C2 20677,c1(CC(=O)NC2C(NC(C(CC)n3ccnc3)=O)CCC2)ccccc1N 20678,c1(N(C(=O)NC(C)CCc2ccccc2C(F)(F)F)CC)ccc(C(F)(F)F)cc1 20679,n1(CC(=O)NC2(C)CN(C(CCCC(=C)C)=O)C2)ncn2nccc2c1=O 20680,C1(C(=O)NCC2CC(O)C(O)C2)(CNC(C2COCCO2)=O)CC12CCC2 20681,N1(C(C(CC)c2cccnc2)=O)CCCN(C(=O)C=Cc2cnccn2)CC1C 20682,c1(C(N2CCN(C(COCC(=C)C)=O)C(CC3CC3)C2)=O)ccsc1S(C)(=O)=O 20683,CN1CC(C(N2CCOCC2CN(C(=O)CC2(O)CCCCC2)C)=O)CCC1=O 20684,CN=c1[nH]cc(C(N2CCN(CC(C)NC(C3(F)CCCC3)=O)CC2)=O)o1 20685,c1(CNCCOC(C(C(C)(C)C)c2cccc(C)c2)=O)cnn2ccncc12 20686,c1(C(=O)NCC2(O)CN(C(CNC=O)=O)C2)ccn(CC(F)(F)F)c(=O)c1 20687,C1(C(CNC(c2c(C)nsc2)=O)O)CCN(C(=O)C(C)C2CCOC2)CC1 20688,C(CCC(C)C(=O)ON(C)C)OC.C12CCC(CC1)CN(C)C2=O 20689,c1(OC(CSCC)=O)ccc(CNCCn2nc(C)oc2=O)cc1[N+](=O)[O-] 20690,N1(C(CC=CC)=O)CCC(NC(C2CCCC(NC(=O)OC(C)(C)C)C2)=O)CC1 20691,C=C=CCCC(=O)NCCCN(C(=O)CC1(N(C)C)COC1)C 20692,c1(OC)nc(C)cc(=NC(=O)C2CCN(C(c3ccc(O)c([N+](=O)[O-])c3)=O)CC2)[nH]1 20693,C#CC1CCCN(C(=O)C(C2CC2)NC(=O)CC2CCCN(C)C2)CC1 20694,C12(C(=O)NC3(CNC(C(C)(C)C)=O)CCCC3)CCCCC1C2 20695,C1(CNC(CCn2c(C)cc(C)n2)=O)CN(C(c2coc(CO)c2)=O)CC1(C)C 20696,Cc1cc(Cl)c(C(=O)NCC2CN(C(c3cc4occc4[nH]3)=O)CCO2)cc1N 20697,N1(C(c2cc(C)c(Br)s2)=O)CCC2(NC(c3cocn3)=O)CC2C1 20698,C(=O)(C(C(C)C)n1cc(Br)cn1)N(CCN1CCC1C(=O)N(C)CCOC)C.CC 20699,N1(C(C(=O)NCC2CCC(C(=O)OC(C)(C)C)CC2)=O)CCc2ccccc21 20700,N12CC(C3CCCN(C3)C(=O)CS1)C2.c1(CC)cc(C)nc(N2CCCC2)n1 20701,N1(C(CC2C(C)C2)=O)Cc2ccccc2C(NC(c2cc(CO)n(C)n2)=O)C1 20702,C1(NC(c2ccc(C)o2)=O)CC(O)CN(C(C2(C)C(C)(C)C2(C)C)=O)C1 20703,c1(CC)[nH]ccc1C(=O)NC(C1CC=CCC1)C(=O)NCC(c1ccco1)O 20704,c1(CCC(=O)NCCC2(NC(C3CC(=C)C3)=O)CC2)cccc(F)c1 20705,N1(C(C2(CC)COC2)=O)CC(n2cc(CNC(c3cscn3)=O)nn2)C(O)C1 20706,c1(OC)ccc(CC(=O)NCC(C2CC2)NC(=O)CCn2cncn2)cc1 20707,CC1CCN(CC(=O)N(CC(C)C(=O)N(C2CCCCCC2)C)C)CC1 20708,c1(COC)nc(-c2nc(Cl)c(CO)[nH]2)n(CCS(N)(=O)=O)n1 20709,C1(NC(CSCC)=O)COC2(CCN(C(c3cc(C)c(C#N)cn3)=O)C2)C1 20710,N1(C(C(C)=C2CC2)=O)CCC(CO)(CNC(C2CCC2(F)F)=O)C1 20711,c1(CC(N2C(C)C(NC(=O)CCC(=O)N(C)C)CCC2)=O)ccc([N+](=O)[O-])c(N)c1 20712,Cn1cc(C(=O)NCC(O)CN2CCc3ccccc32)c(=O)n(C)c1=O 20713,c1(C(N2CC(CNC(c3c(C)cns3)=O)C3(C2)CC3)=O)cc2c(C)cccc2o1 20714,C1(CC)CCN(C(c2cccc(O)c2)=O)C1C(=O)NCC(C1CC1)OC 20715,C(=O)(CCS(N)(=O)=O)N1CC(CC)C(C(=O)N(CC(O)CF)CC)C1 20716,C1(CNc2nccc(OCC)n2)CCCN(C(=O)CN2CCS(=O)(=O)CC2)CC1 20717,c1(C(=O)NCC2(C)CCN(C(C(CC)C)=O)CC2)ccc2nc(C)oc2c1 20718,C1(NC(COC(C)C)=O)CN(C(=O)CCCOC2CCCC2)CC1C 20719,C1(C#N)(C(=O)NC2CC3CC(NC(CC(CC)CC)=O)CC32)CC12CCCC2 20720,C(=O)(CC(C)(C)C(F)F)N1CC(CN(C(C(c2cnn(C)c2)C)=O)C)OCC1 20721,C(C(C)(C)C)N(CC(=O)NCCCNC(C1CC1C(N1CCCC1)=O)=O)C 20722,C(=O)(C1Cc2c(Cl)cccc21)Oc1ccccc1.CC1CN(C)C(=O)C2(CC2)N1 20723,c1(CN(CCOC)C(=O)Nc2cccc(-n3ccnc3O)c2)c(C)cccc1C 20724,c1(CNC(c2nc(O)nc(O)c2F)=O)cccc(C2=Cc3ccccc3C2)c1 20725,c1(OCC)c(C(=O)NCCN(C)C(C2(C)CC(O)CN2C)=O)cccc1F 20726,c1(OC)cccnc1C(=O)NCC1COCC1NC(=O)C=Cc1ccc(C)o1 20727,c1(OC)ccc2c(c1)C(C(=O)NCCNC(=O)CSC1CCC(C)C1(C)C)CC2 20728,c1(C(NC)=O)ccc(N)cc1.CC1CCN(C(c2csc(C)n2)C(=O)NCC(F)F)C1 20729,c1(C(N2CCCC(CN(C(C(C(C)C)F)=O)C)C2)=O)cccc2nc(O)ccc12 20730,CP(C)(=O)c1cncc(C(N2CCC(NC(c3cc(O)ncn3)=O)C2)=O)c1 20731,CN1CCC(C(CO)NC(c2conc2CNC(c2sccc2Cl)=O)=O)CC1 20732,C1(C(=O)NC(C=CC(=O)OC)C)CCCC2(CCC2)C1 20733,CC(F)(F)C(F)C(=O)N1CCC(C(=O)NCc2cc(CO)on2)(CF)C1 20734,CCC(C)(CNC(=O)CNC(=NCCF)Nc1cccc(C#N)c1)C(N)=O 20735,c1(C(N(C)C)=O)ccc(C(N2CCN(C(=O)CCc3nc[nH]n3)CC2)=O)cc1 20736,c1(C(N2C(C(=O)NC(CC#C)C(=O)NC)CC3(CC3)C2)=O)ccc2[nH]ccc2n1 20737,c1(CC)noc(CC)c1CC(N1CC(CNC(C2(C)CC3CC3C2)=O)C(C)C1)=O 20738,C1(OC)CCC(CNC(=O)CCCNC(=O)C(C)Cn2ccc(C)n2)C1 20739,C1(O)(C(C(=O)Nc2ncn(COC)c2)=O)CCOCC1 20740,c1(SC)ccccc1C(=O)N(C)CCN(C(=O)CC1CC(C)(C)CO1)C 20741,C1(C(=O)NCCCCC(C)NC(=O)CCN(S(C)(=O)=O)C)CNC(=O)C(C)(C)C1 20742,c1(C(N(C2CCN(C(c3ccc(OC(C)C)cn3)=O)C2)C)=O)cc(Cl)ccc1N 20743,c1(CC(N2CC(NC(CC(CCC)O)=O)C3(C2)CCC3)=O)cn2cc(F)ccc2n1 20744,C1(C(=O)NCC(C(=O)NC)C)C2CN(C(=O)CCC3CCCN(C)C3)CC12 20745,N12CCC(CC1)CNC(=O)C2=O.N1(CCN(CCC=C)CC)CCOCC1 20746,c1(C(=O)NC(C2CCN(C(C3COC3)=O)CC2)C)ccc2c(F)cc(F)cc2n1 20747,C(=O)(C(Cc1ccccc1)NC(=O)C(=O)NC1COC(C)C1)NCC 20748,c1(C(N2CC(CC(C)NC(C3(CCF)CC3)=O)C2)=O)coc(C(C)(C)C)n1 20749,C1(CC)CCCCN1C(=O)C(Cc1cn[nH]c1)NC(=O)C=Cc1cncs1 20750,c1(OC(C)=O)cccc(OC(C)CN(C)C(C2(OC)CCOC2)=O)c1.C1C(=O)N1 20751,CN1CCC(C(C)NCc2nncs2)C1 20752,N1(C(c2nnn(C)c2N)=O)CCCCC(NC(=O)COc2cccnc2Cl)C1 20753,Nc1c(C(=O)NCC=CCNC(=O)CCc2ccc(Br)cc2)cccc1F 20754,C(=O)(C1CCc2cc(Cl)ccc21)NCC1N(C(C2CCC(C)(O)CC2)=O)CC1 20755,C1(C(=O)NCC2C3CN(C(C4CCC45CCC5)=O)CC23)(OC)CCCCCCC1 20756,N1(C(C(=O)Nc2cc(N)cc(F)c2)=O)CC(S(=O)(=O)C2CCOCC2)C1 20757,C1(CC)C(NC(c2ncccc2SC)=O)CCCN1C(=O)C1=CCCC1C 20758,C(C)(C(C(=O)NCc1cn(CC(=O)NC2CCCC(CO)C2)nn1)N(C)C)OC 20759,CC#CCCC(=O)N(C)CC1CCCN(C(C2CN(C)C(=O)N2)=O)C1 20760,C1(NC(c2c(NC(C)=O)cccc2[N+](=O)[O-])=O)CCCCC(O)CNCC1 20761,C1(C(=O)NCCC(C(C)C)NC(=O)CC2(COC)CC2)CCCCN1N=O 20762,C(=O)(C1=CCC2(COC2)OC1)NC1C(NC(c2c(C)nccn2)=O)CCCC1 20763,C(=O)(C1CCc2cccnc21)NC1CCN(C(CCCSC)=O)CC1O 20764,C1(CN(C(=O)C(=O)NC2CCCCCC2)CC)CCCCC1OC 20765,C1(CCNC(=O)CC2OCCO2)CSCCN1C(c1cc(C2CCC2)[nH]n1)=O 20766,Cc1cc(C(=O)NCC=C2CCN(C(=O)CC(C)C3CCCO3)CC2)cc(C)n1 20767,Cc1ccc(C=CC(=O)NC(C2CCCN2C(=O)C(C)Cn2cccn2)C)cc1 20768,N1(CC(=O)Nc2cccc(CC)c2)CCc2c(ccc(C)c2Br)C1 20769,C12(C(=O)NC3CC(NC(Cc4nc(C)sc4C)=O)C(O)C3)CCC(CC1)CO2 20770,C(=O)(C(=O)CCc1ccccc1)N1C(CNC(COC(C)=O)=O)CC1 20771,N1(C(c2ccc(C)[nH]2)=O)CC=CC(C(N2CCC(O)C2C(C)(C)C)=O)C1 20772,CC(CCC(=O)N(C)C1CC1)NC(=O)CCNC(=O)CO 20773,N1(C(CC(C)(C)CO)=O)CCC2(CCC2)C(NC(C2CC(F)(F)C2)=O)C1 20774,C1(C(N2CCC(COC)(NC(=O)CCCF)C2)=O)OC(C)(C)OC1(C)C 20775,c1(CO)c(Br)cnn1C1CC2(N(C(=O)CCc3nc(-c4cccs4)no3)CC2)C1 20776,C1(C(=O)NCCN2CCNC2=O)CC2(CC2)CN1C(c1cccc(CCO)c1)=O 20777,c1(NC(C(C)NC(=O)OC)=O)oc(CNC(=O)CC2(COC)CC2)nc1C 20778,c1(C(=O)NC2C(C)N(C(=O)C=Cc3ccnn3C)CC2)ccc2c(c1)COC2 20779,c1(NC(C2CC(N(C(C3C(CC)C3)=O)C)C2)=O)ccc(SC)nc1 20780,C1(NC(CCC(=O)NC)=O)CCCCC12CCN(C(c1c[nH]nc1[N+](=O)[O-])=O)C2 20781,C1(NC(C2(CC(C)=O)CC2)=O)CN(Cc2cn(C)cn2)C2(CCOCC2)C1 20782,c1(N2CCN(C(C(Cc3ccc(C)cc3)=O)=O)CC2)ccc([N+](=O)[O-])s1 20783,C1(CN(c2nnnn2CCC2CCOC2C)CC)CCCN1Cc1ccccc1 20784,C(=O)(C#CC1CCOCC1)N1C(CNC(C(C)OCCN(C)C)=O)CC(O)C1 20785,CCCCCS(=O)(=O)CC(=O)NC1CN(C(=O)CCN2CCP(C)(=O)CC2)C1 20786,C1(C)(N(C)C)CCN(C(C2(CNC(C3(O)CCCC3)=O)CC23CCC3)=O)C1 20787,N1(C(C=C(C)C(F)F)=O)CCC(C(C)C(=O)N(C)Cc2cc(C)cs2)CC1 20788,N1(C(C(C2CCC(=O)N2)C)=O)CC(C)CN(C(=O)C=CC2CCC2)CC1C 20789,C1(CC(N2CCCC(NC(C(c3cccc(F)c3)C)=O)C2)=O)CCCCCCC1 20790,N1(C(c2c(COC)nn[nH]2)=O)CCC2(CC2NC(=O)C(C(C)C)NC=O)C1 20791,CC(C)(O)C(F)C(=O)N1CCC(O)(CCNC(C2CC(n3cnnc3)C2)=O)C1 20792,c1(CC)ccc(C(N2CCC(C(C)NC(=O)C(=Cc3ccccn3)C)C2)=O)cn1 20793,CC1(C)CN(C(C2CSC2)=O)CCC1NC(=O)C1=COCCO1 20794,c1(OC)nc(C(N2CCN(C)C(c3nc(C)no3)C2)=O)ncc1F 20795,c1(C(=O)NCC(C2CCOC2)NC(c2scc(COC)c2)=O)ncccc1F 20796,C1(S)CCCCN1C(=O)CNC1CC(N(C)C)C1.C1(NC)CC(F)(F)C1 20797,C12CC3(CC(C3)NC1=O)C2.C1(C(=O)NC)CC2CCC1O2.C1(C(CC)C)CNC1 20798,c1(NCC2CC(c3ccccc3)(OCC)C2)nc2ccccc2n1-c1ccccc1 20799,c1(C(N2CC(F)CC2CNC(CS(=O)(=O)NCC)=O)=O)cccc(F)c1NC 20800,C(C)(CCC(=O)NCc1cccc(C(=O)NC2CCN(CC3CC3)C2)n1)SC 20801,c1(CC)cccc(C)c1NC(=O)CC1CCC(NC(c2ccsc2)=O)C1 20802,Cc1ccc(CC(=O)N(CC(C)NC(=O)C(O)CC2CCCC2)C)c(F)c1 20803,CC1(C)CN(C(=O)Cc2cccnc2Cl)C(CNC(C2(C)CC2C(F)(F)F)=O)CO1 20804,c1(CC)cc(C)c(C(=O)NC2CC(NC(c3cn(CC(O)CC)nn3)=O)C2)o1 20805,c1(CC(=O)NC2C(C)N(C(=O)C3=CC(C)(C)C3)CCC2)c(F)cccc1C#N 20806,CCCCCC(=O)N1CC(O)CC1C(=O)N(CC(C)(CO)CO)C 20807,Cc1nn(C)c(C(F)F)c1C(N1CCC(NC(c2cnsc2)=O)C(F)C1)=O 20808,Cc1cc(F)cnc1-c1cn(CC(C)C(c2n[nH]c(O)n2)=O)nn1 20809,C(=O)(CC(C)CC(C)C)NCc1cccc(NC(c2c(OC)n(C)nc2C)=O)c1 20810,c1(CNC(CN(C(=O)C(C)CO)CC)=O)cncn1C(C)C 20811,c1(C(N(CC(CO)(C)C)C)=O)ccc(C(=O)NC2(OC)CCOC2)cc1.C(N)=O 20812,C(c1ccccc1Br)=CC(=O)NCC1N(C(C2CN(CC)C(=O)C2)=O)CC1 20813,O=C1CC(C(=O)NCCCC2CCN(C(=O)C(O)C(F)F)CC2)NC(=O)N1 20814,C(C)(c1ccccc1)=CC(=O)N(CC(CNC(COCCCC)=O)C)C 20815,C1(C(N2CCC(CC(F)F)C2)=O)(CC)CCN(C(=O)CCOC(C)C)C1 20816,N1(C(C2CCCN(C(=O)C(O)C3CCC3)C2)=O)CCOCCC1C1CC1 20817,Cc1c(Cl)ccc(C(=O)NCC2CCN(C(=O)C(C)n3ccnn3)CC2(F)F)c1N 20818,C1(NC(C(C)SC(C)C)=O)CC(C)(C(=O)NC(C)Cc2cc(C)[nH]n2)C1 20819,c1(C(=O)NC(C(C(=O)NCCOCC(C)C)C)C)cc(F)ccc1F 20820,C1(CNC(Cn2c(C)ccc2C)=O)CC2(CC(NC(C3CCNC3=O)=O)C2)C1 20821,Cn1cc(C(=O)N(C2CCCC(NC(=O)Cc3ccccc3)C2)C)c(O)nc1=O 20822,Cc1cc(C(=O)NC2CCC2CNC(=O)CNS(N)(=O)=O)cc(F)c1 20823,c1(CC(=O)NC(CNC(c2nc(C(C)=O)sc2)=O)C)ccc(C(F)F)cc1 20824,C1(NC(c2cc(SCC)ncc2)=O)CCCN(C(c2c(N)cccc2F)=O)CC1 20825,c1(C(N(CC(CC)NC(c2oc(C)nc2C(F)(F)F)=O)C)=O)cnc(O)cc1C 20826,c1(CC(=O)NCC2(C)CCN(C(CCCC(=O)OC)=O)C2)nnc2n1CCOC2 20827,C1(C(=O)NCCCC(C)(C)NC(C2=CCCC2C)=O)CCCCC(F)(F)C1 20828,C(=O)(C(C)(C)C(C)O)N1CCC(N2CCC(NC(COC(CC)(C)C)=O)CC2)C1 20829,C12(CNC(CCc3n(C)ncc3)=O)CC(CN1C(=O)CC1CCC(=O)O1)C2 20830,c1(CC)c(C(=O)Nc2cc(C#N)ccc2OC)cccc1C1=CCOCC1 20831,c1(N2C(CNC(CS(CC)(=O)=O)=O)CC3CCCC32)ncc(C)c(S(C)(=O)=O)n1 20832,c1(CC(=O)NCCCNC(c2ccc(F)s2)=O)nsc2ccccc12 20833,c1(C(=O)NC(C2CCOC2)CNC(C(CC)CC)=O)ncc(C)cc1C(F)(F)F 20834,N1(C(c2n(CCC)ccc2)=O)CCC(C)C1CNC(=O)CCOC1CCC1 20835,c1(C(N(C2CN(C(C34CC(C(F)F)(CO3)C4)=O)C2)C)=O)cnccc1Cl 20836,c1(C(=O)NC2CCC(NC(C(C=C)(C)O)=O)C2)c(F)cc(F)cc1Br 20837,C1(C(=O)NCC(C(C)(C)C)NC(c2coc(C(C)(C)C)n2)=O)(CC)CCCCC1 20838,C(=O)(CCCCC1CC1)NCCCN(C(C(C)N(C(C)=O)C)=O)C(C)C 20839,N1(C(CCC#C)=O)CC2CN(C(c3ccc(C#N)c(F)c3)=O)CCC2(CO)C1 20840,n1(CC(N2CCCSCC2C2CC2)=O)nc(-c2ccccc2)ccc1=O 20841,CC1(C(=O)NC2CCC(NC(c3ccnc(O)c3)=O)C2)CC2CC2C1 20842,C(C(C)(C)CNC(C12CCC1C2)=O)NC(C1(CC=C)CC1)=O 20843,C(c1cccc(F)c1F)=CC(=O)NCC(CN(C(C(C)c1ccco1)=O)C)O 20844,c1(C(N2CCCN(C(C(C(C)O)(F)F)=O)CC2)=O)nccc2[nH]ccc12 20845,n1(CC(=O)NC2CC(NC(=O)CSCC3CCCCO3)C2)cccc(O)c1=O 20846,C1(NC(c2nc(CCC)sc2)=O)CCN(C(=O)C(C)OCC(C)C)C12CC2 20847,c1(C(N2CCC(COC)(NC(=O)C(C(C)C)N(C)C)C2)=O)cnc(Cl)c(F)c1N 20848,c1(OC)ccc(C(C(=O)NCC(F)F)N(c2cccc(F)n2)CC2CC2)cc1OC 20849,c1(C(N2CC(C(n3cc(-c4ccc(Cl)s4)nn3)=O)C2)=O)cccc([N+](=O)[O-])c1Cl 20850,C(CCCCCC(=O)N1CC(NC(=O)CCc2ccsc2)CC(C)(C)C1)SC 20851,Cc1ccc(CC(N2CCC(F)(CNC(C3CCCOC3)=O)C2)=O)cc1Br 20852,N1(C(C2CC2F)=O)CCC(NC(C2(c3ccc(F)cc3)CCC2)=O)CC1 20853,C(N=c1ccc(S(=O)(=O)N2CCCC(c3cncn3C)C2)c[nH]1)c1c(C)n(C)nc1 20854,C(C)(CCC(=O)N1CCC(C)(CNC(c2cnc(-c3ccccc3)[nH]2)=O)C1)OC 20855,C(=O)(CCCCC(F)(F)F)N1CCC(CNC(C2CCN(CC)C2)=O)C(F)(F)C1 20856,c1(OC)cccc(Cl)c1CC(=O)NC(C)CCNC(c1ccnn1CC#N)=O 20857,N1(C(C(CC=C)(C)C)=O)C2CCC1CC(NC(=O)C=Cc1nc(C)c(C)[nH]1)C2 20858,C1(NC(C(COC)C)=O)CC(C)N(C(=O)CCC(=O)c2ccc(OC)cc2)C1 20859,C(=O)(C(CC(F)F)N(C(=O)Cn1cc(C#N)cn1)C)N(CC#C)CCF 20860,Cc1cccc([N+](=O)[O-])c1NC(C)CCNC(C1CC1C)=O 20861,c1(C(=O)NCCC(=O)NCC(C=C)(O)CCC)c(C)ccc(C)c1N 20862,C=CC(C)(CC)C(=O)NC1CN(C(c2coc(OCC)n2)=O)C(C)(C)C1 20863,C(=O)(C(C)CCC(C)(C)C)N1CCCC(CNC(C(C)c2ncco2)=O)C1 20864,c1(-n2cc(CN(C(c3ccc(CC)cc3)=O)CCO)nn2)cccc(F)c1Br 20865,c1(C(=O)NCCC2N(C(CC3C(CC)C3)=O)CCOC2)c(Cl)cncc1Cl 20866,c1(NCC2(O)CCN(C(Cc3cccc(C)c3F)=O)CC2)cc2nncn2cn1 20867,Cc1ccc(C(=O)N(C2CC(NC(=O)C(F)n3cccn3)C2)C)c2ccccc12 20868,c1(N(C)C)ncc(C(N2CCCC(CNC(=O)C(F)CC3CCCC3)C2)=O)cn1 20869,CC(C(=O)NC(CC1CC1)CC(=O)NCc1ccnn1CC1CC1)C(F)F 20870,C(C(C(C)(C)C)NC(=O)CCC(F)F)NC(C(C1CCC(=O)N1)C)=O 20871,N1(C(C(C(C(CC)C)O)C)=O)CCC2(CC1)CCN(C(C13CC(F)(C1)C3)=O)CC2 20872,C1(NC(c2cnn(CC(F)F)c2)=O)CCC(NC(C2(O)CCOC2)=O)CC1 20873,N1(C(c2cnc(C(C)C)nc2)=O)CCN(C(=O)Cc2cncnc2)C2(CC2)C1 20874,c1(NC(C(=O)NC2C(=C)CC2)=O)ccc(CC(F)F)cc1 20875,c1(OC)cc(C(N2CCC(F)(C(=O)Nc3cnc(C(C)C)nc3)C2)=O)nn1C 20876,Cc1cc(CNC(=O)NCc2cnn(C(C)(C)C)c2)on1 20877,C1(CCNC(=O)C#CC2CC2)CCN(C(C2(C3CCCO3)CC2)=O)CC1(F)F 20878,c1(CC(C)C(=O)NCC2CN(C(=O)CN(C)C)CC2O)ccc(Br)cc1F 20879,N1(C(=O)CSC(F)(F)F)CCC2(CCCCN(C(c3ccc(F)o3)=O)C2)C1 20880,C1(C(=O)NC2C(NC(C3(C)CC=CC3)=O)COC2)CCC2(CCOCC2)O1 20881,C1(C(=O)NCC2C(CNC(COCC=C)=O)C2)CCC(C(=O)OC)O1 20882,C1(C)(NC(C2(C)CCOC2)=O)CCN(C(C2CCNC(=O)C2)=O)CC1 20883,C1(NC(c2nnc(C(C)C)s2)=O)CCC2CN(C(=O)CCc3cn[nH]c3)CC2C1 20884,c1(OCC)ccccc1C(N1CCC(N(C(=O)CC(C)(C)c2cccs2)C)C1)=O 20885,C=CCCN=C(NCC(C(C)(C)C)OCC1CCCSC1)NCC(C)(C)C 20886,CCCCCCCCC(=O)N1CCCC(C(=O)OCc2ccoc2C)C1 20887,C1(C(=O)NC2(CC#C)CC2)CC2C=CC1N(C(=O)C(C)(C)C(=O)N(C)C)C2 20888,Cc1cc(Cl)c2c(c1)CCN(c1nccc3ncn(C)c13)C2 20889,C(=O)(CCC1CCc2ccccc21)Nc1cc(NCC2(C)COC(=O)OC2)ncn1 20890,C(=O)(C1CC(=O)c2c(F)cccc21)N1C2CN(C(c3[nH]c(=N)sc3)=O)C(CC2)C1 20891,c1(CSC(C(=O)NCC(=C)Cl)C)cccnc1N1CCCC1 20892,C(=O)(CC(C1CC1)NC(=O)CCCN(C)C(=O)CC=C1CCCCC1)NC 20893,C=C(C)CCC(=O)N(C1CCN(C(C2(c3[nH]nc(C(=O)OC)c3C)CC2)=O)C1)CC 20894,CCC(C(=O)N1CCC(NC(c2ncccn2)=O)C1)C(C)(C)CC 20895,C(CC(C)C(=O)NC1(CCNCCC(=O)OC)CCCC1)OC 20896,C1(C(=O)NC(CC)CN(C(C2CCCN(C(C)=O)C2)=O)CC)CC(=O)NCOC1 20897,c1(C(CC)OCCN(C(C(=O)NC(=O)C2CC2)C2CC2)C)ccccc1 20898,N1(C(C(C)(C)NS(C)(=O)=O)=O)CCC(NC(C2CCOC2)=O)C1C(C)(C)C 20899,N1(C(CCc2c(C)noc2)=O)CCC(C)(C)C1CNC(c1cc(F)cc(F)c1)=O 20900,c1(C(=O)NCC2CCNCCO2)ccn2c(O)nnc2c1 20901,c1(CC(N2CCC(NC(COC(CC)CC)=O)C2C2CC2)=O)cc(F)ccc1C 20902,n1(CC)ccc(C(=O)NC2CC(O)C2CC(=O)NC2(COC)CCCCC2)c1C 20903,CC1(C)CCC(O)(C(=O)NCC(O)CNC(C2CCC=CO2)=O)CC1 20904,N1(C(CCCC=C)=O)CCC2(CC1)CN(C(=O)C(C)(C)C1CC1)C2 20905,c1(COC)ncc(C(=O)NC(C)(C)C(C)NC(C2C(C)C2C)=O)c(=N)[nH]1 20906,c1(CC)nn[nH]c1C(N1CCC1(C)CC(=O)NCCP(C)(C)=O)=O 20907,c1(C(N2CCC(CNC(C(C)NC(=O)OC)=O)C2)=O)cn(CCC(C)C)nn1 20908,C1(CNC(C2(CC(=O)OC)CCC2)=O)CCCCCN1C(C1CC(=O)CCO1)=O 20909,c1(C(=O)NCCC(C)N(C)C(C2CC(O)C2)=O)c[nH]c2cc(Br)ccc12 20910,c1(N(CC(CN(C)C(C2CCCCN2C)=O)O)C)snc(Cl)c1C#N 20911,Cc1nncc(C(N2CC3CCC3(C(=O)NCC(c3nc[nH]n3)C)C2)=O)c1C 20912,c1(C(N(CC(C)(C)C(=O)NCC2CC2)C(C)C)=O)cn2ccnc2s1 20913,C(C)(C)(CCC(=O)N1CCCC(NC(c2nn(C)nc2Br)=O)C1)OC 20914,CC(C(=O)N(CC(C)(C)NC(=O)C(Cc1ccccc1)C(C)C)C)P(C)(C)=O 20915,CCCCCC(C(=O)NC1CC1NC(=O)CN1CCCCC1=O)C(C)C 20916,c1(C(C(N2CC(C)C(NC(=O)C3=CCCC3C)C2)=O)=O)ccc(F)cc1F 20917,c1(NC(Cc2ncc(C)s2)=O)ccc(F)c(C(F)(F)F)c1C(=O)O 20918,c1(CC(C(N2CC(NC(Cc3nc(C)[nH]n3)=O)(CO)C2)=O)C)ccccc1C 20919,c1(C(N(C)CC2(CNC(C3(O)CCOC3)=O)CC2)=O)ccc(C2=CCCC2)cc1 20920,C1(NC(c2c(C(C)C)cno2)=O)CCC2(CC1)CN(Cc1cnn(C3CC3)c1)C2 20921,N1(C(c2cc(C(F)(F)F)cs2)=O)CC2CCC1CN2C(C1CC1Br)=O 20922,c1(C(C(N2CC(C(=O)NCC(=O)NCC)C(OCC)C2)=O)O)ccc(Cl)cc1F 20923,C(CCOCCO)(C(=O)N(c1ccco1)C)NC(=O)CC.C=CC1CN1 20924,c1(CC)ccc(CN(C(CO)CC(=O)OC)C(C)C)cc1.N12CC3(CC3C1=O)C2 20925,C1(C(N2C(CNC(C34C(C)OC(C)(C3)C4)=O)CCCC2)=O)CCc2ccnn2C1 20926,Cc1ccc2c(c1)c(C(C)NC(c1cc3c(o1)CCCC3)=O)cn2C 20927,C(=O)(C1CCc2ccccc21)NC1(C2CCN(C(C3(C)CC(=C)C3)=O)C2)CC1 20928,C(CS(=O)(=O)CC(=O)NCC1CCCC1NC(=O)C=Cc1ccoc1)OC 20929,C1(C(=O)NCCC(C)N(C)C)C=CC(NC(=O)CC(=O)OC)C1 20930,c12cc(ccc1Cl)CC(=O)C2=O.c1(SC)nnnn1CCS.C1(N)CC1F 20931,FC1CCCCCC1N=c1[nH]c(=NCC2CCCC3(CCC3)C2)[nH]c2c1COC2 20932,N1(C(=O)OCC)CCC(CC(=O)NC(CNC(=O)CCCC2CC2)C(C)C)C1 20933,C1(NC(c2cc(C3CC3)cs2)=O)C(C)CN(C(CN(CC)CC)=O)CC1C 20934,C=CCN=C(NCc1cnn(CC(C)C)c1C)NC1CC12CC2(F)F 20935,N1(C(C(C2CCCCC2)C)=O)CCC(NC(=O)Cc2csc(S)n2)C1C(C)(C)C 20936,CC1C(NC(N)=O)CCCN1C(=O)CNC=O.C12(CC1)CC(=O)N2 20937,C1(C(=O)NCC2(OC)CN(C(=O)C(C)N3CCCC3)C2)CC2(CCO1)CC2 20938,Cc1nn(C)c(C(=O)NC2CC3(C2)CC3NC(=O)C(C)(C)C(=O)NC)c1[N+](=O)[O-] 20939,C1(NC(c2occ(C)c2)=O)CCCCC1CNC(C1CCC(C(N)=O)O1)=O 20940,C1(OC)CC(CCNC(C2CC2(F)F)=O)N(C(c2cnc(C3CCCC3)s2)=O)C1 20941,C1(C(N(CC(CC)NC(c2c[nH]nc2-c2ccco2)=O)C)=O)C(C)C1(F)F 20942,N1(C(c2cc(C)ns2)=O)CC2(CC(CNC(c3ccncc3C(F)(F)F)=O)C2)C1 20943,CCCCC(O)Cc1nc(C2CCCC2)nn1CC(C)CC 20944,CC1(C)CCCC1C1CCN(C(N2CCCC3CC(O)CCC23)=O)C1 20945,C1(C(N2CCC3(NC(CNC(CN(C)C)=O)=O)C(C2)C3)=O)CCc2nnnn2C1 20946,c1(C(N2C(C(N3CCC(O)CC3)=O)CCCC2)=O)cc(Cl)ccc1I 20947,c1(OCC)ccc(C(=O)NC(C)(C)CNC(c2nccc(CO)n2)=O)cn1 20948,C1(NC(=O)C(F)C2CCC2)CCCCN(C(c2cnc(C(F)F)cn2)=O)C1 20949,CC1(F)CC(N=c2[nH]c(N3C4CCCC3COC4)nc3c(F)cccc23)C1 20950,C(N=c1nc(N2Cc3cnn(C)c3C2)c2ncccc2[nH]1)c1c(C)ccnc1O 20951,C1(C(=O)NC2(CCOC)CC2)CCN(C(C2CCCCC2C)=O)C12CC2 20952,c1(N2CCn3c(nc(C)n3)C2)nc(=NC(C)C)[nH]c2c1SCC2 20953,CC1(C)NC(=O)CCC1NC(C1CNC(=O)CN1C(=O)C1=CCCCC1)=O 20954,c1(OC)cc(F)c(C(=O)NCCC(C)NC(=O)CCC2C(=O)NN=C2C)c(Cl)c1 20955,c1(CC)c(C(=O)NCCCN(C(=O)CC(C)(C)SC)CCSC)nnn1CC 20956,c1(C(C(F)(F)F)NCCN(CC(F)F)C)cc(F)ccc1C 20957,C1(C2CCN(C(=O)C(F)(F)CC3CC3)CC2)(NC(c2c(COC)ncs2)=O)CC1 20958,c1(OC)ccc(F)cc1NC(C1CC1C(=O)Nc1ccc(Br)c(F)c1)=O 20959,C#CCC(CC(=O)OCC)NC(=O)CC(=O)OC(c1cc(C(C)(C)C)ccn1)=O 20960,c1(COC)ccccc1C(=O)N(O)Cc1cn(CCCNC(=O)N(C)C)nn1 20961,c1(OCC)cccc(NC(C2CCN(C(c3conc3CSC)=O)CC2)=O)c1 20962,c1(C(=O)NC2(COC)CN(C(=O)Cc3ccsc3C)C2)cnc2c[nH]nc2c1 20963,CC(CC(=O)NCC1CN(C(c2ccc(F)c(F)c2)=O)CC1O)P(C)(C)=O 20964,Cn1cnc2cccc(C(=O)NC3CC(NC(C4(c5cc[nH]n5)CC4)=O)C3)c12 20965,N#Cc1ccc(CCC(N2CCCC(NC(=O)Cc3nccs3)C2)=O)nc1 20966,N1(C(CS(=O)(=O)N(C)C)=O)CC(C(F)(F)F)OCC1CNC(=O)Cn1ccnn1 20967,C(CCCCCCCO)=CC(N1C(CCNC(CCCC#C)=O)CSCC1)=O 20968,N1(C(CCN2CCN(CC)CC2)=O)CC(O)C(O)C1CNC(=O)CCCCCO 20969,C1(NC(C(CC)OCC)=O)C2CCCN(C(c3cncc(F)c3)=O)C2C1(C)C 20970,CCC(C)CC(=O)NC(CNC(=O)C(C)NS(C)(=O)=O)C1CC1 20971,C(=O)(CC(O)c1ccccc1)NC1C(NC(C(F)=CCC)=O)CC1 20972,CC1CCC(F)(C(=O)NC(C)CCC(=O)N2CC(O)C(O)C2)CC1 20973,Cc1cc(OCCCN2CCCC2=O)ccc1N1CCCC1=O 20974,C=CCC(C)(C)CCNC(C1CC(CCNC(=O)C(C)(C)C(=C)C)C1)=O 20975,N1(C(c2c(CCC)nns2)=O)CCN(C(c2ccc(C(C)F)cc2)=O)CC1CC 20976,C(=O)(C1CCCn2cncc21)NC(CNC(c1sc(C)c(O)n1)=O)C 20977,C(=O)(C(O)CC(C)C)NC1CCC(N(C(CCOCCOC)=O)C)CC1 20978,S(=O)(=O)(c1cccc(NC2COCC2C(N)=O)n1)N1CC(C)C(F)C1 20979,C1(C(=O)NCC(N(C)C(C2CC(F)C2)=O)C2CC2)CCOC(C)(C)C1 20980,N1(C(C(C)(C)OC(=O)C(F)(F)F)=O)CCN(C(=O)CC#N)C(C=O)C1 20981,C(=O)(C(C)(C)CNC(C1CC1C#N)=O)OC 20982,C1(C(N2CCC(C(CNC(=O)CCc3cn[nH]c3)F)CC2)=O)CCC(F)(F)CC1 20983,c1(N(C)CC2CN(C(C3(CC)CCCCO3)=O)C2)cc(C)nc2ncnn12 20984,n1(C(C)(C)C)ncnc1CCCC(N)=O.c1(NC(C(=O)N)=O)cnn(C)c1 20985,N1(C(C2CN(S(CC)(=O)=O)C2)=O)CC2CCCC2(NC(C2CC2(C)C)=O)C1 20986,CC1=C(C(=O)NCC2C=CCN2C(C2CCCC(=O)CC2)=O)CCO1 20987,CC(C)CCCC(=O)NC1(CF)CCN(C(c2coc3c2CSC3)=O)C1 20988,CC(C(=O)N1CC2CC2(NC(=O)CC(=O)NC2CC2)C1)C(C)(F)F 20989,C1(CNC(c2[nH]cc(CC)c2)=O)CN(C(c2ccnn2COC)=O)CCN1C 20990,C(=O)(CCCCCCS(N)(=O)=O)NC1CC(NC(C(C)OCC#C)=O)C1 20991,C1(C(N2CC(OC)C(C(N3CCC(C)(N(C)C)C3)=O)C2)=O)CCC2(CC1)CC2 20992,c1(C(N(C2CCN(C(=O)CCC3CC3(C)C)C2)CC)=O)n[nH]c2c1CCC2 20993,C#CCC(O)C(=O)NCC(C1CCCCN1C(C1CC(O)CN1C(N)=O)=O)(C)C 20994,S(=O)(=O)(CC(=O)N1CCC(C2OCCC2NC(=O)C(O)CSC)CC1)NCC 20995,c1(OC)c(CN=C(NCc2nccn2C)NC2CCN(C3CC3)C2)cccc1Cl 20996,N(C1CCc2ccccc21)C(C1CCC(CNC(c2cc(C)nn2C)=O)CC1)=O 20997,C(CC(N)=O)(C(=O)NCC(=O)NC1(Cl)CCC1)NC(CC(C)C)=O 20998,C1(NC(C(C)N(C(C2(CCC=C)CC2)=O)C2CC2)=O)CC(=O)N(C)C1=O 20999,c1(SC)ncccc1NC(=O)CC1CCN(C(c2[nH]c(C)nc2C)=O)C1 21000,C1(CC)CCCN(C(=O)CCN(c2cnccn2)C)C1NC(=O)C=C(C)C(C)C 21001,C1(CNC(C=COCC)=O)CN(C(=O)C(C)CN(C)C(=O)OC(C)(C)C)CCO1 21002,c1(C(N2C(C(N3CC(C#N)(CF)C3)=O)CC2)=O)nc2ccccc2s1 21003,N1(C(CC2CCC(C)CC2)=O)CC2CC(C(=O)NCC3COCCO3)(C2)C1 21004,c1(C(C)(C)C)ccc(F)cc1F.n12cc(nn1)C(=O)NC2C1(C(=O)OC)CCCC1 21005,C12CN(CCC1NC(c1coc(C(F)F)n1)=O)C2=O.C1(C)(C(C)C)CCC(=O)C1 21006,c1(C(=O)NCC(C2CC2)NC(C2(F)CCS(=O)(=O)C2)=O)cc2n(n1)CCCN2 21007,Cn1nc(CNC(C2CC(O)C(F)C2)=O)cc1C(=O)NCCC1(C)CCCO1 21008,c12cc(c3[nH]c(O)nc3c1)NC2=O.N1(C(C=CC)=O)CCC(CCOC)(OC)C1 21009,N1(C(COS(C)(=O)=O)=O)CCC(C(=O)OC)(OC2CC2)C1.C12(CC1)CNC2 21010,CC(C)C(C(=O)N(CCCCN1CCCC1)C)NC(=O)C(C)Oc1ccccc1 21011,CN1CCCC(O)(CC(=O)NC2CC(CO)N(C(c3cc(Cl)ncc3O)=O)C2)C1 21012,c1(C(N(C2CC(NC(C3COC(=O)N3C)=O)C2)C)=O)ncncc1Cl 21013,C1(NC(c2c(Br)cncn2)c2nnnn2C2CCOCC2)COC2(CCC2)C1 21014,CC(C)C(C(=O)Nc1cccc(Cl)c1)c1ccn(C)n1.C12(CC1)CNC(=O)N2 21015,CC(C)CC(O)C(=O)NC1CCN(C(=O)CN2CCN(C)CC2)C1C(C)(C)C 21016,C1(CNC(c2ccc(CC)[nH]2)=O)CC2COCC2N1C(c1c[nH]c(C)cc1=O)=O 21017,N1(C(C)=O)CCC(NC(=O)C(C(C)C)NC(C2CC(=O)C2)=O)CC1 21018,C1(COC)C=CCCN1C(C1CCN1C(=O)C=CCN1CCC1)=O 21019,N1(C(C)=O)CC(NC(=O)CCNC(C2CCCN(CC)C2)=O)CC12CCC2 21020,C1(NC(=O)CC2CC(F)CN2C(c2ccc(CO)o2)=O)CNC2(CCC2)CO1 21021,N1(C(C2CCN(C(C)=O)CC2)=O)CC(C)CN(C(c2cc(N(C)C)no2)=O)CC1C 21022,Cn1c(C(=O)NC2CCCN(C(c3ccc(S(C)(=O)=O)s3)=O)C2)ccc1[N+](=O)[O-] 21023,N1(C(C(C2CCC2)OCC)=O)CCC(C)(CCNC(c2c(Cl)nsc2Cl)=O)C1 21024,C1(NC(c2c(OC)nsc2)=O)CC(C(=O)NC2CCNC(=O)C2)C1(C)C 21025,C1(O)(CNC(C(C=C)(F)F)=O)CCCN(C(C2CCN(S(C)(=O)=O)C2)=O)C1 21026,c1(NC(c2occc2-c2ccccc2)=O)ncc(Br)cc1F.C12CC1CNC2=O 21027,CC1CCCCC1CC(=O)NC12CC(CNC(=O)C(N3CCC(C)CC3)=O)(C1)C2 21028,CC1CCN(CC(=O)NCSc2ccccc2)C(NC(c2nnnn2C)C)C1 21029,c1(C(=O)NCCC2CC(Nc3nc(C)cc(CC)n3)C2)c(O)nnc2c1CCC2 21030,C1(C(=O)N(CC2CNC2)CC2CCCO2)(COC)CCC1 21031,C(CNC(=O)Nc1ccc(N(C)Cc2cncc(C)n2)cc1)(C(F)(F)F)OC 21032,Cc1sc(O)nc1C(=O)N(CC(C)NC(c1cnc(-c2ccsc2)s1)=O)C 21033,c1(COC(=O)CSCC(N2CCCCC2)=O)ccc(Cl)o1 21034,CCCCCCCC(=O)NCC1(F)CCN(C(c2cnc(N(C)C)nc2)=O)CC1 21035,C(c1ccn2ccnc2c1)=CC(=O)NC1CCC(CCNC(C=C(C)C)=O)C1 21036,N1(C(CCC2CCN(C(=O)CCc3nncs3)CC2)=O)CC2CCCCC12 21037,c1(OCC)ncc(C(=O)NCCC(O)CNC(=O)CCC2CCCOC2)s1 21038,N1(C(C(n2ccc(C)n2)(C)C)=O)CCC(C(C)NC(=O)C=CBr)CC1 21039,CCS(=O)(=O)CC(=O)NCC(C)(C)CN(C)C(C1CC2CC(=O)C1C2)=O 21040,C1(CC(=O)NCCCOCCNC(=O)CC2CCOC2=O)Cc2ccccc2S1 21041,c1(C(=O)NCC2(Cn3cc(CO)nn3)CCC2)ncsc1CCCc1ccccn1 21042,C(=O)(C1CCCc2scnc21)NCC1C2N(C(c3ncc(C)cc3F)=O)C(CC2)C1 21043,C(=O)(CC(O)CC(C)C)N1CC(C(NOCC2C(=C)C2)=O)C(O)C1 21044,N1(C(c2cn(CCC)nn2)C(=O)NCc2cccs2)CCCCC1.C1(COC)CC1 21045,CC1(C)NC(=O)OC1CNC(=O)C(c1cccs1)NC(=O)CN1CCNC1=O 21046,N1(C(c2cncc(C)c2C)=O)CCC2CN(C(=O)C(O)C3CC3)CC12 21047,c1(-c2c(C)ccc(C3CC3)c2)ccc2[nH]c(C(N3CCC(O)C(C)C3)=O)nc2c1 21048,C1(NC(C(CCC)OC)=O)CC2CCC1CC2NC(=O)CN(C)CCC 21049,N1(C(C)=O)CCOCC1C(N1CC(CO)(NC(c2cn(C)nc2C(C)C)=O)C1)=O 21050,CCC(CC(=O)N1CCC(NC(=O)Cc2ccon2)C(O)C1)C(C)C 21051,C12(CNC(C(C)OCC=C)=O)CC(NC(=O)C=Cc3ccncn3)(CO1)C2 21052,N1(C(C2C(C(N)=O)C2)=O)CC(CNC(c2ccc(=O)n(CCO)c2)=O)CC(C)(C)C1 21053,C1(CCNC(CC(C)SC)=O)CCN(C(c2cc[nH]c2)=O)CC1 21054,c1(C(N2CC(CNC(c3cccc(OC)c3N)=O)C2)=O)ccn2cnnc2c1 21055,c1(CC)ccc(C=CC(N2CCN(CCNC(C3CCCC3C)=O)CC2)=O)cc1 21056,N1(C(=O)CCCCC2CC2)CCCN(C(C2C3CCC2(c2ccsc2)C3)=O)CC1 21057,C1(CNC(C2(C)CC2)=O)CN(C(=O)COc2ccc(CC#N)cc2)C2(CCC2)C1 21058,c1(C(N2C(C)CCC(CNC(CC(C(=O)OC)C)=O)C2)=O)ccn2cncc2c1 21059,CN1CCOC2CN(C(=O)C3=CCN(C(C4CCOCC4(C)C)=O)C3)CC12 21060,C=CC1OCCC1C(=O)NCCCCC1CN(C(=O)CCc2cncc(O)c2)C1 21061,c1(C(=O)NC2CC(CNC(c3oc4ccccc4c3Cl)=O)C2)ccc2nncn2c1 21062,Cc1noc(Cl)c1CC(N1CC(C(=O)NCc2cc(CC3CCC3)[nH]c2)C(C)C1)=O 21063,c1(C(N2CC(C(N3CCC(O)C(F)C3)=O)CC(C)C2)=O)ccc([N+](=O)[O-])cc1O 21064,c1(C(n2cc(C(c3nnnn3C)NCC(C)C(C)C)nn2)C)ccncc1F 21065,N1(C(C(=O)N(CCCCNC(C2(OC(C)C)CCOC2)=O)C)C)CCN(C)CC1 21066,c1(C(C)O)ccc(C(=O)NCC2CCCCN2C(=O)C(F)=CC2CC2)cc1 21067,C(=O)(CCCC(=O)NCC(C)N(C)C(c1cccc(C2CCC2)c1)=O)OC 21068,N1(C(c2cc(COC)no2)=O)CCCC(N(C)C(C2(C=O)CC2)=O)C1 21069,C1(CNC(c2c(CC)cno2)=O)CN(C(=O)C2=CC(C)(CC)C2)C2(CCOCC2)C1 21070,Cn1[nH]c(=NC(=O)C(C)(C)c2cnn(-c3ccccc3)c2)cc1-c1ncco1 21071,C=CCCCCN(C)C(C1(n2cccc2)CCCC1)=O 21072,C1(COC)(NC(=O)C(c2ccc(F)c(Cl)c2)C)CCN(C(=O)C2=COCC2)CC1 21073,c1(CC)n[nH]cc1CNC(=O)C=CC(C)(C)NC(=O)C(F)=C(C)C 21074,C1(O)(CN(C(=O)CC2CCCO2)C)CCN(C(C2CC3C=CC2C3)=O)CC1 21075,C(CC(C)C(F)(F)F)NC(C(CC1CCC1)NC(c1nc(C)sc1C)=O)=O 21076,C1(C(=O)NCCC(CCNC(C(C)=CC)=O)C)CC1C1(C)CCOCC1 21077,C(C(CC(C)C)C(=O)NC1(C(=O)NCC#CC(F)(F)F)CC1C)OC 21078,c1(C(=O)NC2CC3(C(NC(c4c(C)occ4)=O)C3)C2)cc2c(o1)CCCC2 21079,C1(NC(=O)NCC(CSC)(C)C)CCC2(CC1)CC2C#N 21080,C1(COC)(CNC(C2CCC2(C)C)=O)CCN(C(c2cc(Cl)nnc2O)=O)CC1 21081,C(CC(F)F)(C(=O)N=c1ccn(CC2CC2)[nH]1)N(C(C1C(C(=O)OC)CC1)=O)C 21082,c1(CCC(=O)OCc2ccc(N)cc2)cccc(Br)c1F 21083,c1(C(N(CC(CC)NC(c2sccc2C(F)F)=O)CC)=O)cc(OC)cnc1F 21084,C12(C(N(C(CC)CC)CCO)=O)CCC(CC1)N(C(=O)CSCCC(C)C)C2 21085,C1(N(C(=O)C(=O)NCCOC2CC2(F)F)C)CCCC1C(C)(C)C 21086,c1(C(=O)NC2COCCN(C(C(COC)(C)C)=O)C2)ccc2ccccc2c1F 21087,Cc1ccnc(C(C)NC(=O)C(=O)N(CCn2cc(Cl)cn2)CC2CC2)c1 21088,N1(C(CCc2cnc(C)o2)=O)C(C)CC2CN(C(=O)C(F)F)CC12 21089,C1(C(=O)NCCc2cn(C)cn2)(CNC(C(C=CC)O)=O)CCCCC1 21090,c1(C(N2CCOCC2c2nc[nH]n2)C(=O)NCCC)ccc(C)c2c1CCC2 21091,N1(C(C=Cc2oc(C)c(Br)c2)=O)CC2CCC(C1)N(C(c1ccnn1C)=O)C2 21092,CS(=O)(=O)C1(C(N2CC3(CCN(C(=O)CC(C4CC4)C4CC4)C3)C2)=O)CCCC1 21093,N1(C(CCN(CC=C)C(C2CC2F)=O)=O)CCC2(CCCO2)CC1 21094,C(=O)(CCC(C)(C)NC(=O)CCCC1CCC1)NCCCN(C)CCO 21095,C1(C(=O)NC2C(NC(Cc3nc(COC)sc3)=O)CC2)Cc2ccccc2O1 21096,c1(SCC)cnccc1C(=O)NCCC(C(C)C)NC(=O)C=CC1CCCN1C 21097,Cc1cc(C)c(CC(=O)NC2C=CCN(C(c3n[nH]cc3C)=O)C2)c(C)c1 21098,C1(NC(CNC(=O)OCC=C)=O)C2CC1CN(C(C1(OC)CCC1)=O)C2 21099,N1(C(c2ccn(C)n2)=O)CC(CNC(=O)COc2cnn(C)c2)C2CC12 21100,N1(C(C=C(CCC)C)=O)CCC(C)(C(=O)NC(c2cnn(C)c2)CO)C1 21101,CC12CC(NC(C3CCC3)=O)(C1)C1(CCN(c3ncnc(Cl)c3[N+](=O)[O-])CC1)O2 21102,c1(C(=O)NCC2C(CC(=O)N(CC#C)C)C2)cnc(N)cn1 21103,N1(C(c2cccc(CC=C)c2)=O)CC(C)C(NC(=O)CS(=O)(=O)N(C)C)C(C)C1 21104,CCC(C)(CCC(=O)OC)NC(c1cc(CCN)on1)=O 21105,C1(O)(CC(=O)NCc2ccc[nH]2)CN(C(c2ccsc2)=O)C1 21106,N1(C(CCC)C(=O)NCCCC(=O)OCC)CC(C)CCC12CC2 21107,C(=O)(C1CCCc2nnn(C)c21)NC(CNC(CCC(C)C)=O)CC(F)(F)F 21108,C1(C(=O)NC(CN(CC)CC)C)CCN(C(c2n[nH]c(C)c2Cl)=O)CC1(C)C 21109,C1(CC)CN(C(C2CCCCN2N=O)=O)CC(C)S1=O 21110,N1(C(C(c2cn(C)nc2)NC(=O)NC2OCCCC2(C)C)=O)CCc2ccsc2C1 21111,c1(C(=O)NC2CCN(C(C(CC)NC(N)=O)=O)C2(C)C)ccc2c(n1)CCCN2 21112,C12(C(N3CC(C(CC)CC)OCC3)=O)CC(C1)C(C)(C(=O)O)C2 21113,CCCC(CC)CCC(=O)NC1C(C)(C)C(NC(=O)CN2CCCCC2)C1(C)C 21114,Cc1ccc2c(c1)CC(Sc1nnc(-c3ccc(F)c(F)c3)s1)C2 21115,C(=O)(CC(C)CC(F)(F)F)N(C1CCN(C(C2OCCO2)=O)C1)CC 21116,C1(CC)C(C(=O)NCc2n[nH]cc2C(=O)NC2CC=CC2)CCN1C 21117,N1(C(c2c(COC)nn[nH]2)=O)CC2CC1CN2C(C1CC1OC(C)(C)C)=O 21118,C(CC1=CCN(C(=O)C(C)=C2CC2)CC1)NC(C(CCC)CC1CCCCC1)=O 21119,N1(c2nccc(C)n2)CC(NC(C2CC(n3cc([N+](=O)[O-])cn3)C2)=O)CCC1C 21120,N1(C(C(COC)(C)C)=O)CC2(CCC(CNC(C3(NS(=O)(=O)C(F)F)CC3)=O)O2)C1 21121,c1(C(N2C(CCNC(CCSCCCC)=O)CCC2)=O)cn(C)nc1OC 21122,C(CC(C)(C)C(=O)N1CCC(C(C)(C)C)(CNC(=O)C(F)C(F)(F)F)C1)SC 21123,c1(C2N3CCN(CC3)CCC(=O)C2=O)ccc2cccnc2c1.C(CCF)S.CO 21124,c1(C(N2CCC(Cn3cc(CC(C)C)nn3)C2)=O)nn2c(c1I)CCCC2 21125,C1(NC(N(C)Cc2csnc2Br)=O)CCCN(c2cnn(C)c2)C1=O 21126,C1(CC(=O)NC(C#C)C(C)OC)CN(C(=O)CCC(C)OC)CC1C 21127,n1(CC)cc(CC(=O)N(C(C)CNC(=O)Cc2cnc(C)s2)C)cn1 21128,C(C)(C)(CC(=O)N1CC(OC(=O)NC(CF)C(F)(F)F)C1)NC(C)=O 21129,C(=O)(CC(C)(C)NC(=O)CC1CCCN1C)N(C)CC1CCCC1 21130,c1(C(N2CCC(NC(C3(C)CCC(C)C3)=O)C2C)=O)cnn2c1OCC2 21131,C1(C)(CNC(Cc2nc(CC)sc2)=O)CC(F)(F)CN1C(=O)C(CO)OC 21132,N1(C(C(C)SC)=O)CCC(C)C(CNC(c2nccc(Cl)c2C)=O)C1 21133,c1(C(C(=O)NC(CC=C)c2cn(CC(C)C)nn2)OC)ccc(F)cn1 21134,C12CC(C13CCC3)COC2=O.CC1COCC(C)N1C(=O)OC(C)(C)C 21135,C=CC1(NC(C23CC(CN2C(c2sccc2Br)=O)C3)=O)CCCC1 21136,Cc1cccc2oc(N3CCCC34CCN(C(=O)OC(C)(C)C)C4)nc12 21137,C#Cc1ccc(F)c(C(N2CCC(CNC(C3CCC(C)(C)OC3)=O)CC2)=O)c1 21138,c1(C(C)NC(Cc2cnc(C)o2)=O)ccc(S(C)=O)cc1 21139,N1(C(C(C)Cn2ccnc2)=O)CC2CN(C(C3(C)CC3(F)F)=O)CC2C1 21140,C1CCCC(=O)NCCO1.C(CCC(C)c1cn[nH]c1)NC(C=CC)=O 21141,c1(C(=O)NC(C(C)NC(C2CCCN2C=O)=O)CO)ccc(Cl)c(N)c1Cl 21142,c1(OC)ccc(CNC2CN(C(c3csc(C)n3)=O)CC2C)c(C#N)c1 21143,C(CCN(C)C(C1CCS(=O)CC1)=O)(C(C)C)NC(C1(OC)CC(C)C1)=O 21144,C=CC1CN(C(c2cc(C)c(C)s2)=O)CC1NC(C1C(C)(C)OC1(C)C)=O 21145,C(C)(CCCC(=O)N1CC(N2CCNC2=O)C1)NC(c1[nH]cc(C)c1C)=O 21146,C(=O)(C(CC(F)F)NC(c1ccc[n+]([O-])c1)=O)NC(CCC)CCO 21147,CCC(C)C(O)C(C)C(=O)NC1C2CC1CN(C(=O)C(O)Cc1ccccc1)C2 21148,C1(CNC(CC(C)OCCC)=O)C2CCCC1N(C(c1cccc(O)c1F)=O)C2 21149,C1(CNC(C2CC(O)(NC(=O)OC(C)(C)C)C2)=O)CC2CC(C1)CC(F)(F)C2 21150,CCCC(C)(C)CNC(=O)CC1(NC(=O)Nc2cnn(C(C)C)c2)CC1 21151,c1(C(=O)NC(C23CCC(CC2)C3)CNC(C(C=C)O)=O)ccc2[nH]ccc2c1F 21152,c1(C(N(CC(CNC(C(COC)(C)C)=O)C)C)=O)ccc(Cl)nc1Cl 21153,C(c1ccc(CC)cc1)=C(C(N1C(CNC(CCOCC#C)=O)CCC1)=O)CC 21154,C#CCC(O)C(=O)NC(CC)C(=O)N1CC(OCCC=C)C1 21155,CC1(C)COCC(C(=O)NCC2(F)CCN(C(=O)CCN3CCOC3=O)C2)O1 21156,CCC(CCOC)C(=O)OC1CCN(c2ccccc2C#N)C1=O 21157,Cc1cnn(CC(=O)NC2CC(CNC(c3coc(C(N)=O)c3)=O)C2)c(=O)c1 21158,c1(C(=O)NC2(COC)CCN(C(c3cncs3)=O)C2)c(C)oc2nc(Cl)ccc12 21159,C(=O)(CC1=CCCC1)NC1CCCN(C(c2c(C)nsc2Br)=O)C1 21160,C1(C)(C(=O)NCC2C(NC(C3C(C(=O)OC)C3)=O)C2)CCc2ccccc2C1 21161,C1(CNC(c2c(C)nc(C(C)C)o2)=O)C2CCC(C2)N1C(=O)CCn1cccn1 21162,C1(C(N2C(CNC(CCCCOCC)=O)CC(O)C2)=O)(OC)CCC(C)(C)C1 21163,C1(NC(CC(C)SC)=O)CCC(C)N(C(=O)C(C)CC2CC2)C1 21164,c1(C(=O)NC2CCN(C(CCc3ccc(C)cc3C)=O)C2)ccc2snnc2c1 21165,c1(OCC)ccc(Br)c(NNC(=O)C2Cc3c(F)cccc32)c1 21166,C1(O)(C(F)(F)F)CC(=O)N2CC1C2.Cc1cnc(CCC(=O)OC(C)(C)C)cn1 21167,c1(-n2cc(C(C)NC(C3CC3(Br)Br)=O)nn2)cccc(Br)c1 21168,C1(C(=O)NC2CCC2CNC(=O)C(F)(F)c2ccccn2)CCCC1O 21169,N1(C(c2c(C(C)C)scn2)=O)CCCCCC(NC(=O)C2=CCCS2)C1 21170,CCCCC(C)CCC(=O)NCC(C1CCOC1)NC(=O)CC#N 21171,c1(C(=O)NC)cccc(C(=O)NC(C)CC(C)NC(c2coc(C#N)c2)=O)c1 21172,Cc1cncc(-c2cccc(C(=O)NCCC3(O)CCCC3)c2)n1 21173,N1(CC)CCCCC1C(=O)NCC1CCC1C(=O)NCCCc1nnnn1C 21174,CC1CN2CCN1C(=O)COC2=O.c1(NC(=O)C(F)C2CCC2)ccccc1F 21175,CC(C)(O)C(F)C(=O)N1CCOC(CNC(C2CCCCO2)=O)C1 21176,C(=O)(CCOCCCNC(=O)Cc1cc[nH]c1)CC1(NCC(C2CCCC2)C)CC1 21177,c1(OC)cccc(CNC(c2cccc(NCn3cc(NC(C)=O)nn3)c2)=O)c1 21178,c1(C(=O)NCC2CC2C(=O)N(CC(O)CO)CCO)csnc1Cl 21179,C1(NC(CC=C(C)C)=O)CCCCCN(C(c2ccc([N+](=O)[O-])o2)=O)C1 21180,S1(=O)(=O)C2=CC=CC(=NC3CC3CN1)N2.N1(CCSC(C)C)CCCCC1 21181,C1(NC(=O)C(C2CCN(C(COC3(C)CCCCC3)=O)C2)F)CC2C(C1)C2(C)C 21182,CC1(C)OCc2c1n[nH]c2C(=O)NCC1CC(NC(=O)C(F)CC2CCCC2)C1 21183,c1(C(=O)NC2C(NC(COCCCCC)=O)CCC2)c2ccccc2nn1C 21184,c1(CN(C(=O)CC(C)(C)n2cc(C3CCCOC3)nn2)C)ccc(Cl)nc1 21185,CC1(CO)CNC(=O)CSCC(=O)N1.c1(NC(=O)C(O)CF)cccnc1 21186,c1(C(C)C(=O)NCCCCCCNC(C2(C)CCC2)=O)c(Cl)cccc1Cl 21187,C(=O)(C1CCOc2ccccc21)NCC(C1CCCN1C(C1C=CCC1)=O)(C)C 21188,C(CC(=O)NC(C)CCCCO)(C(C)C)NC(C1(OCC)CCCC1)=O 21189,c1(C(=O)NC2(COC)CCN(C(C3(C)CCCC3)=O)C2)ccnc(Cl)c1O 21190,C1(NC(C2(CNC(=O)CC3CCCC3)CCCO2)=O)CCCCCC1F 21191,c1(NC(=O)C(N2CCC3(C2)CC3(F)F)=O)nc2ccccn2c1C1=CCOCC1 21192,c1(CNC(CSCC#C)=O)cc(C(=O)NCC2(C#N)CC2)no1 21193,c1(C(N2CCN(C(CC=C)=O)C(C)CC2)=O)cc(Cl)cc2nc(C)[nH]c12 21194,N1(c2snc(CC)n2)CC(C2CCCCN(C(=O)CC3(C)CCCO3)C2)C1 21195,S(=O)(=O)(c1ncccc1C#N)NCC1CC(C(=O)OC(C)(C)C)C1 21196,c1(C(=O)NCC2(CCNC(COC(C)C)=O)CC2)cncc2c(O)nccc12 21197,CCC(CC)CC(F)C(=O)NC(C12CCC(CC1)C2)CNC(=O)C(C)(C)O 21198,N1(C(CSC)=O)CC2CCCCC2(CNC(c2cccc(C(=O)N(C)C)c2)=O)C1 21199,C#CCC(O)C(=O)NCCCN(C(=O)C(O)(c1ccccc1)C1CCCC1)C 21200,N1(C(C(CCC)CC)=O)CCCCCC(NC(=O)CN2CCC(C(N)=O)CC2)C1 21201,Cc1cncnc1C(N1CCCC1CC(=O)NCC(C)C#N)=O 21202,C1(N(C)C)CCCC1NC(=O)C(C)(C)C1CCCN1C(=O)CCN(C)C 21203,C1(CNC(c2ccc(OC)nc2)=O)CC(C)CN(C(=O)C(C2CCC(=O)N2)C)C1 21204,NS(=O)(=O)C1(C(=O)NC2CC(c3cn(CC4(O)CC5CCC4O5)nn3)C2)CCC1 21205,Cc1nc2ccc(C(=O)NCC3C4CN(C(c5csc(C)c5)=O)CC34)cc2s1 21206,N1(C(c2cc(Cl)c(O)cc2O)=O)CCC2(CC1)CCN2c1ncnn2cccc12 21207,C1(CC(N2CC(n3cc(CNC(C45CCCC4C5)=O)nn3)C2)=O)CCCCC1O 21208,C1(O)(C(C)NC(=O)CSCc2cscn2)CCN(C(=O)C(CO)N(C)C)CC1 21209,c1(CCC(N2C(C)C(NC(c3coc(Br)n3)=O)CCC2)=O)nc2ccccc2o1 21210,C(CCCCCNC(=O)CCNC(C1CCC1)=O)NC(c1ccc(O)nn1)=O 21211,Cn1nc(C(F)(F)F)c(Br)c1CN1CCC(C)(CO)CC1 21212,C1(NC(C=C(COC)C)=O)CC(=O)N(C2CN(C(=O)Cc3c[nH]ccc3=O)C2)C1 21213,C1(C)(CNC(C=CC(C)(C)SC)=O)CCC(NC(C2(F)CCCC2)=O)C1 21214,C1(C(N(CCCNC(CC=C)=O)CC)=O)CCOC1SC1CCCCC1 21215,C1(C(N2C(C(=O)NCC3CCOC3)CC=CC2)=O)CC2(C1)CC2(F)F 21216,C1(NC(=O)CCn2ccnc2)CCC2(CCN(C(c3csc(Cl)c3Cl)=O)CC2)C1 21217,c1(OC)cccc2scc(C(N3CC4CCCC4(NC(C4CC4(F)F)=O)C3)=O)c12 21218,c1(N(CCCOC(c2ccccn2)C)C)[nH]c(=NC2CC2F)nc2c1ncn2C 21219,C1(C2CCN(C(c3cncnc3CC)=O)C2)(NC(CCC(=C)Cl)=O)CC1 21220,C(CNC(=O)COC1CCN1)(C(F)(F)F)NC(=O)OC.c1(C(C)O)nc(C)no1 21221,CCS(=O)(=O)C(C)(C)C(=O)N1CCOC(C)(CNC(c2cnn(C(C)C)c2)=O)C1 21222,C1(c2c(C(=O)OC)c[nH]n2)CC2N(C1)C(=O)C1(COCC)CC1OC2C.OC 21223,C1(NC(c2cc(C(=O)OC)ncc2)=O)CN(C(=O)C(F)C(F)(F)F)CCC1F 21224,CC(C(=O)NCC1CCN1C(c1cncc(F)n1)=O)C(C)(F)F 21225,c1(OC)cccc(NC(=O)C(c2cc(C)on2)N2CCC(C3OCCO3)C2)c1 21226,C1(C(=O)NCC2COCCN2C(=O)Cn2ccnc2)CCC2(CC1)OCCO2 21227,C1(CNC(C=C(CC)CC)=O)(CO)CCCN1C(C1(CCN(C)C)CC1)=O 21228,C1(C)(C(N(CC(C)NC(C2CCN(C)S2(=O)=O)=O)C)=O)CCC(F)(F)CC1 21229,C(=O)(CC(=O)NCCNC(c1cocc1C)=O)NCC 21230,N1(C(C)C(=O)NC(C2(C)CC(N3CCCC3)C2)C)CCN(C)CC1 21231,N1(C(C(C)(C)C(F)F)=O)CCCC(O)(CNC(C23CCC(C)(CO2)C3)=O)CC1 21232,c1(C(N(CCC(=O)NCC(C)(C)NS(N)(=O)=O)C)=O)cc2cccn2cn1 21233,c1(NCC2CCN(CCCC)C2)nccc(CC(=O)NC)n1 21234,O=C(CCC(=O)c1cccs1)NCC(O)CCNC(c1ccn(C2CCC2)n1)=O 21235,c1(C(=O)NCc2cc(C)oc2C)cc2cc(Cl)sc2[nH]1 21236,c1(COC(C2CCCN(C3CCNC3=O)C2)=O)ccc(I)c(F)c1 21237,C1(NC(C(CC)OC)=O)CN(C(=O)CSC(F)(F)F)CCC1(C)C 21238,C(=O)CC(C)(C)CC(=O)OC.C12CCCN(C1)c1ccc2cc1.CC 21239,C1(NC(CCCc2cc(C)no2)=O)CCN(C(=O)C(C)SC(F)(F)F)CC1O 21240,C(=O)(C1CCCc2ccnn21)N(CCNC(c1nc2nccc(C)n2n1)=O)C1CC1 21241,c1(C(=O)NCC2CCN(C(C=C(C)C(F)F)=O)CC2)ccc2c(C)nn(C)c2n1 21242,c1(-c2ccc(C)cc2)ccc(S(=O)(=O)N(C)Cc2onc(C)n2)cc1.C(=O)O 21243,C1(NC(c2n(C=C)nnc2)=O)CN(C(=O)C2=COCCO2)C(C)(COC)C1 21244,Nc1ccc2c(C(N3CCC(NC(=O)Cc4cnoc4)C(CO)C3)=O)c[nH]c2c1 21245,C1(CNC(C(C)NS(C)(=O)=O)=O)CCCN(C(C2CCC(F)(F)C2)=O)C1 21246,Cn1[nH]c(=NC(=O)C2CCCN2C(C2(CO)CCC2)=O)cc1Cl 21247,C1(CC)N(c2ccc(C3CCCN3C(C)=O)nn2)CC12CCCC2 21248,N1(C(c2c(C)nc(CC)o2)=O)CCOC(C)(CNC(=O)CCOC2CC2)C1 21249,N1(C(Cc2c(C)n[nH]c2)=O)CC2CC(NC(c3nnn(C)c3N)=O)C(C2)C1 21250,N1(C(C(C(C)O)Nc2ccccc2)=O)CC(S(=O)(=O)N2CCCC2)C1 21251,C(=O)(CCC(N)=O)NCc1c(C2CCN(C(C3(C)COC3)=O)C2)n[nH]c1 21252,C1(c2c(OC)cc(Br)cn2)NC(=O)N(CC2CCCO2)C2=C1C(=O)NC(C)C2 21253,C(=O)(CCc1ncc[nH]1)N(C)CC1(NC(CC2(COC)CC2)=O)CC1 21254,C1(CC=C)CCCN(C(=O)N(CCOC)CC2CCCCC2)C1 21255,C1(C2C(C)=CCS2)CC2(CCCC2)C1.Cc1nc(C)c(-c2ccc(C(=O)N)s2)o1 21256,C1(CCOC)CCCCN1C(=O)C(=O)NCc1nccnc1C(F)F 21257,c1(C(CC)C)cc(C(=O)NC(c2ncc(-c3cccs3)[nH]2)C)on1 21258,N1(C(CCC#C)=O)CCc2nc(CNC(c3ccnc(N(C)C)c3)=O)sc2C1 21259,c1(C(=O)NC(C)CCNC(=O)C=CC2CCCC2)cnc2ncnn2c1O 21260,N1(C(C#CC(=O)N(C)C)=O)CCN(C(=O)CCC2CCCCO2)CC1C1CC1 21261,CCC(C(=O)N1CC(OCC(N)=O)C1)NC(c1cc(C(N)=O)[nH]n1)=O 21262,C1(NC(CC(CCC)C)=O)CCC2CN(C(=O)C(C)(C)C)CCC2C1 21263,n1(CC)nnnc1C(CC1C=CCN1C(=O)OC(C)(C)C)NCc1ccccn1 21264,CC(C)(C)C(C#N)C(=O)NCCC1(C)CCN(C(C2CC3(CCC3)C2)=O)C1 21265,c1(CC)cnn(CCNCCC2CC(NC(=O)C(C)O)C2)c1 21266,N1(C(C(C)OCC=C)=O)CCC2CN(C(c3cccc(C)c3OC)=O)CC12 21267,CCC(C)(C)CC(=O)NC1CCCC(NCCNC(c2ccc(F)cn2)=O)CC1 21268,N1(C(CCc2cc(C)no2)=O)CC(N(C(=O)COC(F)F)C)C(O)C1 21269,C1(CCS(=O)(=O)N)CC2CCC1CC2CC(F)(F)F.CC(=O)N(CCCCC)C 21270,Cn1nc(C2CC2)cc1C(C1(CN=[N+]=[N-])CC1)=O 21271,c12cccc(F)c1CN1CC3C(C1)N23.c1(C)ccnc(Cl)c1C.COCO 21272,CC(C)CCCCC(=O)N1CC(C(=O)NCC2CC23CC3)CCC1(C)C 21273,Cc1cc(CC(=O)N(C(C)C(=O)NC2CC=CCC2)C2CC2)no1 21274,CN1CCCC(C(N2CCC(O)(CNC(C3CC3(C)Br)=O)C2)=O)C1 21275,n1(C(C)C(C)(C)C)nc(-c2cccc(Cl)c2)nc1C1CC2CC2C1 21276,C=C=CC(C)C(=O)NC1(C)CCN(C(C2CC(=C3CCC3)C2)=O)C1 21277,Cc1csc2ncnc(N3CC4C(NC(C5CCC(C)(O)CC5)=O)C4C3)c12 21278,N1(C(c2cnn3c2OCC3)=O)CC2CCC(C1)N2C(c1cnc2n1CCC2)=O 21279,C12(CCNC(C3CC(SC)C3)=O)CCC(CC1)N(C(c1cncn(C)c1=O)=O)C2 21280,C(C(=O)NNC(=O)c1[nH]nnc1C1CCNC1)SC 21281,c1(N2CCC(C)(CC)C2)ccc(S(=O)(=O)NCc2ncccc2F)cn1 21282,CCC(C)(C)C(O)C(=O)N1CC(N(C(=O)C(c2ccc(F)c(F)c2)=O)CC)C(C)C1 21283,c1(C(=O)NC2(C)CC(NC(c3c(N)cc(F)cn3)=O)C2)ccc(S(=O)C2CC2)cc1 21284,Cc1ccc(C)c(C(N2CC(CNC(=O)CC=CC(C)(C)C)C(O)C2)=O)c1 21285,C1(OCCC)CCN(C(=O)CC2CC(C)N(C(c3cccc(CO)n3)=O)C2)CC1 21286,c1(CCC)cc(C(=O)NC2CC(CNC(C3(C)C=CCCC3)=O)C2)ccn1 21287,C1(NC(c2c[nH]nc2-c2ccco2)=O)CCN(C(=O)COC2CCCOC2)CC1 21288,c1(CNC(NCc2ccc(C)cn2)=NCCC(C)=O)cc2c(cc1Cl)OCCO2 21289,C1(NC(CCC=CC)=O)CCCN(C(c2cn(CCc3cccs3)nn2)=O)C1C 21290,CN1CCCC(C(N2CCCC(CN(C)C(c3ccncc3F)=O)C2)=O)C1 21291,c1(C(=O)NC2CC(C)(NC(c3cc(CC)c(C)s3)=O)C2)ccn2nncc2c1 21292,C1(C(N2CC(OCC)(CNC(=O)C(C)(C)NC(=O)CC)C2)=O)CCCN1N=O 21293,C1(NC(c2ccc(OC)nc2)=O)C2CCN(C(=O)CCn3cnnn3)C2C1(C)C 21294,c1(C(=O)NC2CN(C(c3c(C)cc(SC)o3)=O)C(C)(C)C2)ccc(F)cc1C#N 21295,C(CCC(C)(C)C(=O)N1CCCC(C(C)C)CC1)NC(C(CCCC)O)=O 21296,C1(CNC(=O)CC2CC=CCC2)CCN(C(C2(C3CCCO3)CCC2)=O)CC1O 21297,c1(NC(c2ccc(-c3ccc(C)o3)cc2)=O)ccc(Cl)c(Br)c1Cl 21298,N1(C(c2c(SCC)cc(C(F)(F)F)cc2)=O)C2CCC1CN(C(C1CC1F)=O)C2 21299,C1(C(=O)NC(C)CN2CCN(C(C3CC4(CSC4)C3)=O)CC2)CCC(=O)C(C)C1 21300,N#CC1CCN(C(=O)CC2(NC(=O)CC3CCOC3)CC2)C1 21301,c1(C(N2CCC(NC(CCCN(C)C)=O)(CO)CC2)=O)ccc2nonc2c1 21302,CC1CC2(CC(NC(=O)CC(C(F)F)NC(c3cccc(Cl)c3)=O)C2)C1 21303,O(N1C(=O)c2ccccc2C1=O)CC(=O)NCC(C)CNC(C1(F)CC1(C)C)=O 21304,c1(C(N(CCN(C(C(CC)SC)=O)C)C)=O)nc(-c2ccco2)sc1C 21305,N1(C(C2N(N=O)CCCC2)=O)CC(NC(=O)C(F)(F)C(F)(F)F)CC2(CC2)C1 21306,N1(C(C(C2CCOCC2)OCC)=O)CCC(C)(NC(=O)C(C)(C)CO)C1 21307,c1(OC)cc(C(N2CCC(C)C(CNC(=O)Cn3cc(C)cn3)C2)=O)c(Cl)cn1 21308,C1(NC(C(CC)=CC)=O)CC2(C1)CC(NC(C1CCC(C)(CC)O1)=O)C2 21309,C1(CC#C)CCCN(C(c2cccc(-c3cnco3)c2)=O)CC1 21310,N1(C(C(=O)Nc2ccccc2)COCCCC2CC2)CCCC(F)CC1 21311,C(=O)(C(C)(F)C(C)(C)F)Nc1c(F)ccc(SC(COC)C)c1 21312,CC1=CC(NC(=O)CCC2CC(NC(C3(C#N)CC3)=O)C2)CCC1 21313,N1(C(c2n(C)ccc2)=O)CCOCC(CNC(=O)CC2CC3C=CC2CC3)C1 21314,C12CCCN(C1)CCCNC2=O.c1(CN(C)C)nc(=N)s[nH]1 21315,CC(CCNC(C1(S(C)(=O)=O)CC1)=O)CCNC(=O)CS(=O)(=O)N1CCOCC1 21316,c1(C(=O)NCC(C)N(C)Cc2ccsc2)cccc2oc(O)nc12 21317,c1(OCC)cc(OC)cc(NC(N2CCN(c3nc(C)ns3)CC2)=O)c1 21318,C(C(C(=O)NC1CC1CN(C)C)C(C)C)NC(CNC(CCC)=O)=O 21319,c1(N2CCC(=C)C2)ccc(S(=O)(=O)NCC(N2CCCCOC2)COC)cc1Cl 21320,c1(C(c2n(CC(=C)C)nnn2)NC(c2ccccc2F)CF)noc2c1CCC2 21321,N1(C(C(CC=C)(C)C)=O)CC(NC(C2(CF)CCC2)=O)CC(C)(C)C1 21322,c1(C(=O)NCCCN(C(C(C(CC)(C)C)OC)=O)C)c(C)cnc2ccccc12 21323,N1(C(c2c(C)cn(C)c2)=O)Cc2[nH]nc(C(N3CCCC3CCN(C)C)=O)c2C1 21324,C(=O)(CCCC(=O)NOC(C)(C)C)NC(C(C)NC(CC=C)=O)C 21325,C1(NC(c2cnnn2C2CC2)=O)CC2CC(C1)N(C(C1SC3C=CC1CC3)=O)C2 21326,c1(C(=O)NC(C2CCN(C(c3cn(CC=C)nn3)=O)C2)(C)C)cc(Cl)cn1C 21327,C1(NC(C(C)(C)n2cccn2)=O)(CNC(=O)C=C(Cl)Cl)CCC(F)(F)CC1 21328,N1(C(CNC(CNC(C)=O)=O)=O)CCCC2CN(C(=O)C(F)=C(C)C)CCCC12 21329,C(C(F)(C(=O)N1CCCCC1CCO)C(C)C)NC(C(C)=NOCC#N)=O 21330,N1(C(C(=O)NCCC(=O)OCC)c2cnc[nH]2)CCC(C)(F)CC1 21331,N1(C(C(C)n2cncn2)=O)CC2(CCCCN2C(=O)CN2CCNC2=O)C1 21332,c1(OC)cnccc1C(=O)NC1CCCCC1NC(=O)COCCN(C)C 21333,C1(NC(Cc2cnc(C)s2)=O)CN(C(C2CC3CCC2O3)=O)CC1C 21334,C12(C(=O)NCC34CC=CC(C3)OC4)CCC(C(=O)OCCF)(CC1)CC2 21335,N1(C(c2ccn(CCN(C)C)n2)=O)CCN(C(c2cc(CN(C)C)on2)=O)CC1 21336,c1(CC)nc(CCNC(=O)CC2CCCC2NC(=O)C(F)(F)C2CCCC2)no1 21337,C=CCC(CNC(=O)CC(CC)C1CCC1)C(=O)N(C)Cc1cnccn1 21338,c1(C(=O)NC(C)CN(C(=O)CC(C)C2CCCCC2)C)nccc2cccnc12 21339,C1(NC(c2ccnc(OCC)c2F)=O)CN(C(c2cc[nH]n2)=O)CC2(CC2)C1 21340,C1(NC(C(CSC)(C)C)=O)CN(C(C2CN(C(C)C)C2)=O)CC2CC12 21341,O(NC(=O)C(CC#CC)NC(=O)C(C)C1(O)CCC1)CC1CC(=C)C1 21342,c1(C(=O)NC2C(OC)CN(C(c3cccc(N)c3C)=O)C2)cccc2[nH]cc(Cl)c12 21343,c1(NC(C2N(C(C)=O)C(C)SC2)=O)c(F)ccc(C(=O)NC(C)(C)C)c1F 21344,c1(CC)noc(CCC(=O)NCC(CO)NC(=O)C(F)(F)c2nccs2)n1 21345,c1(C(=O)NC(CCSC)C(N2CC3(CCCC3)C2)=O)cnc2cc[nH]c2c1 21346,N1(C(C(=Cc2cnc[nH]2)C)=O)CCN(C)C(CNC(=O)CC2CCC(=O)N2)C1 21347,Cc1cc(-c2cc(C(=O)OC(C)Cc3nccn3C)on2)n(C)n1 21348,C(=O)(C(CC(C)C)NC(C)=O)N(CC)CC1CCN(C(=O)Cn2cc(Cl)cn2)C1 21349,c1(C(=O)NC(CCCNC(c2cc(C)nn2C(C)(C)C)=O)C)cccc(=O)n1O 21350,c1(C(C)NC(=O)NCC(=O)N(C2CCOC2)C2CC2)ccncc1F 21351,C(=O)(C1CCCc2cncn21)NC(C)CCNC(=O)C(c1cc(F)cc(F)c1)O 21352,C1(N(C(CN(CCC)C)=O)CC)CC(NC(=O)C=CC(=O)N(C)C)C(O)C1 21353,c1(OCCOC)cccc(C(=O)C(=O)NC(CNC(C2CC2C#N)=O)C2CC2)c1 21354,C1(CC(=O)NCCC2(OC)CN(C(=O)COCCCF)C2)CCCC(C)(C)C1 21355,C(=O)(C1=CCCCC1)N1C(C)(CCC(=O)NCC2(C)CC3CC3C2)CCC1 21356,C(C)(C)(CCC(=O)N1CCC(CCOC)(C(N2CCC2CO)=O)CC1)OC 21357,C1(C(=O)NC2C(NC(=O)CCF)C2)COc2ccccc2C1 21358,C1(O)(CC(=O)N(C2CCN(C)C2=O)CC)CCN(C(c2csnc2Cl)=O)CC1 21359,N=c1cc(C(N2CCCC2CC2NC(=O)NC2=O)=O)c(Br)c[nH]1 21360,C1(C)(CC)CN(C(C2CN(C(=O)CNC(=O)Cc3cnns3)C2)C)C1 21361,c1(C(N2CC3(CN(C(CN(C(C)C)C)=O)C3)C2)=O)cccc2[nH]nc(O)c12 21362,N(C1CCCc2sc(Cl)cc21)C(CCCn1cc(CNC)nn1)=O 21363,c1(N(C)CC2CCCC(O)C2)cccc2c(Br)cncc12 21364,C1(NC(C=Cc2c(C)ncs2)=O)CN(C(c2ncc(F)cc2F)=O)CCC1C 21365,c1(C(=O)NC2CCC(NC(C#CC(C)C)=O)CC2)cccc2nc(O)oc12 21366,C1(C(C)N(c2cc(C(F)(F)F)c[nH]2)C(C=CCC)=O)CCCN1C(c1ccco1)=O 21367,C(=O)(C#CC1(C)CCCO1)NCCOC1CCN(C(C(C2CCOCC2)C)=O)C1 21368,C1(NC(CCN(C(CC2(C)CCOCC2)=O)CCCO)=O)CC2CC1CC2CO 21369,C1(C)(C(=O)NC(C=C)C2CC2)CCN(C(=O)COC2(C)CCC2)C1 21370,N1(C(CS(=O)(=O)NCC)=O)CCN(C(c2scc(C)c2C)=O)CC1CO 21371,Cc1cc(Cl)ccc1N(C(=O)Cc1ccsc1)Cc1ccc(F)cc1 21372,N1(C(C2(N(C)C)CCCC2)=O)CC(C(N)=O)(CN(C(CCOC)=O)C)C1 21373,c1(C(N(CCN(C(=O)CN2CCP(C)(=O)CC2)CC)CC)=O)n[nH]c2ccccc12 21374,c1(OC)cccc(S(=O)(=O)NN=Cc2cnc(C(F)(F)F)nc2C)c1Cl 21375,C1(C(=O)NC2(C)CS(=O)(=O)C2)CCC2(CCN(C(=O)CC3C=NNC3=O)CC2)O1 21376,N1(C(=O)OC(C)(C)C)CCC2CN(C(C34CCC(C3)C(=O)N4)=O)CC2CC1 21377,c1(C(=O)NCCC2OCCN(C(c3cccc(N)c3)=O)C2)ccnc2[nH]nnc12 21378,CC1(C)NC(=O)CC1C(N1CC(NC(C23CCOC(C)(C2)C3)=O)C1)=O 21379,c1(OC)ccc2c(c1)OCC(CN1CCCC(O)(C(F)(F)F)C1)=C2.C(CO)S 21380,C12(C(N3CCC(CCNC(c4[nH]cc(CC(C)C)c4)=O)C3)=O)COC(CCO1)C2 21381,C1(C(=O)NCC(CC(=O)NC)C)CCN(C(c2occc2C)=O)CCO1 21382,C(=O)(C#CC1(C)CCCO1)NCC(C)CNC(c1ccccc1C1CC1)=O 21383,C1(F)(C(=O)NC2CC(CCNC(C=CC(C)C)=O)C2)CCCOC1 21384,N1(c2snc(SC)n2)CCC2(CCCCC2NC(c2cc(C)cnc2F)=O)C1 21385,CCC1=C(C(=O)N2CCN(C(c3c(C)cnn3CC)=O)C(COC)C2)SCCO1 21386,C=CCC(CNC(=O)C(c1ccccc1)F)(C(=O)O)Sc1ncccn1 21387,c1(CC(=O)NC(C)CC(C)NC(c2ncoc2C2CC2)=O)ccc(F)c(Cl)c1F 21388,N1(C(CN(C(C2(C)CC(=C)C2)=O)C)=O)CC(C)C(C)C1C 21389,C(C(C)(C)CCNC(C1CCCN(C(=O)C(c2ccc(F)cc2)=O)C1)=O)OC 21390,c1(C(=O)NC(c2cccnc2)C(N2CCC(CO)C(O)C2)=O)cnn2ccccc12 21391,N1(CCC(=O)NC(CNC(C=CCC(C)(C)C)=O)CO)CCCCC1=O 21392,Brc1c[nH]c2cnc(N3CC4CN(Cc5cc6ccccc6o5)C4C3)nc12 21393,C1(CNC(C(CC)(C)COC)=O)CCC2(CN(C(c3cc(F)cc(Cl)c3)=O)C2)O1 21394,C1(NC(C2CC(C)(C)OC2)=O)CCN(c2ccc(C#N)nn2)CC1O 21395,C1(C(N(CC(N2C(CC)COCC2)=O)C2CCC2)=O)CC(=O)CC(=O)N1 21396,C1(NC(C(=Cc2cccnc2)C)=O)C2CCC1CN(C(c1ccns1)=O)C2 21397,O=C(C#CC1CCCCO1)NC1CN(C(=O)CC2CSC2)CC1c1ccncc1 21398,Cn1nc(Cl)c(C(=O)NC2CC23CCN(C(C2CCSCC2)=O)C3)c1Cl 21399,C(=O)(C1CCCc2nn[nH]c21)N(C1CCCOC1C1CCN(C(C=CC)=O)CC1)C1CC1 21400,C1(C(=O)NCc2ccc(C(=O)OCC)o2)C(Cl)(Cl)C12CC2 21401,C1(C2CC2)(NC(C(c2cccc(C)c2)C)=O)CCN(C(=O)CCN(C)C(C)=O)C1 21402,N1(C(C2CCN(C(C3N(CC(C)C)CCC3)=O)CC2O)=O)CCC(C2CCC2)C1 21403,c1(C(=O)NCC(C)(CO)NC(C=CC=CC)=O)cc(-c2ccccc2)nc(O)c1 21404,Cc1cccc2c1CCCN2C(C)C.C12CCNC1C2 21405,c1(CC(=O)NCCN(C(CC)C)CCCC(O)CF)ccc(C)nc1 21406,c1(C(=O)NCC=CC(=O)N(C2CC(CN3CCOCC3)C2)C)ccc(C(F)F)o1 21407,C1(CC(=O)N(C2CCCN(C(c3nc(OC)c(C)s3)=O)C2)C)CC2CCC1CC2 21408,c1(C(=O)NC(CCNC(C(C(CC)C)O)=O)C)c[nH]c2cccnc2c1=O 21409,N#Cc1ccc2c(c1)C(=CC(=O)NC1(C(O)C(F)(F)F)CC1)C2=O.N1CCC1CO 21410,C=CCC(O)(CC=C)C(C)NC(C1CC(=O)N(C)C1c1cccnc1)=O 21411,C(=O)(C1=NOCC1)N1CC(C(=O)NOC(C)CC)(CC)C1 21412,C(=O)(CCC(=O)C1CCC1)NCCC(C)N(C(=O)CCSC(F)(F)F)C 21413,N1(C(C2(OC)CC2)=O)CC=CC(NC(c2c[nH]nc2C2CC2)=O)C1 21414,CC(C)C(CNC(C1CCC2(CCC2)O1)=O)C(=O)NCc1cccc(F)c1 21415,C1(O)(CNC(C(c2ccoc2)NC(=O)CCc2nc[nH]n2)=O)CC2C=CC1C2 21416,c1(C(N(C23CCC(CC2)C3)C)=O)coc2c1CN(C(C1COCCO1)=O)C2 21417,C1(C)(C(=O)NC(C2CCCO2)CC)CN(C(=O)CCCCNC(C)=O)C(C)(C)C1 21418,N1(C(C2(CC)CN(C(=O)CCC3CC3(C)C)C2)=O)CCCCCCC1C 21419,C=CCCC(F)(F)C(=O)NC(CO)CCCCNC(c1cnsn1)=O 21420,c1(C(C(=O)NCC2C(NC(C3(C(C)C)CC3)=O)C2)C)ccccc1F 21421,CCCCC(O)C(=O)N1CCC(C)(CNc2ccnnc2Oc2ccccc2)C1 21422,c1(C(=O)NC(CN(C)Cc2c(C)non2)C)ncc[nH]c1=O 21423,c1(-c2cn(C(C)CN3CCCC3)nn2)cccc(C(N2CCCC2C2CC2)=O)n1 21424,C1(CC(=O)NC)CN(C(c2cncc(C)n2)=O)CCN1C(=O)C1CC1 21425,N1(C(c2cnc(CCC)s2)=O)CC(C(=O)OC)C(C)C1 21426,c1(OCc2nccc(C)c2)ccc2ncc(Br)cc2c1 21427,c1(C(N2CCC(NC(C(C)OC)=O)C(C)(C)C2)=O)cc2c(c([N+](=O)[O-])c1)OCO2 21428,n1(CC)nc(C)c2cc(C(=O)NCC(C)(C)NC(C3CC4CCC4C3)=O)sc12 21429,N1(CC)CC(CSc2cnc(Cl)c(Cl)c2)CC(C)C1 21430,N#Cc1ccnc(CN2CC3CN(C(c4cc(C(F)(F)F)on4)=O)CC23)c1 21431,C1(CCOC)CN(C(c2cc(Cl)cs2)=O)CCN1C(=O)CC(C)(C)O 21432,C=CCC(C)(C)CC(=O)N(C)CCNC(=O)C(c1ccc(OC)cc1)NC(C)=O 21433,C1(CCNC(C2C(C(=O)OC)CCC2)=O)CCN(C(c2nc(O)c(C)s2)=O)CC1 21434,C1(C2CCN(C(=O)CC(C)(F)F)C2)(NC(C2C(CCC)C2)=O)CC1 21435,N1(C(C2C(CC)CCC2)=O)CCC2(CC1)CCN(C(=O)CNC(N1CCCC1)=O)C2 21436,C(CCN=c1cc(C)[nH]c(=NCC2(COC)CCCCO2)[nH]1)OCC 21437,c1(C(=O)NC2C(C)(C)N(C(C3CN4CCN3CC4)=O)CC2)cnc2nccn2c1 21438,CC1C(C)N(C(=O)C2=CCOC2)CCN1C(=O)CCCCN1C(=O)CCC1=O 21439,c1(-c2c(C)oc(C(=O)N(C)CCN(C)C(C3CC3C)=O)c2)cccc([N+](=O)[O-])c1 21440,CC(C)C(C(=O)NC(C)Cn1cc(-c2cccc(C(F)(F)F)c2)nn1)C(C)C 21441,S(=O)(=O)(c1ccc(Cl)nc1C)NC1(C#N)CCN(C(c2c(OC)ccs2)=O)C1 21442,N1(C(C2(NC(C3CCC(CCC)CC3)=O)CC2)=O)CC2CC(C)(C)C2C1 21443,C(C(CC(C)C)C(=O)NCc1c(C)noc1C)NC(C=CCN(CC)CC)=O 21444,c1(OC)ccc(C(=O)NCC(CNC(=O)CCc2cccnc2F)CO)c(C)c1 21445,CC1(C)COCCC1C(N1CCC1CN1C(C(=O)Nc2cnccn2)CCC1)=O 21446,c1(C(=O)NCC(C)OCC#C)ccc(F)c(-c2ccc(OC)c(OC)n2)c1 21447,C1(CC=C)(NC(=O)CCc2ccc(C)s2)CCN(C(c2cncs2)=O)C1 21448,c1(C(N(C)CC2COCCN2C(c2cn[nH]c2)=O)=O)noc2c1CCCCC2 21449,C1(C(=O)NCC23CC(CNC(C(C(C)(C)C)O)=O)(OC2)C3)Cc2ccccc2O1 21450,Cc1scnc1C(=O)NCC(C)CN(C(=O)CNC(C1CCC1)=O)C 21451,C=C(Br)CC(=O)NCCC1CCN(C(C2CCCC2)=O)C1 21452,N1(C(=O)Cc2cncc(F)c2)CC2CC(C1)N(C(=O)COc1cccnc1)C2 21453,OC1(COc2ccc(-c3nnc(C4CC4)o3)nc2)CC(O)C12CCC2 21454,Cc1cc(C(=O)NC2(CN(C(=O)CC3CCOC3=O)C)CC2)c2ccccc2n1 21455,CCC(CC(=O)NC1C(NC(=O)CCCOCCOC)CC1O)C(C)C 21456,CC1=CC(NC(=O)C(=O)NCCNC(C2(C)CCOC2C2CC2)=O)CCC1 21457,CN1CCN(C(C2COCC2NC(=O)C=Cc2cocn2)=O)CC1=O 21458,c1(C(N2CCN(C(C3(C(=O)OC)CCC3)=O)CC2)=O)cncc(Br)c1C 21459,N1(C(C(=O)Nc2ccc(OC)cc2OC)C)CCn2ncc(Cl)c21 21460,C(CCC(=O)NC(c1cccnc1)C(=O)NCCc1ncccn1)=CC 21461,Cc1[nH]c(C)c(C(=O)NC2CCCCC2NC(c2cc(C3CCC3)on2)=O)c1C 21462,CN1CCc2ccc(NC(=O)Nc3ccc(-c4nncn4C)cc3)cc21 21463,C1(NC(=O)CCc2cncs2)CCOCC1NC(=O)CCC(=O)N1CCCCC1 21464,CC1(NC(=O)COC2CC(NC(=O)CC3CCCC34CC4)C2)CC(C#N)C1 21465,CC1CN(C(=O)COCCOC(=O)Nc2ccccc2)CC(C)S1 21466,c1(OC)nn(C)cc1C(N1CCC(N(c2cc(C(C)OC)ncn2)C)CC1)=O 21467,C(CCC(C)C(=O)NCC1CN(C(C2(N3CCCC3)CC2)=O)CCC1C)OC 21468,N1(C(Cn2c3cccc(C)c3cc2)=O)CCC2(NC(=O)CCF)CCCCCC12 21469,C(=O)(C1=CCCSC1)NC1(C)CC(N2CCC(NC(c3ccccc3)=O)CC2)C1 21470,C1(C(=O)NC2C(OC)C2)COCC1NC(=O)CCc1cnn(C)c1 21471,c1(C(N(CCN(C(CC2CC(OC)C2)=O)C(C)C)C)=O)cc(C)c2n[nH]cc2c1 21472,Nc1cc(C(N2CC(NC(=O)CCNC(c3ccsc3)=O)C2)=O)cc(F)c1 21473,CC(C)CCCC(C)C(=O)NC1CC(C(C)O)C1.C1CC(=O)NC(C)CO1 21474,c1(C(C(=O)NCC(C(C)C)NC(C2CCC(OC)C2)=O)(F)F)ccc(Cl)cc1 21475,N1(Cc2c(C)ccnc2)CCC2(CCN(C(C3CC3c3ccc(Cl)cc3)=O)C2)C1 21476,Cc1cc(Cl)ncc1C(=O)N(C1(C(F)(F)C(F)(F)F)CCC1)CC(C)O 21477,C(=O)(C1=CCN(C(C2(C)CCN(C)C2)=O)CC1)N1CCN(CCOC)CC1 21478,C1(CCCC)CCC(NC(=O)C(=O)NC2(C34CCCC3C4)CC2)C1 21479,CCC1=C(C(=O)NC2CC(NC(c3cc(OCC)cnc3F)=O)C2)CCCO1 21480,C(CCOCC(c1ccccc1)CO)(C(F)(F)F)Oc1ccccc1 21481,CC1C2CCC(C2)C1C(N1CCCC(C)(C(=O)NC2CC23CC(O)C3)C1)=O 21482,C1(CNC(C(C)NC(CC)=O)=O)CCN(C(c2cn(CCCF)nn2)=O)C1 21483,Ic1cnc(CNCC2CCN(c3nncs3)C2)s1 21484,CN1CC(C)(C(=O)NC2CC(NC(c3ccc(C4CC4)cc3)=O)C(O)C2)CC1=O 21485,Cn1ncc2cc(C(N3CC(NC(=O)CC4CCCOC4)C(F)C3)=O)cnc12 21486,N1(C(c2cc(CC)ncc2)=O)CCC2CCCC12C(=O)NC1CCCC(C)(C)C1 21487,C1(SC)CCN(CC(=O)NC(C)(C)C(=O)Nc2ccccc2)C12CCC2 21488,N1(C(C(CCC)O)=O)CCOC2(CCN(c3cc(CCOC)ncn3)CC2)C1 21489,c1(C(=O)NC(CNC(c2cc(C)no2)=O)C(C)C)ccn2ncc(Br)c2c1 21490,c1(C(=O)NC23C(CN(C(C(CCC)O)=O)C2)C3)ccc(S(=O)(=O)CC)cc1 21491,C(CCC)(C(=O)NC(CCC1CC1)C(=O)NC(C)Cn1ccnc1)=CCC 21492,N1(C(C)=O)CCC(CC2(C3CCCO3)CCCC2)CC1.C(=O)(C(C)(O)C1CC1)NC 21493,C(=O)(CN=S(C)(C)=O)NCC(C)(O)OC 21494,c1(C(N2CCN(C(C=COCC)=O)C(CF)C2)=O)ccc2c(c1)CCCC2=O 21495,c1(C(=O)NCc2cccc(CN(C(C(C=C)OC)=O)C)c2)cccc2cccn12 21496,c1(N2CCC(NC(c3n(CCC)nc(C)c3)=O)C2)nc2ccc(F)cc2o1 21497,c1(-c2nc(CCOC)nn2-c2ccn(C(C)C)n2)c[nH]c2cccnc2c1=O 21498,C1(C(N(C2CN(C(=O)Cn3cccn3)CC23CC3)C)=O)C2C3CC4C1C1C2CC3C41 21499,C1(C)(C(N2CC(CCNC(C3(COC)CC3)=O)(OC)C2)=O)CCCOC1 21500,N1(C(c2ccnc(CC(C)C)n2)=O)CCC2(CC1)CC2C(N1CC(N=[N+]=[N-])C1)=O 21501,N1(C(Cc2c(C)non2)=O)CC(O)(C2CCN(C(=O)C(C)(C)CO)CC2)C1 21502,c1(CC)ccc(COC(C2CN(C)CC2C(F)(F)F)=O)cc1Cl 21503,N1(C(c2ccc(SC)o2)=O)CCCCC(CNC(=O)CC2COCCN2C)C1 21504,c1(C(=O)NC(C)(C)CNC(c2nonc2N)=O)csc2nc(-c3cccs3)nn12 21505,c1(CC)c[nH]nc1C(=O)N(CC(C)N(C(=O)CCc1cccnc1)C)C 21506,C1(CNC(C2C(C=C)OCC2)=O)CN(C(=O)CCC(=O)OC(C)(C)C)CC12CC2 21507,C1(COCCN(CC(=O)NCC(F)F)C2CC2)CCCCN1C1CCCC1 21508,N(C1COc2cc(Br)ccc21)C(=O)Nc1cc(C(=O)NCC)c(I)cc1 21509,N1(C(C(CC)CCOC)=O)CCC2(CC2)CC1C(=O)NCC(C)(O)CO 21510,CC(C)CCSCC(=O)N(CCNC(=O)C(O)c1ccsc1)C1CC1 21511,c1(OC)ncccc1-c1ccc(C2CCN(C(c3cnc[nH]3)=O)CC2)cc1 21512,c1(OC)cc(Cl)c(CN2CCCC(Nc3ncc(C#N)cc3F)CC2)cc1Cl 21513,C1(C)(C(N2CCN(CCNC(C(=Cc3cnc[nH]3)C)=O)CC2)=O)CCC(=O)N(C)C1 21514,C1(CCOC)(NC(C2CC3CC3C2)=O)CCN(C(c2ccnc(C)c2)=O)CC1 21515,NCCCCN=c1nc2sccc2c(NC2CCn3cncc3C2)[nH]1 21516,c1(C(=O)NCC(C)(F)CNC(C2CCC3CC3CC2)=O)cnc2ccccn12 21517,C1(C(=O)NCCc2scc(C(C)C)n2)CCCC1S(N)(=O)=O 21518,c1(OC)cc(CNC(N2CCCC2C2(CO)CC2)=O)on1 21519,C=Cc1cc(C(=O)NC2(CN(C)C(C)=O)CC2)cc(F)c1.c12csc(n1)CCC2 21520,n1(C2C(C)OCC2)nc(CCO)nc1-c1ccc(SCc2cccs2)cc1 21521,C(c1ccccc1F)=CC(=O)NCCN(CCC)C(C1CC2(C1)CC2F)=O 21522,c1(C(=O)NCCN(CCOC)C(C2CCC(NC)CC2)=O)sc(C)nc1C 21523,C1(C(=O)NCCCCCOC)CCN(C(=O)C2=C(C)CC2)C1C(C)C 21524,CC1(C(N2CCCC(CNC(=O)COc3ccccc3F)C2)=O)CCC(F)(F)C1 21525,C1(C2(NC(CCOC3(C)CN(C(N)=O)C3)=O)CC2)CCCCN1C(=O)CCCF 21526,N1(C(CN(CC(C)(C)C)C)=O)CCOC(c2cn(CCN(C3CCOC3)C)nn2)C1 21527,c1(C(C(N2CCN(C3CCCC(=O)O3)CC2)=O)(F)F)cc(F)cc(F)c1 21528,N1(C(c2ccn(CCC)n2)=O)CCC(C(C)NC(c2cccc(CO)c2)=O)CC1 21529,c1(C(N2C(CC)CN(C(c3cc(Br)ccc3F)=O)CC2)=O)ccc2n[nH]cc2c1 21530,C(=O)(CC(C)CC(=O)NC(C(=O)NCc1ccc(OC)cn1)C(C)C)OC 21531,C1(C(=O)NCc2cncs2)C=CCN1C(C1CCOC1C1CC1)=O 21532,CC1=NOC(=O)C1CC(=O)NCC1(NC(C2(C)CCOCC2)=O)CC1 21533,C(=O)(C(F)(F)CCn1cccn1)NCC(C)CN(C)C(c1cc(=O)cc[nH]1)=O 21534,c1(C(N2CC(CCNC(C=CC(C)C)=O)OCC2)=O)cccc2c1C(C#N)C2 21535,N1(C(c2n(C(C)C)nnc2)=O)CCC(O)(C(C)NC(=O)CCc2ncco2)C1 21536,O=C(C1CCCc2scnc21)N1CCCNC1=O 21537,CC1CCN(C(C2C(C(=O)O)C2C)=O)CCN1C(=O)CSc1ccccc1Cl 21538,C1(NC(=O)NC(c2onc(C)n2)C)CC=C(C)CC1 21539,C(=O)(C1=CCCC1P(C)(C)=O)NCc1c(CNC(C(CCCC)CC)=O)occ1 21540,c1(OC)ccc(Br)cc1CC(=O)NC1(C)CC(NC(=O)CC2=CCCC2)C1 21541,CC1C2CC(C2NC(=O)CNC(c2ccccc2F)=O)N1C(C1CC12CC2)=O 21542,C(=O)(CS(=O)(=O)CC(F)(F)F)N(CC(C)O)CCNC(c1c(OC)nn(C)c1)=O 21543,Nc1cnc(Br)c(C(=O)NCCNC(=O)CC2(C3CC3)CC2)c1 21544,c1(CNC(C2(C)CCCC2O)=O)nc(CNC(=O)C2=COCCC2)cc(O)n1 21545,C1(CNC(C2CC(CC(C)(C)C)C2)=O)CN(C(C2(F)CC=CC2)=O)CC12CCC2 21546,N(C1c2ccccc2CC1NC(=O)C(=O)N=S(C)(C)=O)C(CCOCC)=O 21547,C(=O)(C(C)(CO)NC(C1CCOC1(C)C)=O)N1CC(OCC)(CO)C1 21548,C1(CCNC(c2ccc(C)s2)=O)CCN(C(C2CC2C(F)(F)F)=O)CC1 21549,CCC(C)(COC)NC(=O)C(CC1CC1)OC(c1cn(CCO)nn1)=O 21550,CC1CC(C(=O)N(C2CCCN(C(=O)CCNS(=O)(=O)C(F)(F)F)C2)C)CCS1 21551,N1(CC)CCCC(ONC(=O)C(C2CC2)N(C)C(C2CC=CCC2)=O)C1 21552,C1(C(=O)NC(C(C)C)(C)C)CC(=O)CN1C(=O)CCc1ccncc1 21553,C1(CNC(CC=C)=O)CCC2CN(C(=O)CCC(=O)NCCC)CCC2C1 21554,c12cccc(c1)CO2.C(=O)(CP(C)(C)=O)NCC(CNC(c1nc(C)[nH]n1)=O)F 21555,N1(C(=O)CCc2nnc(C3(C(=O)O)CC3)o2)CCCC(C2CCCN2)C1 21556,c1(CNC(=O)NC(C(C)C)C2CCC2)cc(Cl)ccc1OCc1ccc(Cl)cc1 21557,c1(CC)ccc(CC(N2CCN(Cc3cc(-c4ccccc4)n[nH]3)CC2)=O)cc1 21558,C(C(C(=O)N1CCN(C(=O)C=C2CCCCC2C)CC1)C(C)(C)C)OCC=C 21559,Cc1nn(C2CCOC2)cc1C(=O)NC(CO)C(C)NC(c1cnc(C2CC2)s1)=O 21560,O=C(C(O)C(F)(F)c1ccccc1)NC1CC(NC(=O)Cc2ccc(Cl)cc2)C1 21561,Cc1cc(C(C)C)nc(N2CCCOC(CNC(C3CCCN3N=O)=O)C2)n1 21562,CC1(C)CC(C(=O)NC2CCCCC2CNC(C2CCCN2C2CC2)=O)=NO1 21563,N1(C(C(C)NS(C)(=O)=O)=O)CCC(C)N(C(=O)CNC(=O)Cc2cnn(C)c2)CC1 21564,c1(C(N(C(=O)C(CC)C(C)C)C(CCCC)CN)=O)cnn2cccnc12 21565,C1(CNC(C(CC)N(C)C)=O)CCC2CN(C(=O)C=C(C)c3cccs3)CC12 21566,N#CC12CC(C(=O)NC3CC(C(N4CCCC4c4ncco4)=O)C3)(C1)C2 21567,c1(C(N(C(C(=O)NCC2(O)CC2)C2CC2)C)=O)cc([N+](=O)[O-])n[nH]1 21568,Cc1ncc([N+](=O)[O-])cc1C(=O)NCCNC(C1CC(C2CCCC2)C1)=O 21569,N1(C(=O)CNc2nccs2)C2CCC1CC(NC(C1CC(n3cnnc3)C1)=O)C2 21570,C1(CNC(=O)COc2ccsn2)(CNC(=O)CN2CCC2)CCOCC1 21571,N1(C(Cc2n(CC)ccc2)=O)CCC(NC(=O)C(C)C2CCCC2)C1C(C)(C)C 21572,n1(CC)nc(C(=O)NCC2(CNC(c3nccn3C)=O)CCC2)ccc1=O 21573,C=CCC(C)(CC)C(=O)N1CC=C(C(=O)NC2CCC(C)CC2)C1 21574,C1(CC(=C)C)CCCC1(c1nnnn1CCCSCCOC)NCC1CC1 21575,C1(CCC(=O)NCC(C)(C)NC(C=C(C)C(C)(C)C)=O)CCCCN1C 21576,N1(C(C2(CC)CCC2)=O)CC(CNC(=O)CCCN(C)C)OC2COCC12 21577,c1(C(=O)NC2CCC(NC(C3NC(=O)OC3)=O)C2)cccc(Cl)c1Br 21578,n1(CC)cnc2c(N3CCC(C)=C(C)C3)[nH]c(=NCc3ccncc3N)nc12 21579,c1(C(N2CCN(C(C(C)SC(F)(F)F)=O)C(C3CC3)C2)=O)nc(O)nc(O)c1N 21580,c1(C(=O)OC)ccc(Cl)c(C(C)OC(c2nc(CN)no2)=O)c1 21581,N1(C(c2n(CC)ncc2)=O)CC2CCCC1(CNC(c1conc1C1CC1)=O)C2 21582,C(c1ccccc1)=CC(=O)NC(C)(C)CNC(=O)CCc1cocn1 21583,Cc1cc(C(=O)N(CCNC(=O)CCCN2CCCCC2)C(C)C)ccc1Br 21584,C1(C(=O)NCC2CC(NC(C(n3ccc(C)n3)C)=O)C2)CCOC(C)(C)C1 21585,N1(C(c2ccncc2)=O)CC2CCN(C(c3nc(Cl)c(Cl)s3)=O)C2C1 21586,C1(C(=O)NC(C2(O)CCN(C(=O)CCCC3CC3)C2)C)CC(C)(C)OC(C)(C)C1 21587,Cc1nc(Br)sc1CNC1(c2nnnn2CC2CC3CC3C2)CC1(C)C 21588,N1(C(C(=O)NCC)=O)CC2(C=C(C(=O)NC(C3CCN(C)C3)C)CO2)C1 21589,c1(OC)cc(C)c(C(=O)NC2CC3(C2)CC3NC(=O)CC2CCCN2C)cc1Cl 21590,C1(C(N(C)CCOCCNC(=O)C=CC2CCCC2)=O)CCCCC1C(F)(F)F 21591,N(C(=NCCc1cccc(O)c1)NCc1ccnn1C)CC1C(C)OCC1 21592,C(=O)(CC1OCCc2ccsc21)N1CCN(C(C(CC=C)N(C)C)=O)C(C)C1 21593,c1(CC(=O)NCCCN(C(=O)CC(C)F)CC)cc(=O)n(-c2ccccc2)[nH]1 21594,CCC(C(=O)NCC1CCN(C(c2cnnn2C(C)C)=O)C1)C(C)(C)CC 21595,N1(C(C(CC=C)NC(C)=O)=O)CCOCC(NC(C2CC(O)CN2C)=O)C1 21596,C(=O)(C(C)(F)C(C)(C)F)NCCCOCCNC(c1cnc(C(C)C)nc1)=O 21597,C1(C(=O)NC(C2CCCN(C(c3ncccn3)=O)C2)C)Cc2n[nH]cc2C(=O)N1 21598,CCC(CNC(=O)CCc1nccs1)(CC)C(=O)NCC(C1CCOC1)CO 21599,Cc1ccc(C2=CCN(C)CC2)c2nc(C(=O)N(C)CC3CC3)cn12 21600,c1(C(N2CCN(C(CS(CC)=O)=O)C3C2C3)=O)cc(F)c(Cl)c(Cl)c1 21601,c1(C(=O)NC2(COC)CN(C(=O)C#CC3(C)CC3)C2)c(Br)ccc(F)c1F 21602,CCC(CC(F)F)C(=O)NC1CCN(C(=O)CCC2CC2)C1 21603,C=C(C)CCC(C)N(C(N1CCC(c2ncc(Br)cn2)CC1)=O)CC 21604,c1(N2C(=O)CC(OC(C3(CC=C)CC(=C)C3)=O)C2)ccc2c(c1)OCCO2 21605,N1(C(c2c(OC)ccc(F)c2)=O)CC2CC(C1)CN(Cc1ccc(SC)cc1Br)C2 21606,C(CCNC(=O)C(C)CO)(C(=O)NCCCN1CC=CC1)OC 21607,c1(CCOC)c[nH]c(=NCC2(O)CCN(C(C3CC4CC4C3)=O)C2)c(C)c1 21608,c1(C(c2nnnn2CC2CC2)Nc2c(OC)nc(C)nc2)[nH]c2ccccc2c1Cl 21609,CCC(C)C(C(=O)N1CCC(C(F)(F)F)C(NC(=O)Cc2ccnn2C)C1)OC 21610,Cc1ccc(CNC(C2CSCCN2C(c2cccnn2)=O)=O)nc1 21611,Cc1csc(=O)n1CCC(=O)C(C(C)N)=O.C(=O)(C(C)(C)NC(N)=O)NCCOCCC 21612,C1(C2CCOCC2)(C(=O)NCC2(O)CN(C(C34C(C(N)=O)(CCC3)C4)=O)C2)CC1 21613,CC1Cc2cc(F)ccc2C1NC(c1cc(Br)ccn1)=O 21614,c1(OC)cc(F)cc(C(N2CCC(N(C)C(C3CC(CC(F)F)C3)=O)C2)=O)c1N 21615,C1(N(C(=O)CC2CC(C)(C)C2)CC)CCCN(C(=O)CC2CCCCCO2)C1 21616,S(=O)(=O)(c1ccc(CC(N2C3CN(C(=O)C(C)(C)C)CC23)=O)cc1)N(C)C 21617,C(CO)(CCCCNC(c1cnc(O)o1)=O)NC(C(C)OCC#C)=O 21618,C1(NC(C(C)(C)N(S(C)(=O)=O)C)=O)CCN(C(=O)Cc2ccncc2Cl)CC1CO 21619,n1(CCC(=O)NC(c2cn(CC(=O)OC)nn2)CC(N)=O)cc([N+](=O)[O-])cn1 21620,n1(CC(=O)NC2C(CNC(n3c(C)ccc3C)=O)CCC2)cnc2c1CCCC2 21621,N1(C(c2nc(=O)cc(N)[nH]2)=O)CCCC(NC(=O)CCCC(N)=O)C(F)C1 21622,c1csc2c1CCNC2.C1(CS(=O)(=O)N)CCCCC1F 21623,CC(CC(F)(F)F)N=c1[nH]c(N2CCC(F)CC2)nc2c1CSC2 21624,c1(C(=O)NCC(CC)(CC)NC(=O)CCC(C)(C)C)ccc(C#N)cn1 21625,c1(C(=O)NCC2N(C(c3c(C)nn(C)c3C)=O)CC2)ccc2c(c1)CN(C)C2 21626,C=CCCCC(=O)NCC1(OC)CN(C(=O)C(C)NC(C2CCC2)=O)C1 21627,C1(NC(=O)Cc2ccc(C(F)(F)F)cc2)CC2CN(C(C3C4COCC34)=O)CC2C1 21628,C1(CNC(C2N(CC)CCC2)=O)C2CCC1CN(C(C1CCC1)=O)C2 21629,c1(CC)ccc(N(C(C)CC(C)NC(=O)COCCCc2cccs2)C)c(C)c1 21630,N1(C(c2cc(C(C)=O)on2)=O)CCC(N=[N+]=[N-])(C(=O)NC2CCN(C)C2)C1 21631,N1(C(N2CCN(C(c3onc(CC)n3)C)CC2)=O)CC(C)C(P(C)(C)=O)C1 21632,c1(CNC(C(C2CCCC2)NC(c2ccsc2Br)=O)=O)ccccc1 21633,C(=O)(CC(C(=O)OC)C(C)C)NC1(CO)CCCN(C(C2(C(=O)OC)CC2)=O)C1.COC 21634,S(=O)(=O)(c1cccc(Cl)c1)N(CC(=O)NCC(C)CNC(C1(C)CC(F)C1)=O)C 21635,c1(C(N2CCC(NC(CCC(=C)Cl)=O)C(C)C2)=O)nc2ccccn2n1 21636,c1(OC)nccc2c(C(=O)OCC3CCOC4(CCC4)C3)c[nH]c12 21637,C1(NC(C2CC2C2CCCC2)=O)CC2CC(C1)N(C(=O)C=Cc1cc[nH]n1)C2 21638,C(=O)(CC(CC1CC1)NC(C1C2CCC(=O)C12)=O)NCCC(=C)C 21639,N1(C(C(C)N(C)C)=O)CCC2(NC(=O)C(c3ccc(Cl)cc3)O)CCCCC12 21640,c1(OC)nc(C(N2CC(C)CC2C(N2CC3CC2CO3)=O)=O)ccc1Br 21641,C(C)(C(=O)N(CCNC(C1CCC1n1ccnc1)=O)C1CC1)OCC=C 21642,CN1CC(C)(C)CC1C(N1C2CCC(C2)C1C(N1CC(CC(N)=O)C1)=O)=O 21643,Cc1ccc(C(N2CC(C(O)C(=O)NC3CCCOC3)C2)=O)c(O)c1 21644,c1(C(=O)NC(CNC(c2nc(CCCC)sc2)=O)C2CC2)ccc(O)c(C)c1 21645,Cc1c(C(=O)NCC2CCCC(NC(C34CCC(C3)C4)=O)C2)cnc2ccnn12 21646,C12CCCN(C1)C2=O.c1(C(C(=O)N(C2CCCC2O)CC)C)ccn(C)c1 21647,N1(CC(N2CC(NC(C3CC3C(F)F)=O)C2)=O)C(=O)CNC1=O 21648,N1(C(C(C)OCCCCCC)=O)CCC(NC(=O)COC(C)(C)CC)C(O)C1 21649,c1(C(N2CC3(CC(N4CCCC5(COC5)C4)C3)C2)=O)cc(I)c(F)cc1Cl 21650,CC1CC(NC(c2cn(-c3ccn(C)n3)cn2)=O)CN(C(c2csc(=N)[nH]2)=O)C1 21651,C12(CNC(C(CC)SC)=O)CCCC1CN(C(C13CCC(O)(CC1)CC3)=O)C2 21652,c1(C(C)O)ccc(C(N2CCC(CF)(NC(=O)CC3CCS(=O)(=O)C3)C2)=O)cc1 21653,Cc1nc(C2CCCC2)sc1C(=O)OCC(=O)NC(c1cccs1)C 21654,CC(C(O)C(=O)NC(CNC(=O)CN(C)C(N)=O)C1CC1)c1ccc(Br)cc1 21655,CC1CC(NC(C2CCC2)=O)CCN1C(=O)C(=C1CCCCC1)F 21656,Cc1cc(C)n(-c2ccc(CNc3cccc(C(F)(F)F)c3)cn2)n1 21657,C12(CNC(c3cnn(C(F)(F)F)c3)=O)CCC1CCN2C(=O)Cc1ccco1 21658,C(C)(CCP(C)(C)=O)(c1nnnn1CCC1COC1)NCCCCOCC(C)C 21659,N1(C(C2=CCC(NC(c3ccnc(CC)n3)=O)C2)=O)CCCC(C)(C#N)C1 21660,C(C(C)CN=c1[nH]c(=NC(C)c2cnn(C)c2)[nH]c2c1CSC2)OC 21661,N1(C(CCCCOC)=O)CCCC(C)C1CCNC(=O)C=CC1CCOCC1 21662,c1(C(=O)OCC)cc2cc(NCC3CCCC3N)ccc2s1 21663,c1(C(=O)NC)nccc2cc(-c3ccc(OC)c(C(=O)OC)c3)ccc12 21664,CC(C)CC(CNC(=O)CC(C)NC(c1ccccc1)=O)NC(C1CC(F)C1)=O 21665,N1(C(C(C=C)C)=O)CCOCC1C(=O)NC1(CCO)CCCC1 21666,Cc1cc(N)ccc1C(=O)NC(C)(C)CCCNC(=O)CCn1ccnc1 21667,N1(C(CCCC#C)=O)CCC(O)(CCNC(c2csc(COC)c2)=O)CC1 21668,CC1CN(C(c2ccn(C3CCC3)n2)=O)CC1NC(c1csnc1Br)=O 21669,Cc1ccc(S(=O)(=O)NCCC(N2CC(NC(=O)C(C)C#N)C3(CC3)C2)=O)cc1 21670,C(C(CC(F)(F)F)NC(=O)CN1C(=O)CCC1=O)NC(CC(C)C1CC1)=O 21671,c1(C(=O)NC(C)CC2CN(C(=O)CSc3nnc(S)s3)C2)cc2scc(Cl)c2[nH]1 21672,c1(C(=O)NCCC2CC(NC(C3ON=C(C(C)C)C3)=O)C2)cncc2c[nH]nc12 21673,S(=O)(=O)(c1cccnc1NCCc1nncs1)NC1C(C)CCCC1 21674,C=CCCCCC(=O)N(C(C)CNC(=O)C(N1C(=O)CCC1=O)CC)C.CCSC 21675,C1(C)(CNC(C(C)c2ccco2)=O)CCCC1NC(c1cnc(C(C)(F)F)s1)=O 21676,C=CCC(C(=O)NCCCN1CCN(C(C2(SCC)CCCCC2)=O)CC1)OC 21677,c1(-n2ncc(CN3CC(C)(NC(CCN(C)C)=O)C3)c2)ccc(F)cc1 21678,c1(SCC(=O)Nc2cc(OC)nc(SC)n2)nc2ccccc2s1.C12(C)CC(C1)N2 21679,CCC(C)(C)C(=O)C(=O)NCC1(C)CCN(C(C2(C(F)F)CCC2)=O)C1 21680,Cc1ncc(N)cc1C(N1CC(CNC(c2ccc(=N)[nH]n2)=O)C(C)C1)=O 21681,c1(SC)ccc([N+](=O)[O-])cc1C(=O)NC(C)C(C(C)C)NC(=O)CC1(CO)CC1 21682,CCCCC(CNC(c1c(C)nsc1N)=O)NC(=O)CCN(CC)CC 21683,c1(OC)ccc(OC)c(C(=O)NCC2CCN(C(=O)C(C)CC(F)F)C23CC3)n1 21684,c1(C(N(CC(C)NC(=O)CC(O)C2CC2)CC)=O)cccc(-c2ccncc2)c1 21685,CC(C)S(=O)(=O)CC(=O)NCCCNC(c1nc(=O)n(C)[nH]1)=O 21686,c1(C(F)(F)Br)cc(C(C2CC2)OCCNCC2CCC2)ccn1 21687,C(=O)(C(COCC)CC)NC1(CNC(CCC2(CCC#C)N=N2)=O)CCCC1 21688,N1(N(C(C)C=CC(N2CC(OC(F)F)C2)=O)CC)CCN(C)CC1C=O 21689,c1(C(C)C)cc(N2CC(NC(=O)CC(C)(C)CCl)C(C)(C)C2)n2ncnc2n1 21690,CC1CC(NC(C2CCN(C(=O)CCC(C)(F)F)CC2CO)=O)CC(C)O1 21691,C(=O)(CC(C)(C)CC(F)(F)F)NCCCNC(c1ncc(OC)nc1)=O 21692,C1(NC(CC=C)=O)(CO)CCCN(C(c2cnn(-c3ccc(Cl)c(Cl)c3)c2)=O)C1 21693,N1(C(C(C)OC2CCOC2)=O)CCCC1C(C)NC(c1ccc(F)s1)=O 21694,c1(CCC(=O)N(CCCNC(C(CCC)NC(C)=O)=O)CC)ccc(C)cc1C 21695,C1(CNC(CCCNC(C)=O)=O)CCC2(CN(C(=O)C(C)C(C)(F)F)C2)O1 21696,c1(C(N2C(C)(CNC(=O)COC3CCOC3)CCC2)=O)ccn2nccc2c1 21697,C=CCCC(C(=O)Nc1cc(Br)ccc1F)NC(=O)NCCC 21698,C1(C=O)CC2(C1)CC(O)C2.C1(CNC(C(C)N(C)C)=O)(CO)CCCO1 21699,c1(C(=O)NC2CN(C(CC=C=C)=O)C(C)C2)cc(Cl)c(Br)cn1 21700,CCC(C(=O)NCC1C2COCC12)N(C)C(c1[nH]ccc1COC)=O 21701,C1(C(=O)NCC2(CO)C(=O)OCC2)C2CN(C(=O)CNC(=O)CN(C)C3CC3)CC12 21702,C1(C(=O)NCCOCCCC)CC2(CCC2)CN1C(=O)CC1CC=CC1 21703,C(=O)(C#CC1CCCOC1)NC1CN(C(C(COCCCCC)=C)=O)CC1SC 21704,C1(NC(c2c(CCC)occ2)=O)CC2CC1N(C(c1cc(Cl)nn1C)=O)C2 21705,C1(CC(=O)NCc2cccc(F)c2)CC2(C1)CN(C(=O)Cc1cnns1)C2 21706,C1(C(=O)NC(C(=O)OCCC)Cc2ccc(F)cc2)CC(=O)N(CCC)C1 21707,c1(C(=O)NCCC(C)NC(C2N(C(C)=O)CCCC2)=O)c2c(c[nH]c1=N)CCC2 21708,N1(C(=O)Cn2cncn2)CC2CN(C(C3(c4cccc(F)c4)CC3)=O)CC2C1 21709,C(c1cc2c(cc1OC)CC(C)O2)=CC(=O)N(CCCNC(=O)C(F)F)CC 21710,c1(C(N(CCCNC(=O)CC(C)C(F)F)CC)=O)cn2cc(C)c(C)cc2n1 21711,C=CCC(C)(C)CC(=O)N1CCC(C)(C)C1C(=O)NC1CCNC(=O)C1 21712,C1(OCC2(CO)N(C(=O)NCC=C(C)C)CC2)COc2ccccc2O1 21713,C1(C(=O)NC2(CCCC(=O)NC3CC4CCC3C4)CCC2)OC2CCC1C2 21714,C12(CC(=O)N(CCCCO)C)CCC1CN(C(C1(C(N)=O)CC1)=O)C2 21715,N1(C(c2cc(OC)no2)=O)CCC(C)C1C(=O)NCC(c1cnc[nH]1)C 21716,c1(NC(C(N2CCC(C(=O)OC)C2(C)C)=O)=O)ccc(N=[N+]=[N-])cc1 21717,CCCCC(O)CC(=O)NC1CCC(CNC(c2ccc3c(c2)C(C)CO3)=O)C1 21718,N1(C(C(CC(C)C)C)=O)CCC2(CCCN2C(=O)C2=CSCS2)C1 21719,C1(C(N2CC(CNC(c3c(C)ncs3)=O)C2)=O)CC(=O)N(C)C1c1cccnc1 21720,C1(NC(CC(C)N(C)C)=O)CN(C(=O)C(CO)C(C)(C)C)CC1C1CC1 21721,n1(C(C)C(N2CC=CC(NC(=O)C(C)(F)F)C2)=O)c(S)nc2ccccc2c1=O 21722,c1(NC(=O)CC2CCN(C(c3ccc(Cl)c(F)c3)=O)C2)nc(Br)cnc1Cl 21723,c1(C(N2CCC3(CNC(=O)C3)C2)C(=O)NCCC#N)cn2cc(Cl)ccc2n1 21724,c1(C(=O)NCCCN(C(C(C2CCOCC2)OC)=O)CCO)cn(C)[nH]c1=N 21725,c1(OC)cc(F)c(C(=O)NC2CC2NC(c2cccc3ccncc23)=O)c(F)c1F 21726,C1(C(=O)NC(CNC(c2sc(CC)c(C)c2)=O)(C)C2CC2)CC2CSCC(C1)C2 21727,C(=O)(CCN=c1[nH]c(=NCCC(C)C(F)F)c2sccc2[nH]1)NCC(C)C 21728,C(=O)(C1CCCn2ccnc21)N1C2CCC(CNC(CC(C)OC)=O)(CC2)C1 21729,N1(C(CNC(c2ccoc2)=O)=O)CCN(C(=O)CSc2cc(Cl)no2)C2CC12 21730,CCCC(C(=O)N(CC(CC)NC(c1ocnc1CC)=O)C)C(C)C 21731,N1(C(C2CCC(OC)C2)=O)CCC(CO)(NC(=O)CSCCC(F)(F)F)CC1.C(C)(=O)O 21732,O=C(CS(=O)(=O)CC1COCCO1)N1CCC(Nc2ccc(F)cc2Br)C1 21733,N1(C(CC(COC)COC)=O)CCCCC12CN(C(c1cc(O)cc(Cl)c1)=O)C2 21734,c1(NC(C(C)C)C(C)NC(c2ccnn2C(C)(C)C)=O)ccc(C#N)nc1 21735,N(C(=NCCCCl)NC1CC(=O)N(Cc2ccccc2)C1)C(C#C)CC 21736,Cc1nn(C)cc1C(C)NC(C1CSCCN1C(=O)CC(C)(C)C1CC1)=O 21737,N1(C(c2n(C)ncc2)=O)CCC(CO)C(NC(c2ccncc2N)=O)C1 21738,C1(C(N(C)CC2(C)CCCO2)=O)C2CC1N(C(C1(CF)CC1)=O)C2 21739,c1(C(=O)NCC2(O)CCN(C(CSCCC)=O)CC2)cc2c(cc1Cl)NC(=O)C2 21740,C1(n2cc(N(C)CC3CC3)nn2)CCN(C(c2cc(C(=O)O)[nH]n2)=O)CC1 21741,C(=O)(C(C1CC1)OC)NC(C1CCCC1)COC.C1(=O)CSCCN1 21742,C(=O)(C(c1cccs1)NC(=O)C(C)n1cccn1)N(CCF)CC 21743,c1(SCCC)nc(Cl)c(CN2CC(C(=O)N=c3nc[nH]s3)CC(F)C2)c(Cl)n1 21744,N1(C(C(C)OCC)=O)CCCC(N(C(c2cc(CC)oc2C)=O)CC)C1 21745,N1(C(C2(OCC)CCOCC2)=O)CC(NC(c2cnccc2C)=O)CC(O)C1 21746,c1(C(N(C)CC2N(C(C(F)=C(C)C)=O)CCCC2)=O)ccc2c(c1)C(=O)C(=O)N2 21747,c1(N(C(C)=O)C)ccccc1C(=O)N(CC(C)CNC(=O)CC1OCCCO1)C 21748,C(C(CC1CC1)C(=O)NOCC=CCl)NC(CCC(=O)N(C)C)=O 21749,N1(C(C(C)c2ccsc2)=O)CCCCCC1CNC(=O)Cc1ccn(C)n1 21750,CC(C)CC(O)C(=O)N1CCCC(C(C)C(=O)NCCC(=O)NO)C1 21751,C(=O)(C(C)(O)CC(C)C)NCC(CNC(c1c(C)nc(Br)s1)=O)F 21752,N1(C(c2c(C)nn(C)c2OC)C(=O)NC2CC(C(=O)OC)C2)CCS(=O)(=O)CC(C)C1 21753,c1(C(=O)NC(C)CCCCNC(C2CC3(CSC3)C2)=O)ccc([N+](=O)[O-])s1 21754,N1(C(C(C)CN(C(=O)COCCNc2ccccn2)C2CC2)=O)CCCC(O)C1 21755,C(=O)(CCC(=O)N1CC(OCCCNC(C2(C)CC2(F)Cl)=O)C1)NC 21756,c1(CNC(CC2CC(=O)NCC2)=O)nnc2n1CCN(C(c1ccsc1Cl)=O)C2 21757,c1(CN(C)C(C2CC3CC3N2C(=O)CC2(N3CCCC3)CC2)=O)oc(C)nc1C 21758,c1(CC(=O)NC2C=CCN(C(c3ccc(Br)o3)=O)C2)ccccc1CO 21759,CC(C(=O)NC1CC(NC(=O)C(C)N2CCC2)C1)S(C)(=O)=O 21760,c1(C(=O)NCC(CN(C(C2(CC)COC2)=O)CC)C)cnc(CC(C)C)[nH]1 21761,C=CCCCCCCCC(=O)NCCOCCNC(=O)C(c1c(C)n[nH]c1C)C 21762,C=CC(C)(CC)C(=O)NCC1(F)CC(NC(=O)C=CC)C1 21763,CCC(CC(=O)NCCC1(O)CCN(C(=O)C(C(C)C)NC(C)=O)C1)OC 21764,c1(C(N2CC(CNC(c3ncc(F)cn3)=O)C3C2C3)=O)ncc2ccccn12 21765,N1(C(C(C)NC(COC)=O)=O)CCCN(C(C2CC2[N+](=O)[O-])=O)CC1C 21766,C1(NC(=O)CC(F)F)(CNC(C2CC23CCOC3)=O)CC(F)(F)C1 21767,O=C(O)CC1=CCN(Cc2cn3ccsc3n2)CC1 21768,C1CCCC(=O)N1.C1(N(C(C)=O)C2CC2)(CO)CCN(C(C2(n3cccn3)CC2)=O)C1 21769,CC1=C(C(=O)NCC2(C)CCC(NC(=O)Cc3cncn3C)C2)COCC1 21770,c1(-c2nc(NC(=O)Nc3scnc3Br)on2)cccc(F)c1 21771,c1(C(=O)NC(=O)CN2CCC2CNC(C2(O)CC(F)(F)C2)=O)ccc(Br)cc1F 21772,c1(C(N2CC(CNC(c3cncc(F)c3)=O)C(O)C2)=O)coc2c1C(O)CCC2 21773,N1(C(C2CCC(=C)CC2)=O)CC2(CC2)CC1C(=O)Nc1ccnn1CCO 21774,c1(C(N2C(C)(C(=O)Nc3cnc(Cl)cc3I)CCC2)=O)c(F)ccc(Cl)c1Cl 21775,c1(C(=O)NCCC2(NC(CS(=O)(=O)NCC)=O)CC2)cc(Br)cnc1O 21776,C(=O)(CCCN=[N+]=[N-])N(CCC(C(C)C)NC(C1(C)CC=CCO1)=O)C 21777,Cc1cc(N(C)CC2CCCCN2C(=O)COCC2CC2)n2nc(C)nc2n1 21778,N1(C(Cn2cc(C(=O)O)nc2)=O)CCCC2C1CCN2C(=O)C=CC1CC1 21779,Cc1cc(C(=O)N(C)CC2CCN(C(=O)C(F)C(C)C)CC2)ccn1 21780,c1(OC)ccc(C(=O)NC23CC(NC(=O)CC45CCCN4CCC5)(C2)C3)c(O)c1 21781,C(=O)(C(C(C)C)n1cccc1)NC(C1CCN(C(c2cc(OCC)no2)=O)C1)C 21782,c1(OCC(N2CCC=C(Br)C2)=O)ccc(-c2ccncc2)cn1 21783,CCS(=O)c1ccccc1CC1C(C(=O)NC2CC(NC(=O)CO)C2)C1 21784,N1(c2nnc(C(=O)OC)s2)CC(C)(C)CC1CNC(c1cccc(F)c1)=O 21785,CCC(C)C(C)C(=O)N1CC2(CC(CC(=O)NCCSCc3ccccn3)C2)C1 21786,c1(CC)nc(C(=O)NC2CN(C(c3noc(C4CC4)c3C)=O)CC2F)c(N)s1 21787,c1(C(N2C(COC)(CNC(=O)CC(C)CF)CCC2)=O)ccn2nccc2n1 21788,C(CCC(C)(C)C(=O)N1CC1)N(C(=O)C=CC(=O)NC=O)C.N1(C=O)CCOCC1 21789,c1(C(N2C(CCNC(C(C3CCC3)OCC)=O)CCCC2)=O)c[nH]nc1[N+](=O)[O-] 21790,CS(=O)(=NC(=O)c1ccc2nc(Cl)nn2c1)c1ccncc1 21791,C(CS(C)(=N)=O)NC(C(n1cc(CCC2CCOC2)nn1)C)=O 21792,O=C(C1=CCCOC1)N(C1C2CN(C(c3ccc(=O)oc3)=O)CC12)Cc1cccs1 21793,C1(CNC(c2ccc(NC)cc2)=O)CC(C(=O)N(C2CC3CC3C2)C)=NO1 21794,c1(C(=O)NC2C(NC(C3N(CC)CC3)=O)CC2)oc2ccccc2c1COC 21795,c1(CN2CCC(C)(C(=O)Nc3[nH]nc(OC)c3C#N)CC2)c(F)ccc(F)c1C 21796,Cc1cc(C(N2CCCC(F)(CNC(=O)C(C)NC(N)=O)C2)=O)cc(C)c1F 21797,c1(CN2CC(C)CC(NC(c3ccc(OC(C)C)cc3)=O)C2)c(Cl)ccc(Cl)c1Cl 21798,CC(C)C(C(C)NC(c1cn(C(C)C)cn1)=O)NC(=O)CCC1CCC1 21799,Cn1cc(C(=O)NC2(CCCCNC(=O)CN(CC(C)(C)C)C)CC2)nn1 21800,C12(NCCC=C=C)CCCC1N(C(=O)Oc1ccc(F)cn1)CCC2.C(C)(C)(C)O 21801,Cc1ccnc(-n2cc(C3N(C(=O)CC4CCC5CC5C4)CC3(C)C)nn2)n1 21802,CC1CCN(C(=O)C(N2CCC3CCOC3C2)=O)CCN1 21803,N1(C(CNC(CC)=O)=O)CCOC(CC(=O)NCC2(O)CCSC2)C1 21804,C1(F)(C(=O)NCCC2(CNC(C3(C(=O)NC)CCC3)=O)CC2)CCCN(C)C1 21805,N1(C(C2CC(C)N(C(c3cc(Cl)c(Br)cc3Cl)=O)CC2)=O)CCC(S(C)(=O)=O)CC1 21806,N12CCC(CC1)CCn1cc(nn1)C1(CCCC1)NC(=O)C2=O.C1(CO)CC1 21807,CP(C)(=O)CC(=O)N1CCOC(CCNC(=O)CC2CCC(=O)O2)C1 21808,c1(C(=O)NC2C(CN(C(C3C(C(=O)OC)C3)=O)C)CCC2)cnc(S)n1C 21809,N1(C(C(CCC)(C)CC)=O)C2CCCC1CN(C(=O)C=CC(C)(C)SC)C2 21810,c1(N(CCN(C(c2ccc(CC(C)C)s2)=O)C)C)ncnc2cccnc12 21811,N1(C(C(CC2CC2)NC(CCC2C(C)(C)C2)=O)=O)CCCC2(CCCC2)C1 21812,c1(C2(CC(N3C(C(=O)NCC(COC)O)CCC3)=O)CC2)cncc(C)c1 21813,C1(CC)C(C(N2CC(=O)NCC2)=O)CCN1C(=O)C(=O)C1CCCC1 21814,c1(OC)cc(F)c(CN=c2[nH]c(CNc3ncnc(OC)c3C)cs2)cc1Br 21815,C12(NC(=O)Cc3cnccn3)CCCN(C(C3CC3(Cl)Cl)=O)CC1C2 21816,c1(-c2c(OCCC)c(F)cnc2)cccc2sc(C(=O)NC3CC(CO)C3)cc12 21817,c1(C(N2CC(O)(CCNC(C3(COC)CCCO3)=O)C2)=O)oc(C2CC2)nc1C 21818,CCC(C)CCCCC(=O)Nc1cnn(C2CN(Cc3cnc(C#N)cn3)C2)c1 21819,C1(CNC(C(C)OCC#C)=O)CN(C(=O)Cc2ccc(Cl)cn2)C2CCCCC12 21820,c1(C(C)C)cc(N2CCCC2(C)CNC(C2CCCN2C)=O)nc(C(C)C)n1 21821,N1(C(C)CNC2CCN(CC(C)(F)F)CC2)CCN(C=O)CC1.C(=O)(C1CC1)OC 21822,CC1CC(CNC(=O)CC(C)(C)C)CCN1C(=O)COc1cncc(Cl)n1 21823,C1(NC(CC2(NC(C(CC)n3ccnc3)=O)CCC2)=O)CN(C)C2(CCC2)C1 21824,C1(CC(=O)NC(CCCNC(COCC(=O)OC)=O)C)CCC(=O)N1C 21825,C(C(=O)Nn1cnn(C)c1=S)C1N(C(COCC)=O)CCCCC1 21826,C1(NC(C2CC(C)C2(C)C)=O)CC2(C1)CN(C(c1cc(C(F)(F)F)nn1C)=O)C2 21827,N1(C(c2n(CCCC)ncc2)=O)CC2CC2(CNC(=O)C=CC(F)(F)F)C1 21828,C(C)(C(CC(=O)N1CCC(CO)C1(C)C)NC(=O)CC1CC=CC1)OC 21829,c1(C(N2CCC(NCC(C)O)C(C)C2)=O)ccc2c(c1)CCC(C)(C)O2 21830,N1(C(CCC2CC(OC)C2)=O)Cc2[nH]nc(C(=O)NCC=CC3CCOCC3)c2C1 21831,c1(C(=O)NCC2(O)CCN(C(=O)Cc3nn(C)cc3CC)C2)cc2n(n1)CCC2 21832,C1(C(=O)Nc2c(C(=O)OC)occc2=O)CC(F)(F)CN1C(=O)OC(C)(C)C 21833,C(=O)(CC(C)(C)COC)N(CC(C)(C)NC(C1C(CC)CCC1)=O)C 21834,c1(CNC(=O)Nc2ncnn2CC)cccc(CNC(=O)Nc2coc(Br)n2)c1 21835,N1(C(C2CN(C(C)=O)C2)=O)CC(NC(=O)CN(C2CCSC2)C)CCC1C 21836,N1(C(Cc2cc(C)nn2C)=O)CC(NC(C2(n3cc(Cl)cn3)CC2)=O)CC(C)C1 21837,c1(N(C)C)cccc(C(N2CCCCC2CNC(=O)CCC2CCCO2)=O)c1 21838,C(=O)(NNc1nc(C)nc2sc(C)c(C)c12)C1CC(COC)CN1O 21839,c1(C(=O)NC(C#C)C)n[nH]c2c1CCN(C(c1cccc(F)c1C)=O)C2 21840,C1(C)(NC(C(CCC)O)=O)CCN(C(=O)CCC2CCC2)CC1 21841,c1(C(N2CC(CNC(CN(CC)CC)=O)(OC)C2)=O)c(C)ccc(F)c1N 21842,Cc1cc(N(C)Cc2nncn2C)nc(NCC(N2CC(CS(C)(=O)=O)C2)=O)n1 21843,c1(C(=O)NCCC2(NC(c3cncnc3)=O)CCC2)ccc2nn[nH]c2n1 21844,C(=O)(CC(Cl)Cl)N(C)CC=CC(=O)N1CCC1 21845,N1(C(C2C(C)C2C)=O)CC2CCC1(CNC(C1CCC(C)(C)C1)=O)CC2 21846,c1(C2C(C(=O)NCC3C(NC(CNC=O)=O)C3)C2)cccnc1 21847,CCCCC(C)CCC(=O)N1CC2CC(C(=O)NCCCCCCO)(C2)C1 21848,N1(C(C(N2CCC(COC)C2)=O)=O)CCC(F)(COCCNC(C)=O)C1 21849,C1(C(=O)NC2CC(N(C(CCNC(C)=O)=O)C)C2)Cc2ccccc2S1 21850,N1(C(CCc2c(C)noc2C)=O)CCC(CNC(c2csc(C#N)c2)=O)C(C)C1 21851,Cc1c(Cl)ccc2c(CC(=O)NCC3CCCN3C(=O)CC(=O)O)c[nH]c12 21852,CC1CC(CNC(c2cc(C(F)F)ccn2)=O)CN1C(=O)C(C)n1cccc1 21853,c1(-c2cncc(C(=O)NCCC(N)=O)n2)ccc(Br)c(O)c1 21854,C1(CNC(CCc2cn(C)nn2)=O)(CO)CCN(C(=O)CCC2CC2(C)C)C1 21855,CN1CCC2(CCN(C(CC3CC(F)(F)C3)C(=O)NC3CCCCC3)C2)C1 21856,N1(C(C=CC(C)C)=O)CCC2CC(NC(C3CC(=O)N3)=O)CCC2C1 21857,O=C(CCCCCNC(=O)CC1COCCO1)NCC12CCC(CC1)O2 21858,C(=O)(n1ncc(OC)c1C(F)(F)F)OCC.C1C(C(F)(F)F)N1 21859,C(=O)(C(O)CC(C)C)NCC1(COC)CN(C(=O)CCC2(C#N)CCC2)C1 21860,c1(CC2CCN(C(=O)NC(c3nc[nH]n3)C)CC2)cccc(Cl)c1 21861,c1(C(=O)NC(CN(C(c2ccnc(OC)n2)=O)CC)C)cc(Cl)cc(Cl)c1 21862,C1(NC(c2cc(CCC)on2)=O)CN(C(c2cccc(N)c2N)=O)CC1(C)C 21863,C1(C(=O)OC23CN(C2)C(=O)C(C)NC3=O)CCC(C)(C)O1.c1(OCC)ccccc1 21864,C(CC(C(C)(C)C)NC(c1coc(Cl)c1)=O)N(C(=O)CC1CCOCC1)C 21865,C(=O)(C1=CC2(CCOCC2)C1)NCC1CCC(CNC(CCC2C(C)C2)=O)CC1 21866,N1(C(c2c(OC)cc(OC)nc2)=O)CC2CC(C1)N(C(C1CCC3(CC1)N=N3)=O)C2 21867,CC1C(C(N2CCC(C3CCCCN3C(c3ccc(Cl)o3)=O)CC2)=O)CCN1C 21868,N1(C(CC2COCC(C)O2)=O)CCN(C(c2cccc(CO)c2)=O)C(CO)C1 21869,C(=O)(C1=NNC(=O)CC1)N(CCN(C(=O)C(c1ccccc1F)C)CC)CC 21870,CC1(C)CCCC(CC(N2CCC3(CC3NC(=O)CCN3CCCC3)C2)=O)C1 21871,C(=O)(C(C(C)C)C1CCC1)NCC(NOCCCC=C)=O 21872,C12CCCCC1NCC(=O)N2.n12cc(nn1)C2.C1C(=O)N1.C(=O)(C1CC1)NC 21873,c1(CC(=O)N(CC(CC)NC(=O)CC2CCC2(F)F)C)ccc(F)cc1 21874,CN1C(=O)C2CN(c3ccc(C(F)(F)F)nn3)CC2C1=O.C12CCN(CC1)C2=O 21875,c1(NC(C(=O)NC2C(C)(C)C(CN)C2)=O)ccc2c(c1)NC(=O)CO2 21876,c12ccccc1OC(CC)CN(C)C(=O)CC2O.C(=O)(CC(C)C)NC1CCCC1 21877,C1(CC=C)(NC(=O)CC(C)OC)CCN(C(=O)CSC(F)(F)F)C1 21878,Cc1cc(=NC(C)c2ccc(Cl)c(F)c2)[nH]c(=NCc2cccc(F)c2Cl)[nH]1 21879,c1(SC)ccc(NC(C2CC(=O)NC(c3ccccc3)C2)=O)cc1Cl 21880,N1(C(=O)CCC2CCC2)CCC2(CC1)CCN(C(C1CC1CF)=O)C2 21881,C(=O)(N=c1ccc2nnnn2[nH]1)Nc1cc(C(=O)OC)n(C)n1 21882,N1(CC)CCS(=O)CC1c1ccccc1.c1(N2CC(C)=CC2=O)ccc(F)cc1 21883,C(=O)(CC(C)C(F)(F)F)NC(CC)CCC(=O)NCC1CC12CCCC2 21884,Cn1cnc(NCC2CCCN(C(c3ccc(C(F)(F)F)s3)=O)C2)c(Br)c1=O 21885,c1(CC(=O)NCC2(OC)CN(C(=O)C=NOC)C2)ccc(-c2ccccc2)cc1 21886,C(C(C)C)(C(C(=O)Nc1ccc(F)cc1)N(C)CCOCC1CC1)OC 21887,C1(O)(CNC(=O)C(=O)NC2CCN(C(=O)Nc3ccccc3)C2)CCOCC1 21888,N1(C(C=C(C)C(C)(C)C)=O)CCC(CCNC(c2ccnn2C)=O)C(F)(F)CC1 21889,C(=O)(C(CCNC(c1ccn(C(C)C)n1)=O)OC)NCC#CCC 21890,C1(C(=O)NCCNC(C(C)SC)=O)CCNC(=O)C1 21891,CN=c1nc(N(C)Cc2cccc(O)n2)[nH]c(=NC2Cc3ccc(Cl)cc3C2)[nH]1 21892,C1(C(=O)Nc2cnc(CC)nc2)CN(C(=O)CC2CCCN2CC)C2(CCC2)C1 21893,c1(OCC)ccc(CNc2cnccc2OC(F)F)c(C(F)(F)F)c1 21894,C1(C(=O)NCC2C(NC(C(C=C)(C)C)=O)C2)CCOC(C)(c2ccccc2)C1 21895,N1(C(C(C)NC(C)=O)=O)c2ccccc2CCC1C(=O)NCC1CCC(C)CC1 21896,C1(NC(C2N(S(C)(=O)=O)CC2)=O)CCC(C)N(C(C2(c3ccc(F)s3)CC2)=O)C1 21897,Cc1ccc(F)c(C(=O)NC2CC3CCC2(NC(C2CCC(C)(C)C2)=O)C3)c1 21898,C1(NC(C2CC(CNC(CC3(N(C)C)CCC3)=O)OC2)=O)C(C)(C)C(O)C1(C)C 21899,C(CC(=O)N(CCNC(C1(n2ccnn2)CC1)=O)C1CC1)=CCC 21900,c1(C(=O)NCCC(C)N(C(C2C(CC)OCC2)=O)C)c[nH]cc(Cl)c1=O 21901,FCCN=C(NCC=Cc1ccco1)NCC(c1ccccc1)N1CCCC1 21902,N1(c2c(Br)cnc(OC)n2)CCC2(CC1)CCN2Cc1ccc(Cl)nc1 21903,c1(OC)cc(C2(C(=O)NCCCC(C)NC(=O)C(O)CSC)CCCC2)ccc1C 21904,c1(-c2ccc(SCC)s2)c(C(=O)NC)nc2ccccn12 21905,c1(C(N(CC#C)C(C)C)=O)cc2ccsc2[nH]1 21906,N1(C(C2C(C)(C)C2)=O)CC2CCC(NC(c3ncoc3C3CCC3)=O)C2C1 21907,C(C(C(=O)NC(C)CNC(=O)C(=O)N(CC(F)F)C)C(F)(F)F)OC 21908,C1(O)(CN(C(CC2(CC)CC2)=O)C)CCN(C(c2ccc(C(C)=O)[nH]2)=O)C1 21909,C1(CNC(c2cncc(NC(c3ccccn3)=O)c2)=O)CCc2ccccc2C1 21910,C1(CNC(COC)=O)CC2CCC1N2C(=O)Cc1ccc(OC)c(O)c1 21911,c1(CN(C(c2conc2C)C(=O)NC2CC(F)(F)C2)CCOC)ccccc1 21912,c1(CC(=O)NCCN(CCC)C(C2CC2(Cl)Cl)=O)ccnc(O)c1 21913,C1(CC)CCCN(c2nnc(-c3ccccc3Cl)n2CCC(C)C)C1 21914,N1(C(C(C)(C)OC)=O)CCN(C(c2ccc(F)cc2Cl)=O)C(C(C)C)C1 21915,Cc1ccc(C(=O)NCC2(NC(C3CC(F)(F)C3)=O)CCOC2)nc1O 21916,N1(C(CC(=O)NCC)=O)CCN(C(c2c[nH]c(=N)o2)=O)C(CC(F)F)C1 21917,CCC(CCC(=O)NC1(CNC(c2ccc(CC)c(O)c2)=O)CCC1)OC(C)=O 21918,N1(C(c2ncc(CC)cn2)=O)CCCC(O)(CNC(C2CCCC(=O)N2C)=O)C1 21919,N1(CCN(C(C)C)C(C(c2ccc(Cl)cc2)C(N)=O)=O)CCCCCC1 21920,N1(C(C2C(C(=O)O)C23CC3)=O)CCc2c(I)n[nH]c2C1 21921,N1(C(CCCCOC)=O)C2CCC1CC(CNC(=O)CC1CC(C)=NO1)C2 21922,CCC(C)C(C(=O)NCC(F)F)N(C(=O)C(=O)NCCOC)C 21923,C1(C(=O)NC)CCN(C(=NCCC(C)C)NCc2ncccc2F)C1 21924,c1(C(N2C(C(N3CCOCC3CCO)=O)(COC)C=CC2)=O)cc(C)cc(C)c1 21925,C(C(C)N=c1[nH]c(=NCC2CC(=O)N(CC)C2)c2sccc2[nH]1)OCC 21926,CC(C)C(C)(O)C(=O)NC(CNC(c1cncnc1-c1ccccc1)=O)C1CC1 21927,CN1CCC2(CC1)CN(C(C1CCN(C(C3(C)CC=CC3)=O)CC1(C)C)=O)C2 21928,c1(C(=O)NCCC(C)NC(c2cc(-c3cccs3)on2)=O)csc(O)n1 21929,C1(C2(O)CN(C(C3(C)COC3)=O)C2)(CNC(c2csc(C)c2C)=O)CC1 21930,c1(OC)cc(Br)cc2c1NC(=O)CCCOC(=O)C2.C(C(F)(F)F)SC(C)(C)C 21931,N1(C(C(C)Cc2ccc(Cl)cc2)=O)CC2CCC(C1)N2Cc1ccc(F)nc1 21932,c1(NC2(C(=O)NC(COC)C(C)C(C)C)CCCCC2)ncc(Cl)cc1[N+](=O)[O-] 21933,CS(=O)(=O)c1ccc(S(=O)(=O)N2CCOC3(CCC(NC(N)=O)CC3)C2)cc1 21934,N1(C(c2ccc(CC)s2)=O)CCC(C2CN(C(c3c[nH]c(C#N)c3)=O)C2)CC1 21935,CCN=C(NCC1CCCCO1)NC1CC(=O)N(C(C)(C)C)C1 21936,N1(C(C=C(COC)C)=O)CCC(C2(NC(=O)C(C)(C)OCC(F)(F)F)CC2)C1 21937,c1(Cc2ncc(SC)cn2)cnn2c1CN(Cc1ncccn1)CC2 21938,C1(COCCC(=O)NC(C(OC)OC)C)CC(=O)N(C2CN(C(=O)OC)C2)C1 21939,c1(C(=O)NCCC(C)NC(Cc2ccc(C)c(F)c2)=O)ccc2c(n1)OCCO2 21940,c1(CC(=O)NCC(CNC(C2(CC)CCNC2=O)=O)C)c(C)nc2ccccn12 21941,C1(C(N(C(C)CNC(c2c(C)cc(C)cc2C)=O)CC)=O)CCCCC12CCC2 21942,C1(C(N(C)Cc2c(CC)noc2)=O)CC(=O)CN1C(=O)Cc1ccon1 21943,C(CCCCC(=O)NC1CCC(NC(=O)CC2CCCC(C#N)C2)CC1)OCC 21944,c1(CNC(C(C2CCC2)NC(c2cc(Cl)n[nH]2)=O)=O)ccncc1F 21945,C(=O)(C(F)CCC(C)C)NC1CC(C(C(=O)NCC2(CC)CCC(=O)N2)F)C1 21946,Cc1ccc(OC(C)C(=O)NCCCC(C)(C)NC(=O)CC2(O)CCCC2)cc1 21947,c1(C(=O)NC(CN(C)C(c2cc(F)cc(F)c2)=O)(C)C)cnc2[nH]cncc1-2 21948,C1(SCC)CCCN(C(=O)CN2CCNCC2)C1 21949,C(=O)(CC(C)(C)C(C)(F)F)N1CCN(C2CCN(C(C)C(=O)NC3CC3)CC2)CC1 21950,c1(C(=O)NC2C(NC(c3c(C)nn[nH]3)=O)CC2)cc(Br)c2ccccc2c1 21951,c1(CN2CCCC(OCCC)CC2)ccc(Cl)c(Cl)c1C 21952,Cc1cc(C)c(C(=O)NCCCC2CCCCN2C(=O)Cn2cnnc2)c(C)c1 21953,N1(C(C2N(C(C(C)=CC3CC3)=O)CCN(C)C2)=O)CCC2CCC(C1)N2C 21954,CCCC(C)(C)C(=O)NCC(C)(O)CNC(=O)CSc1ccc(C(C)C)cc1 21955,C1(Cc2nc(C)sc2)CCN(N2CCOCC3(CC3)C2)C1 21956,N#CC12CCC(C(=O)NCC3CCN(C(C4CC5(CC5)CO4)=O)CC3)(CC1)CC2 21957,N1(C(COCCC)=O)CC2CC2(CN(C)C(C2CC(c3cccc(F)c3)C2)=O)C1 21958,N1(C(CCc2cc(C)[nH]n2)=O)CCCCC1CC(=O)NC(c1csnn1)C 21959,Cc1cnccc1C(=O)NCCC1CCCN1C(C1COC1)=O 21960,c1(CNC(CC(N)=O)C(N2CC3CC3(C(N)=O)C2)=O)cccc(=O)o1 21961,C1(CNC(C2CCC2(F)F)=O)C2CN(C(C3CC4CCC3C4)=O)CC12 21962,Cc1cc(C(=O)N(C(CNC(=O)C(C)CO)C2CC2)C)nn1CCO 21963,CCC1=NOC(C(=O)NC(CCC2CCC2)C(=O)Nc2ccccc2OC)C1 21964,C1(CNC(C(C)SC(F)(F)F)=O)CCN(C(=O)CCS(C)(=O)=O)C1(C)C 21965,Cc1ccc2c(N3CCN(C(C)C)CC3)nc(=NC3CCCCCC3C)[nH]c2c1 21966,C1(CC(=O)N(CCNC(c2c(C)cc[nH]2)=O)C)CCCCN1C 21967,C(=O)(C(C(C)C)N1CCCCC1)N(C1CCN(C(CN(C(C)=O)C)=O)C1)CCO 21968,CC(C)(C(=O)N1CC(C2CN(C(c3cc(C#N)ccc3O)=O)C2)C1)C1=CCSCC1 21969,C#CCC(C(=O)NC(C)Cc1cccnc1)NC(=O)C=CC(C)C 21970,C1(C(N(CC(O)C2CC2)C)=O)CCN(C(c2c[nH]c(C(N)=O)c2)=O)C1(C)C 21971,C1(C)(C(=O)NCC2N(C(COC(C)=O)=O)C3CCC2C3)CC(C(C)C)=NO1 21972,Cc1cccc(CNCCNC(C2CCCN2C(=O)Cc2ccccc2I)=O)n1 21973,N1(C(C2CC3(CCN(C(C(C=C)C)=O)C3)C2)=O)CCCC2(CCCC2)C1 21974,C(=O)(C1=CNS(=O)(=O)N=C1C)N1CC(OC)(CNC(C2(S(C)(=O)=O)CC2)=O)C1 21975,Cc1ccc(C(N2CC(CNC(c3ccccc3C)=O)CC2C)=O)c(C(C)C)n1 21976,C1(NC(c2cc(SC)c(C)o2)=O)CCN(C(c2cccc(F)c2)=O)C12CC2 21977,Cc1cncc(C)c1C(=O)NC1(CO)CCC1.N1(C(C=CC)=O)CCC(CC(N)=O)C1 21978,C(=O)(C(CCOC)NC(=O)CCc1ccc[nH]1)N(CC(CCC)O)C 21979,N1(C(C(COC)NC(=O)C(C)C#N)=O)CC(C)OC(C)(C)C1C 21980,c1(Cn2c(C3C(O)CCC(C)C3)nc(C3CSC3)n2)ccc(S(N)(=O)=O)cc1 21981,N1(C(C)=O)CC2CC(N(C(c3cnsn3)=O)Cc3ccc(NCCC#N)cc3)C1C2 21982,N1(C(c2c(C)c(F)ccc2Cl)=O)CC2CC3CC2C1C3NC(=O)Cc1ccno1 21983,Cc1ccn2ncc(C(=O)NC3CC(C)N(C(c4ccnc(Cl)c4)=O)C3)c2c1 21984,c1(CCNC(c2cccc(NC(=O)NC)c2)=O)c[nH]c2cc(F)c(Cl)cc12 21985,CCC(C)(CNC(c1ccnc(C)n1)=O)C(=O)NCC1C=CCCC1 21986,N1(C(C2(C(F)F)CC2)=O)CCN(CCCNC(C2CC(CC)C2)=O)CC1 21987,CC1CC2(CCN(C(=O)CC3CCCC3)CC2)CN1C(=O)CCCCC(C)(C)C 21988,Cc1cnn(C(C)C(=O)NC2(CCNC(c3ccn(CCF)n3)=O)CC2)c1 21989,C1(O)(CC=C)CCN(C(c2conc2CNC(C2CC(=O)CS2)=O)=O)CC1 21990,c1(C(=O)NC(CNC(CCn2ccc(C)n2)=O)C)ccc([N+](=O)[O-])s1 21991,n1(CC)cnc(C(=O)NC(CNC(=O)CC2(C)CC2(F)F)C2CC2)n1 21992,c1(C(N2CC(O)(C(C)NC(C3CCOC3)=O)C2)=O)coc2c1CCCC2 21993,C1(C(C)C(=O)NCCCc2ccsc2)CCN(C(c2scnc2Cl)=O)CC1 21994,CN1CCC2CN(C(C3CCCN(C(C4CCCN4C=O)=O)C3)=O)CC2C1 21995,C(=O)(CCCC(=O)N1CCN(C(=O)CC2CCCSC2)C(C2CC2)C1)N(C)C 21996,C12COCCC1C(=O)NCCn1cc2nn1.n1(CC(C)C)ccc(C(F)F)n1 21997,c1(C(=O)NCC2(OC)CCC2)cccc(CNC(=O)CCOCC(C)(C)C)n1 21998,c1(C(C(=O)NCC(CC=C)NC(=O)C(C)NC(C)=O)(C)F)ccc(F)cc1 21999,Cc1oc(C2CC2)nc1C(=O)N(C(C)CNC(=O)C(O)Cc1ccccn1)C 22000,c1(CN2CC3C(Nc4cc(OC)ncn4)C3C2)c(Cl)cc(Br)cc1Cl 22001,C(COc1ccccc1)(C(=O)NC(CNC(=O)C(C1CC1)OC)C1CCC1)OC 22002,C(=O)(CCCCC(C)CC)N1CC(NC(CC(=O)NCC#C)=O)C(CC)C1 22003,C(CNC(=O)CN(C)C(C)C)(CCNC(=O)CCc1nccn1C)OC 22004,c1(C(=O)NC2CCC(C)N(C(c3cccnn3)=O)C2)cccc2c1CCCCC2 22005,C(c1c(C)coc1C)=CC(N1CCC(C(C)(C)NC(C2C(=C)C2)=O)C1)=O 22006,Cc1nc(OC2CCCC2)ccc1C(=O)NCCSc1ccc(O)cc1 22007,c1(NCC(C)(C)C2CCOC2)[nH]c(=NCCc2ccn(C(F)F)n2)nc2scnc12 22008,N1(C(CNC(NCC)=S)=O)CC2(C1)CN(C(=O)CC1CCC(=O)N1)CC2CO 22009,C(C(C)(C)CC)(c1n(CCOCCOC)nnn1)NCc1cn(C)cn1 22010,c1(OCC)c(C(N2CCC(NC(c3ccc(C)cc3O)=O)C2)=O)cccc1F 22011,C1(NC(COC)=O)(CNC(=O)Cc2nnc(-c3ccco3)o2)CCCC1 22012,CC(=O)C(C)CC(C)C(=O)N1CCC(C)(C)CC1C(=O)N(CC(O)C1CC1)C 22013,c1(CN2CCC(CC(N3CC4CC4C3)=O)CC2)cccc2ccncc12 22014,C1(CNC(=O)CCN2CCC2)CCN(C(C23CC(C(F)F)(C2)C3)=O)CC1 22015,C12(C(=O)NCc3snc(CC)n3)C(NC(=O)CC3CCOC3(C)C)C3CC1C2C3 22016,Cc1cccc(C)c1C(N1CCC(F)(CNC(C2CCC2C(F)F)=O)CC1)=O 22017,c1(CC)nc(=NCC2CN(C(=O)CCOC(C)C)CCO2)s[nH]1 22018,C(C(C)(C)CCNC(=O)C(F)(F)c1ccccn1)NC(c1cc(COC)on1)=O 22019,c1(OC)cc(Br)c(CC(=O)NCC=CCNC(=O)C(N)=O)cc1O 22020,C1(CC=C)(NC(c2cnc(C(C)(C)CF)o2)=O)CN(C(c2cc(CC)cs2)=O)C1 22021,Cc1cc(C)c(CN2CCC(N(C(=O)C(C)C)C)C2)cc1C 22022,c1(CC)ncc(C(=O)NCC2CCN2C(=O)CC2CS(=O)(=O)C2)c(C)n1 22023,c1(CC#C)onc(C(OC(F)F)C)c1CSc1cccs1 22024,C1(NC(C=CC(N)=O)=O)CC2CCC(C1)N2C(=O)Cc1ccc2c(c1)CCO2 22025,Cc1cccc2c1ccn2CC(=O)OCC(=O)OC1CCC(C)(C)CC1 22026,N1(C(CC2C(C)(C)OCC2)=O)CC2CCC(C1)N2C(C12CCCN1CCC2)=O 22027,CC(C)CC(CNC(=O)CC1CCC(=O)C1C)C(=O)NCC(C)(C)N(C)C 22028,Cc1cc(C(=O)NCCc2ccn(C)n2)nn1C(C)(C)C 22029,c1(C(N2CC(CNC(C3CN(CC(C)C)C3)=O)C2)=O)ccc2c(O)ncnc2c1 22030,c1(CNC(CCOCCC)=O)cnn2c1CN(C(=O)Cn1ncccc1=O)CC2 22031,c1(C(=O)NCCCCC2CN(C(C(C(C)O)(F)F)=O)C2)cc2ccsc2n1C 22032,c1(C(=O)NCCCN(CCCNC(c2ccon2)=O)C)cccc2c1NCC2 22033,N1(C(c2cnn(C)c2Cl)=O)CCC2(CCN(C(C3CCC(C4CC4)CC3)=O)C2)C1 22034,C=C(Cl)CCC(=O)NCC1CCN1C(c1ccnn1CCCC)=O 22035,C(=O)(C1CCc2nccn21)NC(C)C(=O)NOC1CCCCCC1 22036,C(N=c1[nH]c(N2CCC(c3nncs3)C2)nc(=N)[nH]1)c1cn(CC=C)nn1 22037,C1(C(=O)NCC2C(C)CN(C(=O)Cc3ccco3)C2)CCc2ncncc2C1 22038,C12(NC(C(C)=CC3CC3)=O)CCC1CN(C(c1ccsc1C)=O)C2 22039,Cc1cc(NC(C)CC(C)NC(=O)Cc2c(F)cccc2F)n2nc(C)nc2n1 22040,C(=O)(CS(=O)(=O)N1CCOCC1CNC(c1ccc(CF)nc1)=O)OCC 22041,c1(N(C2CCCNCC2)C(c2cc(Br)cs2)=O)ncc2[nH]ncc2n1 22042,c1(C(CC)C(=O)NCC(C)NC(c2ccn(C)c2)=O)ccc(Cl)cc1 22043,CC1CCC(NC(=O)Cc2cn[nH]c2)CN1C(c1ccc(O)nc1Cl)=O 22044,Cc1cc(NC(C23CC2CN(C(c2ccno2)=O)C3)=O)c(F)c(Br)c1 22045,C1(C(N2CC3(CC(=C)C3)C2)=O)COC2(C1)CN(C(c1cccc3ccnn13)=O)C2 22046,N1(C(c2c(OCCOC)cccc2)=O)CCC(NC(=O)C2=CCC2)C(CO)C1 22047,C1(C(=O)NCC(CNC(c2ccn(CC(C)C)n2)=O)(C)F)CCCCC(=O)N1 22048,c1(CNC2CCC(C(=O)NCc3ccn(C)n3)CC2)c(Br)ccc(Cl)c1F 22049,N1(Cc2cc(Cl)sc2Cl)CCC2(CCSCC2)C1 22050,c1(COC(C2(NC)CC2(C)C)=O)cc(Br)ccc1F 22051,C(=O)(CS(=O)CCC(F)(F)F)N1C2(CNC(CC=CCC)=O)CCC1CC2 22052,c1(C2C(C(=O)NCC(C)(C)N)C2)c(F)cccc1F.C(=O)(CCC(=O)OC)CCF 22053,N1(C(CCCC)=O)CCC2CCCC12C(=O)NCc1cncs1 22054,c1(C(=O)NCC2CC(C)N(C(=O)CC3(C)CC3(F)Cl)C2)cnc2occc2c1 22055,C1(C(N(CCCNC(c2c(OC)nsc2)=O)C2CC2)=O)CCSC(C)C1 22056,Cc1cnc(C(N2CCCC(CN(C)CCc3cnn(C)c3)C2)=O)cn1 22057,c1(CC(N2CCCC(NC(c3c(C)nns3)=O)(CO)C2)=O)ccc2ccoc2c1 22058,C(C)(C(=O)N1CCC(CC(=O)NCC(C)CC2CC2)CC1)(C(C)C)OC 22059,C(CCN=[N+]=[N-])CC(=O)NCCN(CCC(C)N(CCC)C)C(=O)C(F)C1CCCC1 22060,C(=O)(CCCCC(=O)NOC(C)(C)C)N1CCC(C(=O)OC2CCNC2=O)(OC)C1 22061,C(=O)(C1=CCCOCC1)N(C(C)CNC(=O)CC1CCC(C(=O)OC)CC1)CC 22062,Cc1cc(C)c(C(=O)NCC2CCCC2NC(c2cccc(O)n2)=O)cn1 22063,c1(C(N2CC(NC(c3ccc(CC)o3)=O)(CO)C2)=O)c(C)nnn1CC 22064,C1(CCNC(C(c2cscn2)N(C)C)=O)CC2CCC(C1)N2C(c1cscn1)=O 22065,N1(C(c2ccc(C(C)=O)nc2)=O)CCC(NC(C2(Br)CC2)=O)C1(C)C 22066,C1(C(=O)NC(C(C)NC(c2cc(C)n(C)c2C)=O)C)CN(C)CCN(C)C1 22067,N1(C(c2c(C)snc2)=O)CCC(NC(=O)CC(C)c2cccnc2)C(F)(F)CC1 22068,C1(CC)CCCCC1C(=O)NC(C)(C)CNc1cc(C(=O)OC)no1 22069,c12cc(ccc1C)C(=O)Nc1ccc-2cn1.CCCCS(=O)(=O)N1CCNCC1 22070,C#Cc1ccc(C(N2CCCC(COC)C2)C(=O)NCC(=C)C)cc1OC 22071,c1(CC)conc1C(N1CCCC1C1CCN(C(c2cnc(C)s2)=O)C1)=O 22072,N1(C(c2c(CNC(CCC(C)OCC)=O)cnn2C)=O)CCCC12CCCC2 22073,Cc1ccc(C(C(=O)NCC=CCNC(=O)CCCC2CC2)SC2CC2)cc1 22074,c1(CN2CCC(N3CCN(CCCOC)CC3)C(C)(C)C2)ccc2nonc2c1 22075,N1(C(C2C=C(C)CS2)=O)CC(F)CC1C(=O)NOCCC(C)O 22076,C1(N(CCOC)C(c2ccncc2)=O)CCN(C(=O)C(C)(C)n2cccn2)CC1 22077,c1(-c2scc(C)c2)cccc(C2(N3CCN(c4nc(=N)[nH]s4)CC3)CC2)c1 22078,C1(CC(=O)NCCCOCCCO)CCC(C(=O)Nc2cccc(F)c2)CC1 22079,C1(NC(c2ccc(NC(C3CCOCC3)=O)cc2)=O)CCC2CC1CN2 22080,c1(C(N(C2CCN(C(C3CC3CN(C)C)=O)CC2)CC)=O)ccc2c(c1)CC2 22081,c1(SC)cc(NC23CCC(CNC(=O)C(C)(C)C)(C2)OC3)nc(SC)n1 22082,c1(C(=O)NCC2CC(C)(C)N(C(=O)CCC(F)(F)F)C2)cccc2c1CCC2 22083,c1(C(=O)NC2(C(N3CC(C)(CC=C)C3)=O)CCCCC2)cnc(C)c(C#N)c1 22084,N1(C(Cc2ccc(C)s2)=O)CCN(C(=O)C=Cc2ccoc2)C(C)C1C 22085,C(=O)(C(CNC(=O)Nc1cnc(S)nc1)C(C)(C)C)N1C(C(N)=O)CCC1 22086,C(=O)(C(C)CCCC(C)C)N1C(C(=O)N(CC(C)(C)N(C)C)C)CC(OC)C1 22087,c1(NCCN2CC(C)C=C(C)C2)cc(=NC(=O)CCOCCF)[nH]n1C 22088,C1(NC(c2ccnc(C)n2)=O)CN(C(c2sccc2Cl)=O)C2(CCCCCC2)C1 22089,c1(C(=O)NCCC(C(C)C)NC(=O)CC2NC(=O)NC2=O)ccc2[nH]ccc2n1 22090,N1(C(C(CC)OC)=O)CC2(C1)CN(C(C1(CCOCCO)CCCC1)=O)C2 22091,C1(C(=O)NCC(COC)O)(NC(=O)Cn2ccnc2)CCOCC1 22092,c1(C(N2CCCC(c3cn(C4CCC4F)nn3)C2)=O)cc2scc(Cl)c2[nH]1 22093,C1(NC(COCC)=O)CCN(C(c2cc(C)n(-c3nccs3)c2F)=O)C(C)C1 22094,c1(NC)cnc(C(N2CC3C(C(=O)NCCn4ccnc4)C3C2)=O)cn1 22095,N1(C(C2CCN(C)C2=O)=O)C2CCC1CN(C(=O)CC(C)(C)c1ccccc1)C2 22096,C12(CNC(C3C(NC(c4c(C)nc(Cl)s4)=O)C3)=O)CC3CC(CC(C3)C1)C2 22097,CCCCCC(C)CC(=O)NCC1CCC2(CN(C(C3CC(C)(CO)C3)=O)C2)O1 22098,CN1CCOc2cc(C(N3CC4CN(S(=O)(=O)CC5CC5)C4C3)=O)ccc21 22099,N1(C(C(C2CN(C(CC=C)=O)C2)OC)=O)CCC2(CC(OC)C2)C1.c1(C)ccn(C)n1 22100,CC1OCCCC1C(=O)NC(C)CNC(c1cccc(OC(C)(C)C)c1)=O 22101,C1(O)(CNC(C=NOC)=O)CCN(C(c2csnc2C)=O)C1 22102,C1(C)(C(=O)NC2CCC(OC)C2)CCN(C(=O)Cc2cnc(C)s2)CC1 22103,N1(C(CCn2ncc(C)c2)=O)CC(CNC(C2CCC(=O)NC2)=O)CC(C)(C)C1 22104,C(C(CNC(C1C(C)C1C)=O)CO)NC(C1C(OCC)C1)=O 22105,CC1c2cc(C(=O)NCCCCN(C)C(c3ncn(C)n3)=O)ccc2OC1C 22106,C(=O)(C(C)(C)CC(=O)NC(C)C(C)NC(c1cc(=O)cc(Cl)[nH]1)=O)OCC 22107,C1(NC(C=C(CC)C)=O)CC(NC(c2ccc(S(C)(=O)=O)o2)=O)C12CCOCC2 22108,c1(CN2CC(F)(C(=O)NCCc3ccc(OC)cc3)C2)cc(F)cc(Br)c1Cl 22109,C(=O)(CC(F)(F)C(F)F)N1CCC(CNC(C2(C)CCNC(=O)C2)=O)(CO)C1 22110,N1(C(c2c(SC)csc2)=O)CC2CCCC2(NC(C2OCCC2(C)C)=O)C1 22111,N1(C(c2ccc(CC)nc2)=O)CCC(NC(=O)CC(C)(F)F)C(C)C1 22112,Cc1cn(C(C)(C)C(=O)NC(C)C)cn1.N1(CC(=O)N)CCOCC1.C1(CN)(C)CC1 22113,C(C(=O)NC1CCC(NC(=O)CN2CCCC2C)CC1)(C(C)(C)C)NC(=O)OC 22114,C1(CNC(C(CCC)OC)=O)CC2(CCOCC2)CN1C(=O)CN(C)C 22115,S(=O)(=O)(CC(=O)NC1(C)CC(NC(C2CC23CCC3)=O)C1)NCC 22116,N1(C(=O)NC)CCN(C(c2cn[nH]c2)=O)CC1C(F)F.C1(C)C(=O)N1 22117,Cc1cc(C(N2CCOCC2C(O)CO)=O)ccc1C#N 22118,N1(C(CC=C)=O)CC(CNC(c2ccc(F)c(Cl)c2F)=O)C2(CCOCC2)C1 22119,C(=O)(C(C)S(C)(=O)=O)NCCN1CCN(C(c2c(OCC#C)nccc2)=O)CC1 22120,c1(C(N2CCN(C(=O)CC3CCN(CC(F)(F)F)C3)CC2)=O)c(F)ccnc1Cl 22121,C1(S(N)(=O)=O)(C(=O)NCC(C)N(C)C(c2cc(Cl)cn2C)=O)CCC1 22122,c1(C(N2CC(CCNC(=O)CC3CCCCCO3)C2)=O)cnn2cnnc2c1 22123,Cc1nc(CCNC(c2cccnc2-n2nccn2)=O)c(C)o1 22124,c1(CC)c(C(=O)NCC(N2CCN(C(=O)CCC#N)CC2)=O)nnn1CC 22125,C1(N(C)C(C2CCOC2)=O)CCCN(C(c2cc(O)ccc2Br)=O)CC1 22126,C(=O)(C(O)CCC(F)(F)F)N1C(CN(C(=O)CCc2nccn2C)CC)CCC1 22127,C1(NC(C2C(C)(C)C2)=O)CC(NC(=O)CNC(C2CCC2)=O)C12CCC2 22128,N(C1CCC(Nc2ncc3c(n2)COC3)c2ccccc21)C(C1CC1(F)F)=O 22129,CC(C)C(CC(=O)NC1CCC2(CCC2)C1)NC(=O)C(C)CC#N 22130,C1(OC)CCCCN(CC(=O)NC23CC(Nc4cccc(OC)c4)(CO2)C3)CC1 22131,c1(-c2nn(C(NOCC)=O)c(CC3CCOC3)n2)ccc(F)c(Cl)c1 22132,C1(CCNC(Cn2ccc(C)n2)=O)CCN(C(C2CC2C(C)(F)F)=O)CC1 22133,C1(C(=O)NCc2ccnnc2)CC2CCCC2N1C(C1CC12CCCC2)=O 22134,N1(C(CNC(c2ccc(CC)cc2)=O)=O)CC2CCCCCC2C1 22135,C1(NC(CCC(N)=O)=O)CC2(CCN(C(c3cncc(OC(F)F)c3)=O)CC2)C1 22136,c1(CC(=O)NCC(C)CNC(=O)Cn2cnc(C#N)n2)cc(F)ccc1F 22137,c1(NC(c2scc(C(C)C)n2)c2nnnn2CCCF)cncn1C(F)(F)F 22138,N1(CC(=O)NC2C(CNC(CCC)=O)CCC2)CCN(C2CC2)C1=O.C(C)(=O)O 22139,CC#CC1CCN(C(=O)CC2CCCC2NC(=O)C(O)C(C)(C)C)C1 22140,C1(CNC(CNC(=O)OC)=O)CCN(C(c2cc3c(ncn3C)s2)=O)CC1(F)F 22141,N1(C(CCOC(C)=O)=O)CCC(C)(CNC(=O)Cc2ccn(C)c2)C1 22142,c1(OC)cccc(F)c1C(=O)NCC1CN(C(c2c[nH]c(C)c2)=O)CCC1C 22143,C(=O)(C(O)CC(F)(F)F)NCC1N(C(CSc2nc(C)[nH]n2)=O)CCCC1 22144,C1(CCNC(c2c(C(C)C)noc2)=O)CCCCN1C(=O)C=CC1CCOCC1 22145,n1(CC)nnc(C(=O)NC2CC(c3c(C(=O)OCCOC)cc[nH]3)C2(C)C)c1C 22146,C1(C(N2CCOC(C3CCC3)C2)=O)(CC)CCN(C(C2CCC(C)(C)CC2)=O)CC1 22147,Cc1c(C(N2CCOC(C(=O)NCCC3OC(=O)NC3=O)C2)=O)cnn1C 22148,C1(NC(C(C)n2cnnn2)=O)CCCCCN(C(c2cn3ccnc3cn2)=O)C1 22149,c1(OC)ccc(C=CC(=O)NC2CCCC2NC(=O)CCN2CCC2)c(OC)c1 22150,Cc1cc(C(=O)NC(C2CC2(F)F)C)cc(F)c1Br 22151,Clc1cc2c(cc1Br)N(CC1CCCN1CC1CC1)CCCC2 22152,c1(C(=O)NC(C)CC(C)NC(=O)Cc2cnn(C)n2)cccc2c1CCCN2 22153,c1(CCC(=O)OCC(CCSCC)=O)ccnc(Br)c1 22154,N1(C(C2CC(=C)C2)=O)CC(CNC(c2ncccc2C(C)=O)=O)C(O)C1 22155,C1(COC)(NC(C2CCCN2S(C)(=O)=O)=O)CCCN(C(c2c[nH]nc2C)=O)C1 22156,C12(CNC(=O)COCC3CCCCO3)CC1CN(C(c1cc(C(F)F)on1)=O)C2 22157,Nc1cc(C(N2CC(NC(c3c[nH]nc3-c3cccc(Cl)c3)=O)C2)=O)cc(F)c1 22158,N1(C(C2N(C(C(C)OCCN(C)C)=O)CC=C2)=O)CCN(C)C(C)C1 22159,CCC(CCC(=O)N(C(C)CC(N)=O)C)NC(C1(C)CCCCC1)=O 22160,C#Cc1cccc(C(=O)NCC2COC(CNC(=O)C(C)(C)c3ccsc3)C2)c1 22161,C1(C(N2CC(NC(CCC(C)OCC)=O)C2)=O)CCC(=C(F)F)CC1 22162,CCCCC(CNC(=O)C=C1CCCC1)NC(=O)CNC(=O)NC1CC1 22163,c1(OC)cc(C(N2CCN(C(c3ccncc3OC(C)C)=O)CC2)=O)cnc1C 22164,c1(CN(C)C(C2CC(NC(CCN(C(C)=O)C)=O)C2)=O)n[nH]cc1C 22165,N1(C(COC(C)C)=O)CCC(C(C)(C)C)(CNC(=O)C(C)Cc2ccncc2)C1 22166,c1(-c2c(F)cc(C)cc2F)ccc2c(C(=O)NCC(C)(C)C)nn(C)c2c1 22167,c1(C(=O)NC(CN(C(c2ccc(COC)o2)=O)C)COC)occ2c1CCOC2 22168,CON1CCC(C(=O)NC2C(C(=O)NC)C2)CC1.C12(CC1(C)C)C(=O)N2 22169,c1(C(=O)NCC2CC(NC(C3(CC)CCNC3=O)=O)C2)cn2cccc(Cl)c2n1 22170,c1(CC)cnc(SCC)[nH]c1=NC1CN(C(c2nc3ccccn3c2F)=O)C1 22171,Cc1cc(CCNC(=O)C(=O)NC2CC(N(C)C)C2(C)C)c(C)s1 22172,CC(CN(C)C)C(=O)NCC(C1(N(C)C)CCC1)N(C)C.n12ccnc1C(=O)N2 22173,C(=O)(CS(=O)(=O)C(C)C)N1CCC(N(C(=O)C(n2ccnc2C)C)CC#C)CC1 22174,c1(NS(CC)(=O)=O)[nH]c(=NC2CC3(C2)C(F)(F)C32CCC2)nc2sccc12.C1CC1 22175,N1(C(c2ccn(C3CC3)n2)C(=O)NCC)CCc2c(cc(C#N)n2CC)C1 22176,C1(C(C(=O)NC(C)(CNC(=O)C=CC2CCCO2)CO)O)CCCCCCC1 22177,CC(c1ccc(F)cc1)=CC(N1CC(NC(c2c[nH]nc2[N+](=O)[O-])=O)C(F)C1)=O 22178,N1(C(CN2CC(C)(C)C2)=O)CCCC2CN(C(c3cc(N)ccn3)=O)CCC12 22179,C(=O)(C1=CC2CC=CCC12)N(CC(CNC(Cc1nc(C)sc1C)=O)(C)C)C 22180,C1(C(N(C)CCOCCCN(C(=O)C(F)(F)c2cscn2)C)=O)CCCC(F)C1 22181,CC1CC(C2CN(C(C3CCC3NC(c3ccnnc3)=O)=O)C2)=NO1 22182,C1(C(N(C)CC2(O)CCN(C(=O)CCC3CCC3)C2)=O)CCC(=C(F)F)CC1 22183,N1(C(c2cc(C)oc2C)=O)CCC2CN(S(=O)(=O)CCC(F)(F)F)CCC12 22184,CC1(C(N2CCC(OCC(=O)NC34CCC(CC3)C4)C2)=O)CCC2(CC1)CC2 22185,c1(OC)nc(Cl)ccc1C(=O)NC(C1CN(C(c2cc3sccc3s2)=O)C1)C 22186,c1(CCS(=O)(=O)NC(c2ccccc2F)C)c[nH]c2cc(Cl)ccc12 22187,N1(C(CCCC(C)NC(c2ccc(C)c(C)n2)=O)=O)CC2(C)CC1CCO2 22188,Cc1cnccc1C(C)C(N1CC(NC(=O)Cc2cncnc2)CC1C)=O 22189,CC1(F)CN(C(c2n[nH]c3ccccc23)=O)CCN(c2ncnc(Cl)c2Br)C1 22190,c1(C(=O)NCCC(C)N(C(c2c(COC)scc2)=O)C)ccc2c(c1)CCC2 22191,c1(C(=O)NC(CC=C)(C)C(F)F)n[nH]c2c1CN(C(c1nnn(C)c1CC)=O)C2 22192,N1(C(CN(C(C)C)C)=O)CCC2(CC2NC(=O)COC2CCCCCC2)C1 22193,CC1(C)CC(O)CCN(C(c2ccsc2Br)C(=O)NC2CCOCC2)C1 22194,c1(C(C(=O)NC2CC(CCNC(c3ccsc3)=O)C2)SC)ccccc1 22195,c1(NC(C)=O)ccc(C(=O)NC2COCC2NC(=O)CCc2nncs2)cc1 22196,N1(C(C(CO)OC)=O)CCC(NC(=O)C2=C(Cl)CCC2)C1(C)C 22197,N1(C(C(C)N(C(C2(C(F)(F)F)CC2)=O)C2CC2)=O)CC(CO)C(O)C1 22198,C1(NS(CCC)(=O)=O)CN(C(=O)CNc2nccc(OC)n2)CCC12CCC2 22199,n1(CC)c(C(=O)NCC2CC3CN(C(C4CC(O)C4)=O)CC23)cc2ccccc12 22200,Cc1c(C(N2CC3(C2)CN(c2nc(Cl)ncc2F)C3)=O)cccc1O 22201,c1(C(=O)NCC(c2ccccc2)NC(C(C(C)C)C)=O)c(N)cccc1Cl 22202,c1(CC2C(CNC(C(C)NC(C3(C(=O)OC)CC3)=O)=O)C2)ccc(C)cc1 22203,CCCCC(C(=O)NC1CC1(F)F)NC(=O)CSCC1CC1 22204,C1(C(=O)NCC(c2ccccc2)N(C)C(c2cscc2F)=O)(OC)CC(C)(C)C1 22205,c1(CNC(Cn2nc(C(=O)OC)c(C#N)c2)=O)cccc2c1C(=O)NC2 22206,N1(C(Cc2cccc(OC)n2)=O)CCC(C)(C)C(NC(c2cccnc2S)=O)C1 22207,c1(C(=O)NC2CC(NC(CCC3COC(C)(C)O3)=O)C(O)C2)ccc(Cl)cc1F 22208,Cc1ccc(C)c(C(=O)N(C)CC2CCCN(C(C34COCC(C3)C4)=O)C2)c1 22209,CC(C(C)C(=O)N1CCOCC1C(C)(C)C)NC(=O)C(C)C#N 22210,Cc1cc(C(=O)NC(CNC(C2(S(C)(=O)=O)CCCC2)=O)C2CC2)ncc1C#N 22211,c1(C(C)NCCC2COCC(C)O2)nc2c([nH]1)CCCC2 22212,Cc1cc(NC(=O)CSCC(C)C)ccc1NC(=O)C(C1CCOCC1)O 22213,C1(C(=O)NCCCOCCNC(C(C)Cn2ccnc2)=O)NC(=O)OC1C 22214,N1(C(C2(CC(C)C)CC2)=O)CC(NC(C2CCCOC2C)=O)C(O)C1 22215,C=CCC(CNC(=O)C(C)OCC1CC1)C(=O)NC1(CO)CC2CCCC12 22216,N1(C(CCN2CCN(C)CC2)=O)CCC2(CC1)CC(N1CCC(F)(F)C(O)C1)C2 22217,c1(C(=O)NCC2CCC(NC(c3sc(CC)c(C)c3)=O)C2)cc(C#N)ccc1F 22218,C(C(F)(F)CNC(=O)CCCN(C(=O)C(O)Cc1ccco1)C)OC 22219,c1(C(N(CCC(C)NC(=O)C(=Cc2c[nH]cn2)F)C)=O)cc2scc(Cl)c2[nH]1 22220,CC(C)C(C)C(CNC(c1cccc(N2CCCC2=O)c1)=O)NC(=O)C=CBr 22221,OC1(F)NC(N=c2[nH]c3c(c(=NCc4cccc(Cl)c4Cl)[nH]2)SCC3)CC1CO 22222,C1(OC)CN(C(C2(CC(C)C)CCC2)=O)CC1NC(=O)CSC1CCOC1=O 22223,c1(OC)cc(C)c(CN2CC(O)(CNC(c3ccsc3Cl)=O)C2)cc1OC 22224,Cc1nn(C)c(C(=O)NCCCC(C)NC(=O)CCCC#N)c1Br 22225,Cc1cc(CC(=O)NCC(C)(CC2CC2)NC(=O)C(O)CN2CCCC2)n[nH]1 22226,c1(C(N2C(C(N3CCOC4CC34)=O)CSC2)=O)cccc2c1CCC2 22227,CC(C)(CO)C(=O)N1CCC(C)(CNC(C2CCOC2c2ccncc2)=O)C1 22228,N1(C(c2sccc2Br)C(=O)NC2CC2)CCN(c2ccc(-c3ccsc3)cc2)CC1 22229,CC1CN(C(c2ccc(OCC(N)=O)cc2)=O)CC1NC(=O)CCC1CC1(Cl)Cl 22230,C1(NC(C(CCCOCC)C)=O)CN(C(c2cc3ccccc3[nH]2)=O)CC(C)(C)C1 22231,c1(NC(c2c(Cl)ccc(OC)c2F)=O)ccc(S(C)(=O)=O)cc1Cl 22232,n1(CC(=O)NCC2CC2NC(=O)CSc2cccc(Cl)c2)cccnc1=O 22233,C12(C(=O)NCCCc3cc(C)no3)CCCC1CCN2C(c1n[nH]c(=N)[nH]1)=O 22234,c1(C(=O)NCC2OCC(CNC(c3nnn(C)n3)=O)C2)ccc(O)c(Cl)n1 22235,C(=O)(C(C(C)C)C(C)C)N(C)CC1(C)C(NC(CS(CCC)(=O)=O)=O)CCC1 22236,N1(C(c2c(COC)ncs2)=O)CC2CC(NC(c3c(C)nn(C)c3C)=O)C2C1 22237,c1(C(=O)NCCC(C(OCC)OCC)O)ccc2cccnn12 22238,C1(C(=O)NC2(N(C)C(C3CCCC3)=O)CCOCC2)(OC)CCS(=O)(=O)C1 22239,N1(C(CCC(C)O)=O)CC(NC(c2coc(C3CCOCC3)n2)=O)CC2(CC2)C1 22240,N1(C(c2cn(CC)nc2C)=O)CC(NC(=O)Cc2ccns2)C(N=[N+]=[N-])C1 22241,Cc1ncnc(N2CC3CC3(CNC(c3cc(F)ccc3Cl)=O)C2)c1Br 22242,C(c1cnc(C)s1)=CC(=O)NC(CC=C)CNC(c1cnc(C2CCOC2)s1)=O 22243,CC(=Cn1ccnn1)C(=O)NNC(=O)C1CCCCN1Cc1cn(C(C)C)nn1 22244,c1(CCC)ccc(S(=O)(=O)N(CC)Cc2ccsc2)cc1Br 22245,Cc1nn(C)c(C)c1C(c1nnnn1C1CC(F)(F)C1)NC(C1CCOC1)C 22246,C1(NC(CCCSC)=O)CCCC(NC(c2ncncc2OC)=O)CC1 22247,N1(C(C(CCC=C)(F)F)=O)CCC2C(CCCN2C(=O)CC(F)(F)CC)C1 22248,C1(O)(CNC(c2c(CNC(CNC(=O)NC)=O)n[nH]c2)=O)CC2C=CC1C2 22249,CC1OC2(C(=O)NCC3CC4CC4N3C(=O)Cn3cnnc3O)CC1C2 22250,c1(CC2(C(=C)F)N=N2)ccc(F)c(CC(=O)NCC2CC2C(F)F)c1 22251,N1(C(C=C(C)Cl)=O)CC2C(NC(=O)CCSc3ccccn3)C2C1 22252,C=CC(C)(C)CC(=O)NC1COCCN(C(C2(c3ccccn3)CC2)=O)C1 22253,Cc1c(C(N2CC3CC2C3C(=O)Nc2csc(C(F)(F)F)n2)=O)cccc1F 22254,N1(C(CN(CC)CC)=O)CC(NC(=O)CN(S(=O)(=O)CC)C)CC2COCCC12 22255,C=CCC(CC(=O)NCCC(O)C1CCCC1)NC(=O)CCCF 22256,C(=O)(CS(=O)(=O)NC)NCCN(C(=O)CC1CC1)CC.C(C)(=O)N 22257,N1(C(C(c2cn(C)nn2)NC(C2CC(C#C)(O)C2)=O)=O)CCC(O)C(F)(F)C1 22258,c1(C(=O)NCC2CC(NC(c3cccnn3)=O)C2)cnc(S)nc1 22259,C12(CCNC(C3(C(F)F)CC(=C)C3)=O)CCC(C1)N(C(=O)C=Cc1cnc[nH]1)C2 22260,n1(CCC)c(C)cc(C=CC(=O)NCC2CCNC3(CC3)C2)c1C 22261,N1(C(=O)CC=Cc2ccccc2)CCC(CN(C(C2COC(=O)C2)=O)C2CC2)C(O)C1 22262,c1(C(=O)NCCN(C(c2c(C)cc(SC)s2)=O)C2CC2)cccc2c[nH]nc12 22263,N12CC3C(C1)(CS3(=O)=O)NC2=O.C1(C(N)=O)CC2(CCN(c3cc[nH]c(=N)n3)C2)C1 22264,CCCCCCC(F)C(=O)NCC1(NC(C2CCC2(C)C)=O)CCC1 22265,N1(C(C=C(C)C)=O)CCC(OCC(=O)N(C2CCCCC2)C(C)C)C1 22266,c1(-n2cc(CSCCNC(Cn3c(C)ncc3)=O)nn2)ccc2c(c1)OCCO2 22267,C1(C(N2C(C(N)=O)CC2)=O)C=CCN(C(=O)CC2OCCCO2)C1 22268,C(=O)(C(C(C)(C)O)NC(=O)Cc1cccnc1C)NCC(C(=O)OC)O 22269,c1(C(=O)NCC2CCN2C(C2CCCCC2O)=O)nc2ncc(CCO)cn2n1 22270,N#Cc1cc(F)ccc1C(N1CCN(C(C2CCSCC2)=O)C2CC12)=O 22271,Cc1ccc(CC(N2CCCC(O)(CNC(=O)C(C(C)O)N(C)C)C2)=O)cc1C 22272,N1(C(c2c(C)cco2)=O)CCN(C(c2cccc(I)c2)=O)CC1c1nccn1C 22273,C(=O)(CCC(CC)NC(=O)C1CC1)NC1C(C#C)CCC1 22274,n1(CC)cc(CC(=O)NC(CO)C2CCC2)cn1.C1(C2CCOC2)C(=O)N1 22275,CC(C1CCCCC1)=CC(=O)NC1CN(C(=O)COC2CC=CC2)CCC1C 22276,c1(C(=O)NC2C=CC(CNC(C(n3ccc(C)n3)(C)C)=O)C2)cccn(C)c1=O 22277,C(=O)(C(C(=O)NC1CC2(NC(c3cnsn3)=O)COC1C2)C(C)C)OCC 22278,n1(CC(=O)NCC(CNC(C(CC)OC)=O)CO)nc(-c2cccs2)oc1=O 22279,c1(C(N2C(CNC(CC(C)OC)=O)C=CC2)=O)ccc(N2CCCC2)cc1 22280,c1(CC(=O)NCC2CN(C(c3scc(OC)c3)=O)C(C)C2)ccc2n[nH]cc2c1 22281,N1(c2n(CC)nnn2)CC2(CNC(=O)C2)C1.N12CCCN(CC1)C(C)(C)C2=O.c1ccccn1 22282,N1(C(CC(C)OC)=O)CCC(O)(C(C)NC(=O)C(CO)NC(=O)C(C)C)CC1 22283,C1(N(C(C=CC(CC)C)=O)C)CCCN(C(=O)CCCn2cccc2)C1 22284,c1(C(=O)NCCN(C(=O)CC2COC3CC2C3)C2CC2)cc([N+](=O)[O-])ccc1Cl 22285,C(C(C)(C)C(=O)NCCC(C)CCNC(=O)C=C1CCCC1)OCC 22286,CC1(C)CN(C(=O)CCOCC2CC2)CC(CNC(c2cc3scnc3[nH]2)=O)O1 22287,Cc1ncc(Cl)c(C(N2CC3C(CNC(=O)CCS(C)=O)C3C2)=O)n1 22288,N1(CC2(F)CCN(C(C3(CCC=C)CC3)=O)CC2)CC(C)N(C)CC1C 22289,c1(C(N2CC(NCc3ccc(OC)nc3)C2)=O)ccc2c(C)noc2c1 22290,c1(C(=O)OC)cc(S(=O)(=O)N2CCCC2C(=O)O)c(C)o1 22291,C(=O)(C1=NN2CCCN=C2N1)N(C1CN(C(CN(CC)CC)=O)CC1(C)C)C 22292,C1(CNC(C(CC)(C)C)=O)C(O)C(O)CN1C(=O)C=Cc1ccc(F)s1 22293,c1(C(=O)NCC2CN(c3cc(COC)ncn3)C2)cc2cnc(Cl)cc2s1 22294,c1(C(=O)NC2C3CN(C(C4CCC4(F)F)=O)CC23)cccc2cnccc12 22295,C1(C2CC2)(C(N(CC(C)(C)OC)C)=O)CN(C(=O)Cn2ncn(C)c2=O)C1 22296,C1(NC(c2c(CC)cccc2)c2nnnn2C2COC2)CCc2nnc(CC)n2C1 22297,N1(C(CNC(C(C)(C)C)=O)=O)CCC2CCCC12C(N1CCCC(C)(CO)C1)=O 22298,Cc1nsc(C(=O)NC2(CCO)CN(C(=O)CC3(C)CC3)C2)c1N 22299,C1(C(=O)OCc2cccnc2)CCCCN1C(=O)Nc1cccnc1 22300,c1(CC(N2CCC(N(C(CC(CC)SC)=O)C)C2)=O)c(F)cccc1Cl 22301,C1(CC(=O)NCC(C23CCC(CC2)C3)NC(c2ccoc2)=O)CCCNC1=O 22302,CC1CN(C(C2(c3ccccc3Br)CCC2)=O)CCN1C(C1C=CCCC1)=O 22303,C1(C)(C(=O)NC(CNC(c2n(CC)nnc2)=O)(C)C(C)C)CCCCNC1=O 22304,C(CNC(C1(c2ncco2)CC1)=O)(CC(=O)N1CCOC(CC(N)=O)C1)OC 22305,N1(C(C(CC)OC)=O)CCOC(C(=O)NCC2(F)CC(CO)C2)CC1 22306,CCC(C(=O)OC)C(=O)NC1CC=C(C(=O)NCCc2nc(C)no2)C1 22307,c1(N(C(=O)CN)CCCl)ncnc2[nH]cc(Cl)c12 22308,Cc1ccc2c(C(=O)NCC(C3CC3)N(C(=O)CSc3nc[nH]n3)C)n[nH]c2c1 22309,C1(COC)(CNC(=O)CC#N)CCN(C(=O)Cc2ncccc2C)C1 22310,c1(C(=O)NCCC2(O)CN(C(C34CCCC3CC4)=O)C2)cnc2n1CCOC2 22311,S(=O)(=O)(c1ccc(-c2ccc(Br)c(C(=O)O)c2)s1)N(CCC)CCO 22312,N1(C(CCC=C)=O)CCCC(NC(=O)CCc2ccc(C(C)C)cc2)C1 22313,C(=O)(C1=CNC2=NCCCC2=C1)N1CC(CN(C(C(C(=O)OCC)(C)C)=O)C)C1 22314,c1(OCOC)cccc(NCCNC(=O)C(C(C)C)n2cnnc2)c1 22315,Cn1cc(C(N2CCC(NC(=O)CCc3cc(Cl)no3)C2)=O)nc1-c1cccs1 22316,N1(C(c2c(C)cc(C)s2)=O)CCCC1C1CCCN1C(=O)CCN(S(C)(=O)=O)C 22317,c1(C(=O)NCC2C(C)CN(C(c3c[nH]c(=N)o3)=O)CC2)ccc2nnc(S)n2c1 22318,C(=O)(C1=C(Cl)CCC(C)C1)NCC1(NC(C2CCCC(C(=O)OC)C2)=O)CCC1 22319,C1(NC(=O)CC2CC(CF)C2)CCCC(C(=O)NCC=Cc2cccc(F)c2)CC1 22320,c1(CC)nc(=NCC(C)(C(C)C)NC(C2CCCCN(C)C2=O)=O)s[nH]1 22321,CC(C(=O)N1CCC(C(O)CNC(C2NC(=O)OC2C)=O)CC1)S(N)(=O)=O 22322,N1(C(c2ccc(C(=O)OC)[nH]2)=O)CC2(CCC2NC(C2CCCOC2C)=O)C1 22323,Cc1ccc(C2(C(=O)N(CCCCNC(C3CC3C#N)=O)C)CCOCC2)cc1 22324,C(=O)(C(CC(F)F)NC(C1CN(C(=O)NC)C1)=O)N1CCCC(OCC)C1 22325,CC1=C(C(=O)NC2COCC2NC(C2NC(=O)OC2C)=O)C(=O)OC1(C)C 22326,CC1CC(NC(=O)C(C)(C)N2CCOCC2)CCN1C(C1C(F)(F)C12CC2)=O 22327,C1(NC(C(C)OCC)=O)CN(C(=O)C=CC2CCOC2)CC12CC2 22328,c1(CC)c(C(=O)NC2CCCCC2N(C(=O)Cc2c[nH]nc2O)C)cccc1C 22329,c1(C(=O)NC2CC3CC(NC(CCCOC)=O)CC3C2)ccc2c(c1)ncn2C 22330,C1(NC(C2N(CC)CCC2)=O)CN(C(c2cccc(=O)n2C)=O)C(C)(C)C1 22331,CCCN=C(NCC1CC1)NCC.S(C)(=O)(=O)NC(N(C)C)=O 22332,N1(CC)CCC(NC(C2CCOCC2NC(C2CC2Cl)=O)=O)C1=O 22333,C12(NC(CC3(OC)CC3)=O)CCCC(NC(=O)CCc3nccn3C)(C1)C2 22334,C(=O)(C(CC)C(C)(C)CC)NCC1(O)CCCN(C(C2(CC=C)CCC2)=O)CC1 22335,C(=O)(C#CC(C)(C)C)NCC(C)(CO)NC(CC(C)c1ccncc1)=O 22336,N1(C(CSC)=O)CCC2(NC(=O)CC3CCCC3C)CCCC12 22337,N1(C(C23CCC(C)(CC2)OC3)=O)CCC(C2(O)CN(C(c3ccsc3)=O)C2)CC1 22338,c1(C(N(CC(C)(C)NC(c2sccc2C#N)=O)C)=O)cc(F)ccc1C(F)(F)F 22339,C1(NC(=O)C(F)CC2CCCC2)CCC2(CCCN2C(c2ccc(Cl)o2)=O)CC1 22340,c1(CNC(c2ccc3nc(C4CCCO4)oc3c2)=O)nc2ccc(Br)cc2n1C 22341,C1(F)(C(NOC(C(=O)NC(c2ncc(C(C)O)s2)C2CC2)C)=O)CCCCC1 22342,c12cn(C)nc1NC2.c1(SC)sccc1C(=O)N(CCCN(C)C)C(C)C 22343,c1(-c2c(C(N(CCNC(=O)COCCF)CC)=O)c[nH]n2)cccc(OC)c1 22344,n1(C(C)C)ccc(C(N2CCC2CNC(c2nc(Cl)cs2)=O)=O)n1 22345,N1(C(CC=C=C)=O)CC(CCNC(c2ccnc(Cn3cnnc3)c2)=O)OC(C)C1 22346,C1(C(=O)NCC2C(C)CN(C(=O)CC3CC(C)(C)C3)C2)C2CCCCCCC12 22347,N1(C(c2ncc[nH]2)=O)CC(C2CCCN(C(C3CC(c4ccccc4)=NO3)=O)C2)C1 22348,Cc1[nH]ccc1C(=O)NCc1cn(CC(N2CCC2CN(C)C)=O)nn1 22349,c1(C(=O)NC(CNC(C(C(C)C)OCC)=O)(C)CC)cc(Cl)c(C)cc1OC 22350,C1(OC)CCN(C(c2ccoc2CNC(=O)C(C)OC2CC2)=O)C(C)C1 22351,c1(C2(C(N(CC(C)(C)CN)C(c3cn[nH]c3)=O)=O)CC2)ncccc1C.CC 22352,Cc1cc(C)[nH]c(=NCC2(N(C)C(c3cccn4c(O)nnc34)=O)CC2)n1 22353,C1(CC(=O)NC(C(C)(C)NC(c2cncc(COC)c2)=O)C)NC(=O)CNC1=O 22354,CC(CC(=O)NC(C)C(C)(C)NC(=O)Cn1cnnc1)n1cccn1 22355,CCCCC(O)CC(=O)N(C1(C)CC(OC)C1OC)C.c12cn(nn1)C2C 22356,n1(CC)cc(Cl)cc1C(=O)NC1(CNC(C23COCC(C2)C3)=O)CCCC1 22357,c1(C(=O)NC2C3CN(C(=O)NC4CCOC4)CC23)cc(Br)cc2cc[nH]c12 22358,c1(C(=O)NC(CC)CNC(=O)C(C)OC(C)(C)C)cc(Cl)cs1 22359,CCS(=O)c1ccccc1C(N1CCN(C(c2cc(C)cs2)=O)CC1)=O 22360,C(C)(C(CC(=O)NOC(C)C)OC)OCCCC(=O)NCC.C1C(=O)N(C)C1=O 22361,N1(C(c2cncc(NCC)c2)=O)CCC(C)C(NC(=O)CN2C(=O)CNC2=O)C1 22362,Cc1ccc2c(c1)C(C(=O)N(CCCN1CCCCC1)C)OCC2 22363,N1(C(CC2N(C(C(CC3CCC3)OC)=O)CCC2)=O)CC(CO)C2(CCC2)C1 22364,c1(OC)ccc(NC(C(C2CC2)N(CCCC(C)C)C2CC2)CCC#N)cc1CO 22365,N1(C(C(CC)(C)C)=O)CCC(NC(=O)Cc2cc(Cl)ccc2O)C(C)C1 22366,c1(C(=O)NCCCNC(c2c(C)nn(C3CC3)c2)=O)cnn2c(N)ccnc12 22367,C(=O)(C(=O)C(C)(C)C)NCCC1(OC)CN(C(c2cccc(=S)n2O)=O)C1 22368,N1(C(C23CC(CO)(CO2)C3)=O)CCCC(CCC(=O)NCC(N2CCOCC2)C)C1 22369,c1(CC(C(N2CC(CCNC(=O)C(C)CO)(OC)C2)=O)C)ccc(C#N)cc1 22370,C(C(CC(C)C)C(=O)NC(C)(CNC(c1cnc(Cl)n1C)=O)CO)OC 22371,Cc1cc(NCC(C2CC2)NC(C2CCCC(C)(C)C2)=O)c(Br)cc1[N+](=O)[O-] 22372,c1(C(=O)NC2CCC(NC(=O)C3=CCSC3)C2)c(Cl)ccc(Br)c1F 22373,C12(NC(CN(C)C)=O)CCCCCC1N(C(c1coc(Br)n1)=O)CC2 22374,Cc1cnn(C)c1CC(N1CC(CCNC(=O)CCC=CBr)C1)=O 22375,C1(C(=O)NC2CC2COC)CCCN(C(=O)CCCN(CCO)CCO)C1 22376,CC1(C)CCc2n[nH]cc2N(C(=O)NC2(C)CC(=O)NC2=O)C1 22377,c1(OC)cc(CCCNCC(C)(C)C2(O)CNC2)cc(F)c1 22378,c1(NC(C(N2CCn3c(C)nc(Br)c3C2)CCCC=C)=O)cccc2c1OCCO2 22379,CC(C)(O)C#CC(=O)N1CSCC1C(N1CC2(CCC1CO)CC2)=O 22380,Cc1cc2nc(NCC3(O)CCCN(C(C4(C)CC(C)(C)C4)=O)C3)cc(=O)n2o1 22381,N1(C(=O)C=CCF)CCC(NC(C2(Cn3cncn3)CC(F)(F)C2)=O)CC1 22382,C1(NC(Cc2ccn(C)n2)=O)CCCCC1NC(c1cc(C(C)(C)C)n[nH]1)=O 22383,N1(C(C2=CCN(C(C(CC)(C)OC)=O)CC2)=O)CCC2(CCC(O)C2)C1 22384,C1(NC(C(c2ccc(F)cc2)C)=O)C2CC(CN(C(C3(C)CC3)=O)C2)C1CO 22385,N1(C(c2ccc(OC)nc2)=O)CCCC(NC(c2cnnc(C3CC3)c2)=O)C1C 22386,C(=O)(C(C)CC(F)F)NC1C(C(=O)Nc2c(C)[nH]c(=N)s2)CCC1 22387,C(=O)(C(C)CC(C)(F)F)NC(CCN(C(Cc1ccc(OC)cc1)=O)C)C 22388,C(CCCC(C)C)NC(CCC1N(C(c2c(C)scn2)=O)CCC1)=O 22389,C1(c2cn(CO)nn2)(COC2CCN(C(CC3N(C)CCC3)=O)C2)CCCCC1 22390,c1(CC(C)NC(=O)Nc2cncnc2Cl)nc2ccccc2s1 22391,N1(C(c2c(C)cc(SC)o2)=O)CC(NC(=O)Cc2coc(C)n2)CC1(C)C 22392,C1(C(N)=O)(CNC(=O)CC(O)C2CCCC2)CN(C(C2CC2C(N)=O)=O)C1 22393,c1(CC(C)C(=O)NCC2CCN(C(=O)COCCO)CC2)ccc(O)c(O)c1 22394,c1(C(=O)NCCN(C(=O)C(=O)NCCC(N)=O)CC)cccc(COC)c1F 22395,N=c1ncn(CC(=O)N(CCC(=O)NCCCCF)CCCO)[nH]1 22396,C1(NC(C2(N(C)C)CCCC2)=O)CN(C(=O)CC2CCC23CCC3)CC1C(F)F 22397,c1(N2C(C)COCC2C)ncnc2c1ncn2CC1CCC2(COC2)OC1 22398,CCC(CC)(CC)C(=O)N1CC(C)(c2cn(-c3ccc(C(C)(C)C)cc3)nn2)C1 22399,CCC(CC)CC(=O)NCC12CC1CN(C(=O)CC1(C)CC1(F)F)C2 22400,C12(C(N3CCC(C)(NC(C=C(CC)C)=O)C3)=O)CCOC1CC(=O)NC2 22401,C(=O)(C(COC)OC)NC(C1C(C(=O)NC2(CC#C)CCC2)C1)C 22402,c1(N(C)CC2C(C)C2)nc(=NC2CC(N3CCCC3)C2)[nH]c2cc[nH]c12 22403,c1(CCOC2(OCC)CN(C)C2)ncnc2c(Br)nn(C)c12 22404,N1(C(CN(C(C)=O)C)=O)CCOCC(NC(c2cc(Br)n(C)c2)=O)C1 22405,c1(C(N2CCCC(C(=O)NCCc3cccnc3)C2)=O)ccc([N+](=O)[O-])o1 22406,C1(NC(C(c2cnn(C)c2)C)=O)CCCCN(C(=O)C(C)(C)C2CCCCO2)C1 22407,C12CCCN(C1)C(=O)N2.n1(C2(C(=O)OC)CC2)cc(CC(C)O)nn1 22408,c1(C(=O)NC2CC(O)(CN(C)C(c3nnc(C(C)(C)C)s3)=O)C2)ccc(=O)n(C)c1 22409,c1(SC)cccc(F)c1C(=O)NCC(C)NC(=O)CCC1CCCN1C 22410,C1(NC(C(=CC2CCCC2)C)=O)CN(c2nnc(C(F)F)o2)CCC12CCC2 22411,N1(C(Cc2c(C)n[nH]c2)=O)CC(CNC(=O)CCC2CCCO2)C(C)(C)C1 22412,C(=O)(CC(C)(C)C(=O)N1CC2C(CNN3C(C(=O)C(N)=O)CC(O)C3)C2C1)OC 22413,O(NC(=O)C(F)C(C)CNC(C1(C(C2CC2)N(C)C)CC1)=O)C(C)C 22414,c1(NCC)ncc(C(=O)NC23CC(CNC(=O)C#CC(C)C)(C2)C3)cc1Cl 22415,c1(CC(=O)NCC23CC(NC(C(COC)N(C)C)=O)(C2)C3)c(O)ncnc1O 22416,c1(C(=O)NC2CN(C(CNC(=O)OCC)=O)CC(F)C2)csc2ccc(F)cc12 22417,CCCC(C)CC(=O)NC(C)C(C)NC(c1onc(OC)c1Br)=O 22418,c1(OCC)cccnc1C(=O)N(CCC(C)NC(=O)C=Cc1ccc[nH]1)C 22419,C1(C)(CNC(C(CC)O)=O)COCCN(C(c2cc(F)c(O)c(Cl)c2)=O)C1 22420,C(C(=O)N1CCCC1CC(=O)OC)(C(C)C)C(=O)NC 22421,N1(C(CC2(C)CCC2)=O)CC2(CNC(c3cnn(C)c3Cl)=O)CC1CO2 22422,C=C(C)C(C)(C)C(=O)NC1CCCCC1C(=O)Nc1cc(C)nc(C(F)(F)F)n1 22423,c1(C(=O)NCC2CC(C)(C)N(C(=O)C(O)C3CCC3)C2)c[nH]c(=N)c2[nH]ccc12 22424,c1(C(N2CCN(C(COC)=O)CC2)=O)cc2ccccn2c1.C12CC(C1)C(=O)N2 22425,CC(C)CC(O)C(=O)NC1(CO)CN(C(C2CCCCN2C)=O)C1 22426,CC(CC(C)(C)C)C(F)C(=O)NCC1C2CN(C(=O)CCn3cnc(=N)[nH]3)CC12 22427,N=c1[nH]c2ccc(C(N3CC(CNC(=O)CC4CCCCC4F)C3)=O)cc2[nH]1 22428,C=C(Cl)C(C)(C)C(=O)N1CCCC1CCC1CCCCN1C(=O)CC=CC(C)(C)C 22429,CCCCCC(O)C(=O)N1CC=CC1CNC(=O)CNC(C1CCC1)=O 22430,c1(C(C)OC(C2CC(CCC)C2)=O)ccc(Cl)nc1 22431,C(=O)(C1=CCCOC1)NCCC1CCC(NC(CC(CC)c2ccccc2)=O)C1 22432,c1(SC)cncc(NC(C2CN(C(C3CC3(F)Cl)=O)CC2F)=O)c1 22433,C1(C(=O)NCc2n(CC)nnc2C)N(C(=O)C(C)n2cccn2)CCCC1(C)C 22434,c1(NC(N)=O)ccc2nc(Cl)nn2c1.c12cn(nn1)CCOCCCC2 22435,c1(C(=O)NC2(CCNC(C(CC)C(C)C)=O)CC2)ncnc2c1CCC2 22436,c1(C(N(CC(CNC(c2c(C)oc(C(F)(F)F)c2)=O)C)C)=O)ccc([N+](=O)[O-])[nH]1 22437,N1(C(C(CC2CN(C(C(CCC)C(C)C)=O)C2)F)=O)CC2CCCC(O)C2C1 22438,N1(C(Cc2cc(C)on2)=O)CCC(C2CC2)(CNC(c2ccn(C(F)F)n2)=O)C1 22439,C1(C(=O)NCC(CC)C)CC(C)CN(C(C2CCC(O)CN2C)=O)C1 22440,N1(C(CN(C(=O)COCC2CCCO2)CC#C)=O)CC2COC(=O)C2C1 22441,N1(C(CCC2CCN(C(C(C)OCC3CC3)=O)CC2)=O)CCCSCC1C 22442,c1(C(=O)NCC#CCNC(=O)COCC2CCCC2)cccc(C(N)=O)c1F 22443,c1(OCC)nc(N2CC(CNC(c3ccccc3SCC)=O)CC2C)ncc1C 22444,C1(C)(C(=O)NCC(=C2CN(C(C(n3ncc(C)c3)C)=O)C2)F)CCCNS1(=O)=O 22445,N1(C(CC(C)(C)C)=O)CCC2CN(C(c3cc(F)cc(F)c3O)=O)CCC2C1 22446,C1(NC(=O)Nc2cnc(I)s2)CCN(Cc2ccc(OC(F)(F)F)cc2)CC1O 22447,C(C(O)(C(F)(F)F)c1ccccc1)NC(CCC(=O)NCCC)=O 22448,N1(C(c2c(CCC)n[nH]c2)=O)CC=CC(NC(c2cnco2)=O)C1 22449,Cc1cc(C)n(CC(=O)N(C2CC3CNC2C3)c2sccc2C)n1 22450,C(=O)(CS(=O)(=O)CC1CCCO1)NCC(C(C)(C)C)NC(=O)C=C1CCCC1 22451,c1(NC(C=CCNC(C2(C=C)CCOCC2)=O)(C)C)cncc2sccc12 22452,C(CCC)(C(=O)NCC(C)CNC(C1(C(F)(F)F)CCCC1)=O)=CCC 22453,c1(-n2cc(NCC3CCCN(C(C(COCC)O)=O)C3)nn2)ccc(C)c(Cl)c1 22454,Cc1cc(C)n(CCCNC(c2cccc(CN3CCOC(O)C3)c2)=O)n1 22455,C12CN(CCC1O)C2=O.c1(NC(=O)NC(C(=O)OCC)C)ccc(CC)s1 22456,N1(C(CCc2ccc(OC)c(C)c2)=O)CC(C)N(C(C2(C)COC2)=O)CC1C 22457,O=C(N=c1ccn(C2CC2)[nH]1)C1CN(C(c2cc(Cl)c(Cl)nc2Cl)=O)CCO1 22458,N1(C(C2C(=C)CC2)=O)CCC(C)(CCNC(=O)CCc2ccc[nH]2)C1 22459,N1(C(=O)NC23OC(C)C(CC2)C3)CC(S(C)(=O)=O)CC1F 22460,CC1(C(=O)NC2CCOC(CNC(=O)CCc3cccnc3Cl)C2)COCCO1 22461,N1(C(CSCC)=O)CC2CCCC2(CNC(=O)C2=NOC(c3ccccc3)C2)C1 22462,c1(NC(=O)NC(c2ccccn2)Cc2cccc(C)c2)cc(F)c(I)c(F)c1 22463,N1(C(c2c(C)nsc2)=O)CC(NC(c2ncc(Cl)c(N)c2Cl)=O)CC2(CCC2)C1 22464,C(CN=c1[nH]c2ccc(O)cc2s1)=CCNC(C(C1CCCOC1)OC)=O 22465,C1(C(=O)NC(CC)C(N)=O)CCN(C(C2CC(=O)NC2(C)C)=O)C12CCC2 22466,C1(N(C)C(C2C=CCS2)=O)CN(C(c2cc(Cl)c[nH]2)=O)CCC1O 22467,C1(N(C(CC(C)(C)C)CNC(C2CC2C(=O)NC2CCCC2F)=O)C)CCCCC1 22468,CC(C)CCCC(C)CCNC(=O)N(C(C)(C)C)C(c1ccc(Cl)cc1)C 22469,c1(C(=O)NCCC2(O)CCN(C(=O)CSC(F)F)C2)cnn2ncccc12 22470,C(=O)(C(C)(O)COc1ccccc1)NC(CNC(c1ccc(CC)s1)=O)CC 22471,c1(NC(CN(C(C(=O)OC)C2CC2Cl)C)=O)cc2c(cc1OC)CCC2 22472,C1(CC)CCC(C(=O)OC2COCCCC2c2ccccc2)CN1CC(=O)OC 22473,Cc1cc(OCCC(=O)N2CCC2Cc2cn(C3CCN(C)C3)nn2)c(C)c(C)c1 22474,N1(C(C2(C)CCCOC2)=O)CCOC2(CCN(C(C3CCC4CC4C3)=O)C2)C1 22475,C1(C(=O)NCC=C2CCSCC2)(NC(C(c2cncnc2)C)=O)CC(O)C1 22476,c1(-c2cn(C(C(=O)Nc3nnc(C)s3)C)nn2)c(C)[nH]c2ccccc12 22477,c1(C(=O)NCC(CNC(=O)CCC2CCCN2C)OC)cccc2c1CCO2 22478,C1(CNC(C2(CC)CN(C(=O)CN3CCCC3)C2)=O)CCC(=O)N1C 22479,C1(COC)(NC(=O)C(C)SC(C)C)CCN(C(c2cc[nH]c(=N)c2)=O)CC1 22480,C1(NC(c2nccc(CC)c2)=O)CC2CC1N(C(c1ccc(F)c(N)c1)=O)C2 22481,c1(C(=O)NC(c2nccn2C)C)ccc(=O)n(CCN(C)C)c1 22482,C=CCC(CNC(c1nnsc1C)=O)C(=O)N(C)CC1CCN(C)C1 22483,C(=O)(C1=CC2(CCOCC2)C1)NCCC(C)CCCNC(=O)C(CO)C(C)(C)C 22484,C(C(C)(C(=O)N(C(C)CCNC(c1n[nH]c(C)n1)=O)C)OC)OC 22485,N1(C(C(C2CCC2)NC(c2c(OC)ccnc2)=O)=O)CCC(C)C(F)(F)C1 22486,N1(S(=O)(=O)c2cnccc2N2C3CCCC2CC3)Cc2ccccc2CC1CO 22487,N1(C(c2c(OC)cc(N)cc2)=O)C2CCC1CN(C(=O)CC1CCCN(C)C1)C2 22488,C1(C)(CNC(C2(NC(C)C)CC2)=O)CCC(NC(=O)C(C)(C)F)C1 22489,CN1CCCC1(C)C(=O)NCc1ccc(C(=O)NC2COCC2O)cc1 22490,N1(C(COC(CC)(C)C)=O)CC(C)CN(C(c2cccc(C(C)C)c2)=O)CC1C 22491,Cc1ccc(C(N2CCCC2CNC(=O)CC2CCCC2C)=O)c(C(C)C)n1 22492,Cc1cc(C(N2CCCCC2C(=O)OC(C)(C)C)=O)cc(CNC(=O)C(C)C)c1 22493,Cc1oc([N+](=O)[O-])cc1C(=O)NCCC(C)(C)NC(=O)C(=Cc1cscn1)F 22494,C(=O)(C1=C(C)S(=O)(=O)CC1)NC1CN(C(C=CCCC)=O)C(C)(CC)C1 22495,C1(C)(C(N2CCC(CNC(c3c(OC)c(F)ncc3)=O)C2)=O)CCCCCCC1 22496,c12ccc(O)c(c1)C(=O)C1CN(C1)C(=O)n1cc-2nn1.C1(C(C)=O)C(C2CC2)C1(C)C 22497,N1(C(Cn2nc(C)c(Br)c2)=O)CCOC2CN(C(=O)Cn3cnnc3)CC12 22498,C1(C(=O)OC)CN(C(c2nc(CNCC34CCCN3CCC4)cs2)=O)CCC1O 22499,c1(C(N(C(CCNC(C(C)OCC)=O)C)C)=O)cc(C)c(Br)cc1C 22500,N1(C(c2nccc(C)c2)=O)CCN(Cc2ncccc2C(F)(F)F)CC1C#N 22501,C#CCC(C(=O)NCC1(NC(=O)C(=CC2CCCCC2)F)CCOC1)C1CC1 22502,C1(NC(C(=O)NC(C)C)=O)CCC2(CC1)CCN(C(C1OCCO1)=O)C2 22503,CCC(CC)(CC)C(=O)N(C)CC1CCC(NC(=O)CS(=O)(=O)CC)CC1 22504,C1(S(C)(=O)=O)(C(=O)NC2CC(NC(c3nc(N(C)C)nc(O)c3)=O)C2)CC(O)C1 22505,C#CC1CCN(C(=O)C(Cc2cn[nH]c2)NC(=O)CCCN(C)C(C)=O)C1 22506,Cc1cn2c(C)c(C(N3CCCC3CN(C)C(c3[nH]ncc3C#N)=O)=O)nc2s1 22507,C1(C(=O)NCCNC=O)CCC(O)CN1C(=O)Cc1cccc(O)c1.C1CC1 22508,Cc1nc(N2CCCC(NC(c3cscc3C(F)F)=O)C2)c2cnn(C)c2n1 22509,c1(N(C(=O)C=CCC2(C(N(C(C=C)C)C)=O)CCC2)CC)ccccc1 22510,CC1COC(CC(N2CCC(N(C(=O)CCc3cscn3)CCO)C2)=O)CO1 22511,C1(NC(c2nn(C)c(CNC(N)=O)c2)=O)CC1C1CCCN(C(=O)OC(C)(C)C)C1 22512,N1(C(CS(CCC)(=O)=O)=O)CCc2nc[nH]c2C12CCN(c1cc(Cl)ncn1)C2 22513,C1(COCC(=O)NCC2CC2C(=O)NCC2(Br)CC2)CCCO1 22514,Cc1nc(CCNC(=O)CCC2(N)CCOC2)c(C)o1 22515,C1(O)(C(C(=O)NC(C#C)CC2CC2)NC(=O)C(C)(C)OC)CCCCC1 22516,C1(NC(c2cc(Cl)nnc2O)=O)CN(C(=O)CSCC(F)(F)F)CC1C1CC1 22517,CC(C)(CC(=O)NCC1CCCCN(C(C2CCC(N=[N+]=[N-])C2)=O)C1)CC(F)F 22518,C1(F)(NC(C=CCOC)=O)CCN(C(C2(C3CCCO3)CCC2)=O)C1 22519,N1(C(C2(CC)CC2)=O)CCC(F)(F)C(CNC(C2(N(C)C)CC2)=O)C1 22520,CC1=CC(C)CN(c2nnc(-c3cc(C)c(O)nn3)n2CCC(=O)N(C)C)C1 22521,c1(C(N2CC(NC(Cc3c(OC)ccnc3)=O)C(C)C2)=O)cncc2nc[nH]c12 22522,C(c1ccc(C#N)cc1)=CC(=O)NCC(CC)NC(c1c(C)cc(Cl)cc1C)=O 22523,C12CCCCN(C1)C2.C1(NC(C=C(CCN(C)C)Cl)=O)CC2(CSC2)C1 22524,c1(C(=O)OC(C(F)F)C2CCCC2)cc(N2CCOC2=O)ccc1F 22525,CCC(C)(C)CCCC(=O)NCCCN1CCC(NC(c2nccc(N)c2Cl)=O)C1 22526,c1(C(N2CC(N(C)Cc3cc(OC)ns3)C2)=O)cc(F)c2ncccc2c1 22527,C1(C(C)C)C(NC(=O)CNC(N)=O)CCN1C(C1CC(F)(F)CS1)=O 22528,C1(CCN(C(=O)Cn2ncccc2=O)C)CCN(C(C2(SC)CC(O)C2)=O)CC1 22529,C(C(C)C(C)(C)C)NC(C1CCCN(C(c2ccccc2)C)C1)C 22530,C1(CC(N2CCC(C(=O)N(C)C)(OC)C2)=O)CCCOC12CCC2.CC(C)CCSC 22531,c1(C(N(C(CNC(C2CC(=O)N(O)C2)=O)C2CC2)C)=O)coc2c(F)cccc12 22532,C1(OC(C2(CCC)CCCN2Cc2ccc(C)c(C)n2)=O)CC(S(C)(=O)=O)C1 22533,CCC(CO)CCNC(=O)C(Cc1cc[nH]n1)NC(=O)Cn1nccn1 22534,C=CCC(CC)C(=O)N1CCCC(C)(Cc2nccc(OCC)n2)C1 22535,c1(C(N(CC(C)O)CCNC(C(C2CC2)OCC)=O)=O)nocc1Cl 22536,c1(NC(N)=O)ccc(CC(N2CC(NC(C3CC4(C3)CC4F)=O)C(CO)C2)=O)cc1 22537,c1(CC)c(C(N2CC(c3cn(CC4CCCO4)nn3)C2)=O)cnn1C 22538,c1(OC)ccc(NC(=O)NCC(C(F)(F)F)N2CCCC2)c(C)c1OC 22539,c1(C(N2C3C(NC(C(c4ccccc4)OC)=O)C(C3)C2)=O)ccc(=O)n(O)c1 22540,c1(C(=O)NCC#CCNC(C2C(C)CC(=O)NC2)=O)ccccc1S(C)(=O)=O 22541,C1(O)(C(C)NC(C2(CO)CCCCC2)=O)CCN(C(c2nccnc2N)=O)CC1 22542,c1(C(=O)NCC2(COC)CN(C(=O)CC3CCOC3(C)C)C2)ccnc(S)c1 22543,CC1=C(C(=O)NCc2ncccc2C(N2CC(C3CCCOC3)C2)=O)CCO1 22544,Cc1cccc(C(N2CC(CC(=O)N(CC(C)C(F)(F)F)C)C(C)C2)=O)c1O 22545,c1(C(=O)NCCC(C)(C)NC(=O)CNC=O)ccnc(F)c1O 22546,N1(C(C(OC)OC)=O)CCC2(CCCCC2NC(C2CCC3(CC2)CC3)=O)CC1 22547,C(CN=C(NC1CCCC1)N1CC(CN2CCOC2=O)C2(CCC2)C1)SC 22548,N(C(=S)N1CC(S(=O)(=O)C(C)(C)C)C1)c1cccc(C(C)C)c1 22549,C(C)(C(C(=O)NC1(CSC)CC1)C(C)C)NC(CC=CC)=O 22550,c1(C(N2CC(NC(c3[nH]n(C)c(=O)n3)=O)C(O)C2)=O)occ2c1CCOC2 22551,C(CNC(c1c(CC)occ1)=O)(CC(C)C)NCc1cc(C(=O)OC)sc1 22552,c1(N(CCC(=O)NC)C)nc(=NCC(CO)C2CCC2)[nH]c2cccnc12 22553,c1(NC(COCC)=O)cccc(CSC2CC2NC(c2nnc(CC)s2)=O)c1 22554,N1(C(CC(=C)Br)=O)CCC(NC(=O)CSCCCC)C(F)C1 22555,c1(CCC2C(C(=C)C)OCC2)cc(=NCC(C)(C)C(N)=O)[nH]c(CSC)n1 22556,N1(C(=O)Nc2c(C)cn(-c3ccc(Br)cc3)n2)CC2CC1CN2S(C)(=O)=O 22557,C1(NC(=O)NCC(N(C(=O)CCC2(C)N=N2)C)C2CC2)CCCC1C(F)(F)F 22558,C(=O)(C1=CCCOCC1)N1CCC(N(C(C2C3CC4C(C3)C24)=O)CC2CC2)CC1 22559,C=CCC(CC)C(=O)NC1CN(C(c2cn(C(C)C)nn2)=O)CC1(C)C 22560,C1(C2CCN(C(c3ccc(C#N)nc3O)=O)CC2)(NC(C(OC)OC)=O)CCC1 22561,c1(C(=O)NC2CC(C)(NC(COC(C)(C)C)=O)C2)cc(F)c2c(c1)CCC2 22562,C(C(=O)NCC1CC(O)CN1C(=O)C=Cc1cnccn1)(C(C)C)OC 22563,c1(CC(N2C(CN(C(CCC(N)=O)=O)C3CC3)CCC2)=O)ccc(F)c(F)c1F 22564,C(CO)(CCCNC(=O)C(c1cnn(C)c1)=O)NC(C(C1CCOCC1)C)=O 22565,c1(C(=O)NC(CCNC(c2n(CC)nnc2)=O)C)cc2c(s1)CCOC2 22566,N1(C(c2ccc(C#C)cn2)=O)CCC2(CC(NC(=O)C3=NOC(C)C3)CO2)C1 22567,c1(C(N(CCCOC(N)=O)C(C)C)=O)nc2cc(F)ccc2s1.CCC1C(=O)N1 22568,c1(C(N2CCC(C(F)(F)CO)CC2)C(=O)NC)ccc(Br)cc1OC 22569,N1(C(C(CCC)F)=O)CC2CCC(C(N3CCc4c[nH]nc4C3)=O)(C2)C1 22570,c1(CC)ccc(C(N2CC(OC)CC2C(N2C3CSCC2C3)=O)=O)cc1 22571,C1(C(=O)NC(C2CCN(C(C3CCOCC3)=O)C2)C)CCCC(CF)C1 22572,C1CCCCCCC(=O)N1.C1(CC=C)(N)CCN(C(c2cn(CC)nn2)=O)C1.CO 22573,C1(CC)(CNC(=O)C(C)O)COCCN1C(=O)CCCN1CCOCC1 22574,C1(OC)CCC2(C(N3CCN(C(C4(COC)CCCCC4)=O)CC3C)=O)CCC12 22575,N1(C(c2ccc(P(C)(C)=O)[nH]2)=O)CCOC2CN(C(=O)CC(F)(F)C(F)F)CC12 22576,N1(C(C(CCC)(C)C)=O)CCC2(CCCN2C(=O)Cc2n[nH]cc2Br)C1 22577,Cc1cnsc1C(=O)NC1(C(=O)NOCC2CC(=C)C2)CCC1 22578,C1(C(=O)NCCNC(=O)NC)CCN(C(c2cc(C)c[nH]2)=O)C1C 22579,N1(C(COC(C)(C)C)=O)CC(O)CC1C(=O)NCCN=[N+]=[N-] 22580,c1(OC)ccc(C(C(F)(F)F)NC(c2coc(C(C)OC)n2)=O)cc1 22581,c1(C(=O)NC2C(NC(=O)CO)CS(=O)(=O)C2)cc2c(c([N+](=O)[O-])c1)OCO2 22582,C1(NC(C(C=C)(C)C)=O)CCC2(CC1)CN(C(C1(CCS(N)(=O)=O)CCC1)=O)C2 22583,c1(C(N2CC(CC=C)(NC(c3nc(C)nn3C)=O)C2)=O)nc(C2CC2)oc1C 22584,N1(CC)CCC(C(N2CC(CCCCNC(=O)CC3CC3(Cl)Cl)C2)=O)C1 22585,C1(CN(C(c2n(CC#C)ccc2)=O)C)CCCCN1C(c1cnsc1)=O 22586,c1(C(=O)NCCN(CCC)C(C2CCC(=O)C(C)C2)=O)cnc(C2CC2)nc1O 22587,C1(CNC(c2c(C(C)C)con2)=O)C(C)CCN1C(=O)C#CC1CC1 22588,C1(C(=O)NC(C#C)CC(C)C)CCN(C(=O)CC2(O)CCCCC2)C12CC2 22589,CC(CS(=O)(=O)N=c1ccn(C2CCOC2)[nH]1)C1CC1 22590,C1(C(C)C)CN(C(C2CCC3(CC3)C2)=O)CCN1C(=O)CN1CCOCC1 22591,C(=O)(CCC(CF)CF)NC(C(C(=O)NC(C)CC1CC1)(C)C)C 22592,Cc1cc(=NC(=O)CSC2NC(=O)N(CC(=O)N(C)C)C2=O)[nH]o1 22593,c1(C(N2CC3C(NC(C(CCC)O)=O)(C3)C2)=O)cc(OC)ccc1C 22594,C12(CC(N3CCC(NC(C4C(OC)CCC4)=O)C3(C)C)=O)CCCCC1C2(F)F 22595,c1(C(=O)NC2CC3CN(C(CCOCC)=O)C2C3)c(F)cc(C)cc1Br 22596,Cc1nnc2cnc(C(=O)NC(C)CCCNC(=O)C(C)(O)CC(C)C)cn12 22597,Cc1oc(C)c(C(=O)NC2CC(F)(CNC(=O)Cc3ccc(O)c(F)c3)C2)c1C 22598,C1(C(N(CCC(=O)NCC(F)CO)C)=O)COCC1C(N)=O 22599,c1(C(=O)NCC2(C(N3C(C(=O)NC)CCC3)=O)CCCC2)cncc2[nH]ccc12 22600,N1(C(CCC(=O)OCC)=O)CCC(CNCN2C(C3CCC3)CCC2)C(F)(F)C1 22601,C1(CNC(CCCCNC(N)=O)=O)CCN(C(=O)CC2CCCOC2)CC1(F)F 22602,c1(OC)ccc2c(C(=O)NC3CC(C)CN(C(c4csc(=N)[nH]4)=O)C3)coc2c1 22603,C1(CC(N2CC(COC)(CNC(C3CNC(=O)N3)=O)C2)=O)CC2CCC1CC2 22604,N1(C(CCSC)=O)CCC(C)(C)C(NC(c2cc(C3(C)CC(C)(C)C3)no2)=O)C1 22605,c1(C(C)N(C(=O)CC(c2cccc(C(F)(F)F)c2)N)C)ccc(F)cc1F 22606,N1(C2C(NC(C(CC)F)=O)CCC2)CCN(C(=O)CC2CC(=O)C2)CC1 22607,C(=O)(C1c2ccccc2CN1Cc1c(C)nc[nH]1)Nc1cc(Cl)ccc1I 22608,C=C(C)CC(C(=O)N1CCC(C)(C(=O)N(CCCO)CCO)C1)OC 22609,CC1CN2CCN1C(C(N1CCN(C(c3cc(Cl)ccc3Cl)=O)CCC1C)=O)C2 22610,N1(C(CCOC(C)C)=O)CC(O)CCC1C(=O)NCCN(C)C 22611,Cc1cc(C#N)nc(=NCC(C)CNC(c2c(C3CC3)cnn2C)=O)[nH]1 22612,N1(C(c2ccc(C)c(Cl)c2Cl)=O)CCCC2CCN(C(c3ccncn3)=O)CC12 22613,c1(OCC)ccc(C)nc1C(N1CC(COC)CC1CNC(=O)C=CSC)=O 22614,N1(C(CSCC#C)=O)CC2CCC1CN2C(=O)Cc1c[nH]c2ncccc12 22615,CCCC(CC)CC(=O)NCC1CC(C)N(C(C2OCC3COCCC23)=O)C1 22616,c1(C(N2CCC(NC(CCn3c(C)ncc3)=O)C2)=O)cc2scc(C)c2[nH]1 22617,C=CC1(C(=O)NCCN(CC)CC)CCN(C(=O)CCCC2CC2)C1 22618,c1(C(=O)NCC2(F)CCC(NC(c3ccn(C)n3)=O)C2)ccnc2ncccc12 22619,C12(C(N3C(CNC(c4cccc(COC)n4)=O)COCC3)=O)CC1CCC2(F)F 22620,N1(C(C(CC)CC)=O)CCCC(C2CN(C(C3(OC)CCCC3)=O)C2)C1 22621,O=C(CS(=O)(=O)c1cccnc1)N=c1cc(CCSC2CCCCC2)[nH][nH]1 22622,c1(CSC)cccc(C(=O)NC2CC2CNC(=O)C(C)C2CCCO2)c1 22623,c1(C(=O)NCC(C)(C2CC2)NC(C2C(OCC)C2)=O)nc(F)ccc1Cl 22624,c1(C(N2CC(C(=O)NCC(C)(C)C3CC3)(COC)C2)=O)ccc2cccnn12 22625,Cc1coc(C2CC2)c1C(=O)NCC1(NC(=O)C=C2CCN(C)C2)CC1 22626,C#Cc1ccc(C(N2CCC(NC(c3cc(O)ncc3Br)=O)C2C)=O)nc1 22627,CC1CCn2c(C(N3CC4C(N(C)C(C5C6CCN5CC6)=O)C4C3)=O)cnc2C1 22628,Cc1ccc2occ(C(N3CC(CCNC(C4CCC(C)NC4=O)=O)C3)=O)c2c1 22629,C1(NC(C(C)CS(C)(=O)=O)=O)CC2(CCCN(c3c(Br)cncc3[N+](=O)[O-])C2)C1 22630,c1(CC)ccccc1CC(=O)NCC(C)(Cn1cccn1)NCN1CSCC1=O 22631,C1(C(N2CC3C(NC(C4(C)CCOCC4)=O)(C3)C2)=O)CN2CCN1CC2 22632,c1(C(=O)NC(CN(C(C2(COC)C=CCC2)=O)CC)C)noc2cc(F)ccc12 22633,n1(CCC(=O)NC(CNC(C23C=CC(CC2)C3)=O)C2CCC2)cc([N+](=O)[O-])cn1 22634,N1(C(c2cc(C(=O)OC)sc2)=O)CC2CCCC(C1)N(C(C1CCC1)=O)C2 22635,CCCCCC(F)C(=O)N1CC2CC1C2C(N1CCC2CC12C)=O 22636,N1(C(C2(COC)CC(=C)C2)=O)CC(NC(c2ccncc2Cl)=O)C(C(=O)NC)C1 22637,C1(NC(COCCOCC#C)=O)CCN(C(c2c[nH]cc2C(C)(C)C)=O)CC1F 22638,N1(C(N2CCC(N(OC)C)CCC2)=O)CCOC2(CCC(F)(F)CC2)C1 22639,N1(CC(=O)NCC2(OC)CN(C(CC3(COC)CCCC3)=O)C2)CCCNC1=O 22640,c1(CCC)ccc(C(C(=O)NC(C)CC)N(CCCCO)C)cc1 22641,CCCC(C(N)=O)NC(=O)NCC(C)(C)CCOC 22642,c1(NC(C(c2ccc(C)o2)NCCN(C(=O)OC)CC)=O)ccccc1C 22643,CC(C)C(O)C(=O)NC1CC12CC(NC(=O)C=Cc1ccsc1Br)C2 22644,C(=O)(C(C)P(C)(C)=O)N1CC2C(C(N(CCOCC=C)C)=O)C2C1 22645,c1(CN(C(c2scc(C(=O)O)n2)=O)Cc2occc2C(=O)O)ncc(F)cc1F 22646,c1(C(N2CC(NC(C(C(C)C)O)=O)C(O)C2)=O)ccc2scc(Br)c2c1 22647,C1(C(N2CCC(CN(C)Cc3ccc(C(C)=O)cc3)C2)=O)CC(C)(C)OC1(C)C 22648,CC1=C(C)CC(C(N2CCCC2C(=O)NCC2(O)CCC(C)(C)C2)=O)CC1 22649,c1(OC(C)C)cc(N(CC(C)CNC(=O)Cc2ccc(Cl)nc2)C)ncn1 22650,C1(Nc2nccc(OC(F)F)n2)CCCN(CC2CCN(C(C)=O)C2)C1 22651,CCC(CC(=O)N1CCC(CCNC(=O)C(C)(CC)OC)C1)C1CCC1 22652,CC1(C)C(NC(=O)CN2CC3CC3C2)CCN1CC(=O)Nc1cnccc1Cl 22653,Cc1ccn2cnc(C(N3CCN(C(C4CCOC4C)=O)C(C(C)C)C3)=O)c2c1 22654,C(=O)(CC(C)(C)CC(=O)N1CCC(CNC(c2csc(CO)c2)=O)(OC)C1)OC 22655,N1(C(C(C)=CC=C)=O)CCC(C(=O)N2CCN(C(C)=O)CC2)=C(F)C1 22656,C1(C(=O)NCC=CC)CC2(CCC2)CN1C(=O)CC(C)NC(=O)NC 22657,O=C(C#CC1CC1)Nc1ncn(-c2ccccc2)n1 22658,C1(C=O)(CC)CCCC1O.N1(N2C(C)(C)CC=CC2=O)CCC(CC(C)O)CC1 22659,C1(NC(Cc2nc(CC)sc2)=O)CCN(C(c2ccncc2Cl)=O)C(C)C1 22660,c1(C(=O)NC(c2ccccc2)CNC(C(C=C)O)=O)nc2ncccc2cc1C 22661,CCCC(O)CC(=O)N(C1CCCN(C(=O)Cc2nccn2C)C1)C 22662,C1(C(N2CC(O)(C(F)C(=O)NC(C)(C)CF)C2)=O)(CC)CCOC1 22663,C1(C(N(CC(CC)NC(c2ccc(CO)cc2F)=O)C)=O)CC2(COCCO2)C1 22664,N1(C(CCCCC(=O)N(C)C)=O)CCC2(C1)CN(C(=O)C(=O)C(C)(C)C)CCO2 22665,N1(CCC(=O)NC(C(C)NC(c2c(C)onc2Cl)=O)C)CCSC(C)(C)C1 22666,S(=O)(=O)(c1ccc(=NCc2csc3cc(Cl)ccc23)[nH]c1)N(C1C(C)C1)C 22667,CCC(CO)(C(=O)N1CC=CC(C(=O)NOC(C)C)C1)OC 22668,Cc1cc(NC(C23CC(CN2C(c2ccc(C)nc2O)=O)C3)=O)c(=O)n(C)c1 22669,c1(OCCC(=O)NCC(C)N(C(=O)C(C)(F)F)C)ccc(F)cc1 22670,C1(CC(=O)NC(CNC(C2(C(=O)NC)CCC2)=O)(C)C2CC2)C=NN(C)C1=O 22671,c1(CC=C)ccccc1C(=O)NC(C)(CSC)C(=O)NCCOC(F)F 22672,C(C(C(C)(C)C)NC(=O)Cn1c(C)ccc1C)NC(C1C(=C)CC1)=O 22673,C(=O)(C(O)C(C)(C)C)N1C(C(=O)NC(COC)COC)CC2CC21 22674,C1(NC(=O)C2CC2)CCN(C(C2(C(F)(F)F)CCCCO2)=O)CC1CO 22675,C1(C2CCC(=O)NC2)(C(N2CC(N(C(=O)C(F)CC3CCCCC3)C)C2)=O)CCC1 22676,C1(CC=C)NC(=O)N(c2ccccc2)C1=O.c12cnn(c1)CCNC(=O)N1CCC21 22677,C1(NC(Cc2cn(CC)nc2)=O)CNCC(O)C1 22678,c1(CC(=O)NCC2CC(NC(c3c(=N)cc[nH]c3)=O)C2)cc(O)nc(O)n1 22679,c1(CN(C)C(C2CC2(C)C)=O)cnn2c1CN(C(=O)COc1cnn(C)c1)CC2 22680,C(C)(C(=O)N(C1CCCC1)CC1CC1)(N(C(C(C)c1cc[nH]n1)=O)C)C1CC1 22681,C1(NC(CNC(CC)=O)=O)CCC2CC1CN2C(=O)C(C)OC(C)=O.C1CCCC1 22682,C1(C(=O)NC(COC)C(C)(C)C)CCCCCCN1C(=O)C(F)CCC(C)C 22683,c1(C(C)NS(=O)(=O)C2CC2)cc(N(C)C)ncc1Br.C1CO1 22684,C1(OC)CC(NC(c2cn(C(=O)C(C)C)nn2)=O)CN(C(=O)CC2C=CCCC2)C1 22685,C(=O)(C(CCF)SC)N(CCCOCCC)SC(=O)OC(C)(C)C.C=CCC(=O)N 22686,C1(CNC(c2cn(CC)nc2)=O)CCC(NC(=O)CN2CCSCC2)CC1 22687,C1(NC(C2CCC(C)(C)OC2)=O)CC1C1CCN(C(c2ccoc2Cl)=O)CC1 22688,c1(C(C(N2CC(OCC)CC2(C)CNC(=O)OC)=O)=O)oc2ccccc2c1C 22689,O=C(CC(Cc1cccs1)NC(=O)Cc1ncc[nH]1)NCc1cccs1 22690,c1(N2CC=CC(NC(CCOC)=O)C2)ncc(C)c(C)n1 22691,c1(C(=O)NCCCCn2cc(C(C)OC)nn2)cnccc1C#N.C(CO)S 22692,CCCC(C(=O)NCC1CCC(NC(C2CC2CC(C)(C)C)=O)CC1)NC(N)=O 22693,N1(C(c2nnc(O)nc2O)=O)CC2CC1CCC2c1cn(CC(F)(F)CO)nn1 22694,c1(OC)ccc(C(N2CC3C(C(=O)Nc4cc(C)cc(C)c4)C3C2)=O)c(C)c1 22695,N1(C(=O)C(O)CC2CCCC2)CCN(C(c2cccc(CO)c2)=O)C2(CCC2)C1 22696,N1(C(c2cn(CCOC)nc2)=O)CCOC2(CCN(C(=O)C3=COCC3)CC2)C1 22697,C1(NC(CCCC#C)=O)CCN(C(=O)COc2ccc(C)cc2SC)CC1C 22698,Cc1c(C(C)NC(=O)C(C2CCOC2)N(C)C)cccc1Cl 22699,CC1CC=C(C(=O)NC(CC2CC2)C(=O)NCCCn2cnnc2)CC1 22700,C1(C)(C(N2CC(SCC)C2)=O)CCCN(C(=O)CC(F)(F)F)C1 22701,c1(C(=O)NCC(C2CC2)NC(C(COC)N(C)C)=O)sc(C)c(Br)c1OC 22702,C1(NC(c2c(C)noc2C(C)C)=O)CCCN(C(=O)C2=CCC2)C1C 22703,c1(C(=O)Nc2cccc(N3CCCS3(=O)=O)c2)cccc(-c2ccccc2)c1F 22704,Cc1c(C(=O)OC(C)(C)C(=O)Nc2ccccc2)nc(O)c2ccccc12 22705,C(=O)(C1=NNC(=O)C1)NC1CC(CNC(C2CCCC(C)C2)=O)C1 22706,c1(NC(C(CNC(c2c(CC)occ2)=O)O)=O)ccccc1C1CC1 22707,C1(CNC(C=CC(C)=O)=O)CC2CCC(C1)N2C(=O)CCCc1cccnc1 22708,C1(CN(C)C(C2COCCN2C(c2cncn(C)c2=O)=O)=O)CN2CCC1CC2 22709,C1(CNC(=O)C(O)Cc2cnc[nH]2)C2CN(C(C3CC(F)(CF)C3)=O)CC12 22710,C1(CNC(=O)OC)CCN(C(C2(CO)CN(CCC(=O)NC)C2)=O)C1.c1nccs1 22711,C12(CNC(=O)Cc3cn[nH]c3)CC(CN1C(c1cccc(C3CCOC3)c1)=O)C2 22712,C1(C(=O)NCC(C(C)(F)F)Cl)CCC(O)CN1C(c1cc(C#N)c[nH]1)=O 22713,c1(C(=O)NC(C(C)NC(C=Cc2ccc(C)cn2)=O)C)ccc(S(N)(=O)=O)nc1 22714,CC(CC(C)(C)C)C(=O)NCc1ncc(C(=O)N(C)CC2(O)CCOC2)cn1 22715,C(CNC(=O)C(=O)NC(c1cc(C)ccc1Cl)C)(CCS(C)(=O)=O)OC 22716,N1(C(C(CC)(C)O)=O)CCCC(CC)(NC(=O)CCNc2cccc(Cl)c2)C1.OCC 22717,C1(CC)CN(C(c2ccc(F)c(F)c2)=O)CCC1NC(=O)CN1CCCCCC1 22718,c1(C(=O)NCCCN(C)C(C2CC2C(F)(F)F)=O)cnn2cccc(Br)c12 22719,N1(CCNC(=O)NC2CCCC2CO)CCOCC1.C12CC(C1)N2 22720,C1(CN(C(=O)COCCF)CC)CCN(C(C2(C3CCCCO3)CC2)=O)C1 22721,CC1CCc2sc(C(N3CCC(NC(=O)CN(S(C)(=O)=O)C)C3)=O)cc2C1 22722,c1(C(=O)OC)c[nH]c(C)cc1=NCC1(C)CCN(C(C2COC3COCC23)=O)C1 22723,C(=O)(CC(O)C(C)C)NC(CC=CC)C(=O)NC(c1ncccc1F)C 22724,C1(CN(C2CCOCC2)CCC#C)CCN(C(=O)C(c2cnn(C)c2)C)CC1 22725,C(=O)(C1=CNC2=NCCCN12)N1CCCCC(NC(C2CC(C)N(C)C2)=O)C1 22726,C1(CNC(c2cnn(CC(C)C)c2C(F)F)=O)CN(CCF)CCC1(C)C 22727,c1(C(N2CCC(CC(NOCC(C)(C)O)=O)CC2)=O)cc(C#N)cn1C 22728,C1(CNC(=O)CC2CC2)CC2(CCN(C(c3ccc4oc(=O)oc4c3)=O)C2)CO1 22729,C(=O)(C(C)CC(=O)NCCCc1cncc(C(=O)OC)c1)OC 22730,c1(NC(C(=O)NC(c2c(OC(F)F)cccc2Cl)C)=O)cccc2c1CCC2 22731,c1(C(C)C)nc(=NCC2CCCCN2C(c2cn(C)cn2)=O)s[nH]1 22732,C1(NC(c2cc(C)ncc2)=O)CCN(C(C2OCCCO2)=O)CC1F 22733,c1(NC(CN(c2nnc(C)o2)CCOC)=O)c(Cl)cc(OC(C)=O)cc1Cl 22734,CCC(C)C(C)C(=O)N(C)CC1CCCCN1C(C1CCCC(C)CC1)=O 22735,CC(C)(C(=O)NCC1CN(C(C2CCS2(=O)=O)=O)C1)c1ccccc1 22736,Cc1cc(N2CCC(NC(C3CCSC(C)C3)=O)CC2)ccn1 22737,n1(CC(N2CCCC(N(C(C3CC3CF)=O)CC)C2)=O)cc([N+](=O)[O-])cn1 22738,Cc1ccc(C(N2CCCC(C)C2CNC(=O)C(F)F)=O)cc1[N+](=O)[O-] 22739,c1(C(=O)NCC2CN(C(CCCC#C)=O)CC2C(F)(F)F)ccc(CC)nc1C 22740,Cc1nc2nccc(C(=O)NC(C3CN(C(C4COCCO4)=O)CCO3)C)n2n1 22741,N1(C(=O)C2=C(Cl)CC2)CCC2(CCCN2C(C2CC3(C2)CC3F)=O)C1 22742,c1(NC(c2ccc(-c3cc(C)c(C)nc3)nc2C)=O)cccc2cc(Br)ccc12 22743,Cc1ccncc1C=CC(=O)NC(C1CN(C(C2CC3C=CC2C3)=O)C1)C 22744,CC(CCCCNC(C1CCOC1C1CC1)=O)NC(c1ccc(F)nc1)=O 22745,C(=O)(C1=C(C)C(C)(C)OC1=O)N1C(COC)CN(C(=O)Cc2ccc(C)s2)CC1 22746,C1(C)(CNC(c2c(C)cc(Cl)cc2)=O)CN(C(=O)C(=O)N(C)C)C(C)(C)C1 22747,C1(C(N(CCN(C(=O)CC2CCC(=O)N2)C(C)C)C)=O)CCNC(=O)C1 22748,N1(C(CCC(C)C)=O)CCC2CN(C(=O)Cn3cc(C4CCCC4)nn3)CC2C1 22749,C1(C(=O)NCC(C)NC(C(C)NC(c2ccco2)=O)=O)C(C)(C)OC1(C)C 22750,CCCC(C(=O)NCC1(O)CN(C(=O)CNS(=O)(=O)CCCC)C1)NC(N)=O 22751,c1(NCC(COC)(C)O)ccc(S(=O)(=O)NCC(C)(C)C)cn1 22752,C1(C(=O)NCC2CCN(C(=O)CC3COCC(C)O3)C2)(CC)CC(C)(C)C1 22753,Cc1nc2cncc(C(=O)NC(C3CN(C(C4C5COCC45)=O)CCO3)C)c2[nH]1 22754,C(=O)(C1=NOC(C)(C)C1)NCC1(NC(C2C(c3c(C)cccc3)C2)=O)CC1 22755,C(=O)(CCCc1ccncc1)N(CC(CC)NC(=O)C(C)(C)SC)C 22756,N1(C(C(C)(C)CF)=O)CCC2(CCCC2CNC(c2ccnc(O)c2)=O)CC1 22757,S(=O)(=O)(c1c[nH]c(C(=O)NCC2CC(C)N(C(C3C4COCC34)=O)C2)c1)NC 22758,CC1CCN(C(C2CC(=O)CC(=O)N2)=O)C(C(=O)NC2C3CCC(F)(F)C23)C1 22759,N1(C(C2(C=C)CCC2)=O)CCCC(CCC(=O)N(C)CCC2CCCN2C)C1 22760,c1(CNC(C23N(C(CSCCCC)=O)CCC2CC3)=O)nccn2nccc12 22761,C(=O)(C1=Cc2ccccc2OC1)N(CC(C)N(C(=O)CN1CCCCC1C)C)C 22762,c1(C(C)=O)ccc(CC(=O)N2CCC2)cc1.c1(C(C2CCCOC2)O)cn(CCN)nn1 22763,c1(CCC(N2C(CC)CN(C(C3(CF)CCC3)=O)CC2)=O)ccc2c(c1)OCO2 22764,c12cc(O)cc(O)c1C(=O)CO2.C12(COC(CC=C)=O)CC1CN(C(C)=O)C2 22765,c1(OC)cc(C(=O)N(CC(C)NC(c2c(C)nc(C)n2O)=O)C)ccc1C 22766,c1(C(=O)NCC2C(NC(C3(CC#C)CCCC3)=O)C2)cnc2[nH]cnc2c1 22767,C(CNC(c1cccnn1)=O)(C(C)C(C)C)NC(Cc1cncc(C)c1)=O 22768,N1(C(C2CCC(C)O2)=O)CC=C(CCNC(c2cc(Br)n[nH]2)=O)CC1 22769,C1(C(=O)NC(C2CCCC2)CNC(C(C)C2CCCO2)=O)CC(=O)NC1(C)C 22770,N1(C(c2cn(CC)nc2)=O)CCC(C)(C)C1CC(N1CC(C)(C#N)C1)=O 22771,S(=O)(=O)(c1cccc(-c2nnc(N3CCCC3C)n2CC(C)C)c1)NC 22772,C1(NC(Cc2c(C)cco2)=O)CN(c2nnn(C)n2)CC2(CC2)C1 22773,C(C1C(C(=O)N(C)CCOCCNC(c2sc(CO)nc2C)=O)C1(C)C)=C(C)C 22774,O=C(CCCC(F)(F)F)NCC1CN(C(C2CC23CCCCC3)=O)CC1O 22775,c1(C(=O)NC23C(CN(C(C4(NC(C)=O)CCCC4)=O)C2)C3)cc2nc[nH]c2cn1 22776,CCC(CCCC(=O)NCC12CCCC1OCC2)NC(C1C2CCCCCCC12)=O 22777,C1(C(=O)NCC(=O)NC(C(C)NC(=O)CCC2CC2)C)CCCCC1 22778,Cc1ccc([N+](=O)[O-])c(C(=O)NC2CCCN(C(c3ccccc3O)=O)C2)c1C 22779,CCC(CC)CCCC(=O)NC(C1(O)CCN(C(c2noc(CC)c2C)=O)C1)C 22780,C1(NC(c2csc(Cl)n2)=O)CC(O)CN(C(c2ccc(OCC3CC3)nc2)=O)C1 22781,C12(NC(c3nsc4ccc(C)cc43)=O)COCCC1CN(C(=O)C=CC(C)C)C2 22782,N1(C(C2CCC(=C)CC2)=O)CC(=O)NCC1C(=O)NCCC(=O)N(C)C 22783,C1(NC(C2C(C)C2)=O)CCCN(C(c2cn(-c3ccc(Br)cc3)nn2)=O)C1 22784,C=CCC(C)(C)CC(=O)NCCC1CCC(NC(c2cc3ncccc3s2)=O)C1 22785,C1(C(N2C(C(C)C)C(C)(C)C2)=O)CN(C(=O)CC2CCC(C)(C)C2)CC12CC2 22786,C(=O)(C1CCCn2cnnc21)NCCC(CNC(c1cnc(CC)o1)=O)OC 22787,C1(C(=O)Nc2ncc(Cc3ccnc(C)n3)s2)CCc2ccccc2O1 22788,C1(C(C)NC(c2cnnn2C)=O)CCN(C(c2cn[nH]c2)=O)CC1 22789,N1(C(c2c(C)c[nH]c2)=O)CCC2(CC1)CC(C(=O)NC(CO)CC(C)C)CO2 22790,c1(OC)c(CC(=O)NCCN(CC(C)O)C(C2CCCCS2)=O)cccc1F 22791,C(CC(=O)N1CCN(CC2(NC(C3=CCC(C)C3)=O)CC2)CC1)(C(F)(F)F)OC 22792,c1(NC(C)=O)ccc(O)c(C(=O)N(C2CCC(NC(=O)CSC3CC3)CC2)C)c1 22793,C(C)(N=c1cc(C)nc(OC(C)C(C)(C)OC(C)(C)C)[nH]1)c1cccc(OC)c1 22794,N12CCC(CF)(C1)CNC(=O)C1(CCC1)C2=O.C1(N)CCCCC1.COC 22795,c1(CC)cc(CNC(=O)C(C)=CCNC(c2cc(OC)n[nH]2)=O)on1 22796,CCC(C)(C)C(C)NC(C1CCN1C(=O)C(C)NC=O)=O 22797,C=CC1OCCC1C(=O)NCC1CC(O)CN1C(C12CCN(CC1)C2)=O 22798,c1(NC(CCC(=O)OC=C)=O)cc(Cl)ccc1NCC(F)F 22799,Cc1cn(C)nc1C(=O)NC(CC1CCCC1)C(=O)NC1CCOCC1F 22800,C(=O)(C1COc2ccccc21)N1C(CNC(c2n[nH]c(C)c2O)=O)CC(F)(F)C1 22801,CC(C)C(O)C(C)C(=O)NCC1CCOC1C(N1CC2CC(O)CC1C2)=O 22802,N1(C(c2[nH]cc(C(C)(C)C)c2)=O)CCC2CN(C(c3ncc(F)cn3)=O)C2C1 22803,C(=O)(CC(O)CC(C)C)N1CCN(C(C(CCCOC)C)=O)CC1c1ccco1 22804,c1(NC)c(C(=O)NC2CN(C(=O)CCSc3nccn3C)CC2F)cccc1F 22805,c1(C(=O)NC2C(NC(=O)CC3CC4(CC4)CO3)CCC2)ccc2c(c1)CNC2=O 22806,C#CCCC(O)C(=O)N1CC(F)CC1CNC(C1(S(N)(=O)=O)CC1)=O 22807,c1(C(=O)NC2C3(CCN(C(C(CC)SC)=O)C3)C2)ccc2nc(C3CC3)[nH]c2c1 22808,C1(NC(CCc2n(C)cnn2)=O)CCCC12CN(C(=O)CC1(O)CCOC1)C2 22809,c1(C(=O)NCCCCC(CO)NC(CCN(C)CCO)=O)ccc(C#N)c(O)c1 22810,N1(C(c2nn(CC)c(O)c2)=O)CCCC(C)(C)C1CNC(=O)C(C)(C)OC 22811,c1(C(=O)NCC2(F)CN(C(C3C4CCOCC34)=O)C2)ccc2ncnc(O)c2c1 22812,CCCCCCCCCCCCCCCN(C)C(C1CC(=O)NC2CCCCC12)=O 22813,c1(CNC(C2CCC(F)C2)=O)ncc(Cl)cc1Cl 22814,c1(-c2scc(C(N3CCC(NC(CCC=C)=O)C3)=O)n2)ncccc1F 22815,C1(C(N(C2CCN(C(c3nc(OC)c(F)cn3)=O)C2)C)=O)CCC2C(C1)C2(F)F 22816,c1(C(=O)OC)cc(C(=O)NCCNC(=O)COCC2CCCCO2)on1 22817,Cc1oc(CNC(C2CN(C)C2)=O)nc1C(=O)N(C)CCC1CCC1 22818,c1(C(=O)NCC2N(C(C3C(C)(C)C3)=O)CCC2)ccccc1S(C)(=O)=O 22819,C12(C(N(CC(CCC)C)C)=O)C(NC(c3cocn3)=O)C3CC1C2C3 22820,N1(C(CO[Si](C)(C)C)=O)CC(O)CC1CNC(C1(C(F)(F)F)CC=CC1)=O 22821,C12(CCC(C(N3C(C(C)(C)C)CCC3)=O)C)CC(C(=O)N(C)SCC)(CO1)C2 22822,C1(CC(=O)Nc2cnsn2)CCCN1CCN1CCC1 22823,c1(OC)cc(CSCC(=O)Nc2noc(C3CCOCC3)n2)cc(F)c1 22824,Cc1nnn(CC(=O)NCCC(C)NC(=O)Cc2ccn(C3CC3)n2)n1 22825,N1(C(C(C)(C)SC)=O)CCC2(CC1)CC2NC(c1cnn(CCCOC)c1)=O 22826,c1(C(N2CC(OC)(CNC(C3(C)CCCNC3=O)=O)C2)=O)nc[nH]c2nccc1-2 22827,Cc1csc(Cl)c1C(=O)NCC1CN(C(=O)C(O)Cc2cccc(Cl)c2)CC1C 22828,c1(C(=O)NC2CCC(CC(=O)NCc3ncc(C)s3)CC2)cc2ccccn2n1 22829,Cc1nnc2n1CC(NC(=O)C(F)C1CCOC1)C2 22830,c1(NC(=O)Nc2nnc(C(C)C3CC3)o2)nn(C)c2ccc(Br)cc12 22831,CC(C)CC(C(=O)N1CCCC(CNc2ncccc2C#N)C1)C(N)=O 22832,N1(C(c2occ(C)c2C)=O)CC2OCCN(C(C3CCCCS3(=O)=O)=O)C2C1 22833,N1(Cc2ncc(C(=O)OC)s2)CCc2c(NC(=O)C(F)(F)F)cccc2C1C 22834,N1(C(CCCCC)=O)CC2(C1)CN(C(=O)CCC1CCCC(O)C1)CC2CO 22835,C(=O)(C(CCCC)C(C)C)N1CCC(C(=O)NCCOCC=C)C1CC 22836,C1(C2(NC(c3c(CCCC)ocn3)=O)CC2)CCCCN1C(=O)C=CC(F)(F)F 22837,Cc1cn2ccc(C(N3CC4CC3CN4C(=O)Cc3cncn3C)=O)cc2n1 22838,CC1(C)C(C(=O)NCc2ccc3c(c2)CC3)CCN1C(c1c[nH]c(=O)cn1)=O 22839,N1(C(C(CCC(C)C)F)=O)CC(C)CN(C(c2cnc(N(C)C)cn2)=O)C(C)C1 22840,c1(C(=O)NC2C(NC(C3=CCCC3C)=O)CCC2)cc2c(s1)CCCCCC2 22841,N#Cc1ccc(C(=O)NCC2CNCCC23CCC3)cc1Cl 22842,N1(C(CC(C(C)C)C)=O)CCC(N(C)C(C2CC3(C2)CC(O)C3)=O)C2(CC2)C1 22843,C(=O)(C(CCC(C)C)NC(C1CN2CCN1CC2)=O)NCC1CCCN(CC)C1 22844,CC(O)CCC(=O)N(C1CCC(NC(=O)CCc2ccccc2C(N)=O)CC1)C 22845,C1(C(=O)N(CC(C)NC(C2C3CCC2CC3)=O)C)(COC)CCCCO1 22846,C1(C)(COC)CC(NC(c2cc(N)ccc2Cl)=O)CN1C(=O)CCCC1CC1 22847,c1(SCC(=O)NCC2CCCC2NC(C2CC23CCC3)=O)ccc(F)c(F)c1 22848,CC(C)CC(C(=O)N(CCC(=O)NCC1CC(C)(C)OC1(C)C)CCO)C(N)=O 22849,C(=O)(CC(CNC(c1ccc(C2CC2)o1)=O)C1CCC1)NCC(CC)(C)O 22850,Cc1ccc(CCC(=O)NC2CN(C(C3CC4(CC4)CO3)=O)CCC2O)cc1Cl 22851,c1(C(=O)NC(CNC(C(CCC)C)=O)CO)c(NC(=O)C2CC2)sc(C)c1C 22852,c1(C(N(CCC(=O)NC(C2CCOC2)C)CC#C)=O)scc(C)c1OC 22853,CCCCC(F)C(=O)NC1CCN(C(=O)C(O)C(C)(C)C)C(C)C1 22854,c1(CC(N2C(C(C)C(=O)O)CCC2)=O)cc(C(F)(F)F)ccc1Br 22855,CC1=C(C)CC(C(N2CCCC(NC(C34COC(CF)(C3)C4)=O)C2)=O)CC1 22856,N1(C(C(COCC)C)=O)CC(N(C)C(c2cnc(SC)nc2O)=O)C2(CC2)C1 22857,c1(OC)cc(CO)c(C(N2CCOCC2C2CCOCC2)=O)c2ccccc12 22858,c1(C(c2n(CC)nnn2)NCC2(c3cc(C)no3)CCCC2)nc(C)c(C)[nH]1 22859,CC1CCN(C(=O)Cn2ccnn2)C(C)C1NC(c1cccc(C2(C)CC2)c1)=O 22860,c1(CCN=c2ccnc(NC3CN(CCOC)C3)[nH]2)oc2ccccc2c1C 22861,C(c1ccc2ccccc2n1)=CC(=O)NCC1C=CC(NC(=O)CCF)C1 22862,N1(C(N2CCCCCC(C)(C)C2)=O)CCC2CC(C(N3CCC(NC)C3)=O)C2C1 22863,C1(C2CCC2)(C(N2CCC(C(F)(F)F)(CNC(=O)Cc3cnns3)C2)=O)CC1 22864,N1(C(c2c(C(C)C)nn(C)c2)=O)C(CNC(=O)COCC2CC2)CC2COCC12 22865,c12ccc3c(c1)CCN3S(=O)(=O)C2.O=C1OCCN1c1ccc(NCC2CC2)s1 22866,CC12CC(C(N3CCC(F)(CNC(=O)C4=CCCOC4)C3)=O)(CCO1)C2 22867,C1(C(=O)NC(C(C)C)C)CCN(C(=O)CCCc2cnn[nH]2)CC1O 22868,N#CC1(C(N2CCC3(CC(NC(C4CNC(=O)N4)=O)C3)C2)=O)CC2(CCC2)C1 22869,C(C)(C)(CCC(=O)N1CCCC(COC)(NC(c2ccc(C)nc2)=O)C1)OC 22870,C12(C(=O)NCC3CN(C(C4CCCC45CCC5)=O)CCO3)C3CC(CC13)C2(F)F 22871,c1(C(=O)NCCN(CCCN(C)C)C(C2C(C)C2C)=O)csc(Cl)c1 22872,N1(C(C#CC2(C)CC2)=O)CCCC2CN(C(c3noc4c3COCC4)=O)CCC12 22873,C=CC(C(=O)NC(C1CCCN1C(C1CC1(C)C)=O)C)OC 22874,CC(C(=O)N1CCC(C(C)C(=O)NCC2(SC)CC2)C1)C(F)F 22875,C(CN=C(NC(CO)CCF)N1CCN(c2ccccc2Cl)CC1)OCC 22876,Cc1ccc(F)cc1CN(C1C2CCC1CNC2)C(c1ccnc(OC(F)F)c1)=O 22877,C(=O)(C(C)(O)CCN(C)C)N1C2C(C(N(CCCCOC)C)=O)C(C2)C1 22878,C1(C(N2C(CN(C(c3c(CC)non3)=O)C)CCCC2)=O)Cc2ccncc2C1 22879,c1(OC)cc(C(N2CCC(SC)CC2)=O)ncc1-c1cccc(N2CCCC2)n1 22880,S(=O)(=O)(c1ccc(F)c(F)c1)N1C(C(=O)NCc2ccc(CO)cn2)CC2CC21 22881,Cc1cc(O)cc(C)c1CC(=O)NCC1CCCCC1NC(=O)Cn1ncnn1 22882,CC1(C#N)CCN(C(=NC2CCC2)NC2CC2c2ccc(OC(F)F)cc2)CC1 22883,CCC(C)C(O)C(C)C(=O)NC(Cn1cncn1)C(N1CCC(O)(CC)C1)=O 22884,c1(C(N2CCC(C3(NC(C(C)=C(C)C)=O)CC3)C2)=O)ccc2ncccc2n1 22885,N1(C(c2n[nH]c(CC)c2Cl)=O)CCCC(O)(CNC(C2CC23CC3)=O)CC1 22886,N1(C(c2c(CC)cns2)=O)CC(N(C(=O)C(C2CC2)OC)C)C2(CC2)C1 22887,N1(C(c2coc(Br)c2)=O)CCN(C(C2(n3ccnn3)CC2)=O)C(C2CC2)C1 22888,c1(NC(CNC(CNC(C(CC=C)C)=O)=O)=O)ccc2ccncc2c1 22889,CCCC(C)(O)C(=O)NCCC1CCCN1C(c1c(OCC)nn(C)c1OC)=O 22890,C1(C(=O)NC2CCC(n3cc(CCP(C)(C)=O)nn3)C2)CC2C=CC1C2 22891,C1(NC(c2ccc(OC(F)F)cc2)=O)CCN(Cc2nccc(C(F)F)n2)CC1 22892,c1(SC)ccc(CN(C(c2cc(C)ns2)C(=O)NCC2CCCO2)C)cc1 22893,C=C(CNC(=O)C(C)(C)C1CCCC1)CCNC(=O)CSCCOC 22894,C(N=c1[nH]c2c(F)cc(Cl)cc2s1)C1CCN(C(c2nc(CC(C)C)sc2)=O)C1 22895,C1(CNC(C(CC=CC)C)=O)CN(C(c2cc(Cl)cs2)=O)CC1(F)F 22896,c1(C(=O)NCCC2CN(C(C3CCC(O)CC3)=O)CCO2)coc2c1COC2 22897,N1(C(c2cn(CC=C)nc2)=O)CC(O)CC1CNC(=O)C(C)OCCOC 22898,Cc1nc2[nH]c(C(N3CCCC(C)(NC(C4(COC(C)C)CC4)=O)C3)=O)cc2s1 22899,N1(C(C(C)NC2CCCC2)=O)CCC2(CC1)CC2CNC(=O)CN1CC(C)(C)C1 22900,Cc1cc(NCCc2ncc(Br)cn2)ncc1S(=O)(=O)NC(C)(C)C1CC1 22901,C1(NC(C2C(NC(CCc3n(C)ccn3)=O)COC2)=O)CCCCC12CC2 22902,N1(C(C(C)(C)C(N)=O)=O)CCN(C(=O)Cc2cnn3ccccc23)CC(O)C1 22903,c1(OC)ccc(F)c(C(c2nnnn2C(C)(C)C)NCC(C)CO)c1F 22904,C1(CNC(=O)CC2=CCCC2)CC2CCC1N(C(=O)CC1CCC3CC3C1)C2 22905,N1(C(c2c(-c3cn(C)nc3)ocn2)=O)CC=C(CCNC(C2CCCS2)=O)CC1 22906,C1(O)(C(C(C)C)NC(C(C)OCCC=C)=O)CN(C(=O)C=Cc2ccc[nH]2)C1 22907,c1(CCC)ccccc1COC(=O)CCC(=O)NCc1cccc(C(F)(F)F)c1 22908,c1(-c2cccc(SCC)c2)cnc(C(F)(F)F)cc1NC(c1cc(C)c(Cl)cn1)=O 22909,c1(C(N2C(CN(C(C(CSC)(C)C)=O)C)COCC2)=O)nsc2ccc(C)cc12 22910,c1(NC(C2C3CC(=O)CC32)=O)cn2nncc2cn1 22911,c1(C(=O)NC(C)CNC(c2cc(-c3c(F)cccc3F)on2)=O)cc2c(s1)CCC2 22912,CC1CCC(C)N1CC(=O)NCc1ccc(C(=O)O)cc1 22913,c1(OC)ccc(C(N2CCCC(CNC(C3(C)CC4CC4C3)=O)CC2)=O)c(N)c1 22914,N1(CCC(=O)NC2CC(C)(NC(C3C=CCCC3)=O)C2)CCCS1(=O)=O 22915,c1(C(=O)NCCCN(C(C(C)OCC)=O)C)cc2ccccc2c([N+](=O)[O-])c1N 22916,Cc1cccc(CCC(=O)NCC(C(C)C)N(C(=O)C(C)(C)c2cscn2)CC)c1 22917,c1(C(=O)NCC2CC2)ccccc1OC1(COC)CN(C(=O)C(C(C)O)SC)C1 22918,C1(C(N2C(CNC(C(C3CC(F)(F)C3)OC)=O)CC2)=O)CCC(F)(F)CC1 22919,CC(C)CC(F)C(=O)NCC1C2CCC(C2)N1C(=O)CNC(C1CCCC1)=O 22920,c1(OC)cc(F)ccc1C(N1CCC(CNC(C2CCSC2)=O)(OC)C1)=O 22921,CCC(C)(CCNC(c1nocc1C)=O)NC(=O)COC1(C)CCCC1 22922,N1(C(C(=O)N(C(C2CC3CC3C2)C)C)=O)CCCC(N(C)C)C1 22923,c1(C(=O)NCCN(C(C2CN(C)CC2c2cccnc2)=O)CC)ncc[nH]c1=O 22924,C1(=O)C(C(C)(C)F)NC(C)(C)C(C)N1.C(C)(C)(C)OC(=O)NC1COC1 22925,N1(C(C(C)(C)NC(C(C)C2CCOC2)=O)=O)CCc2ncccc2C1 22926,N1(C(CC2CCC(=O)NC2)=O)CC2CC3CC2C1C3NC(C1CCC2(CC2)C1)=O 22927,CC(C)(O)C(C(=O)NOCC1CCCCC1)NC(c1cccnc1S)=O 22928,C(=O)(C(O)CCCC)NCC1OCCN(C(C2(C=C)CC2)=O)C1 22929,N1(C(C(F)=CC)=O)CCC2CN(C(C3CCN(c4ccccc4)C3)=O)C2C1 22930,C1(C(N(C(C)CNC(C2CC2C(C)O)=O)C)=O)CCC(N(C)CCO)C1 22931,c1(N(C)CCN2CCOCC2)cc(Br)c(C(F)(F)F)cc1F.c12cccc(c1)S2 22932,N1(C(c2n[nH]c(=N)o2)C(=O)NCc2cccc(OC)c2)CCNC(=O)C1CCO 22933,C12(CNC(C3(F)C(C)C3)=O)CC(NC(C3CS(=O)(=O)C3)=O)(C1)C(C)O2 22934,c1(C(N(C2CCCN(C(CNC(=O)OC)=O)C2)C)=O)cc2c(=O)[nH]c(C)cn2n1 22935,C1(OC)CN2CCCC2(C(=O)NCC2CC(NC(c3c(Cl)cccc3Cl)=O)C2)C1 22936,N1(C(CCc2onc(C)n2)=O)CC2CN(C(=O)CC3CCC(=O)NC3=O)CCC12 22937,C(CO)(CCCCNC(=O)C=CC1CC1)NC(C(CC#C)O)=O 22938,N1(C(C2C(CNC(C3CCCS3)=O)CC2)=O)CC(F)(F)C(F)(F)C1 22939,C#Cc1cccc(C(N2CC(NC(=O)CC(C)CN(C)C)C(C)(C)C2)=O)c1C 22940,CC1=CCSC1C(=O)NC(CNC(=O)CCc1nccn1C)CO 22941,Cc1ncnc(C(N2CCC(NC(=O)CC3C=CCCC3)C2(C)C)=O)c1C 22942,C1(C(=O)NCCCC)(NC(C2CCN2S(C)(=O)=O)=O)CCC(C)(C)CC1 22943,C1(O)(CC=C)CCN(Cc2c(C(=O)OC)c[nH]c(=N)n2)CC1 22944,c1(C(N2C(CNC(C3N(C)CCCC3)=O)CC(O)C2)=O)ccc(N)c(Cl)n1 22945,C1(C(C)NC(=O)CC(=O)NCC2CC2)CN(C(C2(C)CCN(C)C2)=O)CCO1 22946,c1(C(=O)NCc2cn(C3CCN(C(C(C)=CC4CC4)=O)C3)nn2)ccccc1C 22947,Cc1cc(N2CC(F)(F)CC2CCNC(=O)CCc2cncs2)n2ncnc2n1 22948,S(=O)(=O)(c1ccccc1Cl)NCC(=O)NCCN(C)C(c1ccns1)=O 22949,c1(C(N2CCN(CC(F)NC3CCCN(C(C)=O)C3)CC2)=O)csc2nccn12 22950,S(=O)(=O)(c1cccc(=NCC(C)n2cncn2)[nH]1)NC(c1ncc(C)o1)C 22951,N1(C(=O)NC2C(C3C(C)C3)C2)CCC(N=c2nc[nH]n3c(Br)ccc23)C(C)C1 22952,C1(NC(=O)C2CC2)CC(CN)C1(C)C.n1(CCC)cc(C(=O)NC)cn1 22953,C1(c2cccc(C)c2)CN(Cc2cc(C3CC3)nn2-c2ccc(F)cc2)CCN1C 22954,C1(CC)CCC(C(N2CCOC(Cc3cn(-c4ncccc4Cl)nn3)C2)=O)CC1 22955,C1(NC(CCCCCC)=O)CC2CN(C(c3cc(C)n(C(C)CC)n3)=O)CC2C1 22956,c1(C(=O)NC23C(CN(C(C(C)C4CCC4)=O)C2)C3)ccc2c(c1)C(=O)NCCO2 22957,C1(S(N)(=O)=O)(C(=O)NCCCOCCCNC(C2(SC)CC2)=O)CC1 22958,C(=O)(CC(C)C(C)(C)C)NCCN(C(C(CC)CC)=O)CC1CC1 22959,C(CO)(C(F)(F)F)NC(C(Cc1cc[nH]n1)NC(=O)CCn1cncn1)=O 22960,N1(C(C=C(C)c2cnn(C)c2)=O)CCN(C(c2ccc3cc[nH]c3n2)=O)CCC1C 22961,C1(C(N2C(CCNC(c3nc(C4CC4)cs3)=O)CCC2)=O)CCC2(CCC2)C1 22962,c1(OC)cccc(C(N2CCC(CF)(NC(=O)Cn3cccn3)C2)=O)c1 22963,c1(NC(C2CC3CC3N2C(=O)CC2C=CS(=O)(=O)C2)=O)ccc2nncn2c1 22964,N1(C(CC(C(C)C)O)=O)CC(C)(CNC(=O)COCCCN(C)C)CC1(C)C 22965,C#CCCCCC(=O)NCC(CC(=O)N(CC(C)C(=O)OC)C1CC1)C1CCC1 22966,N1(C(CC)=O)CCN(C(c2[nH]ccc2-c2ccccc2)=O)CC1CC1CC1 22967,Nc1cc(Br)ccc1C(N1CCC(NC(c2ocnc2C2CC2)=O)C(O)C1)=O 22968,CN1CC=C(C(=O)NCC(C2CCCN2C(C2CCC(=O)N2)=O)(C)C)C1 22969,C1(C(=O)NCCC2CCN(C(=O)C(F)CC3CCC3)C2)CC(F)C(=O)N1 22970,c1(CNC(c2cnc(CC)s2)=O)ccc(CNC(=O)CN2CSCC2)cc1F 22971,C1(CC(=O)NCC(C)NC(c2nnc(C(C)(C)C)o2)=O)CCOCC1 22972,c12cc(F)ccc1NC2=O.C(C(=O)N(C)CCC(C)CC)OCCOCC#C 22973,C1(C(C)(C)O)CCN(C(C2(C(n3cc(-c4cc(N(C)C)ns4)nn3)C3CC3)CC2)=O)C1 22974,N1(C(CC(CC)C2CC2)=O)CCN(C)CC1C(=O)NOCC(C)CC 22975,CN1CC(N(C=O)CCc2c[nH]c3cc(F)ccc23)CCc2ccccc21 22976,c1(C(=O)NCC(C)(C)NC(C(CC#C)C)=O)cccc(Br)c1SC 22977,c1(C(N2CCC(N(C(c3coc(C)n3)=O)CC)C2)=O)cc(F)c2ncccc2c1 22978,c1(CNC(C)C(C)(C)NC(c2cc(C3CC3)no2)=O)ncc(F)cn1 22979,Cc1ccc(C2CC2NC(C2CC(C)CCN2C(=O)C(O)C(F)F)=O)c(Cl)n1 22980,C(=O)(C1=CC2CCCCCC12)N1CC(N(C)C(C2C3CC4CC(C3)CC2C4)=O)C1 22981,N1(C(CCCOC(C)C)=O)CC2(CC(NC(c3csc4cncn34)=O)C2)C1 22982,C1(N(C(C2C(OCC)C2)=O)CC)CCN(C(=O)Cc2cccc(F)c2)CC1 22983,N1(C(C(=O)NCC)=O)CCC2(CC1)CC2NC(=O)C(C(C)C)NC(N)=O 22984,CN1CC2C(CCN2C(=O)C(=O)NC2Cc3ccccc3C2N)CC1=O 22985,C(CN=c1nc2scnc2c(NCc2ccc(O)nc2)[nH]1)c1c(C)nn(C)c1C 22986,Cc1ccc(C(=O)N(c2cnncc2C)C2CC3(CNC3)C2)nc1 22987,c1(C(=O)NCC2C(C)CCN(C(C34CC(C3)C4)=O)C2)ccc2nn[nH]c2n1 22988,c1(CC(N2CCCN(C(=O)CC3CC4CCC3C4)CC2)=O)ncc(F)cc1F 22989,n1(CC)cc(C(=O)NC(C2CCOC2)CNC(c2cc(C(F)(F)F)no2)=O)nn1 22990,N1(C(c2n(CC=C)ccc2)=O)CCCN(C(=O)CCCOCC)C(C)C1 22991,C1(NC(C2CCOCC23CCC3)=O)CC2CCC1CN(C(=O)Cc1cccs1)C2 22992,c12cc(c(Br)cn1)C(=O)N2.Cc1ccc(OCC2(CC#N)CC2)cc1 22993,C1(C(=O)NCC2C(CNC(Cn3ccc(C)c3)=O)C2)CCC2(CC2)C1 22994,C1(C(C(N2C(C)CC(OCC)C2)(C)C)=O)CC2(C1)CC2C(=O)OC 22995,N1(C(C2COC(=O)O2)=O)C(CNC(C2(CCO)CC2)=O)CC2COCC12 22996,C1(CC(=O)N(c2cccc(N3CCCC(O)C3)c2)CCO)CCC2(CCCC2)CC1 22997,N1(C(c2cnc(C(C)C)nc2)=O)CC(NC(C2CCCC2O)=O)CC(C)(C)C1 22998,N1(C(C(N2CCSCC2)C)=O)C2CCCC1CN(C(c1cc(Cl)c(Cl)s1)=O)C2 22999,CCS(=O)CC(=O)N(CCCCNC(C1COCCN1C(C)=O)=O)C 23000,c1(CC)c(C(=O)NCCC2(NC(C3CCC(C(N)=O)O3)=O)CCC2)nnn1C 23001,C(=O)(C(CNC(c1cnsc1C)=O)CC(C)C)NCc1c(C)nc(C)[nH]1 23002,Cc1cc(C(=O)NC(C)CCNC(=O)C=Cc2cnccc2C)ccc1C#N 23003,c1(C(N2CCc3nn(C)cc3C2)C(=O)NCCSCC)ccc2c(c1)n(C)c(=O)n2C 23004,c1(CNC(c2occc2CNC(C2C=CCCC2)=O)=O)ccc2n[nH]cc2c1 23005,c1(CN2CCN(C(c3ccc(Cl)nn3)C)CC2)nccc2cnn(C)c12 23006,n1(-c2cc(C)on2)c(C)cc(C(=O)NCC(C)NC(=O)C(F)C(C)C)c1C 23007,C1(CCNC(=O)NC(C)CN2CCOCC2)CCCS1(=O)=O 23008,c1(N(C)Cc2nccc(C)c2)nc(=NC2CCN(C)C2)[nH]c2cc[nH]c12 23009,CC(O)C(C)(C)C(=O)N(C)CC1CN(C(C2(CC(C)C)CCCC2)=O)CC12CC2 23010,C1(F)(C(=O)NCC23CC(CNC(C(CC)COC)=O)(OC2)C3)CCC(F)(F)CC1 23011,c1(COC)[nH]c(=N)sc1C(N1CC(CNC(=O)C=CBr)CC1C)=O 23012,C(=O)(C#CC1CCCCO1)O.C(C(C)C(=O)OCC)COC 23013,C1(C(C)C(=O)NCc2cccc(Cl)c2)CCN(C(C2CCC(=O)C2)=O)CC1 23014,C#CC1CCC(N(C(C2CCN(C(c3ccc(C)o3)=O)CC2)=O)CCC)C1 23015,CCC(CCOC)C(=O)NC12CCC(C1)N(C(c1sccc1-n1ccnn1)=O)C2 23016,CC1CN(C(C2CC3C=CC2C3)=O)CC1NC(c1cnn(C)c1N)=O 23017,N1(c2c(S(=O)(=O)N3CCCCCC3)cccc2)CCOCC2(CCCC2)C1 23018,N1(C(=O)Nc2ccc(-c3ccoc3)cc2)CC(c2ccc(Br)cc2)C2(CCC2)C1 23019,N1(C(c2cn(CCC)nn2)=O)CC2(NC(=O)C(c3ccc(F)cc3)F)CC1C2 23020,C1(N(C(c2c(C)ocn2)=O)C)CCCC(N(C)C(c2ccon2)=O)C1 23021,C1(C(NOCC=C(C)C)=O)CCCCCCN1C(=O)C(C)C(=O)OC(C)(C)C 23022,Cc1cccc(C(N2CCOCC2CC(=O)NCC2(CO)CC23CCC3)=O)c1F 23023,C1(NC(C(C2CC(F)(F)C2)NC(c2ccc(CC)s2)=O)=O)CC2(CCC2)C1OC 23024,Cc1onc(Cl)c1C(N1CCC(Cn2cc(-c3nccnc3N)nn2)C1)=O 23025,C1(OC)C2CC1N(C(=O)C(C)OCCC(C)C)C2.c12ccnc(c1)COC2=O 23026,N1(C(c2cc(NC(c3c(C)nn(C)c3C)=O)cn2C)=O)CC2CCC(C1)N2C 23027,C1(CC(NOCC2CC(=C)C2)=O)CN(C(=O)C(C)O)CC1C 23028,C1(n2cc(CNC)nn2)CCCN(C(=O)C(C)(C)c2ccc(Cl)s2)C1 23029,C1(C(N2C(C(CNC(C3C(C)OCCC3)=O)(C)C)CCC2)=O)CC2CC1C1CC21 23030,C1(CC#N)CN(Cc2ccc(Cl)nc2)CCN1Cc1sccc1Cl 23031,c1(C(=O)NCC2(O)CN(C(C(c3c(C)cncc3)C)=O)C2)cc2c(s1)CCSC2 23032,c1(C(=O)NC2CC(C)N(CC(=O)Nc3ccncn3)C2)ccc2c(c1)nnn2C 23033,c1(CC(=O)NCC(CCOC)NC(=O)C(C)N2CCC2)cc(C)cc(F)c1 23034,c1(SCCNC(=O)NC(C)C2=CCCC2)ccc(Cl)c(F)c1 23035,C1(CC)C(NC(=O)C=C2CCC(C)C2)CCN1C(c1oc(C(F)(F)F)nc1C)=O 23036,C1(CC=C)(NC(=O)CCOCC2CCCO2)CCN(C(=O)C(C)=C2CCC2)CC1 23037,c1(NC(c2ccc(CCC(=O)NC3CC(O)C3)[nH]2)=O)ccc2nn(C(F)F)cc2c1 23038,Cc1cc(C(=O)NC2CC2NC(=O)Cc2c(C)cccc2C)cc(C(F)F)c1 23039,C1(C(C)C)C(=O)N2CCC(F)(C2)c2cn1nn2.n1(CC)cc(CC#N)cn1 23040,C(C(CCCC)N)N.C(C)(C(=O)C(=O)CSC(F)F)=C(CC)C 23041,CC(C)CCC(O)C(=O)N(C1CCN(C(=O)C(C)Cc2ccc(O)cc2)CC1)C 23042,N1(C(CCC(CC)NCCOC)=O)CC=C(C(C)(C)C(=O)NCC(C)CN(C)C)C1 23043,c1(NC(N2CC(C)(CC(=O)NCC=CCCC)C2)=O)cc2c(cc1Br)OCCO2 23044,c1(C(N2CC3C(C(=O)NCc4cn(C(C)C)nc4)(C3)C2)=O)cc(I)ccc1O 23045,c1(C(=O)O)ccc(S(=O)(=O)N2CCCCC2C(N2CCCC(F)CC2)=O)cc1 23046,C(=O)(C1CSc2ccccc21)NC(C1CC(NC(c2c(CC)nn(C)c2)=O)C1)C 23047,N1(C(C2COCC2C(N)=O)=O)CCOC(C(=O)NCc2cnn[nH]2)C1 23048,C(=O)(C(F)(F)CC(C)C)N1C2CN(C(C(C(=O)OCC)CC)=O)C(C2)C1 23049,C1(NC(C(CCC)C)=O)CCN(C(c2nc(C(C)C)ncc2NC)=O)CC(O)C1 23050,CC1(C(=O)NC2CCC(n3cc(-c4cncnc4)nn3)CC2)CCCC1O 23051,c1(C(=O)NCC2N(C(c3c(C)cncc3)=O)CCCC2)c(Cl)cccc1[N+](=O)[O-] 23052,c1(N(CC(Cl)Cl)C)nc(=NCC(C(F)F)N2CCOCC2)[nH]c2c1COCC2 23053,C1(CC(=O)NCCCC#C)CCCCN1C(c1c[nH]nc1-c1cccc(Br)c1)=O 23054,c1(CC)cnn(-n2cc(C=CCN3C(c4cn(CC)nn4)C(C)CC3)nn2)c1N 23055,c1(C(C)C)cc(Cl)nc(NC(=O)CN2CCN(CC(=O)N(C)C)CC2)n1 23056,C1(CNC(C(C)(C)SC(C)(C)C)=O)CN(C(=O)CCCC(F)F)CC1(C)C 23057,N1(C(C=C(C)C)=O)CCN(C(C2C3CCC2CC3)=O)CC1c1cccc(Cl)c1 23058,c1(C(=O)NC2(CN(C)C)CC3CCC2C3)nc2ccccn2n1 23059,c1(C(N2C3C(NC(=O)C4=CCCC4)C(C3)C2)=O)nccc2cccnc12 23060,C(CNC(=O)C=Cc1ncc[nH]1)(CCCC)NC(C1(CC#C)CCCO1)=O 23061,C1(CC(=O)N(C(c2ccccc2)C)CCSc2ccccc2)CCNCC1 23062,CC1=C(C(=O)N2CCN(C3CN(C(=O)Cc4csc(C)n4)C3)CC2)CCS1(=O)=O 23063,C#CCCCCCCC(=O)N(CCCCNC(=O)CC(CC)OC)C 23064,CC(CC(=O)NC1CCN(C(c2cc(N)c(O)c(F)c2)=O)CC1)P(C)(C)=O 23065,N1(C(c2ccc(C(=O)OC)o2)=O)CC(NC(=O)C(C)(C)Cc2cnn[nH]2)C(F)C1 23066,CC1=C(C)C(NCc2cnc(C3OCCO3)s2)CCC1 23067,c1(NCc2c(C)nsc2)nccc(N(CCS(C)(=O)=O)C)n1 23068,C12(C(N3CCCC(N(C(c4c(C)cc(SC)o4)=O)C)C3)=O)CCC(CC1)CC2 23069,C1(CCC(=O)N(CC(C(=O)NC)C)C)(NC(=O)CCc2cc[nH]c2)CCCCC1 23070,c1(CNC(C(CSC)n2cc(CNC(C3CCC3)=O)nn2)=O)c(C)ccc(C)c1C 23071,c1(CNC)ccc(C(N2CCCC(CNC(c3cccnn3)=O)C2)=O)cc1 23072,C(=O)(C1=NOC(C2(O)COC2)C1)NC(C)CCCNC(c1ccn(C(F)F)n1)=O 23073,N1(C(C2(CC#C)CCC2)=O)CCN(C(c2coc(-c3cccs3)n2)=O)CC(O)C1 23074,c1(OCC)c(-n2cc(COC(CCC(C)NS(C)(=O)=O)=O)nn2)cccc1F 23075,Cc1ccc([N+](=O)[O-])c(C(=O)NCC2CC2CNC(c2cc(N)c(Cl)cn2)=O)c1 23076,C1(NC(C2C(=C)CC2)=O)CN(C(c2nc(C3CC3)cs2)=O)CC1F 23077,C1(C)(NC(c2cc(OC)ncc2)=O)CCCN(C(=O)CCc2cncc(O)c2)C1 23078,C1(CNC(c2c(Cl)nc(OC)s2)=O)CCCCN(C(=O)C(C)C2CC2)CC1 23079,C1(CC(=O)NC2(C3N(C(C4(C#C)CC4)=O)CCC3)CC2)CCCC(=O)N1 23080,CCC(C)C(C(=O)NC(C)CNC(c1cccc(NC(C)=O)c1)=O)NC(=O)OC 23081,C1C(F)(F)CCC(=O)NCCCc2cn1nn2.c1(CSC)sc(C(C)C)nc1C 23082,c1(C(N(CCNC(CCC#C)=O)CCOCCO)=O)cc2c(s1)CC(C)CC2C 23083,C(=O)(CCC#Cc1ccccc1)NC1CC(NC(c2ccn3nncc3c2)=O)C1 23084,C1(NC(CCc2cc(OC)no2)=O)CCCCN(C(=O)CC2CC(OC)C2)CC1 23085,C1(C(=O)NCCCN(C)C(c2sccc2CC#N)=O)(COC)CC=CCC1 23086,CC1Oc2c(C(=O)NCC3CC(NC(=O)CC4CCCCC4)C3)cccc2C1C 23087,N1(CC(=O)NCc2ccccc2)CCN(C(C2C=CCCC2)=O)CC1 23088,Cc1c(C=CC(=O)NCC2CC(C)CN(C(=O)CC3CCC3(C)C)C2)cnn1C 23089,CCCCCC=CCNC(C(=O)OC)C1CC(N)C1 23090,C1(C)(CC)CCC(CNCc2nc(-c3ccccn3)cs2)O1 23091,C#Cc1cccnc1NC(=O)C(=O)N(C)CC1CC1 23092,N1(C(=O)NC(CC)CNS(C)(=O)=O)CC(=O)NCCNC(=O)c2ccccc21 23093,C(=O)(C(O)CC1CCCC1)N1CC(CC(C)NC(=O)C(C2CCCCC2)O)C1 23094,N1(C(C2(c3c(C)ncs3)CC2)=O)CC2(CCN2C(=O)CCCCNC(N)=O)C1 23095,CCCCC(O)CCC(=O)NC(CNC(c1ccc2nc(S)oc2c1)=O)C(C)C 23096,C1(C2(CC)CC2)CCN(C(=O)CN2CC(C)(C)C2)CC1.C12(CC=CC1)C(=O)N2 23097,N(C1CCc2c(Br)cccc21)C(c1cccc2nc[nH]c12)=O 23098,C1(C(N2CCC(C(=O)Nc3ccc(CC)c(Br)c3)CC2)=O)Cc2ccccc2C1 23099,c1(CNC(Cn2ncc(CC)c2)=O)cccc(C(=O)N(C)Cc2[nH]nnc2C)c1 23100,C1(C(N2CCC(OC)(CN)C2)=O)CC2(CCO1)CC2 23101,c1(C(C)NC(c2ccncc2Br)c2n(CCCOC)nnn2)ccc(F)cc1 23102,c1(OCCC(=O)NCC2CCCN2C(c2nn[nH]c2Cl)=O)ccccc1F 23103,CC1CCCC(C(=O)NCC2CCN(C(C3CC4CC3C4)=O)CC2)C1 23104,N1(C(=O)Nc2ccoc2C2CC2)CCC2(CC1)CC2c1cccnc1 23105,Cc1ncnc(C(=O)NCCN2CCN(CCOOC3CCOC3)CC2)c1C.O 23106,C1(NC(c2cnn(CC)n2)=O)CCC2(CC1)CC2NC(=O)CC1CCOC1=O 23107,c1(CC(=O)NC2COCC2NC(c2cc3n(c2)CCC3)=O)cnc2cccnn12 23108,S(=O)(=O)(c1c(C)sc(C)c1Br)NCc1c(OC(C)C)ccc(OC)c1 23109,C1(CC(=O)NCCCN(C(C)C)C(C2CCC2)=O)CCCC(C)(C)O1 23110,N1(CC)CCC(NC(=O)C(CC2CCC2)NC(=O)CSc2cn[nH]c2)C(C)C1 23111,O=C(C1=CC2(CCOC2)C1)NCC1(F)CCN(C(=O)Cc2n[nH]c(=N)s2)C1 23112,O=C(C1=CCCCCC1)NCC12CCC1CN(C(c1nncs1)=O)C2 23113,CC(CC(=O)NCC1(F)CCN(C(c2cnc(Cl)cc2N)=O)C1)C(C)(C)C 23114,C1(NC(c2cnc(C(F)F)s2)=O)CC(O)CN(C(=O)CCc2ccccn2)C1 23115,c1(C(=O)OC)cnn2c1CC(Nc1nn3cc(CC(C)C)nc3s1)CC2 23116,C(=O)(C(CC(C)C)C(C)C)NC1C(OC)CN(C(c2cc(C)cnc2C)=O)CC1 23117,Cc1ccccc1C1(C(=O)N(CCNC(C2(C)CC2C(F)(F)F)=O)CC)CCCC1 23118,c1(C(=O)NCC=CCNC(c2ccc(C(F)(F)F)cn2)=O)cccc2nsnc12 23119,C12(NC(c3ccc(CC)c(C)c3)=O)CCCC1N(C(C1CC1(C)Br)=O)CC2 23120,c1(C(N2C(CNC(C(N3CCC(O)CC3)C)=O)CCC2)=O)cnn2ncccc12 23121,C(=O)(C1Cc2ccc(F)cc21)NC12C(CN(C(CS(CC(=O)OC)(=O)=O)=O)C1)C2 23122,N1(C(c2cc(N)c(O)cc2F)=O)C=CCCC2CCCCC12 23123,C12(NC(c3c(C)c(F)ccc3)=O)CCCN(C(=O)Cc3cnn(C)c3)CC1C2 23124,C(=O)(C1=NOC(CNC2C3CCC(F)C23)C1)N(C1CCCNC1=O)C 23125,N1(C(CN(C(C2CCCC3CC23)=O)CC)=O)CCN(C)C(C(C)C)C1 23126,c1(C(N(C(C(C)Cc2cnn(C)c2)=O)C2CCCCC2)=O)c(Br)nnn1C 23127,C(=O)(C1=CC2C=CC1C2)N1CCN(CC(C)NC(C2=CCCC2C)=O)CC1 23128,C(F)(c1ccccc1)=CC(=O)NC(CNC(C(COC)OC)=O)CC(C)C 23129,Cc1ncncc1C(N1CC(NC(c2cnc(C(C)(C)C)[nH]2)=O)C(C)C1)=O 23130,C1(CCNC(CN2CCN(C(C(=O)OCC=C)C)CC2)=O)CC2CCC1CC2 23131,C(=O)(C(O)CC(C)(C)C)NCc1cccc(NC(Cn2c(C(F)F)cc(C)n2)=O)c1 23132,C1(NC(c2c(C)nns2)c2nnnn2C2CCOC2)CC2CC(O)C1C2 23133,Cc1ccc2c(c1)C(NC(N1CC(C)CCC1CO)=O)CCC2 23134,C(CN=c1cc(C)nc(-c2ccccc2)[nH]1)N(C(C(=O)NCC)=O)CC 23135,c1(C(=O)NC2(C)CN(C(C3CC3C(N)=O)=O)C2)c(F)cccc1Br 23136,N1(C(CC(C)C)=O)C(C(=O)Nc2cnccc2SCCN2CCCC2)CC2CC12 23137,CC(C)C(C(=O)NCCCCNC(=O)CCC1(C)N=N1)S(=O)(=O)C1CCCCC1 23138,C(=O)(C(F)(CNC(=O)Cc1ccc(C)c(O)c1)C(C)C)NC1CCN(CC)C1 23139,c1(NC)ccc([N+](=O)[O-])cc1C(N1CCC2(CCCN2C(=O)C=CCF)C1)=O 23140,C(C1=CCCNC1)NC(c1ccc(C(=O)Oc2ccccc2)cc1)=O 23141,C1(C(N(CCN(C(c2[nH]cc(CC)c2C)=O)C)C(C)C)=O)CC(=O)NC1(C)C 23142,CC1ON=C(C(=O)N2CC(NC(c3c(Cl)cnn3C)=O)C(C3CC3)C2)C1C 23143,c1(OC)ccc(F)c(F)c1CN1CC(NC(c2ccc(Br)c(CO)c2)=O)C(F)C1 23144,N1(C(CC(=O)NC)=O)CC(C)N(c2nc(C)ncc2C#N)CC1C 23145,C1(NC(C)=O)CCC(C(N2CCC(NC(c3cn(C(C)C)cc3C)=O)C2C)=O)CC1 23146,N1(C(C(OCC)OCC=CC(=O)NC)=O)CC2(COC(C)C2)C1 23147,c1(C(=O)NC(C)CCNC(c2c[nH]nc2-c2ccc(Cl)s2)=O)nnc(S)n1C 23148,N1(C(C=CC=CC)=O)CCc2ccccc2C1CNC(=O)CCc1scnc1C 23149,N1(C(c2ccc(CC)c(F)c2)=O)CC2CCCC2(NC(c2cc(Cl)c(Cl)[nH]2)=O)C1 23150,c1(SC)ccccc1CN1CCCC1CC(=O)Nc1ccc(F)nc1 23151,c1(NC(C(CC)(C)CNC(=O)C(C)SC(F)(F)F)=O)cnc2ccnn2c1 23152,C(=O)(C1=CC2CCCC12)NCCC1N(C(c2cccc(C(C)C)c2N)=O)CCC1 23153,N1(C(C(CC(C)C)C(C)C)=O)CCCC2(CCCN2C(=O)COCP(C)(C)=O)C1 23154,N1(C(C2(CNC(C(C)=NOCC#N)=O)CCCO2)=O)CC[Si](C)(C)CC1 23155,c1(CCCCOC(C)=O)c(-c2cncc(OC3CCC3)c2)ncn1C 23156,Cc1cccc(C(C)NC(=O)NC2(NC(=O)CCSC(F)(F)F)CC2)c1 23157,CC1=C(C(=O)NCC2CCCN(C(=O)CCCc3nccs3)C2)CCC(C)(C)C1 23158,c1(C(N2C(CNC(c3noc(CC)c3C)=O)C=CC2)=O)ccc(P(C)(C)=O)cn1 23159,C1(CCCCCNC(c2c(CC)cno2)=O)CCN(C(=O)C(C)=CC2CC2)CC1 23160,S(=O)(=O)(c1ccc(C#N)cc1)NC(C12CC(NC(c3cnc(C)nc3)=O)(C1)C2)=O 23161,N1(C(CSCc2ccc(C)cc2)=O)CC2CC(N(C)C(C3CCC(=O)N3)=O)C1C2 23162,c1(CC(=O)NC(CNC(C(C)OCCOCC)=O)CO)cc(C)no1 23163,Cn1nc(CN2CCC2Nc2ncccc2C(F)(F)F)c2c1CCCC2 23164,c1(NC(CC)CNC(=O)CCc2ccccc2F)ncc([N+](=O)[O-])cc1Br 23165,C(=O)(C1=CS(=O)CCC1)N1C(C(C)C)CN(C(=O)C(O)Cc2cnn(C)c2)CC1 23166,N1(C(CCc2nc(C)c(C)o2)=O)CCC2(NC(=O)NCCOC)CCCCCC12 23167,C(=O)(CC(C)COC)N(C)CC1CN(C(c2n(CCC)ncc2)=O)C1 23168,N1(C(CC(CCC)NC(c2oc(C)nc2C)=O)=O)CCC2(CCCCC2)C1 23169,CCC(CC(F)(F)F)C(=O)N1CC2CCN(C(=O)CCc3ccc(C)cc3)CC12 23170,c1(C(C)=O)ccc(CC(=O)N(C(C)CN(C(=O)CC2CCCC23CC3)C)C)cn1 23171,c1(C(=O)NCC(CNC(CC2(C=C)CC2)=O)(C)C)cc2sc(C)cc2[nH]1 23172,N1(C(c2cccc(OC)c2F)=O)CC2CCC1CN2C(=O)C=Cc1cccnc1 23173,CC1(C)CCC(CNC(C2(C#N)CCCC2)=O)N(C(C2(C)CCC(=O)NC2)=O)C1 23174,N1(C(c2nc(C(C)C)oc2)=O)CCn2nc(C(=O)Nc3ccccn3)cc2C1 23175,c1(C(=O)NCC2CC2C(=O)Nc2cncc(Cl)c2)ccnc(O)c1 23176,O=C(C1CCCn2c(Br)cnc21)NC12CC(C(=O)N(C)C)(C1)C2 23177,C1(NC(c2cn(CCNC(CC3(C)COC3)=O)nn2)=O)CCc2ncnn2C1 23178,C(C(=O)N=S(C)(C)=O)OCCC1CN(Cc2ccccc2)CC(CC(=O)OC)O1 23179,C#CCCCC(=O)NC1CCOC(C(=O)NC2CC3(CC3)C2)C1 23180,CCS(=O)(=O)CC(=O)N1CCC(N(C(=O)Cc2ccn(CCOC)n2)CCO)C1 23181,N1(C(c2ccc(Br)s2)C(=O)NC2(C)CC2)CCC(n2cnnc2O)CC1 23182,c1(C(=O)NC2C(NC(C3(C)CC4CC4C3)=O)CCCC2)cc2nn[nH]c2cc1F 23183,C1(C2CCCCC2)(C(N2CCCC(NC(c3[nH]cc(C)c3)=O)C2C)=O)CC1 23184,Cc1nc2sccn2c1C(=O)NC(c1ccc(F)cc1F)C(F)F 23185,c1(NC(CSC2N(C(CCCNC(=O)OC)=O)CCC2)=O)ccc(F)cc1 23186,C1(C(NOCCOC)=O)COCCN1C(=O)CC1CC(OC)C1 23187,N1(C(C2ON=C(C)C2)=O)CCC(C(=O)Nc2cnccc2C)C(C)(C)C1 23188,C(=O)(C(O)CC(N)=O)NCCCOCCC(N1CCC(=CCC)CC1)=O 23189,C(=O)(CCC(C)SCC)N1C(CC(=O)N(CCCC)CC(N)=O)CCC1 23190,Cc1ccc(C(C)NC(=O)C(C2(O)CCC2)NC(=O)CCCc2cnn[nH]2)s1 23191,c1(N2CC(O)(CNC(c3nn(C(CC)CC)c(C)c3)=O)C2)cc(O)nc(=O)n1C 23192,N1(C(C(c2ccc(C)o2)C)=O)CC(NC(c2onc(C)c2C)=O)CC(F)C1 23193,C1(CC)(CO)CCCN(C(=O)C(CN(C)C)NC(C2COCC(C)O2)=O)C1 23194,CC(C)CCC(C(=O)N1CCC(N(C)CCO)C1)NC(c1csc(C#N)c1)=O 23195,N1(C(CC(C)C)=O)CCN(C(=O)C(C)NC(=O)OC(C)(C)C)CC2(C)CCCC12 23196,C(CCC(C)C(=O)N1CC(O)(CNC(c2cccc(C3CC3)n2)=O)C1)OC 23197,C1(NC(C2(CC(C)=O)CC2)=O)CCN(C(=O)C(C)CCN(C)C)CC1C 23198,N1(C(c2cn(CCC)nc2)=O)C2CCC1C(CNC(=O)CC(C)n1ccnc1)C2 23199,CC1CCN2N=C(C(=O)N3CC(N(C)C(c4ccnn4CC4CC4)=O)C3)NC2=N1 23200,N1(C(=O)OC(C)(C)C)CC(CNCC2CC(C)(C)CO2)C(F)C1 23201,c1(CN2Cc3c(C(=O)OCC)n[nH]c3C2)cn2c(Br)cnc2s1 23202,N1(C(C(CC)N(CC)CC)=O)CCCC(C)(NC(=O)Cc2ccoc2C)C1 23203,N(C1CCCc2ccc(F)cc21)CC(CC)c1nn[nH]n1 23204,c1(OC(C)(C)C)nccc(=NC(=O)CC2CCCN(C(c3ccsc3C)=O)C2)[nH]1 23205,CC1(F)CC(C(=O)NCCCC(=O)NC2(C(N)=O)CC(O)C2)C1 23206,C(C1CN(C(=O)C(n2cc3c(n2)CCCC3)C)Cc2ccccc21)NC(C)=O 23207,N#CC1CN(C(=O)C=Cc2ccc(O)cc2)CCN1Cc1cc(Cl)ccc1Cl 23208,C1(CC)CN(C(C2CC(O)C(F)C2)=O)CC1C(=O)NCC(N1CCCCCC1)=O 23209,C1(C(=O)NCCN(C(CC(CC=C)(C)C)=O)CCC)CC12CCC1(CC1)CC2 23210,N1(c2nccc(C(=O)Nc3cccc(Cl)c3)c2)CC(C(=O)O)OCC12CCOC2 23211,C(=O)(C1=CS(=O)(=O)CCC1)N1CCN(C(Cc2cc(C)nc(O)c2)=O)CC12CC2 23212,C1(C(=O)NC2CCOC2C(N2CCCC2C(N)=O)=O)(COC)C=CCC1 23213,C1(NC(C(C)CCO)=O)COC2(C1)CN(C(=O)Cn1nc3c(n1)CCCC3)C2 23214,CC1(C)NC(=O)CC1C(=O)NCc1ccc(CNC(C2CC3(C2)CC3(F)F)=O)cc1 23215,c1(OC)ccc(NC(=O)C(=O)N2CC(CNc3sc(Br)nc3C)C2)c(OC)c1 23216,C1(F)(C(=O)NCC(C)N(C(C(c2cc(F)cc(F)c2)C)=O)C)CCN(C)CC1 23217,N1(C(C(C)OCC#C)=O)CC2CCC1C2NC(c1nn(C)c(Br)c1C)=O 23218,Cc1nccc(C(=O)NCCC2(C(=O)N(C3(CCO)CC3)C)CC2)c1N 23219,C#CC1(C(=O)N(CCCCN(C(=O)C(F)(F)c2cnn(C)c2)C)C)CCCC1 23220,C(=O)(C(F)C(=O)N1CC(F)CC1CC(=O)NC(CC1CC1)CC1CC1)OCC 23221,C(=O)(C1=C(F)CN(C(=O)CC(Cl)Cl)CC1)NCc1nn(C)c(CO)c1.N 23222,O=C(C#CC1CC1)NC1CC2(C1)CC2NC(C1CCCCS1)=O 23223,O=C(N=c1[nH]nc2n1CCCC2)N1CCC(Cc2cccnc2)C1 23224,CCCS(=O)(=O)CC(=O)N1CCN(C(=O)CCOc2ccccc2F)C2CC12 23225,Cc1cc(=NCc2cc(C3CC3)on2)[nH]c(N2CCc3ncncc3C2)n1 23226,c1(C(=O)NC(CC=C)CNC(c2ccc(CO)cc2)=O)c(F)ccc2n[nH]cc12 23227,N1(C(C2OCCCO2)=O)CCC(C2CCCN(C(=O)C3=CCCOCC3)C2)CC1 23228,N1(C(CC(CCC)C)=O)CC2CCC(N(C(=O)CCc3ncc(F)cn3)C)C2C1 23229,N=C1NC(=O)C(CC(=O)NCC2(CNC(=O)C(O)Cc3cnc[nH]3)CC2(F)F)S1 23230,C1(CNC(c2c(CC)ncs2)=O)C(O)C(O)CN1C(=O)CN1CCCC1=O 23231,CC12CC(C(=O)NC3CC(O)CN(C(=O)Cc4cnc[nH]4)C3)(C1)C(C)(C)O2 23232,C(=O)(C#CC1CCOCC1)N(CC(C)NC(C1CCC(CC(F)(F)F)CC1)=O)C 23233,C1(C)(C(N(CCNC(C=CC)=O)Cc2ccc(Cl)nc2)=O)CC(OC)CN1C 23234,c1(C(N2CC(NC(c3ccc(CC)[nH]3)=O)C(C)CC2)=O)ncn2c1COCC2 23235,C1(CNC(C(Br)=C(C)C)=O)CC2(CC2)CN1C(C1CC(C2CC2)=NO1)=O 23236,c1(C(N(CC(C)NC(C(CSC)C)=O)C)=O)cc2ccc(Cl)cc2c(O)n1 23237,N1(C(C(c2ccc(C)cn2)(F)F)=O)CCCC(NC(c2ncoc2C)=O)C1C 23238,C1(CNC(c2c(C)[nH]cc2)=O)CN2CCCCC2CN1C(c1ccoc1Cl)=O 23239,c1(C(N2CCC(OCCNC(C(COC)C)=O)C2)=O)cc(O)ccc1C 23240,c1(C(=O)NC2CCN(C(C(CC)NC(N)=O)=O)CC2F)cc2n(n1)CCNC2=O 23241,N1(C(C(=O)NC(C)(C)C)C2CC2(Br)Br)CCCC(C2CCC2)C1 23242,c1(C(=O)NCC2(F)CC(NC(C3CCSC3)=O)C2)cccc(CC(F)(F)F)c1 23243,CC1=NNC(=O)C1CC(=O)NCC1(CN(C)C(c2ccn(CC(C)C)n2)=O)CC1 23244,C(=O)(CCCCC(C)(C)C)N1C(C)CC1C(=O)NCC12CC(C)(CCO1)C2 23245,C(CCC(=O)N1CC(O)(CN(C(=O)C(F)CC2CCCC2)CC)C1)=CCC=C 23246,C1(C(CC)CC)CN(C(=O)C=CC(=O)N(C)C)CCN1C(=O)CNC(=O)OC 23247,CC1CCCN1C(=O)Cn1cc(C2CCCC2O)nn1 23248,C=CC12CN(C1)C(=O)C(CC)COC(=O)C(C)N(C)C(=O)C2.C(C)(=O)OC 23249,N(C(=NCCc1ncnn1C)NC1CCCC1)C(c1ccccc1Br)C 23250,n1(CCOC)cc(C(=O)N(CCCNC(C2(C)CC2F)=O)CC2CCCC2)cn1 23251,c1(N2CCC3(CC(NC(C4(O)CCSC4)=O)C3)C2)nc(Cl)nc2[nH]c(O)nc12 23252,C1(N(C)C(c2coc(CC3CC3)n2)=O)CC2CC1N(C(C1(C)CC=CCC1)=O)C2 23253,c1(C(=O)NC2(CO)CCN(Cc3cn[nH]c3)CC2)c(O)ncc2c1CCC2 23254,N1(C(C(CCSC)(C)C)=O)CC2ON=C(CNC(c3coc(C(F)F)n3)=O)C2C1 23255,c1(C(N2C(C(=O)NC(CCC)C3CCCCC3)C(C)C2)=O)ncc(C)cc1F 23256,Cc1nscc1CC(=O)N(C1CCC(NC(=O)COC(C)C)C1)C 23257,c1(N2C(C)C(NC(=O)CC3(O)CC3)CCC2)ncc2ccnc-2[nH]1 23258,N1(C(C(C(C)(C)O)(F)F)=O)CC2CN(C(c3ccsn3)=O)CC(C1)O2 23259,c1(SCC)cccc(C(=O)NC2(C)CCN(C(c3nnc(S)n3C)=O)C2)c1 23260,CC(C(O)C(F)F)NC(=O)C=CC(C)NC(=O)CC1NC(=O)NC1=O 23261,C(C1=CCCSC1)(c1nnnn1-c1ccc(Cl)cc1)NCC(C(C)C)C(C)C 23262,C1(n2nnc(C(F)(F)F)n2)(OCC)CCOC(Cc2ccc(C)cc2Br)C1 23263,N1(C(C(C)n2ccnn2)=O)CCC(C)(C)C1CNC(=O)COCc1cccnc1 23264,N1(C(COC)=O)CC2CCCC(NC(C3CCC=CCC3)=O)(C2)C1 23265,N1(C(C(CC=C)C(C)C)=O)CC2(CCN(C(c3cc(C)ns3)=O)CC2)CC1C 23266,N1(C(C(C)=C2CCC2)=O)CC2CCN(C(=O)COc3cc(C)ccc3F)CC2C1 23267,c1(NC(C(C)NC(c2coc(C3CC3)n2)=O)=O)cccc2c1OCC2 23268,C(CC(C)(C)CC(=O)NC(CC)CCC(=O)Nc1ccc(O)c(Cl)c1)OC 23269,C1(C(=O)OC)CCCOC12CCN(C(c1ccc(C)c(F)n1)=O)CC2.C=CC 23270,CC1(C)CC(C(=O)NC2(C(=O)NCC3CC(CF)C3)CCSC2)CCO1 23271,c1(OCCOC)ccc(Cl)cc1C(=O)NCC1CN(C(=O)C(O)CF)CCO1 23272,CC(C)C(C)CC(=O)N1CC(C)CCC1C(=O)NCc1nncn1C1CC1 23273,c1(OC)nccc(Br)c1C(=O)N(C)CCNC(C1CCSC(C)C1)=O 23274,N1(c2c(C(=O)OC)cc(Br)cc2)Cc2[nH][nH]c(=NC(=O)c3ccnc(F)c3)c2C1 23275,c1(C(N2CCC(OCCNC(CCC#CC)=O)C2)=O)cc(C)c(O)c(C)c1 23276,c1(C(N(C)CC2N(C(c3cn(CC)nn3)=O)CCC2)=O)[nH]c(C)c(C)c1C 23277,CCCCC(CNC(=O)CCSc1ccccc1)NC(=O)CCC1CCCN1C 23278,C(=O)(C1=NNC(=O)CC1)NC1CN(C(C(CC)CC)=O)CC(C(F)(F)F)C1 23279,C1(O)(CC(=O)OCC)CCN(C(=O)C(O)Cn2cncn2)CC1 23280,C1(CC#C)(C(=O)NC=O)CCCCO1.N12CCN(CC1)c1nc(ncn1)CC2 23281,CC1=C(C(=O)N2CCCC(NC(c3cc(F)ccc3Cl)=O)C2C)CCC1 23282,c1(NC(C)=O)cccc(C(=O)NC(C)CCNC(=O)Cc2cc(C)no2)n1 23283,c1(OCC)ncccc1C(=O)NC(C)CNC(c1cnn(CC2(O)CCC2)c1)=O 23284,C(CO)(CCCCNC(=O)C(O)Cc1cnc[nH]1)NC(CN1CC(C)(OC)C1)=O 23285,C(C(CC1CC1)C(=O)NOCC1CCCO1)NC(c1c(OC)ccs1)=O 23286,c1(CN2CC3CN(C(C=CC=CC)=O)C3C2)cc(F)cc(F)c1O 23287,CC1(NC(=O)CCC2CCOCC2)CCCN(C(c2ccnn2CC(F)F)=O)C1 23288,c1(C(=O)NCC2(O)CN(C(C(C)NC(CC)(C)C)=O)C2)cc(Br)cn1C 23289,CC1CCCC=C1C(=O)NCC1(O)CCCN(C(c2cc(C3(C)CC3)n[nH]2)=O)CC1 23290,c1(CCC(=O)NCCN(C(=O)CN2CCC(C)C2)CC)cnc(O)[nH]1 23291,c1(OC)cccc(C(=O)NCC2(NC(C3CC3F)=O)CCOCC2)c1[N+](=O)[O-] 23292,C1(CNC(C(C)SCCCC)=O)CN(C(c2ccsc2Cl)=O)C2(CCOCC2)C1 23293,C(=O)(CCC(C)(C)NC(=O)Cc1ccccc1C)NCCCC(=C)Cl 23294,c1(C(=O)OCCC(=O)Nc2ccc(OCC)cc2C)cnc2ccccn12 23295,N1(C(C(C(C)C)CNC(C2(C)CC3CC3C2)=O)=O)CCCOC(C)(C)C1 23296,C1(CC)CCC(C)CN1C(c1c[nH]nc1CNC(c1coc(C)n1)=O)=O 23297,C1(N(C(=O)CCc2cn[nH]c2)C)CCCN(C(=O)C(C)(C)c2ccccn2)CC1 23298,C1(O)(CC)CCC(NC(=O)CC(C)(C)CNC(C2CCCOC2)=O)CC1 23299,N1(C(CCNC(N)=O)=O)CCC(NC(=O)CN2CCCC(C(N)=O)C2)C(F)C1 23300,CC1CCN(C(=O)CC=CC(C)(C)C)C1CNC(c1cncc(F)c1)=O 23301,c1(C(=O)NCCC2CCN(C(C3CC34CC4)=O)C2)cc(C2CC2)nnc1O 23302,c1(NCC2C(NC)COC2)cncc(C(=O)Nc2ccccc2)c1 23303,C(=O)(C#CC1CCOCC1)NC1CCC(N(C(CCC=C)=O)C)C1 23304,N1(C(C(C)NC(COC)=O)=O)CC2CC1C2CNC(C1(C)CC1(F)F)=O 23305,c1(-c2nc(Cc3ccc(C)nc3)n(C3CCS(=O)(=O)C3)n2)ccc2nc[nH]c2c1 23306,c1(C(N2CCN(C(C(n3ccc(C)n3)C)=O)CC2CO)=O)ccc(O)c(C)c1C 23307,C1(OC(CC2CCCC(C)C2)=O)COc2ccccc2N(C)C1=O 23308,n1(C)cc(C(=O)N(C2CC2)NC(COCCCOC)=O)nn1.C1(C)CCOC1 23309,C(=O)(C1=NOC2COCC12)NC1C(n2cc(-c3cncc(C(C)C)c3)nn2)COC1 23310,CC1(C)CN(C(C2CC2NC(c2cnc(O)nc2O)=O)=O)CCO1 23311,C1(SCC)COC2(CCCC2)O1.N12C(=O)CC(C1c1cccc(C)c1)CN1CCCC21 23312,C1(C(N(CCCC)CC)=O)CN(C(C2CCCOC2)=O)C(C)(C)C1 23313,C12(OC)CCC(C(N3CCC4C(C(=O)OC)CC34C3CC3)=O)(CC1)CC2 23314,c1(C(=O)NC2CCCN(C(CSCCC)=O)C2C)ccn2ccnc2c1 23315,C(=O)(C(O)(C(C)C)C(F)(F)F)NC1CC(NC(C=C(C)Cl)=O)C1 23316,c1(C(N(C(CNC(c2nc(C(C)C)oc2)=O)C)C)=O)cc2c(cn1)OCCC2 23317,c1(C(C(=O)NCCOCCC#C)NC(=O)COCC(C)C)cccnc1 23318,C(=O)(C(CC(F)F)NC(c1cc(C)cnn1)=O)NCCCOC 23319,N1(C(C(C)C)=O)CCN(C2CCC(NC(=O)C(N3CCC(C)(O)C3)=O)C2)CC1 23320,c1(C(C(=O)NC(CCOC)CNC(c2cc(C)sn2)=O)C)cccc([N+](=O)[O-])c1 23321,N1(C(Cc2nc(=N)[nH][nH]2)=O)CCC(NC(C2CC2F)=O)C12CCC2 23322,C1(NC(C2N(CCC(C)C)CCC2)=O)CN(C(=O)Cn2nccn2)CC1CO 23323,C(=O)(C1SCCc2ccccc21)NCCN1CCN(C(CN(C)CCO)=O)CC1 23324,C1(NC(C=CC(C)(C)NC(C2CC2C(N)=O)=O)=O)CC2(C1)CC(C#N)C2 23325,C(=O)(CC(F)(F)C(F)F)N1CCC(NC(c2cc(COC)oc2C)=O)C(F)C1 23326,C(=O)(C(O)(C(C)C)C(F)(F)F)NCC(C)NC(Cc1c(C)ccnc1)=O 23327,C1(CCC)CN(C(C2(C(C)NC(=O)C(O)C3CC3)CC2)=O)C1 23328,CC1CC(NC(c2cccn2C)=O)CN1C(C1CC1C)=O 23329,C1(CNC(CCNC(c2cccc(C)c2)=O)=O)CCC12CCN(C(=O)CO)CC2 23330,c1(NC(=O)CC2CN(C(=O)CN3CCOC3=O)C2)cnc2ccccc2c1Cl 23331,Nc1cncc(C(=O)NCC2CCCCN2C(=O)CCCn2ccnn2)n1 23332,C1(C(=O)NCC(C)(C)NC(=O)Cn2nccn2)CS(=O)(=O)CC12CC2 23333,Cc1c[nH]cc(C(=O)NCC(C2CCC2)NC(c2ccc(CO)cn2)=O)c1=O 23334,C1(N(C(Cc2ccc(C)o2)=O)C)CN(C(=O)C=CCOc2ccncc2)CC1F 23335,Cc1cc(C(N2CCN(C(c3ccc(Br)c(O)n3)=O)C3CC23)=O)nc(C)c1 23336,Cc1cnc2n1CC(C(N1CCCOC(CNC(C3CCSCC3)=O)C1)=O)CC2 23337,N1(C(CC)=O)CCC(n2nc(-c3cccc(N)n3)nc2-c2cnnn2C)CC1 23338,c1(C(=O)NC2CN(C(C(c3cccc(C)c3)(C)C)=O)C2)ccc(F)c2[nH]ccc12 23339,c1(C(=O)NC(C)CC(N)=O)cccnc1CNC(c1nn(C)cc1Cl)=O 23340,CN1CC2C(C(=O)NC3(CC(=O)N(C)CC4CCCC5CC45)CC3)C2C1 23341,C1(C(=O)NC(CN(C(C2CC(OC)C2)=O)C)(C)C)CCCCO1 23342,c1(OC)cc(OC)nc(N2CC(NC(C3(C)CCCOC3)=O)CCC2C)n1 23343,c1(OC)cccc(CC(N2CCCC2(C)c2cccc(F)c2)=O)n1 23344,N1(C(C2(OC)CCSC2)=O)CCC(C)C(CNC(=O)C(c2cccs2)C2CC2)C1 23345,N1(C(c2cnn(C)c(=O)c2)=O)CC(C(N2C3C=CCC2CC3)=O)CCC1(C)C 23346,CCCCC(C(=O)N(C)CCN(CC(C)(O)COC)C)N1CCCS1(=O)=O 23347,CC(F)(F)CCCC(=O)NC(CNC(C1OCC1(C)C)=O)CO 23348,C1(CC)CCCN(C(=O)CC(C)(C)OC)C1.C12(CCC1)N(C1CC1)C2=O 23349,C(=O)(CCCCCc1ccccc1)NCC(CNC(C(C)CN1CCCC1)=O)O 23350,NC(=O)CCC(=O)NCC1(C(=O)NCc2ccccc2F)CCCO1 23351,CC1(C)CCC(CN)CN1C(N)=O.n1(CC(=O)C(=O)N)cc(CC(C)(C)C)nn1 23352,CC(C)CCCC(=O)N1CCCCC1CCN(C)C(c1cc(CC(C)C)c[nH]1)=O 23353,CC(C)(F)CCC(=O)NCC#CCNC(c1cccc(Cl)c1O)=O 23354,N#Cc1ccccc1C=CC(=O)NCC1(NC(c2n[nH]cc2F)=O)CCOC1 23355,Cc1cc(C#N)nc(NCCN(C(c2ccncc2F)=O)C2CC2)n1 23356,C1(C(=O)NC(C(=O)NCC)CC2CC2)CCN(C(=O)CCC(=O)OC)CC1 23357,CCC(CC(F)F)C(=O)NC(C)(C)CNC(=O)C(C(C)C)NS(=O)(=O)C1CC1 23358,C1(NC(CCCCC)=O)CN(C(c2ccc([N+](=O)[O-])c(C)n2)=O)C2CCCCC12 23359,c1(C(c2n(CCC)nnn2)NCc2ccc(C)c(Cl)c2)cc(F)cc2c1CCC2 23360,Cc1ccc(Cl)c(C(N2CC3(CCC3)CC2CNC(C2(CF)CC2)=O)=O)c1N 23361,c1(OC)cnc(Cl)cc1C(=O)NC1(CO)CN(C(C2CCC(=O)N2C)=O)C1 23362,C(=O)(C(C)(C)N(C)CCN1CCCC1)N(CC(CNC(C(C)NC(N)=O)=O)O)C 23363,N1(C(COCCSC)=O)CCOCC(NC(=O)C(n2cnc(C#N)n2)C)C1 23364,c1(NCC2CCCC2c2ccc(N(CCN(C)C)CC)cc2)nc(O)sc1C 23365,C1(C(=O)NCCN(CCC)C(c2nccnc2Cl)=O)CCC(C)(CC)O1 23366,c1(N2CC3N(C(=O)CC4CCC5CC5C4)C(CC3)CC2)nc2ccc(F)cc2s1 23367,C1(C(=O)NCCCN(C(CC)C)C)CCCN(C(c2cn[nH]c2)=O)C1 23368,CC(CC#N)C(=O)N1CC(=C(F)CNC(=O)Cn2cc[n+](C)c2)C1 23369,C(=O)(CC1=CCN(C)CC1)OCC.CC1CS(=O)(=O)CCN1C(=O)COCC 23370,N1(C(CC2(C)CCCO2)=O)CCCN(C(C2CCC3(C(=O)C4CC4)CCC23)=O)CC1 23371,C1(C(=O)OCC)CN(C(c2ccc(-c3nnc(C)o3)cc2)=O)CCO1 23372,c1(CN(C(C)C)C(=O)NCC2CC(O)C2)ccccc1.C1(C)CCCO1 23373,Cc1sc(=O)n(CCC(=O)NCC2CC2NC(=O)CN2CCCCCC2)c1C 23374,Cc1nc2cncc(C(=O)NC3CCN(C(=O)C(C)(F)C(C)(C)F)CC3)c2[nH]1 23375,C=CC(C)(C)C(=O)Nc1cccc(CNC(c2ccnn2CCC(F)(F)F)=O)c1 23376,c1(OC)c(C)cc(-c2nnc(CNC(=O)NC3CCCC(SC)CC3)o2)cc1Cl 23377,C1(CCOC)(NC(=O)CC2(O)CCOCC2)CCN(C(=O)CC2CCOC2=O)C1 23378,c1(ONC(C2CC(N(C(C(C)OCCOC)=O)C)C2)=O)cc(C)ccc1C 23379,N1(C(Cc2cn(CC)nc2)=O)C2CC1CN(C(C1CCCN1C(C)C)=O)C2 23380,c1(C(N(CCNC(C2C(COC)C2)=O)C)=O)cccc(Cl)c1O 23381,c1(C(=O)NCC2CCCN(C(c3ccon3)=O)CC2)c[nH]c2ccc(Br)cc12 23382,c1(COC)ccccc1CC(=O)NC(C)CNC(=O)Cc1cc(C)nn1C 23383,c1(N(CC(C)C)C(=O)NC(C)(C)C2CC2)cccn(O)c1=O 23384,c1(C(N2CC(SC)C(NC(=O)C(O)C(C)C)C2)=O)cc(S(N)(=O)=O)cnc1C 23385,N1(C(C(C(CC)C)OC)=O)C2CCC1CN(c1ncnc(Cl)c1OC)CC2 23386,C(=O)(C(C)(C)c1cscc1Br)N1CC(CCNC(C)=O)C1 23387,C(=O)(CC1OCCc2sccc21)N(CCCNC(C1CC2C(C1)C2(C)C)=O)C 23388,Cc1csc(C2CCCN2C(=O)CCCOCCN)n1 23389,c1(OC)cccc(-c2cn(CC(C)(C)CNC(=O)C(C)CC3CCC3)nn2)c1C 23390,N1(C(COCCNC(Cc2n(C)nnc2)=O)=O)CC2CC2C2CC12 23391,n1(CCCC(=O)NCC2CC2)ncn(C)c1=O.N12CC(C1)C(=O)NC(C)C=CC2=O 23392,C(=O)(CCC(CF)CF)N(C)CC1CCN(C(C2(C(C)(F)F)CCC2)=O)C1 23393,N1(C(c2occc2C2CC2)=O)CC2C3CCC(C2C1)N(C(=O)CCSC(F)(F)F)C3 23394,N1(C(C2C(C(C)=O)CCC2)=O)CCC2(CCN(C(c3sncc3C)=O)CC2)C1 23395,c1(CC(N2CCC(C3N(C(C=C(C)C(C)C)=O)CCC3)C2)=O)ccc(F)cc1Cl 23396,Cc1cc(Cl)cc(C(N2CCCOC(CNC(C3CC4(CCC4)C3)=O)C2)=O)c1C 23397,c1(C(C(=O)NCC=C)N(C2CC2)CC2CCCC2)ccc(CC(C)C)s1 23398,C1(CNC(C(C(C)OC)O)=O)(NC(=O)Cc2ccc(F)cc2)CCC(F)(F)CC1 23399,N1(C(C(C)(C)OC)=O)CC2CS(=O)(=O)CC2(NC(c2ccc3cccnn23)=O)C1 23400,N1(C(c2[nH]cc(C)c2)=O)CCOCC(NC(=O)C(C)(C)CF)C1 23401,CCS(=O)(=O)CC(=O)N1CCN(C(=O)CC2C=CS(=O)(=O)C2)C(CO)C1 23402,c1(C(C(=O)N(C(C(=O)NCC2(COC)CC2)C)C)O)cncn1C 23403,C1(CC(=O)N(CCCNC(C2CC2F)=O)C(C)C)COCCO1 23404,C1(CC)CN(C(=O)CCC(F)F)CCC1NC(c1nc(-c2ccccc2)sc1C)=O 23405,C1(CNC(CC(n2c(CC)ncc2)C)=O)CC2CCC1N(c1ncnc(=N)[nH]1)C2 23406,C1(O)(C(=O)NCC(C)CNC(=O)C(n2ccc(C(F)(F)F)n2)C)CCCCCC1 23407,C1(CC(=O)Nc2c(CC)noc2C)CN(C(=O)Cc2ncoc2C)CCC1C 23408,c1(CN(c2ccnn2C)C(C2C(COC)CNC2)=O)ccc(O)cc1Cl 23409,CCCC(C(C)(C)C)NC(=O)CC(C)(C)NC(=O)CCOC(C)=O 23410,c1(CC)ccccc1OCC(N1CCCC1CNC(=O)C(C)(C)c1cnco1)=O 23411,CCCC(C(F)(F)F)NC(C1CCCC(NC(c2cc[nH]c2)=O)C1)=O 23412,C12CCN(CC1)C(=O)C1(CC1)C(=O)NCCO2.C1(CC)CCNC1=O 23413,c1(C(N(CC(CNC(c2ccc(CC)[nH]2)=O)O)C)=O)ccc(NC)cc1Cl 23414,N1(C(c2ccc(CC)nc2)=O)CC2(C=C(C(=O)N(CCF)CCOC)CO2)C1 23415,C1(CNC(CC(=C=C)C)=O)CC(NC(c2onc(C)c2C)=O)C12CCC2 23416,c1(C(N2CCC(N(CC)CC)C2)=O)n[nH]c2c1CN(C(=O)CCCC1CC1)C2 23417,Cc1cc(C(=O)N(CCC(C(C)C)NC(=O)CC2CCCO2)C)c(C)nc1C 23418,O=C(CC1CCc2ccccc21)NC1COC2(C1)CN(C(C13CC(CO1)C3)=O)C2 23419,CC1CCN(C(=O)C(F)CC2CC2)CCN1C(=O)CC1NC(=O)NC1=O 23420,c1(C(=O)NC23CC(NC(C4C(CC)C4)=O)(C2)C3)cc(F)cc(F)c1N 23421,CC(C)CS(=O)(=O)CC(=O)N1CC(NC(=O)CCc2cscn2)CC1(C)C 23422,Cc1cccc(-n2cc(-c3c(C)noc3C)nn2)c1O 23423,c1(CNC(CCC2N(C(C(CCC)F)=O)CCCC2)=O)cn2cc(C)ccc2n1 23424,CC1CN(C(=O)CC2CC(C)(C)C2)CC(C)C1NC(c1cccc(N)c1O)=O 23425,C=CCC(F)(F)C(=O)N(CC(CC)NC(c1ccc(Cl)cc1Cl)=O)C 23426,C(=O)(C#CC1CCOC1)N1C(CC)CN(C(c2cc(N)cnc2C)=O)CC1 23427,CCCC(C(=O)OC(CC)C(=O)Nc1ccc(OC(F)F)cc1)c1ccccc1 23428,N1(C(C2(N(C)C)CCC2)=O)CCCC(CNC(=O)CCc2cnco2)C1 23429,c1(NC2CCN(C(c3nc(C(N)=O)sc3)=O)C2)ncc(Cl)cn1 23430,C1(N(C(CCN(C(=O)C(C)N2CCCC2)CC=C)=O)C)CCCC(C)(C)C1 23431,c1(NC(C(N2CCC(CO)CC2C)c2sc(C(=O)OC)c(C)n2)=O)c(C)cccc1C 23432,O=S(=O)(c1ccc(NCC2=CCCC2)cc1Br)NCc1cscc1Br 23433,N1(C(C#CC2(C)CC2)=O)CCC2CN(C(c3snc4ccccc34)=O)CCC12 23434,c1(CNC(C2(N(C(C3CC(C)OCC3)=O)C3CC3)CCC2)=O)cc(F)ccc1O 23435,c1(C(C2CC(C)(NC(CNC(C(C(CC)C)C)=O)=O)C2)=O)cc2cccnc2[nH]1 23436,CCCC(C)(C)C(=O)NCCC1(C)CCN(C(c2cn(C(C)C)nn2)=O)C1 23437,CN1CCCN(C(c2cscc2Br)C(=O)NC2CC2)CCC1 23438,C12CCCC(C1)NC1(CC1)C(=O)N2CC(=O)OC.c1(CN(C)C)ccccc1 23439,Cc1oc(Br)cc1C(N1CCC(O)C1c1ccc(F)cc1)=O 23440,C(C)(C(C(=O)NCC(N1CC(C)C1)=O)N(C)C)OC.n12cc(nn1)CC(C)C2 23441,c1(NCc2nccc(C)c2F)nc(N2CC3CCC(CC3)C2)nc2ncn(C)c12 23442,S(=O)(=O)(c1cnc(N2CCCC(CS(N)(=O)=O)C2)c(Cl)c1)NC1C(OC)COC1 23443,c1(C(=O)NCC(C)N(C(=O)CNC(N)=O)C2CC2)cn[nH]c1 23444,O=C(NNC(=O)C(O)c1cn2ccnc2s1)C1CCCC1c1ccc(F)cc1 23445,N1(C(CC2C(C)(C)C2)=O)CC(C2(NC(c3cccc(OC(F)F)n3)=O)CC2)C1 23446,c1(C(N2CC(NC(c3ccc(CC)cn3)=O)(COC)C2)=O)ccc2occc2c1 23447,c1(C(N(C(C)CNC(=O)C(C)C2CC2)C)=O)cc(Cn2cccn2)cnc1O 23448,N1(CC2CN(S(C)(=O)=O)C2)CCC(c2nc(-c3ccccc3)no2)CC1 23449,C(=O)(C#CC1CCOC1)N(CCNC(CCCN1C(=O)CN(C)C1=O)=O)C1CC1 23450,C1(OCc2ccccc2)CCN(N2CCOC3CCCCC23)C1 23451,CC(N=c1[nH]c(=NCCC2(C(F)(F)F)CC2)[nH]c2ccccc12)c1nncs1 23452,CC(C)(O)C(F)C(=O)N1CCOC(CNC(c2ccc(-c3ccco3)[nH]2)=O)C1 23453,c1(OC)cc(C2CCN(Cc3cncc(C)n3)C2)ccc1C 23454,N1(C(c2cnc(C)o2)=O)CC2CCCC2C1C(=O)NCC(O)CF 23455,C(CCSC)(C(=O)NCCC1(NC(=O)CC2CSCCS2)CC1)OC 23456,c1(C(=O)NCC(C)NC(=O)CN(C2CCSC(C)C2)C)ccc2c(n1)CCC2 23457,c1(NC(C(C)NC(c2ccc(CO)cc2)=O)C)ccn2nccc2n1 23458,CC1(C)CN(C(c2cnns2)=O)CC1NC(=O)CNC(C1CCCC1)=O 23459,C1(C(=O)NCC#CCOC)(CNC(C2CCC(C)(C)C2)=O)CC12CCC2 23460,C(=O)(C1=NOC(CNC(c2cccc(CC)c2)=O)C1)N(CC(=O)NCCC)C 23461,N1(C(CC2(CSC)CC2)=O)CCCC(C)(C)C1CNC(c1ccc(C)c(F)c1)=O 23462,N1(C(C(CC#C)C)=O)CC2CCC(C1)N2C(=O)CC(C)(C)COC 23463,c1(N2CCCCC(NC(C(C)NS(CC)(=O)=O)=O)C2)cc2nnc(CO)n2cn1 23464,C(=O)(C1=CCC(F)(F)CC1)N(CCCNC(C1(COC)CCCOC1)=O)C(C)C 23465,c1(C(N2CC(CC(C)NC(=O)C(C)(F)F)C2)=O)ccc2nc(CO)[nH]c2c1.C(F)(F)F 23466,C1(C(N2CCC(F)(CNC(c3nn(C)c(O)c3)=O)CC2)=O)CC2CCCCN2C1 23467,C1(=O)C(CCC(N)=O)n2cc(nn2)C2COCC2N1.C(CC(=C)C)=CC=C 23468,Cc1cc(Cl)nc(N)c1C(N1CCC2CC1CN2)=O 23469,c1(OC(CC)C)ccc(-n2nc(-c3nccs3)nc2C(C)CC)cc1 23470,C1(C(N2C(CCNC(COCCCCC)=O)CCC2)=O)CCc2nncn2C1 23471,Cc1cc(C(F)F)ccc1-c1cn(CC2CCN2C(c2c(C)nsc2C)=O)nn1 23472,N1(C(C(C)OCCOCC)=O)CC2ON=C(CNC(c3cnn(C)c3)=O)C2C1 23473,C1(NC(C(n2cc(C)nc2)C)=O)CN(C(=O)C=Cc2ccoc2)CCC1CO 23474,Cc1nn(C)c(C)c1C(N1CCCC1CNC(C1CCC(=O)N(C(C)C)C1)=O)=O 23475,C(=O)(C(CC(C)C)N(C(=O)CN1CC(=O)NC1=O)C)NCc1c(C)non1 23476,CCC(C(=O)N1CC(C)(C)C1C1CCN(C(=O)COC(F)F)CC1)C(C)(C)CC 23477,N(C1CCc2ccc(Cl)nc21)CCC1(C)CCCC1 23478,n1(CC)cnc(C(N2CC(CCO)(NC(c3cnn(C(C)C)c3)=O)C2)=O)n1 23479,CCC(C)(C)C(=O)C(=O)N1CCCC1CC(=O)NCC1CC1(C)C 23480,N1(C(CC(OCC)OCC)=O)CC(NC(c2ccc(Br)nc2Br)=O)C(C#N)C1 23481,S(=O)(=O)(c1c[nH]c(=N)c(C)c1)NCCCc1cn(CC2CCC(OC)CC2)nn1 23482,CC(C)S(=O)(=O)CC(=O)N1CCCC(CCC(=O)N(C)C)C1.C1CCC(=O)N1 23483,C1(C(N2CCC(NC(=O)CCF)C23CCCC3)=O)CC(c2ccccc2F)=NO1 23484,N1(S(c2c(C(C)(C)C)n[nH]c2)(=O)=O)CCN2C(=O)OCC2C1 23485,Cc1cncc(CCC(N2CCCC2c2cn(C3CCCC(C)C3)nn2)=O)c1 23486,C1(C(=O)NC(CC(C)NC(c2cn(CCC(C)C)nn2)=O)C)CCC(C(N)=O)CC1 23487,c1(C(C)C)ccc(N)c(C(N2CC(C(N)=O)(CNC(=O)CC(C)C3CC3)C2)=O)c1 23488,N1(C(CC=CC=C)=O)CCC(F)CC1C(=O)NCC(C)C(F)F 23489,C1(C)(C(N(C(CNC(=O)Cc2ccccc2)C2CC2)C)=O)CCCN1C 23490,N1(C(COCCCC#C)=O)CCC(NC(C2CCC(=O)N2CC)=O)C1(C)C 23491,C(=O)(CC(C)(C)CCOC)NCC(CNC(c1cccc(C(=O)OC)c1C)=O)F 23492,c1(NC(C)=O)c(C(=O)NCC2COC(CNC(=O)Cc3ccoc3)C2)cccc1C 23493,C1(NC(=O)CCC2CCOC2)CCC(NC(=O)CCCn2ccnc2)C1 23494,C1(NC(C2CCc3nncn3CC2)=O)C2CC3CN(C(=O)CC(F)F)C1C3C2 23495,c1(C(=O)NOC2CCN(C(c3ncc[nH]3)=O)C2)cnn(C2CC2)c1 23496,c1(NC(C2CC23CN(Cc2scnc2Cl)C3)=O)cc2ccccn2n1 23497,Cc1ccc(C(c2nnnn2-c2ccccc2C)NC(C)(C)C)c(Br)c1 23498,N1(CC(=O)NCCCCN(C)C(c2cc(Cl)c(Cl)s2)=O)CCC(C)(C)C1 23499,CCCC(CC)CC(=O)NCC(O)CN(C)C(c1ccoc1CC)=O 23500,CC(c1cccs1)=CC(N1CCC(CNC(C23CC(C)C2C3)=O)C1)=O 23501,N1(C(C(=O)NCCC)C)CCCC2(CCN(C(c3nn(C)cc3Cl)=O)C2)C1 23502,N1(C(C2CCC(C(=O)OC(C)(C)C)CC2)=O)CC(CC(=O)O)OCC12CC2 23503,C#CCCC(C(=O)NCC1CCSCC1)NC(c1cc(CCC)[nH]n1)=O 23504,CCC(C)(O)C(=O)N1CC(NC(c2cn(C3CC3)nc2C)=O)C(O)C1 23505,N1(C(C(CC(C)C)O)=O)CC(C)N(C(c2ncc(Br)s2)=O)CC1C 23506,Cc1cccc(CCC(=O)NC(=O)CC#N)c1Br.C1C(C(F)(F)F)CC2CN1C2 23507,N1(C(CC2N(C(C=Cc3n(C)cnc3)=O)CC(O)C2)=O)CCC(N=[N+]=[N-])C(O)C1 23508,C(C)(CNC(=O)COCC1CCCC1)(CO)NC(C(C)OCCOC)=O 23509,N1(C(c2c(C)ccnc2)=O)CCN(C(=O)CCC2CCCC(=O)N2)C(C2CC2)C1 23510,c1(C(=O)NC(C2CCN(C(c3cnco3)=O)C2)C)ccn2nccc2n1 23511,S(=O)(=O)(c1cc(C(N)=O)ccc1F)N(C)Cc1c[nH]nc1C(F)F 23512,C12(NC(c3coc4ccccc34)=O)CCCCC1CN(C(c1cnccn1)=O)C2 23513,CCCC(C)(C)CN=c1[nH]c2c(c(=NC3CCC(C(C)C)CC3)[nH]1)CSC2 23514,N1(C(CC2CC(SC)C2)=O)CCN(C(=O)C(F)F)C(C2CCCC2)C1 23515,C1(C#CC(=O)N2CC(NC(C3CCC(C#N)CC3)=O)C(C)C2)(CC)COC1 23516,c1(C(C)C)cccc(C(N2CCC(F)(C(=O)NC(c3ccccc3)C#N)C2)=O)c1 23517,O(C1CCOc2ccc(Br)cc21)C(=O)CCCCc1cnn[nH]1 23518,Cc1cc(C(=O)NC2C3CN(C(c4occ5c4CCC5)=O)CC23)c(O)nn1 23519,c1(CC)ncccc1C(=O)NCc1cnnc(C)c1 23520,N1(C(C=CCOC)=O)CC(NC(=O)CCc2c(OC)cccc2F)CC1(C)CC 23521,C=CCC(CC(F)F)NC(=O)C=CCF.C12CCCCC1NC(=O)C2 23522,c1(N2C(=O)CC(C(=O)Nc3cn(CCS(CC)=O)nc3)C2)cc(F)cc(F)c1 23523,C#Cc1cccc(C(N2CCN(CCNC(=O)CC3CCC(O)C3)CC2)=O)c1C 23524,C12(CC(F)(F)C1)C(=O)N2.n1(CCNC(C(C)OC)=O)cc(C2CCOCC2)nn1 23525,C(=O)(CCCCCC(C)(C)C)NC1CCC(N(C(c2c(C)cc(N)cc2)=O)C)C1 23526,C12(NC(CCCOCCC)=O)CCCC1N(C(c1cc(C)ccc1F)=O)CCC2 23527,CC(C)(C)CC(C1CCC1)NC(=O)NCCn1cccn1 23528,Cc1ccc(Cl)c(O)c1C(N1CC(NC(c2ccc(F)s2)=O)CC(O)C1)=O 23529,N1(C(CCS(C)(=O)=O)=O)CCC2(CC1)CN(C(c1ccc3scnc3c1)=O)C2 23530,C1(CC=C)(NC(=O)CC=CCNC(=O)C(C)CC2CC2)CCCCC1 23531,c1(C(N2C(C(C)(C)NC(C(F)=C(C)C)=O)CCC2)=O)cc2cc(Br)cn2cn1 23532,C(=O)(C(C)C(CC)CC)NC(C1CN(c2nc(N(C)C)nc(C)c2F)CN1)CC 23533,Cc1cc(C(N2CC(N(C(=O)CC3OCCCC3(C)C)C)C(O)C2)=O)cnc1O 23534,C1(NC(C(CC)F)=O)CC2(CCCN(C(c3coc4c3COC4)=O)C2)C1 23535,C12(C(=O)OCC)CCC(C(=O)NC3CN(C(C4(S(C)(=O)=O)CCC4)=O)C3)(C1)OC2 23536,N1(C(CC2CC(C)(C)OC2=O)=O)CC2CC(C1)CN(C(c1cc[nH]n1)=O)C2 23537,C1(C(N2CCCC(c3cn(CCCCF)nn3)C2)=O)COC2(CNC2)C1 23538,C12(CN(C)Cc3ccc(C#N)cc3)CC(C)(C1)OC21CCC1 23539,Cc1cccc(Cl)c1CC(=O)NCCCN(C1CCOC1)C(=O)COCCF 23540,N1(C(c2cc(C)on2)=O)CCC(C)(CNC(C2CC(C)CCO2)=O)CC1 23541,CC(C)C1=NOC(C(N2CC(C)(NC(=O)COc3c(Cl)cccc3Cl)C2)=O)C1 23542,N1(C(C2C(C)C2)=O)CCCCC(NC(C2CC3CCC2CC3)=O)C1 23543,C#Cc1ccc(CNc2cc(NC3COCC3n3cc(OC)cn3)ncn2)cc1 23544,C1(CNC(C(CC)c2ccccc2)=O)CC2CN(c3nccc(CC#N)n3)CC12 23545,c1(C(=O)Nc2c(C)nc(-c3cn(C(C)C(=O)O)nn3)s2)cccc(F)c1Br 23546,Cc1nn(CC(=O)NCC(C2CCCC2)NC(=O)Cn2ccccc2=O)c(=O)o1 23547,CN(C)NC(=O)CCC(=O)N1CCC(NC(C2CC(O)C2)=O)C1c1cn[nH]c1 23548,c1(C(N2CCC(O)(CNC(c3n(C)ccn3)=O)C2)=O)c(O)ccc2ccccc12 23549,C(=O)(C1CCCc2sc(=N)[nH]c21)NCC12CC(NC(CCN(CCC)C)=O)(C1)C2 23550,c1(C(N2CCCC3C(C(F)(F)F)C23)=O)c(O)ccc(Br)c1O 23551,CC(C(=O)NCC1CCCN(C(c2nc3ccccc3o2)C)C1)C(C)S(C)(=O)=O 23552,c1(C(C)=O)cccc(NC(=O)CC2CCN(C(c3occc3C)=O)C2)c1 23553,c1(C(=O)NC2(C)CN(C(C34CCC(F)(CC3)C4)=O)C2)noc2ncccc12 23554,Cc1cc(CNC(c2coc(CNC(=O)CC3CCN(C)C3)n2)=O)sn1 23555,Cc1c(C(N2CCOCC(NC(=O)C(=O)NCCC(N)=O)C2)=O)oc2ccccc12 23556,CC1CN(C(=O)Cc2ccn(C)n2)CC1CNC(=O)CC1(O)CCOCC1 23557,CC(C(F)(F)C(F)(F)F)=CC(=O)N(CCCNC(c1cnn(C)c1Cl)=O)C 23558,N1(C(CC=CC)=O)CCCC(O)(CNC(=O)C=Cc2nccn2CC)CC1 23559,c1(C(N)=O)cc(Cl)cc(Cl)c1NC(C1CNCCN1Cc1cc(Br)cnc1Br)=O 23560,Cc1oc(CO)cc1C(N1CCN(C(C2CNC(=O)C2)=O)CC1)=O 23561,N1(C(Cc2cnc(C)[nH]2)=O)CC2CCC1C1CN(C(=O)C=CC3CC3)CC21 23562,C1(CCNC(CN(C)C2CC2)=O)CCN(C(C2CC3C(C2)C3(F)F)=O)CC1(F)F 23563,C(C#N)(C(C)CC)C1C(OC)CC1.c12ncoc1C(=O)NC2 23564,C1(C(N2CCC(CNC(C(c3cncn3C)C)=O)CC2)=O)CCC2(CCC2)C1 23565,C12(C(=O)NCCCCN(CC)CC)CCN(C(=O)CC(C)(C)C)CC1C2 23566,c1(OC)ncnc(C)c1C(=O)NCC1CCCCN1C(C1CC(F)(F)C1(F)F)=O 23567,c1(C(=O)NCC(C)(CO)NC(CN(S(C)(=O)=O)C)=O)ccc(C)c(C)c1O 23568,c1(C(=O)NCC=CCC(=O)NCC=C)cc(CC2CC2)no1.c1(N)cnn(CCO)c1 23569,C1(C(=O)NCC2=CCN(C(=O)CC3CCCC3)CC2)CCC2(CCOC2)O1 23570,c1(C(C)C)cc(CNC(=O)C(CC2CCC2)NC(=O)C(F)OC(F)(F)F)on1 23571,C1(O)(C(CNC(CCN(C)CC)=O)C)CCN(C(c2cc(CC)n(C)n2)=O)C1 23572,Cc1oc(S(C)(=O)=O)cc1C(N1CCC1CNC(c1cc2c(s1)CCC2)=O)=O 23573,c1(CNC(C2CC(O)(Cn3cc(CO)nn3)C2)=O)nnc(O)o1 23574,N1(C(c2ccc(OC)c(F)c2F)=O)CCCC2(CCCN2C(C2C=CCC2)=O)C1 23575,N1(C(c2cc(C)nc(C)c2)=O)CC(C)CN(C(c2nc(Cl)sc2Cl)=O)C(C)C1 23576,N1(C(C2(C(C)C)CCC2)=O)CC2CCC1C(CNC(=O)CCCC#N)C2 23577,Cc1cc(Br)ccc1CC(=O)NCC1CCCN1C(=O)Cc1ccc(C)s1 23578,c1(CC(=O)NCCCOCCN(C(=O)CC(O)c2ccccc2)C)nocc1C 23579,C1(CC(=O)NCCC2CCN(C(C3(C)CCCC3)=O)C2)CCCC1(F)F 23580,C1(C(=O)NC2CC(COCC)C2)CC2CC1CC2NC(C1CCCN1C)=O 23581,N1(C(C2CCCC(NC(C3C=CCCC3)=O)CC2)=O)CCN2CCCCC1C2 23582,c1(NC(=O)CNC(c2cc(O)cc(=O)o2)=O)ccc2c(c1)COC2=O 23583,N1(C(C)=O)CCCC(C)(C(=O)N(C2(c3ccc(Br)cc3)CC2)C)C1 23584,c1(N2CC3CC(NC(c4ccc(CC(N)=O)cc4)=O)C3C2)ncnc2c1CCO2 23585,N1(C(C)=O)CCC(NC(c2cc(C(F)(F)F)n(C)n2)=O)C(O)C1 23586,N1(C(CCNC(C(CC)NC(N)=O)=O)=O)CCC(O)(C(=O)OCCOC)C1 23587,N1(c2nnc(-c3cc(Br)cc(C)c3N)n2C)CCCc2ncccc2C1 23588,C(C(=O)NOCC1(C)OCCO1)N(C(C1(C)C(C)C1)=O)CC1CC1 23589,c1(OC)cc(F)c(S(=O)(=O)NC2CCCC2P(C)(C)=O)cc1OC 23590,CC(C)CCC(=O)N(C(CNC(=O)Cn1cnnc1O)Cc1ccccc1)C 23591,S(=O)(=O)(c1c[nH]c(=NCC2CC3CCC(C2)S3)cc1C)NCC(COC)C 23592,N12CCCC(O)(C1)C(OC)C2=O.C(=O)C(C)(Cl)Cl.CO 23593,C(=O)(C(O)CC(F)F)NCC(C1CCN(C(Cn2nc(C)c(Cl)c2)=O)CC1)C 23594,C(=O)(C1=CCC(NC(c2cnn(C)c2Cl)=O)C1)N(C)CC1CC(F)(F)C1 23595,CC(C)(C)C(CN=c1ccn2c(Br)cnc2[nH]1)NC(c1ccc(F)o1)=O 23596,c1(C(=O)NCCCN(C(CCCOCC)=O)CC)ccc(N)c(N)n1 23597,C12(CNC(C(C)C3CCC3)=O)CC1CN(C(c1nccn1C)=O)C2 23598,C1(c2nc(C3CCCN3C(c3cccnc3)=O)n[nH]2)CCNC(c2ccco2)C1 23599,N1(C(Cc2ccc(C)nc2)=O)CC(C)(C)C(NC(c2cnc(Cl)s2)=O)C(C)(C)C1 23600,C(CC(F)(F)CF)(C(=O)NCCNC(=O)COCc1ccccc1)OC.c1ncc[nH]1 23601,N1(C(=O)OC(C)(C)C)CC2COCC2(C(=O)NC(C)(C)CN2CCOCC2)C1 23602,c1(CN2CC3CCC(C(=O)Nc4cnc(CC)s4)C3C2)[nH]c2ccccc2c1C 23603,C(CN=c1nc2sccc2c(NC2CN(C3CC3)C2)[nH]1)OC(C)C 23604,c1(CC(=O)NC2C3CC(NC(C4COCCO4)=O)CC23)ccc(F)cc1[N+](=O)[O-] 23605,C1(OCC)CCCN(C(C2CC(C)=NO2)=O)C1.c12nc(cs1)CNC2=O 23606,C(=O)(C(C)(C)CC(C)=O)N(C(C(CC)C)C(=O)N1CC=CC1CN(C)C)C 23607,C1(C(=O)NCC(C)NC(c2snc(C)c2SC(C)(C)C)=O)CN2CCN1C(C)C2 23608,CC1(C)CN(C(C2CC2C#N)=O)CC1CNC(c1cc(C(F)F)[nH]n1)=O 23609,N1(C(C(C)OCCCC)=O)CCCCC(C(N2CC(CO)C2)=O)C1 23610,C(=O)(C#CC1CCCCO1)NCC(C)(Cn1cccn1)NC(c1cccnn1)=O 23611,c1(C(=O)NC(C2CCCCN2C(C2CC(C#N)C2)=O)C)cc2cc(F)ccc2o1 23612,CCCCC(F)C(=O)N1CCCCC1C1CCN(C(c2sccc2F)=O)C1 23613,NS(=O)(=O)c1ccnc(C(=O)NCC2C(CNC(=O)CC3CC=CC3)C2(F)F)c1 23614,Cc1ccc(C(F)F)cc1OC(C)C.C1C(CC(C)C)NC(=O)N1 23615,C1(C(N2CC3(CN(C(c4ncn(C)c4)=O)C3)C2)=O)CCC(S(C)(=O)=O)CC1 23616,N1(C(C=NOC)=O)CCC2C(NC(=O)C=Cc3cc(C)no3)C2C1 23617,CCC(O)CCN=c1[nH]c(N2CCN(C(C)COC)CC2)nc2cccnc12 23618,c1(CC)nc(C(N2CCC(C(C)NC(c3cncs3)=O)C2)=O)co1 23619,c1(C(=O)NC(CC(C)NC(=O)Cn2ccnn2)C)ccc(-c2csnn2)cc1 23620,N1(C(c2cnc(C)o2)=O)CCC2C(C1)CN2C(=O)Cn1c(C)csc1=O 23621,C(CC(C)C(=O)NCC1CCC1NC(c1c(C)nsc1N)=O)OC 23622,C12(NC(C=CC(=O)OCC)=O)CC1CN(Cc1cccc(CO)n1)C2 23623,C1(CC(=O)NCc2cccc(O)c2)CCCCN1C(=O)CN1C(=O)CNC1=O 23624,C1(NC(CC2C(=O)NCC2)=O)CC2CC(C1)N(c1nnco1)C2 23625,C12(C(=O)NCCc3c(CNC(CC=C=C)=O)nco3)CC3CC1C2C3(F)F 23626,N1(C(C)=O)CCCC(C(N2CCSC(C(=O)NCCSc3cccnc3)C2)=O)C1 23627,c1(C(N(CC(C)NC(=O)CC2CC3CCC2O3)C)=O)c(Cl)csc1Cl 23628,CC1CN(C(=O)Cc2cc(C3CC3)no2)CC1NC(c1cc(Br)c[nH]1)=O 23629,C1(=O)C(CCC)N1C.C(C)(C)(CNC)N(C)C.C(C(=O)NCCO)OCC#C 23630,C(=O)(CC(C)C(C)(C)NC(C1CC(C)(CC)C1)=O)NCC1(CCC=C)CC1 23631,N1(CC(C)C)CCC(CC(=O)NC(C)CNC(c2cnn(CC(C)C)c2)=O)CC1 23632,c1(C(C)C)ccc(C(N2CCC(OC3CC3(F)F)C2)=O)nc1 23633,C1(NC(c2cnc(OC)s2)=O)CN(C(=O)CCc2ccc(SC)cc2)CC1O 23634,c1(C(=O)NCCCN(C(C2C(C)=CCS2)=O)C(C)C)cn2cccnc2n1 23635,c1(C(N2CC(N(C(C(CC(=C)C)OC)=O)C)C(O)C2)=O)noc2ncccc12 23636,c1(OC)ccc(Cl)c2[nH]c(C(=O)NC3CCCC3NC(c3coc(C)c3)=O)cc12 23637,c1(OC)ccccc1OCCC(=O)NC(C)(C)CNC(=O)Cc1cn(C)nc1C 23638,CC(CC(=O)N1CCC(CNC(=O)C(c2cc(F)cc(F)c2)O)C1)C(F)(F)F 23639,c1(C(=O)OCC(=O)NC2CC2)cnc2ncnc(O)c2c1 23640,Cc1ccc(COC(C)C(=O)NCCC2CN(C(c3c[nH]c(=O)cn3)=O)C2)cc1 23641,C(C(C)(C)C(F)(F)F)OC(C(N1CC(C(=O)NC)C1)=O)C1CN(C=O)C1.OC 23642,CC1=C(C(=O)NC2CC3CC(NC(=O)C(O)CN(C)C)CC23)SCCO1 23643,N1(C(c2nn(CC)c(O)c2)=O)CCC2(CC1)CC2CNC(=O)CC(O)CC(C)C 23644,C1(C(=O)NC23C(CN(C(CC4(C=C)CCCCC4)=O)C2)C3)CS(=O)(=O)CC(=O)N1 23645,O=C1CCN(C(C23CC(CO2)N(C(=O)C(C)(C)C2CCCO2)C3)=O)CCN1 23646,N1(C(c2c(C)nc(O)[nH]2)=O)CCC(NC(c2cc(C(F)(F)F)no2)=O)CC1C 23647,CC1CC(C(=O)NCc2ccc(C(=O)NCC3(O)CC3)cc2)CC(C)C1 23648,N1(C(Cc2ccn(C)n2)=O)C2CCC(C2)C1C(=O)NCC1(N(C)C)CCCC1 23649,C(CCCCC(=O)NC1CCC(C)N(C(c2[nH]nnc2C2CC2)=O)C1)NC(C)=O 23650,Cc1nn(CC(=O)NCCCC(=O)NCCC2CCCO2)c(=O)o1 23651,C12CC3CC3N1C(=O)N2.O=C1OCCC1C(=O)NCCCn1cc(C(F)(F)F)nn1 23652,n1(CC(=O)NCC(CCOC)NC(C2CC3CCC(C2)O3)=O)nc(C)c(C)c1C 23653,C1(NC(C2(C)CC(NC(CCc3c(C)noc3)=O)C2)=O)CCOC2(CCC2)C1 23654,C1(O)(CN(C(=O)Cn2cncc2Cl)C)CCN(C(c2ccc(CO)o2)=O)C1 23655,c1(C(=O)NC2(CCNC(C3C(C)CCC3)=O)CCC2)cc2c(F)c(F)ccc2[nH]1 23656,c1(C(=O)NCCCCNC(=O)CC2CCC(=O)N2)ccc(C(F)(F)F)cc1O 23657,c1(NC(C2CCC(NC(=O)C(C3CCCCC3)F)C2)=O)cc(-c2cc[nH]n2)co1 23658,C1(F)(CNC(c2c(CCC)[nH]c(CC)c2)=O)CC2CCC(C1)N2C(=O)C(C)OC 23659,Cc1cc(C)n(-c2ccc(-c3nc(-c4ccn(C)c4)n(CCC(C)C)n3)nc2)n1 23660,c1(C(=O)NCC2(O)CCN(C(CCn3ncc(C)c3)=O)C2)cnc2ccsc2c1 23661,C(=O)(C(O)CCNC(C1CCCC1F)=O)NC(C1CCCC1)C#C 23662,C1(CC(=O)N(CC)Cc2ncc[nH]2)COCCN1C(=O)C(=O)N(CCCO)C(C)C 23663,N1(C(C(CSC)C)=O)CC(NC(=O)C(CO)NC(=O)C(C)C)CC(F)C1 23664,c1(C2(C(=O)NC3CC(NC(c4c(C)nn(C5CC5)c4)=O)C3)CC2)ccc(C#N)cc1 23665,N1(C(C=CC=CCC)=O)CC(NC(c2cnc(C)nc2CC)=O)CCC1C 23666,CC(C)CC(F)C(=O)NCC1(C)CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CC1C 23667,N1(C(c2ccnnc2)=O)CCCC2(CCCN2C(c2cnc3ccccn23)=O)C1 23668,C1(COC)(NC(=O)Cc2ccsc2)CCN(C(C23CC4CC2C3C4)=O)C1 23669,N1(C(c2c(C)n(C)nn2)=O)CC2(CC(NC(c3n[nH]c(C)c3[N+](=O)[O-])=O)CO2)C1 23670,c1(OC)cc(Br)c(C(=O)COC(c2cc3c(s2)CCC3N)=O)cc1OC 23671,N1(C(c2c(C)nc(CC)s2)=O)CC(OC)C(OC)C1CNC(=O)CCC(C)(C)F 23672,c1(CC)cc(C(=O)NC2(C)CC(NC(=O)CCOCC(C)C)C2)ccc1C 23673,c1(CCCNC(C2CCOCC2)=O)ccc2nc(O)[nH]c2c1.C12CCCN(C1)C2 23674,C1(C(=O)NC(CNC(C=C(C)c2ccco2)=O)CC(C)C)CN(C)CC(C)O1 23675,N1(C(c2ccc(C#C)cc2)=O)CC(C)CN(C(=O)CCOCC(F)(F)F)CC1C 23676,N1(C(C2C(c3ccc(C)s3)C2)=O)CCC(C2CC2)C1CNC(c1ccsn1)=O 23677,c1(CN2CCC(NC(=O)Cc3cc(F)ccc3Br)CC2)ccc([N+](=O)[O-])c(Br)c1 23678,CCC(CC)CCCC(=O)N(CC(N1CC(O)CC1C(C)C)=O)C 23679,CC(C(=O)NC1C=CC(C(=O)NC(C)C(=O)NCCF)C1)C(F)F 23680,C1(OC)CC(CNC(c2csnc2C)=O)N(C(C2CC(N(C)C)C2)=O)C1 23681,c1(CC(=O)NC2(C#N)CN(Cc3cnccc3Cl)C2)ccccc1OCCO 23682,C(C)(CN=c1[nH]c(N(C)Cc2cccc(N)n2)nc2ccccc12)OCC(C)C 23683,CCCC(C(O)C(=O)NCC1(O)CCCOC1)NC(c1ccccc1CC)=O 23684,N1(C(c2ccc(OC)c(Cl)c2)=O)C2CCCC1CN(C(=O)C(C)CS(C)(=O)=O)C2 23685,C#CCCCC(=O)N1CCC(C(F)C(=O)Nc2cnn(CCC)c2)C1 23686,c1(OC)cnc(C(N2CCC(c3cn(Cc4ncccn4)nn3)C2)=O)nc1 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23722,c1(CC)ncsc1C(=O)NC1(CN(C(=O)CC(F)F)C)CC1 23723,CCCCC(CNC(c1cnccc1Cl)=O)NC(=O)CC1CC(F)(F)C1 23724,C1(NC(CCC2C(C)C2)=O)CC(C)(CNC(=O)CC23CCCC2C3)C1 23725,N1(C(c2c(SC)csc2)=O)CCC2CN(C(c3ncc(C)cc3C)=O)CC12 23726,C1(C(=O)NCCC(C)(C)NC(C2CC=CC2)=O)CC2COCCN2C1 23727,Cc1c(C(=O)N(C2CCCN(C)C2)C)cc([N+](=O)[O-])cc1Cl 23728,CCC(C)C(O)C(=O)N1CCN(CC2CN(C(=O)C3=COCCC3)C2)CC1 23729,c1(C(=O)NCc2cccc(CN(C(C(C)CO)=O)C)c2)onc2c1CCCC2 23730,N1(CC2CCC(C(N(C(C(C)C)=O)CCCCl)=O)CC2)CCC(CO)C(F)(F)C1 23731,C=CC(C)CC(=O)NCCC1(OC)CN(C(=O)CCc2cc(OC)no2)C1 23732,c1(C(=O)NC(CNC(COCCOC)=O)C)ccc(SC(C)(C)C)cc1 23733,c1(OC)nc(Cl)cc(=NC(=O)C2CN(Cc3cccc(I)c3F)C2)[nH]1 23734,c1(C(N(C)CC2(CNC(=O)C=CS(C)=O)CC2)=O)cnn2cccnc12 23735,c1(C(N2CC(C)(CNC(c3c(C)c[nH]n3)=O)OCC2)=O)cc2c(s1)CCCC2 23736,c1(N(C(c2c(C)scc2)=O)C2CC2)ccc(O)c(C)c1.N12CC3C(C3C1)C2=O 23737,S(=O)(=O)(c1cccnc1N1CCC(C)C(C)C1)NC 23738,c1(C(C)=O)ccc(CC(=O)N(CCCCN(C(=O)Cn2nccc2C)C)C)s1 23739,N1(C(C(C)SCCCC)=O)CC(CNC(=O)CN2CCSCC2)CC(C)(C)C1 23740,C1(O)(CN(C(CCC)=O)C)CCN(C(c2n[nH]c(SC3CC3)c2C)=O)C1 23741,C1(C(=O)NC2C(NC(COCC#C)=O)COC2)Cc2cc(F)ccc2C1(F)F 23742,C1(C)(NC(CCN(C(Cc2c(C)noc2C)=O)C(C)C)=O)CC2CCC1C2 23743,N1(C(C=CC(CC)=CC)=O)CC2CCC1C2NC(C1C(C)C1C)=O 23744,C1(N(C)C(c2ccc(C3CC3)o2)=O)CCC2CN(C(=O)Cc3nccn3C)CC12 23745,S(=O)(=O)(c1cnccc1N1CCS(=O)(=O)C(CO)C1)NC(c1ccc(Br)cc1)C 23746,C1(CNC(c2ccc(F)s2)=O)CC(O)C(O)CC1C(N1C(C#C)CCC1)=O 23747,c1(C(N2C(CNC(C3(C)CC=CCC3)=O)CCC2)=O)c(N)cc(F)c(Br)c1F 23748,c1(NC(CC)CO)cc(Br)ccc1S(=O)(=O)NC1CCCN(C)C1 23749,CCCC(C)(O)C(=O)NCCc1ccc(CNC(C2CCCC2OC)=O)cc1 23750,C1(C2CCOCC2)(c2onc(-c3c(C)ccnc3)n2)CC1 23751,N1(C(C=C(C)C(F)F)=O)CCC(NC(c2ccc(F)cc2F)=O)C(O)C1 23752,CCC(c1cccc(Cl)c1)=CC(=O)NCC=CCNC(C1CCC(C2CC2)C1)=O 23753,C(=O)(C(O)CCCC)NCC1(O)CCN(C(CSCCC)=O)C1 23754,N1(C(C(C2CCCC2)OCC)=O)CCC(CCNC(c2cnc(O)o2)=O)CC1C 23755,N1(C(C=CC=CC)=O)CCN(C(=O)Cn2c(C)c(C)sc2=O)C(c2ncc[nH]2)C1 23756,Cc1c[nH]c(C(=O)NC(c2ccccc2)C(=O)N2CC(OCCO)C2)c1C 23757,Cc1cc(C(=O)NC2CCCC(NC(c3ncc(C)cc3Br)=O)C2)cc(F)c1 23758,N1(C(c2nc(C)sc2C)=O)CC(C)OC2(CCN(C(=O)C(N)=O)C2)C1 23759,N1(C(CC2N(C(=O)CCC3CC3(F)F)CCC2)=O)CC=CC12CCCC2 23760,C(=O)(CS(=O)C(F)(F)F)N1CCC(NC(C(CC)=CCCC)=O)CC1C 23761,c1(C(=O)NCC(CC)NC(c2cn(CCF)nn2)=O)c(OC(F)F)cccc1F 23762,c1(C(=O)NCC2CC(CCNC(CCC=C)=O)C2)sc2nc(C)nc(C)c2c1C 23763,Cc1ccc(C(C)C)c(C(=O)NCC(C)(C)NC(c2ccc(F)s2)=O)c1 23764,c1(OCC(N2CC(C3CCN(C(=O)C(F)=CCCF)CC3)C2)=O)cccc(O)c1 23765,Cc1cc(=NCc2cccc(CS(C)=O)c2)[nH]c(N2CC(C)=CC(C)C2)n1 23766,CC1=CC2CCCC(C1)N2C(=O)NCCCCCCN1CCCCCC1 23767,CC#CCC(C(=O)Nc1ccc(O)cc1C)NC(=O)C(C)N(C)C(C)=O 23768,c1(C(N)=O)cccc2c1C1CCC2CC1.C1CCCN2CC(C2)C(=O)O1 23769,N1(C(C2(CCNC(C(CC)C)=O)CCCC2)=O)CC2C=CCC(C2)C1 23770,c1(NCc2ccc(C)cc2)cc(C(=O)O)ccc1N1CCCC1=O 23771,C12(CNC(Cc3ccc(C)c(Cl)c3)=O)CCC(CC1)N(C(=O)C(O)CC(F)(F)F)C2 23772,c1(NCC(C2CCCCC2)NC(CC2C(C)C2)=O)cnc2ccccc2n1 23773,S(=O)(=O)(c1ccc(N2CCC(F)(F)CC2)cc1Br)SCC.C12(CCOC1)CN2C1CC1 23774,c1(ONC(Cc2n(C)ncc2)=O)ccc(Cl)c(C(=O)O)c1.C1(C2CC2)CC1 23775,N12CC(C(C)C1)C2=O.CCCCCC(=O)NCc1cc(-c2ccncc2)nn1C 23776,CCS(=O)(=O)CC(=O)N1CCC(NC(=O)CCCOC(=O)CCC)C1.C(C)(C)C 23777,c1(OC)ccccc1SCC(=O)NCCC1CCCN1C(C1CCC(C)(C)C1)=O 23778,c1(N(CCC)CCNC(=O)CN2CCCS2(=O)=O)ncc2ncn(C)c2n1 23779,N1(C(C(CCCC)C)=O)CCCC2CN(C(C3CN(CC(C)C)C3)=O)CC12 23780,C12(CCN(C)C1)C(=O)N2.Cc1ccsc1CCCC(=O)NCCCN(C)C 23781,C(C)(C(=O)N1CCCC(C)(CNC(=O)C(C2CCCCC2)F)C1)(C(C)C)OC 23782,N1(S(c2c(N3CC(CO)OCC3)nccc2)(=O)=O)CCc2cc(C)cc(C)c2C1 23783,C1(CNC(CN(CCOC)C)=O)CC(OC)CN1C(=O)C=Cc1ncc(C)[nH]1 23784,C(=O)(C1=CCCOC1)NCCC1OCCN(C(C(C)(C)Cc2ccccc2)=O)C1 23785,c1(C(=O)NCC2N(C(C(C(C)C)C)=O)CCC2)c2n(c(=O)n1C)CCCC2 23786,Cc1ccc(C(F)C(=O)OCC(=O)N(C)CC2CCOCC2)cc1 23787,Cc1nccc(CCC(=O)NCC2CCCCN(C(C3(C)CCCCCC3)=O)C2)n1 23788,CCCCC(C(=O)NC)NC(C12CC1CN(C(c1cc(C)ccc1F)=O)C2)=O 23789,c1(NC(=O)NCc2nnc(S)n2CC2C(CCC)CCC2)ncc(OC)cc1C 23790,n1(CCC(C)C)ccc(=NC(=O)c2ccc(C3CCNCC3)s2)[nH]1 23791,C1(C(=O)NC2(C)CN(C(C(C)c3ccco3)=O)C2)CN(C(N)=O)CCO1 23792,C(=O)(CCCCC(F)F)N(CC(C)NC(C(c1ccccc1)OCC)=O)CC 23793,C(=O)(C#CC(C)(C)C)N1C(C)(NCC(N2C(CCCCC)CC2)=O)C=CC1 23794,CC(CN=C(NCC1(C2CCCO2)CCCC1)NCC(F)F)CC(F)(F)F 23795,N1(C(CC2CC(SC)C2)=O)CCC(C(=O)NC2CCN(CCF)C2)C1C 23796,C(=O)(CCC(F)(F)F)NC(C1(O)CCN(C(c2nn(C)cc2Cl)=O)C1)C 23797,C1(C)(NC(CCOc2ccc(C)cc2)=O)CCN(C(C2CC(C)(O)C2)=O)CC1 23798,c1(N(C2CN(C(=O)C(C)C(F)F)C2)C(CC)=O)cc(C(F)(F)F)ccc1I 23799,N1(C(C(CC)OCC)=O)CC2CCC2(NC(C2(c3ccno3)CC2)=O)C1 23800,N1(C(C(C2CCOC2)OC)=O)CC(C)(NC(=O)COC2CCCCC2)C1 23801,C(=O)(C(F)C(C)CNC(c1cncc(OC)n1)=O)NCc1n(CC)cnn1 23802,c1(OC(C(N2CC(O)(CN(C(C(CC(C)C)OC)=O)C)C2)=O)C)ccccc1C 23803,N1(C(CCC(=O)NC(C)(C)C)=O)CC2(C1)CN(C(c1cnn(CCF)c1)=O)C2 23804,N1(C(c2c(C)nn(C)c2C)=O)CC(NC(=O)Cc2nncs2)CC2(CC2)C1 23805,C1(C(=O)Nc2c(OC)nccc2)C2CCCC1N(C(c1ccnc3c1CCC3)=O)C2 23806,CCCCCCCC(F)C(=O)N1CC(O)(CNC(C2CC3CCC2O3)=O)C1 23807,Cc1noc(C)c1C(=O)NC(C1CCCCN1C(c1occc1Cl)=O)C 23808,S(=O)(=O)(c1cccc(=NCc2ncc(Br)s2)[nH]1)NC1CCC(C=C)CC1 23809,N1(C(CN(CC(C)C)C(C2CCCN2C(C)(C)C)=O)=O)CC(F)CC1C 23810,C1(CCC)CN(C(=O)CN(C(=O)C(c2ccccc2)C)C(C)C)CC1CO 23811,C(CNC(=O)Cc1c(Cl)cnn1C)(CCCC)NC(CSCC=C)=O 23812,C(c1ccc(F)cc1F)=CC(=O)NCC1CN(C(c2nc(C(C)OC)sc2)=O)C1 23813,C(=O)(CCCCC(=O)OC(C)(C)C)NC1C(NC(C2CC(C)OCC2)=O)CCC1 23814,C(=O)(C1=CC2C=CC(C1)C2)NCCCN(C(C)C)C(C1CC(O)CN1C)=O 23815,C(C)(C)(CCN=c1nc(C#N)cc(C)[nH]1)NC(Cc1ccc(OC)cn1)=O 23816,C1(C(=O)Nc2nc(C(F)(F)F)cs2)CN(C(=O)CCc2ccccc2)CCN1 23817,C1(C(=O)NC2CC(CNC(Cn3c(C)ccc3C)=O)C2)CC(S(C)(=O)=O)C1 23818,FC1(F)CC12CCC(CSc1ccc(-c3ncccn3)cc1)C2 23819,c1(C(N2CC(C)C(NC(c3ccc(Cl)cn3)=O)C2)=O)c(N)sc2c1CCSC2 23820,CC1SCCCC1C(=O)NC1CCN(C(=O)C=Cc2cnccn2)CC1 23821,N1(C(C(C)(C)O)=O)CCC(C2CCN(C(C3(CF)CC3)=O)CC2)C1 23822,N1(C(C(C2CCOC2)OC)=O)C2CCCC1CN(C(C1CC1C(C)O)=O)C2 23823,N1(C(CCSCCC)=O)CCN(C(=O)Cc2nocc2C(C)C)CCC1C 23824,C=CC(CC)CC(=O)NC(CN(C(c1cn(CCC)nc1C)=O)CC)CC 23825,CCC(C)CCC(=O)N1CCC(CNC(c2cncnc2C)=O)C1(C)C 23826,C(C)(C(=O)N1CC(C(O)C(=O)N(C(C)C(C)SC)C)C1)OCCCC 23827,C#Cc1cc(C(=O)OCCOC2CCCCC2C)cc2c1OCCO2 23828,Cc1nsc(C(=O)NCC2CCCCN2C)c1N 23829,C1(C(=O)NCCC(=O)NCC#C)CCCC(NC(=O)COCCOC)CC1 23830,C1(NC(C(C)C2CC2)=O)CN(C(c2cc3scnc3[nH]2)=O)CC12CCOCC2 23831,c1(C(=O)NCCC(C)NC(CN(C2CC2)CC)=O)cnc2nc(C)ccc2c1O 23832,N1(C(C(CCCC)O)=O)CCOC2(C1)CN(C(=O)C(O)Cc1ccc(O)cc1)C2 23833,C1(C(=O)NC23CC(CC(NOC(CC)C)=O)(C2)C3)CC2CC(=O)C1O2 23834,C1(NC(c2ccn(CC(C)C)n2)=O)CC(NC(=O)C=CC=C(Cl)Cl)C12CCC2 23835,c1(NC(c2cccc(OC)c2)C(=O)OC)cc(Br)cc(C)c1OC 23836,Cc1ncnc(C(N2CCCC(NC(C3(F)CCCOC3)=O)C2)=O)c1C 23837,Cc1noc(C)c1CC(C)C(=O)NCCC1(O)CN(C(C2CC3C=CC2C3)=O)C1 23838,N1(C(COCc2cc(C)no2)=O)CCC(C)(CNC(c2ccncc2)=O)CC1 23839,C1(C(=O)OC)(C(=O)NC2CCN(C(C3CC=CCO3)=O)C2)CC=CC1.C1CO1 23840,C(N=c1[nH]c2ccc(Cl)cc2c(=NCCSC(C)(C)C)[nH]1)C1C(C)(C)OCCO1 23841,CCC(C)(C)CC(=O)N1CCOCC(C(=O)NCC=CC(C)(C)C)C1 23842,n1(CC)cc(C(=O)NC(c2cccnc2)C(=O)NCC2CCCS2)c(C)n1 23843,C(=O)(CCCCCN(C)C)N1C(C(=O)Nc2c(CC)cccc2)CC(C)C1 23844,c1(NC(C2(CNC(=O)CCc3ccsc3)CC(=C)C2)=O)ccc(CO)nc1 23845,C(=O)(NNC(=O)N1CCCC1C(F)(F)F)c1n(C)ncc1 23846,c1(CCC)cccc(C(=O)NC(C)CCCNC(=O)CC2CC3(CC3)C2)c1 23847,N1(C(C2(OC)CCC2)=O)CC(CC(=O)NCCn2nc(C)cc2C)C2(CC2)C1 23848,c1(NC(N2C3CC2CN(Cc2ccccn2)C3)=O)cccc2c1OCCO2 23849,CC(C)C(C)(C)C(=O)NCc1cc(C(=O)NC(C2(CO)CC2)C2CC2)n[nH]1 23850,O=S(=O)(c1ccc(NCCc2ccc(F)c(Br)c2)cc1Br)NC(C1CC1)C1CC1 23851,C1(NC(C(CC=C)CC)=O)CCC2(CC1)CC(NC(c1ccoc1)=O)C2 23852,c1(SCC(=O)NCC2(OC)CCN(C(C(CC)N(C)C)=O)C2)nc2ccccc2[nH]1 23853,c1(C(N2CCN(C(C(CCC)C)=O)C(COC)C2)=O)sc2ccccc2c1Cl 23854,CC1(C)CCCC(CCCC(=O)NCC(C)(O)CNC(=O)CCc2cnco2)C1 23855,CC1CC(C(=O)NCCSCC(N2CCOC(C)C2C)=O)CCC1=O 23856,N1(C(c2cc(OCC)no2)=O)CC(C(=O)NC(c2ccccn2)C)C(F)C1 23857,c1(C(N(C2CCCN(C(c3ccsc3SC)=O)C2)CC)=O)nccc(C)c1N 23858,C1(N(CC(C)CC)C(CCCCCC)=O)CC(C(=O)NCCCCC)C12CCC2 23859,C1(N(C)C(c2ccc([N+](=O)[O-])[nH]2)=O)CN(C(c2cccc(F)c2)=O)CC1(C)C 23860,C1(CC(=O)NC2C(SC)CN(C(=O)Cc3nc(C)sc3C)C2)OCCOC1(C)C 23861,CCS(=O)(=O)CC(=O)NCC=CCNC(c1c(-c2ccccn2)n[nH]c1C)=O 23862,c1(OCC(N)=O)ccc(C(=O)NC(CNC(=O)CC2SC(=N)NC2=O)CO)cc1 23863,Cc1c(CNC(C2CCOCCN2C(=O)CNC(=O)C2CC2)=O)cccc1F 23864,Cc1cccc(CN2CC3C(C2)N3C(c2ccc(F)cc2C(F)(F)F)=O)c1Br 23865,N1(C(CCCCNCCN(CCCCOC)C)=O)CCn2nc(C)cc2C1 23866,C1(N)(C(C)(C)C)CCN(CC2CC(=O)CCO2)C1 23867,N1(C(C2(CC=C)CCOC2)=O)CC2C(NC(c3cnnc(C)c3)=O)C2C1 23868,Cn1nnc2c1C(c1nc(-c3ccc4c(c3)C(O)CCCC4)no1)CCC2 23869,Cn1cnc(C#N)c1-c1cn(CCCCCCCC(=O)NC(=O)CS(C)(=O)=O)nn1 23870,CCC(C)C(C(=O)NCCC1=CCCCC1)NC(c1cccc(OC)c1)=O 23871,c1(C(=O)NC2(CNC(C3N(C)CCC3)=O)CC2)nccc2occc12 23872,C(CSC)(C(=O)NOCC(C)O)NC(C(COCC)(C)C)=O 23873,N1(C(C2C(C)N(C)CC2)=O)CCC2CN(C(=O)CNS(N)(=O)=O)C(C)C12 23874,c1(C(=O)NCCC2N(C(CC#N)=O)CCOC2)cccc2c1OCC2 23875,C(C(=O)N1CC(NC(c2c(F)cncc2Cl)=O)CC(O)C1)(C(C)(C)C)OC 23876,c1(OC)cc(NC(=O)CCOC(c2cc(O)nc(O)n2)(C)C)nc(OC)n1 23877,c1(CNC(C=C)CO)ccc2c(c1)CN(Cc1cnc(O)c(Br)c1)C2 23878,C1(NC(CCCC#C)=O)CN(C(C2(CC=CC)CCC(O)CC2)=O)CC12CCC2 23879,C12(CC(=O)NCC3CCC(NC(C(=O)NCCOC)=O)CC3)CCC(CC1)OC2 23880,CCC(CC)C(C(=O)N1CCC(F)(F)C(CNC(C2CC3(CSC3)C2)=O)C1)OC 23881,N12CCS(=O)(=O)C(C1)CCC2.N1(C(=O)OC(C)(C)C)CC=CCC1CCO 23882,c1(CNC(C2(c3nn[nH]n3)CCCSC2)=O)cc(O)ccc1O 23883,c1(C(=O)NC2CC3C(NC(C(C)n4cncn4)=O)C3C2)c[nH]nc1[N+](=O)[O-] 23884,c1(OC)ccc(C(=O)NC2CC(C)CN(C(c3n[nH]c(C)c3Cl)=O)C2)c(F)c1Cl 23885,O1NC(=O)C(CCSC)NC(=O)CCC1.C1(C(=O)OC)CC1(F)F 23886,C1(C(N2CC(CC#C)OCC2)=O)CCN(C(=O)OC(C)(C)C)C(C#N)C1 23887,c1(C(N2CCN(CC3CN(C(C4=CC(C)(C)C4)=O)C3)CC2)=O)[nH]cc2c1CCC2 23888,C(=O)(C(F)C(=O)NCCCOCCOC)OCC.c1(CCN(C)C=O)ccc(O)cc1 23889,c1(CC(=O)NCc2cnn(CC)c2C)ccc(Br)cc1OCC(F)F 23890,C1(CC)CCCCN1C(c1ccc(CCNCc2ccnnc2)cc1)=O 23891,C1(C(C)C(=O)NC(c2nnnn2CCCC2CC2)C2CCOC2)CCCC(=O)N1 23892,CCC(C)CCCCC(=O)NCC1(C)CN(C(=O)CN2CCCNC2=O)CCO1 23893,Cn1ncc2c(NC(C3CC4CN(C(=O)CC5CC6(CC6)CO5)CC34)=O)ncnc12 23894,C(=O)(CCCCNC(c1ccncc1Cl)=O)NC(C)(CO)CO 23895,CCC(C)CCCCC(=O)NCCCOC1CN(C(=O)CSCC(N)=O)C1 23896,CS(C)(=O)=Nc1ccc(C(N2CCN(C(=O)C(C3CCCO3)C3CC3)CC2)=O)s1 23897,C1(C(=O)NOCC2CCCO2)(CC=C)CCCN1C(=O)C(C1CCOCC1)F 23898,c1(C(=O)NC(CC(C)NC(C(CC)=CC)=O)C)c(C)c[nH]c1CC(N)=O 23899,c1(CN(C)Cc2c(OC)ncc(C)c2)cc2c(OC)cccc2[nH]1 23900,C#Cc1ccc(CNC(=O)C(C(C)(C)C)c2cn(CC3(C(=O)O)CC3)nn2)cc1 23901,Cc1cc(Cl)cnc1NC(NNC(c1ccc(NCC(C)(C)S(C)(=O)=O)cc1)=O)=O 23902,c1(OC)ccc(C2(C(=O)N(CCCCNC(=O)CN(C)C(C)C)C)CCC2)cn1 23903,C1(C(N2CC(C3(NC(C(c4ccnn4C)C)=O)CC3)C2)=O)CS(=O)(=O)CC(=O)N1 23904,N=c1cc(C(N2CCN(C(C3CC3F)=O)C3CC23)=O)[nH]c(=N)[nH]1 23905,Cc1nc(-c2ccccc2)sc1C(=O)NC1(CCNC(C2(C)CC2F)=O)CC1 23906,C1(CCC(C)C)CN(C(=O)C(=O)NC(c2ccc(F)cc2)CN)CCS1 23907,c1(CC(=O)NCCC2(O)CN(C(CC3CC(=C)C3)=O)C2)nnc(S)nc1O 23908,c12ncccc1c2=O.c12nnn(C)c1S2.n1(CCC)ccnc1CCCOC 23909,c1(NC(C)=O)ccnc(C(N2CC(C)(NC(=O)CCCOC(C)(C)C)C2)=O)c1 23910,C1(NC(c2ccc(N(C)C)c(F)c2)=O)CN(C(=O)CCC2CC2)CC1C1CC1 23911,CCCC(CCC)C(=O)N1CCC(CC(C)NC(C2CC(C)CC(C)C2)=O)CC1 23912,C1(C(C(=O)NC(COC)C)C)CCN(C(c2ccns2)=O)C1 23913,n1(CCCOCC)c(N(CCCS(C)=O)C2CCOCC2)nnc1-c1coc(C)n1 23914,c1(C(N2CCN(C(=O)CO)C3CC23)=O)ccc(Cl)c(F)c1.c1ccc(F)cc1O 23915,c1(C(=O)NC(CC)(CNC(C2(C)CSC2)=O)CC)ccc2occc2c1 23916,c1(NC(C2C(NC(C(C(CC)O)(F)F)=O)COC2)=O)cnc2ccccc2c1 23917,N1(C(C(CCC)C)=O)CCN(C(c2cc(C(N)=O)c[nH]2)=O)C2CCC12 23918,C(=O)(C1=C(C)CCC1)NC1CCN(CCCNC(C(CC)O)=O)C1 23919,c1(C(=O)NC2(CCOC)CCN(C(CC)=O)C2)ncc2cc(Cl)ccn12 23920,N1(C(c2ncn(C)c(=O)c2)=O)CCCC2(CCN(C(=O)CC(O)CC3CC3)C2)C1 23921,CP(C)(=O)c1cncc(CNC(=O)NC(c2ncccc2F)c2ccccc2)c1 23922,C#Cc1cnc(C(=O)NC(C)(CNC(C2CC23CCC3)=O)C(C)C)c(C)c1 23923,C=CC(C)(C)CC(=O)NC12COC(C1)C(NC(C1CCCC1(F)F)=O)C2 23924,C(CCCC(=O)NCC(CO)OC=O)N(C(Cc1n(C)cnc1)=O)C 23925,c1(C(=O)NCC(CNC(C2=C(C)OCCS2)=O)CO)ccc2c(c1)OC(C)(C)C2 23926,C1(OC)CCCN(CCNC(C2CC(=O)N(C)C2)=O)C1.c1(-c2ccco2)ccccc1 23927,n1(CC(=O)NC2CN(C(c3ccc(NC(C)=O)nc3)=O)C2)c(C)cc(C)nc1=O 23928,c1(OCCNC(c2ccc(I)cc2)=O)c(F)cc(Cl)cc1F 23929,c1(C(=O)NCC2(OC)CCN(C(CS(CC)=O)=O)C2)cccc2c1OCC2C 23930,c1(C(N(CCN(C(c2sc(C)nc2C)=O)CC)CC)=O)ccc(Br)c(C)c1N 23931,N1(C(CC(C)SC)=O)CCCC(C)(NC(=O)C(=Cc2cnn(C)c2)C#N)C1 23932,C(=O)(CCC(=O)C(C)(C)C)NCC1C(C)CCCN1C(C1CCCCC1(C)C)=O 23933,c1(C(N2CC(CNC(C=CC=CCC)=O)C(F)(F)C2)=O)c(S(C)(=O)=O)cnn1C 23934,C1(CC(=O)NC(CC=C)CNC(=O)C=CCC)COC(C)(C)CO1 23935,N1(C(CCC(C)=O)=O)CCC2(CCCN2C(c2nn(C)c(C)c2Br)=O)CC1 23936,N1(C(CNC(=O)OCC)=O)CC(O)(C(C)NC(=O)Cc2cc[nH]n2)C1 23937,C1(CNC(Cc2c(C)noc2)=O)CCN(C(=O)CC(C)n2ccnc2)C(C)C1 23938,C1(NC(c2ccc(C)n2C)=O)CC12CCN(C(C1COCCN1C1CCCC1)=O)C2 23939,N1(C(C2CC(C)(O)C2)=O)CCC2CC(CNC(=O)CC=C(Cl)Cl)CCC2C1 23940,N1(C(c2ccnc(C)n2)=O)CC2CC(NC(=O)Cc3csc(C(C)C)n3)CC2C1 23941,C1(NC(c2c(SC)csc2)=O)CC2CCC1(NC(=O)CC(C)(C)C#N)C2 23942,C(=O)(C(C)CC(F)(F)F)N(CCCCCNC(c1ccc(OCCC)nc1)=O)C 23943,c1(OC(=O)CNC(=O)NC23CCN(C(=O)CO)CC2C3)cccc2ccccc12 23944,CCCCC(C)CCC(=O)NCC(CC)NC(C1CCN(C)C1CC)=O 23945,c1(NC(=O)CC2CC(O)CN2C(C2CCCSC2)=O)cc(O)cc(F)c1 23946,CC1CN(C(=O)C(=O)NC2CCCNC2)C(C)CN1CC(F)F 23947,Cc1c(NC2CCCCC2CC(F)(F)F)ncnc1N(CCCC(C)C)C 23948,N1(C(c2n(C)c(Cl)c(Cl)c2)=O)CCC2(CCCCC2NC(=O)Cc2cnc[nH]2)C1 23949,CCC(CC(=O)NC1CCC(C)N(C(c2nc(C)sc2C)=O)C1)CC(C)C 23950,c1(C(=O)NC(CCC)C2CC2)coc(CNC(C2(CO)CC2)=O)c1 23951,c1(N(C)C(C2CN(CC(F)(F)F)CCC2O)=O)c(Cl)cc(Cl)cc1Cl 23952,N1(C(CCC2(C)CCC(=O)N2)=O)CC2CCC(C1)C(NC(=O)C(F)C1CCC1)C2 23953,C12(CNC(C=NOC)=O)CCC(NC(c3cc(Cl)cc(C)c3O)=O)(CC1)CO2 23954,C1(CNC)CN(C(c2ncnc(C)n2)=O)CC1C.c1cc(CC(=O)OC)on1 23955,Cc1ccc2c(C(=O)N(C3C4CN(C(C5(CO)CCC5)=O)CC34)C)onc2c1 23956,C=CCCCCCNC(=O)NC(CO)C1CC1c1ccccc1 23957,c1(C(=O)NCC2C(NC(C3C(=C)C3)=O)CCCC2)cc(F)c2[nH]nnc2c1 23958,c1(OC)cc(C(N2CCCC2CNC(C2C(C#N)C2(C)C)=O)=O)cc(Cl)c1 23959,c1(C(N2C(CNC(C(C)CC(N)=O)=O)(CC3CC3)CCC2)=O)cnn2cccnc12 23960,c1(CN2CCCC(N3CCN(C(CCC#C)=O)CC3)C2)n[nH]c2ccc(Cl)cc12 23961,Cc1ncc(C=CC(N2CC(F)(F)CC2CCNC(=O)C(C)C2CC2)=O)c(O)n1 23962,c1(C(=O)NCC(CNC(c2sc(CC)c(C)c2)=O)CO)ccc2cccnn12 23963,C1(C(N2CCCC(N(C(CCCSC)=O)C)C2)=O)C2CC3C(C2=O)C13 23964,c1(CN2CCC(N(C(c3n(CCCOC)nnn3)=O)C)C2)c(Br)cnc(Cl)c1F 23965,C1(NC(C(C)c2ccsc2)=O)CCC2(CC1)CCN(C(=O)OC(C)(C)C)CC2 23966,C#CC1CN(C(C2(O)CN(C(c3cnc(OC)cn3)=O)C2)=O)CCN1C 23967,N1(C(CC(=C)C)=O)CCC(OCCN2CC(NC(c3nccs3)=O)C2)CC1 23968,Cc1ccc(C=CC(=O)NCCCC2CCCN2C(=O)CN(C)C)nc1 23969,C1(CCC(=O)NC(C2CCOC2)C#C)CCCCN(C(c2cc(=N)[nH][nH]2)=O)C1 23970,C(=O)(CCC(C(C)C)NC(c1ccncn1)=O)N1CCC(C(CC)C)CC1 23971,c1(N(C(C)C)Cc2cccc(C)n2)nc(=NCCc2cccs2)[nH]c2c1CCC2 23972,C(CC(COC)N=c1[nH]c(=NCC=CC2CC2)[nH]c2c1COCC2)OC 23973,N1(C(C(CC#C)O)=O)CC2(CNC(=O)CCOCCCOC)CC(F)(C1)C2 23974,CC(C)(C#N)C(=O)NCCc1ocnc1CNC(=O)CCc1nncs1 23975,C1(C(=O)NCCCOCCCNC(CSS(C)(=O)=O)=O)CC2(CCOCC2)CO1 23976,N1(C(CC(=O)OC)=O)CC(NC(C2CC3CC2C3)=O)C(O)C1 23977,CC1C(NC(=O)Cc2c[nH]ccc2=O)CC2CCC1N2C(c1ccc(F)s1)=O 23978,c1(C(N(CCNC(C2CC(C)(CC)C2)=O)C)=O)ccc(NC(N)=O)cc1 23979,C(=O)(C(C)CC(C)(C)C)N(CCC(=O)N(CCCO)C(C)C)CCCO 23980,C1(C(=O)NC(CCCNC(c2nncc(C)c2)=O)C)CCCC(C)(C)CC1 23981,N1(C(C=CC=CCC)=O)CC2(C1)CN(C(c1cc(C)nc(C)n1)=O)C2 23982,c1(OC)ccc(SCC(=O)NC23CC(CNC(C)=O)(C2)C3)cc1 23983,C1(NC(C(CCC=C)NC(=O)CC=C(C)C)=O)CC(C2CC2)(C2CC2)C1 23984,C12(CNC(c3c(C)cccc3)=O)CCCC1CCN2C(=O)Cc1cnn(C)c1C 23985,c1(OC)cc(OC)cc(CN2CCC(O)C(C(=O)NC3CC(O)C3)C2)c1 23986,C1(CC(=O)NC2CC(C)OC2=O)CC(C)(C)CN1C(=O)CCC1CCCCC1 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24073,C(=O)(CCS(N)(=O)=O)NCC(CCNC(=O)C(c1cccc(C)c1)F)OC 24074,c1(OC)cscc1C(=O)NC1CC(N(C)C(c2nccn2C(C)C)=O)C1 24075,Cc1ccn(CC(N2CCC(F)(CNC(=O)CCOC3CC3)C2)=O)c(=O)c1 24076,c1(N(C)Cc2ccc(Cl)nc2)[nH]c(=NCc2cc(N)ccc2F)nc2scnc12 24077,CCC(C)(CO)C(=O)NC(C)C(C)NC(=O)COC1CCCCCC1 24078,N1(C(CCOCC(C)C)=O)CCN(C(=O)CC2CCC(=O)NC2)C2(CCC2)C1 24079,N1(C(C(C)OCC#C)=O)Cc2nccn2CC(NC(=O)C2=CCC(C)(C)C2)C1 24080,C1(C(=O)NC(CNC(C(CC)c2ccccc2)=O)C)CCc2cc(C)ccc2O1 24081,N1(CCC)CCCC(C(=O)NCCC2CN(C(c3ccc(C)nc3)=O)CCO2)C1 24082,c1(CC)cc(C(=O)NC(C2(O)CCN(C(C3(OC)CCOCC3)=O)C2)C)sc1C 24083,C(=O)(CCC(C)NC(c1cn(C)c(C)n1)=O)N(C(C)COC)CC=C 24084,c1(C(=O)OCCC(C)NC(C)=O)ccc(N=Nc2ccc(C)cc2[N+](=O)[O-])[nH]1 24085,CC1CN(C(c2ccc(C(C)(C)C)cc2N)=O)CCC1NC(=O)Cc1cscn1 24086,C1(C(=O)NC2CCC(NC(CC3(COC)CCCC3)=O)CC2)OCC2CCCC12 24087,c1(NC(C2CCN(C(C3(C4CCC4)CC3(F)F)=O)C2)=O)ncc(Cl)cc1[N+](=O)[O-] 24088,N1(C(c2cc[nH]c2)=O)CCCC2C1CCCN2C(c1cc2cccnn2c1)=O 24089,C1(C(=O)NC2C(O)CCN(C(c3n(CCC)ncc3)=O)C2)CCn2cnnc2C1 24090,c1(C(=O)OC)cc(C(=O)NC2CCC(NCC3(OC)CCOC3)CC2)cc(F)c1 24091,C1(C)(CNC(C(C)OCc2ccc(OC)cc2)=O)CN(C(c2cnns2)=O)CCO1 24092,c1(NC(N2CCC(C3CCCN3C(c3ccncn3)=O)C2)=O)cc(O)ccc1F 24093,C1(C(=O)NC(CNC(CCSCCCC)=O)COC)(C(=O)NC)CCOCC1 24094,C1(CCCCNC(=O)CC2CC23CC3)CCN(C(=O)CC2OCCO2)CC1 24095,c1(C(=O)NCC(CC)NC(c2c[nH]c(=O)cn2)=O)ccc(CN(CCC)C)cc1 24096,C(=O)(C(O)C(C)(C)C)N1CCC(CC=C)(C(=O)NCc2cncnc2)C1 24097,C12(N(C)C(C3(NC(=O)C=CC(=O)N(C)C)CCCC3)=O)CC(CN3CCSCC3)(C1)C2 24098,CC1CCn2cc(C(N3CCCNC(=O)C3c3ccccc3)=O)nc2C1 24099,c1(C(=O)NC2CCN(c3c(OC)cncn3)CC2F)cc(=O)n2[nH]cnc2n1 24100,N1(C(C=CCCC)=O)CCCC(CO)(NC(=O)Cc2nn(C)cc2SC)C1 24101,C=CC(C)(C)CCN=C(NCC=C(C)C)NC1CCN(C(=O)OCC)C1 24102,c1(C(N2C(CNC(c3c(C)cc(F)cc3)=O)CCC2)=O)cc2cccn2c(O)n1 24103,C1(C(=O)NCC#CCNC(C(CSC)OC)=O)CCCN(C(=O)OC(C)(C)C)C1 24104,Cc1ccccc1Oc1ccc(C(=O)N(C2CCN(C)C2=O)C)cc1 24105,c1(C2C(C(=O)NC(C)CC3CN(C(=O)CC4CSC4)C3)C2)ccncc1 24106,C(CC(O)CC(=O)NC1CN(C(=O)C(=O)N(C)C)CC1c1cccc(F)c1)SC 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24213,C(=O)(CCCCCN=[N+]=[N-])N1CC(CC)N(C(=O)CC(C)c2cnn(C)c2)CC1 24214,CCC(C)C(O)CC(=O)NCC(CC(=O)N1CCOCC1CC)OC 24215,c1(C(N(CCCNC(C(C)SCCCC)=O)C(C)C)=O)ccn(C(C)(C)C)n1 24216,c1(C(C)C)cccc(C(=O)NC2CC(NC(=O)CC3CCC(C)(C)C3)CC2O)c1 24217,N1(C(c2c(C(C)(C)C)ocn2)=O)CC(NC(c2ncccc2O)=O)C(C)(C)C1 24218,c1(C(=O)NC2(C3CN(C(CS(C(C)C)(=O)=O)=O)C3)CC2)cc2cc(Cl)cnc2o1 24219,CC1(C)CCCOC1CC(N1CCOC(CNC(C2CC(=O)N2)=O)C1)=O 24220,N1(C(C(C2CCC2)OC)=O)CC(CNC(C2CCCCC2O)=O)C(C)C1 24221,Cc1cc(C(N2CCC(CNC(c3ncccc3CO)=O)C(C)C2)=O)[nH]c1C#N 24222,C1(C(N2CCC(N(C(C(c3ccccc3F)C)=O)CCO)C2)=O)C(C)(C)C1(F)F 24223,Nc1ccc(CCCC(=O)NC2CCOC(CNC(=O)CNS(N)(=O)=O)C2)cc1 24224,Cc1ccc(S(=O)(=O)N2CCN(C3CCCN(C4CC4)C3)CC2)nc1 24225,Cc1ncnc(C(N2CCCC(N(C)C(C3CCS(=O)(=O)C3)=O)CC2)=O)c1C 24226,C=CC1CCCCN1C(c1cc(CNC(=O)C(=O)CC(C)C)no1)=O 24227,c1(COC(C(=O)NC2CCC(CCNC(C=CCC)=O)C2)C)ccc(C)cc1 24228,c1(C(=O)NC2CCN(C(CSC(C)C)=O)C(C)C2)cnn2ccccc12 24229,N1(C(C2CCC(C(CCCC)=O)CC2)=O)CC(NCCNS(C)(=O)=O)C2(CC2)C1 24230,c1(N2CC(OC)C(F)C2)nc(Nc2cc(N)ccc2F)c2cnn(C)c2n1 24231,n1(CC)cc(C(=O)NCCC2(NC(=O)CC3CCNC3=O)CCC2)c(C)n1 24232,Cc1ccc2c(C(=O)NC3CCN(C(=O)CC4CCOC4)C(C)C3)n[nH]c2c1 24233,c1(NC(=O)NC2CC(C(=O)OCC)C2)ccc(C)cc1.C12(CC=CC1)C(=O)NC2 24234,c1(C(N(C(CCNC(C2(SC)CC2)=O)C)C)=O)ccc(S(N)(=O)=O)[nH]1 24235,N1(C(c2c(C)ncc(Cl)c2)=O)CC2(CCN(C(=O)C3=CCCCC3)CC2)CC1C 24236,N1(C(COCCCC(C)C)=O)CCCN(C(c2cnc3c[nH]nc3c2)=O)C(C)C1 24237,C1(C(C(=O)NC(CNC(C(C)=C2CC2)=O)C2CCC2)C)CCOCC1 24238,N1(C(Cc2cncc(C)c2)=O)CCCCC1C1CCCN1C(=O)C=CC1CC1 24239,C1(C(N(CC(O)CNC(C2CCNC(=O)C2)=O)C)=O)CCS(=O)(=O)CC1 24240,Cn1cc(C(=O)NC2CC3(C2)CC3NC(C23CC4CC2C3C4)=O)ncc1=O 24241,C(=O)(CC(F)(F)F)NCC(=O)NCCN(CC)Cc1cccs1 24242,CC(N=c1[nH]c(N(C)CC2CCCC2O)nc2c1CCC2)c1nnc2n1CCC2 24243,C(=O)(C1=CCS(=O)(=O)C1)NCC1(CNC(CCC2CCC(=O)N2)=O)CC12CCC2 24244,C1(CNC(c2cnc(CC(C)C)[nH]2)=O)CCC(CNC(C2CCN(C)C2)=O)CC1 24245,FC1(F)CCC1CN1CCOCC1.C1(CC2=NOCC2)c2nnnn2CCN1 24246,C(=O)(C1CCc2c[nH]nc21)N(C(C(NOC(C)(C)C)=O)CC1CCC1)C1CC1 24247,C(C)(CCC(=O)NCC1CCC1NC(c1cnc(-c2ccccc2Cl)nc1)=O)OC 24248,C1(CNC(c2ccc(CC)[nH]2)=O)CC2(CCN(C(C3CC4CCC3CC4)=O)C2)CO1 24249,c12ccc(c(C#N)c1)[nH]2.C=CCC(CC=C)OC 24250,c1(C(N2CC(CC)N(C(C3CCC(=O)NC3)=O)CC2)=O)c(F)ccc(Br)c1Cl 24251,C1(NC(CN(C)CCO)=O)CC2CN(C(=O)C(c3ccccc3)N(C)C)CC2C1 24252,C1(CNC(CCn2ncc(C)c2)=O)(CO)CCN(C(c2sccc2C#N)=O)C1 24253,C12(CNC(C3(C)COC3)=O)CC1CN(C(=O)CCOc1ccccc1Br)C2 24254,n1(CC(=O)NC(CC=C)CNC(=O)C(C)C2(O)CCC2)cc(C2CC2)c(C2CC2)n1 24255,C(=O)(C1=NOC(C)C1)N(CC(Cc1ccccc1)NC(Cc1c(C)cco1)=O)C 24256,C1(C(=O)NC(C)CNC(c2cnoc2CC(C)C)=O)CCCC2(CC2)C1 24257,CC1(C)CC(C)(C(N2CC3OCCOC3C2)=O)CN1C(=O)C=Cc1cscn1 24258,C=CC(CC)CC(=O)N(CCCOCCN(C(=O)C=Cc1ccc(C)cc1)C)C 24259,n1(C(CC)C)ccc(=NC(=O)CC(CC(C)C)NC(C2C=CCCC2)=O)[nH]1 24260,N1(C(CCC=C)=O)CCC(c2ccccc2)(CNC(=O)CC2CCCOC2)CC1 24261,N1(C(c2c(COCC)cc[nH]2)=O)CC2CC(NC(c3ccncn3)=O)CC(C2)C1 24262,N1(CC(=O)NC(C)C)CCC(NC(=O)CC2CC2C)C1 24263,C(=O)(C1CCCc2scnc21)NC12CC(C(=O)NC(CCOCC)C(C)C)(C1)C2 24264,C(C)(CN=c1cnc2cc(F)c(F)cc2[nH]1)(C(C)C)NC(C(COC)C)=O 24265,C(C)(CSC)(C(=O)NC(c1cccnc1O)C)NC(CCc1ccc(C)s1)=O 24266,C1(C(N(CCC(=O)OC)C)=O)CCC(CNC(=O)CCc2nncn2C)O1 24267,C(=O)(C(CCC(N)=O)N(C)C)N(C(C)CNC(=O)CCOCC1CC1)C 24268,C1(C(=O)NCCCN2CCN(C(c3ncn(CC)n3)=O)CC2)CN(C)CC(C)O1 24269,C1(CNC(=O)Nc2ccccc2)COC2(CCCCC2)O1.C1CC(=O)O1 24270,Nc1cccc(C(N2CC(NC(=O)Cn3ncc(Br)n3)C2)=O)c1 24271,C(C(F)(C(=O)NCC1CCCC(C)C1)C(C)C)NC(COCCC=C)=O 24272,N1(C(C2C(C)(C)C2(F)F)=O)CCC(NC(c2ccnc(N(C)C)c2)=O)C12CCC2 24273,N(C(=NCCF)NCCC(=O)N1CCCC1)C(C)CN1CCCCCC1 24274,C#CCCCCCCCNC(=O)C(CC(N)=O)NC(=O)C(C(C)C)NC(C)=O 24275,C12(C(N3CC(CNC(C(C4CCCC4)OCC)=O)C3)=O)CC(C(C)(C)C)(C1)C2 24276,C1(NC(=O)NCC2C(C)(C)C2)COC(=O)N1 24277,C1(CNC(=NCC=C)NCC(C2CC2)C2CC2)CC2(C1)CC(F)(F)C2 24278,N1(C(C(CC=C)(F)F)=O)CCC(C2CCCN(C(=O)C=CC(C)(C)SC)C2)CC1 24279,C12(NC(C3CCC(C)C3)=O)CC(CNC(=O)CCS(C)(=O)=O)(C1)OC2(C)C 24280,c1(C(=O)NC2(C)CN(C(CCc3scc(C)c3)=O)C2)ccc(Br)nc1C 24281,N1(C(C(C(C)C)O)=O)CCCCC(NC(=O)C=Cc2cocn2)C1 24282,C1(NC(c2cnc(CC)[nH]2)=O)(CNC(c2cc3c(s2)CCC3)=O)CC2CCC1C2 24283,c1(C(=O)NC(C2N(C(C(N3CCOCC3)C)=O)CCC2)C)cc2ccccn2n1 24284,C1(C(=O)NCC(C)N(C)C(c2cnn(C3CCOCC3)c2)=O)CCCC12CCC2 24285,C(=O)(C(CO)C(C)(C)C)N1CC(CCNC(=O)Cn2ccc(O)nc2=O)(OC)C1 24286,N1(C(CCCC#C)=O)CCC(C(=O)N(C)C(C2CCCC2)C)C12CCC2 24287,c1(CC(=O)NCCC2CCCN2C(=O)CCc2cn[nH]c2)cn(C2CC2)cn1 24288,c1(NC(CNC(C2N(CC(=O)NCC3CC3)CCC2)=O)=O)cc(Cl)ccc1Cl 24289,N1(C(c2ncc(OC)nc2)=O)CC(CCNC(C2(S(C)(=O)=O)CC2)=O)OC(C)C1 24290,Cn1cc(C=CCNC(C2CC3CC3N2C(=O)C=CCO)=O)cn1 24291,N1(C(c2cnc(C)c(N)c2)=O)CCC2(CCCC2CNC(C2(O)CCC2)=O)CC1 24292,c1(C(=O)NCC2C(CNC(C(C)(C)OC(C)C)=O)C2)cn2c(n1)CCCC2 24293,Cc1c(F)ccc(C(=O)NCC2CCN2C(C2CC3(C2)CC(C)(C)C3)=O)c1N 24294,c1(NC(S(=O)(=O)c2cc[nH]n2)=O)ccc2ccnc(C(C)NC(C)C)c2c1 24295,C(N=c1nc2c(ncn2C)c(NC2CCCC2)[nH]1)c1c(CC)con1 24296,Fc1cc(CCNCCCc2nc(-c3ccccn3)cs2)ccc1Cl 24297,N1(C(c2ncc(CC3CCC3)s2)C(=O)NCCOCC)CCOC(c2cccs2)C1 24298,C1(C(=O)Nc2ccc(OCC)nn2)CCC(C)CN1C(c1cc(OC)n(C)n1)=O 24299,C1(CCNC(c2c(C)ocn2)=O)CCCN(C(C2CCCOCC2)=O)C1 24300,c1(CC=C)cccc(C(N2CC(OC)C(NC(c3cnn(C)c3OC)=O)C2)=O)c1 24301,C1(NC(C(c2cccnc2)C)=O)CC12CCN(C(C1CC(N=[N+]=[N-])C1)=O)C2 24302,C1(CC)(CC)CC(NC(C2CC2C2CC2)=O)CN1C(=O)CCCF 24303,C(C(=O)N1CCC(NC(=O)CCN2C(=O)CCC2=O)C1C)(C(C)C)SC 24304,c1(C(=O)NC(C)CCCNC(c2cn(CC(F)F)cn2)=O)cccc2nc[nH]c12 24305,N1(C(C)(C)C)CC(C(N2CCC2CNC(C2(c3ccsc3)CC2)=O)=O)CC1=O 24306,Cc1ccc(CO)cc1C(=O)NCC1CCCC1NC(=O)CN1C(=O)CCC1=O 24307,N(C(=NCCOc1ccccn1)NCCNC1CCC1)Cc1cccc(N(C)C)c1 24308,CCC(CC(=O)NC1(CCC(=O)NC(CC)CC(=O)OC)CCC1)C(F)F 24309,C1(C(=O)NOCc2cccc(Cl)c2)(CNC(CC)=O)CCCCC1 24310,c1(C(N2CCC(NC(C(C=C)O)=O)C(F)C2)=O)c(C)cc(O)cc1C 24311,Cc1cc(C(N2CCCN(CCNC(=O)CC34CCC(CC3)C4)CC2)=O)cc(N)c1 24312,C1(C(N2CC(NC(COCCC)=O)C(C)C2)=O)CCC2(CC1)CC(O)C2 24313,C(=O)(C1=NNC(=O)CC1)NC1C(NC(c2c(C)ccnc2O)=O)CCCC1 24314,CC1(C)CN(C(=O)C2=CCCCO2)CC1C(=O)NC1CC2C=CC1C2 24315,c1(OC)cccc(C(=O)NCC(C)CNC(c2cnc(CC(C)C)s2)=O)c1N 24316,c1(C(N2CC(NC(CC3ON=C(C)C3)=O)C(F)C2)=O)cnc2ccnn2c1 24317,C#Cc1ccc(C(=O)NCC2(C)CCCN2C(c2ccc(=O)n(O)c2)=O)nc1 24318,C(=O)(CC(C)C(C)(C)C)NCC1CCCC(C(=O)NCC(CC(=O)OC)O)C1 24319,c1(NC(C2C(C(N(CC#C)C)=O)C2)=O)cc(Br)cc(F)c1OC 24320,c1(C(=O)NCC2(NC(CCC(C)SC)=O)CC2)c[nH]c2c(C)c(C)ccc2c1=O 24321,Cc1c(C(=O)NCC2(CN(C(=O)C(C)CS(C)=O)C)CC2)ccc2c1CCC2 24322,c1(C(=O)NC(CCOC)CNC(=O)C=C(C)Cl)cccc(-c2ccncc2)c1 24323,c1(NC(C(CC)NC(CSCCCOC)=O)=O)ccc(OC)cc1 24324,CC1COCC(C(=O)NCC2CCC2C(=O)NCCN2CC(CF)C2)O1 24325,c1(C(=O)NC2CN(C(CSCC=C)=O)CC2C2CC2)c(C)[nH]cc([N+](=O)[O-])c1=O 24326,N1(C(CCSCCCC)=O)CCc2[nH]nc(CNC(C3(C)CC3(F)Cl)=O)c2C1 24327,C1(C(=O)OC)C(F)(F)C12CC(C(=O)N(C1CCN(C(=O)C(F)(F)CC3CC3)C1)C)C2 24328,c1(CC(=O)N(CC(CC)NC(C(C)SCC)=O)C)cccc2ncccc12 24329,Cc1n[nH]c(C)c1C(C)CC(=O)N1CCCC1Cn1cc(CCC#N)nn1 24330,C(=O)(N=S1(=O)CCNC(C2CC2(C(=O)OC(C)(C)C)C)C1)c1c(C)n(C2CCC2)nn1 24331,N1(C(C(=O)NCC)=O)CC=C(C(C)(C)C(=O)NCC2OCCC2(C)C)C1 24332,C1(C(C)NC(c2cn(C3CCOC3)cn2)=O)CCN(C(C2CCC2)=O)CC1 24333,C1(C(=O)NC2CNCC(F)(F)C2)Cc2ccncc2N1 24334,C(CC(C(=O)NCc1ccc(CC)cc1)NC(=O)C(C)n1ccnc1)=CC 24335,C123CC(C1)(OC2C)CNC3=O.CC1CCOC(C(=O)Nc2cc(C(N)=O)c[nH]2)C1 24336,Cc1ccnc(C(=O)NCCc2ncc(C(=O)NCc3cn(C)cn3)cn2)c1F 24337,c1(OC)cc(CN2CCC2C(=O)NCCC2CCCC2)cc(F)c1OC 24338,c1(NC(C(c2cccc(Cl)c2)OC)=O)ccccc1Br 24339,c1(CC(C)(C)C)ccc(C(=O)NC(CNC(c2ccn(C)c2)=O)CO)cc1 24340,c1(C2CCN(C(=O)OC(C)(C)C)CC2)ncnc2c1ncn2C1CCCCO1 24341,c1(CC2CN(C(CS)=O)C2)cn(CCCC)nn1.C#CC 24342,CC1CC(c2nnnn2CCCF)CS1.n1(CCNCCSC)cc(Br)cn1 24343,N1(C(CC2(COC)CCC2)=O)CC=C(CC(=O)N2CC(F)(F)CC2CCO)CC1 24344,N1(C(c2c[nH]cc2Br)=O)CCN(C(=O)CC=C(Cl)Cl)C2(CC2)C1 24345,N1(C(c2nc(C)oc2)=O)CC2(C1)CN(C(=O)CN(C)C(C1CCCCC1)=O)CCO2 24346,C1(C(N(C2CN(C(CCc3nc(C)sc3)=O)C2)C)=O)CCC(O)CN1C 24347,Cc1nc2ccc(-c3cncnc3C(=O)NCc3cncs3)cc2s1 24348,N1(CC(=O)NC(C)CCN(C)C(c2ccc(=O)oc2)=O)CCCCC(O)C1=O 24349,C1(C(=O)NC(C)C(=O)Nc2cccc([N+](=O)[O-])c2)NCCC12CCCCC2 24350,Cc1csc2c(NC3CCC(NC(c4ccccc4CO)=O)CC3)ncnc12 24351,c1(C(=O)NCC2CN(C(CCCOCCOC)=O)C(C)C2)cc(F)cc(Cl)c1O 24352,c1(C(=O)NC(c2cncc(F)c2)C2CCCO2)ccc(-c2nn[nH]n2)cc1 24353,C(=O)(CC(C)(C)C(F)F)N.C1(CCCC)CCN(C(=O)CNC(=O)C)C1 24354,C(CC(CC)C(=O)N1CCCC(OC2CC2)C1)=CC.C1(Cc2cn[nH]c2)C(=O)N1 24355,N=c1[nH]n(CCSc2cn(C3CCCC3)nn2)cc1Br 24356,c1(C(N2CCC(NC(C3(COC)CC3)=O)C2)=O)c(C)nc2sc(C)cn12 24357,C1(NC(Cc2c(C)scc2)=O)CCCC2CN(C(c3cnn(C4CC4)c3)=O)CC12 24358,C1(c2cn(CCCCNC(=O)Cc3n[nH]c(C)n3)nn2)(C(=O)OC)CCCO1 24359,c1(C(N(CCNC(=O)Cc2cnccc2Cl)CC)=O)cnc2n1CCS2 24360,CC(C)C(C(=O)N1CCCC(C(=O)N(CCC#N)CCO)C1)c1ccncc1 24361,CC1COc2c(C(N3CC(CNC(c4ncccc4N)=O)C3)=O)cnn2C1 24362,Cc1cc(NC(=O)CCCN(C(C)(C)C)C(C2CC3CCCC3C2)=O)cn(C)c1=O 24363,n1(CC)nc(C)cc1C(=O)NCc1ocnc1C(=O)NC12CC(C1)C2 24364,c1(C(N2CCCCC(n3cc(C4(CC)CCOC4)nn3)C2)=O)cnc(N)c(Cl)c1 24365,Cc1ccc(-c2ocnc2CNCSc2cncs2)s1 24366,C1(C(N(CC(CNC(CCOCC#C)=O)C)C)=O)COCCN1C 24367,CN=c1[nH]ccc(C(N2CCC(C)(C)C(CNC(=O)COC(F)(F)F)C2)=O)c1N 24368,c1(CC)ccc(CCN2CC(CNC(C=CCNC(=O)CC=C)=O)C2)s1 24369,CCCCC(CNC(=O)Cn1cc(C(C)O)nn1)NC(C1CCN1CC)=O 24370,C#CC1CCCC(c2nnnn2C2CCC2)(NCCCCC(N)=O)C1 24371,c1(CC)cccc(CC(=O)N(CCN(C)C)C(C2CCCC2)C)c1.C1(C)C(=O)N1 24372,c1(C(N2CCCCC(NC(c3scc(OC)c3)=O)C2)=O)cnc2nncn2c1C 24373,N1(C(C2CCCC(OC)C2)=O)CC2(CCN(C(=O)C(C)NC=O)C2)C1 24374,N1(C(CC)=O)CC(OC)CC1CNC(=O)CN(CCC)C(=O)OC(C)(C)C 24375,c1(C(C)=O)ccc(N2CCCC3(NC(c4c[nH]c(C)c4)=O)CC3C2)c([N+](=O)[O-])c1 24376,C1(NC(C=C(COC)C)=O)CN(C(C2CCC(OC(F)(F)F)C2)=O)CC1N=[N+]=[N-] 24377,c1(N(C)Cc2cn(C3CC(O)C3)nn2)ccc2ncccc2c1 24378,C(=O)(C(C)C(F)(F)C(F)F)NC1(CCCNC(c2cc(CC)c(F)cc2)=O)CC1 24379,Cn1c(C(=O)NCC2CCCC(NC(=O)C(C)(C)C3CCC3)C2)cc2ccsc12 24380,c1(C(N(C)CC2CCN(C(C(C3CC3)OC)=O)CC2)=O)cc2n(c1)CCC2 24381,n1(CC(=O)NCC2CC(NC(c3coc(C(F)F)c3)=O)C2)cc(Cl)cn1 24382,CC1CN(C)CC1NC(C1CCN(C(C2CCNC(=O)C2)=O)CC1)=O 24383,c1(N(C(NNC(=O)C2(OC)CCOC2)=O)C)ccc2nncc(C(F)(F)F)c2c1 24384,CC(C)C(C(=O)NCC=CCNC(c1ccc(C2CCOC2)s1)=O)n1cnnc1 24385,C(CC)(CCCC(=O)NC(c1ccc(O)cc1)C)NC(C(C1CCC1)OCC)=O 24386,CCCCC(CO)NC(=O)CC1CC(NC(=O)CN2CCNC(=O)C2)C1(C)C 24387,C1(C(=O)NCCCN(CC)CC)(NC(=O)CCSC)CCOC1 24388,Cc1cc(Cl)c(C(=O)NCC2(C)CCCN2C(=O)CSCc2ccncc2)cn1 24389,c1(OC)cc(NC(C23CC2CN(C(c2cc(C)n(C)c2)=O)C3)=O)ncn1 24390,c1(NC2C(OC)CC(COC)C2)[nH]c(=NCC(CC2CC2)OC)nc2c1ncn2C 24391,CC1CCCC(N=c2nc(N3CC4C=CCC(C4)C3)c3c([nH]2)CCC3)C1 24392,C1(COC)(NC(c2cnccc2C)=O)CCN(C(=O)C(C#N)C(C)C)CC1 24393,C1(C(N2C3CC(N(C(CSC)=O)C)CC2CC3)=O)CCc2cnc(C)n2C1 24394,c1(CNC(C2C(CCC)C2)=O)csc(C(N2CC(O)(COC)C2)=O)c1 24395,CCC(C)C(C(=O)NC(C)CCSC)N(C)C(c1cccc(C)c1C)=O 24396,C1(C(N2C(CNC(C(N3C(=O)CCC3=O)C)=O)CCCC2)=O)CCC=CCCC1 24397,N1(CC)Cc2nccn2CC(NC(c2cccc(-n3cc(C4CC4)nn3)c2)=O)C1 24398,C(=O)(CCC(CF)CF)NCC#CC(=O)NCCC1CC(O)C1 24399,C1(NC(c2c(C)scc2)=O)CN(C(C2CCC2C(C)(C)C)=O)C2(CCC2)C1 24400,C(CS(=O)(=O)CC(=O)NC(C)(C)CC(F)C(=O)NCc1nnnn1C)OC 24401,C1(C(=O)OC(C)(C)C)(C(N2CC(O)CC(O)C2)=O)CC12CCCCC2 24402,c1(C(=O)NCC2(C(=O)NCc3cnc(CC)[nH]3)CCCC2)cccn2ccnc12 24403,Cc1c[nH]c(C#N)nc1=NCc1ccc(F)cc1.C1CC(N)C1 24404,Cc1ncc2n1CCC(C(=O)NCC(C)NC(c1ccc(CF)cc1)=O)C2 24405,C1(NC(C(CCCCC)O)=O)CCN(C(c2cccnc2OC)=O)CC12CCC2 24406,c1(C(C(=O)N(CC(=O)NCC(C)N(C)C)C)C)cccc(O)c1 24407,C(C(CC(C)C)C(=O)N(C)Cc1ccncc1)NC(C(CCC)CC)=O 24408,Cc1cccc(Br)c1CC(N1CCCN(c2cc(O)ncn2)CC1)=O 24409,N1(C(C(CC2CCCC2)NC(C2CCC(=O)O2)=O)=O)CCC2(CCC2)CC1 24410,c1(CCCC(=O)NC(CNC(C2CCOC2)=O)C2CCC2)ccccc1Cl 24411,C(=O)(C1=C(F)CN(C(=O)CN2CCC(OC)C2)CC1)N1CC(CC)OCCC1 24412,C(=O)(CC(C)(C)C1CCCCC1)NCC(CCOC)NC(=O)C(F)OC 24413,N1(C(C2=CCN(C(=O)CCC3CC3(F)F)C2)=O)CCn2ccnc2C1 24414,c1(C(=O)NCCNC(CC2C(C)(C)C2)=O)cocc1Br 24415,N1(C(c2ccc(C)cc2)=O)CCC(NC(C2CCC(CO)CC2)=O)C(F)C1 24416,C=CC1(C(=O)NCc2cnn(C)c2C(N2CCC3(CC3)C2)=O)CCCC1 24417,n1(CC=C)nc(-c2cccc(Br)c2)nc1C1CCCCC1O 24418,C(=O)(CCc1ccco1)OC.n1(CC(=O)NC(C)CC2CC2)cnc(=N)[nH]1 24419,C(=O)(C(C)(C)C(=O)Nc1cc(F)cc(F)c1)NCC1(O)CCN(C(C=CC)=O)C1 24420,Cc1ccc(F)cc1C(=O)NC(C1CCN(C(=O)CC2OCCCC2(C)C)C1)C 24421,C(=O)(C(F)C(F)(F)F)Nc1cccc(NC(CC(OC)Nc2ccccc2)=O)c1 24422,Cc1c(Br)cnn1CC(=O)N(CC(C)NC(=O)C(F)=C1CCC1)C 24423,CC(C)CS(=O)(=O)CCC(=O)NCC(C(C)C)NC(=O)CP(C)(C)=O 24424,CC1(C)CC(CC(=O)NCC2CCCOC2)N(C(N2CC(CO)C(O)C2)=O)C1 24425,C1(CCNC(C2C(COC)C2)=O)CC(F)(F)CN1C(=O)CCc1nc[nH]n1 24426,CCCCCC(CC)C(=O)NC1C2CCC1N(C(=O)C=Cc1cccc(Cl)c1)C2 24427,c1(N2CCC(NC(C(CCC)(C)C)=O)C(O)C2)ncc([N+](=O)[O-])cn1 24428,N1(S(=O)(=O)CC2CC3CCC3C2)CC=CC12CCCCC2 24429,N1(C(c2cc(F)cc(C)c2N)=O)CCOC2(C1)CN(C(=O)OC(C)(C)C)C2 24430,Cc1cc(CCC(N2CCCC(N(C(=O)CC3(CO)CC3)CCO)C2)=O)nn1C 24431,N1(Cc2cn(C(C)C)nn2)CCCC(C(=O)NCC2(n3cccn3)CC2)C1 24432,N1(N(c2nc3ncc(C(=O)OCC)cc3o2)C)Cc2ccc(F)cc2CC1C 24433,C1(C(=O)NCCCNC(c2c(N)cc(Cl)nc2)=O)CCOC2(CCOCC2)C1 24434,c1(C(=O)NCC2CC(NC(CCc3nnc(C)n3C)=O)CC2O)c(C)ncnc1O 24435,c1(N2CCC(S(=O)(=O)NC)C2)ccc(S(=O)(=O)NC(CO)C2(C)CC2)c(Cl)c1 24436,C1(OC)CC2(C1)CN(C(=O)C(O)CCNC(c1cc(C)c(C)[nH]1)=O)C2 24437,C1(C(=O)NCCCC(C)NC(Cc2cccc(OC)c2)=O)CCCC(C#N)C1 24438,CC1(C)CN(C(=O)CCn2ccnc2)CC(C)(C)C1NC(c1ccc[nH]1)=O 24439,C1(NC(=O)C=CCN2CCOCC2)CCN(C(=O)CCc2cn[nH]c2)CC1F 24440,C(=O)(CC(O)CC(C)C)N1C(C(=O)NC2C(OC)C(C)(C)C2)CC(C)C1 24441,C(C1CCN(C(C2CC3(CCO2)CC3)=O)CC1)=CC(=O)NCc1ccccc1O 24442,C1(c2c(C)cco2)NC(=S)N(CC2(CF)CCC2)C2=C1C(=O)NC2c1ccccc1 24443,C(C(=O)N1OC2CCC1CC2)N(C(=O)C(F)C1CCCC1)CCOC 24444,C1CCC2(CC1)OCCO2.Cc1nc(-c2nnc(-c3ccco3)o2)[nH]c(=N)c1Br 24445,C(C)(CCCNC(=O)C(C)Sc1nncn1C)NC(CC1C(OC)CC1)=O 24446,c1(C(C)C)ccc(C(c2nnnn2C2COC2)NCC2(CCO)CC2)cc1F 24447,Cc1cc(O)cc(=O)n1CC(N1CC(CNC(=O)CCC(C)(F)F)C2CC12)=O 24448,C1(NC(C2(CNC(C)=O)CC2)=O)CN(C(C)=O)C(C)(CO)C1.C1(=O)CN1 24449,C=C=CCCC(=O)NCc1cc[nH]c1C(N1CCC(O)CC1)=O 24450,CCCC(C)CC(=O)N1CC(NC(=O)CCCc2ccccc2)C(O)C1 24451,N1(C(C2SCCN(C(CN(C)C)=O)C2)=O)CCN2C(=O)CCC2C1 24452,c1(C(N2CCC(CNC(C(C#C)(C)C)=O)C23CC3)=O)ccc(=O)n2c1CCCC2 24453,N1(Cc2nccc(C(=O)OC)c2)CCC(NC(=O)Cn2cc(Cl)cn2)C(C)(C)C1 24454,C(=O)(C(O)C(C)CC)NC1(NC(CNS(CCCC)(=O)=O)=O)CC1.C[SH](=O)=O 24455,N1(C(C(CC)NC(N)=O)=O)CC2CC2C1C(=O)NCc1nccn1C(C)C 24456,c1(NC(CC(C)F)=O)sc2c(c1C(=O)Nc1cccnc1)CCCC2 24457,c1(OCCNC(N(CC(c2cccc(F)c2)C)C)=O)ccc(Cl)cc1 24458,N1(C(=O)Cc2cnc3cccnn23)CCc2c(Cl)ccc(Br)c2C1 24459,N#Cc1ccc(CN2CCCC(C(=O)Nc3cc(I)ccc3Cl)CC2)cc1F 24460,c1(C(=O)NCCC(C)NC(=O)CCCc2n[nH]c(=N)s2)cnc(N(C)C)nc1 24461,Fc1cc(Cl)cnc1C(N1CC2(CC3CC2C3)C1)c1ccccc1 24462,C(=O)(C(C)(CNC(=O)CCc1nc(O)n[nH]1)CC)NCC(N(OCC)C)=O 24463,C(=O)(C(C)C(C)CC)N(CC(CNC(c1nc(C(=O)NCC=C)sc1)=O)(C)C)C 24464,c1(C(=O)NCC2OCCCN(C(CSC(C)C)=O)C2)cccc2nc(O)[nH]c12 24465,N1(C(CC(=O)OC)=O)CCC2(CC1)CCN(C(=O)Cc1ccc(SC)cc1)C2 24466,C(CC(C(=O)NCCc1cc(C)ns1)NC(C1CCN1C)=O)OC 24467,N1(C(CCCOC)=O)CC2CCCC(N(C(=O)CC3CCCC34CC4)C)C2C1 24468,CC#CCCCC(=O)NCCOCCCN(C(=O)C(c1ccn(C)n1)C)C 24469,C(=O)(C(CCC(C)C)NC(c1ccnn1CCC)=O)NC(C=C)C1CCC1 24470,CCC(O)C(C)C(=O)N1CCCC1C1(C(=O)NCc2cc(C)co2)CC1 24471,c12ccc3nc(sc3c1)N1CC(CO)(C1)N2CC.c1(C(N)=O)c[nH]nc1C1CC1 24472,N1(C(c2c(SC)cn(C)n2)=O)CC(C)(CNC(=O)C(F)(F)C2CC2)CC1(C)C 24473,N1(C(C(CC)F)=O)CC2(C1)CN(C(c1ccc(C3CCOC3)cc1)=O)CC2CO 24474,CCC(C)(F)C(=O)N(C)CCNC(C1CCCCN1C(C)=O)=O 24475,C1(C(N2CCC(CNC(c3ccc(CO)o3)=O)C2)=O)CCC=CCCC1 24476,c1(OC)cccnc1C(=O)N(C(CNC(=O)CSc1nnnn1C)C1CC1)C 24477,N1(C(c2ccc(C)nn2)=O)C2CCC1C(CNC(c1cnc(C(C)C)s1)=O)C2 24478,C(C(C)(O)CC)NC(C1C(=C)C1C(N1CC(C(C=CC2CC2)OC)C1)=O)=O 24479,CC1CCSCCN1C(C(=O)NC1CC(F)(F)C1)C1CCOC1 24480,C(=O)(C(C)(C)C(C)(C)C)NCC1(C(=O)NCc2cccc(C)c2O)CCCCC1 24481,Cc1ncnc(C)c1CC(N1CCC(F)C(NC(C2CCC3CC2CO3)=O)C1)=O 24482,C1(CC=C)(C(=O)NC(C)(C)CCN(C)C)CCN(C(=O)CN2CCCC2C)C1 24483,N1(C(C2C(C)CCN2C(=O)CCC(N)=O)=O)CC2(CCCCCC2)C1 24484,c1(-c2n(CC=C)ccn2)[nH]nc2ccc(C(=O)Nc3cccc(N)c3)cc12 24485,c1(-c2cccc(CO)c2)ccc2c(c1C(=O)NN=c1cccn[nH]1)OCO2 24486,C1(NC(c2c(C)nc(C)[nH]2)=O)CC2CC(C1)CN(C(c1ccc(O)c(C)c1)=O)C2 24487,C1(C(=O)NC(c2cnn[nH]2)C)CC=CCN1C(C1COCC1C(N)=O)=O 24488,CCC(F)(F)C(=O)N1CCOC(CCNC(c2cnnn2C2CCOCC2)=O)C1 24489,N1(C(C(C)C2CCC2)=O)CCOC2(CCCN(C(c3cc(Cl)ncc3F)=O)C2)C1 24490,c1(C(=O)NC(C2CN(C(=O)CC(C)(C)c3ccccc3)C2)C)cccnc1S 24491,N1(C(CCSCCCC)=O)CCC(CCOC)(NC(=O)C(CC)NC(=O)OC)C1 24492,Cc1ccccc1CC(N1CCC(NC(=O)CSc2ccccc2Cl)C2CC12)=O 24493,C(=O)(C1=NNC(C(F)(F)F)C1)NCCNC(COCCCOC)=O 24494,N1(C(CCOCCSC)=O)CC(NC(=O)CC23COC(C)(C2)C3)CC12CCOC2 24495,C=CCCC(C)(C)C(=O)N1C2CCC(C2)C1C(=O)NCc1oc(C(N)=O)cc1C 24496,C1(C(=O)NC2C(CC(=O)NCc3ccsc3)CCC2)OC2CCC1C2 24497,C(CCC(=O)N1CC2(CCC2O)C1)(C(C)C)NC(c1cccc(CC)n1)=O 24498,c1(C(=O)NCC(CC)(CC)NC(=O)C(O)CN(C)C)nc2n(c1Cl)CCCC2 24499,N1(CC(N2CCC(C(C)C(=O)NCCc3ccccn3)C2)=O)CCC(=O)CC1 24500,CC1CC(C(=O)NCCNC(=O)CCN(CCCO)CCO)C1 24501,c1(CN2CCC(C(=O)NCc3cnccc3Cl)C(O)C2)cccc2c1OCCO2 24502,c1(CN(C)Cc2ccnn2C2CCOCC2)cccc2c1OC(F)(F)O2 24503,N1(C(c2c(CC)c[nH]n2)=O)CC2CCCN(C(=O)C(C)O)C2C1 24504,N1(C(CSCC#C)=O)CCn2ncc(N(C)C(c3ccc4nncn4c3)=O)c2C1 24505,C1(C(=O)NC2C(NC(Cc3cn(C)nn3)=O)CC2)CC2CCCC(C1)C2 24506,c1(CNC(C(=O)N(C)CC2CC2[N+](=O)[O-])=O)cncc(F)c1 24507,Cc1cc(C(N2CC(CC(=O)NC3CCCC3(C)C)CC2C)=O)nc(O)n1 24508,N1(c2nc(CC)nc(C)c2)CC2(CCCC2NC(c2ccc3c[nH]nc3c2)=O)C1 24509,N1(C(c2cncc(Cl)n2)=O)CCCC(F)(CNC(=O)C(F)(F)C2(O)CCC2)C1 24510,C1(C(=O)N(CC)CC)(OCC)CCN(C(c2ccc(C)o2)C)CC1 24511,N1(C(C(C)c2ccco2)=O)CCCN(C(c2ccc(Br)s2)=O)CC1CO 24512,C1(NC(c2cnc(C)nc2)=O)CC2(C1)CN(C(C1CCC(C(F)(F)F)CC1)=O)C2 24513,Cc1cc(C(=O)NCCC2(C)CCN(C(c3nnn(C)c3N)=O)CC2)ncc1Cl 24514,C(C1CCN(C(C2CCCC(=O)N2C)=O)CC1)=CC(=O)NC(C1CSC1)C 24515,C1(NC(C(CO)NC(CCCCCOC)=O)=O)CCC(N=[N+]=[N-])CC1 24516,Cc1nn(C)c(C(=O)N(CCCNC(=O)C(C)C(C)C)C)c1Cl.N12CCC(C1)C2 24517,C1(CC(=O)NCCC2CCN(C(C3(O)CC(F)(F)C3)=O)C2)CCCOCC1 24518,c1(C(=O)NC2CC(NC(CCc3cc(C)on3)=O)C2)cc2c(C)cc(F)cc2[nH]1 24519,N1(CC)CCOC(C(N2CCOC(CN(C(=O)CC(F)(F)Br)C)C2)=O)C1 24520,CCN=C(NCc1cccc(C)n1)N1CCC(CC(C(=O)NC)C(F)(F)F)CC1 24521,C(=O)(CC(C(F)F)NC(c1c(O)noc1C)=O)Nc1ccc(OC)nc1 24522,Cc1oc(C)c(C(N2CC(CNC(c3cnn(CCC(C)C)c3C)=O)C2)=O)c1C 24523,Cc1ccc(F)c(C(=O)NNC(=O)N(c2cccc3[nH]ncc23)C(C)C)c1F 24524,N1(C(C2CC(N(C)C)C2)=O)CCC(NC(C2CCC(C)(C)OC2)=O)C(O)C1 24525,N1(C(CN(CCC)C)=O)CC(C(=O)NCc2ccnc(Cl)c2)C2(CCC2)C1 24526,C1(CN(C(=O)C(C)Cc2cnc[nH]2)CC)CCCCN1C(=O)C(C)OCC(F)(F)F 24527,C(C)(C)(CCC(=O)N(C)Cc1ccon1)NC(C(CC)NC(N)=O)=O 24528,Cc1nccc(C(=O)NCCOC2CN(C(C3CCC(C)NC3=O)=O)C2)c1C 24529,c1(C(=O)NCC2C(C)CN(C(c3cccc(C(N)=O)c3)=O)C2)c(F)ccnc1F 24530,N1(C(C(CC)NC(=O)CCc2cnccn2)=O)CCOC(C)CC1 24531,C1(CNC(CSCC)=O)CCC(C)CN1C(c1ccnn1CC(C)C)=O 24532,C1(CNC(=O)CCC2CCCC2)CCCN(C(c2ccc(C(F)(F)F)nc2)=O)C1 24533,C1(N(C(c2occc2C2CC2)=O)C2CC2)CC2CN(C(=O)C=CC3CC3)CC2C1 24534,C(CC(=O)NCC(C)(CC)OC)(C(C)(C)C)NC(c1c(CC)csc1)=O 24535,c1(C(=O)NCC(CC)NC(=O)C(F)(F)c2cnn(CC)c2)cscc1C 24536,C(C1CCc2ccccc21)NC(=NCCC)NCC1CCCCN1C(C)C 24537,Cc1ccc(C(=O)NC2CCN(C(=O)CC3(C)OCCO3)C2)cc1Br 24538,C12(C(N(CC(CN(C(=O)C(=O)Cc3ccccc3)C)O)C)=O)CCOC(C)(C1)C2 24539,Cc1c(NCC(C)N(C)C)ncnc1NCCCOc1ccc(F)cc1 24540,N1(C(CSC)=O)Cc2ccnn2CC(NC(=O)C(C)CC(C)(C)C)C1 24541,C(=O)(C(C)(C(F)(F)F)c1ccccc1)N(CC(C)NC(=O)CC(C)(F)F)CC 24542,N1(C(C2CCC3(CC2)CC3)=O)Cc2ccccc2C(NC(C2CCCCS2)=O)C1 24543,CC(C)C(C)(C)C(=O)NCC(CC1CCCC1)C(=O)N(C1CCCN(C)C1)C 24544,c1(NC(CC(CC=C)NC(=O)COC2CCCC2)=O)ccc2occc2c1 24545,c1(N2CC(CC(C)C)OCC2)nc(=NCC2CCC2)[nH]c2ccc(Cl)cc12 24546,N1(C(CCCOC(C)=O)=O)CCCC(C)(CNC(=O)Cc2csc(C3CC3)n2)C1 24547,C1(n2ncc(C(=O)OC)c2)CCCN(C(=O)C(N2CC(C=O)CC2OC)C)C1 24548,Cc1occc1C(=O)NC1CC(C)(NC(c2ccon2)=O)C1 24549,CC1(C)CN(CC23CC(C2)C3)C1c1nccn1Cc1ccccc1Cl 24550,C1(CCN(C(CC(C)F)=O)C)CCN(C(=O)CC2CCC23CCC3)CC1 24551,c1(NC(C2N(Cc3cnc(C)nc3Cl)C3C(C2)C3)=O)ccc(O)c([N+](=O)[O-])c1 24552,c1(C(=O)NCCC(C)NC(c2cc[nH]n2)=O)cc2c(s1)CCCNC2=O 24553,c1(C(=O)NCC(NOCC)=O)ccnc(CNC(=O)C(C)(O)CC)c1 24554,c1(NC(C)C)ccc(C(=O)NC(C2CCCN2C(c2ncc(Cl)n2C)=O)C)cc1 24555,c1(C(=O)NCC2C(NC(=O)Cc3ccc(F)c(F)c3)CC2)cc2c(s1)CCCC2 24556,C1(F)(C(=O)NC2(CC#C)CC2(C)C)CCN(C(c2ccsn2)=O)C1 24557,C1(CC)C(NC(=O)CC(C)OC(C)C)CCCN1C(=O)COCCOC 24558,N(C(=NCCC(C)=O)NCCc1nc2c(s1)CCCC2)C1C(CC)OCCC1 24559,Cc1cn2c(n1)CC(C(=O)NCC1CC13CCN(C(c1nncs1)=O)CC3)C2 24560,C(=O)(CCCC(F)(F)F)NC1(C2N(C(C3C(C)(C)C(F)(F)C3)=O)CCCC2)CC1 24561,c1(C(CC2CCCC2)NCC(CO)OC)nnnn1C1CCCCC1 24562,N1(C(CC=C(C)C)=O)CCOCC1CNC(C1(c2ccc(Cl)cc2)CCC1)=O 24563,C1(C(=O)NC2CC2)(COC)CCCN1C(=O)COCC(C1C2CCC(=O)C12)=O 24564,N1(C(CCc2n(C)ccn2)=O)CC2(CO)CC1(C(=O)NC1CCCC1(C)CO)C2 24565,c1(C(=O)NC2CCCN(C(C3C(C)C3)=O)C2)ccc2c(c1)CC2 24566,c1(C(=O)NC2(CNC(C(C)SC(C)C)=O)CCOCC2)ccc2c(c1)NC(=O)C2 24567,C1(NC(c2ccc(NC(CC)=O)cc2)=O)CC2(C1)CN(C(c1ncnn1C)=O)C2 24568,C1(CC(C(=O)OC)NC(=O)C(O)COCCOC)CCC(C)(C)CC1 24569,N1(C(COC)=O)CCCC2CN(C(c3ncc(C)cc3C)=O)CCC12 24570,N1(C(c2cc(C(C)=O)oc2C)=O)CCCC2(CCN(C(=O)C(F)CC3CC3)C2)C1 24571,c1(CC)cccc(C(=O)NCCC2CCN(C(=O)CS(=O)(=O)NC)C2)c1O 24572,N1(C(Cc2c(C)cco2)=O)CCCC12CCN(C(C1CC1CC(C)(C)C)=O)C2 24573,c1(CC(=O)NCC(CNC(Cn2ncc(CC)c2)=O)O)ncncc1Cl 24574,N1(CC(CS(CC)(=O)=O)=O)CCC(NC(=O)Cc2ccccc2C)C(F)(F)CC1 24575,C1(C(=O)NCCN(C(=O)CCS(C)=O)CCOC)CCCCC1(F)F 24576,c1(-c2cn(C3CC(NC(=O)Cn4cccnc4=O)C3)nn2)cccc(Cl)c1Cl 24577,C#CCCC(O)C(=O)NCC1CCN(C(c2ccc(F)c(C)c2)=O)C1(C)C 24578,N1(C(c2c(CC)n[nH]c2)=O)CCCN(C(=O)C(COC)COC)CC1C 24579,N1(C(CC(C)(F)F)=O)CC2CC(NC(c3ccnc(C(F)F)c3)=O)CC1C2 24580,C1(NC(C(C)=C2CC2)=O)CC2(C1)CN(C(C1(C(C)C)CC1)=O)C2 24581,CC(C)CC(C)C(=O)NCCNC(=O)CN1CC2C(C1)C2(F)F 24582,C1(CN(C(C2(OCC)CCC2)=O)C)CN(C(=O)CNC(=O)C(C)CC)C1(C)C 24583,N1(C(c2c(C)con2)=O)CCN(C(c2c(C)nn(C)c2F)=O)CC(O)C1 24584,N1(C2CN(CC(N)=O)C2)C=NC2=NC(=O)CN(C3CCC3)N12.C=O 24585,N(C1CCOc2c(F)cc(F)cc21)C(C(C1(COC)CCOCC1)(F)F)=O 24586,N1(C(CCSc2n(C)ccn2)=O)CC(CNC(c2cc(=N)[nH]n2C)=O)C2CC12 24587,N1(C(C(C)O)=O)CC(NC(c2ccc(F)c(SC(C)(C)C)c2)=O)CC(F)C1 24588,C(=O)(C1=CCS(=O)(=O)C1)N1CCC(NC(=O)COCC2CCCOC2)C1 24589,Cc1c(C(=O)NCCC2(O)CN(C(=O)Cc3cscn3)C2)cccc1N 24590,N1(CC(C(C)C)(C)O)CCC2(CC1)CN(C(=O)C(C)NC(=O)C(C)(C)C)CCO2 24591,C1(C(C(=O)NCCC(C)NC(=O)C(Cl)=CCl)(C)O)CCC(F)(F)CC1 24592,CCC(CC(=O)NC(C)(C)C=CC(N1CCC(C(N)=O)CC1)=O)C1CC1 24593,n1(C(C)C)ncc(C(N2CC(O)(CCNC(C3CC(CF)C3)=O)C2)=O)c1N 24594,C1(C(=O)NC(CCSC)C(=O)N(C)CC2COCCO2)CCCCCCC1 24595,c1(CNC(=O)NC2CN(C(=O)OC(C)(C)C)C2)ccc(Cc2cnc(Cl)s2)s1 24596,c1(C(N(C)CCNC(=O)CCc2cocn2)=O)ccc(Cl)cc1N 24597,N1(C(C(C)NC(N)=O)=O)CCN(C(c2ccon2)=O)CC12CC2 24598,c1(CC)nccnc1C(=O)NC(CNC(c1ccccn1)=O)C1CC1 24599,C(=O)(CC(CC=C)c1ccccc1)N(CC(=O)NC1C(C=C)COC1)C 24600,c1(C(=O)NCCCCC2(NC(C(C)n3ccnn3)=O)CC2)cc2cccnc2[nH]1 24601,C1(C(C(=O)OC)F)CCN(S(=O)(=O)CC2CCC(SC(F)(F)F)O2)C1 24602,N1(C(c2c(CC)noc2)=O)CCC(C)(N(C(=O)CC2(n3ccnc3)CC2)CC)CC1 24603,C12(C(N3C(C)(C(C)C)CC3)=O)CC(C)(CN1C(=O)CCCn1cncn1)C2 24604,CC(F)(F)CCC(=O)NN1CCCC1C(N1CC(C)(C)C12CCC2)=O 24605,c1(C(=O)NC2(CC)CCN(C(=O)CN(C)S(N)(=O)=O)CC2)cccc2sncc12 24606,C1(C(=O)NC2CCC(OC)C2)CCN(C(=O)CCc2cnco2)C1C 24607,C1(NC(COCCOCC)=O)C=CCN(C(=O)C=Cc2ncco2)C1 24608,C1(C(N2CCC(N(C(=O)CCC3CCCC3)C)C2)=O)CC(=O)N(C)C1 24609,c1(OCC)ccc(C(=O)NC2CCC2NC(=O)CC(n2nc(C)cc2C)C)nc1 24610,CC1CCC(C(=O)NCC(=O)NCc2ncccc2F)CC1 24611,c1(C(N2CCN(C(c3c(CC)nc[nH]3)=O)C(CO)C2)=O)c[nH]c2nc(F)ccc12 24612,c1(C(=O)NC2CCN(C(c3cccc4nccn34)=O)C2)ccc2c(c1)COCO2 24613,C1(C(=O)NCC(CN(C)C(C2(c3cncnc3)CCCC2)=O)(C)C)CCCC(=O)O1 24614,C123CN(CC1CS(=O)(=O)C2)C3.CCCCN=C(NNC(=O)C1CC1)NC(C)C(C)C 24615,Cc1c(-c2c[nH]nc2C(N2CCCC2C2CC2)=O)cccc1S(C)(=O)=O 24616,N1(C(C#CC)=O)CCC(CCNC(=O)CC(c2ccc(C(F)(F)F)cc2)C)CC1 24617,C(C(=O)N1CCCC1C(C)(C)NC(c1sc(N(C)C)nc1C)=O)(C(C)C)NC(C)=O 24618,Cc1ccc(C(=O)NC2(C)CCN(C(C3(C)CCN(C)C3)=O)CC2)c(C)c1 24619,c1(C(=O)NC2C(CC)N(C(c3cnn4c3OCC4)=O)CC2)ccn2ncccc12 24620,C(CCC(C(=O)NC(C)(C)C)N1CCC(c2nnc(C)s2)CC1)OCC 24621,c1(OC)ccccc1C(N1CC2CC1C2CNC(=O)C(c1ccc(F)cc1)=O)=O 24622,c1(C(N(CCCNC(C2CC3(CC3)CO2)=O)C(C)C)=O)cc(Cl)c(N)cc1F 24623,n1(CCC(N2CC(C(N(CC#N)CC#N)=O)C(O)CC2)=O)ccc2ccccc12 24624,N1(C(=O)NC(c2c(C)ncc(Br)c2)C)CC2(CC(O)c3nccn32)C1 24625,N1(C(C(COCC)C)=O)CCCCC1C1CCN(C(c2cnc[nH]2)=O)CC1 24626,C1(C2CCN(C)CC2)(C(=O)NC2C(OC)CN(C(C3CCCC3(F)F)=O)C2)CC1 24627,C(=O)(C(C)N(OC)C(=O)CCCCCN(C(=O)CSCc1ccccc1)C)OC 24628,CC(C)CCN=C(NC(CC)CCCO)N1CCC(Oc2cccc(Cl)c2Cl)C1 24629,CCS(=O)(=O)C=CC(=O)NC1CC(NC(=O)COc2cnccc2C)C1 24630,N1(C(COC(CCC)=O)=O)CCn2nc(C)c(I)c2C1 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24648,c1(C(N2CCC(NC(C(C=C=C)C)=O)CC2)=O)cc(Br)c2ncccc2c1 24649,c1(NC(C(=O)N(CC(C)NC(c2n[nH]cc2C)=O)CC)C)ccccc1 24650,C1(CC(=O)NC(C2CCCC2)CNC(CCc2n(C)cnc2)=O)CCC=CCC1 24651,Cc1ccc(F)c(OCC(=O)N(CC(C)NC(c2ncn3c2CCC3)=O)C)c1 24652,C1(C#N)(C(=O)NC2C3(CC(NC(CC=C=C)=O)C3)C2)CC12CCC2 24653,n1(CC(=O)N(CC)CC2CN(C(=O)CC3CC3C)C2)cc(CNC(C)=O)nn1 24654,Cc1cc(Br)cc(C(N2C3CCC2(CNC(=O)COC(C)C)CC3)=O)c1N 24655,c1(C(=O)NC2C(C)CCN(C(c3nc(C)sc3C)=O)C2)cc2c([nH]1)CCCC2 24656,N1(C(=O)CC2C=CCC2)CCC2CCN(C(c3ccc(O)nn3)=O)CC2C1 24657,c1(C(N2C(CC(N3CCCC(C#C)C3)=O)COCC2)=O)ncnc2sc(Br)cc12 24658,Cc1c(C(=O)NCCOCCNC(=O)CC(C)n2ccnc2)ccn1C(C)C 24659,CCCC(C(=O)N1CC(NC(N)=O)CC1C(=O)NCCC(C)(C)F)OC 24660,c1(OC)cc(NC2CC2)ccc1C(=O)NC(C)(CNC(=O)C(=O)C(C)(C)C)CO 24661,CC1(C)COc2cc(CNC(N3CCCC3c3nncs3)=O)ccc21 24662,c1(-c2c(C(=O)OC)scc2)cn(C)nc1CNC(c1nccnc1Br)=O 24663,N1(C(c2c(OC)csc2)=O)CC(C)(CNC(C2CC3CCC2CC3)=O)CC1(C)C 24664,C1(C(=O)NCC(CNC(C(C)Cc2cnc[nH]2)=O)F)C2CC3C(C2=O)C13 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24683,c1(C(C(=O)NCC(C)C)N(C)CCC2CCCCN2C)c(Cl)nc2sccn12 24684,N1(C(C2=CCC(NC(C(CCC)=CCC)=O)C2)=O)CC2CCCCC12C 24685,C1(CN2C3CCN(C3)CC2=O)CCS(=O)(=O)C1.C(C)(C)(C)OCC 24686,CC1(C)CC2(CN1)CN(C1CCN(CC(F)(F)F)C1=O)C2 24687,c1(CNC(COC(Cc2cncc(C)c2)=O)=O)cccc2ccccc12 24688,N1(C(c2c(CC)cno2)=O)CC(NC(c2cc(N)cc(O)c2)=O)CC(O)C1 24689,N1(C(C(c2cn(C)nn2)NC(c2ccc(OC)nn2)=O)=O)CCC(O)C(O)C1 24690,CC1CCc2n[nH]cc2C1C(=O)NC1CC2CCC(C1)N2CCS(C)(=O)=O 24691,CCCC(CCC)CCCC(=O)NC(C)(CNC(=O)CC1CC=CC1)CO 24692,n1(CC(=O)NC2C(NC(C(C)C(F)(F)F)=O)CCCC2)ccc(=O)n(C)c1=O 24693,N1(C(C(C)CC(C)(C)C)=O)CCC2(CC1)CCN(C(C1COC(=O)N1)=O)CC2 24694,c1(CC(N2CC(N3CCN(CCO)CC3)C2)C)cc2c(ncn2C)s1.C(=O)C1CC1 24695,N1(C(c2csc(-c3ccccn3)n2)=O)CCC2C(CCCN2C(c2ccsn2)=O)C1 24696,N1(C(=O)NC(CCC)C(=O)OC)CC(OC)CC(C)C1 24697,CC1CCN(C(=O)CSS(C)(=O)=O)CC1CNC(c1nn(C)cc1Cl)=O 24698,C1(c2cc(C)[nH]n2)CCCCCN1C(C(=O)NC1(C)CC1)C1CC(C(F)(F)F)C1 24699,CCC(CC)C(C)C(=O)NC1CCC(C)(CNC(c2cc3[nH]ccc3s2)=O)CC1 24700,c1(CNC(CC2(C)CCN(C(=O)C(F)(F)C3CCCC3)C2)=O)cnc(O)c(F)c1 24701,C1(CNC(CC(C)SC)=O)CCCN(C(c2ccc(NCC(N)=O)cc2)=O)C1 24702,N1(C(C(C)SC)=O)CCC2C(C1)NC(=O)CN2C(c1cncn1C)=O 24703,c1(-c2c(C)cnc(F)c2)cccc2c(C(=O)NCC(C)O)n[nH]c12 24704,C1(C(=O)NC(C)C(C)NC(=O)CNC(=O)CC2CCCC2)CCOC(C)(C)C1 24705,c1(C(N2CCCC(C3N(C(COCC=C)=O)CCCC3)C2)=O)ncc(Cl)cc1O 24706,C1(C(=O)NCC(C(C)C)NC(CCc2ccc(C(=O)OC)[nH]2)=O)CC(C)(C)CN1C 24707,C1(CC(N2CCC(OCC=C)CC2)=O)CN(C(=O)CN2CCOC2=O)CCC1C 24708,N1(C(c2ccc(C#C)cc2OC)=O)CCCC12CCCN(C(c1ccon1)=O)C2 24709,O=C(CCCC(F)F)NCC12CCC1CCN2C(c1cc(Cl)nnc1O)=O 24710,C1(NC(COC2(C)CCCC2)=O)CCC2(CC1)CC2NC(c1ccncn1)=O 24711,N1(C(CCOCC#C)=O)CC=CC1CNC(=O)C(C)OCCN(C)C 24712,Cc1ccn2ncc(C(=O)NCC3(F)CCCN(C(=O)C(C)OCC4CC4)C3)c2n1 24713,N1(C(C=Cc2c(C)ncs2)=O)CCN(C(c2occc2Br)=O)C(C)CC1C 24714,C12(C(=O)NC(C(C)C)(C)CNC(=O)C=CC(F)(F)F)CC(C)(C1)OC2C 24715,Cc1c[nH]c(=NC(=O)C2CCC(NC(=O)Cc3c[nH]c4ccccc34)C2)c(Br)n1 24716,c1(C(=O)NC2(CNC(C3CCCC(OC)C3)=O)CC2)ccc(P(C)(C)=O)o1 24717,c1(C(=O)OC)ccc(C(=O)NCC(C)NC(=O)CCCSC)cc1Cl 24718,c1(C(=O)NCC(C)NC(=O)Cc2cc(F)ccc2Cl)cc(F)c2cn[nH]c2c1 24719,c1(OCC)cccc2[nH]c(C(=O)NCCCN(C(c3ccoc3)=O)C3CC3)cc12 24720,C1(OCC)CC(CCNC(c2ccnc(C)n2)=O)N(C(=O)C(C)OCC(C)C)C1 24721,c1(C(=O)NCC2N(C(C3C(C)CCC3)=O)CCOC2)nn2c(c1Br)CCC2 24722,c1(COC)nc(N2CCC(NC(C3(S(C)(=O)=O)CCC3)=O)C2)cc(C)n1 24723,c1(OC)cc(CN2CCCCC2c2ccc(Cl)s2)cc(C(C)(C)C)c1O 24724,Cc1cnncc1C(=O)NCC1CN(C(c2coc(CC3CC3)n2)=O)CC1O 24725,C1(NC(c2ccncc2Br)=O)CN(C(C2CCCCO2)=O)CC(F)(F)C1 24726,C(=O)(CC(C)(O)C(F)(F)F)N1CC(C(C)NC(c2c(C)cc(C)[nH]2)=O)OCC1 24727,c1(CC(C)NC(CCSCC)=O)ccc(CNC(c2ccncc2F)=O)cc1 24728,CS(=O)c1ccccc1C(=O)NC1CN(C(C2CC3(CCC3O)C2)=O)C1 24729,CC1CN(C(=O)C(F)(F)c2ccccn2)CCC1N(C(=O)CSC(F)F)C 24730,c1(NC2SCCN(C(C(C)OCC=C)=O)C2)c(Br)ccc2n[nH]cc12 24731,Cc1n[nH]cc1CC(=O)NC(CO)C(C)NC(=O)CC(C)n1cccn1 24732,Cc1ncnc(C)c1C(N1CCC(C(C)NC(c2cnn3c2CCC3)=O)CC1)=O 24733,C1(F)(NC(=O)COCC2CCC2)CCC(CNC(c2ccn(C(F)F)n2)=O)C1 24734,C1(C(=O)NC(C2CCCN2C(=O)CC2CCSC2)C)CCC(=O)C1 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24753,c1(CC)nn(C)cc1C(=O)NCC(CC)NC(=O)C(C)Cc1cccc(F)c1 24754,c1(C(N2C(CC)CCCC2)C(=O)NC2CCOC2)cc(=O)n2ccccc2n1 24755,C(c1ccc2cc(OC)ccc2c1)=CC(=O)NCCNC(CCC(=C)C)=O 24756,c1(C(=O)NCC2CCN(C(C(C)=C3CCCC3)=O)C2)cccn2c(C)nnc12 24757,Cc1csc(=NCC(=O)N2CCC3C(C2)CN3C(=O)CCNC(=O)CO)[nH]1 24758,C(=O)(C1CCCc2nc[nH]c21)NCC1(NC(c2cscc2Cl)=O)CC1 24759,C1(C(=O)NCC2C(NC(c3nc(OC)c(C)s3)=O)C2)CCc2ncnn2C1 24760,c1(NC(CCC)c2ccco2)cc(N2CC3CN(c4ccccc4)C3C2)nc(C)n1 24761,C=CCC(CNC(c1ccc(CC)o1)=O)NC(=O)CCSCc1ccccc1 24762,c1(CN2C(C3CCN(C(CCC(C)C)=O)CC3)CCC2)ccc2n[nH]cc2c1 24763,N1(C(c2c(C)[nH]nc2C(F)F)=O)CC(NC(=O)C=Cc2cnc[nH]2)CC(O)C1 24764,C(=O)(C(O)CSc1ccccc1)N(CCNC(C(C)=CC1CC1)=O)CCOCCO 24765,C(CNC(C)=O)(C(C)(C)C)NC(=O)CCCN.C(CC(=O)C(C1C(C)C1)=O)N 24766,C(=O)(C1CCCc2nccn21)NCC(C)(CNC(c1cc(N)ccc1F)=O)OC 24767,C(=O)(CS(=O)(=O)CCOC)N1CCC(C(=O)NC2CCCCCC2O)(CC)CC1 24768,Cc1n[nH]c(C)c1SCC(=O)NCC1CCCN1C(=O)CC1CCOCC1 24769,c1(NC(CC2N(C(C(C)(C)c3cccnc3)=O)CCC2)=O)nc(Cl)c(Br)cc1O 24770,N1(C(CC(C)OC)=O)CCCC(NC(c2ccc(NS(C)(=O)=O)nc2)=O)CC1 24771,C(=O)(C(CN(C)C)CC(C)C)NC1(CC#C)CCC1.C12(CCCCC1)CC(=O)N2 24772,C1(CNC(C(C)n2cccn2)=O)CC2CC2N1C(=O)C=CCN1CCOCC1 24773,Cc1cccnc1CC(=O)NC1CC(C(N2CC(NSC(F)F)C2)=O)C1(C)C 24774,c1(OC)cc(F)c(CN2CCCC(C(C)NC(c3ccc(Cl)cc3)=O)C2)c(F)c1 24775,c1(C(C(=O)NCC2(F)CN(C(C3CC(OC)C3)=O)C2)(C)F)ccc(F)cc1 24776,c1(OC)c(CC(=O)NC2CN(C(=O)CCC(N)=O)CC23CC3)cccc1Br.C(C)(=O)O 24777,c1(NC(C(C)NC(C2CC(C)(CN)C2)=O)=O)cccc(OC(F)(F)F)c1 24778,Cc1ccc(C(=O)NCC(=O)NC(C)CNC(=O)CCc2cc(Cl)no2)c(C)c1 24779,c1(OC)cc(C(=O)NC(C)C(c2ccccc2)NC(=O)CC2CC23CC3)ccn1 24780,c1(CCC)cc(C(=O)NC2CN(C(=O)CNS(C)(=O)=O)CC2C)c(C)o1 24781,C1(C(=O)NC2CCCN(C(=O)CCSC(F)(F)F)C2)CCc2cnnn2C1 24782,C(CCCCCN)N(C(=O)CC1CCC1)C.C1(N)CCS(=O)(=O)C1 24783,C1(NC(C(C)CNC(=O)CN(C)CCO)=O)CCCOC12CCC2 24784,c1(SC)cc(C(=O)NC2CC2CNC(C2(C)CNC(=O)C2)=O)nn1C 24785,c1(CN2CC(F)(CNC(c3cnc(C)nc3Cl)=O)C2)c(F)ccc(Cl)c1Cl 24786,c1(CCC(=O)OCc2ccccc2)cccc(OC(C2CC(Cl)(Cl)C2)=O)c1 24787,c1(C(=O)NCC(CC)NC(C2C3CC(=O)CC23)=O)nc(C)oc1C 24788,C(C(=O)NC(CC1CC1)C(=O)N(C)CC1CCN(CC)C1)(C(C)C)SC 24789,c1(OC)ccccc1OC(C)C(=O)NCCC(C)N(C)C(c1c[nH]c(C#N)c1)=O 24790,C1(OCC(=O)OC)CCN(C(C2CN(C(c3ocnc3C)=O)CCS2)=O)CC1 24791,C12(C(N3CC(=CC)C3)=O)CCCC1CCN2C(c1cnnc(C)c1C)=O 24792,CN1CCC(CC(=O)NC(C)(CNC(=O)CNS(C)(=O)=O)C2CCC2)CC1 24793,N1(C(C2CC23CCCC3)=O)CC2CCC1C(C(=O)Nc1cccnc1)C2 24794,C1(NC(C2(CC)COC2)=O)CC2CC1N(C(C1CCCNC1=O)=O)C2 24795,CCC(C(=O)N1CC(CNC(C2CC2c2ccn(C)n2)=O)C(C)C1)C(C)C 24796,Cc1cc(C(N2C3CC2CN(C(c2cccc(C)c2I)=O)C3)=O)cc(Br)c1 24797,Cc1ccc2cc(C(=O)NC3CCCC3(C)CNC(=O)C(=O)N(C)C)cnc2c1 24798,c1(CC2N(C(=O)NCC3CCC(C(C)C)N3)CCC2)ccc2c(c1F)CCC2 24799,Cc1cc(Cl)c(C(=O)NCC(C2(O)CCN(C(=O)CC3=CCCC3)CC2)C)cn1 24800,c1(OC)cc(C=CC(N2CCC(NC(=O)C(F)CC3CCCC3)C2)=O)sn1 24801,c1(CC(=O)N(c2nccnc2Cl)Cc2cc(F)ccc2Cl)ccc2c(c1)CNC2 24802,N#Cc1ccc(Cl)c(C(N2CCC2CNC(C2CCOC23CCC3)=O)=O)c1 24803,c1(CCOC)n[nH]c(=NC2(CNC(=O)Cc3c(Br)cnn3C)CCCCC2)s1 24804,O=C(C(CC1CCC1)N1CCCC1C1(c2ccccc2)CC1)NCCC1CC1 24805,C1(NC(=O)NCCC2CC(CC)C2)CCC2(CC1)CSC2 24806,c1(C(=O)NCC2C3CN(Cc4cccc(C)c4Br)CC32)ccc2scnc2c1 24807,C1(C(=O)NCc2ccc(C(C)NC(=O)CC)o2)CCC(CC(C)(C)C)C1 24808,Cn1nc(C(N2CC(CNC(c3cnoc3C3CCCC3)=O)C2)=O)cc1Cl 24809,CC1CC2(C(N3CCCC3Cn3cc(CCN(C)C)nn3)=O)CC12 24810,C1(C(=O)NCCC2(CNC(COCC=C)=O)CC2)CC=CCO1 24811,c1(C(=O)NC(CN(C(c2ccc(F)c(O)c2)=O)CC)C)ccc(C)cc1OC 24812,N1(C(c2ccc(C(C)C)s2)=O)CCC(NC(=O)CCN2CCCC2=O)C1(C)C 24813,CC(CC(=O)N1CCC(N(CC(C)C)C(C2CCC(O)C2)=O)CC1)C(F)(F)F 24814,C=CC(CC(=O)NCC1CN(C(c2oc(CC(C)C)nc2C)=O)C1)c1ccccc1 24815,c1(CNC(C(=O)NCCCC(=C)C)=O)nc(Cl)ccc1Cl 24816,c1(OC)ccc(CNC(=O)C(C2CCC2(F)F)N2CCCC2C(C)(C)C)c(C)c1 24817,N1(C(C2CCCCN(C(c3cnc(C)nc3)=O)C2)=O)CCCC(C2CCC2)C1 24818,c1(CN2CCC(NC(C(c3ccnn3C)C)=O)C(O)C2)ccc(F)c(C#N)c1 24819,C12(CNC(c3c(CC)nco3)=O)CCC(Nc3ncc(Cl)c(C)c3C#N)(CC1)CO2 24820,C(C(=O)NCCCC(C)NC(=O)CN(C)C(c1cccs1)=O)(C(C)(C)C)SC 24821,Nc1nc(C(=O)N(Cc2scc(CSC)n2)CCF)ccc1Br 24822,C=CC(C)(O)CC(=O)N1CCC(C(C)(C)C(=O)NC2CCOC2=O)C1 24823,N1(C(Cc2c(C)non2)=O)CCC(C)(NC(=O)COc2cscn2)C1 24824,CC(O)C(C)C(=O)NC1(CNC(=O)CCCc2cccs2)CC1 24825,N1(C(CC2N(CC)C(=O)CC2)=O)C2CCC1CN(C(C1CN(S(C)(=O)=O)C1)=O)C2 24826,C(=O)(CCCCC#N)NCC1CN(C(C=CCOC)=O)C(C)C1 24827,C1(NC(CCN(C)CC)=O)CC2CC(C1)N(C(=O)Cc1ccccc1Cl)C2 24828,c1(OC)nc(Cl)ccc1C(N1CCCCC(NC(C2CCC(C)(C)CO2)=O)C1)=O 24829,C(=O)(C1=CCC(C)(C)CC1)NC1(CCCCNC(c2cc(C)sc2C)=O)CC1 24830,C(=O)(CCCC(N)=O)N1CCC(NC(CC2C(C)C2(F)F)=O)CC1 24831,CCN=c1[nH]cc(C(N2CCCC2CN(C)C(c2cn(C3CC3)nc2C)=O)=O)s1 24832,CCC(C)(COC)C(=O)NCC1CN(C(=O)CC(C)(C)C)CC1c1cncn1C 24833,C1(C)(C(N(C2CCN(C(Cn3c(C)c(Cl)cn3)=O)C2)C)=O)CC2CCC(C1)S2 24834,N1(C(c2nc(Cl)c(Cl)s2)=O)CCc2sccc2C1c1ccccc1 24835,c1(NC(Cc2cccc(OC)c2)(C)CO)ncnc2cccc-2c1N 24836,Cc1cnc(C(N2CC3CC2C3C(=O)N(C)C(C2CCC2)C)=O)c(F)c1 24837,c1(OCC)ccc(C)cc1C(=O)N(CCCNC(C1C2CCC12)=O)CC 24838,c1(OCC)ccc(Cl)c(C(=O)NCC(C)N(C)C(C2CC2c2cccs2)=O)n1 24839,N1(C(CC(C=C)(C)O)=O)CCC(C)(C)C(NC(c2cccc(Br)c2C)=O)C1 24840,c1(CC(=O)NC)ccc(OC)c(OC(F)F)c1.C(=O)(C(C1CCC1)OC)N1CC1C 24841,Cc1cccc(C(CNC(C2CN(C)C(=O)N2)=O)NC(=O)Cn2cnnc2)c1 24842,N1(C(Cc2cncc(C)c2)=O)CC(C)(CNC(C2CCCCO2)=O)CC1(C)C 24843,C1(C(N2CCC(C3N(C(CCC(=C)Cl)=O)CCC3)C2)=O)CCc2cnc(C)n2C1 24844,C=C=CC(C)C(=O)NC1(C(F)F)CC(NC(=O)CCCOCCOC)C1 24845,N1(C(c2ccc(C3CC3)s2)=O)CC2CCCC(N=c3ccn(CCF)nn3)C2C1 24846,CCC(CCCC(=O)N1CC(C)(O)CO1)NC(C12CCCC1C2(F)F)=O 24847,N1(C(CCC(C)OCC)=O)CCN(C(c2cnc(C)s2)=O)CC1CC(C)(C)C 24848,CC1=C(C(=O)NC(C(=O)NCC2(C)CCC(=O)N2)c2ccco2)CC1 24849,N1(CC(=O)N(CC=C)CC2CC2)CC(c2ccccc2C)OCC1C 24850,CCCCC(C)C(C(=O)NCSc1ccccc1)N1CCN2CCC1C2 24851,c1(CC(=O)N(C(CCNC(C=NOC)=O)C)C)cccc2c(C)coc12 24852,C=CC(CCC)CC(=O)N1CCCC1(CC)C(=O)NC(c1ccnc(F)c1)C 24853,C1(NC(C2CC(=C)C2)=O)CC2CCC1CN(C(c1cn(C3CCOC3)cn1)=O)C2 24854,C(=O)(CCC(C)(C)O)NCCCNC(c1ccc(CC(C)C)cc1)=O 24855,C1(COC)(NC(=O)CCNC(N)=O)CCN(C(C2CC3(CSC3)C2)=O)C1 24856,N1(CCC2CCC(C)O2)CCN(CC2CCCC2)CC1 24857,c1(C(=O)NC2CCC(N(C(CCN(C)CC)=O)C)C2)cc(C)ccc1C(=O)OC 24858,C1(NC(CCCOCCOC)=O)C2CCC1N(C(C1(CCF)CC1)=O)C2 24859,c1(C(N(C2CCN(C(=O)CCc3ncco3)CC2)C)=O)ccc(F)c2c1OCC2 24860,O=C(CC1CCOc2ccccc21)NC1CN(C(c2nccc(Br)c2)=O)C1 24861,Cc1cc(-c2cncc(CN3CCOC(C(C)C)C3)c2)c(C)cc1O 24862,C1(C(=O)NCC=CCC(C)C)CCCCC1(C)NC(=O)C=Cc1cncs1 24863,CCC(C)(C)C(=O)N(CCNC(c1ccnc(C(C)C)n1)=O)CC1CC1 24864,C1(NC(=O)CCOCC2CCC2)CN(C)CCCN1C(=O)C(CC1CC1)OC 24865,c1(-c2c(C)cc(C(=O)N=c3cc[nH][nH]3)cc2)ccc2c(c1)CNC(=O)N2 24866,c1(OCCC)ccc(CNCCCCC2CN(C(=O)C(CC)N(C)C)C2)cc1 24867,C1(Sc2ccccc2)CC(C(=O)N(C2CC3CNC2C3)CC(C)C)CCC1O 24868,Cc1cc(CN(C(=O)C(Cc2cn[nH]c2)NC(C2(CO)CCC2)=O)C)no1 24869,c1(CN2C(C(CC)O)CCCC2)ccc(Cl)c(Br)c1 24870,CC1(CNC(c2cc(N)ccn2)=O)CCCN1C(C1CC2CC2C1)=O 24871,C=CC1(C(=O)NCC(C(C)C)NC(c2cncc(OCC(F)F)c2)=O)CCOCC1 24872,c1(C(=O)NCC(CC=C)NC(=O)CCn2ccccc2=O)cc(Cl)ccc1N 24873,CCCC(C)C(=O)NC1CC(F)(CNC(C2(N3CCOCC3)CC2)=O)C1 24874,C1(C(N)=O)CCC(C(N2CC(C(N)=O)(CN(C(=O)Cn3cnnn3)CC)C2)=O)CC1 24875,n1(CC)cnnc1C1CN(C(=O)NOC(C)C(=O)NCCO)C1 24876,N1(CCC(C)C)CC(C(=O)NC(C)(C)C(C)NC(c2ccc(F)cc2)=O)CC1=O 24877,C1(NC(C(CCOC)C)=O)CC2(CCN(C(C3(c4cc(C)on4)CC3)=O)CC2)C1 24878,c1(CCC)ccc(N)c(C(=O)NCC=CCNC(=O)C=CC2CCC2)c1 24879,C1(NC(C(C)N(C(=O)C=C2CCCC2)C)=O)CNC(=O)C1 24880,N1(C(C2=NOC(C)C2)=O)CCCC2CN(c3nc(Cl)nc4c3SCC4)CCC12 24881,C=CCC(CC=C)C(=O)NC(CN(C)C)C(=O)NCC(=O)NCC1CCC1 24882,C1(CNC(C=C(CC)C)=O)CN(C(c2cc(C)[nH]n2)=O)CC12CCC2 24883,C(CC(C)CNC(C1C(NC(C2CC(Cl)(Cl)C2)=O)C1(C)C)=O)OC 24884,c1(CCN)cc(C(=O)NCC(C)(O)C2CC2)sc1Cl.C1(C)CC1 24885,N1(C(C2(C)CC2(F)F)=O)CC(CNC(c2csnc2C2CC2)=O)C2(CCC2)C1 24886,N1(C(C(COCC)(C)C)=O)CC2CC(NC(=O)CCC3CCOC3)C1C2 24887,c1(C(=O)NCC(CN(C(C(N2CCN(C)CC2)C)=O)C)O)ccccc1[N+](=O)[O-] 24888,N1(C(CCCOC(C)=O)=O)CC2CCN(C(C3CCc4n[nH]cc4C3)=O)C2C1C 24889,C1(N(C(CC(C)F)=O)C)CS(=O)(=O)C12CCN(C(=O)CCCF)CC2 24890,c1(C(N2CCC(NC(C3CC4(CC4)CO3)=O)C23CC3)=O)noc2c(F)cccc12 24891,C(=O)(C(C)(C)CN1CCOCC1)NCC(CNC(C1(n2nccn2)CC1)=O)OC 24892,Cc1ccnc2sc(C(=O)NCC3CC3NC(=O)Cc3ccc(O)c(F)c3)c(C)c12 24893,CC1CN(C(C2CCC(C(C)(C)O)CC2)=O)CCC1CNC(C1(C)CC1Br)=O 24894,C1(=O)CCN1.C(=O)(C(c1ccoc1)CC)N(CC)C.C(=O)(CN(C1CC1)CC)NC 24895,C12(C(=O)NCC3C(NC(CN(CC)CC)=O)CCCC3)CCCN(CC1)C2 24896,CC(C)CC(CNC(=O)CCc1ccc[nH]1)C(=O)Nc1ccccc1N=[N+]=[N-] 24897,c1(CC)onc(C(N2CCOC(C(=O)NCC(C)(O)CO)C2)=O)c1C 24898,C1(C(=O)OC)CN2CC12.C1(Oc2ccccc2Cl)CC(=O)C1(C)C 24899,C(C(O)CC(=O)NCCC(C)N(C)C)NC(CCNC(=O)NC)=O 24900,CN1CCC(N=c2[nH]c(=NCC3(CC4CC4)CC3)c3sccc3[nH]2)CC1=O 24901,C(c1c(C)noc1C)=CC(=O)NCC1(CNC(C=C(C)C(C)(C)C)=O)CCCC1 24902,C1(NC(C(C2CC2)OCC)=O)CCN(C(c2cn(CCF)nn2)=O)C1C1CC1 24903,C(CNC(C1(CNC(C2CC2c2csnc2C)=O)CC1)=O)(C(C)C)OC 24904,C(C(=O)NCC1CC(CNC(c2csc(C3CC3)n2)=O)C1)(C(C)O)OC 24905,C1(C(N2CC(C)OCC2)=O)C2CC3C(C2N(C(c2ccccc2F)=O)C2CC2)C13 24906,c1(Nc2nc(-c3ccc(OC)nc3OC)sc2)ncnc2c1ccn2C 24907,C(=O)(C1=Cc2cc(Br)ccc2OC1)NC1CCN(C(C)=O)CCC1(F)F 24908,c1(N2CCN(CC3CN(C(C)=O)C3)CC2)cc(NC(C)CCCCO)nc(C)n1 24909,c1(OC)ccc(C2CC2C(=O)N(C(C)CNC(=O)C(F)(F)c2nccs2)C)cc1 24910,CCC(C)(CC)NC(C1CC(CCNC(=O)CC(=O)N(C)C)C1)=O 24911,C1(NC(c2c(NC)scc2)=O)CCCCN(C(C2CCC(NC3CC3)CC2)=O)C1.CCS 24912,C1(C(=O)NCCCCN(C)C(C2(C(F)(F)F)CC=CCO2)=O)CC12CC(C)(C)C2 24913,C(=O)(C(C)CS(=O)(=O)NC1CCC(CS(N)(=O)=O)C1)OC 24914,CCC(c1ccccc1)=CC(N1CCC(C(C)(O)CNC(=O)CSC(F)F)CC1)=O 24915,C1(C(=O)NCCCN(C(C2CC(C)CO2)=O)CC)CCCOCC1 24916,c1(NC(C(=O)NC(c2ccc(C(F)(F)F)cc2)CC)=O)cc(C)c(Br)c(Cl)n1 24917,N1(C(C2C(OC)CCC2)=O)CCCCC(C(=O)NCCC2(CO)CCC2)C1 24918,N1(C(=O)Cc2cccs2)CCC2(CCN(C(c3cc(Cl)c4n[nH]cc4c3)=O)C2)C1 24919,C1(CC(=O)NCC(C)N(C)C(c2n[nH]cc2C2CCC2)=O)CCn2cncc2C1 24920,C(N=c1cc[nH]c(C#N)n1)C1CN(C(CC2(OC)CC2)=O)CC1C 24921,C1(C(=O)NC2CN(C(C(C)OCC=C)=O)C(CO)C2)CC12CCOCC2 24922,C1(NC2(C(=O)O)C(CC)CN(C(c3ccccc3Br)=O)C2)COCCC1(F)F 24923,c1(CC(=O)N(CCNC(C2C(=C)CC2)=O)C)cc(F)cc(Br)c1 24924,C(=O)(C1SCc2cccnc21)NC(CCN(C(c1cc(COC)[nH]n1)=O)C)(C)C 24925,C(=O)(C1CCc2c(F)cccc21)N1C2CN(C(c3cc4scc(Cl)c4[nH]3)=O)C(C2)C1 24926,C1(c2nc(C3C(SCC)OCC3)on2)CCOC(C)C1 24927,C(=O)(C(C)(C)CNC(=O)CCCOC(C)C)NCC(C1CC1)OCC 24928,c1(C(C)=O)cccc(CC(=O)NCC2CC(C)N(c3nnc(CO)s3)C2)n1 24929,c1(OC)cc(I)c(C(N2C3COC(CF)(C2)C3)=O)cc1OC 24930,c1(COCC(=O)NCC2CC2NC(=O)CCc2cnco2)nncs1 24931,N1(C(C2C(C)(C)C2(F)F)=O)CCC(CNC(=O)Cn2ncc(O)nc2=O)C(O)C1 24932,N1(CCC(=O)NC(CN(C(c2ccncc2)=O)CC)C)CCCCCC1 24933,c1(C(=O)NC2C(C)(C)N(C(=O)CCCC#N)CC2)ccc([N+](=O)[O-])cc1Cl 24934,C=CCC(C(=O)NCC(C)N(C(c1[nH]nc2ncccc12)=O)CC)C(C)C 24935,c1(C(=O)NC2CC(NC(CS(CC)=O)=O)C2)cc(O)nc2cc(F)ccc12 24936,C1(C(N(C(C)CCNC(=O)CN2CCCC2C)C)=O)COCCOC1 24937,C(C(=O)Nc1cn(C)nc1C1CCCN(C(=O)COC2CC2)C1)(C(C)C)SCC 24938,C1(O)(CNC(C(C)c2ccco2)=O)CN(C(=O)CCSCC(F)F)C1 24939,c1(C(N2CC(O)(CNC(c3ncn(C(C)(C)C)c3)=O)C2)=O)ccc2c(c1)COC2 24940,C1(NC(c2cc(C)nn2C)=O)CS(=O)(=O)C12CCN(C(C1CCC=CO1)=O)CC2 24941,CC1(CNC(C2CCC(N(C)C)C2)=O)CCCN1C(=O)CCC1CC1(F)F 24942,C1(CC#C)(C(N2CC(NC(=O)C(C)(CO)NC(=O)NC)C2)=O)CCOCC1 24943,Cc1cc[nH]c(=N)c1C(=O)NC(CNC(=O)C(C)c1cccs1)C1CC1 24944,c1(OC)ccc([N+](=O)[O-])c(C(N2CC(F)CC2C(=O)NCC2CCOC2)=O)c1 24945,C1(CNC(C(C)CCO)=O)COCCN(C(c2cnc3n2CCC3)=O)C1 24946,S(=O)(=O)(c1cc(C)ccc1C)N(C1CN(CC(CC)CC(C)C)C1)C 24947,c1(C(N2CCC(C3N(C(CC4C(C)C4)=O)CCCC3)C2)=O)ccc(CO)cc1F 24948,c1(OC)cc(OCC(N2CCN(CCN3CCC(C)C3)CC2)=O)cc(COC)c1 24949,c1(C(=O)NC(CNC(C(C(C)C)(C)O)=O)C)coc(S(N)(=O)=O)c1 24950,CCCCC(CC)C(=O)N1CCCC(C)(C(=O)NC(c2ccc(C)cn2)C)C1 24951,C1(OCC)CN(C(=O)CCC2CCC(=O)NC2)CC1CNC(C1CC2(CC2)C1)=O 24952,c1(C(N2CCCC(NC(C3CC3(F)F)=O)C2)=O)c(OC(F)F)cccc1Br 24953,c1(C(N2CCC(C(C)NC(c3scc(OC)c3)=O)C2)=O)n[nH]c2ccccc12 24954,Cc1cc(C(=O)NCC2CCCC2C(N2CCCC(C#N)C2)=O)cc(O)n1 24955,c1(NC(=O)COC(CCCn2c(C)csc2=O)=O)ccc2c(c1)CCNC2=O 24956,CC(C)(C)C(C(=O)N1CCC(NC(=O)CC2CCC3CC3C2)CC1)n1ccnn1 24957,Cc1ccc(C)c(C(=O)NCc2ccc(C(=O)N(C3CCCC(O)C3)C)s2)c1 24958,N1(C(CC(C)C2CCC2)=O)CCC2CCCC12C(=O)NCC(=O)NC1CC1 24959,c1(C(N2CC3CN(C(c4ccccc4F)=O)C3C2)=O)ccc2ccccc2c1O 24960,c1(CC)cc(C(=O)NCC(C)N(C(=O)C(C)n2cncn2)C)cn(C)c1=O 24961,N1(C(C(C2CCN(C(CCCOCCC)=O)C2)F)=O)CCCC2C(O)CC12 24962,N1(C(c2snc(OC)c2Br)C(=O)NCC2CCOCC2)CC(C)(C)C(F)(F)C1 24963,c1(C(N2CC(C=C)(CC(N3CC(O)CC(O)C3)=O)C2)=O)ccc(C#N)c(C)c1 24964,C1(NC(C(C)C(C)O)=O)CC2CCCC(C1)C2NC(=O)Cn1ccc(O)nc1=O 24965,C(CCCC(C)(C)C(=O)NNC(=O)C1CSC1)NC(c1cc(C)c(C)nn1)=O 24966,Cc1nc(=N)[nH]c(C)c1C(N1CC(NC(c2ccc(C(C)C)cn2)=O)C(C)C1)=O 24967,c1(C(=O)NC(C)C(C)NC(C2(C(F)F)CCCC2)=O)cccc(-c2cc[nH]n2)c1 24968,C(=O)(CC(C)C(F)(F)F)N1C(C(N2C(COC)COCC2)=O)CC2CC21 24969,C1(F)(CNC(C(C2CCC(=O)N2)C)=O)CCN(C(=O)CC2SC(=N)NC2=O)CC1 24970,N1(C(C2CCCC(C(C)=O)C2)=O)CCCC(C)(CNC(c2cn(CCF)nn2)=O)C1 24971,N1(C(C(CC=CC)C)=O)CCCCC(CNC(c2ccc(C#N)cc2)=O)C1 24972,NS(=O)(=O)CC(=O)NC1CN(C(c2cccc(C3(O)COC3)c2)=O)C2CC12 24973,c1(C2(NC(C34CC(C(=O)NC5C(SC)CCC5)(C3)C4)=O)CC2)ccc(C)cc1 24974,N1(C(=O)C(F)(F)C2(O)CC2)CC(C2CCCNC2)C1.c1(C=O)ccc([N+](=O)[O-])[nH]1 24975,Cc1ccc(C)c(CC(C)N(C)Cc2cc(-c3ccccc3)[nH]n2)c1 24976,c1(C(=O)NCC(C(C)C)NC(C2CCc3c[nH]nc3C2)=O)cncc2ccsc12 24977,C1(NC(c2c(C)ccnn2)=O)C(C)(C)CN(C(c2cnsc2C)=O)CC1(C)C 24978,C(=O)(CC(C)(C)CC(=O)NC1(C2CC2)CCN(C(=O)C(C)(F)F)C1)OCC 24979,C(=O)(C1=NOC2(CCC2)C1)N1C(CNC(c2occc2Cl)=O)CC(O)C1 24980,C(=O)(C(F)CCC(C)C)NC(CC(=C)C)C(=O)NCCCc1cccnc1 24981,N1(C(C(F)=CC)=O)CCCC(CNC(=O)CC(CC)OC)C1 24982,C(=O)(C1CCCc2nccn21)N(CCCNC(Cc1cn(C(C)C)nn1)=O)C 24983,c1(C(=O)NCC=CCNC(C2N(S(C)(=O)=O)CC2)=O)cc(NS(C)(=O)=O)ccn1 24984,NS(=O)(=O)CC(=O)NCCN1CCC(NC(=O)CC(F)(F)F)C1 24985,c1(C(=O)NC2CN(C(C(C)CC(F)F)=O)C2)ccc2c(=O)ccoc2c1 24986,c1(CC)[nH]nc(C(=O)NC(CCC2CCC2)C(=O)NC(c2cnc(C)s2)C)c1C 24987,N1(C(C2C(C)C2)=O)CC2OCC(C(=O)NC(=O)CCSCc3ccccc3)C2C1 24988,CC(c1cccnc1)=CC(N1CCCC1CCNC(=O)CC1CC2CCC1O2)=O 24989,c1(-n2cc(CC(CCOC)NC(C)C)nn2)ccnc(OC(=O)C(=O)NOC)c1 24990,c1(C(N(CCC)Cc2cn(CC3CCOC3)nn2)=O)cc(P(C)(C)=O)cs1 24991,CC(CC(=O)N1CCN(C(c2c[nH]c(C(N)=O)c2)=O)C(C2CC2)C1)C(F)F 24992,CCCC(CC1CCCC1)C(=O)N(CC(O)CNC(=O)Cc1ccncc1Cl)C 24993,c1(OC)cc(F)c(F)cc1C(N1CCC(C)(C(=O)O)CC1)=O 24994,c1(OC)ccc(C(=O)N(CCNC(=O)C(C)S(N)(=O)=O)C2CC2)cc1S(=O)(=O)N(C)C 24995,C(=O)(C(C(C)(C)C)NC(=O)C(C)C)NCCC1(NC(CCC(C)OC)=O)CCC1 24996,C(CNC(C1(CF)CC1)=O)(CC(F)(F)F)NC(c1occc1Cn1ccnn1)=O 24997,c1(C(N(CC(C)NC(c2cc3ccccn3n2)=O)CC)=O)ccc([N+](=O)[O-])cc1Cl 24998,C1(CC(=O)NC2(CCOC)CCC2)CCCN(C(=O)C=CC2CCOCC2)CC1 24999,CCCC(C(=O)NC1CCCN(C(c2ccc(F)c(C(F)F)c2)=O)C1C)C(C)C 25000,Cc1nn(C(C)C)c(C)c1C(=O)NCC(C)(C)OCCNC(=O)CCC1(C)CC1 25001,CC1CCC(NC(c2ccc(C#N)n2C)=O)CN1C(c1cnc(C(F)(F)F)s1)=O 25002,C1(C(N(CCNC(c2ccn(C(C)(C)C)n2)=O)C2CC2)=O)CC2(CCOCC2)C1 25003,N1(C(C(C)(C)CO)=O)CCCC(CO)(NC(c2cnnn2-c2ccccc2)=O)C1 25004,C12(CNC(C3CC(CC)C3)=O)CC(C1)C(NC(=O)C=Cc1nccn1CC)CO2 25005,CC1(C)C(C(N2CC(CNC(=O)C(c3ccccc3)O)C2)=O)CCS1(=O)=O 25006,C1(N(C(C2CC2C(F)F)=O)CC)CCN(Cc2ccc(OCC)cc2)CC1 25007,CC1CN(C(=O)CC(O)c2ccccc2)CC(c2ccc(Br)cc2)O1 25008,c1(C(N2CCC(O)(CNC(c3c(CC)cncc3)=O)C2)=O)cc(C)cc(Cl)c1 25009,C1=C(c2ncc(-c3ccc(-c4ccsc4)cc3)cn2)CCN(C2CC2)C1 25010,C1(C(N(C2CCN(C(CC(C)C)=O)C2)C)=O)Cc2ccccc2N1C 25011,c1(OC)ccc(CN2C(CO)CC(NC(c3cscn3)=O)C2)cc1.C1C(=O)N1 25012,CC(C)(CS(N)(=O)=O)C(=O)N1CC2CCC(Nc3ncccc3C(F)F)CC2C1 25013,c1(-c2ccc(NC(=O)CNC(c3ccncc3)=O)o2)c(F)cccc1Cl 25014,c1(OCC)cnc(F)c(C(=O)N(C(C)CN(C)C(c2cncc(CC)c2)=O)C)c1 25015,S(=O)(=O)(c1cnn(C)c1)CC(=O)NCC(C)CNC(=O)C(C)C(F)F 25016,CCC(C)CC(=O)C(=O)NCCC(=O)NC(C1CCOC1)C 25017,CC1(C)CCCOC1C(=O)NC1CCCCC1NC(c1cccc(O)c1Cl)=O 25018,N12CCCCC(C1)NC(=O)C2.N1(C2C(C(=O)NCCC)CCC2)CCN(C)CC1 25019,C12(c3ccc(F)cc3)CCN(c3cnc4ccnn4c3)CCC1C2 25020,C1(CNC(CCCN(CCC)CC)=O)CCCN(C(=O)Cn2cnc(=N)[nH]2)CC1 25021,CC(C(=O)N1CCC(N(C)C(C2CCCN2CC(F)(F)F)=O)CC1)C(F)(F)F 25022,N1(C(CCOCC#C)=O)CC2CCC1C1CN(C(c3ccnc(CO)c3)=O)CC21 25023,CCCCCCCC(=O)NC1C(C)CCN(C(=O)COc2ccc(F)cc2)C1C 25024,CC1CCN2N=C(C(=O)NCC(C)N(C(=O)C(C)NC(C3CCC3)=O)C)NC2=N1 25025,c1(CN(CCN(C(C23CCC(OC)C2C3)=O)C)C)cc(C)ccc1F 25026,N1(C(C(CCC)F)=O)CC(C(=O)NCC(O)CCOC)CCC1(C)C 25027,C1(C(N(C(C2CCOCC2)C)C)=O)CN(C(C2CCCC2)=O)CCO1 25028,C(=O)(CC(C)CC(C)(C)C)NCC1=CCN(C(c2c(NC(C)=O)cccn2)=O)CC1 25029,C(CC)(C(=O)NC1(C)CC(NC(=O)Cn2ccnc2CC)C1)=CC 25030,Cc1noc(C(F)F)c1C(=O)NCC1CCCN(C(=O)CCc2cnccn2)C1 25031,c1(C(N2CCCC(C)C2CNC(C2CC3(C2)CC3F)=O)=O)ccc2nonc2c1 25032,C1(N(C(c2c(CC)c[nH]c2)=O)C)CCCCN(C(=O)CCOC2COC2)C1 25033,N1(C(C(C)n2cnnn2)=O)CC2CCCC(C1)N2C(c1cnc(F)c(F)c1)=O 25034,c1(CC)n[nH]c(CC)c1CC(N1CCCCC1CNC(=O)CCC=C(C)C)=O 25035,c1(C(=O)NCCC(=C)CNC(=O)CC2CC2)ccc(Cl)c(N2CCNC2=O)c1 25036,C1(=CC(=O)N(CCCCCCNC(=O)Cc2csc(=N)[nH]2)C)CN2CCC1CC2 25037,CC1CCCC(CC(=O)NCC(CC(C)C)NC(=O)CC2(C3CCCO3)CC2)C1 25038,C#CCCC(O)C(=O)NCC(c1ccccc1)NC(c1sc(C)nc1C)=O 25039,Cc1scc(C(=O)N(C)CCOCCCN(C(=O)CC2CC2C)C)c1C 25040,c1(OC)ncc(C(=O)N(C(C)CN(C(=O)C(O)C2CC2)C)C)c(C)n1 25041,O=S(=O)(c1cnn2ccc(=NCCN3CCCOCC3)[nH]c12)NC1(CO)CCC1 25042,C(=O)(CCC1=NNC(=O)CC1)N(CCCNC(=O)CCCC(=O)c1cccs1)C 25043,c1(CNC(c2nc(C)oc2)=O)cc2n(n1)CCN(C(=O)C(C)CC1CCC1)C2 25044,CCCC(C(=O)N1CC(N(C(=O)C(=O)N=S(C)(C)=O)C)C(F)C1)S(N)(=O)=O 25045,CC(CC(F)(F)F)C(=O)NC(C(N1CCC(C(F)F)CC1)=O)c1ccco1 25046,CC1CC(c2ncc[nH]2)CCN1.C(=O)(NNC(=O)CC1CC1)NCc1ccc(CO)o1 25047,CCC(C(=O)N1CC(CNC(=O)CC2CCOC2=O)C1)N(C)C 25048,N1CC(C(=O)NC2(CCN=[N+]=[N-])CC2)OC(C)C1.Cc1cc2oc1C(=O)NC2 25049,N1(C(C(C2(OC)CCCC2)(F)F)=O)C2CCCC1CC(NC(=O)CSC)C2 25050,Cc1[nH]nc2cc(C(N3CC4CC3CN4C(C3CC(=O)N(OC)C3)=O)=O)ccc12 25051,C1(C2CC2)(N(C)C)CN(C(C2CN(C(=O)CCCF)C(C)(C)C2)=O)C1 25052,CC1CCN(CC2CCN(C(=O)OC(C)(C)C)C(C)C2)CC1C 25053,C1(C)(NC(C=CC(C)NC(c2cn(CC)nn2)=O)=O)CC(F)(F)C1 25054,C=CCCC(=O)NCCC1CC(C(=O)NCCCC=CC)C1 25055,N1(C(=O)OC(C)(C)C)CC2CCCC2C1NC(=O)Nc1cc(Br)cc(CO)n1 25056,C1(C(=O)NC(C2C(C(N(C)Cc3nc(C)sc3)=O)C2)C)COCCOC1 25057,C(=O)(C(C)CC(N)=O)N1CCC(C(=O)N(C)CCc2nccs2)(CC)C1 25058,c1(CCC)ccc(CC(=O)N(CC)CC2N(C(=O)C=CSC)CC23CC3)cc1 25059,C(=O)(CC(C(F)F)NC(c1cccn1CC)=O)NC(c1ccc(C)o1)CC 25060,C(CC(C)(C)CC(=O)NC1COCCC1NC(c1cc(C(C)=O)cn1C)=O)OC 25061,Cn1c(C(N2CC3CCN(C(=O)COc4ccsn4)C3C2)=O)cnc1[N+](=O)[O-] 25062,N#Cc1cc(NCCc2cccc(F)n2)cc([N+](=O)[O-])c1Cl 25063,Cc1nc(C(=O)N(CC(C)NC(=O)C(C)(C)CF)C)ccc1[N+](=O)[O-] 25064,N1(C(C(C)N(C(C)(C)CO)C)=O)CCSCC1C 25065,Cn1ncc2ncc(C(=O)NC3CCCCN(C(C4CC4C#N)=O)CC3)cc12 25066,c1(C(N2CC(=C(CNC(C(C)Cc3ccco3)=O)F)C2)=O)cccc(Cl)c1Cl 25067,C(=O)(CCCCNC(c1cnnn1C)=O)N(CCN=[N+]=[N-])C 25068,Cc1cc(O)cc(C)c1C(=O)NCC1CCN(C(=O)CN2CCC(CO)CC2)C1 25069,C1CN(C)CC(C)O1.C=CC(C(=O)NCCCCN(C(=O)C=Cc1ccco1)C)OC 25070,C(=O)(C(CCCCCCC)C(CCC(=O)NNC(=O)c1csc(CC)n1)C=C)OC 25071,Cn1ncc(Cl)c1C(=O)NCC1CCCN1C(C1CN(C2CCOCC2)C1)=O 25072,C1(C)(CC)CCN(C(C2CCCCCN2C(=O)C(C)NC(N)=O)=O)CC1 25073,N1(C(C2(CNC(C3CCCC3C3CC3)=O)CC2)=O)CC2(COC(CO)C2)C1 25074,CN1CC(F)CC1C(=O)NCCCOCCC(N1CCC(F)(CO)C1)=O 25075,CC1CC(NC(c2ccc(I)cc2)=O)CCN1CC1C(C)(C)C1(C)C 25076,C(CC(=O)N1CC(c2ncc[nH]2)C1)(C(F)F)NC(C(C1CCOCC1)C)=O 25077,C1(OC)(CNC(C23CCN(CC2)C3)=O)CCN(C(=O)CN2CCC(C)C2)C1 25078,C(C)(C(=O)N1CC(C(C)NC(c2coc(C(F)F)n2)=O)C1)(C(C)C)OC 25079,C(=O)(C(C(C)(C)C)N(C)C)NC(C(C)C)(C)CNC(=O)Cn1ccnc1C(C)C 25080,C(C(CC(=O)NC1(CCO)CCCCC1)NC(c1cccnc1OC)=O)OC 25081,CC(=O)CCC(=O)NCC(CC(N1CCC(F)(CO)C1)=O)C1CCC1 25082,c1(NC(=O)OC(C)(C)C)ccc(=NCCCOCCC(C)N2CCCC2)[nH]c1 25083,c1(C(=O)NCC(CC=C)NC(=O)CC2CCCN2C(C)C)cc(OC)nn1C 25084,C1(C(=O)NC2(CNC(CC3CC(OC)C3)=O)COC2)CC(C)(O)C1 25085,CON(CCO)C(=O)CC(C(F)F)NC(=O)C(C1CCOCC1)F 25086,C1(C(=O)NCc2c(CNC(=O)CN3CCC(O)CC3)nco2)CCCCC1(F)F 25087,c1(C(=O)NCC#CCNC(c2c(C(C)C)n(C)nc2)=O)cc(Cl)c(Cl)cc1O 25088,C(c1ccccc1)=CCOCC(=O)N(CC(C)N(C(C(C=C)O)=O)C)C 25089,C(c1cc(C)cc(C)c1)=CC(=O)NC(C1CCCN(C(C2(C)CC(=C)C2)=O)C1)C 25090,C1(CNC(=O)CC2(CO)CCC2)CC2CCC1N2C(c1cnc2n1CCC2)=O 25091,C1(NC(c2cnn(C)c2C2CCC2)=O)CC(O)C12CC(F)(F)C2 25092,Cc1ncccc1CC(=O)NC1(C(=O)NCC(C)(C)C(N)=O)CC1C 25093,Cc1c(F)ccc(C(=O)N(C2CCCC(NC(c3c(C)n[nH]c3C)=O)C2)C)c1Cl 25094,c1(C(=O)NCC2(F)CCC(NC(C(C(C)C)O)=O)C2)c[nH]nc1[N+](=O)[O-] 25095,N1(C(c2ccnc(C(F)F)c2)=O)CCC2C(C1)CN2C(c1cncc(Cl)c1Cl)=O 25096,c1(CC)ccc(C(N2CCC(CCNC(c3cn(CC)nn3)=O)C2)=O)c(O)c1 25097,CCC(CC)CCC(=O)Nc1cn(C2CCCN(C(=O)C(C)CC(N)=O)C2)nn1 25098,C(=O)(CN=S(C)(C)=O)N1CC2C(N(C(=O)Cc3ccn(CC(F)(F)F)n3)C)C2C1 25099,c1(CN2CC3N(C(c4c(OC)cncc4)=O)C3C2)c(C)cc(C)cc1C 25100,c1(COC)cc(C(=O)NC(C)(CNC(=O)Cc2nccn2C)C2CC2)no1 25101,O=C1NC(=O)C(CC(N2C(C(=O)NC(CO)C3CCC3)CC3CC23)=O)N1 25102,C(=O)(C1=COCC1)N1CCC(n2cc(C(c3n(CC=C)ccn3)OC)nn2)C1 25103,c1(C(=O)NC2(C(=O)NC(CCC=C)C)CC2(C)C)cc(O)n(CC)n1 25104,C1(CC#C)(C(=O)NCCCOCCC(=O)NC2CCC23CCC3)CCCCO1 25105,N1(C(=O)O)CC2(CCN(CCCl)C2)C1.c1(C(F)(F)C(O)c2ccccc2)ccncc1F 25106,C1(C(C)NC(CC2(CC(=O)OC)CC2)=O)CCCN1C(=O)CCCN1CCOCC1 25107,N1(C(COC(C)(C)S(C)(=O)=O)=O)CCC2(CCC2)CC1 25108,C#Cc1cccc(OCC(N2CCC(CNC(=O)Cc3cccc(O)c3)C2)=O)c1 25109,C1(NC(C2CC(C)(C)OC2(C)C)=O)CCC2(CC1)CN(C(C1(O)CCSC1)=O)C2 25110,C(=O)(C(CC=C)C(C)C)NCC1C=CC(NC(CCC=C)=O)C1 25111,c1(CN(C)C)cc(C(N2CC(Oc3cc(-n4c(C)co4)ncc3)C2)=O)n(C)n1 25112,C1(CC(=O)Nc2cnc(F)cn2)CCCCN1S(=O)(=O)Cc1ccc(Br)cc1 25113,N1(C(COC2CC(CNC(CN(C)C)=O)C2)=O)CCC(O)CC1C1CC1 25114,C1(NC(c2cc(C)on2)=O)CC2(C1)CC2C(=O)NCC(N1CCCCC1)C 25115,CC1(C)CCCC(O)(C(=O)NCC2COCCN(C(C3(n4cncn4)CC3)=O)C2)C1 25116,C(C)(CCC(=O)N(C)C(c1ncccn1)C)NC(CCCOC)=O 25117,N1(CC(=O)NC(C(C)C)CCN(C(=O)C(F)=CCCF)C)CCCCS1(=O)=O 25118,CC1CCN(C(=O)C=C(Cl)Cl)C1CNC(c1cccc(N2CC=CC2)c1)=O 25119,C1(O)(CNC(c2c(C)snn2)=O)CCN(C(c2cccc(Cl)c2)=O)CC1 25120,C(N=c1nc2sccc2c(NC2CC(C)CC(C)(C)C2)[nH]1)c1cc(C)cc(C)c1 25121,CCC(CC)C(C)C(=O)NC(CNC(c1ccc(N)c(C(=O)OC)c1)=O)CO 25122,C1(C(=O)NCCOC2CCN(C(C(c3cccnc3)C)=O)C2)CC2(C1)CC21CC1 25123,Nc1cc(C(N2CCCCCC2CNC(C2(Br)CC2)=O)=O)ccc1Cl 25124,N1(C(=O)NCCC(C=C)(C)O)CC2(CCCC2)CCC1CO 25125,C1(C(N2CCCC(CCC)C2)=O)CCC(C)=C(C)C1.c12occc1CNC2=O 25126,C#Cc1cnn(C)c1C(N1CC(C)(NC(=O)CC2CC(O)C2(C)C)C1)=O 25127,n1(CC(=O)NCC2(CNC(C=CCCC)=O)CC23CCC3)cnc2ccccc12 25128,C(C)(CN=c1nn[nH]n1-c1ccccc1)N(C(F)(F)C(F)(F)F)C(C(=O)OCC)=O 25129,C12(C(=O)NCC(C)(C)OC)CC(CN(C(=O)CC(C)C3CCCO3)C1)C2 25130,C1(C(N(CC(=O)N(C2CC2)C2CC2)C)=O)CC12CCC2.C1C(=O)NOC1 25131,c1(NCc2ccc(OCCC)nc2)scnc1C1=CCN(Cc2cccs2)CC1 25132,N1(C(c2cnc(CC)s2)=O)C2CCC1CC(N(C)C(c1cc(C)ncc1C)=O)C2 25133,CCC(CNC(c1ccc(C2CC2(F)F)cc1)=O)(CC)NC(=O)CC1CCSC1 25134,N1(C(C(C)NC(C2(OC)CCOC2)=O)=O)CC2(CCC(=O)N2)C1 25135,Cc1nn(C)c(N)c1C(N1CCC(OCC(=O)NC(C)C(O)C(C)C)C1)=O 25136,C(=O)(CC(C)(C)C(C)(F)F)N(CC(C)NC(c1ccc(NC(N)=O)cc1)=O)CC 25137,c1(NC(C=C2CCC(C)C2)=O)ccc(C2CC2)nc1.C12CN(C1)C2=O 25138,CCCC(CC(C)C)C(=O)N1C(C(=O)NCCC(=O)OCC)C2CC(O)C1C2 25139,C1(CC(=O)NC(C)Cc2cnc[nH]2)CN(C(=O)C(N)=O)CC1O 25140,N1(CC)CC(NC(=O)CC=CCNC(c2cc[nH]c2C2CC2)=O)CCC1=O 25141,CCCCC(O)C(=O)NC1(C(=O)NCCCN2CCOCC2)CCCC1 25142,Cn1cc(C(=O)NCC(C2CC2)NC(=O)CCC(N)=O)c(-c2ccccn2)n1 25143,S(=O)(=O)(c1c[nH]ccc1=NC1COCC(C)(C)C1)N(CC(CC)C)CC 25144,C1(NC(c2n(CC=C)nnn2)CCC2CCCCC2)CCn2nnnc2C1 25145,C1(C(=O)NCCN(C(C23CCC(C2)C3(C)C)=O)CC)CCCC2(CCCCC2)C1 25146,c1(C(=O)NC(CNC(c2c(C)nc(CC)s2)=O)CC)cc(C)c2[nH]nnc2c1 25147,CC1CC(C(=O)NCCC2CC(NC(=O)C3=CCCCO3)C2)CC(C)C1 25148,C1(=CCNC(=O)CC2CCOCC2)CCN(C(=O)CCOCC(F)F)CC1 25149,c1(C(C)(C)C)[nH]cnc1C(N1CC(CNC(c2cn(CC(F)F)cn2)=O)C1)=O 25150,CC(C)C(C)(CNC(C1SCCS1)=O)NC(=O)Cc1csc(-c2ccoc2)n1 25151,c1(C(N(CCCNC(C(C)OCC#C)=O)CCO)=O)c[nH]cc1-c1cnn(C)c1 25152,C1(NC(c2c(CC)[nH]nc2Cl)=O)CCC(O)CN(C(c2csc3nccn23)=O)C1 25153,N1(C(c2c(C)coc2C)=O)CC2CCCC(C1)N2C(=O)Cc1cc(Cl)ccc1Cl 25154,C1(NC(CNC(c2cc(C)no2)=O)=O)CCCN(CC(=O)NC(C)C)C1C 25155,c1(CN(CCCCOCC#C)CC(=O)Nc2cscn2)cccc(CS(C)(=O)=O)c1 25156,c1(C(N(CCNC(c2ccc(Br)o2)=O)CC)=O)ccncc1Br 25157,C1(C(=O)NCC(C(C)C)OC)(CNC(=O)CCCn2ccnc2)CCN(C)CC1 25158,c1(CC)cc(C(=O)NC2CN(C(=O)CCC)CC2C)ccn1.N1CCOCC1 25159,C1(C(=O)NCC(=O)NC2C(NC(CNC=O)=O)CCC2)CCC(F)(F)CC1 25160,N1(C(COC(c2cccs2)=O)=O)CCC(N(C(=O)C(F)(F)F)Cc2ccoc2)CC1 25161,C1(C2CC2)(C(=O)NCC(C(C)C)OC)CN(C(=O)C=Cc2cn(C)nn2)C1 25162,Cn1ncnc1CNC(c1ocnc1C(F)F)c1nnnn1C1CC1 25163,c1(CC)c(C(N2CC(N(C)C(c3ccnc(OC)c3)=O)C2)=O)cnn1C 25164,c1(C(=O)NC2CC(N(C(C34CC(C(C)C)(C3)C4)=O)C)C2)cn(C)[nH]c1=N 25165,C1(NC(c2ccn(C)c2)=O)CC(NC(c2nnc(S)n2C)=O)C12CCC2 25166,N1(CC)CC2CC1CN2C(C1(COC)C=CCN1C(c1oc(C)cc1C)=O)=O 25167,C1(NC(CCCC#CC)=O)COC2(C1)CN(C(=O)C(c1ccc(Br)cc1)C)C2 25168,C(C)(CNC(C)=O)(C(=O)NOCC(C)(C)C)NC(c1cccc(CC)n1)=O 25169,Cn1ccc2cccc(C(=O)NC3(C)CCN(C4CCNC4=O)C3)c12 25170,C(CCN(C)C(c1c(C)noc1C)=O)(C(C)(C)C)NC(c1cncc(C)n1)=O 25171,C(=O)(CCCCCCNC(=O)C(CO)NC(N)=O)Nc1c(C)ncnc1 25172,CCCCC(C)CCC(=O)NC(COCC)C(=O)NC1(CC)CCCC1 25173,N1(C(C2N(CCC)CCC2)=O)CC(C)(C)C(NC(c2cnc(Cl)[nH]2)=O)C(C)(C)C1 25174,N1(C(C2CCC3CC3C2)=O)CCC2(CC1)CCN(NC(c1onc(C)n1)=O)C2 25175,c1(OC(C)C)ccc(Cl)c(NC(c2cncc(C(C)(F)F)c2)=O)c1 25176,c1(C(N(CCNC(C=C(CC)C)=O)CCOC)=O)cccc(F)c1Br 25177,C12(CC=C)CCN1C2=O.C1(C(=O)NC)CC(C)N1C(=O)OC(C)(C)C 25178,CCC(O)C(F)(F)C(=O)NCC(C1CCN(C(c2ccncc2F)=O)CC1)C 25179,C1(CC)C(C(=O)NC2CCN(C(=O)Cn3nc(C)oc3=O)C2C)CCN1C 25180,C12(CC(N3CCC4CN(C(CC=C)=O)CC4C3)=O)CC3CC(C)(C1)CC(C)(C3)C2 25181,C(=O)(C(C)C(O)C(C)C)N1C(C(C(=O)NCC(COC)C)(C)C)CC1 25182,N1(C(C)=O)CCC(c2nc(-c3ccccc3C)nn2Cc2cccs2)CC1 25183,c1(C(=O)NC(CNC(CC(C)F)=O)C)nc(Br)c2c(F)cccn12 25184,N1(C(CCc2ccc(C)o2)=O)CCCC2CN(C(=O)C(C)(C)C(C)(C)O)CCC12 25185,S(=O)(=O)(c1cccc(Cl)c1F)NC1CC(C(=O)NCc2ccc(O)c([N+](=O)[O-])c2)C1 25186,c1(C(C)NC2CC(C)(CCC)C2)ccc(F)cc1F 25187,C(=O)(CC1CN(C)c2ccccc21)NC(CCNC(CC(CC)C1CC1)=O)(C)C 25188,C(CC(=O)NCC(C)CN(C(=O)CCc1ncco1)C)OCCC 25189,C1(F)(NC(C2CC(OCC)C2)=O)CCCN(C(c2c[nH]nc2C(C)C)=O)C1 25190,c1(C(=O)NC2C3CC4C2C4C3C(=O)NC2C=CCCC2)cc2cccn2cn1 25191,C(CCCCC(=O)NCCC1CCCCN1C(c1ccnn1C(F)F)=O)N(C)C 25192,CC1(C)CN(C(=O)C(C#N)C(C)(C)C)CCN(C(c2c(O)nnc3c2CCC3)=O)C1 25193,C(=O)(C1=C(C#N)CCC1)NC(C1CCCN(C(c2c(C)nc(N(C)C)s2)=O)C1)C 25194,c1(C(N2C3C(NC(=O)CCC4CCCO4)C(C3)C2)=O)n[nH]c2c1CCC2 25195,C1(NC(C(C)OCC(C)C)=O)CC2CC(C1)CN(C(C1(O)CCCCC1)=O)C2 25196,O=C1CC2CN(C(C3CC34CCN(C(=O)C(c3ccccc3)=O)CC4)=O)CC2N1 25197,C=C=CCCC(=O)N1CC(O)CC1CNC(=O)C(CC)n1ccc(C2CC2)n1 25198,n1(CC)cc(Br)cc1C(=O)OCc1nnc(C2CC2)o1 25199,Cn1cc(Cl)c(C(N2CC(O)(CCNC(C34COCC3C4)=O)C2)=O)n1 25200,C1(CC)CCN(C(c2[nH]ccc2CNC(=O)CCCCSC2CC2)=O)C1C 25201,c1(CC2N(c3nc(SC)c(Br)cn3)CCN(C(=O)CC)C2)cc([N+](=O)[O-])ccc1O 25202,C1(C(=O)NCC(C)NC(C=CC(=O)NCC)=O)CCC(OC)CC1 25203,N1(C(c2c(CC)c[nH]c2)=O)CCC(C)C(NC(C2OCCN(C)C2=O)=O)C1C 25204,N(C(=NCCc1cnccc1OC)NC(c1cncc(F)c1)C)CCOC 25205,c1(C(=O)NCC2(C(N3CC4C(C)(CC4)C3)=O)CCC2)cccc2ccnn12 25206,C#Cc1c[nH]nc1C(=O)NC(C)CNC(C1C2CC1N(C(C)=O)C2)=O 25207,C1(C(=O)NCC(COCCC(=O)NC2CCCOC2)CO)CC2(C1)CC(F)(F)C2 25208,C1(CCC)(NC(c2cc(Cl)no2)=O)CCCN(C(=O)CCc2cncnc2)C1 25209,Cc1cc(C)c2c(c1)CCC2NCC1CCN(Cc2cccnc2)C1 25210,C=Cc1cnn(C)c1C(N1CC(COC)(NC(=O)Cc2cccc(OC)n2)C1)=O 25211,C1(NC(c2cc(OC)n[nH]2)=O)CN(C(C2(NC(C)=O)CC(=O)C2)=O)CCC1(C)C 25212,C1(C(N2C(C3(NC(COCC#C)=O)CC3)CCC2)=O)CC(=O)N(CC(F)(F)F)C1 25213,CCCCCC(O)CC(=O)N1CCOC(CCNC(=O)CC2CC=CCC2)C1 25214,c1(OC)cccc(OCCN(CCOC)C(C2CCN(CC3CCOC3)C2)=O)c1 25215,C(=O)(C(Cn1cccn1)NC(=O)CC1CCC1C)NCC(C)OC 25216,C1(NC(c2c(C)nc(OC(F)F)s2)=O)CC2CN(C(=O)C=C3CC3)CCN2C1=O 25217,c1(NC(C2CC2Cc2ccccc2)=O)cnn(Cc2cccnc2)c1 25218,c1(C(C)C)nc(C(N2CCC(CNC(C3(C4CCCCO4)CC3)=O)C2)=O)co1 25219,N1(C(C2N(CC#C)CCC2)=O)CCCC(CN(C(=O)CN2CCC(OC)C2)C)C1 25220,Cc1ccc(CC(=O)NCCCCCNC(C2CN(C)C(=O)CCO2)=O)cc1C 25221,c1(NC(CNC(c2cc(CC)n(CCO)n2)=O)C(C)C)ncnc2cnccc12 25222,c1(C(N2CCC(NC(CN(C)C3CC3)=O)C23CC3)=O)ccc2ncn(C)c2n1 25223,N1(C(CCc2cnn(C)n2)=O)CCC(O)(Cn2cc(CC(C)(C)C)nn2)CC1 25224,c1(CC)nc(=NCc2cc(C(N)=O)co2)[nH]c2ccsc12 25225,N1(C(C=COCC)=O)CC(NC(c2nc3cccnc3s2)=O)CC12CCCOC2 25226,c1(C(N(C(CC)C(=O)O)Cc2cccs2)=O)nc(C)n(C2CC2)c1C 25227,C1(CNC(CC(CCOC)(C)C)=O)CCC2CN(C(=O)C3=COCC3)CCC2C1 25228,C(=O)(C(CNC(=O)Cc1cncn1C)N(C)C)N(C)CC1(N(C)C)CCC1 25229,S(=O)(=O)(c1ccc(NCC(c2cccs2)O)nc1)NC(c1ccc(Cl)cc1)CC 25230,c1(C(=O)NC(CNC(c2c(SC)cc(F)cc2)=O)CO)cc2ccc(F)cc2o1 25231,C(=O)(C1OCCc2c(O)cccc21)NCC1(C)CC(NC(=O)C(N)=O)C1 25232,c1(OC)c(C(N2CCC2CNC(c2cnn(C)c2)=O)=O)cccc1F 25233,C1(NC(CCc2nc(C)c(C)o2)=O)COC2(C1)CN(C(C1CC1C1CCCC1)=O)C2 25234,C(=O)(C1=NOC(C)(C)C1)Nc1cccc(CNC(CC(CC)(C)C)=O)c1 25235,C1(C(=O)NCC23CC(CNC(C4C(CC)OCC4)=O)(OC2)C3)CCCNS1(=O)=O 25236,Cc1ccc2c(c1)C(C(=O)N(C(C)Cc1ccc(C#N)cc1)C)OCC2 25237,CC1(C(N2CCC(C)(NC(c3cc(F)cnc3O)=O)C2)=O)CCCCC1(F)F 25238,Cc1cccc2[nH]cc(C(=O)NCC3CC3NC(c3nnc(O)nc3O)=O)c12 25239,C1(NC(c2c(CC)onc2)=O)CCC2(CCN(C(=O)CC(C)CC(=O)OC)C2)C1 25240,c1(C(=O)NCCCC(N)=O)ccc(NC(C(=O)N(C)C)=O)cc1 25241,C(=O)(C#CC1CCC1)NC1CN(C(CN(c2ccc(N)cc2)C)=O)CC1C(F)F 25242,c1(-c2ccc(C(N3C(C(C)NC(C=CC)=O)CCC3)=O)s2)cccc(F)c1 25243,Cc1cccc(OCC(=O)NC(CNC(=O)C2=CCCSC2)CO)c1C 25244,C1(O)(CCNC(c2n[nH]cc2F)=O)CCCN(C(c2sccc2C(F)F)=O)C1 25245,C1(NC(C(CC=C)OC)=O)CC(NC(=O)CC23COC(C)(C2)C3)C12CCC2 25246,C1(Cn2cnc(C(=O)O)n2)CCN(CCc2cn(CC3COCCO3)nn2)CC1 25247,c1(CNC(C(C=C)O)=O)cc2n(n1)CCN(C(=O)CN1CCCNS1(=O)=O)C2 25248,C1(F)(CNC(=O)C(F)=CC2CC2)COCCN(C(c2ncsc2C2CC2)=O)C1 25249,n1(CCC)ccnc1CNC(=O)C(c1ccco1)NC(=O)C=C(C)C(F)F 25250,O(NC(=O)C(CNC(=O)C(F)CCC(=O)OC)C(C)C)CC(NOC)=O 25251,C1(C)(CC)NC(=O)N(CC(N2CC(F)CC2CNC(=O)C(O)C2CCC2)=O)C1=O 25252,c1(C(=O)NC(CNC(C(CC)F)=O)(C)CO)cccc(N(C)C(C)C)c1 25253,c1(-n2cc(CNC(c3ccc(C(CC)C)cc3)=O)nn2)cc(C)c(F)cc1Cl 25254,N1(C(c2ccc(C(C)C)s2)=O)CCC12CN(C(=O)CC13CCCC1C3)C2 25255,CC1(CNC(C2OCCC2NC(c2ncncc2N)=O)=O)CCCCC1O 25256,C(N=c1[nH]c(=N)[nH]c(=NC(C)CC2CCOC2)[nH]1)C1(OC)CCSCC1 25257,N1(C(=O)OC(CC)CNC=O)CCC(C)C1c1ccccc1.C(C)(C)(C)O 25258,C12(CCCCO1)C(=O)OCCC(=O)NC2.C(C(=O)NC(C)(C)C)N(C(C)C)C.O 25259,C1(CNC(C(C)SC)=O)C2CN(C(c3cn(C)nc3C(F)(F)F)=O)CC12 25260,C(CN=C(NCC1(O)CCN(C)C1)N1CCC(C=Cc2cccs2)C1)SC 25261,C#CC1CN(C(c2nnsc2C(F)F)=O)CCN1C(=O)CC1CCC(C)(C)CO1 25262,N1(CC(C)C)CCC(C(=O)N(CCNC(C2C(F)(F)C23CC3)=O)C(C)C)CC1 25263,N1(C(CCSCCCC)=O)CCOC2(CCN(Cc3cc(=O)on3C)CC2)C1 25264,c1(SC)nc(N2CCN(CCNC(=O)CC(C)CF)CC2)ncc1C 25265,C(C(CC(=O)N1CCCC1)NC1(O)CCCC1)NC(C(c1cccnc1)C)=O 25266,C1(CNC(c2c(C)nn[nH]2)=O)CC(F)CN1C(c1sccc1C(F)F)=O 25267,C1(O)(CNC(c2c(C(C)C)cco2)=O)CCCN(C(=O)CCC2CCC(=O)N2)C1 25268,N1(C(c2c(C)c(Cl)ccn2)=O)CCC(C2CCCN(C(=O)C(C)CO)CC2)CC1 25269,c1(C(=O)NCC2CCCC(CNC(CC(COC)C)=O)C2)cnn2ccccc12 25270,C(=O)(CC1=CCOCC1)NC1N(C(c2cn(CCO)nn2)C)CCN(C)C1 25271,c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)C2)ccc(C(C)C)cc1F 25272,CC1(C(N2CCCC2C2CCN(C(C3SCCS3)=O)CC2)=O)CCNC1=O 25273,c1(NCC2(C)CCCN(C(C(C)OC)=O)C2)c(C#N)cnc2c(Cl)cccc12 25274,Cc1cc(C(=O)NC2CC(NC(=O)C(C)NS(C)(=O)=O)C2)sn1 25275,C(=O)(CCCCC(C)(C)C)NC(C(C)C)CNC(=O)C=Cc1cnn(C)c1 25276,N1(C(c2ccc(C)nc2C2CC2)=O)CC(C)N(C(=O)CN(C)C2CC2)CC1C 25277,CC(C)(CS(C)(=O)=O)C(=O)NC(C1CCN(C(=O)Cn2ncnn2)CC1)(C)C 25278,C1(C(N2C(c3cn(CC4CCC(=O)O4)nn3)CCC2)=O)CC2CCCC2C1 25279,CC(CC(C)NC(=O)COCC1CC1)NC(c1cccn1CC1CCCCC1)=O 25280,C1(COC)CCCCN1C(=O)CCN(C(=O)CCc1ccc[nH]1)C(C)C 25281,CC(C)(F)CCC(=O)NCC1(C)CCCN1C(C1COC(=O)N1)=O 25282,CCCCS(=O)(=O)CC(=O)N1CCC(C)C(N(C)C(c2cc(COC)on2)=O)C1 25283,C1(C(=O)NCC(COC)NC(c2cnc(C3CC3)s2)=O)CNC(=O)N1C 25284,C=CCC(C)(C(F)F)NC(=O)CNC(C1CC1)=O.c1(N)ccc(C)cc1C 25285,C1(CNC(CSC)=O)CN(C(C2(n3cccn3)CC2)=O)CC1C 25286,S(=O)(=O)(c1cn(C)c(C)n1)NC(C(=O)N(C(C)CNC(=O)CNC)CC)COC.OC 25287,Cc1cc2[nH]c(C(=O)NCC(C(C)C)NC(=O)CCCCCN(C)C)cc2o1 25288,c1(C(=O)NCC(C2CCCC2)C)cn(CCNC(c2cc[nH]n2)=O)cn1 25289,N1(C(C=Cc2cnc(OC)nc2)=O)CCC(C2CCN(C(=O)C(=O)NC3CC3)C2)C1 25290,N1(C(C2(COC)C=CCN2C(C2(C)CCCCC2C)=O)=O)CC(CO)CC12CCC2 25291,N1(C(C(C)SC(F)(F)F)=O)CCN(CC2CCCN(C(=O)C=CBr)C2)CC1 25292,c1(C(=O)NCCC2OCCCN(C(CC(CC)(F)F)=O)C2)cc(S(N)(=O)=O)c[nH]1 25293,c1(CN(C(=O)NC(c2cccc(F)n2)C)C)cccc(Cl)c1Cl 25294,Cc1cc(C)c(C(=O)NCCC2CCN(C(=O)C(c3ccccc3)O)C2)s1 25295,C1(C(=O)NCC(CNC(C2CCC(OC)C2)=O)(C)C)C2CCC3(COC(=O)C13)O2 25296,Cc1cnc(C(N2CCC(C)C(NC(=O)Cc3ccc(F)cc3)C2)=O)c(F)c1 25297,C(=O)(C(C(C)O)NC(C1CCCC1)=O)NC(CC)CNC(=O)C(C)SC 25298,C1(CC(=O)OC)CCC(=O)N(CO)C1.N1(CC)C(C=O)CC2CC12 25299,C1(C(=O)NC(C2CCCC2)CNC(c2c(C)scc2)=O)CCC(C)(F)CC1 25300,Cc1nsc(C(N2CCCCC2CCC(=O)NC2(CC(N)=O)CC2)=O)c1N 25301,N1(C(c2c(CC)cc[nH]2)=O)CCCC(C(C)(O)CNC(c2coc(CO)c2)=O)C1 25302,Cc1nc(NCC2CC2(C)C)cc(=NCc2ccc3ncsc3c2)[nH]1 25303,CCC(C(=O)Nc1cccc(-n2cccc(OC)c2=O)c1)C(C)(C)CC 25304,C(CNC(c1cnc(SC)s1)=O)(C(C)(C)C)NC(c1cn(CC(CC)O)nn1)=O 25305,Cc1cc(F)cnc1C(=O)NCC1C(C(=O)NCCC2CC(C)(C)CO2)C1(C)C 25306,C1(CC(=O)NC(C(C)(C)C)CNC(c2cccnc2S)=O)CCCC2(CC2)C1 25307,N1(C(C2N(C(CC(C)c3ccco3)=O)CCC=C2)=O)CCc2nnnn2CC1 25308,C1(O)(CNC(C2CCN(C(C)=O)CC2)=O)CCN(C(C2CNC(=O)N2C)=O)CC1 25309,c1(C(=O)NC2C(C)(CNC(C3CCCOC3)=O)CCC2)nnc(O)cc1O 25310,C1(C(=O)NCC(CN(C(COCCC#C)=O)C)O)Cc2ccccc2S1(=O)=O 25311,c1(NC(CN(C(C(=O)O)=O)CCC)=O)ccc2c(c1)OCCO2.C(C(=O)OC)NC 25312,N1(C(c2c(OC)nsc2OC)=O)CCCC(CNC(c2csnc2Cl)=O)CC1 25313,C(=O)(CCCC(C)(c1nnnn1C1CCCC1)NCc1ncc(Cl)n1C)N(C)C 25314,C1(N(C(CCCOC)=O)C)CC2CCC(C1)N2C(C12CCCC1C2(F)F)=O 25315,C(CNC(C1CC1(C)C(F)F)=O)(CC)NC(C1(CCC)CC1)=O 25316,N1(C(c2cc(CNC(c3ccco3)=O)no2)=O)CC2CC1C(F)(F)C2 25317,N1(C(C(CC(=C)C)C)=O)CCC2CCN(C(c3c[nH]c4nccc-4c3)=O)C2C1 25318,C1(C(N(CCCNC(c2c(C)oc(Cl)n2)=O)C(C)C)=O)CCOC(=O)CC1 25319,C(=O)(C1=C(CC)OCCS1)NCC(C1CC1)NC(c1oc(CC)c(C)c1)=O 25320,C(=O)(CC1COc2ccccc21)NC(C)CNC(=O)Cn1cc(C(F)(F)F)cn1 25321,C(C(C)CC(=O)N1CCCC1C(C)NC(c1cc[nH]n1)=O)OC 25322,N1(C(C2(CNC(c3ccc(C)o3)=O)CCCO2)=O)CCCC(C)CC1 25323,c1(C(=O)O)cncc(C(=O)NC2CC(NC(c3c(C)cns3)=O)C3C2C3)c1 25324,C1(OC)CCC2(NC(N3CCCC(CN(C)C)C3)=O)CC12.c12ccc(cc1)o2 25325,c1(CCC)cc(C(=O)NCC(O)CCNC(=O)Cc2cccn2C)ccn1 25326,CC1c2cc(O)ccc2CCN1Cc1snc(C(F)(F)F)c1Cl 25327,c1(OCC)cc(NC(CC2C3CN(C(c4ccc(CC)o4)=O)CC32)=O)nnc1C 25328,c1(CCC(=O)NC2CN(C(CCC(=C)Cl)=O)CC(C)C2)cccc(S(N)(=O)=O)c1 25329,C1(CNC(CN(C)CCO)=O)CN(C(C2CC3CCCC3C2)=O)CC(C)(C)O1 25330,C1(C(C)NC(=O)CN2CCCC2=O)CCN(C(C2COC(=O)N2)=O)CC1 25331,c1(C(=O)NCCN(C(C)C(C)C)C(c2oc(C)c(CO)c2)=O)cccc(F)c1O 25332,Cc1cc(C(N2CCC(C(C3CC3)N(C3COCC(C)O3)C(C)=O)CC2)=O)ncn1 25333,N1(C(=O)C=CCF)CCC2CN(C(C3CC3C3CCCCO3)=O)C2C1 25334,N1(C(CN(C)CC)=O)CCC2CN(C(=O)Cc3cccc4c3OCC4)CCC2C1 25335,Cn1cccc1CC(N1CCC1(C)C(=O)NCC1CCN(C2CC2)C1)=O 25336,C12(Sc3ccc(C(=O)NC4C(NC=O)COC4)cc3)COCC(C1)C2 25337,N1(C(CCc2onc(CCC)n2)=O)CCC(NC(c2cc(Cl)cn2C)=O)CC1C 25338,N#Cc1c(NC(c2cccc3c2CCC3=O)=O)sc2cccc(F)c12 25339,c1(OC)ccc(CNCCC2(NC(N3CC(C(=O)O)C(C)C3)=O)CC2)cc1 25340,C(=O)(C1SCCc2sccc21)OCC(C(C)C)(c1n(CCC)nnn1)NCC 25341,C12(C(=O)NC(C=C)(C)CC)CCC(NC(=O)Cc3c(C)n[nH]c3C)(CC1)C2 25342,Cn1ccc(=O)c(C(=O)NCCC2CCCN(C(c3coc4c3CSC4)=O)C2)c1 25343,C(=O)(C1CCCc2nn[nH]c21)N1CC2CC(NC(=O)Cn3ncccc3=O)C2C1 25344,Cc1cc(C(N2CCC(NC(=O)CSS(C)(=O)=O)C(CO)C2)=O)cc(C)c1C#N 25345,c1(C(N2CC(NC(c3c(OC)ccc(C)c3Br)=O)C2)=O)cn(C)c2ncccc12 25346,CCCCCC(O)C(=O)N(CC(O)CNC(=O)Cc1ccc(C(C)(C)C)cc1)C 25347,N1(C(c2[nH]cc(C)c2)=O)CC(C)CN(C(c2ccn(C)c(=O)c2)=O)C(C)C1 25348,C12(OC)CN(C1)C(=O)C=CC2(F)F.C(C)(C)(CF)NC(=O)C=CC(=O)N.C(C)(=O)O 25349,c1(CC)c(C(=O)NC2C=CCN(C(C3CC3c3cccnc3)=O)C2)ccn1C 25350,c1(C(=O)NC2C(CNC(c3c(C)snc3)=O)CC2)nc(-c2cccs2)oc1C 25351,Cn1c(NCC2CCCCN(C(c3cc(C(F)F)[nH]n3)=O)C2)cc(=O)n(C)c1=O 25352,c1(NC(CN(C(C2(O)CCSC2)=O)CC)=O)cc(CSC)[nH]n1 25353,N1(C(CC(c2ccccc2F)C)=O)CC2CC(NC(=O)C=Cc3cocn3)C2C1 25354,CC1CCCC1NC(=O)CCCN(C(=O)CC1CCCC1)C 25355,c1(CNC(c2cc(C)[nH]n2)C)ccc(CN2CCC(C)CC2)cc1 25356,N1(C(c2n(C)nc(Br)c2)=O)CCC(NC(=O)CCc2cnco2)C12CC2 25357,C1(CCC)CC(C(=O)NC(C)CCNC(=O)C(C)C)C1 25358,c1(C(=O)NCC(CO)NC(CC(CC)C2CC2)=O)cc(C)ncc1C 25359,N1(C(C(c2ccn(C)c2)C)=O)CCC2CCCC12C(=O)NCCc1ccns1 25360,S(=O)(=O)(c1ccc(C(=O)NCC2(F)CC(CNC(C3(C(N)=O)CC3)=O)C2)cc1)NC 25361,CS(=O)C1CN(C(=O)CC2CCN2C(c2csc(Cl)n2)=O)C1 25362,c1(C(=O)NCC2C(CC)N(C(=O)COCCSC)CC2)cnc2ccoc2c1 25363,C1(C(=O)NC(C#C)C(C)C)CC12CCN(C(=O)C(C)CC#N)C2 25364,C=CC1(C(=O)NC2CCC(NC(=O)C(C#N)=CC(C)C)CC2)CCCCC1 25365,C(=O)(CCCN=[N+]=[N-])N1CCC(N(C)C(c2occc2C(=O)OC(C)(C)C)=O)CC1 25366,CN1CCN(C(=O)CC2CCCC(C)(C)C2)CC1CNC(c1cc(C#N)no1)=O 25367,C1(CNC(CCC#C)=O)C(O)C(O)CN1C(C1CCNC(=O)C1)=O 25368,c1(C(=O)NC2(CNC(C)=O)CC2)cnc2ncccc2c1.N12CCCC1(C)C2=O 25369,C1(N(C(C2(OCC)CCOC2)=O)C)CCCCN(C(=O)Cc2cncnc2O)C1 25370,C(=O)(CC(CC(C)C)NC(C12CCC(C)(C1)OC2)=O)N1CCCC(CCC)C1 25371,N1(C(C)C)C(=O)CCC1C(=O)NCCC(C)NC(=O)CC1CC2(COC2)C1 25372,C1(C)(C(=O)Nc2c3nc(C)[nH]c3ncc2)Cc2ccc(Br)cc2C(=O)O1 25373,Cc1ncnc(C)c1NC(C1CCCC1CNC(c1cc(F)n(C)n1)=O)=O 25374,N12CCN(CC1)C(=O)NC(OCCC1CC1)CN(C)C(=O)C(C)N2CC.SC 25375,C1(C(=O)NCC2(NC(C3CC34CCCC4)=O)CC2)(CC)CNC(=O)C1 25376,Cc1cc(CCC(=O)N(CCNC(=O)CC2(C)CC2(F)F)C(C)C)on1 25377,C1(NC(C(C(C)C)(C)C)=O)CC2CCC1CN(C(=O)CC1CCCCC1O)C2 25378,c1(C(=O)NC2CCC(NC(c3ccc(C)cc3F)=O)C2)cc2ccncc2s1 25379,N1(C(C(Cn2ccnn2)NC(CSCC#C)=O)=O)CCC(F)C(O)C1 25380,c1(CSCC)cc(C(=O)NCCN(CC(C)O)C(C2CCSC2)=O)sc1C 25381,Cc1nn(C)c(C)c1CC(=O)NCCOC1CCN(C(C2CCCOCC2)=O)C1 25382,c1(OCC)cc(NC(c2cc(Br)nc(CNCCO)n2)=O)ccc1OCC 25383,N1(C(CCn2ccc(C)n2)=O)C2CCCC1CNC2 25384,C1(C(=O)NCCCc2nc(C)[nH]n2)CN(C(C2(C)CCCC2O)=O)CC1(F)F 25385,N1(C(C(c2ccc(C)cc2)C)=O)CC2(C1)CN(C(=O)C(C)(C)CF)CCO2 25386,C1(NC(CSCCCC)=O)CCCC2CN(C(C34CC3COC43CCC3)=O)CC12 25387,c1(C(=O)NCCN(C(C(CC#C)O)=O)C2CC2)ccc(OC)c(C)c1 25388,c1(C(=O)NC2CC23CCN(Cc2cncc(Br)c2)CC3)ccc(I)c([N+](=O)[O-])c1 25389,N1(C(C(=O)NC(CC)C)C(C)C2CCC2)CCN(CC2CC2)C(=O)C1 25390,c1(OC)cc(N)c(C(N2CC(NC(=O)Cn3cncn3)C3CC23)=O)cc1F 25391,C1(C(N2CC(S(N)(=O)=O)C2)=O)(NC(CNC(C2C(C)C2)=O)=O)CCC(C)(C)C1 25392,c1(N2CC(N(C(c3ccn(COC)n3)=O)C)C2)ncnc2[nH]c(C)nc12 25393,c1(C(=O)NCC2CCCN2Cc2ccc(N(C)C)nc2)cc2n(n1)CCC2 25394,Cc1ncc(Cl)cc1NC1CCN1C(=O)C(=O)Nc1ccc(C2CCCCC2)o1 25395,c1(C(=O)Nc2ccc(NC(c3cc(C)on3)=O)cn2)ccc(Cl)c(C)c1F 25396,C(=O)(CC(C)C(C)C)NCC(CN(C(C1CCC(CCO)CC1)=O)CC)(C)C 25397,C(=O)(CC(C1=CCCC1)OCC)NCC(CCC)NC(=O)C=CC 25398,C1(C#N)(C(N(CCCCCNC(c2c(C)n[nH]c2)=O)C)=O)C(C#N)C1(C)C 25399,C1(c2nc(C3CCCC(COC)C3)on2)CCCC12CCC2 25400,N1(CC=C)CCCC(C)(C(=O)NC2CC(SC)C2)C1.c12ccc(cc1)CNC2=O 25401,CS(=O)CCC(O)C(=O)NCCCCCCNC(c1ccoc1C(F)(F)F)=O 25402,c1(CC(C)C)cc(N(C2CNCC2(F)F)Cc2cc(Cl)sc2Cl)ncn1 25403,c1(C(=O)OC)ccc2nc(NC(CC(=O)NC)c3cccnc3)sc2c1 25404,C1(CNC(c2ccc(Cl)[nH]2)=O)CC(F)CN1C(C1CCS(=O)(=O)C1)=O 25405,CN1CCC(=CC(=O)NC(C)(CNC(C2CC2C(C)(C)C)=O)CO)CC1 25406,Cc1nc(N2CCCC(Cc3ccc(F)cc3)CC2)ccc1S(N)(=O)=O 25407,CC1(CNC(C2CCOCC2)=O)CN(C(c2cc(Cl)ccc2F)=O)CCO1 25408,C=CCCC(C(=O)N1CCOC(C)(C)C1)NC(=O)CC=C(Cl)Cl 25409,c1(C(N2CC(CNC(c3cc(OC)ncn3)=O)C3C2C3)=O)ccc(F)c(F)c1F 25410,C12(CNC(CC(C3CC3)SC(C)(C)C)=O)CC1CN(C(=O)CCOCC(F)F)C2 25411,N1(C(C(CC)CC(F)(F)F)=O)CCC2(CCC2)C(NC(C23CC(C)(CO2)C3)=O)C1 25412,Cc1cc(C(=O)OC)cc(C)c1.n12nnnc1C(c1ccc(CC3CC3)s1)NCC2 25413,CC(C)(C)CCCC(=O)NC1CC2CCC1CN2C(=O)COc1cccnc1 25414,C1(C(=O)NC(CCSC)C)CCN(C(=O)CCCC2CCCO2)O1 25415,c1(C(N2CCC(NC(C(CCC)OCC)=O)CC2)=O)c(C)nn(C)c1N 25416,c1(C(N2CC3(CCC(NC(CC=C)=O)C3)C2)=O)cc(C)cc([N+](=O)[O-])c1 25417,C(=O)(C1Cc2c(Cl)cccc21)NCC(CNC(c1c2cccc(C)c2sc1)=O)C 25418,c1(C(=O)NCCCN(C(=O)CCn2ccnc2)CC)cc(Cl)c(N)cc1F 25419,C(=O)(C1CCc2cccnc21)NCC1(CC)CN(C(C2(C(CC)(F)F)CC2)=O)C1 25420,c1(C(C(=O)NCCC2(O)CN(C(C)=O)C2)C)cccc([N+](=O)[O-])c1 25421,C(=O)(C(C)(C(C)C)OC)N1CC(N)(CC(=O)OC)C1.C1CO1 25422,c1(C(=O)NC2(CNC(C(C)C3CC3)=O)CC2)cc2c(nc1O)CCCC2=O 25423,C1(CNc2cnn(C)c2)CCN(CC2N(C(CCn3ncc(C)c3)=O)CC2)CC1 25424,c1(OC)cc(CNc2nc(OC)cc(C)n2)ccc1Cl.N12CCCC1CCC2=O 25425,C1(NC(c2nc(F)ccc2Cl)=O)CN(C(c2cc(O)cs2)=O)C2CCCCC12 25426,C=CCC(CNC(C1(CC2CC2)CCC1)=O)C(=O)N1CCC1C(N)=O 25427,C1(N(C(=O)CCc2ccsc2)CC)CCCN(C(=O)CC=C(C)C)C1 25428,c1(COC)nc(NCc2c[nH]nc2C)cc(=NC2CCCC(C)C2)[nH]1 25429,c1(CCN(CCC(=O)NCCCO)C(C)C)ccccc1.C(C)(C)(C)O 25430,C1(OC)CC(CNC(=O)COCCNC(=O)C(F)n2ccnc2)N(C(C)=O)C1 25431,c1(OC)nc(C(=O)NCCC2CN(C(C3(C)CC3)=O)CC2OC(C)C)cc(O)n1 25432,N1(CC(CN(C(C(C)OCCOC)=O)C)O)CCc2sccc2C1 25433,C(CCCCC(=O)NCC(CNC(C1CC(C)(C)O1)=O)OC)OCC 25434,N1(C(C(C)(CO)OC)=O)CC2(C(=O)Nc3cnnc(C4CC4)c3)CC1CO2 25435,N1(C(C2COCC(C)(C)O2)=O)CC(N=[N+]=[N-])CCC1(C)C 25436,C=CCCCCCC(=O)N1CCC2(NC(=O)CC3(OC)CCOCC3)CC2C1 25437,n1(CC(=O)N(CC(CO)(CO)NC(C(CC)C)=O)C)c(C)cc2ccccc12 25438,CC1CCN(CC(C)(C)C(=O)O)CC1.c12ccc(cc1)N(C(=O)C(=O)NC1CC1)C2 25439,c1(N(C(N2CC(CC(C)(C)C)OCC2)=O)CC2CC2)ccc(I)cc1Br 25440,C12CCCC(C1)CNC(=O)COC1(C)CN(C1)C2=O.C(C(Cl)=CCl)OC 25441,CC1(C)COc2c(C(=O)NCc3csc(CNC(=O)C(F)F)n3)cccc21 25442,N1(C(c2c(Cl)ccc(C#C)c2)=O)CC2CCCCC2(NC(C2CCN(C)C2)=O)C1 25443,c1(C(N2CCC(N(C)CC)C2C)C(=O)NCCC(=O)OC)ccc(Cl)c(Cl)c1 25444,C1(CN(C(C2CC2CC(C)C)=O)CC)CCCCN1C(=O)CC1(OC)CCC1 25445,Cc1ccc(C(=O)O)cc1C(=O)NCc1cnn(C2CCC2)c1C 25446,N1(C(c2c(C)cccn2)=O)CC2CCC2(CC(=O)NCc2cccc(O)c2)C1 25447,C(=O)(CCCCCC(=O)NC(C)CNC(=O)CC1CCC2(CC1)CC2)OC 25448,C1(OCC)CCN(C(=O)C=CC(C)(C)NC(=O)CCOC(C)=O)CC1C 25449,C12(CCNC(CCc3c(C)noc3)=O)CCC1CN(C(c1cncs1)=O)C2 25450,Cc1cc(CNC(=O)N(C)Cc2ccc(CC(C)C)cc2)ccc1O 25451,CCCC(O)CC(=O)NC1CN(C(c2ccnn2C(F)(F)F)=O)CC1O 25452,c1(C(=O)NCC2N(C(C(c3n(C)nnc3)(F)F)=O)CC2)cc2cc(Br)cn2cn1 25453,n1(CCOC)cc(C(N2CC3CCC2CN3C(=O)C(C)C)=O)c(=O)cc1C 25454,c1(C(=O)NCCC2CC(NC(c3nn(C)c(O)c3)=O)C2)cnc2ncccn12 25455,C12(NC(C(C)(N(C(=O)C=Cc3ccoc3)C)C3CC3)=O)CCN(CC1)CC2 25456,c1(N2CC(C(C)NC(C(CCCC)C)=O)OCC2)ccc([N+](=O)[O-])cn1 25457,C(=O)(C(F)(F)CC1CCCO1)NC1CC(C)(NC(c2c(C)ccs2)=O)C1 25458,C1(C(=O)NCC2N(C(=O)COCc3ccccn3)CCCC2)(OC)CCCSC1 25459,C1(NC(c2n[nH]cc2Br)=O)CC2CC(NC(C3CC34CC4)=O)C2C1 25460,C1(C#N)(C(N(CCC)CC2(O)CCOCC2)=O)CC2CCC1C2 25461,CS(=O)c1ccccc1C(=O)NC1C=CC(CNC(=O)Cc2ccns2)C1 25462,C(CC(CNC(=O)CN(C)C)NC(=O)CCc1ccn(C)c1)OC 25463,c1(NC(=O)NCC2(C#N)CC2)ccc(C(F)(F)F)cc1Cl 25464,C=CC1(C(=O)OC)CCN(C(C2C(C(=O)OC)CCN2C)=O)C1 25465,Cc1cc(N2CCCC(CNC(C3(C4CCC4)CCC3)=O)C2)nc(C)n1 25466,c1(C(N2CCN(C(C(C)OCc3ccc(C)cc3)=O)CC2)=O)cnc(F)cc1C 25467,c1(O)ccc(Cl)c(Cl)c1.C1(C)(COC)CC1C(=O)NCCN(C(=O)COC(F)(F)F)CC 25468,c1(N(C2CCCC2)C(N2C(CC(=O)OC)COCC2)=O)cnnc(Cl)c1Cl 25469,c1(SCC)ccccc1C(=O)NC1CC(CCNC(C2OCCO2)=O)C1 25470,CCC(C)C(C(=O)N1CCCC1(C)CNC(=O)C(c1ccc(F)cc1)=O)N(C)C 25471,c1(-c2cc(C)sc2)nc(COc2cccnc2)nn1C(c1ccc(F)cc1)C 25472,c1(CC(N2CC(C(C)NC(c3c(CCC)n[nH]c3)=O)C2)=O)cnccc1OC 25473,c1(OC)cc(C(=O)NCCCCNC(=O)C(F)Cc2ccccc2)c(O)c(Cl)c1 25474,c1(C(=O)NC(C(C)C)CNC(=O)C2=CCSC2)c(C(F)(F)F)cccc1F 25475,C(C1CN(C(=O)CC2(N(C)C)COC2)Cc2ccccc21)NC(C(=O)NCC)=O 25476,N1(C(c2c(C)scn2)=O)CC(C)CN(C(c2ncncc2Cl)=O)C(C)C1 25477,N#Cc1cc(C2(CN3CCCC3c3ccccn3)CC2)ccc1F 25478,N1(C(CC(=O)OC)=O)CCC(NC(=O)CCN(C)Cc2ccccc2)C1C 25479,c1(C(=O)Nc2ccc(C(C)O)cc2)cccc2occc12.C123CC1CN(C2)C3=O 25480,Cc1cc(NC(C2CC2C2CN(C(C34CCN(CC3)CC4)=O)C2)=O)cnc1C 25481,C1(N(C(CC(C)C2CCCO2)=O)C)CCC(CNC(=O)CCc2cccs2)CC1 25482,N1(C(CCCCCCC=C)=O)CCC2(CC1)COC(CNC(=O)CNC(N)=O)C2 25483,c1(C(=O)NC2CCC2C(=O)NCc2cccc(Cl)n2)cc2ncccc2o1 25484,C1(CNC(C2(C)CC3CC3C2)=O)CCCCN(C(=O)COCC2CC2)C1 25485,CCS(=O)c1ccccc1C(N1CCCN(CCNC(C2CC2C)=O)CC1)=O 25486,N1(C(C(CC#C)C)=O)CCC2(CC1)CC(NC(=O)C(C)(C)CCC)CO2 25487,C1(NC(c2cc(C)sc2)=O)CCCN(C(=O)CN2CCC(=O)NC2=O)CC1F 25488,Cc1nc(N)c(CC(N2CCC(NC(=O)CC(C)(O)CN(C)C)C2C)=O)c(O)n1 25489,Cc1nc2cc(C(=O)NCC(CNC(c3cn(C)cn3)=O)CO)cnc2[nH]1 25490,c1(C(N2CCCCC(C(=O)NCC3(COCC)CC3)C2)=O)cccc(C#N)c1F 25491,C(C)(C)(CC(=O)N1CC(c2ncccn2)C1)NC(c1c(C)nn[nH]1)=O 25492,N1(Cc2c(CC)cccc2)CCCN(C(c2cccc(-c3cc[nH]n3)c2)=O)CC1 25493,Cc1cc(F)cc2[nH]c(C(=O)NCCN(C)C(c3cnn4c3N(C)CC4)=O)cc12 25494,c1(OCC(=O)NCC2CN(C(C3(C#N)CC3)=O)CC2O)cccc2ccccc12 25495,n1(CC)cnc2c(NCC(C)(C)CC)[nH]c(=NC3CCOC(C)(C)C3)nc12 25496,Cc1ccn2c(CNC(C34CCC(CC3N)C4(C)C)=O)cnc2c1C 25497,N1(C(CC(C(C)OC)NC(=O)CC2C(C)(C)C2(C)C)=O)Cc2cccc(C)c2C1 25498,C1(NC(CC2C(C)=NOC2=O)=O)CCN(C(C2CC2(F)F)=O)C1(C)C 25499,n1(C(C)C)cc(C(=O)NCCCN(C(CNC(=O)CNC(=O)CC#N)=O)C)cn1 25500,Cc1ccccc1OCC(=O)NC1CN(C(=O)CCC2NC(=O)NC2=O)CC1O 25501,c1(C(=O)NC2CC(N(C)C(C3CC34CCCC4)=O)C2)c[nH]c2ccc(Cl)cc12 25502,c1(C(=O)NCCC(C)NC(C2COC(=O)N2C)=O)ccc(SC(F)(F)F)cc1 25503,C1(C(=O)NCCCN(C(C(C)SC)=O)C(C)C)CC(=O)N(c2ccccc2)C1 25504,N1(C(C2C(CC)N(C(=O)C=CCO)CC2)=O)CC2CC1CN2C1CCC1 25505,C(=O)(CC(C)C(=O)N1CCOCC1CC(=O)Nc1cc(Cl)ccc1C)OC 25506,C(=O)(C1=C(Cl)CCC1)N(CCC)CCNC(=O)CNC(c1cnccn1)=O 25507,N1(C(C=C2CCC(C)C2)=O)CCC(C2(NC(c3cc(F)c(F)c(F)c3)=O)CC2)C1 25508,c1(CC=C)ccccc1C(=O)N(C)CCNC(=O)CC1CC(C)OC1C 25509,N1(C(C(=O)N(CCCCCN)c2ccccc2)=O)CCOc2ncccc21 25510,C1(CNC(CCCOCCC)=O)CC(C)N(C(c2cnccc2C)=O)C1 25511,CC(CC(=O)N1CCN(CC(N2CC(F)(F)CCC2C)=O)CC1)C(C)(C)C 25512,c1(C(=O)OC)cc(C)cnc1N(CC(O)CNC(=O)C(=Cc1cccnc1)F)C 25513,c1(C(N2CCC(C3CCCO3)C2)=O)cnc(N2CCNCC2)nc1 25514,C(CN=C(NCc1c(Br)nnn1C)NCC1CCN(c2cnn(C)c2)C1)OCC 25515,C1(CNC(C2(CCCC)CC2)=O)CCCCCN1C(c1ccccc1OC)=O 25516,CN1CCC(C2(C(=O)NC3CCC(n4cc(C5(CO)CC5)nn4)CC3)CC2)CC1 25517,Cc1cc(O)c(C(=O)NCCCN(C(=O)COCCCF)C)cc1Br 25518,C(CC(F)F)(C(=O)NCC1CCOC(C)(C)C1)NC(c1c(CCC)nco1)=O 25519,C=CCN=C(NCC(c1ccc(F)cc1)C)NC1CCN(S(C)(=O)=O)CC1 25520,N1(C(=O)CSC(F)F)CC2CN(C(=O)C3=CCOCC3)CC2C(F)(F)C1 25521,N1(C(=O)CCc2nccs2)CC2CN(C(c3ncc(Cl)s3)=O)CC2C1 25522,Cc1ncnc(C(N2CCC(C(C)NC(c3n[nH]cc3C3CC3)=O)C2)=O)c1C 25523,N1(C(CSCCCC)=O)CCC(NC(C2CCCN2C(=O)CC)=O)C12CCC2 25524,N1(C(C(C)NC(C)=O)=O)CCC(C2OCCC2NC(c2ccns2)=O)CC1 25525,C(C(F)(F)F)(C1CCCCC1)N(CCn1ccnn1)CCOC 25526,N12CC3C(C3C1)CC2=O.CC(C)(C(=O)N1CCC(CN2CC2)C1)n1cnnn1 25527,Cc1cc2ccccc2nc1C(=O)NC1CCC(CNC(c2ccc(CO)s2)=O)C1 25528,c1(C(=O)NCCN(C(C=C(CCN(C)C)Cl)=O)C(C)C)cnc(CC2CC2)nc1 25529,C1(F)(CNC(c2ncccc2N2CCCC2)=O)CCN(C(C2CC2C2CCC2)=O)C1 25530,C(=O)(CCCCC#N)N(C(C(=O)NCc1onc(CC)n1)C1CC1)C 25531,CC(CC(=O)N1CCN(C)CC1)C(C)(C)NC(=O)CCCCN=[N+]=[N-] 25532,C1(O)(CN(C)C(c2scnc2C2CC2)=O)CCN(C(C2(C#N)CC2)=O)C1 25533,CC1CN(C(C2(C(=O)NCCC(F)(F)F)CCC2)=O)CCS1=O 25534,C(CNC(c1ccc(N2CCC(C)(C)C2)cc1)=O)(CCS(C)(=O)=O)OC 25535,C1(C(N2CC3C(CNC(CNC(C(C)(C)C)=O)=O)C3C2)=O)CC2(CCOCC2)C1 25536,C1(CCC)(N(C(=O)COC2CN(C(c3cn[nH]c3)=O)C2)CC)CCC1 25537,C(=O)(C1=NNC(=O)CC1)NCC(CNC(C1CCC(=O)C1)=O)OC 25538,C1(NC(C(C)SCc2ccccc2)=O)CN(C(c2csc3nnsc23)=O)CCC1C 25539,C(C1CCCCC1)=CC(=O)NCC1N(C(C2CC(C(=O)OCC)C2)=O)CCC1 25540,N1(Cc2ccc(C(=O)OC)cc2)CC2CCN(C(C3(C)CCOCC3)=O)CC2C1 25541,c1(OC)cccc(C(F)(F)F)c1S(=O)(=O)N1CC(=O)NC(C)C1 25542,c1(C(N2C(CNC(Cc3c(C)ocn3)=O)CC2)=O)cc2ccccn2c1 25543,Cc1cc(C(N2CC3CC2CCN3C(c2csc(=N)[nH]2)=O)=O)c(S(N)(=O)=O)s1 25544,C(C)(CNC(=O)CC1(CO)CCC1)(CO)NC(C(F)=CC)=O 25545,c1(C(=O)OC)cccc(C(=O)NCC(C(C)(C)C)NC(=O)CCCN(C)C)c1O 25546,N1(C(CC2(C=C)CCC2)=O)CC2COCCC2(NC(C2CC3(C2)CC3(F)F)=O)C1 25547,C(CC(C(=O)NOCC(C)C)NC(=O)C(N1CCCN(C(C)C)CC1)=O)OC 25548,Cc1ccc(F)c(C(=O)NCc2occc2C(=O)NC(C)C(F)F)n1 25549,C1(NC(=O)CN2CCS(=O)CC2)CN(C(=O)CCC2CCCCCC2)CC12CC2 25550,C=CCC(C(=O)NC(C)CCNC1(CO)CCCCC1)NC(C)=O 25551,c1(C(N2CC(O)(C(C)NC(CCC(C)SC)=O)C2)=O)ccc(=O)n(CC(C)O)c1 25552,S(=O)(=O)(c1ccccc1C#N)N1C2CCCN(C(CN(C)C)=O)C2CC1 25553,c1(C(N2C(CNC(c3c(C)cn(C)n3)=O)CN(C)CC2)=O)ccc2nccn2n1 25554,C1(C(=O)NC(CCOC)CNC(=O)CC2(OC)CCC2)Cc2nccn2C1 25555,Cc1nn(C)c(C)c1CC(=O)NC(CNC(=O)Cc1cc[nH]c(=N)c1)C(C)(C)C 25556,C1(C#CC(=O)NC2CC3(C2)CC(C(=O)N(C2CCC(O)CC2)C)C3)(CC)COC1 25557,CC(CCCO)N=c1[nH]c2c(c(=NCC3OCCC3C)[nH]1)COC2 25558,Cc1cc(C(=O)NC2CC3CCC2N(C(C2(CCF)CCC2)=O)C3)cc(C)c1Cl 25559,c1(CNC(C(C2CCCC2)NC(c2c(CC)ncs2)=O)=O)cccc(F)c1O 25560,C1(CC(=O)N(CCNC(Cc2c(C)con2)=O)C)CCOC(C(C)C)C1 25561,C1(NC(C(CC)n2ccnc2)=O)C=C(c2ccccc2)C1 25562,CCCC(CCCNC(C1CC(C)OC1C)=O)NC(c1ccnn1CCC)=O 25563,C1(NC(c2n(CC)ccc2)=O)(CF)CCN(C(=O)CCSC(F)(F)F)C1 25564,N1(C(=O)OC)CC(N(C(=O)CC2CCC=CCC2)C)C(C)C1.C1(=O)CC2(CC2)N1 25565,c1(C(=O)NC2CCN(C(Cc3c(C)cccc3)=O)C2)nc(=N)[nH]c2ccccc12 25566,C(CN=C(NCC1CC1C1CCC1)NC1CCS(=O)(=O)C1)c1cccc(O)n1 25567,C(C(CC(C)C)C(=O)NC1CC(C)(CO)C1)NC(c1cc(C)oc1)=O 25568,C(=O)(C1=NN(C)C(=O)CC1)NC1CCN(C(C(CC=C)CC=C)=O)CC1C 25569,C1(CNC(=O)C=Cc2cccs2)CCN(C(c2cn(C(F)F)cn2)=O)CC1 25570,c1(CNC(C2C(NC(C3CCC(=O)N3)=O)C2)=O)c[nH]c2ccncc12 25571,C(=O)(CCC(C)(C)N(C)C)N1CCC(N(C(c2ncc(OC)cn2)=O)CCO)CC1 25572,N12CC3(CCCCC3)CC1C2=O.C(C(F)F)OC1CC1 25573,C1(CC)CC(O)CN1C(=O)CCCCN(C)C.c12cc(on1)CNC2=O 25574,c1(OC)ccc(CCCNC(=O)NCC2(c3csnc3OC)CCC2)cc1 25575,C1(CC(=O)NCCC(C)SC)CN(C(=O)Cc2cccs2)CCC1C 25576,CCCCC(CC(=O)NC1CC2(C1)CC(C)(C)C2)NC(c1ocnc1CC)=O 25577,CC1CCN(C(=O)CSC(=N)N)C(C)C1NC(c1cc(C(F)F)[nH]n1)=O 25578,C(c1cc2ccccc2o1)=CC(N1CC(COC)(CNC(=O)CSC)C1)=O 25579,c1(C(=O)NCC(C(C)C)NC(C2CC(O)CN2C)=O)c(F)ccc(Cl)c1F 25580,N1(C(C(C2CCOCC2)SC)=O)CCC(C(F)CNC(=O)CNC=O)CC1 25581,c1(OC)cnc(C(F)(F)F)cc1C(=O)NC1(CNC(=O)C(O)COC)CCOC1 25582,N1(CC(=O)NCC2(CN(C)C(C3CCC(F)(CN(C)C)C3)=O)CC2)C(=O)CCC1=O 25583,C=C(Cl)CC(C(=O)NCc1cn(C)nc1C)NC(=O)Cc1ccc(F)cc1 25584,c1(C(=O)NCCN(CC(C)O)C(=O)C=Cc2cnccn2)cc(O)cc(C#N)c1 25585,Cc1ccc(C)c(C(N2CC3C(CN(C)C(c4csc(C5CC5)n4)=O)C3C2)=O)n1 25586,C1(NC(C23OCC(C(C)C)(C2)C3)=O)CN(C(=O)C(C)CC(F)(F)F)C2(CCC2)C1 25587,CC1CN(C(C2CNC(=O)N2)=O)CCN1C(=O)CCCC(=O)c1ccc(F)cc1 25588,CCCC(CCC)=CCSc1nc(C2(C(=O)O)CC2)no1 25589,N1(C(C=CC=CC)=O)CCC12CN(C(c1cncnc1)=O)C2 25590,Cn1nc(C(F)F)cc1C(N1CCCC(CNC(=O)CC2CCNC2=O)C1)=O 25591,N1(C(CCC#C)=O)CC(C(=O)NC(CC2CC2)CC=C)C2(CC2)C1 25592,N1(C(CSCCC)=O)CC(C(N2CCc3c[nH]nc3C2)=O)CC(C)(C)C1 25593,C1(C(N(CCNC(CCOCCOC)=O)C(C)C)=O)CCC(N=[N+]=[N-])CC1 25594,N1(C(c2ccc[nH]2)=O)CCC2CCCN(C(c3ncoc3Br)=O)C2C1 25595,C=CC1COCC1NC(=O)C(CCSC)NC(=O)CC1(CSC)CC1 25596,CC(C)CC(C(=O)NCCOCC(N)=O)ONC(C1C2CCC(F)(F)C12)=O 25597,c1(NCc2cc(Br)cc(C)n2)nc2ccccc2nc1NCC1CSC1 25598,C12(c3cn(CC(=O)NC4CC(O)CN4)nn3)COC(CN1C(C1(C(F)F)CC1)=O)C2 25599,c1(CCC(=O)N(CCCCCC)C(C=C)CO)ccc(C2CC2C)[nH]1 25600,c1(CC(C)NC(CC2(N(C(=O)C=Cc3ccsc3)C)CC2)=O)cccc(C)c1 25601,C(CC(N)=O)(C(=O)N1CCCC1c1ccco1)NC(C(C)C1CCCC1)=O 25602,C1(CCCNC(C(CC)SC)=O)CCCCN1C(=O)CCCCc1cnn[nH]1 25603,c1(C(C)C)ncc(C(=O)NCC2CCC2NC(C2(n3nccn3)CC2)=O)s1 25604,O(NC(=O)CC(CNC(c1c[nH]ccc1=N)=O)OC)CCC(=C)C 25605,C(C(CC)(CC)C(=O)NC1CCN(C(C)=O)CC1C)NC(C1(CCC=C)CC1)=O 25606,C1(C(N(C(CC)CC)CCO)=O)CC=CCN1C(c1cncc(OC)c1)=O 25607,N1(C(C=NOC)=O)CC2CCC1C1CN(C(=O)CCn3cc[nH]c(=O)c3=O)CC21 25608,CN1C(=O)NCC1C(=O)NCC1(NC(c2ccc(O)nc2)=O)CCCCC1 25609,C#CCCC(O)C(=O)NC1CC(C)(NC(=O)C2=CSCCO2)C1 25610,O(P1(=O)Cn2cc(nn2)CO1)CC.C1(C(=O)OC)CC(C)CO1 25611,Nc1nccnc1C(=O)NCC1CN(C(=O)Cc2cn[nH]c2)CC1C(F)(F)F 25612,CC1C(NC(=O)CC2(C(F)(F)F)CC2)CC2CCC1N2C(C1CN(C)C1)=O 25613,c1(OCC(N2CCC(NC(C3(CC)CC3(F)F)=O)CC2)=O)ccc(F)c(F)c1 25614,c1(C(N2CCCC(NC(C3(C)CCN(C(C)=O)C3)=O)C2)=O)ccn2ncccc12 25615,C1(NC(C(F)(F)Sc2ccccc2)=O)CC2CCC1(CC1(C(=O)OC)CCCO1)C2 25616,N1(C(C2(NC(C3CC(CC)C3)=O)CCCCC2)=O)CCCCC(CC(N)=O)C1 25617,C(COC(C)C)(C(=O)Nc1conc1C)NC(C=CC(CC)C)=O 25618,N1(C(CCCN(C)C)=O)CCC(NC(c2cc(CF)on2)=O)C12CC2 25619,c1(C(N2CCCC(F)(CNC(c3ccns3)=O)C2)=O)cccc2nn[nH]c12 25620,Cc1nc(C(=O)NCC(c2ccccc2F)NC(=O)C=Cc2cc[nH]n2)c(C)s1 25621,N1(C(c2cc(C3CC3)on2)=O)CCOC(CO)C(O)C1.N12CCCC(CC1)C2=O 25622,N1(CCNC(=O)Nc2cccc(I)c2)CCCC(O)(c2ccccc2)CC1 25623,n1(CC)ncc2cc(C(=O)NC(CNC(c3nocc3Cl)=O)CC(C)C)cnc12 25624,c1(-c2nc(C(CC)CC)nn2Cc2cccs2)cnc2n1CCCCC2 25625,C(CCC(=O)NC1(CCNC(c2nc(C3CC3)cs2)=O)CCC1)C1C(C)C1 25626,C#CCCCCC(=O)N1CCC(CO)C(NC(c2cccnc2C)=O)C1 25627,C12CCN(C3(CC3)C1)S(=O)(=O)C2.c1(C(CC(=O)O)N2CCCC2)ccccc1Br 25628,CCCC(C(=O)NCc1cc(C)ns1)NC(=O)CC1CCOC1(C)C 25629,C1(c2c(C(=O)N(C)C)n[nH]c2)CC(C(=O)NC2C(C)C(O)C2)=NO1 25630,CCCC(CCC)CC(=O)NC(C(=O)NCC(F)Br)C1(O)CCC1 25631,c1(CCC(=O)NC2CN(C(C(CCC)N(C)C)=O)C2)nc2ccccc2[nH]1 25632,c1(C(N(CC(C)CNC(=O)CC2CCCN2C)C)=O)cc2cccnc2cc1F 25633,N1(C(CCC(C)SC)=O)CC(NC(c2csc(C(F)F)c2)=O)C(C2CC2)C1 25634,C1(NC(CC=CC=C)=O)CC(C(=O)N(C)Cc2cc(C)no2)C12CCC2 25635,C1(NC(Cc2cc(C)sc2)=O)(COC)CCN(C(=O)C(c2ccncc2C)C)C1 25636,N1(C(CC2C(C)(C)C2)=O)CCC(OCCNC(=O)Cc2sccc2Cl)C1 25637,C1(NC(C2CC(C)CC(C)C2)=O)CCOC12CCN(C(=O)OC(C)(C)C)CC2 25638,C1(C(NOCCCOCC)=O)CN(C(c2ccsc2C#N)=O)C2(CCC2)C1 25639,c1(C(=O)NC2C(NC(C3(Cl)C(C)(C)C3)=O)COC2)cccc(OCC(F)F)n1 25640,C(CCN=c1[nH]c(=NCC2COC(C)(C)C2)[nH]c2c1CSC2)NC(C)=O 25641,c1(NC(=O)CN(C(=O)C(C)C)C)[nH]c(O)nc1C.C1(CC)CCCN1C(C)=O 25642,c1(N(C)CC2COC(=O)N2)nc(=NCC2CCCO2)nc(N2CCOCC2)[nH]1 25643,c1(C(C)=O)ccc(C(=O)NC(C)CNC(=O)C=CC(N2CCC(C)C2)=O)s1 25644,c1(C(N2CC(CNC(C=Cc3c(C)cccn3)=O)C2)=O)cn2cnnc2cn1 25645,C(=O)(C(CCC=C)NC(c1cc(C)cc(O)c1)=O)NC(CC#C)C(=O)NC 25646,N1(C(CNC(COCCCC(C)C)=O)CC)CCN(C(c2ncnn2C)=O)CC1 25647,Cc1nc2ccccc2c(C)c1CC(=O)NC(C)CCNC(=O)C(C)P(C)(C)=O 25648,c1(OC)ncc(Br)cc1CN1CCC(NC(=O)CCCCC(F)(F)F)CC1 25649,c1(OC)cccc2c1NC2=O.C1(COC)CCN(CCCCO)C1 25650,Cc1cccc(C(C(=O)O)NC(c2ccccc2C(C)C)=O)c1 25651,C1(CNC(C(C)Nc2ccccn2)=O)CN(C(C23CC(C2)C3)=O)CC1(F)F 25652,N1(C(C2CCCC(=O)C2)=O)CC=C(C(=O)NCC(c2cccnc2)O)CC1 25653,CCCCC(C(=O)Nn1cnnc1C)NC(c1ccc(C#N)s1)=O 25654,C(=O)(C1=NOC2(CCC2)C1)N(CC(O)CNC(C1CCN(C2CC2)C1=O)=O)C 25655,CC1CCN(C(c2cc(Cl)nnc2O)=O)CCN1C(C1C2CCC1CC2)=O 25656,N1(C(CC(C=C)C)=O)CCCC(O)(CNC(=O)CSCc2ncc[nH]2)C1 25657,N1(C(C(C=C)CC)=O)CC(CC(=O)NCCSC)CCC1C 25658,C(=O)(C(O)CC(C)(C)C)NCC1(CNC(CCCN(C(C)=O)C)=O)CCCS1 25659,Cn1cc2c(C(=O)NC3CCCN(C(=O)CCc4nc(=N)[nH][nH]4)C3)cccc2n1 25660,CC1CC(N(C)C(CC(c2cccs2)=O)=O)C1 25661,C(N=c1[nH]c2c(c(=NC3CCC4CCC34)[nH]1)CCCCC2)C1(COC)CCCC1 25662,c1(NC(CC2N(C(C(c3cnn(C)c3)C)=O)CC2)=O)ccc(O)cc1F 25663,S1(=O)(=O)c2ccc(nc2)N1.c1(NCC2(CC)CC2)cn(C)nc1C1CC1 25664,n1(CC(C)NC(C(C)NC(CC)=O)=O)cc(CNC(=O)Cc2cc[nH]n2)nn1 25665,N1(C(C)C(=O)NC(C2CCN(CC(=O)Nc3ccccc3)C2)=O)C(=O)CNC1=O 25666,Cc1nc2ccsc2c(=NCCNC(=O)C(c2ccc(F)cc2)O)[nH]1 25667,C1(C(=O)NCC(C)CNC(C2CN(C(C)=O)CC2OC)=O)(COC)CCCCC1 25668,N1(Cc2cccc(C#N)c2)Cc2ccc(NC(c3cc(Cl)c(Cl)cn3)=O)cc2C1 25669,C1(N(C(C=C(CCC)CCC)=O)C)CC2CCC(C1)N2C(=O)C1=NOC(C)C1 25670,CCC(CC)CCC(=O)N1CCOC(C(C)NC(=O)C#CC2CCC2)C1 25671,N1(C(c2cc(C)on2)=O)CCC2(CC1)CCN(C(C1COC(C)C1)=O)CC2 25672,N1(C(C(C)N(C(=O)CC(C)(C)C)CCC)=O)CC2C3CCC(O3)C2C1 25673,C1(C2CCC2)(SCC(C2CCCC2)OC)CC1 25674,c1(C(=O)NCCCC(C)NC(=O)Cc2ccc(F)cc2)ccc2c(c1)CC(=O)N2 25675,N1(C(c2c(C)sc(Cl)n2)=O)CCN(C(c2ncc[nH]c2=O)=O)CC(O)C1 25676,N1(C(C(CC2CCCC2)NC(=O)C=Cc2ccccc2)=O)CCC(F)C(O)C1 25677,c1(C(=O)Nc2cc(F)ccc2F)n[nH]c2c1CN(C(C1(F)CC1)=O)CC2 25678,C12(Cc3ccccc3C1)CC(C)NC2=O.c1(NC(N)=O)cc(I)c[nH]1 25679,CCCCCC(C)CC(=O)NC1CC1NC(=O)CNS(N)(=O)=O 25680,c1(C(=O)NC(CNC(c2c(C)cccn2)=O)C(C)(C)C)ccc(F)c2occc12 25681,c1(SC)cc(C(N2CCC(CCNC(=O)C(c3cnn(C)c3)O)C2)=O)oc1C 25682,c1(OC)cncnc1C(N1CC2C(CNC(C3CCOC3C3CC3)=O)C2C1)=O 25683,C(CO)(CCCCNC(C1CC(F)(F)C1)=O)NC(c1ccn(C(F)(F)F)n1)=O 25684,N1(C(c2n(C)ncc2[N+](=O)[O-])=O)CCCC1C1CCCCN1C(c1cc[nH]n1)=O 25685,CCS(=O)CC(=O)NCCCC(C)(C)NC(=O)C(C(C)C)NC(C1CC(C#N)C1)=O 25686,CC1CN(C(=O)C=CSc2nc[nH]n2)CCCN1C(c1cncc2ccsc12)=O 25687,CN1CCN(c2nccc(Cc3ccccc3)n2)CC1(C)C 25688,c1(C(N2CC(CNC(c3c(C)ncn3O)=O)C3C2C3)=O)cccc2[nH]ccc12 25689,C(c1ccc(F)c(F)c1)=CC(N1CC(NC(c2cnnc(O)c2)=O)CC(C)C1)=O 25690,C1(CNC(C(C)CN(C)C)=O)CCN(C(C23CC4CC2C3C4(F)F)=O)C12CCC2 25691,c1(CC)cc(C(=O)NC2CC23CC(NC(c2nn(C)cc2C)=O)C3)n(C)n1 25692,c1(C(=O)NCCCCCNC(c2c(CC#N)cccc2)=O)cc2ncccc2[nH]1 25693,N1(C(C=C(C)C(F)(F)F)=O)C2CCC1CC(N(C(=O)C=Cc1nc(C)cs1)C)C2 25694,c1(C(N(C(CNC(C23CCCC2C3(F)F)=O)C2CC2)C)=O)cccc(O)c1Cl 25695,CCC(F)(F)C(C)(C)C(=O)NC(CO)CCCCNc1ncc(C(F)F)cn1 25696,CCCCCO.C12(CCC1)C(=O)NC(C)CNC2=O 25697,c1(C(=O)NC23C(CN(C(CSC)=O)C2)C3)c(Cl)oc2ccccc12 25698,C(=O)(CCCCCC#N)NC(C)CC(C)NC(c1cccc(OC(F)F)c1)=O 25699,C(=O)(C1=C(Cl)CCOC1)N(CCNC(C1(NCC(CC)C(C)(F)F)CCCC1)=O)CC 25700,C(=O)(CC(C)(C)O)NCCOCC(=O)NC(C)Cn1cncn1 25701,CC1(C)CC(NC(=O)CCC2CCOCC2)CN1C(=O)CN1CCCCCC1 25702,N1(C(c2nc(C)oc2)=O)CCN(Cc2cc(Br)ccc2I)C(C)C1 25703,C1(C(C(C)C)NC(=O)C(Cl)=CCl)CN(C(=O)C=Cc2cn(C)cn2)CCO1 25704,n1(CCC(=O)NCC(C2CC2)NC(=O)CC2CCCCC2)cnc([N+](=O)[O-])c1 25705,C1(C(C)NC(C(C)(C)OC)=O)CCCN(C(=O)CC(C)(F)F)C1 25706,C=CCCC(C(=O)N(C(C)C(C)(C)O)C)NC(c1cc(Cl)ns1)=O 25707,c1(C(N2CC(CCNC(C(CCCC)C)=O)C(C)C2)=O)nccn2cc(C)nc12 25708,N1(C(C(=O)NC2CC2)c2cn[nH]c2)CC2C3C=CC(O3)C2C1.c1(C(N(C)C)=O)cc(O)ns1 25709,C1(c2nnc(C)o2)CN(C(c2coc(C3CC3)n2)C(=O)NC(C)(C)C)CCO1 25710,N1(CCN(C)CCO)CC2(Br)CC2(CN(S(C)(=O)=O)C)C1 25711,C1(C)(C(=O)OC)CC(NC(=O)C(C2CCSCC2)N(C)C)C1 25712,C1(NC(CC2N(C)CCC2)=O)CS(=O)(=O)CC1NC(=O)C=CSc1ccccc1 25713,Nc1cc(F)ccc1C(=O)NCC(O)CNC(C1CCC(C(F)(F)F)CC1)=O 25714,C1(NC(c2c(CC)cno2)=O)C(C)CCN(C(c2nc(C)c(C)nc2C)=O)C1C 25715,CS(=O)(=O)CC(=O)NCC12CC1CN(C(c1cccc(C(N)=O)n1)=O)C2 25716,N1(C(C=CSC)=O)Cc2nccn2CC(NC(c2cc(C)nn2C(F)F)=O)C1 25717,c1(C(=O)NC2CCCCCN(C(CC=C=C)=O)C2)n[nH]c2cc(Br)ccc12 25718,Cn1cnc(I)c1NC(CN1CCC(c2nc(C(N)=O)cs2)CC1)=O 25719,C1(CNC(c2ccc(C#C)o2)=O)CN(C(c2csc(C(N)=O)n2)=O)CC12CCC2 25720,Cc1[nH]nc(C(=O)N(C)CC2CN(C(c3ocnc3C(F)(F)F)=O)CCO2)c1F 25721,C(=O)(CCCC(C)O)NCC(Cc1ccccc1)N(c1nccc(CC)n1)C 25722,N1(C(c2cc(COC)no2)=O)CC2CN(C(=O)C(C)CS(C)(=O)=O)CC2C1 25723,c1(C(=O)NCC2CC(C)(C)CN2C(=O)Cn2cnc(=N)[nH]2)cc2c[nH]cnc-2n1 25724,Cc1c(C(N2CCN(C(=O)C(O)C3CC3)CC2)=O)sc2ccccc12 25725,c1(C(=O)NC2CC(NCc3c[nH]c4ncc(Br)cc34)C2)n[nH]c2cc(Cl)ccc12 25726,N1(C(C(C)NC=O)=O)CCC(NC(c2cc(C(C)(C)C)n(C)n2)=O)C1C1CC1 25727,N1(C(CSCC(=O)OC)=O)CC2CC1C2NC(=O)C(C)(C)n1ccc(C2CC2)n1 25728,CC1CCn2cc(C(=O)NCC(CO)NC(c3c[nH]c(Br)c3)=O)nc2C1 25729,N1(C(C(N2CCOC2=O)C)=O)CC=CC(CC=C(C)C)C1.c1(C(=O)N)ccc(SC)nc1 25730,CCCCS(=O)(=O)CC(=O)N1CCC(OCCNC(=O)C2=CS(=O)CCC2)C1 25731,C#Cc1ccc(C(=O)NC(C)CN(C)C(c2cscn2)=O)c(OC)c1 25732,C1(CNC(C2CN(C(N)=O)C2)=O)CN(C(c2cc(F)ccc2Cl)=O)CC12CC2 25733,C1(C(=O)NC(CNC)(C)C)C2CC2CN1C(=O)C(C)OCC(C)C 25734,C1(NC(C2=NOC(C(C)(C)C)C2)=O)CN(C(C2(C)CC(F)(F)C2)=O)CC2(CC2)C1 25735,N(C1COc2ccccc21)N(C(C)C(=O)NC(CCC1CCCC1)C(=O)NC)CC.CC 25736,c1(C(C)(C)C)cccc(C(c2nnnn2C2CCCC2)NCCC2CCOC2)c1 25737,N1(C(CC2C(OC)COCC2)=O)C2CCC1C1CC1(NC(=O)COC(F)(F)F)C2 25738,N1(C(C(Cc2c(C)ncs2)NC(=O)OC(C)(C)C)=O)CCCC(N(C)C)C1 25739,C(C)(C)(C#Cc1cn(CC2(OCC)CCC2)nn1)NC(C(CC)CC(C)C)=O 25740,C(C)(CCCCNC(C12CC(C)(C1)C2)=O)NC(c1c(C)ocn1)=O 25741,C1(CC(=O)NCC2CC2CNC(c2sncc2Br)=O)CN2CCC1CC2 25742,c1(C(N2C(CNC(C(CCC)CC)=O)COCC2)=O)cc(F)c(O)c(Cl)c1 25743,Cc1cccc(C2(C(=O)NC(CNC(C3CN(C)C(=O)N3)=O)C(C)C)CCC2)c1 25744,C1(NC(CC2(OCC)CCCC2)=O)CCOC(NC(=O)CNC(=O)CC)C1 25745,N1(C(C(CC)SC)=O)CCC2(CC1)CCN(C(c1cnn(C3CCC3)n1)=O)C2 25746,c1(C(=O)NC(C2CN(C(=O)CCCCC(N)=O)CCO2)C)cc(Cl)c(F)cc1F 25747,c1(C(N(CCC)OC)=O)ccn2c(-c3ccc(Cl)cc3Cl)nnc2c1 25748,c1(C(=O)NC2CCCCN(C(CC(=C=C)C)=O)C2)c(F)cc(O)cc1F 25749,c1(C(N2CCC(N(C(=O)C3=CC(C)(C)C3)CC)C2)=O)ccc2c(c1)C(=O)NC2=O 25750,c1(OCCC(=O)NC2(CC=C)CCN(C(C3C=CCC3)=O)C2)cc(Cl)ccc1Cl 25751,N1(C(CCN2C3CC(N)C2CC3)=O)CC(=O)Nc2ccccc21 25752,c1(COC)nn(C)cc1C(=O)NCCN(C(=O)C=C1CCCC1)C(C)C 25753,c1(OC)ccc(F)c(C(N2CCC(CNC(C3CCC=CCCC3)=O)CC2)=O)c1 25754,C1(NC(CCc2c(C)noc2)=O)CC(C)N(c2nc(-c3ccccc3)ns2)C1 25755,N1(C(C2C(NC(=O)Cc3cscn3)C=CCC2)=O)CC(O)C(O)C1CO 25756,S(=O)(=O)(c1ccccc1F)NCC(=O)NCCCNC(CCCCNC(C)=O)=O 25757,N(C(=NCc1ccccc1)NC1CC1(c1ccccc1)C)C1C(C)C1 25758,c12ccc(cc1)S(=O)(=O)N2.Cc1cc(CN(CCCCCO)C(C)C)cc(Cl)c1 25759,C1(C(=O)NC(CC)C)CN(C(c2ccc(O)nc2Cl)CC)CC1(C)C 25760,C1(NC(C2CCC(CCCC)C2)=O)CCN(C(C2CC3CC3C2)=O)CC1CC 25761,C(c1cn(C)c(=O)n(C)c1=O)=CC(=O)N(C1CCN(C(C(C)OC)=O)C1)C 25762,N1(C(c2nnn(C)n2)=O)C2CCC1CC(NC(=O)CCCC1CC1)C2 25763,C(=O)(C1CCc2nccn21)NCC1CCC(C(=O)NC2CCC(C)CC2)CC1 25764,C12(NC(c3cc(C)[nH]n3)=O)CCC(C(=O)NCCSC3CC3)(CC1)CC2 25765,C1(CNC(c2cc(C(C)C)no2)=O)CC(C)CN(C(=O)C(CO)N(C)C)C1 25766,c1(-c2occ(-c3c(CO)cccc3)n2)c(O)ccc(Cl)c1F 25767,c1(C(=O)NC(C)C(C)NC(=O)C(C)c2cncs2)cc2occc2s1 25768,C(=O)(C(CO)C(C)(C)C)NCC1(C(=O)NC(C=C)C(F)(F)F)CC1 25769,c1(OC)ccc(C(N2CCCC2CN(C)C(c2csnn2)=O)=O)c(Br)n1 25770,C=CC(CCC)CC(=O)NC1C2CCN(C(C3CCCC3F)=O)CC12 25771,C(C(O)CC(=O)N(C)CC1(O)CCC1)NC(CNC(CC(C)C)=O)=O 25772,N#Cc1cnccc1N1CCCCC1CNC(=O)CSCCO.C1(C)CCCO1 25773,c1(C(=O)NCC2C(C)CN2C(=O)CC2OCCC2(C)C)cc2ccccn2c1 25774,c1(C(N2CC(CC=C)(C(N3CCCC3CC)=O)C2)=O)c[nH]c(=NC)o1 25775,C(=O)(C1CCCn2nccc21)N(CC(CN(C(CCC=C=C)=O)C)O)C 25776,N1(C(c2cc(F)ccn2)=O)CCC2C1CCN2C(C1CC(O)C1)=O 25777,c1(NC(c2c(CCC=C)cc(Br)cc2)=O)ccc(S(=O)(=O)N2CCOCC2)cc1 25778,CC(C)CC(CNC(=O)C1=C(Cl)CCC1)C(=O)NC1CCCC(O)CC1 25779,Cc1ccc2[nH]cc(CCC(N3CCC(C)C3CNC(c3cccs3)=O)=O)c2c1 25780,c1(CNC(CC(=O)NCC)=O)cccc2c1CN(C(=O)CC1CCSCC1)C2 25781,N1(c2[nH]c(=NCC3COc4ccccc4C3)cc(C)n2)CCCc2c(O)cccc21 25782,C(=O)(CS(=O)(=O)C(C)(C)C)N1CC(O)(CNC(C2(C)CC3CCC2O3)=O)C1 25783,c1(SC)ccc(C)c(C(N2CCCCC2CCN(C)C(c2nnc(C)s2)=O)=O)c1 25784,N1(C(COCCC=C)=O)CCN(C2CCCN(C(=O)CSC(F)(F)F)C2)C(=O)C1 25785,Cc1ncc(CC(=O)NCC(C(C)C)NC(=O)C(C)CSC(F)(F)F)[nH]1 25786,c1(Oc2nc(-c3cc(OC)ncc3)nn2C)c(F)cccc1Br 25787,N1(CC(=O)NCCCN(C)C(c2ccc(CO)o2)=O)C(=O)c2ccccc2C1=O 25788,c1(NC(C2CCCC(NC(c3n(C)cnc3)=O)C2)=O)cc(Cl)ncc1[N+](=O)[O-] 25789,c1(C(N2CCCC(NC(c3c(CC)c[nH]c3)=O)C2C)=O)ncnc2c1CCCC2 25790,CCCC(C)(C)CC(=O)NCCC1(O)CN(C(c2ccsc2-n2cnnn2)=O)C1 25791,Cc1ccc2cc(C(=O)N(C3CCCN(C(c4sccc4C)=O)C3)C)nn2c1 25792,C1(OC)CN(C(=O)CC2(O)CCOCC2)CC1NC(c1coc(C2CCC2)n1)=O 25793,c1(C(=O)NC2C3CC(NC(CC(CC)C(C)C)=O)CC32)c[nH]c2cccc(Cl)c12 25794,CN1CC2C(NCC(=O)N=S(C)(C)=O)CCCN2C1=O 25795,c1(C(N(CC(CN(C(C2(NOCC)CC2)=O)C)O)C)=O)sccc1Cl 25796,c1(C(N(CC(CN(C)C)O)C)=O)sccc1C1CC1.c12cnn(c1)CNC2=O 25797,C1(NC(CN(C(=O)CC(C)n2cccc2)CCC)=O)CC12CCOCC2 25798,c1(NCC2CCC(=O)NC2)ccc(S(=O)(=O)NC(Cc2cccs2)CO)cn1 25799,C1(C(=O)Nc2c(C)nc[nH]2)C2CCC(C2)N1Cc1cncs1 25800,CN1CC2CCC(OC(c3ccc(COc4ccccc4)cc3)=O)C2C1 25801,c1(CC(=O)NC(C=CC(=O)NCC(C)CC2CC2)C)cnn(C)c1 25802,c1(CN(C(c2ccnn2CC(F)F)C(=O)NCC2CCOC2)C)ncc(CO)[nH]1 25803,c1(C(C2(F)CCC2)N(C(C(N2C(C(=O)NCC#C)CCC2)=O)=O)CC)cccc(C)c1 25804,N1(C(c2ncc(OCC)nc2)=O)CC2CN(C(=O)CCc3cccc(C)n3)C2C1 25805,c12c(cnn1C)C1CCCN(C1)C2.CN1CCC(NC(=O)OC(C)(C)C)C1 25806,CCCC(C(=O)NC(C(=O)N1CCC(CC(=O)OC)C1)C(C)OC)OCC 25807,C1(CN(C(C2(COC)CCOC2)=O)C)CCN(C(=O)CC(C)c2ccco2)CC1 25808,Brc1cc(I)c(C(F)(F)F)cc1NCC1CC12CCC2 25809,n1(CC(=O)NC(C)CC2CN(C(=O)CC3CC3)C2)ccc2ccccc12 25810,N1(C(Cc2cc(C)ncc2)=O)CC(C(=O)NCC=C2CCC(C)CC2)C(C)(C)C1 25811,c1(C(=O)OC(C(C)SC)C)ccc(NCCC(F)(F)Cl)cc1 25812,Cc1nc(O)nc2ccc(C(=O)NC3CCCC3NC(c3ccncc3Cl)=O)cc12 25813,c1(OC)ccc(N2CCCC2)cc1N1CCOCC1.N12CCOC(C1)NC2=O 25814,Cc1nnc(O)c(C(N2CCCC(CN(C(=O)CC#N)C)C2)=O)c1C 25815,CC(Cc1cccs1)N=c1[nH]c(N(C)Cc2ccc(Cl)cc2Cl)nc2c1CSC2 25816,Cc1cccc(C(=O)NC2CC(O)CN(C(=O)Cc3csc(C4CC4)n3)C2)c1C 25817,N1(C(c2n(C)ccn2)=O)CC2(CC(NC(C3(CCF)CC3)=O)CO2)C1 25818,c1(C(N2C(C)CCC(NC(Cc3c(C)nc(S)s3)=O)C2)=O)cc2c(ccn2C)[nH]1 25819,c1(C(N2CC3CC(C2)N(C(C2CCCOC2)=O)C3)=O)c(Cl)ccc2c1OCO2 25820,c1(C(=O)NCC(C)(C2CC2)NC(C2CCCN2CC(F)F)=O)ccccc1CO 25821,C(CC(C)(C)C)(C(=O)NCC1CCN1C(c1cc(C)[nH]c(=N)n1)=O)OC 25822,c1(OC(N2CCC(C(=O)O)C2)=O)ccccc1OCC1CCCO1 25823,C(C(C)(O)C(=O)N1CCC(CF)(NC(c2cccc(OC(F)F)n2)=O)C1)OC 25824,C1(CC=C)(NC(c2cocn2)=O)CC2CCC(C1)N2C(=O)CCSC(F)(F)F 25825,N1(Cc2ccc(C#C)s2)CCCN(C(c2nocc2Cl)=O)CC1 25826,N(C1CN(C(=O)C(c2cncn2C)N(C)C)Cc2ccccc21)C(C1C(=C)CC1)=O 25827,C(=O)(C(C(C)(C)C)NC(C1CN(C(c2ccc(C)c(F)c2)=O)CC1(F)F)=O)NC 25828,C(C(C)(C)CN(C(c1nnn(C)n1)=O)C1CC1)NC(C1CN(C(C)=O)C1)=O 25829,c1(OC)cncc(C=CC(=O)NC2(CN(C(=O)CN3CCCC3C)C)CC2)c1 25830,Cc1cc(C(=O)NCC(C)(F)CNC(c2ccnc(O)c2F)=O)nc(O)n1 25831,c1(C(=O)NCC(C)(C)NC(=O)C(F)F)ccc(OC(F)(F)F)nc1.c1(O)ccccc1 25832,c1(CC)cc(C(=O)NCC(CC)NC(C2CCCCC2(C)C)=O)ccc1OC 25833,c1(C(N2CC(C(=O)Nc3cc(Br)cc(Br)c3)C(O)CC2)=O)cccc2c1CCC2 25834,CCC(CCC(=O)NCC(CC(=O)NCC(C)(CC)CO)C1CCC1)OC 25835,C1(CNC(C(=CC2CCCC2)C)=O)CCCN(C(c2cc(C(C)(C)C)c[nH]2)=O)C1 25836,C(C1=CCN(C(C2CCC(F)CC2)=O)CC1)NC(C(C)C1CCCO1)=O 25837,C(=O)(CCCCCCCCN(C)C)NCC(C)NC(c1cc(C(F)(F)F)no1)=O 25838,c1(OC)cc(OC)c2c(c1)CCN(C(=O)C(C)Sc1nccn1C)C2(C)C 25839,c1(SC)ncc(N)c(C(N2CCC(F)(CNC(c3ncoc3C)=O)C2)=O)n1 25840,CCCCCCCCCCCCn1cc(CNC(=O)CCOCCO)nn1 25841,c1(C(N(C2C(C)CCC2)CCc2ccccc2)=O)cn2c(n1)CCCC2 25842,CC(C)(CNC(=O)CN1CCCC1=O)C(=O)NOCC=C1CCOCC1 25843,c1(CC(=O)NC(CC2CN(C(C(F)=CCC)=O)C2)C)ccc2c(c1)CCO2 25844,C1(C(N(C)CC2(O)CN(C(=O)CCn3ccnn3)C2)=O)COCC(C)(C)O1 25845,c1(-c2ccnc(CC(=O)OC(C(=O)OCC)C)n2)cccc(S(C)(=O)=O)c1 25846,C1(C(=O)NC2C(C(N(CC)Cc3ccoc3)=O)COCC2)CC2(C1)OCCO2 25847,c1(C(N2CCC(N(C(=O)CCc3cccnc3C)CC)C2)=O)cc(C)ccc1N 25848,C12(C(=O)NC3CCCN(C(C(CSC)OC)=O)C3)C3C4C1C1C2C3C41C(N)=O 25849,C1(NC(C2CCOC2=O)=O)C2CC3C(C2)C13C(=O)NC(CC1CCC1)CO 25850,c1(C(N2C(C)C(NC(=O)CC(C)(C)O)CCC2)=O)cc2c(nc1O)CCOC2 25851,CCC(C)(C(=O)N1CCC(C)N(C(c2cc(N)c(F)cc2F)=O)CC1)C(F)F 25852,C(=O)(C(C)(C)Cc1ccccc1Br)NCCN(C(=O)C=CC1CCOC1)C 25853,C(CN=C(NCSC(C)C)NC1CCC=CCC1)Sc1c(C)cccc1 25854,CC1(C)CN(C(=O)C=Cc2cncs2)CC(CNC(=O)C(F)(F)CC2CC2)O1 25855,N1(C(CC2(C)CCOCC2)=O)CC2CC(NC(=O)CCN3CCOCC3)C(C2)C1 25856,Cn1cnc2c1CN(C(C1(NC(c3cc(O)nc(O)n3)=O)CCCC1)=O)CC2 25857,Cc1ccc(F)cc1NC(=O)CC1(C)CN(Cc2ccc(Cl)cc2Br)C1 25858,C(=O)(C(=O)N=c1cc(C)o[nH]1)NC1C(F)(F)CCN(C(C(C)OCCOC)=O)C1 25859,c1(C(=O)NCCC(CCC)C)cc(C(N)=O)cc([N+](=O)[O-])c1 25860,Cc1ccc(F)c(C(N2CC(NC(c3ccc(C(C)(C)C)s3)=O)C(O)C2)=O)c1 25861,N1(C(c2c(C(=O)OC)cc3c(n2)CCC3)=O)CC(NC(=O)C(C)O)C2CCCC2C1 25862,C(=O)(C(CNC(=O)Cc1coc(C)n1)CC1CCCC1)NCCCCOCC 25863,N1(C(C)=O)CC(NC(C2(c3ccc(C)cc3)CCCC2)=O)CC1CO 25864,c1(OC)ccccc1NC(=O)C(=O)NC(CNc1ccc(C#N)s1)CO 25865,C12(CNC(=O)C(C3CC3)C3CC3)CCCCC1N(C(=O)Cn1cnnc1)CCC2 25866,Cc1nc(NCCNC(=O)CC2NC(=O)NC2=O)ncc1[N+](=O)[O-] 25867,C1(C(C)(C)O)(CNC(c2ccnn2CC(F)F)=O)CN(C(c2ccccc2)=O)C1 25868,c1(CN=c2ccnc(N(C)C3CC3)[nH]2)cc(N)ccc1S(C)(=O)=O 25869,c1(CC(=O)N(CCC)CCNC(C2CCS(=O)CC2)=O)ccc(C#N)nc1 25870,c1(CN(C(C2C(CC)C2)=O)CCNC(=O)Cc2ccsc2)ccc(Cl)cc1 25871,C1(C(N2CCC(CN(C(=O)CCP(C)(C)=O)C)C2)=O)CC(C)(C)OC(C)(C)C1 25872,c1(C(C)NC(=O)COC)coc(NC(=O)COC2CC2)n1.C(CC)OC 25873,C1(C(N(CC(=C)C)CC)=O)CCN(C(c2cnn(C)c2Cl)=O)C1(C)C 25874,CC(C)S(=O)(=O)C1CCN(C(CCCCC#N)c2nnnn2CC2CC2)CC1 25875,C1(CNCc2cc(SCC)no2)CC2(CO1)CN(c1ncc(C#N)cc1Cl)C2 25876,C1(NC(C2(C#C)CCN(C(c3cc(CC)nn3C)=O)C2)=O)CC2C(O)C(O)CC12 25877,c1(C(N2C(CNC(C3COC4(CCC4)C3)=O)COCC2)=O)coc2c1COC2 25878,c1(C(C(=O)NCC(C)(C)OCCNC(Cc2ccc(C)s2)=O)C)cccc(F)c1 25879,N1(C(C(C(C)O)(F)F)=O)CCC2(CCN(C(c3ccc4nc[nH]c4c3)=O)C2)C1 25880,N1(C(c2scc(CNC(C3(CC)CCC3)=O)c2)=O)CCCC2CC2C1 25881,N1(C(C(COC)N(C)C)=O)CCC2CN(C(=O)Cc3ccnc(C)c3)C(C)C12 25882,C(C)(C(=O)NOCC(=O)N(C)C)N(C(c1c(CC)[nH]cc1)=O)C 25883,C=CCCCCCCCC(=O)NCC(C1CC1)NC(=O)CCOC.c1(C)nccn1C 25884,c1(C(N2CCC(NC(=O)C(O)C(F)(F)F)C2)=O)n[nH]c2c1CCCC2 25885,C1(CCNC(CC2N(CCC)CCC2)=O)CCCN(C(=O)CCNC(=O)OC)CC1 25886,C(=O)(C(C)(C)C(F)F)NC(C(C)C)CNC(=O)CCN(C)CCO 25887,c1(C(=O)NCC(CN(C(C(CCC)C(C)C)=O)C)C)cccc2c1ncn2C 25888,C1(C#N)(C(=O)NCCC2N(C(C3(C)CCC(=O)N3)=O)CCCC2)CC(F)(F)C1 25889,c1(C(COC(C2CC2CC2CCCC2)=O)=O)cnn(C)c1 25890,C(CNC(=O)C(C)OC)(C(C)(C)C)NC(c1c(CC)scc1)=O 25891,C12(C(N3CCCCC3c3ccc(CO)cc3)=O)CC(CO)(C1)OC21COC1 25892,N1(C(C(CCC)OCC)=O)CC2(C1)SCCC2N=c1[nH]cc(C#N)c2ccsc12 25893,c1(C(=O)NC2CN(C(COC(C)(C)C)=O)CC3(C2)CC3)cc(F)cc2c1NCCC2 25894,C(C1=NOC2CN(C(=O)C(F)(F)C3CC3)CC12)NC(c1nccc(CC)c1)=O 25895,C=CC(CC(=O)NCC(C)(Cn1cccn1)NC(=O)CCOCC)c1ccco1 25896,C(=O)(C1=NN2CCC(C)N=C2N1)NC1CCCC(NC(C(C)=CC)=O)C1 25897,c1(OC)ccc(CO)cc1C(=O)NCC(C)(C(C)C)NC(C1CC1C)=O 25898,C1(NC(c2cnc(CC)o2)=O)CCCN(C(C2(c3ccno3)CC2)=O)CC1F 25899,Cc1nc(NC(C2CCCN2C(c2ccncc2O)=O)=O)cnc1Cl 25900,C1(CC(=O)NCCCN(C(=O)CC2CCCC23CC3)C)CCC(C)(C)CO1 25901,N1(C(C(c2cn(C)nc2)NC(CCC(F)CN=[N+]=[N-])=O)=O)CC(O)CC12CCOC2 25902,N1(N2C(C(=O)Nc3ccc(Cl)c(Cl)c3)COCC2)CC2CC1CC2(F)F.C=O 25903,C1(NC(CN(C(COC)=O)C)=O)CN(C(=O)CN(C)C2CC2)CC2(CC2)C1 25904,O=C(C#Cc1ccccc1)N1CCC(c2ccccc2)(N)C1.c1(N)ncncc1F.CC 25905,N12CC(CC13CCOCC3)NC2=O.N1(C(C2CC2)=O)C2CCCC1CC2 25906,c1(C(=O)NC(C)(C)CCCNC(=O)CC2(C#N)CC2)ccc2nonc2c1 25907,c1(N2CC(C)C=C(C)C2)nc(NCCc2c[nH]ccc2=N)c2ccsc2n1 25908,C(=O)(CC(CC1CC1)NC(=O)C(O)COC)NCC1(C2CC2)C(C=C)C1 25909,N1(C(c2cc(OC)cc(OC)c2)=O)CC(O)CC12CCN(C)CC2 25910,C(C)(CN=c1[nH]c(=NC2CC2c2cccs2)c2ccccc2[nH]1)c1ccc(C)cc1 25911,N1(C(c2c(CNC(c3csnn3)=O)c[nH]n2)=O)CC=C(CO)CC1 25912,C1(CC)C(NC(c2cc(O)nc(Cl)c2)=O)CCCN1C(=O)CC(C)(C)F 25913,c1(OCC(CCC)(F)F)ccc(Cl)cc1N1CCOCC1 25914,CN1CCCCC(C(N2CC=CC(NC(c3csc(C(F)(F)F)c3)=O)C2)=O)C1=O 25915,CCCC(CC)C(=O)NCCCN1CCN(C(=O)C(C)C(=O)OC)CC1 25916,CCC(F)(F)C(=O)NOC(CC(C)C)C(=O)NC1(c2nn[nH]n2)CC1 25917,N1(C(C2C(CC)OCC2)=O)CC(OC)C(NC(=O)CC23CCCC2C3)C1 25918,c1(CC(C(=O)NCCC(C)N(C)C(c2ocnc2C2CC2)=O)O)ccccc1Cl 25919,N1(C(C(C)N(C)C)=O)CC2CCC1C(NC(C1CCCN1Cc1ccccn1)=O)C2 25920,C=CC1CCCN1C(C1C(NC(=O)CSC(C)(C)C)CC1)=O 25921,N1(C(=O)NCC(=O)Nc2cncs2)CC2C(C(=O)NCC3(O)CCCCC3)C2C1 25922,c1(N(C(C)CNC(=O)C(C)S(N)(=O)=O)C)cc(C(F)(F)F)ncc1[N+](=O)[O-] 25923,c1(CC(N2C(CNC(c3c(C)ocn3)=O)CCCC2)=O)cc2ccccc2s1 25924,Cc1ccc(NC(=O)Cc2csc(NC(c3ccc(F)cc3Cl)=O)n2)nc1Br 25925,c1(CCOC(C2CC(C)N(C(=O)NC(C)(C)C)CC2)=O)ccccc1[N+](=O)[O-] 25926,C(=O)(C(CC(C)C)ONC(C1CC2(CCN1)CC2)=O)NCCC 25927,C1(C(=O)NCCN(CC(C)O)C(c2ccns2)=O)CCCCN1S(C)(=O)=O 25928,[N-]=[N+]=NC1COCC1NC(C1CC(F)(F)CN1C(=O)C(=O)N(C)C)=O 25929,CCCCCC(O)CC(=O)NCC1CC(NC(=O)C2=CCCC2(C)C)C1 25930,C1(C(=O)NCCC2CN(C(=O)CC(C3CCC3)C3CCC3)C2)(COC)C=CCC1 25931,c1(NCCc2ccc(CCN(C3CC4CC3CN4)C(N)=O)cc2)ccc(O)cc1 25932,c1(N(CC(C)C(C)(C)C)C)nc(N2CCCC(C)(F)C2)nc2ccc(Cl)cc12 25933,C1(C(=O)NCC2(CC(C)(C)C)CC2)CCCC(NC(C2(F)CC=CC2)=O)CC1 25934,c1(CC)ccc(F)cc1NC(=O)CCN(C(C12CCC(C1)C2)=O)CC1CC1 25935,CN1CC2CCC(C1)N2c1cc(NCCc2cn(C)cn2)nc(C(F)(F)F)n1 25936,CC1=C(C(=O)N2CCC(NC(c3cnn(CC(F)F)n3)=O)C(C)(C)C2)CCCO1 25937,N1(C(Cn2c(C)cc(C)n2)=O)CCOC2CN(C(=O)CN3CCCC3)CC12 25938,c1(CC(=O)NCC(CC)(C)NC(c2ncoc2C)=O)cc(Br)ccc1F 25939,c1(C(=O)NCCCOCCNC(CCC#C)=O)[nH]c(Sc2ccccc2)nc1C 25940,C(=O)(CC(C)(C)CC(=O)OC)NC1(CO)CN(C(CCc2ccc(CC)[nH]2)=O)C1 25941,c1(C(=O)NCC2CCN(C(C(C)C3(O)CCC3)=O)C2)ncc(N)cc1Cl 25942,C1(C(C)C)CN(C(=O)CC2CC=CC2)CCN1C(=O)COc1ccc(F)c(Cl)c1 25943,C1(CC=C)(NC(=O)Cc2ccnc(OC)c2)CCN(C(=O)C(C(C)C)OCC)C1 25944,Cc1cc(C(C)NCC(O)COc2ccccc2C)cc(C)c1 25945,N1(CC)CCOC(C(=O)NC2CCCC2NC(c2sccc2OC(C)C)=O)C1 25946,c1(C(N2CC(NC(C(CC)CC3CCC3)=O)C2)=O)c([N+](=O)[O-])c(C)nn1C 25947,N1(Cc2ccc(SC)s2)CCN(C(c2cc(Cl)cnc2F)=O)C(C#N)C1 25948,c1(OC)cc(C(=O)CCN2CCCCC2=O)cc(Br)c1.N1CCCC(O)C1 25949,N1(C(C2OCCN(CC)C2)=O)CCCC(C2CC2NC(C2CCCN(C)C2)=O)C1 25950,N1(C(CN2C(=O)CCC2)=O)C2CN(c3ncccn3)CC12 25951,N1(C(CCNC(CCNC(c2[nH]cc(C#N)c2)=O)=O)=O)CC(O)C(C2CC2)C1 25952,N1(C(C(CCC#C)O)=O)CC2(CCCCN(C(c3cc(C)on3)=O)C2)C1 25953,N1(C(C(C)=C2CCC2)=O)CCCCC(NC(=O)C(CN(C)C)C(C)C)C1 25954,Cc1cnc(C=CC(=O)NC2COCC2NC(=O)CC2COCC2O)[nH]1 25955,c1(OC)cc(C)ccc1C(=O)NCCCC1CCN(C(=O)CC=CC(C)(C)C)C1 25956,N1(C(CC2C(OC)CC2)=O)CCN(C(c2cocn2)=O)C(c2ncc[nH]2)C1 25957,C1(CNC(C=CC=CC)=O)CCC2(CN(C(=O)Cn3ccnn3)C2)O1 25958,C(=O)(C1CCc2c[nH]nc21)NC1(C(=O)NC(C2CCCCC2)C)CSC1 25959,N1(C(CCC#CC)=O)CCCC(C(=O)N(C)CC2CCOC2)CC1 25960,c1(C(=O)NCCC2N(C(Cn3c(=N)nc[nH]3)=O)CCCC2)cc(S(N)(=O)=O)c[nH]1 25961,Cc1[nH]nc(C(=O)NCC2CCCN(C(C3CC3C)=O)C2)c1C 25962,C1(CCOC)CN(C(=O)C(C)C(=O)OC)CCN1C(=O)CCc1cncs1 25963,c1(C(=O)NCCCCN(C)C(C2CC2c2cccs2)=O)c[nH]nc1C(C)(F)F 25964,N1(C(C(CC)NC(N)=O)=O)CCCC2(NC(=O)CCc3ncc(C)[nH]3)CC2C1 25965,c1(CCC)nc(=NC(C(C)NC(=O)CC2CCC(C(F)(F)F)O2)C(C)C)s[nH]1 25966,N1(Cc2c(C)ccnn2)CCCC(C(=O)NCC2CCCO2)CC1 25967,c1(CC(=O)NC2CN(C(C(C)OCC3CC3)=O)C(CO)C2)ccc(F)c(Cl)c1 25968,c1(-c2ccc(COC)cc2C)ccc2oc(C(N3CCCC3)=O)cc2c1 25969,c1(N(C)C)noc(CNC(=O)CONC(=O)CC2CCSC2)n1 25970,c1(NC(c2c(OC)cncc2)C)ccc(S(=O)(=O)NCC2C3CCCOC23)cn1 25971,c1(C(N2CC(NC(c3c(C)scn3)=O)C(C(F)(F)F)C2)=O)[nH]nc([N+](=O)[O-])c1Cl 25972,N1(C(C(CC)=CC)=O)CCN(C(C2CCOCC2)=O)CC1c1cccc(Cl)c1 25973,C1(CCNC(CCC(=O)C2CC2)=O)CCCN(C(=O)COc2cccnc2)CC1 25974,c1(C(N2CCC(=CCNC(C(C(C)C)C)=O)CC2)=O)c(F)ccc2occc12 25975,O=S1c2ccccc2CC1CCNc1nccc(=NCCSCC(F)(F)F)[nH]1 25976,C1(CCC)CN(C(=O)C(F)n2cccn2)CCN1C(=O)CN1CC(C)(OC)C1 25977,c1(C(N2CC3C(NC(C45C(C)(C)OCC4C5)=O)(C3)C2)=O)cc(Cl)cc2c1CCC2 25978,C#Cc1cccc(C(=O)N(CCNC(C2(COC)CCC2)=O)C2CC2)c1C 25979,C(=O)(C1=COCCO1)N(C)CC1CCN(c2cc(COC)ncn2)CC1 25980,N1(C(C2N(C)CCC2)=O)CCC(CCCCCNC(C2CC3CCC3C2)=O)CC1 25981,C1(c2nnnn2-c2c(C)noc2C)(NC(CCC)C)CCOCC1OC 25982,C(C(=O)NC12CC(NC(=O)CC(C)(F)F)(C1)C2)(C(C)C)NC(=O)OCC 25983,C1(C(=O)OC)OC2(C)CC1(COC(=O)NCCOc1ccccc1F)C2 25984,c1(N(C2CCCN(C(=O)C(C)(O)C3CC3)C2)C)ccc(Cl)cc1[N+](=O)[O-] 25985,C1(OC)COCCC1N(C(C1CCCOCC1)C(N1CCOCC1)=O)C1CCOC1 25986,c1(C(=O)NC2C(NC(CSC(C)(C)C)=O)CS(=O)(=O)C2)ccc2nncn2c1 25987,N1(C(C=CC(C)NC(C(C)NC(=O)NC)=O)=O)CCC(CO)C1(C)C 25988,C12CCN(C1)C(=O)CONC2=O.c1(COCCCOC)ncccn1 25989,S(=O)(=O)(c1ccc2ccccc2c1)CCCCNC(C(c1ccn(C)n1)(C)C)=O 25990,C(=O)(CP(C)(C)=O)NCC(CN(C(=O)C(C)O)CC)(C)C 25991,CCCCCCC(CC)C(=O)NCC1COCCN(c2nccn3nnnc23)C1 25992,C(N=c1[nH]c(=NC(CCO)c2ccccn2)[nH]c2c1CSC2)C1(C)CCCS1 25993,C1(n2c(C(c3ccc(C)o3)NCCC(=O)NCC)nnn2)CCC(F)(F)CC1 25994,N1(C(c2cnc(CO)nc2O)=O)CCC2C(CCCN2C(c2cnc(O)s2)=O)C1 25995,C(=O)(C1CCCc2nccn21)N(C)CC1OCCN(C(CC=C)=O)C1 25996,CCS(=O)CC(=O)NC(C)(CNC(=O)CN(c1cccc(Cl)c1)S(C)(=O)=O)C1CC1 25997,CCC(C)C(C)(O)CNC(C1CC(C)CN(C(=O)Cc2ccc[nH]2)C1)=O 25998,c1(SC)nc(=NCC2(NC(C3CC3(C)Br)=O)COC2)s[nH]1 25999,CCCCCCCCC(=O)NC(C)CN(C(=O)Cn1cc(F)ccc1=O)CC 26000,C1(NC(C(=O)NC(C)C)=O)CCC(F)(CNC(c2csc(Cl)c2)=O)C1 26001,C1(C(=O)NC2CC3(CN(C(CC(C)(C)C)=O)C3)C2)CCCC1S(C)(=O)=O 26002,C1(CNC(C(C2CCC(=O)N2)C)=O)N(C(c2cc(Cl)cc(F)c2)=O)CCC1(C)C 26003,c1(OC)ccc(Cl)c(C(=O)NCCC2(O)CN(C(=O)Cc3ccc(O)cn3)C2)c1 26004,C1(C(=O)NCC2N(C(CC3(CC)CCC3)=O)CC(F)C2)CC1C1CCCC1 26005,N1(C(CC2(C=C)CC2)=O)CC2CC(NC(=O)C(C)(C)F)CC2C1 26006,N1(C(C(C)CO)=O)CCCCC1CC(=O)Nc1ncc(Br)s1 26007,C(=O)(CC1=NN(C)C(=O)C1)NCCNC(c1cc(OC)cc(C)c1)=O 26008,N1(CC)CCC(n2nc(-c3cncc(F)c3)nc2COC)CC1 26009,C1(C(=O)NC)CCCCN1C(c1ccc(-c2cnn(C)c2C)o1)C(=O)NC(C)C 26010,C12CC(=NO1)C(=O)N(C)CCNC2.N1(CC)CCC(C(=O)OC(C)(C)C)C1 26011,C1(CC(=O)NC2CC2NC(c2cncc(CO)c2)=O)CN2CCN1CC2 26012,C1(C(=O)OC)CC2CC(C(=O)OCC3(O)CN4CCC3CC4)C1C2 26013,[N-]=[N+]=NC1(C(=O)NC2(CCCCO)CC2)CCN(C(=O)CC2CCOC2=O)C1 26014,S(=O)(=O)(CCC(F)(F)F)NC(C1CC1(F)F)=O.C12CN(CC1F)C2 26015,c1(NCc2c(OCC)ccc(F)c2)c(I)cc(F)c(Br)c1F 26016,C(CCCCCN=c1ccnc(NCCCc2ccccc2)[nH]1)OC 26017,C1(OC)(OC)CCC(C(c2nnnn2C)OC(C2CCCC2)=O)C1.C(C)(CC(C)C)N 26018,N1(C(C2(C)CCN2C(=O)CC2CC(F)(F)C2)=O)CCOC(C)(CC(N)=O)C1 26019,C1(SCC=CCNC(CCOCC(=O)OC)=O)CC(=O)c2cc(F)ccc2O1 26020,N1(C(c2cnc(CCCC)s2)=O)CC2CC(NC(c3cc4sccc4[nH]3)=O)C1C2 26021,N1(C(=O)N(C2(CCC)CCCC2)Cc2ccccn2)CCNC(=O)C1CC1CC1 26022,C1(NC(COC2C(C)CCCC2)=O)CCN(C(=O)CS(C)(=O)=O)CC1O 26023,C1(NC(C(CC)C)=O)CCC2(CC1)CN(C(=O)Cc1occc1C)CCO2 26024,C(CC(C)NC(=O)CC1(OC=O)CC1)N(C(=O)CCC1CCCC1)C 26025,C(c1cc(F)cc(F)c1)=CC(N1CC(C(C)NC(C2CCCCS2)=O)C1)=O 26026,c1(C(N(CCCNC(=O)CN2CCOCC2=O)C(C)C)=O)cc2ccsc2n1C 26027,c1(OC2CS(=O)(=O)C2)cccc(F)c1.CC1CCNC(=O)NO1 26028,CC(N=[N+]=[N-])C(=O)N(CCC(=O)NC1CCN(C)C1=O)C1CC1 26029,C1(NC(C2N(CC)CCC2)=O)CC2(CCN(C(c3nc(C)ccc3NC)=O)C2)C1 26030,Cc1cccc(C(=O)NCC2(CNC(=O)C=Cc3cncs3)CCCC2)c1O 26031,C1(CC)C(C(=O)NCC(O)COC)CCN1C(c1csnc1Cl)=O 26032,c1(C(=O)NC2CCN(C(c3nc(C)oc3)=O)C2C2CC2)ccc2c(c1)CCCC2 26033,C1(NC(C2(CNC(=O)Cc3cn[nH]c3)CC(=C)C2)=O)CCCCC1C(N)=O 26034,Cc1ccc(CC(=O)NC(CNC(C2CC(n3ccnc3)C2)=O)C2CC2)cc1C 26035,c1(NC(CN(C(c2csc(C)c2C)C(=O)NC)CCC)=O)cccc(OC)c1.N(C)C 26036,C1(CC)CC(C(=O)Nc2ccccc2Oc2ccccc2F)CN(C(=O)C2CC2)C1 26037,CCC(C)CCC(O)CC(=O)N1CC(O)(C(C)NC(=O)C(C)(C)S(C)(=O)=O)C1 26038,c1(C(N2C(CCNC(C3CCO3)=O)CCC2)=O)csc2ccc(F)cc12 26039,N1(C(c2c[nH]c(=NC)s2)=O)CC(NC(=O)C(Br)=C(C)C)CC(C)(C)C1 26040,c1(C(=O)NC23CCN(C(COCC#C)=O)CC2C3)c(Cl)c([N+](=O)[O-])nn1C 26041,C1(NC(c2cc[nH]n2)=O)CCCC2CN(C(=O)Cc3csc(C(F)(F)F)n3)CC12 26042,C1(C)(C(=O)Nc2cn(CCNC(CNC(=O)NC)=O)nc2)CNC(=O)N1.C1C(=O)N1 26043,c1(C(N(CC(O)CNC(C2(S(C)(=O)=O)CCCC2)=O)C)=O)ccc2c[nH]nc2c1 26044,c1(CC)c(C(=O)NC(C2CCOC2)CNC(=O)CN2CCCC2=O)cccc1F 26045,c1(OCc2occ(C)c2)cccc2oc(C)nc12 26046,N1(C(C2C(NC(c3ccccc3)=O)CCCC2)=O)C2CCC1CC(O)C2 26047,c1(OCCOC)ncccc1C(=O)NCC1CCC1NC(c1ccc(Cl)s1)=O 26048,C1(CNC(C(CCC)C)=O)CCN(C(=O)C(c2ccc(=O)n(C)c2)(F)F)C1(C)C 26049,n1(CCN(C(N2CC(O)(NCc3ccccc3)C2)=O)C)cc(Cl)c(C(F)(F)F)n1 26050,C1(C(=O)NCCN(C)C(=O)OC(C)(C)C)CCN(C(C2CCCOC2)=O)C1 26051,c1(C(=O)NC(C(C(C)C)N(C)NC(C=CC)=O)C)ccc(OC)nc1OC 26052,C12(CNC(CC3(C=C)CN(C(C4NC(=O)OC4C)=O)C3)=O)CCCN1CCC2 26053,C1(C)(CNC(c2ccc(SC)cc2)=O)CCC(NC(C2CC3CC3C2)=O)CC1 26054,c1(CCCC(=O)NCCC(C)NC(C2COCCO2)=O)ccc(F)c(F)c1 26055,CC1CCN(C(C2(N=[N+]=[N-])CCN(C(C3SCCS3)=O)C2)=O)CC1O 26056,C(C1CN(C(c2coc(C(F)F)c2)=O)CC1C(=O)NCC1CC(C)(O)C1)=CC 26057,CCCCC(CC)C(=O)NC1CN(C(c2cccc(C(N)=O)n2)=O)CC12CC2 26058,C(=O)(C(CO)C(C)(C)C)N1CCC(C(=O)Nc2ccsc2COC)(OC)C1 26059,C(=O)(CS(=O)(=O)C1CC1)NCC1N(C(c2c(C)cco2)=O)CCCC1C 26060,c1(OC)ccc(C(C)NC(=O)N(C)CC2(F)CCOCC2)cc1S(N)(=O)=O 26061,N1(C(C2CC(CC)C2)=O)CC2(C1)C(NC(=O)C(CC)C(C)C)CCS2(=O)=O 26062,Cc1nc2c(C(=O)Nc3ccc(C)c(-c4nn[nH]n4)c3)cccn2c1Br 26063,N1(C(C(C2CCCC2)OC)=O)CC(C2CCCCN(C(=O)C(C)(C)C(C)C)C2)C1 26064,CON1CCC(C(N2CCN(C)C(CNC(c3ccccc3SC)=O)C2)=O)CC1 26065,C1(NC(=O)CCC2CC(NC(=O)CC(Cl)Cl)C2)C=CC(C(=O)O)C1 26066,c1(OC)cc(OC)cc(CNc2nc(COC)oc2-c2ccncc2)c1.c1cn[nH]c1 26067,CC1CCC(CNC(=O)COCC2CCCO2)CN1C(=O)C=Cc1nccs1 26068,Cc1sc(Cl)c(C(N2CCN(C(=O)C(C)Cc3ccccn3)C(CO)C2)=O)c1C 26069,N1(C(c2cc(C)nc(O)c2)=O)CCN(c2snc(Cl)c2C#N)CC(C)(F)C1.C1C(=O)N1 26070,C1(CNC(=O)COCC2CCOC2)CN(C(c2cc(N)ccc2O)=O)CCCO1 26071,C(=O)(CC1=NNC(=O)C1)NC1CC(C)(NC(c2c(C)cc(F)cc2)=O)C1 26072,c1(C(N2CC(NC(C)=O)CC(C)(C)C2)=O)nnn2cc(C)nc(O)c12 26073,N=c1ncc(C(=O)NCC2(CO)CCN(C(=O)C(CO)c3ccccc3)C2)c[nH]1 26074,C(=O)(C1=NOC2(CCC2)C1)N1CCC(C)(CNC(C2(CC=C)CCOC2)=O)C1 26075,N1(C(C(CC)C(F)(F)F)=O)CC2(C=C(C(=O)NCC3CCSC3)CO2)C1 26076,Cc1cc(C)n(CC(=O)NCC(C2CCN(C(=O)Cn3cc(Cl)cn3)CC2)C)n1 26077,C(C#N)(C(=O)C(C)(C)C)c1cn(C(C)C(=O)NC2CC(C3(C)OCCO3)C2)nn1 26078,c1(OC)cc(C(=O)NC23CCC(CN(C(C4CC4(F)F)=O)C2)C3)sc1S(N)(=O)=O 26079,N1(C(C=CC=CC)=O)CC(O)(C2(CNC(c3ccc(=NC)[nH]c3)=O)CC2)C1 26080,Cc1nsc(C(=O)N(C)CC=CC(=O)NCCN2C(=O)CCC2=O)c1N 26081,N1(C(C(C)C2CCOC2)=O)CC(C(C)(C)O)(CNC(=O)CCCNC(N)=O)C1 26082,c1(N2CC(CNC(C3(CC)CCC3)=O)(OC)C2)ccnc(C(C)C)n1 26083,S(=O)(=O)(c1cn(C)nn1)NCCN(C(C(=O)Nc1cccc(C)c1)=O)C 26084,c1(C(=O)NCC(C)NC(=O)COc2ccc(F)cc2)cnc(Cl)cn1 26085,C(Cn1ccnn1)(C(=O)NCCc1nc(O)n[nH]1)NC(C1C(C)CC1)=O 26086,c1(C(=O)NC2C(CNC(C(CCC)(C)CC)=O)CC2)ccc2nccc(C)c2c1 26087,c1(CC(=O)NC(CO)C2CC2)cc(Cl)ccc1Br.c12ncccc1NC2=O 26088,C1(NC(C(C)(C)OC)=O)CC2CN(C(C3CC3(C)Br)=O)CC12 26089,C(CC(C(=O)N1CCCC(C(F)F)C1)NC(c1cccc[n+]1[O-])=O)N(C)C 26090,c1(C(N(CC(CC)NC(c2nonc2N)=O)C)=O)cccc(C)c1N 26091,C1(CCC)CN(C(=O)Cc2csc(Cl)n2)CCN1C(=O)C(C)OCC 26092,N=c1[nH]c(CCC(=O)NC2(CNC(=O)C(=O)NCC3CC3)CCC2)cs1 26093,Cc1cc(S(=O)(=O)N2CCCC(NC(C)(C)C(=O)O)C2)c(C)cc1-c1ccncn1 26094,C1(C(=O)NCC2N(CC)CC2)C=CCN(C(=O)CN2CC(=O)NC2=O)C1 26095,CCCC(C(=O)N(C(C)C(=O)NCC(C)(CC)CC)C1CC1)N(C)C 26096,N1(Cc2c(C)ncnc2)CCc2ccc(NC(C3(c4ccccc4)CC3)=O)cc2C1 26097,n1(CC(=O)NC2C(NC(c3c(C)ncn3C)=O)CCC2)ccc2ccccc12 26098,c1(NC(=O)NCC(=O)N(C)CCNC(C2CCCC(=O)O2)=O)cc(F)cc(F)c1 26099,N1(C(C2C(C)C2C)=O)CC(N(C)C(c2cccc(F)c2F)=O)C(C)(C)C1 26100,C1(CCNC(C(C)(C)SC)=O)CN(C(=O)Cc2nnc(O)s2)CC(C)O1 26101,c1(CN(C(C(C2CC=CCC2)NC(C(SC)SC)=O)=O)CC2CC2)ccccn1 26102,CC(CC(N)=O)C(=O)NC1CC(NC(c2cc(C3CC3)nn2-c2ccccc2)=O)C1 26103,N1(C(c2n(CC#C)ccc2)=O)CC2CCC2(CC(=O)N(CC)CC)C1 26104,c1(N2CCN(C(=O)NC(C)CCCC#N)CC2)nc2cc(Cl)ccc2s1.C(C)(C)O 26105,N1(C(C(C(C)OCC)C)=O)CC(C2CC2)OC(C)C1.C12(CCC1)C(=O)N2 26106,Cc1cc2c(cc1C)C(C(=O)N1CCC(C(C)CNC(C3(F)CC3)=O)CC1)CO2 26107,C1(CC)CN(C)C(=O)CN1C(c1ccc(F)c(CO)c1)=O 26108,Cc1cccc(C)c1CCC(=O)NC1CC12CC(NC(=O)CC13CCCC1C3)C2 26109,CCC(C)C(O)C(=O)NC1CCN(CCNC(=O)C(F)(F)C2CCCC2)CC1 26110,CC1(C)CC2(CC(C(N3CCN(C(=O)C=Cc4ncc[nH]4)CC(O)C3)=O)C2)C1 26111,CC(C)C(CN(C)C)C(=O)N1CCOCC(NC(=O)CCCN=[N+]=[N-])C1 26112,c1(C(N2CC3C(CNC(C(C)=CC)=O)(C3)C2)=O)cccc2cccc(O)c12 26113,c1(C(N2CCC(c3cccc(C#N)c3)C2)=O)c(F)ccc2c1OCO2 26114,c1(OC(CC)CNC2CC2c2ccc(C)o2)ccccc1OC(F)(F)F 26115,Cn1cc(NC(=O)NCCC2CC2(F)F)c(C2CCOCC2)n1 26116,C(=O)(CC(O)CC(C)(C)C)N(C(CC(=O)NC(CCC)C1CC1)C)C 26117,N1(C(C(C)C2CCCO2)=O)CC(C2CN(C(=O)C(C3CCC3)C3CCC3)C2)C1 26118,C1(NC(Cc2cnc(C)s2)=O)CCC(F)(CNC(C2CCN(CC3CC3)CC2)=O)C1 26119,CC(C)C(F)(F)CC(=O)N1CCCC(N(C)C(c2ccc(Cl)cc2)=O)C1 26120,c1(OC)cc(C=CC(N2CCCC2C(C)NC(c2cocc2C)=O)=O)ccc1F 26121,Cc1cc(C(=O)NC2CCN(c3nc(Cl)ncc3Br)CC2F)c2[nH]cnc2c1 26122,n1(CC)c(C(C)Cc2nccs2)nnc1-c1cnc(C2CC2)[nH]1.C1C(=O)N1CC1CC1 26123,C1(C(=O)NCCCN(C(c2ccc(CC(C)C)s2)=O)C(C)C)CCCCCCC1 26124,c1(CC(=O)N(C2(O)CCN(C(=O)CNS(N)(=O)=O)C2)C)cn(C)c2ccccc12 26125,N1(C(C(CC)(C)O)=O)CCC2(CCCC(CNC(C3(CCl)CCC3)=O)O2)CC1 26126,c1(C(N2CC3N(C(Cn4nnc(=N)[nH]4)=O)C(C3)C2)=O)cncc([N+](=O)[O-])c1 26127,C1(COC)CCC2(CCN(C(C3CCC(C(N)=O)CC3)=O)CC2)O1 26128,c1(C(N(C)CCNC(c2ccc3sncc3c2)=O)=O)cnn2cc(Br)cnc12 26129,N1(C(c2n(CCC)ncc2)=O)CC2C(CNC(c3ccc(Br)o3)=O)C2C1 26130,c1(OC)cc(C)c(C(=O)NCC2(F)CCN(C(C3COC(C)(C)C3)=O)C2)cn1 26131,C1(NC(c2cc(-c3ccccc3Cl)[nH]n2)=O)CN(C(C2(Cl)CC2)=O)CC12CCC2 26132,C1(NC(c2c(C)nc(CO)s2)=O)(CNC(=O)COC(F)(F)F)CCCCC1C 26133,C=CCC(CC=C)C(=O)N1CCC(C(=O)NC2(C)CCC(C)(C)CC2)CC1C 26134,Cn1nnc2c1CC(C(N1CCC(NC(=O)COCc3nc[nH]n3)C1)=O)CC2 26135,C1(C(N2CC(C(=O)NCC3(CF)CCC3)C2)=O)CCCOC1 26136,c1(OCC)ccc(C(C(=O)NCCC2(C)CC2)N(c2cccc(Cl)c2)C)nn1 26137,c1(C(=O)NCC=CCNC(C2N(CCC)C(=O)CC2)=O)nccc2nn[nH]c12 26138,c1(C(=O)NC2CCC23CCNCC3)nn(CCO)c(=O)c2ccccc12 26139,C(=O)(C1=C(Cl)CCOC1)NCC(C1CC1)NC(C1(C(=O)OC)CCCO1)=O 26140,N1(CC(=O)NCC(=C)C)CC(CSc2cnnn2C=C)C(O)C1 26141,C1(CCN(C(c2n(CC#C)ccc2)=O)C)CCCCN1C(=O)COCCOC 26142,c1(CC(=O)N(C2CCN(C(=O)C(C)(Cl)Cl)C2)C)cnn2c1OCCC2 26143,CC1(C)CN(C(=O)CC2(CO)CCC2)CC1NC(c1ccccc1F)=O 26144,N1(C(C=Cc2ccc(C)cn2)=O)CCC2(CC1)CC2NC(C1CC2C=CC1O2)=O 26145,c1(OC)cc(F)cc(F)c1-c1ccnc(OC(F)(F)F)c1F 26146,c1(C(=O)NCc2cc(C(=O)NCCN(C)CCO)sc2)cnnn1C 26147,C(=O)(CCC(F)F)NCC(Cc1ccccc1)N(C(COC)=O)C 26148,C(c1cccnc1C(F)(F)F)=CC(=O)N(CCN)C(C1CSC1)=O.C(=O)(C(C)S)OC 26149,Cc1nc(=N)[nH]cc1C(N1CCC(N(C(=O)C(C)O)C)C1)=O 26150,c1(C(C(=O)NC2CCC(NC(C3C(C)(C(F)(F)F)C3)=O)C2)O)cccc(Cl)c1 26151,C1(c2cn(Cc3cc(C)on3)nn2)CN(C(=O)CC2(C)CNC(=O)C2)CCO1.N(C)C 26152,C1(CNC(CC=CCC)=O)CN2CCCCC2CN1C(c1ccncc1)=O 26153,Cc1cc2cc(C)c1CC(=O)N1CCC(=CC(=O)N2)CC1.C1(=O)CCN1C.C1(CO)CC1 26154,N1(C(c2cccc(OCC)c2)=O)CC2(CC(NC(=O)C(C)(C)C3CCOC3)C2)C1 26155,N1(C(C(C=C)(C)O)=O)CC(C2CCCN(C(=O)C(c3ccccc3)F)C2)C1 26156,C1(C(=O)NC(CCOC)COC)CN(C(C2CC(C)=NO2)=O)CC1(C)C 26157,Cc1ncnc(C)c1C(=O)NCc1cccc(NC(=O)C(C)C(C)n2cccn2)c1 26158,O=C1Cc2c(C(N3CC4(CC4)CC3CNC(=O)C(F)C3CCC3)=O)cccc2N1 26159,C1(NC(C(C2CC2)OCC)=O)CCN(C(C2CC(N(C)C)C2)=O)CC1COC 26160,c1(C(N(CCCNC(CC(CCC)C)=O)CCC)=O)csc(=NC2CC2)[nH]1 26161,c1(CC(=O)NC2C3(CC(NC(C(CC)SC)=O)C3)C2)ccc(Cl)cc1F 26162,C(=O)(N1CC(O)CCO1)C1CCCN(C(c2cncc(CO)c2)=O)CC1 26163,C(C1(C)CCOCC1)=CC(=O)N(CCNC(C1C(C)(CC)C1)=O)C(C)C 26164,c1(C(=O)NC2CCC2NC(C(C)NC(=O)OC(C)(C)C)=O)cn(C)nn1 26165,Cc1cc2ncc(C(N3CCOC(Cn4cccn4)C3)=O)c(C)n2n1 26166,n1(CCOCC)cc(C(=O)NC(CNC(=O)OCCC(F)(F)F)CO)cn1 26167,Cc1sc(C(=O)NC2CCC(CCNC(=O)Cc3ccn(C)n3)C2)cc1Br 26168,N1(C(CCc2[nH]c(=N)sc2)=O)CC(NC(=O)COCCCF)CCC(O)C1 26169,c1(OCC(=O)NC(CC(C)NC(Cc2ccc(C)cc2)=O)C)cc(C)ccc1F 26170,C1(CNC(C(C)SCCCC)=O)CCCC(CNC(=O)CCc2nc(C)c(C)[nH]2)C1 26171,N1(C(CN(C)CC)=O)CC2CCCC1C2CNC(=O)C(C)(C)n1cccn1 26172,N1(C(c2n(C)ncc2I)=O)CC2(C1)SCCC2NC(C1CC12CCSCC2)=O 26173,c1(C(=O)NCCOCCCN(C(=O)CCCc2ccncc2)C)ccc(OC)cc1 26174,c1(C(N2CCC3CCN(C(=O)C(F)(F)C4CC4)CC23)=O)cc2cc(F)ccc2o1 26175,c1(C(=O)NC2C3(NC(c4cc(C)nn4C)=O)CCC(C2)C3)cccc2[nH]ncc12 26176,CCC(O)C(F)(F)C(=O)N1CCCC(C(=O)NC(CCO)C2CC2)CC1 26177,Cc1cnc(C(N2CCOC(CCNC(=O)C(C)(C)CF)C2)=O)nc1 26178,c1(CNC(NCC(C=C)(C)C)=NCCN2CC3CCC2C3)cn(C)c(=O)nc1O 26179,CCC(CC)(CCNC(=O)C=NOC)NC(C1CCC1n1cccn1)=O 26180,c1(N(N2CCCC2c2cnn[nH]2)C)ccc2nnn(C(C)(C)C)c2c1.CCO 26181,c1(C(=O)NC2C(NC(c3c(C)cc(O)cc3)=O)CCC2)[nH]nc2c1COC2(C)C 26182,C(C1=CCN(C(C2(C)CCN(C(=O)CCNC(C)=O)CC2)=O)CC1)OC 26183,C(=O)(CCC(C)N(C)C)N(CC(C)NC(CN(CC(COC)(C)C)CC)=O)C 26184,C1(C(N(C)CC2N(C(c3c(CCC)n(C)nn3)=O)CCC2)=O)CC2CC1C1CC21 26185,CCCCC(CC)CCCC(=O)N1CCC2(CCN(C(C3CCC(=O)O3)=O)C2)C1 26186,N1(C(C2(CNC(CCn3cnc(=N)[nH]3)=O)CC23CCC3)=O)CCC(C2CCC2)C1 26187,C(=O)(CCCS(C)(=O)=O)NC1COCCN(C(C2CCC(C)(C)C2)=O)C1 26188,C1(n2cc(C3CCN(C)C3)nn2)C=CCC(C(N2CC(n3ccnn3)C2)=O)C1 26189,C(C(C)(CNC(c1cscc1Cl)=O)OC)NC(C(C)OCCC=C)=O 26190,CC(C)C(CCNC(c1ccc(N(C)C)cn1)=O)NC(=O)CCN1CCCCC1 26191,c1(C(N2CCC3CN(C(C4(O)CC(F)(F)C4)=O)CC23)=O)ccn2ccnc2n1 26192,N1(C(c2c(C)nc[nH]2)=O)CC(CNC(=O)Cc2cnc(C(F)(F)F)s2)C(C)C1 26193,N1(C(C(C(C)C)C(C)C)=O)CCC2CCN(C(=O)NC3(n4ccnn4)CC3)CC12 26194,CCCCC(C)C(=O)NCCCC(O)C(=O)NCCCC(=O)NO 26195,N1(C(c2c(N)cnc(Cl)c2)=O)CCC2CC(NC(C3CCCCO3)=O)CCC2C1 26196,c1(C(N2CCC(O)(C(=O)NCCC(=O)NC(C)(C)C)C2)=O)c(O)cccc1[N+](=O)[O-] 26197,n1(C(C)C)ccc(C(=O)NCc2cc(C(=O)NCCNC(=O)C(C)(C)C)cs2)n1 26198,CNS(=O)(=O)NCC(=O)NCC1COCC1n1cc(COCP(C)(C)=O)nn1 26199,C(CC(CC)C(=O)N(C1CN(C(C2CC(n3ccnc3)C2)=O)C1)CCO)=CC 26200,C1(NC(c2n(CC)ccc2)=O)CN(C(=O)C(C)C2CC2)CCC12CCOCC2 26201,C1(F)(C(=O)NCC(C)(C)CNC(C2CC23CC3(CCC)C)=O)CCCCCC1 26202,C12CC3CCC1CC3NC(=O)N(CC)CC(=O)N2.C(=O)(CC1CC1C)OC 26203,c1(C(N(CCN(C(=O)CCc2ccnc(Br)c2)C)C)=O)ccccc1C#N 26204,C1(C(C)C(=O)NCC2CCOC2=O)CCN(C(=O)CCOC2CCCC2)CC1 26205,c1(C(=O)NCC(CN(C(COCCCC)=O)C)C)ccc(F)c(C(F)(F)F)c1 26206,CCC(C)(C)CC(=O)N1CC2CC(NC(=O)C(c3ccc(C)cc3)=O)C1C2 26207,C1(NC(C23CC(C)(C2)C3)=O)CCC2(CC1)CCN(C(=O)CC1(C#N)CC1)C2 26208,Cc1c(C(=O)N(C2CCCNC2)C)cccc1Br 26209,c1(OC)c(Cl)ccc(Cl)c1CN1CCC(N)CC1.c12ccc(cc1)C(C)NC2=O 26210,C1(C(=O)NC2C(CNC(C(F)=CCC)=O)CCC2)CCCNS1(=O)=O 26211,Cc1ccc(C)c(C(N2CC(C(C)NC(=O)CSc3nncn3C)C2)=O)c1 26212,c1(C(=O)NCC2C(CNC(c3cn(CCC(C)C)nn3)=O)C2(F)F)ccc(C#N)o1 26213,N=c1[nH]cc(C(=O)NCC2CC(O)(CNC(C3(C(F)F)CCC3)=O)C2)o1 26214,Cc1oc(-n2cccc2)c(C#N)c1C(=O)NCC(O)CNC(C1CCC(=O)O1)=O 26215,Cc1ccc(N)c(C)c1C(N1CC2CCCC2(NC(C2CCC(O)C2)=O)C1)=O 26216,C1(CNC(CN(CC)CC)=O)CCCC(N=c2[nH]c3ccc(Cl)cc3s2)C1 26217,c1(C(N2C(CNC(c3ccc(F)cn3)=O)CC(OC)C2)=O)ccc2ccsc2c1 26218,N1(C(C(CCC)O)=O)CC2(CCN(C(C3CCCCO3)=O)CC2)CC1C 26219,Cc1cc(C(N2CCC(C)C2CNC(=O)Cn2ccnn2)=O)cc(F)c1 26220,C1(C(N2CCC(NC(c3ccc(CSC)o3)=O)C2)=O)CC(C)CC(C)(C)C1 26221,c1(CC(=O)NCC(C2CC2)NC(C(C)OCCC=C)=O)ccc([N+](=O)[O-])c(N)c1 26222,C=CC(CC)CC(=O)NC(C)C(CO)NC(=O)C(c1ccccc1)=O 26223,N1(C(C(=O)NC(C(CC)OC)C2CC2)=O)CC2(C(F)(F)F)CC2(CC(C)(C)C)C1 26224,CCCCC(O)C(=O)N1CC(NC(=O)CCc2ncccn2)C(n2ccnn2)C1 26225,N1(C(CC2C(NC(c3n(C)nc(O)c3)=O)CCCC2)=O)CCOC2CCCC12 26226,Cc1ccc(F)cc1C(F)(F)C(=O)NCC(C)CN(C)C(C1CC2(CSC2)C1)=O 26227,N12CCC(C1(C)C)CC2=O.Cn1nncc1C(=O)NCCNS(N)(=O)=O 26228,C1(CNC(C=CCCC)=O)CC2CC(C1)N(C(=O)CCc1cccnc1)C2 26229,CC(C)(CCCNC(c1sc(OC(F)F)nc1Cl)=O)NC(C1CCC(=O)O1)=O 26230,c1(C(N(CCC)CCNC(=O)CCSc2ccc(Cl)cc2)=O)cccc(F)c1 26231,N1(C(C=CCN(C(C(C)(C2CC2)NC(C)=O)=O)C)=O)CC(C)CC(C)C1 26232,Nc1c(C(=O)NCCCCN(C(C2C3CC4C(C3)C24)=O)C2CC2)ccc(Cl)c1O 26233,c1(C(NNC(=O)c2ccccc2Cl)=O)cnc2ncnc(O)c2c1 26234,C1(OC)CCC(C(=O)NC2CC2CNC(=O)CCc2cccs2)C1 26235,c1(CC)cc(C(=O)NCC(O)C(=O)NC(C(=O)OC)C2(C)CC2)no1 26236,C(=O)(CC1COCc2ccccc21)N1CCC(NC(CN(C)C(N)=O)=O)C1(C)C 26237,CCCCCCCC(=O)N1CCC(NC(=O)COc2cc(F)cc(F)c2)C12CC2 26238,c1(Cc2nc(CNC(CCC3CCC(C)O3)=O)sc2)cccc(P(C)(C)=O)c1 26239,c1(C(=O)NCC(CC)(C)NC(=O)C(C)C)cc(F)cc(Br)c1 26240,N1(C(=O)Nc2ccc(-c3n(C)ncc3)nc2)CC2CCN(CNC(C)(C)C)C2C1 26241,N1(C(c2ncc(C)nc2)=O)CCC2(CC1)CN(Cc1nccs1)CCO2 26242,C1(CN(C(C(C2CCCC2)OCC)=O)CC(=O)NCC(C)C)COCCO1 26243,c1(CC)nn[nH]c1C(=O)NCC(O)C(=O)N1CCC(c2cnn[nH]2)C1 26244,CC#CCC(C(=O)NCC(C)(O)CCO)NC(=O)C(C)CC1CCC1 26245,C1(c2n(C(CC)(C)C)nnn2)(NC2CCCC2)CCN(Cc2c(C)cnn2C)C1 26246,C1(NC(CCN(CCC)C)=O)CCCN(C(=O)CCCSC)C1 26247,c1(C(C)C)ccc(C(N2CCC(F)(CNC(c3cnco3)=O)CC2)=O)c(O)c1 26248,c1(C(=O)NCCN(C(=O)C=CCO)C)cc(I)cnc1O 26249,c1(CN2CCC(O)(NC(CNC(CC(C)C)=O)=O)C2)ccc2ncccc2c1 26250,C1(NC(CCC2(C)CC2)=O)CCC12CN(C(=O)NC1CC(=C3CCCC3)C1)C2 26251,CC1(CC(=O)NCCC2CCCN2C(c2csc(Cl)n2)=O)CC1(F)Cl 26252,C12(CNC(CC(C)(C)C)=O)CN(C(=O)C=Cc3ccc(F)nc3)CC1CCO2 26253,C1(NC(c2cc3sccc3s2)=O)CCN(C(=O)CC2=CCOCC2)CCC1CO 26254,S(=O)(=O)(c1ccccc1)NCC(=O)N(C)CC1NC(=O)CC1OC(=O)CO 26255,C(=O)(C1CCCn2ccnc21)NC1CC2(C(NC(CC(C(C)C)(F)F)=O)C2)C1 26256,c1(OC)cc(C(=O)N(C)CC2CCCN2C(c2ccn(C3CC3)n2)=O)sc1Cl 26257,C(=O)(C(CC)CCC1CCCC1)NC1C(CC)CN(C(c2cocn2)=O)C1 26258,c1(C(=O)NCCC(CNC(c2c(CC)onc2)=O)O)cccc2ncc(C)n12 26259,Cc1ocnc1CC(=O)NC(C)(CNC(C1(C)CCCS1)=O)CO 26260,c1(C(=O)NCCN(CCCN(C)C)C(C2C(C)C2C)=O)nc(N(C)C)nc(=N)[nH]1 26261,c1(OC)cc(F)c(C(=O)NCC2CCC(NC(=O)C(CO)N(C)C)CC2)c(F)c1 26262,c1(C(C)=O)cccnc1N1CCCC(=C(F)CNC(=O)C(C(C)C)N(C)C)C1 26263,CC(C)C(F)(CNC(=O)CC1CCCSC1)C(=O)N1CCCC(C)(N(C)C)C1 26264,c1(CC)nc(C(=O)NC2CCC(NC(=O)COCc3cc(C)on3)C2)co1 26265,C#Cc1ccc(CC(N2CCCC(NC(C3(F)CCS(=O)(=O)C3)=O)C2C)=O)cc1 26266,N1(CC(N2CCC(NC(CCc3onc(C)n3)=O)C2)=O)CCCC(C)C1 26267,C1(C(=O)NCCOCCCC)C2CC2CN1C(c1[nH]ccc1CC)=O 26268,Cc1csc2ncc(C(=O)N(CC(O)CN(C)C(C3(Cl)CC3(C)C)=O)C)c(=O)n12 26269,c1(OC)ncnc2[nH]cc(C)c12.c12ccc(cc1F)[nH]c2=O.C12(COC1)CN2 26270,N1(C(Cn2nc(C)oc2=O)=O)CCCC1C1CCCN1C(c1cc(C)n(C)n1)=O 26271,C1(C(=O)OC)CC(C)N1C(C1(NC(c2cnc(C(C)C)o2)=O)CC1)=O 26272,c1(C(N2CCCC(N(C(=O)C3=NOCC3)C)C2)=O)ccc2c(c1)C(=O)CCN2 26273,c1(CC)cc(C(N2CC(NC(=O)CC=C(C)C)C(C)C2)=O)cc(O)n1 26274,c1(SC)ccccc1CC(=O)NCC(O)CNC(=O)CC#N 26275,C1(NC(C(C)(C)OC)=O)CN(C(c2cncc(C(C)(F)F)c2)=O)CC1CO 26276,C1(CC)CCN(C(=O)Cc2cc(C)on2)C1C(=O)NC(c1nncs1)C 26277,c1(C(=O)NC2C(C(=O)NCC(COC)C)CCC2)ccc2ccccc2c1 26278,C(C(O)CC(=O)NC1(CNC(c2c(C)coc2C(C)(C)C)=O)CCOC1)SC 26279,C1(C(=O)NCC(CC)NC(C2CCCCCCC2)=O)OC2CCC1CC2 26280,C1(N(C(=O)C(C)c2ccco2)CCC)CCN(C(=O)Cc2coc(C)n2)CC1 26281,c1(CC)cn2c(n1)CCC(C(=O)NC1CC(CNC(C3(C)COC3)=O)C1)C2 26282,C(=O)(C(C)(C)CC(=O)NCc1nc(CNC(=O)CCc2csnn2)cs1)OCC 26283,C(=O)(C(CCS(C)=O)N(C)C)NC1CCN(C(CCCOC)=O)C1(C)C 26284,C12(C(=O)NC(C)CNC(C3COC(=O)N3C)=O)CC3CC(C)(C1)CC(C)(C3)C2 26285,C1(NC(C(CC=C)C)=O)CCN(c2ncc(C(F)F)cn2)CC1C 26286,c1(OCCOC)ccc(C(=O)NC2CC2NC(C2SCCCS2)=O)cc1N 26287,c1(C(N2CCN(C(CNC(CCC)=O)=O)C(C(F)F)C2)=O)c[nH]c2cnccc12 26288,c1(C(c2n(C)nnn2)NCc2cnoc2C(F)(F)F)nn(C)cc1I 26289,c1(OC)c(C)cc(NC(=O)Cc2csc(NC(=O)C(C)(C)CCl)n2)cc1C 26290,Cc1ccc(C2CC2)c(NC(=O)N(C)Cc2c(C)noc2-c2ccc(Br)cc2)c1 26291,C1(NC(CNC(C)=O)=O)CCN(C(C2CCCCS2)=O)CCC1(F)F 26292,C(CCS(=O)(=O)NCC(=O)NC1CCC(CNC(=O)COCCN(C)C)C1)OC 26293,c1(-c2cn(C(C(=O)NCCN(C3CC3)CC)C)nn2)cccc(N)c1C#N 26294,C1(OCC)CCCC1CNC(c1ncoc1CNC(c1sccc1CC)=O)=O 26295,c1(OC)c(C(=O)NC2CCC2NC(C23CC(F)(C2)C3)=O)cc([N+](=O)[O-])cc1Cl 26296,C(CCCC(C)(C)C)NC(C1CC=CC(NC(C(CC=CC)C)=O)C1)=O 26297,C1(COC)CCCCN(C(=O)C(N2CCSCC2C)=O)C1 26298,CC1CC(NC(=O)C=Cc2ccc(Br)cc2)CN(C(=O)C(C)NC(N)=O)C1 26299,c1(NC(c2ccc(Br)c(Cl)c2)c2n(CCSC)nnn2)ccc(Br)c(C)c1 26300,N1(C(C(C)C2CCCC2)=O)CCC(C2CCN(C(=O)C(C)(O)C3CCC3)C2)CC1 26301,c1(OCC)ncc(S(=O)(=O)Nc2cc(C#N)ccc2Cl)s1 26302,CCC(F)(F)C(=O)NCC(O)CCNC(c1nc(Cl)sc1Cl)=O 26303,N(C(=NCC1CCN1c1ccc(F)cc1)N)CC1(n2cnnc2C2CC2)CC1 26304,C=CCCCC(C(=O)NOCCOCC)NC(c1nscc1C)=O 26305,C=CCCCC(=O)NCC1(CNC(C2CCC(C)CC2)=O)CC1(F)F 26306,c1(C(N(CC(C)CNC(=O)CC(C)P(C)(C)=O)C)=O)ccc(F)c2ncccc12 26307,C(=O)(C(CC(F)F)N(C(=O)CCC1CCCOC1)C)NCCCOC(C)C 26308,c1(OC)cccc(CC(O)C(=O)NCC2CN(C(=O)CCC3CCC(=O)N3)C2)c1 26309,c1(C(N2CCCC2c2ccc(F)cc2)C(=O)NC2CC2)cc(C2CC2)ccc1Br 26310,N1(C(c2cnn(C)c2C2CC2)=O)CCC(NC(C2(C)CC=CCO2)=O)CC(O)C1 26311,C1(C)(C(=O)OC)CN(CC(=O)NC2OCCC2c2ccccc2)CCO1 26312,C1(c2cn[nH]c2)C(C2CC2)CCN1N(c1coc(Br)c1)C(c1c(C)cco1)=O 26313,N1(C(C2(CC)CCCC2)=O)CC(NC(C2CN(C(C)=O)C2)=O)CC1(C)C 26314,N1(C(CC(=O)OC)=O)CCC2C1CCCN2C(c1ccc([N+](=O)[O-])c(C)c1)=O 26315,C1(C(C(=O)NCC(=C)C)N(CC(C)OC)CC)CCSC1(C)C 26316,CCCCCC(O)C(=O)NCC1CN(C(=O)C(=O)NCCOCCOC)CCO1 26317,N1(C(c2cc(OC)nn2C)=O)CC2CC(O)C1C2NC(=O)CC(C(F)(F)F)OC 26318,c1(C(N2CC(NC(C(CC=C)C)=O)C(C)C2)=O)cc(F)ccc1Cl 26319,C1(C)(C(N(CC(C(=O)OC)C)C)=O)CCN(C(=O)C(C)COC(C)C)C1 26320,C12(NC(C3C(C)C3C)=O)CN(C(c3cc4c(s3)CCC4)=O)C(CN(C)C)(C1)C2 26321,C(C#N)(C(=O)C(O)c1ncc(F)cc1F)n1c(C(=O)OCC)ccc1 26322,c1(-n2cc(C(N(C3CN(C(=O)C=CC(C)(C)C)C3)C)=O)nc2)cccc(Cl)c1 26323,CC(C)C(F)(F)CC(=O)NC1CC(CNC(c2ccc(O)nn2)=O)C12CCC2 26324,c1(C(CC)O)ccc2c(c1)CCN(C(C1(C)CCN(C(=O)OC(C)(C)C)C1)=O)C2 26325,N1(C(C)=O)CC2COCCC2(NC(c2cccc([N+](=O)[O-])c2Br)=O)C1 26326,C1(CN2CC(N(C(C(CC)n3nccc3C)=O)C)C2)CCC(OC)CC1 26327,c1(C(=O)CN2CCC(CCNC(c3c(C)c[nH]c3)=O)C2)cncc(OC(F)F)c1 26328,c1(NCC2(COC)CC2)nc(=NC2CCCSCC2)[nH]c2c(C)nn(C)c12 26329,N1(C(C2(C)COC2)=O)CCC2(NC(c3ccc(-c4cccs4)[nH]3)=O)CC2C1 26330,c1(C(CNC(c2c(C)cncc2)=O)NC(c2ncccc2N)=O)cc(F)cc(Cl)c1 26331,C1(C(N2CCC(CCOC)C2)=O)CCC(C)(C)N(C(=O)C#CC(C)C)C1 26332,n1(CC(=O)NCCCNC(=O)N(C2CC2)C(C2CCC2)=O)cc2ccccc2n1 26333,c1(C(N(CCCNC(C2ON=C(C)C2C)=O)CC)=O)cnc2sccc2c1 26334,C#CC1CC2CCC1N(C(C1(C#C)CN(C(c3cnn(C)c(=O)c3)=O)C1)=O)C2 26335,CC1(C)OC2(C(N3CC(OCCNC(=O)CCn4cccn4)C3)=O)CCC1CC2 26336,C1(C(=O)NC2CN(C(CC)=O)C2)C(C)CCN1C(=O)CCC#N 26337,C1(C)(CNC(C(CC)SC)=O)COCCN(C(c2ccn(CCOC)n2)=O)C1 26338,C1(NC(C=C(CCC)C)=O)(CNC(=O)Cc2nc([N+](=O)[O-])n[nH]2)CCCCCC1 26339,C1(C(=O)NCC2CC(O)CN2C(c2cn(C)c(C)n2)=O)(COC)CCOCC1 26340,N1(C(c2cccc(OCC)c2)C(=O)NC2CCCC2)CC(C(N)=O)C2(CC2)C1 26341,C12(CSCC)CC(C(N3CCC(C)(CCNC(=O)CC=C(C)C)C3)=O)(CO1)C2 26342,c1(C(=O)NCCCN(C(Cc2c(CC)con2)=O)CC)cc(Cl)ncc1O 26343,C1(C(N2CC(F)C2)=O)C(C)CCCN1C(=O)CC1CN(C2COC2)C1 26344,C1(NC(CN(CCC)C)=O)(CNC(C2(CC=C)CCOC2)=O)CCCC1 26345,CC1CC(C(=O)NCC2(NC(=O)CS(N)(=O)=O)CCCCC2)CCS1(=O)=O 26346,C(=O)CCCC(F)F.Cc1ccc(OCCCC2N(CC(CO)O)CCC2)cc1 26347,C1(F)(CNC(C2C(C)(C)C2)=O)CC(NC(c2cnsc2Br)=O)C1 26348,C1(CNC(C(=O)NCC(CO)OC)=O)CCCOCC1 26349,C=C(C)CCCC(=O)NC(C)CCCCNC(=O)C(C(C)(C)C)N1CCNC1=O 26350,c1(CNC(CC2CC(NC(=O)CC3CCCO3)C2)=O)ccncc1CO 26351,CC1CCN(CC(=O)NCCCN(CCCNC(C2CCSCC2)=O)C)C1 26352,C(CCCCCF)OCCNC(=O)N(CCCF)CC 26353,c1(NC(=O)NC2C=CC(CC)C2)cc(Nc2csc(C)n2)ncn1 26354,c1(C(=O)NC2(C)CN(C(c3nc(NC(C)=O)cs3)=O)C2)cncc(N=[N+]=[N-])c1 26355,CCC(C)(CC)C(=O)NCC1CN(C(=O)CC2CC(CC)=NO2)C1 26356,N1(CC)CCCCC1C(=O)NCC1CCCCN1C(C1NC(=O)OC1C)=O 26357,CC(O)CCCCCC(=O)N1CCN(C(=O)CC2CCC2)C2CCC12 26358,c1(C(C)(C)C(=O)NCC2CCC(NC(C3CC=CC3)=O)C2)cccc(Cl)c1F 26359,c1(C(=O)NCCC2N(C(C3=CCCC3C)=O)CCSC2)n[nH]c2ccc(F)cc12 26360,N1(c2cc(N(C)CC3CCOCC3)ncn2)CCC(O)(NC2CCCCC2)CC1 26361,C1(C(=O)NC)CN(C(=O)CN(C)C(=O)C2CC2)CC1(C)C 26362,C1(CNC(Cn2c(C)ccn2)=O)CN(C(=O)CC2C=CCC2)CC1(C)C 26363,c1(NC(C(C)NCC2CCCC2N2CCOCC2)=O)ccc(N)cc1 26364,c1(C(=O)NC(C2(O)CN(C(=O)CC3CCC3(C)C)C2)C)cnccc1Cl 26365,C(=O)(C1SCc2cccnc21)NC1(CNC(C2CCN(CC)C2)=O)CC1 26366,c1(CCC(N2CCCN(c3ccccn3)CC2)=O)ccc2c(c1)CCC2 26367,c1(OCC)cccc(F)c1C(=O)NCCC(O)C(F)(F)F 26368,c1(NC(C2CCCC(NC(Cc3c(C)cccc3)=O)C2)=O)c(Cl)cc(Cl)nc1Cl 26369,CCC(CC)(C(=O)N(C1CC(NC(C2CC(C)(C)CO2)=O)C1)C)C(C)C 26370,C1(NC(C(=O)NCCOC)=O)CCC(CNC(=O)CC2CCOC2)C1 26371,c1(OC)cc(CNCC(C(=O)O)OC)cc(I)c1OC(F)F 26372,C1(NC(Cc2c(C)nn(C)c2)=O)CCS(=O)(=O)C12CN(C(c1[nH]cnc1C)=O)C2 26373,c1(OCC)cc(C=CC(=O)NCC2CCCC(C)(C)O2)ccc1OC(F)F 26374,c1(CC)cc(C(N2CC(CC(F)C(=O)NC(C)CCC3CCCO3)C2)=O)ccn1 26375,C1(NC(C2CC(C)(CC)C2)=O)CCCC2CN(C(=O)C=Cc3ccccc3)CC12 26376,c1(CC(=O)NC2CC(NC(C3CC(Cl)(Cl)C3)=O)C2)cnc2ncccn12 26377,CCCCCC(CC)C(=O)NCC1CCOC1C(=O)NCC1CCC(=O)NC1C 26378,C(=O)(C(C)(C)CCSC)NCCC1CCN(C(C(CCSC)NC(C)=O)=O)C1 26379,C1(C(=O)NCCN(C(=O)CC(F)F)CC(C)O)(COC)CCCCC1 26380,CCCCC(CNC(=O)CC1(OC)CCCC1)NC(=O)C(C)=CC1CC1 26381,Cc1cccc(CC(C)N(C)C(c2c(C)nsc2N(C)C)=O)c1 26382,N1(C(CC(=C)C)=O)CCC(NC(c2ccnc(CC)c2)=O)C(CC)C1 26383,c1(N2CC3(C)C(C2)CS(=O)(=O)C3)nc(=NCC2CCCCO2)[nH]c2cccnc12 26384,c1(N2CCCC(CNC(C3(C=C)CCOCC3)=O)CC2)ncccc1[N+](=O)[O-] 26385,c1(C(N2C(C(C)C)(C(=O)NCC(C)C(C)(C)C)CCC2)=O)cccc2ccoc12 26386,C(=O)(C(C(=O)N1CCC(CN(C)C(c2cncn2C(C)C)=O)C1)OC)OC 26387,C1(CC=C)(NC(c2snnc2C(C)C)=O)CCCN(C(c2ccnc(F)c2)=O)C1 26388,c1(C(=O)NC2C(NC(c3c(C)cco3)=O)CCC2)c(Br)ccc2c1CCC2 26389,C1(NC(C(c2ccccn2)C)=O)CN(C(c2cccc(Cl)c2)=O)C2CCCCC12 26390,C(CCOC)(C(=O)NCCCCCN(C)C(C)C)OC(CCN(CCC)C)=O 26391,c1(C(=O)NC2C=CCN(C(C3CN(S(=O)(=O)C(F)F)C3)=O)C2)sc([N+](=O)[O-])cc1Cl 26392,Cn1nc(C2CC2)cc1C(=O)NC1(C)CN(C(=O)CN2CCC2)C1 26393,C(CN=c1cc(C)nc[nH]1)(C(=O)OC)NC(C1C(C)(CC)C1)=O.C1CC1 26394,C1(C(=O)NC(CNC(=O)CN2CC3CC3C2)C2CC2)CC2CCCC(C1)C2 26395,c1(C(=O)NCC(CNC(c2ncc(C)c(C)c2)=O)O)ccn2ccccc12 26396,C1(C(=O)NC2CC(NC(c3sc(CC)c(C)c3)=O)C(O)C2)CC2C(C1)C2(C)C 26397,S(=O)(=O)(c1ccc(NCc2cncs2)c(C#N)c1)N(C)Cc1ncc(Br)s1 26398,c1(C(=O)NC)nccc(-c2noc(C3(O)CCN(C)CC3)n2)c1F 26399,C(=O)(CCCC(=O)OC)N(C)CC1OCCN(C(C(C(C)C)SC)=O)C1 26400,c1(CC)nc(N2CC3CC(NC(=O)C(C)C)CC3C2)c(C)c(Cl)n1 26401,C#CC1CCCN(C(C2(CNC(=O)C=Cc3ccoc3)CCC2)=O)C1 26402,c1(OC)cc(F)ccc1C(N1CC(C)(C)CC1CNC(=O)CCCC1CC1C)=O 26403,c1(C(N2CCC(NC(CN3C(C)CC3)=O)CC2C)=O)cccc2[nH]ccc12 26404,Cc1ccnc2nc(C(=O)N(C3CCCN(C(c4cccnc4O)=O)C3)C)nn12 26405,Cc1ccc(C(=O)NCCCCC(CO)NC(=O)C=C2CCC2)cc1S(N)(=O)=O 26406,C(=O)(CC(C)C(C)(C)C)N1C(C(C)C)CN(C(=O)CCCc2ccsc2)CC1 26407,N1(C(CC(CC)C)=O)CCC(CNC(=O)C=Cc2ccc(Cl)s2)C12CC2 26408,N1(C(C(COC)OC)=O)CC(C(=O)N(CCCC(C)(F)F)C)CCC1C 26409,C(=O)(C#CC1(C)COC1)N1CC(CC(=O)NCc2cc(C)nn2C)OCC1 26410,c1(C(=O)NCC2CC(C(=O)NC(c3nncs3)C)C2)cccc(C#N)c1 26411,c1(C(N2CC(C(C)NC(C(COC)(C)O)=O)OCC2)=O)cncc2[nH]ccc12 26412,CC(C)CC(C)CC(=O)NCc1nccn1C.C12CCC(CC1)CC(=O)C(=O)N2 26413,C(=O)(CC(O)C(C)CC)NCCCCC1CN(C(C(C=C)(C)CC)=O)C1 26414,CCC(C)C(C(=O)N1CCC(n2cc(CCN3CCCC3)nn2)C(O)C1)N(C)C 26415,N1(C(Cc2c(C)nn(C(F)F)c2C)=O)CCN(C(C2CCC2C)=O)CC(C)(C)C1 26416,C1(N(C(=O)CO)CC)CCCN(C(C2C=CCCC2)=O)C1 26417,C1(NC(C2(c3ccc(C(=O)OC)cc3)CCC2)=O)CC2(COC(=O)N2)C1 26418,N1(CC#C)CCN(C(C2(CNC(c3csc(-c4cccs4)n3)=O)CC2)=O)CC1 26419,c1(C(N2C(CC(=O)NC3CC=C(C)CC3)CCC2)=O)ncn2ccccc12 26420,CP(C)(=O)CC(=O)N1CC2(NC(C3CCC3)=O)CC1C2.N1(C(=O)C2CC2)CCCC1 26421,C1(CNC(=O)C=C2CCCC2)CCCC1NC(=O)CCC1CC1(F)F 26422,c1(OC)cc(OC)c(C)cc1C.c1(OC)ccc2c(c1)NC(=O)C21CC1 26423,C1(N(C(=O)C(C)c2ccsc2)CC)CCN(C(=O)CC2CCCN(C)C2)CC1.C1(C)CC1 26424,CCC(C(=O)NC(C)(CNC(c1cc(C2CC(F)(F)C2)[nH]n1)=O)CO)C(C)C 26425,N1(C(C(=O)NCCCSC)c2cnsc2)CCC(C2CCCCC2)CC1 26426,c1(C(=O)NCC2(F)CC(NC(C(CC)(C)O)=O)C2)cccc(F)c1Cl 26427,C1(NC(=O)COC(=O)CO)CCN(CCNC(c2cocn2)=O)CC1 26428,c1(C(N(CCCNC(C(COCC)C)=O)CC)=O)cccc(S(C)(=O)=O)c1 26429,CC1CC(C)C1C(=O)NC1(CNC(=O)C(=O)NCC2CC2)CCCC1 26430,N1(CCC(=O)OCC)CCC(CC(C)C)C1.c1(C=O)cn(C)nc1C(C)C 26431,CC1CC(NC(C2CCC2)=O)CCN1C(c1cnn(C2CC2(F)F)c1)=O 26432,c1(CNC(c2ccsc2C(=O)NCc2cccc(F)n2)=O)cc(Cl)cc(Br)c1 26433,n1(C(C)CNC(c2cc(CCN)cc(Cl)c2)=O)cnc2c(N)ncnc12 26434,C1(CC(=O)NC)CC(C)(C)CCC1CN.C(=O)(CC(C)(C)C)C(C(C)OC(C)(C)C)=O 26435,c12cccc(c1)N2.CCC(CN(C(=O)C=CC(=O)N(C)C)C)NC(=O)C=CCF 26436,C1(C(=O)OC)CC(NC(=O)Nc2ccnc(-c3ccccc3)c2)C(OC)C1 26437,c1(OC)ncc(Cl)c(C(N2CC(N(C)C(c3ccccn3)=O)C(O)C2)=O)c1Cl 26438,c1(C(N(CC(c2ccc(OCC)cc2)C)CC)=O)ccc2c(c1)C(CN)CCC2 26439,C1(NC2(CC(=O)OC)CC2)CC(NC(=O)C(C)=CCO)C1 26440,C#CC1(CO)CCN(C(C2(C3CCCN3C(=O)CCOCCOC)CC2)=O)C1 26441,c1(OC)ccc(F)cc1CC(N1CC(C)C1CNC(c1cc(O)nn1C)=O)=O 26442,C1(C(=O)NCC(C)(C)C#N)CCCC(NC(=O)CC(C)(C)C)CC1 26443,c1(C(=O)NCC2CCCN(C(c3ccn(CCOC)n3)=O)C2)cccc(F)c1N 26444,C1(NC(C2(C#C)CC2)=O)C=CCC(C(=O)NC2CC(CC(N)=O)C2)C1 26445,C=CCC(CNC(C1(C2CC2)CC1)=O)NC(c1c[nH]nc1-c1ccc(Cl)s1)=O 26446,C1(CC(=O)NCc2cnc(OC)nc2C)CCn2cncc2C1 26447,C1(C(N(C(CNC(C2(O)CCOCC2)=O)C2CC2)C)=O)C2CCCCCC12 26448,CCCC(C#N)C(=O)NCC1(O)CCCN(C(c2c(C)cnn2C)=O)C1 26449,C(=O)(CCC(C)(C)C(=O)N(CCO)CCNC(C1CCCCC1F)=O)OC 26450,N1(C(C2CC(=C)C2)=O)CCN(C2CCC(NC(=O)Cc3ncccc3C)C2)CC1 26451,c1(NC(C(C(C)NC(=O)CC(C)(C)C2CC2)(C)C)=O)cc2ccccn2n1 26452,N1(CC(=O)NC(c2c(C)cc(C(N)=O)cc2)=O)CCc2ccc(Br)cc2C(C)C1 26453,c1(C(N(C2CN(C(C3C(CC)CCCC3)=O)C2)C)=O)cc2c(C)ccc(F)c2[nH]1 26454,C(c1ccccc1OC(F)F)=CC(=O)NC1CC1CNC(C1CC1SC1CC1)=O 26455,N1(C(C=CCC)=O)CC(CC(=O)NC2CC2c2nn[nH]n2)CC1(C)C 26456,N#Cc1c(Cl)ccc(CN=c2[nH]c(C(=O)NCc3cccc(Br)c3F)cs2)c1Cl 26457,C(CCCC(C)(C)NC(=O)C(C)Sc1ccccn1)NC(c1cc(C)c(C)s1)=O 26458,N1(Cc2cccc(C)c2)CCC(C)C(NC(c2cc(-c3cccs3)nn2C)=O)C1 26459,C1(NC(COCC=C)=O)CCCC(NC(c2cccc(CCN(C)C)c2)=O)C1 26460,CCC(C)(C#N)C(=O)NC(C)CN(C(=O)Cc1ccccc1C(N)=O)CC(C)C 26461,c1(NCc2c(F)cccc2I)ncc(CO)cc1Br.N12CC(CC(F)C1)C2=O 26462,c1(N(C(N2CC(=C(C)I)C2)=O)CC2CC2)cccc([N+](=O)[O-])c1 26463,N=c1nc[nH]n1CC(=O)NCC1(CC(N)=O)CC1.C12CCCC1NC2=O 26464,N1(C(C(C2CCC2)OC)=O)CC(CNC(=O)CC2(N(C)C)CCCCC2)C(C)C1 26465,N1(C(c2c(OC)cccc2O)=O)CCN(C(=O)CN2CCCC2=O)CCC1C 26466,CN1CCCC(CN(C)C(C2CCN(C(=O)Cc3cnoc3)CC2)=O)C1 26467,N1(C(c2c(OC)cccc2)=O)CC2CCC1C(CNC(=O)CCOCC(F)F)C2 26468,c1(NC(N2CCCC(N(CC(C)O)C)C2=O)=O)cccc([N+](=O)[O-])c1 26469,C1(OC)(CNC(=O)C(C2CCOCC2)C)CCN(C(=O)CC2CC(OC)C2)CC1 26470,S(=O)(=O)(CC(=O)NCC1(CNC(c2cc(CC3CC3)on2)=O)CC1(F)F)NC 26471,CCC(CCCC(=O)N1CC2(C1)CC2(F)F)NC(C1(O)CCSC1)=O 26472,c1(C)csc(C(=O)NNC(CNC(=O)NC(C)(C)C)=O)n1.C1(CSC)CC(O)C1 26473,c1(C(C=O)NCCC#N)cn(C)nc1Cl.C1(C2(CC(F)F)CC2)CCCC1 26474,C1(CNC(C(CCC=C)(C)C)=O)CCC2(CCC2)CN1C(=O)Cc1ccns1 26475,C(=O)(C#CC(C)(C)C)NCC1(NC(c2ccc(OC)s2)=O)CCCCC1 26476,CCS(=O)c1ccccc1C(N1CCN(C(c2csnc2C)=O)CC1CCO)=O 26477,C1(c2cn(C(C)C)nn2)C(C)CCN1C(c1ccc(C(SC(F)(F)F)=O)o1)=O 26478,C(c1ccccc1)=CC(C(=O)NC1CCN(C(C(=O)Nc2nc(=N)s[nH]2)=O)C1)=O 26479,c1(OC)ccc(S(=O)(=O)N2CCOCC2C2CCCCC2=O)cc1-c1cc[nH]n1 26480,CCCCCC(F)C(=O)N(CC(N1CCc2nn[nH]c2C1)=O)CCOC 26481,C1(NC(C2CCCC(C(=O)OC)C2)=O)CCCN(C(=O)C(C)n2ccnc2)CC1 26482,c1(CC(=O)NCC(C)(C)NC=O)ccc(C(F)(F)F)cc1 26483,N1(C(COCCCC)=O)CC2(C=C(C(=O)N3CC(F)CC3C(N)=O)CO2)C1 26484,C1(C(N(CC(COC)(C)C)C)=O)CCN(C(C2CC(F)CN2C)=O)CC1 26485,C1(O)(CCNC(CCOCCCNC(CC2C(C)(C)C2)=O)=O)CCOC1 26486,c1(OC)ccc(N)c(C(N2CCC(N(C(=O)CCc3ccc(F)cc3)C)C2)=O)c1 26487,C1(C)(C(=O)NCC2(C)CC(NC(=O)Cc3ccncc3Cl)C2)CC(C#N)C1 26488,N1(S(c2ccc(C(=O)OC)cc2)(=O)=O)CC(C)CN(C(=O)CS(C)(=O)=O)CC1C 26489,c1(C(N(C2CCN(C(c3ccc(OC)c(C)c3)=O)C2)C)=O)cc(C)c(N)cc1Cl 26490,c1(C(=O)NC(CN(C(C2(NC)CCCCC2)=O)CC)C)cc2cc(C)ccc2[nH]1 26491,C(=O)(CC1=CCOCC1)N1C(C(C)NC(C(C)(c2ccccc2)OC)=O)CCC1 26492,C(=O)(C(C)(CC)CCC)NC1(CCCC(N2CCC(C#C)CC2)=O)CCC1 26493,c1(-c2nc(C(CC)CC)nn2C2CCS(=O)(=O)C2)cc(F)cc2nccnc12 26494,C1(CNC(CCC)=O)CCC12CCN(C(=O)COc1ccc(Cl)cc1C)CC2 26495,C(=O)(C(CNS(C)(=O)=O)c1ccccc1)N(CCN(CC)CC)CC 26496,c1(NC(C2CC2C(=O)Nc2cc(Br)cnc2Br)=O)c(Cl)cnnc1Cl 26497,c1(NC(c2scc(-c3c(F)ncc(C)c3)n2)=O)cc(Br)c(F)cc1C 26498,N1(C(CCC(C)C)=O)CCN(C(c2cc3n(n2)CCNC3=O)=O)C2COCC12 26499,c1(C(N2CCC(C(C)(C)NC(c3c(CC)scc3)=O)C2)=O)n[nH]c2c1COC2 26500,N1(C(C=CC=CC)=O)CCC2(C1)CN(C(C1CCCSC1)=O)C2 26501,N1(C(C(CC)C)=O)CCC2CN(C(=O)C3=C(C)OCC3)CC2CC1 26502,C(=O)(C1=CC2C=CC(C1)C2)N1CC2CC(CNC(c3c(C)oc([N+](=O)[O-])c3)=O)C2C1 26503,C(=O)(C(F)(F)C(C)(C)O)N1CCC(CN(C(=O)C(=Cc2c[nH]cn2)F)C)C1 26504,C1(F)(CNC(C2C=CC=CC=C2)=O)COCCN(C(=O)CC23CCC(CC2)C3)C1 26505,C#CCC(C)(CC)C(=O)NCCN(C(c1cnc(C2CCC2)o1)=O)C(C)C 26506,C#Cc1ccc(C(=O)NC(Cn2cncn2)C(=O)NCC2C=CCC2)cc1 26507,Cc1c(O)ccc(C(=O)NC2(C3CN(C(=O)CC(C)C(C)C)C3)CC2)c1C 26508,c1(C(=O)NCC23N(C(C4C(C)(C)CCC4)=O)C(CC2)CC3)ccsc1S(C)(=O)=O 26509,c1(C(N2CC(CC(C)NC(C3CCC(F)C3)=O)C2)=O)ccnn1CCN(C)C 26510,c1(C(=O)NC2C=CCC2)cccc2nc(O)ccc12 26511,CC1(C)CCN(C(c2cncnc2)=O)CC1NC(c1cc(-c2ccoc2)[nH]n1)=O 26512,c1(C(N2CCC(N(C(=O)CCCCC(C)(C)C)C)C2)=O)cc2ccncc2cc1F 26513,c1(-c2scc(OCC)c2)nc(CSc2cccc(F)c2)nn1-c1ncnn1C 26514,c1(C(=O)NC2C(CNC(C(n3ncc(C)c3)C)=O)CC2)cncnc1C(C)(C)C 26515,C1(CNC(c2cnn(C(F)F)c2)=O)CCCC(NC(c2snc(Cl)c2Cl)=O)C1 26516,N1(C(C)=O)CC(C)(C)C1Cn1cc(CCCc2ccccc2C)nn1 26517,C1(C(=O)OCC)CN(C(=O)C(=O)NC(c2nc[nH]n2)CC)CCC1(C)C 26518,c1(OC)cc(C(=O)N(CCNC(=O)CC2(O)CCCC2)C2CC2)cc(Br)c1 26519,C12(NC(CCS(C)=O)=O)CCC(CNC(c3cc(F)ccc3Cl)=O)(C1)OC2 26520,C(C(=O)Nn1nnc2c1CCCC2)(C(C)O)NC(CC(C(C(C)C)=O)C)=O 26521,C(=O)(CCC(C(C)C)NC(c1ocnc1C(C)C)=O)N(CC(C1CC1)OC)C 26522,C1(NC(CCC)=O)CCN(C(=O)CCN(C(C2CCOC2C2CC2)=O)CC)C1 26523,N1(C(c2n(CC)ncc2)=O)C2CCC1C(NC(=O)Cc1nn(C)cc1Br)C2 26524,N1(C(c2c(C)n(C)nc2)=O)CCC2(CCCN2C(=O)CCCn2cccc2)C1 26525,CC(C)CC(C(=O)NC(CC1CCC1)C(=O)N1CC(C(N)=O)C1)NC(=O)CO 26526,C1(C)(CC)CC(C(N2CCC(OCCNC(c3sc(C)c(C)c3C)=O)C2)=O)CCO1 26527,c1(NC(C(=O)NCC(=O)NC(C(=O)OC)C(C)C)=O)ccc2nc(C)cc(Br)c2c1 26528,S(=O)(=O)(c1ccc(Br)cc1NCc1cccc(Cl)c1)NCC1OCC(C)C1 26529,N1(C(CCC(=O)OCC)=O)CC(NC(=O)CC2CC=CCN2C)CC(F)C1 26530,c1(C(=O)NC23CC(CNC(C(C)=C(CC)C)=O)(C2)C3)cn(C)cc1C(F)(F)F 26531,C12(C(=O)NCCCC(C)NC(c3c(C)n[nH]c3C)=O)CCC(CC1)C(C)O2 26532,N1(C(Cn2ccc(C)n2)=O)CC(NC(c2ccc(-c3ccco3)s2)=O)C2(CC2)C1 26533,c1(C(N(CC(CC)NC(=O)C(O)CC2CCCC2)C)=O)cc(F)n(C)n1 26534,N1(C(C(CCC)N(C)C)=O)CC2CC(C(=O)N(C(C)C(C)(C)C)C)C(C2)C1 26535,C(C1=CCN(C(=O)C(F)(F)Cc2ccccc2)CC1)NC(Cc1nnc(C)s1)=O 26536,N1(C(C(C2(O)CN(C(C(C(C)C)SC)=O)C2)F)=O)CC2CN(C)CC2C1 26537,c1(C(N(CC(O)CNC(=O)CN2CCNC(=O)C2)C)=O)cc2nc[nH]c2cc1F 26538,N1(C(=O)O)C2CCC1CC(Cc1cn(CC3C(CCOc4ccccc4O)C3)nn1)C2 26539,C(=O)(C(C)(CC)C(=O)OC)NC(CNC(c1c(CC)n(C)nc1)=O)CO 26540,c1(C(=O)NCC(CNC(Cc2n(C)ccn2)=O)F)cnn(C)c1S(C)(=O)=O 26541,CCC(CC(C)C)C(=O)N1CC(C(=O)NCc2ccccn2)C2(CC2)C1 26542,Cc1ccc(Br)c(CCC(=O)NCC23CC2CN(C(c2csc(O)n2)=O)C3)c1 26543,C1(CNC(c2c(C)nco2)=O)CN(C(C2CC2c2sccc2C)=O)CC12CCC2 26544,c1(NC(C(=O)NCCCCSC)=O)ccc(Br)cc1SC 26545,C1(C2(O)CN(C(=O)CC3CNC(=O)O3)C2)(CNC(=O)CCc2cnco2)CC1 26546,CN1CCCC(C)(CNC(=O)C(N2CC(CO)C(C(F)(F)F)C2)=O)C1 26547,C1(OC)CC(C(=O)OC)N(C(=O)NC(C)C(C)NC(C)=O)C1 26548,c1(CC)[nH]c(C(=O)NCC(C)(CO)NC(c2cc(C)nn2C)=O)nc1Cl 26549,c1(NC(C2(F)CN(C(CCOCC)=O)C2)=O)ccccc1N(C)C 26550,C1(CNC(C(=O)NC2C(c3n(C)nnc3)C2)=O)CCC(C)(C)CO1 26551,c1(OCC=C)cccnc1C(=O)NC1CCC(N(C)C(c2csc(Cl)c2C)=O)C1 26552,c1(CC)noc2ncc(C(=O)NC3CC4CC(C3)N(CC(C)OC)C4)cc12 26553,Cc1cnc2n1CC(C(N1CC(N(C)C(C3SCCCS3)=O)C3(CC3)C1)=O)CC2 26554,N1(C(=O)CC2(O)CCOC2)Cc2n[nH]cc2C1C(=O)N1CC2CCCC2C1 26555,c1(C(N2C(C(C)NC(C3CC3CF)=O)CCC2)=O)c[nH]c(=S)cn1 26556,c1(OC)ccc(C=NOCC(=O)N(CC(C)NC(=O)Cc2cc(C)cs2)C)cc1 26557,c1(OC)cc(C)c(C(N2CCCC(NC(C3(C4CC4)CCCO3)=O)C2)=O)cn1 26558,N1(CCOC(=O)CSCCSCC=C)CCCCC1=O 26559,c1(C2C(N(C)C(=O)OC(C)(C)C)C2)ccc(F)cc1.C1(=O)C(C2CCC2)CO1 26560,C1(C(=O)NCCc2cncc(C)n2)CCN(C(C2CCCN2C=O)=O)CC1(C)C 26561,Cc1nn(C)cc1CC(=O)NC(CNC(=O)C(C)Sc1ccc(Cl)cc1)C1CC1 26562,CC(C(=O)C12CC(C1)CN(C)CCOCCCN(C)C2=O)C1CCC1 26563,c1c(I)ccnc1F.c1(C(CN(C(C)C)C=O)(C)O)cccc(Br)c1 26564,N1(C(c2cccc(C(=O)Nc3cnn(C)c3C(F)F)c2)=O)CC2(CNC(=O)C2)C1 26565,C1(CC(=O)NCC(C(C)C)NC(=O)C=CC(N)=O)CC(C)OC(C)C1 26566,N1(C(c2c(F)ccc(C)c2)=O)C2CCC1CC(F)(CNC(C1CC3CC3C1)=O)C2 26567,C1(C(=O)NC(CN(C(c2c(C)scn2)=O)C)(C)C)CCCC(F)C1 26568,N1(C(CCc2ccn(C)n2)=O)CCC(O)(Cc2nc(-c3ccncc3)cs2)C1 26569,C(=O)(C(O)CC(C)(C)C)NC1(C)CCN(c2snc(CCOC)n2)C1 26570,C1(NC(COCC#C)=O)CCN(C(=O)CCOCC2(CF)CC2)CC1CC 26571,N1(C(C2CCC(CC)C2)=O)CC2(C1)CN(C(=O)Cc1ccc(Cl)c(F)c1)CCO2 26572,c1(C(=O)NC23CCCC(NC(C=CC=CCC)=O)(C2)C3)ccc(Cl)c(F)c1N 26573,c1(N2CCCC(CN(C(C3(OC)CCCOC3)=O)C)C2)cccc(F)c1[N+](=O)[O-] 26574,C1(C(=O)NCCNC(C23COCC2C3)=O)(CN2CC([SH](C)C)C2)CC12CCC2.C(=O)N 26575,c1(C(=O)OC)cc(C(=O)NCC2(CN(C)C(c3ccn(C)n3)=O)CC2)nn1C 26576,N1(C(c2nccc(C)c2)=O)C2CCC(C2)C1CNC(=O)COc1ccccc1F 26577,c1(C(=O)NCCN(C(=O)Cc2cc(Cl)ccc2F)C)cncc([N+](=O)[O-])c1 26578,N1(CC(N2C(C(N3CCC(CO)C3)=O)C=CC2)=O)C(=O)CCC1=O 26579,C(=O)(C1OCCc2ccccc21)N(CCNC(CC(C)OC)=O)C(C)C 26580,C=Cc1ccc(C(=O)NCC2CN(C(=O)C(C)(C)C#N)C2)cc1 26581,C1(NC(C(COC)O)=O)CN(C(C2CC(S(C)(=O)=O)C2)=O)CC12CCC2 26582,Cc1cc(C(N2CC(OCCNC(=O)C=CCF)C2)=O)c(C)cn1 26583,C1(C(=O)NCCSC(C)C)CN(C(=O)CCCSc2ccccc2)CCO1 26584,C#CCC(CC(=O)N1CCCC1C(C)CC)NC(c1cc(O)ccc1F)=O 26585,N1(C(CCCC(C)C)=O)CC2(CCN(C(=O)C(c3ccccn3)C)C2)C1 26586,c1(C(N2CCC=C(Br)C2)C(=O)NCCCOC2CC2)ccc(F)cc1Cl 26587,C12(NC(c3c(C)nsc3)=O)CCN(C(c3cnc(N)cn3)=O)CCC1C2 26588,C1(CCN(C(COCc2onc(C)n2)=O)C)CCCCN1C(C1CC1F)=O 26589,CCC(C(=O)N(C)CC1CCN(C(=O)Cn2cc(S(C)(=O)=O)cn2)C1)C(C)(F)F 26590,CC1CC2(CC2)CN1C(C1OCCC1CNC(=O)Cc1cccnc1O)=O 26591,S(=O)(=O)(c1ccc(C(=O)NC(C)(CNC(=O)C=CBr)C2CCC2)o1)NC 26592,N1(C(C(CCC)OC)=O)CCC2(CC1)CC(NC(=O)CC(C)CC)C2 26593,C1(C(N(CC(C)C(=O)NC2CCOC2)C)=O)CCC(O)CN1C 26594,C=CCCCC(C(=O)NC1CN(C(=O)OC)C1)NC(=O)C(C)CC(=C)C 26595,CC(C)(C)CC(O)C(=O)OCCc1cccc(O)n1 26596,c1(C(C)NC(=O)NNC(=O)c2nccn2C)nc2ccccc2o1 26597,N1(C(c2c(CC)ccs2)=O)CCOCC1CNC(=O)C(C)Oc1ccc(F)cc1 26598,c1(C(N2CC3N(C(CCCCSC)=O)C(CC3)C2)=O)n[nH]c2c1CC(F)(F)CC2 26599,C(CN=c1cc[nH]cc1S(=O)(=O)N1CCCS(=O)(=O)CC1)C1C(C)NC(=O)O1 26600,C(CC(=O)NC1CC(NC(=O)CCn2cnnn2)C1)=CC 26601,c1(C(=O)NC(C)CCNC(C2COCCN2C)=O)cccc2nc(O)[nH]c12 26602,c1(C(N(CC(C)NC(C2CCC2(C)C)=O)C)=O)cc(O)no1 26603,c1(C(C(=O)NCc2n(CCCC)cnc2)N(C)C)ccc(OC)cc1 26604,C1(OC)CN(C(=O)CCn2cnnn2)CC1NC(=O)CCNC(=O)OC 26605,N1(C(C2C(C)(CC)C2)=O)CC2CC3CC2C1C3NC(c1ccccc1OC)=O 26606,C1(NC(C2C(C)=CCS2)=O)CCN(C(=O)CCc2ncnn2C)CC1O 26607,c1(-c2cnc(CC)s2)nc(-c2cccc(C)c2)nn1C1CCCCC1C 26608,C(C(F)(F)C(=O)NCCCCC1(C)NC(=O)NC1)OC 26609,C1(NC(C2C(NC(C3(OC)CCOC3)=O)CC2)=O)CCCCC1(F)F 26610,C(CC(C)(C)CC(=O)NCCOC1CCN(C(c2cc(N)ccc2Cl)=O)C1)OC 26611,Cc1cccc(C(N2CC(NC(=O)CN3CCOCC3)C3CC23)=O)n1 26612,C=Cc1cc(C(=O)NCC(CNC(c2cc(C#N)on2)=O)C(F)(F)F)cc(F)c1 26613,Cc1cn2ccc(C(=O)NCCC3CC(NC(C4CCCC4C)=O)C3)cc2n1 26614,c1(C(=O)NC(C)(C)CCNC(c2ccccc2Cl)=O)c[nH]c2ccc(O)cc12 26615,Cn1cnc2c(N3CCSC(NC(N4CCC5(CCCC5)CC4)=O)C3)ncnc12 26616,CCC(CCOC)C(=O)N1CCN(C(=O)C(=O)C(C)(C)C)CC1c1ccnn1C 26617,C1(COC)(CNC(=O)CC(F)(F)Cl)CCCN1c1nccc(CC(=O)OCC)n1 26618,N1(CC)CCN(C(C2CC(NC(C3CCC3(OC)OC)=O)C2(C)C)=O)C(C)C1 26619,CC1(C)CN(C(C2CCCCS2(=O)=O)=O)CCC1NC(c1cc(F)cnc1Cl)=O 26620,c1(C(=O)NCCC(=C)CNC(=O)CCCN=[N+]=[N-])ccc(S(=O)(=O)C(C)C)cc1 26621,N1(C(CC=C=C)=O)CCC(C2CCN(C(c3cc(C#N)c[nH]3)=O)CC2)C1 26622,Cn1cc(C(=O)NCC2CC(NC(=O)CCc3cccnc3)C2)c(C2CCC2)n1 26623,C(=O)(C1=CCCCCC1)N(CCC1N(C(C(CC(=C)C)C)=O)CCCC1)C 26624,c1(COC)ccc(C(N2CCC(C)(NC(c3cc(C)ccc3O)=O)C2)=O)cc1F 26625,C1(NC(C(CC=C)C)=O)CN(C(c2cccc(F)c2NC)=O)Cc2ccnn2C1 26626,N1(C(c2cc(COC)sc2)=O)CCCCC1C(C)NC(c1ccc(C)n1C)=O 26627,N1(C(CCNC(=O)NC)=O)C2CCC1CC(C(=O)Nc1cccc(N=[N+]=[N-])c1)C2 26628,C1(NC(CC(CN(C)C)O)=O)CCN(C(c2cc(F)ccc2Cl)=O)C12CC2 26629,C(=O)(C1=CCCCC1)NC(CNC(c1c(OC)csc1)=O)C(C)C 26630,C=CCC(C)C(=O)N1CCOC(CNC(=O)CCc2nncs2)C1 26631,c1(C(C(=O)NCC(C)CNC(c2ccco2)=O)O)ccc(Cl)c(Br)c1 26632,c1(C(N(C(CN(C(c2ncn(C(C)C)c2)=O)C)C)C)=O)cccc2c1CCOC2 26633,c1(C(=O)OC)cc(Cl)ccc1S(=O)(=O)Nc1ccc(-c2csnn2)cc1 26634,C(C(C)(C)CC(=O)NCC(=O)NC1CC1)NC(c1cc(C)[nH]c1C)=O 26635,C1(CNC(C2CC2C(F)(F)F)=O)CC2(CC2)CN1C(=O)C(F)(F)c1cscn1 26636,N1(CC=CC)C(=O)CCC1CC(=O)NC1COCC1CNC(=O)CS(C)(=O)=O 26637,C(=O)(CCCC(=O)N(C)C)N1CC(C(C(=O)NC2CN(CC)CC2C)OC)C1 26638,N1(C(c2cccc3sccc23)=O)Cc2ccc(Br)cc2CC12CCC2 26639,c1(C(=O)NC2(CNC(c3ccc(OC)cc3)=O)COC2)cc2c(nn1)OCCS2 26640,c1(C(N2CC(NC(C3C(C)(C)CC3)=O)CC3(C2)CC3)=O)[nH]c2ccccc2c1Cl 26641,CC(C(C)Cc1ccccc1)NCc1cnn(C)c1 26642,c1(CC(C(N2CCC(CNC(C3CC(C(F)(F)F)C3)=O)C2)=O)O)cc(Cl)cc(Cl)c1 26643,C(=O)(C1=CCCCC1C)N1CC2C(C(N(C(C(C)C)=O)C3CC3)=O)C2C1 26644,c1(C(N(CCNC(=O)Cc2sc(O)nc2O)CC)=O)c[nH]c(C)c(Br)c1=O 26645,C1(NC(CCNC(=O)CO)=O)CCC2(CC1)CCN(C(C1CCC1)=O)C2 26646,Cc1snnc1C(=O)NCC(C1CC1)NC(=O)C=CCOC(C)(C)C 26647,N1(C(c2cn(C)nc2)=O)C2CCC1CN(C(=O)CCSCC(N)=O)C2 26648,c1(CC(=O)N(CCC(=O)N(C(C=C)C2CC2)C)C)cc(C)on1 26649,c1(CNC(CC)=O)ccc(CC(C)NC(=O)CC=CC(C)(C)C)cc1 26650,c1(C(=O)NC2CN(C(Cn3nnc(C)n3)=O)C(C)CC2)cnn2ccc(O)nc12 26651,N1(C(C(COC)N(C)C)=O)CC(CNC(=O)Cc2c(C)n[nH]c2C)C(C)C1 26652,c1(CCNC(C2N(C(CCN(C)C)=O)CCSC2)=O)c(Cl)cc(Br)cc1Cl 26653,c1(CC(=O)NCCCN(C(=O)CNS(C)(=O)=O)C(C)C)nccc2ccccc12 26654,C1(NC(C2CCC(O)CN2C(=O)CN2C(=O)CNC2=O)=O)CCOC12CCCC2 26655,c1(C(n2cc(COCC(N3C(CC(=O)O)CC3)=O)nn2)C2CCCC2)ccccc1 26656,C(CC(=C)C)(C1CC1)NC(CCOCCN(C(CC=CC=C)=O)C)=O 26657,CON(CCC(=O)NCC1(CC)CCC1)C(=O)c1c[nH][nH]c1=N 26658,n12cc(nn1)CCNC(=O)C2C.C(=O)(CCn1ccnc1)N(C(C)C)C1CC1 26659,N1(C(CSCCC(C)C)=O)CCCCCCC1C(=O)N(C)CC1CC1C 26660,c1(OC)cc(Br)c(NC(=O)NCC(C)(C)C(N)=O)cc1C 26661,C(=O)(C(C(C)(C)C)N1CCNC1=O)N1C(C)C(NC(c2cc(N)ccn2)=O)CC1 26662,n1(CC)nnc2c1CCC(C(=O)Nc1nccnc1C#N)C2 26663,c1(C(c2nnnn2C2CCCC2)NCCC(=O)NC(C)C)cc(Cl)cc(Cl)c1Br 26664,O=S1(=O)CCC2(CCN(S(=O)(=O)c3ccc(N4CCOCCC4)c(Cl)c3)CC2)C1 26665,Cn1nc(O)cc1NC(C1CC1NCc1csc(Br)c1)=O 26666,CC1CN(C(c2cccc(C#N)c2)=O)C(C)CN1C(c1ccnc(C(F)F)n1)=O 26667,c1(CC(=O)NC2C(NC(C(C)CC(C)(F)F)=O)CC2)cc(F)cc2c1OCOC2 26668,C(=O)(CC(C)CF)N(CC(C)CNC(c1c[nH]nc1-c1cnn(C)c1)=O)C 26669,N1(C(C2(COC)CN(C(c3c[nH]c4cccnc34)=O)C2)=O)CC2(C1)OC(=O)NC2C 26670,C=CCC(C)(C)CNC(C12CC(CNC(c3cnccc3CC)=O)(C1)C2)=O 26671,CN=C(NCC1(O)CCOCC1)N1CCN(CC(F)(F)F)C(=O)C1 26672,CCCCC(C(=O)N(CCCCCCNC(=O)C(F)=C1CCC1)C)N(C)C 26673,C1(C(=O)NCC(=O)OCC=C)CC12CC(NC(c1ccoc1)=O)C2 26674,N1(C(Cc2c(C)scc2)=O)CC2COCC2(C(=O)NCC(C)CN(C)C)C1 26675,Cc1cc(C(=O)NCCC(=O)N2CCC2C(CCCO)=O)nc(O)c1 26676,c1(C(=O)NC(c2ccccc2)CNC(C(CCSC)O)=O)cccc2c1OCC2 26677,Cc1nc(O)nc(C)c1C(=O)NC1CCCCC1CNC(c1ccc(N)c(Cl)n1)=O 26678,CC1CN(C(=O)COCc2ccnc(O)c2)CCC1N(C(=O)CCC(C)(F)F)C 26679,C(=O)(CCC(=O)NCC1OCCC1C(=O)NC1(C)CC1(C)C)NCCC 26680,CC1CN(C(=O)Cc2cccc(F)c2)CCC1NC(=O)Cc1nnn(C(C)(C)C)n1 26681,C1(F)(C(=O)NC(C(C)C)CNC(c2csc(-c3cnccn3)n2)=O)C2CCCC12 26682,N1(C(C2C(C)C2C)=O)C2CCCC1CN(C(C1CC1c1ccccc1)=O)C2 26683,c1(CC)cc(C(N2CCOCC2)C(=O)NCc2ccc(C)cc2)cc(N=[N+]=[N-])c1 26684,N1(C(C(C)=CC)=O)CCCC(NC(C2CC(=O)N(c3ccccc3SC)C2)=O)C1 26685,N1(C(=O)Nc2ccc3nncn3c2)CCOCC2(CCC2)C1 26686,C=C(Cl)CCC(=O)NC1CCN(C(c2cncc(N(C)C)n2)=O)C1 26687,N1(C(c2c(CC)ccc(C)c2)=O)CC2CCC1C(CNC(=O)C(SC)SC)C2 26688,N1(C(C(C(CC)O)C)=O)CCC2(CC1)CC(NC(c1cc(Br)c(O)cc1F)=O)C2 26689,c1(C(N(CC(CN(C(C(=O)N(C)C)=O)C)O)C)=O)ccnc2c1CCO2 26690,C(=O)(C(CC(C)C)C(C)C)NC(C1CCN(c2nc(COC)nc(C)c2)CC1)C 26691,c1(C(=O)NCC2(O)CN(C(=O)CCc3cn[nH]c3)C2)csc2cccc(F)c12 26692,c1(C(=O)NCC2(C(C)(C)C)CN(C(=O)CC3CCCC3(F)F)C2)cccc(=O)n1C 26693,c1(C(N2C(CNC(CC(C(=C)C)O)=O)CCCC2)=O)cn2nc(OC)ccc2n1 26694,CC1CC(C(=O)NCC2CCN(C(=O)COc3ccn(C)n3)CC2O)=NO1 26695,N1(C(c2c(C)nc(CO)o2)=O)CCC2C(C1)CN2C(=O)Cn1nnc(C2CC2)n1 26696,C1(CC)CC(C(=O)N(CC(C)(C)NC(c2ccc(C3CC3)cc2)=O)C)CC(=O)N1 26697,C(CC1=CCOCC1)NC(C1CC(=O)CN1C(C1C2CCC(F)C12)=O)=O 26698,c1(C(N2CCCC(NC(C(CC)NC(C)=O)=O)C2)=O)cc2cccnc2[nH]1 26699,CCC1=NOC(CC(=O)NCC2C=CCN2C(c2csc(C)c2)=O)C1 26700,Cc1ncc(C(=O)NC(C2CCCC2)CNC(=O)C(F)Cc2ccccc2)[nH]1 26701,N1(C(COCCC)=O)C(CNC(=O)CC2(COC)CC2)CC2CCCCC12 26702,c1(NC(C(C)N(C(C=CCOC(CC)(C)C)=O)CCO)=O)cccc(F)c1 26703,c1(CC(=O)NCCCC(C)NC(C2OCCCO2)=O)c(Cl)cccc1Br 26704,O=C(CN=c1cc[nH]cc1)NCCCNC(c1ccc(O)nn1)=O 26705,N1(C(c2nc(OCC)oc2)=O)CCN(C(=O)Cc2ccsn2)CC1C(F)F 26706,S(=O)(=O)(c1cc(C(=O)O)c(C)o1)N1CCCC(C(CC)NC(=O)C(C)(C)C(N)=O)C1 26707,c1(NC(C2(F)CCN(C(C(c3cccc(C)c3)=O)=O)C2)=O)cc(Br)c(Cl)cc1F 26708,C1(CC(=O)NC2(CCNC(C=CC(=O)OCC)=O)CCC2)CCOC1(C)C 26709,c1(C(N2CC3CCN(C(CCOC)=O)C3CC2)=O)oc2ccccc2c1C.C(C1CC1)N 26710,CCC(C)(COC)C(=O)N1CCOC(C(=O)NCCCCO)C1 26711,c1(C(=O)NCC2C(NC(c3ccc(-c4ccccc4)[nH]3)=O)C2)ccccc1F 26712,N1(C(CCC(C#C)(C)C)=O)CCC2CCN(C(=O)CSc3nncs3)CC2C1 26713,C=CC(C)(O)CC(=O)N1CC(OC)CC1CNC(c1cc(Br)cn1C)=O 26714,C(=O)(C1=C(C#N)CCC1)N1CCC(C(N2CCC(CN(C)C)C2)=O)(CO)CC1 26715,c1(C(C)(C(=O)NC2CN(C(c3cncc(Cl)c3)=O)C2)N(C)C)ccc(F)c(F)c1 26716,c1(C(N(C)CCNC(=O)CSCC(F)(F)F)=O)cccc2c1COC2 26717,C1(C(=O)NCCn2cc(C(N(CC(CC)O)CC)=O)nn2)CCSC(C)C1 26718,C(c1cccnc1)=C(C)C(=O)N(C1CN(C(=O)C=CC2CCC2)CC1F)C 26719,C(CCC(C)(F)F)N(C(=O)CN(C(=O)CC1CC2CC2C1)C1CCC1)C 26720,C12(CNC(=O)CCn3ccnn3)CC1CN(C(c1nccnc1C(F)(F)F)=O)C2 26721,C(CN=c1[nH]c2c(c(=NCc3noc4c3COCC4)[nH]1)SCC2)OC 26722,O=C(Nn1ccnn1)C1(c2ccccc2)CC1 26723,C(=O)(C(CC(C)C)CC(C)C)N1C2(CNC(C(CC=C)(C)C)=O)CCC1CC2 26724,C=CCC(CNC(=O)COC(C)(C)CNC(C1(c2ccno2)CC1)=O)CC(C)C 26725,C(CC1=CCN(c2nc(C3CC3)nc(=N)[nH]2)CC1)NC(C(C)CC1CCCC1)=O 26726,Cc1ccc(C(=O)CCC(=O)N(C)CC2CN(C(c3cnccn3)=O)C2)cc1 26727,Cc1oc([N+](=O)[O-])cc1C(=O)NCCC(C)N(C)C(c1cnn(C)c1N)=O 26728,Cc1cc(C(=O)NCC2CN(C(c3ccc(F)cc3)=O)CCC2C)cc(C)c1O 26729,C#CCCCC(=O)N1CCN(CC2CN(C(c3ocnc3C)=O)C2)CC1 26730,C(=O)(C(F)(F)C(O)C(C)C)NC1(OC)CCN(C(C2(COC)CC=CCC2)=O)C1 26731,C1(CNC(C(C)Sc2ccccn2)=O)COCCN(C(c2ccn(C)n2)=O)C1 26732,N1(C(=O)Nc2ccc(CCCC)cc2)CC(C(=O)O)OCC1C 26733,N1(C(c2c(C)ccnc2)=O)CCC(NC(=O)C(F)(F)c2cscn2)C(O)C1 26734,c1(C(c2cc(C)ccc2I)NCC(CCNC(C)=O)F)c(C)cccc1C 26735,C1(C)(C(N(C2CCC(NC(=O)CC(C3CC3)C3CC3)C2)C)=O)COC(=O)OC1 26736,CCC(C)C(C)C(=O)NCC(=O)NC(C1CN(C(=O)C(C#N)CC)C1)CSC 26737,C(C1=NOC2CN(C(c3cc(O)cc(=O)o3)=O)CC12)NC(=O)C1=CCS(=O)(=O)C1 26738,CON(CCC(=O)OC(C(C)(C)C)=O)C(=O)C1CNCC(C)(C)O1 26739,C(N=c1ccn(CCOC)[nH]1)(c1n(CC=C)nnn1)C1CC1.c1nnnn1CCCF 26740,CCC(C)C(C(=O)NCC=CCNC(=O)C(c1ccc(C(F)(F)F)cc1)(C)C)OC 26741,N1(C(COC(C)C)=O)CC2(C1)C(NC(=O)CC1CCSCC1)CCS2(=O)=O 26742,Cc1cccc(C(C)C)c1C(N1CCC(C(C)NC(C2C=CCC2)=O)C1)=O 26743,CCC(C(=O)NC(CC1CCCC1)C(=O)NCCC(C)COC)C(C)C 26744,CCC(C)(C#N)C(=O)NCCCOCCN(C(=O)CC1CCCC(CF)C1)C 26745,C1(C(=O)NCC(c2ccccc2)NC(=O)Cc2ccoc2)CCCCO1 26746,N1(C(CC=C)=O)CCN(C(c2cnc(CC)s2)=O)C(CC2CC2)C1 26747,Cc1cc2cc(C(N3CC(CNC(c4cnc(Cl)[nH]4)=O)C(C)C3)=O)c(Cl)cc2[nH]1 26748,C1(C(N2C(C)CN(C(CCN(CC)CC)=O)C(C)C2)=O)(OC)CC2CCC1CC2 26749,N1(CCC)CC(C(N2CCCC(c3nnc(C(=O)OC)s3)C2)=O)CC1=O 26750,O=Cc1ccc(-c2cn(CCNc3ccn(Cc4ccccc4)n3)nn2)cc1 26751,C1(N(C)C(C2(O)COC2)=O)CC(C(=O)OC(C)(C)C)C1.C12CCC1N(C)C2=O 26752,C1(NC(c2sc(C)c(Br)c2)=O)CN(C(c2ncccn2)=O)CCC1F 26753,N1(C(c2cc(OC)no2)=O)CCCCC(CNC(c2cc(OC)cc(C)n2)=O)C1 26754,C(C(CC(C)C)NC(=O)C(C)Oc1ccccc1OC)NC(C(F)OC)=O 26755,C1(C(N2CCN(CC)CC2)=O)CNC(=O)CN1C(c1ccc[n+]([O-])c1)=O 26756,C1(n2cc(CN3CCCC(CCCN(C)C)C3)nn2)CC2CCC1N2C 26757,c1(CC#N)ccc(Cl)c(OCCCC2CCC23CCC3)c1 26758,N1(C(C(C)CC2CCC2)=O)CC2(CCCN(C(=O)C=CC3(C)CCOCC3)C2)C1 26759,c1(OCC(=O)C(=O)NC(c2nc(C)no2)CC)ccc(F)nc1.C(CN(CCO)CC)N 26760,c1(OC)ccc(CC(=O)NC2(C)CN(C(C3(Br)CC3(C)C)=O)C2)cc1F 26761,C(=O)(CC(C)(C)C(F)F)NCCOC1CCN(C(CC(C)(C)C)=O)C1 26762,C#Cc1ccc(C(=O)NC(CNC(c2cccn2C)=O)CC)o1 26763,c1(C(N2CCC(CN(C(c3nc(CC)oc3C)=O)C)CC2)=O)cc(C)nc(O)n1 26764,C1(CNC(CC(c2c(C)noc2C)C)=O)CC2CCC1N2C(=O)CC(C)(C)C 26765,N1(C(C(C=C)O)=O)CCC(CCCCNC(=O)C(n2ccc(C)n2)C)CC1 26766,S(=O)(=O)(c1cc(C(=O)NC2CC3(C2)CN(C(C24CC(C)(C2)C4)=O)C3)co1)NC 26767,Cc1cc(C(N2CCC(C)(NC(=O)CC3CCC(C)(C)O3)C2)=O)ccc1Cl 26768,c1(C(N(CCNC(C2CC3CC(O)C(C2)C3)=O)CC)=O)cc2cc(Cl)cnc2o1 26769,CCC(C)(COC)C(=O)N1CCCC(CNC(c2nocc2C)=O)CC1 26770,C(C(=O)NOCC(N1CCC(C(C)(C)C)C1)=O)=C(C)C 26771,C12(C)CC(NC(c3[nH]nnc3C)=O)CN1C2=O.C1(COC)CN(C2CCC2)C1 26772,c1(NC(c2c(C)cccn2)C)nc(N(C)CC2CCC(=O)N2)c2ccsc2n1 26773,N1(Cc2cccc(OC)c2F)CC(C(=O)Nc2cnc(Cl)c(C#N)c2)CC(F)(F)C1 26774,N1(c2c3ncn(CC4CCC(C)C4)c3ncn2)CC=C(c2ccc(Br)cc2)CC1 26775,CC1CN(C(=O)CCNc2ccc(OC(F)F)c(OC(F)F)c2)CC(C)O1 26776,C1(CC)(NC(c2cc(N(C)C)ccc2F)=O)CCCN(C(C2(C)CCCS2)=O)C1 26777,c1(CC)ncccc1C(=O)N(C(C)CNC(=O)CC1CCC(C)CO1)C 26778,c1(OCOC)cc2c(cc1NC(c1nccn1-c1ccc(C)c(F)c1)=O)OCO2 26779,c1(CC)cccc(OCC)c1.c1(C(C(=O)N)C)ccccc1.C1C(=O)NCCN1CC 26780,Cc1cc(F)ccc1C(F)(F)C(=O)NCC1(C(F)F)CCN(C(=O)CC(C)C)C1 26781,CC1CCN(C(=O)C(C)Cn2cccn2)CC1.C(=O)(CS(=O)(=O)N)N1CC(CN)C1 26782,N1(C(CCC#C)=O)CCCCC2C1CCCN2C(=O)Cc1n[nH]c2c1CCCC2 26783,C1(NC(CC2C(C)=NN(C)C2=O)=O)CN(C(=O)CCC2CCC2)CC1C1CC1 26784,Cc1cc(C(=O)N(CCCNC(c2cnn(C3CC3)c2)=O)C)cn1C(C)C 26785,C(CCC(C(=O)Nc1csnc1C1CC1)NC(c1cc(C)ccc1F)=O)OC 26786,CCCC(C(=O)NCC(N1CCCC(C(C)(C)O)C1)=O)OC.C1C(=O)N1 26787,N1(C(COCC(CCCC)=O)=O)CC(=C(F)CN)C1.C(CO)O 26788,c1(CNC23CCC(C(N=c4ccn(C)[nH]4)=O)(CC2)CC3)c(Cl)ccc(Br)c1F 26789,c1(C(N2CC(CNC(Cc3cc(CC)on3)=O)C(C)C2)=O)ccc(N)c(Cl)n1 26790,C(=O)(C1=C(C)CCCC1(C)C)N1CCC(NC(C(c2ccccc2Cl)OC)=O)C1 26791,Cc1ccc(C=CC(N2CCCC(CCNC(=O)CC(C)F)C2)=O)cc1Cl 26792,Cc1c(C(N2CC(F)CC2CNC(=O)CCS(C)=O)=O)nnn1C 26793,c1(C(=O)OC)nccnc1C(=O)N(C(C)C(N1CCC(O)C1)=O)C1CC1 26794,C1(CC)CN(C(=O)Cc2ccno2)CCC1NC(=O)CC(C)(F)F 26795,N1(C(CN(C(C(n2ccc(C)n2)C)=O)CCO)=O)CC2(C)COCC2(C)C1 26796,c1(C(=O)NC2C(NC(C(C)C(F)(F)F)=O)C2)ccc2c(c1)NCCC2 26797,C1(NC(C(CC)OCC)=O)CN(C(c2ccc(OC(F)F)cn2)=O)CC12CC2 26798,CCC(CC)(CC)C(=O)N1CCC(CC(=O)N(C2CCCC2(C)O)C)CC1 26799,c1(CNC(C2ON=C(CC)C2)=O)nn(C)c2c1CN(C(=O)C=C(C)C(F)F)CC2 26800,C1(C(N2C(CN=c3nc(CC)[nH]s3)CCCC2)=O)CCC2(CC1)CC(O)C2 26801,Cn1cc2cc(C(=O)NC3C=CC(CNC(=O)C(F)CC4CCC4)C3)ccc2n1 26802,C(CCC(C(=O)N(C)Cc1nncn1C)NC(c1csnc1Cl)=O)OC 26803,c1(-c2cc(C(=O)NCC(CC)OC)no2)ccccc1C#N 26804,Cc1ccc(C(=O)NCCC(O)CNC(C2CC(O)C2)=O)c(N)n1 26805,c1(CCC(=O)NCC2(C(=O)CNC(=O)NCC3CCCCC3)CC2)nc(O)n[nH]1 26806,N1(C(c2ccc(C)cc2)=O)CC2CCN(C(=O)C(CO)N(C)C)C2C1C 26807,C(CCCC(=O)N(C)CC=CC(=O)NC(CCF)C(=O)OC1CC1)OCC 26808,N1(c2ccnc(C)n2)CCC(C)C(NC(C2CC3CC3C2)=O)C1C 26809,C1(NC(C2(C#C)CC2)=O)CCN(CCNC(C2(OC)CCCCC2)=O)CC1 26810,c1(COC2CCCN(C(CNC=O)=O)C2)cccc2cncn12 26811,N1(C(C2C(=C)C2)=O)CC=C(C(=O)NCC2Cc3nccn3C2)CC1 26812,c1(OCCC(=O)NCCC(C)NC(C2C(F)(F)C23CC3)=O)cccc(F)c1 26813,c1(C(C)C)cc(C(N2CC(C)(CCC(N3CC(O)(CCO)C3)=O)C2)=O)n[nH]1 26814,Cc1nc(C=CC(=O)NCC2(NC(=O)CC3(CO)CCC3)CC2)cs1 26815,C1(C)(C(=O)NCC(CN(C)C(c2csc(-c3ccco3)n2)=O)O)C(C)(C)C1(C)C 26816,C1(C(=O)NCCC#CCC)CCN(C(=O)CC(C)N(C)C)C12CC2 26817,C1(C)(CC(=O)NCCOC)CCN1C(C1CC1C(C)C)=O 26818,C1(C(=O)OC(C)(C)C)(NC(=O)C(c2ccc(Cl)nc2)(C)C)CC2CC1C2 26819,N1(C(c2cc(CC)[nH]n2)=O)CC2CN(C(c3ccc(C)nc3)=O)C2C1 26820,C1(NC(C(C)(C)NC(C)=O)=O)CCCC1(C)NC(=O)C=C(C)C 26821,C1(c2nnnn2-c2ccccc2Br)(NCc2ccc(CC)nn2)CCCC2(CC2)C1 26822,C1(C(=O)NC2(CC)CCN(C(c3cc(CO)[nH]n3)=O)C2)CCc2c(n[nH]c2C)C1 26823,N1(C(C2(C(=O)OCC)CCC2)=O)CCC(CNC(=O)CC2CCC2)C(O)C1 26824,CCCCCCCC(=O)NC(CCOCC)C(=O)NCC1CC=CCC1 26825,C1(C(=O)NCC2CCN(C(=O)CCc3cc[nH]n3)C2)CCCC1C1CC1 26826,CC(C)S(=O)c1ccc(C(=O)NCC2(NC(C3COC(=O)N3C)=O)CC2)cc1 26827,N1(C(C(C)N(C(C)=O)C)=O)CCC12CN(C(=O)C(C)(C)N(S(C)(=O)=O)C(C)C)C2 26828,O=C1Cc2c(C(N3CC(O)(CCNC(C45CCCCC4C5)=O)C3)=O)cccc2N1 26829,C1(NC(C)=O)CCN(Cc2ccc(C#N)s2)CC1C 26830,C1(NC(CCSC)=O)(CNC(C2(N3CCOCC3)CCC2)=O)CCCCC1C 26831,C1(NC(C(CSC)C)=O)CCN(C(c2cc[nH]c(=N)n2)=O)C1(C)C 26832,c1(C(=O)NC2CCCC(CNC(C(CC#C)O)=O)C2)cccc2nc(CO)[nH]c12 26833,N1(C(C2C(C)OCC2)C(=O)NCc2ccco2)CCCC(C)(CNS(C)(=O)=O)C1 26834,c1(C(N2CCC(NC(C3CCCCS3)=O)CC2)=O)ccc([N+](=O)[O-])cc1O 26835,N1(C(c2c(C)n(C)nn2)=O)CC(F)(F)CC1CCNC(=O)C1=CSCS1 26836,c1(CSC)cc(C(=O)NC2CC2CNC(=O)C2=C(C)OCC2)ccc1F 26837,N1(C(c2c(C(C)C)onc2)=O)CC2CCC1CN2C(c1cccc2nccn12)=O 26838,C1(NC(C=C(COC)C)=O)CN(C(c2cnc(O)cc2C)=O)C2(CCOC2)C1 26839,N1(C(C2C3(CC(C)(C)C3)C2)=O)CC2(C1)CN(C(=O)C=C1CCCCC1)CC2CO 26840,C1(C(N(CC(C)NC(C2(F)CC2)=O)C)=O)CC2CC2C1 26841,n1(CCc2onc(-c3ccc4ccn(C)c4c3)n2)cnc2ccccc2c1=O 26842,c1(N2C(CNC(c3csnn3)=O)CC(F)(F)C2)ncnc2c(F)c(F)ccc12 26843,C1(C(=O)OC)(C(=O)NCC(C)(C)NC(c2cc(C#N)c[nH]2)=O)CCCCO1 26844,C(=O)(C(C)(C)CS(C)(=O)=O)NC1CC(C)CN(C(=O)Cn2nc(O)ccc2=O)C1 26845,C(N(C)N1CCC(C)(CC(=O)OC)CC1)c1cccc(OCC)c1 26846,N1(C(CC2CCC(=O)N2)=O)CCCC(F)(C(=O)N(C2CCCC2)CCO)C1 26847,N(C1CCOc2ccc(F)cc21)C(C(c1ccc(C)nc1)N)=O 26848,NS(=O)(=O)c1ccc(C(N2CCC(CCNC(C3CC3c3ccsc3)=O)C2)=O)o1 26849,c1(C(=O)NC(CCN(C(CCCC(C)=O)=O)C)C(C)(C)C)cc2c([nH]1)CCCC2 26850,c1(C(C(=O)NC2CC(F)(F)C2)N(CC(=O)NC)CC)nc(Cl)cc(Cl)c1C 26851,c1(OCCOC)ncccc1C(=O)NC1CCC(NC(=O)C(C)(C)O)CC1 26852,N1(C(c2ncn(C)n2)=O)CCC2(C(N3CCN(CC(F)F)CC3)=O)CC2C1 26853,N1(C(COC(CC)C)=O)CCC(CNC(=O)Cc2cnsc2)C(CC)C1 26854,c1(OC)cc(Br)c2c(c1)CCN(C(=O)NCC1(OC(C)C)CCOCC1)C2 26855,N1(C(C(CC#C)NC(c2cnncc2)=O)=O)CC2CC(C)(C)C2C1 26856,N1(C(C2(CCCC)CC2)=O)CC(NC(=O)CC2CC(N(C)C)C2)C(CC2CC2)C1 26857,CCCC(C)(CC)C(=O)NC1CN(C(c2cccc(C(=O)OC)n2)=O)CC1N=[N+]=[N-] 26858,Cc1cc(N)c(C(=O)NC2CC(N(C(=O)C(C)CC(C)(C)C)C)C2)cc1C 26859,C(CN(C(=O)CCc1nncs1)C)(CO)(CO)NC(C(C)C)=O 26860,N1(C(c2ccc(C(C)=O)cn2)=O)CCC(CNC(=O)C(C)C2CC2)C(F)(F)C1 26861,S(=O)(=O)(c1ccc(C(=O)N(C)C)cc1)NC1CCC(CC)CC1 26862,C1(CC#C)CCN(C(C2CC(O)(CNC(=O)COc3cccnc3)C2)=O)CC1 26863,CC1(C(=O)N2CC(NC(c3sccc3Cl)=O)C3(CCC3)C2)COc2ccccc21 26864,c1(C(=O)OC)ccccc1C(N1CCCC1CC(=O)N(CC1CCCCO1)CC)=O 26865,CCCCCCC(CC)NC(C1CCCCCN1C(=O)C=Cc1ccncn1)=O 26866,N1(C(C2N(C)CC(C)(C)C2)=O)CC=C(CC(=O)NCC23CCCC2C3)CC1 26867,N1(C(CC(CC)C2CC2)=O)CCC2C(C1)CN2C(c1csc(Br)n1)=O 26868,C1(CN(C(=O)C=Cc2ccc[nH]2)C)CN(C(=O)CCNc2cnccn2)CCO1 26869,CC1CCC(=CC(=O)NC(C)(C(=O)NC(c2cscn2)C)C2CCC2)CC1 26870,CCC(CC(=O)NCC(CC)NC(C1CCN(OC)CC1)=O)C(C)C 26871,C1(NC(c2c(C)nco2)=O)C2CCCN(C(c3cccc(F)c3C)=O)C2C1(C)C 26872,c1(SCC(=O)OCC(C2CC(C)NC2)=O)ccc(N2CCCCC2)cc1 26873,N1(c2ncnc(OC)c2OC)CCC2CN(C(=O)CCC(C)C)C2C1 26874,N1(C(C2N(C(C(CC)N(CC)CC)=O)CC(C)(C)C2)=O)CCn2c(C)nnc2C1 26875,C1(C)(NC(C2N(C(C(C=C)C)=O)CC(F)(F)C2)=O)CCC(C)=C(C)C1 26876,C1(C(=O)NC(C(=O)NC2CC(C(=O)NC)C2)C)CCC2(CCC2)C1 26877,C(=O)(C1=CCCC1P(C)(C)=O)NCCN(C(CC(C=C)(C)C)=O)CC(C)O 26878,C(=O)(C(CC1CC1)N(C(=O)CCC1CCCC1)CC)N(CCN=[N+]=[N-])CC 26879,C(C)(C(N)CC(=O)N1CCCC1CCc1cccs1)OCC 26880,N1(C(C(C2CC2)OCC)=O)CC2(CCC(NC(c3ccnn3C(C)C)=O)CC2)C1 26881,N1(C(C(=O)N(CCN(C(CSC)=O)C(C)C)C)CC)C(=O)c2ccccc2C1=O 26882,c1(NC)ccc(C(=O)N(CC(C)(C)NC(C2CCC3CC23)=O)C)cn1 26883,C(=O)(C1=NOC2(CCC2)C1)N(CC(CC)NC(c1cc(C#N)oc1C)=O)C 26884,CC(C)(O)CC(=O)N1CCC(N2CC(C(=O)NC3(C4(C)OCCO4)CC3)C2)CC1 26885,CC1(C)CC(C(=O)NCC23COCC(C2)C3)N(C(=O)COC(C2CCCC2)C2CC2)C1 26886,CS(=O)(=O)c1ccc(C(=O)NC2CCN(C(=O)C(F)C3CCC3)CC2)cc1 26887,C1(CNC(CCN(C(CCC)C)C)=O)CC(NC(c2cnn(C3CC3)c2)=O)C(O)C1 26888,c1(C(=O)NC(C(=O)NC)C(C)(C)C)coc2c1CN(C(c1ccc(C(C)=O)[nH]1)=O)C2 26889,c1(C(=O)NCC(C)(CC)NC(CC=CC=C)=O)cc(OC)cc(OC)c1 26890,CC1(C)CC(Sc2ccccc2Cl)(Oc2ccc(Br)c(F)c2)CO1 26891,C(=O)(C(C)C(F)F)N(CC(C)C(=O)NCC1(CO)CCCO1)C 26892,c1(C(N2C(CNC(C(CCC)=CCC)=O)CCCC2)=O)cnc2ncccn12 26893,N1(C(C2(C(=O)OCC)CC2C)=O)CCc2cc(NC(C3CC(O)C3)=O)ccc2C1 26894,c1(C(=O)NC2C(NC(CC(C=C)(C)C)=O)CCC2)ccc(C)c(Br)c1N 26895,c1(C(=O)NCCN2CCC(NC(C(C(C)O)C)=O)CC2)cc2n(c1)CCCC2 26896,c1(C(=O)NC(c2cccn2C)C)cc2c(cnn2C)nc1C(F)F 26897,c1(C(N2C(CNC(C3C(CCC)C3)=O)CC(CC)C2)=O)cccc(OCC)c1 26898,N1(C(Cc2cc(C)sc2)=O)CCCC(C)(C(=O)NCC2CCC(=O)NC2C)C1 26899,N1(C(CCN(C(CCCCOCCC#C)=O)C)=O)CC2CCC2(CC(=O)O)C1 26900,n1(C2(C(=O)NC(C)C(C)NC(=O)Cc3cc(C4CC4)on3)CC2)cc(Br)cn1 26901,c1(CC(=O)NC2CCCC(NC(C(C=C)O)=O)C2)cc(F)ccc1Cl 26902,N1(C(c2c(C)cco2)=O)CC2CCC1C1CN(C(c3occc3F)=O)CC21 26903,c1(CC(=O)NCC(O)CNC(C23CCC(C2)C3)=O)cccc(Cl)c1 26904,C12C(CCN1C(c1csc(CC)n1)=O)CC(C#C)NC2=O.CC.NC 26905,N1(C(c2nnc(C(c3ccccc3)C)o2)=O)CCCC(c2nnc(O)o2)C1 26906,N12CCC(C3(CC3)NCCCC1=O)CC2.c1(C(C)=O)ccc(C(=O)O)cc1 26907,C1(CC(=O)NCCOCCNC(C2(C)C3CCC23)=O)CC2(CCC2)CO1 26908,Cn1c(C(N2CCC(O)(CNC(C3(C)CCNC(=O)C3)=O)C2)=O)ccc1C#N 26909,C1(NC(C(CCC)OCC)=O)CCCN(C(=O)Cc2cnoc2)CC1 26910,N1(C(c2nc(C(C)OC)sc2)=O)CCCC(N(C(=O)CC2CCC(=O)N2)C)C1 26911,C1(N(c2c(OC)ccs2)C(C2C3CCCOC23)=O)CCNCCC1C 26912,c1(C(=O)NCCCCN(C(C2ON=C(C)C2)=O)C)ccnc2c(I)cccc12 26913,C1(NC(c2cncc(C)c2)=O)COC2(CCN(C(=O)CC34CCCC3C4)CC2)C1 26914,C1(C2CC2)(C(N2CCC(NC(CCC(=O)OCC)=O)C2)=O)CCOCC1 26915,C(=O)(C1CCc2nccn21)NC1C2(OC(C3CN(C(C)=O)C3)=O)CC2CC1 26916,c1(OCC)cncc(N2CCCC2Cc2ccc(C)cc2)n1 26917,c1(C(N2C(CNC(c3ncncc3Cl)=O)C=CC2)=O)ccc2scnc2c1 26918,c1(C(=O)NC2CC(CCC(=O)NCCCCC(=O)NC)C2)cc(C)nc(C)c1 26919,C(=O)(C(C)C(=O)OC)N(CCC)CCNC(=O)COCCC(C)C 26920,c1(C(=O)NCCNC(c2c(C)nc(CC)o2)=O)c(F)ccc(Br)c1Cl 26921,c1(C(=O)NCCC2CCN(C(c3cnc(C(=O)OC)s3)=O)C2)nnn(C)c1C 26922,N(C(=NCC1CC2CCC2C1)NC1CCC1)C(COC)C.S(C)(=O)(=O)N 26923,N1(C(Cn2ncc(C)c2)=O)CC(C)(CNC(C2CC2C2CC2)=O)CC1(C)C 26924,C1(NC(CCNC(C(=O)OC)=O)=O)OC(C)(C)OC1C(=O)N(C)C1CC1 26925,c1(C(=O)NCCCCC(C)NC(CSCC=C)=O)ccc2n[nH]cc2n1 26926,C(=O)(C1=CSCCO1)NCC1CC(C)N(C(c2ccn(CC(F)F)n2)=O)C1 26927,C(=O)(C(=O)CC(C)CC)Nc1ncoc1C(=O)NCCC=CCCC 26928,Cc1c(C(N2CC3C(CNC(=O)C4=COCC4)C3C2)=O)cnn1C(C)C(C)C 26929,N1(CC(=O)NC(C)C(c2ccccc2)NC(=O)C2=CCC2)CCCC1CO 26930,N1(C(C2(CC(C)C)CC2)=O)C2CCC1CC(NC(C1(C#N)CCOCC1)=O)C2 26931,CC1CCC(CNC(C23CC(C2)C(C(F)(F)F)O3)=O)N(C(=O)CNC(N)=O)C1 26932,N(C(=NCCc1ccc(Br)cc1)NCC(=O)NC(C)(C)C)C(CC)C 26933,CC1C2CCC(C2)C1C(=O)NCC1CCC(CC(=O)NCCc2nc[nH]n2)CC1 26934,N=c1nc(O)c(-c2cn(C3CC(CNC(=O)C(O)Cn4cncn4)C3)nn2)c[nH]1 26935,CCCS(=O)(=O)C(C)C(=O)NCCCOCCCNC(=O)CSc1nccn1C 26936,C1(NC(c2c(C)cns2)=O)CC2CC1CN(C(=O)C(C1CCCCCC1)O)C2 26937,CCC(F)C(=O)NCCN(C(=O)CC1CC=CC1)C 26938,c1(CNC(c2c(-n3cc(CC(C(C)C)O)nn3)cccc2)=O)cccc(F)c1F 26939,N1(C(C(c2cccc(F)c2)C)=O)CC(CNC(c2n[nH]c(O)n2)=O)C(C)C1 26940,N1(C(C2C(C=C)C2)=O)CCCN(C(c2ccnn2CC)=O)CC1COC 26941,C(=O)(C1=CC2(CCN(C(C34C=CC(CC3)C4)=O)C2)C1)N(CC(F)Cl)C 26942,C1(CC(=O)NCCC(=O)OCC)N(C(=O)CC2CC(C)(C)C(=O)N2)CCC1(C)C 26943,N1(C(N2CCN(CC(=O)NC3C(C#C)C3)CC2)=O)CCn2ccnc2C1 26944,C=CCCC(C(=O)NCC(CC)C(N)=O)NC(=O)CO.C(=O)CC(C)C 26945,c1(C(=O)NCC(C)NC(=O)CN(C)C(C)C)cc(Cl)c2n[nH]cc2c1 26946,Cc1coc(C(C)C)c1C(N1CCCC(c2ccc(=N)[nH]c2)C1)=O 26947,c1(NC(=O)C=CC2CC2)cccc(C(F)(F)F)c1.c12nc(cs1)CC(=O)N2CCO 26948,C1(CNC(C(C2CCCC(=O)N2)C)=O)CCC(NC(c2cnns2)=O)CC1 26949,c1(C(N2CCC(C(=O)NCC3CC(OC)(OC)C3)C2)=O)ccc(C(C)(C)C)cc1 26950,C1(CCC)CN(C(c2ccc(C(O)CF)cc2)=O)CCN1C(C1CC1OC)=O 26951,c1(C(=O)NC(CC)CN(C(=O)CC2CCOC2)C)ccnn1C(F)F 26952,C(C)(CCCC(=O)N1CCC(CC(C)O)CC1)NC(C(C)OCCCC)=O 26953,C1(NC(=O)CN2CCCC2)CN(C(c2ccc(C3CC3)nc2O)=O)CC1(F)F 26954,N1(C(c2cc(CCOC)on2)=O)CC2CCC2(CC(=O)NCCC(=O)N(C)C)C1 26955,c1(CCC)onc(C)c1C(=O)NCC1(C)CCN(C(C2(C#N)CCCO2)=O)C1 26956,C=CC1CN(C(=O)C2=CCN(C)C2)CC1NC(c1c[nH]c(-c2ccccc2)c1)=O 26957,C1(C(=O)OC)CN(C(C2CC2c2cccc(C)c2)=O)CC(=O)N1 26958,CC1CCC=C1C(=O)NCCCOCCNC(C1CC1c1cncn1C)=O 26959,Cn1cc(C(N2CC(OC)CC(NC(=O)CCNC(=O)CO)C2)=O)ccc1=O 26960,c1(C(N2CCC3CN(C(C4CCCS(=O)(=O)C4)=O)C3C2)=O)cccc2c[nH]nc12 26961,CN=c1ccc(C(=O)NC(C(=O)NCC2CCOC(C)(C)C2)C(C)C)c[nH]1 26962,c1(C(=O)NCC(C)(CO)NC(c2cc(CCC)[nH]n2)=O)ccc(C)cc1OC 26963,N1(Cc2c(=N)cc[nH]c2)CCCC(C(N2CC3CCCC2C3)=O)CC1 26964,Cc1cccn2ncc(C(N3CC(O)(CN(C)C(C4CNC(=O)N4C)=O)C3)=O)c12 26965,C1(C(=O)NCCN(C(=O)CCCCOCC)CCC)CC2(C1)CC(C)C2 26966,N1(C(CCC#CC)=O)CC(CNC(c2ncccc2CC)=O)C2(CC2)C1 26967,C1(CC(=O)N(CCCN(C(C=CC(C)(C)OC)=O)C)C)CCC2CC2C1 26968,CN1CC(F)CC1C(=O)NCC1CCC(NC(C2CC2CC(C)(C)C)=O)C1 26969,C1(NC(C2N(C(C(C)OCOC)=O)CC2)=O)CC2(C1)CN(C)C2 26970,C12CCCN1C(=O)CCOC2.C1(CC(N2CC(OCC#C)C2)=O)C=CCCC1 26971,c1(C(=O)NCC2(C)CC(NC(c3c(C(C)C)ocn3)=O)C2)ccc2c(c1)CCC=C2 26972,C1(C(=O)NCCCCN(C(C2(COC)CC=CC2)=O)C)CCC(C)(C)CO1 26973,C1(C(=O)NCCC(CNC(c2csnn2)=O)O)CCCCC(=O)N1 26974,c1(C(=O)NC2CCN(C(c3sccc3Cl)=O)C2)nnn2c1C(=O)NCC2 26975,C(=O)(C1=NOCC1)N1CCC(N(C(C(CC)N(c2ccccc2C)CC)=O)CC)C1 26976,C(C(CC1CC1)C(=O)NCC1(F)CC1)NC(C(CC)n1cncn1)=O 26977,c1(OCC)ccc(NC(c2cc(CNC(c3cc(O)nn3C)=O)[nH]n2)=O)cc1 26978,C1(C(=O)NC(C)CC2CN(C(=O)CCc3cnoc3)C2)CCc2nncn2C1 26979,C1(CN)(NC(=O)Nc2c(C(C(N3CCCC3)C3CC3)=O)cccn2)CCOCC1 26980,c1(NC(C(c2ccccc2)NC(c2cccc(F)n2)=O)=O)cc(CO)cc(O)c1O 26981,C(=O)(C(F)CC(C)(C)C)NCCN(C(c1ncccc1N)=O)CC 26982,Cn1nc(Br)c2ccc(C(N3CC[Si](C)(C)C3)C(=O)NCC3CCOC3)cc12 26983,N1(C(C(CC(CC)C)C)=O)CC(C)CN(C(c2cccc(CSC)c2)=O)CC1C 26984,C12(CNC(C(=O)NCC34CCCC3C4)=O)CCC(CC1)O2 26985,Cc1ccc(C(N2CCOC(C#N)C2)C(=O)NCCOCC2CC2)c(F)c1 26986,N1(C(C(C=C)CC)=O)CC2(C=C(C(=O)N(C3CC(OC)C3)CCC)CO2)C1 26987,N1(C(C(C(=O)OC)C)=O)CC(C(=O)N(C)CCc2nccs2)CCC1(C)C 26988,C1(=O)CCCCCNCC(C)N1C.C(c1cnc(C)s1)=CC(=O)N(CC)CC 26989,C(CC(C)(C)C(=O)NC(C(=O)NCCOC1CCOC1)C1CCCO1)OC 26990,S(=O)(=O)(c1cc(F)cc(F)c1)NC1CN(C(=O)CCCCc2cccs2)CC1F 26991,C(=O)(CC1OB(O)c2ccccc21)N1C(C)CN(C(=O)C=C2CCCC2)CC(C)C1 26992,C(C1=CCN(C(C2CCC3(CC2)CC3)=O)CC1)NC(C(CC=C)OC)=O 26993,c1(OC)cc(CN=c2ccnc(NC3COCC3C3CC3)[nH]2)c(F)c(F)c1F 26994,C1(C(N2CCC(CCC)C2)=O)CC(O)CN1C(c1ccc(Cn2ccnc2)o1)=O 26995,n1(CCNC(N2CCOCC(CC(C)C)C2)=O)nc2c(n1)CCCC2 26996,C1(C(C)NC(C2CCN(C(C)=O)CC2)=O)CN(C(=O)C=CCN(C)C)CCCO1 26997,c1(N2CCC(C)C2)nc(Cl)ncc1C1CCN1C(c1ccc(CCN(C)C)s1)=O 26998,c1(C(=O)NC2C(NC(=O)CCn3c(O)nnc3O)CC2)n[nH]cc1[N+](=O)[O-] 26999,CC1(Nc2ncccn2)CC(NC(=O)CSCC2CC2)C1 27000,N1(C(C(C)(C)O)=O)CCN(Cc2sc(Br)nc2Br)CC1c1ccccc1 27001,C1(C(=O)NCCN(C(C)C)C(C2CC23CCC3)c2ccccc2)CC(F)(F)C1 27002,N1(C(c2n[nH]c(C)c2O)=O)CCC2CN(C(=O)CCc3nc(C(C)C)no3)C2C1 27003,Cn1c(=O)n(C)c2cc(CN)ccc12.C12CC3(CCC(CC3)N1)C2 27004,C(CN=c1cc[nH]cc1S(=O)(=O)N1CCCC(CF)C1)c1c(C)c(Cl)c(Cl)cc1 27005,c1(OCC(=O)NC(C2CN(C(C(CC)F)=O)C2)C)ccc([N+](=O)[O-])cc1 27006,c1(C(=O)OC2CC(C)(C)C2)cc(Br)cnc1OC(F)F.C(=O)(C(=O)NC)NC 27007,N1(C(CC2C(C)OCC2)=O)CCOCCC1C(=O)Nc1cnc(C(C)C)nc1 27008,CCC(F)(F)CC(=O)N1CCC(C)C(NC(=O)Cn2cnc(Br)c2)C1 27009,C(CNC(=O)Cn1cc(N)cn1)(C(C)(C)C)NC(C1(CC=C)CCC1)=O 27010,c1(C(N(C2CCCCN(C(C3CC3CF)=O)C2)C)=O)cc2cn[nH]c2cn1 27011,C1(NC(C2CCC(CC)O2)=O)CCN(C(c2cc(C)cc(Cl)n2)=O)CCC1CO 27012,C1(CNC(C2(CC)CCCCO2)=O)CCN(C(c2cnn(C)c2)=O)CC1O 27013,N1(C(c2cncc(OCC)c2)=O)CCC(F)(CNC(=O)CN2CCCOC2=O)C1 27014,C(CNC(C1CC1c1cccc(Cl)c1)=O)(C(C)(C)C)NC(C12CC(C)C1C2)=O 27015,C1(COC)CN(C(=O)C=Cc2cccnc2)CCN1C(c1csc(COC)n1)=O 27016,N12CCCC(N(C)C)(C1)C(OC)c1cn(nn1)CC2=O.CCS(=O)(=O)C(=O)OC 27017,C1(C(N2CC(O)(CCC)C2)=O)CCN(C(=O)CCN=[N+]=[N-])C(C)(C)C1 27018,N1(CCCC#N)CCCC(C2CCN(C(C3CC34CCOC4)=O)CC2)C1 27019,C1(NC(C(c2ccccc2)OC(C)=O)=O)CC2CC(N(C)C)CC12 27020,N1(C(c2n(CC)ccc2)=O)CCOC(CC(=O)N(C)CCN2CCOCC2)C1 27021,Cc1ccc(C(C)C(=O)NCC(O)CNC(c2ccc(N)cn2)=O)cc1 27022,c1(CC(=O)NCC(C(C)C)NC(C(C(C)C)F)=O)c[nH]c2cc(Cl)ccc12 27023,C(=O)(CCCCN=[N+]=[N-])N(C(C)C(=O)Nc1cccc(CC2CCC2)c1)CC#C 27024,O=C(C(O)CCC1CCCC1)NC(CNC(=O)C=Cc1cccs1)C1CCC1 27025,C(=O)(C(C)C(O)CC)NC(CC=C)C(=O)Nc1ccc(CO)cc1O 27026,C(C(C)C(=O)NOCC1CCOCC1)NC(C(COC)(C)OC)=O 27027,CC(=O)CCCC(=O)NCCN(C1CCCCC1)C(C1CCCC1P(C)(C)=O)=O 27028,N1(C(c2ccn3c2CCCC3)=O)CC2CCCC(O)C2C1 27029,N1(C(C2(CCOCC)CCCC2)=O)CCC(O)(CN(C(=O)C=C(C)C(C)C)C)C1 27030,c1(C(=O)NCC(CN(C(C2=NOC(C)C2)=O)C)(C)C)cc2cc(Cl)ccc2o1 27031,c1(C(N(C)CC2CCCN(C(C(C(C)O)(F)F)=O)C2)=O)c(F)cc(F)c(F)c1F 27032,c1(C(N(C(CCNC(C2C(=C)C2)=O)C)C)=O)cc(N(C)C)ccc1N 27033,C(=O)(C1CCOc2c(F)cccc21)NC1(C(=O)NCCNOCCC(C)C)CCC1.O 27034,c1(N(C)C)cnc(C(N2CCC(NC(C3C(C(F)F)C3(C)C)=O)C2)=O)nc1 27035,Cc1c(C(=O)NC(CNC(=O)CC2CCC(=O)N2)CO)nn2ccccc12 27036,N1(C(C2C(C)C2)=O)CC(NC(=O)C2=CCCCO2)CC12CCC2 27037,n1(CC(=O)NCC2CC2CNC(C2CCC(CCO)CC2)=O)ccc(O)nc1=O 27038,N1(C(Cc2c(C)cc(C)s2)=O)CCC(CO)C(NC(=O)Cc2cccnc2C)C1 27039,C1(C(=O)NC2CC(CNC(C3(C)COC3)=O)OCC2)CCCCN1N=O 27040,c1(OCCC)cccnc1C(=O)N(C)CC1CN(C(=O)C=CCOC)CCO1 27041,c1(OC)cccc(C(=O)NCC2CC(NC(=O)CCCC(N)=O)C2)c1O 27042,N1(C(C2C(OC)CC2)=O)CCC(CO)(NC(=O)CCc2cc[nH]n2)CC1 27043,C1(NC(c2c[nH]nc2CCNC(c2cccc[n+]2[O-])=O)=O)CC1C1CCC1 27044,CCC(C(=O)NCC12CC(NC(=O)C(F)OC(F)(F)F)(C1)C2)n1ccnc1 27045,c1(C(N(C)CC2CCCN2C(=O)CC2(O)CC2)=O)cc(OC)cc(Br)n1 27046,Cc1cc(C)c(CNC(=O)C(=O)Nc2n[nH]c(C(C)C)n2)c(C)c1 27047,Cc1ccc(C(=O)N(CCCNC(C2C3CCCCCC23)=O)C)c(O)c1C 27048,c1(CC)nc(NC2CN(C(=O)CC3CCCC34CC4)CC2(C)C)c(C#N)cc1C 27049,C1(CNC(=O)CCCC2(NC(c3cccc[n+]3[O-])=O)CCC2)CCCC2(CC2)C1 27050,C1(NC(CCSCCC)=O)CC2CCC1CC2NC(c1csc2nccn12)=O 27051,c1(C(=O)NCc2cccc(COC)c2)oc2cccnc2c1NCC1(CC)CC1 27052,N1(C(N(c2ccnc(C(=O)O)c2F)CC)=O)CCC(C2CCNCC2)C1.C(C)(C)(C)OC 27053,C1(C(=O)NCC(=C)C)CCCN1C(c1ccc(Cl)o1)=O.C(=O)OC 27054,c1(CCC(N2CC(NC(C3CCOC3)=O)CC(C)C2)=O)ccc2ccn(C)c2c1 27055,C1(F)(C(=O)NC(c2onc(C)n2)C)CCCN(C(=O)CC2CCC2)C1 27056,Cc1c(O)ccc(C(N2CCCC(C(C)NC(C3(CF)CCC3)=O)C2)=O)c1C 27057,C1(NC(CCc2cc(C)on2)=O)CC2CCC(C1)N2C(C1CC1C(F)F)=O 27058,C(=O)(C1=CCCCO1)N1CC2C(NC(C3(COC)CCCOC3)=O)C2C1 27059,C(=O)(CC1OCc2ccccc21)NCC1N(C(=O)C(F)CC2CCC2)CC1 27060,C1(C(N2CCC3CN(C(CC(=C)C)=O)CC3C2)=O)C2Cc3c(Cl)cccc3C12 27061,C1(C)(C(N2OCC(=C)C2)=O)CN(C(=O)CCC(C)OC)C(C)(C)C1 27062,CC1CN(C(=O)C(C)Cc2cccc(F)c2)CCC1CNC(=O)C1=C(Cl)CC1 27063,CC1CC(NC(C2(C)CSC2)=O)CCN1C(C1(N(C)C)CC1)=O 27064,N1(C(C2N(C(CCC(C)N(C)C)=O)CCCC2)=O)CCN2CCCC2C1 27065,c1(C(N(C2CN(C(C3CC(CF)C3)=O)CC2F)C)=O)cnc2c(C#N)cnn2c1 27066,CC1(C)CC(NC(C2CC(F)(F)C2)=O)CN(C(=O)CSC(F)(F)F)C1 27067,Cc1cccc(CNC(C2CC2c2ccccc2-c2cncn2C)=O)n1 27068,c1(C(C(=O)NCC2CCCO2)N(C)CC2C(C)C2)cc(Br)cc2nc[nH]c12 27069,C1(C(=O)NCC2CCN(C(C3OCCN(C)C3)=O)C2)CCC(=O)N(C)C1 27070,c1(C(N2CCC(NC(CC(CC)SC)=O)C2)=O)cc2ccccc2n1CC1CC1 27071,C(C(O)CN=C(NCCOC)NC1CCOc2ccccc21)N(C(C)C)CC 27072,c1(CCC)nnc(S)n1CC(=O)NCC=CCNC(c1cnc(C2CC2)o1)=O 27073,C1(NC(C2CCCN(C(C)=O)C2)=O)CCCC12CN(C(c1ccn(C)c1C)=O)C2 27074,C=CC1CCN(C(C2CCN(C(c3cc(C)nc(O)c3)=O)C2)=O)CC1 27075,N1(C(c2cc(SC)c(C)o2)=O)CCC2CN(C(C3CC(N(C)C)C3)=O)CCC2C1 27076,N1(C(C(CCOC)(C)C)=O)CCCC(C2CN(C(C3(S(C)(=O)=O)CCC3)=O)C2)C1 27077,c1(C(=O)NCC(C(=O)N(C(C=C)C)C)(C)CC)cn2ccccc2n1 27078,C12(CC(=O)NC(COC)CO)CCC1CN(C(c1csc(C)c1)=O)C2 27079,c1(C(N(CCOCCNC(CC(CCCC)O)=O)C)=O)cccc2c1OCC2C 27080,C1(C(=O)NCC2CN(C(C(CC)(O)c3ccccc3)=O)C2)C2CCCC(F)(F)C12 27081,CCCCCC(O)C(=O)NCC1CN(C(C2COCCN2C)=O)C1 27082,N1(C(C(CCNC(C(C)OCC)=O)O)=O)CCCCC(C)(F)C1 27083,c1(C(=O)NCCCN2CCC(NC(c3cc[nH]n3)=O)C2)cc(F)cc([N+](=O)[O-])c1 27084,C12(CNC(c3c(OC)c[nH]n3)=O)CCC1CCN2C(c1cnc(O)s1)=O 27085,C1(NC(CCN(C)CC)=O)CN(C(=O)C(N2CCN(C)CC2)C)CCC1C 27086,CC1C(C(N2CCN(CCNC(=O)CC(F)(F)F)CC2)=O)CCN1C 27087,CCC(CNC(C1CC(OC)CN1C(=O)CSc1ccccn1)=O)CC(C)C 27088,N1(C(C2N(C(CC(=O)NC)=O)CCC2CC)=O)CC(C2CCCC2)C1 27089,C(C)(C)(CC(C)NC(C1(NC(=O)C=Cc2cc[nH]n2)CSC1)=O)OC 27090,c1(C(=O)NCCN(C(C2(CC)CCOC2)=O)C)ccc(C(C)C)nc1O 27091,c1(CNC(C(CC)OC)=O)nnc2n1CCN(C(c1ccc(C)c(N)c1)=O)C2 27092,Cc1sc(C(=O)NC2(CCCCNC(=O)CCC3CC(OC)C3)CC2)nc1O 27093,c1(C(N(C)CCNC(C2CCCOCC2)=O)=O)ccc2c(c1)CCCC(=O)N2 27094,C1(CNC(C(=O)NC(c2ncccc2Br)C)=O)CCCOC1C(C)(C)C 27095,N1(C(CC=C=C)=O)CCCC(NC(c2coc(Cl)c2)=O)CCC1 27096,Cc1cc(O)cc2c1CN(C(C1CC1C(=O)Nc1cccc(Br)c1)=O)CC2 27097,c1(N2C(CNC(COCCN(C)C)=O)CC(F)C2)nc2cc(Cl)ccc2s1 27098,n1(CCC)cc(C(=O)N(C2CC(NC(=O)CCc3cccn3C)C2)C)c(C)n1 27099,C1(C#N)(CC)CCN(C(=O)CC2(NC(c3cccc(=O)o3)=O)CCC2)CC1 27100,c1(OC)cccc2c1CN(N1CCC(CCSC)CC1)C2 27101,CC(C(CO)NC(c1cnc(C2CC2)[nH]1)=O)NC(=O)C(c1cccn1C)=O 27102,c1(C(N(CCNC(c2n(CC)c(O)nc2)=O)C2CC2)=O)sc(C)c(Br)c1C 27103,Cc1ccc(C(N2CC=CC(NC(c3cccn3C)=O)C2)=O)c(F)c1F 27104,c1(CC(=O)N(C2CCN(C(C3C(=C)C3)=O)C2)C)c(C)c2cc(O)ccc2oc1=O 27105,c1(CC(=O)NC(CC=C)CNC(=O)Cc2cccc(Cl)c2)ccc(C)cc1Cl 27106,c1(C(=O)NC2CCN(C(c3c(C(C)C)ccs3)=O)C2)cc2c(cn1)OCCC2 27107,C1(CCC)(NC(c2cn(CCC)nn2)=O)CCCN(C(=O)CCn2cnnn2)C1 27108,CCC(CC)C(C)C(=O)NCCCC(C)(C)NC(=O)CCC1CCC(C)O1 27109,N1(C(c2c(C)c(C#N)[nH]c2)=O)CCC(F)(F)C(NC(C2CC3CCC2CC3)=O)C1 27110,c1(C(=O)NC2(C)CC(NC(C3(C)N(C)CC(O)C3)=O)C2)cc(F)c(Cl)cc1F 27111,N1(C(C(CSC)C)=O)CCCCCC(NC(c2cc(C)cnc2C)=O)C1 27112,c1(C(N2CC(NC(C(C(C)O)(F)F)=O)C(F)CC2)=O)ccc2c(c1)N(C)C(=O)C2 27113,Cn1cc(S(N)(=O)=O)cc1C(N1CC(NC(=O)CCCN=[N+]=[N-])CC(C)(C)C1)=O 27114,N(C(=NCCCCSC)NCC(C)(C)C#N)CC 27115,C1(C)(CCNC(COC(CC)C)=O)CCN(C(c2ncoc2-c2cccs2)=O)C1 27116,C(CN=c1ccnc(N2CCC(c3cccnc3)CC2)[nH]1)c1cc(O)n[nH]1 27117,C1(NC(C(C)NS(CC)(=O)=O)=O)(CF)CCN(C(c2c[nH]nc2C(=O)OC)=O)C1 27118,C(=O)(CC(=O)N(CC(=O)N(C1CC1(C)C)C)C1CC1)NCC 27119,c1(C(C)CC(C(CCCNC)=O)CN(C)C(C2CCC3CC23)=O)ccccc1 27120,C(C(CC(C)C)C(=O)NC(c1ccccc1)C#N)NC(c1cnn(C=C)c1N)=O 27121,CCC(CC(=O)NCC1COCCN(C(=O)C(F)C2CCC2)C1)CC(C)C 27122,CCC(C)(C)CCCC(=O)NC1CCN(C(=O)CNS(=O)(=O)CC)C(C)C1 27123,Cc1ccc(NCC(=O)NC2CCC(CNC(=O)COc3ccsc3)CC2)cc1 27124,Cc1cc(C)c(C(=O)N(CC(C)C(=O)NCC(O)C2CCC2)C)s1 27125,C1(OC)(CNC(=O)C(Cc2ccccc2)C2CC2)CN(C(=O)CC2(C)CCC2)C1 27126,C1(CCNC(CSCC=C)=O)CCCN(C(=O)C(C)Cn2ccc(C)n2)C1 27127,C(=O)(C#CC(C)(C)C)N(C1CCN(C(c2ccccc2-n2cccn2)=O)C1)C 27128,c1(C(=O)NC(C2(O)CN(C(=O)C(C)n3ccnc3)C2)C)cn(CC2CC2)nn1 27129,C1(NC(C2C(=C)C2)=O)CN(C(c2cc(C)n(C3CCCCC3)c2C)=O)CC12CC2 27130,Cc1ncc(C(=O)NCC2CC(F)CN2C(=O)CC2CCOC2=O)n1C(F)F 27131,c1(N2CCC(OCC=C)CC2)nc(=NCc2cc[nH]c(=N)c2)[nH]c2c(C)nn(C)c12 27132,CCCCC(F)(F)C(=O)NCCC1CCCN1C(=O)CCC1CNC(=O)N1 27133,C(CC(C)C(=O)NCc1ocnc1C(=O)NCCCC1CCC1)OC 27134,c1(N(C)CC2CCC2)nc(=NCC2NC(=O)CC2(C)C)[nH]c2c(F)cc(F)cc12 27135,C1(C(=O)NCC2C(C)CCN2C(c2cccc(CC#N)c2)=O)CC12CCSCC2 27136,c1(CC)cc(CC)nc(N2CC3C(CNC(=O)C(c4cnn(C)c4)SC)C3C2)n1 27137,N1(C(CSCC#N)=O)CC2CCC(CNC(C3CC3C3CCC3)=O)(C2)C1 27138,C(C(CO)C(C)CC)NC(C1C(CCC)CN(C(=O)C(C)(C)OC)C1)=O 27139,C1(C(C)CNC(=O)Cc2cc(Cl)n(C)n2)CCN(C(C2CCC(=O)N2C)=O)CC1 27140,C12(C(N3CCC(C(C)NC(c4cccc(N)n4)=O)C3)=O)CC3CC1(CO)CC3C2 27141,C1(NC(c2nc3c(s2)CCC3)=O)CCN(c2nnc(O)s2)CC1F 27142,CC(C)S(=O)c1c(NC(=O)Nc2ccnn2CC2CCCO2)cccc1C 27143,C(=O)(CC(C(C)(C)C)NC(c1cc(F)ccc1F)=O)N(CCN=[N+]=[N-])C 27144,N1(C(C2C(=C)C2)=O)CCN(C(c2sc(-c3nc[nH]n3)nc2C)=O)CC1CCO 27145,N1(C(C(C)(C)O)=O)CCCC(C(N2CCC(COC(F)(F)F)CC2)=O)CC1 27146,Cc1nn(-c2ccncc2)cc1C(=O)N(CCCNC(=O)C(C)(C)CF)C 27147,C(=O)(CCC(=O)N(CCCNC(=O)CCCCN1CCCCC1)C)N(C)C 27148,CCCCCC(C)CC(=O)NCCC1CN(C(=O)COc2cccc(C)c2C)C1 27149,C(=O)(CC(CC)CC(C)C)NC(CCC(=O)NCCC(=O)NC(C)C)C(C)C 27150,N1(c2ccnc(C)n2)C2CCC1(CN(C(c1cccc(F)c1F)=O)C(C)C)CC2 27151,c1(C(N(CC(C)NC(CCCn2c(C)nc(C)n2)=O)C)=O)cc2ccsc2n1C 27152,c1(NC)ccc(C(N2CCN(C(c3c[nH]ccc3=O)=O)C(C)C2)=O)cc1F 27153,CCC(CCC(=O)NC(C1CC(O)C1)C)NC(c1cn(C(C)C)cn1)=O 27154,C1(NC(C(C)c2ccco2)=O)CN(C(=O)C=CC2(C)COC2)CC1C1CC1 27155,N1(C(CCC(C)(C)C)=O)CCOCC(C)(CNC(C2CNC(=O)C2)=O)C1 27156,Cc1cnc(C(=O)NC2(CCO)CCCC2)o1.c1(C2C(=O)N2)ccn(C)n1.C(=O)(C)N 27157,C12(CNC(COCCOCC)=O)CCCCC1CN(C(=O)CCCS(N)(=O)=O)C2 27158,N1(C(C(C)n2cncn2)=O)CC2CC2(C(=O)NOCCF)C1 27159,CC(c1ccccc1)=CC(=O)NCC1(NC(C2CC3CC2C2CC32)=O)CCCC1 27160,c1(C(=O)NC(CNC(CC(C)(C)OC)=O)CC(C)C)cccc(F)c1C 27161,C1(C(=O)NC2(c3scc(C)n3)CC2)CCCN(C)C1 27162,c1(C(C(=O)NCC2CCN(C(=O)C=Cc3nccs3)C2)O)cc(Cl)cc(Cl)c1 27163,C1(NC(c2c(C)ncnc2)=O)(CO)CCCN(C(c2ccccc2Br)=O)C1 27164,C=CCCCCCC(=O)N1CCCC(CC(=O)N(C(C)C(C)C)C2CC2)C1 27165,Cc1sc2ncc(C(N3CC(CC(C)NC(C4(C)CCCC4C)=O)C3)=O)n2c1C 27166,C1(SC)CN(C(C2(OC(C)C)CCCCC2)=O)CC1NC(=O)C=C(C)C 27167,C(=O)(C1=NOC(C)C1C)N1CC2C(NC(CC3(COC)CCCCC3)=O)(CC2)C1 27168,N1(C(CCC(C)(F)F)=O)CCc2sc(CNC(=O)C(=C3CCCCC3)F)nc2C1 27169,C1(C(=O)NC23C(CN(C(C4N(C(N)=O)CCC4)=O)C2)C3)CS(=O)(=O)CC12CC2 27170,c1(C(N2CCN(C(C(C(C)C)C)=O)CC2C)=O)cccc2ccnn12 27171,N1(C(CNC(C(C)(C)C2CCCC2)=O)=O)CCN2C(=O)CCC2C1 27172,C#Cc1cncc(CN2CCN(C(=O)CN3C(=O)CSC3=S)C(CC)C2)c1 27173,N1(C(CCOCC)=O)CCC(C)C(NC(=O)Cc2ccc(NC(C)=O)cc2C)C1 27174,c1(CCC)ccc(C(=O)N(CC(C)N(C(=O)CC)C)CC(C)C)cc1[N+](=O)[O-] 27175,C1(C(N2CCC(C(C)CNC(c3csnn3)=O)CC2)=O)CCCC1C1CC1 27176,CC(C)CCCC(C)CNC(C1CC(C)CN(C(c2cncc(F)c2)=O)C1)=O 27177,CCCCC(C)(F)C(=O)NCCCOCCCNC(=O)CC1(C)CCCC1 27178,c1(C(=O)NC(C)CCN(C(=O)CCS(=O)(=O)N(C)C)C)ccc([N+](=O)[O-])cc1 27179,c1(C(=O)NCC2C(C)(C)C(NC(=O)C=CC3CCC3)C2)cncc2[nH]ccc12 27180,C(=O)(C(F)(F)C1(n2cc(Cl)cn2)CC1)NCCNC(C1(C2CCCO2)CCC1)=O 27181,N1(C(C(COC)C)=O)CCCC(O)(CNC(c2ccc(C(F)(F)F)cc2Cl)=O)C1 27182,C(=O)(C(C)C(C)(C)O)N1CCC(CCCNC(c2c(OC)c(C)cs2)=O)CC1 27183,c1(C(=O)NCCCC2N(C(CC(C)SC)=O)CCCC2)cccc2nncn12 27184,c1(C(C)C)n[nH]cc1C(=O)NCC(O)CNC(=O)CCc1ccsc1Cl 27185,C1(NC(c2csc(C)c2C2CC2)=O)CCCC12CN(C(=O)Cn1ccnc1C)C2 27186,C(=O)(CC(C)(C)C)NCC(N1CCC(c2cn(CCCC(=O)OCC)nn2)C1)=O 27187,c1(C(CNC(CC2CC(=O)C2)=O)NC(c2cnccn2)=O)ccccc1 27188,C1(CNC(C(C(C)C)(C)C)=O)CN(C(c2ncccc2Cl)=O)CC2(CCC2)O1 27189,N1(C(c2c(C)noc2)=O)CCCC12CCC(NC(=O)CNC(=O)C(C)(C)C)CC2 27190,C(CC(F)F)(C(=O)NC(C)Cc1cnc[nH]1)N(C(C1C(C)=CCS1)=O)C 27191,N1(C(C)C(=O)N(C2CC(F)(F)C2)C(c2ccoc2C2CCC2)=O)C(C)CCC1C 27192,CC(C(CO)NC(c1cncn1C)=O)NC(c1cn(CC2CCCO2)nn1)=O 27193,c1(CNC(c2ccccc2Br)C)ccc2c(c1)CNC2=O 27194,C1(NC(C(CSC)C)=O)CCSC12CN(C(=O)CCc1ccc(O)c(F)c1)C2 27195,CCCCCCCC(=O)NCC1COCC1NC(c1cc(C=CCCC)[nH]n1)=O 27196,c1(CN2C(C(=O)Nc3cccc(N(C)C)c3)CCC2)cc(Cl)cnc1Cl 27197,C(=O)(C(CN=[N+]=[N-])NC(=O)C(C)NC(c1ccoc1)=O)NCC(C)OC 27198,C1(C(N2CCC(CNC(C3(C)CCC(F)(F)C3)=O)CC2)=O)CCC2(CCC2)OC1 27199,c1(OC)ccc(C(=O)NCC(C)CNC(c2cc(C)cc(F)c2)=O)cc1C1CC1 27200,CC1(CNC(=O)CN2CC=CC2)CC(NC(c2ncsc2Br)=O)C1 27201,Cc1noc(C(C)C)c1C(=O)NCCNC(c1c(C)coc1C)=O 27202,c1(C(N2CCCC(CN(C)C(C3(Cl)CC3)=O)C2)=O)ccc(Cl)c2occc12 27203,C12(C(NOCC=C)=O)CCCC1CCN2C(=O)CC(C)(C)C=C 27204,C1(C(C(=O)OC)O)CCN(C(=O)Nc2c(COC)c[nH]n2)CC1 27205,CC1CN(C(=O)C2=CCCCC2)CC(C(=O)NCc2ccns2)O1 27206,c1(C(=O)NC2CC2NC(c2noc3c2CCCC3)=O)ccc2cccnc2c1 27207,C(CCCCCO)S.N1(C(CCN(CCCO)CC)=O)CCCC1C(C)(C)C 27208,c1(NC)ccc(C(N2CCC(CC)C2C(N2CC(OC(=N)O)C2)=O)=O)cc1 27209,C(=O)(CCCCC(=O)N1CC(CNC(=O)CC2CC2CN)C(F)(CO)C1)OC 27210,CC1(F)CCC(C(N2CCC(CCNC(=O)C(F)=CC3CC3)C2)=O)CC1 27211,CC(C)C(CNC(=O)CN(CC(C)C)C(c1cc(C)n(C)n1)=O)C(C)C 27212,CC#CCCCC(=O)NC1(C)CCCN(C(=O)C(CC)C(C)O)C1 27213,c1(CNC(C(C)O)=O)ccc2c(c1)CCN(C(c1coc(SC)c1)=O)C2 27214,C1(C)(C(N(CCN(C)C)C)=O)CCCN(C(c2cc(CCO)on2)=O)C1 27215,C1(C(=O)NCC2N(C(c3cc(C)oc3)=O)CCC2C)CCc2nncn2C1 27216,CCCCC(C)(F)C(=O)NCC(CC(=O)Nc1ccc(C2CC2)nc1)OC 27217,c1(CC)c(C(=O)N(CC(C)NC(=O)CC2(O)CCCC2)CC)cnn1C(C)(C)C 27218,Cc1ccc(C(=O)NC2CC(CNC(=O)CS(C)(=O)=O)C(O)C2)c2c1CCCN2 27219,C(C)(C)(CC(=O)N1CCCC(C(=O)NC2(CO)CCC(C)C2)C1)OC 27220,C(=O)(C1=COCCO1)N(CCN(C(CCC(=O)NCC(C)O)=O)C)C(C)C 27221,C(=O)(C(CO)NC(=O)CCN(C)C)N(C)CCC1CCCN1C 27222,c1(C(=O)NCC(CCOC)(C)C)cc(O)nc(C(F)F)n1 27223,C1(CC)CN(C(c2cc(C)oc2C)=O)CCC1NC(c1cnn(CC(F)F)c1)=O 27224,Cc1ncnc(C)c1OCC(=O)NCC12CC1CN(C(=O)CN(C)C1CC1)C2 27225,c1(N2CCN(C(c3c(OC)cncc3)=O)CC2C)ncnc2ccccc12 27226,c1(NC(C)=O)cccc(C(N2CC(O)(C(C)NC(C3CC34CCCC4)=O)C2)=O)n1 27227,Cc1cc(C)c(C(=O)NC(C)CCCCNC(=O)CCCC2CCC2)[nH]1 27228,CCCC(C)(C)C(=O)N1CCC(C)(NC(=O)CN2CC3CCC2C3)C1 27229,C1(C(=O)NCc2ccc(F)nc2F)CC12CCN(C(c1cc[nH]n1)=O)C2 27230,C#Cc1cccc(NC(=O)COC(C)(C)CNC(=O)C(C)(C)C(F)F)c1 27231,C#Cc1cn(C)nc1C(N1CC(NC(=O)CC2CC3CC(=O)C2C3)CC(O)C1)=O 27232,C(=O)(CCC(=O)c1ccncc1)N1CC(OCCN(C)C(C2CCNC2=O)=O)C1 27233,C1(C(=O)NCCNC(c2c(OCC)oc(C)n2)=O)CC1C1CC(F)(F)C1 27234,c1(SCCC(=O)NC2CC(C)(NC(C(CCN(C)C)O)=O)C2)cc(F)ccc1F 27235,C(CC#C)(C(=O)NC1CCC2(CC2)C1)NC(C=CC#C)=O 27236,C(=O)(CC(O)CC(C)C)NC(C(=O)NC(C#C)C)C1(C)CC1 27237,Cc1ccccc1OCCCC(=O)NC(c1nccs1)C1CCC1 27238,Cc1cc(C)c(C(=O)NC2(CNC(c3cnc(C(F)(F)F)nc3)=O)CCOC2)o1 27239,c1(OC)ncccc1-c1cn(C(C)CNC(c2occc2CO)=O)nn1 27240,c1(C(=O)NCC#CCC(=O)NCCC(COC)O)ccc2c(c1)CCC2 27241,C1(C(N2CC(C(=O)NC(C#C)CC3CCC3)(CC)C2)=O)CCCC(O)C1 27242,c1(C(N(C2C(N(C(C=C(COC)C)=O)C)CCCC2)C)=O)cnc2sccn12 27243,N1(C(C)C)CCN(C(=O)C(c2ccoc2)NC(=O)C(N2CCOC2=O)C)CC1 27244,CC(C)C(C(=O)NC1CS(=O)(=O)C1(C)C)C(C)NC(c1cncc(C#N)c1)=O 27245,C1(CNc2cccc(NC(=O)NC(=O)C3=NOCC3)c2)COc2ccccc2O1 27246,C(=O)(C(C)CC(N)=O)NCc1cn(CC2N(C(COCCOCC)=O)CC=C2)nn1 27247,C(=O)(C(C)CN(C(=O)CC1CNC(=O)O1)C)NC1CC(CSC)C1 27248,N1(C(C)C)CCOC(C(=O)NC2CCC(NC(=O)C(N3CCOCC3)C)CC2)C1 27249,C1(CC(N2CCC(CC=C)C2)=O)CN(C(c2cc(O)n(C)n2)=O)CC1C 27250,Cc1c(C(=O)NCC(C(C)C)NC(=O)COC(F)F)cnn1CCC(C)C 27251,CC(C)CCC(C)N=c1cc(NCc2c(Br)cnn2C)nc(C(C)C)[nH]1 27252,c1(C(N(CC(C)(C)CNC(C2(CC)CCCC2)=O)CC)=O)cc(C)cc(O)c1 27253,c1(C(=O)NC(C)CCCNC(=O)CC2CC2(Cl)Cl)ccc(N)cn1 27254,N1(C(c2cn(CC=C)nc2)=O)CC(NC(c2onc(CC)c2C)=O)CC1CO 27255,C=CC(C)C(C)C(=O)NCCCN(C)C(c1cncc(C#N)c1)=O 27256,C1(C)(N)COCCO1.c1(C(=O)NCCNC(C(C)(C)C)=O)ccccc1OC1CC1 27257,CC1(C(=O)NCCn2cnnn2)CC(O)CN1C(=O)Cc1nc[nH]n1 27258,Cc1cccc2cc(C(=O)NC3CCN(C(C4CC45CC(O)C5)=O)CC3F)nn12 27259,c1(CN2CCC(N(C(=O)CC3CCCCN3C)C)C2)n[nH]c2ccccc12 27260,c1(OC)ccc2ccccc2c1CNC12CC(NC(C3CC3C)=O)(C1)C2 27261,C1(C)(CNC(c2ccc(C#C)cn2)=O)CC(F)(F)CN1C(C1COC(=O)N1C)=O 27262,c1(OCC)ncccc1CN1CC2CC2(C(=O)NCc2ccccc2Br)C1 27263,C1(N(C)C(c2ccc(CO)nc2)=O)CCN(C(C2(C3CC3)CCCO2)=O)CC1 27264,C1(N(C(=O)CC2CCCC2)CC)CCCN(C(c2oncc2CC)=O)C1 27265,N12CCC(C(C)(C)C1)C2=O.C(C)(C)(CCC(=O)NCC1C2CCCC12)OC 27266,C(C)(C)(CCCCC(=O)NCC1C=CCN1C(=O)C=Cc1nc(C)c(C)[nH]1)OC 27267,N#Cc1ccc(S(N)(=O)=O)c(OCc2nnc3ccc(Cl)cn23)c1 27268,C1(O)(CCNC(=O)CNC(C2CN(C(C)C)C2)=O)CCN(C(c2cccs2)=O)C1 27269,n1(C(C)C)cnc(C(=O)NCC(C)(C)NC(=O)C(C)NC(c2cccs2)=O)n1 27270,C(C1CCCCCC1)=CC(=O)NCC1N(C(CCCc2onc(C)n2)=O)CC1 27271,C1(O)(CNC(CCCN(C)C)=O)CCCN(C(=O)CC2CCC(C)(C)CO2)C1 27272,Cn1cc2c(NC(c3ccc4occc4n3)=O)cc(C(F)(F)F)cc2n1 27273,N1(C(C2(COC)CN(C(C3CC(F)(CF)C3)=O)C2)=O)CCS(=O)C(C)C1 27274,CC1CN(C(c2c(C(C)(C)C)oc3ccccc23)=O)C2COCC2O1 27275,c1(-c2scc(CN3C(CNC(CCOCC)=O)CCC3)n2)cccc(OC)c1 27276,CC1(C)COC(C(=O)NC2CCC(CC(N3CCOCC3CO)=O)C2)C1 27277,C1(NC(C(C)CC2CCCC2)=O)CCN(C(C2CC(C)(F)C2)=O)CC1C 27278,c1(C(=O)NCCC(C)NC(c2cc(Cl)cnn2)=O)ccc2c(c1O)CCC2 27279,C=CCC(CC=C)C(=O)N1CCC(NC(C23CC(C#N)(C2)C3)=O)CC1C 27280,CC(C)C(CC(=O)N1CC2C=CC2C1)NC(c1cnn(C)c1C#N)=O 27281,N1(C(c2c(C)n(CC(F)F)nc2)=O)CCN(CC2CCC(C)C2)CC1C 27282,N1(C(C2CCC(=O)OCC2)=O)CC2(CCCN(C(C3CN4CCC3CC4)=O)C2)C1 27283,N1(C(COC2(C)CCC2)=O)CCOC(C(C)NC(c2ccc(C(N)=O)[nH]2)=O)C1 27284,C1(Cl)(CN(C(=O)Cc2cccn2C)CC#C)CCCCC1 27285,C1(NC(c2cc(COC)no2)=O)CCN(C(=O)C(F)(F)C(F)(F)F)CC12CCC2 27286,c1(C(N2CCC(F)(CNC(C(=O)NCC3CC3)=O)C2)=O)cccc2oc(O)nc12 27287,Cn1nc(C(=O)NC(Cc2ccccc2)CCO)c2c1CNCC2 27288,C(=O)(C1CCCn2cnnc21)NC1CC2CN(Cc3cccs3)CC2C1.O=C1CN1 27289,C1(CNC(c2cccc(OC)n2)=O)CN(C(=O)CNC(c2cscn2)=O)CCN1C 27290,C(CCCC(=O)NC1CC(CNC(c2cn(CCN3CCCC3)nn2)=O)C1)SC 27291,CC(C(=O)NC1COCCN(C(C2CN3CCN2CC3)=O)C1)S(C)(=O)=O 27292,C(CC(=O)NC(c1ccccc1C)C)(C(F)(F)F)NC(CC(C=C)C)=O 27293,CC1(C(=O)NCC2CCCC(NC(=O)CNS(=O)(=O)C3CC3)C2)CNC(=O)C1 27294,C1(CC=C)(C(=O)N(CC(C)NC(C2CCCN2CC(C)C)=O)C)CCCCC1 27295,c1(C(N2C(C3CC3)CCC2)=O)ccc(OC)c2ccsc12.CCC1CC(=O)N(C)C1 27296,c1(CN(CC(=O)NCC(C)(C2CC2)NC(C(C)=C(CC)C)=O)C)ccc(C)s1 27297,C1(CNC(Cc2c(C)non2)=O)CCCN(C(C2SCCS2)=O)CC1 27298,N1(C(c2c(C)ccc(N)c2)=O)CC2CC1CCC2NC(C1C2CC3C(C2)C13)=O 27299,c1(OC)ccc(O)cc1C(=O)NCC(C)CNC(=O)CC(C)F 27300,c1(N(CC(CNC(CC(COC)(C)C)=O)C)C)ncc2c(ncn2C)n1 27301,c1(N2CCN(C)C(CNC(c3cccc(C4CC4)n3)=O)C2)ncc(C#N)cc1F 27302,c1(SC)ccsc1C(=O)N(CC(=O)N(C1CCSC1)C)CC1CC1 27303,c1(CC(=O)NCCC(C)N(C(=O)Cc2cc(C3CC3)ccn2)C)ccc(Cl)cc1 27304,c1(C(N2CC(CC(=O)Nc3cncc(Cl)c3)OCC2)=O)cnn2ccccc12 27305,C1(CC(N2CCN(CCOC)C2)=O)COCCN1C(=O)COc1ccn(C)n1 27306,C(=O)(C#CC1CCCC1)N1CCN(C)C(C(N2CCC(F)(CF)C2)=O)C1 27307,N1(C(c2cc(C)sc2C)=O)CC2CCCC2(CNC(=O)CCCC(C)=O)C1 27308,Cc1[nH]c(C)c(C(=O)NCC(C)(C)CNC(=O)CC2CCC(C3CC3)O2)c1C 27309,c1(OC)ccc(CCC(=O)NC2CC(C)(NC(C3CCCC3(C)C)=O)C2)cc1F 27310,C1(NC(C=C(C)Cl)=O)CC1C1CCCN(C(=O)C(C)SC(C)C)C1 27311,N1(C(CC2C=CC(NC(c3ccn(CC)n3)=O)C2)=O)CCC2C(C(N)=O)C2C1 27312,Cc1cnn(CC(=O)NCC2CCN2C(c2c[nH]nc2-c2cccnc2)=O)c1 27313,c1(C(=O)NCCCN(C(c2nc(Cl)cs2)=O)CC)ccnc(C(C)(F)F)c1 27314,CC1(CCC(=O)NCC2CCC(=O)C2)CN(C(c2cnn(C(F)F)c2)=O)C1 27315,C(CCC(O)C(=O)NC1CCOCC1)NC(C(C)(C)C1CCCO1)=O 27316,N1(C(c2cc(CNC(C3N(C)CCCC3)=O)on2)=O)CC2(CNC(=O)N2)C1 27317,n1(CCOC)nc(C)c(NC(=O)C(N2CCC(C)(c3nc(C)no3)CC2)=O)c1Cl 27318,CCCCCCC(C)(CC)C(=O)NCC(CCCC)NC(c1ccc(O)nn1)=O 27319,S(=O)(=O)(c1ccc(NCCCCS(C)=O)nc1)N(C)Cc1cc(C)sc1 27320,Cc1ccc(C(N2CCSCC2C(N2CCC(OCC(C)C)C2)=O)=O)nc1O 27321,C(=O)(CCCS(C)(=O)=O)N(C)C(CC(CNC(=O)CCC1CCCC(=O)N1)(C)C)=O 27322,C1(CC(=O)NCCC(=O)NC)CCN(C(c2ncccc2Cl)=O)C1(C)C 27323,c1(C(N2CCOCC(C(=O)NCCC(=O)N(C)C3CC3)C2)=O)cccc2ccoc12 27324,C1(CC(=O)N(CC(O)CNC(=O)C=Cc2cccs2)C)CCC(F)(F)CC1 27325,c1(NC(C2N(Cc3ncc(C)cc3F)CC2)=O)ccc2c(c1)CCC2 27326,c1(C(N2CCC(N(C(=O)CC3C=CCC3)CC#C)C2)=O)ncc(OC)nc1OC 27327,C1(NC(CN(C(C)C)C)=O)(CNC(c2ccn(C3CCCCC3)n2)=O)CCOC1 27328,CCCCC(CC)C(=O)NC1(CCF)CC1.C12CCOC1C(=O)N2C1CC1 27329,c1(NCCN(c2nccc(NC3C(C)CSC3)n2)C)ccc(Br)cc1[N+](=O)[O-] 27330,CC1(C)OCCC1C(=O)NCCn1ccc(C(N2CCC3CC23)=O)c1 27331,C1(NC(C=CC)=O)CC=C(C(=O)NCc2cnc(CC)[nH]2)C1 27332,C(=O)(CC(C)(C)C(=O)N(CCCN(C(=O)C(C)CNC(C)=O)C)C)OC 27333,c1(OC)cc(Br)cc(I)c1NC(N1CCC(C(c2ccccc2)CO)CC1)=O 27334,C(CCCC)(C(=O)N1CCC(CC(=O)OC)C1)NC(CCC=CC)=O 27335,c1(C2(C(c3n(CC=C)nnn3)C3CCCC3)CC(CC)C2)cccc(Br)c1 27336,C1(NC(CCCOCC)=O)CC(NC(c2cc(C(N)=O)ccc2C)=O)C12CCC2 27337,c1(C(N2CCC(N(C(C34COCC3C4)=O)CC)C2)=O)ccc2c(=O)ccoc2c1 27338,C(=O)(C(C)CC(C)C)N1CCC(C(=O)NC2(C(=O)NC(C)C)CC2)C1C 27339,Cc1c(NC(c2oc(CNC(=O)CC3CCC(C)C3)nc2C)=O)cnn1C(C)C 27340,c1(C(CCC(=O)NCCN(CCCCCC2CC2C)C(C)C)C)ccc(F)c(F)c1 27341,C(=O)(CN=c1cc[nH]cc1)NCC(C)C(F)C(N1CC2(CCCN2C)C1)=O 27342,C1(CC=C)(NC(C)=O)CCCN1C(c1ncn(CC)n1)=O.C1(=O)CN1 27343,Cc1cccnc1C(C(C)C)NC(=O)CCC(c1ccc(F)cc1)=O 27344,c1(N2CCc3n(cc(C)n3)C2)nc2c(F)cccc2c(=NCCSCC2CCC2)[nH]1 27345,C1(NC(c2n(C)ncc2C2CCC2)=O)CN(c2ccncn2)CC1N=[N+]=[N-] 27346,Cc1cc(Cl)c(C(N2CCN(C(=O)CS(C)(=O)=O)CC2C)=O)c(Cl)c1 27347,C(C(C)(CCO)NC(=O)C(CCC1CC1)NC(c1snc(C)c1N)=O)OC 27348,c1(OCCC(=O)N(CCN=[N+]=[N-])CCOC)ccc(C)cc1Br 27349,C1(CNC(c2n(C)c(O)nc2)=O)CCCCCN1C(c1cc(Cl)cs1)=O 27350,c1(CNC(C=CCC2(NC(c3n(C)ncn3)=O)CCC2)=O)cc(=O)cc[nH]1 27351,CC1(C)CN(C(=O)OC(C)(C)C)CCC1O.C12=NNC(=NC(=O)N1)C=C2 27352,c1(C(N2CC3C(NC(C4C(CCC)C4)=O)(CC3)C2)=O)cc(S(C)(=O)=O)co1 27353,N1(C(CCC)C(=O)O)CCC(O)C(C(N2CCCC(C(=O)NCCO)C2)=O)C1 27354,c1(C(=O)NCC(CCOC)NC(C2(NC(C)C)CCC2)=O)cc(=O)n(C)o1 27355,CC(C)C(CNC(=O)COCCc1ccccc1)NC(=O)CCc1cc(Cl)no1 27356,c1(OC)cc(C(N2CCC(CNC(c3ccc(CF)cc3)=O)C2)=O)cc(F)n1 27357,C(=O)(C(C)CC(=O)OC)NC(CC=CC)C(=O)NC1(C(O)CO)CC1 27358,C1(C(=O)N(C)CC2CCCN2C)(COC)C=CCN1C(=O)CC1COCCOC1 27359,CCC(CC(=O)NC1CCC(NC(c2cc(F)cc(Cl)c2)=O)CC1)C(C)(C)C 27360,N(C1COc2ccccc21)C(CC1CCN(C(c2cnc(C)n2C)=O)C1)=O 27361,CCCC(C(=O)N(C(C(=O)NOCCCN(C)C)C1CC1)C)C(C)C 27362,Nc1c(C(=O)NC2CCCCC2NC(C2NC(=O)C3CC23)=O)cc(Cl)cc1F 27363,c1(CC(C)(CO)N(C(C)(C)Cc2ncc[nH]2)C)cccc(Br)c1 27364,C#Cc1cc(C(=O)N(C)CCNC(=O)Cc2ncn(C)c2C)cc(C(F)(F)F)c1 27365,C12(CC)CCC(C(=O)NNC(=O)NCC3=CCS(=O)(=O)C3)(C1)OC2 27366,N1(C(c2cc(C(C)C)nn2C)=O)CCN(C(=O)CCOCC2CC2)CC1C(C)C 27367,c1(OCC)[nH]c(=NC(=O)c2c[nH]c(=N)c(C)c2)ccc1Cl 27368,C1(CNC(CCC)=O)CCCC2CN(C(=O)CC3CCN(C)C3=O)CC12 27369,C1(COC)(NC(c2cc(-c3ccco3)on2)=O)CN(C(=O)CC(C)OC)C1 27370,c1(C(=O)NCC(O)CNC(C2(F)CCOC2)=O)ccc2ccccc2n1 27371,C1(CNC(CC(C)OC)=O)CC2(CCC2)CN1C(C1CN(CC(F)(F)F)C1)=O 27372,C1(C(=O)NCC2(CN(C(C3C(C)C3(F)F)=O)C)CC2)C(F)(F)C12CCC2 27373,c1(C(=O)NCCC2N(C(CC(C)C(F)F)=O)CCCC2)c([N+](=O)[O-])cnn1C 27374,CC1CCC(C)(C(=O)NCCOC(C)(C)CNC(=O)CCc2cc(Cl)no2)C1 27375,C1(C(=O)NC2COCCN(C(=O)Cc3ccoc3)C2)CC2(C1)CC(F)(F)C2 27376,CC1(C)CN(C(=O)CC2CCCCCO2)CC(CNC(=O)CC2CCCCCC2)O1 27377,c1(C(=O)NC)ccc(C(=O)NC2CN(C(C3COCCN3C)=O)CCC2F)cc1F 27378,C1(CNC(C2CCC(CC)O2)=O)CC2(CC2)CN1C(=O)CCCc1cnccn1 27379,C1(NC(C(=Cc2cccs2)C)=O)CCCCC12CCCN(C(=O)C(C)C)C2 27380,CCC(CO)CN=c1[nH]c(=NCc2cc(F)cc(Cl)c2)c2sccc2[nH]1 27381,C#CC(C)(C)C(=O)NCCCC1CN(C(c2ccc(CC(C)C)cc2)=O)CCO1 27382,c1(CCC(N2CC(CNC(=O)Cc3cscn3)OCC2)=O)cccc2[nH]ccc12 27383,c1(OC)cc(C(N2CC(NC(c3cnc(Cl)s3)=O)CC(F)C2)=O)cc(F)n1 27384,c1(C(=O)NC(CNC(C(C2CC2)SC)=O)CO)cc(C(F)(F)F)cc(Cl)c1 27385,c1(C(N2CC(NC(C(C)CC(N)=O)=O)(CO)C2)=O)cnc2c(c1)NC(=O)CO2 27386,c1(C(=O)NCC(CCCC)NC(C2CC2OCC)=O)c[nH]c2cc(F)ccc12 27387,Cc1cc(C(=O)NC2CCOC(C(=O)NC34CC(F)(C3)C4)C2)c(C)o1 27388,Cc1nc2c(o1)CCCC2CC(=O)N1CC2CCC1CN2CCCn1cncn1 27389,C1(C(=O)NCC2(C)CC3(CC3)C2)CCCCCCN1C(=O)CCc1ccco1 27390,C(=O)(CCCC(F)(F)F)NC(C1CCCN1C(c1cnoc1C1CC1)=O)C 27391,CC(CC(=O)NCCC1CN(C(=O)CNC(C2CCC2)=O)C1)C(F)(F)F 27392,C1(CNC(C(C)(C)C)=O)CCCC2(CN(C(=O)C3CC3)C2)O1 27393,C1(CC)CN(C(=O)CCC2CCCCCCC2)CCN1C(C1CC1C)=O 27394,c1(C(N2CCC(c3cccc(C)c3)C2)=O)cnc(Cl)cc1C(=O)NCCNC 27395,CC1CC(C)N(C(c2c[nH]nc2F)=O)CCN1C(c1cncc([N+](=O)[O-])c1)=O 27396,C1(CCC(=O)NC23CC(NC(C4CC4(F)Cl)=O)(C2)C3)CCCCC1 27397,c1(C(=O)NCC2N(C(c3cccc(OCC)c3)=O)CCC2)scc2c1OCCO2 27398,C1(NC(CCn2c(C)ccc2C)=O)CC(NC(=O)Cc2nc[nH]n2)C12CCC2 27399,N1(C(=O)OCC)CCN(C(=O)C(CNC(=O)C=C(C)C(F)F)N(C)C)CC1C 27400,N1(C(=O)Cc2ccc(Cl)nc2)CC(C(=O)NCC2CC23CCC3)C2(CC2)C1 27401,N1(C(CN(C(CNC(=O)OC)=O)Cc2ccco2)=O)CCn2cnnc2C1 27402,C12(NC(C3OCC(C)C3)=O)CCC(CC1)N(C(c1nccn3cnnc13)=O)C2 27403,N1(C(CSCC)=O)CCCC2CN(C(c3nccc(C)c3F)=O)CC12 27404,C(=O)(CCCCN=[N+]=[N-])N1CCCC(CN(C(C(C)Sc2nncn2C)=O)C)C1 27405,C(=O)(C(O)CC(=O)OC(C)(C)C)NCC1N(C(C(CCC)C)=O)CCCC1 27406,N1(C(C2C(C)(C)CC2)=O)CCCCC(CNC(c2cccc(F)c2N)=O)C1 27407,Cc1cccc(F)c1CNC(C1CCC2(CC2)N1C(C1(CO)CCC1)=O)=O 27408,Cc1nc(C(=O)NCC(C)(O)CNC(=O)Cc2nc(=N)[nH][nH]2)c(C)n1C1CC1 27409,CC(CC(=O)NC1CC(CNC(=O)CC2(CO)CC2)CC1O)P(C)(C)=O 27410,N1(C(C=CCCC)=O)CC(C(=O)NCC2(CN3CCCC3)CCCC2)CC(O)C1 27411,C(=O)(C(C)(C)CCCF)N1CCCC(N(C(C(c2ccc(C)cc2)C)=O)C)C1 27412,C(c1cccc(N)c1)=CC(=O)NCC(CNC(=O)CCN1CCOCC1=O)OC 27413,C(CCCCC(=O)NCC(c1ccc(F)cc1OC)NC(=O)CCC1CC1)=CC 27414,CC(=O)CCC(=O)N1CC=CC1(C(=O)N(CCc1csc(C)n1)CCO)C(C)C 27415,Cc1cn2c(CC(N3CCC(CNC(c4c(C)cccc4F)=O)C3)=O)csc2n1 27416,c1(CCC)c(NC(C2CC2NC(=O)NC(C)CN(C)C)=O)cccc1Br 27417,C(=O)(CCCCC(C)CC)N.C(=O)(CC(CC#C)C1CC1)NCCCOCC#C 27418,C1(C(=O)OC)CCC(NC(=O)CCCNC(C)(C)CNC(=O)C(C)(C)C)C1 27419,Cc1cc(O)cc(=O)n1CC(=O)NCC1CC2CN(C(C3(C)CCCS3)=O)CC12 27420,c1(C(N2CC(NC(C(C(CC)O)(F)F)=O)C(C)C2)=O)cc(S(N)(=O)=O)oc1C 27421,C1(C(=O)NCCC=CC(=O)NC2C(CCOCC)C2)COCCN1CC 27422,Cc1cnc(Cl)cc1NC(C1CCCN(C(c2cccnc2C)=O)C1)=O 27423,c1(OC)ccc(F)c(C(=O)NCC2CCCN2C(C2CCC(C)(C)OC2)=O)c1F 27424,N1(C(C2C(C#C)C2)=O)CCN(C(=O)CSCc2ccccn2)CC(C)(C)C1 27425,c1(C(N2CC(CN(C(=O)C(O)C(C)(C)C)C)OCC2)=O)ccccc1C#N 27426,C1(C(=O)NC(CC=C)CNC(=O)CCS(C)(=O)=O)C2CCC1(C)C2(C)C 27427,c1(C(N(C)CC2CCCN(C(C(C3CCC3)OCC)=O)C2)=O)ncnc(O)c1F 27428,N1(C(c2nc(C)[nH]n2)=O)CCCCC(CNC(c2nc(C)nn2C)=O)CC1 27429,c1(N(C)CC2(CC)CC(F)(F)C2)nc(N(C)C(C)C)nc2c1SCC2 27430,C12(CNC(C3(C)C(C)C3)=O)CC1CN(C(=O)CCOc1cccc(Cl)c1)C2 27431,C(=O)(CN=c1cc[nH]cc1)N(C)CCN(C(=O)CC1CCCCO1)C 27432,c1(OC)ccc(C(=O)N(CC(C)N(C(=O)Cc2ccoc2C)C)C)nc1 27433,C1(C(=O)NCC(C)S(N)(=O)=O)C(C)OCCN1C(C1CN(C)C1)=O 27434,Cc1nc(CO)ncc1C(=O)NC1CN(C(=O)C(C)(C)F)CCC1C 27435,N1(C(COCCCOC)=O)CCCC(NC(c2cc(CO)on2)=O)C1C 27436,C(=O)(C(F)C(C)CNC(C1C=CCCC1)=O)NCC(N1CC(C(CC)CC)C1)=O 27437,CC1CN(C(c2ccc(-c3ccco3)s2)=O)CC(C)C1NC(=O)CCC1CCC1 27438,C1(Cc2cc(OC)on2)NC(=O)N(CCC23CCCC2C3)C1=O 27439,Cn1c(C(=O)NC2(CNC(=O)CS(C)(=O)=O)CC(F)(F)C2)cc2sccc12 27440,c1(C(=O)NCC2(F)CN(C(=O)C(F)F)C2)c(C(F)(F)F)cncc1F 27441,Cn1ncc([N+](=O)[O-])c1C(=O)NCCC12CC(NC(C3CCC(C)(C)C3)=O)(C1)C2 27442,C1(NC(c2c(CC)con2)=O)CC(CC(=O)NCc2[nH]ccc2C2CC2)C1(C)C 27443,N1(C(C(CCCC)C)=O)CCC2CCN(c3ncncc3C)CC2C1 27444,c1(C(C)C)nc2ccc(NS(=O)(=O)c3cc(Cl)sc3Cl)cc2s1 27445,C1(NC(COCc2cc(C)no2)=O)CC(F)CN(C(=O)CCn2cncn2)C1 27446,c1(C(=O)NC(C2CCN(C(C(CSC)(C)C)=O)CC2)C)[nH]c(C)c([N+](=O)[O-])c1C 27447,C1(N(C(=O)CC(F)(F)F)C)CC2CCC(C1)N2C(=O)CC1=CCCCC1 27448,C12(NC(c3coc(CO)c3)=O)CCN(C(c3cc(C(F)(F)F)c[nH]3)=O)CCC1C2 27449,Cc1c(S(N)(=O)=O)sc(C(=O)NCCN(C)C(C2(CN(C)C)CC2)=O)c1Cl 27450,c1(C(N2CCC(C)(O)C2)=O)cc(-c2ccco2)cc2[nH]ncc12 27451,C1(C(N2CCC(F)(CNC(=O)CCc3cncnc3)C2)=O)CC2C=CC1CCC2 27452,N1(C(=O)Cc2c[nH]c3cccnc23)CC2CC(N=c3ccnc(Cl)[nH]3)C2C1 27453,c1(CNC(=O)Cc2ncc(Cl)s2)nc(CNC(=O)C(F)CC2CCC2)cc(O)n1 27454,C(=O)(C(C(C)CC1CCC1)N1CCC(C2OCCO2)C1)NCCC 27455,n1(CC)ccc(C(=O)NCC2CN(C(c3ncc(F)cc3N)=O)CC2C)cc1=O 27456,c1(C(N(C)CC2CN(C(c3cc(O)cc(F)c3)=O)C2)=O)ccc(=O)n2c1CCC2 27457,CC(C)C(CCN(C)C(C1CCCC(=O)N1)=O)NC(=O)C(C1CCCCCC1)C 27458,c1(C2C(=C)C2)cccc(N)c1.N(C(=NC)NCC(F)F)C 27459,CC(F)(C(=O)NC1CC2CC(C1)N(C(=O)Cc1cc[nH]n1)C2)C(F)(F)F 27460,C1(C(=O)NC(C2CN(C(C3CCCS(=O)(=O)C3)=O)C2)C)CCC2CC(C)CN2C1 27461,N1(C(C2COCC(C)O2)=O)CCCC(O)(CCNC(=O)C(C)(C)CC2CC2)C1 27462,S1(=O)(=O)c2ccc([N+](=O)[O-])cc2N1.C(=O)(C=CCOC)OC 27463,N1(C(C(C)NC(=O)NCCNS(C)(=O)=O)=O)CCc2ccsc2C1 27464,N1(C(c2nnc(C(C)C)s2)=O)CCC2CN(C(=O)C(C)C3CCC3)CC2CC1 27465,c1(C(=O)NC(C2(O)CCCCC2)C(=O)NCC(C2CC2)OCC)c[nH]ccc1=O 27466,N1(C(CSCC(=O)OC)=O)C(C(=O)NCc2conc2C(C)C)CC2CCCC12 27467,c1(NC(C2(CC=C)CCN(C(=O)C=CC(C)CC)C2)=O)ccc(OC)c(OC)c1 27468,C12(C(=O)OC)CC(OCCO)C1C2.c1(CO)ccccc1 27469,N1(C(c2c(CN(C)C)cccc2)=O)CCN(C(C2(C(C)(F)F)CC2)=O)CC12CC2 27470,c1(CC(=O)NCc2cccnc2Br)n[nH]c2cc(C3=CCCCC3)ccc12 27471,C(=O)(C1=CC2CCCCCCC12)N1CC(O)(CNC(c2cc(=N)[nH]c(Cl)n2)=O)C1 27472,Cc1cccc(CC(=O)N(C2CCC(NC(C3CSCN3C(C)C)=O)C2)C)c1F 27473,Cc1nocc1C(=O)NCC(C1CCCC1)NC(=O)C(C)c1cccs1 27474,N1(C(=O)CCCCN2CCCCC2)CNS(=O)(=O)c2cc(Br)ccc21 27475,N1(C(Cc2cc(CC)nn2C)=O)C2CCC1C(NC(=O)C(C)OC1CCCC1)C2 27476,S(=O)(=O)(c1ccc(CCC(=O)O)cc1)N1CCC(C)CC1C(N)=O 27477,CCCCC(F)C(=O)N1CCCCC(C(=O)NCCc2ccc(C)c(C)c2)C1 27478,N1(C(c2cnc(C(C)C)s2)=O)CCCC2(CC(NC(=O)CC(F)(F)F)CO2)C1 27479,N1(C(C=CC)=O)CC2CCCC2C1C(=O)N(CCCCCC)C 27480,C1(NC(CC2CCN(C)C2)=O)CCC(C)(NC(c2cc(N)cc(N)c2)=O)CC1 27481,C(c1ccccc1SC=O)=CC(=O)NCC1(NC(COCC)=O)CC1.C(F)(F)F 27482,c1(C(N2C(C)(CNC(c3cc(OCC)n[nH]3)=O)CCC2)=O)c(C)nn(C)c1F 27483,CC1CCC(CS(=O)(=O)Nc2nn(C)c(=O)n2C)CC1C 27484,N1(C(CNC(=O)OC)=O)CC(CNC(=O)CC(C)C(F)F)C(F)(CO)C1 27485,C(=O)(C(O)CC(C)C)NC1(CCNC(C(c2ccc(CCCC)cc2)C)=O)CC1 27486,C1(C(=O)NC2(COC)CC2)CC12CCN(C(c1ccc(NC(C)=O)cn1)=O)CC2 27487,CCC(C)C(O)C(C)C(=O)NC1(C(=O)NOCCc2ccccc2)CCC1 27488,C(C)(C(C(=O)NCCc1ncccc1C)C(C)C)NC(c1ccnc(C)n1)=O 27489,Cn1ncc(C#N)c1C(=O)NCc1ccnc(C(N2CCC(CO)C(O)C2)=O)c1 27490,C1(CC)CC(C(=O)NCC(C)N(C(=O)C(F)OC)C)CC(=O)N1 27491,NS(=O)(=O)c1csc(C(N2CCC3C(NC(=O)CCCn4cncn4)CC23)=O)c1 27492,c1(CC)cc(C)c(C(=O)NCC(C)(C(C)C)NC(=O)Cc2cscn2)o1 27493,c1(C(=O)NCC(C2CC2)NC(C(OCC)OCC)=O)cc(CF)on1 27494,N1(C(C(CCC)OC)=O)CCN(C(c2cnc(O)o2)=O)CC(CO)C1 27495,c1(NC(C)C(=O)NCC=CCOC=O)ccc[nH]1.C(COC(C)(C)C)=CBr 27496,C(CC(=O)NCC1CN(C(=O)CN2CCCNC2=O)CCO1)(C(C)C)OCC 27497,c1(OC)ccc(NC(C2(CCNC(=O)C=CC(F)(F)F)CCC2)=O)c(F)c1 27498,C1(CC)CCN2C1C(=O)N(C)C(=O)NCCC2=O.c1(CNC)scnc1C 27499,N1(C(c2c(SCC)cccn2)=O)CCN(C(=O)CCc2ncccc2Cl)CC12CC2 27500,c1(C(N2CC(CCC)C(C(=O)NC3CCSC3)C2)=O)ccc(=O)n(C)n1 27501,c1(C(=O)NCC(=O)N(C(CCNC(C(C)OC)=O)C)C)cccc(F)c1 27502,c1(C(=O)NCCC2N(C(C3CC=C(C)CC3)=O)CCOC2)cc(C)c(C)cc1C 27503,CCCC(C(=O)N1CCOCC1CCNC(C1CS(=O)(=O)C1)=O)OC 27504,CC1CC(C(=O)N2CCC(N(C)C)(CNC(C3(C)CC(O)CN3C)=O)C2)=NO1 27505,N1(C(C=CSC)=O)CC(C)CN(C(=O)C(c2cccc([N+](=O)[O-])c2)C)C(C)C1 27506,c1(C(=O)NCC(=C2CN(C(Cc3cccc(C)c3)=O)C2)F)[nH]c(C)c(C)c1C 27507,C(=O)(C1=CCCCO1)NCCCCCNC(=O)Cn1ccc(C(F)F)n1 27508,Cc1cccc(CNC(=O)CC2CCN2C(=O)CSC(C)(C)C)c1F 27509,CC1(CNC(=O)C(O)C2CCC2)CCCN(C(=O)C=CC2CC2)C1 27510,C(C(C(=O)N(C(C)C(C)(C)C)C)C(C)(C)C)NC(c1n(C=C)ncc1)=O 27511,C(=O)(C1=COCCC1)N(C1(NC(c2ccccc2F)=O)CC(O)C1)C1CC1 27512,CC1CN(C(c2nnn(C)c2N)=O)CCN1C(c1cccc(CCN(C)C)c1)=O 27513,C(=O)(C1CCc2c(Cl)cccc21)NCC(CCCC)NC(=O)CS(=O)(=O)C1CC1 27514,C#Cc1cc(C(=O)NC2CCC2C(=O)NC(C2(O)CCCCC2)C)ccc1C 27515,N1(C(C2(OCC)CCOC2)=O)CCC(C(N2CC3CC=CC2C3)=O)C(O)C1 27516,N1(C(c2nc(CCC)oc2)=O)CC2(CCN2C(C2C(C#N)C2(C)C)=O)C1 27517,Cn1ccc2cc(C(N3CCCCC(N4CCCC4)C3)C(=O)NCCO)ccc12 27518,C(=O)(C(F)CCC(C)C)N1CCC(NC(C=CCC=C)=O)CC1C1CC1 27519,c1(C(c2n(CC=C)nnn2)NCCC2CC3(CCC3)O2)nc(C)c(C)s1 27520,N1(C(C(CCC)C#N)=O)CCCC(C)(C)C1C(=O)NCC1CC(CC)C1 27521,C1(C(N2CCC(NCC)C2)=O)CC(=O)N(C2CCCCCC2)C1 27522,N#CCCCC(=O)N1CCCC1C1CCN(C(C2(C(=O)NC3CC3)CC2)=O)CC1 27523,Cc1cc(C)n(CCNC(C2CN(C(C)C(=O)NCC3CCCO3)CCO2)=O)n1 27524,c1(C(C(=O)NC(C)C)N(C)Cc2nc(C(=O)OC)nn2C)ccc2nonc2c1 27525,C12(CNC(c3cc(C)ncc3)=O)CCC(CNC(c3cscc3Cl)=O)(CC1)CO2 27526,N1(C(c2ccsn2)=O)CC2C3CCC(C2C1)N(c1nccc(Cl)c1O)C3 27527,c1(CNC(c2ccc(C#C)o2)=O)nc(CNC(=O)CC2CC(C)C2)cc(O)n1 27528,c1(CN(C(N(CCOC)CCN2CCCC2)=O)C)cncc(OC)c1 27529,N1(C(c2cc(C)c(C#N)cc2)=O)CCC2CN(C(=O)CCP(C)(C)=O)CCC2C1 27530,c1(CC(=O)N(CCCNC(C2(CCC)CC2)=O)CC)c(CC)noc1CCOC.CCC 27531,C1(C(=O)NC(C(C)NC(C2CCCSC2)=O)C)CC2C=CC1CC2 27532,c1(C(=O)NCC2CN(C(CC(=O)NCCOC)=O)CC2C)cc(N)c(C)cc1C 27533,c1(SC(C)C)ccc(C(=O)NCCOC2CN(C(=O)C(C)N(C)C(C)C)C2)cc1 27534,C12(C(=O)OC)CCC(CC1NC(=O)CSc1cccc(N)c1)C2(C)C 27535,N(C1CCCn2ccnc21)C(c1cc(CNC(Cc2ccc(C)o2)=O)ncc1)=O 27536,C1(NC(=O)CCn2cc(Cl)cn2)CC2CCC1(NC(C13CCCC1C3(F)F)=O)C2 27537,CC(C)CC(CCCC#N)O.N1(CCO)CCCC1CC(F)F 27538,CCCC(O)C(=O)N1CC(CNC(=O)C(C)OCCC(C)C)C1 27539,C1(C)(COC)CC(NC(=O)CC(C)(C)O)CN1C(=O)CCc1cnn(C)c1 27540,c1(C(N2CCC(NC(c3c(C)cns3)=O)C2C2CC2)=O)cc(S(N)(=O)=O)c[nH]1 27541,c1(NCC(C)(C)n2ccnc2)[nH]c(=NCC2CCC(CO)O2)nc2scnc12 27542,N1(C(=O)NC(c2c(C)cccc2)C)CCCCC1(C(C)C)C(=O)O 27543,C(=O)(CC(C(F)F)NC(=O)C(C)(C)CCSC)NCC1(CCC)CCC1 27544,C1(CC(=O)N(CCCS(N)(=O)=O)C)CCC1C1CC1 27545,Cc1ccc(Cl)cc1C(=O)NC1COCCC1NC(=O)CC1(O)CCCOC1 27546,C12(NC(C(C)n3ccnn3)=O)CC(C(=O)NCCC(F)(F)F)(C1)C2 27547,Cc1cnc(C(=O)NC2CCCN(C(=O)C(C)NS(C)(=O)=O)CC2)c(C)c1 27548,N1(C(C(C(C)C)SC)=O)Cc2ccnn2CC(NC(c2cc(C)ccn2)=O)C1 27549,Cc1c(C)c(C)c(C(=O)N(C)CC2CN(C(=O)CC3CCNC3=O)C2)c(C)c1C 27550,C1(CSC)CC(N(C(CC2(C(=O)N(C3CCC3)C)CC2)=O)C(C)C)C1 27551,C1(NC(C(=O)C(=O)Cc2ccccc2OC(F)F)=O)CS(=O)(=O)C12CCCOC2.OC 27552,CC1CN(C(=O)CC2(O)CCCCCC2)CCN1C(C1COC(=O)O1)=O 27553,C1(N(C(=O)Cc2cscn2)C)CCN(C(C2(NCCN(C)C)CC2)=O)C1 27554,C1(C(=O)NC(C)CN(C)C(c2cnn(C)c2Br)=O)C2CCC1(C)C2(C)C 27555,N1(C(C=NOC)=O)CCOC(C(C)NC(c2csc(C(F)F)n2)=O)C1 27556,c1(C(=O)NC2(C)CC(NC(C3CC(C#N)C3)=O)C2)ccc(-c2cc[nH]n2)cc1 27557,c1(C(=O)NC2C(C(N(CC(F)(F)F)C(C)C)=O)CCCC2)cc(O)cc(F)c1 27558,c1(C(C)C)ccc(C(N2CC(C(C)NC(c3cnoc3C3CC3)=O)C2)=O)s1 27559,c1(CNC(N2CCCC2C2CCOCC2O)=O)c(O)cccc1Br 27560,C1(NC(=O)CCCCc2cnn[nH]2)CC2CCC1N(C(c1ccc(=O)oc1)=O)C2 27561,C1(CC(=O)N(C2CC2)CC2N(C(c3ccc(OC)cn3)=O)CC2)CC2C=CC1CC2 27562,N1(C(c2c(C)c(=O)cc[nH]2)=O)CCC12CCOC(C)(C)C2 27563,Cc1nn(CC(=O)NC(C)(CNC(C2CC3(CCC3)C2)=O)C2CC2)c2ncccc12 27564,N1(C(C(=O)NCCOC)=O)CC(NC(C2CC23CC(F)(F)C3)=O)CC(C)(C)C1 27565,C1C(C(C)(C)C)C(=O)N1.C(CCCCC(=O)N1CCC1N1CCOC1=O)OC 27566,N1(C(CC(COC)C)=O)CCC2C(NC(c3cc(N)cc(F)c3)=O)C2C1 27567,C1(CNC(c2ccn(CCCC)n2)=O)CC(NC(C2CC2F)=O)CC1O 27568,C12(NC(c3cc(C)c(O)cc3)=O)CCCC1N(C(c1cc(O)nn1C)=O)CCC2 27569,N1(C(C(C)c2ccsc2)=O)CC(CC(=O)NC2CN(C(C3CCC3)=O)C2)CC1(C)C 27570,CC(C)CC(CCO)CN=c1cc(NCC2CCC(F)(F)C2)nc[nH]1 27571,N1(CC(=O)N(CCCC)CCCC)CC(OC)CC(OC)C1 27572,N1(C(C(C)CF)=O)CC(C2CCN(C(C3(CO)CCC3)=O)CC2)C1 27573,C(=O)(CC(C(=O)N1CCOCC1N(C(=O)CC(=O)N(C)C)C)N(C)C)OC 27574,c1(C(N(CC(CNC(c2c(C)nns2)=O)O)C)=O)ccc2c(F)cc(F)cc2n1 27575,c1(CC)cc(C(N2CCC(NC(c3occc3C3CC3)=O)C2C)=O)nn1C 27576,c1(C(N2CCC3(NC(=O)CCCCC4CC4)C(C2)C3)=O)ccc2nnc(S)n2c1 27577,C(=O)(C#CC1CCOCC1)N1CCC(=C)CC1C(=O)Nc1cnccc1SC 27578,C1(NC(c2c(OC)n[nH]c2)=O)CC1C1CCN(C(=O)Cc2cnc[nH]2)CC1 27579,C12CC(=O)N(C1)C2.c1(CC(=O)N(CC(C)C)CCC)ccc(Cl)s1 27580,c1(NC(C(CC)(C)C)C)ccc(C(N)=O)c([N+](=O)[O-])c1.C(C(O)COC)S 27581,n1(CC(=O)NC(CCNC(CC(C=C)CC)=O)C)ccc(=O)n(C)c1=O 27582,N1(C(c2cc(OC)n[nH]2)=O)CC(C(=O)NC23CC(F)(C2)C3)C2(CCC2)C1 27583,N1(C(C2CCCCC(=O)N2)=O)CCC(C2CCN(C(=O)CC(O)C3CC3)CC2)C1 27584,Cc1ccc(NC(C2CCCCC2CN2CCC(C(N)=O)CC2)=O)nn1 27585,c1(C(=O)Nc2nc(SCC)nc(Cl)c2)cnc2[nH]cnc2c1 27586,N1(C(C=C)=O)CCOCC(CNC(C2CCCN2C(=O)C(F)(F)F)=O)C1 27587,c1(OC)cc(OC)c(NC2CCCN(CC(F)(F)F)C2)c(OC)c1 27588,C(CC)(C(=O)NCC(C)(O)CNC(=O)CCOCC(F)(F)F)OCCOC 27589,C(=O)(C1COc2ccc(F)cc21)N1CC2CCN(C(C(COC)(C)C)=O)CC2C1 27590,N1(C(C2(CC)CCCC2)=O)CCC(C2(NC(C3COC4(CCC4)C3)=O)CC2)CC1 27591,C1(C(=O)N(C2C3CCCOC23)c2cccs2)COCCN(C(=O)CC2CC2)C1 27592,Cc1cnc2n1CCCC2C(=O)NC1CCCC1NC(c1cncn(C)c1=O)=O 27593,c1(CCCC)nc(C)c(C(=O)NCc2ncoc2CCNC(=O)CO)s1.C1(C)CC1 27594,C1(OCC)CCN(C(=O)CC2(C)CCN2C(=O)CC2CC(OC(C)=O)C2)CC1 27595,c1(OC)ccc(C(=O)NC2(C)CCCN(C(C3(CN(C)C)CC3)=O)C2)cc1Cl 27596,N1(C(C(CC)CO)=O)CCN(C(C2CC(=O)NC2(C)C)=O)C(C)C1 27597,N1(C(=O)CC2(CO)CCCC2)CCC2(CCC2)C(NC(C2CC3C=CC2C3)=O)C1 27598,N1(C(C2N(C(C(CC)SC)=O)CCC2CC)=O)CCC2C(O)CC12 27599,c1(C(=O)NCC2CCC(C(N3CC4(CCOC4)C3)=O)O2)nccc2cc[nH]c12 27600,c1(C(=O)NCCN2C(CCC)CCC2)c[nH]c2cccc(Cl)c12 27601,C12(C(=O)NCC3N(C(C4SCCCS4)=O)CC(F)C3)CCCC(CO1)C2 27602,CC(C)(C)CC(=O)N1CCSCC1C(=O)NC(CO)C(N)=O 27603,C(=O)(C(C)S(C)(=O)=O)N1CCN(c2cc(C=CCOC)sn2)CC1 27604,c1(C(=O)NC2CC(N(C(=O)CC3CCCO3)C)C2)cnc2c(c1)CCOC2 27605,C(=O)(C(C)CC(C)(C)C)NC(c1ccc(F)cc1)CNC(c1onc(C)c1C)=O 27606,c1(C(C)C(=O)NC(C)(C)CNC(C2(C(C)(F)F)CC2)=O)cncc(F)c1 27607,C1(O)(CN(C)C(c2cnnn2C)=O)CCN(C(=O)CC2CCCN2C)C1 27608,N1(c2ncnc3n[nH]c(C)c32)CCC2CC(NC(c3ccno3)=O)CCC2C1 27609,Cc1cncc(CC(=O)NC2(CC(=O)NC3CCSCC3)CCCCC2)c1 27610,c1(C(=O)NCC2OCCN(Cc3c(C)ccs3)C2)cccc2c1COC2(C)C 27611,C1(C(=O)NCC#CCNC(C2C(C)(C)COC2)=O)CCC2(CCC2)C1 27612,C(=O)(CC1=CCOCC1)N(CCCC(=O)N(C1CCN(C2CC2)C1)C)C 27613,C(CC)(C(=O)N(CCC(O)CNC(c1cc(-c2ccco2)c[nH]1)=O)CC)OCC 27614,c1(CC)cc(C(=O)N(C(C)CNC(C2(c3ccccc3)CCCC2)=O)C)c(C)o1 27615,N1(C(C2CC(CNC(C3(O)CCCCCC3)=O)C2)=O)CCCCC(F)(F)C1 27616,CC1CN(C(=O)CC2CCC(=O)NC2=O)CCN1C(C1(NC(N)=O)CC1)=O 27617,C=CCCC(C)(C)NC(c1nnnn1CCOC)(C1CCCCC1)CC 27618,c1(C(=O)NCC2N(C(Cc3nnc(C)s3)=O)CC(O)C2)cnn2cnnc2c1 27619,c1(C(=O)NC(C(C)NC(C2CNC(=O)C2)=O)CO)cnc2nccn2c1 27620,c1(C(=O)NC2(CO)CN(C(Cc3c(OC)ccc(F)c3)=O)C2)cc(F)c(O)c(Cl)c1 27621,C12(NC(CCCCC=CC)=O)COCCC1CN(C(=O)Cn1nc(C)nc1C)C2 27622,c1(-c2cccc(Sc3cc(C4(N)CCOC4)ccc3F)n2)cc2ncccc2o1 27623,c1(C(N2C3C(C(N4CCN(C)CC4)=O)C(C3)C2)=O)ccc2[nH][nH]c(=N)c2c1 27624,C1(NC(c2cc(C)[nH]n2)=O)CCCC(N(C(=O)C(F)=CC2CC2)C)C1 27625,C1(NC(c2noc(CC)c2C)=O)CN(C(c2c(C)noc2N)=O)CC1S(C)(=O)=O 27626,C(=O)(C1CSc2ccccc21)N1CCC(C(C)NC(c2ccnnc2Cl)=O)CC1 27627,Cc1cc(NC(=O)CC2CCCN(C(=O)CC(O)C(C)C)CC2)cc(Cl)c1 27628,c1(C(N2C(C(=O)NCCSCCC=C)CCC2)=O)cccc(=O)o1 27629,N1(C(c2cc(C)n(C)c2)=O)Cc2[nH][nH]c(=NC(=O)C3CC4CCC3O4)c2C1 27630,N1(C(C(COC)NC(=O)C(SC)SC)=O)CC(C2CCCCC2)C1 27631,C1(COC)(N)CCOC1.N12CCC(C1)C2=O.c1(CCC(=O)NC)cnc(C)o1 27632,c1(C(C)(C)NC2CN(C(CC(C)(C)C)=O)C2)ccc(OC2CCCCO2)c(F)c1 27633,c1(CC)c(C(=O)NC(C)CCN(C)C(C2CCOC2)=O)nnn1CC 27634,C1(CCNC(CN(C2CC2)CC)=O)(NC(=O)CCc2csc(=N)[nH]2)CCCC1 27635,c1(C(=O)NCC2CC2(F)F)cc2n(n1)CC1(CC1)C2 27636,C1(N(C)C(C2CCC(=O)C2)=O)CCCN(C(=O)CSc2nnc(S)s2)CC1 27637,c1(C(=O)NC2CN(C(C3(C)CC3(F)Cl)=O)C2)cccc(NC(N)=O)c1 27638,C1(C(CC)NCC2CNC(=O)C2)CCN(Cc2ccc(C)o2)CC1 27639,C(C)(C)(C(C)(C)O)N(C(C(n1c(C)ccn1)C)=O)C(CC12CC(COC)(C1)C2)=O 27640,C1(C(=O)NC2CC3CN(C(c4ccc(C)o4)=O)C2C3)CCn2nncc2C1 27641,C=C(CNC(=O)CC1CCCC(NC(C2CC2(Cl)Cl)=O)C1)C1CCOCC1 27642,C1(C(=O)OCC)(NC(c2ccc(Br)cc2)C2CC2)CCOCC1.C1C(=O)N1 27643,N1(CC(=O)N(C2CCCCN(C(CCOCC)=O)C2)C)CCc2ccccc21 27644,c1(C(C2CCOCC2)(CC)NC(C=C)COC)nnnn1CCCOCC1CC1 27645,C1(C(N(CC#C)CCOC)=O)(NC(=O)Cc2ccccn2)CC1(C)C 27646,N1(C(c2n(C(C)C)ccn2)=O)CCN(C(C2CC3CCCCC23)=O)C(C(C)C)C1 27647,C1(C(=O)NCC(N2CC=CC2)C)CSCCN1C(=O)C(=O)NCC(F)F 27648,c1(C(=O)NCCCN(C)C(C2(n3cncn3)CC2)=O)cn(CC(N)=O)nn1 27649,N1(C(C(CCC)(C)CCC)=O)CCC2(CC1)CC(NC(C1CC(=O)N1)=O)CCO2 27650,C(=O)(C(CC=C)CC(C)C)NC(CC#C)CC(=O)NC1COCC1SC 27651,CC1(C)CC(CNC(=O)CC2(CO)CC2)CN(C(=O)C(=O)Cc2ccccc2)C1 27652,C1(NC(C2C(C)CCC2)=O)CC(=O)N(C2CN(C(C3(CC4CC4)CCCC3)=O)C2)C1 27653,N1(C(C2(OC)CCCCC2)=O)CC(C)CN(C(c2cccc(=O)n2O)=O)C(C)C1 27654,N1(C(=O)CCc2cncs2)CC2CC1CN2C(C1C2(CC2)C12CC2)=O 27655,c1(C(N2CCC(C)(NC(C(CC=C)C)=O)C2)=O)c(C)ccc2ncccc12 27656,C1(SCC(N2C(CNC(C3(C)CCCC3)=O)CC2)=O)CCS(=O)(=O)C1 27657,c1(C(N2CC3CC(NC(c4c(O)cc(C)nn4)=O)C3C2)=O)ccc(C#N)nc1C 27658,C1(CN(C)C(C2CCCCO2)=O)CCCN1C(=O)CSC(F)F 27659,N1(C(c2c(OC)c(F)ccc2)=O)CCC2CN(C(=O)CCC(C)N(C)C)CC12 27660,c1(OC)ccc(C(=O)Nc2ncoc2-c2cccs2)c(Br)c1 27661,C1(C2CCN(C(=O)CS(=O)(=O)N(C)C)CC2)(N(C(C(C)SCCCC)=O)CC)CC1 27662,C(=O)(C1=C(Cl)CCC1)NC(C(=O)N(C)CCc1cccs1)CCF 27663,c1(OCC)cc(F)c(F)cc1C(=O)NC1CC(NCc2c(F)ccc(C)c2Cl)C1 27664,N1(C(C(C(=O)OC)OC)=O)CC(F)(F)CC1CNC(C1CCCN(C(C)C)C1)=O 27665,C#CC1CN(C(c2cccc(C)c2)=O)CCN1C(=O)CCNC(=O)C=CCl 27666,C1(C(=O)NC2(C(=O)NCC=C=C)CC2)CCNC1=O 27667,C(=O)(C(C)(C)C(C)O)Nc1cccc(-c2cn(C(C)C(=O)O)nn2)c1 27668,C(=O)(C(C(C)NC(=O)CC(C)F)C(C)C)N(c1onc(C)n1)C(C)C 27669,c1(CNC(C2CNCCN2Cc2ccc(Br)c(Cl)n2)=O)ccc(O)c(O)c1O 27670,CN1C(=O)NC2(CCC(NC(c3ccc4nccnc4c3)=O)CC2)C1=O 27671,C(=O)(C(CC)CC(F)(F)F)NCc1cccc(CN(C(CCC(=C)C)=O)C)c1 27672,c1(COCC(=O)NC2CN(C(C(C)OCCOCC#C)=O)C2)ccc(C)nc1O 27673,c1(NC(C)=O)nc(-c2ccccc2)sc1C#N.N12CCN(CC1)CC=CC2 27674,CC1CC(CNC(=O)CCc2cnn[nH]2)CN(C(=O)C2=CSCS2)C1 27675,c1(NS(c2c(C)ccc(C)c2)(=O)=O)ncc(S(=O)(=O)N(C)CC2CSC2)cc1Cl 27676,CC1(C)CC(C(=O)NC2CCCNC2=O)CN1C(c1ccc(F)c(O)c1)=O 27677,Cc1nccc(C(N2CCN(C(=O)C(O)Cc3cnc[nH]3)CC2C)=O)c1N 27678,C1(C(=O)NCC2(CCO)CC2)(CNC(=O)CC2CC3CC3C2)CC12CCC2 27679,Cc1[nH]c2ccccc2c1CC(=O)NC1(O)CCN(C(=O)CSCC(N)=O)CC1 27680,c1(NC(=O)NC(c2cn3cccnc3n2)C)c(F)cc(C(N)=O)cc1F 27681,c12nc(nn1C1CCOC1(C)C)-c1cc(ccn1)C2.n1(CC=C)cc(Br)cn1 27682,C1(COCC(=O)NC(C)CC2CN(C(C3CC(F)C3)=O)C2)CCCCO1 27683,c1(C(=O)NC2C(CO)CCN(C(C(C)OCC=C)=O)C2)cc(OC)c(N)cc1F 27684,C1(C(N(CCCNC(C2(N(C)C)CCCC2)=O)C2CC2)=O)CCC12CCC2 27685,Cc1[nH]nc(C(F)(F)F)c1C(N1CCC(CCNC(=O)CC2CCCC2C)C1)=O 27686,c1(CC)nn(C)c(CC(=O)NCCCC(C)NC(=O)C(C)C(F)(F)F)c1Cl 27687,Cc1cc(NC(=O)NC2CCSC2)cc(C(=O)N(C)C)c1 27688,n1(CC)ccc(CC(=O)NC(c2ccccn2)C(C)C)n1.c12cc[nH]c1C(=O)N2 27689,Cc1c(C(N2CCC(N(C)C(c3cnoc3)=O)C2)=O)oc2c(C)cccc12 27690,CON1CCC(C(=O)NC2CCC(C)N(C(=O)CCc3ccc(Cl)s3)C2)CC1 27691,CCCC(C)C(=O)NC1CC(C)(NC(=O)CCc2ccccn2)C1 27692,C1(O)(C(=O)NCC2(O)CN(Cc3cnc(C)o3)C2)CCCC(C)CC1 27693,c1(SC)ccc(C(=O)NC(CO)C(C)NC(=O)C(c2cnn(C)c2)N(C)C)cc1 27694,C1(C(=O)NCC2(C)N(C(C(C)NC(C)=O)=O)CCC2)CCc2nc(C)ncc2C1 27695,C(=O)(C(=O)C(C)(C)C)N1CC(C(=O)NC(CC(C)C)C)C(F)C1 27696,C1(O)(CN(C)C(c2cnns2)=O)CN(C(=O)CCN2CCC2)C1 27697,C1(C(=O)NC2CCC(NC(C(OC)OC)=O)CC2)CC(F)(F)CCC1(C)C 27698,N1(C(C(CSC)C)=O)CC(CC(=O)N(CCn2cc(C)cn2)C2CC2)CC1(C)C 27699,c1(C(N(C2CCN(C(C(COC)(C)OC)=O)C2)CC2CC2)=O)cncc(F)c1Cl 27700,c1(C(N2C(CCNC(=O)C(O)CC3CC3)CSCC2)=O)ccnc2ccsc12 27701,c1(C(N2CCCC(Cn3cc(C(C)(C)OC)nn3)C2)=O)cncc(F)c1C 27702,c1(C(=O)NCC2N(C(Cc3nc(=N)[nH][nH]3)=O)CC3CC32)csc2ccccc12 27703,c1(C(=O)NC(C(C)(C)NC(CCC2CC(OCC)C2)=O)C)ccc(Cl)nc1 27704,Cc1cc(Cl)c(-c2nc(C3CCOC3)nn2Cc2ccccc2F)cc1F 27705,Cc1cc(C(=O)NC2C(CCC(N3CCC(C(N(CCC)CCC)=O)C3)=O)C2)cs1 27706,C(=O)(C#CC1CC1)NC1(CNC(C=CCOCCOC)=O)CCCC1 27707,c1(OC)cnc(C(=O)N(CCCNC(=O)Cc2sc(C)nc2C)C)c(OC)n1 27708,c1(-c2cn(CC(CNC(c3ccc(CCC)[nH]3)=O)OC)nn2)c(F)cccc1F 27709,C#CCCC(C(=O)OC)NC(=O)CC1(NC(=O)CC(C)(C)SC)CC1 27710,C(C1c2ccsc2CCN1C(=O)C=CBr)NC(C(C)CC(N)=O)=O 27711,c1(C(=O)NCC(CN(C(C(C)C(F)(F)F)=O)C)O)cccc2c1N(C)C(=O)CO2 27712,O=[N+]([O-])c1ccc(N2CCC(c3nc(=N)[nH][nH]3)C2)c2ccncc12 27713,CC(C)C#CC(=O)N(CC(C)N(C)C(c1cnn(C)c1CC(C)C)=O)C 27714,CC1(C)CN(C(=O)C(c2ccc(Cl)cc2)O)CC1NC(c1ccccc1CO)=O 27715,C(CN=[N+]=[N-])(C(=O)NC12CCC(CC1O)C2)NC(CC=C)=O 27716,OC1CCCCC(NC(C23CCC(CC2)C3)c2nnnn2C2CCCC2)CC1 27717,N1(C(c2cn(C(C)C)nc2)=O)CCCCC1C(C)(C)CNC(C1CS(=O)(=O)C1)=O 27718,C1(NC(C2(CC#C)CCCC2)=O)CCN(C(c2ccc([N+](=O)[O-])s2)=O)CC1C 27719,N1(C(CN(C(=O)CN(C)C)CC#C)=O)CCCC1CO.C1(C#C)(N)COC1 27720,CC1CCC(C)(C(N2CC3CC2CS3=O)=O)CC1.C1C(=O)NCCO1 27721,c1(C(=O)NCCN(C(C=CCC)=O)CCCN(C)C)cncc(CC(C)C)c1 27722,CC1(C)C(C(=O)NCC(CO)NC(=O)CNC(N)=O)CC1(F)F 27723,CC1=NC(C)(CNC(c2coc(C(C)NC(c3cnc(C)o3)=O)n2)=O)CS1 27724,C(=O)(CC(C(F)(F)F)NC(c1[nH]ccc(=O)c1C)=O)N(C(CC)CSC)C 27725,C(=O)(C(CC(=O)OC)N(C)C)N1CC(CCCCNC(C(C)OC)=O)C1 27726,c1(C(c2nnnn2C)NC2C(CC)C2)nnsc1Br 27727,C1(NC(c2cc(CO)on2)=O)CN(C(c2c[nH]nc2C2CC2)=O)CCC12CCC2 27728,C1(c2c(C(N)=O)nsc2Br)NC(=S)N(CC2CCCCC2)C2=C1C(=O)N(C)C2C 27729,n1(CC=C)cc(CNC(=O)C(F)CC2CN(C(=O)CSC(C)C)C2)nn1 27730,CCC(C)C(C(=O)NCc1cc(C)ncn1)NC(C1C2CCC(F)C12)=O 27731,c1(SC)ncc(C#N)c(N2CCN(c3ncc(C)cn3)C3CC23)n1 27732,C(=O)(CC1=CCN(C)CC1)NCCCCN1CCCN(C(C(C)=C(C)C)=O)CC1 27733,N1(C(c2c(CC)ocn2)=O)CCCN(C(c2cc(C#N)oc2C)=O)CC1C(C)C 27734,c1(C(=O)NCC2CCCC(NC(CC(=O)OC)=O)C2)cc(N)ccc1Br 27735,C(F)(C(=O)NN1CCCC1C(=O)N(C)CC1CCCOC1)=C(C)C 27736,CCC(C)CCCCC(=O)N1CCC(C)(C(=O)NCC2CC=CC2)C1 27737,S(=O)(=O)(c1ccc(C(=O)NC2CCC(CO)C2)cc1)NCCCOC 27738,N1(CC)CCC1C(=O)N(C1(C(=O)NC2(c3cc[nH]n3)CC2)CC1)C 27739,c1(C(=O)NCC2N(C(CC=C(C)C)=O)CC(F)(F)C2)cn2c(n1)C(C)CCC2 27740,C1(N(C)C(C2CC2c2ccncc2Cl)=O)CCCN(C(C2(F)CC=CC2)=O)CC1 27741,C=CCC(C)(C)C(=O)N(CC(O)CNC(C1CN(C)CC1C(F)(F)F)=O)C 27742,C1(C(=O)NC2CCC(NC(c3ccc(CC)o3)=O)C2)CCOC1(C)C 27743,c1(OC)ccc2c(c1)CCN2C(C1CCCC(c2ccccc2)C1)=O 27744,C(CO)(CCCCNC(c1cc(C)[nH]n1)=O)NC(C=C(CC)C)=O 27745,Cc1nc2c([nH]1)CC(C(N1CC3C(N(C)C(c4cnc[nH]4)=O)C3C1)=O)CC2 27746,Nc1cc(O)c([N+](=O)[O-])cc1C(N1CCC2(CC1)CC2NC(=O)C1=CCC1)=O 27747,CCS(=O)(=O)CC(=O)N1CC(CNC(c2cnc3n2CCC3)=O)C2(CC2)C1 27748,c1(C(=O)NC2CN(C(C(CCC)O)=O)C3(C2)CCC3)coc2cc(OC)ccc12 27749,C1(C(N2CCC(O)(CNC(c3cnc(C)o3)=O)C2)=O)CC(C)(C)CN1C 27750,Cc1ccc(N(C(c2ccc(C(N)=O)cc2)=O)Cc2cc(Br)ccn2)cc1 27751,C1(CNCC(C2(C(=O)OC)CC2)=O)C2CN(C(=O)Cc3cncc(Cl)n3)CC12 27752,CCC(CC(=O)N1C2CCC1CC(CNC(=O)CCCS(N)(=O)=O)C2)C(C)C 27753,N1(C(C2(C)CCCC2)=O)CC2(CC(CC(N3CCOC(C#N)C3)=O)C2)C1 27754,N1(C(C(CC)c2ccccc2)=O)CCC2(CC1)CC2C(=O)NCc1cnc(C2CC2)[nH]1 27755,CC(CS(C)=O)C(=O)NCCCCN1CCCN(C(=O)CCSC(F)(F)F)CC1 27756,c1(C(N2CCC(NC(CCCNC(C)=O)=O)C2)=O)cccc(C)c1N 27757,C1(C)(CNC(c2cnc(CC(C)C)[nH]2)=O)CCCN1C(C1CCN(C)C1C)=O 27758,N1(C(CCC2CCCN(C(C(CCC=C)(C)C)=O)C2)=O)CCc2c(O)noc2C1 27759,Cc1ccc(O)cc1C(=O)NC(C)C(c1ccccc1)NC(=O)C(C)NC=O 27760,C(CC(C(=O)NC1CCC(C)CC1)NC(=O)CC1(CSC)CC1)SC 27761,C(C(=O)NCCCc1c[nH]nc1C)(C(C)(C)O)NC(c1c(CC)n(C)cc1)=O 27762,C1(C(N(c2c(C)n[nH]c2)C)=O)CC12CC2(F)F 27763,C1(OC)CC(CNC(c2ncc(F)cn2)=O)N(C(c2cnc(C(C)(C)C)o2)=O)C1 27764,C1(NC(=O)CCCCN2CCCC2)CC2CCC1N(C(=O)Cc1ccccc1)C2 27765,C1(NC(CCc2onc(CCC)n2)=O)CC12CCN(C(=O)C(C)(C)C1CC1)CC2 27766,N1(C(C(CC)(C)OC)=O)Cc2cccc(CNC(c3ncc(C4CC4)s3)=O)c2C1 27767,C(CC(C)C(=O)NCC(C)(C)N(C(=O)CC1(CSCC)CC1)C)=CCC 27768,Cc1nc(O)nc(C)c1C(=O)NCCCCCCNC(c1cc[nH]c1)=O 27769,S(=O)(=O)(c1ccc(OC)c(-c2cc(NC(C)C(C)C)cc(F)c2)c1)N(CC)CC 27770,N1(C(c2ccn(CC)n2)=O)CCC(C)C(NC(=O)CCc2ccon2)C1 27771,C1(NC(c2ccc(C(=O)OC)[nH]2)=O)COC2(C1)CN(C(=O)C1=CS(=O)CCC1)C2 27772,C1(N(C(c2ccc(CC)s2)=O)CC)CCCN(C(C2CC3CC2CC3O)=O)CC1 27773,c1(CC(=O)NCCNC(c2nc(COCC)sc2)=O)ccc(S(C)(=O)=O)cc1 27774,c1(OC(c2ccoc2CNC(N2C(CC)CCC2)=O)=O)cc(F)cc(F)c1 27775,C1(C(=O)NC2CCC(n3cc(CCC(C)(C)CO)nn3)CC2)(OC)CC(C)(C)C1 27776,c1(C(N2CC(Oc3cccc(F)c3)C2)C)ccc2c(c1F)OCCO2 27777,c1(NC2CN(C(c3occ(C)c3)=O)C2)ncnc2sc(C)c(C)c12 27778,N1(N(C2CCCCCCCC2)C(c2ccc(SC)s2)=O)CCC2(CCCCC2)CC1 27779,C(=O)(CCCCNC(=O)COC1CC(CC)C1)NCc1cc(CC)[nH]n1 27780,c1(C(=O)NC2CN(C(c3ccc(CO)c(F)c3)=O)C2)ccc2cc(F)ccc2n1 27781,N1(C(C2C(CC)OCC2)=O)CC2(CC(CC(=O)NC(COC(C)=O)CO)C2)C1 27782,C1(c2ccc(C)cc2)(C(F)(F)F)NC(=O)C2=C1C(c1ccccc1)CNC2=O 27783,c1(NCC2CCC(NC(c3c(CCC)nco3)=O)C2)ncccc1C#N 27784,C1(CNC(=O)NCC(CCSC)OC)CC2(C1)CC1(CCC1)C2 27785,Cc1nnc2n1CC(C(N1CCOC(c3ccc(Cl)cc3)C1)=O)CC2 27786,c1(C(=O)NCCC2(OC)CN(C(C3CCCC3C)=O)C2)c(C)nn(C(C)C)c1C 27787,C1(C(N2CC(CC(F)(F)F)C2)=O)CCN(C(=O)Cc2cncnc2O)C12CC2 27788,C1(NC(CCc2cnc(C)s2)=O)CCN(CCC2CCOC2)CC1(C)C 27789,c1(C(=O)NC2(CC=C)CCN(C(CC(=C)C)=O)C2)ccc(N)c(Cl)n1 27790,C1(F)(CNC(c2c(CCC)nco2)=O)CCC(NC(c2conc2C)=O)C1 27791,C1(O)(CNC(C(C)OCCOCC)=O)CCN(C(c2scc(C)c2C)=O)C1 27792,c1(C(=O)NCC(C)N(C(c2ccoc2)=O)CC)cocc1C 27793,c1(SCC)nccnc1C(N1CC(OC)CC1CCNC(c1ncoc1C)=O)=O 27794,O=C1CCc2ccc(C(=O)NC3CCCC(NC(c4n[nH]cc4Cl)=O)C3)cc2N1 27795,c1(OC)ccnc(CNC2CCCCC2C(=O)O)c1C 27796,C(C(=O)NCC1CCC2(CC2)C1)(C(C)(C)C)NC(c1c(C)ccnc1)=O 27797,C1(C(=O)NC(C)C(C)NCc2ccoc2)C2CC3CC(C2)CC1C3 27798,N1(Cc2c(C#N)c(F)ccc2)CCC2(CC1)CCN2C(c1cc[n+]([O-])cc1)=O 27799,c1(CCC)[nH]nc(C(=O)NCC2CCN(C(C3CC3C)=O)C2(C)C)c1[N+](=O)[O-] 27800,N1(C(C2(SC)CCC2)=O)CC2CCC(NC(=O)C=Cc3ccc(C)s3)CC2C1 27801,C=CCCCC(=O)NC(c1ccc(OC)cc1)CNC(C1CNC(=O)N1C)=O 27802,N#Cc1cc(C(=O)NCC2CCC2NC(c2ccn(-c3cccnc3)n2)=O)c[nH]1 27803,N1(C(C2(C#C)CN(C(c3cn(CC)cn3)=O)C2)=O)CCOC(CC)CC1 27804,O=C(CC(C(F)(F)F)NC(c1ccns1)=O)NC1C2CCC(C2)C1CO 27805,N1(CCC2CCN(C(=O)CCc3ccccc3)C2C(=O)OC)CCC(F)(F)CC1 27806,C1(C(N2CC(c3ccc(Cl)cn3)C2)C(=O)NC(CCC)C)CCCC(CF)C1 27807,C1(C(=O)NC2C=CCN(C(C(C)S(N)(=O)=O)=O)C2)CN(C)CCN(C)C1 27808,N1(C(C2CCC(NC(C)=O)O2)=O)CCN(C(c2ccc(C)cc2)=O)C(C)C1 27809,C1(OC)CC(CC(C)(C)COC(C)(C)C)N(C2CC2)C1.c12ccc(cc1)oc2=O 27810,C1(CNC(C2(CCOC)CCCC2)=O)CCN(C(c2nnc(C)s2)=O)C12CC2 27811,Cc1ccc(F)c(C(=O)NC2CCN(C(c3cn(CCF)nn3)=O)C2C)c1F 27812,C1(C(C)NC(=O)C=CBr)CCCN(C(=O)CNc2cnn(C)c2)C1 27813,N1(CC(=O)NC(=O)NCC=C)CC(NC(C2CCCC2O)=O)Cc2ccccc21 27814,N#Cc1ccc(-c2cn(C3CCN(C(=O)CCc4cc[nH]n4)CC3)nn2)cc1 27815,c1(C(=O)NC(CNC(c2c(C)occ2)=O)CO)cc(Cl)cc(Cl)c1O 27816,CC1(C)CCN(CC(=O)NCC(C)(O)CNC(c2cc(C#N)c[nH]2)=O)C1 27817,Cc1ccc(NC(CC(=O)NCCc2cnn(C)c2)c2ccccc2)cc1C 27818,C1(CC(=O)NC(C2(O)CN(C(c3cc(C(=O)OC)no3)=O)C2)C)CCCCN1C 27819,C1(NC(c2c(CC)[nH]cc2)=O)C2CC(NC(C3(C)CCSCC3)=O)CC12 27820,Oc1nc(NS(=O)(=O)CCc2cccnc2Cl)oc1Cl 27821,N1(C(C2CC(C)OC2)=O)CCN(C(=O)CN2CCC(CN(C)C3CC3)CC2)CC1 27822,C#CCCCCC(c1nnnn1CCOC)NCC1COC1 27823,c1(CN2CCCC(N(C)C)C2)ccc(C(=O)Sc2ccccc2)c(F)c1 27824,CC(C)(C)C(C(=O)NCc1cccc(F)c1F)NC(c1ncoc1C1CC1)=O 27825,C1(C)(COC)CC(NC(c2c[nH]nc2OC)=O)CN1C(c1n[nH]c2c1CCC2)=O 27826,C(=O)(C(C(C)(C)O)NC(c1nocc1C(C)C)=O)NCCCc1nnc(C)s1 27827,C1(CNC(c2n(C=C)ncc2)=O)CC2CCC(C1)N2C(C1(C2CC2)CCCO1)=O 27828,c1(C(N2CC(CNC(C3OC4CCC3CC4)=O)C(O)C2)=O)cn2c(n1)CCC2 27829,c1(CC)cc(C(=O)NCC2(C(N)=O)CN(C(=O)C(=O)NCC(N)=O)C2)cc(Cl)n1 27830,c1(C(=O)NCC2C(NC(c3cc(C)nc(C)n3)=O)CCC2)cnc2ncccn12 27831,C(=O)(C1CCc2scnc21)N1C2CN(C(C(C)c3cc[nH]n3)=O)C(C2)C1 27832,O=C1CCCC(C(=O)N(CCCNC(C2(c3cc[nH]n3)CC2)=O)C2CC2)O1 27833,Cc1ccc(C(=O)NC(C)CCCNC(C2C=CCC2)=O)c(C)c1 27834,CCCCCCNC(=O)C(Cc1cnc[nH]1)NC(C1CC1c1cn[nH]c1)=O 27835,c1(C(N2CCC(C3CCCN3C(c3occc3Cl)=O)C2)=O)ccc2ncnn2n1 27836,N1(C(c2c(OCC)nccc2)=O)C2CCC1CN(C(c1noc(C)n1)=O)C2 27837,Cc1cnc(Cl)c(C(N2CCC(CC(C)NC(c3ccc(F)nc3)=O)CC2)=O)c1 27838,c1(C(=O)NCC(C)(CO)NC(C=C(C)C2CCCCC2)=O)cccn2nnnc12 27839,C(N=c1[nH]c(C)c(C(=O)NC(CCO)C(C)C)s1)c1c(F)ccc(OC)c1 27840,Cc1cc(C(=O)NCC2C(C)CCN2C(c2ccnc(Cl)c2O)=O)cnc1C 27841,c1(C(=O)NCC(Cc2ccccc2)CO)csc(=NCc2ccc(O)c(Cl)c2)[nH]1 27842,Cc1cc(C(F)F)oc1C(=O)NC(C)CC(C)NC(c1ccncn1)=O 27843,Cc1ccc(C(=O)NCC2CN(C(c3nncn3C)=O)CC2C)c2ccccc12 27844,c1(C(N2CCC(O)(NC(c3cccnc3)=O)C2)=O)ccc(OCC(F)F)cc1 27845,N1(C(Cn2ncn(C)c2=O)=O)CC2CC(NC(c3cncc(C4CC4)c3)=O)C2C1 27846,C1(NC(CCC=CC)=O)CC2CC(NC(c3cc(OC)cnc3F)=O)CC2C1 27847,N1(C(C(C2CCCC2)SC)=O)CC(F)(NC(=O)CN(c2ccncc2)C)C1 27848,c1(C(N2CC(COC)(CNC(=O)C(F)F)C2)=O)ccnc(S(N)(=O)=O)c1 27849,C12(CNC(C(CCC)N(C)C)=O)CN(C(=O)CN=S(C)(C)=O)CC1CCO2 27850,CC1CN(C(C2C3CC4C(C3=O)C24)=O)CCC1C(=O)NCC(O)C(C)(C)O 27851,N1(C(C(C(C(C)C)O)C)=O)CCC2(C=C(C(=O)Nc3ccnc4cc[nH]c34)C2)C1 27852,CCCC(C#N)C(=O)NC1C2CN(C(c3cnn(CCCOC)c3)=O)CC12 27853,c1(NC(Cc2nc(CC)sc2)=O)cccc(NC(=O)C(C)SC(F)(F)F)c1 27854,Cc1ccc(-c2cn(C3CC3NC(=O)C(C)OCCC(C)C)nn2)cn1 27855,C1(NC(c2n(C=C)nnc2)=O)CCN(C(=O)Cc2cc(C3CC3)nn2C)CC1C 27856,N1(C(C(COC)(C)C)=O)CCOC2(C1)CN(C(=O)CCc1cnc[nH]1)C2 27857,C1(NC(CN(C(C)C)C)=O)CC(O)CN(C(=O)CN2CCC(O)CC2)C1 27858,Cc1nnc(N(CCCNC(c2nc(Cl)sc2Cl)=O)C2CC2)nc1C 27859,N1(C(CCCC(C)=O)=O)CCC2OCCN(C(c3ccsc3Cl)=O)C2C1 27860,C1(C(=O)Nc2c(C)nc(-c3ccccc3)s2)CN(C(=O)CCN(C)C)CC(F)(F)C1 27861,N1(C(c2cc(OC)c(C)cc2)(c2nnnn2C)OC)CC2CCC(C1)C(=O)N2 27862,c1(CNC(=O)NCC2CC(F)(F)C2)c(C(F)(F)F)cccc1F 27863,c1(C(N(C(C)C(N2CCn3ncnc3C2)=O)CC)=O)ccc(C#N)c(C)c1 27864,C1(NC(c2c(CC)con2)=O)CCOC(CNC(=O)Cn2nccn2)C1 27865,c1(C(=O)NC(CNC(C(CCC)(C)O)=O)(C)Cn2cccn2)ccc(S(C)(=O)=O)s1 27866,C1(NC(c2ccoc2)=O)CCCCC12CCN(C(c1cc3n(n1)CCCN3)=O)C2 27867,N1(C(CSC(CC)C)=O)CC2C(NC(=O)CNC(=O)CON3CCOCC3)C2C1 27868,N1(C(C(C)N(C)C)=O)CCC(C(=O)NC(c2cc(C3CCCN3)no2)C)C1 27869,C1(CC#C)(C(=O)NCCC(C)NC(c2coc(Br)n2)=O)CCOC1 27870,N1(C(c2ccc(CC)cc2C)=O)CC(C)N(C(c2cnc(S)[nH]2)=O)CC1C 27871,C1(NC(C2(C)CC=CCC2)=O)C2CC3C1C3C2C(N1CCCC(C(C)(C)C)C1)=O 27872,Cc1oc([N+](=O)[O-])cc1C(N1CC2CCC1C(CNC(c1cnoc1C)=O)C2)=O 27873,c1(C(=O)NCC2C(C(=O)NCC(CO)OC)C2)ccc2ccccc2n1 27874,Cc1oc(CO)cc1C(=O)NCC1(C)CCCN1C(C1CC12CC2)=O 27875,N1(C(C2(C(F)F)CC(=C)C2)=O)CC(NC(c2ccc(C)nc2O)=O)C(C#N)C1 27876,CC(C)(CCC(=O)NC1CCCC(O)CC1)NC(=O)CCCC1CCCO1 27877,CC1CCN(C(C2(O)CCCN(C(=O)OC(C)(C)C)C2)=O)C(C2CC2)C1 27878,C1(c2cn(CCCCNC(c3cnc(CCC)s3)=O)nn2)CCCCC1O 27879,c1(C(=O)NCC2C(C)CN(C(c3cccc(=O)o3)=O)C2)cnc(P(C)(C)=O)cn1 27880,O=C(C(O)C(F)(F)F)N1CCN(CC2CN(C(C3(C(F)F)CCCO3)=O)C2)CC1 27881,N1(C(C(CCC)OC)=O)CCCC(F)(C(=O)NC2(CC(C)(C)C)CC2)C1 27882,c1(C(N(CCC=C)CC)=O)cc(N(C(=O)CNC(=O)OC(C)(C)C)C)ncc1F 27883,C1(CC#C)(C(=O)NCc2ccc(Cl)cn2)CCN(C(=O)CCSC)C1 27884,c1(C(=O)NCC(COC)F)cccc(C(=O)NC2(c3ccc(F)cc3)CCC2)c1 27885,c1(SC)nc2ncnc(NC3(NC(=O)CCCC4CCCC4)CC3)c2s1 27886,C1(CNC(COCCOCCOC)=O)CC(CO)CCN1C(=O)CC(C)F 27887,c1(OC)ccc(OC)c(C=CC(=O)NC2CC2NC(c2cc(OC)n(C)n2)=O)c1 27888,Cc1ccc(C(=O)NC2CCOCC2NC(=O)CCc2ccoc2)cc1N 27889,C1(C(N(c2ccn(C)n2)CC)=O)CCCCC1(C)NC(c1c[nH]c(=NC)s1)=O 27890,c1(CN2CCCC(C(=O)OC)C2)ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=O 27891,N1(C(c2n(C(CC)C)ncc2)=O)CCN(C(C2CC(OC)CN2C(C)=O)=O)CC1 27892,C(=O)(C1=C(C)CC(C)(C)CC1)N1CCN(C(C(CCC)O)=O)C(C2CCCC2)C1 27893,CCCS(=O)(=O)C(C)C(=O)NC1CCCCC1CNC(c1cc2sccc2n1C)=O 27894,N(C1CCc2c(Br)cccc21)c1cc(NC(C(n2ncc(C)c2)C)C)ncn1 27895,c1(SC)ccc(NC(N(CC(F)(F)C(C)C)C(CC)C)=O)c(C)c1 27896,c1(C(N(C(CNC(CCC(=C)C)=O)C)CC)=O)cc(OC)c(OC(C)C)c(Cl)c1 27897,c1(C(C(=O)NCCNC(CC(C)CO)=O)O)ccc(Cl)c(F)c1 27898,N1(C(c2c(CC)sc(=N)[nH]2)=O)CCCOC(CNC(=O)C2=COCC2)C1 27899,CN1C(C(c2nnnn2C2COC2)NC2CCCSCC2)CCS1(=O)=O 27900,c1(C(C(F)F)NC(=O)CCCCc2ccc(Br)cc2)ccc(F)cc1Cl 27901,N1(C(CN(C)Cc2ccccc2)=O)CC(CNC(c2cc[nH]n2)=O)C(O)C1 27902,CN1c2ccc(C(=O)NCCCNC(c3coc(Cl)c3)=O)cc2C(C)(C)S1(=O)=O 27903,C1(NC(C2C(C)C2C)=O)CCN(C(c2cnn(CCC(F)(F)F)c2)=O)C1C1CC1 27904,N1(C(C(N)=O)=O)CC2(CCC2CNC(C2CCCS2)=O)C1 27905,c1(C(C(=O)NC)N(C)Cc2ncc(C)cc2F)ccc(OC)cc1Cl 27906,C(C1COCc2ccccc21)NC(=O)NCC(CC)(CC)C(N)=O 27907,CN=c1[nH]cc(C(=O)N(C2CCN(C(=O)CCc3ccncn3)C2)C)s1 27908,c1(C(=O)NCC2C(NC(CCSCCC)=O)C2)[nH]c(C)c([N+](=O)[O-])c1C 27909,N1(C(C2(C=C)CCCCC2)=O)CC2(C1)CN(C(=O)CN(CC)CC)CCO2 27910,c1(CCCC)ccc(CC(=O)NCCN(C(=O)CCCCSC)CC2CC2)cc1 27911,c1(C(C)NC(C2C(C#N)C2(C)C)=O)ccc2nc(O)[nH]c2c1 27912,C(=O)(CC1=CCN(C)CC1)NCCSC.C#CC1CO1.C12CC1CNC2=O 27913,c1(C(N2CCN(C(CSCCCC)=O)CC2C(C)C)=O)cccc2cncn12 27914,CC1C(CS(C2CC(Oc3ccccc3)C2)(=O)=O)CCN1C 27915,C1(CNC(C2N(C(C)=O)CCC2)=O)CN(C(c2cc(C#N)oc2C)=O)CCN1C 27916,C1(CNC(c2c(COC)n(C3CCC3)nc2)=O)CC2(CC2)CN1C(=O)C(C)C#N 27917,N1(C(c2c(O)ccc(C#N)c2)=O)CCC2(CCCC2NC(C2CC(=O)N2)=O)CC1 27918,c1(C(N(CCCNC(C2(CC(F)F)CC2)=O)C)=O)cc(C(C)(F)F)ccn1 27919,c12ccc(C)nc1C(=O)N1CC(OC)C(C1)C(=O)N2.c1(SCC)cscc1OC 27920,C(=O)(C(C(C)(C)C)SC)NCCN(C(=O)CCC1CNC(=O)N1)CCC 27921,Cc1[nH]nc2c1CCC(C(=O)NCCNS(=O)(=O)c1ccc(Br)cc1)C2 27922,C1(O)(C(=O)NC2C(N(C)C)CC2)CCN(C(c2ccccc2N2CCCC2)=O)C1 27923,c1(NC(=O)C(N2CCN(c3ccnnc3)CC2)=O)ccccc1-n1ccnn1 27924,C1(OC)CC(NC(=O)C(C(C)O)NC(C)=O)N(C(=O)CSc2nccn2C)C1 27925,c1(C(=O)NC2(CNC(=O)C3=CCC3)CC(OC)C2)cc(N=S(C)(C)=O)ccn1 27926,N1(C(C(C(C)C)NC(C)=O)=O)CCCC2(NC(c3ocnc3C)=O)CC2C1 27927,C1(C(C)C)CN(C(=O)C(CC(F)F)C2CCC2)CC(=O)N1 27928,CCCCS(=O)(=O)NC(C)C(N1CC(O)(CNC(=O)C=Cc2cccnc2)C1)=O 27929,C(=O)(N1CC=CCO1)C1(CC=C)CN(C(C2CCN(C(N)=O)CC2)=O)C1 27930,c1(OC)ccc(C(N2CCOC(C)(CNC(=O)C(F)(F)C3CC3)C2)=O)cc1F 27931,S(=O)(=O)(c1[nH]c(=NCCCCC(C)(C)SC)ccc1Br)NCCCC=C 27932,Cc1cn2ccc(C(=O)NCC3CCCC3NC(c3sccc3C)=O)cc2n1 27933,N1(C(C(C)(C)NS(C)(=O)=O)=O)CCOCC(NC(c2conc2Br)=O)C1 27934,Cc1cccc2[nH]cc(C(=O)NC3(C)CCN(C(C4CCCSC4)=O)C3)c12 27935,C=CC1CN(C(=O)C(C)(C)NC(=O)CCCCCC)CCO1 27936,CCC(C)(C)CCCC(=O)NC(C)Cn1cc(CCc2ccccc2)nn1 27937,Cc1cc(Br)oc1C(=O)NC1CCOCC1NC(=O)C(C)N(C)C 27938,C1(Cc2cn(CCOC)nn2)CCCCCN1C(c1cc(OC)ccn1)=O 27939,c1(-c2ccc(CNC(c3c(N)nc(C(=O)O)cc3)=O)s2)ccc2nonc2c1 27940,CCC(C)C(O)C(C)C(=O)N1CCOCC1CCNC(C12CCCN(CC1)C2)=O 27941,C1(CC)OCCC1C(=O)NCC1C(CNC(=O)Cc2cnsc2)C1(F)F 27942,C1(CCC(=O)NCC2CC2NC(c2cc(Cl)ccn2)=O)NC(=O)NC1=O 27943,Cn1cc(C=CC(=O)NCC2CC(NC(=O)C(=O)NCC(F)(F)F)CCO2)nn1 27944,C1(CC(=O)NC2(CF)CCN(C(CCC(C)C)=O)C2)COC(C)(C)CO1 27945,N1(C(CCC(CC)CC)=O)CC(C2CCCCN(C(C3CCSC3)=O)C2)C1 27946,c1(C(N2CCC(NC(C(CC)N(C)C)=O)C(CO)C2)=O)cc2ncccc2[nH]1 27947,C12(C(=O)NC3CCCC(NC(CC4(C)CCC4)=O)C3)CC3CC(C(=O)N1)C2C3 27948,C12(CNC(c3[nH]c(CC)c(Cl)n3)=O)CCC(C1)N(C(C1CCC(OC)CC1)=O)C2 27949,C1(CC(=O)NC(C(=O)NC)CC2CCCC2)CCNC2(CC2)C1 27950,N1(C(c2c(CC)noc2C)=O)CCC(CNC(=O)CCc2cnc[nH]2)C(C)C1 27951,C12(C(N(C(CN(C(CNC(CCC)=O)=O)C)C)C)=O)CC1COC2(C)C 27952,C1(C(N2CCC(C(N3CCN(c4nncs4)CC3)=O)C2)=O)CCC(F)(F)C1O 27953,C1(COCC)CCCN(C(C2(C)CCN2C(c2ccnc(F)c2)=O)=O)C1 27954,C(C(C)(C)C(=O)N1CCCC(N(C(=O)CCCc2cccs2)CCF)C1)N(C)C 27955,C(C[Si](C)(C)C)NC(CCN(CC#C)C(c1cc(Cl)cs1)=O)=O 27956,C(CC(N)=O)(C(=O)N1CC(CO)CC1CO)NC(c1nccc(COC)c1)=O 27957,c1(C(=O)NC2C(NC(C3(CC#C)CCC3)=O)C2)cc(C(F)(F)F)cnc1O 27958,C1(NC(COCCOCC#C)=O)CN(C(=O)C(C)CF)CC1F 27959,N1(C(CC2CCC(=O)C2)=O)CCC(C2CCN(C(c3ccc(F)cc3Cl)=O)C2)C1 27960,c12cccc(c1)C2.Cc1sccc1CC(=O)NC1COCC1n1cc(C(=O)O)nn1 27961,c1(C(CC(=O)N(C)CCNC(c2ccc(C(C)(C)C)s2)=O)=O)cc(F)ccc1F 27962,N1(C(C(C)NC(C)=O)=O)CCC(CCNC(C2(CC(C)C)CCC2)=O)C1 27963,c1(-n2cc(C(C(OC)OC)C)nn2)ccc2ncc(Br)cc2c1 27964,N1(C(Cc2c(C)ccs2)=O)CCC(NC(c2cn(CC(=O)N(C)C)nn2)=O)CC1C 27965,N1(C(Cc2n(C)cnn2)=O)CCC(CNC(C2CC(n3cnnc3)C2)=O)C12CC2 27966,C12C3CCCC3CN1C(=O)C2.CC(CNC(c1ccccn1)=O)CC(F)(F)F 27967,CCCCCCC(C)(c1nnnn1CC1CCCO1)NC1CCC(C)CC1 27968,C=CC(C)(O)CC(=O)N(C1CCCCN(C(c2nc(OC)cc(OC)n2)=O)C1)CC 27969,c1(N2CC3C(NC(C4N(S(CC)(=O)=O)CCCC4)=O)C3C2)nnc(C)c(C)n1 27970,C=C(C)C(C)(C)C(=O)N1CCC(CN(C)C(c2cn(C)nc2SC)=O)C1 27971,N1(C(c2cccc(C)c2F)=O)CCC2(C1)CN(c1ncc(Br)cn1)CCO2 27972,c1(CN=C(NC(C2CCCO2)=O)NC2CCS(=O)(=O)C2)ccc2c(c1)OCCCO2 27973,N1(C(CCCCCNC(Cc2c(C)n(C)cn2)=O)=O)Cc2cccnc2C1 27974,N12CC3CCCC(C3C1)NCC2=O.N=c1[nH]c(CCO)cs1.C1(CNC(=O)CO)CCCO1 27975,N1(C(=O)Cn2cncn2)CCC(F)(C(N2CCCCC2c2ccncc2)=O)CC1 27976,C#CCCCC(C(=O)Nc1ccc(C(=O)OC)cc1)N(C1COC1)C 27977,c1(-c2onc(CC(C3CCS(=O)(=O)CC3)O)n2)ccnc2c(I)cnn12 27978,Cc1c(C(=O)NCC2CCN(C(=O)C(F)=C3CCC3)C2)cnn1CCO 27979,c1(OC)c(C(=O)N(CCCNC(=O)CC2CCC(=O)N2)C2CC2)cccc1Cl 27980,CC1CN(C(c2ncnc(O)c2Cl)=O)CC(C)N(C(c2cnn3c2SCC3)=O)C1 27981,C(=O)(C(F)C(C)CNC(c1ccc(C)o1)=O)N(C(CC)C(=O)OC)C 27982,N1(C(C2(C)C(C)C2)=O)CCC2(CC1)CN(C(c1c(F)cncc1F)=O)CCC2O 27983,c1(CN(C(Cc2ccccc2)C(=O)NC2CC2)C)ccsc1S(C)(=O)=O 27984,N1(c2c(C#N)cnc(C)n2)Cc2ccc(NC(=O)C(c3ccccc3)F)cc2C1 27985,Cc1ccc(N)c(C)c1C(=O)N(CC(O)CNC(=O)CC(C)C1CC1)C 27986,CCC(CC(=O)N(CC(C)C(=O)NC(C)CC1CC1)C)CC(C)C 27987,C1(NC(C=C2CCN(C(C3(COC)COC3)=O)CC2)=O)CC(=O)N(C)C1=O 27988,C1(CNC(C(CCCC)C)(C)c2nnnn2CCCF)Cc2ccccc2CO1 27989,c1(C(=O)NC2C=CCN(C(CC3N(C(C)=O)CCC3)=O)C2)n[nH]cc1[N+](=O)[O-] 27990,N1(C(CCc2cnc(C)o2)=O)CC(C(=O)NCC(Cl)=CCl)C(C)(C)C1 27991,CON(C(=O)C#CCNC(c1cc(=O)cc[nH]1)=O)C1CCOCC1 27992,C(=O)(C1=CC2C=CC1C2)N1CCCC(C(=O)Nc2c(C(C)C)nccc2)CC1 27993,C12(CC(=O)NCc3ccncc3)CCC1CN(C(c1ccc(CO)c(Cl)c1)=O)C2 27994,C(CCN(C)C)(C(=O)N(C1CC1(Cl)Cl)CC)NC(Cn1ncc(CC)c1)=O 27995,C#Cc1cccc(CNC(C2(CCNC(=O)C(c3cnccn3)C)CCC2)=O)c1 27996,N1(C(c2cnco2)=O)CC2CCN(C(c3ccc(-n4cnnn4)cc3)=O)C(C2)C1 27997,CC1(C)OCCC1(O)C(=O)NC1CCCCC1NC(c1cn2ccsc2n1)=O 27998,c1(C(=O)NCC2C(C)CN(C(c3nsc(C(F)(F)F)n3)=O)C2)cc(C#N)cn1C 27999,C(=O)(C1=CCCCO1)NC1(CC=C)CCN(C(c2ccc(=NC)[nH]c2)=O)C1 28000,CC(C)(C)CCNC(C1CCCN(C(c2ncccc2C2CC2)=O)C1)=O 28001,N1(C(c2cnn(CC)n2)=O)CCCC(C2CCCCN2C(=O)CNS(C)(=O)=O)C1 28002,c1(CC(C)C)ccc(C(N2CCCC(CNC(=O)Cn3cc[n+](C)c3)C2)=O)cn1 28003,CN(S(=O)(=O)N1CC(O)C(O)C1)CC(c1ccccc1)O 28004,Cc1csc(CC(=O)NC(C(=O)NCC2(S(C)=O)CC2)C2CCCC2)c1 28005,C123CCC(F)(CN(C1)C2=O)C3.c1(SCCOCC(F)(F)F)ccccc1 28006,C(=O)(C(O)CCn1cncn1)NC(C(C)NC(c1coc(CC2CC2)n1)=O)(C)C 28007,C1(OC)(CNC(=O)Cc2cccs2)CCN(C(C2C3CCC(F)C23)=O)C1 28008,C(=O)(C#CC1CCOCC1)N1C(C2(NC(C3CCS(=O)(=O)N3C)C)CC2)CCCC1 28009,C(=O)(CS(=O)(=O)CCOC)NC1(CF)CCN(C(C(CC)(C)O)=O)C1 28010,c1(NC(C)=O)ccc(N)c(C(=O)NCCC(F)Cn2cc(C3(O)CCC3)nn2)c1 28011,C1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)(C)N(C)C)CCCC(=O)N1C 28012,n1(CCCC)cc(C(=O)NCCC2CN(C(c3ns[nH]c3=O)=O)CC2C)c(C)n1 28013,c1(CC)ccc(C(=O)NCC(C)CNC(c2cccn2CC)=O)cc1Cl 28014,c1(C(N2CC3CC(NC(C(C)N4CCC4)=O)CC3C2)=O)ccc2c(n1)CCCC2 28015,Cn1ncc2ccnc(C(=O)NC(CNC(=O)C(O)P(C)(C)=O)C(C)(C)C)c12 28016,c1(N(C2CN(C(=O)CC(C3CCCCC3)C3CC3)C2)C)cnnn1C 28017,Cc1nc(O)sc1C(=O)NC(C)(CNC(=O)C(=O)NCC(F)F)C(C)C 28018,N1(C(COC2(C)CCC2)=O)CCCC2(NC(=O)C(C)(C)C3CCC3)CCCC12 28019,CC(C)C(C(=O)N1CCN(C(c2ncccc2O)=O)CC1CC1CC1)C(C)C 28020,C(=O)(C(CCSC)NC(=O)CC1CC(O)C1)NC(CC=C)C1CC1.SCC.OC 28021,C1(NC(c2n(C)ncc2)=O)Cc2ccccc2C1NC(=O)CC1CC12CC2 28022,c1(CNC(c2cc(OCC)n[nH]2)=O)ccccc1CCBr.C1(C)(C2CCC2)CN1 28023,c1(N(CCN(C(c2c(C(C)C)cco2)=O)C(C)C)C)ncc(Cl)c(C)c1C#N 28024,c1(C(N2C3(CN(C(C4CN(C(C)C)C(=O)C4)=O)C3)CC2)=O)cc(F)cc(F)c1F 28025,N1(C(CCc2cnn(C)n2)=O)CCC2(CC1)CCN(C(C1CC(O)C1)=O)CC2 28026,c1(C(N2CC(C)C(NC(c3cccc(F)c3Br)=O)C2)=O)ccn2ccnc2c1 28027,C(c1csc2ccccc12)=CC(=O)N(C1(N2CCCCC2)CNC1)C1CC1 28028,c1(C(C)NC(C2COCCN(c3ncc(C)cn3)C2)=O)cccc2c1OCCO2 28029,CC(C)CCCCCC(=O)NCC1(CNC(=O)Cn2cc(C(F)(F)F)cn2)CC1 28030,c1(C(CC)NC(=O)C(=O)NCc2c[nH]nc2-c2ccccc2)cc(F)cc(F)c1 28031,c1(OC)ccc(N(C)C)cc1.C12CC(C)(C1)NCC(=O)N1CCCC1C(=O)N2 28032,C1(OC)CC(CNC(=O)C(=O)NC(C)Cc2cccnc2)C1(C)C 28033,C1(CCC)CN(C(=O)C=Cc2ccc(CC)o2)CCN1C(=O)CCC(C)(C)F 28034,N1(C(C2C(OC)C2)=O)Cc2n[nH]cc2C1C(=O)N1CCCC(NC(=O)C2CC2)C1 28035,C1(C(=O)NC2C(NC(C(C3CCC3)OCC)=O)CC2)CC(c2cccnc2)=NO1 28036,N1(C(c2cccc(CCC)c2)=O)CCC2CN(C(=O)Cc3cn[nH]c3)C2C1 28037,Cc1c(C(N2CCC(C(C)NC(C3CC(=O)N(CC4CC4)C3)=O)C2)=O)ncn1C 28038,N1(C(CS(N)(=O)=O)=O)CCOCC(NC(=O)C(O)Cc2ccccc2)C1 28039,Cc1nc(Cl)ccc1CC(=O)N(CC(O)CN(C)C(c1ccn(C)c1)=O)C 28040,Cc1ccc(CNC(N2CCC(NC(C34CC(CO3)C4)=O)C2)=O)cc1 28041,c1(OC)ccc(C(N2CC(O)CC2C(=O)NCc2ccc(Br)c(Br)c2)=O)cc1I 28042,C1(C(=O)NC2CCC(NC(CC3C(C)(C)CCO3)=O)C2)CCOC(=O)CC1 28043,c1(C(=O)NCC(C)(C)NC(c2cnc(C)[nH]2)=O)ccc(OC(F)(F)F)nc1 28044,C12(CC(N3CCC(CO)C(O)C3)=O)CCC1CN(C(=O)CCCCC1CCCO1)C2 28045,C1(N(C(CC(C)C)=O)C)CCCN(C(C2(C#N)CC2(C)C)=O)CC1 28046,C1(COCC(=O)NC(C2CN(C(=O)CCc3ccon3)C2)C)CCCCO1 28047,c1(CC(N2CCC(NC(CC3C(C)CCC3)=O)C2C)=O)ccc2oc(O)nc2c1 28048,N1(C(c2c(C)cncc2C)=O)CCC2C(CCCN2C(=O)C(F)CC(C)C)C1 28049,c1(NC(c2c(CNC(c3ncc(F)cc3F)=O)ccs2)=O)ccc(Cl)c(O)c1 28050,C1(NC(C2CC(=O)NCC2)=O)C2CC(O)C1N(C(=O)CC1CCC1)C2 28051,CC1C(NC(=O)CCCC(=O)N(C)C)CCCN1C(C1CCC(=O)N1C)=O 28052,N1(C(c2nc(OCC)sn2)=O)CCC(C2(NC(c3ccoc3)=O)CCC2)CC1 28053,CC(CNC(=O)CCc1ccncc1)C(=O)N(C1CCCC1)C 28054,C1(NC(C(C)Sc2nncn2C)=O)CC(C)N(C(c2cc[nH]c2C2CC2)=O)C1 28055,N1(C(CSCC)=O)CCC(C2CCN(C(c3cc(-c4cccn4C)[nH]n3)=O)C2)C1 28056,c1(C(=O)NC2(CCCNC(c3cncc(C=C)c3)=O)CC2)cnc2scc(C)n12 28057,S(=O)(=O)(c1c[nH]ccc1=NCC1CCC(C)(C)CO1)NC(c1ccncc1)C=C 28058,N1(C(c2cncc(OCC)c2)=O)CCC(CNC(=O)C(C)c2ccsc2)C1(C)C 28059,c1(N2CC(C(N3CCN(CCC)CC3)=O)C(O)CC2)cnc2cc(Cl)ccc2n1 28060,c1(CC(N2CC(OC)C(NC(=O)C(C)S(N)(=O)=O)C2)=O)ccc2c(c1)NC(=O)C2 28061,C1(CNC(C=CC)=O)CN(C(=O)C(c2cccc(OC(F)F)c2)C)C(C)(C)C1 28062,CC1=C(C(=O)NC23CCN(C(=O)CC(C)(C)C)CC2C3)CCC1 28063,N1(C(c2c(CC)csc2)=O)CCC(CNC(=O)Cn2nc(C)oc2=O)C(C)C1 28064,C(=O)(CCCC(C)(F)F)N1C2C(NC(c3cc(C)c(C)nn3)=O)CC(C2)C1 28065,c1(C(=O)NC(C(=O)NCC2(C)CCCC2O)CN(C)C)cc2cc[nH]c2cn1 28066,C(=O)(CCCCCN(C(=O)CC1CCC1C)C(C)C)N(CC(C)C)CCC 28067,C(C)(C)(CC(F)C(=O)NCCCc1cccnc1)NC(Cc1scc(C)c1)=O 28068,c1(C(N2CCCC(NC(C(C)n3cnnn3)=O)C2)=O)ccc2c(c1)COC2 28069,C(CC(=O)N1CC(CC(C)(C)C)C1)N(C(=O)C=CC(F)(F)F)CC 28070,C(C(C)(C(C)C)NC(=O)Cc1csc(N(C)C)n1)NC(CNC(CC)=O)=O.C1CC1 28071,C1(NC(C(C#C)(C)C)=O)CCC(C)(CNC(c2coc(C(F)F)n2)=O)CC1 28072,c1(C(N2CC(CCNC(c3cnsn3)=O)(OC)C2)=O)cccnc1SC(F)F 28073,CC1CCC(C)(C(=O)Nc2cn(C3C4C(=O)OCC34Br)nn2)C1 28074,c1(C(N2CCC(OCCNC(Cn3c(C)c(Cl)cn3)=O)C2)=O)ccn(C)c(=O)c1 28075,C1(C(=O)NCCC2CCCN2C(=O)CC2CCCC23CC3)(OC)CCS(=O)(=O)C1 28076,C1(NC(CSS(C)(=O)=O)=O)CCN(C(c2ccnn2C(F)F)=O)CC1(C)C 28077,CC1CCCCC1C(=O)NC(C)(C)C=CC(=O)NCC(F)Cl 28078,c1(C(N)=O)ccc(CC(N2CCOCC2CNC(=O)CCC2CCCO2)=O)cc1 28079,C1(CNC(C(C(CC)C)O)=O)CCCC2(CN(C(=O)Cc3cccc(Cl)c3)C2)O1 28080,Cc1c(C(=O)NCC2CN(C(=O)CC3CCSC3)CCO2)nn(C)c1N 28081,Cc1cccc2c(C(N3CCCC(N(CCF)C(C4CC4(F)F)=O)C3)=O)coc12 28082,N1(C(CN(C(COC)=O)C)=O)CCCC1(C)NC(=O)CSC1CCOC1=O 28083,N1(C(C(C(C)C)OC)=O)CCN(C(=O)Cn2nnnc2C(C)C)CC12CC2 28084,Cc1cccc(CC(=O)NCC(C)N(C)C(c2cnc(CC(C)C)[nH]2)=O)c1C 28085,c1(C(=O)NC2CCNC2=O)cc2c(s1)CCN(Cc1cc(Cl)ccc1Cl)C2 28086,C(=O)(C(F)(F)C(O)C1CC1)NCC(C)N(C(c1ccnc(Br)c1)=O)CC 28087,c1(C(=O)OC)ccc(N(C)C)cc1C.n12cc(nn1)CNC(=O)C(=O)NC(C)C2 28088,CC1(C)CC(CC(=O)NCC(C)(C2CC2)NC(=O)COc2ccon2)C(=O)O1 28089,N1(C(C(C)=CC2CC2)=O)CC2CCCCC2(CNC(=O)C(C)c2cccs2)C1 28090,C#Cc1ccc(C(=O)NCC2CC3CCC2N3C(C2C3CCCC23)=O)nc1 28091,CP1(=O)CCN(NC(=O)CC2COCCC2O)CC1 28092,C#CC1CN(C(c2cc(Cl)ccc2O)=O)CCN1C(c1cnc(CC)[nH]1)=O 28093,C(=O)(CCCCCCCCCOC(c1cc(Br)c(Cl)s1)=O)OC 28094,N1(C(CN(C(C(F)=CCOC)=O)C(C)C)=O)CC(C(=O)OC)CCC1=O 28095,c1(OC)ccc(CCC(=O)NCCCCNC(c2cccc(CO)c2)=O)c(C)c1 28096,C#CCC(C)(C(=O)NCC(C)S(N)(=O)=O)NC(c1cccnc1NC)=O 28097,Cc1c(F)ccc(C(=O)NC2CC2C(N2CCC(n3cccn3)C2)=O)c1Cl 28098,CCCC(CCC)C(=O)NCCN(C1CCCCC1)CCOC1CCC(C)O1 28099,c1(C(=O)NC(CNC(c2cc(SC)oc2)=O)(C)CO)ccc([N+](=O)[O-])s1 28100,n1(CCC(N2CCC(CNC(c3ccc(CCC)[nH]3)=O)C2)=O)ccc(O)nc1=O 28101,CCCC(C(=O)OC)C(=O)N1CCC(C)(C)C(C(=O)NC(C)C(C)(C)OC)C1 28102,C1(Cl)(C(=O)NCC(C)CNC(c2nncn2C)=O)CC12CCC2 28103,C(=O)(CCN(OC)C(=O)C(CN(C)C)NC(c1ncc[nH]1)=O)NCC(=O)NC 28104,c1(NC2(CNC(C3(C)CNC(=O)C3)=O)COC2)ncnc2sc(C(F)(F)F)nc12 28105,C(=O)(C1=NOC(C)(C)C1)N1CC(C(=O)NCC(COC)C(C)C)C(F)C1 28106,N1(C(c2cnnn2C2CC2)=O)CCN(CC2COCC2O)CC1 28107,c1(N(C(C2CC(C(=O)OC)C2)=O)C)cc(CNC(=O)C(F)C2CC2)on1 28108,C(=O)(C(C)(C)C(F)F)N1CCCC(CNC(C2C(C)(C)C2(F)F)=O)C1 28109,N1(C(CN(C)CC)=O)CCCC12CCN(C(C1CCC(C)=C(C)C1)=O)C2 28110,N1(C(c2c(CC)nco2)=O)CCCC(C(C)NC(c2c(C)nnn2C)=O)C1 28111,C(CCCCCNC(=O)C(Br)=C(C)C)N(C(c1c(CC)cco1)=O)C 28112,c1(C(=O)NC(CNC(=O)C=CC2CCCO2)CO)cc2ccccn2n1 28113,c1(C(=O)NC(C)(CNC(=O)CCS(N)(=O)=O)CO)ccc2c(c1)CCC2(F)F 28114,S(=O)(=O)(c1ccc2c(c1)COCC2)CCC(N1CC2C(C)(C)C2C1)=O 28115,C1(COC)(CNC(c2ccc(CF)cc2)=O)CCCN1C(c1cncnc1)=O 28116,C[Si](C)(C)CCNC(=O)NC1CC1c1ccccc1 28117,Cc1ccccc1CC(C)C(=O)NCCNC(=O)CCN(S(C)(=O)=O)C(C)C 28118,CS(=O)(=NC(=O)CC1CCCCS1(=O)=O)c1ccccc1 28119,c1(NCc2cn(C3CCCN(C(C4C(C)C4)=O)C3)nn2)c[nH]cc(F)c1=O 28120,C12(NC(CC(CC)C(C)C)=O)CCCC(CN(C(c3cccn3C)=O)C1)C2 28121,N1(C(C(C)(C)Cc2cnn[nH]2)=O)CC2CCC(C1)N2C(=O)Cc1csnn1 28122,c1(NCC(=O)NCCCN(C)C(=O)NC)cccc(C(C)=O)c1 28123,Cc1nnc2n1CCN(C(=O)NCc1ccc(C3CCC3)nc1)C2 28124,N1(C(C2CC(C(C)C)OCC2)=O)C2CCCC1CN(C(c1cccc(O)n1)=O)C2 28125,C1(NC(C(C)(C)C)=O)CC2CC(NC(C3CCCN(c4nccs4)C3)=O)C1C2 28126,C(=O)(C(CCCOC)NC(c1ccn(CCF)n1)=O)NC(c1n(CC)ncc1)C 28127,CCC(CC)CC(F)C(=O)N(C(C)CNC(=O)C(C)(C)C1CCOC1)C 28128,CCC(CC(=O)N1CCC(CCO)CC1)NC(C1CCCO1)=O 28129,NS(=O)(=O)CCC(=O)Nn1cc(CC(CO)c2cccs2)nn1.C12CC(C1)C2 28130,Cc1nc(C(N)=O)ccc1CNC(=O)C=CC(C)NC(C1CC1(C)C)=O 28131,N1(C(C2(CCOC)CC2)=O)CCC2C(C1)CN2C(=O)CC1(C(F)(F)F)CC1 28132,C#CC1CN(C(=O)CCOCCN(C(=O)C(C)CC(C)C)C)CCN1C 28133,N1(C(CCC2CCN(C(C(CCC)C)=O)C2)=O)CCCC(C)(CO)C1 28134,Cc1ccc(CN2C(C(=O)NCCC3CCCN3C)CC3CC23)c(Cl)c1Cl 28135,C1(C(N2CCC(OCCNC(C(COC)(C)C)=O)C2)=O)CCc2nccn2C1 28136,N(C1CC(C)n2ccnc21)C(CN(C(C(CNC(COC)=O)O)=O)C)=O 28137,C1(CNC(C2CN3CCC2CC3)=O)CCN(C(=O)Cc2c[nH]nc2O)C12CC2 28138,C(=O)(C1Cc2ccc(Cl)cc21)NC1C2CN(C(C3(C)COC3)=O)CC1COC2 28139,C1(CC(=O)NCCC(N2CCN(C(c3ncccn3)C)CC2)=O)CC2(CCC2)C1 28140,C1(C(C(=O)NCc2ccccc2)N(CCOC)C2CC2)CCOC(C)C1 28141,N1(C(c2ccc(CNC(c3cc(C)sc3N)=O)cn2)=O)CC2CCCCC2C1C 28142,C(=O)(C(C)(C)C(F)(F)F)NCCC1CCC(NC(CCC(=O)NCC)=O)C1 28143,CCCCCCCC(=O)N1CC(C(=O)NCc2ccc(Cl)cc2Cl)C(C)C1 28144,C1(N(C)C)CCCCC1C(=O)NC1CC(C)(NC(=O)CCC2(C)CC2)C1 28145,C1(NC(CCCCN(C(C)C)C)=O)CC2C1CCN2C(C1CCNC1=O)=O 28146,N1(C(c2ccc(C)cn2)=O)CCC2(CC1)CC2(CO)CNC(C1(Cl)CC1)=O 28147,N1(C(C(CC)C#N)=O)CCCC(C(=O)NC2COCC2CO)CC1 28148,N1(C(c2cccc(OC)c2N)=O)CC23CCCC2(C1)CN(C(c1ccc[nH]1)=O)C3 28149,Cc1ccccc1C1CC1C(N1CCCC(C(=O)Nc2cncn2C2CC2)C1)=O 28150,c1(OCC#C)cncc(CN2CCC(SC)CC2)n1 28151,C(CC(C)(C)CC(=O)NCC1CC(C)CCN1C(c1ccc(F)cc1Cl)=O)OC 28152,c1(C(N2CCC(CC=C)(NC(=O)CSCCC(C)C)C2)=O)cnc(C)c(C)c1 28153,CC1C2CCC(C2)C1C(N1CCC(CCC(N2CCC(CO)(CF)C2)=O)CC1)=O 28154,C(C1CCc2nccn21)NC(C1CC(C)(NC(=O)C2=CCCC2)C1)=O 28155,c1(CN2C(C(=O)Nc3ncc(-c4cc[nH]n4)cn3)CC2)ccc(Cl)c(F)c1 28156,c1(N(S(=O)(=O)CCN2CC(=O)NC2=O)C)ccc(C(c2ccccn2)OC)nc1 28157,c1(C(N2CC(C(=O)OCC)C2)=O)cncc(CNC(C2CCCNC2=O)=O)c1 28158,C(C(C(=O)N1CCCC(C(C)(C)O)C1)C(C)C)NC(c1nc(CC)oc1C)=O 28159,C(C(CC1CCCC1)C(=O)NCCCC1CCSC1)NC(CNC(CC)=O)=O 28160,CC(C)(C)C(CC(=O)NOCC1CCOC1)NC(C1CCC1)=O 28161,N1(C(C2C(C(C)(C)C)CC2)=O)CCN(C(=O)CNc2ccccc2Cl)CC(O)C1 28162,CCC(C(=O)OC)C(=O)NC1(CNC(c2cccc(SC(F)(F)F)c2)=O)CCC1 28163,C1(C(=O)NC(C2CCCN2C(c2cnn(C(F)F)c2)=O)C)C2CCC(F)(F)C12 28164,c1(-c2nc(C)c(NCc3cccc(O)c3C)s2)cc(F)c(C(=O)N(C)C)c(F)c1 28165,N1(c2cc(CC)nc(C)n2)CCOC2(CCCN(C(=O)CC3CCC(C)C3)C2)C1 28166,C1(NC(C(C)C2CCC2)=O)CN(C(c2cncn(C)c2=O)=O)CC12CCC2 28167,C1(NC(CCC(C)C2CCC2)=O)CC=C(C(=O)N2CCC(C(F)F)CC2)C1 28168,C(C(C)C(=O)N(C(C)CC(=O)N(CC(C)O)C)C)OCC 28169,N1(C(C(C)NC(N)=O)=O)CCN(C(=O)COCC2CCOCC2)C2CCC12 28170,C(=O)(C(F)CC(C)(C)NC(=O)C=C1CCC1)NC1CON(CC)C1=O 28171,N1(C(C2COCCN(C(c3nn(C)c(CC)c3Cl)=O)C2)=O)CCC(C)C(F)(F)C1 28172,N1(C(C2N(C(C3(C)CCCN(C)C3)=O)CC(=O)C2)=O)CC2(CNC(=O)C2)C1 28173,N1(C(C(C)CS(C)(=O)=O)=O)CCN(C(C2(C)CCN(C)C2=O)=O)CC(C)(C)C1 28174,N1(CC(=O)NCCCN(C)C(=O)NC(C2CCCC2)=O)CC(C)(C)C1c1ccco1 28175,C1(CNC(CCCCOCCC=C)=O)(NC(c2snnc2C)=O)CCCCC1C 28176,C=CCC(CC(F)F)NC(=O)C(CCC1CC1)NC(c1ccncc1CC)=O 28177,C1(CC(=O)NCCCCCNC(C#CC(C)C)=O)CC2(CCOCC2)CO1 28178,C1(NC(C(c2ccc(Cl)nc2)(C)C)=O)CN(C(C2CC(C)(C)C2)=O)CC(F)(F)C1 28179,CCS(=O)CC(=O)N(C)CCOCCN(C)C(c1cccc(=O)o1)=O.C(CCSC)O 28180,n1(CC(=O)NCC2C(CNC(C3CC(CC)C3)=O)C2)ccc2ccccc2c1=O 28181,CC1=C(C(=O)NCCCCC2CN(CC(=O)NCC3CC3)C2)Cc2ccccc2O1 28182,O(NC(=O)CN=c1nc2c(ncn2C)c(NC2C(C3CC3)C2(F)F)[nH]1)CC 28183,c1(C(N2CC(O)(CCNC(C(c3c(C)noc3C)C)=O)C2)=O)ccc(F)c(O)c1 28184,c1(C(N2CC(OC)C(NC(C3(CCF)CCC3)=O)C2)=O)cc2ccnc(C)n2n1 28185,c1(C(=O)NC2CCCC23CN(C(=O)Cc2cccs2)C3)ccc2nccnc2n1 28186,C1(C)(C(N2CC(NC(C(CCC)=CCC)=O)C(F)C2)=O)CCS(=O)(=O)CC1 28187,C(=O)(C(C)(C)CCC(=O)OC(C1CCCN(C(C2CC(=C)C2)=O)C1)C)N(CC)CC 28188,C1(C(N(C2CC(CO)C2)C)=O)CCOC1C(=O)NC1CCCC1F 28189,C1(CNC(c2ccc(C#N)o2)=O)CCCN(C(=O)C(Cn2cccn2)OCC)C1 28190,C(=O)(Nn1nnc2c1CCCC2)C1(C#C)CC1.C1(=O)CC2(CC2)N1 28191,C(=O)(C1=CC2(CCOC2)C1)NCC1N(C(C(CCC(C)C)O)=O)C2CCC1C2 28192,c1(C(=O)O)cccc(Br)c1NC1CCCC(n2ccnc2)C1 28193,c1(C(=O)Nc2cccc(OCCC(C)(C)OC)c2)cccc2c(C)coc12 28194,c1(C(=O)NC(CCOC)CNC(=O)CC2COCC2(C)C)cc2nccnc2[nH]1 28195,C(=O)(CS(=O)C(F)(F)F)NCC(C1CCC1)NC(CCNC(CC(C)(C)C)=O)=O 28196,C1CCC(C)(C)C(=O)N(OC)CCC(=O)N1.C#CCCCOC 28197,N1(C(C2C(CC)OCCC2)=O)CCN(c2nnc(C(C)(C)C)o2)CC(O)C1 28198,CCC(C)C(O)C(C)C(=O)N1CCCC(CCNC(c2cscn2)=O)CC1 28199,N1(C(C2C(OCC)C2)=O)CCCC(C)(C)C1CNC(c1cnn(CC)n1)=O 28200,C1(NC(C(CC=CCC)C)=O)C2CCC1CN(C(=O)CC1CC(F)C1)C2 28201,N1(C(CC2(NC(c3c(CC)ccs3)=O)CCC2)=O)CCC(O)(CO)C1 28202,c1(C(=O)OC)csc(C2CCCN2C(=O)C(N)CSC(F)(F)F)c1 28203,C1(C(=O)NC(CCC)(CC)CC)CCN(C(c2cncc(C#N)c2)=O)C(C)(C)C1 28204,c1(C(=O)NC2C(CC)N(C(c3ccccn3)=O)CC2)ccc(OC)c(Cl)c1F 28205,CC12COCCN(C1)C2=O.c1(NC(C2CC2OC(C)(C)C)=O)cnc(O)c(F)c1 28206,C1(C(=O)NCCC(C)N(C)C(c2ccc(C3CC3)o2)=O)C2CC(F)(F)CC12 28207,Cn1nnc(C(=O)NCCC2CCCCN2C(=O)CCc2ncc[nH]2)c1C(F)F 28208,Cc1nc(NCC2C3CC4CC2CC(Cl)(C4)C3)c2c(n1)SCC(=O)N2 28209,CCC(C#N)(CC)C(=O)NCCC1(C)CCN(C(C2C=C(C)CS2)=O)C1 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28227,c1(OC)cc(C(=O)NCC2(F)CN(C(c3cc(O)no3)=O)C2)c(F)cc1F 28228,C(CCC(=O)N(C)CC1CN(C(c2occc2Br)=O)C1)N(C(C)=O)C 28229,Cc1nc(C)c(C(=O)NCCCN2CCC(NC(=O)CS(N)(=O)=O)CC2)[nH]1 28230,Cc1ccc2c(C(=O)NCC3CC(NC(C4CCS4(=O)=O)=O)C3)csc2c1 28231,C1(C(N(CCOCCNC(c2c(CC)nc[nH]2)=O)C)=O)CN2CCN1CC2C 28232,Cc1ncnc(C)c1CNC1CCCN(CCC(C)(C)C)C1=O 28233,N1(C(C(C)=C(C)C)=O)CCN(C(c2cc(C#N)ccc2C)=O)C2CCC12 28234,C1(OC)CC2(C1)CC(C(=O)NC1CCN(C(c3cnn(CC4CC4)c3)=O)C1)C2 28235,C1(C(N2CC(C(=O)NC)(Cc3ccccc3C)C2)=O)(CC)CCCCC1 28236,N1(C(C2CC(O)(CC#C)C2)=O)CCC(NC(=O)CCC(C)(C)O)C(C)C1 28237,N1(C(CNC(C)=O)=O)CCCC(N(C)C(C2COCC(=O)N2C(C)C)=O)CC1 28238,C1(C(=O)NCC2CC(F)CN2C(c2cc(Br)c[nH]2)=O)CCCC12CCC2 28239,c1(C(N(CCOCCNC(C2(SC)CC2)=O)C)=O)ccnnc1C1CC1 28240,c1(C(N2CC3C(NC(c4c(CCC)nco4)=O)(CC3)C2)=O)cc(N)c(C)cc1Cl 28241,c1(C(N2CC(N(C(CCCOCC=C)=O)C)C3(C2)CC3)=O)cc(C)c(C)cc1C 28242,c1(NCC(CC)N(C)C)ccc(S(=O)(=O)NCC(N2CCOCC2)C)cc1Br 28243,c1(OC)ncnc(N(C2CNC2)C(c2cc(CC(C)C)on2)=O)c1C 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28261,N1(C(c2ccc(C)c(Cl)c2)=O)CCC2(CC1)CC2NC(C1(C)CC=CCO1)=O 28262,C1(CNC(C(C2CCCCC2)OCC)=O)CN(C)CCN1c1cnc(C#N)cn1 28263,C1(C(C)NC(c2cc(Cl)c[nH]2)=O)CCCCN1C(=O)CCc1cccs1 28264,N1(Cc2cc(C)no2)CCC(NC(C2CCC3CCCCN23)=O)C(C)(C)C1 28265,CC1COCCC1NC(C1CC12CC(NC(=O)C(=O)N(C)C)C2)=O 28266,N1(C(C(=O)Nc2scc(C(=O)OCC)c2)=O)CCC2(CC1)CC(O)(C(F)F)C2 28267,c1(C2C(C(=O)NCCN(C(C=CC(C)C)=O)C)C2)cscc1OC(F)F 28268,C1(NC(=O)NC2CC(CO)N(C(=O)CCC3CCCC3)C2)COCCC1CO 28269,N1(C(C2C(C)CC2)=O)CCOC(CC(=O)N(C2CCCCC2)CC2CC2)C1 28270,N1(C(C=C2CCN(C)C2)=O)CCC2CN(C(c3ccc(C(=O)C4CC4)s3)=O)CC12 28271,Cc1cc(C(=O)NCC2COCCN2C(c2cc(C3CC3)nn2C)=O)cc(F)c1 28272,N1(C(CC2(C(F)(F)F)C(C)C2)=O)CC2(C(=O)O)CC2(CO)C1 28273,CC(C)CCC(F)C(=O)NCC1CC(NC(=O)CCC2CC2(F)F)C1 28274,C(CCCC(=O)NCC(C)(O)CNC(c1cccnc1NC1CCCC1)=O)OC 28275,C1(C(N(C(C)C(=O)NCCC2CCCC(C)C2)C2CC2)=O)C2CC3C(C2=O)C13 28276,Cc1ncn(C)c1C(=O)NCC1(C)CCN(C(=O)C(C)N(C)C)C1.NC 28277,C(=O)(CC(F)(F)C(F)F)NCC(CCNC(C1CCC2CC2C1)=O)OC 28278,N1(C(CC=C)=O)CCC2(C(=O)NCCCCCCO)CCCC12 28279,c1(CNC(=O)NC(C2C(c3ccccc3)CCC(=O)C2)=O)nnc2ccccn12 28280,C1(NC(C2(CC)CN(C(=O)Cc3cc(C)ccc3C)C2)=O)C(=O)NCCC1C 28281,C#CCC(C(=O)NC(c1ccccc1)CC)NC(c1ccc(CO)nc1)=O 28282,c1(OC(CC)C)ccc(NC(c2ccc(N3CCC3)c(F)c2)C)cc1C 28283,c1(C(C)N(C(=O)NC2C(C)C2)C(C)C)csc(C(=O)OCCc2cn[nH]c2)n1 28284,C1(NC(C(C)NC(CC)=O)=O)CN(C(=O)CN2CCC(O)CC2)CC2(CC2)C1 28285,c1(C(=O)NCCC(C)N(C)C(c2cccnn2)=O)csc2ccc(F)cc12 28286,c1(OCC)ccc2c(c1)CCC2NC(=O)NC(c1nnc2n1CCNC2=O)C 28287,C(C1=NOC2CN(C(=O)C#CC3CCCC3)CC12)NC(=O)CC1(CO)CC1 28288,c1(C(=O)NCC2(O)CCN(C(c3c[nH]c(=N)s3)=O)C2)ccc2ncnn2c1 28289,C1(C)(NC(CNC(CNC(c2cnc(C(C)C)o2)=O)=O)=O)CCCC1(C)C 28290,CCCCC(C)CCC(=O)NCC1(C)COCCN(C(=O)Cc2cnoc2)C1 28291,N1(C(CCc2cc(C)sc2C)=O)CC(C)OC2(CCN(C(=O)C3CC3)CC2)C1 28292,c1(N2CCC(C=C)CC2)nc(=NCCC2(C)CCCO2)[nH]c2c1cnn2C 28293,C(=O)(C1CCCc2c1ncn2C)NCC(C)(CO)NC(CCc1cc(C)on1)=O 28294,N1(C(c2ccc(CSC)o2)=O)CCC(NC(C2CCN2C(C)(C)C)=O)C1C 28295,c1(NOC(=O)OCc2ccccc2)cc2n(n1)CCCO2.C12(CCCC1)NC2 28296,c1(OC)cc(C(=O)NC2CCC(NC(C3(Cl)CC3)=O)C2)c(C)c(Br)c1 28297,C1(CC(=O)NCCNC(C)=O)CC2(C1)CN(C(c1cc(C)cs1)=O)C2 28298,C1(C(N2C(C(N3CCC3C(C)O)=O)CC(OC)C2)=O)CC2(C1)CC(O)C2 28299,C1(CC(N2CC(=C(CNC(=O)CCC3CCOC3)F)C2)=O)CCC2CC12 28300,N1(C2c3csc(n3)CCNC2=O)CCC(C(C)OC)CC1.n1(CC)cccc1 28301,N1(C(C2CC(NC(C3(O)CCSCC3)=O)CCO2)=O)CCC(F)(F)C(O)C1 28302,CCCCC(C)(F)C(=O)NCCCCCC.C12CC(C1)NC(=O)OCC(=O)NC2 28303,c1(NC)ccc(C(C)NC(C)CC2CCNCC2)cc1 28304,C1(CNC(c2ccc(Cn3cc(-c4ncon4)nn3)o2)=O)CCCOCC1 28305,N1(C(C(C(=C)C)(C)C)=O)CCC2(CCN(C(=O)C(CCC)S(N)(=O)=O)C2)C1 28306,C1(c2ccccc2)(CN2CCC(c3cc(Br)ccc3Cl)(N)C2)CCS(=O)(=O)CC1 28307,n1(CC)cnc2c(NCC3CC3(Cl)Cl)[nH]c(=NCC3(C)CCC(C)(C)CC3)nc12 28308,c1(N(C)C)cc(CNC(=O)C(c2ccc(-c3nn[nH]n3)cc2)O)cc(F)c1 28309,c1(C(=O)NCC(CN(C(c2ccc(SC)o2)=O)CC)(C)C)cnnc(C)c1 28310,C#CCCCCC(C(=O)NCc1ccco1)N1CCC2CCC(C1)S2 28311,C1(NC(C=CC)=O)CN(C(c2ccc(C(=O)OC)cn2)=O)C2CC12 28312,C(COC)(CC(=O)NCCOC)NC(C(CC)=CCC=C)=O.C1(=O)N(C)CCN1 28313,C1(C(C)NC(CN(CC)CC)=O)COCCN1C(c1ccn(C(C)(C)C)n1)=O 28314,C(=O)(C1=CN(C)S(=O)(=O)N=C1C)N(C)CC1N(C(C(C(CC)O)C)=O)CCCC1 28315,C(=O)(CS(=O)(=O)CC(C)C)NCC1C(C=C)CN(C(=O)C(C)(CO)NC(C)=O)C1 28316,Cc1ccccc1-n1ncc(C(=O)NCC2CCCC2NC(=O)C=CCO)c1N 28317,CCN=C(NCCC(=O)NC(=S)SCC)N1CCC(O)CC(C)(C)C1 28318,N1(C(CC2(C)CN(C(c3cccc(-n4cccc4)c3)=O)C2)=O)CC2CCCC2C1 28319,c1(CC(=O)N(CCC(C)NC(=O)CCCCSC2CC2)C)ccc2c(c1)CCO2 28320,C1(NC(N2CC(C)(C)OC(CC(F)(F)F)C2)=O)CCCC1C1CCCC1 28321,c1(C(=O)NCC2CCC(NC(CCCOC(C)C)=O)C2)ccc(C(F)(F)F)cc1 28322,N1(C(c2cc(CC)on2)=O)CCCC2(CCN(C(c3cc(N)cc(O)c3)=O)C2)C1 28323,C1(NC(c2n(CC)ncc2)=O)CC2CN(C(c3cccc4c[nH]nc34)=O)CC2C1 28324,C1(CNC(=O)NC(c2cccc(OC3CCC3)c2)C)CCCCC1C 28325,C12CCC1C(=O)N2.C(=O)(C(C)n1cccc1)NCC1(OC)CC1 28326,N1(C(c2c(CC)con2)=O)CC(NC(c2ccc(C(C)C)nc2)=O)CC1C 28327,N1(C(C(N2CCP(C)(=O)CC2)C)=O)CC2CCC1C(NC(=O)C1=CSCS1)C2 28328,C1(C(N2CCC(CNC(C(C)NC(N)=O)=O)C2)=O)CS(=O)(=O)CC(=O)N1 28329,C(=O)(C(CO)C(C)(C)C)NCCCN(C(c1cnn(CC)c1C)=O)CC 28330,c1(C(=O)NCCC(C)NC(C2CCC(C)(CC)O2)=O)cc(O)nc2c1CCCC2 28331,C1(C(=O)OC)CCCN(CC(=O)NC2CCC(NC(c3ccncc3)=O)C2)C1 28332,CCCC(O)C(CO)NC(=O)C(CCC1CCC1)NC(=O)Cc1cccn1C 28333,CC1=CCCN(C(C2CC(=O)CN2C(C2CC(O)C(F)C2)=O)=O)C1 28334,N1(C(CCOCC)=O)CCC(CO)C(NC(=O)Cc2cccc(C(=O)OC)c2)C1 28335,c1(CC(N2CCC(O)(CNC(C(c3cccs3)SC)=O)C2)=O)cc(F)cc(F)c1 28336,N1(CCCNC(C2(CNC(C(C)NC(=O)NC)=O)CC2)=O)CCCCCC1 28337,c1(C(=O)NCC(C2CCCC2)NC(c2cnn(C)c2Cl)=O)c(F)cc(Cl)cc1F 28338,N1(C(C(CC=CC)C)=O)CCN(C(c2cc(C)n(CC(F)(F)F)n2)=O)CC1CF 28339,O=C1NC(C(N2CCC(n3ccnc3)C2)=O)CO1.c12ccc(s1)CC(=O)N2 28340,C1(NC(C2(CNC(C3C4(CC4)C34CC4)=O)CCCC2)=O)CCN2CCCCC12 28341,CCCC(CC)C(=O)NCC1(F)CCN(C(c2cc(Cl)c[nH]2)=O)CC1 28342,N1(C(C=CC(C)(C)C)=O)CCC(CCNC(C2CN(C(N)=O)C2)=O)C1 28343,N1(CC(=O)NCC2(CN(C)C(C3CCCC34CCC4)=O)CC2)C(=O)NC(C)(C)C1=O 28344,N1(CCNC(C(C)CC2CCCC2)=O)CCC(NC(C2CCOC2(C)C)=O)CC1 28345,Cc1nn(C)c(C)c1C1OCCC1n1cc(OCCO)nn1 28346,c1(C(C(=O)NC2CCOC2)N2CCC2C(=O)NC2CCCC2)ccc(Br)cc1 28347,C(C(C)(C)CN=C(NCc1cccs1)N1CCCC2(CCSC2)C1)OC 28348,C(C)(C(C)C(=O)NCc1noc(C)n1)NC(CN(CCOC)C)=O 28349,C1(COC)CC(CNC(=O)C(C)Cc2ccnn2C)N(C(c2cccn2C)=O)C1 28350,Cc1ccc(CN2CCC(CNC(c3ccn(C4CCCC4)n3)=O)C2)o1 28351,c1(C(N(CC(C)CNC(C2(CN(C)C)CC2)=O)C)=O)coc(Br)c1 28352,CC(C)CC(C(=O)NC(CC1CC1)C(=O)NCCC(C)N1CCCC1)C(N)=O 28353,C12(CNC(=O)C3=C(Cl)CC3)CC3CC(CC(C3)C1NC(=O)CCc1ccoc1)C2 28354,CCCC(C)(CC)C(=O)NC(C1CCCCC1)CNC(=O)C1=CCSC1 28355,c1(C(=O)Nc2cocn2)cc2c(s1)CCN(C(c1cc3ncccn3n1)=O)C2 28356,C12(CC(N3C(COC)(CNC(c4ccn(C)c4)=O)CCC3)=O)CCC(CC1)OC2 28357,C(CC(=O)N1CCN(C(c2ccc(C)s2)=O)C(C(F)F)C1)(C(F)(F)F)OC 28358,C1(CC)(CC)CC(NC(=O)COc2ccsn2)CN1C(=O)CN1CC(C)C1 28359,C1(NC(C=CCCC)=O)CN(C(C2(C)CCN(CCSC)CC2)=O)CCC12CCC2 28360,CCCC(C)(CC)C(=O)N1CC(CC(N2CCCC2C(C)O)=O)(OC)C1 28361,C(C)(C)(C(CO)CO)NC(C1C(CCC)CN(C(=O)C=CC(C)CC)C1)=O 28362,c1(C(N2C(C(=O)NCCCOCCNC(CSC)=O)CCC2)=O)ccc(C#N)cc1 28363,c1(C(N(C(C)CN(C)C(C2CC(CSC)C2)=O)C)=O)cccc(C2CC2)c1 28364,Cc1cncc2cc(C(=O)NC3CCCC3NC(C3CC(=O)NC3(C)C)=O)sc12 28365,N1(C(c2c(C)c[nH]c2)=O)CCC2(C=C(C(=O)NC3Cc4ccccc4C3)C2)C1 28366,CCCC(CNC(C1CCCC1O)=O)C(=O)NCC1CCC1(F)F 28367,N1(C(c2c(C)n(C)nc2)=O)CCC(C2CC(NC(C3(C)CCCS3)=O)C2)CC1 28368,CC1CC(CCNC(=O)CCOC2CC2)CCN1C(=O)CC(Cl)Cl 28369,Cc1cc(C(=O)NCC2(C(N3CC(N4CC(F)C4)C3)=O)CC=CC2)ncc1F 28370,CC(C)CC(F)(F)C(=O)NCC1CC(C)CCN1C(C1CCCCC1(C)C)=O 28371,C1(NC(C(CCCCC)O)=O)CCN(C(c2ncc(C)cc2C)=O)CC12CCC2 28372,C1(CC)OCCC1C(N1CCC(CN(C)C(c2coc(CO)c2)=O)C1)=O 28373,CC1CCC(CNC(c2ccc([N+](=O)[O-])[nH]2)=O)CN1C(C1CCC(=O)O1)=O 28374,c1(OC)ccnc2c(Cc3csc(=NCc4cocc4C)[nH]3)cccc12 28375,C(=O)(C(C)(O)C(F)(F)F)NCC(CC(C)C)(C)NC(=O)CCn1cnnn1 28376,N1(C(c2c(COC)scc2)=O)CCN(C(C2CCCOC2)=O)CC1C1CC1 28377,CC(C)C(CNC(=O)CCc1cc(Cl)no1)NC(C1CCCOC1)=O 28378,Cc1ccc(N)c(C(=O)N(CC(C)(C)NC(=O)C(C2CCCCC2)F)C)c1 28379,C(CNC(=O)C=CCF)(CC(=O)N1CCCC1C1(C)CC1)OC 28380,c1(C(=O)NCC(CCNC(C2(C)CC3CC3C2)=O)O)ccc2oncc2c1 28381,c1(OC)cc(NC(=O)CN2CCC(NC(=O)CC(C)(C)O)CC2)ccn1 28382,N1(C(c2cc(CCNC(C3CC4CCCC4C3)=O)on2)=O)CCC12CC(O)C2 28383,N12CCCC(CC1)C(=O)NC(C1CCC1)C2=O.N1(CC)CCC(N2CC=CC2)C1 28384,c1(C(=O)NC(CCOC)CNC(=O)Cn2cccc2)ccn(C(C)C)c1C 28385,Cc1cccc(C(O)C(=O)NCCC2(NC(=O)CCc3ccsc3)CC2)c1 28386,C1(C(=O)NCC2C(C)(C)C2)CN(C(C2C3CCCCC23)=O)CC1(F)F 28387,C(=O)(C(C)(C)C(C)O)N(CCOC)CCNC(c1ccncc1N(C)C)=O 28388,CCC(CCC(=O)NC1C=CCN(C(=O)CCc2ccc(C)s2)C1)OC 28389,Cc1csc(=O)n1Cc1cn(-c2cccc(N)c2)nn1.C12CC(C)N(C1)C2 28390,CC1(C)CN(C(=O)CC2CCC3(CCC3)O2)CCN(C(C2CCOC(=O)N2)=O)C1 28391,C1(CCC)(C(=O)NC)CCCN(C(=O)C(c2ccccc2OC)OC(C)C)C1 28392,Cc1n[nH]cc1CC(N1CC(F)(CNC(C23CCC(C2)C3)=O)C1)=O 28393,n1(CC)nnc2cc(C(=O)NCC(O)CNC(C3CC(CCO)C3)=O)ccc12 28394,C1(CCCC)CN(C(c2c[nH]c(=NC)o2)=O)CCN1C(c1cccnc1)=O 28395,C(=O)(C1=CCCOC1)N(C)CC=CC(=O)NC(C1CCCC1)CNCC 28396,C=CCCC(F)(F)C(=O)NCC1CN(C(c2cnn(CCC)c2C2CC2)=O)CCO1 28397,c1(C(=O)NCC2C(NC(c3c(OCC=C)cccn3)=O)C2)cc2cc(O)ccc2[nH]1 28398,c1(C(N(C2CCN(C(=O)CSC3CC3)C2)CC#C)=O)cc(Cl)n(C)n1 28399,N1(CC#C)CC(NC(c2ncoc2COC)=O)C2(CCOCC2)C1 28400,C1(C(N2CCC(c3cccc(F)c3)CC2)=O)CC2CC2N1C(C1CC1F)=O 28401,c1(SC)ccc(CC(=O)NC2CCCC(NC(=O)Cc3ccc(Cl)cn3)C2)cc1 28402,C1(O)(CN(C)C(C2CCC3(CCC3)C2)=O)CCCN(C(c2nc(=O)n(C)[nH]2)=O)C1 28403,c1(C(=O)NC(C2CCCC2)CNC(C(CC=C)CC)=O)cccn2nccc12 28404,C1(C(C(=O)NCCC(C)N(C(=O)CC2(C)CC2)C)OCC)CC(F)(F)C1 28405,C(CC(=O)NC1CCCN(C(C2(OC)CC2)=O)C1)(C(N)=O)OC.N1(CC)CCOCC1 28406,c1(C(=O)NC2CCN(C(C3C4CC(=O)CC43)=O)CC2O)cc(O)c(Br)c(O)c1 28407,c1(NC(C2(CNCc3c(C)cccc3)CC2)=O)cccc2nscc12 28408,C(=O)(CC(F)(F)F)NC1(COC)CN(C(=O)C(F)(F)c2cscn2)C1.C1(=O)CN1 28409,c1(C(N(CC(O)CN(C)C(c2ccnc(C(F)(F)F)n2)=O)C)=O)cncc(N)c1 28410,c1(OC)cc(C(=O)NC(CNC(C2CC(=C3CC3)C2)=O)C2CC2)c2occc2c1 28411,C(=O)(CC(O)c1ccccc1)NCC(C)N(C)C(C1(C)CCCC1)=O 28412,CCC(C)(C)CCCC(=O)NC1(CNC(c2ccc(CC(C)C)cc2)=O)CCCC1 28413,c1(C(N2C3C(NC(CSCC=C)=O)CC(C3)C2)=O)cccc2nccnc12 28414,c1(C(=O)NCc2ccsc2C(N2CCC2C2CCC2)=O)n[nH]cc1[N+](=O)[O-] 28415,C(=O)(C(F)(F)F)NC(C)C(=O)NC1CN(C(C2CSC2)=O)C1 28416,CCC(C(=O)NCC1CN(C(c2ccc(C)nc2C)=O)CC1(F)F)C(C)C 28417,c1(NC(C)=O)c(C(N2CCC(NC(=O)CCC3CC(C)C3)C2C)=O)cccc1C 28418,C#CC1CN(C(=O)CCc2cc[nH]n2)CCN1C(c1cnc(O)o1)=O 28419,CN1CCC(C(=O)NN2CCC(C(=O)NC3C(O)CC3O)O2)=NC1=O 28420,c1(C(=O)NC2C3CN(C(C4(SC)CC4)=O)CC32)ccc(F)c(C(C)C)c1 28421,C1(C(=O)NCc2nc(CNC(c3csc(C)n3)=O)cs2)(CC)CCN(C)CC1 28422,N1(C(C(C)NC(=O)CNc2ccccc2)=O)CCOCC(NC2(C)CC2(F)F)C1 28423,C1(C(C)OC(OC=CC(=O)NC)=O)CCCCN1C(C1(C2CCCCO2)CC1)=O 28424,N1(C(CCC=C(C)C)=O)CCOC2(C1)CN(C(=O)C(C)Oc1ccccc1)C2 28425,CC1CCC(C)(C(=O)NCCCN(C2CCCC2)C(=O)CN2CC3CC3C2)CC1 28426,Cc1ccnc(O)c1C(=O)NCC1CN(C(=O)CC(C)C)CC1C 28427,S(=O)(=O)(c1ccc(C)c(C)c1)N(CCCNC(=NCC)NC(C)C1CC1)C 28428,C1(NC(=O)Cn2cccn2)C2CC3C1C3C2C(=O)NC1(c2ccc(Cl)o2)CC1 28429,CC1CN(C(c2cncnc2C2CC2)=O)CC1NC(c1ccc(CC(N)=O)cc1)=O 28430,Cc1ccc(O)c(C(N2CCN(C(=O)CSc3cnn(C)c3)C(C3CC3)C2)=O)c1 28431,CC1CCCCCN1C(=O)CSCCNC(c1cncn(C)c1=O)=O 28432,N1(C(C#CC(C)C)=O)CCCC(C)(NC(c2cc3n(c2)CCC3)=O)C1 28433,c1(C(=O)NC(C)CNC(C2(Cc3cncnc3)CC2)=O)ncc(Cl)cc1F 28434,C1(C(N2CC(C(=O)Nc3c(C)non3)N(C)CC2)=O)CCc2nnc(O)n2C1 28435,C1(NC(CCOCC(C)C)=O)CC2CN(C(c3ccc(F)c(O)c3)=O)CCN2C1 28436,C1(C)(NC(CC2CCN(C(C3CCN(C)CC3)=O)CC2)=O)CCC(C)(C)C1 28437,c1(C(=O)OCC)cccnc1C(N1CC=CC(CNC(=O)C=C2CCCC2)C1)=O 28438,c1(CC(=O)NCC2(F)CN(C(Cc3cc(C)on3)=O)C2)cnc(Cl)cc1C 28439,C1(O)(CC(=O)N(C(C)CNC(=O)C(c2ccc(Cl)s2)C)C)CCCCCC1 28440,CC1=C(C(=O)NC(C2CCN(C(c3coc(C)n3)=O)CC2)C)CCCO1 28441,c1(C(=O)NC2CC(C)(C)N(C(C3COCCO3)=O)C2)cc(F)cc2nn[nH]c12 28442,C1(NC(c2csnn2)=O)C2CC1CN(C(C1CC3(C1)CC31CC1)=O)C2 28443,C(=O)(C(C)(C)COC(C)=O)N(CC(=O)NCCCCO)CC=C.C1(O)CCCC1 28444,C(c1cccc(F)c1)=CC(=O)NCC(C)(C)OC1CN(C(=O)CCCC(N)=O)C1 28445,c1(C(N(CCCCC)CCNC(=O)CC2CCOC2(C)C)=O)cc(C)ncc1C 28446,CC1(C(=O)N2CCC(C(C)(C)NC(c3cn[nH]c3)=O)C2)COc2ccccc21 28447,C(=O)(CCS(=O)(=O)CC(C)C)N1CC(NC(Cc2cc(C)on2)=O)C(CO)CC1 28448,c1(C(=O)NCCC2(C)CN(C(c3cnc(C(F)F)nc3)=O)C2)cc2n(n1)CCC2 28449,CC(CN(C)C)CC(=O)NCC1CCCCC1NC(=O)C(F)(F)C1CC1 28450,N1(C(C2ON=C(CC)C2)=O)CCC(O)C2(CCN(Cc3ccncc3Br)CC2)C1 28451,c1(C(N2CC(CNC(c3c(OCC)scc3C)=O)C2)=O)ccc(=O)n(C2CC2)c1 28452,CC(=NO)C1CC(C(N2CC(NC(=O)COC3CCCC3)C(O)C2)=O)C1(C)C 28453,Cc1cccnc1C(N1CC(CC(C)NC(c2cncc(C(C)(F)F)c2)=O)C1)=O 28454,N1(C(CCC2N(C(c3ccc[nH]3)=O)CCCC2)=O)CCc2ccncc21 28455,Cn1nc(C(=O)NC2CC2NC(C2CC3(CC3)CO2)=O)cc1C1CC1 28456,c1(-c2ccc(CN3CCN(CCC(=O)OC)CC3)cc2)ccc(Cl)c(CO)c1 28457,c1(CCC(=O)NCC2C(C(N(CC(C)(C)N(C)C)C)=O)CC2)ccccn1 28458,C1(C(N(CCCNC(=O)C(O)P(C)(C)=O)C(C)C)=O)CCn2nccc2C1 28459,c1(C(C)C)ccncc1C(=O)NC1COCCC1NC(C12CSCC1C2)=O 28460,c1(OC)ccc(F)c(C(N2C3CCC2C(C(=O)NCC(C)OC)C3)=O)c1 28461,C1(CN)CC(Cn2ccnc2)CN1C(=O)Cc1nc[nH]n1.n12cc(nn1)C2 28462,c1(C(=O)NCC(C)=CC(N2CC(C)CCC2C)=O)cccc2cc[nH]c12 28463,C(CC(=O)N1CCC(CCNC(c2cn(C3CC3)nn2)=O)C1)(C(C)C)OCC 28464,c1(-n2ccc(C)n2)ccccc1C(=O)NCC(F)CNC(C1CCOCC1)=O 28465,C1(NC(CN(C(CC2CCC(C)(C)O2)=O)C2CC2)=O)CC2(CCCC2)C1 28466,N1(C(Cc2cncc(C)c2)=O)CC(F)(F)CC1CNC(c1nc(C)ccc1C)=O 28467,c1(C(N(CCN(C)CC2CCC(C)(C)CC2)C)=O)occ2c1CCC2 28468,N1(C(C2C(CCC)C2)=O)CC(NC(=O)C=C2CCCCC2(C)C)C2CCCC12 28469,c1(NC(CCOC2CN(C(C3C(C)(C)COCC3)=O)C2)=O)ccc2cc[nH]c2n1 28470,O=C(Cn1cccc1)N=c1cc(C2CNC2)[nH][nH]1.c1(C=O)ccsc1Cl 28471,C(C(=O)OC)(C(C(=O)OC)N(C1CC1)C1CC1)Sc1ccc(C(=O)OC)cc1 28472,C(=O)(C(SC(F)(F)F)C1CC1)N(C)CC1(NC(=O)CSC(F)F)CC1 28473,c1(C(N2CCC(NC(c3c(C)noc3)=O)C(C)C2)=O)scc2c1CCCC2 28474,C1(CC)CCC(C(=O)N(C2(C(N3CC(C(F)(F)F)C3)=O)CC2)C)CC1 28475,C1(CNC(CC)=O)CN(C(=O)CCc2ccc(C(=O)OCC)cc2)CCO1.C(=O)N 28476,c1(NC(C(C(=O)OC)OC)=O)ccc(NC(=O)COCCCF)c(C)c1 28477,C1(C(N2CC(c3cn(CCOC)nn3)(O)C2)=O)CCC(C(=O)NCCO)CC1 28478,n1(C(C)C)ncc2cc(-c3ccc(NC(=O)CN4CCOCC4)cn3)cnc12 28479,CCC(C(C)c1nn[nH]n1)NC(=O)CC1(NC(=O)C=CC2CC2)CCC1 28480,C#CCCCCC(=O)NC1CCN(CCNC(=O)CC2CCCS(=O)(=O)C2)CC1 28481,N1(C(C2(OCC)CCC2)=O)CCCCC1CNC(=O)C(c1cccc(F)c1)O 28482,Cc1cn2cc(C(N3CCN(C4CN(C(=O)C=CS(C)(=O)=O)C4)CC3)=O)sc2n1 28483,C1(C(=O)NC(C=C)CO)CCCCN1C(c1cncn1CC)=O 28484,c1(C(=O)NC(CNC(C(C)NC(C)=O)=O)(C)CO)cccc(CS(C)=O)c1 28485,C1(NC(CC2(NC(C)=O)CC2)=O)CN(C(=O)C(C)CC(=O)OC)CC(C)(C)C1 28486,CC1(C)CC1(C#N)N(CCOCc1cccc(Cl)c1)C(=O)NC1CC1 28487,Cc1cnc2cc(C(N3C4CCC3C(CNC(=O)COCC(C)C)C4)=O)ccn12 28488,c12c[nH]c3cc(cnc13)-c1ccc(cc1)CN(CC)C2.c1(NC)ccccc1C 28489,C(=O)(CC(C(F)F)C(C)(C)C)NCCCN(C(c1cccc(OC)c1)C)CC 28490,c1(C(=O)NCC2C3CN(C(COCCCC)=O)CC32)c[nH]c(=N)nc1C(F)(F)F 28491,C1(C(=O)NC2C(OC)CCC2)(C)CC12CCC2.C12(CCCC1)C(=O)N2.C(C)(C)S 28492,C1(C(=O)NC(C)(C)CNC(c2[nH]ccc2-c2ccccc2)=O)CCC2(CCC2)O1 28493,C(C)(C(=O)NC(C1CCC1)CO)N(C(=O)C=CCF)CC 28494,c1(C(=O)NC2CCCN(C(C(C)c3cc[nH]n3)=O)C2)ccc(N)c(Cl)c1O 28495,c1(C(=O)NC2CCCC23CCN(c2nnco2)CC3)ccnc2ccc(Cl)cc12 28496,C(=O)(CC(C)(C)C1CCCCC1)N(CCNC(C1CCC(C(N)=O)N1C)=O)CC 28497,N1(C(C=COCC)=O)CCCC2(CCC(NC(c3cc(C)c(C)nc3O)=O)C2)C1 28498,n1(CC)nccc1C(c1nnnn1C1(C)CC1)NC1CCN(c2ccccn2)C1 28499,c1(C(=O)NC2CC3(C(NC(Cc4n(C)ncc4)=O)C3)C2)cccc2c1C(=O)NC2 28500,Cc1cc2[nH]c(C(=O)NCC(C)N(C)C(C34CC(C3)C4)=O)cc2s1 28501,C1(NC(C(CCCC)O)=O)CC2CC(NC(C3(S(N)(=O)=O)CC3)=O)CC2C1 28502,c1(CC(c2ccc(C)o2)O)nc(C2CC2C(F)(F)F)nn1C1CCS(=O)(=O)C1 28503,C12(CC(=O)NCC3C(CNC(CCCCCSC)=O)C3)CCC(CC1)C2(C)C 28504,N1(C(CC)=O)CCc2cc(C(=O)NCCNC(C3(C)CCC34CCC4)=O)ccc21 28505,N1(C(Cc2c(C)ccc(C)c2)=O)CC2CCC(C1)C2CC(N1CCC(C)C1)=O 28506,c1(C(=O)NCC2(C)C(C)CN(C(C3COC(=O)C3)=O)C2)nnn2c1CCCC2 28507,CC1CN(C(=O)OC(C)(C)C)CC(CNC(=O)Nc2nc(CCO)ncc2N)O1 28508,C1(C(N2CCOC(CNC(=O)C=Cc3ccccc3)C2)=O)(OC)CCC(C)CC1 28509,C(=O)(C(C)(F)C(C)(C)F)NCc1ccc(CNC(CCS(C)=O)=O)cc1 28510,Cc1ccc2c(c1)CC(C(=O)NCC(C)N(C(=O)CCSc1nccn1C)C)O2 28511,N1(C(C2C(CNC(CC(CC(C)C)C)=O)CCC2)=O)CC2C(=O)NC(=O)C2C1 28512,Cc1sc(C(N2CCC(OCC(C)(C)NC(=O)C(C)CN(C)C)C2)=O)c(C)c1C 28513,N1(C(CCC=CC)=O)CCOC(C)C1C(=O)NC(C)CNC(N)=O 28514,C(=O)(CCCCC(=O)NC(C(=O)N(CC(=O)N(C)C)C)C1CCCO1)OC 28515,C=C(C)CCCC(=O)NC(CNC(=O)CC1(O)CCCCCC1)C(C)C 28516,C(CC(C(=O)NC1CCCN(C(c2cccc(C(N)=O)c2)=O)C1)OC)OC 28517,N1(C(C(C)=C2CCC2)=O)CCC2(CO)CN(C(=O)Cc3cccc(F)c3)CC2C1 28518,CCC(CC(=O)NC(C)(C)C(C)CC(=O)N1CCCC1C1(CO)CC1)C(F)F 28519,c1(C(=O)NC2CC(CCNC(C(C)C3(O)CCC3)=O)C2)coc2c1C(=O)NCC2 28520,N1(C(CCC=C(C)C)=O)CCN(C(=O)C(C)(C)CCF)CC1c1ncc[nH]1 28521,C1(NC(COCCCOC)=O)CCN(C(C2CC2C2CC2)=O)CC1F 28522,C(C)(CNC(=O)C(Cl)=CCl)(CC(C)C)NC(C1(C=C)CC1)=O 28523,Cc1c(C(=O)NC(C)(CNC(=O)C(C)CC2CCC2)C(C)C)nnn1C(C)C 28524,c12ccc(o1)CNC2=O.n1(C(C)C(=O)O)cc(-c2ccccn2)nn1 28525,c1(C(=O)NC(C)(Cc2ccccc2)C(=O)O)ccc([N+](=O)[O-])cn1 28526,C1(OCCNC(C23CC(F)(C2)C3)=O)CN(C2CC2)CC12CCC2.C(C(=O)C(=O)N)NC 28527,N1(C(=O)NC2CC(c3ccc(Br)cc3)C2)CCC12CC1CCC2C1 28528,C1(C)(C(=O)NC(CN2CCN(C(C=CC(C)C)=O)CC2)C)CC2CCC(C1)S2 28529,c1(CNC(CC(=O)NCCC2(OCC#C)CC2)=O)ccc2c(c1)C(=O)CCC2 28530,C(=O)(CCCC(=O)OC(C)(C)C)NC1CCCC(NC(c2c(C)scc2)=O)C1 28531,c1(C(=O)NC2C(NC(CCOCCN(C)C)=O)CC2)ccc(C(C)(C)C)nc1 28532,C1(NC(c2cc(C)c(C)[nH]2)=O)CS(=O)(=O)C12CCN(c1ncc(Cl)cn1)CC2 28533,c1(NC(c2cncc(Nc3nc(SC)c(Br)cn3)c2)=O)c(C)cc(C)nc1Br 28534,c1(-c2ccc(OCC#C)cc2)ccc2c(NC(=O)C3CC3)cnn2c1.C1(CC(=O)OC)CCO1 28535,c1(CC(=O)N(C(C(=O)NCCN(C)C)C2CCC2)C)cccnc1 28536,C(=O)(CC(CC)OC)NCC(C(=O)NCC(C=C)(C)C)C1CCC1 28537,C1(NC(C(CCC)O)=O)CCN(C(c2cc(NC(C)=O)ccc2C)=O)C12CC2 28538,c1(NC(C2(C(C)(C)O)CC2)=O)ccc(O)cc1.C12CC(C)(C1)CNC(=O)C(=O)N2 28539,CCCCC(CC)C(=O)NCC(C)C(N1CCC2(CC(F)C2)C1)=O 28540,C1(C)(c2cn(CC(=C)CC)nn2)CCCN(C(C)=O)C1.Cc1sc(Br)cc1 28541,N1(CCC)C(=O)CCC1C(=O)NCC(C)(C)CN(C(=O)Cn1nc(C)nc1C)C 28542,c1(CC)cn2c(C(=O)NC3CCN(C(c4ccoc4)=O)C3C3CC3)cccc2n1 28543,Cc1c(CS(N2CCCC(OC3CCOC3)C2)(=O)=O)cccc1Br 28544,CC1CN(C(c2ccn(C)c(=O)c2)=O)C(C)CN1C(C1CCNC1=O)=O 28545,C1(N(C(=O)COCc2ccncc2)C)CCCN(C(=O)CCOCC(F)F)C1 28546,C1(CC)(NC(=O)C(F)F)CCN(C(=O)C(C)(C)C)CC1 28547,c1(NC(=O)NCC2C(CC)C2)ccc([N+](=O)[O-])cc1-n1cnnn1 28548,CCC(CC)CC(F)C(=O)N1CSCC1C(=O)NC1(c2cc[nH]n2)CC1 28549,c1(C(=O)NC(C)CN(C)C(c2ccns2)=O)cccc2c1NCCNC2=O 28550,c1(C(=O)NC(CC)CNC(C2(C)CC(C)=NO2)=O)sc2cncn2c1C 28551,c1(C(=O)NC2CCN(C(C(CC)n3ccnc3)=O)C23CC3)cccc2[nH]ncc12 28552,c1(C(C(=O)N(C2CCCO2)CCCF)N2CCC2)cc(Cl)ccc1F 28553,C(=O)(C1=CCC(NC(C2(O)CCCCC2)=O)C1)NC(CC)C1CC1 28554,n1(CC)nc(C)c([N+](=O)[O-])c1NCC1CC(NC(C2CCCCC2O)=O)C1 28555,C1(NC(c2c(OCC=C)cccn2)=O)CN(C(c2cc[nH]c2C)=O)CC2(CC2)C1 28556,N1(C(Cc2c(C)scc2)=O)CCC(C)(O)C1C(=O)NC(c1nnc(O)o1)C 28557,c1(C(=O)NC2C(NC(C(C)Oc3ccc(Cl)cc3)=O)CC2)cccc(C(F)F)n1 28558,CC(C)CCC(F)C(=O)NCC1CC2CCCC2N1C(=O)C=C(Cl)Cl 28559,N1(C(C=CC(C)(C)C)=O)CCCC(C2CCN(c3nc4ccccc4o3)C2)C1 28560,C1(CNC(CSCC=C)=O)CC(NC(=O)C(c2cccc(Cl)c2)N(C)C)CC1O 28561,C1(C(=O)OC)CC(F)(F)CN1C(c1cc(C)c(C)s1)C(=O)NC(C)C 28562,C1(CNC(C(CC)(C)C)=O)C2CCCC1N(c1ccc(-c3cnco3)cn1)C2 28563,C1(NC(CC(CC=C)(C)C)=O)CC2(CCC(CNC(C3C4COCC34)=O)CC2)C1 28564,n1(CC)cc(C#N)cc1C(N1CCCCC1)C(=O)NCC1CCCCCC1 28565,CCCC(C)(C)CC(=O)NCC(=O)OCCn1cc(COC)nn1 28566,N1(C(c2c(COC)nn[nH]2)=O)CC(CNC(C2(C)CCN(C)C2=O)=O)CC(C)C1 28567,C(=O)(C(O)CC(C)(C)C)NCC(C)C(F)C(=O)NCc1cnn[nH]1 28568,c1(C(N2CCC(N(C(c3cnsn3)=O)CC)C2)=O)cc(Cl)cc(Cl)c1F 28569,c1(OC)nccc2c(C(N3CC4C(NC(c5cc(C)oc5C)=O)C4C3)=O)c[nH]c12 28570,N1(C(CCCc2nc(C)sc2)=O)CCCCC(NC(c2n[nH]c(C)c2F)=O)C1 28571,C12(CNC(=O)NC(C(C)C)c3ncc[nH]3)CC3CC(CC(C3)C1)C2 28572,c1(C(C(=O)NCCC(C)NC(Cc2cc(CC)no2)=O)(C)F)ccccc1F 28573,CC1(CC(N2CC(NC(C3(O)CC3)=O)CC3CC23)=O)CCS(=O)(=O)N1 28574,C(C1CCCN1C)=CC(=O)NC(c1ccccn1)C(=O)NCC1CC(=C)C1 28575,CC(C)(C(=O)N1CCC(N(c2ncccn2)C2CCC2)C1)c1ccsc1 28576,C12(NC(C(=O)NCCNC(C)=O)=O)CCC(NCC=Cc3ccnn3C)(C1)OC2 28577,c1(CNC(c2n(C)cc(Cl)c2)=O)ccc2c(c1)CN(C(=O)Cc1cc[nH]n1)C2 28578,c1(C(=O)NCCCC2N(C(CSCCOC)=O)CCCC2)cccn2nncc12 28579,N1(C(C=CCCC)=O)CCCC(C(=O)NCc2conc2C)CC1 28580,c1(C(N(C2CN(C(c3cc(Cl)cnc3O)=O)CC2F)C)=O)ccc2nonc2c1 28581,C1(NC(=O)Cc2nc(C3CC3)cs2)CN(C(c2cc(Cl)ns2)=O)CC12CCC2 28582,C(=O)(CCCCN1CCCC1)N(C1CN(C(=O)CC2CCC3CC23)C1)C 28583,c1(CC(N2CC(OCC)C(n3cc(C4CCC4)nn3)C2)=O)cc(C)cc(Br)c1 28584,Cc1ccc(C(=O)NC(C)(CNC(=O)C(F)F)C(C)C)c(=O)n1C 28585,c1(C(C(=O)NCCC(CNC(c2c(CC)csc2)=O)OC)SC)ccccc1F 28586,c1(C(=O)NC2CC(NC(C(c3scc(C)n3)C)=O)C2)cc2nccnc2cc1C 28587,c1(OC)ccccc1C(=O)NCC1CCC1NC(C1(C)CC=CCC1)=O 28588,C(=O)(CCCCCS(N)(=O)=O)N(C)CCN(C)C(C1(O)CN2CCC1CC2)=O 28589,c1(C(c2n(CCCC)nnn2)NCc2ccccc2C)nnc2n1CCC2 28590,c1(C(=O)NC2(C(=O)NCC(C3CCCCC3)O)CCSC2)cc(F)ccc1F 28591,c1(OC)ccc(CN(C=O)C(C)C)c(NC(=O)COc2ccccc2Br)c1 28592,C1(C(=O)NC2CCN(C(c3c(C)nc(C4CC4)o3)=O)CC2)CC2CCCCCC12 28593,C1(C(=O)NCC2=CCN(C)CC2)COC2(C1)CN(C(C1(N(C)C)CC1)=O)C2 28594,N1(C(CC2(C=C)CCC2)=O)CC(NC(C2(CC)CCCC2O)=O)C(CO)C1 28595,c1(OC)ccc(C(C)CNC(C2CCC2(C)C)=O)cc1 28596,c1(C(N2CCC(NC(CSCCCC)=O)C2C)=O)cc2cccnc2cc1F 28597,c1(C(N(CC(C)NC(=O)COCC2(F)CC2)CC)=O)c(F)cc(OC)cc1F 28598,c1(C(NOCC2(C)CC2)=O)cccnc1C(=O)NCC1CC(O)C1(C)C 28599,CC1CCC(C(=O)N(CCNC(c2cncc(C(F)F)c2)=O)C2CC2)CC1 28600,C1(C(F)(F)F)(OC)CC(NC(=O)NC2C=CCC2)C1 28601,Cc1csc(=O)n1CC1CCC2CC12.c12ccc(cc1)COC2=O 28602,C12(CNC(Cc3cncc(C)c3)=O)CCCC(CN1C(c1nc(O)c(C)s1)=O)C2 28603,N1(C(C2CN(CCC)C(=O)C2)=O)CCN(C(C2CCC2)=O)C(CCO)C1 28604,CC(C)CCC(=O)NC(c1ccccc1F)CNC(c1ccco1)=O 28605,N1(C(=O)CSc2cccc(F)c2)CCC2C3CCC(C3)C12 28606,Cc1cc(O)c(C(=O)NC(C2(O)CCN(C(=O)CN3CCC(C)C3)CC2)C)nn1 28607,CCC(CCC(=O)NCC1(C)CC1(C)C)NC(=O)CCN(C)CC 28608,C1(C(N(CCN(C(=O)CC2CC(C)(C)CO2)C(C)C)C)=O)CCC(O)CN1C 28609,C1(OCC)CC2(CCC(C(=O)NNC(=O)NC3CCC4CCCCN4C3)CC2)C1 28610,N1(C(CCc2ccc(C)nc2)=O)CCC(C)C(NC(c2ncc(F)cc2C)=O)C1 28611,c1(C(=O)NCCCN(C(C(C)OC)=O)CCO)csc2ccc(F)cc12 28612,N1(C(CC2(OC)CC2)=O)CCCC(C)(CNC(C2CC(C)CO2)=O)C1 28613,C(CCO)(C(=O)N1CCCC1Cc1cn(C(C)CN2CCCC2)nn1)N(C)C 28614,c1(NC(=O)NCC(c2ccccc2Cl)SC(C)(C)C)nccc2nn[nH]c12 28615,CCCC(F)C(=O)NC(CC1CC1)C(=O)N(CCO)CCOC 28616,Cc1nnc(O)c(C(N2CCCC(C)(NC(=O)C(O)C(C)C)C2)=O)c1C 28617,N1(C(C2C(OC)CCOC2)=O)CCC(CO)(CNC(C2(F)CCCC2)=O)CC1 28618,C=CCCCC(=O)NCC(=O)N(Cc1cnc[nH]1)CC1CCCO1 28619,c1(C(N2C(C3(O)CN(C(=O)CO)C3)CCC2)=O)cnc2n1CCCC2 28620,C12CCCCCN(C1)C(=O)N2.c1(CC2(OCC)CC2)ccccc1.C12CC1C(=O)N2 28621,c1(C(=O)NCC(CNC(c2cc(C)no2)=O)S(C)(=O)=O)ccn2ncnc2c1 28622,C(=O)(C(O)C(C)(C)C)N(CC)CC1CCN(C(c2cc(C)no2)=O)CC1 28623,C#CCS(=O)(=O)CCNC(=O)C(=O)NC1(C#N)CCCCC1 28624,C(=O)(C(=O)C(C)(C)C)NCC1(OC)CCN(C(=O)CCn2ccccc2=O)C1 28625,C1(CNC(C2(C)CC2(F)F)=O)CN(C(c2cn(CCO)nn2)=O)CC1(C)C 28626,c1(NC(C2CC(NC(CNC(CCC)=O)=O)C2(C)C)=O)n[nH]c2ccccc12 28627,c1(OC)nn(C)cc1C(=O)NCC12CC1CN(C(c1sccc1CC#N)=O)C2 28628,C(=O)(C(C)(C(C)C)NC(C)=O)N1CCC(CCNC(C(CCC)OC)=O)CC1 28629,CCC(COC(c1ccn(-c2ccccc2)n1)=O)CC(F)(F)F 28630,N1(C(C=CCC)=O)CC(C)(CNC(C2CCCC(C)(C)C2)=O)CC1(C)C 28631,c1(OC)ccc2[nH]c(C(N3CC=CC(NC(=O)CC4CCC4)C3)=O)cc2c1OC 28632,N1(C(CNC(CC)=O)=O)CC2CC(O)C1C2NC(=O)COCCN1CCCCC1 28633,N1(C(C2N(C)CCC2)=O)CCCC2(CCN(C(c3n[nH]cc3Cl)=O)C2)C1 28634,C(=O)(C1=CCCCO1)NC1C(C)(C)C(CC(=O)Nc2ccc(CO)nc2)C1 28635,c1(C(=O)NC2C(NC(C3(C(=O)OCC)CC3)=O)C2)occc1C 28636,N1(C(C(c2ccccc2F)OCC)=O)CCCC(CO)(CC2C3COCC23)C1 28637,C(=O)(CCC(C)(C)[N+](=O)[O-])NCC1(NC(C2CCC(C(=O)OC)O2)=O)CCOC1 28638,C1(C(C)(C)C)(CNC(C(OC)OC)=O)CCN(C(c2nc(C(C)C)oc2C)=O)C1 28639,c1(NC(CN(C(=O)C(CC)=CCCC)CC=C)=O)ccc(N(C)C)cc1 28640,C(=O)(C(CC(C)C)NC(c1coc(CSC)n1)=O)N(C)Cc1[nH]nc(CC)n1 28641,N1(C(C2(C)CCN(S(=O)(=O)C3CCCCC3)CC2)=O)CCc2ccc(F)cc2C1 28642,C(=O)(C(C)(C)CCC(=O)OC)NC1CN(C(c2ccc(NC)cc2)=O)CC(O)C1 28643,C(=O)(CC(C)C(C)(C)C)NC1CC=C(C(=O)NC2CCN(CCOC)CC2)C1 28644,Cc1nc2ncc(C(N3CC4C(NC(C5CC=CC5)=O)C4C3)=O)cc2o1 28645,C1(C(C(CC2CC(=O)C2)=O)=O)CC(O)C1NNCC(=O)NC1CCC1 28646,c1(C(c2nnnn2C2CCC2)NC(CC)=O)csc(C2CC2)n1.C1C(=O)O1 28647,N1(C(CC2CC(C)C2)=O)CCC(C)(NC(c2cccc(N3CCOC3=O)c2)=O)C1 28648,CC(C)CS(=O)(=O)CC(=O)N1CC(O)CC1CNC(c1ccccc1)=O 28649,C(=O)(CCC(c1ccccc1)NC(=O)CC1(C)CCCCC1)OCC 28650,CC1(C)CC(CC(N2CC(NC(c3ccc(Cl)o3)=O)C(C)(C)C2)=O)CCO1 28651,N1(CCNC(c2cnn(-c3ccccn3)c2C(F)(F)F)=O)Cc2nccc(Cl)c2C1 28652,c1(C(=O)NCCN(CCC)C(c2cccc(CF)c2)=O)nn(C)c2c1CCC2 28653,N1(C(CCC(=O)NCC#C)=O)CCN(CCOCC=C)CC1=O 28654,n1(CCCOC(=O)C(O)Cc2cnc[nH]2)cc2ccccc2n1 28655,c1(OC)ccc(C)c(NC(C2COCCN2C(c2ccncc2C)=O)=O)c1 28656,C12(CCC)CN(C(=O)C3CC(=O)O3)CC(C(F)(F)F)(C1)C2.C(C)(C)(C)OC(C)=O 28657,CC(=O)CCN=C(NCc1cc(C)ccc1O)NC1CC(C)(C)C1 28658,C1(C(N(CCCNC(C2CCN(C)C2)=O)CC)=O)CC12CC(C)(C)C2 28659,C(C1C(C(=O)OC(C)(C)C)C1(C)C)=C(C)C.c1(C2C(=O)O2)ccccc1 28660,N1(C(c2cn(CCNC(C3C(OC)CCC3)=O)nc2)=O)CC(C)C1(C)C 28661,c1(N(C)Cc2c(C)n[nH]c2)ccc(CN2CCC(C(F)(F)F)C2)cc1 28662,N1(C(c2c(OC)nccc2)C(=O)Nc2ccc(F)cc2)CCCC(C)(O)CC1 28663,CC(Cl)(Cl)C(=O)NCC(C1CCOC1)NC(=O)C=Cc1cc[nH]n1 28664,C1(C(=O)NCc2nnnn2C2CC2)CN(C(c2cccnc2NC2CC2)=O)CC1O 28665,c1(CC)nc(C)c(C(=O)NC(C)(C)CNC(c2cn(C(F)(F)CO)nn2)=O)s1 28666,CCCC(C(=O)N1CC(O)(C(F)C(N2CCC23CC(C(N)=O)C3)=O)C1)C(C)C 28667,c1(C(=O)NC(CN(C(c2cc(C)[nH]c2)=O)C)C)cc(C#N)ccc1C 28668,c1(CSCC(C)OC)cc(C)c(-c2ccccc2)s1 28669,c1(NC(C)C)ccc(C(=O)NCCCCNC(=O)CC2CC(C(F)F)C2)cn1 28670,C1(CNC(C(C=C)OC)=O)CN(C(c2ccn(C3CCC3)n2)=O)CC1(C)C 28671,c1(OC)ccc(Cl)c(C(=O)NC23COC(CNC(c4cccnc4N)=O)(C2)C3)n1 28672,N1(C(C2(CCC)CC2)=O)CC(NC(=O)Cc2ccccc2O)CC(C)(C)C1 28673,C1(C2CCC2)(C(=O)NCC2N(C(=O)Cc3ccccc3F)CC2)CC1(F)F 28674,c1(NC(C(CCC)CNC(C2(C#N)CCOC2)=O)=O)ccc2nncn2c1 28675,C1(CCNC(C=C(CC)C)=O)CCN(C(=O)COc2cncc(Cl)n2)C(C)C1 28676,C1(c2nnnn2C(C)(C)C)(NCC2(SC)CCCC2)CCCC2CC12 28677,C(=O)(C(F)C(C)CNC(c1cc(C)cc(O)c1)=O)NCCOC 28678,CCC(C(=O)NCCC1(OC)CCC1)NC(c1cc(O)cs1)=O 28679,Cc1cc(F)ccc1CC(=O)N(C)CC1CN(C(c2cocc2C)=O)CC12CC2 28680,C=CCCCCCN(C1CC2CC1CN2)C(=O)CC(O)c1ccccc1 28681,C(CCCCC(=O)NC1CCC1CNC(C1CCCN(C(C)C)C1)=O)OC 28682,C1(NC(CCS(C)=O)=O)CCC2(CCN(C(=O)CNC(=O)CC3CCCC3)C2)C1 28683,Cc1cccc(CC(N2CC(O)(C(C)NC(C3CCC(C)(O)CC3)=O)C2)=O)c1F 28684,C1(O)(CC(=O)N(C)CC2CCN(C(C3C(CC)OCC3)=O)CC2)COC(C)(C)C1 28685,C1(C(N(C2CC3CC3C2)C)=O)CC(NC(=O)C=CC2CC2)C12CCC2 28686,N1(C(C2N(CC)CCCC2)=O)CC(C)(C)CC1C(=O)NCC1(C)CCCCCC1 28687,N1(C(CCc2n(C)ccn2)=O)C(C(=O)NC2CCOC2)CC2CCCC12 28688,c1(C(C(=O)NC2CN(C(C=CCN(CC#C)C)=O)C2)C)cccc(Cl)c1 28689,C1(NC(CCC)=O)CCC(CCCC)CC1.c12cccc(c1)CNC(=O)C2 28690,c1(OC)cc(C(=O)NC2CCCC2NC(C2(F)CC2)=O)cnc1O 28691,C(=O)(CCCCCNC(N)=O)NCC(CNC(CC1(COC)CC1)=O)O 28692,c1(-c2c(OC)ccc(C(C)C)c2)cncc2sc(C(=O)Nc3conc3C)cc12 28693,c1(OC)c(C(=O)C(=O)C)cccc1Br.C1(CC(C)N)CN(C(C2CCC2OC)=O)C1 28694,C1(C(N2CC(C(C)O)C2)=O)CCC(O)CN1C(c1sccc1CO)=O 28695,C(=O)(N=c1[nH]nc(-c2ccc(F)cc2)s1)c1cn(C(C2CCCC2)C)nc1 28696,C(CCC(C)(C)NC(C1CSCN1C(=O)C(C)OCCN(C)C)=O)OC 28697,C12(NC(C(C)Sc3ncccn3)=O)CCCCCC1N(C(=O)CC(C)(F)F)CC2 28698,N1(c2sc(C#N)c(Cl)n2)CCC2(NC(c3ccc(Cl)cn3)=O)CCCC12 28699,Cc1cc(C(N2CC3CC(NC(c4ccc[n+]([O-])c4)=O)C2C3)=O)n2nccc2n1 28700,c1(C(N(c2scc(C)n2)C)C2CC2)nc(-c2ccccn2)c(C)o1 28701,N1(C(c2c(CNC(C3(C)C(C)CCC3)=O)cco2)=O)CC2CCCCC2C1 28702,C1(C(=O)NCC2CC2)(C(=O)NCCO)CC=CC1.CC1C(=O)N(C)CCCO1 28703,C(C(=O)NCC1CCC(F)(F)C1)(C(C)CC)N(C(c1c(CC)cno1)=O)C 28704,C1(C(=O)NCc2cn(Cc3cccs3)nn2)CC12CCOc1ccccc12 28705,N1(C(CC=CC)=O)CCC2CCCC12CNC(=O)CCc1ccc(CC)cc1 28706,C1(C(N(C2CCN(C(C3(CC)CCC3)=O)C2)CC)=O)CC(C)(C)CN1C 28707,C1(O)(CCNC(c2c(C(C)C)ocn2)=O)CCCN(C(=O)C(F)(F)C(F)F)C1 28708,N1(C(CCC2OCC(C)C2)=O)CCC2CN(C(c3cnc4cc[nH]c4c3)=O)C2C1 28709,c1(C(=O)NCCC2CC(NC(C3CCC3)=O)C2)cnoc1-c1ccccc1 28710,c1(C(=O)NCC2CC(NC(C(C)=C3CCC3)=O)CC2O)ccnc2c1ccn2C 28711,c1(CNC(CC(=O)NCC(C)C)Cc2cccs2)cccc(F)c1I 28712,C1(N(C)C)(C(=O)OCCCC2CCC2)CC2CCC1C2 28713,C1(OCC)CC(NC(C2CC23CCC(F)(F)CC3)=O)C12CCCCC2 28714,C(=O)(C1=CC2(CCOCC2)C1)NCC(C)(C)CNC(C1CC1c1ccccc1)=O 28715,N1(C(c2c(C)cco2)=O)CCN(C(c2csc(-c3ncc[nH]3)n2)=O)C2CC12 28716,N1(C(CC(=O)NCC)=O)CC(C(=O)NCC(F)CO)CC12CCC2 28717,C1(O)(CCNC(c2c(CC)c[nH]n2)=O)CCCN(C(C2CC(O)(CC)C2)=O)C1 28718,CCCCC(C(=O)N1CC(O)(C2CC2)C1)NC(C1CC(O)C1)=O 28719,c1(C(=O)NC2C3(CC(NC(CCC(=O)NC)=O)C3)C2)oc2ccccc2c1Cl 28720,c1(C(C)NCC(C2CCCC2)OC)nnnn1C1CCOCC1 28721,C#CCC(C(=O)N1CCCC(CC(N2CC(C(=O)OCC)C2)=O)C1)C1CC1 28722,C12(C(=O)NC3C(C)(NC(c4c(C)nn[nH]4)=O)CCC3)CC=CCN1CCC2 28723,N#Cc1cccc(F)c1NC(C1CCC(NCc2cnccc2Cl)C1)=O 28724,C1(c2c(C(N(C3CN(C(C4(C)CCCO4)=O)C3)C)=O)nco2)CCC(F)(F)CC1 28725,C(=O)(CC(C)CC(F)(F)F)NCC#CCNC(c1ccc(OC)cc1F)=O 28726,C(=O)(C1CCCc2nn(C)cc21)NCCN(C1CCS(=O)(=O)C1)C(CC)=O 28727,C1(F)(C(N2CCN(CCCCCNC(C=CCC)=O)CC2)=O)C2CCCCC12 28728,Cc1cc(CO)cc(NC(C2CN(C(=O)NCc3cccnc3)C2)=O)n1 28729,c1(Sc2ccc(NC(=O)NCC3CCC(OC)CC3)cc2)cnc2[nH]cncc1-2 28730,N1(C(COCC(C)=O)=O)CCC(C(N2CC3CCC(C2)N3C)=O)C12CCC2 28731,Cc1ccnnc1C(=O)N(C)CCOCCN(C(=O)C#CC(=O)N(C)C)C 28732,N1(C(C2(CC)CCCN(C(C3CCCN3C)=O)C2)=O)CC2(CCCCC2)C1 28733,C(CNC(C1CC(NC(c2ncsc2CC)=O)C1)=O)(C(C)C)OCC 28734,C1(N(C(C2C(NC(CCC=C(C)C)=O)C2(C)C)=O)C)COCC1(C)C 28735,CC1CCN(C(c2ccc(Cl)cc2N)=O)CC1N(C(=O)CSc1ccccc1)C 28736,C=CC1(CNC(=O)NCCN(C)C(C)C)CCC1 28737,C12(CNC(C(C)CC(N)=O)=O)CCC(CN(C(c3ccc4occc4n3)=O)C1)C2 28738,N1(C2CCN(CC(C)F)CC2)CCN(C(=O)CCc2cccnc2)C(=O)C1 28739,C=CCC(CC)C(=O)NCC1CNC(=O)CN1C(=O)CC1CCOC1=O 28740,N1(C(C(c2cccs2)SC)=O)CCC2(CCN(C(=O)Cc3cc[nH]n3)CC2)C1 28741,C(CC(=O)NCC1CC2CCC(C1)C2)(C(C)CC)NC(C(C)=CC=C)=O 28742,N1(C(Cc2ncn(C)c2)=O)CC2CC(N(C)C(C3CCC4(CC3)CC4)=O)C1C2 28743,Cc1nccc(C(=O)NC2C3CN(C(c4ccccc4)=O)CC23)c1O 28744,C#Cc1ccc(C(N2CCN(C(=O)Cc3ccoc3C)C3CC23)=O)cc1F 28745,CC1=NOC(=O)C1CC(=O)N(C)CC1CCN(C(c2cnc[nH]2)=O)CC1 28746,N1(C(c2cc(COC)n(C)n2)=O)CC2CC1CN2Cc1ccc(C(=O)OC)cc1 28747,C(=O)(C#CC1CCOCC1)NC(C1CCCCC1)C(=O)NC1C(C)C1C 28748,c1(C2(C(=O)NCc3cccc(C(F)(F)F)n3)CCCC2)ccc(Br)cc1 28749,N1(C(C(N2CCOCC2)C)=O)C2CCCC1CN(C(=O)CN1CCCCCC1)C2 28750,C1(C(c2ccccc2F)C(=O)O)C(C(O)=COc2nn[nH]n2)=NOC1 28751,c1(C(C)=O)ccc(C2CN(C(c3ncnn3C)C(=O)NC3(C)CC3)CCO2)cc1 28752,N1(C(c2ncc(Br)cc2C)C(=O)NCCCSCC)CCC2(CO)CCCC12 28753,c1(NC(c2n(CC(=C)C)nnn2)c2cccs2)ccc(SC)cc1OCCC#N 28754,Cc1cccc(CNC(C2(C)CC(NC(=O)C(C)S(C)(=O)=O)C2)=O)c1O 28755,c1(C(=O)NC2(CCCCNC(C3CC4(CC4)CO3)=O)CC2)cccc(CO)n1 28756,N1(CC(CCC)O)CCOc2cccc(OC(F)(F)F)c2C1 28757,C1(C(=O)NCC2(CNC(C3COCCOC3)=O)CC2)CCC=CCC1 28758,C=C(C)CC(C(=O)N(C)C)NC(c1nocc1OCC)=O 28759,C(=O)(CC(CC)C1CCC1)NCC1N(C(C(=O)NCCOC)=O)CC1 28760,C1(CS(N2CCCC(c3cnc[nH]3)C2)(=O)=O)CC2CCCCC2O1 28761,CN1CCC(O)(CNC(c2cc(CNC(c3cc(Cl)no3)=O)[nH]n2)=O)C1 28762,N1(C(C2(C)CCC(=O)C2)=O)CCC(C)(C)C(NC(c2ccc(F)s2)=O)C1 28763,C1(CCNC(CCc2c(C)cccn2)=O)CN(C(C2CCOC2=O)=O)CCCO1 28764,C(N=c1[nH]c(=NCC2=CCCCC2)c2cccc(F)c2[nH]1)C1CCCC(CC)C1 28765,c1(C(c2nnnn2C)NCc2n(CC)ncc2)sc(Br)c(C)c1C 28766,Cc1cnc(NC(=O)C(=O)Nc2ccnn2C2CCCCC2)c([N+](=O)[O-])c1 28767,c1(NC)ccc(Cl)c(C(=O)NC2CN(C(c3cc4n(n3)CCC4)=O)C3CC23)c1 28768,C1(N(C)C(C2CC2c2cn(C)nn2)=O)CCCN(C(c2cnn(C)c2Cl)=O)C1 28769,N1(CC)CC(C(=O)NC2(CCO)CCCC2)C(C)C1.C(=O)C=CCO 28770,C(=O)(CCC(F)(F)CN=[N+]=[N-])NCC1(O)CCN(C(c2ccn(CCC)n2)=O)C1 28771,C1(CNC(COCCOC)=O)CC(C)N(C(C2CCC(F)(F)C2)=O)C1 28772,C1(C(N2CCC(NC(CCC(N)=O)=O)CC2)=O)C2C3CC4C1C1C2CC3C41 28773,c1(SCC)ccccc1CC(=O)NCCC1CCN(C(C2CC3(CC3)C2)=O)CC1 28774,CC1(C)CCC(C(=O)NC2C3CC2N(C(=O)C=Cc2nccs2)C3)CC1 28775,C(=O)(CCCC(C)(C)C)N(CCC(=O)NCCC(O)C(C)C)CC=C 28776,N1(C(c2nc(C(C)C)sc2)=O)CC2CC(NC(=O)CN3CCOC3=O)C2C1 28777,N1(C(c2[nH]c3cc(C)oc3c2)=O)CCCC2CN(CC3(C)OCCO3)CCC12 28778,C(=O)(CCC(C)(F)F)NCC(CNC(c1cccc(OCCOC)c1)=O)OC 28779,CCC(C(=O)NCC1(OC)CN(C(=O)CC(C)F)C1)N(C)C 28780,Cc1sc(NC2CC2)c(C(N(CC(C)NC(C2CC2C)=O)C)=O)c1C 28781,c1(CN(C(=O)C(n2cc(-c3cncnc3)nn2)C)CC)cc(C)ccn1 28782,C=Cc1ccc(C(=O)NCC2CCC(F)(CNC(c3ccns3)=O)CC2)cc1 28783,CN1CCCC(F)(C(=O)NC(C)CCN(C(=O)CCCc2cccnc2)C)C1 28784,c1(CNC(C2C(NC(CC(C)(C)OC)=O)CCOC2)=O)cnc(C)cc1C 28785,Cc1cc(CNC(=O)COCCNC(C2CC=CCO2)=O)sc1C 28786,C1(NC(CS(=O)(=O)NC)=O)CN(C(=O)CCC2CC(F)(F)C2)CCC1O 28787,C1(NC(COCCC=C)=O)CC(C2CCN(C(=O)C=Cc3cccc(C)c3)C2)C1 28788,c1(CC)nccn1C(C)CC(=O)NCC1(NC(=O)CCc2ccccn2)CC1 28789,c1(C(=O)NC2(C(C=CC(N3CC(CC(C#C)C)C3)=O)OC)CCC2)ccc(F)s1 28790,c1(C(N(CCCN(C)C(C2CSCCS2)=O)C)=O)ccc(-n2cccn2)nc1 28791,N1(C(CCc2cncc(OC)c2)=O)CCC(NC(=O)CCc2nc[nH]n2)C(O)C1 28792,C1(C(N(C2CCCN(C(c3cnn(C)n3)=O)C2)CC)=O)CCC(C)CC1 28793,c1(CC(=O)N(C2CCN(C(=O)CNC(=O)C3CC3)CC2)C)ccc(=N)[nH]c1 28794,C(=O)(C1=CCCN(C(c2ccc(OC)cc2)=O)C1)NC12CC(C(C)(F)F)(C1)C2 28795,CCC(CC(C)C)(c1nnnn1C)NCCn1nnnc1-c1cc(Cl)ccc1Cl 28796,C=C(Cl)C(C)(C)C(=O)NC1CCN(C(c2ccc(CN3CCCC3)o2)=O)C1 28797,O=C(C1=CCS(=O)(=O)C1)NCC1CCN(C(c2ccsc2Cl)=O)C12CC2 28798,C1(C(=O)NCCCn2ccnc2)CCCN(CC(C)Oc2ccccn2)CC1 28799,Cc1ccc(F)c(C(N2CC(NCc3cc(Cl)ncc3Br)C(F)C2)=O)c1 28800,C(CCS(C)=O)(C(=O)N1CCC(CCNC(c2ccc(Cl)c(F)c2)=O)C1)N(C)C 28801,C(=O)(C1=CCC(C)CC1)N1CC(CC)(NC(C23CCCC2C3(F)F)=O)C1 28802,C(=O)(CCCCC(=O)Nc1ccccc1N(C)C)c1ccc(OC)cc1 28803,C12(CO)CCN(CC1)C(=O)c1cccc(Cl)c1CC=CCC(=O)N2.CO.SC 28804,c1(SCCC(=O)NC(CCNC(C2(OCC)CCC2)=O)CC)ncnc2[nH]cnc12 28805,C1(NC(CC(=O)NCC#C)=O)CCC2(CCN(C(C3(SC)CCC3)=O)C2)C1 28806,C1(CNC(Cc2c(C)noc2Cl)=O)CC(O)CCN1C(=O)Cc1cnc[nH]1 28807,N1(C(c2c(C)nn(CC(F)(F)F)c2)=O)CCN(C(C2(C)CC3CC3C2)=O)CC1C 28808,CC(CCCO)(N=c1ccn(C(F)F)[nH]1)c1nnnn1-c1ccc(F)cc1 28809,C1(CC(=O)NC(c2c(C)nccc2)C)C2CCCC2N1C(=O)C(C#N)C(C)C 28810,C(=O)(CC(O)CC(C)(C)C)NC1C(OC)CN(C(c2c(CCC)n(C)nc2)=O)C1 28811,C(c1cccc(F)c1Cl)=CC(=O)N(C(CN(C(CCNC(COC)=O)=O)C)C)C 28812,c1(C(N(C2CCOC2)CCNC(C(C2CCCC2)OC)=O)=O)ccccc1 28813,c1(C(N2CC(c3c(CNC(c4ccon4)=O)nco3)C2)=O)cccc(C(F)F)n1 28814,C1(C(=O)NC2(COC)CCN(C(=O)CCCC(F)(F)F)C2)CC2C=CC1CCC2 28815,c1(CC(=O)N=c2cc(C3CCCCC3F)[nH][nH]2)cc2c(cc1Br)CCC2=O 28816,c1(CC(=O)NCC(C)N(C(=O)C(C)n2cccc2)C)cn(C)nn1 28817,c1(NC(=O)CCN(c2ccc(Cl)o2)CCCO)ccc(Cl)cc1F 28818,CC(C)CC(C)(CNC(=O)C=CS(C)=O)NC(c1cnc2ccsc2c1)=O 28819,c1(C(=O)OC)cc(C)cnc1N1CC(NC(C2CC(=O)N(C)C2)=O)C1 28820,Nc1cc(C(N2CCCCCC2c2cccnc2)=O)c2c(c1)OCCO2 28821,c1(CC)cccc(C(=O)N(CCCNC(=O)CCSCC(N)=O)CC)n1 28822,N1(Cc2c(OC)ccc([N+](=O)[O-])c2)C(=O)Nc2cc(Cl)ccc2S1(=O)=O 28823,S(=O)(=O)(c1ccc(N2CCn3ncnc3C2)cc1Br)NCCOCCC 28824,C#Cc1ccc(Cl)c(C(=O)NC2CCCC(NC(c3cnsc3C)=O)C2)c1 28825,c1(OC(C2CCC(=O)N2)=O)ccccc1-c1ccc(NCCC2OCCO2)s1 28826,C1(C(N(C2CCC(C)C2)C)=O)CCCN(C(c2coc(C3CCCC3)n2)=O)C1 28827,c1(NCc2c(F)cccc2F)cccc2c(Br)cccc12 28828,C1(NC(=O)CONC(=O)CC2C=CCCC2)(CF)CCOCC1 28829,C(N=c1[nH]c(=NCC2CN(C3CCC3)C2)[nH]c2ccsc12)c1c(C)cccc1Cl 28830,c1(C(=O)NC2(CNC(C(C)(C)c3ccno3)=O)CCC2)c[nH]nc1[N+](=O)[O-] 28831,N1(C(c2c(OC)nccc2)=O)CC2CC(NC(c3cc(C(N)=O)[nH]n3)=O)CC1C2 28832,C(=O)(C1CCCc2nncn21)N1CC2CN(C(c3cc(Cl)cc(Cl)c3)=O)CC2C1 28833,N1(C(C(C=C=C)C)=O)CCN(C(c2cc(C)ns2)=O)C(c2ccnn2C)C1 28834,c1(CC)ccc(-n2nc(CCOc3ccccc3)nc2C2CC2F)cc1 28835,c1(C(=O)NCCC(=C)CNC(=O)CCn2ccnn2)c(Br)cnn1C 28836,C(N=c1nc2scnc2c(N2CCOCC(F)(F)C2)[nH]1)c1n(C)nnn1 28837,C1(C(=O)N(C)CC2(C)CCCO2)(NC(C(CO)OC)=O)CCCCC1 28838,CC1(C)C=C(C(=O)Nc2cccc(NC(C3CC3c3cccc(Cl)c3F)=O)c2)C1 28839,c1(OCC(=O)NC2CC(C)N(C(C3CCOCC3)=O)C2)cncc(C#N)c1 28840,c1(C(N2CCC(NC(C(CCC)OCC)=O)C2(C)C)=O)cc(F)cc(Cl)c1N 28841,c1(C(=O)NCC2(F)CN(C(=O)C=C3CCC3)C2)cc2cccc(Br)n2c1 28842,c1(C(N2CC(N(C(=O)C(c3ccnn3C)O)C)C2)=O)cccc(C#CC2CC2)c1 28843,C(c1nc2cc(Br)cnc2o1)=C(C)C(C)(C)C 28844,CC1(CNC(c2ccc(CNC(c3cccc(F)c3F)=O)o2)=O)CCCCC1O 28845,c1(CNC2CCCN(C(=O)Nc3cc(Cl)c(Br)cn3)C2)ccccc1[N+](=O)[O-] 28846,C(=O)(C1=C(Cl)CCOC1)N1CCC(C(N2CC(CC)NC(=O)C2)=O)C1 28847,Cn1ncc2nc(Cl)nc(N3CCCC3(C)C(=O)NCC34CCCCC3C4)c12 28848,N1(C(c2ncc(Br)s2)C(=O)NC2CCCC2)CCCC2OC(c3ccccc3)CC12 28849,c1(CC)cn2c(n1)CC(C(=O)NCC(C)N(C)C(c1cc(C)cc(O)c1)=O)CC2 28850,N1(C(C(C)Oc2ccccc2)=O)CC2CC2(NC(c2ccn(C3CCC3)n2)=O)C1 28851,c1(CC)ccc(F)c(C(N2CCN(C(=O)CCOCC(F)(F)F)C3CC23)=O)c1F 28852,n1(CCC(N2C(CCCNC(C(C)OC)=O)CCC2)=O)ccc2ccccc12 28853,C1(C(=O)NC2CN(C(C=C(C)C(C)(C)C)=O)C3C2C3)(CF)CCC(F)(F)CC1 28854,CCCCC(C)CCC(=O)NC(CNc1snc(Cl)c1C#N)C(C)(C)C 28855,C(=O)(C1=C(C)OCCS1)N1CC(OCC)C(CNC(C2CCC(C)(C)OC2)=O)C1 28856,N1(C(C(C)Oc2ccc(OC)cc2)=O)CC2CN(C(=O)C(C)C)CCC12 28857,N1(C(C2=CC(C)(CC)C2)=O)CC2CC(C1)CN(C(c1cc(Br)c[nH]1)=O)C2 28858,c1(OC)ccc(C(C(=O)NCCOC(C)(C)C)N(CC(F)F)CCO)c(Cl)c1 28859,N#CC1CCN(C(C2CN(C(c3ccnc(O)c3F)=O)CCC2O)=O)CC1 28860,c1(C(c2n(CCOC)nnn2)NCCS(C)=O)ccc2ccn(C)c2c1 28861,c1(C(=O)NC2CC(NC(c3c(CC)n(CC)nn3)=O)C2)ccnc2ccncc12 28862,C(=O)(C1=CCOCC1)NCCC(CNC(C1CCN(C)C1=O)=O)OC 28863,CN1N=C(C(=O)Nc2cccnc2C(=O)NCC(N2CCCC2)=O)CCC1=O 28864,c1(C(N2C(C)C(NC(=O)CCc3csc(=N)[nH]3)CC2)=O)csc2c(F)cccc12 28865,c1(C(C)C)ccc(CN2CCN(C(C)C(=O)NCC(c3cnoc3)=O)CC2)cc1 28866,c1(OC)nc(C)ccc1C(=O)NCC1(C)CN(C(c2c[nH]nc2F)=O)CCO1 28867,c1(C(N2CC(CC)N(C(=O)CCC(=O)OC)CC2)=O)cc2c(C)nn(C)c2s1 28868,c1(SCCC)cccc(C(=O)N(CC(C)(C)NC(C2CCOC2=O)=O)C)c1 28869,CC1CC2CN(C(=O)C(CO)C(F)(F)F)CC2N1C(=O)CCC(=O)C1CC1 28870,c1(CCC)cc(C(N2CC(C(C)(C)O)(CNC(C3CC3(C)C(F)F)=O)C2)=O)no1 28871,Cc1noc(C)c1C(C)C(=O)NCC1(CNC(C2(C)CNC(=O)C2)=O)CC1 28872,n1(CC)nc(C(N2CCN(C(c3ccco3)=O)C(C(C)=O)C2)=O)c(Br)n1 28873,c1(C(=O)NC2C(SC)CN(C(=O)CC3CCCC3O)C2)cc2c(cn1)OCCC2 28874,Cc1cc(C)n(CC(=O)NCCCCNC(=O)CC2CC(C)(C)CO2)n1 28875,c1(NCC)cc(C(=O)N(C2CC(NC(=O)C(C)(C)CO)C2)C)cnc1OC 28876,c1(N(C(C)CNC(c2ccc[nH]2)=O)C)scnc1NC(=O)OC(C)(C)C.C=CC 28877,CCCC(C)(C)CC(=O)NC1C(C)(C)C(NC(=O)CN2CSCC2=O)C1(C)C 28878,Cn1cccc(C(=O)NCC2CN(C(C3(F)C4CCCC34)=O)CC2O)c1=O 28879,C1(NC(CSS(C)(=O)=O)=O)CCN(C(=O)CCN2CCCC2=O)CC1C(N)=O 28880,c1(C(=O)NC(C(C)(C)C)CNC(C2CC3(CSC3)C2)=O)cc(Cl)ccc1F 28881,C1(NC(C=CC)=O)CN(C(=O)C(O)Cc2cccc(Cl)c2)CC2(CCOCC2)C1 28882,C1(C2CCN(C(C34CCC(CC3)C4(C)C)=O)C2)(NC(c2c(C)snn2)=O)CC1 28883,C12(COC)CCNCC1CN(C(=O)CCOC(C1CCN(C(C)=O)CC1O)=O)C2 28884,c1(CN(C(C(C=C)OC)=O)C)cc2c(=O)[nH]c(C)cn2n1.C1CC(C(C)C)N1 28885,N1(C(C(C)C2CNC2)=O)CCCOCC1.CC(C)O 28886,C1(C(=O)NCCCC2(NC(=O)C=CCF)CC2)COc2c(F)cc(F)cc2C1 28887,c1(CNC(C(COC)C)=O)ccccc1CN(C(=O)C=CSC)C 28888,C(C(C(=O)N1OC2CCC1C2)NC(=O)CNCc1cccnc1)SC 28889,C1(CC)CCN(C(c2cccnn2)=O)C1C(=O)NC(C1(O)CCC1)C 28890,N1(C(C)=O)CCCC1(C)C(=O)NCC1C=CCN1C(=O)CCOCC1CC1 28891,C1(CC(=O)N(CC(O)CO)C(C)C)CCN(C(C2OCCC2(C)C)=O)C1(C)C 28892,c1(C(=O)NCC(=C2CN(C(c3nc(OCC)oc3)=O)C2)F)cccc(C(C)C)c1 28893,C(=O)(CCCC1CC1)N(C(C1(C(=O)NC(CC)C2CCC2)CC1)C)C 28894,Cc1[nH]c(C)c(C(=O)NCCCNC(c2cccc(N(C)C)c2)=O)c1C 28895,c1(C(N2C(C)(CCC)CC2)=O)cccc(-c2n[nH]cc2CC2CCCC2)c1 28896,c1(C(=O)NCC2(O)CCN(C(C3(CC4CC4)CC3)=O)C2)csc2ccc(F)cc12 28897,C1(NC(C(C)SCC)=O)CC(C(=O)N2CC=CC2(C)CO)=CC1O 28898,c1(C(N2CC(OC)C(NC(=O)C=Cc3cnc[nH]3)C2)=O)sc([N+](=O)[O-])cc1Cl 28899,CC1CCN(C(=O)C(O)C2CCCC2)CC1NC(=O)CC=Cc1ccccc1F 28900,C1(NC(c2c(CC)ocn2)=O)C(C)CN(C(=O)C2=C(C)CCCC2)CC1C 28901,C1(NC(CSCC(C)C)=O)CCN(CCCNC(C2CCS(=O)(=O)C2)=O)CC1 28902,N1(C(=O)Nc2c(C(=O)OC)ccs2)CCN(C(c2cnccc2C)=O)CC1C#N 28903,c1(N(CC=CCC2CCN(C(=O)CC(F)(F)F)CC2)CC)cccc(OC)c1C 28904,C1(CCC)CCC(C(=O)NCC(C)N(C)C(c2cnc(OC)s2)=O)CC1 28905,c1(C(C)C)ncc(C(=O)NC(C)C(C)(C)NC(C2CC(n3ccnc3)C2)=O)s1 28906,CCCCC(O)C(=O)NCC(CC1CC1)C(=O)NC12CCC(CC1)C2 28907,C1(NC(CC(C)C)=O)CCCCCN(C(C23CC(CC(F)F)(C2)C3)=O)C1 28908,c1(CC(=O)NCC(Cn2cc(-c3ccn(C(F)F)n3)nn2)OC)cccnc1F 28909,c1(C2(N(C(C)CNC=O)C)CC2)ccccc1OC.c1(OC(C)(C)C)ccccc1F 28910,C(CC(C(=O)NC(C(C)(C)O)C1CC1)NC(=O)CCc1ccc(C)o1)=CC 28911,N1(C(C(C)=CC2CC2)=O)CCC(C(=O)NC2(CO)CCC2)(CF)C1 28912,Cc1sc(-c2ccccc2)nc1C(=O)NC1CN(C(C2CCCO2)=O)C1 28913,C1(C(=O)NCC(CN(C(c2c(C)occ2)=O)C)C)C2CCC1(c1ncco1)C2 28914,C1(C(N(CCNC(C2(C)C(C(=O)OCC)CCC2)=O)C)=O)CCN(C)C(=O)C1 28915,N1(C(CCNC(c2cncc(OC)c2)=O)=O)C2COCC1CC(F)C2 28916,C(=O)(C1COc2ccccc21)NCC1(C)CCN(C(c2cc(F)ccc2N)=O)C1 28917,C1(C=O)CCCC(=O)C1.C1(COC)(NC(=O)CC2(N(C)NC)CC2)CCOC1 28918,C1(NC(C2(CC)CCC(O)CC2)=O)CCCCN(C(c2ccnnc2S)=O)CC1 28919,CCCCC(=O)C(=O)NCCCN(C(c1nnc(S)n1C)=O)Cc1cccnc1 28920,C=CC(F)(F)C(=O)NCCCN(C)C(C1COC(C)(C)C1)=O 28921,c1(NCC2N(C(C3CC(SC)C3)=O)CCCC2C)nc2c(C)cccc2o1 28922,C12(C(N3CCC(C(C)(O)CNC(=O)Cc4cncs4)CC3)=O)CCC(F)(CC1)C2 28923,C1(C(N2CC(NC(C(C)NC(C)(C)C)=O)(CO)C2)=O)OCCOC1C(F)(F)F 28924,c1(NC(CNC(C2N(CC)CCC2)=O)(C)CO)nc2cc(Cl)cc(Cl)c2o1 28925,c1(N2CCN(CC(=O)NC)CC2)nc(=N)[nH]c(=NCCc2cn(C)nn2)[nH]1 28926,c1(N(C(CNC(c2ccc(OCC#C)cc2)=O)C)C)nc(Cl)c2ncnc-2[nH]1 28927,C12(C(=O)NCC3CCN(C(C(=O)NCC)=O)C3)C=CC(CC1)C2 28928,C1(NC(C2CC(C#C)(O)C2)=O)CCCC(C(=O)N(C)Cc2occc2C)CC1 28929,CC(C)(F)CC(=O)N1CCCCC1CCC(=O)NCC1=NOCC1 28930,CC1(C)CCCC1(O)CNC(=O)C(F)C1CC(NC(C2OC3CCC2C3)=O)C1 28931,CCCCC(O)CCC(=O)NC1CC(C)N(C(=O)Cc2cnn(C)c2C)C1 28932,Cc1noc(Cl)c1CC(=O)NC(C)(C)CCCNC(=O)C(n1cnc(C#N)n1)C 28933,c1(CC(N2CC(NC(C3CCC3)=O)CC(C)C2)=O)ccccc1S(=O)(=O)C(F)F 28934,C1(NC(C2N(CCC)C(=O)CC2)=O)CCCCN(C(=O)C(F)C2CCC2)C1 28935,Cc1cccc(C(=O)N(C(C)CNC(C2(C)CCN(C)C2=O)=O)C)c1C#N 28936,CCCC(CCCNC(=O)C(O)Cc1ccc(Br)cc1)NC(C1CCC1)=O 28937,CC1(C(=O)NCCN(c2ccccc2F)CC2CC2)COCCO1 28938,C(=O)(C1=C(Cl)CCC1)NC(CCCCNC(C(CC)(C)C)=O)C 28939,n1(C(C(=O)NCC(C)(C)NC(C(C)NC(=O)NC)=O)C)nccc1C 28940,CC(C)(C)CCCCNC(=O)C(CCC1CC1)NC(=O)C(C1CCOCC1)F 28941,C1(CNC(CN2CC(CC)C2)=O)CN(C(c2cnn(C)c2N)=O)CCC1(F)F 28942,CC1CC=C(C(=O)NCc2cncc(C(=O)NC(c3nnc(O)n3C)C)c2)CC1 28943,C(=O)(CC(C)(C)C(=O)N(CCCN(C(=O)C(=Cc1cccnc1)C)C)C)OCC 28944,C(CCCCC(=O)NC1CC(NC(=O)CC2CC(F)C2)C12CCC2)OC(C)C 28945,c1(C(=O)NC2CC(C)(NC(C(F)OC)=O)C2)ccc(Cc2cnn(C)c2)cc1 28946,N1(C(C(CC(=O)OCC)C)=O)CCC2CN(C(C3CN(C(C)=O)C3)=O)CC12 28947,c1(N(C)C)cc(F)c(NC(C2CCN(c3ccc(Cl)cc3)C2=O)=O)cc1[N+](=O)[O-] 28948,c1(C(=O)NCCCOCC)cccc(Cl)c1OCC.c1ccc(F)cc1.C1(=O)CN1 28949,C1(CC(=O)NCC2(F)CC(NC(C(C#N)C3CC3)=O)C2)NC(=O)NC1=O 28950,C1(C(N2CC(O)(CC(=O)NCCC(C)(C)F)C2)=O)(SC)CC(=O)C1 28951,N1(C(c2n[nH]cc2Br)=O)CC(NC(c2ccc(C3CC3)o2)=O)C2(CC2)C1 28952,c1(C(=O)NC(CN(C(Cn2ncc(CC)c2)=O)C)(C)C)cc(N)c(Cl)c(O)n1 28953,C(CN=C(NCC(N1CC=CC1)=O)N1CCS(=O)(=O)CC1)NCC.C(C)=O 28954,c1(C(=O)NC(C2CCN(C(CSCC)=O)C2)C)cc2c(C)ccc(F)c2o1 28955,C(c1ccco1)=C(C)C(N1CCC(CC(=O)NC(c2nccs2)C)C1)=O 28956,CCC(C)(O)C(=O)N1CC(C(C)NC(C2(O)CCC2)=O)C1 28957,N1(C(CNC(C=C)=O)=O)CC(C)(C)OCC1C(=O)NCC12CCCC1OCC2 28958,C1(C)(C(=O)NCCc2cc(C)ns2)CCCN1C(c1cnc(C)s1)=O 28959,C(=O)(C#CC1CCOC1)N1CC(C(=O)NCCN2CCOCC2C)CC(C)C1 28960,C1(CNC(c2c(CC)c[nH]n2)=O)CC2CCC(C1)N2C(=O)C(COC)OC 28961,CC1CN(C(=O)C=Cc2cncc(F)c2)CC1(C)CNC(c1ncncc1F)=O 28962,N1(C(C2C(C(N)=O)C2)=O)CCCC2(C1)CN(C(c1cc3cn[nH]c3cn1)=O)CCO2 28963,Cc1cc(C(=O)N(CCNC(c2ccn(CCOCCO)n2)=O)C(C)C)sc1C 28964,CC1(C)CC2(CC(C(N3CCC(CNC(=O)CCS(N)(=O)=O)C3(C)C)=O)C2)C1 28965,CCCCC(C)(C)C(=O)N1CC2C(C(=O)NCC(=O)NC3CC3)C2C1 28966,N1(C(c2ccc(COC)o2)=O)CCCCC(CNC(=O)C(CBr)=CC2CC2)C1 28967,c1(C(=O)NC2(CNC(C(CC(C)C)(C)C)=O)CCCC2)cn2cc(Cl)cnc2n1 28968,C(=O)(C(C)C(F)(F)F)NC(C(C)NC(Cn1c(CCC)nnc1S)=O)C 28969,C1(CNC(c2cnc3sccn23)=O)CC2CCC1N2C(C1CC2CCC1CC2)=O 28970,C(c1cccc([N+](=O)[O-])c1)=CC(=O)NC1C(C(N2CC(C)(O)C2)=O)C1 28971,c1(OC)ccc(NC(C2CCCN2C(C2CCC2)=O)=O)cn1 28972,Cc1c(CC(N2CCCCC2c2cn(-c3ncn(C)n3)nn2)=O)nc(Br)n1C 28973,C1(C(=O)NCC(C)(O)CNC(c2ccn(-c3ccncc3)n2)=O)CCC(=O)NC1 28974,Cn1nc(C(=O)NC2CCN(C(C34CC(C)(C3)C4)=O)C2)cc1Br 28975,C1(CNC(C2(Cc3ccccc3)CCOC2)=O)NCC12CCC2 28976,N1(C(C=C(C)Cl)=O)CCC(NC(=O)Cc2sc(O)nc2O)CC1c1ccccc1 28977,c1(SCC)ccc(C(C(=O)OC)NC(N2CCCC2N(C)C)=O)cc1Br 28978,c1(C(=O)NC(CCCC)CNC(=O)CN(C)CCC)ccc(Cl)c(S(N)(=O)=O)c1 28979,n1(CCC(=O)NC2CCN(C(CNC(CC)=O)=O)CC2)c(C)c(C)sc1=O 28980,c12ccccc1-n1cc(nn1)C(=O)NC2.C(C)(c1cccs1)=CCOCC=C 28981,Cc1nccc(CC(N2CC(NC(c3ccc(N(C)C)nc3)=O)CC2C)=O)n1 28982,C1(O)(CN(C(=O)C(N)=O)C)CCN(C(c2ncccc2Br)=O)C1 28983,c1(C(N2CC3N(C(CC(C)C(F)(F)F)=O)C(CC3)C2)=O)cnn(C)c1S(N)(=O)=O 28984,C1(c2ccn(C)n2)(CNC(C#C)(C)C)CNC(=O)O1 28985,C1(C)(CC)CC(C(=O)N(CC(C)N(C)C(C2CNC(=O)C2)=O)C)C1 28986,N1(C(C2CC(n3cc(-c4nccs4)nn3)C2)=O)CCOCC12CCS(=O)(=O)C2 28987,N1(CC(N2CC(C(C)NC(C(CCC)C)=O)C2)=O)C(=O)NC2(CCCC2)C1=O 28988,C1(NC(c2n(C=C)nnc2)=O)CC2CC1CN(C(=O)C(C)(C)c1cncnc1)C2 28989,N1(C(c2c(COC)ccs2)=O)CCN(C)C(CNC(c2ncc(C)cn2)=O)C1 28990,O=S(=O)(c1cc2sc(=NCCCCO)[nH]c2cc1Cl)NC1CCCc2sccc21 28991,N1(C(C2(n3cc(C(C)C)nn3)CCC2)=O)CCC(CCC#N)CC1 28992,Cc1cc(=NC(Cc2ccc(Br)cc2)C(C)C)nc(-c2ccn(C)n2)[nH]1 28993,c1(NC(C(=O)OC)C)cccc(OCc2ccccc2)c1 28994,C1(Nc2ccnc(C)n2)CCN(C(=O)C2=CC(C)(C)C2)CC1C 28995,C(=O)(C(CC(C)C)NC(=O)C=Cc1cnccc1C)NCC1CC(OC)C1 28996,CC1=C(C)CC(C)(NC(C2CSCCN2C(c2coc(C)n2)=O)=O)CC1 28997,c1(N2CCC(NC(=O)NCc3cc(Cl)ncc3Cl)C2)ncc2c(n1)CCC2 28998,c1(CC(=O)N(CCC)CCNC(=O)CNC(C)=O)cc(F)ccc1OC 28999,O=C(CCCCNC(C1C2CCCC12)=O)NC1(CF)CCC1 29000,Cc1noc(Cl)c1CC(=O)NC1CCCCC1NC(C1(F)CC=CCC1)=O 29001,c1(CCC(=O)NC(C(C)C)CNC(C2(C(C)(F)F)CC2)=O)ccc(F)cc1F 29002,Cc1ccn(C)c1C(=O)NCC1CN(C(=O)C=Cc2ccsc2)CC1C(F)(F)F 29003,C1(C)(CNC(CCC#C)=O)COCCN(C(c2ccc(CC)cc2)=O)C1 29004,c1(C(=O)NCC(COC)C(F)(F)F)sc2ncn(C(C)C)c(=O)c2c1C 29005,c1(OC)ncnc(C(=O)NCC2(O)CCN(C(c3ccc(C#N)cc3)=O)C2)c1F 29006,N1(C(c2c(C)nsc2)=O)CCC=CC1C(=O)NC1C(=O)OCC1CO 29007,c1(C(=O)NC2CC(CNC(Cc3nc(C)sc3)=O)C2(C)C)ccc(CO)c(Cl)c1 29008,Clc1ccc2c(c1)CCC2NCCCCn1cccn1.c12cn(nn1)CCCS2 29009,O=C1NCCC2(CN(C(C3(NC(C4CCC4)=O)CC(O)C3)=O)C2)O1 29010,CN1CCC(C(N2CCCC(SCCc3cn(CC4CNC(=O)CO4)nn3)C2)=O)CC1 29011,c1(N(C)C)ccc(C(=O)NCC23COC(CF)(C2)C3)cc1.C12CCN1C(=O)C2.C(N)=O 29012,Cc1nc(S)sc1CC(N1CCC(F)(CNC(c2cncc(F)c2)=O)C1)=O 29013,C1(N(C)CC)CN(C(c2ccc(C3CCC3)cn2)C(=O)NC)CC12CCC2 29014,C1(NC(c2cc(CN(C)C)on2)=O)CCCCC1CNC(=O)C(C)(C)C1CCC1 29015,Cn1ccc2cc(CNC(N3CCCC3C3CCOC3)=O)ccc12 29016,c1(CNC(c2cccc(Cl)c2Cl)C(=O)OCC)scc2c1OCCO2 29017,c1(C(N2C(C)CC(NC(C(CCC)(C)O)=O)C2)=O)c(F)cc(F)cc1F 29018,c1(C2(C(N3C(CNC(c4c(C)cns4)=O)CC3)=O)CC2)ccccc1C 29019,C1(CC(=O)N(CC(C)SC)C)CCCCN1C(=O)COc1ccsn1 29020,N1(C(C=CC=CC)=O)CCOC(CC(=O)NCC(C)C(C)C)C1 29021,CCCCC(C)(F)C(=O)N(CC(C)NC(c1cc(N(C)C)ccn1)=O)C 29022,N1(C(c2coc(C3CCC3)n2)=O)CCC2C(C1)CN2C(C1CCCCC1(F)F)=O 29023,C1(C(N2CCC(COCC)C2)=O)CCCCN1C(=O)CCOCc1ccccc1 29024,N1(C2CCN(C(CCC)=O)CC2)C2CCC1CN(C(c1csc(C(F)(F)F)n1)=O)C2 29025,C(C(F)(F)C(=O)N1CCC(C(C)NC(=O)C(C)OCc2ccccc2F)C1)OC 29026,c1(C(=O)NC(C2CCOC2)CNC(C2(C)CC2(F)F)=O)cc2nc(F)ccc2o1 29027,C=CCCC(c1nn[nH]n1)OCCOCC1CCCO1.C1(=O)C(C)O1 29028,O(C1CCOc2ccc(Br)cc21)C(c1cc(F)c(OCC)c(F)c1)=O 29029,C=C(Cl)CCC(=O)N1CC(NC(=O)C(CC)NC(=O)NC)C(CC)C1 29030,C(=O)(C1=C(Cl)CCC1)N1C(C(=O)NCCCOC(C)C)CCC1 29031,N1(C(c2ccc(CC)cc2)=O)CC2CCC1CN2C(=O)C(c1csc(C)n1)=O 29032,c1(CC(=O)NC2(CO)C(C)C2)csc(-c2cccnc2)n1 29033,C1(CC(=O)NC(C2CCN(C(=O)C(F)CC3CCCCC3)CC2)C)SC(=N)NC1=O 29034,C1(NC(c2c(SC)cn(C)n2)=O)C2COCC1CN(C(C1CCCO1)=O)C2 29035,c1(C(=O)NC23CCN(C(C=C(C)C4CC4)=O)C2CCC3)ccc2c(c1O)CCC2 29036,C1(CCCNC(c2cnsn2)=O)CCCCN1C(=O)CCC1CC1 29037,CC(C)C(C(C)NC(c1nocc1Cl)=O)NC(=O)CCNC(=O)C=CCl 29038,n1(CC)nc(C)cc1C(=O)N(C)CC1CCCC1NC(C1(C)CC1C)=O 29039,c1(CCC(=O)NC2C(CNC(CCOC)=O)C2)ccc(Br)cc1 29040,c1(C(N2CC(C)(NC(CC(c3ccccc3F)C)=O)C2)=O)cc2c(s1)CCCCC2 29041,c1(C(C)NC(N(C)Cc2ncc(C)o2)=O)cc(Cl)c(Cl)c(Cl)c1 29042,C1(N(C(c2cccc(Cc3c(C)n(CCO)nc3)c2)=O)C)CCN(C)CC1C 29043,c1(C(=O)NCC(F)CNC(C2(CO)CC2)=O)cc2sc(Br)cc2[nH]1 29044,Cn1c(C(=O)N(CCNC(C2CC2F)=O)CC2CC2)cc2occc12 29045,Cc1nc(O)[nH]c1C(N1CC(NC(c2cscc2C#N)=O)C1)=O 29046,N1(C(COCCCCC)=O)CC2CC(C(=O)NC(C)CC3CC3)(C2)C1 29047,C1(C(N2CCN(C(=O)Cc3cccnc3)CC2)=O)CC12CCCOC2 29048,c1(OC)cccc2c1CC(C(=O)NCC1CN(C(C34CC(CO3)C4)=O)CCO1)O2 29049,C(c1ccc(Cl)cc1F)=CC(=O)NC1CCC(CNC(c2n(CC)ncn2)=O)C1 29050,C(C)(CCC(=O)N(C)CCNC(=O)CCc1ccc(OC(F)(F)F)cc1)CC.C(C)O 29051,c1(C(N(CC(CC)NC(C2CC23CCOCC3)=O)C)=O)ccc(C)c(COC)c1 29052,c1(OC)ccc(Cc2cn(-c3ccc(C(=O)NOCC)cc3)nn2)cc1 29053,c1(C(=O)NCCN(C)C(c2nocc2Cl)=O)cncc2c1CCC2 29054,c1(NCc2c(C)nc(C)s2)cc(=NCCS(=O)(=O)N2CCCC2)[nH]c(C)n1 29055,c1(C(N2CC(C(C)NC(CC(COC)C)=O)C2)=O)ccc2c(c1)CCO2 29056,N1(CCC(N2C(C(C)NC(=O)CCc3ccc[nH]3)CCC2)=O)CCCCC1=O 29057,c1(OC)ccc(-c2cn(CC(F)CCNC(=O)Cc3nnc(C)s3)nn2)nc1 29058,Cc1cccc2c1ccn2CC(N1CC(O)CCC1C)=O 29059,C1(OC)COc2c(CNC(C34CC5CC(C(=O)N3)C4C5)=O)cnn2C1 29060,Cc1nccn1CC(=O)NC1(C(=O)NCCN2CCC(C)C2)CCC1 29061,N1(C(C2(O)CCCC2)=O)CC(N=c2cc(C3CCCC3)nc(Cl)[nH]2)C2(CCOCC2)C1 29062,C1(NC(=O)NCC2(NS(C)(=O)=O)CCC2)CC(C2CCCC2)C1 29063,CC1(NC(c2cc(C(F)(F)F)n[nH]2)=O)CCCN(C(c2cncn2C2CC2)=O)C1 29064,N(C(=NCCS(=O)(=O)c1ccc(Br)cc1)NCC1(O)CCSC1)CC(=C)C 29065,CC1(C)CCC2CC(NC3CCCOC3)c3cccc1c32 29066,c1(NC(C(CC2CCCC2)NC(C2CCC(=O)C2)=O)=O)cnc(F)nc1 29067,N1(C(CC=CC(C)(C)C)=O)CCCC2CN(C(=O)Cc3cncc(C#N)c3)CCC12 29068,c1(CC(C)NC(C(=O)NC(c2ncc(Cl)n2C)C)=O)noc2ccccc12 29069,C(C(=O)N1CC(n2cc(CNC(C3CCCS3)=O)nn2)C1)(C(C)(C)O)NC(C)=O 29070,c1(CC(=O)NC(CN(C(CC(C)(C)CO)=O)CC)C)cccnc1 29071,c1(CN2C(C(=O)NCc3nc(C(F)(F)F)cs3)CC2)csc2ccccc12 29072,Cc1cnn(C)c1CC(=O)NCc1ccc(C(=O)N(C)CC2CCCS2)cc1 29073,c1(C(N2C(C(=O)NCCc3c(C)nn(C)c3)CC2)=O)cc(C#N)cn1C 29074,Cc1ccc2c(c1)CC(C(N1CCCC1CCCNC(c1cc(C)sn1)=O)=O)S2 29075,C12(C(=O)OCC)CCCC1CCN2C(=O)CN1CCOCC1=O 29076,C=CCCCC(=O)NCC1(NC(=O)C(F)CNC(C2CCC2)=O)CCCC1 29077,C1(NC(CC2CCCC(C(N)=O)C2)=O)CC12CCN(C(c1ccc[nH]1)=O)CC2 29078,C=Cc1ccc(C(N2CC(O)CC2CNCc2ccc(Cl)cc2Br)=O)cc1 29079,CCCCN=C(NCc1ccccc1C(F)F)N1CCC(O)C1 29080,c1(N(C2CCN(c3nnnn3C)CC2)C(CC(C)F)=O)cc(Cl)c2c(c1)OCCCO2 29081,CC(C)CCC(C(=O)NCC1(O)CSC1)NC(=O)C(O)C(C)(C)C 29082,c1(CCC(=O)NC2CN(C(C(CC#C)O)=O)CC2(C)C)cncc2ccccc12 29083,C#CCC(C(=O)NC1(CC)CN(C(=O)C(C)CC)C1)C1CC1 29084,c1(C(C(=O)N(C2CC3CNC2C3)C(CC)=O)C)ccc(C(F)(F)F)cc1 29085,N1(C(C=Cc2cn(C)nc2)=O)C2CCC(C2)C1C(=O)NCc1ncn(C)n1 29086,c1(NC(C(COC)(C)C)c2nnnn2CCSC)ccc2nsnc2c1 29087,N1(C(C2CCC(C(C)=O)CC2)=O)CC2CCC1CN2C(c1cc(C(N)=O)n(C)n1)=O 29088,N1(C(CCCNC(=O)OC)=O)CCC(NC(c2cc(C3CC3)ns2)=O)C(CO)C1 29089,C1(C(=O)NCCOC2CCN(C(CC3CN(C)CC3O)=O)CC2)CCCCCCC1 29090,C=C=CC(C)C(=O)N1CC(CNC(=O)CCN2CCCCC2C)C(C)C1 29091,c1(C(=O)NCC(C)Nc2cc(=O)n(C(C)C)c(O)n2)ccc2c(c1)COCC2 29092,N1(C(c2nc(CN3CCOCC3)no2)CC#C)CCC(N2CCCC2=O)C1 29093,CCS(=O)(=O)c1ccc(F)c(C(=O)N(CCC(C)NC(=O)Cc2cccs2)C)c1 29094,C12(NC(C(C)c3ccsn3)=O)CCC(CC1)N(C(=O)Cn1cnc([N+](=O)[O-])n1)C2 29095,C#CCC(C)(C(=O)N(CCCOC)C)NC(=O)CC1CC(=O)C1 29096,C1(C(=O)NC(CC)CN(C)C)CCCCN1C(C1CC2C=CC1O2)=O 29097,C(C(C)(O)CC(=O)N1CCC(F)(NC(=O)CNC(=O)C(C)(C)NC(C)=O)CC1)OC 29098,N1(C(C2C(OC)CC2)=O)CC2C(C(=O)N(C)CC3CCCS3)C2C1 29099,c1(C(=O)OC)cc(C(=O)NC(C)CNC(C2(C)CCNC2=O)=O)cc(C)c1 29100,N1(C(C2C(=C)C2)=O)CCCC1C(C)NC(=O)CCc1nc(-c2ccoc2)no1 29101,c1(C(N2C(C)(CNC(=O)C3=C(Cl)CC3)CCC2)=O)cc(=O)n2ccccc2n1 29102,N1(C(c2cnc(C(C)OC)s2)=O)CCCC(N(C)C(c2c(C)nsc2C)=O)CC1 29103,N1(C(c2ccc(C(C)C)cc2)=O)CC2CC(NC(C3CCCC(C)C3)=O)CC2C1 29104,CN1CC=C(CC(=O)NC2(CC(N3CCC4OCCCC4C3)=O)CCC2)CC1 29105,c1(C(N2C3(CNC(C4NC(=O)OC4)=O)CC(C2)C3)=O)cn2cc[nH]c(=O)c2n1 29106,S(=O)(=O)(c1c[nH]ccc1=NCc1ccc(C(C)(C)C)o1)NCC(CC)N1CCCC1 29107,C=C(C)CC(C(=O)NC(C)CNC(c1ccsc1)=O)NC(C)=O 29108,C1(C)(C(N(C2CCN(C(C3(n4nccn4)CC3)=O)C2)CC)=O)CC(C2CC2)=NO1 29109,Cn1cc(-c2nc(C(N3CC(F)(CNC(C4CCOC4)=O)C3)=O)co2)cn1 29110,C1(C#CC(=O)N2CCC(OCCNC(C3CC3(F)Cl)=O)C2)(CC)COC1 29111,C1(C)(NC(C=CC)=O)CCN(C(c2oc(-c3ccccc3)nc2C)=O)C1 29112,C1(CNC(CC(CC)SC)=O)CCCCCN1C(=O)COc1cc(C)ccc1C 29113,n1(CC(N2CCC(NC(c3n(C)nc(O)c3)=O)C(F)C2)=O)nnc2c1CCCC2 29114,N1(C(CNS(CCCC)(=O)=O)=O)CC2CCCN(C(=O)C(C)C(F)F)C2C1 29115,S(=O)(=O)(c1ccc(=NCc2ccc(S(C)=O)cc2)[nH]c1)NCc1c(C)nccn1 29116,N#CCCCN=c1[nH]c(N2CCC3(CC(=O)NC3=O)C2)nc2c1CCCC2 29117,Cc1oc(C(=O)NCCNC(C2CCCCN2C2CCCC2)=O)cc1S(N)(=O)=O 29118,C(=O)(C(C(=O)OC(C)(C)C)SC1CN(C(=O)C=CC2CCCC2)C1)OC(C)(C)C 29119,C(=O)(CCC(C)(C)NC(c1cc[nH]c(=N)n1)=O)N(C)Cc1onc(CC)n1 29120,c1(CN2C(C(=O)NCC(C)(C)F)CCC2)c[nH]c2ccc(Br)cc12 29121,c1(C(=O)NCC2CCCC(NC(CCCSC)=O)C2)coc2c(F)cc(Cl)cc12 29122,c1(C(N2CCN(C(C3(COC)CCC(=O)N3)=O)CC2)=O)cc(N)c(Cl)cn1 29123,N1(C(C(c2cccc(O)c2)C)=O)CC(NC(=O)COC2CCOCC2)C(C)C1 29124,c1(OCC)ncccc1CC(=O)NC1(CCNC(=O)C=C=C(C)C)CC1 29125,N1(C(Cn2ncc(C)c2)=O)CCCCC1C1CCN(C(=O)C(C)C)C1 29126,C(c1cnc2ccccc2n1)=CC(=O)NC1CC2CC1N(C(c1cocn1)=O)C2 29127,C1(C(N(CCCCC(=O)NCC2CC(F)(F)CO2)C)=O)CC2COCC2C1 29128,N1(C(C2CCCN(C(=O)OC)C2)=O)CC2(CCC2NC(=O)C(F)=C(C)C2CC2)C1 29129,C1(CNC(CS(=O)(=O)NC)=O)CN(C(=O)CC2(C)CCOC2)CCC1C 29130,C1(=O)C(=O)NNC(=O)C2(CCOC(C)(C)C2)N1.C1(CC)COCC1NC(=O)C(C)C 29131,c1(C(=O)OC(CC#C)COC)sc2ccccc2c1C(C)=O 29132,C1(C(N2C(CN(C)CC=Cc3cn[nH]c3)CCC2)=O)CCCC2CCCN12 29133,CCN=c1cc(C(N2CC(NC(=O)C=C3CCC(C)CC3)C3(CC3)C2)=O)cc[nH]1 29134,c1(NC(N2CCC3CN(S(=O)(=O)C4CC4)CC23)=O)cccc2ccccc12 29135,C1(NC(C(=O)N(C)Cc2cccc(C(=O)OCC)c2)=O)CCC(P(C)(C)=O)C1 29136,C1(O)(CC(=O)NC(C2CCCCC2)CC)CN(C(=O)Cc2nocc2C)C1 29137,c1(NC(C(CC)NC(=O)CN)=O)cc(S(=O)(=O)N(C)C)ccc1F 29138,CC1CC(C)N(C(c2cccc(NC(=O)CO)c2)=O)CCN1C(=O)CC(C)(C)O 29139,C1(O)(CN(C(=O)C(C)P(C)(C)=O)CC)CCN(C(c2cc(C(F)(F)F)c[nH]2)=O)CC1 29140,N1(C(c2c(C)csc2C(F)(F)F)=O)CC2CCC2(CCNC(=O)CCC2CC2)C1 29141,c1(Cc2nc(CC(=O)OC(=O)CC3CN(CC)C3)sc2)ccc(Br)cn1 29142,N1(CCC(C(=O)O)n2ccnc2C2CC3(CCC3)C2O)Cc2cccnc2C1 29143,C1(C)(OC)CC(NC(C2(C)CN(C(C3(OC)CCOC3)=O)C2)=O)C1(C)C 29144,Cc1ncc(Br)c(N2CCOCC2C(=O)Nc2ncc(Br)cc2I)n1 29145,CC1CC(=O)NC(C(=O)N(C(C)CNC(c2ccc(CO)cn2)=O)C)C1 29146,C1(NC(CCC#CC)=O)CC(O)CN(C(=O)CCC2CC2)C1 29147,c1(C(=O)NCCC(C)NC(C2N(C(C)=O)CC(O)C2)=O)ccc(=O)n(C)c1 29148,C(=O)(C1=CCCOC1)NCC1CCC(NC(c2ccc(OC)s2)=O)CC1 29149,c1(CNC(c2nnnn2CCCF)(CSC)C)cccc(OC(C)(C)C)n1 29150,c1(C(=O)NCC2N(C(C3N=C(C)SC3)=O)CC2)cc(C)c(F)cc1Br 29151,n1(CCCC)nc(C)c(C(N2CC(CCCCNC(=O)CC(C)SC)C2)=O)c1Cl 29152,N1(C(C)=O)CCN(CC(c2cccc(S(C)(=O)=O)c2)=O)CC12CCCCC2 29153,N1(C(C(C)=C2CC2)=O)CCCCC1C(N1CCC(C)C1C)=O 29154,C#Cc1ccc(C(N2CCN(C(C3C4CCCC34)=O)CC2CN(C)C)=O)nc1 29155,C(=O)(C(C)CCCOC)NCC12OCC(NC(Cc3cn(CC)nn3)=O)(C1)C2 29156,C1(NC(=O)C(C)(C)C)CCC(C)N(C(C2CN(C(=O)NC)C2)=O)C1 29157,C12(NC(C(CCC)C)=O)CC(CNC(c3n[nH]cc3C#N)=O)(C1)OC2C 29158,c1(C(N2CC(OC)C(NC(=O)C(C)(O)C(C)C)C2)=O)cccc2ncsc12 29159,c1(C(=O)NCc2sccc2F)cc(NC(N2CCC(c3cnccn3)C2)=O)[nH]n1 29160,CCCC(C(=O)NCc1ccc(F)cc1)NC(C1CN(C(=O)C(C)C)C1)=O 29161,N1(C(=O)NCC2Cc3c(cn(C)n3)CC2)CC(N=[N+]=[N-])CCC1(C)C 29162,c1(C(N)=O)cc(C(N2CC(NC(c3cnns3)=O)CC2CO)=O)ccc1O 29163,c1(C(CCC)NC(=O)CC2CN(Cc3ccco3)CCO2)cc(Cl)ccc1OC 29164,C1(CNC(C2(C(C)(F)F)CC2)=O)CN(C(=O)CCCOc2ccccc2)CCN1C 29165,C(=O)(C(CN=[N+]=[N-])NC(=O)CCC(C)(C)F)Nc1c(CC)csc1 29166,C(=O)(CCCCC(=O)NC)N(CC(CNC(C(CCC)c1ccccc1)=O)C)C 29167,C12(NC(CCOC(CC(C)C)C)=O)COC(C1)C(NC(c1cccc(CO)c1)=O)C2 29168,C1(OC(Cc2nc(C(CC)(C)C)on2)=O)CCC(=O)NC1 29169,C1(C(=O)N(CC(C)NC(C2(C#N)CCCC2)=O)C)(COC)CC=CCC1 29170,C1(NC(c2c(CC)n(C)nc2)=O)CN(C(=O)CCNC(C)=O)C(C)(CC)C1 29171,N1(C(Cc2ccc(N(C)C)cc2)=O)C2CCC(C2)C1CC(=O)NCCS(C)(=N)=O 29172,c1(OC)ncccc1CC(=O)NCC1C2CC1N(C(=O)CN1CCCC1C)C2 29173,N1(C(C(=O)NCc2c(CC)nn(C)c2)=O)CCC(O)CC1c1ccc(F)cc1 29174,CC1CC(NC(c2cccc(O)n2)=O)CN(C(=O)CCNS(=O)(=O)C(F)(F)F)C1 29175,N1(C(COC(CNC(c2cc(C)c(C)nn2)=O)(C)C)=O)CC2CCCCC2C1 29176,C(=O)(C(C)(O)C(C)C)N(CC(CNC(Cc1ncc(C)[nH]1)=O)C)C 29177,c1(NC(C2CCN(C(c3ccc[n+]([O-])c3)=O)C2)C)nc(O)c2ccccc2n1 29178,c1(N2CCCC(CN(C(C)=O)C)C2)nc(Nc2cnco2)c2ncn(CC)c2n1 29179,C1(C(N2C3COCC2C3)=O)CC(O)CN1Cc1ccncc1Br 29180,C1(CC(=O)NCCC2CCN(C)C2)C2CCCC2N1C(C1(N(C)C)CCCC1)=O 29181,C(=O)(CCCC(=O)N(CCCCN(C(=O)Cc1ccno1)C)C)NCCC(C)C 29182,Cc1cccc(C2(C(=O)NC3CCCC(CNC(c4cocc4C)=O)C3)CC2)c1 29183,C(=O)(C1=C(CNCC(CNC(=O)OC(C)(C)C)CO)NC(=O)NC1C)OC 29184,c1(CC(N2CC(O)(CCNC(c3[nH]c(=N)sc3)=O)C2)=O)cnc2cccnn12 29185,C1(NC(C(=O)NCC2CCN2Sc2ccccc2)c2ccco2)CC2CCC1CC2 29186,c1(C(=O)NC2CCC(NC(CC=C(C)C)=O)CC2)[nH]nc([N+](=O)[O-])c1Cl 29187,N1(C(c2c(C)ocn2)=O)C2CCC1CN(C(c1cccc(C(F)F)n1)=O)C2 29188,C1(CCOC)CN(C(c2[nH]c(C)nc2C)=O)CCN1C(c1cc(C)ncc1C)=O 29189,c1(C(=O)NCCC2N(C(c3c(OC)nsc3)=O)CCCC2)ccc(C)c(C)n1 29190,C(=O)(CCCC(=O)N1CC(CNC(C2(F)CCOC2)=O)CC1C)NC(C)C 29191,C(C#Cc1cc(Cl)cnc1F)C(N1CCC(O)(CCOC)C1)=O 29192,C1(C(N(CCNC(c2ccc(C)cc2)=O)C)=O)CCC2CC2CC1 29193,N1(C(C2CCC(C)O2)=O)CC2CCCC1(CNC(c1ccc3c(c1)CCO3)=O)C2 29194,c1(C(N(C(CNC(c2c(OC)ccc(O)c2)=O)C)C)=O)cc2n(c1)CCSC2 29195,C12(C(N3CC(C)C(NC(c4cnn(C)c4Cl)=O)C3)=O)CCCCN1CCC2 29196,N1(C(c2cc(C#N)[nH]c2)=O)CCOCC(NC(C2CC3CCCCC23)=O)C1 29197,CC1(C)C2CN(C(c3ccc(OC(F)(F)F)cc3Cl)=O)CC12 29198,C#Cc1ccc(C(=O)NCC2(NC(c3cncc(N(C)C)c3)=O)CCCCC2)o1 29199,CCCC(C)CC(C(=O)c1ccc2cc1OCON2)NCP(C)(C)=O 29200,C1(NC(CC(COC)C)=O)(CO)CCCN(C(=O)CCc2conc2C)C1 29201,c1(C(N(C2CCCN2C)CCOC)=O)cn(CCNC=O)nn1.c1ccc(C)s1 29202,N1C(=NCCCc2ccccc2)N2CCC(C2)C1.C[Si](C)(C)C1CCCCC1 29203,c1(CN2C(C(=O)Nc3nccc4occc34)CC(C)C2)cccc2c1OCO2 29204,C1(CNC(C(C)C2CCC2)=O)CCCC12CCN(c1nc3ccccc3o1)CC2 29205,C1(CC)CCN(C(C2CC=CC(O)C2)=O)C1CNC(c1cc(F)n(C)n1)=O 29206,S(=O)(=O)(c1ccc(OC)cc1)N1CCC(N(C)CCC2CCN(C(=O)NC)CC2)C1 29207,C1(C(=O)NCC2N(C(c3c(C)occ3)=O)CC=C2)CSC(c2ccccc2)=N1 29208,c1(CN(C(CN(C(C(c2cncnc2)C)=O)C2CC2)=O)C)ccnn1C 29209,c1(C(N2CCC(CCNC(C(C)=CC)=O)CC2C)=O)cccc2c1ccn2C 29210,C1(NC(C)=O)CCCN(C(c2cnc(CNC(C3CCCC(C)C3)=O)nc2)=O)C1 29211,n1(CC)ncc(C(=O)N(CCCNC(=O)COCP(C)(C)=O)C2CC2)c1Cl 29212,C12CCCC(C1)CNC2=O.c1(NC(C)=O)ccc(C)cc1.C1(=O)C(=O)NCCN1 29213,C1(C(N2CCC(c3cn(-c4ccncc4)nn3)C2)=O)(SC)CC(=O)C1 29214,CC1CN(S(=O)(=O)CCNC(c2ccccc2)=O)CCC1(O)C(F)(F)F 29215,c1(CC)ccc(C(=O)NCC2(C)CCCN(C(c3csc(=N)[nH]3)=O)C2)c(O)c1 29216,C1(C(=O)NCc2ccc(C(N3CCC(O)C3)=O)cc2)(CC2CCOC2)CC12CCC2 29217,N1(C(c2c(CNC(C(C)C3(O)CCC3)=O)n[nH]c2)=O)CCOCC(O)C1 29218,C1(NC(C2CCCO2)=O)CC2CC1CC2C(=O)NC(Cc1ccco1)CO 29219,O=C(CC(O)CC(F)(F)F)NCCCNC(C1Cc2c(F)cccc2O1)=O 29220,Cc1ccc2c(N3CCC(C(F)(F)F)C3)nc(=NCC=CCl)[nH]c2c1 29221,c1(C(N(C2CCN(C(c3snnc3CC)=O)C2)CCC)=O)ccnc(S)c1 29222,c1(C(=O)NCC2(OCC)CC2)ccc(C(=O)OC(F)C(=O)C2CCCO2)cc1 29223,N1(C(C(c2ccccc2F)C)=O)CCCC(CO)(NC(c2cccn2C)=O)C1 29224,CC(C)(O)C(F)C(=O)NCCC1CC(F)CN1C(=O)C1CC1 29225,C(C(C(C)(C)C)NC(=O)CCc1nc(C(C)C)no1)NC(C1C(COC)C1)=O 29226,c1(NC(CC(C)NC(=O)C(C)Cc2cnc[nH]2)=O)ccc(Cl)nc1 29227,c1(C(C)=O)nccc(=NC(=O)c2cc3ccc(-c4cnn(C(F)F)c4)cc3o2)[nH]1 29228,N1(C(=O)NC2CC2C2CCCCC2)CCOc2cc(Cl)ccc2C1 29229,c1(NC(C2CN(S(CC)(=O)=O)C2)=O)cc(C2CCCC2)nn1C 29230,CC1CCN(C(=O)Cn2[nH]cnc2=N)C(C(N2CCCC(CO)(CO)C2)=O)C1 29231,C1(CNC(c2ccc(CCCCC)o2)=O)CCN(C(=O)C(C)(C)CF)CC1C 29232,N1(C(C(C=C)(C)O)=O)CCc2nc(CNC(C3CC(C)CC(C)(C)C3)=O)sc2C1 29233,c1(C(=O)NCC(CNC(CN(C2CC2)CC)=O)F)nn2c(c1Br)OCCC2 29234,CCCCCC(C(=O)OC)NC1CC2(C1)CC(C(F)(F)F)C2 29235,C(CN=c1ccc(N2CCc3nncn3CC2)n[nH]1)Oc1cccc(OC)c1 29236,N1(C(CCc2c(C)nn(C)c2)=O)CCN(C(=O)CC2CCOC2(C)C)C(CF)C1 29237,N1(C(CSS(C)(=O)=O)=O)CC2CCCC(C1)N2C(=O)CC1CC(C)(C)C1 29238,C(C(CC1CCCC1)C(=O)Nc1ccc(SC)cc1)NC(CC(=O)NCC#C)=O 29239,c1(C(=O)NC(CCCNC(CC(C)N(C)C)=O)(C)C)cnc(N)c(N)c1 29240,c1(C(N2CCN(C(CNC(C(C#C)(C)C)=O)=O)CC2)=O)ccnc2c1nnn2C 29241,CC(C)C(CNC(=O)C(F)CC1CCCCC1)NC(c1nocc1Cl)=O 29242,C(N=c1cc(NCc2ccccc2OC)nc(C)[nH]1)C1(F)CC(NC(COC)=O)C1 29243,N1(C(c2c(C)c(Cl)cnc2)=O)CCCC(C2CN(C(=O)COC3COC3)C2)C1 29244,c1(N(CC(=O)NCCC2=CCCCC2)C)ccc([N+](=O)[O-])cc1 29245,c1(CN2CCC3(C(C(=O)NCc4ccc(F)c(Br)c4)C3)C2)cc(Cl)cc(Cl)c1O 29246,c1(C2CC(C(=O)NCCCN(C(=O)Cc3ccoc3)C(C)C)C2)cccnc1 29247,C1(CC(C)NC(c2csc(C#N)c2)=O)CCN(C(=O)CCc2cn(C)cn2)CC1 29248,C(=O)(CCCCCNC(C1C2CCCC12)=O)NCCC(=O)NCC 29249,C1(CC)CC(C(=O)NCC(c2ccsc2)O)CCN1C(c1csc(C)n1)=O 29250,C12(CC(N3CC(C4N(C(=O)COCCF)CCC4)(O)C3)=O)CCC(CC1)C2 29251,N1(C(C(C)=CCC)=O)CCN(C(c2nn[nH]c2C(F)(F)F)=O)C2(CCC2)C1 29252,Cc1cc(CCC(N2CCCC2CCNC(C2CC3CCC2C3)=O)=O)c(C)o1 29253,C1(C(=O)NCCC2CC(NC(CNC(=O)OC)=O)C2)CCCCC(C)(C)C1 29254,Cc1nn(C)c(Cl)c1C(=O)NC1(CNC(c2ncnn2C)=O)CCCCC1C 29255,C1(NC(c2ccnc(C)n2)=O)CCCCCN(C(c2ccc(C3CC3)cc2)=O)C1 29256,c1(CCN(C(C)C)Cc2nc(C(F)(F)F)cs2)ccc(F)cc1 29257,c1(C(N(C)CC2N(C(C(CC=C)(F)F)=O)CCC2)=O)ccc(C)c(OC)c1F 29258,C1(NC(C2(C(C)C)CCN(C(C(CC)C#N)=O)C2)=O)CC2(C1)CC(C)(C)C2 29259,C(=O)(C1=C(C)OCCC1)NC1CC(CCNC(C2C(CC)C2)=O)C1 29260,C1(C(=O)NCC2(NC(C(CC)CC3CCCC3)=O)CNC2)CC12CC(F)(F)C2 29261,N1(C(=O)NCC(O)C2CCC2)CC2CC1(Cc1ccc(C(F)(F)F)cc1)C2 29262,C(C(CCC(F)(F)F)Nc1ccc(Br)cc1F)OC(C(C)C)=O 29263,C(=O)(C1=NOC(C)(C)C1)NC1CC(NC(CCC(c2cc(C)sc2C)=O)=O)C1 29264,C(CC(CC)C(=O)NCC1CN(C(=O)CN2CCN(C)CC2)CC1(C)C)=CC 29265,C1(C)CCCC1C(F)(F)F.CC(Cn1cccn1)CNC.C12CN(C1)C2=O 29266,C1(NC(C=CC2CCN(C(C(CC)CN(C)C)=O)CC2)=O)CCn2nccc2C1 29267,c1(NC(c2cnn(-c3ccccn3)c2)=O)ncnc2cc(I)sc12.C12CN(C1)C2 29268,C(=O)(C1=CCCCCC1)N1C(C)C(NC(c2sccc2OC(F)F)=O)CCC1 29269,CC(C)C(C(F)F)NC(C1CCN(c2cccc(F)c2)CC1)=O 29270,c1(CNC(C(C(CC)C)C)=O)c(C)nn2c1CN(C(=O)CC(C)(C)OC)CC2 29271,N1(C(C=CC)=O)CCOC(C(C)NC(c2sc(-c3nc[nH]n3)nc2C)=O)C1 29272,C(=O)(C1=C(C#N)CCC1)N(C1CCCC(NC(=O)CCC2CC(F)(F)C2)C1)C 29273,CCC(CC)(C(=O)NCC1CN(C(c2n[nH]cc2C=CC(C)C)=O)CC1C)OC 29274,C12(NC(=O)C#CCNC(=O)C=Cc3cscn3)CCCC1CCC2 29275,CC1CN(C(=O)CCCCc2ccccc2OC(F)(F)F)CC(C)N1 29276,C(=O)(CN=c1cc[nH]cc1)N1CC(CC=C)(C(=O)NC2CCCCC23CC3)C1 29277,C(=O)(CCC(C)(C)C)N1CC(NC(C(CC)C)=O)C(C)C1 29278,C1(C(N2CC(O)(CCNC(C(C=CC)O)=O)C2)=O)COc2ccccc2O1 29279,c1(OC)cc(C(=O)NC2CCCCC2NC(c2ncccc2N)=O)cc(F)c1F 29280,Cc1nc(C)c(C(=O)NC(C2CCN(C(C3CCCC3CF)=O)CC2)(C)C)[nH]1 29281,c1(CCNC(CC2(C)CN(Cc3cc(F)ccc3Cl)C2)=O)cc(F)ccc1C#N 29282,c1(CC(=O)NC2(CCNC(CCCSC)=O)CC2)ccc(O)c(F)c1 29283,C1(NC(c2ccc(C(C)=O)[nH]2)=O)CC2CC1CN(C(=O)CC1CCN(C)CC1)C2 29284,C1(C(=O)OCCCC2(O)CCC2)Cc2nnsc2S1 29285,C12(CNC(c3cc(C(C)C)nn3C)=O)CN(C(=O)C=CC3CC3)CC1CCO2 29286,C1(NC(C2CCOCC2)=O)CS(=O)(=O)C2CN(C(c3ncccc3Cl)=O)CC12 29287,C1(CC)CCN(C(c2cnn(C)c2OC)=O)C1CNC(=O)C(CC)OC1CCCC1 29288,c1(C(N(c2nc(C)sc2)CC2CC2c2cccc(Br)c2)=O)cc(F)ccc1O 29289,C1(F)(CNC(CNC(=O)OC)=O)CCCN(C(=O)CCCn2c(O)nnc2O)C1 29290,N1(C(c2nn[nH]c2Cl)=O)CCN(C(=O)C=CBr)C2CCCCC2C1 29291,C1(CNC(COCCCCC)=O)CC(CNC(C2CC(CC)C2)=O)CO1 29292,O=CN1CCCN(C(=O)CC2CC=CCC2)CC1 29293,C#CC1(O)CCN(C(=O)C(CC(=C)C)NC(c2ccccc2C#N)=O)C1 29294,N1(c2nnc(-c3ccc(OC)s3)n2CC2CC2)CCc2nc(Cl)ccc2C1 29295,c1(C(=O)NCCN(C(c2cn(C3CCC3)nn2)=O)CC)coc2c(F)cc(Cl)cc12 29296,Cc1occc1C(=O)NCC(O)CCNC(=O)CC1(O)CCOC1 29297,CN1C(=O)CCC1CC(N1CCCCC1CCNC(c1csc(Cl)n1)=O)=O 29298,c1(NC(c2cccc(OCc3ccc(OC)c(Cl)c3)c2)=O)cc(Br)c(Cl)cc1F 29299,O=C(C=CC(=O)NCC12CCN(CC1)C2)N=c1[nH]oc2ncccc12 29300,C1(C)(C(=O)OC)CCN(C(=O)CCCCc2ccccc2)C1.C123CC(C1)(C2)NC3=O 29301,c1(C(N(C)CC2CCCN(C(C(C)S(C)(=O)=O)=O)C2)=O)ccc(S(C)(=O)=O)s1 29302,C1(C(=O)NCc2n(C)ccc2)CCN2CCOCC12.c1ccc(F)cc1Cl 29303,C(=O)(C(CO)C(C)(C)C)NC(CNC(c1ccc(C#C)o1)=O)CC(C)C 29304,C1(CNC(c2c(CC)onc2)=O)CN(C)CCN1C(=O)CCc1ccn(C)c1 29305,N=c1[nH]c(CC(N2CC(NC(C3CC3C3CC3)=O)C2)=O)cs1 29306,c1(C(N(CCCCC(=O)NC)C)=O)cc(Br)c(CC)cc1OC 29307,C1(CNC(C(C)OC2CCCC2)=O)CCN(C(=O)CCc2cccnc2)CC1C 29308,C1(NC(C23CC(C)(OCC2)C3)=O)CCC2CN(C(=O)C(C)(C)C3CCC3)CC12 29309,c1(C(=O)NCCOc2ccc(C#N)cc2)c(Br)cc(F)c(F)c1F 29310,c1(C(=O)NC2C(CNC(C(C)(C)c3ccc(Cl)s3)=O)CCC2)cc2n(n1)CCO2 29311,N1(CCOCCCC#C)C(=O)CCN(CC2CCCc3nc[nH]c32)C1=O 29312,O=C(C1CCCc2nccn21)Nc1cnn(C2CCNC2)c1 29313,C(=O)(C(C)CCCC(C)C)NCC1C(CC(=O)NCC2(CC)CCCCO2)C1 29314,CONC(=O)C(=O)NC1CN(C(=O)COCP(C)(C)=O)CC1C 29315,C(=O)(C(C)(C)CCCNC(=O)CS(=O)(=O)NC)N1CC(O)(CC(=O)NC)C1 29316,n1(CCNC(c2n(CCCCCC)nnn2)c2cnccn2)c([N+](=O)[O-])cnc1C 29317,Cc1coc(C)c1C=CC(=O)NCCSCC(O)CN(C)C 29318,CCC(CC(=O)N1CCOCC1CCNC(=O)C=Cc1nccs1)C(F)F 29319,CC(C)(C)C(CO)NC(=O)C(C1CCCCC1)NC(=O)CCc1ccoc1 29320,C1(CCC)(C(=O)NC2(CO)CN(C(C)=O)C2)CCNC1=O.C12(CC1)C(=O)N2 29321,C(CC(=O)NC1CC2OC(=O)CC12)(CC(C)C)NC(CC1(NC(C)=O)CC1)=O 29322,N1(C(c2c(OC)ccc(C)c2)=O)CC2CCCC2(CNC(=O)Cc2cnsc2)C1 29323,Cc1cc(C(=O)N(C)C)c[nH]c1=NCc1ccc2c[nH]nc2c1 29324,C1(CC)(NC(c2scnc2COC)=O)CCN(C(=O)CCc2cscn2)C1 29325,c1(NC)ccc(C(=O)C(=O)NCCCCC(C)NC(c2ccc(F)o2)=O)cc1 29326,C(C(F)(C(=O)NCC1CC2CCC(C1)C2)C(C)C)NC(CCC(CC)=O)=O 29327,C=CCCCC(C(=O)N(CC(O)COCC)CC)NC(=O)Cc1ccc(C)nc1 29328,c1(CC)cc(C(N2CCC(N(C(=O)CC3CCCC(O)C3)C)C2)=O)c(C)o1 29329,C(=O)(C1(C)CCn2c(C)nnc21)N1C(CNC(C(C(=O)NC)(C)C)=O)COCC1 29330,C(=O)(C1CCCn2ncnc21)N(C1CCN(c2nccc(OC)n2)C1)C 29331,c1(OC)cc(C)c(C(=O)NCC2CC(O)CN2C(C2CCC(=O)N2C)=O)c(C)c1 29332,N1(C(c2[nH]cc(CC)c2)=O)CCN(C(c2sc(C(C)(C)C)nc2C)=O)CC1C 29333,C1(C(=O)NCC(CC)NC(c2cnc(C)cc2Cl)=O)CCc2ccnn2C1 29334,C1(C(N(CC(C)NC(c2nn(CC)c(C3CC3)c2)=O)C)=O)CCc2nccn2C1 29335,Cc1nc(C(C)(C)C)nc(C)c1C(=O)NCC(C)(C)NC(C1CC(O)C(F)C1)=O 29336,C(=O)(C(O)Cc1cnn(C)c1)N(C1CC(NC(=O)Cc2ccc(Cl)s2)C1)C 29337,C1(CN(C)C(C2COC(=O)N2)=O)CCCCN(C(c2ccc(C3CC3)cc2)=O)C1 29338,c1(CC(=O)NCC2CC(NC(C(CC#C)O)=O)C2)cccc2c(C)csc12 29339,N1(C(CSCC)=O)CC(CN(CCCC(=O)NC(=O)C(C)(C)C)CC(CC)CC)C2CC2C1 29340,c1(OC)ccc([N+](=O)[O-])c(C(N2CCCC(CNC(c3c[nH]c(=N)s3)=O)C2)=O)c1 29341,N1(C(c2cc(OC)ncc2)=O)CCC2CN(C(c3cnn(C)c3Br)=O)CC12 29342,c1(C(COC)NC(c2nnsc2C)=O)ccc(Cl)cc1 29343,c1(OC)c(F)ccc(C(N2CC(NC(c3ccc(Cl)o3)=O)CC2C)=O)c1F 29344,CC(CCC(=O)N1CCC1c1ccccc1Cl)Nn1cc(C2CC(=O)CO2)nn1 29345,c1(C(=O)OCC)nc(C(=O)NCC2(C)CCN(C(=O)Cc3cnsc3)C2)c(C)s1 29346,O(NC(=O)CC(C)(C)OC)C(C(=O)OC)NC(=O)C(CO)OC 29347,C1(CCF)CC1N=c1[nH]c(N2CCCC(c3cccnc3)C2)nc2c1CCC2 29348,NS(=O)(=O)C1CC(C(=O)NCc2cccc(CNC(C3CC3CF)=O)c2)C1 29349,c1(CC(N2CC(CNC(CCNCC=C)=O)C2)=O)csnc1C 29350,C#Cc1ccc(C(N2CCC(C(=O)NCC3(n4nccn4)CC3)C2C)=O)cc1C 29351,C1(F)(CN(C(C2CC(NC(CCNC(C)=O)=O)C2)=O)C(C)C)CCCCCC1 29352,c1(CC)c[nH]c(C(N2CCCC2Cn2cc(-c3cc(C(=O)O)ns3)nn2)=O)c1 29353,c1(OCc2onc(-c3ccc(OC)cc3)n2)c(Cl)cc(Br)cc1Cl 29354,c1(Cn2c(-c3c(F)nc(Cl)cc3)nc(-c3cscn3)n2)cc2ccccc2o1 29355,C(=O)(CC1=NN(C)C(=O)C1)N1CCC(C)CC1CNC(C1CNC(=O)C1)=O 29356,C(CC(C=O)NC(c1csc(CNC(=O)CC2OCCC2(C)C)c1)=O)OC 29357,C1(N(C)C(c2cc(C(C)(F)F)ccn2)=O)CN(C(C2CCNC2=O)=O)CC1(C)C 29358,N1(C(c2c(OC)n[nH]c2)=O)CC(C)(C(=O)NCCc2ncc[nH]2)CC1(C)C 29359,C1(CC(N2CC(O)(COC)C2)=O)CCCC12CC2.C1(=O)NCCN1 29360,C(C(N=c1ccnc(C)[nH]1)C1CC1)OC(C1(OC)CC(C2CCC2)C1)=O 29361,c1(OC(C(=O)N2CCCC2)=O)ccc(OCCSc2ccc(Br)cc2)cc1 29362,Cc1nc(Br)sc1C(=O)NC1CCC(NC(=O)CCc2cccn2C)CC1 29363,N1(C(C2C(C(N)=O)C2)=O)CCC2CCN(C(=O)COC(F)F)C2C1 29364,C1(C(N2CC(CCO)(NC(CC=CC=C)=O)C2)=O)CCCC2(CCC2)O1 29365,C(=O)(CC(C)(C)CC(=O)NCC1CC1CNC(C1CC2(CCC2)C1)=O)OC 29366,C(CC(C)C)(C(=O)NCC(CC1CC1)C(=O)NC1COCCOC1)OC 29367,CN=c1nc(C(=O)N(CC(C)N(C(=O)CCc2ccsc2)C)C)cc(C)[nH]1 29368,C1(NC(=O)CN(C(C(C)P(C)(C)=O)=O)C2CCCC2)CC2CCC(C1)N2C(N)=O 29369,C=CCCC(C(=O)NOCC(C)(C)C)NC(=O)CNC(=O)CCCN=[N+]=[N-] 29370,c1(C(C)(C)C)ccc(C(N2CCC(C)(NC(=O)Nc3cncnc3Cl)C2)=O)nc1 29371,C1(COC)CC(Cn2cc(C3CC(=O)C3)nn2)N(C(=O)C(C)(C)F)C1 29372,C(N=c1[nH]c(=NCC2CC2)c2[nH]ccc2[nH]1)C1CC(C(F)(F)F)C1 29373,c1(C(N2CCC(C(F)(F)F)C(C(=O)C3CC3)C2)=O)cc2ccsc2s1 29374,c1(CC)ccc(C(=O)NC2COCC2NC(=O)Cc2nnc(O)nc2O)cc1N 29375,N1(C(c2ccccc2Cl)=O)CC2CCC(C1)C2NCc1cc(Cl)ccc1Cl 29376,N1(C(C(C)=C(CC)C)=O)CC2CC(NC(C3CNC(=O)C(C)(C)C3)=O)C(C2)C1 29377,c1(CC(n2cc(CCC3CCCN3C)nn2)C)cccnc1 29378,c1(C(=O)NC2CC(C)(CNC(CS(CC)=O)=O)C2)cc(Cl)n[nH]c1=N 29379,N1(C(C2(C(F)(F)F)CCC(=C(C)C)CC2)=O)CCOc2cccc(C(=O)O)c2C1 29380,C1(O)(C(C(N2CC(O)(CC)C2)=O)NC(c2ccc(NC)cc2)=O)CCCCC1 29381,N1(C(C2OCCN(C)C2=O)=O)CC(NC(C2CCC(F)CC2)=O)CC2(CC2)C1 29382,C1(NC(CNC(CNC(c2ccc(C(C)=O)o2)=O)=O)=O)COCC(C)(C)C1 29383,C(C(COC)C(=O)NC(Cc1ccco1)C(=O)N(C)C(C1CCCO1)C)OC 29384,C(C)(CO)(C(=O)N1CC(CCNC(=O)CNC(=O)C(F)(F)F)(CO)C1)OC 29385,N1(C(c2c(C)sc(O)n2)=O)CC(C)C(NC(c2cc[n+]([O-])cc2)=O)C(C)C1 29386,c1(C(N2CCC3CCN(C(C)=O)C3C2)=O)cc(C)c(F)c(S(=O)(=O)NC2CC2)c1 29387,C1(OCCC)CCCCC1C(=O)NCCNC(=O)C(F)(F)C1CC1 29388,c1(CC(=O)N(CC(CC)NC(=O)CN(CC(F)F)CC2CC2)C)csc(Cl)n1 29389,c12cccc(c1)CNC(=O)C(C1CC1)SN(CC)C2=O.c1(SCC)ccccc1 29390,C(=O)(CCCCCC)N(C1CC(NC(CSCCC)=O)C1)C 29391,Cc1ncc(F)c(=NCC2CCN(C(=O)CC3CCC(C)C(C)C3)CC2)[nH]1 29392,N(C(=NCCOC(C)(C)C)NCCc1ccoc1)CC1(CC(C)C)COC1 29393,C1(C(N2CCC(CNC(C(CCC)c3ccccc3)=O)C2)=O)CCC(F)(F)CC1 29394,c1(C(=O)NC(C)(C)CNC(=O)CC2(C)OCCO2)cc(Cl)ccc1-n1ccnc1 29395,C=CCN=C(NCc1nnn(C)c1C(F)(F)F)NCC(CO)C(C)C 29396,Cc1ccccc1CC(C)C(=O)NCC(COC)NC(=O)Cn1ccnn1 29397,C1(CNC(C2(N(C)C)CCCC2)=O)C2CC1N(C(C1CCS(=O)CC1)=O)C2 29398,C(c1ccc(C)c(Cl)c1)=CC(=O)N(CCCNC(CSc1ccc(C)cc1)=O)C 29399,c1(NC(C(c2cccs2)N(CCOCC)CC)=O)c(C)nc(O)nc1O 29400,C1(C(N2C(CCNC(=O)CCC3CCCC3)CSCC2)=O)COCCC1(F)F 29401,N1(C(c2cnn(C)c2C(F)(F)F)=O)CC2CC(NC(C3CCSCC3)=O)CC1C2 29402,c1(C(=O)NCC2CCC(C(N(CC#CC)CC#C)=O)O2)c[nH]c2cnccc12 29403,S(=O)(=O)(c1ccc(NC2CC(C3CC3)C2)c(Br)c1)NCC(C)C 29404,N12CCC(C1CC)NC(=O)Cc1c(cccc1)C2=O.n1(CCC)cc(C(F)F)cn1 29405,C1(CNC(C2(SC)CC(O)C2)=O)CCN(C(=O)CCC2CC2(F)F)CC1 29406,n1(C(C)C)ccc(=NC(=O)C23CC2CN(C(=O)CCC(C)OC(C)(C)C)C3)[nH]1 29407,Cc1cnc(CNC2CC(CCN)C2)n1-c1ccccc1 29408,C1(C)(OCCC)CCCN(C(=O)C(O)C2CN(C(=O)Cc3ccccc3C)C2)C1 29409,C(=O)(C1=CCC(NC(c2ccc(C#N)cc2)=O)C1)NC(C)CC1CC1 29410,C1(c2nc(C)no2)(C(=O)O)CCN(C(C)=O)C1CO.C(C)(C)(C(C)(C)O)NC(=O)OC 29411,C1(C2C(=O)N2C)CC(F)(F)C1.N1(C(=O)NCC#C)CC(C(=O)NC2CCCC2)C1 29412,Cc1coc(C=CC(=O)NCCCC2CCCN2C(=O)C(F)n2ccnc2)n1 29413,C(=O)(CCS(N)(=O)=O)N1CCCC(CCCC(=O)N(C)Cc2onc(CC)n2)C1 29414,N1(C(C(CC=C)CC)=O)CCC2(CCCN2C(=O)CCCC2CC2)C1 29415,CCCCC(CNC(c1ccc(OC(C)(C)C)cc1)=O)NC(C1CCCCO1)=O 29416,c1(C(=O)NC2CCN(C(=O)C=CC=C(Cl)Cl)CC2O)ccc2c(c1)NC(=O)C2 29417,CC1(C)CN(C(=O)C(F)(F)F)CCS1.C1CCCCCn2cc(nn2)COC1 29418,C1(CNC(C(C(C)C)N(C)C)=O)CN(C(=O)C=CC(F)(F)F)CCC12CCC2 29419,C1(C(=O)NCC(CNC(C2CC(C)C2)=O)O)CC(c2cnn(C)c2)=NO1 29420,C1(NC(C2(CCOC)CCCC2)=O)CC(C)N(C(c2ncncc2Cl)=O)C1 29421,C1(C(=O)NCc2nc(CC)on2)CC(O)CN1C(=O)Cc1cncc(C)c1 29422,C(=O)(C1=CS(=O)CCC1)N1CCC(N(CC(C)NC(=O)CC(C)(C)C)C)CC1 29423,N1(C(C2CCCCC2(C)C)C(=O)NCC)CCSC2CCCCC12 29424,C=C1CC2(C1)CC(C(N1CC(CNC(C3CCOC(COC)C3)=O)C1OC)=O)C2 29425,C(=O)(CCCNC(C1CCC1)=O)NCC(=O)Nc1cc(Cl)c[nH]1 29426,N1(C(C(C)(C)Nc2ccccc2)=O)CCN(C(C2CC(F)(F)C2)=O)CC(O)C1 29427,N1(C(C(C)SC(F)(F)F)=O)CCC2(CCC2)C(NC(c2csc(S)n2)=O)C1 29428,N1(C(C2CNC(=O)C2)=O)CC2CC1CN2C(=O)COCC1CCC1 29429,CC(CC(=O)NC(C)Cc1cnn(C)n1)S(=O)(=O)c1ccc(F)cc1 29430,N1(C(CC=CC)=O)CCC2(CCC2)C(CNC(c2ccc(N)c(Br)n2)=O)C1 29431,O=S(=O)(c1cccnc1NCCn1cnnc1)N1CCC2C(C1)C2(F)F 29432,CCC(C)C(C(=O)NCCN(CC)CC)N(C(=O)CCc1cnc(C)o1)C 29433,N1(c2ccnc(C(CC)C)n2)CCCCC(CNC(c2ccc(C)nc2)=O)C1 29434,c1(C(=O)NC2CC(C(NOCC=CCSC)=O)C2(C)C)cnn(C)c1C#N 29435,N1(C(CC2CC(OC)C2)=O)CCCC(O)(CNC(=O)C=Cc2ccc(C)o2)CC1 29436,Cc1noc(CCCOC)n1.C1(CNC=O)CCN(Cc2nc(CC(C)C)no2)C1 29437,N1(S(c2c(C)nc(C)s2)(=O)=O)CCCC2(CCS(=N)(=O)C2)C1 29438,C1(C(=O)NCC=CCNC(=O)COC2CCCCO2)CCS(=O)(=O)N1 29439,CC1(NC(=O)CC2CC(NC(C3CCCSC3)=O)C2)CC(F)(F)C1 29440,c1(C(=O)NC(C2CCN(C(c3cc(C(C)=O)oc3)=O)C2)C)cnn(C)c1C 29441,c1(CNC(c2ccc(C)cc2)CF)ccc(O)cc1.C1(CCC)(O)CCC1 29442,c1(Nc2nccc(COCC=CC3C(C)(C)C3(C3CC3)C)c2)cnn2c1CCC2 29443,c1(C(=O)NCC2(C)CCC(NC(C3CC(C#C)(O)C3)=O)C2)cccc(SC)c1Cl 29444,c1(OC)ccc(C(C)=CC(N2CC(OC)CC(NC(C3(O)CCC3)=O)C2)=O)cc1 29445,c1(C(=O)OC)c(C)[nH][nH]c1=NC(=O)c1ccc(CNC(=O)OC(C)(C)C)o1 29446,Cc1ccncc1C=CC(=O)NC1CC(C)N(C(c2cc(N)cc(F)c2)=O)C1 29447,C12(NC(C=Cc3ncc(C)[nH]3)=O)CCOCC1CN(C(c1nccnc1C)=O)C2 29448,c1(NC(C2CCOCC2)CC)nc(NCc2ccnc(OC)n2)c2ccsc2n1 29449,S(=O)(=O)(CCC)COCCNC(CN)=O.CC(C)(C)N.C1(CCOCCO)CCC1.C 29450,N1(C(CCCC(N)=O)=O)CCCC12CCN(C(c1cnc3nccn3c1)=O)C2 29451,C1(C)(CNC(CC=C(C)C)=O)COCCN(C(C2CCC3(CCCC3)C2)=O)C1 29452,N1(c2ncn(C(C)C)c2)CCC(O)(C(=O)N(C)C)CC1 29453,Cc1cccc(C)c1OCC(=O)NCC1CC(NC(C2(C)CC3CCC2C3)=O)C1 29454,C12(C(N3C(C)(C)C(CNC(=O)CC4CCCS4(=O)=O)CC3)=O)CCC(CC1)OC2 29455,CC1(OCC(=O)NCC2(C)CC(F)C2)CN(C(CCC(O)CO)=O)C1 29456,C1(NC(C=CC(N)=O)=O)CN(C(=O)CCn2ccnc2)CC12CCC2 29457,C1(n2cc(COC(=O)NCC3CC3)nn2)CC2CCC(C1)N2C(=O)Cn1cnnn1 29458,CC1CCCCC1(C)C(=O)NCCCN(CC(=O)NC1CC(C)N(C)C1)C 29459,N1(C(=O)Cn2cccnc2=O)CC2CCC1CN2C(c1nc(Cl)ccc1Cl)=O 29460,c1(C(N2CC(NC(C3(CC)CC3)=O)C(CO)CC2)=O)cccn2nnnc12 29461,C(CCS(N)(=O)=O)NC(C(C1CCN(C(=O)CCn2ccnn2)CC1)(C)C)=O 29462,C12(OC)CC(C1)C(=O)N2.C1(C(=O)OC)(C(=O)OC(C)(C)C)CC1C 29463,N1(C(c2occ(C(N)=O)c2)=O)CCC2(CCCCC2NC(=O)CSC2CC2)CC1 29464,Cc1c[nH]c(CC(N)=O)c1C(N1CCCC1c1cn(C2CCC(O)CC2)nn1)=O 29465,N1(C(Cc2nc(C)[nH]n2)=O)CCC2(CC1)CCN(C(C1CC3CCC(C1)N3C)=O)C2 29466,c1(C(N2C(C)CC(CNC(CCC3CCC(C)O3)=O)C2)=O)ccc(N)c(O)c1 29467,C1(C(N2C(C(=O)NCCC3CCCCC3)C=CCC2)=O)CC2CCC(C1)C2 29468,c1(OC)cccc(CC(=O)NC2CC3N(C2)C3)n1.c1(C(=O)OC)cnco1 29469,C(=O)(C(C)(C(F)(F)F)c1ccccc1)NC1C(c2ccc(C)cc2)C1 29470,C1(C(=O)NCC(C)CC2CCCC2)CCCN(C(c2ccc(CO)o2)=O)C1 29471,N1(C(CC=CC=C)=O)CC2CC1CC2NC(=O)C(C)(C)C1CC1 29472,C1(c2scc(C)n2)CCCN(C(=O)CC(C)(C(N)=O)C2CC2)C1.S 29473,Cn1cnc2c1CCCC2C(=O)N1CC2C(NC(C34CCCN(CC3)C4)=O)C2C1 29474,C#CCCC(=O)N(C(C)C(C)COC)C1(C(=O)OCC)CCC1 29475,Cc1ccc(C(O)C(=O)NC2CC(NC(c3cnc(O)n3C)=O)C2)cc1 29476,Cc1cccc2[nH]c(C(N3CCOCC3CNC(=O)CCc3cnc[nH]3)=O)cc12 29477,CC(C)CC(CNC=O)CC(=O)NC1CC1NC(c1ccc(CCO)cc1)=O 29478,C(=O)(CCCCN1CCCCC1)NCCC1(NC(COCC(=O)NC)=O)CCC1 29479,CCCC(CCC)NC(=O)NCCCCCc1cn(C2CC(F)(F)CO2)nn1 29480,C1(C(=O)NC2CC(CCNC(c3c(C#C)cnn3C)=O)C2)CC2(COCCO2)C1 29481,CCS(=O)(=O)CC(=O)NC1CCN(C(=O)CCC#N)CC1C 29482,C(=O)(C1=CCC(NC(c2cc(C(C)=O)on2)=O)C1)NCCCOCCOC 29483,CC1CC(CCNC(c2cc[nH]c2)=O)CCN1C(c1ccc(C(N)=O)[nH]1)=O 29484,N1(C(c2c(OC)noc2C)=O)CCCN(C(=O)CN2CC(=O)NC2=O)CCC1 29485,C1(CCC=C)(NC(c2cccc(C(F)F)n2)=O)CCN(C(C)=O)CC1 29486,c1(CNC(C(N2C3(C(=O)OC)CC3CCC2)=O)=O)ccc2c(c1F)CCC2 29487,C1(N(C(CSC)=O)C(C2C(c3n(CC)ccn3)OCC2)=O)CC2CCC1O2 29488,c1(OC)ccc(OCc2ccn(C)c(=O)c2)cc1F 29489,C1(C(=O)NC2(CN(C)C(c3nccn3C)=O)CC2)C2CCC1(c1ccccc1)C2 29490,Cc1ccc2c(c1)C(NCCCC(N)=O)C(C)C2 29491,C1(CCOC)CCN(C(=O)C(F)CC2CN(C(c3cnc[nH]3)=O)C2)CC1 29492,N1(C(C2COc3ccccc3C2)c2cn(C)cc2)CC(O)C2(CCS(=O)(=O)CC2)C1 29493,N1(C(CSC)=O)CCc2sc(CNC(=O)Cn3nnc(=N)[nH]3)nc2C1 29494,N1(C(C(Cc2cccc(C)c2)=O)=O)CCC(C(=O)Oc2ncc(Br)cn2)C(C)C1 29495,N1(C(C(C(C)(C)C)OC)=O)CCC2(CC1)CCN(C(C13CC(C1)C(C(F)(F)F)O3)=O)C2 29496,c1(CC(=O)OC)cccc(Cn2nnnc2C(N2CCC3CC23)=O)c1 29497,C(C(CC(C)C)NC(C1(C(F)F)CCOCC1)=O)NC(C1(COC)CC1(F)F)=O 29498,c1(N(C23CC(CO)(C2)C3)C)ccc2c(n1)CCCC2=O 29499,Cc1sc(O)nc1C(=O)NCC(C)(CO)NC(=O)C(C)(C)CN1CCOCC1 29500,N1(C(c2c(C)cc[nH]2)=O)CCC(NC(c2ccc(C(=O)N(C)C)cc2)=O)C1(C)C 29501,CC(CC(C)(C)C)C(=O)NC1CC(O)CN(C(c2cscc2C(F)F)=O)C1 29502,N1(C(c2c(CC)non2)=O)CCC(C(C(C)C)NC(C2(C)CCCCC2)=O)CC1 29503,C(C)(C)(CC(=O)N1CCCCC1C(C)NC(=O)CCc1ccc(C)s1)SC 29504,O(NC(=O)C(C)CN(C(c1cccc(F)c1)=O)C(C)C)CC 29505,CC1CC1N=c1nc2c(ncn2C(C)C)c(NCCc2cc(Cl)ccc2Cl)[nH]1 29506,c1(N)cccc(P(C)(C)=O)c1.N1(C(NC)=O)CCN(c2ncc(Cl)cn2)CC1 29507,Cc1ccc(O)cc1C(=O)NCC1CC1NC(c1cn(C(C)(C)C)cn1)=O 29508,C1(C(=O)NC2CCCC(CNC(C3CCCN(CC)C3)=O)C2)CN2CCN1CC2 29509,Cc1cccc(OCCCC(=O)NCCCCCNC(c2cc(C)[nH]n2)=O)c1 29510,C(CC(N)=O)(C(=O)N1C(CO)CC1C)NC(C1CC(=C)C1)=O 29511,c1(CC)cccc(C(=O)NCC(C)CNC(=O)C(c2cccc(O)c2)(C)C)n1 29512,n1(CC)nnc(C(=O)NCCCCC(=O)NCC2(F)CCN(C)C2)c1C 29513,C12(C(=O)NCC3N(C(=O)Cc4cnccn4)CC3)CCOC1CC(=O)NC2 29514,c1(C(=O)NCC2(CNC(Cc3scc(CC)n3)=O)CC2)cc(OC)ncn1 29515,c1(C(N2CCCC(C(=O)NCC3(CC)CC3)C2)=O)cnc2[nH]ncc2c1 29516,c1(C2(C(N(CCCNC(C3CCCCO3)=O)C)=O)CC2(C)C)cccc(Cl)c1 29517,C1(CNC(=O)CC(C2CC2)C2CC2)CC2(CCC2)CN1c1nc2ccccc2o1 29518,Cc1cncc(CCNC(c2oc(CC(c3c[nH]c(C(N)=O)c3)=O)nc2C)=O)n1 29519,C(=O)(C(C)P(C)(C)=O)N(CCNC(C12OCC(C(=O)NC)(C1)C2)=O)CC1CC1.CC 29520,C1(NC(c2n(C)ncc2)=O)CC2CCC1(NC(c1cc(C(N)=O)co1)=O)C2 29521,N1(C(=O)OC(C)(C)C)CC2CCC(F)(c3nc(CCC4CC4)no3)C1C2 29522,C1(NC(c2cn(CC)nc2C)=O)CC12CCN(C(=O)Cc1nc(=N)[nH][nH]1)C2 29523,c1(OC)ccc(CC(C)C(=O)NC(C)CCNC(=O)Cc2sccc2C)cc1F 29524,C1(NC(C2CN(CC)C(=O)C2)=O)CC2CCC(C1C)N2C(c1cc(C)c(C)o1)=O 29525,C1(C(=O)NCc2c(CNC(C3CCCC(OC)C3)=O)ocn2)C2CCC3C(C2)CC13 29526,C(C)(C)(CC(F)C=O)NC(C(COC)COC)=O.C(C(C)C)N(C)CCO 29527,C(CC1=CCN(C(C2(C)CCCO2)=O)CC1)NC(C(C(C)C)n1cc(C)nc1)=O 29528,c1(C(=O)NCC2CCCC(NC(=O)CCn3cnnn3)C2)cncc(Cl)c1Cl 29529,N1(C(C=CSC)=O)CC2C3CCC(C2C1)N(Cc1n[nH]c(C)n1)C3 29530,c1(OCCC)cccc(CC(=O)NC(C)C(C(C)C)NC(c2cncnc2)=O)c1 29531,N1(C(CCC=C=C)=O)CCCC(C(=O)NC2CN3CCC2CC3)C1C 29532,C(=O)(C1CCCn2nccc21)N1CCC(C2(SCc3n(C(C)C)cnc3)CC2)CC1 29533,Cc1cc2c(cc1C(=O)NC1CC(C)(NC(C3CC4(CC4)C3)=O)C1)OCO2 29534,N1(C(c2cc(OCC)n[nH]2)=O)CCC(C(=O)Nc2cccc(Cl)c2)C12CC2 29535,n1(CC(=O)NC2CC(C(N(C(C)(CO)C3CC3)C)=O)C2)cnc(C#N)n1 29536,c1(C(N2CC(CCNC(c3cc(C)c(N)cn3)=O)C2)=O)ccc2c(n1)OCCO2 29537,C(CC(Cc1ccccc1)NC(C1(Br)CC1)=O)NC(c1cnns1)=O 29538,c1(C(N2CC(CCNC(C3CC=C(C)CC3)=O)C(C)C2)=O)cccc2nc[nH]c12 29539,C1(NC(Cc2c(C)cccn2)=O)CN(C(=O)C(C)OCCN(C)C)CC2(CC2)C1 29540,C1(NC(C(CCC)F)=O)CC2CC1CN(C(c1cc(OC)cs1)=O)C2 29541,C(=O)(C(CCC(C)C)NC(c1cnn(C)c1Cl)=O)N(CC#C)Cc1ccco1 29542,c1(C(=O)NCCC(C)N(C(CC)=O)C)cccc2c(I)n[nH]c12 29543,C(c1ccc2ccccc2n1)=CC(=O)N(C)CC1CCN(C(C(C)O)=O)C1 29544,C#CCCCCCC(=O)N1CC2(CC(C(=O)NC3CC(=O)N(C)C3)CO2)C1 29545,c1(C(N)=O)cc(C(=O)NCC2CCCC2NC(=O)CCOC2CCCC2)ccn1 29546,Cc1nnc2cnc(C(=O)NC3CC(CNC(c4ccc(Cl)[nH]4)=O)C3)cn12 29547,c1(NC(=O)NCC(=C2CCCCC2)Br)ccc(I)c(Br)n1 29548,C1(C(=O)NC2C(C(=O)NC(c3c(C)nns3)C)CC2)CCC(C)CC1 29549,c1(CC)conc1CC(=O)N(C(C)CC(=O)NC1COCC1CN(C)C)C 29550,C(=O)(C(CC1CCCC1)NC(c1cc(F)c[nH]1)=O)N1CC1.C1(COC)CCC1 29551,n1(CC(=O)NCC(C)N(C(c2ncn(CC)n2)=O)CC)cc(C)ccc1=O 29552,C1(NC(CNC(=O)NC)=O)CN(C(=O)CN2CC3CCC2C3)C2CCCCC12 29553,C(=O)(CCCCC(N)=O)N1C(C)CC(NC(=O)C(CCN(C)C)N(C)C)CC1 29554,c1(CNC(C(C)C#N)=O)cccc(CN(C(=O)CCC2CC(C(F)F)C2)C)c1 29555,C1(C2CC2)(NC(CN2CC(CCN(C)C)OCC2)=O)CCCCCC1 29556,CC1(C)CN(C(=O)Cc2ccc(OC(F)F)cc2)CC1c1cc[nH]n1 29557,Clc1ccccc1C(c1ccccc1)ON1CCN(c2nccc(C3CC3)n2)CC1 29558,C(=O)(CCN=[N+]=[N-])N(CCCN(C)C(C1(N(C)C)CCCC1)=O)C 29559,C1(NC(c2nc(C)oc2C)=O)CCN(C(=O)C(F)C(C)C)CC1CO 29560,C1(CNC(c2cc(O)ncn2)=O)CCN(Cc2c(F)cncc2F)CC1(F)F 29561,c1(C(=O)NCC2(F)CC(CNC(C3(C)CCC3)=O)C2)ncccc1N 29562,N1(Cc2ccccc2)CC2CC=CC1C2.c12ccc(nc1)n(C1CCOCC1)c2=O 29563,CC(CCc1ccc(F)cc1)C(=O)NCC(CO)NC(=O)C=Cc1cn(C)nn1 29564,C(=O)(C#CC1CCCCC1)N1CC(C(C(=O)NCC(CCC)CCO)OC)C1 29565,CCC(CCC(=O)NOC(CC(C)C)C(=O)N(C)Cc1ccc(C)nc1)OC 29566,Cc1nn(C)c(C(=O)NCC2CN(C(=O)COC(F)F)CCCO2)c1Cl 29567,S(=O)(=O)(c1cccc(Cl)c1)NCC(=O)NC1CC1NC(=O)C1=COCCC1 29568,C=CC1OCCC1C(N1CCN(CC2(NC(=O)Cn3ccnc3C)CC2)CC1)=O 29569,C1(NC(c2n(C)nc(Br)c2)=O)COC2CN(C(=O)Cc3ccno3)CC12 29570,C1(CC(N2C(CNC(c3ccc(C)n3C)=O)CCC2)=O)COc2ccccc2O1 29571,c1(C(C)(C)NC(C(N2CC(C)=C(C)CC2)=O)=O)ccc([N+](=O)[O-])c(F)c1 29572,C1(NC(c2nn(CC)c(C3CC3)c2)=O)CCN(C(=O)C(=O)NCC2CCC2)C(C)C1 29573,C=CCC(C(=O)NC1CCCN(C(c2snnc2CC)=O)C1)OC 29574,C(=O)(C(C)(C)C(F)F)NCC1(C(C)NC(C(C)OCC(C)C)=O)CC1 29575,CCC(C)(CNC(=O)C(C1CC(F)(F)C1)O)NC(c1snnc1C1CC1)=O 29576,c1(C(N2C(C(=O)NC34CC(C(=O)OCC)(C3)C4)C3CC3C2)=O)ccc(O)c(C)c1 29577,c1(CC(C(=O)NC23CC(CC(=O)OCC)(C2)C3)C)cccc(F)c1 29578,c1(C(N2CC(CC=C)(CNC(C3CC3F)=O)C2)=O)ccc(S(=O)(=O)CC)cc1 29579,C1(COC)CN(C(c2cc(F)c[nH]2)=O)CCN1C(=O)CCc1ccc(O)cc1 29580,N1(C(C2CC(SC)C2)=O)CC2CC(NC(=O)C(C3(O)CCCC3)F)CC(C2)C1 29581,c1(CNC2CCN(Cc3c(-c4ccc(Cl)o4)n[nH]c3)CC2)cccc2c1OCO2 29582,c1(OC)ccc(OC)cc1CN1CCCC1C(N1CCCC(C)C1)=O 29583,c1(OC)ccccc1C(N1CCCC1)CNC(c1sc(C)cc1C(N)=O)=O 29584,Cc1cc2ccc(C(N3CCC(N(C(=O)CSc4n[nH]c(O)n4)C)C3)=O)cn2c1 29585,N1(C(C2N=C(C)SC2)=O)CCOCC(CNC(=O)Cc2cccc(N)c2)C1 29586,C1(C(N2CC=CC(C(=O)NCC3CC(F)(F)C3)C2)=O)C2CCC(F)(F)C12 29587,C(=O)(C(C)CC(F)(F)F)NCCC(C)NC(c1cc2n(n1)CCC2)=O 29588,c1(C(=O)NC(C(C)NC(c2c(C)cc(F)cn2)=O)CO)cnc2c(c1)COCC2 29589,C1(C(N2CC(CNC(CN(C)C3CC3)=O)C2)=O)CC(=O)N(c2ccccc2Cl)C1 29590,c1(C(C)NC(C(C2CC(NC(C=C(C)C(F)F)=O)C2)F)=O)ncc(C)s1 29591,c1(C(N2CCN(c3cc(C)c(F)cn3)CC2)=O)cc(C(=O)O)cc(S(C)(=O)=O)c1 29592,C1(C)(C(=O)NCC2CC2C2CCN(C(CCCCOC)=O)CC2)CC(=O)N(C)C1 29593,c1(C(N(CCCNC(C(CC)C)=O)Cc2ccccc2)=O)nc(C)ccc1F 29594,c1(SC(C)(C)C)ccc(Cl)c(Cl)c1.c12ccccc1NCCS2 29595,CCCCC(O)C(C)C(=O)N(CCCC(=O)NCCN(C)C)C(C)C 29596,N1(C2CC2)CC2C(NC(c3c(COCC)c[nH]n3)=O)C2C1.C12CC1N(C)CC2=O 29597,C1(O)(CNC(c2c(C(C)C)occ2)=O)CCCN(C(C2(S(C)(=O)=O)CC2)=O)C1 29598,C(=O)(C(C(C)(C)C)NC(N)=O)N1CC(C)(c2cn(C3CCC4(CCC4)C3)nn2)C1 29599,CC(C)C(F)(F)CC(=O)NCC1(C)CN(C(C2CCOC2(C)C)=O)CCO1 29600,C#Cc1ccccc1CC(=O)NC(CNC(=O)C(O)C(C)(C)O)C1CC1 29601,Cc1cc(C)n2nc(CNC3C(CN)CCC34CCC4)cc2n1 29602,C1(CNC(c2scc(C)c2C)=O)CN(C(c2ccc(C(N)=O)cc2)=O)CCC1C 29603,N1(C(=O)NC(c2cnn(C)c2)C(C)C)CCOC(C)(CO)C1 29604,c1(-n2c(CC(C=C)C)nc(C3CCCCC3)n2)ccnc2ccccc12 29605,C1(NC(CCC(=O)OC(C)(C)C)=O)CC2CC1CN2C(c1cnc(C(N)=O)s1)=O 29606,CC(O)C(C(=O)NCC(C)(C)C#N)NC(=O)C(c1ccccc1)C 29607,c1(-c2nc(CC)nn2-c2cccc(NC(C)=O)c2)cnn2ccc(O)nc12 29608,N1(C(C2CCn3nccc3C2)=O)CCCC2(CCN(C(C34CC(F)(C3)C4)=O)C2)C1 29609,C=CC1(CC(N2CCC(NC(c3cscc3C)=O)C(CC)C2)=O)CCOCC1 29610,C1(NC(c2cn(CC=C)nc2)=O)CCCN(C(=O)CC2CC(O)C2(C)C)C1CC 29611,CCCCCCC(=O)NCC(CC)NC(C1CCCSC1C)=O 29612,C(=O)(C#CC1CCC1)NCC1(C(=O)NC(C(C)C)C(N)=O)CC(C)(C)C1 29613,c1(CNC(C(CCCC)ON=C(C)C)=O)c(C)nc2sc(C)cn12 29614,C(CCC(C)C(=O)NCC12CC(CO1)N(C(=O)CCc1nc(O)n[nH]1)C2)OC 29615,c1(C(=O)NC(CNC(C(c2cccc(C)c2)(F)F)=O)C)ccnc(C)c1C 29616,C1(CNC(C(C)SC(F)(F)F)=O)C(C)CCCN1C(=O)CC1(O)CCCOC1 29617,c1(N(C)C(C2CSCCN2C(c2ccc(Br)nn2)=O)=O)cccc(O)c1F 29618,c1(C(N2CC(O)(CCNC(c3c(C)cc(F)s3)=O)C2)=O)cc2ccc(Cl)cc2o1 29619,N1(C(CNC(CC)=O)=O)CCCC2CN(C(=O)C(c3ccc(C)cc3)C)CC12 29620,C(C(CC1CC1)C(=O)NC(C)COC(F)(F)F)NC(C(C1CC1)OC)=O 29621,n1(CC(C)CO)nc(-c2ccc(C(F)(F)F)cc2)nc1-c1nc(Cl)cs1 29622,N1(C(C(CNC(c2ccc(C)nc2O)=O)O)=O)CC2OCC(C)C2C1 29623,c1(NC2CC(C(=O)Nc3snc(C)c3C#N)C2)ccc2c(O)nc(C)nc2c1 29624,CCC(C#N)(CC)C(=O)NCC(O)CNC(C1(OC)CC1)=O 29625,C(=O)(CCCCCCNC(C1(C#N)CCCOC1)=O)NC(C)C(C)n1cccn1 29626,c1(C(N2CCC(CNC(=O)C(O)c3ccco3)C2)=O)cncc2nc[nH]c12 29627,N1(C2C3CCC(C3)ONC(=O)CNC2=O)CCOC2COCC12.COOC 29628,C1(COC)(CNC(c2csc(C)c2N)=O)CCN(C(=O)C(C#N)C2CC2)CC1 29629,C1(CC)CN(C)C(=O)CN1C(C1(NC(C2CCCC2)=O)CCCCC1)=O 29630,C1(NC(C2C(C)C2)=O)CC2(C1)CC(NC(c1ccc(C(C)(C)C)nc1)=O)C2 29631,c1(CC(=O)N(C2C(N(C(C3(C=C)CC3)=O)C)CCCC2)C)cc(C)nc(O)c1 29632,N1(C(c2cocn2)=O)CC2C(NC(C3(CO)CC(F)(F)C3)=O)C2C1 29633,C(N=c1cc(C(F)F)nc[nH]1)C1(CNC(C(C(C)C)N2CCCCC2)=O)CC1 29634,c1(CN(C(=O)C(=O)NCCc2ccc(C#N)cc2)C)sccc1S(C)(=O)=O 29635,c1(OC)ccnc(C(=O)NCC2CCCCN(C(c3csnc3C)=O)C2)c1F 29636,c1(C(=O)NCC(C)CNC(c2cc3nc[nH]c3cn2)=O)cncc2sccc12 29637,c1(OCC(c2[nH]c(C)c(C(=O)OC)c2C)=O)ccc2c(c1)CCC(=O)N2 29638,C1(C(=O)NCCCC=C)(NC(=O)C(F)OC(F)(F)F)CCCC1C 29639,CN1CCN(C(=O)CCC2NC(=O)NC2=O)C(CNC(=O)CCc2nncs2)C1 29640,c1(N2CCC(CCNC(=O)C(c3ccccc3)O)CC2)ncc2cccnc2n1 29641,N(C(=NCCNC(c1cccc(F)c1)=O)N1CCCC2(CC2)C1)C(CC)C 29642,C1(NC(C2(CC)CN(C(Cn3ncc(CC)c3)=O)C2)=O)CC(CO)N(C)C1 29643,C(=O)(CC(C(=C)C)OC)NC1(CNC(c2cn(CCC=C)nn2)=O)CCCCC1 29644,c1(C(=O)OC)ccc(C(=O)Nc2cccc(C(=O)Nc3cncnc3Br)c2)cn1 29645,C1(C)(C(N2C(C(C)NC(C(c3cccc(C)c3)C)=O)CCC2)=O)C(C)(C)C1(C)C 29646,C1(NC(C=C(C)C(C)C)=O)C2CC1N(C(=O)CC(c1ccccc1)NC(N)=O)C2 29647,C(N=c1[nH]cncc1Cl)C1(NC(c2c(C)n[nH]c2C)=O)CCOCC1 29648,CCCC(C#N)C(=O)NCC1(F)CC(NC(=O)Cc2cncn2C)C1 29649,C(=O)(CC(C(F)(F)F)NC(=O)C(C)(O)COC)NC(C#CC)(C)C 29650,N1(C(c2cc(CNC(c3c(C)occ3)=O)sc2)=O)C(CO)CCC1C 29651,c1(OC)ncnc(N2CCC3(CC3C(=O)Nc3ccc(O)cc3C(C)C)C2)c1C 29652,N1(C(C)=O)CCC(C2CCCN(CCC3CC3)C2)C1 29653,N1(C(C2(C)CCCCC2)=O)CC2CCC(C1)N2C(c1cc(I)c(O)c(I)c1)=O 29654,C1(C(=O)NCCNC(c2cnn(C)c2C(C)(F)F)=O)Cc2ccccc2CO1 29655,c1(CN2CCC(NC(=O)NCc3ncc(C)s3)CC2)cc2ccccc2[nH]1 29656,CCC(C)C(C(=O)NCc1cc(C)on1)NC(=O)CC(C)N(C)C 29657,CC(C)CCCC(C)C(=O)NC1C2CC3C(C2)C13C(=O)N(C(CO)C1CC1)C 29658,c1(C(N(C2CCN(C(C(=CC3CCCC3)C)=O)C2)C)=O)nc(Cl)c(Cl)s1 29659,C1(C(=O)NC(c2ccccc2)(C)C)CC(F)CN(C(=O)Nc2cncc(F)c2)C1 29660,CCCCC(C(=O)N(CCCCC(=O)N1CCC1CF)C)N(C)C 29661,C1(C(=O)Nc2ccc(-c3n(C)cnn3)cn2)CCC2(CCC2)NC1 29662,c1(C(=O)NC2(CNC(c3ccc(N)c(Cl)n3)=O)CCCC2)ccc2ccnn2c1 29663,C(=O)(CS(=O)(=O)C(C)(C)C)NC12CC(NC(C(CC)OC)=O)(C1)C2 29664,CCCC(CC)C(=O)N1CCC(CNC(c2csc(CC)n2)=O)C12CC2 29665,C(=O)(CCC(F)(F)C(=O)N1CCCCC1CNC(C1(C)CNC(=O)C1)=O)OCC 29666,N1(CCNC(CN2CCC(C)C2)=O)CCC(NC(=O)C(Cl)=CCl)CC1 29667,Cc1nc(C(C)(C)C)sc1C(=O)NCC1(NC(C2CCCC2)=O)CCCC1 29668,C(=O)(CC(O)CC(C)(C)C)N1CCC(CCNC(Cc2cncc(C)c2)=O)C1 29669,c1(C(=O)NC2CCN(C(=O)C3=COCCO3)CC2)cccc2c3c([nH]c12)CCC3 29670,C(CO)(CCF)NC(C(C)N(C(=O)C=C1CCC1)C1CC1)=O 29671,Cc1cccc2c1c(CC(C)NC(C)CC(F)(F)F)cn2C 29672,c1(C2(C(=O)NC(C)CN(C)C(C3(C)CC3Br)=O)CC2)ccccc1 29673,Cc1oc(C#N)cc1C(=O)NCC1(C)CCN(C(C2CCCC(F)C2)=O)CC1 29674,CCC(CC(=O)N1CCOCC1C1CCOC1)C(C)(C)C 29675,CC1(C)OCCC1CC(=O)NC1CCCC1NC(c1ncccc1O)=O 29676,N1(C(c2onc(C)c2C)=O)CCCCC(NC(c2ccc(CO)s2)=O)C1 29677,Cc1ccc(O)nc1CNC(C1CCCN(CC2CCSC2)C1)=O 29678,N1(C(CC(=O)OCC)=O)CCC(NC(=O)Cn2nnc(C)n2)CC(C)(C)C1 29679,N1(C(c2c(C)nn(C(C)(C)C)c2)=O)CC2CCC1C2NC(Br)NC(=O)CC1CC1 29680,C1(C(=O)NC2CN(C(c3c(C)onc3)=O)CC2(C)C)Cc2ccccc2S1 29681,C(C1=NOC2CCCC12)n1cc(N(C(Cc2ccc(C)cn2)=O)C(C)C)nn1 29682,C=C(C)C1CCC(C)=CC1C(N1CCCCC1C=CC(=O)O)=O 29683,c1(C(=O)NC23CN(C(c4c(CC)nccc4)=O)C(C2)C3)ccnc(Cl)c1OC 29684,CCCC(CC)C(=O)NCC1CCC1NC(=O)COCC1CCCC1 29685,C12(CNC(C(CC)N(CC)CC)=O)CC(CN1C(=O)CC1CCC1)C2 29686,C(=O)(CC(C)P(C)(C)=O)N(CCCNC(CSCC(=O)OC)=O)C(C)C 29687,C(=O)(C1=CCCN(C(C2CCC=CCC2)=O)C1)NCCc1n(C)nnc1 29688,CCC(C)(CCNC(=O)C=CC1CCCCC1)NC(=O)C(C1CCCCC1)F 29689,N1(C(c2ccc(C)cc2C)=O)CC2=C(C1)CN(C(C1(C)CCCS1(=O)=O)=O)C2 29690,C12(C(=O)NC3(C(=O)OCC)CC3)CCC(CN(C(=O)C3=NOCC3)C1)C2 29691,CCCC(C)(CCC)C(=O)NC1CN(C(=O)CCNC(N)=O)CC1C1CC1 29692,C(CC1=CCN(C(c2cc(C#N)c[nH]2)=O)CC1)NC(C(C)SC1CCCCO1)=O 29693,c1(C(=O)NCC2CC(C)(C)CN2C(C2CC(=O)N2)=O)cnc(O)c2ncccc12 29694,Cc1nc2ccnn2c(C)c1C(N1CCN(C(c2cnc(O)n2C)=O)C(C)C1)=O 29695,Cn1cnc(CNC(C2CC(C)(NC(=O)CCCc3cnn[nH]3)C2)=O)c1 29696,Cc1ccc(C(=O)NC2CC(CCNC(c3cc(O)n(C(C)C)n3)=O)C2)nc1 29697,N1(C(CCC2N(C)CCC2)=O)CCN(CCN(C(=O)CCCCC2CC2)C)CC1 29698,C1(CNC(c2c(C)cco2)=O)CN(C(=O)CCCCN2CCCC2)CC12CCC2 29699,c1(C(=O)NC23CC2CN(C(C2CC4(C2)CC(O)C4)=O)C3)cn2cc[nH]c(=O)c2n1 29700,C1(CNC(c2n(C)cc(Br)n2)C(=O)Nc2cccc(I)n2)CCC(F)(F)CC1 29701,C1(c2nc(-c3n(C)cnn3)on2)(NCc2ccc(C(F)(F)F)o2)CCOCC1 29702,c1(C(=O)NCC=CCNC(C2CC3CCC2CC3)=O)ccc2nn[nH]c2c1 29703,CC1OC2(C(N3CCCC(NC(c4cc(C#N)no4)=O)C3)=O)CCC1C2 29704,N1(C(C#CC2(CC)CC2)=O)CCN(C(=O)CSC2Cc3ccccc3O2)CCC1C 29705,C1(C(=O)NCCCCC(C)NC(c2c(C(C)C)ccs2)=O)C2CCC3C(C2)CC13 29706,Cc1c(Br)c(C(N2CCC(CNC(=O)C(C)N(C)C)C23CC3)=O)nn1C 29707,C1(C(=O)NCC2CCC(NC(Cn3c(C)c(Cl)cn3)=O)C2)CCC2(CCC2)CC1 29708,C(=O)(C1=CC2C=CC(C1)C2)NCc1occ(C(=O)NC2(CC=C)CCC2)n1 29709,C1(CC(=O)NC(C(C)C)CNC(=O)CCN2CCCC2=O)CCCS(=O)(=O)C1 29710,c1(C(=O)NCCCCNC(CSCCOC)=O)cc(C)ccc1C1CC1 29711,c1(CC)cccnc1C(=O)NC(C)CN(C(=O)C(=Cc1ccccc1)C)CC 29712,Cc1ccc(C(N2CCCCC2CCC(=O)Nc2ccnc(F)c2F)=O)c(I)c1 29713,N1(C(Cc2cccc(CC)c2)=O)CCC(NC(C2CC(=O)N(C)C2)=O)C(O)C1 29714,C(=O)(CC(C)(C)CN(C)C)N1CCCC(N(C(CCC(=C)C)=O)C)C1 29715,C1(C(COC(c2c(C)nc3ccccn32)=O)=O)CCC2(CC1)OCCO2 29716,n1(CC)nccc1C(=O)NC(C1CCCN1C(c1cc(CCO)on1)=O)C 29717,C12(NC(c3ccc(C)nc3)=O)COCCC1CN(C(=O)C=C1CCCC1)C2 29718,C12(C(=O)NCCc3cncc(C)n3)CC(CN(C(c3c(C)noc3N)=O)C1)C2 29719,CC(CC(=O)NC(C)C=CC(N1CCC(CO)C(C)(C)C1)=O)C(C)(C)C 29720,C(=O)(C1=COCCC1)N1CCC(c2cccc(F)c2)(NC(C2CC(OC)C2)=O)C1 29721,c1(OC)ccc(C2CCN(C(=O)NC(C)C(C)(C3CC3)OC)CC2)cc1 29722,N1(C(c2nn(CC)nc2C)=O)CCC(NC(c2cc(Cl)sc2Cl)=O)C(CO)C1 29723,N(C(=NCCCCl)N1CCC(C)(C2CC2)CC1)CC(c1ccccc1)NC(C)=O 29724,C(C)(CO)(C(=O)NCCC1CC(NC(c2cnc(C(C)C)[nH]2)=O)C1)OC 29725,C1(C(=O)NC(COCc2ccccc2)C2CC2)CC(O)CN1C(C1CCC(O)C1)=O 29726,c1(NC(C2CCC(CCC)O2)=O)c(C(=O)OC)ccnc1OC 29727,C1(C)(COC)CC(NC(=O)C(C)(C)C2CC2)CN1C(c1cnc(S)n1C)=O 29728,c1(OCCC)cc(Cl)ccc1C(=O)NCCN(C)C(C12CC(CO1)C2)=O 29729,C(CCC)(C(=O)NC1CCN(C2CCN(C(=O)Cc3cnc[nH]3)C2)CC1)=CCC 29730,Cc1cc(C(N2CCC(CF)(NC(=O)CC(C)F)C2)=O)cc([N+](=O)[O-])c1 29731,C1(C2CC2)(CNC(CNC(CN(C)C)=O)=O)CCN(C(C2(C)CCOC2)=O)C1 29732,C1(CC(N2CC(C)C(NC(=O)Cc3nncn3C)C2)=O)CCC(F)(F)CC1 29733,C1(NC(c2csnn2)=O)CN(C(=O)C(Cl)=CCl)C2(CCCCOC2)C1 29734,N1(C(c2cc(C(=O)O)ncn2)=O)CC2(CC(NC(C3COCCC3(F)F)=O)C2)C1 29735,C#CC1CCC(C(=O)NCCC(C)N(C)C(c2ccc(C3CC3)c(F)c2)=O)CC1 29736,C1(C(N2CCC(N(CCC)C(C3CC(C(F)(F)F)C3)=O)C2)=O)CC(C)(C)CO1 29737,c1(C(=O)NCCC(C)NC(=O)C=Cc2ccc(F)cc2)cc2c(Cl)cccc2[nH]1 29738,N1(C(COC(CC)C)=O)Cc2[nH]nc(C(=O)NCc3cc(C)sc3C)c2C1 29739,c1(OC(CC=CCC(C(=O)N2CC(COC)(OC)C2)C)=O)cc(C)ccc1F 29740,Cc1cc(C(=O)NCC(=O)OCCCN(CCC(C)C)C)c[nH]1 29741,CC1CC(C(C2CC3CC3C2)Nc2nnnn2C2CCCCC2)(CO)C1.C1CC1 29742,C(=O)(C(CC=C)CC(C)C)NC(C(=O)NCC(=O)NCC#C)CCF 29743,c1(CC)[nH]nc(C(=O)NCC2(C)CCCN2C(C2CC(=C3CC3)C2)=O)c1[N+](=O)[O-] 29744,CC1CCCN(C(c2cnc(C#N)s2)=O)C1CCNC(=O)CCF 29745,N1(C(c2c(C(C)C)con2)=O)CCCC(N(CCO)C(c2csnc2Cl)=O)C1 29746,C1(OC)CCCN(C(C2C3CCC(C3)N2C(=O)C(C)CC2CC2)=O)CC1 29747,c1(C(=O)NC(CNC(C2CCCOC2)CC)(C)C)ccc(C)o1 29748,C1(C(=O)NC2C(NC(CC3(CC=C)CCCC3)=O)COC2)CCS(=O)CC1 29749,N1(C(C(c2cccnc2)C)=O)CCC(N(C(=O)C=CCF)C)CC1 29750,CC(C)(C)CCC(F)C(=O)N1CC(CNC(=O)CC2C=CS(=O)(=O)C2)C1 29751,Cc1cc(=NC2CCC(=O)N(C)C2)[nH]c(N2CCC(CO)(Cc3ccccc3)C2)n1 29752,C1(C(=O)NCC(CC(C)C)NC(CC(CC)OC)=O)CC12CCS(=O)(=O)CC2 29753,C1(C(=O)NCc2nnnn2C2CC2)C=CC(NC(=O)CCn2cncn2)C1 29754,CC1CSCC1NC(=O)CN(C(=O)CC1(O)CCCC1)CC1CC1 29755,C1(CCNC(c2c(C)cc[nH]2)=O)CN(C(c2ccnn2C(F)F)=O)CC1C 29756,C(CCCC(=O)NC(C1CCCCN1C(=O)CC1CC(F)(F)C1)(C)C)N(C(C)C)C 29757,C1(N(C(=O)C=Cc2cc[nH]c2)C)CCC(NC(c2ccc(CO)cc2)=O)CC1 29758,C1(NC(C(C2CCN(C(=O)CCN(C)CCO)C2)C)=O)(CO)CC2CCCC12 29759,c1(C(N2CC3C(CNC(CC)=O)C3C2)=O)oc2ccccc2c1CS(C)(=O)=O 29760,C1(C(=O)NC(CC2CN(C(c3nc(C(C)=O)sc3)=O)C2)C)CCCCN1C 29761,c1(C(=O)OCC)cc(C(=O)NC2CC(C(C)N)C2)cnc1C 29762,C12(C(N(CC(C)NC(C(CCC)O)=O)CC)=O)C3CCC(CC13)C2(F)F 29763,CC1C(NC(c2ccc[n+]([O-])c2)=O)CCN1C(=O)C(C)c1cccs1 29764,C12CCN(C3(CC3)C1)C(=O)NC2.c1(C(CC)=O)ccc(OC(F)(F)CF)cc1 29765,C(CC(C)(C)C)(C(=O)N1CC(CC(=O)NCCC(C)(C)N(C)C)C2(CC2)C1)OC 29766,C1(CC(=O)NC(C)C(=O)NCCNC(=O)CN(C2CCC2)C)(OC)CCOCC1 29767,Cc1ocnc1CC(=O)NCC1CCC(NC(=O)Cn2cnnc2O)C1 29768,c1(C(N(CC(C)NC(=O)C=CCO)CC)=O)ccc(OC)cn1 29769,C#Cc1cccc(C(N2CCC(CN(C)C(C3CC(=O)NC3(C)C)=O)C2)=O)c1F 29770,Cc1noc2nc(C(=O)NOC(=N)O)ccc12.n12cc(nn1)CC1(CCC1)C2 29771,N1(C(C(=O)N(C)C)=O)CCCC(CO)(NC(=O)Cc2nc(Br)n(C)c2C)C1 29772,c1(CN2CCC(CC(N3CCC(N4CCCC4)C3)=O)CC2)cccc2nonc12 29773,CCCC(CC(C)C)C(=O)NC1CC(C)N(C(=O)CCCC(F)(F)F)C1 29774,C(=O)(CCCC(=O)NC1CC(NCCNC(C2CC3(C2)CC(O)C3)=O)C1)N(C)C 29775,N1(C(C=CC(CC)C)=O)CCC2C(NC(c3ccc(F)cc3)=O)C12 29776,CCCCCC(C)CC(=O)NCC1(F)CC(NC(=O)C2=NNC(C(F)(F)F)C2)C1 29777,Cc1noc(N)c1C(=O)NCc1cn(CC(N2CC3CC3(CN(C)C)C2)=O)nn1 29778,C(CNC(=O)C(O)CN(C)C)(CC(=O)Nc1ccccc1Cl)OC 29779,C(=O)(C(CC)C(=O)NC(C)Cn1cccn1)OCC 29780,CC1CN(C(=O)CCn2ncn(C)c2=O)CC1CNC(=O)CSCC(N)=O 29781,Cc1cc2ccc(C(=O)NCC3(O)CCN(C(=O)Cc4ccoc4)CC3)cc2o1 29782,N1(C(c2c(C)snn2)=O)CCC(C(C)CNC(C2(P(C)(C)=O)CC2)=O)CC1 29783,N1(C(CC(C)N(C)C)=O)CCC2CCN(C(c3cc4n(n3)CCNC4=O)=O)CC12 29784,c1(C(=O)NC2CC(N(C(c3c(CC)nc[nH]3)=O)C)C2)cccc2ncnn12 29785,c1(C(N2CCN(C(C(=O)NCC3CC3)=O)CC2C2CC2)=O)nccn2ccnc12 29786,C1(OC)CC(C(N2CCOC(C(N)=O)C2)=O)N(C(=O)CC2CCCCC2)C1 29787,C1(NC(C2CCC(NC(CCC(=O)OC)=O)CC2)=O)CCN2CCC1C2 29788,C1(C2CC2)(CNC(COCCCC)=O)CCN(C(c2cnn3c2OCCC3)=O)C1 29789,C=C(C(=O)NCC(O)COc1ccc(OC(C)(C)C)cc1)C(C)(C)C.C(C)(C)O 29790,CC1(C)CNC(=O)C2=C(C1)N(C1CC1)C(=O)NC2c1ccccc1F 29791,Cc1ccc(-n2nc(-c3ccncc3)nc2CC2CCN(C)C2)cc1Cl 29792,O(S(=O)(=O)CC1(Cl)CCCC1)CC1CN(C(=O)OC(C)(C)C)C1 29793,c1(C=O)nccc2ccn(C)c12.CCC(C)(C)C 29794,C(=O)(C(C(C)C)NC(N)=O)NCC(CNC(=O)Cn1nnnc1C(C)C)OC 29795,C(CCNC(c1ccc(CC(C)C)s1)=O)(C(C)C)NC(C1(CC#C)CCCO1)=O 29796,c1(OC)cc(CCC(N2CC(O)(CO)C2)=O)on1.c12coc(c1)CCNC2=O 29797,N1(C(c2ccc(C)nc2)=O)CCCOC(C(=O)NCCC2(C)CC2(F)F)C1 29798,c1(NC(CNC(=O)NC2CCCC(c3n(C)ncc3)C2)=O)ccc(C#N)cc1 29799,C1(c2cc(C(=O)NCC3CCCN(C(C=C(C)C)=O)C3)on2)CC(F)(F)C1(F)F 29800,c12ccc(cc1)s2.N1(C(COC(C)=O)=O)CC(CO)(NC(C2CCCN2C)=O)C1 29801,C(=O)(CC1=CCOCC1)NC(C(=O)NCc1cccnc1O)C1(C)CC1 29802,C(=O)(C1c2c[nH]nc2CN1C(c1cc2n(n1)CCC2)=O)N1C(C)COCCC1 29803,C1(C#N)(CNC(C)=O)CCN(C(=O)CC2CCOC2=O)C1 29804,CCC(CC(=O)NC1CCN(C(=O)Cc2ccc(C#N)cc2F)C1CC)C(F)F 29805,C(=O)(CC(O)CNC(=O)C(C)c1cccs1)NCC(CC)CC 29806,c1(OC)ccc(F)cc1C(=O)C(=O)NC(C1CC(OCC(F)(F)F)C1)C 29807,c1(NC(C2C(NC(C3(CC4CCCCC4)CC3)=O)C2)=O)ccc2ncoc2c1 29808,C(=O)(C(F)CN(C)C)NC(C)CN(C(=O)CCOC1CC1)C 29809,Cc1cnc(C(=O)NC2CCCCC2C(=O)Nc2cscc2C(N)=O)cn1 29810,C1(C)(CNC(C2CC(C)C2)=O)CN(C(=O)CNC(c2ccc(F)c(F)c2)=O)CC1C 29811,C(CC1=CCN(C(=O)CCF)CC1)NC(C1CCCN1c1ccccc1)=O 29812,N1(C(C(CCOC)C)=O)CCCC(NC(=O)CCOc2cccc(Cl)c2)CCC1 29813,Cc1c2cccc1CN(C)C2=O.C1(N)CC(CO)N(C)C1.c1ccccc1 29814,CC1CCCN(C(c2cnc(C(C)O)s2)=O)C1CCNC(=O)CCNC(N)=O 29815,c1(CC)ccc(F)c(C(=O)NCC(O)CNC(c2c[nH]c(=N)o2)=O)c1 29816,C1(CNC(c2[nH]nnc2C2CC2)=O)C=CC(NC(=O)CC2CCCC2)C1 29817,c1(N(CCOC)CCNC(=O)Cn2cnc([N+](=O)[O-])c2)ncnc2scc(C)c12 29818,C(C(CNC(C1CCC(C)(C)CC1)=O)S(C)(=O)=O)NC(CN1CC(C)(OC)C1)=O 29819,CC1CCCCC1OCC(=O)OCc1ocnc1C(=O)NCCC(C)N(C)C 29820,N1(C(c2cccc(C)c2O)=O)CCCN(C(C2(C)CCS(=O)(=O)CC2)=O)C(C)C1 29821,CCCC(C)(CC)C(=O)NCC1=CCCN(C(c2nscc2C)=O)C1 29822,c1(C(N2CC(C(=O)NC(Cc3cnc[nH]3)CO)(CC)C2)=O)cccc2occc12 29823,c1c(F)c(F)c(Cl)c(F)c1F.OC1CN(Cc2cncc(Br)c2)CC1N 29824,c1(OC)ccc(F)cc1C(=O)NCCC1CCCN1C(C1CCS(=O)(=O)C1)=O 29825,c1(C(N(CC(C)O)CCNC(C2(C(C)C)CCC2)=O)=O)cccc2c1CC(=O)N2 29826,C12(CNC(C3(SC)CC3)=O)COCCN1CCN(C(=O)C1CC1)C2 29827,C1(OC)(CNC(c2ccn(C3CCC3)n2)=O)CCN(C(c2ccns2)=O)C1 29828,N1(C(C(C2CCCCC2)=O)=O)CC2CCCC2(C(=O)N)C1.c1(N)ccc(F)cc1 29829,CC(=O)CCN=C(NCCC1(CO)CCC1)N1CCN(c2cccc(F)n2)CC1 29830,c1(CC(CN(C(c2cccnc2OC)C(=O)NCC)C)CO)ccc(Br)c(F)c1 29831,c1(C(N2C(CNC(C3(CCOC)CCCC3)=O)CC2)=O)ccc(F)cc1N 29832,OCCC(N=c1[nH]c2c(Br)ccc(C(F)(F)F)c2s1)C1CCCC1 29833,C#Cc1ccc(C(=O)NCC2(COC)CCCN2C(=O)CCSC2CC2)c(C)c1 29834,C(=O)(CN1C(=O)CCc2ccccc21)NC(CN(C(=O)CSC)CC)C 29835,Cc1nc(CNC(c2nnnn2-c2ccccc2)C2CC23CCC3)sc1C 29836,c1(OC)ccc(Cl)c(C(N2CC(CNC(=O)CCC(C)C)C3(CC3)C2)=O)n1 29837,N1(C(CCCCCNC(C(C)C#N)=O)=O)CCc2c(C#N)cccc21 29838,C1(C(C(=O)NC2C(NC(C3(C(=O)OCC)CC=CC3)=O)C2)C)CCC(C)(O)CC1 29839,C1(C(=O)OC)C2CC1N(C(C1C=CCCN1C(=O)Cc1ccsn1)=O)C2 29840,n1(C(C)(C)C)cc(CCC(=O)NCC(C2CC2)NC(C2(C)CCCO2)=O)cn1 29841,c1(CSCC(N)=O)cn(C)cn1.c1(C(N2CC(C(C(=O)N)F)C2)=O)cocc1C(N)=O 29842,C1(CNC(CN(C(C)=O)C)=O)CN(C(=O)COc2cccc(F)n2)CCO1 29843,C(=O)(CCCCC(N)=O)N1CCCC(CCCCNC(C(CN(C)C)O)=O)C1 29844,c1(COC)cnc2ccc(C#N)cn12.C123CCC(C1)N(C2)C(=O)N3 29845,c1(N2CCC(OCCO)C2)[nH]c(=NCc2ccc3ccsc3c2)nc2scnc12 29846,Cn1cnc2c(N3CCC(CNC(c4cn(CC5CCOC5)nn4)=O)C3)ncnc12 29847,C(CCCC(C)(C)C(=O)NNC(=O)CCCCC(C)C)NC(C(C=C=C)C)=O 29848,N1(C(C2N(C(c3ccc(OC)cc3)=O)C3(CC2)CC3)=O)CC(C)CCC12CC2 29849,N1(C(CC)=O)CC(OC)CC1CNC(=O)C(c1cccnc1)N1CC(OCC)C1 29850,c1(CC(=O)NC(C(C)C)CNC(=O)C=CSc2nc[nH]n2)nn(C)cc1Cl 29851,c1(C(N(C2CN(C(C(CC)OC)=O)CC2O)C)=O)cc(F)cnc1O 29852,c1(C(C)(C)C#N)cncc(C(=O)NCCNC(c2ccns2)=O)c1 29853,N1(C(C(CCC)C)C(=O)NCC2CCCO2)CCc2ccc(C#N)cc2C1 29854,C(C(C(=O)NCC(F)F)N(C1CCC1)CCN(C)C)(C1CCCC1)OC 29855,C(c1cc(Cl)ccc1Br)=CC(=O)NC(CC(C)NC(C1(C#C)CCCC1)=O)C 29856,Cc1cc(C(=O)NC2CCN(C(=O)COCCCC(C)C)C2)nnc1O 29857,C1(NC(C2C(NC(C(C)=CC3CC3)=O)COC2)=O)CC(C)(C)C12CCC2 29858,c1(C(N(C(C(C)NC(C(C)NC(CC)(C)C)=O)=O)C)C)ncccn1 29859,c1(C(=O)NCC2(F)CCC(CNC(C3C(C)C3)=O)C2)n[nH]c2c1CS(=O)(=O)CC2 29860,CCC(C(=O)NC(C1CN(C(=O)CC2(C)CCCC2)C1)C)NC(=O)OC(C)(C)C 29861,N1(C(c2c(C)nccn2)=O)CCC(C(=O)NC2C=CC(C)(C)CC2)CC1(C)C 29862,c1(C(C(=O)NCC(C)N(C(=O)C(O)P(C)(C)=O)C)=O)cc(Cl)cc(Cl)c1 29863,c1(N(CC(C)(C)C)C)cccc(S(=O)(=O)NCCCCCOC(=N)O)n1 29864,CC(C)CCC(O)C(=O)NC1CCC(CC(=O)NCCOCC(O)CO)CC1 29865,C(=O)(CCC(C)(C)c1ccccc1)OC(CC)C(C)C 29866,c1(CC)cc(C(N2CCC3CN(C(=O)CC4(CSC)CC4)CC23)=O)cn(C)c1=O 29867,C(CCCCNC(c1occc1Br)=O)N(C(C(C)N1CCC1)=O)C 29868,C(CCCC(=O)NC(CNC(C1(CO)CC1)=O)CCO)OCC 29869,c1(C(=O)NCCN(C2CCCC2)C(c2c(COC)cc[nH]2)=O)ccn(C)c(=O)c1 29870,CCCCC(O)C(=O)N1CC(NC(=O)CCc2ccc(F)cc2)C2(CC2)C1 29871,CC1C(C(=O)NCC(C)NC(c2cc(CO)cn2C)=O)CCN1C(=O)OC(C)(C)C 29872,C1(F)(CNC(=O)CN2CCCC2=O)CCC(NC(C2CCCN2C(=O)C2CC2)=O)C1 29873,C1(CCC)CC(C(=O)NCCOCCNC(=O)CCC(=O)N(C)C)CCO1 29874,N1(C(Cc2ccc(C)o2)=O)CC(CNC(c2ccc(CO)s2)=O)CCC1C 29875,C(c1cc(F)c(F)c(F)c1)=CC(=O)N(C)CC1N(C(CC(=O)OC)=O)CCOC1 29876,c1(OCC)ncccc1C(=O)NCCOCCNC(=O)C(CC)c1ccncc1 29877,O=C1CN(C(c2cc(O)nc(O)n2)=O)CC2CCCN12 29878,Cn1ccc(C(=O)NCC2(NC(=O)C(F)COC3CC3)CC2)c1C1CCC1 29879,C1(C(=O)NCC(C)NC(=O)OC)CC2(CCN(C(=O)C3=CCCC3C)C2)C1 29880,c1(C(=O)NC2CCC(CNC(C3(CC4CC4)CCCC3)=O)C2)[nH]nc2ncccc12 29881,Cc1cc(F)ccc1S(=O)(=O)N1CCC(C)CC(C(=O)NCc2cnns2)C1 29882,N1(C(C(CCC)OC)=O)CCN(C(c2sccc2C(F)F)=O)CC1C 29883,C1(CC(=O)NC2(CCCO)CCC2)CC1(Br)Br 29884,CC(O)CCCCCC(=O)N1CC(CNC(c2ccon2)=O)C2(CC2)C1 29885,CCN=c1[nH]cc(C(c2ccccc2)=O)s1.C(=O)(CC(C(C)C)OC)N1CCNCC1 29886,C(=O)(C1=CCCC1)NCC(CO)NC(c1cc(CC)on1)=O 29887,c1(C(N2CCN(C(c3coc(C(F)F)c3)=O)C(CO)C2)=O)cc2cnccc2o1 29888,C1(C(=O)NCCC(C)N(C(c2ccc(C)o2)=O)C)CC=CCC1C 29889,c1(C(=O)NC2C(NC(c3nc(COC)sc3)=O)CCC2)cnc2sc(C)c(C)n12 29890,c1(OC)cc(C)c(F)cc1S(=O)(=O)N1CCCC2C1CCN2Cc1cncs1 29891,C1(C)(CN(C(COCCC=C)=O)C)CCCC1NC(c1sccc1SC)=O 29892,CC(C)(C)CCC(=O)NCC12CCC(NC(=O)CCC3CCCCO3)(CO1)C2 29893,N1(C(C2(CC(C)=O)CC2)=O)CCC2(CC1)CC(CNC(c1cc(O)ccc1F)=O)C2 29894,N1(C(c2ccc(C=C)cc2)C(=O)NCC(C)C)CC(C)CC2CCCCC12 29895,Cc1ccc(C(N2CCC(CCC(=O)NC(C3CCCC3)CO)C2)=O)cc1 29896,n1(CCC)nc(C)c(C(=O)N(CCC(N2CCCC2Cc2nn[nH]n2)=O)C)c1C 29897,N(C(=NCCS(=O)(=O)N1CCCC1)NCC1CC1C)CCOC 29898,c1(C(=O)NC2CC2)c(C)nsc1N.C(C(C)=CC(=O)C1(CCNC)CC1)OC 29899,C1(C(=O)NCCN(C)C=O)(OC)CC(C)C1.C1(CC(=O)N)C=CCC1 29900,C(CNC(=O)CCCc1cc(C)no1)(C(C)C)NC(CCCCOC)=O 29901,c1(CN2CCCCC(NC(c3ccc(C(F)F)o3)=O)C2)cc2cc(O)ccc2[nH]1 29902,C1(CC(=O)N(C)CCOCCCNC(=O)CC2COC(=O)C2)OCCC1(C)C 29903,N1(C(Cc2n(C)ccn2)=O)CC2CC1C2NC(=O)CC1CCC1 29904,Cc1ccc2nc(C)c(C(=O)NCC(O)CN(C(=O)CC#N)C)cc2c1 29905,N1(CC=C)CCc2nc(C(=O)NCC3(CCOCC)CCCC3)cn2CC1 29906,CC(=O)n1cc(CN2CCC(C(c3ccc(O)c(C)c3)=O)C2)nn1 29907,CN1CC(C)(C)CC1C(N1CCC(CN(c2ccccc2)CC2CC2)C1)=O 29908,CCC(N=c1[nH]c2c(c(=NC(C)c3ncc(C)s3)[nH]1)CSC2)C1CCCC1 29909,Cn1cc(-c2ccc(CNc3cccc4[nH]cc(C#N)c34)nc2)c2ccccc12 29910,CCC(CC)C(F)C(=O)N1CC(F)CC1CC(=O)NCc1ccc(F)c(C)c1 29911,n1(CC(=O)NCCCCCNC(CCC=C=C)=O)ccc(=O)n(C)c1=O 29912,CCC(CC)CC(=O)N1CCC(O)(c2cn(Cc3cncc(Cl)c3)nn2)CC1 29913,c1(C(N2C3CN2CCN3)=O)ccc2c(c1)CCC2.c1(CC)nc(C)ccc1O 29914,c1(OC)ccc(F)c(CNC2CCCC2NC(c2ccc(F)cc2C#N)=O)c1Br 29915,CCCCC(O)C(C)C(=O)NC1(C)CCCC1NC(=O)C=CC1CCCC1 29916,C(=O)(C#CC1CCCOC1)N1CCC(NC(C2CCC(CC)O2)=O)C(C)C1 29917,c1(C(=O)NCCCC(C)NC(C2(CC)CCCO2)=O)c(C)nc(O)nc1S 29918,C12(C(=O)NCC3CCC=CCC3)CCCC1N(C(c1sccc1F)=O)CC2 29919,Cc1ccc(C(=O)NC(C(=O)NOC2CC3CCC2C3)c2cccnc2)nc1C 29920,Nc1c(C(N2CC(F)(F)CC2CNC(=O)CCF)=O)cccc1[N+](=O)[O-] 29921,C1(OC)CC2CC1CN(C(C1CC(C)N1C(c1sncc1C)=O)=O)C2 29922,c1(C(=O)NC2(CNC(CN(C3CCC3)C)=O)CCCC2)ccnc(N(C)C)c1 29923,c1(NC(=O)NCC(=O)NC2CC(NC(c3cocn3)=O)C2)ccc(Cl)cc1 29924,CP(C)(=O)C(O)C(=O)NC1CCCN(C(=O)CSc2cccc(Cl)c2)C1 29925,c1(N(CCCN2CC2=O)C(C2CCC2F)=O)ccccc1.C=CCCOC 29926,CC(CC(=O)NC1CCC(C(C)(C)C)C1)C(=O)OC(=O)C1=CCCC1 29927,N1(C(C(C)OCC(C)C)=O)C2CCC(C2)C1CNC(c1cncc(F)c1)=O 29928,C1(C(=O)NCC(CN(C)C(C2CNC(=O)N2)=O)O)(N(C)C)CCCC1 29929,C1(C2C(C(C)C#N)C2)C2CC1N(C(=O)CC1CCOC1)C2 29930,Cc1cc(C(=O)NC(CNC(c2ncn(C)c2C)=O)CO)c(Br)s1 29931,C1(NC(C(CCC)C)=O)CN(C(=O)C2=CCC(C)(C)CC2)CC2(CCC2)C1 29932,N1(C(=O)NCc2nc(C)on2)CCc2ccccc2C1C(N)=O 29933,C(=O)(CC(O)CN(C)C)NCCC(C)(C)NC(c1c(-c2nc(C)sc2)c[nH]c1)=O 29934,N=c1nc[nH]c(=NCCOC2CCN(C(=O)C=C3CCC3)CC2)[nH]1 29935,N1(Cc2scc(-c3c(C#N)scc3)c2)CC(O)C(C#N)C1 29936,n12cc(cn1)C1C(C1)NC(=O)C2.C1(C(=O)NCCN2CC3CC3C2)CCCCC1 29937,c1(C(=O)NCC(=O)NCC(C)(C2CCC2)NS(C)(=O)=O)ccnc2ccncc12 29938,c1(C(=O)NCCC(=O)NCC2CN(C(=O)C=C3CC3)CCO2)ccc(F)cc1Cl 29939,c1(C(=O)CC2(C(=O)NCc3nnsc3CO)CCCC2)cc2n(n1)CCCO2 29940,O=S(=O)(c1sccc1I)N.N1(C(CN)C2CC2)CCOCC1 29941,Cc1nc(=N)[nH]cc1C(=O)NCCNC(C1CCN(CCF)CC1)=O 29942,C(CC(CNC(=O)C(CSC)N(C)C)NC(=O)CC(C)=C(C)C)OC 29943,N1(C(C=CCN(C(=O)CCC2CCCC2)C)=O)CCC(c2nncs2)C1 29944,c1(C(CO)NC(=O)Nc2nccc(SC)c2)cc(Br)ccc1C 29945,C(=O)(CCCCCNC(N1CCOCC1CC(=O)OC(C)(C)C)=O)NCCOC 29946,CCC(C)C(=O)C(=O)N1CC(C)C(C)(C(=O)NCCN(C2CCCCC2)C)C1 29947,N1(C(=O)CN2CSCC2=O)CCC2(CCN(C)C2)C1.C(C=O)NCCC 29948,C12(C(N(OC)C)=O)CC1CN(c1ccnc(NCC3CCCCO3)n1)C2 29949,C(=O)(C(CCC)C(=O)OC)NC1C(CC(=O)NCCC#C)CCC1 29950,c1(C(=O)NCC2(NC(CCn3ccc(C)n3)=O)COC2)cn2ccc(Br)cc2n1 29951,N1(C(CCc2c[nH]c(=N)[nH]2)=O)CCC2(CC1)CC2C(N1CCC(CF)CC1)=O 29952,C=CC(C)(CC)NC(c1cc(CNC(c2scnc2C)=O)[nH]n1)=O 29953,N1(C(C)CNC(c2cc(C(N)=O)c[nH]2)=O)CCN(C(=O)CN2CCOC2=O)CC1 29954,CC(C(c1cccs1)NC(=O)CCc1nccs1)NC(=O)COCC1CC1 29955,CC1CN(C(=O)C(C)(C)C2CCCCO2)CC(C)C1Nc1ncnc(O)c1Br 29956,Cc1nn2ccccc2c1C(=O)NCC1(CNC(C2CCCC2(F)F)=O)CCC1 29957,N(C(=NCCC1CCN(CC(F)(F)F)C1)NCC1CC1)Cc1cccc(C)c1.O 29958,c1(C(N2CCN(C(c3scc(C#N)c3)=O)C3C2C3)=O)ccc2ccccc2c1 29959,Cc1nc(C(F)(F)C(=O)N2CCCC2CNC(=O)CC2C=CCCC2)n[nH]1 29960,C(=O)(CCCS(N)(=O)=O)N(CCC(c1cccs1)NC(C(C)OCCCC)=O)C 29961,C1(NC(C(COC)O)=O)CN(C(=O)C(C)(C)n2cncn2)CC2(CCC2)C1 29962,c1(C(N2CCC(C)(CNC(C(CCCC)O)=O)CC2)=O)cc(OC)c(O)c(N)c1 29963,C(C)(CCC(=O)NCC1OCCC1C(=O)NCC1(C#N)CCC1)OCC 29964,c1(C(N(C2CCN(C(C3CC3OCC)=O)CC2)CCC)=O)ccc(F)cc1Cl 29965,C1(N(C(C(N2C(=O)CCC2=O)C)=O)C)CCCN(C(=O)Cn2cnnc2O)CC1 29966,Cc1ccncc1CC(N1CC2C(CNC(C3(CO)CCCO3)=O)C2C1)=O 29967,Cc1cnc(C#N)nc1N1CC(CO)(NC(C2CCC3CC23)=O)C1 29968,CC1CC(=O)NC1C(=O)NC1CCCC1NC(c1cc(-c2ccco2)[nH]n1)=O 29969,CCCC(O)(CCC)CC(C=O)N1CCC12CC(C(=O)OC)C2(C)C 29970,C1(NC(Cc2ncc(C)o2)=O)CC2CC(NC(=O)CC(F)(F)C(C)C)CC2C1 29971,N1(C(CCNC(CC(C)C)=O)=O)CCC2CN(C(c3cn(C)nn3)=O)C2C1 29972,N1(C(c2cc(C)ncc2)=O)CCC2CCN(C(=O)C(C)OCC(F)(F)F)CC12 29973,n1(CC(=O)NCCn2cccn2)ccc(=NC(=O)c2cccnc2O)nc1O 29974,C(CC(C(=O)N1CCC1CN=[N+]=[N-])NC(c1nc(C)sc1C)=O)OC 29975,C(=O)(C(CC(C)C)NC(C1CCC1)=O)NCC(CC)NC(=O)Cc1cccs1 29976,c1(C(=O)NC2CCC(N(C(C3(C)CC(=C)C3)=O)C)C2)onc(C)c1C(F)(F)F 29977,c1(C(=O)NCCCN(CCOC)C(C2SCCC2C)=O)cc(C2CCC2)nn1C 29978,C(=O)(C(C)(C)CN1CCOCC1)N(CCN(C(C1C(=C)C1)=O)C)C 29979,C(C(O)C(=O)N(CC(C)C(=O)NCC1CSCCO1)C)SC 29980,C(C(=O)NC(CO)C(CC)NC(=O)Cn1cc(C(C)=O)nn1)(C(C)C)SCC 29981,N1(C(C2C(C=C)C2)=O)CCC(CNC(c2ccnn2C(C)CC)=O)(COC)CC1 29982,N1(c2ccnc(C)n2)CC23CCCC2(CN(C(C2(CC4CC4)CC2)=O)C3)C1 29983,N#CC1CCCC(CC(N2CCN(C(=O)CCCc3cccs3)CC2C2CC2)=O)C1 29984,c1(C(=O)NCC(CCCC)NC(C2CC(C)=NO2)=O)cc2nccc(Cl)c2s1 29985,C=C1CCN(C(=O)CC=CC)C(C(N2CCC(CO)CC2)=O)C1 29986,c1(C(=O)NCC(C2CCCC2)NC(C(C)SC)=O)noc(-c2ccccc2)c1C 29987,C1(CC(=O)NCC2(NC(C(C(C)C)C)=O)CCCC2)COC(C)(C)CO1 29988,c1(C(=O)NCCC2(O)CCN(C(=O)C3=CCSC3)CC2)cc2c(nn1)CCC2 29989,C1(C(=O)NC2CCCC2CNC(=O)CSCc2ccsc2)(CC)CCOC1 29990,C(=O)(C(C)S(=O)(=O)C(C)C)N1CCC(C(CNC(C(COC)(F)F)=O)F)CC1 29991,CCC(C)C(C(=O)NCC1CCN(C(=O)CCCCNC(C)=O)CC1O)OC 29992,c1(C(=O)NC2CCCC(CNC(C3(N(C)C)CCCC3)=O)C2)cc(F)cc(F)c1 29993,N1(C(CC(C)CN(C)C)=O)CCCC(CC(=O)NCCN2CC3CC3C2)CC1 29994,C1(C(N2C(CCNC(COCCC#C)=O)CCCC2)=O)CCOCC1(C)C 29995,N1(C(c2c(C)nc(C(C)C)s2)=O)CC(C2CCCCN(C(=O)CSC(F)(F)F)C2)C1 29996,C(C1=NOC2OCCC12)NCC1(c2ccccc2)C(C#N)C1 29997,C1(C(=O)NCCCc2ncn(C)c2)CCN(C(=O)C2(CO)CCCO2)O1 29998,N1(C(C(C)OCC)C)CCC(O)(CO)CC1.CCCN(C)C 29999,N1(C(C(C)OC)=O)CCCCC(CNC(c2cnoc2C)=O)C1 30000,C1(OC)CCCC1NC(=O)C(C1CCCC1)Nc1ccnn1C 30001,CCCC(CC(=O)N(C)CCN(C)C(=O)NC1CC1)OCCc1cn(CC)nn1 30002,C(=O)(CCC(=O)N1CCOC(CNC(C2(n3cccn3)CC2)=O)C1)OCC 30003,c1(C(=O)NCCCN2CCN(C(C3(O)CC3)=O)CC2)cc([N+](=O)[O-])ccc1Br 30004,N1(C(=O)C2=COCCO2)CCCN(C(c2cc[nH]c3nccc2-3)=O)C(CO)C1 30005,C1(C(N2CCN(C(c3c(C)onc3)=O)C(C(C)C)C2)=O)CCc2ncccc2C1 30006,Cc1ccc2c(CNC(=O)COC(N3CC(C(F)F)C3)=O)coc2c1 30007,N1(C(c2cccnc2S)=O)CCC2(CCCN2C(c2ccc[n+]([O-])c2)=O)C1 30008,c1(CNC(C(=O)N(c2cccc(OCC)c2)CC)=O)c(C)nn(C(C)(C)C)c1C 30009,C1(C(=O)Nc2nccs2)CN(C(c2ccc(Br)cc2Br)=O)CCC1O 30010,N1(Cc2cccc(I)c2)CCC12CCCCC2 30011,c1(C(=O)NCC2CC(NC(c3cn[nH]c3)=O)C23CCC3)cc2c(Br)coc2cn1 30012,N1(C(c2c(CC)nn[nH]2)=O)CCC2(CCCN2C(=O)CC(C)C2CCCO2)C1 30013,c1(C(N2CCC(O)(CNC(Cn3c(C)ncc3)=O)C2)=O)nnn2c1CCCCC2 30014,Cc1cccc(N2CCC(C(=O)OCC3OC(=O)CC3C(F)(F)F)C2=O)c1 30015,C(=O)(CCCCCN(C)C)N(CC(CC)NC(=O)CSc1n[nH]c(C)n1)C 30016,C1(NC(c2c(C(=O)OC)[nH]cc2)=O)CCC(N(C(=O)CSCC(F)(F)F)C)CC1 30017,Cc1cc(C(N2CC3CCC2C3NC(C2CCC2)=O)=O)c(N)c(F)c1 30018,C(CC)(CCC(=O)N1CCOC(CF)C1)NC(c1c(CCC)nco1)=O 30019,CC(C)CC(C)C(=O)N(CC(O)CN(C(=O)C(C)Oc1ccc(CO)cc1)C)C 30020,c1(C(N2CC(NC(C34CCN(CC3)CC4)=O)C2)=O)ccc([N+](=O)[O-])[nH]1 30021,c1(C(=O)NCC23CC(NC(Cn4ncc(C#C)c4)=O)(C2)C3)cc(Cl)c(Cl)n1C 30022,C(CC1=CCN(C(c2ccc(C)c(C#N)c2)=O)CC1)NC(C(CC=C)OC)=O 30023,N1(CCCC(=O)N(C2CC(NC(C3OCCO3)=O)C2)C)CCc2ccccc21 30024,N1(C(C2(OC)CCOC2)=O)CC(C(=O)N(C)CC=CC(=O)NC)CCC1(C)C 30025,C#CCCCC(=O)NC(Cc1ccoc1)C(N1CC2C=CC2C1)=O 30026,C1(NC(C2=C(C)CC2)=O)CC=C(C(=O)NC2(C(N)=O)CCSC2)C1 30027,Cc1cccc(F)c1C(=O)NC1CCC(NC(C2CC23CC3)=O)CC1 30028,N1(C(C(C)(C)c2ccc(Cl)s2)=O)CCCC(O)(CNC(c2ccc(CO)o2)=O)C1 30029,CCC(CC(=O)NOCc1cn(C(c2ncccn2)C)nn1)C(C)(C)C 30030,N1(C(CCOCCOC)=O)CCC(C(=O)NC(CCO)c2ccco2)(CC)CC1 30031,n1(CC(N2C(C)CC(CNC(=O)CC3CS(=O)(=O)C3)C2)=O)nnc2c1CCCC2 30032,c1(C(=O)Nc2c(C#N)cc(Br)cc2)cnc2c(-c3ccc(CO)s3)cccc2c1 30033,c1(C(N2CC(NC(c3ccc(F)cn3)=O)C3C2C3)=O)ccc2cnccc2n1 30034,C1(C)(OC)CCN(C(=O)C(O)CNC(c2occc2C(=O)OC)=O)CC1 30035,N1(CC)CCCCC1C(=O)N(C)CCN(C)C(c1cnn(CCOC)c1)=O 30036,N1(C(=O)OC(C)(C)C)C2CCC1CC(COCC1CCC(O)CC1)C2 30037,C(=O)(C(CN1CCCCC1)C(C)C)NCCCCCNC(c1cc(C)n(C)n1)=O 30038,C1(C(=O)NC(CC=CC)C(=O)N(C)CC2(F)CCCC2)C2CCC(C2)C1C 30039,c1(-c2n(C)cnc2)ccc2oc(C(=O)Nc3cc(O)ccc3Br)cc2c1 30040,c1(C(N2CCCC(NC(C(C)OCCOC)=O)C2)=O)cnc(OC(C)C)nc1C 30041,C(CCC(=O)N1C2COCC1C2)(C(C)C)NC(CC(COC)(C)C)=O 30042,c1(C(=O)NCC(CC)NC(=O)C(CC)Nc2nc(C)cs2)cccc(=O)o1 30043,Cc1c(C(N2CCN(C(=O)CC3C=CCCC3)CC2CO)=O)nn(C)c1Br 30044,CC(F)(F)C(C)(C)CNC(=O)NC1(NC(=O)OC(C)(C)C)CCCC1O 30045,N1(C(C)C)CCCC1CC(=O)NCC(C)(C1CC1)NC(=O)CSC(F)(F)F 30046,Cc1cc(C(=O)NC2CC23CN(C(=O)COC2CCCC2)C3)nc2nccn12 30047,CN1CCOC(C(=O)NCC2(F)CCC(NC(=O)CSc3ccccc3)C2)C1=O 30048,c1(OC)ccc2c(C(=O)NC3CC(O)(CNC(=O)C(C)C)C3)cnn2c1 30049,C1(SCC(N2CCCCC2Cn2cc(C3CCC3)nn2)=O)CCCC(CCO)C1 30050,C1(CNCc2c(F)ccc(C(=O)NC)c2)COC(C)(C)CN1C(=O)OC(C)(C)C 30051,C#CCCCCCC(=O)N1CCCOC(CNC(=O)CCSC2CCCC2)C1 30052,C1(C(=O)OC)COC2(CCC2)CN1C(c1cc(OC)c2occc2c1)=O 30053,CC1CN(C(=O)CC(C)(C)CCC2OCCO2)CCC(C2CCNC2)O1 30054,c1(SC)ncc(C#N)c(N2CC3C(C2)N3C(C2CC2C)=O)n1 30055,c1(C(=O)OCC)ccc(C2CCCCN2C(=O)C(=O)NCCc2ccsn2)n1C 30056,Cc1ccnc(CNc2c[nH]nc2C(=O)Nc2nccnc2C(F)(F)F)c1 30057,C1(C(CC)O)CCCN(C(=O)C(C2CCCO2)NC(=O)Cn2cnc(=N)[nH]2)C1 30058,c1(C(N(CCN(C(C2(CC)CCCC2)=O)C)C(C)C)=O)cc(OC)c2sccc2c1 30059,N1(C(CCNC(C(C=C)C)=O)=O)CC=CCC1C(=O)NC 30060,N1(C(c2cc(C(C)C)n(-c3ccccc3F)n2)=O)Cc2cccc3c2C(CCC3)C1 30061,n1(C(CC)C)ncc2cc(C(=O)NC3CCCCN(C(=O)CO)C3)cnc12 30062,CCC(CNC(=O)CSC1CC1C(=O)OC)NC(=O)Cn1cncn1 30063,c12cc(on1)C(=O)NC2.C1(C(=O)NCCOCCOCCO)CCCC1 30064,C=CCC(C)(CO)CN=c1[nH]c(=NCc2nc(SC)ns2)[nH]c2c1COC2 30065,c1(CC(=O)NCC2(C)CCN(C(Cn3nnc(C)n3)=O)C2)c(F)cncc1Cl 30066,Cc1ccc(C(N2CCN(C(=O)CSS(C)(=O)=O)C(C)C2)=O)c(C(C)C)n1 30067,Cc1c(C(=O)NCCOCCNC(=O)C(C(C)C)n2cncn2)noc1C1CC1 30068,c1(CN(C(CC(=O)O)c2ccccc2)CC)c(Cl)cccc1Cl 30069,N1(C(=O)OC(C)C)CCN(C(=O)C2=CCCN(S(C)(=O)=O)C2)CC2CCCCC12 30070,S(=O)(=O)(CCC(=O)NCC1CC(O)CN1C(c1cccc(=O)n1C)=O)N(C)C 30071,c1(C(=O)NC(CC)CNC(=O)CN2CCN(C)CC2)cnc2ccccn12 30072,C(CCOCC(C)C)(C(=O)N(C1CCC1(C)C)C)NC(c1c(C)ocn1)=O 30073,C1(C(N(CC(C)NC(C23CCCC(C)(C2)OC3)=O)C)=O)CNC(=O)CC12CCC2 30074,C=CC1OCCCC1C(=O)NC1CCN(C(c2c(OC)nsc2OC)=O)CC1 30075,N1(C(CC(C)(F)F)=O)CCn2ncc(CNC(C34CCC3C4)=O)c2C1 30076,C12(C(N(C(CNC(CC(C=C)C)=O)C)CC)=O)C3CC(CC13)C2(F)F 30077,C1(CNC(C(CC)SC)=O)CCN(C(=O)Cc2scnc2C)C12CCC2 30078,N1(C(CNS(CC)(=O)=O)=O)CCCC(C)(CNC(c2ccoc2)=O)C1 30079,CCC(C)CCC(O)CC(=O)NC(C)CN(C(=O)C1=CCC(C)CC1)C 30080,CC1CCN(C(=O)CCn2cnnn2)CC1NC(C1COC(C)(C)C1)=O 30081,Cc1ccc(C#N)cc1C(N1CC(CCNC(=O)Cc2ncc(C)s2)C(C)C1)=O 30082,Cc1cccnc1C(N1CCC(C)C1CNC(C12CC(C1)C(C)O2)=O)=O 30083,C1(CNC(c2csc(CNC(c3ccnnc3C)=O)c2)=O)CCCC12CC2 30084,c1(NC(N(C)Cc2cc(OC)ncc2)=O)cc(F)c(Cl)cc1I 30085,c1(C(=O)NCC2C(NC(Cc3cccc(CC)c3)=O)C2)c(C)cc(C)oc1=O 30086,c1(CC)nn(C)c(CC)c1C(=O)NCC1CCN1C(c1ocnc1C(F)(F)F)=O 30087,c1(C(=O)NC2CC(CCNC(c3cscn3)=O)C2)ccnc(O)n1 30088,c1(C(=O)NCC(C)(C2CC2)NC(C(C)OCCCC)=O)cc(O)cc(C#N)c1 30089,C1(C(=O)NCCC=C)CCCC1NC(=O)C(CC)N(C(C)=O)Cc1ccccc1 30090,N1(C(COCCNC(CC(C)n2ccnc2)=O)=O)CCCN(C2CC2)CC1 30091,C(C(CC1CC1)C(=O)NOCC1CCCS1(=O)=O)NC(C1CCC(=O)C1)=O 30092,C1(C(=O)NC2CC(CNC(C3C(CC)OCC3)=O)C2)CCCCC(F)(F)C1 30093,CCC(C(=O)NCC1CC2(CC(NC(=O)C=CCOCCOC)C2)C1)C(C)C 30094,N1(C(CC(C)(C)C#N)=O)CCC(O)(C2CCN(C(C3CC(=O)N(O)C3)=O)CC2)C1 30095,C1(C2CC2)(C(=O)NCC(C2CN(C(=O)Cc3nccn3C)C2)C)CCC1 30096,c1(C(N)=O)ncn(CC(=O)NCC2CCC(NC(=O)C(=O)NC3CC3)C2)n1 30097,N1(CCCC(=O)NC(C)C(C)NC(c2sccc2Cl)=O)C(=O)NC(C)(C)C1=O 30098,c1(C(N2CCCN(C(C3(OC(C)=O)CC3)=O)CC2)=O)ccc2c(c1)CCCS2 30099,C1(C)(NC(COCCCOC)=O)CCN(C(=O)CCCN2CCCC2)C1 30100,c1(OC)ccc2sc(C(=O)N(C(C)C(=O)NO)Cc3ccc(C)c(C)c3)c(C)c2c1 30101,Cc1cn(C)nc1C(=O)N(CCC(C)NC(C1CCCN1S(C)(=O)=O)=O)C 30102,c1(CCC(=O)NC2CCN(C(C=CCC)=O)C2C)nc2ccccc2[nH]1 30103,CC1C(NC(=O)COC2CCOC2)CCN1C(=O)C=CC1CCC1 30104,N1(C(=O)CCCl)CCC2(CC1)CC(C(N1CCC(O)C1)=O)C2.c1(CN)ccccc1 30105,C=C(C)C(C)(C)C(=O)NC1CCC(NC(c2ccccc2C(F)(F)F)=O)CC1 30106,S(=O)(=O)(c1ccccc1F)NCC(=O)NC1CC(O)C12CCOCC2 30107,c1(C(N(CC(=O)NCCC(=C)C)C)=O)ccn(C)n1 30108,CC1CN(C(=O)C(=O)NC2CC2)CCCN1C(=O)CC12CCC(CC1)OC2 30109,CC1OCCC1C(=O)NCC1CCOC1C(=O)NCCc1cnnn1C 30110,C1(CNC(=O)NC)CCN(C(=O)Cn2ccnc2C(C)C)CC1 30111,C(C(C)(C)C(=O)N1CCCCC1CC(N)=O)NC(CC(C)=CCN)=O 30112,Cc1sc(=O)n(CC(N2CCCC2CCNC(c2cc(Cl)c(Cl)n2C)=O)=O)c1C 30113,C(C)(CO)(C(=O)N(C)Cc1cn[nH]c1)NC(C(c1cnn(C)c1)C)=O 30114,C=C(Cl)CC(C(=O)N=c1cc(C)n(C(C)C)[nH]1)NC(=O)C1=CC2CCC(C1)C2 30115,C(=O)(C1=NOC2(CCOC2)C1)NCCOCCNC(C1(c2c(C)c[nH]n2)CC1)=O 30116,CC1C(=O)N(CC(=O)NC(C)(CNC(c2ncnc(O)c2Cl)=O)CO)C(=O)C1C 30117,C1(C(=O)NCC(CN(C(=O)Cc2cc[nH]n2)C)(C)C)CC(F)(F)C12CCC2 30118,C1C(=O)N=C2C=CN(N2)CC(=O)NO1.C1(C(NOC)=O)CN(C)CCO1 30119,N1(C(CCC(C)OC)=O)CCC2(CCC(NC(=O)CCc3ccoc3)C2)C1 30120,C1(CCC)CCC(C(=O)NC23CC(NC(C4(CSC)C=CCC4)=O)(C2)C3)CC1 30121,C1(CNC(C=C(C)C)=O)CC(CNC(=O)CCOC2COC2)CO1 30122,C(=O)(C1CCC(=O)c2cccn21)NCC(C)(CNC(C)=O)OCC(=O)OC 30123,C1(C(N2CCC(C)(NC(c3cccc(Cl)c3)=O)C2)=O)CCCC1S(C)(=O)=O 30124,C(=O)(C(CCF)NC(=O)CC1CCCSC1)NC1C(C)CC1 30125,C(CCC(C)C)(C(=O)N1CCC(F)(CO)CC1)NC(C(=CC1CCCC1)C)=O 30126,C1(C(=O)NCCN(C2CCCCC2)C(=O)C(C2CCCCC2)O)CCCS1(=O)=O 30127,C(=O)(C(C)CCC(C)(C)C)N1CC(CCCNC(C=C(CC)CC)=O)C1 30128,c1(C(=O)NC2CCN(C(C(CNC(C)=O)(C)C)=O)C2)n[nH]c2ccc(F)cc12 30129,N1(C(c2ncn(C)n2)=O)CCOC2CN(C(=O)CC3CCC(C)(C)O3)CC12 30130,c1(C(=O)NC(C2(C(=O)NCc3ccncn3)CCC2)C)ncccc1N 30131,N1(CCOC)CC(NCCCCCN(C(=O)OC)C2CC2)CC1=O 30132,S(=O)(=O)(c1ccc(C#N)c(NCc2nccn2C)c1)N1CC2C(=C)CC(C2)C1 30133,c1(SC(C)C)ccccc1C(=O)NCC(C)(C)CN(C(=O)CC(C)(C)F)C 30134,C1(CNC(c2cnsc2)=O)COC(CNC(c2cnc(-c3cccs3)s2)=O)C1 30135,c1(NCCOCOC(CC(C)C)C)c[nH]c2cc(F)c(F)cc12 30136,c1(C(=O)NC2CC(NC(Cn3c(C)nnn3)=O)C2)cccc2c1OCC2(C)C 30137,CC(C)CC(C(=O)NC1CC2CC(NC(=O)CSc3nnnn3C)C1C2)C(N)=O 30138,C(=O)(C1C(=O)N1)OCC.C(=O)(CCSC)NC(C)CCOCC1CC1 30139,C1(CC)CCC(NC(=O)C(N2CCC(O)(c3ccc(Br)cc3)C2)=O)CC1 30140,N1(C(c2ccn(CCNC(C3N(C)CCN(C)C3)=O)c2)=O)CC2(CNC(=O)N2C)C1 30141,c1(OC)ccc2nc(N3CCC(NC(=O)Cn4cc(C(C)O)nn4)C3)sc2c1 30142,N1(C(c2ccc(OC)cn2)=O)CC2(CCCN(C(c3cc(O)nn3C)=O)C2)C1 30143,C1(COC)CN(C(=O)Cc2cncc(F)c2)CCN1C(=O)CC(C)OC 30144,C(C(CC(C)C)C(=O)NC(C)(C)CNC(C1(C)CC1)=O)OC 30145,c1(N2CCC(COC)C2)ncc(C)cc1S(=O)(=O)N1CCC1(C)C(=O)OC 30146,C(=O)(C1=CCCC1C)NCC(CC)(C)NC(=O)CCCc1n[nH]c(=N)s1 30147,Cc1ccc(C(C(=O)NC2CNC2)N(C2CCC2)C2CCC2)cc1C 30148,N1(C(c2c(C)nsc2C)=O)CC2(CO)CC1(C(=O)NCC1(C)CC1(C)C)C2 30149,N1(C(COCCCC(C)C)=O)CC2CCC2(CCNC(=O)C=C2CCCC2)C1 30150,C1(NC(c2nc(C#C)sc2)=O)CS(=O)(=O)CC1NC(=O)CC1(N(C)C)COC1 30151,C12CC3CCC(C1)N3C(=O)C(C)c1ccccc1CC(=O)N2.CCC(C)(C)OC 30152,CC(C)CC(O)CC(=O)N1CCC=CC1C(=O)NCC1(C)CC1(F)F 30153,C1(CNC(C2CCOC2)=O)CC2COCC2N1C(=O)CCc1ccc(Cl)nc1 30154,N1(C(C)C)C(=O)CCC1C(=O)NC(C)(CNC(c1c[nH]c(=N)o1)=O)C1CC1 30155,CC1c2ccc(Cl)cc2CCN1C(=O)CN=c1c(F)c[nH]cc1Br 30156,CC1=C(C(=O)NC2CN(C(=O)CC(C)C3CC3)CC23CCC3)C(C)(C)CCC1 30157,C(=O)(CC(CC)C(C)(C)C)N(CCC)CCNC(c1nc(C)c(C)s1)=O 30158,C(=O)(C1=CCC(C(F)(F)F)OC1)NCCCCCN(C(=O)Cc1ccc(F)cc1)C 30159,c1(C(N2C(CNC(c3c(CCC)cccc3)=O)CCC2)=O)ccc2cncn2c1 30160,C1(CNC(Cn2c(CCC)ncc2)=O)CC(F)CN1C(c1cnncc1OC)=O 30161,C(=O)(CC(F)(F)C(F)F)N1CC(NC(=O)C=Cc2ccsc2)C(F)C1 30162,c12ccnc(c1)-n1cc(nn1)NC2=O.C1(OCC)COCC1N(CC)CC 30163,C#CCCCCCC(=O)N1CCC(NC(=O)Cc2cn[nH]c2)CC1C1CC1 30164,c1(CNCCNC(c2cccc(OCC)c2)=O)cccc(I)c1.C(F)(F)(C(F)F)O 30165,N1(C(CC2(C=C)CC2)=O)CC(CNC(=O)CC(C)(C)OC)CC1(C)C 30166,c1(C(N2CC(N(C(=O)CC(C)(C)C3CC3)CCC)C2)=O)ccc2c(c1)CCC2 30167,N1(C(=O)Cc2cccc(F)c2)CCCC(c2cn(CC3COCC3CO)nn2)C1 30168,c1(CN(C(C(=O)N(C(c2nccs2)C)C)=O)C)csc2ccccc12 30169,Cc1cccc2c1c(CN1CCC(C#N)(NC(=O)C(C)n3cccn3)C1)cn2C 30170,C1(C(=O)NCCCCNC(=O)CC2CCCCO2)(COC)CCCCO1 30171,C1(NC(=O)CC(O)c2ccccc2)CN(C(c2ccsc2Br)=O)CC12CC2 30172,N1(C(CCC2C(C)=NOC2=O)=O)CCCCC(NC(=O)COc2cc(C)on2)C1 30173,C1(C(C)NC(c2c(C)c[nH]c2)=O)CCN(C(c2c[nH]ccc2=O)=O)CC1 30174,C=C=CCCC(=O)NC1CC(CC(=O)NCCn2ncccc2=O)C1 30175,CN1CCC2CN(C(C3CC(NC(C4(O)CCC4)=O)C3)=O)CC2C1 30176,N1(C(C2CCC(N(C)C)CC2)=O)C2CC1CN(C(C1(C)CNC(=O)C1)=O)C2 30177,N1(C(C(=O)N(C2(C)CC2)C2CC2)c2nccs2)CCC(C2=NOCC2)C1 30178,C1(NC(CCCOC)=O)CC=C(C(=O)NC2(C(C)O)CC2)C1 30179,C1(C(N(C(C)C(N2CCC(CC(N)=O)C2)=O)CC)=O)CCOC1(C)C 30180,n1(CCC)cc(C(=O)N(C2(CC(=O)NC3CCCC3C(C)C)CC2)C)nn1 30181,C1(NC(c2c(N)cncc2)=O)CC(NC(c2coc(Cl)n2)=O)C12CCC2 30182,N12CC(CC1=O)C2.C1(F)(C(N2CC(NC(C(C)C)=O)C2)=O)CC1(Cl)Cl 30183,CC1C(C)N(C(=O)Cn2ncnn2)CCN1C(c1cc2ncccn2n1)=O 30184,Cc1cccc2cc(C(=O)NC3CCCC3NC(=O)C#CC3CC3)oc12 30185,N1(C(c2ccc(OC)c(OC)n2)=O)C2CCC1CC(NC(C1(C)CCCO1)=O)C2 30186,c1(C(C)(C)Cc2cn(C3COC3)nn2)cccc(O)c1 30187,c1(C(=O)NC(CNC(c2c(C)nncc2)=O)(C)C(C)C)ncc(C#N)cc1Cl 30188,CC12COC(C(=O)NCCC3CSCCN3C(=O)CC3CCC(=O)N3)(C1)C2 30189,c1(C(N2CCNC3CC23)=O)cccc(C2(C(F)(F)F)CC2)c1Cl 30190,Cc1cc(C(=O)NC2CCCC(C(N3CCC(O)C(O)C3)=O)C2)cc(O)n1 30191,Cc1cnc(F)cc1C(=O)NC12CC(NCc3cc(Cl)ccn3)(C1)C2 30192,N1(C(C(C)c2ccco2)=O)CCC(C)(C(N2CCC(CCCO)C2)=O)C1 30193,C1(C(=O)NC(CC#C)C(=O)NCCCc2nc[nH]n2)CC2(CCO1)CC2 30194,c1(OC)ccccc1NC(C1C=CC(NC(c2csc(Br)c2)=O)C1)=O 30195,C(=O)(CCC(=O)NN(C)C)NC(C1C(C(=O)NCC(CCC)C)C1)C 30196,C1(CCOC)(NC(C23CC(C2)C(C)(C)O3)=O)CCN(C(C2CCCN2C)=O)CC1 30197,n1(CC)cnnc1C(=O)NCC(O)CN(C)C(c1cc(C(C)(C)C)on1)=O 30198,C1(NC(c2c(CC)nc(C)n2C)=O)CCN(C(=O)Cc2cnoc2)CC1(C)C 30199,N1(C(CNC2CC(CS(C)(=O)=O)CO2)=O)CCc2ccc(F)c(F)c2C1CN 30200,N1(CCOCC)CCC(=O)N(C2CCOC(C3CCC3)C2)C1=O 30201,Cc1ccc(F)cc1C(=O)NC1CCCN(C(=O)C(n2ccc(C(F)(F)F)n2)C)C1 30202,N1(C(c2cn3ncc(C)c3nc2)=O)CCCc2ccc(S(C)(=O)=O)cc21 30203,C(=O)(C(C)(C)C(C)O)NC(C1CCN(CC(F)F)CC1)C.C12CC(C1)C(=O)N2 30204,C(Cc1ccoc1)(C(=O)N1CCCCCO1)NC(C1CN2CCC1C2)=O 30205,CCC(COC)C(=O)NC(C)C(C)(C)NC(c1cc(Cl)cnn1)=O 30206,CCCCCC(O)CC(=O)NCC1CCCCN1C(c1nc(Br)c[nH]1)=O 30207,C1(C(=O)NC(C)CCNC(=O)C(n2cc(Cl)cn2)C)CC2CCCCCN2C1 30208,C1(CCCOC)CCN(c2nnc(C3CC(F)(F)C3)n2CCC#N)CC1 30209,C#CC1(C)CCCN(C(=O)C(CC(=C)C)NC(c2cc(C3CC3)[nH]n2)=O)C1 30210,C1(CNC(Cc2[nH]cc(C)c2)=O)COCCN(C(c2csc(CO)n2)=O)C1 30211,C(=O)(C(C)(C)CCNC(C1C(CC)C1)=O)NCC1CC(F)(CNOC(C)(C)C)C1 30212,CC(C)N(NC(=O)c1ccccc1C(=O)Nc1ccc(Br)cn1)C(N)=O 30213,c1(CC)ccc2c(c1)CN(c1nnc(-c3ncc[nH]3)n1CCC#N)CC2 30214,c1(C(N(C2CCNCC2)CC=C)=O)nn[nH]c1Cl 30215,Cc1ncc(COc2ccc(CN)cc2)c(NC(=O)C(=O)OC(F)F)n1 30216,Cc1cccnc1OC1CC(NC(=O)NC2CCC(C)(C)C2)C1 30217,c1(NC(C2C3COCC23)=O)ccc(-n2cc(-c3c[nH]nc3F)nn2)cc1 30218,N1(C(c2cnc(CC)s2)=O)CCCCC(NC(=O)C(O)CC2CCOCC2)C1 30219,C1(OC)CCCCC1C(=O)NCC(C)(C)OCCNC(=O)Cc1cc(CC)no1 30220,c1(C(N2CCC(F)C(NC(C3CC3C)=O)C2)=O)cc(SC)ccc1Cl.CO 30221,C(=O)(CCCCC(=O)N(C)CCNC(=O)Cn1cc(Br)c(C)n1)OC 30222,c1(NC(C2CC3CC3N2C(C2CCCCCC2)=O)=O)ccc2c(O)n[nH]c2c1 30223,N1(C(C(CO)N(C)C)=O)C2CCC1CN(C(c1cccc(C(C)(C)C)c1)=O)C2 30224,c1(C(=O)OC)cc(Cl)nc(Cl)c1NC(C1(C)CCN1C(=O)Cc1cscn1)=O 30225,c1(C(=O)NCC2CCCN2C(C23C=CC(CC2)C3)=O)ccc2c(c1)COC2=O 30226,C(=O)(CCCC=O)N1CC(C2CCC2)C(C(C)(C)O)C1.CN 30227,N1(c2nnc(C(CC)(C)C)o2)CCCC(C)(NC(=O)C(C)=C(C)C)C1 30228,C1(C(=O)NCC2CC3(CC3)CN2C(c2ccc[nH]2)=O)CCC(C2CC2)CC1 30229,C1(C(C)(C)C)(CSC)CCN(C(C2C3CC(=O)CC23)=O)C1.c12sccc1NC2=O 30230,N1(C(c2cn(C)nn2)=O)CC2(C1)CN(C(C1CC3(C1)CC(O)C3)=O)C2.CS(=O)(=O)N 30231,c1(C(=O)Nc2ccccn2)cccc(N(CCNC(C23CC(C(=O)O)(C2)C3)=O)C)c1 30232,C1(C(=O)NCC2(C(C)(C)C)CCN(C(C=CCCC)=O)C2)CCC(O)CN1C 30233,N1(C(c2c(C(C)(C)C)ocn2)=O)CCC(F)C(NC(C2(F)CC2(C)C)=O)C1 30234,C1(NC(C2C(C)(C)OC(=O)C2)=O)CC2CN(C(=O)CCF)CC2C1 30235,C1(C(C)NC(C(C)NC=O)=O)CN(C(=O)C(C2CCCO2)C2CCCC2)CCO1 30236,C1(N(C(=O)Cc2ccsn2)CCC)CCN(C(c2nc[nH]n2)=O)C1 30237,N1(C(C#C)C)CCN(C(=O)COCCNC(C2CCCN2C)=O)CC1 30238,N1(C(C(CC)(C)O)=O)CCC2CC(CNC(c3coc(Cl)n3)=O)CCC2C1 30239,Cc1nc(CC2CCCC2)sc1C(=O)NCC(n1cccc1)C 30240,Cc1ncc([N+](=O)[O-])n1CC(N1CCN(C2CCCC2O)CC1)=O 30241,c1(NC(C)=O)ccc(F)cc1NC(N1CCCOC(CCS)C1)=O 30242,C1(NC(C(CC(=C)C)OC)=O)CN(C(=O)C(C)SC)CC1S(C)(=O)=O 30243,N1(CC(NNC(c2ccc(OC)cc2OC)=O)=O)C2CCCC1CC(O)C2 30244,c1(C(=O)NC2(CC=C)CN(C(=O)C(C)SCC)C2)cn(C)nc1C 30245,CC1C(C(=O)N(C(C)(C)CC(=O)NCC2CCCC23CC3)C)=NOC1C 30246,N1(C(c2ccc(CC)o2)=O)CCN(C(c2cc(Cl)cn2C)=O)CC1CC(F)(F)F 30247,CC1CN=C2NC(C(=O)N3C4CCC3C(CNC(c3cccnn3)=O)C4)=NN2C1 30248,C(C1=CCN(C(C2CCC(C(N)=O)CC2)=O)CC1)NC(c1nnn(C)n1)=O 30249,Cc1cc(C(=O)NCC2C(CNC(c3cc(C)oc3C)=O)C2(F)F)c(C)[nH]1 30250,CC(C)(C(=O)NC1CC(F)(CNC(c2cc(C3(C)CC3)on2)=O)C1)C(N)=O 30251,c1(CCC(=O)N(CCC(=O)NCCS)C(C)=O)ccc(Cl)cc1.C(=O)(CO)OCC 30252,c1(C(=O)NCCCNC(c2snc(COC)n2)=O)cnc(C(=O)OC)cn1 30253,C(=O)(C1=NOC(C)C1C)N1CCC(C(=O)NCCC(=O)NC)C1 30254,CC1C(C(N2CCN(CC3(NC(C4(C)CCCN4C)=O)CC3)CC2)=O)CCN1C 30255,c1(CC)nc(C(N2CCC(NC(=O)CCCc3sccc3C)CC2)=O)c(C)o1 30256,C1(C(=O)NCCOCC(N2CC(C)(C(N)=O)C2)=O)CC12CCOCC2 30257,c1(C(=O)NC(CNC(C(CC=C)CC)=O)CC)ccc2c(c1)COCO2 30258,c1(C(C(=O)NCCC)N(CC=C)CC2CC2)ccc(CC)cc1 30259,c12cc3ccccc3n1CC(=O)NCC1CN(CCN1C)C2=O.C(C)(=O)OC 30260,c1(SC2ON=C(C)C2)cccc(CC(=O)N(C)C(c2ccccc2)C)c1 30261,C1(NC(C(CCC)C)=O)CCC12CN(C(=O)CCCCN1CCCCC1)C2 30262,c1(C(=O)OC(CCC(=O)OCC)C(=O)O)cc2ccc(OC)cc2o1 30263,C(=O)(C(C)Cc1cn(CCC(N2CCCC2C(C)(C)O)=O)nn1)OCC 30264,CCC(C)C(C(=O)NC1CCC(C)(C)C1)N(C)C(c1csnc1OC)=O 30265,c1(C(C(C)CCC2C3CN(C(=O)C(C)(C)c4cnccn4)CC23)=O)ccc(Cl)cc1 30266,C=CCC(CC(=O)NCc1nn(C)c(=O)o1)NC(=O)CSC(F)(F)F 30267,CC(C)(O)C(F)(F)CNC(=O)C(CNC(=O)Cn1ncccc1=O)CC1CC1 30268,c1(C(N2CCN(C(CN=[N+]=[N-])=O)CC2)=O)cc2c(F)ccc(F)c2s1 30269,c1(C(=O)OCC)ccc(NC(=O)OC(C)(C)C)nc1Cl.C12(CC(F)(F)C1)NC2 30270,c1(OC)ccc(SCCCC(=O)NCCN2C(C)C2=O)cc1.C1(CO)CCCC1 30271,c1(C(N2CCCN(C(C3CCCCO3)=O)CCC2)=O)cnc2c(c1)CCCO2 30272,c1(C2(C(C3CC3)NCCC(C)NC(=O)CC3CSCCS3)CC2)cccc(Cl)n1 30273,CN1CCCCC1c1ccc(CNc2ccccc2-c2nncn2C)s1 30274,c1(C(=O)NC2CCCC(CNC(C3CC(CF)C3)=O)C2)cn2ncccc2n1 30275,C1(NC(C2CCCOC2)=O)(CO)CCCN(C(c2cnn[nH]2)=O)C1 30276,C(=O)(CC(C)(C)C(F)F)N1C2C(NC(c3nnn(CC)c3C)=O)CC(C2)C1 30277,C1(NC(CCNC(C)=O)=O)CCN(C(=O)Cc2csc(Cl)n2)C1C(C)C 30278,C(=O)(C1=CS(=O)CCC1)N1C(C(C)C)CN(C(=O)CCc2nncs2)CC1 30279,C1(NC(c2ccc(CC(C)C)nc2)=O)CC(NC(=O)CNC=O)C12CCOCC2 30280,C1(COC)(NC(C2CCN2C(C)(C)C)=O)CN(C(=O)CCCN2CCCC2)C1 30281,C1(CNC(CC(COC)C)=O)C(C)CCCN1C(c1cc(=O)c(OC)co1)=O 30282,c1(C(N(C(C)C)CCN(C)CC2NC(=O)NC2=O)=O)ccc2c(c1)C(C)(C)CO2 30283,C1(C(N2CCC(C)(NC(C(CC)C)=O)C2)=O)C2Cc3ccccc3C12 30284,C1(NC(CCc2nc(C)c(C)o2)=O)CCC2CN(CC(=O)N3CCC3)CC2C1 30285,NC(CNC(C1(N2CCOCC2)CC1)=O)CC1CCc2ccccc21 30286,CC(C)C(C)(O)C(=O)N1CCC(CCC(=O)NC(CN(C)C)CCO)C1 30287,C1(C(=O)NCCCN(c2cc(CC(C)C)nc(O)c2)CC)CCc2nncn2C1 30288,c1(CNC(CC)Cc2ccc(Cl)cc2)cc(OC)cc(Br)c1OC 30289,O=C(NNc1ccc(S(=O)(=O)NCCC2CCNC23CCOCC3)cc1)C1CC1 30290,C1(C2(C(=O)OC)CCC2)CCN(C(=O)NCc2ccc(I)cn2)CC1 30291,C1(C)(CNC(CN(C)C)=O)CCCN(C(c2cccc(F)c2Cl)=O)C1 30292,C1(C(=O)Nc2ccc(C(F)(F)F)nc2)CN(C(=O)CCCCCBr)CCC1F 30293,C1(CNC(COCCOCCOC)=O)CCOCC1NC(C1OCC1(C)C)=O 30294,C1(CCC(C)(C)NC(C2CC2(F)Cl)=O)CCN(C(=O)OC(C)(C)C)CC1 30295,C=Cc1ccc(CNCC23CC2CN(C(C2Cc4ccccc4N2)=O)C3)cc1 30296,C(=O)(CC(C)n1cccc1)N(c1ccccc1)CCNC(C1C(C)C1C)=O 30297,CC1CN(C)CC1C(=O)NCC1(NC(c2ccc(-c3cccs3)s2)=O)CCC1 30298,c1(C(N(C(C(=O)NCCOCC#C)C)CCC)=O)coc(OC)n1 30299,C(=O)(CCCCN=[N+]=[N-])N1C(C)CN(C(=O)C(c2ccc(F)cc2)O)CC1 30300,CN1CCC(CC(=O)NC2(C(=O)NC3CC3)CCC2)C1.c12ccc(s1)[nH]c2=O 30301,c1(C(=O)NC(C2CN(C(C3CCC3)=O)C2)C)ccc(N(C)C)cn1 30302,C1(CNC(c2cnn(C(C)C)c2N)=O)CCN(C(=O)C(C)(C)N(C)C)C1(C)C 30303,N1(C(C2C(CC3(NC(C4N(C)CC(O)CC4)=O)CC3)C2)=O)CC(O)CC12CCCC2 30304,C#CCCCC(C)Nc1c(-n2c(C3(Cc4ccccc4)CCSC3)nnn2)cccc1 30305,N1(C(C(CC)C)=O)CC2C(C(=O)OC)C2C1.C12(CC3(CC3)C1)C(=O)NC2 30306,Nc1ccc(C(N2CC(CO)C(O)C2)=O)nc1F.C12CCCC1C(=O)N2 30307,C12CC(F)CN1C(=O)CNC2=O.c1(CSc2nc[nH]n2)ccc(C(F)(F)F)cc1 30308,c1(C(=O)NCC(CC)NC(c2cccn2C)=O)cc(O)ncc1Br 30309,Cc1cc(=NCC2CC(C)(C)CCO2)[nH]c(NC2COCC2F)n1 30310,C=CCC(C(=O)N(C(C)CNC(c1ccc(Cl)nc1N)=O)C)C(C)(C)C 30311,N1(C(CCC2(C)CC2)=O)C(CC(=O)NCCC23CCCC2C3)C2CCCC12 30312,c1(C(N2CC(C)C(CNC(=O)C(F)=C3CCC3)C2)=O)c[nH]c2c(F)cccc12 30313,c1(OC)ncnc(C(N2CCC(CF)(NC(=O)CC34CCC(CC3)C4)C2)=O)c1F 30314,C1(C(N2CCN(C)CC2)=O)CCC2(CC2)N1C(C1(CF)CCC1)=O 30315,C1(NC(c2c(CC)cno2)=O)CN(C(c2cocc2C)=O)CC12CCCC2 30316,N1(C(CCC2CC(OC)C2)=O)CCC2CCN(C(=O)C(C)CSC)CC2C1 30317,c1(NC(C2(O)CN(c3cc(C(=O)OC)ncn3)C2)C)cc(S(C)(=O)=O)ncn1 30318,C(=O)(C(C)(C)CC(F)F)NCC(C(C(C)C)C)NC(c1ccsc1Cl)=O 30319,C1(C#N)(Cc2nn(-c3ccccc3)c(Cn3cncn3)n2)CCOCC1 30320,N1(C(C2(C#N)C(C)C2)=O)CC(CNC(=O)C=CCOC2CCOCC2)C2(CC2)C1 30321,Cc1cncc(C(=O)NC2CC3CCC2(NC(C2CC2C(=O)N(C)C)=O)C3)c1C 30322,CCC(CCO)CN=c1cc[nH]cc1S(=O)(=O)NCC1(CO)CCCCC1 30323,CC1(C)CCC(NC(C2CC=CCO2)=O)CN1C(=O)C=Cc1ccncc1 30324,CC(C)C(C)(CN=c1cc(F)nc[nH]1)NC(c1ccc(F)c(Cl)c1F)=O 30325,c1(C(N2C(C(=O)Nc3ccc(C)nc3)C=CCC2)=O)ccc2c(c1)CCCC2 30326,C12(C(NOCC(CC)(C)O)=O)CCC(CC1)N(C(=O)CCC1CC1(C)C)C2 30327,c1(C(=O)NC2C(C)CN(C(C3CCCN3N=O)=O)C2)[nH]nc2c1COC2(C)C 30328,N1(C(C2CCC(=O)C2)=O)CCc2ccccc2C(NC(=O)Cc2ccc(Cl)s2)C1 30329,N1(C(C(c2cnn(C)c2)NC(c2c(CC)occ2)=O)=O)CCCN(C)CC1C 30330,Cc1cc([N+](=O)[O-])ncc1C(=O)NCCOCCCN(C)C(C1CCCS1)=O 30331,c1(OC(=O)NCC)cccc(C(N2CCCCC2c2ccco2)=O)c1 30332,c1(-c2nc(C(CC)C)nn2C23CC(C2)C3)ccc(Cl)c(S(C)(=O)=O)c1 30333,c1(OC)cc2cc(C(=O)N=c3nc(-c4ccccc4Cl)[nH]o3)[nH]c2cc1OC 30334,N1(C(C=CS(C)=O)=O)CCN(C(c2ccccc2C(N)=O)=O)CC1c1cn[nH]c1 30335,c1(NC(c2ccc(C(=O)NC)cc2)c2nnnn2C)cccc(OC(F)F)c1 30336,Cc1ccc(Br)c(O)c1CN1CC2CN(S(=O)(=O)C(C)CCc3ccccc3)CC12 30337,N1(C(CC(C)SC)=O)CC(NC(c2cc(C)cc(F)c2)=O)CC(F)C1 30338,c1(C(N(C(C)CNC(=O)C(F)(F)C(F)F)CC)=O)ccc2c(c1)COC2 30339,N1(C(C=Cc2cnc(C)s2)=O)CC(CO)C2(C1)CN(c1nc(C)ncc1C)C2 30340,C(=O)(CC(CC1CC1)NC(=O)CS(=O)CC)NC(CCC)C1CCCC1 30341,c1(N(C)CCN2CCC(C(C(=O)OC(C)(C)C)F)C2)cc(F)cc(F)c1 30342,c1(NC2CCCN(C)CC2)[nH]c(=NCC23CC2CN(C)S3(=O)=O)nc2sccc12 30343,C1(C(=O)NC(CCNC(c2nc(C)oc2C)=O)C(C)C)CCOC2(CCC2)C1 30344,N1(C(C(CN(C(c2ccc(C)cc2)=O)C)C)=O)CCCC(C(=O)O)C1C 30345,c1(C(N2CC(CCNC(C(CCC)OC)=O)C(C)C2)=O)c(F)ccc2nc[nH]c12 30346,C(=O)(C(F)C(C)C)NC(CCOC)CNC(c1cnc(-c2ccc(Cl)s2)s1)=O 30347,c1(C(=O)NC2(CC)CCN(C(c3cncs3)=O)CC2)ccc2c(c1)nc(O)n2C 30348,C1(C(N(CCCCNC(=O)Cc2sccc2Br)C)=O)CC(C)(C)CO1 30349,CCC(C)(CNC(C1(C(C)C)CCN(C(=O)CC(C)SC)C1)=O)CO 30350,C1(N(C(=O)CC2CCC(=O)O2)C)CCN(C(C2CCC2C(F)(F)F)=O)CC1 30351,CC(O)(C(=O)NC(Cn1cccn1)C(=O)NCCCc1ccco1)C1CC1 30352,C(=O)(CC(C)C(F)(F)F)NCC1=CCCN(C(C2=CCCC2C)=O)C1 30353,C1(C(=O)NC2CC(F)(F)C2)(CC)CN(C(c2sccc2F)=O)C1 30354,C(C(CC(F)(F)F)NC(=O)CC(Cc1ccccc1)CC)NC(CN(C)CC)=O 30355,C1(CNC(C2COC(=O)N2)=O)CCN(C(C2CCC23CCC3)=O)CC1 30356,CC(C)(CC(=O)NC1CN(C(=O)CC2CCn3cncc3C2)CC1CO)C(F)F 30357,C(=O)(C1=C(Cl)CCC1)N1C(CNC(c2c(C)ncs2)=O)CCC1 30358,C1(NC(CC(=O)NC)=O)CCC(NC(=O)C(C)(F)F)CC1 30359,S(=O)(=O)(c1cc(C)c(Cl)cc1F)N1CC(CC)OCC1 30360,Cc1cc(=NCC2CCc3nccn32)[nH]c(=NCc2sccc2S(C)(=O)=O)[nH]1 30361,C(=O)(CCCCCCNC(c1ccccc1OC)=O)NC(c1ccccc1)CC 30362,c1(C(N2CC3C(CNC(=O)C=CC4CC4)C3C2)=O)ccc(F)c(F)c1 30363,Cn1ncc(C2CC2)c1N(C(=O)Cn1cc(CCS(C)(=O)=O)nn1)CC1CC1 30364,CC1CC(C(N2CCCC(CN=[N+]=[N-])C2)=O)CN(C(=O)CCOCC2CCC2)C1 30365,c1(C(=O)NCC(CC=C)NC(C2(F)CC=CC2)=O)[nH]c2ccc(Cl)cc2c1Cl 30366,C1(C(=O)NCCC)CC2CC2N1Cc1ccncc1Br 30367,N1(C(c2ccnc(C)n2)=O)CC2C3CCC(C2C1)N(C(C1(N(C)C)CCC1)=O)C3 30368,CC1CCC=C1C(=O)NCCC(O)C(=O)NCCC1CCCCCCC1 30369,C1(C(=O)NC2CCOCC2)CC(O)CN1Cc1ccccc1OCCO 30370,c1(OCC=C)ccc(Cl)c(C(=O)NCC#CCNC(C2CCC(C3CC3)C2)=O)n1 30371,C(C(N=c1nc(C2CC2)[nH]s1)C1CCC1)NC(CCC(=C)C)=O 30372,N1(C(=O)NCC)CCC(N2CCC(C(=O)NC3CCCC3NC(C)=O)CC2)CC1 30373,c1(C(N(CCC(C)NC(c2c[nH]nc2C2CCC2)=O)C)=O)ccc(C(F)(F)F)s1 30374,C1(CNC(CN(C(C(C)NC(C2C(C)C2)=O)=O)C)=O)(CO)CC12CCC2 30375,c1(C(N2CCN(C(CCOCC)=O)C(CCO)C2)=O)oc2ccccc2c1CC 30376,C(=O)(C(C)(C)CO)NCC(CC)(C)NC(C1(c2ccc(C)s2)CC1)=O 30377,c1(-c2scc(C(=O)Nc3cc(C)[nH]n3)n2)cncc(OC)c1.c1ccccc1 30378,c1(-c2c(C(N(C3CCCC3)CC(=O)OCC)=O)nccn2)ccc2c(c1)CCO2 30379,C1(N(C(CCCOC(C)C)=O)CC)CCCN(C(=O)CSCC2CCCOC2)C1 30380,C1(CN(C(CCN(C(c2nccn2C2CC2)=O)CC)=O)C)CCOC1C 30381,c1(C(N2CC(O)CC(NC(CC=CC=C)=O)C2)=O)nc2ccccc2nc1C 30382,CC(C)(C(=O)NC(CC1CCC1)C(=O)NCCN1CCCC1=O)C1CCCC1 30383,C(C(C(=O)NCCN1CC=CCC1)NC(c1ccn(C(F)F)n1)=O)OC 30384,N1(CCCNC(C(CC)OC2CCCCC2)=O)CCN(C(=O)CC2CCC2)CC1 30385,C1(C)(C(=O)NC2C(NC(CCOCCC)=O)CCCC2)CCCCCCC1 30386,C(C1CCCCCC1)=CC(=O)NCCCC(C)NC(C1CC(C(C)C)C1)=O 30387,N1(C(c2c(CC)con2)=O)CCC(NC(c2[nH]nc(C(F)(F)F)c2C)=O)C(C)C1 30388,C(C)(CCCC(=O)NC1CCC(C)CC1)NC(c1c(NC)scn1)=O 30389,c1(C(=O)NC(C(C)NC(C(C2CCC2)OCC)=O)C(C)C)scc2c1OCCO2 30390,C(=O)(CC(C)CC(=O)NC1CCN(C(C2(C3CC3)CCOCC2)=O)C1)OC 30391,C(C(N=c1[nH]nc(C#N)s1)C(C)C)NC(c1cc(OC)c(F)c(F)c1)=O 30392,C12(NC(c3c(COC)cc[nH]3)=O)CCC1CN(C(=O)Cc1csc(C)c1)C2 30393,N1(C(C=COCC)=O)CCOC2CCN(C(=O)C=CC(C)C)CC12 30394,N1(C(C=CCNC(C(C)c2cc[nH]n2)=O)=O)CCCC(C)C1CCO 30395,C(=O)(C(C)CC(F)F)N1CC(CC(C(=O)NC(CCOC)COC)F)C1 30396,CC1CCN(CC(C2(c3ccc(Br)cn3)CCOCC2)=O)CC1 30397,C12(C(=O)NC(CN(C(c3nc(OCC)oc3)=O)C)(C)C)CCCCC1C2 30398,CC1CCC(C(=O)NCc2cncnc2)CN1C(=O)CCCOc1cccnc1 30399,c1(NC(C2(NC(CN(C)CCO)=O)CC2(C)C)=O)ccc2ccoc2c1 30400,C(C(C(=O)NC1COCC1NC(=O)C(C)(C)c1cocn1)OC)OC 30401,N12CC(F)CC1C2=O.n1(C(C)C)cc(CNCc2csc(Br)n2)nn1 30402,N1(c2nc(OC)nc(C)c2)CCC(F)(F)C(CNC(=O)Cc2sc(S)nc2C)C1 30403,CC1CCN(C(C2(NC(=O)CC3CCCSC3)CCC(C)(C)C2)=O)CC(C)O1 30404,CC1(C)CCN1CC(=O)NC1CCCC1NC(C1(c2cccnc2)CCCC1)=O 30405,C(CCCCC(=O)N1CC2(CC(CC(=O)NC3CN(C)CC3O)C2)C1)NS(C)(=O)=O 30406,c1(CC(=O)NC(C(C)NC(COCCCCC)=O)CO)ccc(C2CC2)cc1 30407,c1(Cc2onc(COC(c3cc(OC)no3)=O)n2)ccc(O)cc1 30408,C1(CCOC)C=CC(NC(C2(CNC(=O)CC3CC(=O)C3)CCC2)=O)C1 30409,Cc1cnn2cc(C(N3CC(O)CC3c3ccc(F)cc3)=O)cnc12 30410,CC1CN(C(=O)CN2CCCCCC2)CCCN1C(C1CCCC(C#N)C1)=O 30411,C1(CC(=O)NCC(C2CCCC2)NC(C2CC(F)(F)C2)=O)CCCCC1F 30412,C1(C(=O)OCC)CN(C(=O)CNC(=O)Nc2ccccc2)CC(C)S1(=O)=O 30413,N1(C(c2c(CC)nn[nH]2)=O)CC2(CCC2)CC1CNC(=O)CNC=O 30414,c1(NCC(=O)NCC(=C)CCNC(=O)C(C(C)C)n2cncn2)ccc(Cl)c(C)c1 30415,O(C1CCCc2ccccc21)CC(=O)NC1CCN(C(c2cnc(C)o2)=O)C1C 30416,c1(C(=O)NC2CN(C(c3c(NC)cccc3)=O)CC2C)cc(N)ccc1F 30417,C1(C(=O)NCC2(O)CN(C(C3C=CC=CC=C3)=O)C2)CC2CCC(C1)S2 30418,N1(C(c2ccc(CNC(C(CC)COC)=O)cn2)=O)CC(O)CC1(C)C 30419,c1(C(=O)NCC(N(C(CC(CCC)C)=O)C)C2CC2)cnc2scc(C)n2c1=O 30420,N1(C(COCC)=O)CC(OC)CC(NC(c2ccc(CC(C)C)cc2)=O)C1 30421,C(C(C(=O)NCCc1cn[nH]c1)C(C)C)NC(C1CC(CCC)C1)=O 30422,C(N=c1cc(C(C)C)nc[nH]1)C1CN(C(C(C=C)O)=O)C(C)C1 30423,c1(C(=O)NC(C2N(C(C(C)c3cncs3)=O)CCC2)C)n[nH]c2ccc(Cl)cc12 30424,Cc1cnnc(O)c1C(=O)N(CCCCCNC(=O)CC(C)NC(N)=O)C 30425,C(=O)(CCS(=O)(=O)c1ccccc1)NC1C(C)CN(C(=O)Cc2cc[nH]c2)CC1 30426,C(=O)(C1=NOC2(CCC2)C1)N1CC(=C(CNC(=O)C2=CCCCC2)F)C1 30427,C1(OC)CN(C(c2ncc[nH]c2=O)=O)CC1NC(=O)Cc1sc(S)nc1C 30428,CC1(C)CCC(C(=O)NCC2(C)CCCN(C(c3ncoc3C(F)F)=O)C2)OC1 30429,c1(C(=O)NCC2CCC(NC(=O)COCC3CCC3)C2)ncccc1Cl 30430,c1(OCC(=O)NCC2CCN(C(C(CSC)C)=O)C2)cccc([N+](=O)[O-])c1 30431,Cc1cc(C(N2CCCC(CC(=O)NC3CN(C)CCC3O)CC2)=O)cnc1O 30432,Cn1c(O)nc2cccc(C(=O)NCC(C)(CO)NC(C3CCCO3)=O)c12 30433,c1(NCCN2C(=O)CCCC2)nccc(=NCc2ccc(Br)cn2)[nH]1 30434,C12(C(=O)NCC3(F)CC(CNC(c4ccc(C)s4)=O)C3)CCOC1CS(=O)(=O)C2 30435,c1(CC(N2CCC(C(C3(CC4CC4)CCCC3)C)C2)=O)c(F)cccc1Cl 30436,c1(OC)ccc(C2CCCN2C(=O)C=CCCc2ccccc2)c(F)c1F 30437,C(=O)(C(F)C(C)CNC(c1ccsc1CC)=O)N(CC(COCC)O)C 30438,c1(C(N(C2CC(C(=O)NC3CC3(F)F)C2)C)=O)ccccc1S(C)(=O)=O 30439,C=CCC(C(=O)NC(C)CC(C)NC(c1cnn(C)c1OC)=O)C(C)C 30440,c1(OC)ccc(C(N2CCC(CNC(c3ccc(CO)o3)=O)C(C)C2)=O)c(F)n1 30441,C1(NC(CCOCCN(C)C)=O)CC12CCN(C(c1csc3cncn13)=O)CC2 30442,c1(CC(=O)N(CCC(C)SC(F)(F)F)CC)c(C)n[nH]c1C.C12CC(C1)NC2=O 30443,C1(C(N(C(C=C)C2CC2)C)=O)CCC(C)(C)N(C(=O)C(CCC)NC(C)=O)C1 30444,c1(C(N(C2CN(C(=O)COCC3CCCO3)CCC2F)C)=O)cc2cnn(C)c2s1 30445,N1(C(c2cc(C(C)C)on2)=O)CCC(C)N(C(c2ccc3sncc3c2)=O)CC1 30446,N12CCCC(C1)C(=O)NCC2=O.C1(NC(C(C)SC)=O)CCC(O)C1 30447,CCCCCCN(C(c1sccc1Cl)C(=O)NCC1CC1)C1CC1 30448,Cc1ccc(CC(=O)N(CCCNC(c2coc(C)c2)=O)C2CC2)c(C)c1 30449,N1(C(c2c(C)c(Br)cnc2)=O)CCCN(C(=O)C(C)NC=O)CC1C 30450,Cc1noc(C)c1NC(C1CCCC1CNC(C1(N(C)C)CCC1)=O)=O 30451,n1(CC(=O)NC(C2(CNC(c3c(C)ccnn3)=O)CC2)C)cnc2ccccc12 30452,CC1=C(C(=O)NCC2CCC(C)N(C(=O)CCOc3ccc(O)cc3)C2)CCO1 30453,c12cc(nn1C)C(C(=O)OC)N(C)CC2(C)C.C1(CC2COC2)CCOCC1 30454,c1(CCC(=O)N(CC(=O)NCC2CNC(=O)C2)CCOC)cnn(C)c1 30455,n1(C(C)C)cnnc1CC(N1CCCC1CCNC(=O)CN1CC2CC2C1)=O 30456,C1(NC(Cc2cnc(C)s2)=O)CC2CC1CN(C(C1(O)CC1)=O)C2 30457,C1(CNC(C2(CC=C)CC2)=O)CCN(C(=O)CSc2cccc(C)c2)C12CCC2 30458,C1(C(N(CCCCC)CC(N)=O)=O)CC12CCc1cc(Br)ccc12 30459,CCC(=O)CCC(=O)NC(C)C(C)NC(c1cocc1C(N)=O)=O 30460,N1(C(COCCC)=O)CC(C2CC2)(C(=O)NCc2csc(C)c2C)C1 30461,C1(NC(c2ncc(F)cn2)=O)CCC2(CCN(C(C3CCOCC3)=O)C2)C1 30462,c1(C(=O)OCC)cncc(NC(=O)C(=O)NCCCCSC)c1 30463,N1(C(CCN2C(C)CCCC2)=O)CCc2ccccc2C1CNC(=O)CNC=O 30464,c1(C(=O)NC2C=CC(CNC(CCCC)=O)C2)ccc(OC(C)C)c(N)c1 30465,C1(NC(C2CCN(C)C2)=O)CCC12CN(C(=O)C=CCF)C2 30466,N1(C(C(CCC)NC(C)=O)=O)CC2CCC(NC(=O)CSC(F)(F)F)C2C1 30467,Cc1snnc1C(=O)NCC(C)NC(=O)CC1(Oc2ccccc2)CC1 30468,N1(C(C(CC(=C)C)NC(c2nccnc2C)=O)=O)Cc2nncn2C(C)C1 30469,N1(C(CCC(=O)NC)=O)CC(NC(C2(C(F)F)CCCCC2)=O)CCC1C 30470,Cc1cccc(C)c1OCC(=O)NCC(C1CCC1)NC(c1nocc1Br)=O 30471,CCC(F)(F)C(=O)N1CCC(C(C)CNC(=O)CCC2CC(F)(F)C2)CC1 30472,N1(C(C(=O)NCCC)C(N2CCC(C)CC2CC)C)CCOC2(CCSC2)CC1 30473,N1(C(C2CCCN(C(c3cc(C)c(O)nn3)=O)CC2)=O)CC2CCC1C(CO)C2 30474,S(=O)(=O)(c1ccc(NC(c2ccccc2)C(C)OC)nc1)N(CCC=C)C 30475,N1(C(c2c(OC)csc2)=O)CC(CNC(C2CN(C3CCCCC3)C2)=O)C(O)C1 30476,c1(C(=O)NCCN(C(c2c(CCC)nns2)=O)C(C)C)cccc2ccncc12 30477,c1(C(=O)NCC(N2C(CSC)CCCC2)(C)C)cc(C)n(CC2CC2)c1C 30478,C(=O)(C#CC1CCOCC1)N1CC(CCCCNC(c2n(CC)c(O)nc2)=O)C1 30479,C(=O)(CCC(=O)C(C)(C)C)N1CCC(C)C1CNC(=O)C(c1ccccn1)O 30480,N1(C(c2csc(CNC(=O)C(c3cccnc3)O)c2)=O)CCN2C(=O)CCC2C1 30481,CC(C)C(C)C(CNC(c1cc(N)ccc1F)=O)NC(c1cnn(C2CC2)c1)=O 30482,C(=O)(C(C)(F)C(F)(F)F)NC(C1CCN(C(C2(C(=O)OC)CC2)=O)CC1)C 30483,S(=O)(=O)(c1cccc(C(=O)NC23CC(NC(=O)Cc4conc4C)(C2)C3)c1)NC 30484,Cc1cc(CCNC(=O)CN(C(=O)CC2CC(C)C2)C(C)C)nn1C 30485,C(=O)(C1CCCn2nccc21)N1CCC(C(C)NC(CCCC(=O)OC)=O)CC1 30486,C(CNC(c1ccc(C#N)s1)=O)(C(C)(C)C)NC(c1cnc(COC)s1)=O 30487,N1(C(C(C(C)(C)C)O)=O)CC2(C(=O)NCCCn3ccnc3)CCC1CC2 30488,C12C3CCN(CC13)C2=O.C1(CC(=O)N(CCCC=O)C)CC2C(C1)C2(C)C 30489,c1(C(C)(F)F)cccc(C(=O)NCC(C2CC2)NC(=O)Cc2ccccc2Cl)c1 30490,C1(NC(c2n[nH]c(C)c2C)=O)CC2CC(NC(=O)CCn3cnnn3)CC2C1 30491,Cc1nc(C(C)C)ccc1C(=O)N(C)CC1(O)CN(C(=O)COc2ccon2)C1 30492,c1(C(N(C)CC2CCCN2C(c2cc3occc3s2)=O)=O)c(F)ccc(N)c1F 30493,CCC(F)(F)CC(=O)NC1CC(C(=O)NC2CNC(=O)C2)C1 30494,N1(CCCNC(C2C(C)=C2)=O)CCN(C(=O)C(C)Cc2cccc(F)c2)CC1 30495,c1(CNC(C2(COC)CC2)=O)cc(C)c(C(=O)NCCN2CCCNC2=O)o1 30496,N1(C(COCC=C)=O)CCC(N(C(=O)C(F)(F)c2cscn2)CC)CC1 30497,C1(F)(CNC(C=C(C)C(F)F)=O)COCCN(C(=O)CC2CCOC2)C1 30498,S(=O)(=O)(c1cccnc1)NCCC(=O)NCC(C1CCCC1)NC(=O)C1=CCC1 30499,Cc1cncc(NC(c2ccc(O)nc2)(C)C)c1 30500,C(=O)(CCCCN(C(=O)C(C)(C)C1(O)CCC1)C)NCC(C)CCO 30501,S(=O)(=O)(c1ccc(=NCCC(F)(F)Cl)[nH]c1)N(CC#CCC)C 30502,c1(C(C(=O)NC)N(C2CCCN(C(C3CCCC34CC4)=O)C2)C)ccc(C)cc1C 30503,CC(C)C(C(=O)N1CCC(C(=O)NCCCCCN(C)C)CC1)NC(N)=O 30504,C1(NC(C2CCCN(C(C(N3CCNC3=O)C)=O)C2)=O)CC2(C1)CC(O)C2 30505,c1(OC)nccc(C(=O)NC2CCC2CNC(=O)CC2COCCN2C)c1F 30506,N1(C(C(=O)N(C)CCC(=O)OC)C)CCC2CCC12C.CC1CCCCN1CC 30507,c1(NC(COC2CN(C(COCCOCC#C)=O)C2)=O)c(F)ccc2nc[nH]c12 30508,C(=O)(C(CCC(N)=O)n1cc(-c2cncc(Cl)c2C)nn1)N(C(CCCC)C)C 30509,N1(C(c2nc(CS(C)(=O)=O)oc2)=O)CCN(C(c2cncc(O)c2)=O)C2(CC2)C1 30510,c1(C(=O)OC(C)=O)ccc(C=CC(N2CCCC(c3nnc(CC)n3C)C2)=O)o1 30511,Cc1c(C(=O)NC2C=CCCC2C(=O)NCCNC(C2CCCC2)=O)nnn1C 30512,c1(C(=O)NCC(C)(C(C)C)NC(CCc2cc(C)[nH]n2)=O)cc(Cl)c(F)cc1N 30513,CCCCC(=O)C(=O)NCCC1CN(C(C2CC23CCOCC3)=O)CC1C 30514,c1(CC(=O)NC(c2ccccc2)C(C)NC(C2SCCS2)=O)nnc(O)s1 30515,c1(-c2ccc(SC)cc2)ccc2[nH]cc(CC(=O)NCCc3cccs3)c2c1 30516,C1(NC(C(=O)N(CC(N)=O)C)=O)CCN(c2ncccn2)C1 30517,C=CC1(C(=O)N(C)Cc2cncs2)CCN(C(c2ccn(C)c2)=O)C1 30518,c1(C(=O)NCC2(NC(CC(CC)C3CC3)=O)CCOCC2)ccc(N)cc1Cl 30519,N1(C(C2CC(C3CCC3)C2)=O)CC(NC(c2ccccc2CC#N)=O)C(F)C1 30520,O(NC(=O)C(CCF)NC(c1ccco1)=O)CCCC(=O)OC 30521,c1(C(=O)NC2CCN(C(Cc3nc(C)oc3)=O)CC2)ccc2nncn2c1 30522,Cc1nc(C)c(C(=O)NC(C2CCN(C(c3cc(C(F)(F)F)no3)=O)CC2)C)[nH]1 30523,N1(C(C(CC)C)=O)CCCN(C(c2ccc(Cl)cc2)(c2ccccc2)OC)CC1C 30524,c1(-n2cc(CSCCNC(C(CC)NC(C)=O)=O)nn2)cc(F)c(F)c(F)c1 30525,c1(C(N(C2CCC(NC(c3cc(=O)cc[nH]3)=O)C2)C)=O)ccc(CO)nc1 30526,C(=O)(CC(C)P(C)(C)=O)NC12CC(NC(C(c3c(OC)ccc(F)c3)=O)=O)(C1)C2 30527,C1(C(=O)NCC(C)N(C(=O)C(=O)NCC2CC2)C)CC2CSCC(C1)C2 30528,C1(N(C(c2cnns2)=O)CCO)CN(C(=O)CC2OCCO2)C2(CCC2)C1 30529,C(C(C)(CO)NC(=O)CCCSC(F)(F)F)NC(C1C(COC)C1)=O 30530,C1(C(N(CCC(C(C)C)NC(=O)C(C)c2ccco2)C)=O)CN2CCCN1CC2 30531,Cc1cc(C(=O)NC2CCOC(CNC(=O)C3=CCC3)C2)n(-c2ccccc2)n1 30532,C#Cc1ccc(C(=O)NC2CC(NC(c3c(OC)ccc(F)c3F)=O)C2)c(C)c1 30533,Cc1c(-c2nc(-c3cccnc3O)nn2CC2CCOC2)cnn1CC(C)C 30534,C12(CNC(=O)CC3CC3(Cl)Cl)CC3CC(CC(NC(=O)C(O)C(F)(F)F)(C3)C1)C2 30535,N1(C(C(CC)(CC)OC)=O)CCN(C(C2CCCCN2C)=O)C2(CC2)C1 30536,CC1CN(C(C2CCC3(CCC3)C2)=O)CCCN1C(=O)CCc1cn(C)nn1 30537,C12(C(=O)NC(C)CCNC(=O)C=Cc3cnc[nH]3)CC1CCC2(F)F 30538,n1(CCS(CC)(=O)=O)c(=NCCc2nc(C3CC3)n[nH]2)[nH]c2cc(Cl)ccc12 30539,C1(C(C)C)CCN(C(=O)C(C2CC2)N(C(=O)CCc2ccnn2C)C2CC2)CC1 30540,N1(CCCC(N2CCC(C)(C)CC2)=O)C(=O)C2CC=CCC2C1=O 30541,CON=CC(=O)NCCC1(NC(=O)C(C)N(C(C2CCCC2)=O)C(C)C)CC1 30542,C1(N(C(=O)CCCN(C)C)CC)CCN(C(=O)CCOc2cccc(O)c2)CC1 30543,C(C(=O)NCC(C)OC(F)F)(C1CC1)NC(COCCC#C)=O 30544,c1(C(=O)NC2C(NC(c3nnc(C)s3)=O)CCC2)cccc2c1COC2 30545,c1(C(N2CC(CC(C(=O)N(CC#C)CC3CCCO3)F)C2)=O)ncncc1Cl 30546,CC1Cc2ccccc2N1C(C1NCCC1C1CC1)=O 30547,N1(C(C(CC)NC(C)=O)=O)CCN(C(c2n[nH]cc2C)=O)CC1CCO 30548,n1(CC)cc(CC(N2CCCC(CNC(=O)Cc3cc(C)nn3C)C2)=O)c(C)n1 30549,c1(CC(C)CC2CC2)nc(-c2ccc(N(C)C)cc2)nn1CC1CCSC1 30550,c1(OC)ccc2nc(C)c(C(=O)NCC(CNC(=O)C(O)CC(C)C)OC)n2n1 30551,C1(NC(c2c(SCC)cccc2)=O)CN(C(=O)Cc2ncccc2C)CCC1C 30552,c1(C(N2C(CC=C)CCC2)C(=O)NC2CCOCC2)cc(C)cc(OC)n1 30553,Cc1cnc(C(N2CCSCC2CCNC(C2CCCCS2)=O)=O)cc1C 30554,Cc1ncc(C(N2CC(O)CC2CNC(C2(C)CCCN(C)C2)=O)=O)c(=N)[nH]1 30555,c1(-c2cn(CCSC3C(CC)CC3)nn2)cccc(N)c1 30556,N1(C(Cc2nc(C)[nH]n2)=O)CCCC12CCN(C(=O)CCc1nncn1C)CC2 30557,C(=O)(CC(CCC)NC(=O)CC1CCCC(=O)N1)Nc1cc(OCC)n[nH]1 30558,C1(C)(CN2CCN(C3CCN(C(C(C)n4cncn4)=O)C3)CC2)NC(=O)NC1=O 30559,C1(NC(=O)NC2CNCC2O)CCOC2(CCCC2)C1 30560,N1(C(c2ccn(COC)n2)=O)CCC=C(C(=O)N2CC3CCC2C3)C1 30561,n1(CCC)ncc(CN(C(=O)CN2CC(CC(C)(C)C)C2)C2CC2)c1C 30562,c1(C(N2CCCCC(NC(C(CCC)C#N)=O)C2)=O)noc2ncccc12 30563,c1(C(N2C(C)C(NC(c3cc[nH]n3)=O)CC2)=O)cc2c[nH]cnc-2n1 30564,C(=O)(CCC(=O)N1CC(NC(=O)CC(O)CN(C)C)CC1C)N(C(C)C)C 30565,C1(OC)C=CCN(C(c2ccc(OC(F)F)nn2)=O)C1 30566,c1(CC(=O)NC23C(CN(C(c4cncc(C)c4)=O)C2)C3)cccc(F)c1F 30567,C1(N(C)C)(C(=O)NCCCCCn2cc(-c3cc(C#N)cs3)nn2)CCCCC1 30568,c1(CCOC)ccc(Cl)c(S(=O)(=O)N2C3CCCC2CC(O)C3)c1 30569,C1(C(N)=O)C2CC3CC(C2)CC1(C(=O)ONC1CCCc2c[nH]nc21)C3 30570,C1(OC)(CNC(C2(C)CCCCCC2)=O)CCN(C(c2[nH]c(O)nc2C)=O)CC1 30571,CC1(C#CC(=O)N2CCC3C(NC(=O)CSCC(F)(F)F)C3C2)COC1 30572,C1(NC)CCCC2CN(C(c3ccc(C)o3)C(=O)NCCc3ccccc3)CC12 30573,C1(N(C)C(c2ccnc(S)c2)=O)CCCCN(C(=O)Cc2c(O)ncnc2O)C1 30574,C(C)(C(CC(=O)N(C1CC1)CC1CCOC1)NC(=O)C1=COCCC1)OC 30575,C(C)(C)(CC(=O)N1CC(C)(C(=O)NCCCc2ccncc2)C1)OC 30576,c1(-c2nc(C3COCC3c3nc(C4CSCCS4)no3)on2)cccc(Cl)c1.OC 30577,c1(C(=O)NC2C3CN(C(Cc4cccc(C#C)c4)=O)CC32)ccc(F)c(C#N)c1 30578,c1(C(=O)NC(C2Cc3cc(Br)ccc3O2)C2CCCO2)ccc2c(n1)OCCO2 30579,C#Cc1cn(C)nc1C(=O)NC1CCCC(C(=O)NCc2ccns2)C1 30580,C1(CC=C)(NC2CCCCC2C(F)(F)F)CCCNC1 30581,C(=O)(CCCS(C)(=O)=O)NCC1(C(F)F)CCN(C(C(n2c(C)ccn2)C)=O)C1 30582,CCC(O)(C(=O)NCC1CC2CC2N1C(C1OCCO1)=O)c1ccccc1 30583,C1(NC(c2occc2Br)=O)CCC2CN(C(C3=C4C(CN=C3)C=CC=N4)=O)CC2C1 30584,CC1CCCCN1CC(N1CCC(CCC(=O)NCCC(O)C2CCC2)CC1)=O 30585,C1(CCCC)CCC(NC(=O)Nc2c[nH]nc2-c2ccccc2Cl)CC1 30586,c1(N(C(C)C(C)=O)Cc2ccc(OC)cc2)nc(O)c2c(C)c(C)sc2n1 30587,N1(C(C(C)OCCOC)=O)CCC(N(C(C2CCC2C)=O)CC2CC2)C1 30588,c1(C(N2CC3(CNC(C)=O)C(C(F)(F)F)(C2)C3)=O)cc(C)c2nc(C)cn2c1 30589,c1(NC(=O)OC(c2c(Cl)cc(C)s2)=O)cnc(C2CCCC2)[nH]c1=N 30590,c1(C(C)O)ccc(NCc2ccc(NC(c3cccc(I)n3)=O)nc2)cc1 30591,N1(C(Cc2ccc(C)cc2)=O)CC2CC(NC(=O)CC3CCOCC3)CC1C2 30592,N1(CC)CCN(C(=O)CC2CCN(C(=O)C(n3ccnc3C)C)CC2)CC1 30593,C12(NC(c3cccc(C)c3)=O)CC(CNc3ncnc(C)c3Br)(C1)OC2(C)C 30594,C1(C(=O)NC2CCN(CCOC)C2)CCC(CNC(C2CCOC2C)=O)CC1 30595,C1(OC)(OC)CC(C)(C(=O)N(CC(O)CNC(=O)CC2C(C)(C)C2(C)C)C)C1 30596,c1(C(=O)NC2(C3N(C(c4nncc(OC)c4)=O)CCC3)CC2)c(Cl)cccc1Cl 30597,c1(SC)cc(C(=O)NCC2(O)CN(C(=O)CC(c3ccccc3F)C)C2)c(C)o1 30598,c1(CCCC(=O)N(C2CCN(C(CC=C(C)C)=O)C2)C)ccccc1Cl 30599,CCC(CC(C)C)C(=O)N1CCC(CO)C(NC(=O)CC2CCCC(C)C2)C1 30600,c1(C(N2CC3C(CNC(C(CCN(C)C)O)=O)(C3)C2)=O)c(Cl)cncc1Cl 30601,Cc1cc(CC(=O)N)ccc1O.N1(CC=O)CCN(c2ncc(F)cn2)CC1 30602,N1(C(C(CCCC)O)=O)CC(CNC(=O)C(=C2CCCCC2)F)OC2(CCC2)C1 30603,N1(C(C=C2CCC(C)C2)=O)CCC(O)(CCNC(=O)CN2CCNC(=O)C2)C1 30604,c1(NC2CCN(CC=C)CC2)ncc(S(=O)(=O)N2CCCC(C)C2)cc1Cl 30605,CCC(CCOC)C(=O)NCC1CCC1NC(c1nccc(OC)c1O)=O 30606,C1(C(=O)NCc2c(C)nco2)C2CC2CN1C(=O)CC1COCCO1 30607,CN1CCCCC1C(N1CCC(CC(=O)NCCc2cscn2)CC1)=O 30608,Cc1cc(C(=O)NCCC2(NC(=O)CC3CCCO3)CCC2)cc2nc[nH]c12 30609,c1(CC(=O)NCC2COCC2NC(C2CCCCS2)=O)cccnc1Cl 30610,Cc1cc(Cl)cc(C)c1C=CC(N1CCC(CNC(=O)C(O)C(C)C)C1)=O 30611,c1(NCC(C)S(N)(=O)=O)ncccc1S(=O)(=O)NC(CC(N)=O)C1CC1 30612,c12nnc(n1CC1CC1)N1CCCC1CC2.OCC(F)CCCC1CC1 30613,Cc1ccc(C(N2CC3(CCN(C(c4ncsc4C)=O)C3)C2)=O)cc1C#N 30614,CN1CCCC(CNC(C2CSCCN2C(c2ccc(C#N)cn2)=O)=O)C1=O 30615,c1(C(N2CCN(c3ncnc(CC)c3F)CC2)=O)cc2ccc(C)cc2o1 30616,C1(C)(C(N2CCCC2COC)C(=O)NCCCC)CCN(C(=O)NC(C)C)CC1 30617,C1(C(N2CCC(N3CCN(C(c4cscc4Cl)=O)CC3)C2)=O)CCCCC1(F)F 30618,C(=O)(C(C)CC(F)F)NCC1CC(CNC(c2ccn(CCCC)n2)=O)C1 30619,CCC(C)C(=O)OC(C(=O)NC1CC2CC2C1)C1CC(OC)C1 30620,c1(-c2cccc(C(C)NCC3CC3)c2)ccc(S(=O)(=O)N(C)C)cc1 30621,C12CCCN(C1)N(C)C2=O.n1(CC)ccnc1CNc1ncc(C(=O)O)o1 30622,C(=O)(N=c1ccn(CCN(C)C)[nH]1)c1cncc(NC(CC(C)CN(C)C)=O)c1 30623,C(=O)(C(C)=NOCC#N)N1CC(OCCNC(CCCCCCC)=O)C1 30624,CCC1=C(C(=O)NCC2CCN2C(C2CCc3n[nH]c(C)c3C2)=O)CCCO1 30625,C1(NC(c2c(C)cccn2)=O)C2COCC1CC(NC(=O)C1=NOC(C)C1)C2 30626,N1(C(COCCC)=O)CC(C2CN(C(C3CCCC(N(C)C)C3)=O)C2)C1 30627,C1(COC)(NC(=O)C(F)CC2CCCC2)CN(C(=O)Cn2cc(Cl)cn2)C1 30628,CCC(CCC(=O)NCCSCC(=O)NC(c1n[nH]c(C2CC2)n1)C)OC 30629,Cc1c(O)ccc(C(=O)NCCCCN(CCCNC(=O)CCC(C)C)C)c1C 30630,C1(C)(C(=O)NC2CC(CNC(C(C)OC3CCCC3)=O)C2)CCC(F)(F)CC1 30631,c1(C(=O)NC(CCCCNC(C2(C)ON=C(C)C2)=O)C)c(C)nc(O)nc1C 30632,c1(OC)cc(CN2CC3(CC(C(=O)Nc4cn(C)cn4)C3)C2)cc(F)c1 30633,C(CCCCCC(=O)NC1(CC2CCCC2(C)O)CC1)n1cc(C(CC)(C)O)nn1 30634,C(CC(=O)NCC1C(C)CCN1C(=O)CSCCN(C)C)(C(F)(F)F)OC 30635,CCCC(CNC(c1nc(C(C)(C)C)no1)(C)C)C(=O)O 30636,O=C(CC1=CCOCC1)N1CCC(C2CCCN2C(c2cnn(CCO)c2)=O)C1 30637,N1(C(C2C(C)CCC2)=O)CC2(CC2)CC1CNC(=O)Cn1cncn1 30638,CC1(C(=O)NCCOCCNC(C2CCCCNC2=O)=O)CCCNC1=O 30639,C1(CNC(CC(C)n2cccc2)=O)C2CN(C(=O)CCc3nc(=N)[nH][nH]3)CC12 30640,C(=O)(CCCCCCCC=C)NCC(C)N(C(COCCC#C)=O)C 30641,c1(CC)cc(C(N2CC(F)(c3cccnc3)C2)=O)no1 30642,C(=O)(C1=NNC(C(F)(F)F)C1)N1CC(C)(NC(C(C(C)O)C)=O)C1 30643,c1(CC)ccc2c(CC(=O)NC3(CNC(=O)C4CC4)CCCCC3C)coc2c1 30644,C(=O)(C1c2ccccc2CN1C(c1cnc(O)c(Cl)c1)=O)NC1CC(=O)NC1=O 30645,Cc1nc(C(N2CCC(CC(N3CCC(C(C)(C)O)C3)=O)C2)=O)c(C)s1 30646,C1(C(=O)NCCC)CCN(C(=O)C#N)CCC1C(=O)OC 30647,c1(C(N(CCC(C)NC(CCc2onc(CSC)n2)=O)C)=O)cnnc(C)c1C 30648,c1(C(=O)NC(CN(C(CC(CC)CC)=O)CC)C)ccc(F)c2ccoc12 30649,CCCC(CCCNC(=O)CCc1ccc(C(C)(C)C)cc1)SC(C)CC(N)=O 30650,C1(CC=C)(NC(c2coc(O)n2)=O)CCCN(C(=O)CC2CCC(C)(C)CC2)C1 30651,C(=O)(CCC(CF)CF)Nc1cccc(C(=O)Nc2ccc(OC)nc2C)c1 30652,N1(C(C(N2CCCC(C)C2)=O)=O)CCC(CO)C(NC(=O)C(C)C2CC2)C1 30653,N1(C(C(C(C)C)SCC)=O)CC(NC(c2cnnn2C(C)C)=O)CC1(C)C 30654,c1(C(N2CC(C)(C)C(NC(=O)C(F)=CCCF)C2)=O)cc(F)c(O)c(F)c1 30655,c1(C(=O)NCC(C)CNC(c2ccnc3ccnn23)=O)cc2c(s1)CCCCC2 30656,c1(C(=O)NCC2OCC(CNC(Cc3cn(C)nc3)=O)C2)ccnc2ncnn12 30657,C(CC(F)F)(C(=O)NC1CC2(CCCC2)C1)N(C(c1c(CC)con1)=O)C 30658,c1(C(=O)NC2CN(C(c3cccc(CCC)n3)=O)CC2SC)[nH]nc2cnccc12 30659,c1(OC)cccc(C(N2CCCC(F)(F)C2)C(=O)Nc2ccccc2Cl)c1C 30660,c1(N(C(CC)C)CC(=O)OC(C)(C)C)ncc(Br)cc1[N+](=O)[O-] 30661,C1(C)(C(=O)NCC)CCCN(Cc2c(CC)cccc2C)C1 30662,CC1(C2CC2C(=O)NC2CC(CC(=O)Nc3cncc(C(N)=O)c3)C2)COC1 30663,NS(=O)(=O)N1CCCC(C(=O)NC2(C3CN(C(=O)CCC(N)=O)C3)CC2)C1 30664,NS(=O)(=O)c1ccc(O)c(C(=O)NC2CC(NC(c3nn[nH]c3Cl)=O)C2)c1 30665,C1(NC(C(C)NC(=O)NC)=O)CN(c2nccc(C#N)n2)C2CCCCC12 30666,C1(CNC(c2ccc(OC)nn2)=O)CC2(CC2)CN1C(=O)Cc1cccc(C)c1 30667,C1(C(=O)NC(C(=O)OCC)C)CCN(C(=O)CCCC#N)C1CC 30668,C(c1cccc(Cc2n[nH]cc2C(N2CCC(C3CCCN3CC)C2)=O)c1)=CC 30669,S(=O)(=O)(c1cnccc1N1Cc2cnn(N(C)C)c2C1)NCC1(CC(C)C)CC1 30670,CC1(C)CC=C(C(=O)N2CC3CCCN(C(c4ncc[nH]c4=O)=O)C3C2)CC1 30671,C(CC(C)(C)C(=O)N1CCC(CN(C(=O)COCCc2ccccc2)C)C1)OC 30672,CCC(C(=O)N(C1(C(N2CCC3CCC23)=O)CCC1)C1CC1)C(F)(F)F 30673,N1(CCCNC(C(CC)C)=O)CCN(C(=O)CN2CCC(C)(O)C2)CC1 30674,Cc1[nH]c2ncnc(N3CCC(C)(NC(=O)CC4COC5CC4C5)C3)c2c1C 30675,C1(C)(C(C)(C)C)CCCN(C(C2CCCN2C(=O)CC2CCNC2=O)=O)C1 30676,N(C(=NCCSC1CC1)NCC(=O)OC1CCCC1)C(c1cnccn1)C 30677,C(=O)(CS(=O)(=O)C1CCCC1)NC(C)Cc1cc2ccccc2o1 30678,c1(C(N2CCOC(CCNC(C3CC(C(F)F)C3)=O)C2)=O)ccc2nnnn2c1 30679,C1(NC(C=CCCC)=O)CN(C(=O)C(c2cccc(C)c2)(C)C)CC1O 30680,C1(C(=O)NC(c2onc(C)n2)C)CC(NC(=O)OC(C)(C)C)C(O)C1 30681,C=CC1(CO)CCN(C(=O)C(C)(CSC)NC(=O)COc2cccnc2)CC1 30682,Cn1cc(CC(O)C(=O)NCCCN(CCCNC(=O)C=Cc2cnc[nH]2)C)cn1 30683,C1(NC(=O)CCN2CCCC2)CC12CC(NC(C1CC13CC3)=O)C2 30684,c1(C(=O)NC(C2CCN(C(=O)C(F)=C3CCC3)CC2)C)ccc(N)cc1[N+](=O)[O-] 30685,c1(C(=O)NC2C3(NC(CCSCC)=O)CCC(C2)C3)cccc2c1NCCC2 30686,C(=O)(N=c1nc2ncc(Br)cn2[nH]1)NCc1ccc(NC(C)C)cc1 30687,n1(CC)nc(C)c(CC(N2CCCCC2C(C)NC(=O)CC2=CCCC2)=O)c1C 30688,N1(CCCC=C)CCC2C(CCCN2C(=O)C(c2cnn(C)c2)C)C1 30689,Cn1c(=O)oc2c(-n3cc(CCCNc4n[nH]c(=N)s4)nn3)cccc12 30690,O(NC(=O)C(Cc1cc[nH]n1)NC(c1nonc1CC)=O)CCCC 30691,N1(C(CC2(C=C)CCC2)=O)CC(NC(=O)C(C)NS(C)(=O)=O)CC(C)(C)C1 30692,N1(C(C(C)NC(C)=O)=O)CC2(CCN(C(=O)C(F)=C(C)C)CC2)CC1C 30693,c1(C(=O)NCC=C2CCN(C(c3cc(CC)ncn3)=O)CC2)ccn2cncc2c1 30694,N12CCC(CC1)C(C)(C)SCC2=O.C(=O)(C(C)Cc1ccnn1C)NCC#C 30695,c1(OC)cccc(F)c1C(N1CCCC(CN(C(=O)COC2(C)CCC2)C)C1)=O 30696,N1(C(CCOC(C)=O)=O)CCC(O)(CCNC(C2CCN(CC(C)C)CC2)=O)C1 30697,C1(NC(=O)CN2CC3CC3C2)COC2CN(C(=O)CCSC3CCCC3)CC12 30698,N1(C(c2ccn(CCOCC)n2)=O)CCCN(C(C2CCCN2C)=O)CCC1 30699,N1(C(CC(C)n2ccnc2)=O)CCC2(CC1)CC2NC(C1(C(F)F)CC1)=O 30700,c1(C(N2CC(O)(CNC(C3(C)C(CC)CCC3)=O)C2)=O)ccc2oc(=N)[nH]c2c1 30701,C12(NC(Cc3cc(CC)no3)=O)CCCCCC1N(C(c1nnsc1N)=O)CC2 30702,CC#CCCC(=O)N1CC(n2cc(CNS(C)(=O)=O)nn2)CO1 30703,N1(C(c2c(C)ccs2)=O)CC2(CCC2)CC1CNC(=O)CCOC1CCOC1 30704,n1(CC=C)nnnc1C(c1csnc1OC)NCCn1cccn1 30705,CCCCCCC(=O)NC1C=CC(C(N2CCC3CC2C3)=O)C1 30706,c1(-c2ccccn2)cc(-c2noc(C3CCC(F)C3)n2)ncn1 30707,C(=O)(CCS(N)(=O)=O)NC(CNC(CCC(C)SC)=O)(C)C(C)C 30708,c1(CN(C(c2cc(C)no2)C(=O)NC(CC)(C)C)C(C)C)ccccc1Cl 30709,C(C(=O)NC(C)(C)CCNC(c1nc[nH]c1C(C)(C)C)=O)(C(C)C)SC 30710,C1(CC(N2CCC(NC(=O)CCN3C(=O)CCC3=O)C2)=O)COc2ccccc2O1 30711,C1(C(C#C)NC(=O)N(CCCN(C)C)C)CC(F)(F)C1 30712,S(=O)(=O)(c1cc(F)ccc1F)NCc1ccc(-c2c(OC)nc(Cl)s2)cc1.C1(C)CC1 30713,C1(CNC(c2cn(CCC)nn2)=O)CCCCC1NC(c1ccoc1Br)=O 30714,c1(CN2CC3C(C(=O)NCCc4ccc(Br)cc4O)C3C2)cc2ccccc2o1 30715,Cc1ccn(C)c1C(=O)N(CC(C)N(C)C(C1CCN(CC(F)(F)F)C1)=O)C 30716,N1(C(=O)C(c2cc(F)ccc2OC(F)F)=O)CCCS(=O)(=O)CC1C1C(=O)CCC1 30717,C1(=O)C(O)C(C(C)C)NC2C(CC)CCN12.C(C(C)(CO)CC=C)OC 30718,c1(C(N2CCC(NC(CCN(CC)CC)=O)C2C2CC2)=O)cc(Cl)c(F)c(Cl)c1 30719,c1(OC)ccc2c(c1)C(C(=O)NC(c1ccc(C)cn1)C)CC2.C12CC1C(=O)N2 30720,C1(C(=O)NCC2(C)CCN(C(C3(C)C(C)C3)=O)C2)CCC12CCOCC2 30721,N1(C(c2cn(CCCOC)nc2)=O)CC(NC(c2ccoc2Br)=O)C(O)C1 30722,c1(C(N2C(C)C(NC(C3C(C)(C)C3(F)F)=O)CCC2)=O)cc2c(cc1O)OCO2 30723,N1(C(C=C(C)c2cccs2)=O)CC2CC(NC(c3cc(N)ccc3C)=O)C(C2)C1 30724,c1(C(N2CCCC(C(C(=O)NCC(CCSC)O)C)C2)=O)ccn2nccc2c1 30725,c1(C(=O)NCCCCCCNC(C2N(CC)CCC2)=O)c(C)ccc(C)c1F 30726,C1(C(=O)NC(C2CC2C(N2CCC3CC23)=O)C)CC=CC(O)C1 30727,C12(CNC(c3cc(C(F)F)ccc3Cl)=O)CCC(CC1)CN2C(=O)C(F)(F)CO 30728,CC1CCN(C(C2(C)CC2(F)F)=O)CCN1c1nccc(C#N)n1 30729,Cc1nn(-c2cccc(F)c2)cc1C(=O)O.C1CCCC(C)N1C(=O)CS(C)(=O)=O 30730,c1(CC(=O)NC2C(C)N(C(=O)C3=CSCCO3)CC2)c[nH]c(=N)nc1O 30731,Cc1cnncc1C(=O)NC1(C)CC(NC(C2CCCSC2)=O)C1 30732,N1(C(C(C)OCCCCCC)=O)CC(NC(c2ccnnc2C)=O)CC(C)(C)C1 30733,N1(C(C(CNC(c2c(C)cns2)=O)(C)C)=O)CC(O)(C2CCC2)C1 30734,C1(CNC(C(COC)(F)F)=O)CC2CCC1N2C(c1cscc1Cl)=O 30735,CCCCCC(O)C(=O)NCC1CN(C(c2cnc(NC)cn2)=O)CC12CCC2 30736,n1(CC)ccc(C(=O)NCCN(C(=O)Cc2nocc2C)CCOCCO)n1 30737,C1(CNC(C(CC)=CCCC)=O)CN(C(=O)COC)CCN1C 30738,N1(C(CC(C)C(F)F)=O)CCOC2(C1)CN(C(C1(c3ccccc3F)CC1)=O)C2 30739,C=CCCC(CO)N(c1cncnc1C)C(=O)CN1CCC(OC(C)=O)C1 30740,c1(COc2c(C(N(C)C3CC3)=O)cc(Cl)cc2)ccc(Cl)c(C#N)c1Cl 30741,n1(C(C)C(N2CCC(F)(CNC(=O)CCNC(N)=O)C2)=O)cc2ccccc2n1 30742,C(c1ccncc1)=CC(N1CCC(CCC(=O)NCc2cc(Cl)no2)CC1)=O 30743,c1(C(=O)NCCn2cc(-c3ccc(CN(C)C)cc3)nn2)c(O)ccc(F)c1F 30744,C1(=O)C(CO)N1.c12[nH]ccc1CNC2=O.C1(C(C(=O)OC)OC)CC(F)(F)C1 30745,C1(n2ccc(C)n2)CCN(C(=NCC2CC3(CCOCC3)CO2)NCC(F)F)C1 30746,C1(C(=O)NCC2(CCC=C)CC2)(NC(C2SCCS2)=O)CC(CO)C1 30747,c1(OC)cc(C)c(Br)cc1C(N1CCC2(CC2C(=O)Nc2cc(O)ncn2)C1)=O 30748,N1(C(CC(COC)NC(=O)CCCF)=O)CCN(C)CC1C(=O)OC 30749,CON(CCC(=O)N(CC(C)CN(C)C)C)C(=O)C1CC2CCC1CC2 30750,C12(NC(C3(CC#C)CCCCC3)=O)CCC1CN(C(c1ccnc(OC)n1)=O)C2 30751,N1(C(C2C(CC)CCC2)=O)CCC(CCOC)(C(=O)N(C2CCC2)C)CC1 30752,c1(-c2ccc(NCC#N)cc2)ccn2nc(C(=O)NCC3(C#N)CC3)cc2c1 30753,C=C1CCN(C(=O)C(C)OCC2CCC2)C(C(=O)NCC2CC(C)(C)C2)C1 30754,Cc1nc2c(s1)CCCC2C(=O)N1CCCC(NC(c2c[nH]c3c2CCC3)=O)C1 30755,c1(CC)oc(C)cc1C(=O)NC(CSC)CCO 30756,c1(C(=O)NCC2N(C(C3(C#C)CC3)=O)CCC2)c[nH]c(=O)c2ccnn12 30757,N1(c2cc(NCC3(C)CN(C)C3)ncn2)CCCC2(CCCCCC2)C1 30758,C(CCC1CCC1)(C(=O)NCc1cnn(C)c1O)NC(c1c(C)ocn1)=O 30759,c1(NC(C)CNC(=O)C(C)CCOc2ccccc2F)ccc2nnnn2n1 30760,c1(C(N2CC(NC(COCC(=C)C)=O)C(C)C2)=O)cc(N)nc(Br)c1 30761,C(C(=O)NNC(=O)NCc1cn(C)nc1-c1ccc(F)cc1)SCCCC 30762,N1(C(c2c(C)nsc2N)=O)CC(C2CN(C(=O)CCC3CCCOC3)C2)C1 30763,N1(C(C2CNC(=O)N2)=O)CCCC2(CCN(C(c3cocc3C(N)=O)=O)C2)C1 30764,C(=O)(C1CCc2cccc(F)c21)NC(C)CN(C(=O)Cn1ccc(=O)cc1C)C 30765,C=CC1(C(=O)OCC23CCC(C2)OC3)CCN(C(C)=O)C1 30766,CCC(C)CCCCC(=O)NCC(CC)NC(=O)Cn1cc(C)cn1 30767,N1(C(c2ccn(CCC)n2)=O)CC2CCC(C1)N2C(c1cnc(SC)s1)=O 30768,c1(C(=O)NC2C=CC(CNC(C(C(C)C)C)=O)C2)nn(C)c(Cl)c1Br 30769,N1(C(C2C(=C)CC2)=O)CC(Oc2cccnc2)CC(N(C(=O)CCOC)CC)C1 30770,C(=O)(C(COC)COC)NC1(CNC(CC2C(CC)C2)=O)CCC1.C(C)(C)O 30771,C(=O)(C(CC(C)C)N1CCCCC1C(=O)NC)Nc1nc(CCC)oc1 30772,C1(C(C(=O)NCC(C)NC(C2(C)COCCO2)=O)=O)CCCCCC1 30773,c1(C(=O)NCC(C2CCCCC2)NC(C(C(C)C)F)=O)csc([N+](=O)[O-])c1 30774,C1(c2cn(C(C(C)O)C)nn2)CCN(C(=O)CCC2CCCOC2)CC1 30775,C(C(=O)N(C)CCF)(C(C)(C)O)NC(C(CC)C#N)=O 30776,N(C(=NCCc1cnc(C)cn1)N1CCC(CS(C)(=O)=O)C1)C(CC)C 30777,C1(CNC(CC(=O)OCC)=O)CN(C(C2CC(F)C2)=O)CC12CCOCC2 30778,N1(CC(=O)NC2CN(C(CC3C(C)=NNC3=O)=O)C2)CCOc2ccccc21 30779,C(=O)(C(C)(CC)C(=O)N1CC(NC(c2cc(OC)ns2)=O)C(C2CC2)C1)OCC 30780,c1(NCC(CCC)C)nccc(=NC(CCOC)c2ccccc2Br)[nH]1 30781,c1(N2CCN(C(c3c(N)cc(F)cn3)=O)CC2)ncc([N+](=O)[O-])cc1Cl 30782,c1(C(N2CC3(CC(CNC(=O)CC(O)C4CC4)C3)C2)=O)cccc2c1SCCC2 30783,N1(C(CNC(=O)OC)=O)CCCC1(CNC(c1ccnn1C(C)(C)C)=O)CC1CC1 30784,c1(OC(CC(=O)OC)c2ccccc2)cc(CO)cc(F)c1 30785,N1(C(C(C)=CC2CC2)=O)CCN(C(c2n[nH]c(C)n2)=O)C2(CCC2)C1 30786,N1(C(CCC(=O)OC)=O)CCc2cc(NS(=O)(=O)c3cc(Br)ccc3Br)ccc2C1 30787,CC1CCC(NC(c2csc(C(F)(F)F)c2)=O)CN1C(c1c[nH]ccc1=N)=O 30788,C1(NCCNC(C(CC)(C)O)=O)CCC(=O)N(CCOC)C1 30789,CC1CN(C(=O)NCCC23COC(C2)C(O)C3)C(C)CC(C)O1 30790,c1(C(=O)NC2(CC=C)CCN(C(=O)C(F)CC3CCOC3)C2)c(C)cccc1F 30791,C(=O)(C1CCCc2nn[nH]c21)N1C(C)CC2CN(C(c3c(C)coc3C)=O)CC21 30792,N1(C(CCCC(C)=O)=O)CC2CCCN(C(=O)CC3(C)OCCO3)C2C1 30793,N1(C(c2c(OC)nsc2)=O)CC(N(C(=O)C(C)OCC(F)(F)F)C)C2(CC2)C1 30794,c1(CC)cc(C(=O)NCCCCCNC(=O)C(C)(C)n2cnc(C)c2)c(C)nn1 30795,C1(NC(C=C(C)C)=O)CCN(C)C12CCCN(C(C1CCCN1C1CC1)=O)C2 30796,c1(C(=O)NCC2(NC(c3cc(CCC)on3)=O)CC2)cc(Cl)c(Cl)n1C 30797,n1(CC)cc(C(=O)NC2CC2NC(=O)COCC2CCCCO2)c2ccccc12 30798,N1(C(C2(CCOCC)CCC2)=O)CC(CNC(=O)C(N)=O)CC(C)C1 30799,N1(C(c2c(CC)nccc2)=O)CC2(CCN(C(C3CCN3CC)=O)CC2)C1 30800,c1(N2CCC(NC(c3cc(SCC)no3)=O)C(F)C2)ncc(C#N)cc1C(C)=O 30801,C(=O)(CCN=C1NCCN2C(=O)CN1C2=O)NC1CCC1.CC(C)(C)C 30802,c1(OC)cc(C(=O)NCC2CCCCN2C(c2nccnc2Br)=O)ccc1O 30803,C1(C(=O)NCC(COC(C)C)O)(CNC(c2cscn2)=O)CC2(CC2)C1 30804,C(CC(=O)NCC(C)(C1CC1)NC(=O)CONC(=O)OC(C)(C)C)SCCC 30805,Cc1ccc(F)c(C(=O)NC(c2cn(-c3cc(C)cc(Cl)c3)nn2)C)c1 30806,N1(C(CN(C)CC)=O)CCC2C(CCCN2C(c2cc3nc[nH]c3cn2)=O)C1 30807,N1(C(CC(C)(C)OC)=O)C2CCC1CN(C(c1cncc([N+](=O)[O-])c1)=O)C2 30808,c1(C(=O)NCCC(C)NC(=O)CCc2nc(O)n[nH]2)c(F)ccc(F)c1N 30809,C1(C(=O)NCCN(C(C2(C)N(C(C)=O)CCC2)=O)C)COc2cc(Cl)ccc2O1 30810,C1(CC(=O)NCC(CC)NC(C2CCN(CC3CC3)CC2)=O)CCCC1(F)F 30811,N1(C(CSCCC)=O)CCC(CO)(NC(=O)C(O)C(C)C)C1 30812,CCC(CC(=O)NC(CCN(C(=O)C(C)Cc1ccccc1C)C)C(C)C)SC 30813,c1(C(N2CCCC(N(C(CSCCOC)=O)CC3CC3)C2)=O)ccc(O)cc1C 30814,c1(NC(=O)CNC(=O)C(C)(C)CC(F)F)cccc(N2CCCC2)c1[N+](=O)[O-] 30815,N1(C(CCOCC#C)=O)CCC2(CC1)CC2(CO)NC(=O)CNC(C1CCC1)=O 30816,CC1(C)CC(CNC(c2cncc(Cl)n2)=O)N(C(=O)CC2COC(=O)C2)C1 30817,c1(C(N2CCC3C(CCN3C(c3cc(Cl)no3)=O)C2)=O)nn2cccnc2c1Cl 30818,C(=O)(C(C)(F)C(=O)NC1CC(CNC(c2cc(Cl)cc(Cl)c2)=O)C1)OC 30819,N1(C(CNC=O)=O)CCN(C(C2CCCC23CCC3)=O)C2CCC12 30820,C(C1=CCN(C(=O)CC2CCC3CC3C2)CC1)NC(C(C)n1cncn1)=O 30821,C1(NC(c2ccsc2Cl)=O)CN(C(=O)C(F)=CC2CC2)CC12CCOCC2 30822,N1(C(=O)COCCF)CCN(C(C23CCCC2C3)=O)C2(CC2)C1 30823,C1(COc2cccc(C(N)=O)c2)CC(NC(=O)NCCF)C12CCC2 30824,c1(C(N2C3(CNC(CC(CC)O)=O)CC(C2)C3)=O)cc2cc(C)cc(C)c2[nH]1 30825,C(CS(=O)(=O)CC(=O)NC1CC1NC(c1nc(C)c(C)nc1C)=O)OC 30826,N1(C(C(C)(C)SC)=O)CCC(NC(c2cscc2Br)=O)C2(CCC2)C1 30827,c1(C(=O)NC2C(NC(C(CC(C)C)NC(C)=O)=O)CC2)cc2ncccc2s1 30828,Cc1ccc(F)c(C(=O)NCC(C2CCN(C(=O)CC3NC(=O)NC3=O)CC2)O)n1 30829,N1(C(c2cc(C)cc(F)c2)=O)CC(C)CN(C(C2Cc3cscc3C2)=O)CC1C 30830,CC1CCCCCC1NC(=O)C=CC1CCCN1C(=O)C=CC1CCCCC1 30831,N1(C(C(CC=CC)NC(=O)C=CC(C)(C)SC)=O)CCC2(C=CCO2)CC1 30832,C=C(CNC(c1cccc(O)c1)c1nnnn1CCOC)c1ccccc1F 30833,C12(C(C)NC(C(=O)Nc3c(CCC)onc3C)=O)CC3CC(CC(C3)C1)C2 30834,C(CC(C)C)(C(=O)N1CCCN(C(=O)Cn2ccnn2)CC1)OC 30835,CC1CC(NC(C2CCN(C3COC3)C2)=O)C(=O)N1c1ccccc1 30836,C#Cc1cc(C(=O)NCC(C)CNC(c2cc(Cl)cc(F)c2F)=O)cc(N)c1 30837,C(=O)(C(C)(CC)CC#C)N1CC(CC(=O)NCC2(OCC#C)CCC2)C(C)C1 30838,c1(CC)ncc(C(=O)NC2C(C(=O)NC3COC(C4CC4)C3)C2(C)C)cn1 30839,c1(C(=O)NCC=CC(=O)N(C2(COC)CC2)C)ccc([N+](=O)[O-])o1 30840,C(C)(C)(C(=O)NCCC(C)(C)NC(=O)CSc1nccn1C(C)(C)C)OC(C)=O 30841,c1(C(N2CC(C)C(NC(=O)C(c3ccc(F)c(F)c3)O)C2)=O)nc(Cl)ccc1N 30842,C=C=C(C)CC(=O)NCC1(CNC(=O)C(C)(CC)OC)CCOCC1 30843,c1(C(N(CCNC(C2CC(C)OC2)=O)Cc2ccccc2)=O)c[nH]c(=O)cn1 30844,N1(C(C(CC=C)OC)=O)CCC(C2CC2)C1C(=O)NCc1ccc(F)cc1 30845,c1(NCC2C(OC)CC2)c(C(=O)NC(=O)C(C)C(C)(F)F)cccc1F 30846,c1(C(=O)NCCC2(C)CCN(C(C3(OC)CC3)=O)C2)cc2n(n1)CC(C)NC2=O 30847,CC1CN(C(C2C3(CC3)C23CC3)=O)CC2(CCN(C(=O)CC3OCCO3)C2)O1 30848,N1(C(CSCC#C)=O)CCC2(CC1)CN(C(=O)Cc1nonc1C)C2 30849,C12(C(=O)NC3CCC(C(CC)(C)C)CC3)CCC(CC)(C1)OC2 30850,C12(CNC(=O)CC3CCN(C(C4CC(O)C(F)C4)=O)C3)CCC(CC1)C2 30851,N1(C(C2CC3(CCCC3)C2)=O)CCC2CN(C(c3cncnc3)=O)CCC12 30852,CCCC(C)=CC(=O)NC(C(=O)NCCOC1(C)CCC1)c1cccs1 30853,c1(N2CCC(CN(C)C)CC2)nc(=NCc2cocn2)[nH]c2c1COCC2 30854,C1(NC(C2(Br)C(C)(C)C2)=O)CCCN(C(c2ccc(F)o2)=O)C1 30855,c1(C(N2CC(COC)N(C(c3cccnc3)=O)CC2)=O)cccc2c1OCCO2 30856,Cc1cc(C(=O)NCC(C)NC(=O)COc2cccc(O)c2)ccc1F 30857,C(CCCCCCC)C(N1C(CNC(C(CC=C)OC)=O)C(CC)CC1)=O 30858,c1(CNC(=O)Cc2cc(C3CCCC3)no2)ocnc1-c1cn(CCCO)nn1 30859,C(=O)(C(=O)CCC(C)C)NC1CCN(C(C(=O)Nc2c(SC)cc(C)cc2)C)C1 30860,N1(C(c2cc(C(C)(C)C)on2)=O)CC(NC(C2(CO)CC2)=O)Cc2ccccc21 30861,N1(C(c2ccc(OC)s2)=O)CC(NC(c2ccc(CO)nc2)=O)C(F)C1 30862,c1(CCNC(=O)C(=O)NCC2(F)CC3(CNC3)C2)ccc(Br)cc1Cl 30863,N1(C(CC(C)SC)=O)CCCCC1C(=O)N(CCCC1CC1)C 30864,CC1(C)CC(CNC(=O)CNS(N)(=O)=O)CN(C(=O)C=C(Cl)Cl)C1 30865,C(c1cc(C(F)(F)F)ccc1Cl)=CC(N1CC(CNC(=O)CCF)OCC1)=O 30866,C#Cc1cn(C)nc1C(=O)NC1COCCC1NC(=O)CCCCCSC 30867,CC12CCC(C(=O)NCC3CN(c4nc5ccccc5s4)CCN3C)(CC1)CO2 30868,C1(NC(C(C2CCN(C(C3CC(=C)C3)=O)C2)F)=O)CCCCC1(C)O 30869,n1(CC)nc(C(=O)NC(C)CC(C)NC(=O)C(c2ccc(F)cc2)=O)c(C)n1 30870,C1(C(N(C2CC(C#N)C2)CC(=O)NCc2c(C)ocn2)=O)CC(=O)NC(C)C1 30871,Cc1cc2[nH]c(=O)c(C(=O)NCC3CN(C(C4(Cl)CC4)=O)CC3C)cn2n1 30872,Cn1c(C2CC2)nn(CC(=O)NC2CC2CNC(=O)Cn2cnnc2O)c1=O 30873,N1(C(c2cncc(CC)c2)=O)CCCC(F)(C(=O)NCc2ccccc2C#N)C1 30874,O(NC(=O)N(CC(F)(F)F)CCCO)CSCC(=O)NCCOC(C)C 30875,C(C(=O)N=c1cc(C)o[nH]1)OC(=O)C(=O)NC(C)(C)C.C(C1CCC(=O)O1)OC 30876,N1(C(CC(C)OC)=O)CC(CCNC(=O)CCc2cncc(Br)c2)C(C)C1 30877,CCCC(C(O)c1nc(C(c2ccc(Oc3cccc(C)c3)nc2)C)no1)OC 30878,C(C(CNC(C1(C)CC1(F)F)=O)C(F)(F)F)NC(c1c(CC)nccc1)=O 30879,C1(C)(C(=O)NCC2(CNC(c3c(C)ncnc3)=O)CCOCC2)CCCCC1C 30880,CC(C(=O)NCCCN(C(c1cc[nH]n1)=O)CC1CC1)NC(c1ccco1)=O 30881,Cc1ccc(S(=O)(=O)Nc2cccc(C)c2-c2cnc(COC(C)C)s2)c(F)c1 30882,c1(C2C(NC(=O)NCCc3cc(OC)ncc3)C2)cc(C)cc(Br)c1 30883,CCCC(C)CCCC(=O)NC(CNC(c1ncc(OC)cn1)=O)C(C)(C)C 30884,S(=O)(=O)(CCC(=O)NCC1CCCN(C(=O)COc2ccc(F)cn2)C1)N(C)C 30885,C1(C)(CC)CC(CC(=O)N(C23CC2CN(C(C)C(=O)NCCC#N)C3)CC)=NO1 30886,N1(C(c2c(OC)nn(C)c2)=O)CCCC(NC(c2ccc(O)nn2)=O)CC1 30887,N1(C(c2c(C)nn(C)c2Cl)=O)CC2(CCN(C(=O)CCc3cncc(O)c3)C2)C1 30888,C1(C(=O)NC2CCN(C(CCCC#C)=O)C2)COCCN1C=O 30889,c1(C(=O)NCC(CCCC)NC(=O)C=C(C)C(F)F)ncc(OCC)cc1F 30890,O=C(N=c1c(Cl)c[nH]cc1Br)C12CC1CN(Cc1cscc1Br)C2 30891,N1(c2cc(C)nc(Cl)n2)CCCC(C2CCN(C(=O)C(C)(C)S(C)(=O)=O)CC2)C1 30892,CC(CC(=O)N1CCN(C(=O)CC(O)C2CC2)C(CCO)C1)C(F)(F)F 30893,c1(C(=O)NCC2OCCN(CC(COCCOC)O)C2)cc(C)nc(C)n1 30894,CC1C(NC(c2cc(F)ccc2F)=O)CCCN1c1ncc(C(F)(F)F)cc1Cl 30895,N1(C(c2cccc(COC)c2)=O)CCCN(C(c2cccc(=O)n2C)=O)C(C)C1 30896,c1(C(N2C(CN(C(CSCCC(C)C)=O)C)CCC2)=O)ccccc1CC(C)C 30897,C(=O)(CCCC(=O)N1CCC(C(C)NC(c2ncoc2C)=O)C1)NCCC 30898,CC(=O)CCCCCN1CCC(N2CCC(O)C2)C1 30899,c1(C(=O)NCC(CC=C)NC(c2cc(OC)ccc2O)=O)cnn2cnnc2c1 30900,N1(C(C2(OC)CCC2)=O)CC(OC)CC(CNC(=O)CN(C)C(C)=O)C1 30901,C12(CNC(Cn3nnc(C)n3)=O)CCC(n3cc(CC(C)O)nn3)(CC1)C2 30902,c1(OC)c(C(N2CC(CO)(NC(c3ccc(=O)oc3)=O)C2)=O)cnn1C 30903,Cc1c(C(=O)NC2(CNC(C3CC4(C3)CC43CC3)=O)CCCCC2)cncc1F 30904,n1(CC)ccc2ccc(NC(N3CCC(C(F)(F)F)(C(=O)OC)C3)=O)cc12 30905,n1(CC(=O)NC(C)CN(C)C(C2CSC2)=O)cc(C2CC2)nn1 30906,CN1CC2(CCCN(C(=O)Cc3ccsc3[N+](=O)[O-])C2)OCC1=O 30907,N1(C(C[SH](CCC)CC)=O)CCCC1C(C)NC(=O)CCCOc1cccnc1 30908,C(CN=c1ccc([N+](=O)[O-])c[nH]1)N(C(C(C)(O)C(F)(F)F)=O)CCO 30909,CC1(C)CCN(C(C2CC2(C)C)=O)C(C(=O)Nc2ccc(F)c(O)c2)C1 30910,c1(CC(=O)NC2C(NC(CSCCC)=O)CCC2)cc(OC)c(Br)c(OC)c1 30911,C1(NC(CCC2CC(NC(CCN(CCC)C)=O)C2)=O)CCSCC1 30912,c1(NC(CCC)=O)ncc(C)s1.c12cc(cs1)N(C(C1CC(O)C1)=O)C2=O 30913,CC(CCCNC(C1(C2CCCO2)CCCC1)=O)NC(c1ccon1)=O 30914,CC1CN(C(c2sccc2F)=O)CC(C)CN1C(c1cnn(C)c1C(F)(F)F)=O 30915,C1(C(=O)NCC(C)N(C(C(C)NC(CC)=O)=O)C)CC(OC)C(OC)C1 30916,N1(C(Cn2ncc(C#C)c2)=O)CCCC(COC)(NC(=O)CSCCC#N)C1 30917,C(=O)(C(CN=[N+]=[N-])NC(=O)C(F)C1CCCC1)NCc1c(C)nc(C)s1 30918,C1(NC(C2CN(S(CC)(=O)=O)C2)=O)CCC(C)N(C(=O)Cc2ccns2)C1 30919,C1(C(=O)NC2(C)CC(NC(COC3(C#C)COC3)=O)C2)CCCC(OC)C1 30920,C1(CNC(C(COC)O)=O)CCN(C(C2(c3cccc(F)c3)CC2)=O)C1(C)C 30921,N1(C(C2CC(CNC(=O)CSCc3cccs3)C2)=O)CCc2cccnc2C1 30922,c1(C(N(CC(=O)NCC(C)NC(CCOC(C)C)=O)C)=O)ccccc1Cl 30923,C(=O)(C1CCc2c(Cl)cccc21)CC1CCC(C)(C)O1 30924,CC1=NOC(=O)C1CC(N1CCOC(C(C)NC(C2CN(C)CCO2)=O)C1)=O 30925,c1(N2CCN(CCOC)CC2)ccc(CNC(c2cnn(C)n2)=O)cc1C 30926,Cc1ccc2c(CNC(=O)N=c3[nH]onc3C3CCC(C(=O)O)C3)onc2c1 30927,N1(C(c2c(C)cc(F)s2)=O)CCC2CN(C(=O)C(C)Cc3ccnn3C)CC2C1 30928,C(C)(CO)(C(=O)NCC[Si](C)(C)C)N.Cc1ccn(C(C)C=O)n1 30929,N1(C(CNC(C)=O)=O)CCC(C)(CCNC(c2cccc(OC(F)F)c2)=O)C1 30930,c1(CN(S(C(C)C(F)F)(=O)=O)C2(C(C)(C)C)OCCS2)cnc(N)c([N+](=O)[O-])c1 30931,C#CCC(C)(C(=O)NC1CN(C)CC1O)NC(C1CCCCN1C)=O 30932,C1(C)(C(=O)NC(CNC(Cc2nc(C(C)C)sc2)=O)C)COC(=O)C1 30933,Cc1ccc(N)c(C(N2CCCC2CCNC(=O)C(c2cccnc2)O)=O)c1 30934,C1(CCC(=O)N(CCC)CC2CC2)CN(C(=O)CCOCC(C)C)CCC1C 30935,n1(CCOC)ncc(C(=O)N(C)CC2(NC(C3(C)CCSCC3)=O)CC2)c1C 30936,c1(C(N2CC(C)(NC(C3N(C(=O)OC)CC(O)C3)=O)C2)=O)cc(O)ncc1F 30937,CC(C)C(O)C(C)C(=O)NCC1(F)CN(C(=O)Cc2ncn3c2CCC3)C1 30938,c1(C(N(CC(C)NC(C(C2CC(F)(F)C2)OC)=O)C)=O)coc(C#N)c1 30939,c1(CC(=O)NCC(C)CN(C)C(C2CC2c2ccccc2)=O)c[nH]c(=N)nc1O 30940,c1(CN)ccccc1CNC(C1(Cn2ccnc2)CC1C(F)(F)F)=O 30941,c1(CCC(=O)NC(CN(C)C(c2ccc(F)s2)=O)(C)C)ncc(F)cn1 30942,c1(OC)ccc(C(N2CCCC(C)C2CNC(=O)C(F)(F)C(F)F)=O)c(N)c1F 30943,N1(C(C(CC)(C)O)=O)CCN(C(c2ccc(C(=O)OC)c(F)c2)=O)CC2(CC2)C1 30944,c1(C(=O)NCC2(NC(CS(CC)=O)=O)CCCCC2)cc(C)[nH]c(=NC)n1 30945,c1(CC(=O)NCC(C)NC(C2(CS(C)(=O)=O)CC2)=O)ccc(C2CC2)c(F)c1 30946,C(=O)(C1CCc2nccn21)N1C(C)(C)CC(NC(C2(c3cccs3)CC2)=O)C1 30947,c1(C(N2CCC(COCc3ccc(F)cc3)C2)=O)ccc2c(c1)CCN2 30948,CC1=C(C(=O)N2CCCCC2CNC(c2ccc(F)c(F)c2F)=O)CCS1(=O)=O 30949,CC(CNC(C1(O)CCOCC1)=O)C(F)C(=O)NC1(C(C)O)CC1 30950,C#Cc1ccc(C(=O)NC2CCOC2C(=O)NC)nc1.N12CCC(C1(C)C)C2 30951,N1(C(c2c(F)ccc(OC)c2)=O)CC(C(=O)NCCN2CCC2)C2(CCC2)C1 30952,C(=O)(C(F)CC(C)(C)NC(c1ncc(C)cc1C)=O)N1C(CC)(CC)COCC1 30953,C1(C)(CC)CC(O)CN1C(N1CCCC(CC2CC2)C1)=O 30954,C1(CNC(C2C(CCC)C2)=O)(CO)CC12CCN(C(c1cnnn1C)=O)CC2 30955,CC1(C)CC(NC(C2CC3CCC2CC3)=O)CN1C(C1CC(CCO)C1)=O 30956,c1(NC(C)=O)ccc(F)c(C(=O)NCC(C)(C(C)C)NC(=O)C(O)CN(C)C)c1 30957,[N-]=[N+]=NC1CN(C(C2CCC(NC(c3c[nH]ccc3=O)=O)C2)=O)C1 30958,C1(C)(C(=O)NCC2C(NC(c3c(C(C)=O)cn(C)n3)=O)CCC2)CCCS1(=O)=O 30959,N1(C(C2CN(C)C(=O)C2)=O)CCC(C2CC2)(NC(c2cc(F)c(F)cc2F)=O)C1 30960,N1(C2CN(C(Cc3nnc(C)o3)=O)C2)CCN(C(C23CCC(CC2)O3)=O)CC1 30961,C(=O)(CCC(C)(C)F)N1CCCC(CN(C(=O)Cc2nnn(C(C)(C)C)n2)C)C1 30962,C(CN=c1[nH]c(=NCCc2cccn2C)[nH]c2cc(C)ccc12)OCC 30963,C=CC(CC)CC(=O)NC(C1CN(C(C2(n3nccn3)CC2)=O)C1)C 30964,c1(N(C(N2CCC(CC3(F)CC3C)C2)=O)CC)ccnc(N2CCC2)c1 30965,C(C1(C)OCCc2ccccc21)CC(=O)OC.c1(O)cc(Br)c(F)cc1S(=O)(=O)N 30966,C1(C)(CNC(C(CSCC)C)=O)CN(C(c2cccc(O)c2C)=O)C(C)(C)C1 30967,C1(NC(=O)C2=COCCC2)CCN(c2ncc(Br)c(O)n2)CC12CCC2 30968,N1(C(C(C)c2cccs2)=O)CCCC(CCNC(=O)COc2ccccc2)C1 30969,N1(C(Cc2n(C)cnn2)=O)CC2CC(NC(c3cn(CCO)nn3)=O)CC1C2 30970,N1(C(c2cn(C(C)(C)C)nn2)=O)CCC2(CCN(C(C3CC3CF)=O)C2)C1 30971,n1(CC)nc(C)cc1C(=O)NCCC(C)NC(C1(C)CC=CC1)=O 30972,Cc1nc(C(=O)NC2C3CN(C(=O)C=CC4CCC4)CC23)c(=O)[nH]c1C 30973,c1(C(N(C2CCCN(C(C(=Cc3ccco3)C)=O)C2)C)=O)c(N)cc(F)cc1Cl 30974,C1(NC(COCC(=O)NC)=O)CCCC1NC(C1CC(Cl)(Cl)C1)=O 30975,C(=O)(CS(=O)(=O)CC(C)C)N1CCCN(C(c2oc(CC)c(C)c2)=O)C(C)C1 30976,c1(C(=O)NCC(CC=C)NC(C2(C)CCOCC2)=O)nc2ccccc2cc1C 30977,Cc1cc(C)c(NC(=O)CN(C)CCN(C)C(C2CNC(=O)CC2C)=O)c(C)c1 30978,C1(Nc2cnc(OC)nc2)COC2(CCN(Cc3cc(Cl)ccc3Br)CC2)C1 30979,c1(C(N2CC(OCC)(CNC(C3CCC(CC)O3)=O)C2)=O)c(Cl)nn(C)c1Cl 30980,C1(NC(c2cc(OC)n[nH]2)=O)CC2CCC(C1)N2C(C1CCCC1CF)=O 30981,N1(C(C(CC)C(C)O)=O)CC2(C1)CN(C(=O)Cc1ccc(O)cc1)CCO2 30982,C1(NC(C(C)(C)C2CC2)=O)CN(C(C2CCC3(C2)N=N3)=O)CCC12CCC2 30983,CCCCCC(O)CC(=O)NC1CN(C(=O)CCn2ccc(=O)c([N+](=O)[O-])c2)C1 30984,c1(C(C(=O)NCC2(C(=O)NC(c3cccs3)C)CC2)C)ccccc1 30985,C(C(F)(F)CCC(=O)NNC(=O)c1cnccn1)n1cc(CCOC)nn1 30986,c1(CC(N2CC(C(C)NC(CCOCCCC)=O)C2)=O)nc(CSC)n[nH]1 30987,C12(CNC(c3ccc(O)nc3Cl)=O)CCCCC1CN(C(=O)Cc1cc[nH]c1)C2 30988,N1(C(CC=C)=O)CCCCC1CN(C)C(C1(n2cccn2)CCOCC1)=O 30989,C1(n2cnnn2)(C(N2CCC(N(C(C3C(OC)C3)=O)CC)C2)=O)CCCCC1 30990,C1(C(=O)NCCOCCCNC(c2ccc(C(C)C)s2)=O)CN2CCCC1C2 30991,c1(NS(C)(=O)=O)ccc(NC(=O)NCC2CNC(=O)CO2)cn1 30992,C1(C(c2n(C(CC)C)nnn2)NCc2ccno2)CC(OC)C12CCOCC2 30993,N1(C(CN(CCC#C)C)=O)CCC2(COC(CNC(=O)CC3OCCCO3)C2)C1 30994,c1(C(=O)NCC(=O)NC2C3C=CC(C3)C2C2CC2)cc2ccccc2o1 30995,N1(C(C2N(C)CCOC2)=O)CC2(CC(NC(C3(C)CCNC3=O)=O)C2)C1 30996,N1(C(CCC(C)(C)O)=O)CCC2(CC1)CCN(C(=O)C(C1CCCO1)C1CC1)C2 30997,n1(CCCC)cc(C(N2CCC(C(C)NC(c3nc(C)oc3C)=O)C2)=O)c(C)n1 30998,O=C(CN1CCCC1)N1CCC(S(=O)(=O)NCc2ccccn2)c2ccccc2O1 30999,C(=O)(C(C)(C)CC(F)(F)Br)NC(C)CNC(c1cc(C#N)ccc1Cl)=O 31000,C1(C(=O)NC(CNC(c2c(C)ncn2C)=O)C(C)C)CCCCN(C)C1=O 31001,N1(C(C2CCC2(F)F)=O)CCC(F)(CNC(C2(c3cccnc3)CCC2)=O)C1 31002,C(=O)(CC(C)CC(=O)NC(CNC(=O)CCn1cc(C)cn1)CO)OC 31003,N1(C(CCCCC=C)=O)CC(C(=O)NCC2C(CO)C2(C)C)CCC1(C)C 31004,C1(C(C(=O)N(CCN=[N+]=[N-])C)F)CCN(C(C2(c3cc[nH]n3)CC2)=O)C1 31005,C(CN=c1[nH]c(Cl)nc2ccccc12)NC(C(C(C)C)NC(C)=O)=O 31006,C(C(C(C)(C)C)NC(C1(C)COC(=O)C1)=O)NC(Cc1cn(C)nc1)=O 31007,c1(C(=O)NCC2CCC(NC(C3C(OC)CC3)=O)CC2)cc([N+](=O)[O-])c[nH]1 31008,C1(NC(C=CCC)=O)(CO)CCCN(C(=O)C(C)N(C(=O)CC)C2CC2)C1 31009,c1(C(C)C)cncc(C(=O)NCC2CC(NC(=O)CCc3cccn3C)C2)c1 31010,c1(C(N(CC(CC)NC(c2cccnc2)=O)C)=O)c(C)oc(C)c1C 31011,N1(C(C(C)Cc2cnn(C)c2)=O)CCC2(CCCN2C(C2CC2(C)C)=O)C1 31012,c1(C(N(CC(C)O)CCNC(C2(C)CC=CC2)=O)=O)ccc(-c2cnn[nH]2)cc1 31013,C1(NC(CS(=O)(=O)NCC)=O)CC2CC1CN(C(c1nc(C)sc1C)=O)C2 31014,C(=O)(C(F)(F)C(F)(F)C(F)(F)C(F)F)NC1C(C)(C)C(C(=O)O)C1 31015,c1(-c2ncc(C(=O)NCC(CC)NC(=O)C(F)CC3CC3)s2)ccc(F)cc1F 31016,N1(C(c2c(CC)nc[nH]2)=O)CC2(CC(NC(=O)C(C)C(C)CC)C2)C1 31017,C1(NC(CCCC=C)=O)CCN(C(=O)Cn2cncc2C(=O)OC)CC1C 31018,N1(C(C2(CC)COC2)=O)CC2CCC(C1)CC(C(=O)NCC13CCC(CC1)C3)C2 31019,c1(SC)c(C(=O)NC2CCN(C(C3CCCN3C)=O)CC2F)cccc1F 31020,CC(CNC(=O)COC(F)(F)F)CNC(=O)C(F)C1CCCC1 31021,C1(NC(c2cc(-c3ccns3)on2)=O)COCCN(Cc2ccccc2)C1 31022,N1(C(C)=O)CC(NCCc2cc(-c3ccc(-c4ccccc4)cn3)[nH]n2)CC1(C)C 31023,c1(C(N2C(C)CC(CNC(=O)Cn3cnc(=N)[nH]3)C2)=O)ccc2c(c1)nnn2C 31024,c1(C(=O)NC2(C(=O)NCCOC(C)=O)CCCC2)ccc2ccccc2c1 31025,C1(Nc2nc(CC)cc(CC)n2)CC2CCC1N(C(=O)CCC(C)SC)C2 31026,O=C(C1=COCC1)NC1(CNC(=O)CC2CCC(C3CC3)O2)CCCCC1 31027,C1(CC(=O)NC(c2ncc[nH]2)CC)CCC(NC(c2cnn(CCOC)c2)=O)C1 31028,Cc1ccc(C(=O)CC(=O)N2CCC2CNC(c2nn(C)c(Cl)c2Cl)=O)cc1C 31029,C(C(C(=O)N(C)CC1CCCN1C(c1ncoc1C)=O)C(C)(C)C)OCC=C 31030,C1(NC(CCOCCOC)=O)CN(C(c2ccsc2)=O)CC1C 31031,CC(C)CC(C)(C)C(=O)NCC1CC(C)CN(C(=O)C(Cl)=CCl)C1 31032,C1(C(N(CC)Cc2nnnn2C)=O)CC(=O)CN1C(=O)CC1CCCC1 31033,C1(C(N2CC(CNC(c3c(C)nc[nH]3)=O)C(C)C2)=O)CCc2ncncc2C1 31034,C1(C2CC2)(C(=O)NCC(CC)(CC)NC(c2cnn(C)c2Br)=O)CC=CC1 31035,N1(C(c2cc(OC)c(O)nc2)=O)CC2(CCN(C(c3nc(C)n(C)n3)=O)C2)C1 31036,CCCCCC(O)CC(=O)NC12CCC(CNC(=O)C=CCOC)(C1)OC2 31037,c1(C(C)C)nccc(C(=O)NC(C2CN(C(c3ccccc3F)=O)C2)C)n1 31038,N1(CC(c2c(C)c3c(s2)cccc3)=O)CCC2(CCOC2=O)CC1 31039,C1(C(C(=O)NC(CN(CCOC)C)C)(C)C)CCCCN1C(C)=O 31040,C1(N(N2CCCC2c2ccccc2)C)(C=O)CCCNC1.C(C)(C)(C)ONC 31041,C1(C(=O)NCCC(CNC(=O)CCOCC(F)F)O)CC(c2ccccn2)=NO1 31042,C(N=c1[nH]c(=NCC23COCCN2CCC3)[nH]c2c1COC2)c1c(Cl)c(Br)ccc1 31043,C(CCCCC(=O)NCCC(C)NC(c1cccs1)=O)NC(=O)NC 31044,CCCC(CNC(C1CCC(=O)N1C(C)C)=O)CCO.c12cccc(c1)C2 31045,c1(CC)c(C(=O)NCCN(C(c2cccc(CCO)c2)=O)C2CC2)nnn1C 31046,C(=O)(C(C)(C)C(O)C(C)C)N(CCC(C)NC(c1cc(C2CC2)n(C)n1)=O)C 31047,c1(-n2ncc(C(N(CCNC(C(CC)SC)=O)C3CC3)=O)c2)cccc(C#N)c1 31048,c1(CC)cnc(O)c(C(=O)OCCNC(c2cc(CO)ccc2OC)=O)c1 31049,C(CO)(CCCNC(=O)C=Cc1ccoc1)NC(Cc1scc(C)c1)=O 31050,c1(NC(C(=O)NCC)=O)ccc2c(c1)CCN(C(c1ccc3ncnn3n1)=O)C2 31051,c1(C(c2ccc(O)s2)=O)ccc(C=O)cc1.N(C)(CC1CC1)N(C)CCOCCO 31052,C1(O)(CNC(c2cccc(-n3ccnc3)n2)=O)CCN(c2nnc(CO)s2)CC1 31053,C1(NC(Cc2n(C)ccn2)=O)CCCC12CCN(C(c1cc(N)nc(O)c1)=O)C2 31054,c1(C(N2CC(CCNC(=O)C(C#N)C(C)C)(OC)C2)=O)cc(S(C)(=O)=O)co1 31055,N1(C(COCCOC)=O)CCCN(C(=O)C(N2CCCCCC2=O)C)CC1CO 31056,CC1(C)C(CC(N2CC(CNC(=O)Cc3ccc(O)nc3)C2)=O)C1(C)C 31057,CC1CC(NC(C2CC3CCC(C2)S3)=O)CCN1C(c1cc2occc2s1)=O 31058,N1(c2nnc(C(=O)OCC)s2)CCC2(CCC2)C(NC(=O)C2=COCCC2)C1 31059,CC(C)C(C)C(CNC(C1(Br)CC1(F)F)=O)NC(=O)Cc1cnc[nH]1 31060,C(=O)(C(=O)C(F)(F)F)NCC(C)CNC(=O)CN(C)C(=O)C1CC1 31061,N1(C(CC=O)=O)CCCCC(C2CN(CCC3CC3)C2)C1.CC=O 31062,N1(C(c2c(C)snc2)=O)CCC(C2CCCCN2C(=O)CSCC(F)(F)F)CC1 31063,Cc1cc(Br)cc(C)c1OC(=O)CCOCC1CC1 31064,Cc1cc(CN2CCOC(C(N3CCC(CO)C(O)C3)=O)C2)c(C)cc1Br 31065,c1(C(=O)NCC23C(CN(C(C4(C(=O)OCC)CC4)=O)C2)C3)c(C)ccc(C)c1O 31066,CCCCCCN(C(=O)CCC=C(C)C)CCCC.C1(=O)C(C)N1 31067,N1(C(C(C)SCC)=O)CCOCC12CNCCOC2 31068,c1(C(N2CC(C)(c3cn(-c4ccc(Cl)nc4)nn3)C2)=O)nccc2cccnc12 31069,C(=O)(CCCCCN(C(=O)CC=CC(C)(C)C)C)N(C)CC1CC1(C)C 31070,c1(CNC(C(C)c2ccsc2)=O)ncc(C(=O)NCC23CC(CO)(CO2)C3)cn1 31071,c1(C(=O)NCCN(CCOC)C(C2CCS(=O)(=O)C2)=O)cc(Cl)n[nH]c1=N 31072,c1(C(N2C(CC(N3CC(=C)C3)=O)COCC2)=O)cccc(C)c1C#N 31073,C(=O)(C1=C(C)CCOC1)N1CCC(F)(C(N(CCCCCC)C2CC2)=O)C1 31074,C1(COC)(NC(=O)CCC2CCCC2)CCN(C(C2COC2)=O)C1 31075,CS(=O)(=O)c1cc(C(N2CC=C(CCNC(=O)C3=C(Cl)CC3)CC2)=O)cc(F)c1 31076,C(=O)(C1=CCC(F)(F)CC1)NC1CCN(C(C2CCC(C(F)(F)F)O2)=O)C1 31077,N1(C(c2c(C)scn2)=O)CC2C3CCC(C2C1)N(C(c1cccnc1O)=O)C3 31078,C(CCS(=O)(=O)NCC(N1CCCCC1CCN(C)C(C1CC(F)C1)=O)=O)OC 31079,N1(C(COC2CN(C(C)=O)C2)=O)CCC2CN(C(=O)Cn3ccc(C)n3)CC12 31080,c1(CN(C(=O)C(F)(F)C2(O)CCC2)C)cccc(C2CC2)c1.C12(O)CN(C1)C2=O 31081,c1(CC)cc(C(N2CCC2C(N2CCC2C2CCCC2)=O)=O)ns1 31082,c1(C(=O)NCCC(C)N(C(c2n(CC)ncc2)=O)C)cc2c(Cl)cccc2[nH]1 31083,c1(OC)cc(N)c(F)cc1C(=O)NC1CCC1NC(=O)Cc1cc(C2CC2)on1 31084,C#Cc1ccc(C(N2CCC(N(C(=O)Cc3ccn(C(F)F)n3)C)C2)=O)cc1F 31085,C1(C(=O)OCC2CCC2)CCN(C(C2CC=CCC2)C(=O)NC2CC(F)(F)C2)C1 31086,C1(NC(C2(CCNC(=O)C(O)c3cnc[nH]3)CCC2)=O)COCCC1(F)F 31087,c1(CC(=O)NC2(C)CCN(C(c3n(C(C)C)cnn3)=O)C2)nnc2n1CCCC2 31088,C12(NC(C3CCC4(CCC4)CO3)=O)CCCC1N(C(c1cncs1)=O)CCC2 31089,N1(c2cc(NCCC3ON=C(C)C3)ncn2)C2CCC1CN(C)C2 31090,CC1CC(C(=O)NCC2(C(=O)NCC(F)Cl)CC2)=NO1 31091,C1(NC(C2CCC(C)C2)=O)CC2(NC(=O)CCCc3nc(C(C)C)no3)COC1C2 31092,C(C)(CCCC(C)C)NC(CC(CNC(C(COC)(C)OC)=O)C1CCC1)=O 31093,c1(OC)ccccc1CN1CCC(CNC(c2cc(C#N)c[nH]2)=O)C1 31094,c1(C(C(=O)NCCCN(C(Cn2nc(C)c(Cl)c2)=O)C)(F)F)ccc(F)c(F)c1 31095,c1(CCO)cccc(OCCNc2cc(I)ccn2)c1 31096,C1(NC(C2(CC)CC2)=O)CC=CCC1C(=O)N(CC(F)(F)Cl)C 31097,C1(NC(c2cc(Br)ccc2F)=O)CCCN(C(c2ccc(I)c(O)c2)=O)CC1 31098,c1(-c2[nH]nc(C(=O)NCC3(CO)CC34CCC4)n2)ccc(F)c(Cl)c1 31099,N1(C(c2ncn(CC)c2)=O)CCC(C)C1CNC(=O)C=Cc1ncco1 31100,c1(C(=O)NC(CC(C)NC(c2cccc(C(C)=O)c2)=O)C)cc(C)c(C)nn1 31101,C1(NC(C2CCC3(CN(S(=O)(=O)CCCCl)C3)O2)=O)CCc2ccccc2O1 31102,c1(N(C(C(C)CCCc2cn(CCCF)nn2)=O)C)cccc(S(C)(=O)=O)c1 31103,CC(F)(C(=O)N1C2CCC1CN(C(c1ccc3cnoc3c1)=O)C2)C(F)(F)F 31104,C(C)(C(=O)NC(C)COCC(C)(C)C)(C1(C)CC1)OC.c12cn-1nn2 31105,N1(C(CN(CC(=O)NC(C)CCC=C(C)C)CC=C)=O)CCCCCC1 31106,C1(NC(c2c(C)cc(F)nc2)=O)CCC2CC1CN2c1nc(Cl)ncc1Cl 31107,C(=O)(CCO)NC(N)=O.C(=O)(C(C)n1cncn1)NCC(C)NC(c1cccs1)=O 31108,C(CCCC(CO)NC(C1CC2CC2C1)=O)NC(C1(CC)CCC1)=O 31109,C1(C(c2nnnn2C2CCC2)NC2C(C)CSC2)(CCl)CCOCC1 31110,C1(c2n(CC(=C)C)nnn2)(NC2CCCCCC2CO)CC2COC1C2 31111,c1(CC(N2CCCC(N(C(=O)COC3CC3)CC)C2)=O)ccc(Cl)c(C)c1F 31112,C1(C(N(CC(C)NC(c2c(C(F)(F)F)cccc2O)=O)C)=O)CC(F)(F)C1(C)C 31113,N1(C(C)=O)CC2CCC(NC(c3ccnc(C(N)=O)c3)=O)(C2)C1 31114,c1(C(=O)NCC23C(CN(C(C=C4CCN(C)CC4)=O)C2)C3)ccnc2ncnn12 31115,c1(C(=O)NCCN(C(CC(C)O)=O)CC(C)O)cnc2c(c1)NCC2 31116,c1(CC)nc(C)c(C(=O)NC(C)CNC(c2nnsc2SC)=O)o1 31117,c1(C(=O)NCC#CCNC(=O)C=C(Cl)Cl)c(F)ccc(F)c1F 31118,C1(CNC(C(F)=CC)=O)CCC(C)(C)CN1C(=O)C=Cc1nc[nH]n1 31119,N1(C(C(CC=C)C)=O)CCC2C(CCCN2C(c2cccnc2N)=O)C1 31120,c1(CN2C3CN(C(c4sc(CCC)c(CC)c4)=O)C(C3)C2)ccc2[nH]ccc2n1 31121,C12(C(=O)NCCCC(C)NC(C34CC3COC4(C)C)=O)CC3CC(C(=O)N1)C2C3 31122,c1(CN2CCN(C(=O)Cc3nc(C4CC4)cs3)C3C2C3)cnc2c(c1)COC2 31123,c1(NC(C2CCCN(C(c3c(OC)ccc(Cl)c3)=O)C2)=O)cc2ccoc2cn1 31124,c1(OCC)cnc(C(=O)NC2COCCC2NC(c2cc(CO)on2)=O)c(Cl)c1 31125,CCC(F)(C(=O)OC)C(=O)N(C)CCN(C(=O)C(c1ccc(F)c(F)c1)(C)C)C 31126,c1(C(N2C3CC(NC(COCCC#C)=O)(C3)C2)=O)cc(C)c(C(=O)OC)o1 31127,C1(C(=O)NC(C2CC2C(=O)NCC(F)(F)C(N)=O)C)CC(O)C(F)C1 31128,C=CC1(c2ccc(OC)cc2)COCCN1C(=O)C(=O)NC1(Br)CCC1 31129,N1(C(c2ccc(OCOC)cc2)=O)CC(NC(=O)CC2C(C)C2(F)F)CC(F)C1 31130,C1(C)(CCNC(C(N2CC(C)C2)C)=O)CCN(C(c2cnnn2C)=O)C1 31131,c1(C(N2CCC(NC(C3CCC(C)O3)=O)CC2C)=O)ccc2ncccc2c1F 31132,C1(C(=O)NC2CCCC2CF)COC2(C1)CN(C(=O)Cn1ncnn1)C2 31133,CC(CC(=O)NC(CNC(=O)C1=CSCS1)CC(F)(F)F)CC(F)(F)F 31134,C1(C(=O)NC(c2nocc2C(=O)NC2(CN(C)C)CCC2)C)CC=CC(O)C1 31135,Cc1cc(NC(C2CCN2C(=O)Cc2ccc(Cl)s2)=O)cc(Br)c1 31136,C1(C(=O)NC2CC(OCC(=O)NC(C=C)COC)C2)CC(=O)NC(C)C1 31137,c1(OC)nc(C)cc(=NC(C)CC(C)NC(=O)C=CC(=O)N(C)C)[nH]1 31138,C(=O)(C1=CCCCO1)N1CCC(OCC(=O)N(C)Cc2ccccc2F)C1 31139,N1(C(C(c2c(C)cccc2C)O)=O)CCN(C(c2cnc(=N)[nH]c2)=O)CC(CO)C1 31140,c1(C(=O)NCC2CC(NC(COCC)=O)C2)ccccc1SC(C)C 31141,CCCCCCCC(F)C(=O)N1CCOCC12COC2 31142,C(=O)(CCN=C(NCC(C1CCCCO1)(C)C)NCC1C=CCC1)N(C)C 31143,CC1(C)CN(C(=O)Nc2cc(OCc3ccccc3)ccc2Cl)CCC1CO 31144,Cc1scc(C(=O)NCC(C)(O)CNC(c2cccn2C2CCCC2)=O)c1N 31145,C(=O)(C(CC(C)C)N(C)C(=O)N(C)C(C)C)NC(c1ccccc1OC)C(CC)C 31146,C(=O)(C(C)(O)C(C)C)N(CCCOCCN(C(c1ccc(OC)s1)=O)C)C 31147,Cc1oc2cc(C(=O)NCC3CC3NC(c3nccc4n[nH]cc34)=O)[nH]c2c1C 31148,c12ccc(cc1)CNC2=O.c1(C(N(C(C2CCOC2)C)C)=O)coc(N(C)C)n1 31149,C1(C(=O)NC2CCN(C(=O)CCc3ncco3)C2C2CC2)CCCS(=O)(=O)C1 31150,C1(NC(c2c(N)c(F)ncc2)=O)CC2CN(C(=O)CC(F)(F)F)CCN2C1=O 31151,CCC(C)CC(=O)NCC(CC1CCCC1)C(=O)NCc1ncnn1C(C)C 31152,C1(C(N2CCCCC(NC(CCC(=O)NCCC)=O)C2)=O)CC2(CCCC2)CO1 31153,c1(C(N(C(C(=O)N(CC(C)O)CCOC)C2CC2)C)=O)ccc2c[nH]nc2c1 31154,Cc1ccc(N)cc1C(N1CCCC(NC(=O)C=C2CCN(C)CC2)C1)=O 31155,N1(C(CNC(=O)OCC)=O)C2CCCC1C(NC(=O)CC1CCN(OC)CC1)C2 31156,CCC(C(=O)NCCC1CCN(C(=O)CN2CCN(C)C(=O)C2)CC1)C(F)(F)F 31157,C1(NC2CCN(C(c3n(CCC)ccc3)=O)C2)C2CCC(C2)C1CO.C(=O)C1CC1 31158,C1(c2scc(CC(=O)NC(C(C)NC(CCCC)=O)C)n2)CCCCCC1 31159,C(C)(C(=O)N1CC(C(O)C(=O)NCCn2ccnc2)C1)OCC=C 31160,C(=O)(C(O)CC(N)=O)N1CCC(CC=C)(NC(c2ccc(SC)s2)=O)C1 31161,N#Cc1c[nH]c(C(N2CCC(C(N3CCN(c4cnccn4)CC3)=O)CC2)=O)c1 31162,C1(NC(c2ccc(CC)s2)=O)CCCN(C(=O)C=C2CCCCC2(C)C)CC1F 31163,N1(C(C(c2cnn(C)c2)SC)=O)CCc2ncc(CO)cc2C1 31164,c1(C(=O)NC2CC3CC2N(C(C2CCCS2)=O)C3)noc2c1CC(F)(F)CC2 31165,CCCC(O)C(=O)NCC12CC(NC(C3CCCN(CCC)C3)=O)(CO1)C2 31166,C1(C(C)(C)C)(CNC(CN(S(CC)(=O)=O)C)=O)CCN(C(=O)C(F)C2CC2)C1 31167,c1(-n2cc(C3N(C(c4ccn(-c5ccccc5)n4)=O)CC3)nn2)cc(Br)c(O)cc1Br 31168,CCC(CCC(=O)N1CCC(C)C1COC)NC(=O)C=CCN1CCC1 31169,C12CCCCC1N=C1C=C(C)NC(=NCCN2C)N1.c1(CSC)ccccc1 31170,N1(C(C)=O)CCC(C2(NC(C3COC(=O)O3)=O)CCC2)CC1 31171,C1(CC(N2CCCC(OC)CC2)=O)C2CCC1CN(Cc1cncs1)C2 31172,c1(OCC(=O)NCC2C(NC(c3c(C)cno3)=O)CC2)cccc(Br)c1C#N 31173,C(C(C)(O)CNC(=O)C=CC=NCC#C)NC(CCNC=O)=O.C(C)=C 31174,c1(CCC)c(C(=O)N(C2CCCN(C(=O)C(F)=C(C)C)C2)C)nnn1CC 31175,c12nc(Cl)ncc1O2.C(C)(C(=O)NCCN(CC)CC)OCCC=C 31176,CC1(CNC(=O)CC2COCC2O)CCCN1C(c1ccc(OC(F)F)cc1)=O 31177,Cc1ccc2c(C(=O)NC3CCC4CCN(C(c5cccs5)=O)CC34)n[nH]c2c1 31178,N12CCCCC1C2=O.C1(OC)CCCC1C(=O)NOCC=CCl 31179,C(=O)(C(CC)CC(F)F)N(CC(CNC(C(C)OCCOCC)=O)(C)C)C 31180,N1(C(CC2(C)OCCO2)=O)CC(F)(F)CC1C(=O)NCCC1CCCC12CC2 31181,C1(CNC(C(C)C2CCC2)=O)CCC(F)(CNC(c2cncc(C#N)c2)=O)CC1 31182,C1(C)(C(=O)NCC(C2CCCCC2)NC(Cc2c(C)con2)=O)CCCCO1 31183,N1(C(CCCC#C)=O)CCC(NC(=O)C=Cc2ccc(C(N)=O)cc2)CC1C 31184,C1(CCC)(NC(c2ccnn2C(C)C)=O)CCCN(C(c2n[nH]c(CO)n2)=O)C1 31185,CC1(C)CN(C(=O)Cc2ccccc2Br)CC1NC(c1cnnc(O)c1)=O 31186,c1(NCC(CC=C)C2CCC2)ncc(S(=O)(=O)NCCSc2ccco2)cc1Cl 31187,c1(COC(c2c(C)nc(C(C)SC)s2)=O)cc(F)c(F)cc1Br 31188,C(=O)(C#CC1(C)CCCO1)NCC1(CCNC(c2cccc(C)c2)=O)CC1 31189,C1(NC(=O)OC(C)(C)C)CN(N2CC(SC3CC3)C2)Cc2cc(CO)nn2C1 31190,Cc1cc2c(C(=O)NC3CCCOC3C)cccc2o1 31191,C1(NC(C2C(CC)C2)=O)CC(C)CN(C(c2ccc(-c3nnc(S)o3)cc2)=O)C1 31192,C(=O)(C1=NOC2(CCC2)C1)NCCCC(=O)NCCCOC1CCCOC1 31193,N1(C(COc2cn(C(C)C)nc2)=O)CCCCC(NC(=O)C(C)n2ccnc2)C1 31194,C(=O)(C1=CCS(=O)(=O)C1)N1CCC(NC(C(C(=C)Cl)(C)C)=O)C(F)C1 31195,C(C)(CNC(C1CCCS1)=O)(CNC(C1(CC(C)C)CC1)=O)OC 31196,N1(C(=O)NCCCCCF)CCN(C(c2cnc(C3CC3)o2)=O)CC1 31197,C1(C#N)(C(=O)NCCC(CC)(C)NC(=O)CC2(O)CCC2)CC12CCC2 31198,N1(C(CC(C)(C)C2CC2)=O)CCN(C(C2C3CN(CC(F)(F)F)CC23)=O)C(C2CC2)C1 31199,C1(CC)CN(C(=O)CC(F)F)CCC1NC(=O)CN(C)C(=O)Nc1ccccc1 31200,N1(C(CCCn2ncc(C)c2)=O)CC2CC3CCCN3C2C1 31201,c1(C(C)=O)c[nH]c(C(N2CCC(O)(C(C)CNC(c3csc(C)c3)=O)C2)=O)c1C 31202,CC1(C)C(NC(=O)C2=NOCC2)CC1CC(=O)NC1CCOCC1F 31203,C1(CNC(C2(SC)CCC2)=O)CCCN1C(C1CCC(=O)C1)=O 31204,C1(CNC2(C(=O)NC(COC)C3CC3)CCC2)C2CCCCC12 31205,N1(C(CNC(=O)OC)=O)CC(CC(=O)NCCn2ccnc2)C(C)C1 31206,n1(CCCC)cc(C(=O)NC(CNC(C23CCC(OC)C2C3)=O)C(C)C)c(C)n1 31207,C1(NC(CCc2c(C)n[nH]c2C)=O)COC2CN(C(c3ocnc3C)=O)CC12 31208,c1(CCC)ncc(NC(=O)C(O)CCNC(C2(F)CCOC2)=O)cn1 31209,c1(CC)nc(C(N2CC(CO)(NC(c3scnc3C(C)C)=O)C2)=O)cs1 31210,C(=O)(CCCCC(C)(C)C)NC1CC(O)(CNC(C2CCCN(CC)C2)=O)C1 31211,n1(CC(=O)NCCOCCN(C)C(C2(n3cnnn3)CC2)=O)cnc(=N)[nH]1 31212,N1(C(CN(CC(C)C)C(c2c(CC)cno2)=O)=O)CC(F)(F)CC1CO 31213,c1(CN2CCC(N3CCCC3)C2)c[nH]ccc1=NC(=O)C12CC(C(=O)OC)(C1)C2 31214,c1(-c2cc(C)[nH]n2)cccc(C(=O)N(CCCNC(=O)C(O)CSC)CCO)c1 31215,S(=O)(=O)(c1ccc(Br)cc1NCC1OCC1(C)C)N1CCCC(CCC)C1 31216,c1(SCC)nccnc1C(=O)NCC(O)CCNC(C1(CC)CCC1)=O 31217,CC1C(NC(C2CCC2)=O)CC2CCC1N2C(=O)CC1CC(F)(F)C1 31218,C1(CC(=O)NCC2CCC(NC(Cc3c(C)ccnc3)=O)CC2)CCCS(=O)(=O)C1 31219,C(CC(=O)N1CC(CNC(=O)C(C)c2ccsc2)C1)(C(F)(F)F)OC 31220,c1(C(=O)NCC2(F)CCC(NC(C3CCS(=O)(=O)N3)=O)C2)ccc2nn[nH]c2c1 31221,Cc1ccncc1CCC(=O)NCCCC(CO)NC(c1ccncc1)=O 31222,c1(C(N2CCC(CNC(C(C)SC)=O)C23CCC3)=O)ccc2ncc(=O)[nH]c2c1 31223,C1(CC(=O)NC(C2CN(C(c3cn4ccsc4n3)=O)C2)C)COCC1(C)C 31224,C1(NC(c2cc(OC)n[nH]2)=O)CCCN(C(C2CC3C=CC2C3)=O)C1C.C1CO1 31225,C(N=C(NC1CCS(=O)(=O)C1)N1CCn2c(cc3c(Cl)cccc23)C1)C1C(C)(C)C1 31226,C(=O)(CCC(C)OC(c1ccc(C2CCC2(C)C)cc1)=O)OCC 31227,CC(CN=c1cc(CCNCCCOC(F)(F)F)nc[nH]1)c1ccccn1 31228,c1(CC(=O)N(C)CCNC(C2CC3CC3C2)=O)ccc(S(=O)(=O)C(F)(F)F)cc1 31229,C1(CNC(c2cnsn2)=O)CC2CN(C(C3(n4cnnn4)CCCCC3)=O)CC12 31230,c1(C(N2C(C(=O)NCC3CCCOC3)COCC2)=O)ccc(O)c(F)c1 31231,CC1SCCC1N=c1[nH]c2c(c(=NCc3ccnc(N4CCCC4)c3)[nH]1)CCC2 31232,c1(OC)ccccc1CNC1CCN(C(c2ccnc(S)c2)=O)C1 31233,C1(C(=O)NCC2(CC)CCCC2)CC=CCN1C(=O)CC1(C)CCC1 31234,C1(F)(CNC(C(F)=C(C)C)=O)CCCN(C(=O)CCCC2CCC2)CC1 31235,CCC1=NOC(CC(=O)N(CC(C)NC(=O)CCc2ccncc2Br)C)C1 31236,C(C)(CCC(=O)NC(Cc1cc[nH]n1)C(=O)NCC(c1nccs1)C)OC 31237,C1(C(CNC(CC(C)F)=O)(C)C)CCN(C(c2cnn(C)c2C(F)(F)F)=O)CC1 31238,C1(CNC(CCSCCC)=O)CCCCN(C(C2(C)CSC2)=O)C1 31239,C(CC(=O)NCCC1(C(=O)NC2CC2c2cnc[nH]2)CC1)OCC 31240,N1(C(c2cncc(SCC)n2)=O)CC(NC(c2cc(OC)nn2C)=O)CC(O)C1 31241,N1(C(CC2C(C)(C)CCCC2)=O)CC23CCCC2(C1)CN(Cc1csc(=N)[nH]1)C3 31242,N1(C(c2c(C)ncc(Br)c2)=O)CC2CCCC(C1)N2C(=O)C#CC(=O)O 31243,C(=O)(C1=CS(=O)CCC1)N1CC(O)(CCNC(C2(OC)CCCCC2)=O)C1 31244,Cc1cc(C)c(C#N)c(NC(C2CCCN2C(C2CCCN2S(C)(=O)=O)=O)C)n1 31245,c1(OC)ccc(C=CC(=O)NC2CCN(C(C3(C)CC3(F)F)=O)CC2O)cc1Cl 31246,c1(C(=O)NC2C(NC(COCCC)=O)COC2)sc([N+](=O)[O-])cc1Cl 31247,c1(C(N)=O)cccc(C(=O)NCC2CCC(CNC(C3(F)CC3C(N)=O)=O)C2)n1 31248,c1(OC)cnc(F)cc1C(=O)NCCCC(C)NC(C1CCC(F)(F)C1)=O 31249,C(C)(C)(CC(=O)NCC1CCOCC1C)N(C(CCOCCC)=O)C 31250,N1(C(C2CCC(C)(CC)O2)=O)CCC2CCN(C(=O)C(CC)(CC)OC)CC12 31251,c1(C(N2CCN(C(C3CN(C(C(C)(Cl)Cl)=O)C3)=O)CC2)=O)nccn2nccc12 31252,c1(NC(=O)NCCC2CC3CCC2C3)cc2ccc(F)cc2cn1 31253,C1(n2cc(COCC)nn2)CCN(C(=O)NC2CCCC2C(N)=O)CC1 31254,c1(C(N2C(CNC(=O)COCC3CCOC3)C=CC2)=O)nccc2cc[nH]c12 31255,c1(C(c2n(C(CC)(C)C)nnn2)NC2CC3(CC3)C2)sccc1S(N)(=O)=O 31256,c1(C(=O)Nc2cccc(-c3cccnc3)c2)cc2cncn2c(O)n1 31257,N1(C(c2c(N(C)C)nccc2)=O)CC2(CCCCN2C(C2OCCO2)=O)C1 31258,C12(NC(C(C)(C)C3CC3)=O)CC(CNC(C3(Cl)CC34CCC4)=O)(C1)OC21CCC1 31259,C1(NC(CC2(NC(c3cc(SC)oc3)=O)CC2)=O)CCCCC1CCO 31260,c1(OC)c(C(=O)NCC2(CCC(=O)N)CCC2)nc(O)nc1O.C1(=O)CN1.OC 31261,C1(C(=O)NCC(CC)NC(=O)CC2CCCO2)(OC)CCS(=O)(=O)C1 31262,N1(C(=O)NC(C2CCC3(CC3)N2C(=O)OC(C)(C)C)C)CCCc2ccccc21 31263,c1(CC(=O)NC2C(NC(Cn3c(C)ccn3)=O)COC2)ccc2cccnc2c1 31264,c1(C(=O)OC)nn(C)c(NC(C2CN(C(C3CN(C)C3)=O)CCS2)=O)c1Cl 31265,CCCCN=C(NCCOCC1(COC)CC=CC1)NC1CCS(=O)(=O)C1 31266,N1(C(Cc2nn(C)c(Cl)c2)=O)CCC2C(C1)CN2C(C1CCCNS1(=O)=O)=O 31267,C1(NC(C2N(C(c3cc(C)no3)=O)CCOC2C)=O)CCOC2(CCC2)C1 31268,Fc1cc2c(cc1F)CN(c1ccncc1S(=O)(=O)N1CCC3(CCCC3)C1)C2 31269,C1(C(=O)NCC(C)(CO)NC(c2c(OC)n(C)nc2)=O)CCN(C)C(=O)C1 31270,N1(C(C=C2CCC(C)C2)=O)CCC(F)C(NC(c2coc(CC3CC3)n2)=O)C1 31271,C(=O)(C(C)CC(C)C)N1CCC(Cc2nc(CC)on2)C1.n12cc(nn1)C2 31272,N1(C(c2c(-c3ccc(OC)cc3)scc2)=O)CCC2CN(C(=O)CC(=O)OC)CC12 31273,c1(C(N2C(C(N3CCC(CN(C)CC)C3)=O)C=CC2)=O)ncccc1Cl 31274,N1(C(=O)NC)CCC(C(=O)NCC#CCNC(c2sccc2-n2cnnn2)=O)C1 31275,CCC(CCOC)C(=O)N1CC2CC(C1)C2NC(C1CN(C)CC1C(F)(F)F)=O 31276,c1(NC(CC)=O)cccnc1C(N1CCOC(C(C)NC(=O)CCNC(C)=O)C1)=O 31277,C(=O)(CC1=CCN(C)CC1)NC(CCC)C(O)C(=O)NC1COCCC1(F)F 31278,Cc1nc(C)c(C(=O)NCC2CCOC2C(=O)Nc2ccc(C(C)C)nc2)s1 31279,CC(CC1CCCO1)C(=O)N(CCCOCCNC(c1csc(O)n1)=O)C 31280,C1(C(=O)N(CCN(C(C2(COCC)CC2)=O)C2CC2)C)CCCC(F)(F)C1 31281,C1(C(N(C(C)C(=O)N2CC(O)C2)CCC)=O)CC(OC)(OC)C1 31282,C1(CC)CCN(C(c2cc(C)on2)=O)C1CNC(c1n[nH]c(C)n1)=O 31283,C(=O)(C(C)(C)C(F)F)NC1CCC(F)(CNC(c2ccc(CC(C)C)s2)=O)C1 31284,C1(NC(c2c(OC)nn(C)c2)=O)CCN(C(=O)Cc2coc(C)n2)CC1O 31285,c1(CC(=O)NCC(CN(C(CN2CCC(C)C2)=O)C)C)ccc2[nH]ccc2c1 31286,O=C(C1=C(Cl)CCOC1)NC(CC(F)F)C(=O)NC1CC2(CCOC2)C1 31287,CCC(CNC(C1CCOC(C)C1)=O)(CC)NC(c1ccnnc1)=O 31288,C1(C(N2CCC(C(=O)NCCc3ccsc3)(CO)C2)=O)(CC)CNC(=O)C1 31289,CN1CC(F)CC1C(N1CC(OCCNC(C2CC2[N+](=O)[O-])=O)C1)=O 31290,C1(COC)(CNC(C2(C)CC(C)C2)=O)CCN(C(c2cnc(C)[nH]c2=N)=O)CC1 31291,C1(CNC(C(CC)(C)COC)=O)CC2CCC(C1)N2C(=O)C1=NOC(C)(C)C1 31292,C1(O)(CNC(c2c(CC)occ2)=O)CCCN(C(=O)C(C)(C)C2(C)CC2(F)F)C1 31293,C1(C(=O)NCC2CC3N(C(CN(C)C)=O)C(CC3)C2)CCc2c(nnn2C)C1 31294,C1(NC(c2ccnc(C(C)C)n2)=O)CC2CC1N(C(=O)Cc1nc[nH]n1)C2 31295,N1(S(CCCOCC)(=O)=O)Cc2[nH][nH]c(=NC(=O)c3cc([N+](=O)[O-])ccc3F)c2C1 31296,c1(COC(C2C(C(=O)OC(C)(C)C)CC=CC2)=O)cc2c(o1)CCCC2 31297,Cc1c(C(=O)N(CCCCNC(C2C3CC3C3CC23)=O)C)cccc1C#N 31298,C1(CNC(=O)NCc2n[nH]c(C3CC3)n2)CC(C(F)(F)F)CO1 31299,C1(CC=C)(CNC(N2CCCC2)=O)CN(C(=O)C=CCCC2CCCC2SC)C1.OC.C 31300,Cc1sc(Cl)c(C(=O)NCC2CCCN(C(=O)C=CC(C)(C)C)CC2)c1C 31301,C#Cc1cncc(C(=O)NCC(CCNC(c2ccc(CC)[nH]2)=O)OC)c1 31302,N1(C(CCC(C(C)C)NC(CC(C=C)CCC)=O)=O)CCC2(CCC(OC)C2)C1 31303,c1(NC)cccc(C(C(=O)NCC2CCCCC2)N(CC(N)=O)C)c1 31304,C(C1CN(C(C2CC(C)C2)=O)CC1C(=O)Nc1cnc(CC)nc1)=CC 31305,c1(COC(C)=O)ccc(C(=O)NC(C)(C)CCCNC(=O)CC2CCOCC2)cc1 31306,C(=O)(N=c1cc(-c2cn(C)nc2C(F)(F)F)o[nH]1)NC(C)CN1CCCC1=O 31307,c1(C(C)C)ccc(N)c(C(N2CCN(C(=O)C3=CCC3)C(C(C)C)C2)=O)c1 31308,N1(C(CSC)=O)CC(NC(=O)CN2CCC(N(C)C)CC2)CCC1C 31309,CC1CCN(C(c2sccc2S(N)(=O)=O)=O)CC1NC(=O)C(F)C1CC1 31310,Cc1cc(C(=O)NC2CC(NC(C3CCC(C(N)=O)O3)=O)C2)cc(N)c1O 31311,C(CC(CC)C(=O)N1CCCC1C(C)(C)NC(=O)CCCC1CCOCC1)=CC 31312,C12(CNC(Cc3[nH]c(=N)sc3)=O)CCC(CN(C(=O)C3=COCC3)C1)C2 31313,c1(C(CNC(=O)C(C)Cc2cnn(C)c2)NC(C(=O)NC)=O)ccccc1CO 31314,N1(C(C2(C#C)CC2)=O)CC(C2CN(C(c3cc(N)cc(F)c3)=O)C2)C1 31315,C1(C(N2CC(N(C(=O)CC3(O)CCC3)C)C2)=O)C2C3CCC(C3)C12 31316,C(=O)(CCCC(C)C)N(CC1CCN(C(C=CC=CC)=O)C1)Cc1ccoc1CC 31317,C(=O)(C(F)CCC(C)C)NC(C(=O)NCCCOCC=C)CC1CC1 31318,CC(O)C(O)CNC(=O)CCC1CCC(NC(C2(C)CSC2)=O)C1 31319,c1(C(N2CCCC(CC)(NC(=O)COC)C2)=O)cccc2c1ccn2CC(C)C 31320,C1(C)(CC)C=C(C(=O)NC(C)CCNC(c2ncc(Br)cc2N)=O)C1 31321,C(=O)(C=CS(C)=O)N(CC(=O)NC1C(OCC)COC1)CC 31322,C1(C)(C(N2CC(CNC(c3ccc(C(N)=O)nc3)=O)C(O)C2)=O)CCCS1(=O)=O 31323,N1(C(C2(C)CC2F)=O)CCC2(CC1)CCN(C(c1nncc3c1CCCC3)=O)C2 31324,C(=O)(C1=NOC2(CCC2)C1)NC1CN(C(CC2C(CC)C2(F)F)=O)CC1CO 31325,c1(C(=O)NCc2cn(CC(=O)NCC(C(C)O)O)nn2)ccc(Cl)nc1O 31326,C(=O)(CS(=O)(=O)CCOC)NCCN(C(c1cc(CCCO)on1)=O)CC 31327,CC(C)CCCC(=O)NC1COCCN(C(C2CCC(c3ccccc3)C2)=O)C1 31328,n1(CC(=O)NC(CNC(COCCC=C)=O)C2CCC2)cc(CO)nn1 31329,CC(C)C(C)(CNC(=O)CN1CC2CCC1C2)NC(=O)CN1C(=O)CNC1=O 31330,c1(CC(N2C(CNC(c3c(C)cc[nH]3)=O)CCC2)=O)ccc(C(F)(F)F)cc1Br 31331,c1(C(N2C(CNC(Cc3cc(C)on3)=O)CC(F)(F)C2)=O)noc2c1COCC2 31332,c1(C(N(CC(C)NC(=O)C(O)CSC)CC)=O)cccc(NC(N)=O)c1 31333,C(C(C(=O)NC1(CC)CCN(C(=O)C(CN(C)C)CC)CC1)C(C)(C)C)OCC=C 31334,C(=O)(CCCC(N)=O)NCC(C1CCN(C(c2cccc(N)c2)=O)CC1)(C)C 31335,CC(C(=O)NCCC1(O)CN(C(=O)CC2CCC(F)(F)CO2)C1)S(N)(=O)=O 31336,c1(CC(=O)OCC2(c3cc(O)nnc3O)CC2)cc(F)c(F)cc1Br 31337,c1(C(N2CCC(C)(NC(=O)Cc3nnc(O)s3)C2)=O)ccc(Cl)c2cccnc12 31338,CC(CCCNC(c1cc(Cl)c[nH]1)=O)NC(=O)CCOc1ccccc1 31339,Cn1nc(C(F)F)cc1S(=O)(=O)NCCc1cccc(Cl)n1 31340,C(C(=O)NCC(=O)NC1CC1)(C1CCOC1)NC1(C(=O)OC)CC1 31341,C1(CC#C)(C(=O)N(C2CC(N(C(=O)CN3CCOCC3)C)C2)CC)CCCC1 31342,C(=O)(CCC(F)(F)F)N1CC(NC(=O)CSC2CCC2)C(C(F)F)C1 31343,C(=O)(C(C)(C)C(C)(C)O)NC1C=CC(CNC(C(C)C2CCC2)=O)C1 31344,Cc1nc2ccccc2cc1CC(=O)N(C1CC2CC1N(C(=O)C(C)(C)C)C2)C 31345,c1(C(=O)NCCC2N(C(C3C(C(=O)OC)CCO3)=O)CCC2)nc(OC)c(C)s1 31346,O=C1CCC(NC(=O)CCCC2(NC(c3conc3C3CC3)=O)CCC2)C(=O)N1 31347,C(=O)(CC1OCCc2ccccc21)NC12C(CN(C(C3C(C)(C)C3(F)F)=O)C1)C2 31348,C1(C(=O)NCC(C)(CC(C)C)NC(CCC(=C)Cl)=O)CCOC2(CCOCC2)C1 31349,C1(C(=O)NCC2(CC)CCCC2)CCN(C(=O)C(C)(C)C2CCCO2)C(C)(C)C1 31350,c1(CN(C(=O)C(=O)NCC2COCCO2)CCC)ccc(OC(F)F)cc1 31351,Cc1[nH]nc(C(N2CC3C(CNC(c4occc4Cl)=O)C3C2)=O)c1F 31352,C1(C(C)O)(CO)CCN(C(c2ccc(CNC(=O)Cc3nocc3C)o2)=O)C1 31353,c1(C(C)C(=O)NC(C)(C)C)ncc(-c2ccccn2)s1.N1(CCOCCO)CC1 31354,c1(OCC)ccc(C(N2CC(F)CC2C#N)C(=O)NCCCC2CC2)c(C)c1Br 31355,C#Cc1ccc(C(=O)NCC2(C)CCC(NC(c3cc(OC)nn3C)=O)C2)cc1 31356,c1(C(N(C(C)CN(C(=O)CC2CSC2)C)C)=O)cc(=O)c2ccncc2o1 31357,c1(OC)ncc(C(=O)O)c(C)c1Br.N12CCCC1NCC2=O 31358,CC1(C)CNc2cccc(Cl)c21.c1(CN(CC)CC2CC2)cccc2cc(C3CC3)[nH]c12 31359,N1(C(c2cc(C3(C)CC3)n[nH]2)=O)CCCCC1CN(C(C1CCOC1=O)=O)C1CC1 31360,c1(CC)nnsc1C(=O)NCC1(C(N2CC(C)(F)C2)=O)CCCO1 31361,N1(C(C2CC(SC)C2)=O)CC(C2(NC(c3cnc(S)nc3)=O)CC2)C1 31362,Cc1cccn2cc(C(=O)NCC3C(O)C(O)CN3C(C3(F)CCOC3)=O)nc12 31363,c1(C(=O)NC2CC(NC(c3c(OC)nsc3OC)=O)C2)ccc(C#N)n1C 31364,N1(C(c2c(CC)c[nH]c2)=O)CCCC(COC)(NC(=O)CC2CC=CCC2)C1 31365,Cc1nc(C#N)c(N(CCC(N2CCN(C(=O)C(C)(C)C(N)=O)CC2)=O)C2CC2)o1 31366,C1(C(N2CCC(CNC(C(C)=C(CC)C)=O)C2)=O)CCc2[nH]nc(O)c2C1 31367,N#CC1CCCC1NC(=O)C(Cn1cncn1)NC(C1CC1C(F)(F)F)=O 31368,c1(C(=O)NC2CC(CNC(C(CC=C)C)=O)C2)ccc(Cl)cc1-c1ccccc1 31369,Cc1ccc(CNC(=O)C(=O)N(CCOCCC2CC2)C)c(Cl)c1 31370,C1(CCNC(C(C)C#N)=O)CCCN(C(c2conc2C2(C)COC2)=O)C1 31371,O=C1OC2CC(C(N3CCC3CNC(c3cnc4[nH]ncc4c3)=O)=O)CC2O1 31372,C(C)(CCCCNC(c1ccc(F)cn1)=O)NC(CC1N(C(C)C)CCC1)=O 31373,Cc1ccnnc1C(N1CC(CNC(=O)CNC(C2CCOCC2)=O)C(C)C1)=O 31374,c1(C(C)C)nc(NCCCn2cc(C)cn2)cc(=NC2CC3CCCCC2C3)[nH]1 31375,N1(C(CC2C(=O)NC(=N)S2)=O)CC(NC(C2CCC3(CCC3)C2)=O)CC(O)C1 31376,c1(OCC)cccc(C(C(=O)OC)NC2CCCCC2C(=O)NC2CC2)c1 31377,CCC(C(=O)NCC(O)CCNC(=O)Cc1csc(SC)n1)NC(C)=O 31378,n1(CC)nc(C(N2CCOC(CNC(=O)C(C)CCOC)C2)=O)cc1C(F)(F)F 31379,C12(NC(c3ccc(C)c(F)c3)=O)CCOCC1CN(C(=O)C1CC1)C2 31380,C(=O)(C#CC(C)(C)C)NCC(C(=O)NC1CC2CC(O)C1C2)N(C)C 31381,c1(C(N(CC(=O)NC(C)CN=[N+]=[N-])C)=O)ccncc1F 31382,Cc1ccc(F)c(C(=O)NCCC(C)NC(c2cncnc2C(C)(C)C)=O)c1Cl 31383,c1(C(=O)NCC2CCN(C(c3cc(Br)c[nH]3)=O)C2)cnc2c(Br)cccc2c1 31384,c1(NC(C2(C#C)CCN(C(=O)CC(C)SC)C2)=O)ccc2occc2c1 31385,n12cc(nn1)C(=O)C(=O)c1cc(cs1)C2.CC(C(=O)NCC(C)NC1CC1)N(C)C 31386,c1(OC)ccc(C)c(CNc2ncnc(N3CCC(C)(CN(C)C)CC3)c2C)c1 31387,c1(C(N(C2CCN(C(c3cncn3C)=O)C2)CC)=O)c2c(nn1C)CCCC2 31388,c1(C(C)=O)cc(C(=O)NCC(C2CC2)N)ccc1C.C1(C)CCCN1C1CC1 31389,C=CC(C)(C)CC(=O)NCc1n[nH]cc1C(=O)NC1C=CCCC1 31390,C1(CC(=O)NC(C2(O)CCCCC2)C(=O)N(C2CC(F)(F)C2)C)CC2CCC1C2 31391,n1(CC)nc(C(N2CC3(NC(C45CC(C)C4C5)=O)CCC2C3)=O)c2c1CCOC2 31392,c1(CNC(CCN(C(=O)Cc2ccsc2)C)=O)cncc(F)c1 31393,CCC(C)CC(=O)C(=O)N1CCCC1C(=O)NC(C)Cc1cnccn1 31394,c1(OC)ncc(NC(=O)CN2CCOCC2=O)cn1.C12CCOC1CONC2=O 31395,c1(C(=O)OC)ccc(-c2nc(Br)ccc2Cl)cc1C 31396,c1(CC)c(C(N2CC(N(C)C(c3ccc(Cl)s3)=O)C2)=O)cnn1C(CC)CC 31397,N1(C(CN2CCN(C(c3c(OCC)scc3)=O)CC2)=O)CC(C)OC2(CCC2)C1 31398,c1(C(=O)NCC(CCOCC)NC(C2(CO)CCCO2)=O)cccc2c[nH]nc12 31399,Cc1cccc(C(N2CCN(C(=O)C(O)C(C)(C)C)C(C)C2)=O)c1Br 31400,C=C(C)CCC(=O)NCC1CCOC1C1CCN(C(C2CCCN(C)C2)=O)CC1 31401,C(N=c1[nH]c(=NCc2ccc(F)cc2)[nH]c2cc[nH]c12)c1cc(C(C)C)[nH]n1 31402,CC1CN(C(C2C3(CC3)C23CC3)=O)CCC1NC(c1ccc(O)nc1)=O 31403,C(=O)(C(F)CC1(OCC)CC1)NCC(CNC(CCSCCC#C)=O)OC 31404,N1(C(CCCCSC)=O)CC2CCCN(C(=O)CCc3cc(C)[nH]n3)C2C1 31405,C=CCCCCCCCCC(O)Cn1cc(CCO)nn1.C(=O)C=CC=CC 31406,c1(CN(C2CN(C(c3ccc(I)c(F)c3)=O)C2)C)cc(Cl)c(O)cc1F 31407,C1(CC)(CNC(C2(CNC(=O)CC3OCCCO3)CC(C)(C)C2)=O)CCC(=O)N1 31408,C(N=c1[nH]c2cc(F)ccc2o1)C1(CNC(c2cc(Br)n3ccccc23)=O)CC1 31409,Cc1cc2ccnc(OC(=O)C(F)C3CCOC3)c2cc1C 31410,C1(C(=O)OCC)(NC(c2cn(C)nc2C)=O)CCS(=O)(=O)C1 31411,N1(C(Cc2cncc(C)c2)=O)CCC2CN(C(CCS(=O)(=O)N(C)C)=O)CC2C1 31412,C(=O)(C(F)(CNC(=O)Cn1ccnc1)C(C)C)NC(C#C)C(C)OC 31413,c1(Sc2ccc(C=CCc3n(CC)ccn3)cc2)ccc2c(c1)OC(F)(F)O2 31414,CC(CC(C)(C)O)NC(C1CCN1C(=O)C=CCF)=O 31415,Cc1nn(C)c(NC(=O)C(n2cc(CCCCCCO)nn2)C)c1C=O 31416,N1(C(C(C(C)O)C)=O)C2CCC1CC(CNC(c1cc(C3CC3)ncn1)=O)C2 31417,C1(C(=O)NC(CCC)CO)Cc2nccnc2CN1C(=O)Cc1ccc(F)cc1 31418,CCC(C)C(O)C(C)C(=O)N1CCC(CCC(=O)NCCSCCOC)C1 31419,c1(C(=O)NC2CCN(C(CN(CCOC)C)=O)C2C)ccnc2[nH]c(C)nc12 31420,C12(CNC(CCc3cnc(C)o3)=O)CCC(CC1)CN2C(=O)CC1CCOC1 31421,C(=O)(CC(F)(F)C(F)F)NC1C(NC(CC(n2c(C)cc(C)n2)C)=O)COC1 31422,C(=O)(C(C(C)(C)C)OC)NCCC1(NC(c2cc(CC(C)C)[nH]n2)=O)CCC1 31423,C(=O)(C(C)(F)C(=O)N(C)CCOCCCN(C(=O)CC1CCCN(C)C1)C)OC 31424,c1(CC)noc(C)c1NC(=O)NCC1(c2ccc(C(F)(F)F)nc2)CC1 31425,C(=O)(CCCCNC(c1occc1COC)=O)NCC(C#C)CC 31426,C=CC1CN(C(=O)C(CCC)OCC)CC1NC(=O)Cc1ccc(O)nc1 31427,Cc1cccc(C(C)C)c1C(=O)NCCC1COCCN1C(C1CCCS1)=O 31428,N1(C(c2c(CC=C)cccc2)=O)CC(C)CCC1CNC(=O)CNC(C)=O 31429,c1(C(=O)NCC(CCOC)NC(c2cnc(SC)s2)=O)ccn(C)c(=O)c1 31430,c1(CCC)noc2ncc(C(N3CCC(NC(=O)C(C)=C4CCC4)C3C)=O)cc12 31431,c1(C(C(=O)NCCOC)N(C(C)COC)CC=C)ncn(C)n1 31432,c1(C(C)NC(C(=O)N(CC(C)(C)CN(C)C)C(C)C)=O)ccc(C(F)F)o1 31433,C1(CC)C=CCCN1C(=O)CCC1(C)CCCN1C(=O)COCCCOC 31434,c1(OC)cc(C(=O)NC2CCCN(C(=O)CC(C)F)C2)c2ccccc2n1 31435,c1(CC)cc(C(=O)NCC2(F)CC(NC(=O)CC3CCCCO3)C2)n(C)n1 31436,c1(SCC(=O)NCC2N(C(CC(C=C)C)=O)CC=C2)ccccc1[N+](=O)[O-] 31437,C1(NC(CC(CC)OC)=O)COC2CN(C(=O)Cc3ccc(F)c(F)c3)CC12 31438,C(=O)(CC1=CSC2=NCCN12)N1C(C)CN(C(C23CC(CO2)C3)=O)CC1 31439,C1(C(=O)NC2C(NC(=O)COC3CC(F)(F)C3)CCCC2)CCC(F)(F)CC1 31440,CCCCC(C(=O)NC1(CCOC)CC=CC1)NC(=O)C(O)CC(C)C 31441,N1(C(c2c(C)cns2)=O)CC=CC(CNC(=O)CCCNS(C)(=O)=O)C1 31442,C1(CC=C)(NC(=O)CC2CSCCS2)CC2CCC(C1)N2C(=O)C(C1CCC1)OC 31443,C1(CNC(c2cn(C)nc2C2CC2)=O)CCN(C(=O)C(C)(C)OC(F)F)CCC1 31444,c1(CN=C(NCC(O)C(O)c2ccccc2)NC2CCC2)ccc2c(c1)CCO2 31445,c1(COC)cccc(C(=O)NCC2CCC(F)(CNC(=O)CC3CCCO3)C2)c1 31446,N1(C(C2CN(C(Cc3c(C)nn(C)c3C)=O)CC(F)C2)=O)CCOC2(CCC2)C1 31447,c1(C(=O)NC2C(CNC(=O)COC(F)F)C2)cc2ccc(Br)cn2n1 31448,c1(SCC(N2CC(O)(NC(c3cnc(OC4CC4)s3)=O)C2)=O)ccccn1 31449,c1(C(N(C)CC2COCCN2C(C2CC(C#N)C2)=O)=O)cnc(S(C)(=O)=O)s1 31450,N1(C(C2C(C(C)C)C2)=O)CCCC(C)(NC(=O)CCCc2ccc(Cl)cc2)C1 31451,Cc1cc(CC(=O)NC2CC2CNC(c2cccc(O)c2C)=O)ccc1Br 31452,C1(C(N(CC#C)CCF)=O)C(NC(=O)CCC2CC(OC)C2)C1(C)C 31453,C=CCCN=C(NCC1(CCOC)CCC1)NC1CCCC(OCC(F)(F)F)C1 31454,N1(C(C(c2cnccn2)C)=O)CCc2[nH]nc(CNC(=O)C=CBr)c2C1 31455,c1(C(C)(C)C)ccc(C(=O)NC2(CNC(C3CCCOC3)=O)CCC2)[nH]1 31456,N1(C(c2c(F)cn(C)n2)=O)Cc2ccccc2CC1C(=O)Nc1cccc(CF)c1 31457,c1(C(=O)NCC(C)N(C)C(c2cc(C3CCC3)no2)=O)ccc(C(C)(C)C)[nH]1 31458,c1(C(=O)NCCOC2CC(NC(CC(C)C(F)F)=O)C2)cc(N)cc2ccccc12 31459,N1(C(c2ccc(C)c(F)n2)=O)CC2CCN(C(=O)CC3CC4CCC3C4)C(C2)C1 31460,c1(C(=O)NC2(CCC#C)CC2)c(CC)c2ccccc2[nH]1 31461,CC(CC(=O)N1CCCOC(CNC(C2CC(F)(F)C2)=O)C1)C(F)F 31462,CC1(C)CC(CNC(c2ccco2)=O)CN1C(c1ccccc1C1CCCC1)=O 31463,C1(NC(C2CCC(NC(CSCCCC)=O)C2)=O)CCN(C)C1(C)C 31464,c1(OCC)ccccc1C=CC(=O)NC(C)CC(C)NC(c1coc(C(C)=O)c1)=O 31465,C(=O)(C(CNC(=O)CC1CCC(=O)NC1)C(C)(C)C)N1CC(CN(C)C)C1 31466,c1(CCC2(C(N3CC(OCCNC(C4CCCO4)=O)C3)=O)CC2)ccccc1 31467,C1(C(N2CC3CC3(NCC(SC)Sc3ccccc3)C2)=O)CCC(F)(F)CC1 31468,c1(C(C)=O)ccc(C(N2CCCC2C(C)(C)NC(=O)CCC2CCOC2)=O)o1 31469,N1(C(c2cnccn2)C(=O)NCCSC)Cc2cc(Cl)c(Cl)cc2C1 31470,c1(C(=O)Nc2scc(CC(N3CCC(CO)C3)=O)n2)nc2ccccn2n1 31471,CC(C)CC(C(=O)NCC1(O)CC(O)C1)N(C)C(C1CCC1Cl)=O 31472,N1(C(C=CC(CC)C)=O)CCn2nc(CNC(=O)C=Cc3ccnn3C)cc2C1 31473,C1(O)(CNC(C2CC2Cl)=O)CCCN(C(c2cccn2CCN2CCCC2)=O)C1 31474,N1(C(CC)=O)CCCCC1C(=O)NC1C=CCN(C(C2CCC2(F)F)=O)C1 31475,c1(CN)cccnc1N.Cc1occc1COC(F)F 31476,C(CCC(C)(C)NC(=O)C(=Cc1cn(C)nn1)F)NC(C(n1c(C)ncc1)C)=O 31477,C1(C(N2CCOC(C(C)NC(=O)CN3CCCC3=O)C2)=O)(COC)CC=CCC1 31478,C1(C(=O)NCCCOC(=N)O)C2CCC(C2)C1NC(=O)CCCn1nccn1 31479,CC1(C)CN(C(=O)CCC(C)NC(c2csc(F)c2)=O)C2COCC12 31480,CC(C)CC(F)C(=O)NC12CCC1CN(C(c1cccc(OCC(F)F)n1)=O)C2 31481,N1(C(C(C)OC2COC2)=O)CCC2(CC1)CN(C(C1C3CCC(C3)C1(C)C)=O)C2 31482,c1(C(=O)NCc2c(C(N(C)Cc3cccnc3)=O)cccc2)cc(N)c(Cl)cn1 31483,c1(C(=O)N(CCN(C)C)CC2CC2CF)ccc(-c2cccc(O)n2)cc1 31484,c1(C(=O)NCC(CC=C)NC(c2cnn3cnnc3c2)=O)ncc2[nH]ncc2n1 31485,C1(NC(C(CSC)O)=O)CC12CC(NC(c1cnn(C)c1)=O)C2 31486,CC1(F)CCCN(C(C2CCOCCN2C(=O)Cc2ccc3c(c2)CC3)=O)C1 31487,C(=O)(C(C#N)C(C)(C)C)N1CCC(N2CCN(C(CN(C3CC3)CC)=O)CC2)C1 31488,C1(C(=O)NC(C2(O)CCC2)C)CCOCC1NC(=O)C(C)(F)c1ccon1 31489,Cn1cnc2ccsc2c1=NCC1CCCN1C(c1cc(Cl)c[nH]1)=O 31490,Cc1[nH]nc(C(N2CC3CC3(C(N3CCN(C(=O)C(C)C)CC3)=O)C2)=O)c1O 31491,Cc1nc(N(CCCNC(c2cc(C3CC3)nn2C)=O)C)c(C)c(C)n1 31492,N1(C(C(C(=O)OC)C)=O)CCC(CNC(=O)C(=Cc2ccccc2Cl)C)CC1C 31493,c1(CC(=O)OCC2CCSC2)cccc(NC(c2cnco2)=O)c1 31494,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NCCN(C(=O)CC(C)CF)CCOC 31495,c1(C(=O)NCC#CCC)[nH]c(NC(=O)CC2(OC)CC2)c(C)c1C(=O)OC 31496,N1(C(c2cc(C)on2)=O)CCC2(CC1)CN(C(c1cccc3c1OC(C)C3)=O)C2 31497,c1(C(N(CCOC)CCNC(c2cc3sccc3s2)=O)=O)c2ccccc2nn1C 31498,C=C(CNC(=O)C(F)C(C)CNC(=O)C=Cc1ccco1)C1CCOCC1 31499,c1(C(N2C(CNC(C3N(C)CC(C)(C)C3)=O)CC2)=O)ccc2c(O)nc(S)nc2c1 31500,C1(NC(C(C)OCC(C)C)=O)CCCCCN(C(=O)CCCC2CCCCC2)C1 31501,c1(-n2cc(CCCOC)nn2)ccnc(F)c1C(=O)O.C12CN(CCO1)C(=O)C2 31502,N1(C(C(N2C(=O)CCC2=O)CC)=O)CCC(c2cn(CC(C)(C)C)nn2)CC1C 31503,c1(OC)cc(C(=O)NCCCN2CCN(C(c3ccc(C)s3)C)CC2)ccn1 31504,N1(CC#C)CCN(C(C2CCN(C(C3CC(=O)N(CC)C3)=O)C2C)=O)CC1=O 31505,CN1CC2CC1CN2C(=O)CCC(=O)Nc1ccc(COc2cccnc2)cc1 31506,C(=O)(C1OCCn2ccnc21)NCCNC(c1cc(CC2CCCC2)on1)=O 31507,N1(C(COCCC=C)=O)CCC(NC(c2nn(CC)cc2Cl)=O)C(F)C1 31508,C1(CNC(C2(C)CC2)=O)CCC2CN(C(=O)Cn3c(F)cccc3=O)CCC2C1 31509,c1(C(=O)OC)cccc2nc(C(=O)N(C)CC3SCCS3)cn12 31510,Cc1cnc(F)cc1C(N1CCN(C(=O)CCC[N+](=O)[O-])C(C)C1)=O 31511,C1(C(N2CCCC(OCCC)C2)=O)CCC2(CC2)N1C(=O)CC1(CSC)CC1 31512,c1(CNC(CONC(c2cnn(C)n2)=O)=O)ccccc1O 31513,C(=O)(C#CC(C)(C)O)NC(C1CC1C(=O)NCC(c1ccnn1C)O)C 31514,C(COC1C=CCC1)(C(=O)OC(c1ccccc1)C)OC(C)=O 31515,C1(NC(CCCCSC)=O)CCC2CN(C(=O)Cn3nccc3N)CC2C1 31516,Cc1ccc(F)c(C(=O)N(CCCCNC(C2(C)C=CCCC2)=O)C)c1Cl 31517,N1(C(c2cc(OCC)n[nH]2)=O)CC(C(=O)NCC(C)(C)COC)C(F)(F)C1 31518,c1(C(=O)NC(C2(O)CN(C(CC(C)OC)=O)C2)C)ccnc(C2CC2)n1 31519,C(=O)(C1CCCc2cc(O)ccc21)N(C1CCN(C(C2CCNC2)=O)C1)CC 31520,c1(C(c2cn(CC(N3CC(CN4CCCCC4)C3)=O)nn2)N(C)C)ccc(Br)cc1 31521,C12CCCCCN1C2=O.N1(CC)CCN(C(C2CCCN2C(C)=O)=O)CC1 31522,C(=O)(CC1=CCCCC1)Nc1ccc(CC2CN(C(CC(CC)SC)=O)C2)nc1Cl 31523,O=C(C1CCCc2nn[nH]c21)N1CCC(OC2CN(Cc3ccns3)C2)CC1 31524,C(=O)(C(COC)N=[N+]=[N-])N(CCC(=O)NC1CC2(C1)CC2CO)CC#C 31525,C12(C(N3C(C)(CNC(CC4N(CC)C(=O)CC4)=O)CCC3)=O)CCC(C)(C1)OC2 31526,C1(O)(CC(C)NC(CCC)=O)CCN(C(=O)CN2CCC(O)CC2)CC1 31527,C1(NC(C2NC(=O)OC2)=O)CCCN(C(=O)Cc2nc[nH]n2)C1 31528,O=C(CC(O)CNC(c1csnn1)=O)NCC1CCN(C2CC2)C1 31529,C(=O)(C(C)(O)C(F)(F)F)OCCOC1CN(C2(C)CCC2)C1 31530,C(C)(CCC(=O)N(CC(=O)NCc1ncc[nH]1)C)NC(C(C)C)=O 31531,N1(C(Cc2cc(C)sc2C)=O)CCCC(CO)(CNC(C2OCCC2(C)C)=O)C1 31532,Cc1ccc(F)c(C(C(=O)NC2COC2)N(C)CCc2cccs2)c1 31533,N1(C(CC2(C=C)CC2)=O)CCCC2(CCN(C(=O)CN3CCSCC3)C2)C1 31534,C(=O)(CC1C(=O)Nc2ccccc21)N1CCC(C(=O)NCC(COC)(C)O)CC1 31535,C1(CC(=O)NC(C(C)(C)C)CNC(=O)Cc2cc[nH]n2)CCCC2(CC2)C1 31536,c1(C(=O)NC2C(C)CN(C(=O)C=Cc3ccccc3)C2)c2c(c[nH]c1=N)CCC2 31537,N1(C(CCC#C)=O)CC(C(=O)N(c2ncccc2C)CC#C)CC(F)C1 31538,C1(CC#C)(C(=O)NC2CC2CNC(=O)C#CC2CC2)CCCCC1 31539,c1(C(=O)NCC2C(C)CCN(C(c3c(CC)ncs3)=O)C2)cnc([N+](=O)[O-])cc1C 31540,N1(C(CC(C=C)(C)O)=O)CC(C2CN(C(=O)CCC3CCC(=O)N3)C2)C1 31541,C1(NC(c2cc(C)nn2C)=O)CCSC12CN(C(c1ccc(N)cc1O)=O)C2 31542,C12CN(CC1(C)C)C2C.c1(C(=O)OCC)nn(C)nc1Br 31543,C1(N(C(=O)Cc2csc(C(C)CC)n2)CCC)CCN(C(C23CCC2C3)=O)CC1.OC 31544,N(C(=NCCc1ccc(F)cc1)NCCSC1CN(CC)CC1SC)CC=C 31545,c1(CC(=O)NC2(CO)CN(C(CC(CC)C3CC3)=O)C2)cnc2ncccn12 31546,C1(C(=O)NCC(C)NC(C2(c3cccnc3)CC2)=O)CCc2nnc(O)cc2C1 31547,c1(C(N2CCC(C)C2CNC(C23CC4CC2C3C4)=O)=O)cccc(O)c1Cl 31548,C1(C(N2CC3C(NC(c4ccncc4Cl)=O)C(C3)C2)=O)COc2ccccc2O1 31549,N1(C(C(CC)NC(N)=O)=O)CCN(C(=O)CCc2ccc(Cl)nc2)CC1CC 31550,N1(CC(=O)N(CC(O)CO)C(C)C)CCN(C(c2cnncc2C)=O)CC1 31551,CCC(CN(C)C)CC(=O)NCC1C(C(=O)NCCCC2(O)CC2)C1(C)C 31552,C1(C(=O)NC2CCC(CNC(C3(C)CC3C)=O)CC2)(NC(C)=O)CCCCC1 31553,N1(C(C(CC)C#N)=O)CC(C(=O)NCC2(O)CCN(C)C2)CC(C)C1 31554,c1(C(N2CC(NC(C3CC(O)C3)=O)C3(CC3)C2)=O)cc2c(F)c(Cl)ccc2[nH]1 31555,C12(NC(CCCC(=O)N(C)C)=O)CCCC1(F)CN(C(C1CCC(O)CC1)=O)C2 31556,C1(C(=O)NC(N)=O)CCN(C(=O)CC)C1(C)C.c1(SCC)ccc(N)cc1 31557,c1(C(N2C3CCN(C(C(C)CN)=O)C3CC2)=O)ccc2c(c1)NCCC2 31558,c1(C(=O)NCC23C(CN(C(c4n(C=C)ncc4)=O)C2)C3)cnc(O)c(OC)c1 31559,C1(C(N(CC(=O)NC2CC(CC(N)=O)C2)CCOC)=O)C(C)C1C 31560,N1(C(C)C)CC(C(N2CC(c3cc(CNC(C4SCCS4)=O)no3)C2)=O)CCC1 31561,CCC(O)C(C)C(=O)N(C1CCCCC1NC(=O)CCC1CCCO1)CC 31562,c1(C(=O)OC(c2ncc(Br)cn2)C)cc(Cl)c(N)c([N+](=O)[O-])c1 31563,c1(C(C(C2CCOCC2)C)NCCSC(F)(F)F)nnnn1C1CCCCC1 31564,N1(C(C2(C)CCCCO2)=O)CCOC2(C1)CN(C(=O)Cn1ccnn1)C2 31565,C1(CCC(=O)N(CC(C)N(C)C(C2CSC2)=O)C)CC(C)(C)CO1 31566,C(C)(C(=O)N1CCCC(CC(=O)NCc2ccoc2)C1)(C(C)C)OC 31567,C1(C(N2CC(COC)(NC(=O)CC3C=NN(C)C3=O)C2)=O)CC1C1CCCCC1 31568,Cc1oc(-c2ccccc2)nc1C(=O)NC1CC(NC(C2CC(C)OC2=O)=O)C1 31569,Cn1nc(CNC(=O)C(C)(C)NC(C2CCCCN2C)=O)n(C)c1=O 31570,N1(C(C(C)C2(O)CCC2)=O)CC=CC1CNC(C1(Sc2ccccc2)CC1)=O 31571,Cn1cc(CC(=O)NC2COCC2NC(=O)Cc2cnns2)cn1 31572,CC1CN(C(=O)Cc2cc[nH]n2)CC2(CCN(C(C3(O)CCCCC3)=O)C2)O1 31573,C(=O)(C(F)C(F)(F)F)NCC1(F)CC(NC(c2nnc(S)nc2O)=O)C1 31574,C12(NC(=O)CSCc3ccccc3)CCCC1N(C(=O)COc1cn[nH]c1)CC2 31575,C(CC1=CCN(C(=O)Cc2cccc(F)c2)CC1)NC(C(=O)NC(C)C)=O 31576,C(CCCC(=O)NC(C)CCC(C)C)NC(C(COCC)C)=O 31577,c1(N2CCC(N(CCC)C(C3CCCC3(F)F)=O)C2)cc(CC)ncn1 31578,c1(C(=O)NCC2CCC(NC(C3(CCCC)CC3)=O)C2)[nH]nc2ncnc(O)c12 31579,C12(NC(C(C)CF)=O)CCCC1N(C(=O)COCCc1cccs1)CCC2 31580,C(=O)(CCCCC(C)(C)C)NC1COC2CN(C(COCCCCCC)=O)CC21 31581,Cc1ccc(SC(C)C(=O)NC2CCCC2NC(c2csnc2C)=O)cc1 31582,C=C(C)C(CC(=O)N(C(C)C(=O)NN)C1CC1)OC(c1c[nH]ccc1=O)C 31583,c1(C(=O)NC(CNC(Cn2c(C)cc(C)n2)=O)(C)CO)c(C)c(Cl)cc(C)c1N 31584,C1(NC(CC)=O)CCC(C(N2CCOC(C(c3nc[nH]n3)OC)C2)=O)CC1 31585,C(C(=O)N(CC(C)C)C(C)C)(C(C)C)NCCCNC(C(CC)C)=O 31586,c1(C(=O)NC(CC=C)CNC(c2c(C)ncn2O)=O)cc(Cl)ccc1OC 31587,C(=O)(CC(C(F)F)NC(c1ccnc(C)n1)=O)NCCOCCC=C 31588,C1(C(N(CCCCCC)CC(=O)OC)=O)CC=CCC1C.C12C=CC(C1)C(=O)N2 31589,N1(C(Cc2cnc(C)o2)=O)CC2CC(NC(c3ccc(C(C)(C)C)o3)=O)CC1C2 31590,CC1CCCn2ncc(C(=O)NCCNC(C3CC4C=CC3C4)=O)c21 31591,Cc1cccn2c(C(=O)NC3(C)CC(NC(=O)C(F)CC4CC4)C3)cnc12 31592,C12(NC(CC3(COC)CCC3)=O)CC1CN(C(c1ccsc1OC)=O)C2 31593,C1(CNC(c2cnc(OC)nc2)=O)CC2(CC2)CN1C(=O)CC1CC(F)C1 31594,Cc1oc2ccccc2c1C(N1CCCOCC1)C(=O)NC1CCOCC1 31595,N1(C(C(C=CC)O)=O)CCN(CC(=O)NCCC2(C)N=N2)CC1 31596,CP1(=O)CCN(CCNC(=O)NCCNc2cccnc2O)CC1 31597,N1(NC(C2CCN(CC(C)C)C2)CCO)CCN(c2ccccc2O)CC1 31598,c1(C=O)c(C)nc(C2CCCC2)nc1O.Cc1cc(Cl)c(C(=O)NC2(C)CC2)s1 31599,c1(C(N2CCCC(NC(C3(OC)CCOCC3)=O)C2)=O)[nH]c(=N)ccc1C 31600,CC1CN(C(C2(CC3CC3)CC2)=O)CC(C)N(C(=O)C(C)Cc2cnc[nH]2)C1 31601,C1(CNC(C(N2CCN(C)CC2)C)=O)CN(C(=O)CC2CCN(C)C2)CCO1 31602,C1(C(N2CCSCC2)=O)(CC)CCCN1C(=O)Cn1cnnc1O 31603,c1(CC)cc(Br)cc(C(=O)NC2CCN(C(=O)Cc3nc[nH]n3)CC2F)c1N 31604,Cc1c(C(N2CCC(C)(C(=O)OC)C2)C(=O)NCC2CCCO2)cccc1Cl 31605,CC12CCOC(C(=O)NCCCCNC(=O)C(=O)Nc3cnn[nH]3)(C1)C2 31606,C1(CC)CN(C(=O)CCN(C(c2nonc2CC)=O)C2CC2)CC1O 31607,c1(C(C)C)cn(C)nc1C(=O)NCCN(C(C1CCC1C)=O)CC1CC1 31608,c12ccc3c(c1)C(=NC1CC2=CC=C(F)C=C1O)NC(N(CC(C)C#N)C)=N3.CO 31609,c1(C(N(CC(CNC(Cc2c(C#C)cccc2)=O)O)C)=O)cc2cccnc2o1 31610,c1(NC(C)=O)cccc(OCC(=O)NC2CC2NC(=O)Cc2cc[nH]c2)c1 31611,C(=O)(CC(O)CC(C)(C)C)NCC(CNC(CCCc1ccc(C)c(C)c1)=O)O 31612,c1(C(N(C)Cc2c(CNC(C3C(C)CCO3)=O)cccc2)=O)c(Cl)cncc1Cl 31613,c1(C(N(C)CCOCCNC(=O)CC2(C)CCCC2)=O)c(F)ccc2n[nH]cc12 31614,C1(C(=O)NCCCCCNC(=O)CC2COC3CC2C3)CCCCC(F)(F)C1 31615,Cc1cc([N+](=O)[O-])cnc1N1CC2CCN(C(c3cnc(C4CC4)o3)=O)CC2C1 31616,C1(N(C(C(C2CCCC2)NC(C)=O)=O)C)CCN(C(c2ccc(C(F)F)s2)=O)C1 31617,c1(CONC(C2(CC=C)CN(C(=O)C(C)C#N)C2)=O)sc(C)cc1C 31618,Cc1cc(C#N)cnc1C(=O)NC1(C)CCCN(C(c2cncn(C)c2=O)=O)C1 31619,C12(C(=O)NC3CCN(C(c4cncc(N)c4)=O)CC3)CCOC1CC(=O)NC2 31620,N1(C(COC2CCN(C(CC3CCCN(C)C3)=O)C2)=O)CC2CC2C2CC12 31621,C1(C(=O)NCC2C3CN(C(Cn4c(N)cc(C)n4)=O)CC32)CN(C)CCN(C)C1 31622,C1(NC(C2CC(C)NC(=O)C2)=O)CN(C(=O)CC2CC(F)(F)C2)CC12CCCC2 31623,C(=O)(C1(C)c2ccccc2-c2ccccc21)N1CCC(CNC(C(C)SC)=O)C1 31624,C#CCCCC(=O)N(C1CN(C(C2CN(C3CCCCC3)C2)=O)C1)C 31625,c1(C(N(C2CN(C(C(C)OC)=O)C2)C)=O)c(NC(C)=O)c[nH]c1C 31626,c1(NC(N(C2CN(C(=O)CC3CCC(=O)NC3=O)C2)C)=O)cc(O)cc(C#N)c1 31627,CC1CN(N(Cc2ccc(F)cc2Cl)Cc2ccn(C3CCCC3)n2)CC1F 31628,N1(C(C(COCC)C)=O)CCC(C)C(CC(N2CC(F)(F)CC2CO)=O)C1 31629,CCC(CNC(=O)C=CCF)(CC)C(=O)N(C1CC1(C)C)C 31630,CCCC(CC)CC(=O)N1CC(N(C(=O)CSCc2cccnc2)C)C2(CC2)C1 31631,C1(CC)CN(C(C2(NC(=O)CCC3CCOC3)CCCCC2)=O)CCCO1 31632,C(C(C)C)(C(O)C(=O)N1CCOCC1CC(=O)NC1(CF)CC1)OC 31633,CCC(CC)C(C)C(=O)N1CC(NC(=O)Cc2cc(F)ccc2OC)CC(F)C1 31634,C1(N(C(=O)C(CO)NC(N)=O)C)CCN(C(=O)C(C)(C)n2cnnn2)CC1F 31635,C(COC)(C(=O)NC1(CCCC(=O)N(CC(CO)C)C)CCC1)NC(=O)OC.C.OC 31636,C#Cc1ccc(C(=O)NCC(O)CCNC(=O)C(C)(CC)C(=O)OCC)c(C)c1 31637,CCC(C)(C(=O)NCC1CCN(C(C23CCC(O)(CC2)CC3)=O)C(C)C1)C(N)=O 31638,Cc1ccc(CC(N2CCN(C(=O)CCS(N)(=O)=O)CC2C(F)F)=O)cc1Cl 31639,N1(C(C(C)CC2CCCCC2)=O)CCC(O)C(NC(=O)C=CC2CC2)C1 31640,C(C(C)(F)CNC(c1nsnc1O)=O)NC(COCC(=C)C)=O 31641,C12(C(C)(C)C)CCC(C(=O)NC3CN(C(C4CCC(O)C4)=O)CC3F)(CC1)CO2 31642,C1(CC(=O)NCC(=O)NCC)N(C(c2cc(C)[nH]c2C)=O)CCC1(C)C 31643,Cc1cnc(F)cc1C(=O)NC(C1CCCN(c2ncnc(Cl)c2Br)C1)C 31644,c1(C(=O)NC(C2CCOC2)CNC(c2ccc(C)nc2)=O)c[nH]cc(F)c1=O 31645,C(=O)(CC1=CCCCC1)N1CC(CC(=O)NCC2(C)CCC(C)CC2)OCCC1 31646,c1(C(N(C)CC2CN(C(=O)C=C(Cl)Cl)CC23CC3)=O)c[nH]c2ncccc12 31647,c1(C(C)NC2(c3nnnn3C3(C)CC3)CC(COCC(C)(C)C)C2)cccc(Cl)c1 31648,CCC(C(=O)OC)C(=O)NCc1cnn(C)c1C(=O)NCC1CCN(C(N)=O)C1 31649,Cc1ncc(N)cc1C(N1CC(C2(NC(c3ccnnc3Cl)=O)CC2)C1)=O 31650,C1(C(N2CCC(CC=C)C2)=O)N(C(C2COCCO2)=O)CCC1(C)C 31651,CCC(CC)CC(=O)N1CC(C(O)C(=O)Nc2c[nH]nc2C)C1 31652,Cc1cc(C(=O)NC2CCC(CNC(C3CCCOC3)=O)C2)ccc1O 31653,C1(NS(CC)(=O)=O)CCCN(c2nnc(-c3nn(C)cc3Br)n2C2CC2C)C1 31654,c1(OC)cccc(NC(C2(O)CCN(C(c3ccc(O)c(F)c3)=O)C2)=O)c1C 31655,N1(C(C23CC(NC(c4c(CCC)nco4)=O)(C2)C3)=O)CCC(O)CC12CC2 31656,CCC(O)CC(=O)N1CCCCC1OC(C1CCOC1)=O.C12CN(C1)C2=O 31657,N1(C(C2(CF)CC(=C)C2)=O)CCN(C(c2cccn3ncnc23)=O)CC(C)(C)C1 31658,c1(CC(=O)NC23CCC(C2)N(C(=O)C(F)n2ccnc2)C3)cc(F)cc(F)c1 31659,N1(C(C(=O)OCC)=O)CC(F)(F)CC1C(=O)NCc1nn(CC)nc1Br 31660,C1(CCN(C(=O)COC(c2ccccn2)=O)C)CCCCN1C(=O)C(C)(C)C 31661,CCC(CC)C(=O)N1CC(C(=O)NCCNC(C2CCNC(=O)C2)=O)C1 31662,N1(C(c2n(C)ccc2)=O)CCC(OC2CN(C(C3(C#N)CCC3)=O)C2)CC1 31663,c1(CC)nc(C)c(CNC(=O)C(C)N(C(=O)C(C)C(=O)OC)CC)o1 31664,c1(CC)ccc(CNC(C2CN(C(=O)C3=C(Cl)CCC3)CCN2C)=O)cc1C 31665,N1(C(C=CCCC)=O)CCC(O)(C(C)NC(c2snnc2COC)=O)CC1 31666,C(=O)(C(F)C(C)(F)F)NCCCCCCNC(CCC(=O)N(C)C)=O 31667,N1(C(c2nc(C(=O)OCC)oc2)=O)CC(NC(=O)COC2CCOC2)C(C)C1 31668,C1(C(=O)NCC(C)(C(C)C)NC(CCCOCC)=O)CC2(C1)CC(C)C2 31669,C1(C(N(C(C)C)CCN(C(=O)CCCN(C)C)C)=O)CCCC(C)C1 31670,C1(C(=O)NCC2CCC=CCC2)CN(C(=O)CCc2ccccc2)C2(CCC2)C1 31671,c1(OCC)cc(C(=O)N(CC(O)CN(C(=O)CCc2cc[nH]n2)C)C)on1 31672,N1(C(CCCCC#C)=O)CC(C)CN(c2cc(=O)n(C)c(O)n2)C(C)C1 31673,C1(NC(C(C)N(C)CC)=O)CCN(C(c2cnc(C(C)C)nc2)=O)C1C(C)C 31674,c1(C(=O)NCC2CCN(C(C3CC(OC)C3)=O)CC2C)csc(=NC2CC2)[nH]1 31675,C1(CC(=O)NCCOCCCC)CCN(C(c2cc(C(C)C)[nH]n2)=O)CC1 31676,C1(NC(=O)CN2CCOC2=O)CC(C2CCN(C(=O)COC3CCCC3)C2)C1 31677,Cc1ccn(C)c1C(=O)NC1CC(O)(CNC(=O)Cc2cnc[nH]2)C1 31678,Cc1cccnc1CN(CC(=O)O)C(c1cncc(NC)c1)=O.C12COCCN1C2=O 31679,N1(C(C(=O)Nc2ccc(C(=O)OC)cc2)C2COC2)CCC2(CCC(O)C2)C1 31680,C(=O)(C1CCc2c(Cl)cccc21)NC(C)CNC(c1ccc([N+](=O)[O-])s1)=O 31681,c1(C(=O)NC2(C)CCN(C(C3CCC(COC)C3)=O)C2)cc(C#N)cc(C)n1 31682,C1(NC(c2ccc(C)nc2O)=O)CC2(C1)CC2N=c1[nH]c2ccc(Br)cc2s1 31683,C1(CNC(C(C)O)=O)CN(C(C2(CC(F)F)CCC2)=O)CCN1C 31684,CCCCC(C(=O)NC1CCSCC1)NC(=O)C=CCCC(C)C 31685,C1(NC(C2CC2CF)=O)CC2CC1N(C(=O)Cn1ccccc1=O)C2 31686,CC1N(C(c2cccc(CNC(=O)Cc3ccc(O)cn3)n2)=O)CCOC1(C)C 31687,c1(C(=O)NCCC(C)NC(=O)C(CO)N(C)C)cc(Cl)ccc1[N+](=O)[O-] 31688,C1(C(=O)NCC(CNC(C2(COC)CCCCO2)=O)(C)F)CCCC1S(C)(=O)=O 31689,C1(C(=O)NC(C(=O)NC)C(C)C)CC12CCN(C(=O)C(O)C(F)(F)F)C2 31690,N1(C(=O)NC(C)(C)C)CC2CC(NC(=O)Nc3cccc(OC(F)F)c3)C(C2)C1 31691,CCC(C#N)C(=O)N1CC(NC(=O)C(C)c2cccs2)C1 31692,N1(C(CCC=C(C)C)=O)CC(F)(F)CC1C(=O)NCc1ccc(C)o1 31693,c1(C(N2CC(NC(C3C(OC)C3)=O)C(O)C2)=O)sc2sccc2c1Cl 31694,c1(NC(C2CCC(CNc3ccc(-n4ccnc4)cn3)C2)=O)ccc(Br)cn1 31695,C(C)(C(CC(=O)NCc1ccc(C#N)s1)NC(C1CCC(C)(C)C1)=O)OC 31696,C(=O)(C(C)(C)C(=O)NCC)NC(CNC(C=CC(CC)=CC)=O)CCOC 31697,n1(CC)cc(Oc2ccc3ccc(=NCC)[nH]c3c2)c(=O)c2cc(Cl)ccc12 31698,c1(C(=O)NCCCN(C(c2n[nH]cc2CC)=O)CC)nccc2ccn(C)c12 31699,c1(N(CCNC(=O)COCC)C(C2CCC(O)CN2C)=O)ccc(C)c(C)c1 31700,CC(C)CC(F)(F)C(=O)Nc1cn(CCN2C(=O)C3CCCOC23C(C)C)nn1 31701,C(CCCCC(=O)Nc1cncc(C(N2CCCC2CC(C)O)=O)c1)SC 31702,C1(NC(CCCC#CC)=O)CCN(C(=O)CC2CCCCO2)C12CCC2 31703,c1(C(=O)NCCNC(C2CC(CCF)C2)=O)ccc(C2CC2)cc1 31704,CC1CCN(C(c2ccnc(-n3ccnc3)c2)=O)C1CNC(=O)C=C(Cl)Cl 31705,C(CC(C(=O)NCc1ncc(C(N2CCC(C)(C(N)=O)C2)=O)cn1)OC)OC 31706,C(COC)(CC(=O)N1CCC(CC(C)(C)C)C1)NC(C1(COCC)CCCC1)=O 31707,Cc1ccncc1C(=O)NCC(CO)NC(=O)CCOc1ccccc1OC 31708,c1(C(N2CCC(C)(NC(C(C)NS(CC)(=O)=O)=O)C2)=O)ccc2c(c1O)CCC2 31709,C1(CN(C)C)CN(c2ccc(Cl)cc2)CCC1(C)C.C12CCN(CC1)CC(=O)N2 31710,N1(C(c2c(C)ocn2)=O)CC(C(=O)NC2CCCC(O)C2)CC1(C)C 31711,C1(OC)=NC=C(NC)[SH](CC(=O)NC(C)COCCCNC(=O)COC(F)F)C1 31712,c1(CN(C)C(C2CCCN(C(=O)C(c3ccc(F)cc3)O)C2)=O)cccnc1Cl 31713,O=S(=O)(C1CCCCC1)NCCN1C(CC(=O)Oc2cccnc2)CCC1 31714,CC(C)CC(O)CC(=O)N1CCCCCC1C(N1CC(N(C)C)C1)=O 31715,c1(C(=O)NCC(=C)CCNC(C2CCS2(=O)=O)=O)cccc2c1NC(=O)CC2 31716,C1(NC(C=CC(=O)OCC)=O)CCCCCC1C(=O)Nc1cc(C)ccc1OC 31717,C(=O)(C1OC(=O)c2ccccc21)N1CCC2(C(NC(c3c(C)occ3)=O)C2)CC1 31718,C1(C(N(C2CCN(C(C3CN(S(C)(=O)=O)C3)=O)CC2)CC#C)=O)CCCCCC1 31719,CC(C)CC(C(=O)NOC(c1ccc(Cl)cc1)C1CCCCC1)N(C)C 31720,CC(C)C(O)C(=O)NC1(c2ccc(F)cc2)CCN(C(=O)C2=CCOC2)C1 31721,C1(CCCCCNC(C2C(C=C)C2)=O)CCN(C(=O)CC2CCC(=O)N2)CC1 31722,C(CS(=O)(=O)C(N)=O)N(C(CN1CC(CNC(C2CC23CCC3)=O)C1)=O)CCO 31723,c1(C(=O)NC2(C)CCN(C(C3C(CC)C3)=O)C2)n[nH]c2ccc(C(F)(F)F)cc12 31724,c1(C(C)C)cccc(C(=O)NCCN(C(=O)Cc2nnn(C(C)(C)C)n2)C)n1 31725,CCC(CCCC(=O)NCc1ccnc(O)c1)NC(C1CC(N(C)CC)C1)=O 31726,CC1CNC(=O)CN1C(C1CC12CCN(C(=O)CN1CC3CC3C1)C2)=O 31727,N1(C(CC(COC)(C)C)=O)CC2CC(O)C1C2NC(=O)CCC1CCCO1 31728,N1(C(=O)CO)CCC(C2(NC(c3cccc(C4CCC4)c3)=O)CC2)CC1 31729,Cc1nsc(CCNC(=O)NCC(F)(F)C(F)F)c1N 31730,c1(C(=O)NCCN2CCN(C(CC=CC)=O)CC2)cccc2c1OCCC2CCO 31731,N1(C(Cc2ccc(C)s2)=O)CCC2C(C1)CN2C(=O)Cn1cc([N+](=O)[O-])nc1C 31732,C=C(Cl)C(C)(C)C(=O)NCC1(NC(=O)C(C)OCC(C)C)CCCCCC1 31733,CC(CC(F)(F)F)C(=O)N1CCC(C(=O)NCc2cc(O)ns2)C12CCC2 31734,C1(NC(C(C)NC(C(=O)NC(C)C)=O)=O)C2Cc3cc(Br)ccc3C12 31735,c1(CCC)cnnc(C(=O)NC2CCC2NC(=O)CCC(C)C)c1 31736,c1(C(CN(CCS(C)(=O)=O)CC)=O)cc2cccnn2c1 31737,N1(C(C(C(CC)C)O)=O)CCCC12CCCN(C(=O)C(C)CN)CC2 31738,C1(CC)(NC(=O)CCN2CCC(F)(F)C2)CCCN(C(=O)C(C)C2(O)CCC2)C1 31739,C12(CNC(C3C(C)C3)=O)CCCC1CN(C(C13CCC(C(N)=O)(CC1)CC3)=O)C2 31740,C1(CNC(=O)COCC2CC2)CC(NC(C2(CCF)CCC2)=O)C1 31741,CCC(C)(CC)CN=c1nc(N2CC(F)CC(F)C2)c2cc(F)cc(F)c2[nH]1 31742,N1(C(CN2CCN(C(c3cc(Cl)c[nH]3)=O)CC2)=O)CC(C(F)(F)F)OC(CF)C1 31743,C(C(F)(C(=O)NCc1ocnc1CC)C(C)C)NC(C(C=C)(C)O)=O 31744,C(=O)(C(O)CCC)N(C1(CC(=O)NC2C(C)C2)CCC1)C.N(C)N(C)C 31745,C(=O)(C1COc2ccccc21)NCC1CN(C(CCC#CC)=O)C2C(O1)COC2 31746,N1(C(C2C(C)(C)C(NC(=O)Cc3ccns3)C2)=O)CCC2(CC1)CC2C#N 31747,N1(C(CCOC)=O)CCC(C2CCC2)(CNC(=O)CC=C(Cl)Cl)CC1 31748,C1(C)(C(=O)NC2(CNC(C(COC)(C)C)=O)CCCCCC2)CC(C)OC(C)C1 31749,C1(NC(=O)Cc2coc(C3CCCC3)n2)CC(O)CN(C(=O)C2=NOCC2)C1 31750,CCC(C)CCCC(=O)N1CC(CNC(=O)CCc2cccn2C)CC1(C)C 31751,c1(CC)cc(NC(C2(F)CCN(C(c3cc(Br)ccc3F)=O)CC2)=O)ccc1F 31752,C(C1CN(C(=O)C(C)C2CCC2)CC1C(=O)NC(C)C(F)(F)F)=CC 31753,c1(N(C)CC2CC2)nc(N2CCCC(Cc3ccncn3)CC2)c2c(n1)CSC2 31754,C(=O)(C1CCN1)NCc1c(C)csc1.C1(NC(N)=O)CCCC1.C12(CC1)C(=O)N2 31755,N1(c2nc(C)cc(OCC)n2)Cc2nccn2CC(NC(c2coc(C)c2)=O)C1 31756,Cc1ccc(O)c(C(N2CC(O)CCC2C(=O)NCCOCCN=[N+]=[N-])=O)c1.C1(N)CC1 31757,c1(C(=O)NC(CNC(c2c(C)ccnc2)=O)(C)C(C)C)onc2c1CCCC2 31758,S(=O)(=O)(c1ccc(Br)cc1NCC1(CCOCC)CC1)NCCC(C=C)(C)C 31759,c1(CC)noc(C)c1C(=O)NCCCN(C(C1CC1C1CC1)=O)CC 31760,C(=O)(C=C1SCC(=O)N1C)NCC(CN(C(c1cc(C)cc(C)n1)=O)C)(C)C 31761,Cc1nc2cc(C(=O)NCC3CN(C(C4CCOC4)=O)CC3C)cc(Br)c2o1 31762,Cc1noc(CNC(=O)NC2CCC(C)(C)C2)c1[N+](=O)[O-] 31763,Cc1cc(C(N2CCN(CC(C)(C)NC(=O)CC3CNC(=O)C3)CC2)=O)oc1C 31764,N1(C(c2c(C)cc(CC)o2)=O)CC2(CCN(C(c3c(C)cnn3C(C)C)=O)C2)C1 31765,C(=O)(C(C)(C)C(F)(F)F)NC1CCCN(C(Cc2cccc(OCC)n2)=O)C1C 31766,C(=O)(C1(C)COC(=O)NC1)OC.c1(NC(C)(C)C)cc(C(=O)O)ncc1Br 31767,C(=O)(C(C(C)CC)C1CC1)N(CCNC(C1(CCCC)CCCC1)=O)C 31768,C1(NC(c2sc(CCC)c(CC)c2)=O)CCC(C)N(C(=O)Cc2ccc(C)s2)C1 31769,C1(CNC(c2c(C)cco2)=O)CCCN(C(=O)CCc2c(C)noc2Cl)C1 31770,N1(C(Cc2c(C#C)cccc2)=O)CCN(C(=O)CCC2CCCCC2)C(C)C1C 31771,CCC(CCCC(=O)NC1CC(F)(F)C1(C)C)NC(=O)CC(C)n1cccc1 31772,c1(C(=O)NCCCN(C(=O)CC2CCN(C)C2=O)CC)cc(OC)c(Cl)s1 31773,N1(C(c2ncccn2)=O)CC2CCN(C(C3Cc4ccncc4C3)=O)C2C1 31774,CC1(C)COCCC1C(N1CC2CC(NC(c3cnoc3C3CCC3)=O)C2C1)=O 31775,c1(C(N2C(CNC(CCOCC(C)C)=O)CC3(CC3)C2)=O)nsc2ccccc12 31776,c1(C(=O)OC)ccc(CC(=O)NC2CCCC2CNC(c2sccc2Cl)=O)cc1F 31777,n1(CC)nncc1C(=O)N(CCC(C)NC(C12CC(CO)(C1)C2)=O)C 31778,C1(CC)CCC(NC(=O)C(Cn2ccnn2)NC(=O)C(C2CCOCC2)C)CC1 31779,c1(CC(=O)N(C2CN(C(CC(C)c3cnn(C)c3)=O)C2)C)ccc(C#N)nc1 31780,c1(CN2CCC(N(C)C(c3c(I)ccnc3Cl)=O)C2)cc(F)ccc1[N+](=O)[O-] 31781,c1(C(C2C3CCCCCC23)ONC(C2C(C)(C)OC(=O)C2)=O)cc[nH]c2nccc1-2 31782,Cc1cccnc1C(=O)NCC1(C(=O)NCC(c2ncc[nH]2)C)CC2(CC2)C1 31783,n1(C(C)C)ncc(F)c1C(=O)NC1CCCC1CNC(=O)CCc1cnn(C)c1 31784,C1(CNC(CCN(C(=O)COC)CC#C)=O)CC2CC1CC2O.c1(N)nc[nH]n1 31785,C(=O)(CC1OCc2ccccc21)NCC(=O)NC1CC(c2ccncc2)=NO1 31786,Cc1cnc2n1CCC(C(=O)NCCN(C)C)C2.C(=O)(C(F)=CC1CC1)C=O 31787,N1(C(C23OCC(C)(C2)C3)=O)CC=C(CNC(c2ccc(=N)[nH]n2)=O)CC1 31788,N1(C(CNCCS(CC)=O)=O)CCN(C(c2ccccc2)=O)C2(CCC2)C1 31789,C1(NC(C(C)NS(C)(=O)=O)=O)CC2CCC(C1C)N2C(C12CC(CO1)C2)=O 31790,c1(C(c2cnc(C3CC3)o2)=O)cc(Cl)nnc1N1CCCC1 31791,CC1CCC(CCNC(=O)C(N2CCCCC2)C2CCCCC2)O1 31792,CC(CC(=O)N1CC(NC(C23CCC(C2)C3(C)C)=O)C1)CC(C)(C)C 31793,c1(CC(=O)N(C(CCNC(C(COC)COC)=O)C)C)cnn2ccccc12 31794,C1(OCCCNC(C(C)c2cccs2)=O)CCN(C(c2c[nH]ccc2=O)=O)CC1 31795,CCCC(C)(O)C(=O)NCC(C)(C)CNC(c1ccnc(Cn2cnnc2)c1)=O 31796,N1(C(CN2C(=O)CCC2=O)=O)CCC2CCCC12C(N1CCC2C(CO)C12)=O 31797,C(=O)(C(C)(C)C(N)=O)N1CCC(CCN(C)Cc2nc(O)n[nH]2)CC1 31798,C1(CC(N2CC(C)(NC(=O)CCCc3ncco3)C2)=O)CCCCC1O 31799,N1(C(c2cncc(N)c2)=O)CCC(C2CC2)(CNC(c2ocnc2C(F)F)=O)C1 31800,CC(C)CCCC(C)C(=O)NCCOC1CCN(C(=O)C(C2CCCO2)C)CC1 31801,c1(C(=O)NCC2CCN(C(C(CC)O)=O)CC2)cc(Br)cc2[nH]ccc12 31802,Cc1ncccc1CC(=O)N(C1CC(NC(=O)CC2COC(C)(C)C2)C1)C 31803,C1(OCC(N2CCN(C3CC(C)OC3=O)CC2)=O)CCC(F)(F)CC1 31804,C(CC(CC)C(=O)N1CCC(CCC(N2CC=C(C)CC2)=O)CC1)=CC 31805,Cn1cc(CNC(=O)NC2CC3CC(NC(=O)OC(C)(C)C)CC23)c(O)nc1=O 31806,c1(CC(C)NC(=O)NC2CC(C)(Nc3ccc[n+]([O-])c3)C2)cnc2n1CCCC2 31807,c1(C(N2CC3CN(C(c4nc(OC)oc4)=O)C3CC2)=O)[nH]cc2c1CCS2(=O)=O 31808,CC(=O)C(C)(C)CC(=O)N1CC=CC1(C)C(=O)N(C1CC(C)(C)C1)C 31809,N1(C(CC2(N(C)C)CCCC2)=O)CC2CC1CC2NC(c1ccc(F)c(O)c1)=O 31810,c1(C(=O)NC(C(NOCCCOC)=O)c2ccnn2C)ccc(C#N)c(C)n1 31811,c1(C(=O)NCC2C3CN(C(Cc4c(C)cccc4)C)CC32)ccn2cncc2c1 31812,C1(NC(C2C(C(=O)OC)CC2)=O)C2CCN(C(=O)C(C)(C)COC(C)C)C12 31813,c1(C(=O)NC2C=CCN(C(C3(C=C)CCCCC3)=O)C2)cn2c(C)nnc2cn1 31814,N1(C(CNS(C)(=O)=O)=O)CCCC1CCNC(=O)NCCO.C(N)=O 31815,Cc1ccnc(C(=O)NCC(C)(C)CCNC(=O)C(N2CCOCC2)C2CC2)c1 31816,N1(C(COC(CC)C)=O)CCC(CC(C)NC(c2scnc2C2CC2)=O)CC1 31817,c1(C(N2CC(NC(CCC(=C)Cl)=O)C(C)(C)C2)=O)cc(N)c(N)cc1F 31818,C1(NC(c2cscn2)=O)COC2(CCCN(C(=O)C=Cc3cncnc3O)C2)C1 31819,c1(OC)ccc(O)cc1C=O.N12CCOCC1c1n[nH]c(n1)NC(=O)C1N2CC1 31820,C1(C(=O)NC(C(=O)N(CCC(=O)OC)C)c2cccs2)CCC(=O)N1 31821,C1(CC)(COC(=O)C(Cc2ccccc2)N(C(C2CCCC2)=O)C(C)C)CCCC1 31822,C(CC(C(=O)NC1(C)CC1)NC(=O)C=CC1CCCN1C)N(C)C 31823,c1(SC)ccc(C(=O)NC(c2ccccc2)CNC(C2CCOC2=O)=O)o1 31824,N1(C(C(C)OC)=O)CC2CN(C(=O)C(C3CCCCC3)C)CC2(C)C1 31825,CC1CC(CNC(C2(C(F)F)CC2(F)F)=O)=NO1 31826,c1(C(N2CCC3(CCOC3)C2)=O)ncnn2ccc(Br)c12.C12(CCC1)CC(=O)N2 31827,CC(CN(C)C)CCC(=O)N1CC2CC(C1)C2NC(C1CC2CC1C1CC21)=O 31828,c1(CSCC(=O)NC(C)CCCNC(=O)C(C)(C)F)ccc2ccccc2c1 31829,Cc1cn2c(n1)CC(C(=O)NC1CC1CNC(c1ccnc(C)c1)=O)CC2 31830,C(=O)(C(O)CNC(N)=O)NCC1(CN(C(=O)Cn2cnnn2)C)CC1 31831,c1(C(C(=O)OC)=O)ccc(CCC2CCN(C(C3N(C(C)=O)CCC3)=O)C2)s1 31832,C1(NC(N(C2CC2(C)C)C)=O)COCCC1C1CCN(c2nccnc2Br)CC1 31833,C(=O)(C(C)S(=O)(=O)C(C)C)NCC(C1CCC1)NC(c1cc(C)ns1)=O 31834,Cc1cc(C(=O)NCC(C)CNC(=O)C(F)(F)C2CC2)c2cccnc2c1C 31835,C(=O)(CCCCN1CCCC1)N(CCCNC(CCC=C)=O)CC1CCCC1 31836,c1(C(=O)NC2CN(C(C3N(CC)CC3)=O)C(C)CC2)cc(OC)cc2c1OCC2 31837,C(=O)(CC(F)(F)C(F)F)NC(C1(C(=O)NCC(CC=C)CO)CC1)C 31838,C1(C(N2CC(CCNC(C3CC(C)(F)C3)=O)C2)=O)CCN(CC(F)(F)F)CC1 31839,C(=O)(C(C)CC(F)(F)F)NCCCC(C)NC(C1CC(N2CCCC2)C1)=O 31840,N1(Cc2cn(C)nc2)C(C(=O)NC2(c3ncc(Br)cn3)CC2)CC2CC12 31841,C#Cc1cncc(C(=O)NCCC2CCC(NC(c3ccc(C)c(C)n3)=O)C2)c1 31842,C1(C(=O)NCCN(C(=O)C(O)c2cnc[nH]2)C2CC2)CCC(OC(F)(F)F)CC1 31843,C1(c2cn(C(CC=C)CC)nn2)COCCN(C(=O)CCCCCOC)C1 31844,C1(CC(=O)NC2(C(=O)NOCCCCCSC3CC3)C(C)C2)CC2CCC1C2 31845,C1(NC(C2CC(=C)C2)=O)CCCCC12CCN(C(c1cnc3cccnn13)=O)CC2 31846,N1(C(C=CC=CC)=O)CCC=C(C(=O)NCC2(OCC)CCCCC2C)C1 31847,c1(C(=O)NC(C(C)NC(C(COC)C)=O)CO)c(C)ccc(Cl)c1N 31848,c1(C2C(=O)NC(C)CCCN2C)ccc(CC2CC2)cc1F.C1CC1.SC 31849,C1(CC(=O)NCC(C)CNC(c2cc(Cl)c(Cl)[nH]2)=O)CCCC(F)(F)C1 31850,CCC1=NOC(CC(=O)NC2CCCC2NC(c2cnc(CC(C)CCC)[nH]2)=O)C1 31851,c1(C(=O)OC(C)(C)C)cccc(Nc2ccccc2-n2cc(CCCO)nn2)c1 31852,N1(C(COCCC(C)C)=O)CC(C2CN(C(=O)CN3CCCCCC3)C2)C1 31853,CCC(CC(C)C)C(=O)NC(CNC(c1cn(Cc2cccs2)nn1)=O)C1CC1 31854,C1(C(N2CC(C(N3CCC(COC)C3)=O)(CC)C2)=O)COCC(C)O1 31855,c1(C(=O)NC2C3CN(C(C4C(C)=CCS4)=O)CC2C3)cc2cccc(C)c2o1 31856,c1(NC(C2CCC(CNC(C3(O)CCC3)=O)O2)=O)cncc(F)c1 31857,C(CCCCNC(=O)CCC1CCC1)N(C)C(C1SCCS1)=O 31858,CC1(C)CCC(NC(=O)C=CCC2(NC(=O)CC3CC4C=CC3C4)CCC2)CC1 31859,C=CCN=C(NCc1nnc(CO)s1)N1CCC(OC(C)(C)C)C1 31860,C1(=O)C(CCC(C)C)N1.C#CC(C(C)OC)NC(=O)C=C(C)C(C)(C)C 31861,n1(CC(N2C3(CNC(=O)COCC4CC4)CC(C2)C3)=O)cc(Br)c(O)nc1=O 31862,n1(CC)nc(C(=O)NC(C)CCCNC(=O)CCn2cc(C)cn2)cc1C 31863,Cc1oc(C(F)(F)F)nc1C(=O)NCC(O)CNC(=O)C=Cc1ccncn1 31864,c1(C(N2CCSCC2C(c2ccccc2)O)=O)cnc2c[nH]nc2c1 31865,C1(NC(c2cc[nH]n2)=O)CCC2CCN(C(=O)C#CC3CCCCO3)C1C2 31866,C(C)(CN=c1cc(C)c(C#N)c[nH]1)NC(C(CC(C)C)OC)=O 31867,C(=O)(C1CCCc2scnc21)NCC1CN(C(CCCCC(=O)NC)=O)CC1C 31868,CCCCCC(C)CC(=O)N1CC(C2CN(C(c3nccn4nccc34)=O)C2)C1 31869,C(=O)(CC1=CCCC1)NC1CCN(Cc2c(CN3C(=O)OCC3)cccc2)C1 31870,C(=O)(CC(C)C(=O)NC1C=CC(CC(=O)N(C2CC2C2CC2)C)C1)OCC 31871,C1(COC)CC2(CCN2C(c2cccc3cncn23)C(=O)NCC2CC2)C1(C)C 31872,C1(CNC(C2(C)CC(=C)C2)=O)CC(C(C)C)CCN1C(=O)C(C)Cn1ccnc1 31873,c1(CC)ccc(C(=O)NCC2(NC(C3CCC(C)S3)=O)CCCCC2)c(C)c1 31874,c1(C(CNC(C2C(C)C2)=O)NC(c2cccc(C3CC3)c2)=O)cccc(Cl)c1 31875,C1(C(=O)Nc2ncc(Br)nc2I)CC(F)CN(Cc2cc(-c3ccco3)no2)C1 31876,C1(NC(=O)CC2(N3CCCC3)CC2)C(C(=O)NCCSCCC=C)C1(C)C 31877,CC1CN(C(c2cnncc2O)=O)CC1(C)CNC(=O)C1=CCCC1 31878,c1(OCC(=O)NC2CC(Cn3cc(CC(CC(C)C)O)nn3)C2)ccc(F)cc1F 31879,C(=O)(CCC(=O)N(CCSC1CC1)C)NC1CCN(C(COCC)=O)C1 31880,N1(C(Cc2c(C)n[nH]c2C)=O)CCN(C(=O)CC2(O)CCOCC2)C(CO)C1 31881,N1(C(c2ncc(C)cn2)=O)CC2CCC1C(CNC(c1ccc(F)c(Cl)c1)=O)C2 31882,N1(C(C2(CC3CC3)CC2)=O)CC2(C1)CN(C(C1CC(F)(F)C1(F)F)=O)CCO2 31883,C(=O)(C(C)CC(C)C)NCc1cccc(C(N(C)Cc2nc(C)on2)=O)n1 31884,CN1C(=O)CC(CN2CC(CCS(C)(=O)=O)C2)C1=O.C1(=O)CCN1 31885,c1(C(N2CCC(C(C)NC(=O)C3=CCCC3)C2)=O)ccc2c(c1)nc(CO)n2C 31886,C=CCCCCCC(=O)N1CCCC1(C(=O)NCC12CCC(OC)C1C2)C(C)C 31887,c1(C(=O)NCC2(F)CC(NC(C3(C)CCOC3)=O)C2)ccc(S(C)(=O)=O)s1 31888,c1(CC(N2C(CNC(c3cc(CC)oc3C)=O)CCC2)=O)c(OC)cccc1F 31889,C(=O)(CCCCCN(C)C(C1CNC(=O)N1)=O)N1CCC(CSC)C1 31890,N1(C(C(CCCC)O)=O)Cc2ccccc2CC1CNC(=O)COCC(F)(F)F 31891,c1(C(C)=O)ccc(Cl)cc1NC(C1CCCN(Cc2ccc(Br)[nH]2)C1)=O 31892,c1(C(c2ccccc2)N(CCOC)C)ncccc1S(=O)(=O)NC1CNC1 31893,Cc1ccn(CC(C)(O)C(=O)NCC=CCNC(=O)Cn2ccc(C)n2)c(=O)c1 31894,CC1CCc2[nH]nc(C(=O)NC34CCCC3CN(C(=O)CCC=CBr)C4)c2C1 31895,N1(C(c2n(CC=C)ccn2)=O)CC=CC(NC(=O)C=CS(C)=O)C1 31896,C1(CNC(c2c(CNC(C(CC)SC)=O)cccn2)=O)CC(C2CCC2)C1 31897,C1(NC(c2cc(C)ncn2)=O)CC2(C1)CC(C(N1CCN(C(C)C)CC1)=O)C2 31898,c1(OC)ccc(F)c(F)c1CN1CCOC(C(=O)Nc2ccc(C#N)cc2O)C1 31899,C12(CCCC1)C(=O)N2.C(C(C)(C)NC(=O)CC1CC(CF)C1)N(C(C)=O)C 31900,c1(C(=O)NCCOc2ccc(C)cc2)ccc(C#N)cc1.C=C1CC2(C1)C(=O)N2 31901,Cc1cc(C(N2CCCC(CO)(NC(=O)CC3CN(C)C3)C2)=O)c(O)nn1 31902,C(c1ccncc1)=C(C)C(=O)NCC#CCNC(C1CCCCC1C)=O 31903,c1(C(=O)NC(CNC(c2c(OC)cccn2)=O)CO)ncnc2c1ccn2C 31904,C1(CNC(c2c(CC=C)cccc2)=O)CCN(C(C2CC(F)CN2C)=O)C12CC2 31905,C(CCF)(C(=O)NCC(F)F)NC(C(C)OCC=C)=O 31906,CC1CN(C(C2(n3cnnn3)CC2)=O)CC(C)C1NC(=O)C=Cc1cnn(C)c1 31907,Cc1csc2nc(CC(N3CC(NC(C4(C(N)=O)CC4)=O)CCC3C)=O)cn12 31908,C1(C(=O)NC2CC(CNC(C(c3ccncc3)C)=O)C2)COCCN1C 31909,c1(OC)ccc2nc(C(N3CCOCC3C3CC3)C(=O)NCC(C)C)ccc2c1 31910,N1(C(CC(=C)C)=O)CC(NC(c2ccnnc2O)=O)CC(F)C1 31911,c1(SC2C(CC(C(=O)OC)COC3CCC(=O)C3)C2)ccc(OS(C)(=O)=O)cc1 31912,C1(C(N2CC(C)(CCC(=O)NCc3ccc(F)cc3)C2)=O)C2CCC(F)C12 31913,c1(COC(=O)CO)[nH]c2ccccc2c1NC(=O)Cc1ccc(CCOC)cc1 31914,C(=O)(C1=CC2C=CC1C2)N(CCCCCNC(=O)CCC1CCCOC1)C 31915,N1(C(c2ccc(C(N)=O)o2)=O)CC2(CC(NC(=O)CCc3csnn3)C2)C1 31916,C12(C(=O)NCc3ccc(C)cc3C)C3CCC(CC13)C2(F)F 31917,c1(-c2nc(Cc3c(OCC)noc3C)n(CCCC)n2)ccc2ncsc2c1 31918,c1(CNC(COCC=C)=O)ccc(C(=O)NCCCC2CCCO2)o1 31919,C1(C)(CC)C=C(C(=O)N2CC3CC3(CNC(c3cnc(C4CC4)s3)=O)C2)C1 31920,C(CCCN1CCC(O)CC1)(C(=O)O)NC(CSc1c(CC)cccc1)=O 31921,C1(CC)CC(C(=O)NC(C)(C)CCF)CCN1C(c1cc(CCO)on1)=O 31922,CCCCCS(=O)(=O)CC(=O)NCC(C)NC(=O)C#CC1CCCCC1 31923,c1(C(=O)NCCC2CSCCN2C(=O)CCN2CCOCC2)ncc[nH]c1=O 31924,C1(NC(CCCC)=O)COC2(C1)CN(C(=O)Cc1c[nH]c(=N)nc1O)C2 31925,C(=O)(C(CNC(=O)C(F)C1CCC1)CC(C)C)NC(C#C)(C)C1CCCC1 31926,CC1(CCNC(=O)CC2CCC(=O)O2)CCN(C(c2cnoc2C2CCC2)=O)C1 31927,C(C(CC(F)(F)F)NC(c1cnc(O)o1)=O)NC(CCC1CCC(=O)NC1)=O 31928,N1(C(CN(C(c2ccoc2C(F)(F)F)=O)CC)=O)CCCC(C(C)N(C)C)C1 31929,c1(CC)c(C(=O)NCC2(F)CC(NC(c3cc(N)ccc3C)=O)C2)cccc1C 31930,N1(C(C)C(=O)NC2CCCC2C(=O)NC2(CO)CC2)CCCCC1=O 31931,c1(C(N(C)CC2(NC(c3c(CC)nccc3)=O)CC2)=O)cc(O)ccc1C 31932,N1(C(C2=C(C)CCC2)=O)CC(NC(=O)COCCCF)C(C2CC2)C1 31933,c1(C(C(=O)O)NC(CCNC(c2c(Br)sc(C)c2C)=O)=O)cc(F)c(O)c(F)c1 31934,c1(C(c2n(CCCCCC)nnn2)NCc2cccs2)cnc(C2CCC2)nc1 31935,c1(C(N2CCCC(CNC(C(CCC)C)=O)C2)=O)ccc(Br)cc1C(C)=O 31936,CC1(C)OCCOC1CC(=O)NCC1CC(NC(c2cncn2C(F)(F)F)=O)C1 31937,CCC(C)(C)CCCC(=O)NC1C(C)CN(C(c2cnn(CC)c2C)=O)CC1C 31938,CC(C)(CCCNC(=O)C(O)CC1CCCC1)C(=O)NCC1(C2(O)CCC2)CC1 31939,C(CN=S(C)(C)=O)NC(CC1CCN(C(c2c(OC)csc2)=O)C1)=O 31940,CN1CCC(C2(C(=O)NC3CC4CC(NC(=O)C(C)(C)CC#N)CC4C3)CC2)C1 31941,C1(C(=O)OC)CCCN(C(=O)Cn2cnnc2)C1C.C1(CC)CCCN1 31942,C#Cc1cccc(C(N2CCSCC2C(=O)N(C)C(C)C2CC2)=O)c1 31943,C(=O)(C1=C(C)NC2=NCCCC2=C1)N(CCNC(=O)CC1(C)CCCCC1)CC 31944,CCC(CNC(C1(CO)CCCCO1)=O)N=c1[nH]nc(C2CC2)s1 31945,N1(C(C2CN(C(C(F)=C(C)C)=O)CC2(F)F)=O)CCN2CCOCC2C1 31946,c1(CC(=O)N(C2CN(C(c3nonc3N)=O)CC2F)C)cncnc1O 31947,C(=O)(CC(O)CC1CC1)NC(CNC(CCSCC(C)C)=O)C(C)C 31948,c1(CC)ccc(C(=O)NC2CN(C(=O)CSC(F)(F)F)CC2CC(C)(C)C)cn1 31949,c1(N2CCC(C)(CO)C2)ccc(S(=O)(=O)NC2(CO)CCC2)cc1Br 31950,C1(C(=O)NCC23CC2CN(C(=O)C(F)Cc2ccccc2)C3)C2CCCCCC12 31951,c1(OC)cc(C)c(C(N2CCC(NC(=O)CCOC(C)=O)CC2C)=O)cc1OC 31952,C1(C(N2CCC(CNC(=O)CCC=CBr)C2)=O)(CO)CCCCO1 31953,n1(CCS(C)(=O)=O)ccc(=NC(=O)C2COC(C)(C)C2)[nH]1 31954,c1(C(=O)NCC(C)N(C(C(C)C(N2CCCCC2)=O)=O)C)[nH]ccc1C1CC1 31955,c1(C(C(=O)NCCCCN(C(C(C2CCCC2)SC)=O)C)F)ccccc1 31956,CC(=O)CCCC(C)C(=O)N1CC(C)CC1C(=O)NCC(C)OC(F)F 31957,C(=O)(C(C(C)C)n1cncn1)N(CC(CNC(C(CC)n1cncn1)=O)(C)C)C 31958,C(=O)(C(O)CC(C)(C)C)NC(CCCNC(c1c(C)n(CC(C)C)nc1)=O)(C)C 31959,c1(NC(C2CN(C(c3ccccc3O)=O)CCC2O)=O)ccc(F)c([N+](=O)[O-])c1 31960,C1(C(=O)NCCCCNC(c2ccc(C(C)C)cc2)=O)CCCCC(F)(F)C1 31961,N1(C(c2ncn(CC)c2)=O)CCC(C)C(N(C)C(c2ncc(OC)cn2)=O)C1 31962,C1(O)(CC(=O)NC2C(OC3CC3)CN(C(CNC(=O)NC)=O)C2)COC(C)(C)C1 31963,C1(C(=O)NC2CCN(c3ccc([N+](=O)[O-])cc3)C2)CCCC2(C1)CC2(F)F 31964,CCCCC(O)C(=O)NCCC(C)NC(=O)C(=O)NCC(F)(F)F 31965,C(C(C)(C)CNC(=O)CCc1ccnn1-c1ccccc1)NC(CSCC=C)=O 31966,c1(C(N(CC(CNC(c2n(C=C)ncc2)=O)C)C)=O)ccc(C(C)=O)nc1C 31967,c1(NC(C)=O)ccc(CNC(=O)NCC(C)(C)C(F)F)c(F)c1 31968,C(C)(CCCNC(=O)C(F)(F)c1nccs1)NC(C(C)NC(C)=O)=O 31969,C12(C(=O)NC(CCCCC)C)CCC(CN(C(=O)CC3(CSC)CC3)C1)C2 31970,Cc1c(C=CC(=O)N(C)CC2CCCN2C(C2CCOCC2)=O)cnn1C 31971,Nc1ccc(-c2cn(CCCNC(c3cnc(C4CC4)o3)=O)nn2)nc1 31972,C1(C(=O)NCC2CC3(CCC3)C2)CC(O)CN1Cc1nc(Br)sc1Br 31973,C(=O)(CCC(=O)NCCN(C(=O)C(Cl)=CCl)CC1CC1)N(C(C)C)C 31974,CCC(CC)(CC)C(=O)NC1CC2CC1N(C(C1CC1c1ccccc1Cl)=O)C2 31975,c1(C(=O)NCC2CCC(C#C)CC2)c(Cl)cc(C(F)(F)F)cc1Br 31976,Cc1ccncc1C1CC1C(=O)OCF.N12CCCCC1COC2=O.C(C)(C)(C)O 31977,CC(C)(O)C(C)(C)C(=O)NCC1(CNC(C2CCCO2)=O)CCC1 31978,c1(C(=O)NCCCC(C)NC(=O)C(C)CF)cncc(C(=O)OC(C)(C)C)c1 31979,C1(C(N(CCCCC=C)C)=O)CC2CCC1N(C(c1cc(C(C)(C)C)on1)=O)C2 31980,C1(C(F)F)(CNC(C2CC=C(C)CC2)=O)CCN(C(c2ccccn2)=O)CC1 31981,C1(SCC(=O)NCCN(C(c2cn(C(F)(F)F)cn2)=O)C2CC2)CCOC1=O 31982,c1(CN2CCC(NC(c3cc(Cl)ccc3Cl)=O)C(O)C2)cncc2ccccc12 31983,C1(NC(C(CC(C)C)N(C)C)=O)COC2(C1)CN(C(=O)Cc1ccncc1Cl)C2 31984,CC1P(C)(C)(O)CN(C(=O)NC(C2CCCO2)CO)C1 31985,C1(CCNC(=O)Cn2cccc2)CCCN(C(c2sc(Cl)cc2Cl)=O)C1 31986,c1(C(N2CC(CC(C#C)C)C2)=O)cc(F)c(C)cc1Cl 31987,N(C1CCc2ccccc21)c1nn(C)c(Oc2nccc(C=O)c2Br)c1 31988,C1(CCC)CCC(C(=O)NCCC(C)N(C(=O)CCC(C)SC)C)CC1 31989,C(=O)(C(F)(F)C(C)O)NCC1(F)CC(NC(c2c(C(=O)OC)nn(C)n2)=O)C1 31990,Cc1cn2cc(C(=O)NC3(CF)CCN(C(=O)CNS(=O)(=O)CC)C3)ccc2n1 31991,c1(C(=O)NC23C(CN(C(C(C=C)(C)CC)=O)C2)C3)ccc([N+](=O)[O-])c(N)n1 31992,N1(C(c2ccc(C)cc2)=O)CCCN(C(=O)C(C)c2ccon2)C(CO)C1 31993,C1(C(=O)NCCCC=C)CC(=O)CN1C(=O)CCc1cccn1C 31994,C1(NC(C(CCC)(C)O)=O)CC(C2CCN(C(=O)C=Cc3ccncc3)CC2)C1 31995,C1(CC(=O)NCC(C2CCCCC2)NC(c2ccco2)=O)CCC2CC12 31996,C(CC(=O)NCC(O)CN(C(=O)CC1CC(=O)C1)C)OCC#C 31997,Cc1csc2c(C(=O)NCCCNC(=O)C(N3CC(C)CC(C)C3)=O)ncnc12 31998,c1(N(C2CCN(C(C(C(C)C)O)=O)C2)C)ncnc2ncc(Br)cc12 31999,c1(C(N(CC(C)CNC(=O)CCn2cnccc2=O)C)=O)ccc(N)c(Cl)c1O 32000,CCC(C)CCCC(=O)NCC1=CCCN(C(C2CN3CCC2(C)CC3)=O)C1 32001,Cc1c(C2CC2)nc2ccc(Br)cc2c1NCCC1CN(C(=O)C(F)(F)F)CCO1 32002,c1(SC)ccc([N+](=O)[O-])cc1C(=O)NC1CC(NC(=O)C#CC2(C)CC2)C(O)C1 32003,CC1(C)c2[nH]nc(C(F)(F)F)c2CN1C(=O)Nc1cc(F)c(Cl)cc1[N+](=O)[O-] 32004,C1(C(=O)OCC)(C(=O)NCC2CC(O)CN2C(c2cnn(C)c2)=O)CCCCO1 32005,c1(C(=O)NCC(CC)NC(c2cnccn2)=O)nonc1N 32006,Cc1nc2c([nH]1)CC(C(=O)N(C)CCNC(c1ccc(C(C)C)o1)=O)CC2 32007,Cc1ncc(C(=O)NCCC2CCN(C(=O)CC(C)C(F)F)C2)c(=N)[nH]1 32008,Cc1ncc(NC(C2C3CN(C(=O)C(N4CCOC4=O)C)CC23)=O)cc1Br 32009,Cc1cc(N2CCC(NC3C4CCC3CC4)C(F)C2)nc(S(C)(=O)=O)n1 32010,c1(C(=O)NC2CC(CNC(C(C)(O)C3CCC3)=O)C2)cc(Cl)nc(Cl)c1 32011,C=C(C)CC(C(=O)C(=O)CCN)NC(C1CC(C)(C)C1)=O 32012,c1(C(=O)NCC2CCCN(C(C(C)(C)CC#N)=O)C2)cc(F)cc2nc[nH]c12 32013,C(=O)(C1CCCc2cncn21)N(CCCCN(C(C(C)NS(C)(=O)=O)=O)C)C 32014,Cc1noc(CCC(=O)NCc2nc(CNC(=O)C(C)C3CC3)cs2)n1 32015,C#CCC(C)(C=O)NC(C=CC(=O)NCC(CC1CC1)OC)=O.OCC 32016,c1(C(=O)NC(C2CC2C(=O)N(C)Cc2ccsc2)C)c[nH]nc1C(F)F 32017,C1(NC(CC)=O)CCCC(NC(c2cc(-c3ccc(C)s3)[nH]n2)=O)CC1 32018,N1(C(C(C=C)O)=O)CC(C(N2C(C(=O)OC)CC2C)=O)CC(C)C1 32019,Cc1coc(C(=O)NC(C)(C)C(=O)NCC2COCCO2)c1 32020,C1(C(=O)NC2CN(C(c3cccc(Cl)c3Cl)=O)C2)CCC2CC2CC1 32021,CCCCCCCCCCC(=O)NC(C)CN(C(=O)C(c1ccc(Cl)cc1)O)C 32022,c1(C(N2C3CCN(C(c4ncon4)=O)CC2CC3)=O)cc2cccc(F)c2o1 32023,c1(C(N2CC(N(C(C=CC(C)C)=O)C)C(F)C2)=O)cc2nccn2c(O)n1 32024,C1(CNC(CCC(C)C)=O)CC2CCC(C1)N2C(=O)NC1CC1c1cccnc1 32025,c1(OC(C(=O)NC2(C=C)CC2)C)ccccc1Br 32026,c1(C(N2C(C#C)CCC2)C(=O)NC2CCCCC2)cccc2[nH]ncc12 32027,c1(C(N(C)CC2COCCN2C(=O)COC2CCC2)=O)cnn2ccn(C)c12 32028,CC1(C(=O)NCCCN(C(C2OC3CCCC23)=O)C2CC2)CCCCO1 32029,CCCCC(CNC(C1CC(OC)(OC)C1)=O)NC(=O)CC1CCC(=O)N1C 32030,C1(CNC(=O)CCC2CCC(=O)N2)CN(C(=O)C2CC2)CCC12CCC2 32031,c1(C(=O)NCC2CC(NC(CC3CCN(OC)CC3)=O)C2)cnc2ccccn12 32032,c1(CC(=O)N(CC(CNC(C(C)n2ccnc2)=O)F)C2CC2)cccc2cn[nH]c12 32033,CC1(C)C(C(=O)O)(C(=O)NCC(O)CC2CCC2)C1(C)C 32034,C(=O)(C#CC(=O)NCC1(F)CN(C(=O)C=Cc2cncn2C)C1)N(C)C 32035,C1(N(C(CC(C)OC(F)(F)F)=O)C)CCN(C(=O)C(C)(C)NC(N)=O)CC1 32036,c1(NC(CC2CN(C(=O)OC(C)(C)C)C2)=O)ncnc2c1ccn2CC(C(C)(C)C)=O 32037,c1(-c2c(OC(C)=O)cc(C)cc2)cccc2[nH]nc(C(=O)Nc3conc3C)c12 32038,Cn1ccc(S(=O)(=O)NCC(=O)NCCCNC(=O)CCC(C)(C)[N+](=O)[O-])c1 32039,C#CCCCC(C)C(=O)N(C1CCCC1)CCNC(C1CCC(=O)NC1)=O 32040,N1(C(C2CN(C)C2)=O)CCC2C(CCN2C(=O)CCc2ccc(F)cc2Cl)C1 32041,C1(NC(C(C)OC)=O)CCN(C(c2cnc(-c3ccccn3)nc2)=O)CC1O 32042,N1(C(CCC=C(C)C)=O)CCN(C(=O)C=Cc2cccnc2C)C(CC2CC2)C1 32043,c1(OC)cc(C)cc(C(=O)NCC2CC(O)CN2C(=O)CC(=O)N(C)C)c1C 32044,c1(C(=O)OC)cc(C)nnc1NCC1CN(C(c2cc(F)ccc2C2CC2)=O)C1 32045,c1(C(N2CC(C(=O)NOCC=CCl)(OC)C2)=O)sc(O)nc1C 32046,c1(OC)nccc(C(=O)NC2(CO)CN(C(=O)C(CCSC)NC(=O)C3CC3)C2)n1 32047,C1(CC(=O)N(C2CCN(CC)C2)CC)CC2(C1)CN(C(=O)C(C)NC(=O)C1CC1)C2 32048,Cc1c(C(N2CC3CC3(C(N3CC(=O)NCC3C(N)=O)=O)C2)=O)cccc1F 32049,N1(C(C2(C#C)CN(C(C3CCOCCN3C)=O)C2)=O)CCC2(CC1)CSC2 32050,C12(C(=O)OC)CC(C(=O)OC)C(C1)C2.CCCC1CO1 32051,C1(NC(C(CC)CC)=O)CC2CC(NC(C3CN(C(=O)NC)C3)=O)CC2C1 32052,C1(N(OC)Cc2ccc(C)o2)(CC2CC2)CCN(c2ccc(Cl)c(O)n2)CC1 32053,Cc1nc(NCC(F)(F)F)cc(N2CCOC(Cn3cc(C4CC4)nn3)C2)n1 32054,C(=O)(C1=C(C(=O)NC2CCC(C)N(C(c3cnccc3OC)=O)C2)CCC1)OC 32055,N1(C(C2N(C)CC(O)C2)=O)CCOCCC1C(=O)NCCCN=[N+]=[N-] 32056,c1(C(c2nnnn2CSc2ccccc2)NC(C(C)SC)C)sc(C)c(Br)c1C 32057,c1(OC)cnc(NC(C2CC23CN(Cc2cc(C)[nH]n2)C3)=O)c(F)c1 32058,N1(C(C2(COC)CCOCC2)=O)CCN(C(=O)C(C)c2ncco2)CC12CCC2 32059,C(=O)(C1=NOC2COCC12)NC(C)CN(C)C(C1C2(CC2)C12CC2)=O 32060,C(CC(=O)N1CCC(OC(F)F)C1)(CC(C)C)NC(C(COC)NC(C)=O)=O 32061,N1(C(C2C(C=C)C2)=O)CCC(O)C(NC(=O)Cc2csc(-c3ncccn3)n2)C1 32062,CC(CC(N)=O)C(=O)NC12CC(C(=O)NCC(C)(C)CC(C)O)(C1)C2 32063,Cc1cc(F)cc(C(=O)NCCN(C(=O)CC2CCCC(O)C2)C(C)C)c1N 32064,N1(C(C(c2scc(C)n2)C)=O)CCC(CNC(=O)C#CC(C)(C)C)C12CC2 32065,Cc1ccc(C(=O)NCCN(C(=O)C2=NNC(=O)C2)CC(C)O)c([N+](=O)[O-])c1 32066,CN1CCC(C)(CNC(=O)C(O)c2ccco2)C1.C1(=O)C(F)CC2CN1C2 32067,C(c1ccc(C(N)=O)o1)=CC(=O)NCC(CCC)NC(=O)CC1(O)CCC1 32068,c1(C)cc(Cl)ccc1Cl.c1(C(=O)NCC2CCCCN2C(=O)N)cccc(F)c1O 32069,CC1CN(c2nnnn2C)CCC1NCc1ccnc(OC(F)F)c1 32070,C1(C(=O)NC2CC(NC(C3(CO)CC(C)(C)C3)=O)C2)CCn2nncc2C1.C(N)(=O)N 32071,C1(C(N2CCN(C(C34CCCC(C)(OC3)C4)=O)CC2)=O)CCc2[nH]nc(O)c2C1 32072,C1(C(=O)NCCOC2CN(C(c3c(C)ocn3)=O)C2)CCCCC1O 32073,N1(C(C(CCSC)NC(N)=O)=O)CC2(CCN(C(C3CCCN3N=O)=O)CC2)C1 32074,CCC(C(=O)NCC(COC)NC(c1cccc(C)c1F)=O)C(C)(F)F 32075,C1(C(=O)NCC(C)N(C(=O)CC2(NC(=O)OC(C)(C)C)CC2)C)CC2C(C1)C2(C)C 32076,C1(NC(C(CC)N(CC)CC)=O)CN(C(c2ccc(Cl)c(C)c2)=O)CC12CC2 32077,c1(C(C)C)cc(C(=O)NCCNC(c2csc(O)n2)=O)on1 32078,C(CC(C)C)(C(=O)N1CCCC(C)(C(=O)NC2CCOCC2C)C1)NC(C)=O 32079,c1(C(=O)NC2CC(C)N(C(=O)CN3CC=CC3)CC2)cncc(N=[N+]=[N-])c1 32080,N1(C(c2n(C)c(S)nn2)=O)C2CCC1CN(C(c1ccc(N)c(O)c1)=O)CC2 32081,C(=O)(N=c1[nH]nc(N2CCCC(C)C2)s1)NCC(C)OC 32082,C1(CCNC(CCN(C)CC)=O)CCCCN1C(c1ocnc1C1CC1)=O 32083,c1(C(=O)NC2C(C)(C)C(NC(=O)CC3(CO)CC3)C2(C)C)ccc(Cl)c(Cl)c1O 32084,c1(C(=O)NCC(CC)NC(=O)COCc2cccnc2)cnn2c1C(=O)NCC2 32085,c1(C(=O)NCC2(C)CC(NC(C3C4CCCC34)=O)C2)cnc2nccnc2c1 32086,n1(CC)cc(Cl)c(C(=O)NC2(CO)CCN(C(=O)CSc3cnn(C)c3)C2)n1 32087,C#CC1CC1C(=O)NCCCOCCN(C)C(C1(CCN(C)C)CC1)=O 32088,N1(C(c2c(C)nsc2)=O)CC2(CC(C(=O)NCC(C)(O)C3(C)CC3)CO2)C1 32089,Cn1nc(O)cc1C(N1CCCC(OCCNC(=O)CCOC2COC2)C1)=O 32090,CC(C)(C)CC(F)C(=O)N1CC(C(=O)NC(C)(C)CNC(N)=O)C(F)(F)C1 32091,CC1(C(N2CC(C3CCCO3)C2)=O)CN(C(C2CCC(=O)C2)=O)C1 32092,Cc1cc(CC(=O)NCC2CCCN2C(C2CCOC(=O)N2)=O)ccc1C(F)F 32093,N1(C(c2cnn(C(C)(C)C)c2)C(=O)NCCOC)CCC2CC12C.C1(C)CCOC1 32094,c1(CC(=O)NC2CC(NC(c3ccnnc3O)=O)C2)cc(F)cc(F)c1Br 32095,N1(C(CC(C=C)(C)C)=O)C(C)CC2CN(C(C3COCCC3C(F)(F)F)=O)CC12 32096,C(C(F)(F)CC(O)CO)NC(C1=CCCSC1)c1n(CCC(=O)OCC)nnn1 32097,Cc1c(S(N)(=O)=O)cnc(NCCCNC(c2cccnc2)=O)c1Br 32098,c1(C(=O)NC(CCCC)CNC(c2cc(OC)ns2)=O)c(F)cc(F)cc1Cl 32099,C1(C(NOCCCOC)=O)C2CC3C(C2NC(=O)CCCCC2CC2)C13 32100,c1(CC(C(=O)OC)NC2CC(n3ccnn3)C2)ccc(OC(F)F)cc1 32101,c1(CN2C(C(=O)NCc3c(C)ccc(Br)c3)C3CCC2C3)ccc2nc[nH]c2c1 32102,C(C(=O)Nc1cncnc1C)(C(C)(C)C)NC(CCSCCCC)=O 32103,N1(C(c2cnc(CC)[nH]2)=O)CC2CCCC2(NC(=O)Cc2cn(C)cn2)C1 32104,c1(C(N(C(C)C)CCNC(c2cc[nH]c2)=O)=O)nccc2ccn(C)c12 32105,C1(NC(C=C(C)C)=O)CN(C(c2snnc2C(C)C)=O)CC1C 32106,C1(CC)CN(C(C23CCC(OC)C2C3)=O)CC1C(=O)NCCC(C)(O)CC 32107,N1(C(C(CCCC)O)=O)CCN(C(C2CC(OC)C2)=O)C2(CCC2)C1 32108,C1(C)(C(=O)NCC2(O)CN(C(CCCOCCC)=O)C2)CCCS1(=O)=O 32109,C1(CC(N2C(CNC(C3(C)CCCO3)=O)CCC2)=O)COCCN1CC(F)(F)F 32110,c1(C(N(CC)CC2CCN(CCCc3cnccc3C)C2)=O)cnc(C)nc1 32111,CC1CC2CCC(C(N3CCC(F)(CNC(c4ccccc4)=O)CC3)=O)CN2C1 32112,N1(C(c2ccc(C(=O)OC)cn2)=O)CC2(CCN2C(=O)C2=CCOCC2)C1 32113,C1(C(=O)NCC2(C(N)=O)CN(C(C(C)C#N)=O)C2)CC2(CC(=O)N2)C1 32114,O=C1C=C2CN(C(C3CN(Cc4ccc(OC(F)F)cc4)CCO3)=O)CCC2S1 32115,C1(CNC(=O)CCCN2CCCC2)CC(F)(F)CN1C(c1cncs1)=O 32116,c1(C(C(=O)N(CCNC(C(C)n2cccn2)=O)C2CC2)C)ccnn1C 32117,C(c1cnc2ccccc2n1)=CC(N1CCC(NC(C2C(C)C2)=O)C12CC2)=O 32118,S(=O)(=O)(c1ccc(NC2CCOC(CO)C2)cc1Br)NCC(C)(C)OCC 32119,c1(C(=O)NCC(CNC(C(CC(=C)C)C)=O)(C)O)cn2cc(C)ccc2n1 32120,C1(CC(C)O)CCCCN1C(c1ccc(CNC(c2nc(Cl)cs2)=O)cn1)=O 32121,c1(NC(c2c(OC)n[nH]c2)=O)ccc(C2CCNCC2)c(F)c1 32122,C1(CNC(CC=C(C)C)=O)CC2(CCN(C(c3cn(C(C)C)cc3C)=O)C2)CO1 32123,CCC(C(C)(C)O)NC(c1cnn(CCNC(C2CCC(=O)C2)=O)c1)=O 32124,C(=O)(CCCCC(N)=O)NC(C(=O)N(C1CCCN(C)C1)C)CO 32125,C(N=c1[nH]c(=NCCC2(C3CC3)CCCO2)[nH]c2ncn(C)c12)c1n(C)ccc1 32126,C#Cc1ccnc(C(N2CCN(C(=O)C(CC)CC=C)C(C3CCC3)C2)=O)c1 32127,C1(F)(CNC(C(CCCC)C)=O)CCCN(C(=O)Cc2ccc3occc3c2)CC1 32128,CC1(C)CC(CC(N2CC3C(C(N4CCOC(C(C)(C)C)C4)=O)C3C2)=O)CCO1 32129,C(=O)(CCC(C)S(C)(=O)=O)NC(CNC(c1c(C)nn(C2CC2)c1Cl)=O)C1CC1 32130,CCC(C)C(C(=O)NCC1(C(N2CCC(O)CC2)=O)CCCC1)OC 32131,c1(NC(=O)CCOC2COC2)cccc2sccc12.CC1C2CCN1C2=O 32132,CC(c1ccccc1Cl)=CC(=O)N(C)CCN(C(=O)COc1ccc(C)cc1)C 32133,Cc1ccc(O)c(C(=O)NCCNC(=O)CCc2ccn(C)n2)n1 32134,c1(C(=O)NC2CC2)cc2n(n1)CCCN(C(c1cnn(-c3ccccc3)c1)=O)C2 32135,N1(C(C(C)OCC=C)=O)CC(C(N)=O)(CNC(=O)CC(C)SC)C1 32136,c1(CC(=O)NCCCN(C(CCCN(CCC)CCC)=O)C)nn(CC)cc1Cl 32137,N1(C(c2ccc(CCC)[nH]2)=O)CC(NC(c2cccc(N)c2)=O)CC1(C)COC 32138,C1(NC(C2(CC#C)CCOC2)=O)C2CC1N(C(c1ccc(C(F)(F)F)s1)=O)C2 32139,c1(N2CCN(C)C(C)(C)C2)nc(N2CCCC(C)(CO)C2)nc2c1SCC2 32140,N1(C2CCC2)CC(C(=O)N(CCNC(c2ccnc(OC)c2)=O)C(C)C)NC1=O.CS 32141,C(CCC(O)C(=O)NC(c1cc[nH]n1)C)NC(C(CNC(C)=O)(C)C)=O 32142,N1(C(c2cnc(C(C)=O)s2)=O)CCCC2(NC(=O)CNC=O)CC2C1 32143,C(CC(=O)NOCCC(C)O)(C(C)(C)C)NC(C1(COCC)CC1)=O 32144,c1(C(N2CCC(C)(NC(c3nc(C)c(C)[nH]3)=O)CC2)=O)cnc(O)c2ccsc12 32145,C(CC(C(=O)NCc1ncc(Cl)s1)NC(=O)Cc1ncoc1C)=CC 32146,C1(CNC(c2cc[nH]n2)=O)CN(C(c2ocnc2C2CC2)=O)CC12CC2 32147,C(CNC(c1c[nH]nc1OC)=O)(CCC)NC(C(C)=C(CC)C)=O 32148,C12(C(N(CCN(C)C(C3(n4ccnn4)CC3)=O)C)=O)CC(C1)C(C)(C)O2 32149,C1(OC)CN(C(c2csnc2Cl)=O)CCC1NC(c1cnn(C(C)C)c1)=O 32150,N1(C(C2C3CN(C(CC4CCC(C)(C)C4)=O)CC32)=O)CC2(CCOCC2)C1 32151,O=S(=O)(c1ccc(NCC2CC(F)(F)C2)c(Br)c1)N1CCOCC1C(F)(F)F 32152,N1(C(C(C)NC(N)=O)=O)CCC(C2CCCN(C(=O)Cc3ccncc3Cl)C2)C1 32153,Cc1cnc(N(C)CN2C3CNCC(C)CN32)nc1C.C12CCC(CC1)CC2 32154,C(=O)(CCCCCF)N1CCC(CCOC)(NC(C2CC(CSC)C2(C)C)=O)C1 32155,C12(CNCCC(COC(S(C)(=O)=O)=O)N)CC3CC(CC1C3)C2 32156,N1(C(c2cc(CC)[nH]n2)=O)CCCC(N2CCN(C(C3(O)CC3(C)C)=O)CC2)C1 32157,Cc1ccnc(C(C)(C)C(=O)NC(C)CN(C(=O)C(F)OC(F)(F)F)C)c1 32158,N1(C(C(C)O)=O)CC(NC(c2cc3ncccc3[nH]2)=O)CC12CCCCC2 32159,C#CCCCCC(=O)NC1CC1CNC(c1ccc[n+]([O-])c1)=O 32160,c1(C(N2CCCC(C3CCCN3C(c3ns[nH]c3=O)=O)C2)=O)cccc(O)n1 32161,N1(C(C#CC(OCC)OCC)=O)CCC(NC(=O)CSc2nncn2C)C(O)C1 32162,C(=O)(CCC(C)(C)N1CCOCC1)N1CCCC(CCNC(CC(CC)OC)=O)C1 32163,C1(C(N2CCCC2CN(C(=O)CC2COC(=O)C2)CC)=O)CCC(=O)NC1 32164,c1(C(N2C(C)CC(NC(=O)COc3ccsc3)C2)=O)cc(F)cc2nc[nH]c12 32165,CN1CCCC1C=CC(=O)NCC1(O)CCN(C(c2cscn2)=O)C1 32166,c1(SCc2n(-c3c(CCn4cnnc4)cccc3)ccn2)ccc2c(c1)CCC2 32167,C1(C(N(C2CN(C)C2)C)=O)CC12CCN(C(c1cscc1Cl)=O)CC2 32168,C(=O)(CCCCCC#N)NCc1ccc(C(N2CCC(C#CC)C2)=O)cc1 32169,N1(C(C(Cn2cncn2)NC(CCCOC)=O)=O)CC2C(C1)C2(C)C 32170,c1(C(=O)NC2C(CNC(COCCC=C)=O)CCC2)cc(C)nc2ccnn12 32171,N1(C(CCCc2c(C)ccs2)=O)CC(C2CN(C(c3cc4ncccc4s3)=O)C2)C1 32172,C12(C(N(CC)CC3CCCO3)=O)CC1CN(C(=O)C(C)=NOCC#N)C2 32173,c1(C(N2CCCC(N(C(=O)C(F)C(F)(F)F)CC)C2)=O)cc(C)nc(Cl)c1N 32174,C1(CC#C)CCCCN1C(=O)C(C)N(C)C(c1ncccc1F)=O 32175,C1(C)(C(N(C2CC(C#N)C2)CC(=O)NCCC2(C)N=N2)=O)CCOC1 32176,C(C(O)C(=O)NC1CCC(C(=O)N(CC(=O)NC)CC)C1)=CCCC 32177,Clc1ccc(CC(c2nn[nH]n2)Nc2ccccc2)cc1Cl 32178,C(CC(=O)NOCCO)C1(OC)CCC1.C1(=O)CN1.C(C)(C)(C)S 32179,C1(O)(CNC(CCc2onc(CC)n2)=O)CCN(C(c2snnc2C2CC2)=O)C1 32180,N1(C(C2CC(Cl)C2)=O)CCCCCC1.C1(NC(=O)COC)CCCC1CF 32181,CCCCC(C)C(=O)N1CCN(C(c2cc(CC)[nH]n2)=O)C(C(F)F)C1 32182,N1(C(C(C)(C)NC(C)=O)=O)CC2(C(=O)N(CCCF)C)CC1CO2 32183,c1(SC)nc(N2CCC(NC(c3cncn3C)=O)C(F)C2)cc(C(F)F)n1 32184,C(=O)(C1=COCCC1)NC1CCN(C(c2c(C)nsc2)=O)C1 32185,N1(C(C2CCN(C3COC3)CC2)=O)CC(NC(=O)CSC(F)(F)F)C(O)C1 32186,C1(NC(N)=O)CCC(C(F)(F)F)CC1.C1(C)C(=O)OC(C)CO1 32187,Cc1cnc(C)c(C(=O)NCC2CCCN2C(=O)CCCNS(C)(=O)=O)c1 32188,c1(N(C(C)CCNC(=O)CCc2nc(SC(F)F)no2)C)cc(Cl)ncc1Cl 32189,C1(CNC(CCCCC#C)=O)CCCC2CN(C(C3(C(F)F)CC(=C)C3)=O)CC12 32190,c1(OC)ccoc1CNC1CC(C(N2CCCC2C(F)(F)F)=O)C1 32191,C12(NC(Cn3c(C)ccn3)=O)CCC1CN(C(c1cc(O)nc(C3CC3)n1)=O)C2 32192,S(=O)(=O)(C1CS(=O)(=O)c2ccccc21)Nc1ccc(OCCC)c(OCC)c1 32193,CCN=C(NCc1ccccc1CO)NC1CCC(C(=O)OC)C1 32194,C12(C(=O)NCC(=O)NCc3ccccc3F)CC1CN(C(=O)COC1CCC1)C2 32195,O=C(N=c1cc(-c2ccc3c(c2)CCC3)[nH][nH]1)c1csc(=NCc2cc[nH]n2)[nH]1 32196,N1(C(C(=O)NCC)=O)CC(CNC(C2CCC(N(C)C)CC2)=O)C(O)C1 32197,C12(NC(C(CC=C)CC=C)=O)CCCCC1N(C(C1CC=CCO1)=O)CC2 32198,C1(CNC(C2C(c3n(C)ccn3)C2)=O)CN(C(c2ccc(=N)[nH]c2)=O)CC1(F)F 32199,c1(C(N(CCCCNC(=O)COC2CCOC2)C)=O)c(Cl)ccc(O)c1N 32200,c1(OCCN(C2CCC2)CCOC)ccccc1Cl 32201,N1(C(CCc2ccc(OC)nc2)=O)CCN(C(=O)C2=CCSC2)C2CCCCC12 32202,N1(C(C2N(C(c3c(C)oc(CO)c3)=O)CC(=O)NC2)=O)CCOC2(CCC2)C1 32203,C#Cc1ccc(C(=O)NC(C)C(C(C)C)NC(=O)CN(C)CCC)c(F)c1Cl 32204,C1(NC(CCOCCCC)=O)CCC2(CC2)N1C(=O)NC1(C2(C)OCCO2)CC1 32205,C(C1=NOC2CN(C(C34CCC(F)(CC3)C4)=O)CC12)NC(c1nn(C)c(O)c1)=O 32206,C(=O)(C1Cc2ccccc21)N1C(CN(C)C(c2csc3cncn23)=O)COCC1 32207,Nc1[nH]c(=O)c(Cl)nc1C(N1CCC1CNC(c1occc1Br)=O)=O 32208,Cc1cccc(C(=O)NC2(C(=O)NC3(C4CCCCO4)CC3)CCCCC2)c1Cl 32209,N1(C(CCC2CC(NC(C3CC=C(C)CC3)=O)C2)=O)CCC(C)(O)C(O)C1 32210,N#Cc1cnccc1-c1cncc(C(N2CC3CC3C2)=O)n1 32211,CC(CF)CC(=O)NC1CC(NC(c2ccc(-c3cccc(F)c3)o2)=O)C1 32212,n1(CC=C)ccnc1C(=O)NCCCC1CCCN1C(=O)CN(S(C)(=O)=O)C 32213,C(CC(C)C)(C(=O)NC1CN(Cc2ccccc2C(F)(F)F)CC1C#N)NCC 32214,N1(C(N2CCC(Cc3nccc(C)n3)CC2)=O)Cc2c(F)cccc2C(C)(C)C1 32215,C12(NC(CC(C)O)=O)CCCC1CN(C(=O)C(C)(F)F)C2 32216,CC1CCCC(NC(N2CCNC(=O)C2C)=O)CC1 32217,C=CCC(CC)C=O.C1CC(n2cc(CC3CCC3)nn2)C(O)C1 32218,Cc1cc(C(=O)NC(Cn2ccnn2)C(=O)NCCNC(N)=O)ccc1O 32219,C12(CNC(C(C(C)C)F)=O)CC(NC(=O)CCC3CCCCC3)(C1)C(C)O2 32220,c1(SCC(=O)N(C2CCN(C(C3CC3C3CC3C)=O)C2)C)nc(C)cc(C)n1 32221,c1(C(CNC2(c3n(CCC)nnn3)CC(CC(=O)OC)C2)CC)cccc(C)c1 32222,N1(C(CCN(CC)CC)=O)CCCN(C(=O)C2=CCOCC2)CCC1 32223,c1(C(=O)NCC(CNC(C=CCOC)=O)OC)cn2ccnc2cn1 32224,N1(C(=O)OC(C)C)CCCC(C(=O)NCCCCCc2ccccc2)C1 32225,c1(NC(C2(C)CCN(C(CCSNC(C)(C)C)=O)C2)=O)ccc2c(c1)CNC2=O 32226,c1(C(=O)NCC(CNC(C(C2CCCOC2)OC)=O)O)c(F)ccc(F)c1F 32227,c1(C(=O)NC2(C)CN(C(c3c(O)cc(C)nn3)=O)C2)cc(F)cc2c1NCCC2 32228,C1(NC(c2c(C)cc(C)s2)=O)CCN(C(=O)C(c2cccc(Cl)c2)(C)C)CC1O 32229,C1(C)(CN(C(=O)C(N)=O)C)CCN(C(=O)CCC2CCC(C(N)=O)O2)C1 32230,C1(NC(c2ccc3occc3c2)=O)CCCC12CCN(C(c1cncs1)=O)CC2 32231,c1(C(N(CC(CNC(C2(COC)CCOCC2)=O)C)C)=O)nc(C)ccc1OC 32232,C1(CNC(C2N(C)CSC2)=O)C2CCCC1N(C(=O)CC1CCCCC1)C2 32233,C(=O)(C(Cc1ccc(O)cc1)C(F)(F)F)NCCCC(C)NC(C(C)=C(CC)C)=O 32234,C(=O)(C1=CCCOC1)NCC1CC(NC(C2CC(OCC)C2)=O)C1 32235,Cc1cc(C(=O)NC(CNC(c2cc(C(N)=O)[nH]n2)=O)C2CC2)cnc1O 32236,CC1C(C(=O)NC2CCN(C(=O)C=Cc3cnc[nH]3)C2)OC2CCCCC12 32237,CC(=O)CCCC(=O)NCC12CC1CN(C(c1ccc(C)n1C)=O)C2 32238,C1(C(=O)NCC(C)N(C(=O)CN2C(=O)CNC2=O)CC)CCCC(F)(F)CC1 32239,CCC(F)(F)C(C)(C)C(=O)N1CCC(C(C)NC(C2(C#N)CC3CC3C2)=O)C1 32240,c1(C(N2CCC(NC(c3cn[nH]c3)=O)C(O)C2)=O)cnc(O)c([N+](=O)[O-])c1 32241,C(=O)(CCOC(=O)Cc1cnsc1)OC(C)(C)C 32242,c1(C(=O)NC2CCN(C(=O)Cc3c[nH]nc3O)C2)ccc2c(c1)CCC2(F)F 32243,CC(C(C)CO)N(CC(=O)Nc1ccc(Br)s1)Cc1scnc1Br 32244,Cc1cc(NC(=O)CC2CCN(C(c3cc(Cl)ccc3O)=O)C2)nc(Cl)c1 32245,N1(C(C(C)C)=O)CC(NC(c2ccc3ncoc3c2)=O)C(S(C)(=O)=O)C1 32246,c1(OC)ccc(C(=O)NC2CCCCN(C(=O)C3CC3)CC2)c(OC)c1OC(F)F 32247,C(=O)(C1=NOC2(CCC2)C1)NC(C1N(C(CCC=CC)=O)CCCC1)C 32248,Cc1cn2ccc(C(=O)NC3CC(C(=O)NC(C)CN(C)C)C3(C)C)cc2n1 32249,N1(C(CC2(C)CC2(Cl)Cl)=O)CCC2(CCN(C(C3(C(=O)C4CC4)CC3)=O)C2)C1 32250,N1(C(CCCSC)=O)CC(NC(C)(CCN2CCC(C)C2)c2cccs2)CCC1C 32251,c1(C(=O)NCC(C2CCOC2)OC)cc(CO)c(C)o1 32252,N1(CC(C)C)C(=O)c2ccccc2C1=O.c1(-c2cn(CC)nn2)ncccc1Cl 32253,c1(OC)ccc2c(c1)C(=O)CCN2C(c1ccc(Br)cc1)C(=O)NCc1cccs1 32254,N1(C(c2c(CC)non2)=O)C2CCCC1CC(NC(c1cnnc(O)c1)=O)C2 32255,C1(C(C)C)CN(C(C2CC2c2cnc[nH]2)=O)CCN1C(=O)CS(C)(=O)=O 32256,C(=O)(CN=c1[nH]c(C)cs1)NCC(CNC(C1(SC)CC(O)C1)=O)C 32257,c1(C(N2CC(O)(CNC(C3(F)CCOC3)=O)C2)=O)cc(F)ccc1Br 32258,C1(CNC(CC(C)(C)OC)=O)C(C)CCCN1C(=O)C(CO)N(C)C 32259,N1(C(c2c(C)cc(CNC(C3CC34CCCC4)=O)o2)=O)CCCC2C(=O)NCC12 32260,N1(C(CNC(CSCC=C)=O)=O)CCCNCCC1.C(=O)(COCCOC)N 32261,C1(C(N2CCC(O)(CNC(=O)CC3(C)CCOCC3)C2)=O)(COC)CC=CCC1 32262,C1(NC(CC2C(OC)COCC2)=O)CCCC2CN(C(=O)CCCC(F)F)CC12 32263,C1(NC(CC(C)C(F)F)=O)COC2(C1)CN(C(C1CC=CC1)=O)C2 32264,N1(C(CC2(OC)CC2)=O)CC(NC(=O)CCc2ccc(OC)nc2)C(C)(C)C1 32265,c1(CC)nc(Cl)nc(N2CCC(OCCNC(C3(C)C=CCC3)=O)C2)c1Cl 32266,N1(C(Cc2ccn(C(C)C)n2)=O)CCC(C)C1CNC(=O)CCC1CC1 32267,c1(C(=O)NCC2(CC(=O)Nc3cncc(CO)c3)CC2)c[nH]ccc1=O 32268,CC(C)CC(C)(CNC(=O)C=Cc1ccn(C)c1)NC(c1cn2ccnc2s1)=O 32269,n1(CC)nc(C)c(C(=O)ONC(c2n(CC)nnn2)C2(C#N)CC2)c1C 32270,O=S(=O)(c1ccc(F)c(Br)c1)N1CC2CC1CN2c1nccn2ccnc12 32271,C#CCC(CO)NC(C1(C(C)NC(=O)CCOC2CC2)CCC1)=O 32272,C1(CC(=O)NC2CCN(CC(C)C)CC2)CC2(C1)CN(C(=O)CC1COCC1O)C2 32273,C=CC(O)C(C)(C)C(=O)NC1CCN(C(C2CCCNC2)=O)C1 32274,C1(NC(c2ccc(CC)cc2O)=O)CN(C(=O)CCS(C)=O)C2(CCC2)C1 32275,c1(OC)cc(C(=O)NC(C)CCN(C(=O)CC2CNC(=O)C2)C)cc(Cl)c1 32276,c1(C(=O)OC(CCCC)CCCC)cc(F)cc2c1CCC2 32277,C12(CNC(C(CC=C)NC(C)=O)=O)CCC(CC1)N2C(=O)C(C)OCOC 32278,c1(C(C(=O)Nc2ccc(OC)cc2)N(C2CCOC2C)C)cc(C)ccc1Br 32279,c12cccc(c1)C(=O)NC1CC(C1)NC(=O)C(=O)N2.CN1CC(O)(CO)C1.C(C)(C)C 32280,CC(C)C(C)C(=O)NCCN(C)C(c1ccc(OC(F)F)cn1)=O 32281,N1(CC(=O)NCCCN(C(C2C(C)COCC2)=O)C)CCCc2sccc2C1=O 32282,c1(C(N2CCCC(N(C(=O)C(C#N)C3CC3)C)C2)=O)cccc(C(F)F)c1F 32283,CC1=C(C)CC(C(=O)NCC2(O)CC(C(=O)NC3CNC(=O)C3(C)C)C2)CC1 32284,NS(=O)(=O)c1ccsc1C(N1CC(O)(CNC(=O)CCc2cc(Cl)no2)C1)=O 32285,c1(C(N(C(C(=O)NC2(CCC)CC2)C)C(C)CC)=O)c[nH]c(=N)c(C)c1 32286,CCC(C)(C)C(C)NC(c1n[nH]cc1CNC(=O)CCNC(=O)NC)=O 32287,C1(C(C)NC(C=C(COC)C)=O)CCN(C(C2CC(O)(CC(C)(C)C)C2)=O)C1 32288,C(=O)(C(C)(C)CCC)N(CC(=O)N(CCC)CCC)CCCN(CCOC)C1CC1 32289,N1(C(c2cc(-c3cccc(OC(C)C)c3)[nH]n2)=O)CCC2SC(=O)C=C2C1 32290,c1(C(=O)NCC(C2CCC2)NC(C(C=C)O)=O)cccc2c1CCC2 32291,Cc1cc(S(N)(=O)=O)cc(C(=O)NCC(C)NC(=O)CCCCC#N)c1C 32292,N1(C(C2CCN(Cc3cccc(F)c3I)C2)=O)Cc2ccc(C(F)(F)F)cc2C1 32293,Cc1ccc(C(CNC(C2(F)CC2)=O)NC(N2CCCC(N(C)C)C2)=O)cc1 32294,C1(=O)N=C2C=CN(N2)CC2CCCC12.C(=O)(CCCn1ccnc1)N(C)C 32295,CCC(F)(F)CC(=O)N1CCCC(NC(=O)CCCC2CCCC2)C1C 32296,c1(C(C2CC2)NC(=O)NC2CC(N)(C(F)F)C2)ccc(Oc2ccccc2)cc1 32297,c1(C(N2CCC(CC(=O)Nc3onc(C)c3Br)C2)=O)cc(F)ccc1[N+](=O)[O-] 32298,CCN=c1ccc(C(=O)NC2CC2NC(c2ccc(C(F)(F)F)s2)=O)c[nH]1 32299,N1(C(C2(OC)CCN(C(c3cc(OC)c(C)nc3)=O)C2)=O)CCCC(F)(F)CC1 32300,C(C(CC(F)(F)F)NC(=O)C(C)=CC1CC1)NC(CC(CC)n1cccn1)=O 32301,C1(C(=O)OC)CC2(CC(OC(C3(OC)CCNC3=O)=O)C2)C1 32302,C(=O)(C#CC1(C)COC1)N1CCCC(NC(c2n(C(C)C)ccn2)=O)(CO)C1 32303,C=CCC(CC(F)F)C(=O)NCC(C1CC1)NC(=O)C(CC)CC=C 32304,N1(C(C2C(C)(C)CC2)=O)CCC2(CCN(C(c3cnc(C(N)=O)cn3)=O)CC2)C1 32305,c1(C(=O)NCC(CNC(C2CC=CCO2)=O)CO)ccc(-n2cncn2)cn1 32306,N1(C(c2ncn(C)n2)C(=O)NS(C)(=O)=O)CCC(C(=O)NCC2CCCO2)CC1 32307,N1(C(CCOC)=O)CCC(C2OCCC2NC(c2cccc(N)n2)=O)CC1 32308,CC1CN(C(=O)CN(CC(F)F)C)CC1NC(=O)C(C)Cc1cccc(N(C)C)c1 32309,c1(OCC)cc(C(=O)NC(C(=O)NC2(C(=O)OC(C)(C)C)CC2)C2CCC2)[nH]n1 32310,c1(C(=O)NCC(CC)NC(C2CCN(C)C2)=O)nncc2ccccc12 32311,Cc1ccc(O)c(C(=O)NC(c2cnn(C)c2)C(N2CCC3CC23)=O)c1 32312,c1(OC)ncnc(C(=O)NCCCOCCNC(C2CCNC2=O)=O)c1F 32313,Cc1ccc2ncc(C(N3CCC(C)C(NC(=O)C(C)(C)CC(F)F)C3)=O)n2c1 32314,C1(NC(c2c(C)oc(Cl)n2)=O)COC2(CCCN(C(=O)CS(=O)(=O)N(C)C)C2)C1 32315,CCCC(CCNC(=O)CN(C(=O)CC1(OC)CCOC1)CC)CCC 32316,CCCC(CCC)CC(=O)NC1CCC1C(N1CCC(O)CC1COC)=O 32317,C(CCCCCC(=O)NC1(CC2CC2)CC1)NC(c1n(CC)ccc1)=O 32318,C1(CCC)(NC(c2cccc(=O)n2C)=O)CCCN(C(c2csc(C)c2N)=O)C1 32319,c1(C(=O)NCC23CC(NC(CC)(C)C(=O)OCC)(CO2)C3)cc(OC)ncc1Cl 32320,N1(C(Cc2c(C)nc[nH]2)=O)CC(NC(=O)C2=CCOCC2)CC12CCOCC2 32321,C(C(=O)OCCCCc1nnn(C(C)(C)C)n1)(C(C)C)OCC 32322,c1(C(=O)NC2C(CNC(C(C)c3ccsc3)=O)C2)ccc(Cl)c(F)c1O 32323,C1(C)(NC(C2C(CCC)CCC2)=O)CN2CCC1CC2.C1C(=O)N1C(C)C 32324,Cc1cnccc1C(C)C(=O)NCCN1CCC(NC(=O)C(N)=O)CC1 32325,c1(COC)cccc(C(=O)NC(C)C(C(C)C)NC(c2csc(C(C)C)n2)=O)c1 32326,n12cnc3c(ncnc13)N(C1COC1)C(C)C2.C(=O)(C(C1CCOC1)OC)OC 32327,c1(CC(=O)NCCOCCOCC#C)csc(Cl)n1.N12CC(C1)OCC2=O 32328,C1(C(=O)NC(CC)CNC(=O)CCN(S(C)(=O)=O)C)CCOC1CC 32329,C1(O)(C(=O)NCC(CC)(CC)c2ccccc2OC)CCCC(C)CC1 32330,C(=O)(C(C)(C)C(=O)NCC1CN(C(=O)CCCCc2ccccc2)C2CC12)NC 32331,c1(CCC(=O)OC2CC(C(=O)NC3CC3NCC)C2)nncn1C(C)C 32332,Cc1c(SCC2CC3(c4nc(Cc5ccccc5)no4)CC23)cccc1Cl 32333,Cc1cccc2c1c(CN1CCC(C(N3C4COCC3CC(O)C4)=O)C1)cn2C 32334,c1(C(C)NCc2cc(C(=O)OC)c(C)o2)ccc([N+](=O)[O-])cn1 32335,c1(C(=O)NCC2CN(C(=O)CCC(F)F)C3(CCC3)C2)cnc2ncccc2c1 32336,c1(C(=O)NCCNC(c2c(CC)ncs2)=O)cc(O)nc2cc(OC)ccc12 32337,N1(C(c2cc(C)n(C)n2)=O)CC(N(C(=O)CSCc2ccccn2)C)C(C)(C)C1 32338,N1(C(C(C)=O)=O)CC2CC1CN(C(=O)C(C(C)C)NS(=O)(=O)c1cnn(C)c1)C2 32339,C1(CNC(=O)C(F)C2CCC2)CN(C(=O)CCc2cc(Br)no2)CCO1 32340,N1(C(C2CC(=C)C2)=O)CC(CNC(=O)C=Cc2cc(Cl)sc2Cl)OC(C)(C)C1 32341,C1(NC(CCC(=C)Cl)=O)CC12CCC(NC(c1ccsc1)=O)CC2 32342,CC1(C)OCCC1NC(=O)C(C1CCCCC1)NC(=O)CSCC(F)F 32343,N1(C(C=CC(C)(C)N(C(=O)Cn2cccc2)C)=O)CCCC(CN2CCCC2)C1 32344,C(=O)(CCC(=O)NC(CNC(c1sc(N(C)C)nc1Cl)=O)C1CCC1)OC 32345,C1(CNC(C2CCCC(C(N)=O)C2)=O)(NC(c2cc(CO)[nH]n2)=O)CCCCCC1 32346,C1(NC(C#CC(C)C)=O)CCCC2CN(C(c3nc(=O)n(C)[nH]3)=O)CC12 32347,C1(C(N2CC(N(C(C(CC)=CC)=O)C)C(O)C2)=O)OC2CCCCC2C1C 32348,CC1CC(NS(=O)(=O)c2ccccc2CN(C)CN2CCOC2=O)c2nccn21 32349,N1(C(C2(CC#C)CCCCO2)=O)CCCCCC(NC(c2ccoc2Cl)=O)C1 32350,C(CC(C)(C)CC(=O)NCC(C1CC1)NC(c1coc(SC)c1)=O)OC 32351,c1(C(=O)NCC23CC2CN(C(=O)C(C2CCCCC2)O)C3)ccn2ccsc12 32352,N1(C(Cn2ccc(C)n2)=O)CCC(NC(=O)Cc2ccccc2Cl)C(C)C1 32353,N1(C(C2CC(F)(F)CS2)=O)CCN(C(=O)CCCCCF)C(CO)C1 32354,Cc1cnc(C(N2CCC(O)(CNC(=O)Cc3csc(C)n3)C2)=O)c(Br)c1 32355,N1(C(CC2C(=O)NC(=N)S2)=O)CCC2(CNC(=O)O2)C1 32356,c1(CCC(=O)NCC2N(C(c3cc(C)nn3C)=O)CC=C2)ccccc1[N+](=O)[O-] 32357,C1(NC(=O)C(O)c2ccsc2)CCN(C(=O)Cc2cnn(-c3ccccc3)n2)C1 32358,C1(CC(=O)N(CCNC(C2CSC2)=O)CC)CCC(=O)N1 32359,CC(C)=C=CC(=O)NC(C)CC(C)NC(=O)C(=O)Nc1ncc[nH]1 32360,C(c1ccnc2ccccc12)=CC(=O)NC1CCCC1NC(C1CC2CC2C1)=O 32361,S(=O)(=O)(c1cncc(Br)c1)NC1CN(C(C(c2ccccn2)C)=O)CC1F 32362,C(CCCCC(=O)NCC1CCN(C(C2CCCC(C)(C)C2)=O)C(C)C1)SC 32363,c1(C(N2CC(CCNC(CS(CC)=O)=O)C(C)C2)=O)ccc(C)cc1C 32364,c1(CCC(=O)N(C)CCOCCN(C(=O)CCC2CCOC2)C)cccnc1 32365,CC1CCC(C(=O)NCCN(C(=O)CSCC(N)=O)C2CC2)S1 32366,c1(OC)ccc(S(=O)(=O)N2CCOCC2)cc1C(=O)NC(C)(C)COC 32367,C1(COC)CCCN(c2ccccn2)C1.C12(CN(C(C)=O)C1)C(=O)NC2 32368,N1(C(c2c(CC)nns2)=O)CCC(C)(C)C1C(=O)NC(c1ccc(C)cc1)C 32369,c1(C(=O)NC2(C)CC(NC(C(CO)N(C)C)=O)C2)ccc(F)c2[nH]ccc12 32370,c1(C(=O)NC2(C)CC(NC(c3c(C)ncnc3O)=O)C2)cc(F)cc(Cl)c1N 32371,CC1CN(C(=O)C=CCF)CC(C)N(C(=O)C(F)(F)C2CC2(F)F)C1 32372,C1(C(=O)NC(CC(=O)NC)c2ccccc2)CCCN(C(c2ccccc2Cl)=O)C1 32373,c1(OC)ccc(NC(N2CC(C(F)(F)F)CCC2C)=O)cc1OC1CCCCC1 32374,Cc1ccc(C2CC2)c(C(=O)NCCCCN(C)C(C2(C)CCCS2)=O)c1 32375,N1(C(c2c(C#C)c[nH]n2)=O)CC(F)(F)CC1(C)CNC(c1c[nH]cc1C(F)(F)F)=O 32376,C=C=CC(C)C(=O)N(CC(=O)N(C)CC1COC(=O)N1)C1CC1 32377,Nc1cc(C(=O)N(CCCNC(c2nc(C3CC3)cs2)=O)C2CC2)cc(F)c1 32378,c1(OC)cc(C(=O)NCC2CN(C(C3CCC(C)(C)OC3)=O)C2)cc(C2CC2)c1 32379,Cc1c(NC(C2CN(C(=O)NCC34CCCC3CCC4)CCO2)=O)cccc1Cl 32380,c1(CC)nn[nH]c1C(=O)N(CCCNC(c1ccc(CN(C)C)s1)=O)CCO 32381,N1(C(CCOCC#C)=O)CCc2cc(OC)ccc21.N12Cc3[nH]nc(c3C1)C2=O 32382,N(C(=NCCn1cnc(C#N)n1)NCCOC)CC(=C)C 32383,C1(CNC(C=CC=CC)=O)CCCC(NC(=O)CCCCc2cnn[nH]2)C1 32384,C12(COc3ccc(CN(c4cccc(OC)c4)C)cc3Cl)CC3CC(CC(C3)C1)C2 32385,C1(C)(CNC(c2c(OC)nsc2OC)=O)CN(C(=O)CCC(C)C)C(C)(C)C1 32386,C(CN=C(NCc1ccncc1OC)NCc1ccncn1)OC 32387,C(=O)(C(=O)C(C)(C)CC)N(CCC(=O)NCC(C)(C)CCCO)CC#C 32388,Cc1cc(C(N2CC(F)CC2C(=O)NCC2CC(=C3CC3)C2)=O)nc(O)n1 32389,C(=O)(C(C(C)(C)C)n1cc(C2CCN(C)CC2)nn1)OC.C12CC(C1)NC2=O 32390,C1(C2CCCOC2)(NC(CC(CNC(C(CCC)CC)=O)(C)C)=O)CC1 32391,C1(C(=O)OC)CC(F)(F)CN1C(C(=O)NCc1cccs1)C1CC1C 32392,C(=O)(CC1=NNC(=O)C1)NC(C)CCCNC(C1(n2ncc(Br)n2)CC1)=O 32393,C1(C2(C)CC2)(C(=O)NC(C2C(C(N(CC#C)CC#C)=O)C2)C)CC1 32394,c1(N(C(C)=O)C2CCC2)cccc(S(=O)(=O)NC2CCN(C)C2)n1 32395,CCC(CC(=O)NCC(C)NC(c1ccc(SC(F)(F)F)nc1)=O)C(F)F 32396,c1(C(=O)NCCCCC(CO)NC(c2c(C=C)cnn2C)=O)c(F)cc(F)cc1Cl 32397,c1(C(N2CC3CC(C2)CN(C(=O)C(F)F)C3)=O)cnn2c1OCC1(CC1)C2 32398,N12CCOCC1C2=O.Cn1ccc(C2CC2NS(=O)(=O)CC2CCC2)n1 32399,C(=O)(CC(CCC)CCC)N1C(CNC(c2cn(CC=C)nc2)=O)C(C)CC1 32400,CC(CCO)N=c1nc2sccc2c(N(C)Cc2nccn2-c2ccccc2)[nH]1 32401,N1(C(c2cc(C)c(F)cc2)=O)CC2CN(C(=O)C(=O)C(C)(C)C)CC2C1 32402,Cc1ccc2c(c1)C(C(=O)NC1CCC(NC(=O)COCC3CCCC3)C1)C2 32403,CS(=O)(=O)CCC(CO)NC(=O)Cc1cccc(F)c1O 32404,C1(CNC(C(C)CNC(=O)Cc2ccc[nH]2)=O)CC12CCOCC2 32405,c1(CC(=O)NC(C2CC(C)(C)C2)C(=O)OC)c(F)cccc1F 32406,c1(C(=O)NCC2(CN(C(C(CC=C)CC)=O)C)CC2)ccc(Cl)c(OC)c1F 32407,CCC(C(=O)NCCN(C(=O)C(C)C1CCCC1)CCCN(C)C)C(C)C 32408,Cc1ccc(C(=O)NCCCCCC(=O)NC(c2csnn2)C)c(O)n1 32409,N1(C(c2cc(C)on2)=O)CCCC(C2CC2NC(c2cccc3ccoc23)=O)C1 32410,c1(NC(C2C(C(N(C(c3cccnc3)(C)C)C)=O)C2)=O)cc(Br)cc2[nH]ncc12 32411,c1(CNC(=O)NCC2CCC(C)(C)O2)ccc(F)c2c1CCC2.CC 32412,CC1(C(N2CCCC(NC(=O)CSC3CC3)CC2)=O)CCCS1(=O)=O 32413,C1(C(=O)NCC(C)(C)NC(c2ccc(CC(C)C)s2)=O)Cc2cccnc2C1 32414,Cc1cc(C(=O)OCC)nc(C)c1.C1(=O)C(C)N1C1CCOC1.C(C)(C)(C)O 32415,C1(N2CCN(c3nncs3)CC2)CC2CCC(C1)O2 32416,C1(NC(N2CCC(=CBr)CC2)=O)CCCN(C(C2CCOCC2)=O)CC1 32417,c1(OCC(N2CCC(N(C(CCOC(C)C)=O)C)C2)=O)cccc(Br)c1 32418,N1(C(c2c(SC)c(Cl)ccc2)=O)CCC(C)=C(c2ccco2)C1 32419,C1(CNC(CS(CC)=O)=O)CC(C)(C)CN1C(c1ccc(SC(F)F)cc1)=O 32420,Cn1ncc2nc(Cl)nc(NCC34CCC3CN(C(=O)CC3(C5CC5)CC3)C4)c12 32421,C1(C(=O)NC(C)CCNC(C2(C)CCC(=O)N2)=O)CC12CCCCC2 32422,C1(C)(C(N2CCC(CNC(C(c3ccccc3)C)=O)C2)=O)CCN(C)C1 32423,c1(N2CCN(C(C(=O)N(CC#C)CCC)C)CC2)ncnc2sc(C)nc12 32424,c1(C(=O)NCC(=O)NCC(C(C)C)NC(=O)C(F)=C2CCCC2)ccccc1F 32425,c1(C(=O)NCCC(C)(C)O)cccc2c1CNC(=O)C2=O 32426,C(=O)(CC(Cl)Cl)NC(CNC(C1(C(=O)NC)CC1)=O)C 32427,O=S(=O)(c1cc2sc(=NCC3CCCO3)[nH]c2cc1Cl)N1CCCCC1C1CC1 32428,c1(C(=O)NC2CCC(NC(c3c[nH]nc3C3CC3)=O)CC2)ccc(F)c(O)c1F 32429,CC(C)(C)CC(F)C(=O)N1CCC(CCNC(c2ccnn2C2CC2)=O)CC1 32430,c1(OC)ncc(C(=O)N(CCNC(c2cccc(O)n2)=O)C(C)C)cc1Cl 32431,N1(C(C2C(=C)C2C(=O)OC)=O)C(C(=O)NCCOCCO)CCC12CC2 32432,Cc1nc2ccc(C(N3CC(NC(C4CCC(=O)O4)=O)C3)=O)cc2n1C 32433,c1(OC)nc2cc(Cl)ccc2cc1-c1nc(C)nn1-c1cc(C)cc(C)c1 32434,n1(CCC)ccc(C(N2CC(NC(=O)CCC3CC3(F)F)C2)=O)n1 32435,N1(C(c2sc3cc(C)sc3c2)=O)CCC(C2CCN(C(=O)CC#N)CC2)C1 32436,C1(O)(CNC(C2(CC)CC2(F)F)=O)CCCN(C(c2ccc(O)cc2Cl)=O)CC1 32437,C1(CNCC(Br)=C(C)C)CNCCC1c1nccn1C 32438,N1(Cc2c(OCC=C)cccc2)CC2CN(C(C3CC4CCC3O4)=O)CC12 32439,C1(CNC(C(C)C#N)=O)C2CN(CC(=O)NC3(c4ccc(F)cc4)CC3)CC12 32440,n1(CCC2(C)CC2)cc(C(=O)NC2CCC2NC(=O)C(c2ccccc2)=O)nn1 32441,CCC(F)(F)CC(=O)N1CCC(CCNC(C2(C3CCCCO3)CCC2)=O)CC1 32442,N1(C(C2C(C)(C(F)F)C2)=O)CCN(C(=O)CCC2CC2)CC12CC2 32443,c1(SC(C)C)cccc(CNC(=O)Nc2ccccc2C(=O)N(C)C)c1 32444,N#Cc1cccc(Cl)c1NC(C12CC(NCc3ccc(-n4cncn4)cc3)(C1)C2)=O 32445,Cc1cnn(C)c1CC(=O)OC(C)OC(C)(C)C.C1(=O)CCOCCCN1.C.O 32446,Cc1ncnc(C)c1C(=O)NCC1CCC1NC(c1c(C)cc[nH]c1=N)=O 32447,C=C(Cl)CCC(=O)N1CC(CCNC(C2CC3CCC2C3)=O)(OC)C1 32448,C1(C)(C(=O)NCC2N(C(CCC(C)C#N)=O)CC2)CCCCNC1=O 32449,c1(CC)ccc(C(=O)OC)cc1CC1CCC1CSC.C12CCCC1CNC2=O 32450,c1(CNC(N2CCN(c3nccs3)CC2)=O)ccc(F)c(Br)c1 32451,C(=O)(C1=CC(C)(C)C1)NC(CCN(C(c1c(OC)nsc1)=O)C)C 32452,C1(NC(C(OC)OC)=O)CCN(C(=O)C2=CCC2)CC1C 32453,c1(C(=O)NC(C)CCCCNC(=O)Cc2cn[nH]c2)cnc2ncnn2c1O 32454,C=CC(CC)CC=O.N1(C(C)(C)C)CCCCC(C)C1.N12CCCC(C1)CC2=O 32455,c1(CC)nn(C)c(CC)c1C(=O)NCC=C1CCN(C(=O)C(C)S(C)(=O)=O)CC1 32456,c1(NCCC(N2CCCC(CO)C2)=O)ccc[n+]([O-])c1 32457,N1(C(CC)=O)CCN(C(c2cnn(C)c2Cl)=O)C(C)C1C 32458,C1(C2=CCCCCC2)(C(N(CCCNC(c2c(C)onc2CO)=O)C)=O)CC1 32459,C1(N(C(CCN(C(=O)CC=C(C)C)CC=C)=O)C)CCCC(O)C1 32460,c1(C(=O)NC(C2CCCN(C(c3csc(O)n3)=O)C2)C)cc(C#N)c(O)nc1N 32461,c1(C(=O)NC(CNC(c2ncn(CC)n2)=O)C(C)C)ccc(F)c(OC)c1F 32462,N1(C(C(C2CCCN(C(C(CCC)F)=O)C2)C)=O)CCn2ccnc2C1 32463,N1(C(C(C(=O)OCC)SC)=O)CCC(O)(CN(C)C(C2CCN(C)C2)=O)CC1 32464,c1(-n2cnc(NC(N(CC=C)C(C)C)=O)n2)cccc(C)n1 32465,C1(CC)CCCCCN1C(C1(c2c(F)cccc2F)CC(=O)C1)=O 32466,c1(NC(C2CSCCN2C(c2ccnc(Cl)c2F)=O)=O)cc(O)cc([N+](=O)[O-])c1 32467,c1(CCC(N2CC(NC(C(C(C)C)=O)=O)C(C)(C)C2)=O)cnc2ccccc2c1 32468,C1(C(=O)NC2C=CCN(C(c3ccccc3Br)=O)C2)CC2CC(O)C(C1)C2 32469,C=CCCCCCCC(=O)NCC1CC(F)CN1C(=O)CC1CC(F)C1 32470,N1(C(CC#C)=O)CC2C1CN(C(=O)Cc1ccc(O)c(F)c1)C2 32471,Brc1ccc2c(c1)CCN(c1cc[nH]c(=NCCc3ncccn3)n1)C2 32472,C1(NC(=O)CNc2cccc(Cl)c2-n2cccn2)CCc2ccccc2C1 32473,C12(CN(C(C3(CCC)CCC3)=O)CC)CCC1CN(C(=O)C1=CCCCC1)C2 32474,c1(C(C(=O)NC23C(CN(C(CC=CCC)=O)C2)C3)(C)C)ccc(Cl)cc1Br 32475,c1(C(N2CCC(N(CCC)C(c3ccoc3C)=O)C2)=O)occ(C)c1C(F)(F)F 32476,C(=O)(CC(C)C1CC1)NCC(CC)NC(=O)C(c1ccncc1)C 32477,N1(C(CCC2CCN(C)CC2)=O)CC2(NC(C3COC(=O)N3)=O)CCCC2(F)C1 32478,c1(OC)cc(OC)c(C(N2CCCC2CNC(=O)CC2CSC2)=O)c(N)c1 32479,Cc1cc(Br)c2ncnc(N3CCCC(c4ccno4)C3)c2c1 32480,Cn1cc(Cl)c(C(N2CC=CCC2C(=O)NCCC(O)C(F)F)=O)n1 32481,c1(C(=O)OCC)cc(CNCCc2cccc(SC)c2)c(C)s1 32482,N1(C(c2ccc(CSC)o2)=O)CC2CCC(C1)N2C(=O)CCC1CCCO1 32483,n1(CC(=O)N(C2CCC2)C)nnc(CNC(=O)CN2CCCC2C2(O)CC2)n1 32484,C1(CC(=O)NC2CCCC2)CC=CCC1.C(C(Cc1nn[nH]n1)CO)NC1C(=O)N1 32485,CC1CC(NC(c2ccc(=O)n(C)c2)=O)CN(C(c2cc(Cl)sc2Cl)=O)C1 32486,N1(C(COCCC)=O)CCC(NC(c2ccc(F)cc2SC)=O)C(CO)C1 32487,C(=O)(C(F)(F)CCn1ccnn1)NCC(C)(C)NC(=O)CC1CC(O)C1(C)C 32488,C1(NC(C(=Cc2ccncc2)C)=O)CCN(C(C2CC2C(F)F)=O)C1(C)C 32489,C1(NC(CC2C(CC)C2)=O)C2CCCN(C(=O)CN3CC(COC)C3)C2C1(C)C 32490,Cc1cccc(C2(C(=O)NCC=CCNC(c3ccc(NC(N)=O)cc3)=O)CC2)n1 32491,C12(CNC(c3ccsc3Cl)=O)CC(CN1C(=O)COCC1CCCC1)C2 32492,n1(CC)nc(C)c(C(N2CC(NC(C3(O)CCSC3)=O)C(SC)C2)=O)c1Cl 32493,C1(N2CCOCC2)(C(N(CCN(CCO)CC)C(C)C)=O)CCCC1 32494,C(C)(CO)(C(=O)NCc1ccccc1Cl)NC(CC=CC)=O 32495,C1(CNC(=O)C=Cc2ccoc2)CC2CCC1N2C(=O)CCc1cccc(F)c1 32496,c1(CC(=O)NCCCCCNC(C2C3CC3C3CC23)=O)cnc2ncccn12 32497,N1(C(c2n(COC)ncc2)=O)CCN(C(=O)C(F)(F)COC)CC(CO)C1 32498,Cc1ncnc(O)c1CC(N1CCC1CNC(C1(O)CC(F)(F)C1)=O)=O 32499,C1(C(=O)NC(C)CC(C)NC(C2(C#N)CC2)=O)OCC2COCCC12 32500,C1(CCC(N)=O)C(=O)N2CC(C)(C2)c2cn1nn2.C1(CC)(CC)COC1 32501,Cc1c(C(N2CC(OCCNC(=O)C(n3nccc3C)C)C2)=O)c(Cl)nn1C 32502,N1(C(c2cc([N+](=O)[O-])c[nH]2)=O)CCC2CN(C(=O)C(F)(F)c3ccccc3)CC12 32503,C1(CNC(C2CN(C(C)C)C2)=O)CC(C(=O)NC2C(CN(C)C)CCC2)CO1 32504,n1(CC)ccc(CC(N2CC(NC(c3ccsc3Br)=O)C2)=O)n1 32505,Cn1cc(C(=O)NC2CCCC2NC(C2COC(=O)C2)=O)c(=O)c(Br)c1 32506,CCC(C)N(OC)C(=O)C1CCC1CNC(=O)C=Cc1cocn1 32507,CC(C)C(CCCC(F)(F)F)NC(c1csc(C(F)(F)F)c1)=O 32508,N1(C(Cn2ncc(CC)c2)=O)CC(C2CC2C(=O)NC2CCN(C(C)(C)C)C2)C1 32509,c1(NC(C2N(C(C(C)=C3CCCC3)=O)CCC2)(C)C)cncc(OC(C)C)c1C 32510,c1(C(=O)NCC2(NC(c3c(CC)onc3)=O)CCC2)cc2cccn2cn1 32511,N1(C(C2(C)CCN(C(C3(N(C)C)CC3)=O)C2)=O)CC(CO)C2(CC2)C1 32512,c1(C(=O)NC23CCC(NC(=O)CC(F)F)(CC2)C3)noc2c1CCc1sccc1-2 32513,C(CC(C)C)(C(=O)NCC(c1ccccc1)CNC(=O)CSc1ccncc1)OC 32514,C(=O)(CCC(C(C)C)NC(c1cc(C(C)C)[nH]n1)=O)NC(C(=O)NCC(C)C)C 32515,C(=O)(C#CC1CCCOC1)NC1CC2CN(C(c3n(CC#C)ccc3)=O)CC21 32516,c1(C(C2CCCC2)NC)nnc(N2CCN(CCOC)CC2)n1CC1CCOC1 32517,c1(C(=O)NC2CCC(NC(C(C)SCC)=O)CC2)ccc(F)c(CC)c1 32518,C1(CCNC(C2N(CCC)CCC2)=O)CSCCN1C(=O)Cn1cc(C)cn1 32519,C(C(C(=O)N1CC2CC2C1)C(C)C)NC(C=CCCC)=O 32520,c1(NC(=O)Nc2c(CC)cns2)cc(-c2cccnc2)ncn1 32521,C1(NC(C(=O)NCCC=C)=O)CC(C)(C)C1OCC1CNC(=O)C1 32522,N1(n2c(C#C)ncc2)CCOC2(CCCN(C(=O)C(F)C(F)(F)F)C2)C1 32523,CC(O)C(F)(F)C(=O)N1CCC(N(CCO)C(c2cnn(C)c2C(C)(F)F)=O)C1 32524,C1(C=O)CC2(CCC2=O)C1.C12C3CN(CC13)ONC2=O.c1(OC)cnncc1N 32525,N1(C(c2c(COC)scc2)=O)CC(C2CN(C(=O)CN3CCCCCC3=O)C2)C1 32526,N12CC3(CC(C3)n3nnnc31)C2.c1(C(F)(F)F)cnc(C2CCC2)s1 32527,N1(C(C(C)NC(CC)(C)C)=O)CC2(CC(CNC(=O)Cc3ncc(C)s3)C2)C1 32528,c1(C(=O)NCCCC(C)NC(C2CC(CF)C2)=O)cccc(N)c1F 32529,N1(C(CC(C)SC)=O)CCN(C(c2cc(C)on2)=O)CC1c1cc(F)ccc1F 32530,C=CCC(C(=O)NCC1CCCO1)NC(=O)CC1OCCO1 32531,c1(C(=O)OC)c(NC(C2CCCN(C(=O)CC3CCCCO3)CC2)=O)sc(C)c1C 32532,CC(C)CC(C)CC(=O)N1CC(C)N(C(=O)Cc2cn(C(C)C)nn2)CC1C 32533,Cc1ncc(Cl)c(C(N2CCC(O)(CNC(C3CC4COCC4C3)=O)C2)=O)n1 32534,Cc1cc(C(N2CC(CCNC(C3(S(N)(=O)=O)CC3)=O)C2)=O)cnc1C(F)(F)F 32535,c1(C(N2CCC3(CN(C(=O)CCOC4COC4)C3)C2)=O)cc2n(n1)CCCC2O 32536,c1(C(=O)NCC2CCN(Cc3c[nH]c4cccnc34)C2)ccc2c[nH]nc2c1 32537,c1(C(=O)N(C2(C(=O)NC)CC2(C)C)CC(=O)NOC)cccc2[nH]ccc12 32538,c1(OC)nccc(C(N2CC(NC(=O)C=C(C)C)C(C(F)F)C2)=O)n1 32539,CC1CCC(C)(C)N1C(C1(C)CCN(C(C2CCC(CO)CC2)=O)CC1)=O 32540,c1(C(COC)COC)ccc(NC(c2c[nH]nc2NC(=O)CCC(C)C)=O)cc1 32541,CC1CCN(C(=O)Cc2csc(NC=O)n2)C(C)C1NC(c1ccncc1)=O 32542,c1(C(N2CC(N(C(c3cc(OCC)ncc3)=O)C)C2)=O)nc2cc(F)ccc2s1 32543,C1(C(=O)NCCCC(C)NC(c2cc(C(C)(F)F)on2)=O)Cc2ccccc2O1 32544,CC(C)(O)C(F)C(=O)NCC1CN(C(C2CC(=O)N2)=O)C1 32545,c1(C(=O)OC)ccnc2c1OCO2.c12cc(C)cnc1N1CC3(C1)CN(C3)C2=O 32546,c1(C(N(CCCNC(CCC)=O)CCOC)=O)ccccc1-c1ccccc1 32547,c1(C(=O)NCC2(F)CCN(C(c3c(C)cc(C)o3)=O)C2)c(C)nn(CCO)c1C 32548,c1(CN(C(CCC)=O)C)cnn2c1CN(C(=O)C=CCBr)CC2 32549,CC1CCC(NC(c2cccnc2O)=O)CN1C(=O)CC1(NC(N)=O)CC1 32550,CC(CN=c1[nH]c(=NCC2CC23CCCSCC3)[nH]c2c1CCCC2)c1ccsc1 32551,C1(OC)CCC(CC(N2CC3CC3(NC(=O)CC3CC(C)C3)C2)=O)CC1 32552,C1(CNC(CCC)=O)CCC2(CO1)CC(NC(C1Cc3cc(F)ccc3C1)=O)C2 32553,C1(CC(=O)NC(C)Cn2cc(CCN(C)C)nn2)CCC(C(C)(C)C)CC1 32554,N1(C(c2nc(C(C)OC)sc2)=O)CCCC1(C)CNC(c1ccnn1C)=O 32555,CC1(C)CC(C(N2CCN(C(C3CNC(=O)C3)=O)C(CO)C2)=O)C(C)(C)O1 32556,C12CCCC(C1)NC2=O.C1(C(CC)C)CN(C(=O)C(C)S)C1 32557,C1(n2cc(CC(=O)N(N3CCC3)C(CC)C)nc2)CCN(C(=O)OC(C)(C)C)CC1 32558,c1(C(=O)NC2CCCC(NC(c3c(N)c(F)ccc3)=O)C2)cccc2sccc12 32559,c1(C(N(C(C(C)NC(C2(COC)CCCC2)=O)C)C)=O)ccc2cnc(C)n2c1 32560,CCCCC(O)CC(=O)NC(C)(C)C=CC(N1CCCC(C)C1)=O 32561,N1(C(C2CCC(=O)N2)=O)CCCN(C(C23CCC2C3)=O)CC1 32562,C1(NC(CC(COC)C)=O)CC2CC1CN(C(c1ccncc1Br)=O)C2 32563,C(c1ccc(C(F)F)o1)=CC(=O)NCC(CCNC(Cc1cn(C)nc1)=O)O 32564,N1(C(c2ccc(OC)c(C)c2)=O)C2CCC1CN(C(=O)C(C)(C)C1CCCO1)C2 32565,N(C(=NCCCF)N1CCC(c2nccc(C(F)(F)F)n2)CC1)CCC1C(C)C1 32566,N1(C(c2ncc(CC)cn2)=O)CCCC(n2cc(C3CCOCC3)nn2)CC1 32567,CC(CCCc1cccs1)C(=O)N1CCC(NC(=O)C(C)Cc2ccccc2)CC1 32568,c1(OC)cc(C(N2C3CCC2C(NC(=O)CC2CCCN2C)C3)=O)c(Cl)cc1Cl 32569,Cc1ccc(F)cc1C(N1CCOCC1CCNC(C1(F)CCCN(C)C1)=O)=O 32570,C(=O)(C1=NOC(CNC(=O)NC2(n3nccn3)CC2)C1)Oc1c(C)cccc1 32571,Cc1cc2ccc1NC13CC(C1)(C3)C(=O)N2.n1(CCC(=O)N(C)C)cnc(=N)[nH]1 32572,C1(C2=CCOCC2)(C(=O)Nc2sccc2S(=O)(=O)N2CCOCC2)CC1 32573,C(=O)(C(CC(F)F)N(C)C(C1CC(O)C1)=O)NC(c1ncc(C)cn1)C 32574,c1(OCC)c[nH]nc1-c1nc(C)no1.C1(C(C2CCCC2)N)CCCCC1 32575,Cc1ccc(C(=O)NC2CC(NCC(=O)N(C3CCC3)C)C23CCC3)cc1O 32576,c1(CC)nc(C)c(C(=O)NC2(C)CCN(C(=O)CCC(C)SC)C2)c(C)n1 32577,C1(C(=O)NC(C#CC)CNC(=O)OC(C)(C)C)(CN)CCC(=O)N1.C(C)(C)(C)O 32578,c1(CC)nc(C)c(CC(=O)NCCCCNC(C2CS(=O)(=O)CCO2)=O)c(C)n1 32579,c1(OC)ccc(CCC(=O)NC2CCCCC2Cc2ccccc2)c(O)c1 32580,N1(C(C2N(CCCC)CCCC2)=O)CC(NC(=O)Cc2cc(C)nn2C)C(C)(C)C1 32581,C(=O)(C1=CCCN(C(=O)CC=C(Cl)Cl)C1)N1CC(C)(OC)C1 32582,C1(C)(C(=O)NCCN(CC(C)O)CCOC)CCN(S(C)(=O)=O)CC1 32583,c1(C(=O)NC(CC)CNC(=O)C=CS(C)=O)cnc2cnc(Cl)cc2c1 32584,N1(C(c2c(C)coc2)=O)CCC2(CCN(C(=O)CC3COCCOC3)C2)C1 32585,c1(C(N2C(CN(C)C(c3nccnc3N)=O)CCC2)=O)cncc2nc[nH]c12 32586,C=C(Cl)C(C)(C)C(=O)NCC1CCCN(C(c2ncn(C)c2C)=O)C1 32587,C(CC(O)CNC(c1n[nH]cc1Br)=O)NC(C1CC(C(=O)OC)C1)=O 32588,c1(CC)conc1C(=O)N(CCNC(=O)CC(O)c1ccccc1)C(C)C 32589,C1(C(=O)NCC2C(C)CC2)CCCCCN1C(C1COC(=O)N1)=O 32590,C(=O)(C(C)(C)C(=O)N1CCOCC1)NC1CC(N(C)C(c2cscc2F)=O)C1 32591,c1(C(N2CC(CNC(c3cc(C)on3)=O)C3C2C3)=O)cc(F)c(C#N)c(F)c1 32592,CC1CN2CCCC2N1C(C1CCN1C(C1COCC1C(N)=O)=O)=O 32593,c1(CC(C)NC(C2CC(CCNC(=O)CC3(N4CCCC4)CC3)C2)=O)cnc[nH]1 32594,C(CCCCNC(c1ccnn1CC(F)F)=O)N(C(CC1C(C#C)C1)=O)C 32595,c1(C(=O)NC(C2CCCN(C(=O)CCNC(=O)C=CCl)C2)C)ncnc(O)c1F 32596,CC(CO)(C1CCC1)NC(=O)NC1CCC1OCCCN 32597,C1(C(C)C(=O)NCC(C2CC2)C2CC2)CCN(C(=O)COC2CCCOC2)C1 32598,N1(C(C(C)OCCC=C)=O)CC(CO)C2(C1)CN(C(c1ccc(CCC)s1)=O)C2 32599,C=Cc1ccc(C(=O)NCCC2CCN(C(=O)CSC(C)(C)C)CC2)cc1 32600,C1(CCNC(c2c(C)nns2)=O)CCCCN1C(=O)CCC1CCOC1 32601,N1(C(CCC(=C)Cl)=O)CCN(C(c2ncc(F)cc2N)=O)C2CC12 32602,C=C(Br)CCC(=O)N1CCN(CCCNC(c2snnc2C)=O)CC1 32603,c1(CC(=O)N(CCNC(CCC(C)OC)=O)C(C)C)cc(Cl)ccc1[N+](=O)[O-] 32604,N1(C(C=C(CCC)CCC)=O)CC2CCC(C1)N2C(=O)C1=CC(C)(CC)C1 32605,C1(N(C(CCNS(CC)(=O)=O)=O)Cc2ccn(C)n2)CC2CCC(C1)N2 32606,C1(NC(C2(OC)CCCCC2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)CC1C 32607,n1(C(C)C)ccnc1C(=O)NC(C)(C)CC=CC(=O)NC1(c2cccnc2)CC1 32608,S(=O)(=O)(c1cc(C)ccc1Br)NC(=O)CC1(C)N(C(=O)C(F)(F)F)CC(OC)C1 32609,c1(C(N2CC3C(NC(C=CCOC)=O)CC(C3)C2)=O)ccc2cc(Cl)ccc2n1 32610,c1(C(=O)NC2CCCC(N(C(=O)C3=CCCOC3)C)C2)cccc2nccn12 32611,Cc1nnc(CCC(=O)NC2(CCNC(c3ccc(Cl)cc3)=O)CCC2)n1C 32612,C(=O)(CCC(C)(C)NC(c1cccc(F)c1N)=O)N(CC(C)(O)C1CC1)C 32613,N1(C(=O)NC2C(CC)CCCC2)CCC(C#N)(NC(c2cc(F)cc(I)c2)=O)C1 32614,C(CCO)(C(C)(C)O)NC(c1cc(COC)on1)=O.C12(CCCC1)C(=O)NC2 32615,CCC(O)C(F)(F)C(=O)N(C)CC1CN(C(=O)C(C)CCCc2ccccc2)C1 32616,c1(NC2CC(C)CN(C(c3ccncc3)=O)C2)ncc2cc(Br)ccc2n1 32617,N1(C(Cc2c(C)noc2C)=O)CCC2C(NC(c3c(C)nn(C)c3Br)=O)CC12 32618,Cc1cc(Cl)ccc1C(N1CC(CNC(c2cnc3n2CCC3)=O)C2(CC2)C1)=O 32619,c1(C(=O)NCC23N(C(C(C)=C4CCC4)=O)CC(C2)C3)ccc(C)cc1N=[N+]=[N-] 32620,c1(C(N(CCNC(=O)COc2ccc(C)cc2)CC)=O)nccc2c1NCCC2 32621,c1(N2C(CNC(=O)C(C)(C)SC)CC(OC)C2)ncc([N+](=O)[O-])cn1 32622,CC(C)(C)CC(=O)NCC12COC(CNC(=O)CSc3cccc(F)c3)(C1)C2 32623,c1(COC)nc(NC(C)C(OC)OC)cc(N2CCC(CCCO)CC2)n1 32624,N1(CC(N2CC3C(NC(CC4(NC(C)=O)CCCC4)=O)(C3)C2)=O)C(=O)CCCC1=O 32625,c12ccccc1N2.C(=O)(CCC(F)F)NC(CSC1CN(C(C(C)(C)C)=O)C1)=O 32626,C1(C(N2CC(O)(CN(C(c3c(C)cc(CC)o3)=O)C)C2)=O)CCCCCN1C 32627,CC1OCCCC1C(=O)N(C)CCN1CCN(C(=O)CC2OCCO2)CC1 32628,Cc1cc(=NC2CN(Cc3nc(O)n[nH]3)C2)[nH]c(NCC2CCOC2C)n1 32629,CCC(CC)CCCNC(=O)C(O)CNC(=O)C=Cc1cc[nH]n1 32630,C(C(C)C)(C(O)C(=O)NCC=CC(=O)NCC1CCC(C)(C)CC1)OC 32631,C1(C(=O)NCc2occ(C)c2)CCC(C)N(C(C2OCCOC2C)=O)C1 32632,N1(C(c2cc(COC)no2)=O)CCC2(CCCCN(C(=O)C(C)C(F)F)C2)C1 32633,Cc1cc(N)cnc1C(=O)N(CC(O)CN(C)C(c1cnsc1C)=O)C 32634,CC1CC(NC(c2cnc(-c3cccnc3)s2)=O)CN(C(=O)CC2CC=CC2)C1 32635,C(C)(C)(CCC(=O)NCCCCOC(C)C)NC(C(COCC)C)=O 32636,C1(CC(C)NC(C(C)OC(C)C)=O)CCN(C(=O)CSc2cccc(Cl)c2)CC1 32637,C1(NC(c2cn(CC=C)nn2)=O)CCC(C)(CNC(c2cc(C)ns2)=O)C1 32638,C12(NC(c3cnn4ccn(C)c43)=O)CCCCC1CN(C(=O)Cn1cncn1)C2 32639,N1(C(C(CC=C)C)=O)CCC2CN(C(=O)Cc3ccccn3)C(C)C12 32640,C(CCC(C(=O)N1CCN(CCF)CC1)NC(=O)CC(C)n1cccc1)OC 32641,C1(C(N2CC(N(C)C(c3cnn(C)c3)=O)C(C)(C)C2)=O)(OC)CCCCCCC1 32642,C1(C(=O)NCC(C(C)C)NC(C2CCN(C)C2=O)=O)CC(=O)OC1(C)C 32643,C1(C(=O)NCC2N(C(c3c(SC)scc3)=O)CCCCC2)CSc2ccccc2O1 32644,CC1(C)OC2CC(C(N3CCC(C)(CNC(=O)Cc4ccsc4Cl)C3)=O)CC2O1 32645,n1(CCCNC(CCC)=O)cc(CN(C)C)nn1 32646,N1(C(CS(CCOC)(=O)=O)=O)CCC2(CC1)CN(C(C1CCC1OC)=O)CCO2 32647,C1(NC(=O)NCC(C)(C)CS(C)(=O)=O)C(C(=O)O)C2CCCCCCC12 32648,CCCC(CNC(=O)CC1CC(C)=NO1)NC(=O)C=C(C)C(C)C 32649,C1(NC(c2ccc(C)cc2C)=O)CN(C(=O)Cc2csc(C)n2)C2(CCCC2)C1 32650,C1(NC(C2N(CC)CC2)=O)CC2CCC1C(NC(c1cc(C#N)cs1)=O)C2 32651,c1(C(=O)NCC(C)O)ccc2c(c1)CCN(Cc1ccc(F)nc1F)C2 32652,c1(C(N(CCCC)C(=O)C2CC2)=O)ccc(O)cn1.N1(C(C(=O)N)C2CC2)CCOCC1 32653,CCCC(C)(c1nnnn1C(C1(C)CC1)C)NC1CCC1(C)C 32654,C1(NC(CCn2c(C)cc(C)n2)=O)CC2CCC(C1)N2C(c1ncccc1C)=O 32655,c1(CC)oc(C)cc1C(=O)N(CCCC(=O)NCCC(F)F)C 32656,c1(C(=O)NC2CCCN(S(=O)(=O)C(F)F)C2)cc2nc(F)ccc2o1 32657,Cc1sc(=O)n(CC(N2CC(O)(CNC(C3CCC(C)CC3)=O)C2)=O)c1C 32658,N1(C(=O)CCCc2ccccn2)CCC2CCN(C(=O)CC34CCCC3C4)C2C1 32659,c1(C(=O)NC(C)C(CO)NC(C2CCCS2)=O)cccc(-c2ccsc2)c1 32660,C(=O)(C1CCCc2nnn(C)c21)N1CCCN(C(C(C2CC2)OCC)=O)CC1 32661,N1(C(C(n2c(C)cc(C)n2)C)=O)CC2(CNC(C3CCC(=O)N3)=O)CC(F)(C1)C2 32662,CC1(C)CCOC1C(=O)NC1COCCC1C(=O)NCCOCC(F)F 32663,c1(C(N(C(C)CNC(=O)CCCc2cncs2)C)=O)cc2c(O)ncnc2cn1 32664,Cc1cc(NC(c2ncoc2CNC(C2(C#N)CCOC2)=O)=O)cc(CO)c1 32665,C(=O)(C1Cc2ccc(C)cc21)N1CCN(C(CNC(CCC)=O)=O)CC(O)C1 32666,N1(C(C(C=CCCC)O)=O)CC2(CCN(C(c3c(C)occc3=O)=O)CC2)C1 32667,N1(C(CN(C)CC)=O)C2CCC1CC(CNC(c1cnn(C)c1CC)=O)C2 32668,C(=O)(C(C(C)(C)C)OC)NCC(CN(C(CCSc1ccc(OC)cc1)=O)C)C 32669,C(=O)(C(F)CC(C)C)NCC(CC)(C)NC(C)=O.C12CCN(CC1)C2=O 32670,C=CC(CC)CC(=O)N1CCC(C)C(NC(=O)C=Cc2cnc(OC)cn2)C1 32671,C1(NC(CCn2ccc(C)n2)=O)C2CC3CN(C(C4OCCCO4)=O)C1C3C2 32672,C1(C(=O)NCCCN(C)C(C2(CCO)CC2)=O)CC12CCC(=O)CC2 32673,C1(NC(=O)CN2CCOCC2=O)CC(C2CC2)N(C(=O)COCCF)C1 32674,C(=O)(CC(O)CCSC)N1CCC1Cn1cc(-c2cn(CCC)nc2)nn1 32675,C12(NC(c3nc(C(C)C)oc3)=O)CCCN(C(=O)C3=CCC3)CC1C2 32676,c1(CNC(C2CCCCO2)=O)cccc(Cn2cc(CNC3CCOCC3)nn2)c1 32677,c1(NC)c(C(=O)NC(C)(C)C(C)NC(c2ccccc2SC)=O)cccc1F 32678,c1(SC)cccc(C(N2CCOC(C3CN(C(=O)C(C)C4CCCC4)C3)C2)=O)c1 32679,CC1(C(=O)O)CN(C(c2cc3cccnc3s2)=O)CC1(F)F 32680,N1(C(Cc2nnc(C)o2)=O)CCC(NC(=O)CCC2CCCN(C)C2)CC(O)C1 32681,c1(N(c2nccc(N3CCCC3)n2)C(C2CNCCOC2)=O)cc([N+](=O)[O-])cs1 32682,c1(CNC(CC2N(C(CS(CC)=O)=O)CCCC2)=O)c(C)cccc1F 32683,C1(C)(C(=O)NCCN(C(C2CCc3ncnn3C2)=O)CC)CC(C2CC2)=NO1 32684,N1(C(C(C)(C)OCC)=O)CCN(C(c2c[nH]cc2CC)=O)CC(O)C1 32685,O=S(=O)(c1ccc(CO)cc1OCCCC(=O)O)N1CC=CS1(=O)=O 32686,c1(C(=O)NCC2(C)CCCN2C(c2cc(C(N)=O)c[nH]2)=O)ccn2ccnc2n1 32687,Cc1onc(-c2cccc(Cl)c2)c1C(=O)N(C)CCNC(c1coc(Cl)n1)=O 32688,c1(NC(C2C(CNC(Cc3n(C)ccc3)=O)C2)=O)cnc2[nH]cnc2c1 32689,c1(C(N(C(C)C)CCN(C(=O)CCOC2CCOC2)C)=O)cc(Cl)ccn1 32690,c1(-c2cn(CC3N(C(CC(CC)C(F)F)=O)CC3)nn2)ccc2nccnc2c1 32691,C(=O)(CCS(=O)(=O)c1ccc(OC)cc1)NCC(C)NC(C(CCCC)(C)F)=O 32692,c1(C(C(=O)NC)N(CC)Cc2cccc3ccsc23)ccc2c(c1)CCOC2 32693,N1(C(Cc2cc(C)no2)=O)CCCC(C2CC2NC(c2cc(C(N)=O)c[nH]2)=O)C1 32694,c1(C(=O)NC2CN(C(C3CCN(C)C3)=O)CC2F)cccc2c1CCC2 32695,N1(C(C2C(C)(C)C2(F)F)=O)CCCC(C2(NC(=O)CCC3CCCN3C)CC2)C1 32696,c1(C(N2CC(OCCNC(C3C(C)(C)OCC3)=O)C2)=O)n[nH]c2ccc(Cl)cc12 32697,c1(C(=O)NCCCN(C(C(COC)N(C)C)=O)C)ccc2c(c1)C(C)CO2 32698,C1(C(=O)NC(C(=O)NCCCCN=[N+]=[N-])c2ccoc2)CC2(C1)CC(O)C2 32699,C1(C(N2CCC(NC(c3c[nH]c(C(F)(F)F)c3)=O)(CO)C2)=O)C(C2CC2)C1(F)F 32700,c1(-c2c(C)cc(C(N3CC(C)(C)OCC3C3CC3)=O)s2)ccc2c(c1)ncn2C 32701,CCC(C(F)F)NC(=O)CC(C1CC1)NC(=O)CC1CC(OCC)C1 32702,CC(C)C(C)C(CNC(c1cc(=O)n(C)o1)=O)NC(=O)CC1CCCCC1 32703,N1(C(C(C)(C)NC(C)=O)=O)C(CC(N2CC(O)(C(N)=O)C2)=O)C2CCCC12 32704,C(=O)(C1=CC2(CCOC2)C1)NCC1(NC(C2CC3(CSC3)C2)=O)CCCCCC1 32705,Fc1ccc(Cl)c2oc(CNC(=NCC3CCOC3)NCC3CCCO3)c(C)c12 32706,N1(C(=O)Nc2c(C)c3c(cn2)cccc3)CCOc2cc(Cl)ccc2C1 32707,c1(C(=O)NCCC(C)NC(=O)Cc2cnsc2)cccc(N)c1 32708,C1(C(=O)NCC(C2CC2)NC(c2scc(C)c2Br)=O)CCn2nnnc2C1 32709,C1(NC(Cn2ncc(C)c2)=O)C2CC1N(C(=O)CC1CC3(CCC3)C1)C2 32710,CC(=O)C(C)(C)CC(=O)NCC1(C(=O)NC2CS(=O)(=O)C2)CC1 32711,C1(C(=O)NCC(C2CCC2)OC)(CNC(=O)CNC2CCCO2)CCCO1 32712,C1(CC=C)(NC(=O)CC(C)CF)CCN(C(=O)C=Cc2ccccc2)CC1 32713,c1(C(C2CC2)NC2(CC=C)COC2)nnnn1C(C)CC 32714,C1(NC(Cc2c(C)sc(Br)n2)=O)CC2CC(C1)N(C(C1CN(C)C1)=O)C2 32715,N1(C(C2C(C=C)C2)=O)CCC2(CC1)CCN(C(C1CCCC1(C)C)=O)CC2 32716,C1(=O)C(N2CCCC(CC(=O)OC(C)(C)C)C2)C(C)N1.C(CNC(C)=O)OC 32717,C(=O)(CCCN(C)N=O)NC1(CC)CCCN(C(=O)Cc2ccc(Br)cc2)C1 32718,N1(CC)CCCC(ONC(=O)CC2C=NN(C)C2=O)C1.C1(=O)C(C)(C2CCC2)N1 32719,c1(CCCCC(=O)NC2CC(CNC(=O)CCc3ccoc3)C2)ccc(Cl)cc1Cl 32720,CC1(NC(C2CCN(C(CNC(=O)CNC(=O)C(F)(F)F)=O)C2)=O)CCCC1 32721,C#Cc1ccc(NC(=O)C(F)C(C)CNC(C2CC(F)(F)C2)=O)c(C)c1 32722,CC(F)(F)C(F)C(=O)NCc1ccc(C(=O)O)s1.C1C(=O)N1 32723,Cc1nccc(C(N2CCC(CNC(=O)CCOCC3CC3)C2(C)C)=O)c1O 32724,C1(NC(c2cc(COC)[nH]n2)=O)C2CC(CN(c3nnc(C4CC4)s3)C2)C1CO 32725,C1(CNC(C(=O)NCCOC)=O)CC(C(=O)N2CCC(CO)(OC)C2)=NO1 32726,C=CCC(CNC(c1cnn(CC)c1C)=O)C(=O)N=c1cc(C)n(C(C)C)[nH]1 32727,CCCCC(C)CCC(=O)NCC1(CNC(c2cc(C)c(N)cc2Cl)=O)CCC1 32728,C1(CNC(C2CC(=C3CC3)C2)=O)CN(C(C2CC(F)(CF)C2)=O)CCCO1 32729,C(=O)(C(C)CCCc1cccs1)N1CC(N(C)CC)C1.C1(=CC=O)CN2CCC1CC2 32730,c1(NC(C)=O)ccc(C(F)(F)F)cc1.C12CCN(C1)C(=O)CSC(C)C(=O)N2C 32731,C(=O)(C(C)S(N)(=O)=O)NCC(C)(C)NC(C(CC)OC)=O 32732,N1(C(C(c2cccs2)SC)=O)CCN(C(=O)Cn2nnnc2C2CC2)CC1C 32733,c1(C(N2CCC(C)C(CNC(=O)CCc3ccoc3)C2)=O)scc2c1CCCC2 32734,C1(C)(CC)CC(NC(c2ccccc2C)=O)CN1C(c1c[nH]nc1OC)=O 32735,N1(C(c2ccc(CC)cn2)C(=O)NC2CC(F)(F)C2)C(C)CCC1(C)C 32736,C1(OC)CC2(C1)CN(C(c1csc(CNC(C3(CF)CC3)=O)c1)=O)C2 32737,c1(C(=O)NC(CN(C(c2ccn(CC)n2)=O)C)C)ccc(C2CCC2(C)C)cc1 32738,CCC(C)C(C(=O)N1CCC(O)CC1C(N1CC(F)(CC)C1)=O)OC 32739,C(CC1=CCN(C(c2cc(N)nc(Cl)c2)=O)CC1)NC(C(N1CCSCC1)C)=O 32740,C(CC(C(=O)NCC1CCOC1=O)NC(=O)C(Br)=C(C)C)SC 32741,N1(C(c2ccccc2)=O)CCCC(C2CCCN(C(C3CC(O)CN3)=O)C2)C1 32742,N1(C(COCC)=O)CCCC(C)(CNC(=O)C2=CCCC2C)C1 32743,C=C(C)CCC(=O)NCCCN(C(C1CCN1S(C)(=O)=O)=O)Cc1cccnc1 32744,c1(C(=O)NCCCNC(CC(C)c2ccncc2)=O)ncc(Br)cc1N 32745,c1(C(N2CCC(F)(CNC(C3CC4(CC4)C34CC4)=O)C2)=O)ccc(Cl)c(F)c1 32746,C1(C(=O)NC2(CCOC)CCC2)CC1C1CN(C(C2CCSCC2)=O)C1 32747,N(C(=NCC1CC1Cl)NC1CCCC1)C(C1(OC)CC1)C 32748,Cc1ccc(C(=O)NC(C)CCN(C(=O)COCC2CCCO2)C)c(N)c1F 32749,c1(CCCC(=O)N(C)Cc2cn(CC3CCCCC3F)nn2)ccccc1Cl 32750,C1(NC(c2coc(-c3ccsc3)c2)=O)CCN(C(C2CC2C(F)(F)F)=O)CC1C 32751,c1(C(=O)NC2CC(NC(c3ccc(COC)cc3)=O)C2)csc2cccnc12 32752,C(=O)(C(O)C(F)(F)F)NC(=O)CC(C)(C)C.CC1CC2(C1)CC2 32753,CCC(Cc1ccccc1)C(=O)N1CC(C)(CC(F)(F)F)C1.C1(=O)CCC(=O)N1 32754,Cc1nc(O)ccc1C(N1CCC(C)C1C(=O)Nc1cnn(C(C)C)c1)=O 32755,C1(NC(CC(C)OC)=O)CCN(C(c2cnncc2C)=O)CC12CCC2 32756,c1(OC)ccc(C(=O)NCC2CN(C3CC3)C(=O)O2)nn1 32757,CCCC(F)C(=O)NCCOCCCN(C)C(C1CCC1C#N)=O 32758,C(c1cnn(C)c1)=CC(=O)NCC1C(C(NOCCOC)=O)CCO1 32759,CC(C)CC(CC(=O)NCC1(O)CCN(C(=O)C(F)OC(F)(F)F)CC1)CC(N)=O 32760,CN1CC(c2cn(C3CN(C(=O)C4=NNC(=O)C4)C3)nn2)CCC1C(F)(F)F 32761,c1(C(C)NC(N2C3CC(C(=O)OC)CC2CC3)=O)nc2ccc(C)cc2[nH]1 32762,C1(CNC(C(C)(C)SC)=O)CN(C)CCN1C(c1cc(Cl)sc1Cl)=O 32763,C1(=CCNC(C(C)C2CCOC2)=O)CCN(C(=O)CN2CCCCCC2)CC1 32764,CC(F)(F)C(C)(C)CC(=O)N1CC(NC(c2cccc(O)n2)=O)CC12CCC2 32765,C(=O)(C1Cc2ccccc21)NCC(CCCC)NC(=O)CC1(OC)CCOCC1 32766,c1(C(N(CCC(=O)NCCSC)CCC)=O)cn(C2CC2)nc1C 32767,N1(C(=O)NCc2nc(N(C)CC)sc2)CC2(CCC(C(=O)O)O2)C1 32768,C1(C(N(CCCNC(c2ncccc2F)=O)C2CC2)=O)CCC2(CC2)C1 32769,C1(O)(CN(C(C2CCN(C)C2)=O)C)CCN(C(=O)CCc2cnn[nH]2)CC1 32770,c1(NC(c2ccn(CC)n2)c2nnnn2Cc2cccs2)cccc2[nH]ccc12 32771,C1(C)(COC)CC(NC(=O)CCc2cnc[nH]2)CN1C(C1CN2CCN1CC2)=O 32772,CCCC(CCC)NC(=O)CC1CN(C(c2ccsc2)=O)CCO1 32773,c1(C(N(CCN(C(C2C(CCOC)C2)=O)C)C)=O)cncc(Cl)c1C 32774,N1(C(c2c(CC)scn2)=O)CC2CC(C)N(C(c3cn(C)nc3Br)=O)C2C1 32775,c1(-n2cc(C3C(OC)CN(C(=O)CCCN=[N+]=[N-])C3)nn2)cc(F)ccc1Cl 32776,c1(C(N2CC3(CC(NC(C4CC4CF)=O)C3)C2)=O)ccc2nc(O)oc2c1 32777,C#Cc1cc(F)c(CN2CCN(C)C(CO)C2)c(F)c1 32778,N1(C(c2c(C)n(CCC#N)nc2)=O)CC2CCCC2(NC(=O)C(F)=CCCF)C1 32779,C1(C(=O)NCC#CCNC(c2cscc2C(F)(F)F)=O)CC2(CC2)CO1 32780,c1(N(C(C(C)Sc2ccccn2)=O)CC2CCCO2)ccnc2ncnn12 32781,CC(C)(Cc1ccccc1)C(=O)N1CCCC1CC(=O)Nc1c[nH]ccc1=O 32782,C1(C)(C(=O)NCC(COC)OC)CCCN1C(c1c[nH]c(=O)cn1)=O 32783,C(=O)(N=c1ccn(CC2CC2)[nH]1)C1C(=C)C1.N1CC(C)(CCC(=O)OC)C1 32784,C(=O)(CCCCN=[N+]=[N-])NCC=C(C(N1CCC(C(=O)OC)CC1)=O)C 32785,Cc1cc(C(=O)NC2C3CC2N(C(=O)C(C)OCc2ccncc2)C3)cc(C)n1 32786,N1(C(CC=CCOC)=O)CCC2(CC(NC(=O)C(c3c(C)cccc3C)O)C2)C1 32787,Cn1nncc1CC(=O)NCC(C)(O)CNC(=O)Cn1cc(NC(C)(C)C)cn1 32788,c1(C(N2CCC(C(N(C3CC3)CC)=O)C2)=O)ccc(CO)cn1.c1(C=O)cncs1 32789,C1(NC(c2ccsn2)=O)C2CC3C1C3C2C(N1CC(n2cccn2)C1)=O 32790,N1(C(c2c(OC)noc2C)=O)CCCC(N(C(=O)CCCSC)C)CC1 32791,C(=O)(C(O)C(F)(F)F)N(C)CC1COCCN1C(=O)C1=NOCC1 32792,c1(C(=O)NCC2(CN(C(C3(C(=O)O)C(C)C3)=O)C)CC2)ccc(OC(F)F)nn1 32793,c1(N(C)CCn2cccn2)ccnc(NC(C2CCCO2)C)n1 32794,C1(N(C(C2(CC)CCC2)=O)C)CC2CCC(C1)N2C(c1occ2c1CCC2)=O 32795,C1(OC)CC(C(=O)NCC2CC3CC3C2)(NC(=O)CC2CCCC2C)C1 32796,C=CCCCCCCCCC(C(=O)NC1CCC1)N(C)CCc1cnn(C)c1C 32797,N1(C(C(CC2CN(C(CC=CC=CC)=O)C2)F)=O)CCc2c(C)cccc21 32798,N1(CC)CCC(C(=O)NCC(c2ccccc2)NC(=O)CC2CC(=O)C2)C1 32799,c1(CNC(C(C2CC2)SC)=O)cn(CCCNC(=O)CN2CCCC2)nn1 32800,c1(C(=O)NCC2CCCN2C(C(C)CN2CCOCC2)=O)cccc(O)n1 32801,S(=O)(=O)(c1ccc(Br)cc1)NCC(=O)NCCNC(c1cccc(CO)c1)=O 32802,N1(C(c2c(CSCC)cccc2)=O)CC(C2CN(C(=O)CCCCC(N)=O)C2)C1 32803,N1(C(c2cnc(Br)n2C)C(=O)NCC)CCCC(CN2CCCC2)C1 32804,N1(C(=O)OC(C)(C)C)CC(C(=O)O)C(C2CCOCC2)C1.C1(CN)C(C)(C)C1(C)C 32805,c1(CC(=O)NC(CC)CN(C(=O)C(CCC)SC)C)cc(F)ccc1C 32806,N1(C(c2ccc(CC)c(O)c2)=O)CCCN(C(=O)C(C)NC(C)(C)C)C(CO)C1 32807,c1(-c2cc(C(=O)NCC(CC=C)NC(=O)C(C)NC(C)=O)no2)ccc(O)cc1 32808,C(C(C(C)(C)C)NC(C1(C)CCCO1)=O)NC(=O)Cc1csc(C(F)(F)F)n1 32809,CCC(C)(C)CCNC(=O)C=CC(C)(C)NC(=O)C(C)C(F)F 32810,c1(CCC)ccc(C(NC(=NC)NCc2nc(-c3cccs3)n[nH]2)C)cc1 32811,Cc1c(CC(C)NC(CC(C)C)c2nnnn2C2CCCCC2)cccc1Br 32812,N1(C(C2C3(CCN(C(C4CN(C(C)=O)C4)=O)CC3)C2)=O)CCCC(C2CC2)CC1 32813,C(CCF)(C(=O)N(CC(=O)N(c1ccccc1)C1CC1)C)NC(C(CC)C)=O 32814,C(=O)(C1=C2CCCN=C2NN1)NC(CCCOC)c1ccccc1 32815,C1(C(N2CCC(=CCNC(C(CCC)NC(N)=O)=O)CC2)=O)CCCS(=O)(=O)C1 32816,C1(COC)CN(C(c2cc(C#N)oc2C)=O)CCN1C(=O)C1=C(Cl)CCC1 32817,C1(NC(C=C(C)CNC(C2OCCC2C)=O)=O)CCn2nnnc2C1 32818,C(c1cncnc1O)=CC(N1CCC(C(C)NC(=O)CC(F)(F)F)C1)=O 32819,N1(C(c2c(C)nc(C)o2)=O)CCOCC(C)(CNC(C2CCCCC2CF)=O)C1 32820,N1(C(Cc2n(C)cnc2)=O)CCOC(CCNC(C2CC(n3cccn3)C2)=O)C1 32821,C1(CC)CCC(C(=O)N(CC(C)O)CCN(C(=O)CCc2csc(C)n2)C(C)C)O1 32822,N1(C(C(C(C)C)C#N)=O)CC2CCC1(CNC(C1CC3(CCC3)C1)=O)CC2 32823,c1(C(=O)NC(CCCNC(C(CCC)O)=O)C2CC2)cc(F)cc2c1NCCC2 32824,C1(C(=O)NCC(CN(C(=O)CCC2CC2)C)O)CCCC1P(C)(C)=O 32825,c1(C(=O)NCC2(CNC(C3C(C)CCS3)=O)CCCC2)cc2ncn(C)c2cn1 32826,c1(CC(=O)NC(C2CN(C(=O)CCCNC(N)=O)C2)C)ccc2nonc2c1 32827,Cc1cc(C(C(=O)NC2CCCC2)N(C)CC2CCN2C(C)(C)C)c(C)cn1 32828,Cc1nn(C2CCCCC2)c(C)c1S(=O)(=O)Nc1cc(Br)nn1C 32829,CC(C(C)(C)C)=CC(=O)NCCCOCCC(=O)NCC1=CCCC1 32830,c1(C(N(C(C)(C)C)Cc2cccc(OCC#C)c2)=O)cc2nc(F)ccc2o1 32831,C1(CNC(CCc2onc(C)n2)=O)CN(C(=O)CCc2ccco2)C2(CCC2)C1 32832,[N-]=[N+]=NC1CCCN(C(c2csc3ccc(Br)cc23)=O)C1 32833,C(c1cnc2ccccc2n1)=CC(=O)NC1C2CN(C(C(C)(C)CO)=O)C1CC2 32834,c1(C(=O)NCCC(C)N(C(c2ccccn2)CC)C)cc(Cl)cs1.C1(=O)CCN1 32835,Cc1cc(C)c2cc(C(=O)N(C3CCN(C(C4CCC(=O)C4)=O)C3)C)[nH]c2c1C 32836,C1(C(N(C)CC2CN(C(C3(O)CCCCC3)=O)CCO2)=O)(CF)CCC(O)CC1 32837,C(=O)(CCC(C)CN1CCCC1)NC1CN(C(c2ccc(CC)[nH]2)=O)C1 32838,C(c1cccc(F)c1)=CCC(=O)NC1COCCC1NC(c1cccnc1)=O 32839,c1(OC)ncnc(C(=O)N(C2CCCN(C(=O)C(F)(F)C(O)C3CC3)C2)CC)c1F 32840,Cc1cc(C#N)cnc1C(N1CC=CC(C(N2CCCC(C)C2CO)=O)C1)=O 32841,N1(CC(=O)NC2CCOC2C(N2CC(N3CC(F)C3)C2)=O)CCC(F)C1 32842,N1(C(CC(CC=C)(C)C)=O)CC(NC(C2CC2(F)F)=O)C2(CCOCC2)C1 32843,c1(C(N2CC(C=C)C(NC(c3[nH]nnc3C)=O)C2)=O)nn(C)c2c1C(O)CCC2 32844,N1(C(c2cnc(C)n2C)=O)CCn2ncc(CNC(C3C=CCC3)=O)c2C1 32845,N1(C(C2C(C)CC(=O)N2)=O)CCC2(C1)CN(C(=O)CC1CCCC(F)(F)C1)C2 32846,c1(CNC(=NC)N(C)Cc2ncnn2CC)cccc2c1OCCO2 32847,c1(C(=O)NC2C(C(=O)C(F)CSC)C2)ccc(OC)cc1.C(C(=O)NC)OCCC 32848,CC(CC(C)(C)C)C(=O)NCC1CCC(C)(C)CN1C(=O)CCC(=O)N(C)C 32849,C1(C(N2CC(F)(CNC(C3OCCN(C)C3)=O)C2)=O)CC2CCC1CC2 32850,n1(C(CC)C)ncc(C(N2CC(N(C)C(c3nnc(C(C)(C)C)s3)=O)C2)=O)c1C 32851,N1(C(c2nc(C)sc2)=O)CCC(C(F)(F)F)CC1CNC(=O)C(F)(F)C(F)F 32852,C(=O)(C(C)(O)C(F)(F)F)NC1CCN(CCCc2n(C)nnn2)CC1F 32853,C(=O)(C(C)CC(F)(F)F)NCC1CN(C(c2c(C(C)=O)cn(C)n2)=O)CC1(F)F 32854,N1(C(C2N(C)C(=O)NC2)=O)CCC(CO)(NC(c2ccc(F)s2)=O)CC1 32855,CCC(CC)CCCC(=O)NC(C1CCCC1)CNC(C1CC(=O)N(OC)C1)=O 32856,N1(C(C(CC(C)C)O)=O)CCc2nc(O)cc(C(=O)NCCc3nccs3)c2C1 32857,C(=O)(CCCS(N)(=O)=O)NCC1CC(NC(C=Cc2ncc(C)[nH]2)=O)CC1O 32858,N1(C(Cc2c(OC)ccnc2)=O)CCOCC(NC(C2CCCC(OC)C2)=O)C1 32859,c1(CNC2CN(c3cc(OC)ncn3)CC2C)cc(Br)ncc1Br 32860,C(=O)(C(CC(C)(C)C)OC)NC1C(OC)CN(C(=O)CSC2CC2)C1 32861,c1(C(N(C(C)CNC(=O)Cc2cn3ccsc3n2)C)=O)cc(F)c2cn[nH]c2c1 32862,Cc1nc2sccn2c1C(N1CCC(C)(CNC(C2CC3CC3C2)=O)C1)=O 32863,C1(CNC(CC(C)(C)C)=O)CN(C(=O)CSc2ccccn2)CCCO1 32864,c1(C(=O)NCC(C2CC2)NC(CC2(C#N)CCC2)=O)ccc2nc(O)[nH]c2n1 32865,C1(NC(=O)CCc2ccccn2)C2CC3C1C3C2C(=O)NC(C1CC1)C1CC1 32866,C(=O)(C(C(C)C)n1cc(Br)cn1)N(CCCNC(=O)CSC(C)C)CC 32867,CC(=NOCC#N)C(=O)N1CCN(CCN(C(=O)Cc2cc(C)[nH]n2)C)CC1 32868,N1(C(CCC)=O)CC(OC)CC1(C)CNC(c1ccc(C)nc1O)=O 32869,C1(CSC)CCCN(C(=O)Cn2cc(C3CCCCNC3=O)nn2)CC1 32870,C1(O)(NC(CC(=O)NCC#C)=O)CCN(C(=O)COCCCC(C)C)CC1 32871,C1(CNC(c2nnc(CCC)o2)C)(OC(C)C)CCCOC1 32872,C(C(C)(O)CC(=O)N1CC2(CC2)CC1CC(=O)NCC(C)CO)OC 32873,N1(C(COCc2c(C)ncs2)=O)CCC(C)C(NC(C2CC(C)(C)C2)=O)C1C 32874,c1(C(=O)NC2C(NC(C3(CCC)CCC3)=O)COCC2)cnc2c(c1)OCCN2 32875,c1(C(=O)NCC2(OC)CN(C(C(CSC)(C)C)=O)C2)cc(C)c2nc(C)nn2c1 32876,C#CC1(C)CCCN(C(=O)C(C)N(CCC)C(c2cccc(C(C)=O)c2)=O)C1 32877,N1(C(C2CC(OC)C2)=O)CC(NC(c2cc(C)cc(O)n2)=O)C2(CCC2)C1 32878,N1(C(c2n(CC)ncc2)=O)CC2CC(C1)CN(C(=O)COC1CC1)C2 32879,C1(CC(=O)N(CC(C)NC(C=C(CCC)C)=O)CC)CCCC(F)(F)C1 32880,C1(NC(C(CCC2CCC2)NC(c2c(C)noc2C)=O)=O)CCCCN(C)C1=O 32881,C1(COC)(NC(=O)CC2CCCO2)CCN(C(c2cnn(C)c2F)=O)CC1 32882,N1(CC(C)O)CC2CCC(C1)N2C(c1nccc(C2OCCO2)n1)=O 32883,CC(C)CCC(C(=O)N(C(C)CO)C)NC(=O)CCc1cccnc1 32884,Cc1cc(Cl)c(C(=O)NC2CC2NC(=O)Cn2cnc([N+](=O)[O-])c2)c(Cl)c1 32885,CCCC(C)CNC(=O)C(C)N(C(=O)CC(C)n1cccn1)CC 32886,C1(C(=O)NCCCN(C)C(C23CCCC2C3)=O)CCc2ncccc2C1 32887,c1(C(N2CCCCC23CC3)C(=O)NCCOC)cc2c(Br)cccc2o1 32888,c1(C(N2CC(CNC(C=C(C)C(C)(C)C)=O)C3C2C3)=O)cccc2c1CCC2=O 32889,C12CN(C(c3cc(C(=O)C(F)(F)F)c[nH]3)=O)CCN1C(=O)CNC2=O.C1(C)CC1 32890,C1(CNC(=O)Cn2cncn2)CN(C(=O)CC2CC3CC(=O)C2O3)CC1(F)F 32891,c1(C(=O)NCC(C)NC(c2c(F)cc(OC)c(OC)c2)=O)cn2nc(C)sc2n1 32892,c1(CC(=O)NC2CC(NC(Cc3ccn(C)n3)=O)C23CCC3)ccc2sccc2c1 32893,Cc1cc(C(N2CCOCC(NC(c3cnc(F)c(Cl)c3)=O)C2)=O)nc(C)n1 32894,CN1N=C(C(=O)NC(C(N2CCCC(NC(N)=O)C2)=O)c2ccco2)CCC1=O 32895,C(=O)(CCC(F)(F)F)NC1(CCOC)CCN(c2ccnc(C(=O)OC)n2)C1 32896,N1(C(C2(OC)CC2)=O)CCCN(C(c2cc(CO)c(C)o2)=O)CC1C 32897,N1(C(C(C)SC)=O)CC2CN(C(=O)C(n3ccc(C(F)(F)F)n3)(F)F)CC2C1 32898,Cn1c(C(=O)NC(CNC(c2ccc(F)cc2)=O)C2CC2)cc(Cl)c1Cl 32899,C1(NC(C(C)CN(C(=O)CN2CC(=O)NC2=O)C)=O)CN(C)NC1=O 32900,c1(C(=O)NCC(C(C)C)NC(C(CC#C)C)=O)cccc(S(=O)(=O)C(F)F)c1 32901,C1(CCn2cc(CCNC(C)=O)nn2)CN(C(C2C(C)CCC2C)=O)CC(C)O1 32902,C(CC(C(C)C)NC(=O)C(c1ccc(Cl)nc1)(C)C)N(C(CSCC=C)=O)C 32903,c1(C(=O)NCC2CCN(C(C#CC(=O)N(C)C)=O)CC2)cc(Br)ccc1OCF 32904,N1(C(CN(CC#C)C(C)=O)=O)CC2CC1CN2C(C)Cc1ccco1 32905,C(=O)(C(C(C)C)Nc1ccc(C(C)(C)OC)cc1)NC.C12CCN(CC1)C2=O 32906,c1(C(=O)NCC2C(NC(C(C)OCC=C)=O)CC2)c[nH]c2c(C#N)cccc12 32907,N1(CC(=O)NC(CC)(C)CNC(c2cn(C(C)C)nn2)=O)C(=O)CC(C)(C)C1=O 32908,c1(C(N)=O)cc(C(=O)NCCNC(=O)CCC2CC2Cc2ccccn2)ccn1 32909,Nc1cc(Cl)ccc1C(N1CC2(C1)CN(C(c1cocn1)=O)C2)=O 32910,CCCCC(O)C(=O)N1CCCC1C(C)NC(c1ccncc1C)=O 32911,c1(CCN(c2cc(Cn3cc(CNC=O)nn3)cs2)C)ccc(C#N)cn1.CSC 32912,c1(COC(c2nc(C3CC3)cs2)=O)cccc(I)c1 32913,C1(OC)CN(C(c2ncn(C)c2C)=O)CC1NC(c1ccnc(OC(F)F)c1)=O 32914,Nc1c(F)ccc(F)c1-c1cn(C(C2CCCCC2)N)nn1.C1(C)NC(=O)NC1=O 32915,c1(SCC(N2CC(N(C(C3(Cc4nnc(C)o4)CC3)=O)C)C2)=O)ccc(F)cc1 32916,Cc1nc(C(C)(C)C)[nH]c(=NC2CC(NC(=O)CCC34CCC(CC3)C4)C2)c1C 32917,C1(NC(C=CCCC(C)C)=O)CCC(C(=O)NCC2CC2)OC1.c1cnn(C(C)C)c1 32918,Cn1nc(-c2cn(CC3CC4(CCO4)C3)nn2)cc1N 32919,c1(N2CCC3(CC(NC(C(CC)C)=O)C3)C2)ncnc2ccc(S(C)(=O)=O)cc12 32920,CC1(CNC(c2cc(C(F)F)no2)=O)CCN(C(C2(C3CCCO3)CC2)=O)CC1 32921,c1(C(C)NC(N)=O)csc(CCCc2ccon2)n1 32922,c1(C(=O)NC(c2nc(C(=O)OC)c(N)s2)C)cnn2c1CC(C)CC2 32923,c1(C(N2CC(N(C(=O)CCc3cnco3)C)C2)=O)ccc(Oc2cccs2)cc1 32924,c1(C(=O)NC2CC(C(C)O)C2)ccc(CNC(=O)CC(Cl)Cl)nc1 32925,C1(NC(C(N2CCNC2=O)C)=O)C2CC1N(C(C1CCSC1)=O)C2 32926,C1(C(N(C(C#C)C2CCC2)C)=O)CN(C)CCN1C(=O)Cc1ncccc1C 32927,C(c1cccc(F)c1)=C(C(=O)NC1C=CCN(C(c2c(CC)onc2C)=O)C1)F 32928,Cc1cccc(CC(N2CCOC(CNC(=O)Cc3nnc(C)s3)C2)=O)c1 32929,N1(C(C2(CC)COC2)=O)CCC(N=c2nn[nH]n2C)CC1C 32930,C1(CCC)CCC(C(=O)NCCN(CCC)C(C2CCCN2S(C)(=O)=O)=O)CC1 32931,C1(C(=O)NCCCC2OCCN(C(C(C)(C)N(C)C)=O)C2)CCCCC12CCC2 32932,C(CC(O)CC(=O)NCCN(C(=O)C(C(C)(C)C)C1CCC1)C1CC1)SC 32933,c1(CC(C)C)cc(C(=O)NCC(C)NC(=O)CCc2cccnc2F)cc(O)n1 32934,c1(C(=O)NC)ccc(CNC(c2csc(NC(=O)OC(C)(C)C)c2)=O)nc1 32935,CCCCC(C(=O)N1CCCOC(CCNC(=O)CCc2scnc2C)C1)N(C)C 32936,Cc1ccc(C(N2CCC(N(C(=O)C(O)Cn3cncn3)C)C2)=O)cc1 32937,Cc1scc(CNC(=O)CCCC2(NC(=O)C=CCF)CCC2)c1C 32938,c1(OC)ccccc1C(=O)NCCCC1CCCN1C(C1CCC(C)O1)=O 32939,C1(n2cc(C(C(C)(C)C)O)nn2)CCCN(C(=O)COCC2CC2)C1 32940,c1(OC)cccc2c1CCC(N=c1cnc(F)c[nH]1)C2 32941,c1(OC)ncccc1S(=O)(=O)N1CCN(C(=O)CCc2ccsc2)CC1C(C)C 32942,N(C(=NC(C)C)N1CCC(F)C1)Cc1nn(CC)nc1C 32943,N1(C(c2c(OC)cc(C)cn2)=O)CC(NC(=O)CN2CCOC2=O)C(N=[N+]=[N-])C1 32944,C(=O)(C#CC1CCCOC1)N1CCC(CNC(c2cc(C(=O)OC)c(F)cc2)=O)C1 32945,c1(C(N2CCC(C(C)NC(=O)CCc3cncc(F)c3)C2)=O)cnc(N)c(N)c1 32946,Cc1ccc(C(=O)N(C)CC2CCCN2C(=O)CC2CC(CF)C2)cc1N 32947,c1(C(N2CCC(O)(N(C(=O)CN3CCC(O)CC3)CC)C2)=O)ccc2c(c1)CC2 32948,C#CCCC(C(=O)NC1(CO)CC(C)(C)C1)NC(C1CC2(C1)CC(C)C2)=O 32949,N1(C(C(n2ncc(C)c2)C)=O)C2CCC1C(C)C(NC(c1ccc(CO)o1)=O)C2 32950,c1(C(=O)NCC2N(C(c3c(C)con3)=O)CC(O)C2)ccc2nc[nH]c2n1 32951,N1(C(C2CCC(CC)C2)=O)CCCN(C(c2cnn(CC)c2)=O)CCC1 32952,N1(C(CCC=C)=O)CCOC(CC(=O)N(C2CC2(C)C)C)C1 32953,C12(NC(C3CCc4cnnn4C3)=O)CCCC1N(C(=O)C=Cc1cscn1)CC2 32954,N1(C(c2n(CC#C)cnn2)=O)CC2CCCC2(NC(=O)CCc2n[nH]c(=N)s2)C1 32955,C1(N(C(C)C(=O)OC(C)(C)C)C(C)=O)CCN(C(c2ncoc2C)=O)CC1 32956,C1(NC(C(C)NS(CC)(=O)=O)=O)CN(C(C2CCS2(=O)=O)=O)CCC1CO 32957,C(CC(C(=O)NC1CCN(C(C)=O)C1)NC(C1CCCSC1C)=O)=CC 32958,CC1(NC(=O)Cc2ccsc2)CN(C(C2(C)CC2(C)C)=O)C1 32959,C1(F)(CNC(c2c(C)nco2)=O)CCCN(C(c2ccnn2C2CCC2)=O)C1 32960,CCC(C)C(CO)NC(=O)C(Cc1ccco1)NC(c1cc(C#N)cs1)=O 32961,CCC(C)CCCCC(=O)NOCC=CCl.C1(C)C(C(=O)OC)N1 32962,C(=O)(C(C)(C)CO)NC(C)C(C)NC(=O)CCOc1cccc(Br)c1 32963,C(=O)(CCCCC1CCCCC1)N(CCCN(C(CCCNC(=O)OC)=O)C)C 32964,C1(NC(CC(CC)C)=O)(CC)CCN(C(=O)CC23CCC(CC2)CC3)CC1 32965,Cc1nscc1CCC(=O)NCC(C)(CO)NC(c1cn(CC(N)=O)nn1)=O 32966,C1(C(=O)Nc2c(OCC)cccc2)CCN(Cc2cccc(N)n2)CC1O 32967,CC1CC(NC(c2cc(CCCO)on2)=O)CN1C(C1CCC(C(F)(F)F)O1)=O 32968,c1(CC(=O)NCC(CSC)NC(C=CCCC)=O)cc(C(F)(F)F)ccn1 32969,N1(C(c2cccc3ncsc23)=O)CCOC2(C1)CN(C(=O)C(O)CCl)C2 32970,n1(CC#C)c(C)cc(C(=O)NC2(CF)CCN(C(C3CC(F)C3)=O)C2)c1C 32971,N1(C(c2n(C(C)C)ncc2)=O)CCOC2(C1)CN(C(=O)C(C)CS(C)=O)C2 32972,CCC(C(=O)OC)C(=O)NCC(CC)N(C)C(C1(c2cc[nH]n2)CCC1)=O 32973,c1(CCN(C)C(C2(CCNC(C3CCC4CC34)=O)CCC2)=O)ccncc1 32974,N1(C(C2(CC)CCOC2)=O)CCCC(C)(CNC(c2csc(CC(C)C)n2)=O)C1 32975,C(=O)(C1=C(Cl)CCCC1)NC1C2(C(=O)NC(CCCC=C)C)C3CC1CC23 32976,C(=O)(CC1OCCc2sccc21)NC1C(C)CCN(C(=O)CCC(N)=O)C1 32977,C1(CS(C2CC(F)C2)(=O)=O)CC2CCC(C1)N2c1nccc(Br)n1 32978,c1(C(N(C2CCCN(C(C3CNC(=O)C3)=O)C2)C)=O)cc(Br)cc2nc[nH]c12 32979,N1(C(CSCCN(C)C)=O)CC2(C1)SCCC2NC(=O)CC1(O)CCCOC1 32980,O=C(C1=CCCCO1)N1CCCCN1Cc1cc(Br)ccc1F.c12ccc(cn1)NC2 32981,c1(CC(=O)NCC(CC)(C)NC(=O)C(C)(O)COC)cncc(C#N)c1 32982,c1(OC)nccnc1C(=O)NC1C=CC(C(=O)N(C2CCCCC2)C2CC2)C1 32983,CCC(C#N)(CC)C(=O)N1CC2CC1(CNC(=O)Cn1nc(C)ccc1=O)C2 32984,c1(C(=O)NCCC(=C)CNC(C23CCCCC2C3)=O)cc(C)cc(C)c1C 32985,N1(CCC(C(=O)OC)C)CC(C(=O)NOCCCN(C)C)C(C)(C)C1 32986,C1(NC(CC(CC2CC2)NC(c2cc(C)[nH]n2)=O)=O)CC2C(O)C(O)CC12 32987,c12nccc(c1F)C(=O)N2.C(=O)(CCCC(=O)NC)N(C1CCC(SCC)C1)C 32988,C(C)(CCC(=O)N1CCOC(CN(C(=O)CCCN2CCCCC2)C)C1)OCC 32989,c1(CCC(=O)N(CC(CN(CCC(C)C)C)O)C)cc(Br)cc(F)c1F 32990,N1(C(CCSC)=O)CCCC2(CCN(C(c3c(N)cc(Cl)cc3Cl)=O)C2)C1 32991,CN1N=CC(CC(N2CCOCC2CC(=O)NCCc2cccc(F)c2)=O)C1=O 32992,C1(CC(=O)NOCC2CCCO2)(CC#C)CCN(C(c2cccnc2)=O)C1 32993,c1(C(N(CCCNC(=O)Cc2cc(Cl)cs2)C)=O)csc(S(N)(=O)=O)c1 32994,Cc1cc(N(C(C)C(F)(F)F)C)nc(NC(c2cc(Cl)sc2Cl)C)n1 32995,c1(OCC)cc(C(N2CC(c3ccccc3F)C2)=O)cnc1O 32996,c1(C(N2C3CC(CNC(C(CCC)(C)C)=O)C2CC3)=O)cc2n(n1)C(C)CCC2 32997,c1(C(=O)NC2(C(=O)NCc3ccc(C)cc3)CC2C)ccc(F)c(F)c1 32998,C1(CC)CCC(=O)N1.c1(NC(c2cc(OCC)no2)=O)cc(F)ncc1O 32999,C(CC(=O)NCc1cc(C(F)F)[nH]n1)(C(F)(F)F)NC(=O)CN1CC=CC1 33000,N1(C(C(NCP(C)(C)=O)C)=O)CC2CCCC2(C(C2C3CCC(F)C23)=O)C1 33001,c1(C(C)OC)nc(CN(C)C(c2ccc(F)cc2)C)n(C)n1 33002,N1(C(CC(C=C)(C)O)=O)CC(NC(c2cnn(C(C)C)c2Cl)=O)C(N=[N+]=[N-])C1 33003,C1(C)(CNC(CC2C=CC(NC(CC(C)SC)=O)C2)=O)CC(C)=NO1 33004,N1(C(C(C2CC2)OC)=O)CCCC12CCCN(C(C1(NC(C)=O)CCCC1)=O)C2 33005,C1(OCC)CCN(CC(=O)N(C2CN(C(=O)CCSCC(F)F)C2)C)C1 33006,Cn1cc(C(=O)NCC2CCC(NC(=O)CCN3CCCCC3)CC2)ccc1=O 33007,C(=O)(CC(C(F)(F)F)N(C)C1CC1)NC(CC)(CNC(c1coc(Cl)n1)=O)CC 33008,c1(OCC(=O)N(C2CC(NC(C3CCOC(=O)N3)=O)C2)C)c(Cl)cccc1Cl 33009,CCCC(C(=O)NC1(CCF)CCC1)NC(C1CC2CC2C1)=O 33010,C1(NC(c2cnc3[nH]cnc3c2)=O)CC2CN(C(C3CC3(F)F)=O)CC2C1 33011,c1(C(N2CCCC(Cc3ccc(CCC(=O)OC)cc3)C2)=O)c(C=O)cnn1C 33012,C1(C(N2CCC(CCCC)C2)=O)N(C(c2scnc2Cl)=O)CCC1(C)C 33013,c1(CC)ccc(C(N2CC(CNC(C3NC(=O)OC3C)=O)(COC)C2)=O)cc1F 33014,c1(C(=O)NC(CCCC)CNC(=O)CCCCC(C)C)coc2cc(F)ccc12 33015,c1(OC)cc(C#N)ccc1CN1CC2CC(C1)N2C(c1ccc2c(c1)OCO2)=O 33016,C1(C(=O)NC2CC(CCNC(c3cn(C)c(=O)cn3)=O)C2)CCCC1S(C)(=O)=O 33017,CC1CCC(CO)(NC(C2CCNC(C)C2)=O)c2ccccc21 33018,C(CS(=O)(=O)CC(=O)NC1CN(C(=O)CCc2ccncn2)CC1(C)C)OC 33019,C1(NC(=O)C=CC2CCOC2)CC2CC1CN(C(c1noc3c1CCCC3)=O)C2 33020,C(=O)(C1c2c[nH]nc2CN1C(=O)C(c1ccn(C)n1)C)NCC(C)S(C)(=O)=O 33021,C(=O)(C1=C(Cl)CCOC1)NC1C(C)CCN(C(c2n(CC)cc(Br)c2)=O)C1 33022,C1(NC(c2c(C)nco2)=O)CCCC(NC(c2cc(Br)co2)=O)C1 33023,N1(C(CSC)=O)CCC2(CC1)CN(C(=O)Cc1ccc(CC#N)cc1)CC(C)O2 33024,N1(C(=O)OC)CCN(C(C(=O)NC(C)C)C2COC2)CC1(C)C 33025,C12(NC(C(CC3CCCC3)NC(C3C(C#N)C3)=O)=O)CCCCC1OCC2 33026,N1(C(C=CC(C)C)=O)CCC(NC(C2CCS(=O)(=O)C2)=O)C12CCC2 33027,CCCC(C(=O)NOC)NC(C1CC(O)CN1C(=O)OC)=O 33028,C1(NC(CSCCC#N)=O)CC2(C(N3CCC(F)(F)C3)=O)COC1C2 33029,c1(C(C)NC(=O)C(N2CCCC(C3CCCN3C)C2)=O)cccc(O)c1 33030,Cc1nc(NC2CC(C)N(C(=O)CCC(C)C3CC3)C2)c2c(C)c(C)sc2n1 33031,C1(C)(C(=O)NCC(C#C)OC)CC(O)CN1C(c1cnnn1CC)=O 33032,C1(CN2CCC(c3cn(CC)nc3C(F)(F)F)CC2)COC2(CCC2)CO1 33033,C1(C2(O)CN(C(c3oc(SC)cc3C)=O)C2)(CNC(C(C=C=C)C)=O)CC1 33034,c1(CNC(CNC(=O)OCC)=O)cc(OC)c(Cl)cn1.C12CC(C1)NC(=O)C2 33035,N1(C(Cc2ccc(C(=O)OC)s2)=O)CC(C)CN(C(=O)CSCC(F)F)CC1C 33036,c1(N2C(CCNC(c3n[nH]cc3Cl)=O)CCC2)cc(C(F)F)ncn1 33037,c1(C(N2CCN(C(=O)C=CBr)C(C3CCC3)C2)=O)cccc2nonc12 33038,C1(CNC(CSCC)=O)N(C(c2cc(C(C)(C)C)on2)=O)CCCC1(C)C 33039,C1(C(=O)NCCCCN(CCCNC(C(C)OCC)=O)C)CC(=O)N(OC)C1 33040,N1(C(C(CC)NC(C)=O)=O)CCCN(C(c2ncccc2C(=O)OC)=O)CC1C 33041,C1(CNC(CSCC=C)=O)CC(C)N(C(c2cn(C)c(O)n2)=O)C1 33042,C1(CCC)CCCN1S(=O)(=O)CCC1CCOC1 33043,C1(C(=O)NC2CCC(OCC)CC2)C2CCC(C2)C1NC(=O)C1=CCCC1C 33044,N1(C(C=COCC)=O)CCC(NC(c2cc(Br)c(C(F)F)s2)=O)CC1C 33045,c1(C(=O)NCC2(O)CCN(C(c3ccc(C)nc3)=O)C2)c(C)cc(F)cc1Br 33046,N1(CC(=O)NC2(c3ccsc3)CC2)CCC(C2CNC2)CC1 33047,N1(C(c2n(CC)ncc2)=O)CC2CCCC1C2CNC(C1(C)CCCO1)=O 33048,C1(C(=O)NCC(CCC)(C)O)CCC2(CC2)N1C(C1CC2CCC2C1)=O 33049,Cc1ccc(NC(C2CN(C(c3sccc3Cl)=O)CCC2O)=O)c(C#N)c1 33050,Cc1cc(CC(=O)NC(C)CNC(C2(CN3CCOCC3)CCCC2)=O)c(C)s1 33051,C1(NC(C2(CC)CCCCC2)=O)CC(O)CN(C(=O)C=Cc2ccccc2F)C1 33052,C(=O)(C(O)C(C)(C)C)N1CC(C(C(=O)NC2CC(C(=O)NCC)C2)OC)C1 33053,C1(C(=O)NCC2=CCN(Cc3n(C)ncn3)CC2)C2C=CC(CC2)C1C(F)F 33054,Cc1ccc(C(F)(F)C(=O)NCC2CN(C(C3CC(O)C3)=O)CCO2)cc1 33055,n1(CCCOC)cc(NC(=O)NCc2c[nH]nc2-c2cnn(C)c2)cn1 33056,C(C)(C(CCc1ccccc1)OC(C)(C)C)OCC.C1(=O)C(F)(F)CN1 33057,Cc1cnc(C(=O)NCC(C2CCCN(C(c3cncnc3C)=O)C2)(C)O)nc1 33058,C12(CC)CCCN1C(=O)C1(CC1)C(=O)NC2.c1(NC(c2cnsn2)=O)ccccc1 33059,Cn1ccnc1C1CC1C(=O)NCC1(O)CN(C(c2ccccn2)=O)C1 33060,c1(C(N2CCC(NC(CC(C)(C)C3CC3)=O)C(O)C2)=O)ccc2sncc2c1 33061,N1(C(CC=C=C)=O)CCC2CCC12CNC(=O)CCOc1ccc(F)c(Cl)c1 33062,CCC(F)(F)CC(=O)N1CC(CC(=O)NCC2CC(=O)NC(C)C2)(OCC)C1 33063,N1(C(C2N(C(=O)COc3ccn(C)n3)CCC(C)C2)=O)CCCC(C2(C)CC2)C1 33064,N12C3CCC1CC(C3)C(=O)NCC2.C(CCN1CCC1)SCC 33065,C1(C(=O)NCC(CC)CO)CC(NC(C2CCCN2C(C)C)=O)C(O)C1 33066,Cn1cnc2cc(CC(=O)NCC3CC(NC(C4CC4F)=O)C3)ccc12 33067,C(C(=O)N(CC(C)(C)CNC(c1nocc1C1CC1)=O)C)(C(C)C)SCC 33068,C1(C(N2CC=CC2(C)COC)=O)(COC)C=CCN1C(=O)C=CC(C)(C)SC 33069,CN1N=C(C(=O)NC2CS(=O)(=O)CC2NC(c2ccnn(C)c2=O)=O)CCC1=O 33070,C1(CC(=O)N(CCN2CCN(C(C3(CCC)CC3)=O)CC2)C)CCCC(C)(C)O1 33071,C1(C)(C(N2CC(CC)C(NC(C3(C(=O)NC)CC3)=O)C2)=O)CC2(CCC2)C1 33072,c1(C(=O)NCC(CC=C)NC(=O)C(C)(C)C(=C)C)cc2nc(C)cc(C)n2n1 33073,C1(C(N2CCC(N(C(=O)C(C)(C)C3CCCCO3)C)C2)=O)C(C)(C)OC1(C)C 33074,N(C1CCc2c1ccc(Cl)c2Cl)C(c1c(OC)c(Cl)cc(C)c1)c1nnnn1C 33075,N1(C(c2c(C)ccnn2)=O)CC(F)(F)CC1CCNC(=O)CN1CSCC1=O 33076,n1(CC#C)cnnc1C(=O)NC(C1CCOC1)CNC(=O)CNS(=O)(=O)CCC 33077,c1(CC)nc(C)c(CC(=O)NCC(C2CCC2)NC(=O)C=CS(C)=O)c(C)n1 33078,c1(C(=O)NCC2(CCNC(c3cc(C)ncc3)=O)CC2)cc(N(C)C)nc(Cl)c1 33079,CCS(=O)(=O)CC(=O)N1CC(CNC(c2cc(F)n(C)n2)=O)CC1C 33080,N1(C(C=C(CCN(C)C)Cl)=O)CCOC2(C1)CN(C(C1CCCN1N=O)=O)C2 33081,c1(C(=O)NCC(=C2CN(C(C3CC3(F)F)=O)C2)F)n[nH]c(C2CC2)n1 33082,C1(CC(=O)NCc2c(CNC(CC(C)(C)O)=O)cccc2)CN2CCN1CC2 33083,N1(C(CC(C(F)(F)F)NC)=O)Cc2ccnc(Cl)c2C1 33084,C(=O)(C1CSc2ccccc21)NCC1CN(c2ccc(C(C)=O)cc2[N+](=O)[O-])C1 33085,Cc1ccc2[nH]cc(CC(N3CC(NC(C4(C(N)=O)CC4)=O)CC(O)C3)=O)c2c1 33086,c1(NC(C#C)C2CCC2)ccc(CC2CCCC2OCc2ccccc2)cn1 33087,C1(C(=O)NC2(COC)CN(C(c3ccc(F)c(Cl)c3)=O)C2)CC2C(C1)C2(C)C 33088,C1(C(N2CC(CNC(C)C(=O)OC)C2)=O)(CC2CC2)CCCCC1.n12cc(nn1)C2 33089,C1(NC(CCC=C=C)=O)CCCN(C(c2cscc2C#N)=O)C1C 33090,c1(C(=O)OC(C)(C)C)cnc(NC2CC(NC(=O)C3CC3)C2)s1 33091,N1(C(C2CC3CC3C2)=O)CCC2(C1)c1[nH]cnc1CCN2C(C1(O)COC1)=O 33092,CC(C)(C)C#CC(=O)NC1CCN(C(=O)CC2(O)CCCC2)CC1 33093,c1(NC(C)C)cccc(C(=O)NC2CN(C(=O)C(C)=C3CCC3)CC2C)c1 33094,CCCC(CCCNC(=O)CC1CCCCCO1)NC(=O)CNC(=O)C(C)(C)C 33095,N1(C(c2scc(CNC(c3c(C)ocn3)=O)c2)=O)C2CCC1COC2 33096,Cc1cc(C(=O)NC(C)C(C)(C)NC(=O)CSCCN(C)C)c(C)nc1C 33097,c1(C(N(C2CC(NC(C3CCC(C)CC3)=O)C2)C)=O)cccc2nncn12 33098,C1(F)(Cn2cc(CCN(C)CC)nn2)CCN(C(c2ocnc2C2CC2)=O)C1 33099,N1(C(C2C3(CN(C(c4c(C)nn(C)c4C)=O)C3)C2)=O)C2CCC1CN(C)C2 33100,c1(CC(=O)OC)cccc(Br)c1NC(=O)C(=O)NCc1ccn(C2CC2(F)F)n1 33101,CC1(C)Cn2[nH]c(=NC(=O)NC(C3CC(F)(F)C3)C(=O)O)cc2CO1 33102,CN1CCC(NC(=O)CCC2CCC(NC(=O)C=CC3CC3)C2)C(C)(C)C1 33103,c1(C)cc(Br)c([N+](=O)[O-])cc1Br.C1(C(=O)NN2CCCC(O)C2)CCN(C)CC1O 33104,C(=O)(CC(C)(C)C)NC(C)C(N1CCC(C(=O)N(c2cccc(Cl)c2)C)CC1)=O 33105,N1(C(CNC(C)=O)=O)CCOCC1CCN1CCN(C(=O)C2=CCSC2)CC1 33106,C(CCN=C(NCC1CCCS1)NCC(C)(C)CN1CC(C)OC(C)C1)SC 33107,c1(C(=O)NCC2N(C(C(COCC)(C)C)=O)CCC2)cccc(C(F)(F)F)c1C 33108,c1(C(N(C(CC)CNC(=O)C(F)OC(F)(F)F)C)=O)cccc2nsnc12 33109,C(CCC(=O)N(C)CCOCCCN(C(=O)C(C)CSc1ccccc1)C)=CC 33110,C1(C(=O)NCCN(C(c2cnsc2)=O)CC)CCc2nnc(O)n2C1 33111,c1(C(N(CCCN(C)C(C2CCC(CCO)CC2)=O)C)=O)cc2sccc2[nH]1 33112,N1(C(C2(CC#C)CC2)=O)CCC2(CC1)CC2C(=O)NC1CC2(CCC2)C1 33113,C1(C(=O)OC)CN(C(C2CCC(C)CN2C(=O)OC(C)(C)C)=O)CCN1C 33114,N1(C(c2nncc(C)c2)=O)CC(C)CN(C(=O)C(C(C)C)N(C)C)CC1C 33115,C(=O)(C(C)(O)CC)NCC1(C(=O)NCC2CCCC2)CC1.C(CCC=O)N(C)CCOC 33116,C1(NC(C2C(CCC)C2)=O)CN(C(c2ccc(-n3cnnn3)cc2)=O)C(C)(C)C1 33117,C(CC)(CCC(=O)NOCCC(C)O)NC(=O)COC(C(CC)(C)C)=O 33118,c1(CC)onc(C(=O)NCC(C(=O)NCC2CCC=CCC2)N(C)C)c1C 33119,C1(C(N(CCN2CCN(C(C(C)OC)=O)CC2)C)=O)C2CCCCCCC12 33120,Cc1nccnc1-c1cn(CC2CC(NC(=O)COCCOCCO)C2)nn1 33121,c1(C(=O)NCCCN(C(=O)CP(C)(C)=O)CC)c(C)nc2ccccn12 33122,c1(C(N(CC(CC)NC(CSCC(C)C)=O)C)=O)cccc(C#CCO)c1 33123,C(CC1=CCOCC1)NC(C(C1CCCCN(C(=O)C=CCO)C1)C)=O 33124,N12CCC(CC1C)SCC2=O.c1(C=O)cc(C(C)(C)C)[nH]c1C.C(=O)NCC 33125,C1(C(=O)NC2CCCCNC2=O)CN(C(C2CC(O)C2)=O)C2(CCC2)C1 33126,N1(C(C(CC=C)(C)O)=O)CC=C(C(=O)NC(c2nc[nH]n2)C2CC2)CC1 33127,CC(=Cn1ccnn1)C(=O)NCC12CCC(CN(C(c3cccnc3O)=O)C1)C2 33128,N1(C(c2cc(C)sn2)=O)CC2(CCN(C(=O)CCC3CCCC(O)C3)CC2)C1 33129,c1(OC)cncnc1C(=O)NC(C(=O)N(C1CCCCC1C)C1CC1)C1(C)CC1 33130,C1(N(C(C2N(CC)CCC2)=O)C)CCN(CC(=O)NCC2CC2)CC1 33131,c1(C(=O)NC(CN(C(C2N(C(C)=O)CSC2)=O)C)C)cc2c(O)ccc(F)c2[nH]1 33132,c1(-n2cc(-c3cc(CC(C)(C)C4CCCO4)on3)nn2)cc2c(nn1)CCCC2 33133,C(=O)(C(C(C)(C)C)NC(c1ccnc(CNC(c2cnc(Br)s2)=O)c1)=O)NC 33134,CCN(Cc1ccc(C(C)C)cc1)N1CC(OCCO)C(C)C1 33135,c1(C(=O)NC2CC3N(C(C4CCN(C)CC4)=O)C(CC3)C2)c[nH]c2ncc(Br)cc12 33136,N1(C(C2CC(C)C2)=O)C(C(=O)N)CCC12CC2.N1(CCC2CC2)CCCC1C 33137,C1(NC(=O)CCc2ncc[nH]2)CCSC12CN(C(c1cnn(C3CCC3)n1)=O)C2 33138,CC1(C(=O)NCC2CCCCN2C(c2ccn(C3CCC3)n2)=O)CC2CCC1C2 33139,CCC(CC(F)(F)F)C(=O)NC(C)C(=O)NCCCN(C)CCOC 33140,N1(c2n(CC=C)c(C(O)CCOC)nn2)CCC(C)CC(C)C1 33141,C1(NC(c2c(C)con2)=O)CN(C(=O)Cc2ccns2)CCC12CCC2 33142,Cc1cc(C(N2CCN(C)C(CNc3ncccn3)C2)=O)nc(C2CCC2)n1 33143,Cc1nc2sc(CNC(c3cc(C4(C)CC4)n[nH]3)=O)nn2c(=O)c1F 33144,C1(NC(c2cnc(C)o2)=O)CCOC12CCN(C(c1cc(Br)c[nH]1)=O)CC2 33145,N1(C(c2nc(CCC)sc2)=O)CC2ON=C(CNC(c3nc(C)oc3C)=O)C2C1 33146,CC(C)CC(CN(C)C)NC(C1(F)CCN(C(=O)CCCC2CC2C)C1)=O 33147,CCCC(C)(O)CC(=O)N1C2CCC1C(CNC(=O)CN(C)C(C)C)C2 33148,N1(C(N2CCOC3CC23)=O)CCCCC1CCC(F)(F)F 33149,c1(CC(=O)NC(C(C)NC(c2cc(C)c(C)nn2)=O)C)ccc2ncsc2c1 33150,c1(C(C(=O)N(C2N(C(COCCSC)=O)CCC2)C)O)cccc(C)c1 33151,N1(C(C(N2CCC(OC)(NC(c3ncoc3C)=O)C2)=O)(C)C)CCS(=O)(=O)CC1 33152,N1(C(CC(=O)NC2CC2)=O)CCC(C(=O)NCc2cccc(F)c2)C12CCC2 33153,N1(C(CC(CC)O)=O)CCCCC2(CCN(C(=O)OC(C)(C)C)C2)C1 33154,c1(NC(CN2CCCC(CNC(C(C)C)=O)C2)=O)ccc(F)c(Br)c1 33155,c1(C(N2C(C(N3CCC(C(=O)OCC)C3)=O)CNCC2)=O)ccc(F)c(Cl)c1Br 33156,Cc1cc(CN2CC(F)(F)CC2C(=O)Nc2nc(Cl)ccc2O)cnc1Cl 33157,C=CC(CCC)CC(=O)N1CCC(NC(=O)C(O)CC(F)(F)F)C12CC2 33158,N1(C(CCC(=O)OC)=O)CCC2CN(S(=O)(=O)CC3CCC3)CCC12 33159,N1(Cc2nc(CC)sc2Br)CC(CC2CC2)OCC12CC2 33160,C(C)(C)(CCCNC(=O)C(CCSC)NC(C1CCN1C(C)C)=O)OC 33161,CCCCCC(O)CC(=O)N(CCCCN(C)C(c1ccccc1N)=O)C 33162,C1(OC)CC(CC(=O)NCC2CN(C(=O)CC(C)CF)CCO2)C1(C)C 33163,N1(C(Cc2scc(C)c2)=O)CCC2(CC1)OCCC2NC(=O)Cc1coc(C)n1 33164,C(=O)(CCC1=NNC(=O)CC1)NCCC(=O)NC1(C)CC(NC(=O)CO)C1 33165,S(=O)(=O)(c1cc(F)cc(Br)c1)N(C(COc1cc(OC)c(NC)cc1)=O)NC1CCC1 33166,N1(C(C(CSC)O)=O)CCC=CC1C(=O)NCC1CC1CN(C)C 33167,c1(N2CCC(NC(c3ccc(C)c(C(F)(F)F)c3)=O)CC2)ncc2ccsc2n1 33168,C(C)(C)(CCCCNC(=O)Cn1nccn1)NC(C(CSC(C)(C)C)NC(C)=O)=O 33169,c1(C(C)C)nn(C)c(Cl)c1C(=O)NCC(C)(C)CNC(C1CCOCC1)=O 33170,c1(C(=O)NC(C(=O)NCCc2cc(CC)no2)C)cncnc1CC 33171,c1(CN2CC(F)(C(=O)NC3CCCN(C)C3)C2)ccc(F)cc1O 33172,C1(C#N)(OC)CC(C(=O)NC(CNC(c2c(Cl)n[nH]c2C)=O)C(C)C)C1 33173,N1(C(CCCCCCC)=O)CCc2ccccc2C1CCNC(=O)CN(C)CC 33174,N1(C(CCCCCN(C)C)=O)CC(NC(C2OCCCO2)=O)CC12CCCCC2 33175,C1(C2CC2)(C(=O)OC)CCN(C(=O)C2=C(C)OCC2)C1.C12(CCCC1)C(=O)N2 33176,C=CC1CN(C(=O)C(CN(C)C)N(C)C)CC1NC(=O)C(F)C(C)C 33177,c1(CSC)cccnc1C(=O)NCC(C)NC(=O)Cc1cnc(C)[nH]1 33178,CCC(O)C(F)(F)C(=O)NCC1CCCN(C(=O)Cc2c(C)cc(C)cc2C)CC1 33179,N1(C(c2c(CC)csc2)=O)CCCC(N(C(=O)CC2(C)OCCO2)C)C1 33180,C(=O)(CS(=O)(=O)C1CC1)NC(C(C)C)CCN(C)C(c1ccncc1N(C)C)=O 33181,Cc1cncc(C(N2CC(CN(C)C(c3cnc(C(C)C)n3C)=O)C2)=O)c1 33182,C(CC1=CCN(C(c2cccc(Cl)n2)=O)CC1)NC(CCCCCOC)=O 33183,CN1CC(C(=O)NCC(C)(C)NC(=O)C=CC(N)=O)CCC1=O 33184,N1(C(c2ccc(CN(C)C)[nH]2)=O)CCC2(CCN(C(C3CSC3)=O)C2)C1 33185,c1(CNc2cc(OC)c(C(C)(C)C)cc2)nc2ncc(Br)cn2n1 33186,C1(C(=O)NC(C2CCCN(C(c3cnn(CCO)c3)=O)C2)(C)C)CC(F)C(=O)N1 33187,C1(CNC(C2N(CC)CC2)=O)CCC2(CCC2)CN1C(=O)C(Cl)=CCl 33188,c1(CC)nnsc1C(=O)NCC(F)CNC(c1cn(CCF)nn1)=O 33189,c1(NC(=O)CCCNC(=S)NCCC)cccc(C#N)c1 33190,C1(CCNC(c2cscc2)=O)CCN(C(c2cc(O)ncc2F)=O)CCC1(F)F 33191,c1(C(N2C3C(OC)(CCCC3)CC2)=O)cccc2ccn(C)c12 33192,Cc1cc(Cl)nc(Cl)c1C(=O)NCC1CC(C)CCN1C(C1CCCS1)=O 33193,C(=O)(CCCCCSC1CCN(C(C2CC23CCCCC3)=O)C1)N(C)CC 33194,Cc1ccc(CNC(C2C3CN(C(=O)CC(O)c4ccccc4)CC23)=O)c(O)n1 33195,c1(C(=O)NC2CC(F)(CNC(c3sc(CC)c(C)c3)=O)C2)cccc(OC)c1F 33196,CCCC(C#N)N(C)C(C12CC(NC(=O)CC(C)C3CCCO3)(C1)C2)=O 33197,C1(C(N(CCCNC(c2ccnn2C(C)C)=O)CC)=O)CCCC(C(C)C)C1 33198,C(c1ccoc1)=CC(N1CCC(NC(=O)C(Cl)=CCl)C1)=O 33199,C1(OC)CC(CO)(NC(C2CN(C(=O)COc3cccnc3)C2)=O)C1 33200,N(C1CCCc2c(F)ccc(Cl)c21)C(C(c1c(OCC)cccc1)N)=O 33201,c1(N2CC(C)C(N(C)C)CC2)nccc(=NCCc2nc(C(C)(C)C)cs2)[nH]1 33202,c1(NCCC2(NC(CCOCC)=O)CCC2)nccc(Oc2ccccc2F)n1 33203,c1(C(=O)NCCN(C(Cn2c(C)c(Br)cn2)=O)C2CC2)cnc2sccc2c1 33204,C(C(CC(F)(F)F)NC(c1cccc(O)c1Cl)=O)N(C(COC(CC)C)=O)CC 33205,N1(c2onc(-c3occ(C)n3)n2)CC(=O)NCC1C(C)(C)C 33206,C#Cc1cc(C(=O)NCC2CCC(C)CN2C(c2nccnc2C)=O)cc(N)c1 33207,C1(C(N2CCC(C)(NC(c3cc(C)c(C)o3)=O)C2)=O)CCCC2(CCC2)O1 33208,N1(C(c2ncccc2C)C(=O)NC)CC2CC3CC2C1C3O 33209,C1(CNC(c2cnnn2C2CC2)=O)CN(C(C2C3(CC3)C23CC3)=O)CC12CC2 33210,CC1CC(C(=O)N2CC(NC(=O)C#CC3CCC3)CC2CC2CCCC2)=NO1 33211,CC1CN(C(=O)C(c2ccc(Cl)cc2)O)CC1NC(=O)C(C)C1CCOC1 33212,C1(CNC(c2cnco2)=O)C=CCN1C(=O)CCCc1cncs1 33213,c12ccccc1CC(=O)NC1CC(CO1)NC(=O)CO2.CC(C)OCOC1CC1 33214,c1(C(=O)OC)ccc(N2CCCC(CCNC(C3CCCOC3)=O)C2)nc1C 33215,C1(NC(c2c(CC)noc2C)=O)CC2CC(NC(=O)CCC3(C)CC3(F)F)C2C1 33216,Cc1cccc(C(=O)NCC2CC(C(=O)N3CC(CC(F)(F)F)C3)=NO2)c1F 33217,Cc1ccc(C(=O)NC2C=CCN(C(C3CCC(C)(C)OC3)=O)C2)c(O)n1 33218,N1(C(C(C#N)C2CC2)=O)CCOC2(C1)CN(C(c1c(F)cccc1F)=O)C2 33219,C#CCCCCCC(=O)NC(C)(CNC(C1CC1c1ccccc1Cl)=O)C(C)C 33220,c1(OC)cc(F)c(C(N2CC(C)(C(=O)NC3CCOCC3)C2)=O)c(F)c1F 33221,C(=O)(CC(C(F)F)NC(c1conc1C)=O)N1CC(F)(CC)C1 33222,N1(C(c2cncc(OC)n2)=O)CC(C(=O)NCC(O)C(C)(C)C)CC(C)C1 33223,N1(C(C(C)=C2CC2)=O)CC(N(C(=O)Cc2c[nH]nc2C)C)C(C)(C)C1 33224,N1(C(C2CCc3nncn3C2)C(=O)NN2CCOCC2)C2CCC1C1CCC2O1 33225,CC1=C(C)CC(C(=O)NC2CCCC2CC(N2CCC2c2ccccc2)=O)CC1 33226,N1(C(C(C2CCOC2)NC(c2nc(CCC)oc2)=O)=O)CCC12CCCC2 33227,c1(CC)ccc(CCC(=O)N(C(C)CNC(c2coc(Br)n2)=O)C)cc1 33228,c1(COCC)nc(C(=O)NC(CNC(c2ccc(Cl)o2)=O)CO)cs1 33229,c1(NC(C2CN(C(=O)C=Cc3cccnc3)CCS2)=O)c[nH]c2cccc(Br)c12 33230,Cc1ncnc(C(N2CCC(C)(NC(c3cccc(Br)c3)=O)C2)=O)c1C 33231,C(C(C)C(C)C(=O)NCC(C)NC(C)=O)OC.C(C)(C)(C)ON 33232,C1(C(=O)NCCn2c(C)cnn2)CCC(C)(C)N(C(=O)COCCCN(C)C)C1 33233,C1(O)(CCNC(=O)C(O)C2CCCC2)CCN(C(=O)CCCc2cccs2)C1 33234,c1(C(N2C3C(NC(c4c(Cl)ccc(SC)c4)=O)C(C3)C2)=O)c(N)ccc(F)c1C 33235,C1(C(=O)NC(CC)(CNC(c2n[nH]c(C)c2N)=O)CC)CCC2CC2CC1 33236,C12(NC(CN(C(C)=O)C)=O)CN(C(C3CC3F)=O)CC1CS(=O)(=O)C2 33237,C1(NC(c2c(OC)noc2C)=O)CC2CC1CN(C(c1ccccn1)=O)C2 33238,C1(NC(C(C)OCC#C)=O)CC2CC(C1)N(C(C1CC(C(C)=O)C1(C)C)=O)C2 33239,C(=O)(C1=CCOCC1)NC(CNC(C1CC(=C2CCC2)C1)=O)C1CC1 33240,C1(CN(C(C2CCN(C(C)=O)C2)=O)CC)CCCN(C(c2cscc2C#N)=O)C1 33241,C1(NC(c2cnc(CC)[nH]2)=O)(CC)CCCN(C(c2scnc2C)=O)C1 33242,C1(C(=O)NCC(C)CNC(c2ccc(N3CC=CC3)cc2)=O)CC(=O)N(O)C1 33243,Cc1ccc(C=CC(N2CC(NC(C34CC3COC43CCC3)=O)C(C)(C)C2)=O)cn1 33244,Cc1cn2cc(C(=O)NCC3CC(F)(F)CN3C(=O)C(C)N(C)C)cc(F)c2n1 33245,c1(C(=O)NC2(CNC(C(CSC)O)=O)CCOC2)cnc2c(c1)NC(=O)CN2 33246,C(=O)(CC(O)CC(C)(C)C)N1C2CN(CC(=O)Nc3nc(OC)nc(O)c3)C(C2)C1 33247,C1(C(N2CC(c3ocnc3CNC(=O)CC(C)CSC)C2)=O)(COC)CCCOC1 33248,C1(CC=C)(NC(C2CC(N(C)C)C2)=O)CN(C(c2cc(C3CC3)on2)=O)C1 33249,C1(CC#C)(C(=O)N(CC(C)O)CCNC)CCCC1.C1(C)CC1 33250,Cc1cc(C(N2CC(C(N3CCC(O)(CN(C)C)C3)=O)CC2(C)C)=O)ncc1F 33251,C1(C(=O)NCC2CC(NC(c3cccc(CC)n3)=O)C(O)C2)NC(=O)OC1(C)C 33252,CCC(C)C(C(=O)NC(CCO)CC(C)C)NC(c1c(C)cnn1C)=O 33253,N1(C(C(CC)NC(N)=O)=O)CCN(C(=O)CC2(C#N)CC2)C(C2CCCCC2)C1 33254,C(C)(CCC(=O)NC1CC(C(C)O)C1)NC(C1(OCC)CCSC1)=O 33255,c1(CC)ncc(C(c2nnnn2CC(F)F)NC(C2CCCCC2)C)[nH]1 33256,N1(C(C(OC)OC)=O)CCCC(O)(CCNC(C23CC2COC3(C)C)=O)C1 33257,c1(C(C(=O)NC(C)CC)N(C(C#C)C)C)cc(Br)c(OCC)cc1O 33258,N1(C(C)=O)CCC(NC(=O)COc2cccc(F)n2)C(c2ccc(F)cc2)C1 33259,c1(C(N2CCCCC(n3cc(CCCC)nn3)C2)=O)nccc2cc(Br)ccc12 33260,CC1=C(C(=O)NC(C)CC2CCN(C(C3(C)CCCO3)=O)CC2)C(C)(C)CCC1 33261,c1(NC(C(CSC)O)=O)ccc(Cl)c(C(F)F)c1.C12CC(C1)CNC2=O 33262,C(=O)(CC(C)C(F)F)N(CCC(C)NC(=O)Cc1cccc(C(F)F)c1)C1CC1 33263,c1(CNC(C2CC(NC(CCc3cc(C)no3)=O)C2)=O)ccc(I)c(O)c1 33264,CN1CCN(C(c2ncc(Cl)n2C)=O)CC1CNC(=O)CN1C(=O)NC(=O)C1=O 33265,C(C1CCCc2cccnc21)c1n(-c2c(OC)cccc2)cnn1 33266,c1(OC2CCN(C(C3(c4ccncc4)CCC3)=O)CC2)cc(F)ccc1F 33267,c1(C(C(=O)NC2C(CC)C2)NC(=O)CSCCSCC)cc(F)cc(Cl)c1 33268,N1(C(C(C)(C2CCC2)NC(C(C)NC=O)=O)=O)CCn2ccnc2C1 33269,c1(C(C2(C(N3CC(CNC4C(OC)CC4)C3)=O)CCC2)=O)nc(CC2CC2)co1 33270,n1(CC(=O)NC2CCC(NC(=O)C(O)CC(F)F)CC2)cc([N+](=O)[O-])ccc1=O 33271,C1(C(=O)NC(C)CC(C)N(C)C(c2scnc2Cl)=O)(Cc2cnn[nH]2)CCOCC1 33272,C12(C(=O)NC(c3cccc(C)c3)C)CC(CO)(CN1C(C1(C)C=CCC1)=O)C2 33273,c1(NC(C(=O)NCc2cccc(CCF)c2)=O)cccc(F)c1Br 33274,C1(CCC)(NC(=O)C2=CCCOC2)CCCN(C(C2CCCN2C(=O)C2CC2)=O)C1 33275,CC(C)C#CC(=O)NCC12CC1CN(C(c1ncncc1Br)=O)C2 33276,c1(NC(N(CC(C)C)C)=O)ccccc1SCCn1cnnn1 33277,N1(C(CN(CC(=O)NC(CC(C)(C)C)C)C)=O)CC(C(F)(F)F)C(F)C1 33278,N#Cc1cnc(C(F)(F)F)cc1N1CCN(C(=O)C=Cc2cccc(F)c2)CC1 33279,C#CCCCC(C)C(=O)NC1CCN(C(c2ccc3c(n2)CCC3)=O)C1 33280,C1(C(=O)NC2CCC(CN(C)C(C34CC(CO)(C3)C4)=O)CC2)CCOCC1(C)C 33281,CCC(CNC(=O)C(C)OCOC)N(C(=O)C=CC(=O)OC(C)(C)C)C 33282,c1(C(N2CC3C(NCC4(OC)CCC4)C3C2)=O)cc(C(F)F)ccc1[N+](=O)[O-] 33283,c1(C(CN2C3(CCCC3)C2=O)O)cccnc1.c1(C(=O)NCCO)cc(Cl)no1 33284,c1(C(N(CC(CC)NC(=O)C(=O)NCC)CC)=O)ccnn1C(C)(C)C 33285,c1(NC(C2C=CCN(C(=O)CCc3nccs3)C2)=O)cc(F)c(CO)c(F)c1 33286,N1(S(=O)(=O)Cc2ccccn2)CC2CN(Cc3ccc(Br)c(O)c3)CC2C1 33287,CC1CCCCN1N1CCC(C(=O)OC(c2ccco2)=O)C1.C12CC(C)(C1)NC2=O 33288,c1(C(=O)NCC2COCC2O)ccnc(C2(n3cc(C4CC4)nn3)CC(OC)C2)c1 33289,c1(C(C)C)nn(C)c(NC(C2CCCC(NC(c3cccnc3)=O)C2)=O)c1Cl 33290,c1(OC)cc(Cl)c(Cl)cc1C(=O)NCCC(C)NC(C1CCC1C)=O 33291,C1(C(=O)OCCNC(COC(CC)(C)C)=O)CCC2(CC2)N1C(=O)C1CC1 33292,C1(C)(N(C)C)CCN(C(C2CC(=O)CN2C(C2CN(C(N)=O)C2)=O)=O)C1 33293,C1(C(N2C(CNC(=O)Cc3cnns3)CC(OC)C2)=O)Cc2ccc(C)cc2S1 33294,c1(CC(=O)NC(CC)CN2CC(CN(C)C(C)C)C2)c[nH]nc1C 33295,C=C(Cl)C(C)(C)C(=O)NCC(O)CCNC(C1CC1CCC)=O 33296,C1(CC(=O)NCC(CNC(CN(C)C2CC2)=O)F)CC2(COC2)C1 33297,c1(CC)c[nH]cc1C(=O)NC(CO)C(=O)NCCCn1cncn1 33298,CC1SCCCC1C(=O)N(CCCN(C(=O)CC1(OC(C)C)CC1)C)C 33299,C(=O)(C(C)(C)OC)N1CC(C(C(=O)NCC=CC2CC2)OCC)C1 33300,CC1=NS(=O)(=O)NC=C1C(=O)NC1CC(C)N(C(C2CCCC3CCCN23)=O)C1 33301,c1(C(=O)NCC2CCCC(CNC(C(C)=C3CCC3)=O)C2)cc([N+](=O)[O-])c[nH]1 33302,C12(C(N(C(CCNC(C=C(CCC)CCC)=O)C)C)=O)CC1CCC2(F)F 33303,Nc1ccc(F)c(C(=O)NC2CN(C(=O)Cc3ccoc3)CC3CC23)c1 33304,C1(NC(c2cc(F)c(F)c(F)c2)=O)CC1C1CCCN(C(c2coc(O)n2)=O)C1 33305,C1(NC(=O)CCc2cc(F)ccc2Br)CN(C(C2(F)CC2)=O)CC(F)(F)C1 33306,N1(C(C(C(C)C)n2cnnc2)=O)CCN(C(=O)C(N)=O)CC(O)C1 33307,CC1CN(C(=O)CCc2cn[nH]c2)CCC1NC(=O)CCc1cnn(C)c1 33308,c1(C(=O)NC2CC(NC(=O)CC3C=CS(=O)(=O)C3)C2)ccc2c(c1)NC(=O)CN2 33309,c1(C(N2CC(N(C)C(c3cc(F)cnc3O)=O)C(F)C2)=O)c(F)ccc(F)c1Cl 33310,c1(C(N(C(C)CCNC(=O)C=CC2C(C)C2(Cl)Cl)C)=O)n[nH]c2c1CCCC2 33311,c1(CCNC(=O)C(C)NS(C)(=O)=O)ncccn1.C(CN1CC1)OC 33312,C(=O)(C1COc2ccc(Cl)cc21)NC1C(NC(c2c(CC)occ2)=O)CCC1 33313,N1(C(C=CCNC(C2CCC(CC)O2)=O)=O)CCC(O)C(F)C1 33314,C1(C(N2C(C(C)NC(C(C=C)O)=O)CCC2)=O)(OC(C)=O)CCCCC1 33315,N1(C(C(C)CC(F)F)=O)CC(NC(c2cnn[nH]2)=O)C(S(C)(=O)=O)C1 33316,c1(C(N2CCC(C)C2CNC(=O)Cc2cnsc2)=O)cnc(O)c([N+](=O)[O-])c1 33317,C(=O)(C1c2c[nH]nc2CN1C(C1CCC(F)CC1)=O)NCc1c(C)cc(C)nc1 33318,C1(C(=O)NCCCN(C(c2c(C)cno2)=O)C)CC2CCC1CC2 33319,c1(N2CCc3c(ccs3)C2)nc2ccsc2c(=NC2CC(Cc3nccs3)C2)[nH]1 33320,CCC(C)C(O)C(C)C(=O)NCC12CC(CO1)N(C(C1(C)CCC(=O)C1)=O)C2 33321,N1(C(c2cn(C)c(=O)cn2)=O)CCCC(C)(C)C1CNC(=O)C1=NOCC1 33322,CC(C)(C)CCC(=O)NCCCC1CCCCN1C(C1CCC2(CCC2)C1)=O 33323,C12(CNC(c3cc(CO)on3)=O)CCC(CC1)CN2C(=O)CC1C=CS(=O)(=O)C1 33324,Cn1ccnc1C(=O)NC=O.C12CCN(C1)C2=O.c12cc([nH]n1)C1CCCN1C2=O 33325,C1(CNC(CCc2ncc(C)[nH]2)=O)CC(NC(c2sc(C)cc2Cl)=O)C1(C)C 33326,n12cc(nn1)CC(C1CC1)NC(=O)C2C.C(CCCOC)OC 33327,C1(C(=O)NCC(CNC(c2cn(C(C)C)nn2)=O)C)CCCC(=O)O1 33328,C1(NC(C(C(C)C)N(CC)CC)=O)CC2(CCN(C(=O)C=C(Cl)Cl)C2)C1 33329,Cc1nc(CC(=O)NC(C)CCN(C)C(c2cnc(Cl)s2)=O)c(C)s1 33330,C1(OC2(ONC(C(C)NC(CC)=O)=O)CCC2)C2CCCC1COC2 33331,C(=O)(C(O)CCS(C)=O)N(C(C)C)CCNC(c1sccc1OC(F)F)=O 33332,C1(C(C)C)C(NC(=O)Cc2cncs2)CCN1C(C1OCCO1)=O 33333,Cc1nn(CC(=O)NC2CC2NC(C2(C)CC(C)(C)C2)=O)c(C)c1Cl 33334,c1(C(=O)NC2(CNC(CP(C)(C)=O)=O)CC2)cc2cc(Cl)cnc2[nH]1 33335,c1(CC(=O)NCC(C)(O)CNC(=O)CCc2cnc[nH]2)c(F)cccc1F 33336,C1(C(N2CC3C(NC(C4CC5COCC5C4)=O)(C3)C2)=O)CC2(C1)CC(F)(F)C2 33337,c1(CC(=O)NCC=CCNC(C2C(Br)(C(=O)OCC)C2)=O)cccnc1 33338,C1(N(C(c2oc(CC)c(C)c2)=O)C)CCCC2CN(C(=O)C(C#N)C(C)C)CC12 33339,N1(Cc2cn(CCC)nc2C)CC(=O)N(C(c2ccc(Br)cc2)(C)CO)C1=O 33340,C(=O)(C(CNC(=O)CC1CCCO1)N(C)C)NC(C)C(=O)NCCF 33341,c1(C(N2CC(NC(c3cc(COC)sc3)=O)C(C)C2)=O)nc(OC)ccc1F 33342,c1(C(=O)NCC2N(C(CC(=O)OC(C)(C)C)=O)CCOC2)cc2ncccc2s1 33343,c1(OCCC)cccc(OC)c1CNC(=O)CCCCOc1ccc(C)cc1Br 33344,c1(C(C)C(=O)OCc2cc(C(F)(F)F)no2)ccc(C(F)(F)F)cc1 33345,C1(C(C)C)C(C(=O)NCCN2CCNC(=O)C2)CCN1C(=O)CC1CCSC1 33346,C(=O)(CCCN(C)N=O)N1C(C2CCCN(C(CN(C(C)=O)C)=O)C2)CCC1 33347,C1(C(N2CC3(CCN(C(c4ccc([N+](=O)[O-])o4)=O)C3)C2)=O)CC2CC(O)C(C1)C2 33348,C(CCCCCNC(C1CCC(C(=O)OC)CC1)=O)NC(CCOCCC)=O 33349,CCCCC(CC)C(=O)N1CCC(=CCNC(C2(CC3CC3)CCCO2)=O)CC1 33350,N1(C(CC(CC#C)NC(=O)CC2CCCCC2O)=O)CC(=O)NC2(CC2)C1 33351,N1(C(c2cccc(C)c2)=O)CCN(C(c2ccn(CCO)c2C)=O)C2CCC12 33352,c1(C(=O)NC2CN(C(C(CO)NC(C(C)C)=O)=O)C2)ccc2c(c1)CCN2C 33353,C1(O)(N(C2CN(C(=O)OC)C2)C)CCN(C(c2ccc(F)c(C(F)F)n2)=O)CC1 33354,C(=O)(CC(C)(C(F)F)N(C)C)NC(CN(C(c1ccc(C)cn1)=O)C)C 33355,Cc1cc(CC(N2CCCC2CNC(c2ccn(C)n2)=O)=O)ccc1Cl 33356,C1(C(=O)NC(C)(C)CNC(=O)C=CC2(C)COC2)CS(=O)(=O)CCO1 33357,c1(CC)cc(C)c(C(=O)NC2COC(C3CCNCC3)C2)o1 33358,CC1(CCNC(c2cnn(-c3ccc(F)cc3)c2)=O)CCN(C(=O)C(Cl)=CCl)C1 33359,c1(SC(C(=O)NC(CNC(c2cc(CCC)on2)=O)C)C)ccc(F)cc1 33360,C1(CN(CCCO)CC)SC2(CCC2)C1O 33361,C(=O)(CC(C)(C(F)F)Nc1ocnc1-c1nc(C2CC2(F)F)no1)N(C)C 33362,N1(C(C2N(C(C)=O)CSC2)=O)CCCC1(C)c1cn(CC=C(C)C)nn1 33363,N1(C2CCN(C(CC=C)=O)C2)CCN(C(C2CC23CCOC3)=O)CC1=O 33364,C12(C(=O)Nc3cccc(C)c3)CCCN(c3ncc(F)cn3)CC1C2 33365,C1(CC#C)CN(C(=O)COC2CN(C(=O)CSC(C)C)C2)CCO1 33366,c1(CCCOC)noc(-c2cnn(-c3cncnc3)c2)n1.C1C(=O)O1 33367,C(C(CC(F)(F)F)NC(=O)C1=NOC(C)C1)NC(C(NOC)=O)=O 33368,c1(CNC(c2nc(CC)oc2C)=O)ccc2c(c1)CN(C(=O)C(=O)N1CCCC1)C2 33369,N1(C(C(C2CCCO2)OC)=O)CCC(N(C(=O)C=CC2CCCCC2)CCO)CC1 33370,c1(CC(=O)N(C)CCNC(=O)Cn2nnc(=N)[nH]2)cccc(C2(C#N)CC2)c1 33371,N1(C(C2N(CCC)CCOC2)=O)CCCCC(NC(c2cccc(CO)c2)=O)C1 33372,C(=O)(CCC(C)(C)NC(=O)C(F)C1CCC1)N(CCN1CC=CC1)CC 33373,c1(OC)cncc(C(=O)NC(CN(C(C2CN(C)CCO2)=O)C2CC2)CC)n1 33374,C1(NC(=O)Cc2ccon2)(CO)CCN(C(C2CCCCC2O)=O)C1 33375,C(=O)(C#CC1CCCCC1)NC(CC)CNC(=O)CC(C)(O)COC 33376,N1(C(=O)C2=COCCO2)CCOC2(CCS(=O)(=NC(=O)CCC3CCC3)CC2)C1 33377,Cc1cc(O)nnc1C(=O)NC1CC(CNC(c2oc(CC(C)C)nc2C)=O)C1 33378,C1(C(N(CC(CO)(CO)NC(CC2CN(C)C2)=O)C)=O)CCn2cncc2C1 33379,C1(NC(c2[nH]c(=NC)sc2)=O)CN(C(c2ccnnc2O)=O)C2(CCCCC2)C1 33380,C1(COC(C(c2ccc(C(F)(F)F)cc2)(C)C)=O)CC1C1CCOCC1 33381,CCCCS(=O)(=O)CC(=O)NC1CCOCC1NC(c1cccn1C(C)C)=O 33382,N1(C(CCCCN(C)C)=O)CCC2(CCCN2C(=O)Cc2cccs2)CC1 33383,N1(c2nc(C)c(Br)cn2)CC(NC(c2ncc(Cl)s2)=O)CC(C)(C)C1 33384,N1(C(c2c(OC)oc(C)n2)=O)CCC12CN(C(C1CC3(C1)CC3F)=O)C2 33385,C(=O)(CCC(=O)C(C)(C)C)N1C2C(C(N(C)Cc3c(C)nsc3)=O)(CCC2)CC1 33386,Cc1ccc(C)c(OCC(N2CCC(O)(C(=O)NCc3csc([N+](=O)[O-])c3)C2)=O)c1 33387,C1(Cn2cc(C(CC)OC)nn2)CN(C(c2ccc(C(C)C)s2)=O)CC1C 33388,Cc1ncc(C(F)(F)F)cc1C(N1CC(CNC(C2CCCC2)=O)CCC1C)=O 33389,c1(CN(C2CCN(C(C)(C)C)C2)C(=O)NCc2c(CC)ocn2)oc(C)nc1C 33390,c1(C(=O)NCC2(NC(c3c(CC)nns3)=O)CCCC2)cc(C2CC2)nn1C 33391,c1(C(=O)NC2CCC(NC(c3cn(CCC)nn3)=O)CC2)ccc(O)nc1Cl 33392,CCC(C(=O)NCCC(O)CNC(=O)C(C1(C#N)CCCCC1)=C(C)C)C(F)(F)F 33393,N1(C(CNC(=O)CC2CCCC2)=O)CCN(CCC23CC(Br)C2C3)CC1 33394,Cc1ncccc1CCC(=O)NC(C)CNC(c1cn(CCO)nn1)=O 33395,C1(CN(C(=O)Cn2cncn2)C)CCC(CNC(=O)C=CC)CC1.[nH]1cnnc1 33396,Cc1nn(C2CC2)cc1C(=O)NCC1CCN1C(=O)C(F)(F)CN(C)C 33397,CCCCCC(C)CC(=O)NC1CCCCC1N(C(=O)Cc1cncs1)C 33398,N1(C(C=Cc2cn(C)nn2)=O)CCN(C(c2ccsc2C#N)=O)CC(CO)C1 33399,C(=O)(C#CC1CCCO1)N1CCCC(CN(C(=O)CCOC2CCCC2)C)C1 33400,c1(OC)cc([N+](=O)[O-])c(CC(=O)NCc2ncc(C)c(OC)n2)cc1Br 33401,C(=O)(C(C)C(F)(F)F)N1CC(C2CC2)(CNC(C(c2c(C)cccc2)C)=O)C1 33402,C1(NC(C=CC=CC)=O)CCCC12CN(C(c1cccc(C(F)(F)F)n1)=O)C2 33403,c1(C(=O)NCC=CCNC(c2n[nH]c(CSC3CC3)n2)=O)cc2cnccc2o1 33404,C1(NC(COCC(=O)OC)=O)CCCCN(C(c2cc(Br)sn2)=O)C1 33405,C(CCCOC)(C(=O)N1CC(C(C)C)C1)NC(c1nn(CC)c(O)c1)=O 33406,c1(CN(C)CC2CCN(C(=O)Cn3ccc(C(F)F)n3)C2)cc2cnccc2o1 33407,N(C(=NCCCCl)NCc1ncoc1-c1ccccc1Cl)CC1CC(=O)NC1 33408,C1(OCCCOC(=O)OC(COC)CF)CCOC1 33409,N1(C(C(N2CCC(C)C2)=O)=O)CCC(O)(C(=O)N(c2ccccc2)C)CC1 33410,C1(NC(C(=O)NCC)=O)(CO)CCCN(C(c2ccccc2Cl)=O)C1 33411,c1(C(=O)OC)nc(=NC2CC(F)(CNC(=O)C3CCc4ccccc43)C2)cc[nH]1 33412,Cc1c(Cl)cc(C(N2C3CCC2CN(C(c2c(Br)cccc2Br)=O)C3)=O)cc1Cl 33413,CCC(C(=O)N1CC(NC(c2csc(C)c2OC)=O)C1)C(C)C 33414,C1(CC)CN(C(=O)CC(C)C(C)C)CCN1C(C1CN(C)C1)=O 33415,C1(NC(CC(C)(C)SC)=O)C2CCC1N(C(=O)COCc1ccncc1)C2 33416,CCC(C(=O)N1CC(CN(C)C(c2cccc(NC(=O)C3CC3)c2)=O)C1)C(C)O 33417,C#CC1(NC(=O)CCCC(C)NC(C2CC2c2ccccc2)=O)CCCCC1 33418,C1(NC(c2ccccc2C2CC2)=O)CN(C(C2CC2(F)F)=O)CC1n1ccnn1 33419,C(=O)(C1=C(Cl)CCCC1)N1C(C(=O)NCCNC(COCC)=O)CC(F)C1 33420,C1(NC(c2nc(C(C)NC(CC(C)C)=O)oc2)=O)CCN2CCC1C2 33421,C(CC(O)CCc1cn(Cc2cccs2)nn1)NC(=O)CCCc1cncs1 33422,CCC(C)C(C(=O)OC)N(C(=O)CCCN(C)C(C1COCCN1C)=O)C 33423,N1(C(C2C(C)C2)=O)CC2CC(NC(=O)C(F)(F)Cc3ccc(Br)cc3)C1C2 33424,C1(CNC(C(CCOC)C)=O)CCC2(CN(C(C3CCOC(C)C3)=O)C2)O1 33425,C(=O)(CCc1ccc[nH]1)NCC(C)NC(=O)CCOCC1CCCC1 33426,c1(CC)ccc(C(=O)NCCC2(NC(=O)Cn3ncnn3)CC2)c(O)c1 33427,c1(OC)ccc(C(F)(F)C(=O)NC2CN(C(=O)Cc3ncccn3)CC2F)cc1 33428,N1(c2ccc(C)cc2)CCCC(NC(=O)NC2(C(F)(F)F)CCOCC2)C1=O 33429,C#Cc1ccc(CCC(=O)N(C2(CCN3CCC3)CC2)CC)cc1 33430,Cc1cc(C(=O)Nc2ccc(NC3CCC(=O)C3)c(C)c2)cc(=O)o1 33431,CC(C)(CS(N)(=O)=O)C(=O)N1CCN(C(c2cnc3n2CCC3)=O)CC2(CC2)C1 33432,C(C(CC(C)C)C(=O)NCC(C)(C)NC(=O)CCC1CCCN1C)OC 33433,C=CC(C(=O)NCC1CCN(C(=O)Cc2cnccn2)C1)NC(=O)OC(C)(C)C 33434,C(N=c1nnc(C)c(C)[nH]1)C1C(NC(c2ccc(C)c(F)c2)=O)CCC1 33435,N1(CC2(C(=O)OC)CCC2)CC(CC(=O)NCC(=O)NC)C2(CC2)C1 33436,N1(C(c2cc(OC)sc2)=O)CCN(C(=O)C(C)(C)c2cccs2)CC1C1CCC1 33437,c1(N2CCC(C)(CC)CC2)nc(=NCC(C)SC)[nH]c2cc(OC)ccc12 33438,c1(C(N(CC(C(=O)N(C(C(=O)OC)C)C)C)C)=O)cccc(O)c1 33439,C(CC(C)C(=O)NC1CCN(C(C2CC2n2cc(Cl)cn2)=O)C1)=CC.C1C(=O)O1 33440,C1(C(=O)NCC(C)NC(c2cc(Cl)ncc2N)=O)CCc2cc(F)ccc2O1 33441,CC1CC(NC(=O)C=C2CCC(C(C)(C)C)CC2)CN(C(=O)C2=CCCCC2)C1 33442,CCCC(CCCNC(=O)C(N1CCCC(O)C1)C)Nc1ncnc(C)c1F 33443,Cc1cccc(C)c1NC(=O)C(c1cc(Br)ncc1F)N1CCC(C(F)F)CC1 33444,C(=O)(CCCCC(=O)NCc1ccc(NC(c2cccc(Cl)c2)CO)nc1)OC 33445,CC(C)CCC(F)C(=O)NC1CC1CNC(c1cc(C(N)=O)n(C)n1)=O 33446,c1(SCC(=O)NCCC2CCCN(C(C=C(C)C)=O)C2)nc2ccccc2s1 33447,Nc1nc(C(N2CC(NC(c3cnns3)=O)CC(O)C2)=O)cnc1Br 33448,C(=O)(C(C)(F)CC)NCCC(=C)CNC(c1ccc(OC(C)C)nc1)=O 33449,c1(CN(CC(C)C)NCc2cnns2)nnc2n1CCOCC2 33450,c1(N2CCC(=O)C2)cccc(Cl)c1Cl.N12CC3(CC3C1=O)C2.N12CC3C(C3C1)C2=O 33451,c1(C(N(CC(CC)NC(C2(C(C)C)CCC2)=O)C)=O)c(C)nc2sc(C)nn12 33452,C1(CNC(c2cc(COC)no2)=O)CCCCN(C(=O)Cc2cncn2C)C1 33453,CCCC(CC)C(=O)N1CC2C(CC(=O)NC3CCN(CCO)CC3)C2C1 33454,N1(C(c2nc(CCC)sc2)=O)CC(CNC(=O)C=CC2CC2)C2CC12 33455,Cc1cccc(OCC(=O)NCCN(C)C(C2CC(C)(C)CCO2)=O)c1C 33456,N1(C(CC(C)OC)=O)CCN(C2CCCN(C(C3CCCC(O)C3)=O)C2)CC1 33457,CC1(C)CC(C(N2CCOC(CF)C2)=O)CCN1C(=O)CCc1nncs1 33458,C1(NC(C(C)(C)C2CCC2)=O)C2CC(NC(=O)CC3CCCSC3)CC12 33459,CC1CCN(C(=O)C(=O)NCC(c2cnn(C)c2)C)CCS1 33460,c1(NC(C2C(C)CCCC2)=O)cnc2ccc(F)cc2c1 33461,CC1(C)CC(C(=O)NCCNC(c2cc(C3(C)CC3)n[nH]2)=O)C(C)(C)O1 33462,c1(C(C)(C)NC(=O)NC2CC2NC(C2CCN(C)C2)=O)cccc(C(F)(F)F)c1 33463,c12ncnc(c1C)NC1CCN2C1.C(CN1CCCCC1)(C(C)C)SC 33464,C1(O)(CNC(c2cccnc2)=O)CN(C(C2CC2[N+](=O)[O-])=O)C1 33465,c1(C(N(CC)CC2CCCN(C(=O)CC(C)(C)OC)C2)=O)cnc(C)c(N)c1 33466,Cc1cnc(C(N2CCC(CO)(NC(=O)OC(C)(C)C)C2)=O)cc1C 33467,C1(CC(=O)NCC2(F)CCN(C(c3cc(C)[nH]n3)=O)CC2)CCCC2(CCC2)O1 33468,Cc1cc(F)cc(C)c1C(=O)NC1CCC(CNC(c2ccc(C(N)=O)cc2)=O)C1 33469,c1(CCC(=O)NC2CCCC(C(=O)O)CC2)nc2ccc(Br)nc2[nH]1 33470,N1(C(c2cn(C)nc2)=O)CC=CC(NC(C2CCCC2(C)C)=O)C1 33471,Cc1cc(C(=O)NC(Cn2cncn2)C(=O)O)on1.c12cn(nn1)CC(=O)N2 33472,c1(C(N(CC(CO)(CO)NC(C2C(C)C2C)=O)C)=O)n[nH]c2c1CCCC2 33473,C1(CNCC23C(CN(C(=O)Cc4cnc[nH]4)C2)C3)COc2ccccc2O1 33474,C#Cc1ccc(C(=O)NC2CCCC(NC(C3CC(CC)=NO3)=O)C2)nc1 33475,C=CCCCC(=O)NCC(CC=C)NC(=O)C(=C1CCCCC1)F 33476,c1(C(=O)NC2(CO)CN(C(C3C(C)(CC)C3)=O)C2)oc2ccccc2c1C 33477,N1(C(c2nc(CC)oc2C)=O)CCC2CN(C(c3cn(C)nc3OC)=O)CC12 33478,C=C(C)CCC(=O)NCC(CO)NC(=O)CC(C)C 33479,C(=O)(C(C)(C)C(C)O)NCC(C)N(C(Cc1ccc(C(C)C)cc1)=O)C 33480,C1(NS(=O)(=O)CCOC2CCOC2)CCCC12CCCO2 33481,C(=O)(C1=NOC2COCC12)NCCCCCCNC(C(C(=O)NC)(C)C)=O 33482,c1(C(=O)NC2C(C)N(C(=O)Cn3ncnn3)CC2)cc2c([nH]1)CCOC2 33483,CC(C)(CCC(=O)NC1CCCC1N1CCC1)NC(=O)CC1CC=CCN1C 33484,CCCCC(CCCC)C(=O)NC1(CNC(=O)C(O)CC(C)C)CCCC1 33485,Cc1nncc(C(N2CC=C(CNC(C3CCO3)=O)CC2)=O)c1C 33486,C(C)(CNC(C1CCCN1C(C1(C)CCCS1)=O)=O)(CO)OC 33487,C1(OCC)CCCCCC1NCCc1ccc(C)nc1 33488,c1(CCC(N2CCC(C)(CNC(C(C)SCC)=O)C2)=O)nc2ccc(C)cc2[nH]1 33489,C(CC(C(C)(C)C)NC(=O)CN1CCN(C2CC2)C1=O)N(C(C1CC(=C)C1)=O)C 33490,c1(CC(C)NC(C(=O)NC(c2c(OC)cccc2)C(C)N)=O)ccc(C)c(C)c1 33491,C=CC(CC)CC(=O)N1CC(O)(C(C)(C)CNC(C2CCCN(C)C2)=O)C1 33492,c1(S)ccc(OC(C)C2CC2)cc1.Cc1nnc(CNC(=O)C(=O)N)o1 33493,CC1(C(=O)NCC2CC(NC(=O)CCc3cnoc3)C2)CC(C#N)C1 33494,c1(OC)ccc(Cc2cc(C)c(-c3ccc(CN(C)C)cc3)cc2O)cc1C 33495,C1(N(C)C)(C(=O)NCC(O)CCNC(=O)CCC2CCC2)CCOCC1 33496,C12(NC(C(CC)n3nnc(-c4cc(Cl)ccc4Cl)n3)=O)CCC(C1)N(C(C)=O)C2 33497,c1(OC)cc(C(=O)N(CCCn2cc(C3(OC)CCOC3)nn2)C)ccn1 33498,C1(C2CCCC2)(NC(C2C(C)CCN2C(=O)C(C)n2ccnn2)=O)CC1 33499,C(C(=O)N1CC(COC)(CNC(c2cnc(C3CC3)s2)=O)C1)(C(C)(C)C)OC 33500,C(=O)(C1=NOC2(C1)CN(C(c1cc3cncn3c(O)n1)=O)C2)OCC 33501,c1(N(C)Cc2ccoc2)ccc(S(=O)(=O)NC2CC3CCC(C2)S3)cc1F 33502,c1(C(=O)NCCCN(C(C(CSC)O)=O)C)ccc2c(c1)CC(=O)NC2 33503,C=CC(C)(O)CC(=O)N(C)CCOCCCNC(=O)CNC(=O)CN(C)C 33504,C1(NC(c2n(C=C)nnc2)=O)CN(C(=O)C(O)Cc2[nH]cnc2C)C2(CCC2)C1 33505,C1(CNC(C(C)Sc2nncn2C)=O)CCCC(NC(=O)C2CC2)C1 33506,N1(CC)CC(C(N2CC3CC2C3NC(=O)CSc2n[nH]c(C)n2)=O)CCC1=O 33507,N1(CC)CCCCC1C(=O)N(C1CCN(C(=O)CCSc2ccccc2C)C1)C 33508,c1(C(=O)NCCC23C(CN(C(CCOCC)=O)C2)CC3)sc2ccccc2c1C 33509,c1(OC2CC(C(=O)NC3CC(C(C)CCO)C3)C2)ccc(Cl)c(F)c1 33510,c1(N2CCC(NC(C3ON=C(C)C3)=O)C2)nc(C)c(C#N)cc1Cl 33511,c1(-c2cnc(OC)nc2)ccc2[nH]c(C(=O)NCC3(C(F)(F)F)CC3)nc2c1 33512,N1(C(C)C)CC(C(=O)NC2CC(CCNC(C3CCC(=O)N3)=O)C2)CC1=O 33513,c1(CC(N2C(C)CC(CNC(c3cnc(O)s3)=O)CC2)=O)c[nH]c2cccnc12 33514,N1(C(c2nc(C)n(C)c2)=O)CCCC(NC(c2[nH]ncc2C#N)=O)CC1 33515,CCCC(CC)C(=O)NC1(CNC(c2ccc(C)cn2)=O)CCCC1 33516,N1(C(c2ccc(OC)o2)=O)CC(NC(C2CCS(=O)CC2)=O)C(O)C1 33517,N1(CC(=O)NC(c2nc(C)on2)C)CCCC1(C)C 33518,c1(C(N2C(CNC(CS(CCC)(=O)=O)=O)CC2)=O)cc(C)ccc1S(N)(=O)=O 33519,CC(C)(C)C(C(=O)NC1CC(NC(C23CCCC2C3(F)F)=O)C1)C1CCCC1 33520,CC1CN(C(C2CC(F)(CO)C2)=O)CC(C)CN1C(c1cccn(C)c1=O)=O 33521,CN(C)S(=N)(=O)N1CCCC1C(=O)NCCC(O)CNC(c1sccc1Cl)=O 33522,c1(C(=O)NC2CN(C(C)=O)C2)ccnc(C2CC2)c1.N12CC(C1)C2=O 33523,C1(CCC(=O)NCCC(C)N(C(C(C)=C(CC)C)=O)C)CCC(=O)NC1 33524,C1(NC(=O)NC(C(C=C)Sc2cn(C3C(CN)C3)nn2)=O)CCC2(CCC2)C1 33525,C(=O)(C(O)CC(C)(C)C)N1CC(CNC(c2cc(N(C)C)ncc2)=O)C(O)C1 33526,N1(C(c2cc(CNC(c3cc(C)sn3)=O)[nH]n2)=O)CC(C)(C)OC(C)(C)C1 33527,Cc1cnc2c(C(=O)NCC(C)NC(C3CC34CCCCC4)=O)cnn2c1 33528,CS(=O)C=CC(=O)NCC1C2CN(C(C3CC(O)(c4cccnc4)C3)=O)CC12 33529,c1(C2(C(N(C3CC(n4ccnn4)C3)C)=O)CC2)ccc(N)o1 33530,CC1Cc2cccc(NC(=O)Nc3nccnc3OC3CCCCC3)c2O1 33531,c1(C(N2CC(F)(CNC(C(c3scc(C)n3)C)=O)C2)=O)cncc2nc[nH]c12 33532,c1(C(N(CC)Cc2nnnn2C)=O)ccc(CNC(C2CC2(F)F)=O)o1 33533,c1(C(=O)NC(C(=O)NC(C(=O)NCC)C)C2CC2)ncncc1C 33534,C1(C(=O)OC)(NC(C2CCCC2CNC(C2CCCS2)=O)=O)CC(F)(F)C1 33535,S(=O)(=O)(c1ccn(C)n1)N(C)CC1CN(C(c2cc(C)nc(C)c2)=O)C1 33536,C(c1cccc(F)c1Cl)=CC(=O)NCCCCCNC(Cc1cn(C)nn1)=O 33537,c1(C(c2ccccc2)NC(=O)NC(CCOC)COC)cc(C)ccc1C 33538,c1(CNC(C23CC(NC(c4ccncn4)=O)(C2)C3)=O)cnc2ncccn12 33539,C1(O)(C(C)N(C(=O)CC(C)C2CCCO2)CC)CCN(C(=O)CC(C2CC2)C2CC2)C1 33540,CCCC(CCCNC(=O)CC1COCC1(C)C)NC(c1cnc[nH]1)=O 33541,C1(NC(C(CC)CC)=O)CCC(C)N(C(=O)C(c2cccc(Br)c2)C)C1 33542,c1(OC)c(C(N2CCC2CNC(c2cc(C)ncn2)=O)=O)cc(Cl)cc1Cl 33543,Cc1cccc(Br)c1C(C(=O)N(CC(C)(F)F)C)NC(c1nn(C)cc1C)=O 33544,c1(C(=O)NCC23CCCC(CCC2)C3O)ccc2c(c1)C1(CC1)C(=O)N2 33545,Cc1cccc2c1OCCC2N(C)Cc1csc(CN)n1 33546,CCCS(=O)(=O)C(C)C(=O)NCC1CC2(C1)CN(C(C1CC1(C)C)=O)C2 33547,C1(C(N2CCC(N(C(COCCC#C)=O)CCC)CC2)=O)CC2(C1)CC1(CC1)C2 33548,c1(C(=O)NC(CNC(c2cc(CC)n(C)n2)=O)CO)cc(C(C)C)ccc1N 33549,c1(C(N2CCC(Cn3cc(-c4cc[nH]n4)nn3)C2)=O)ncc(Cl)s1 33550,C1(CNC(C2CC(C)N(C)C2)=O)CCC(F)(CNC(=O)CC2=CCCC2)CC1 33551,CC(CC(F)(F)F)C(C(=O)NCC1CCCO1)N1CCCC1CCCO 33552,C=CC1(C(=O)N(C2C3CCCC23)C)CCN(C(c2cccnn2)=O)C1 33553,C1(NC(c2ccc(N)c(CO)c2)=O)CCCCCC1NC(C1(N(C)C)CC1)=O 33554,C1(COC)(CNC(=O)COC(C)C)CCN(C(=O)COc2ccncc2)CC1 33555,c12cnc(o1)C2.O=C(CCNC(C1CCC1)=O)C1CC1.C12CC1CNC2=O 33556,Cc1ncc(C(=O)N(CC(C)NC(=O)CSc2n[nH]c(O)n2)C)cc1C(F)(F)F 33557,c1(OC)ccc(C(F)(F)F)cc1C(N1CC(NC(C2COC(C)CO2)=O)C1)=O 33558,C(=O)(N=c1cc2ccccn2[nH]1)C1(C)CCCN(C(C2CCCCN2C)=O)C1 33559,c1(N(C)C)ccc(CNC(C2CCN(CC3CC3(C)C)C2)=O)cn1 33560,c1(C(=O)OC(NOCC(C)(C)OC)=O)cnoc1C1CCOCC1 33561,N1(C(CSC(C)(C)C)=O)CCN(C(=O)C(F)C(C)(F)F)CC1c1cn[nH]c1 33562,Cc1cc(C(=O)NCC(C)(CO)NC(=O)C=Cc2nccs2)ccc1Cl 33563,C1(OC)(CNC(=O)CCCn2cncn2)CN(C(=O)CCc2ccc(C)s2)C1 33564,c1(SCc2c(C)nc(F)cc2)c(C(N2CC3CCC2C3)=O)[nH]c2ccccc12 33565,C(C)(C(=O)NC1CC1NC(=O)COCC1(F)CC1)OCC=C 33566,c1(CCC(=O)NCC2CCCN2C(=O)C=Cc2cscn2)ccncn1 33567,CN1C(=O)CCC(NC(=O)CN(C(c2csc(CO)n2)=O)C2CC2)C1=O 33568,N1(C(COCCCC)=O)CCC(C)(CCNC(C2CC(C)C2)=O)C1 33569,Cc1nn(C)c(C)c1C(N1CC2CC2(CNC(C2(C)CC2(F)F)=O)C1)=O 33570,C1(CCNC(=O)Cc2ccon2)CCN(C(=O)CC2CCC3(CCC3)O2)CC1(F)F 33571,C1(C(N(C2CCCC2)CC#C)=O)CN(C(c2cc(C)ncn2)=O)C(C)(C)C1 33572,N1(C(c2c(CC)[nH]cc2)=O)CC(C(N2CCCC(COC(C)=O)C2)=O)C2(CC2)C1 33573,Cc1ccnc(C)c1CNC(=O)C(C)(CC1CCC1)NC(C1COCOC1)=O 33574,C1(N(C(c2cc(C(CC)C)no2)=O)C)C2CN(C(=O)CCN3CCCC3=O)CC12 33575,c1(SCC)cccnc1C(N1CCOC(CNC(=O)CCCN2CCCC2)C1)=O 33576,S(=O)(=O)(c1cccnc1N1CSC(C)C1)NCC(C)(C)NC1CCCOC1 33577,CCCCC(F)C(=O)NCCC1CCC(NC(c2c[nH]c(=N)c(C)c2)=O)C1 33578,CCC(C)(C)C(=O)C(=O)N1CC(F)(C(=O)N(C2(CCO)CC2)C)C1 33579,c1(C(=O)NC2C(CNC(C3C(c4c(C)occ4)C3)=O)CCCC2)cn(C)c(=O)cn1 33580,c1(C(N(C(CNC(C2CCC(=O)O2)=O)C2CC2)C)=O)cc2ccccn2n1 33581,N1(C(COc2c(C)cccc2)=O)CCC(C)(C)C(CNC(=O)Cc2csnn2)C1 33582,c1(CC)cccc(N(C)C(c2cc(CNC(=O)CC3CC=CCC3)no2)=O)c1 33583,C(=O)(C(C)(C)NC(=O)NC1CC=CC1)NCCOCCC#C 33584,C1(OC)CCCC(CNC(=O)C=CCN(C(=O)Cn2cncn2)C)C1 33585,C1(C(=O)NCC2(NC(c3cncc(-c4ccccc4)c3)=O)CC2)CCCS1(=O)=O 33586,C(=O)(C(O)C(F)(F)F)N1C(CN(C(c2ccc(CC(C)C)s2)=O)C)CCC1 33587,CC1COCCCN1C(=O)COCCNC(c1cccc(F)c1F)=O 33588,Nc1cnc(Cl)c(C(N2CCOCC(NC(c3ccc(F)s3)=O)C2)=O)c1 33589,c1(SC(CC(=O)NC(CNC(c2ncn(CC)c2)=O)C)C)cccc(OC)c1 33590,c1(C(N(C)CCC2CCN(C(C3CCCN3C)=O)CC2)=O)cc(O)c(O)c(O)c1 33591,Cc1ccc(Br)cc1C(N1CCC(N(C(=O)C=C2CCC2)C)C(C)C1)=O 33592,C1(c2n(CC=C)nnn2)(NCC23COC(CF)(C2)C3)CCN2CCCCC2C1 33593,C1(CNC(C2(CC)CCN(C(C3CCCSC3)=O)C2)=O)CCC(C)(C)CC1 33594,c1(C(C)C(=O)Nc2cccc(N(C)C(c3ccc[nH]3)=O)c2)ccc(Cl)c(Cl)c1 33595,N1(C(CCC(=C)C)=O)CCN(C(=O)C(F)C2CC2)C(CS(C)(=O)=O)C1 33596,c1(C(=O)NC2C=CCCC2)cnc(C(=O)O)[nH]c1=N 33597,c1(C(=O)NCC2CN(C(=O)C=CCF)C2)cccc2cncn12 33598,C#Cc1cc(C2CCCN2C(=O)NCC2CC[Si](C)(C)C2)cc(F)c1 33599,N(C(=NCCOc1ncccn1)NCc1nc(C2CCC2)no1)C(C#C)C 33600,C1(c2n(C(CC)F)nc(-c3nc[nH]n3)n2)CCC(F)(F)CC1 33601,c1(C(N2C(CNC(C(C3CCCOC3)OC)=O)CCC2)=O)ccc2c(c1)COC2 33602,c1(N2C(C(N(C(C)CC)Cc3ccccc3)=O)CC(=C)C2)nc(C)cc(Cl)n1 33603,C1(N(CC(=O)N(C)C)C)COCCC1NC(=O)Nc1cccnc1-n1nccn1 33604,c1(C(=O)NC2CC(CCC(=O)NC(=O)NCCC3C(OC)CC3)C2)ccc(Cl)o1 33605,C=C1CCN(C(=O)CC(C)OC)C(C(=O)NC2(CF)CCC2)C1 33606,Cc1ccc(C(=O)NCc2cc(C(=O)NCC3CCCC3)no2)c(O)n1 33607,c1(NC(C2(F)CN(C(COCCOCC#C)=O)C2)=O)cccc(OC)c1 33608,c1(C(N2CCC(Oc3ccncc3)C2)C(=O)NC)cnc(Br)n1C 33609,C(=O)(C1=NNC(=O)CC1)NC1C(NC(c2ccc(CC(C)(C)C)cc2)=O)C1 33610,c1(CC(=O)NCC(Cn2cc(CCO)nn2)OC)cc(Cl)cc2c1OCC2 33611,CC1(C)OCCOC1C(=O)NCC1(O)CN(C(c2cccnc2)=O)C1 33612,C1(c2n(C(CC)(C)C)nnn2)(NCC2=CCCC2)CCC2(CCC2)CC1 33613,N1(C(c2c(CC)cc[nH]2)=O)CC(NC(=O)CC(C)(C)C)CCC1C 33614,C1(CNC(c2cnc(-c3ccccc3)o2)=O)CN(C(=O)C(F)F)C2COCC2O1 33615,C1(C)(OC)CCCN(C(=O)C(C)(CNC(c2nc[nH]n2)=O)CC)C1 33616,CN1CCOCC1C(=O)NCCOCCCN(C)C(c1cc(C2CC2)no1)=O 33617,CCC(CC(C)C)C(=O)NCCN(c1ncc([N+](=O)[O-])cn1)CCCN(C)C 33618,N1(C(C(C(CC)C)OC)=O)CC2CCC(C1)N2C(=O)CN1CCN(C)CC1 33619,C1(C(=O)NC2CC(C)N(C(=O)Cn3ncccc3=O)CC2)CS(=O)(=O)CC(=O)N1 33620,C(=O)(C(CC(C)C)NC(c1c[nH]c(C#N)c1)=O)NC(C(CC)CC)C 33621,C1(C(=O)NCC2C(C)CN2C(=O)C2=COCC2)CCC(C2CCC2)CC1 33622,C1(CC(=O)NCC(CNC(=O)CCc2nccs2)O)CCCCC12CC2 33623,N1(C(C(C)c2ccsc2)=O)CC(CNC(=O)CC(C)(F)F)C2(CC2)C1 33624,c1(C2C(C(=O)NC3C=CC(CNC(C(COC)OC)=O)C3)C2)cccc(O)c1 33625,c1(C(=O)NC2CCCC(NC(CNC(=O)NC)=O)C2)cc(C)cc(F)c1 33626,c1(CNC(C2(CC(C)C)CC2)=O)ccc(CN(C)C(C2C(F)(F)C23CC3)=O)cc1 33627,c1(C(=O)NC2CC(CNC(CCC=C(C)C)=O)C2)cc(C#N)c(Br)s1 33628,CC1CCN(C(C2(CS(C)(=O)=O)COC2)=O)C1CNC(=O)CC1CCC(C)(C)O1 33629,N1(C(C23CC2CNC3=O)=O)CCC(Nc2cc(-c3ccc(C)cc3)no2)C(C)C1 33630,C1(COC)(CNC(=O)Cc2c[nH]nc2C)CCCN1C(C1CNC(=O)N1)=O 33631,c1(C(N2CC(C3N(C(CC(C=C)C)=O)CCC3)OCC2)=O)c[nH]c2ccncc12 33632,c1(SCC)ccc(CC(=O)NC2CC(NC(=O)Cc3cccnc3)CC2O)cc1 33633,Cc1ccc(CCC(N2CC(C)(NC(c3cc(Cl)c(Cl)[nH]3)=O)C2)=O)cc1Cl 33634,C1CCC(C)N(C(=O)C(N2CCOC2=O)C)CC(C)C(=O)N1.Cc1nccs1 33635,Cc1nnc2n1C(C(=O)N1CCN(C(=O)Cc3csc(C4CC4)n3)C(C)C1)CC2 33636,N#Cc1cnn(CC(=O)NCC2CCN2C(c2ccc(Cl)cc2)=O)c1 33637,FCCN=C(NCC1CCCO1)N1CCCCC(N=c2ccnc(Cl)[nH]2)C1 33638,C1(CNC(C2N(C)C(=O)NC2)=O)C(O)C(O)CN1C(c1ccc(F)cc1)=O 33639,c1(CC(C)C(N2CCN(C(c3ccccc3CO)=O)CC2C)=O)cc(Cl)cc(Cl)c1 33640,O=C(C1=CCCC1)NC1COCC1NC(C12CC(CN1C1CC1)C2)=O 33641,C1(C(N2CCC(NC(C3CC=CC3)=O)(CO)C2)=O)CN2CCN1CC2 33642,C=CCCC(C(=O)Nc1cnc(F)nc1)NC(c1cc(C)n(CC)n1)=O 33643,N1(C(c2ncc(OCC)nc2)=O)CCCC(NC(=O)CCc2csc(C)n2)CC1 33644,Cc1cccc(C(N2C(CNC(=O)C3=NOC(C)(C)C3)CCC23CCC3)=O)c1F 33645,c1(CN2CCC(N(C(C=CC(C)C)=O)C)CC2)ccc([N+](=O)[O-])cc1O 33646,C(CCCC(=O)NC1(C)CCN(C(=O)C(C)(CC2CCC2)SC)C1)OCC 33647,c1(C(=O)NCC(C)NC(CC(=C)Br)=O)ncccc1S(=O)(=O)CC 33648,N1(C(CC2C(=O)NC(=O)N2)=O)CCC2(CC1)CC2C(=O)Nc1c[nH]nc1C(F)F 33649,c1(C(N2CC(C)(C)N(Cc3ccccc3)CC2)=O)nc2c(F)cc(Cl)cc2s1 33650,N1(C(c2c(CC)con2)=O)CCC(NC(=O)CCCN(C)C)C1c1ccccc1 33651,Cc1ccc(C#N)cc1NC(=O)C(C)OCC(=O)NC(C)Cc1ncc[nH]1 33652,C(CC(C)C(=O)NCC1CC1NC(c1ccnnc1C)=O)=CCC 33653,Cc1cc(Cl)c(Cl)cc1C(=O)NCC1CCCCN1C(C1CC12CCCC2)=O 33654,N1(C(c2cc(CC)no2)=O)CCCOC(CNC(=O)C(C)=CC(C)(C)C)C1 33655,c1(OCC)cc(Cl)ccc1C(=O)NCC1(CO)CCCN1C(=O)C(C)OCOC 33656,C1(C(=O)NCCOCCC=C)CNC(=O)CN1C(=O)CCCC(=O)NCC 33657,C(CC(CC)C(=O)N(C)CCNC(=O)C=CSCc1ccco1)=CC 33658,C1(CC(N2CC(NC(C3CCC(CC)CC3)=O)C(C)C2)=O)CC2CCC(C1)N2C 33659,N1(C(C2(CCC)CC2)=O)CC2(CCN(Cc3nnc(C)o3)C2)C1 33660,C12(CNC(c3c(C)nccc3)=O)CC(NC(=O)CC3(C4CC4)CC3)(C1)C(C)(C)O2 33661,c1(OC)ccc(C(F)(F)C(N2CC3CC3(CNC(=O)C(C)C3CCC3)C2)=O)cc1 33662,C1(CC)CN(C(=O)C=CC(N)=O)CCC1N=c1cc(Cl)nc[nH]1 33663,C#CC1CCCCN1C(=O)C(c1cn(C)nn1)NC(C1CCS1(=O)=O)=O 33664,CCC(CC(=O)NCc1csc(CNC(=O)C(C)(C)CC)n1)CC(F)(F)F 33665,C1(C(N(CC(CC)(C)OC)C)=O)(C(C)C)CCN(C(c2coc(C3CC3)n2)=O)C1 33666,C1(CC(=O)NC2(CNC(CN(C)CCO)=O)CC(C)(C)C2)CC2CCC1CC2 33667,c1(C(=O)NC(C)CCN(C(=O)C2=NNC(=O)C2)C)ccc2nc(Br)nn2c1 33668,S(=O)(=O)(c1cc(C(=O)N(C)CC2CCCN(C(=O)C3=COCCC3)C2)co1)NC 33669,N1(C(C(C)OCCCC)=O)CC2CC2(C(=O)NC2CC3CCC2O3)C1 33670,C1(NC(c2c(C)cc(F)cc2)=O)CC2CC(NC(=O)C(C)(C)C3CCC3)CC2C1 33671,c12[nH]c3ccccc3c1CC1(CC)COCC(CCCNC2=O)CNC1=O 33672,N1(C(CCCOCC)C(=O)NC(CC)C(=O)OC)CCC(S(N)(=O)=O)C1 33673,c1(OC)cc([N+](=O)[O-])cc(CN2CCC3C(C(N)=O)C3C2)c1O 33674,C1(C)(C(=O)OC)CC(NC(=O)C(C)C2CCN2C(=O)Cc2ccn(C)c2)C1 33675,CCC(O)(CC)CCN=C(NCCc1ccc(C(N)=O)o1)NC(C)CCC1CC1 33676,N1(C(CCNC(C)=O)=O)CCOCC(NC(=O)CC2(C)CCCO2)C1 33677,c1(C(=O)NCC2CN(C(C3(C(=O)NC)CC3)=O)C2)cc(Cl)c(OC)cc1Cl 33678,C1(C(=O)NCC(N(C(C(C)C2(O)CCC2)=O)C)C2CC2)CCC2(CC1)CC(O)C2 33679,c1(C(=O)NCC(C)NC(c2sccc2C2CC2)=O)ccc(OC(F)F)nc1Cl 33680,Cc1c(I)c(OCCOC(c2cccc(F)c2)=O)nn1CC1CCOC1 33681,O=C(CCS(=O)(=O)N1CCOCC1)N1C2CC2C2CC12 33682,Cc1cc(C(=O)NCCCN(C(=O)CC(=O)NC2CC2)CC2CC2)ccc1O 33683,C(C)(C(CO)NC(c1cscn1)=O)NC(C1(C(C)C)CC1)=O 33684,c1(-c2nc(CC)sc2)cc(CN2CCC=C(C(=O)N(C)N(C)C)C2)ccc1OC 33685,c1(OC)c(C)ccc(C)c1C(N1CC(NC(c2ccncc2N)=O)C1)=O 33686,c1(C(N2CCN(C(C(CC)C)=O)C3C2CC3)=O)cnc2c(c1)CCC(=O)N2 33687,CC1CCC(CNC(c2ccc(N)cn2)=O)N(C(c2csc(C(F)F)n2)=O)C1 33688,N12CC3CCCC1(C3)COC(OCC)CC2=O.C1(C(=O)OCC)C(O)C1(C)C 33689,CC1CCC(c2cn(CCCC(=O)N3CCCC3)nn2)CC1.C[Si](C)(C)C 33690,C(=O)(C(F)CC(C)(C)NC(=O)CC1CCC(C)O1)N(C1CCCC1O)CC 33691,Cc1ccc(C=NOCC(N2CCN(C)CC2c2nn[nH]n2)=O)cc1 33692,Cc1c(N)ccc(C(=O)N(C2CN(C(c3csc(-c4cn[nH]c4)n3)=O)C2)C)c1C 33693,N1(c2ncc(OCC)cn2)CC2CC1CN2C(c1ccc(CCO)cc1)=O 33694,N1(C(C(CCC)CC)=O)CC2(CNC(=O)C(F)OC(F)(F)F)CC1CCO2 33695,CC1CC(CCNC(c2cc(C(N)=O)c[nH]2)=O)CCN1C(=O)C1=CCCC1 33696,c1(C(N2C(CNC(=O)Cc3ccccc3F)CC2)=O)cnc2cnc(Cl)cc2c1 33697,C(c1ccc(OC)c(O)c1)=CC(=O)NCCC1CCN(C(C(CC#C)(C)C)=O)C1 33698,CCCC(C(=O)NCC1(C(=O)NCC2(CO)CCCC2)CC=CC1)C(C)C 33699,CCCC(C(=O)OC)C(=O)N(CCC(=O)NCc1[nH]ccc(=O)c1O)C(C)C 33700,C1(NC(C=CCC)=O)CC(O)CN(C(c2cnn(-c3nccs3)c2)=O)C1 33701,C1(CC(=O)NC(c2ccccc2)C(=O)N(C)CC2(C)CC2)CCCOC1 33702,N=c1nc(N2CCC(C3CC3)C2)[nH]c(=NCc2ccc3c(c2)CCCC3)[nH]1 33703,Cc1cc(C)c(C(=O)NC2CCN(C(c3ccco3)=O)C2)c(=O)o1 33704,Cc1n[nH]c(=NCC2CN(C(=O)C(C)C(C)C)CC2Cc2ccccc2)s1 33705,C(CC(F)F)(C(=O)NCCN1CCC(O)C1)NC(c1cc(CCC)on1)=O 33706,C1(NC(C2CC(OC)C2)=O)CC2CCC1N2C(c1sc(NC(C)(C)C)cc1C)=O 33707,C1(C(N2C(C(=O)NC3(C(N)=O)CCCCC3)CC=CC2)=O)CC2CCC1CC2 33708,C1(CCNC(CCN(C(=O)CC2CSCCO2)CC)=O)CC2CCC1O2 33709,CCC(F)(F)CC(=O)N1CC2(CNC(c3nnn(C(C)(C)C)n3)=O)CCC1C2 33710,CCC(CC(=O)N1CCC1COC(=O)CCc1ccccc1O)SC 33711,c1(CC)ncc(Cl)c(C(=O)NC2(CN3CCN(C(=O)CC(C)O)CC3)CC2)n1 33712,C1(O)(CCNC(c2c(CC)occ2)=O)CCN(C(=O)CC2CCC(C)(C)O2)C1 33713,CC1(C)OCCOC1CC(=O)NC(C)(C)CNC(c1ccccc1O)=O 33714,C1(C(N(CCN(C)C)Cc2c(F)cccc2Cl)=O)C2(CCC2)C12CCC2 33715,c1(C(=O)NC(c2cccnc2)CC)cc2n(n1)CCN(C(=O)COC(C)=O)C2 33716,N1(C(CC2(OC)CN(C(c3c(C)ncn3OC)=O)C2)=O)CC2CCCCC2C1C 33717,O=C(C1=NOC2(CCC2)C1)NC12CC(NC(=O)CCc3cncc(F)c3)(C1)C2 33718,c1(C(=O)NCC2(NC(=O)C=CC3CCC3)CC2)ccc2nc(S)oc2c1 33719,N1(c2nnc(CCC)s2)CCCC(C)(CNC(=O)CSc2ccccc2)C1 33720,N1(C(c2ccc(CCCCC)o2)=O)CC2C(C(=O)NC(c3ncc[nH]3)CC)C2C1 33721,C1(NC(c2cccc(C(C)=O)c2)=O)CC(O)CN(C(=O)Cn2nccc2C)C1 33722,C1(CC)CN(C(c2ccc(OC)c(OC)c2)C(=O)NC(C)C)C(C)CO1.C(C#N)S 33723,Cc1nccc(C(N2CC(CCNC(C3CNC(=O)N3C)=O)C2)=O)n1 33724,N12C(CCC13CC3)C(=O)N(CCCC(=O)OC)CC2=O.C(COC)OC 33725,C(=O)(CCCC(=O)N1CCOCC(CNC(=O)C(C)CC(F)F)C1)OCC 33726,C1(O)(C(=O)NCC2C3CN(C(C=C4CCC(C)CC4)=O)CC32)CCCC(C)(C)C1 33727,CC(C)C(C)C(CNC(=O)CCc1cscn1)NC(c1cnc[nH]c1=N)=O 33728,CC1OC(C)(C)OC1(C)C(=O)Nc1cc(N2CCN(C(=O)OC(C)(C)C)CC2)on1 33729,C(CC(N)=O)(C(=O)NCC1CC1(F)F)NC(CN(C(C(C)C)=O)C)=O 33730,Cc1cc(Cl)ccc1CC(N1CCC(NC(=O)CCNC(=O)C2CC2)C(F)C1)=O 33731,C#CCC(C)(C(=O)NCC1COCC1(C)C)NC(C12CC(F)(C1)C2)=O 33732,c1(C(=O)NCC(CNC(CSCC#C)=O)OC)cnc2sc(C)cn2c1=O 33733,c1(NC(C23CC(C2)C3)=O)ccc(CC2(C(C3CC3CC(F)F)=O)CCCC2)cc1 33734,N1(C(c2cnn3c2CC(C)CC3)=O)CCC2(CC1)CN(C(=O)CC(C)(C)O)C2 33735,c1(NCCN(CC)CC)[nH]c(=NC(C)c2ncccc2F)nc2sccc12 33736,N1(C(=O)CCCn2ccnc2)CCOC(C(F)F)C1.c1(C)ocnc1C(=O)O 33737,c1(OCC)ccc(C(=O)NCC2(CNC(C3(C)CC3(C)C)=O)CCCC2)cn1 33738,c1(C(=O)NC(CC=C)CNC(C2CC3(CCC3O)C2)=O)ccc(F)c(C)c1O 33739,CC(C)CC(C)CC(=O)NC(CNC(=O)Cn1cc(CN(C)C)nn1)CC(F)(F)F 33740,c1(C(N(CCCNC(C2CC(CCC)OCC2)=O)C2CC2)=O)cc(=N)[nH]c(Cl)n1 33741,C=CCC(CC(=O)NCCC1CC(OC)C1)NC(=O)C(N1CCNC1=O)C 33742,C(=O)(C#CC1CC1)NCC1COC(CNC(C(c2ccc(Cl)s2)C)=O)C1 33743,N1(C(=O)NC2CCOC2c2ccccc2)Cc2ccccc2C(CO)C1 33744,N1(C(c2cc(C)no2)=O)CCN(C)CC1CNC(c1nocc1C1CC1)=O 33745,Cc1nc(NC(C2CC(NC(C3C4CC(=O)CC34)=O)C2)=O)sc1C 33746,C1(C(=O)NCc2snnc2C2CC2)CC(F)(F)CN1C(c1ccccc1O)=O 33747,Cc1c(NCc2cscc2Cl)ncnc1N1CCSCC(C)C1 33748,C1(C)(NC(C)=O)CN(c2ncccn2)C1 33749,N#CCC(C(=O)NCC1CN(C(=O)CC23COC(C2)C3)CCO1)c1ccccc1 33750,C1(CNC(COCCCC#C)=O)CCC(CN(C(=O)CC(C)(F)F)C)CC1 33751,C1(NC(=O)OC(C)(C)C)CC2(C1)CC(Nc1cncc(-c3cnn(C)c3)c1)C2 33752,CCC(CC(=O)N1CCN(C(=O)CCC(C)(C)OC)C(COC)C1)C(F)F 33753,C1(C(C)C)COCCN1C(=O)N(c1cc(-n2cccn2)ccn1)C.C(C1CC1)C1CC1 33754,N1(C(C(=Cc2cnc[nH]2)C)=O)CC2(CCC2)CC1C(=O)NC1CN(CC(F)F)C1 33755,C1(OC)CC(CNC(=O)C(F)C(C)C)N(C(C2CC(F)C(=O)N2)=O)C1 33756,C1(N(C(CC2(OC)CCC2)=O)C)CCCCN(C(c2ncccc2O)=O)C1 33757,CC(C)C(C)(C)CNC(=O)C(c1ccccc1)NC(c1ncc(F)cn1)=O 33758,Cc1cc(C(N2CC3CC(NC(c4cocn4)=O)CC3C2)=O)ccc1C#N 33759,c1(OC)cccc2c1CC(C(N1CC(C)N(C(=O)CCCF)CC1C)=O)CO2 33760,C#CCC(O)C(=O)NCCN(CC(C)O)C(C1CC(=C2CCC2)C1)=O 33761,C1(NC(C(C(=O)OC)OC)=O)CC2CN(C(c3ccc(CO)nc3)=O)CC2C1 33762,CC(CC(=O)NCCN(C)C(c1cnc2sccc2c1)=O)P(C)(C)=O 33763,N1(C(CC)=O)CCC(C2CCN(C(c3cc(F)c(N)c(F)c3)=O)C2)CC1 33764,C(=O)(C(C)S(N)(=O)=O)N1CCC(C)(NC(C=Cc2ccc(C)s2)=O)C1 33765,c1(-n2cnc(CC)n2)ccccc1S(=O)(=O)N1CCC(=C2CCC2)C1 33766,C(C(C)CC(=O)N1CC2C(CNC(c3ccncc3COC)=O)C2C1)OC 33767,C1(CS(=O)(=O)NCC2CCN2S(C)(=O)=O)CC2C(C1)C2(F)F 33768,C(=O)(C1CCc2scnc21)N1CC(NC(=O)COc2cccc(Cl)c2)C2(C1)CC2 33769,N1(C(CSSC)=O)CCc2nc(CNC(C3CCC4C(C3)C4(F)F)=O)sc2C1 33770,C1(NC(c2n(C)ncc2)=O)CC2CC1CN2C(c1ccncc1F)=O 33771,c1(C(=O)NCCNC(c2ccc(N)c3c2cncc3)=O)ccc(F)cc1[N+](=O)[O-] 33772,c1(N2CCC(N(C(C)=O)C)CC2)cc(C)c(S(=O)(=O)NCC2CCCCO2)cn1 33773,N1(C(CCOC)=O)CC(NC(c2nn(CCOC)cc2Br)=O)CC12CCCC2 33774,N1(C(c2cc(OCC)n[nH]2)=O)CCC2(CCCN(C(=O)CC3(CO)CC3)C2)C1 33775,C1(NC(Cc2cc(C)c(F)cc2)=O)CCN(C(=O)Cc2ccnn2C)CC(O)C1 33776,C1(O)(CNC(c2ccc(F)c(CO)c2)=O)CCCN(C(c2cnn[nH]2)=O)C1 33777,c1(C2(C(N3C(C4(O)CN(C(=O)CC5CCCO5)C4)CCC3)=O)CC2)ccnc(Cl)c1 33778,C(=O)(C(C)(C)O)N1CC1CC.C=C(C)COCC(=O)NCCOC 33779,c1(NC(C=CC)=O)c(C)cccc1F.c12ccc(cc1)CCC=CCn1cc-2nn1 33780,CC(C)CC(CC(C)C)C(=O)N(C)CC1CN(C(C2OCC2(C)C)=O)CC12CC2 33781,C1(NC(C=Cc2cc(OC)ns2)=O)CC2CCC(C1)N2C(=O)Cc1c[nH]nc1C 33782,c1(C(N2CCC(COC)(CNC(=O)C(F)C(C)C)C2)=O)cn2c(n1)CCC2 33783,CC(C)CCC(C)N=c1[nH]c(=NC2COC3(CCN(C(C)C)CC3)C2)[nH]c2c1COC2 33784,CP(C)(=O)CC(=O)NCC(O)CNC(c1ccc(C(F)(F)CF)cc1)=O 33785,N1(C(CCc2cnn(C)n2)=O)CCCC(C2CCN(C(C3(C(N)=O)CC3)=O)C2)C1 33786,C1(OCC(=O)NCC(F)F)CCC(F)(F)CC1.C1(=O)C(=O)N(CCC)CCN1 33787,c1(C2CCNC(c3n(C(CC)(C)C)nnn3)(C)C2)ccc(C)cc1C.C1CCC1.OC 33788,C12(CNC(C3CCN(C(CCOCCOCC)=O)C3)=O)CCC(CC1)OC2 33789,c1(CC(C)C)ccc2cc(C(=O)NC3CCN(CCO)C(=O)C3)[nH]c2c1 33790,c1(C(=O)NC2CCCCN(C(C(CC)OC)=O)C2)cc2c([nH]1)CCOC2 33791,N1(C(C)C(=O)NCC2C3CN(C(C4CCC4)=O)CC23)C(=O)NC2(CCCC2)C1=O 33792,c1(CC)ccc(C2C(C(F)(F)F)(CNC(=O)COC(=O)CC)C2)cc1 33793,N1(C(=O)CC2CCC2)CC2(CCN(C(C3(CC4CC4)CCCO3)=O)CC2)C1 33794,C1(C(C)NC(CCSC)=O)CN(C(=O)C2=CCCC2)CCO1 33795,C1(C(=O)NC2C(C(C)C)CN(C(=O)COc3cnn(C)c3)C2)CC1C1(C)COC1 33796,C(C(=O)NC1CC2(C1)CC2C(=O)NCC1(C#N)CC1)(C(C)C)NC(C)=O 33797,CC1CCC=C1C(=O)N1CCN(CCCNC(C2CC2Br)=O)CC1 33798,c1(C(C(=O)NC2C3(CN(C(c4n(C)cnc4)=O)C3)CC2)O)cccc([N+](=O)[O-])c1 33799,Cc1csc(C(=O)NCCC(C)NC(c2c(C(C)C)cnn2C)=O)c1Cl 33800,c1(CNC(C2CCN(C)C2)C)cc(I)ccc1N1CCOCC1 33801,N1(C(C=COCC)=O)CCN2C(=O)C(NC(=O)CCn3cc(Cl)cn3)CC2C1 33802,CC(C)(C)C(C)(O)C(=O)N1CCCN(C(c2coc(C(F)(F)F)n2)=O)C(CO)C1 33803,c12ccnc(n1)NC2.C1(NC(=O)C(C)(O)C2CC2)CCCCC1C(C)(C)C 33804,C1(N(C(c2c(CC)oc(C)c2)=O)C)CCCN(C(=O)COc2cnn(C)c2)CC1 33805,c1(C(c2nnnn2C2(C)CC2)Nc2cnn(CCC)c2C)cc([N+](=O)[O-])ccc1Cl 33806,C1(NC(c2c(C)n(C)nc2)=O)C(C)CN(C(=O)CC(C2CC2)C2CC2)CC1C 33807,C1(CC)CN(C(c2ccc(C3CC3)s2)=O)CCN1C(C1C(C(F)F)C1(C)C)=O 33808,CC1(C)CN(C(N)=O)CCC1CNC(=O)NC(N)COCc1ccccc1 33809,C1(CNC(c2c(C)scn2)=O)CC(NC(=O)Cc2sccc2Cl)C1(C)C 33810,c1(OC)cc(C(=O)NCC2CNCCN2S(=O)(=O)CCCCl)c(Br)cc1Br 33811,C(c1cccc(F)c1)=CC(N1CCC(CCOC)(NC(=O)C(C)C2CC2)C1)=O 33812,CCC(C(C)C)C(C(=O)NC1CCC1)N1CCn2c(C(F)(F)F)nnc2C1 33813,C1(C(=O)NCCCC2(NC(C(=O)NC(C)C)=O)CC2)CC(=O)N(C(C)C)C1 33814,C1(CC)CN(C(=O)C(F)OC(F)(F)F)CC1C(=O)N(C)Cc1ccc(F)cc1 33815,Cc1ccc2c(C(=O)N(C)CCN(C)C(C3SC4C=CC3CC4)=O)c[nH]c2c1 33816,N1(C(CN(C)C)=O)CCN(CCNC(C2(CC3CC3F)CC2)=O)CC1 33817,C1(NC(C2(C#C)CC2)=O)CC(CNC(c2coc(N(C)C)n2)=O)C12CCC2 33818,N1(C(Cc2cccc(C)c2)=O)CCN(C(=O)CCc2ccccc2F)CC(CO)C1 33819,C1(NC(C2CC(OC)C2)=O)CCN(C(=O)CNC(c2ccc(C)nc2)=O)CC1F 33820,N1(C(C=Cc2cn(C)nc2)=O)Cc2ccccc2C1CNC(c1cnnn1C)=O 33821,c1(SC)nc(N2CCN(C(c3ccccc3-n3nccn3)=O)CC2)c(Br)c(C)n1 33822,c1(OC)cccc(-n2cc(CNC(=O)CN3CC(C)(C)C3)nn2)c1C 33823,c1(OC)ccc(C(=O)NC2CC(NC(c3[nH]nnc3C)=O)C23CCC3)c(F)c1 33824,c1(C(=O)NC2CCN(C(c3occc3F)=O)C2C2CC2)cc2cc(Cl)cnc2o1 33825,C1(C(=O)NC(COC)C)CC(O)CN1C(=O)CN1CCOCC1 33826,n1(CC)cc(Cl)cc1C(=O)NC(C)CCNC(=O)CCc1cncn1C 33827,N1(C(C2(COC)CCC2)=O)CC2CCCC2(C(=O)NCC(F)F)C1 33828,C1(C(=O)NC2CN(C(C3(SC)CC3)=O)CC2CC2CC2)CC(C)(C)OC1(C)C 33829,N1(C(CCSC)=O)CCC2C(NC(=O)C(c3ccnn3C)C)CC12 33830,C1(CN(C)C(c2cnn(CCO)c2)=O)CCCN(C(c2[nH]nnc2C(F)F)=O)C1 33831,N1(C(CC(C)C(F)F)=O)CC2(CCN(C(=O)C=Cc3ccn(C)c3)C2)C1 33832,C1(CC=C)(NC(C2CCCC(C)C2)=O)CCN(C(=O)CCNC(=O)CO)C1 33833,C#CCCCC(C)C(=O)NC1CC(C)(NC(c2cc(F)c(CC)cc2F)=O)C1 33834,N1(C(CN(C)Cc2ccccc2)=O)CCCCC1CCNC(c1cnccn1)=O 33835,C1(CC)COC2(CCC2)CN1CCC(C(=O)NC)c1ccccc1 33836,N1(C(=O)CCN2CCC2)CCC(CCNC(C2(c3ccccc3)CC2(F)F)=O)C1 33837,N1(C(c2ncc(F)cc2F)=O)CC2CCN(C(C3CC4CCC3O4)=O)C2C1 33838,C12(CNC(c3ccc(Cl)cn3)=O)CC1CN(C(c1cccc(F)c1)=O)C2 33839,N1(C(C2(SCC)CC2)=O)CC(NC(c2cnc(CC3CC3)s2)=O)C2(CC2)C1 33840,N1(C(C2=NOC(C)C2)=O)CC2(CCCC2)CN1C(=O)CC1(CSC)CC1 33841,c1(C(=O)NC2CC(NC(CCCC)=O)C23CCC3)cc2cnc(Cl)cc2s1 33842,c1(N2CCC(CC(C)(C)C)C2)ccc(S(=O)(=O)NCc2cccc(CO)c2)cn1 33843,c1(NC(C2N(C(CN3CC(NS(N)(=O)=O)C3)=O)CC2)=O)cc2cccnn2c1 33844,c1(C(=O)NC2CCC(CNC(c3cc(C)oc3)=O)C2)ccc([N+](=O)[O-])n1C 33845,C12(NC(C(C)OCC=C)=O)CCCC1(F)CN(C(c1[nH]nc([N+](=O)[O-])c1Cl)=O)C2 33846,N1(C(c2c(CC)nn[nH]2)=O)CCC(C)C(NC(=O)COCCOC)C1C 33847,c1(OC)cccc(C(N2CCC(N(C(=O)C=Cc3ccsc3)CCO)C2)=O)c1F 33848,C1(C(N2CCC(O)(C(C)NC(CC(C)(C)C)=O)CC2)=O)CC2CCC(C1)C2F 33849,CC1CN(C(=O)CCCOCCN(C)C)CCCN1C(=O)CNc1ccccc1 33850,C1(N(C)C)(C(=O)NCC(CNC(=O)C(F)=C2CCCC2)CO)CCCOC1 33851,C#CC1(C(N(CCCC(=O)OC)C(=O)CC2CC3(CC3)CO2)OC)CCCCC1 33852,N1(C(C2(C)CCCCNC2=O)=O)CCOC2(CCN(C(=O)C=CC(N)=O)C2)C1 33853,C=CC(C)(O)CC(=O)N(CC(C)O)CCNC(c1sc(C)cc1C)=O 33854,c1(OCCC)ccc(Cl)cc1C(N1CC2C(NC(=O)C3=C(Cl)CC3)C2C1)=O 33855,c1(NC(C2CCN(c3ccc([N+](=O)[O-])cc3)C2=O)=O)ccnc2cc(F)cnc12 33856,c1(OC)ccc(C(C)NC(C(C)(C)OC)c2nnnn2CC(F)F)cc1C#N 33857,O=C1CCCC(NC(C23CCC(CC2)N3)=O)C1 33858,C1(NC(=O)NCc2cccc(-n3cc(CC(=O)O)nn3)c2)CC2(C1)CC(F)(F)C2 33859,c1(C(=O)NCC(CC)NC(=O)CN(C)CC2CC2)ccc(C2CCCCC2)cc1 33860,C1(COC(C2(C)COC2)=O)Cc2ccc(Br)cc2N1C(=O)OC(C)(C)C 33861,C(=O)(C(C(=O)Nc1cccc(NC(=O)C(CSCC)OC)c1)C(C)C)OCC 33862,N1(C(C2CCCCN(C(c3nc(CC)oc3)=O)C2)=O)CCC2(CCCCO2)C1 33863,C#Cc1ccc(C(=O)NCCCN(C(c2ccc(Cl)c(C)c2)=O)C(C)C)nc1 33864,c1(C(=O)NC2C(NC(CCOC)=O)CC2)c(Cl)c([N+](=O)[O-])nn1C 33865,N1(C(C2CC23CCOC3)C(=O)NC(C)C)CCc2ccc(F)c(F)c2C1 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33883,N1(C(C2C(=C)C2)=O)CC(C(N)=O)(CNC(c2cc(Cc3ccccc3)c[nH]2)=O)C1 33884,c1(C(=O)Nc2c(C)c(=O)[nH]c(=O)[nH]2)ccc2c(c1)CN(CCN(C)C)C2 33885,Cc1c(CC(N2CCCC2C2(C(=O)NCC3CCOCC3)CC2)=O)cnn1C 33886,c1(N2CCC(C(N3C(CC=C)CCCN3)=O)CC2)cnc(Br)cc1O 33887,C1(NC(C2CCC3(CC2)CC3)=O)CCCN(C(c2cc(F)c[nH]2)=O)CC1F 33888,N1(C(CC=C)=O)CCCC2(C1)CN(C(C1OCCOC1(C)C)=O)CCO2 33889,C(N=c1ccc(-c2ccccc2)c[nH]1)c1c(C)cc(Cl)cc1 33890,C1(NC(COC(C)C)=O)CCOC(NC(=O)CN(CC(C)(C)C)C)C1 33891,c1(CC2(C(=O)NCCN(C(CCN(CCC)C)=O)C3CC3)CC2)nn(C)cc1Br 33892,Cc1nsc(C(=O)NCC2CCCN(C(=O)C(F)(F)C3CCOCC3)C2)c1N 33893,CCC(C)CCC(=O)N1CCC(CNC(=O)C=C(C2CC2)C2CC2)(OC)C1 33894,CCC(CC(=O)Nc1ncccc1C(C)=O)OC.C1CCCC2CN(C2)C1=O 33895,C1(C(C)NC(C2(OC)CC2)=O)CCCN(C(c2ccc(=N)[nH]c2)=O)C1 33896,N1(C(CS(CC)=O)=O)CC(CNC(=O)C(F)(F)c2nccs2)CC(C)C1 33897,C1(C(=O)NC2CCC(C(N(CC)Cc3ccccc3)=O)CC2)CC(C2CC2)=NO1 33898,C=CC(C)(CC)NC(c1c[nH]nc1NC(C)=O)=O 33899,N1(C(C2(N(C(=O)CC3CCC=CCC3)C)CC2)=O)CCCC(C2CCC2)C1 33900,N1(C(C2CC(=C)C2)=O)CC2CCC(N(C)C(c3cc(F)ccc3OC)=O)C2C1 33901,C1(N(C(=O)C(=O)NC2CC2)C)CCC2CCN(C(c3ccccc3C(F)F)=O)C1C2 33902,c1(C(=O)NC(CCC)CNC(=O)CCC(F)(F)F)cnc2c(c1)nc(C)n2C 33903,C1(CCNCc2cc(C(=O)OCC)c(OC)cc2)CNC(=O)C(C)(C)C1 33904,C(=O)(CS(=O)(=O)C(C)C)N1C(CNC(C=CC=CCC)=O)(COC)CCC1 33905,c1(NCC(C(C)C)(C)NC(C2COCCO2)=O)ncnc2scc(C)c12 33906,C1(NC(=O)CNC(C2CCCC2O)=O)CCC=CCC1 33907,Nc1nc(Cl)ccc1C(N1CC2CC2(CNC(=O)CCC2CC2(Cl)Cl)C1)=O 33908,N1(CCC(=O)Nc2ccc(Cl)cc2)CCC2COCCC12 33909,CCC(C)(C)C(C(=O)N1CC(OC)C(CNC(=O)Cc2ccc(F)cc2)C1)OC 33910,C#CC1(NC(C2CC(NC(c3cnc(O)c(F)c3)=O)C23CCC3)=O)CCCCC1 33911,N1(C(c2cncc(OCC)c2)=O)C2CCC(C2)C1CC(=O)NC(CO)C(C)(C)C 33912,C1(O)(C(C)C)CCN(C(c2ccc(Cl)cc2)c2ccsc2Br)C1.C(=O)N(C)CCO 33913,C1(C#N)(C(=O)NC(C)C(CO)NC(c2cccnc2C(F)(F)F)=O)CC1(C)C 33914,Cc1csc(Cl)c1C(=O)NCCCN1CCN(C(=O)CN2C(C)CCC2C)CC1 33915,c1(NCCC(=O)NCCCOc2cc(C)cc(C)c2)ccc2c(c1F)OCCO2 33916,Cc1c(C(=O)NCCC(C)(C)NC(C2CC2(C)C(F)F)=O)cnc2ncnn12 33917,n1(CC(=O)NCC(CNC(CC(CC)OC)=O)C)cccc([N+](=O)[O-])c1=O 33918,c1(OC)ccccc1OCC(=O)NCCCN(C)CC1CC(C)CO1 33919,O=C(C(c1cccs1)=Cc1cccs1)NCC1CCC(CO)O1 33920,C1(NC(C(CN(C)C)N(C)C)=O)CCN(C(=O)CC=C(Cl)Cl)CCC1CO 33921,C(=O)(C1=CCCCO1)NCCCC(C)NC(C1C=CC=CC=C1)=O 33922,c1(Cc2n(-c3cnc(C)s3)nc(COC3CCCN3C)n2)ccc2ccccc2n1 33923,N1(C(C(C)SCC)=O)CCC2CCCC12C(=O)N(C)CC1CC(F)C1 33924,C(=O)(C(C)(CNC(c1nn(C)cc1Cl)=O)CC)NCCOCC 33925,N1(C(C2ON=C(C)C2)=O)CCC2C(C1)CN2C(=O)CCCN1C(=O)CCC1=O 33926,c1(C(=O)NC2C(C)CCN(C(=O)CC3CC=CC3)C2)cc2occc2n1C 33927,CC1C(NC(C2CCCCS2(=O)=O)=O)CCCN1C(C1CCCC1)=O 33928,C1(CC)CCC(C(=O)N(C)CC2CCCN2C(c2cnsc2)=O)CC1 33929,c1(C(=O)NCC2CCCN2C(C2CC(CCO)C2)=O)cc2c(F)c(Cl)ccc2[nH]1 33930,c1(C(=O)NCC(COC)NC(c2cnnn2C2CC2)=O)cnc(Cl)n1C 33931,C(=O)(C1=CCCCC1C)N1CCCC(C(N(CC(C)C)CC(C)C)=O)CC1 33932,N1(C(c2cnn3ccn(C)c32)=O)CC2(CCN(C(=O)CSC(F)F)CC2)C1 33933,C(=O)(CCC(C)CN(C)C)NCC(CO)NC(CSCC=C)=O 33934,C1(C(=O)NC(CCC)C)CCC2(CC1)CN(C(=O)C(C1CC1)OC)C2 33935,C1(C(=O)NCc2cc(C(N3CC(OCC(=O)NC)C3)=O)n[nH]2)CCCCN1C 33936,C1(F)(CNC(C(CC)NC(N)=O)=O)CCN(C(c2cnccc2OC)=O)C1 33937,N1(C(CC2C(NC(C3(C)C(C)(C)C3)=O)CCC2)=O)CC(CO)C2(CCC2)C1 33938,c1(C(=O)NCC(C)NC(=O)C(c2ccccc2F)C)cccc(N)c1Br 33939,C1(NC(N2CCCC(n3ccc(C)n3)C2)=O)CCC(F)(F)C(C)(C)O1 33940,c1(C(=O)NCC(CCOC)NC(C2CC3CC3C2)=O)oc(COC)nc1C 33941,CC1CCCCN1CCNC(=O)C(CC1CC1)NC(c1ccc(CC#N)cc1)=O 33942,C(=O)(C(CC(C)C)N(C)C)N1C(C(N2CCCC(CCC#C)C2)=O)(CC=C)CCC1 33943,N1(C(c2ccc(CCC)cc2)=O)CCCC(C)(NC(=O)C(C)OCOC)C1 33944,C(=O)(C1=C(NC(=O)Nc2cc(Br)c(SC)cc2C)CCCC1)OC 33945,N1(C(C2N(C(CC3CCC(C)O3)=O)CC3CC32)=O)CC(CO)C1(C)C 33946,c1(C(=O)NC(C)CN(C)C(c2cnc3sccn23)=O)c(F)ccc2n[nH]cc12 33947,N1(C(C(CC)N(C)C)=O)CC(NC(c2cc3c([nH]2)CCC3)=O)C(C)(C)C1 33948,c1(C(N2C(CN(C(C(C)OCC(C)C)=O)C)CCC2)=O)noc2cc(Cl)ccc12 33949,N1(C(C2N(C)CCN(C(CN(CC)CC)=O)C2)=O)CCCC(C)(C)CC1 33950,C1(CC(C)(C)C#N)C(=O)N1.N1(CCS(C)=O)CCC(SC(F)(F)F)CC1 33951,Cc1ccncc1C=CC(=O)NCC(C)(C1CCC1)NC(C1CCNC1=O)=O 33952,c1(-c2cc(C3CCCCC3)no2)nc(C2CC2)nn1CC1CCCCC1 33953,C1(CNC(c2c(C)cccc2C2CC2)=O)CCN(C(=O)CSC2CC2)C12CCC2 33954,C(=O)(C=CS(C)=O)N(CC(CC)NC(c1ccn(CCN(C)C)n1)=O)C 33955,C1(C(N2CCCC(Cn3cc(CN)nn3)C2)=O)CCc2nc(O)[nH]c2C1 33956,c1(NC(C)=O)ccc(NC(c2nnnn2CC2CC2)C2CC=CC2)cc1 33957,CC(C)C(C)C(C(=O)NCCCNC(C1(C(F)(F)F)CC1)=O)NC(N)=O 33958,CCCC(O)C(=O)NCCCC1CCN(C(=O)CC2OCCO2)CC1 33959,N1(C(C(CC)CCOC)=O)CC(C(N2CCCN(C)CC2C)=O)C2(CCC2)C1 33960,C1(NC(C(COCC)(C)C)=O)COC2CN(C(=O)C(F)C(C)(F)F)CC12 33961,C(=O)(C1CC(=O)c2ccccc21)N1C(C)(CNC(C2(CC(C)(C)C)CC2)=O)CCC1 33962,Cc1cc(C(=O)N(C2CN(C(C3(C)CCCCCC3)=O)CC2(C)C)C)nc(C)c1 33963,C=CC(C)(CC)C(=O)NCCCN(C(=O)COc1ccc(F)cc1)CCOC 33964,Cc1cncc(C(N2CCC(C)(CNC(=O)CCc3cccnc3Br)C2)=O)c1 33965,c1(C(=O)NCC(C)(Cn2cccn2)NC(=O)C(F)=CC2CC2)cc(Cl)ccc1O 33966,C1(C(=O)NC(C)Cn2cccn2)CN(C(=O)CN2CSCC2=O)CC(C)(C)C1 33967,Cc1oc(Cl)nc1C(=O)NC1(CCCC(=O)NC2CC(CC(C)(C)C)C2)CC1 33968,CC1CC(NC(=O)C(C)(F)C(C)(C)F)CN(C(=O)CCS(C)(=O)=O)C1 33969,N1(C(=O)CCc2ccccc2)CCC2CCN(C(C3CCCCC3O)=O)CC2C1 33970,N1(C(CC=CC)=O)CC(NC(c2cccc(C(N)=O)c2C)=O)C2CC2C1 33971,C1(NC(CCC=CC)=O)C(C)(C)CN(C(c2cnc(S(C)(=O)=O)s2)=O)CC1(C)C 33972,C1(NC(CN(C2CCCC2)C)=O)CC(F)CN(C(c2c[nH]nc2C(C)(C)C)=O)C1 33973,C1(NC(CC(C)(C)NC(C)=O)=O)CN(C(C2(c3ccccc3)CC2)=O)CC12CC2 33974,C(=O)(CCC(=O)Nc1nccs1)NC1CC(CNC(c2cn(CCC=C)nn2)=O)C1 33975,CC(C)CC(C)(O)C(=O)N1CC2CC(C1)N2C(c1cnn(C(C)C)n1)=O 33976,C(=O)(C(C)(C)Cc1cnc[nH]1)N1CC(CNC(c2cc(COC)[nH]n2)=O)(OC)C1 33977,c1(COC)ccn(C)c(=O)c1.c12cc(n(C)c1)C(=O)NC1(CO)CCN(C1)C2=O 33978,CC1=CC(O)CN(C(c2nc(CNC(=O)Cc3ccn(C)n3)oc2C)=O)C1 33979,C1(SC)CC(F)(F)CN1c1ccnc(C2CC2)n1.c12nccnc1NC2=O 33980,C(=O)(C(CO)C(C)(C)C)NC1COCCN(C(CC2OCC(C)(C)C2)=O)C1 33981,c1(CC)ncc(C(=O)NC(CO)C(C)NC(c2ccncc2C)=O)c(O)n1 33982,Cc1cc(Br)ccc1C1(CN2CCN(C(c3ncc(Cl)nc3Br)=O)CC2)CC1 33983,C1(NC(C2C(C(N)=O)CC2)=O)CCCC1NC(c1cnc(-c2ccco2)s1)=O 33984,C(=O)(C(F)C(=O)N=c1[nH]nc(-c2ncccc2C(=O)OCC)s1)NCC 33985,c1(CC)cc(C2CCCN(C(C3(c4ncco4)COC3)=O)C2)cnc1F 33986,C1(C(=O)NCCN(C(=O)C(C)N2CCC2)CC)CCC(NC(N)=O)CC1 33987,c1(CC)noc(C(=O)N(C2CCN(C(C3CC(OC)C3)=O)CC2)C)c1C 33988,c1(C(=O)NCC(C)CNC(=O)Cc2cccc(F)c2O)cnc2c(c1)nnn2C 33989,c1(C(=O)NCCN(C(c2cccc(OC)c2)=O)CC)cn(C(C)(C)C)nc1C 33990,CCC(O)C(C)(C)C(=O)N1CCN(C(=O)C(C)(Cl)Cl)CC(O)C1 33991,C(CNC(C1CCC=CC1NC(C1CCSCC1)=O)=O)(C(C)(C)C)OC 33992,c1(C(C)C)cc(C(c2nnnn2CC(F)F)N(CCC(N)=O)CC#N)cc(Br)c1 33993,Cc1ccsc1C=CC(=O)NCC(CO)NC(c1cn(C2CC2)cn1)=O 33994,C1(Nc2ccc(Nc3ccc(OC)cc3OC)cn2)CC2(CC(=O)CC(=O)C2)C1 33995,N1(C(C(CC=C)NC(C)=O)=O)CCCCC12CN(C(c1cc(C)nn1C)=O)C2 33996,O=C(C1Cc2ccccc21)N1CCC(N2CCN(C(C3(CO)COC3)=O)CC2)C1 33997,N#CC1(CNC(=O)CSCCNC(=O)CC2CC2C2CC2)CCSCC1 33998,N1(C(C)=O)CCC(NC(c2c(CNC(=O)COC3(C)CCCC3)c[nH]n2)=O)CC1 33999,N1(C(C(CC2CCC2)OC)=O)CC(O)CC1CNC(C1CC=CCC1C)=O 34000,c1(C(N2CCC(Cn3cncn3)CC2)C(=O)NCC(C)C)nn(C(C)C)nc1Br 34001,Cc1cc(Br)cc(C(=O)NC2(CCO)CN(C(C3C=CCCC3)=O)C2)c1C 34002,N1(S(CCOCCC#C)(=O)=O)CCCCC(C)C1 34003,C1(C)(C(N(CCN(C(c2c(C)occ2C(F)(F)F)=O)C)C)=O)OC(C)(C)OC1C 34004,C(=O)(C1Cc2ccccc21)NC(C)(C)CCC(=O)NCCc1cccnc1 34005,C1(C(=O)OC)CC12CN(C(=O)C(Cc1ccco1)NC(c1c[nH]c(=S)cn1)=O)C2 34006,C1(C(=O)NC2CC3(CN(c4ncc(C)cn4)C3)C2)CCc2cnnn2C1 34007,N1(C(=O)CNc2ccc(O)cc2)CCCC2(C1)CN(C(=O)Cc1cnco1)C2 34008,N1(C(c2cnc(C3CC3)s2)=O)CCN(C(c2cnn3c2OCC3)=O)C(CCO)C1 34009,c1(SC)ncc(C(=O)NC2CC3CN(C(c4ocnc4C4CC4)=O)CC23)c(O)n1 34010,CC1(C)CCCC(C(N2CC3(CC(CC(=O)Nc4cncnc4O)C3)C2)=O)C1 34011,C(C(=O)NCC1CC(NC(=O)CNc2cccc(F)c2)CCO1)(C(C)C)SC 34012,c1(C(=O)NCC(CC=C)NC(c2cnc[nH]2)=O)n[nH]c(C)c1C(F)(F)F 34013,C1(OC)(CNC(c2cncnc2C)=O)CCN(C(=O)C=C(C)C(C)(C)C)C1 34014,C(C1=NOC2COCC12)n1cc(C2CCCC(C#N)C2)nn1.N12CCCCC1C2 34015,C1(CNC(C(C)(C)OC(C)C)=O)CN(C(=O)Cc2coc(C(F)F)n2)CC1C 34016,N12CCCC(C)(C1)N(C)CC2=O.c1(C(=O)NC2CCCCO2)csc(Cl)c1Cl 34017,CC1CC(NC(=O)CC(C)(C)F)CN(C(=O)CC2CCC(=O)CC2)C1 34018,c1(C(=O)NCC2CCN(C(C(CCOC)OC)=O)C2)cnn2c1CCC2 34019,c1(NCC2CC3CC3N2C(N(C)C)=O)cccc(C2CCCOC2)c1 34020,N1(C(CC=C=C)=O)CC2CC1C2NC(c1ccccc1)=O 34021,N1(C(c2n(CCOC)ncc2)=O)CCCC1(C)C(C)(C)CNC(=O)C(F)C1CCC1 34022,c1(C(=O)NC2C(NC(C3(CN(C)C)CCCC3)=O)CCC2)nnn(C)c1N 34023,C1(OC)(CO)CCCN(C(C(=O)NCCCF)c2nccs2)C1 34024,c1(C(=O)NCC(C)N(C(=O)Cn2ncc(C#N)c2N)C)nnc2n1CCCCC2 34025,C1(CNC(c2c(C)nsc2)=O)C2CN(C(C3C4CC5C(C4)C35)=O)CC12 34026,CCC(CCOC)C(=O)N1CCC(CN(C)C(C2COC(=O)N2C)=O)C1 34027,C(=O)(C(C)(C)CC(F)(F)F)NCCCC(CCC)Nc1ncc(O)cn1 34028,N1(C(C(c2cccc(Cl)c2)C)=O)CCN(C(c2ccc(Cl)cc2N)=O)CC1C 34029,c1(C(=O)NCC2N(C(CC(C)OC)=O)CC(C(F)(F)F)C2)cnc(C)cc1Cl 34030,C1(CC(=O)OC)COCCN1Cc1cc(-c2ccncc2)no1 34031,c1(C(=O)NCC2(O)CCN(C(C(C)N(C(C)=O)C)=O)C2)cccc(=S)n1O 34032,CC1(C)CN(CC(N2CCC(CNC(C3CCC(c4ccccc4)O3)=O)C2)=O)C1 34033,c1(C(N2CC(NC(C3N(C)C(=O)CC3)=O)C(O)C2)=O)cc2nccnc2cc1F 34034,C=Cc1cncc(C(=O)NC(C2CCOC2)CNC(c2c(C)cnnc2O)=O)c1 34035,N1(C(COC)=O)CCC2CN(C(C3CCN(c4ccc(F)c(F)c4)C3)=O)CC12 34036,c1(CSCC(=O)N(C2CCN(C(c3cscc3C#N)=O)CC2)C)ccc(Cl)cc1 34037,c1(C(C)C)nc(-n2cccc2)sc1C(=O)NC1CCCN(C(=O)C(O)C(F)F)C1 34038,c1(OC)c(F)ccc(F)c1C(N1CC(NC(C2CC2C2CCCO2)=O)C1)=O 34039,C1(C(=O)OCC2(C)CC(F)(F)CNC2)CCc2n[nH]cc2C1 34040,c1(CC(=O)NC2CC(Nc3cc(O)ncn3)C23CCC3)coc2ccccc12 34041,C(=O)(C(F)(CNC(C1(C#N)CCCOC1)=O)C(C)C)NC(C(=O)N(CC)CC)C 34042,N1(C(c2c(C)onc2Cl)=O)CC(NC(c2cccc3nc[nH]c23)=O)C2(CCC2)C1 34043,C(C(CC(C)C)C(=O)Nc1cnc(C)c(C#N)c1)NC(C1(OC)CC1)=O 34044,N1(C(=O)NCC2(COC)CCCO2)CCC2(CC1)CNC(=O)C2O 34045,c1(C(N2CC(OCC)OCC2)C(=O)NCC2CCCO2)ccc2nc[nH]c2c1 34046,C1(CC)CCCC1NC(=O)CC=CCNC(=O)C1=CCC1 34047,CN1CCCC(C(N2CCOC(CNC(C3(C)COC(=O)N3)=O)C2)=O)C1 34048,C(CC(C)(C)C(=O)NC1(C(O)CO)CC1)NC(COC(CC)CC)=O 34049,CC(C)CCC(F)C(=O)N(CCC(C)NC(c1cccc2sccc12)=O)C 34050,Cc1cnc2ccccc2c1C(=O)OCC=CCN=S(C)(C)=O 34051,CC1OC(=O)NC1C(=O)NC1CCCC(NC(c2cc(Br)sn2)=O)C1 34052,c1(C(=O)NC2(CNC(=O)C(=C3CCCCC3)F)CCOC2)cnn2ncccc12 34053,N1(C(C2CC(C#N)C2)=O)CCC2CCN(C(c3cc4sc(Cl)cc4[nH]3)=O)CC12 34054,Cc1noc(C)c1C(C)C(=O)NCCC(C)NC(=O)C(C)C1CCCO1 34055,c1(NC(CSCC(N2CCOCC2)=O)=O)cnncc1Cl 34056,N1(C(CC2(C)N(C(C=CC(C)C)=O)CC2)=O)CC23CCC2(COC3)C1 34057,c1(C(=O)NCCC(C)NC(C(c2cncnc2)C)=O)cnc2cnn(C)c2c1 34058,CC(N=c1cc[nH]cc1S(=O)(=O)N1CCCC(COC(F)F)C1)c1ccc(Br)o1 34059,Cc1ccc2nc(C(=O)NC3COCCN(C(C4CCOC(=O)N4)=O)C3)cn2c1 34060,C(=O)(CC(CNC(C1CC1(C)C)=O)C1CCC1)N(C1(COC)CCC1)C 34061,C1(NC(c2n(C(C)C)nnn2)(C2CCCOC2)C)CCC2(CC1)CSC2 34062,N1(C(c2c(C)noc2)=O)CCC2C1CCCN2C(c1sccc1Cl)=O 34063,C(CC(O)C(=O)NC1(CC=C)CN(C(=O)CCc2cc(C)on2)C1)OC 34064,c1(C(N(CC(C)CNC(c2cc(CC3CCC3)c[nH]2)=O)C)=O)nc(Cl)sc1Cl 34065,C=CC(CC)C(=O)NCC1(C(=O)NCC2C=CCCC2)CC12CCC2 34066,C(CC(C(=O)NC(CCO)c1ccco1)NC(C1CN(C(C)=O)C1)=O)SC 34067,S(=O)(=O)(c1ccc2cccc(Cl)c2c1)C(=O)OCC1(C)CCCC(F)(F)C1 34068,c1(CC(=O)NC(C)(CNC(=O)CC2CC(F)C2)C2CC2)cccc(C(F)F)c1 34069,c1(NCCN(C(C(CC)(C)C)=O)C)cccc(C#N)c1 34070,N1(C(C(C)O)=O)CCC(C2CC(NC(=O)CCc3ccn(C)n3)C2)CC1 34071,C1(C(C)(C)C)CC(C(=O)N2CCCN(C(C34CC(CN3C3CC3)C4)=O)CC2)=NO1 34072,c1(CN2CCC(C(=O)Nc3cc(Cl)ccc3F)C2)nc2ccccc2o1 34073,C(=O)(C(C)(C)S(C)(=O)=O)NCC1(OC)CCN(C(c2c(OC)cccc2)=O)C1 34074,C(=O)(C1=CCCC1(C)C)NCCC1N(C(c2ccc(NC(C)=O)s2)=O)CCOC1 34075,C1(NC(C2(CC)CCOC2)=O)CCCCCC1NC(=O)C(F)(F)c1csc(C)c1 34076,C1(C)(COC)CCN(C(C2(NC(=O)Cc3nonc3C)CC(C)(C)C2)=O)C1 34077,N1(C(COCCCC#C)=O)CCC(F)(F)C(CNC(c2sccc2COC)=O)C1 34078,C(N=c1ccn(C2CCC2)[nH]1)(c1ccc(OCC)cc1)C(C)C 34079,C(=O)(C(C#N)C(C)C)N1CCCC(NC(Cc2c(C)cnn2C)=O)C1 34080,C1(CC)CN(C(C2(CO)CCCC2)=O)CCN1C(c1csc(-c2cccs2)n1)=O 34081,c1(C(C(=O)NCC(CC=C)NC(C2CC(=C3CC3)C2)=O)=O)cc(F)ccc1C 34082,N1(C(C(C=CC)O)=O)CC=C(C(C)(C)C(=O)NCC2CC(C3CC3)=NO2)C1 34083,C=CCC(CN(C(=O)C(C)OC)CCNC(=O)CC1(NC=O)CCC1)OC.C1CC1 34084,C1(OC)(CNC(c2cnoc2C)=O)CCN(C(=O)C2=COCCC2)CC1 34085,N1(C(c2c(CC)cncc2)=O)C2CCC1C(CNC(=O)C=CCn1cncn1)C2 34086,N1(C(C2CN(C(c3c(CC)con3)=O)CC2C)=O)CCC12CCSCC2 34087,c1(CC(=O)N(CC(C)C)CCN(c2ccccc2)C)ccccc1-c1nn[nH]n1 34088,C1(C(=O)NC2CN(C)NC2=O)CN(C)CCN1C(c1ncc(F)cn1)=O 34089,Cc1ncnc(O)c1CCC(=O)NCC1CC2CCC1N2C(=O)COCC(F)F 34090,c1(C(=O)NCC2CCN(C(c3n(C)ccc3)=O)C2)n[nH]c2ccc([N+](=O)[O-])cc12 34091,N1(C(CC2N(C(CN(C(C(C)C)=O)C)=O)CC(O)C2)=O)CC2(C)CC1CCO2 34092,N1(C(C2SCCN(Cc3c(OC)ccc(Br)c3)C2)=O)CCC2(CC1)CN(C)C2 34093,NS(=O)(=O)CCCNC(c1nnnn1C1CC(F)(F)C1)c1nnnn1C1CCOC1 34094,C1(CNC(C2CC(C(C)(C)C)C2)=O)CC2(CC2)CN1C(=O)CNC(=O)C(F)(F)F 34095,Cc1nccc(C(N2CCC(NC(c3cc(Cl)cnc3O)=O)C(C)C2)=O)c1C 34096,C1(C(=O)NCC(CC)(C)NC(c2cn(C)c(C(F)F)n2)=O)CCC(C)(C)C1 34097,C1(NC(Cn2nc(C)n(C)c2=O)=O)CC12CCN(C(=O)CC1OCCC1C)CC2 34098,N1(C(c2c(O)ncc(CC)c2)=O)CCN(C(C2CCCC(=O)C2)=O)CC(O)C1 34099,Cc1coc(C(=O)NCCCOCCCNC(c2c(C)noc2C(C)C)=O)c1C 34100,CCC(C(=O)NCC(C)CN(C(=O)C1=NOC(C)C1)C)C(C)C 34101,c1(CC(=O)NC(C2(O)CCN(C(c3c(C)nn(C)c3)=O)C2)C)c(Cl)cccc1Cl 34102,CCCN=C(NCc1ccc(C(=O)OCC)cc1)NC(C1CCCS1(=O)=O)C 34103,C1(NC(C(N(C(=O)CSC(F)F)C)C2CC2)=O)C2CCC3C(C2)CC13 34104,C1(NC(c2c(C)nccn2)=O)CN(C(c2cnc(S)nc2)=O)CC12CCC2 34105,C(=O)(C1=C(C)OCCS1(=O)=O)NC1CN(C(C(CC)CC(F)F)=O)CC1C 34106,c1(C(=O)NC2CN(C(C(C)N(C)C)=O)CC2C)cc(F)c2nc(O)ccc2c1 34107,C1(CC)CCC(C(N2CCCC(CNC(c3nnn(C(C)(C)C)n3)=O)C2)=O)CC1 34108,C1(NC(C2CCCC2)=O)CN(C(=O)C(c2ccc(F)cc2)F)CC12CCC2 34109,C(C(C)C(=O)NC(C(=O)N(CCCC1CC1)C)C1CC1(C)C)OC 34110,C12CC13CCN(CC3)C(=O)C(=O)NC2.C=CC(CC)CC(=O)NCC(F)F 34111,Cc1cc(Br)ccc1-c1nnc(NCC2(O)CCCN(S(C)(=O)=O)C2)o1 34112,c1(CCNC(C2(CC)CCOCC2)=O)ncc(Br)cc1CCn1cccn1 34113,C1(C(=O)NC(CNC(c2c(C)cc(C)s2)=O)(C)C)CC12CCCOC2 34114,CC1(C)COC(C(=O)NC(CC2CCOCC2)C(=O)NCCC2COCCO2)C1 34115,C=CCC(C)(C)C(=O)NC(C)C(C(C)C)OCC(F)(F)F 34116,C1(NCC=C(CC)CC)CCCC1C(=O)N(C)C 34117,Cc1nc2cc(C(N3CCCC(F)(F)CC3)=O)ccc2n1C(C)CO 34118,C1(SCC)CCCN(C(C2(NC(C(=O)NCC)=O)CC2)=O)CC1 34119,N1(C(CCC(=O)OCC)=O)CCC2(CCCN2C(=O)Cn2cc(C)cn2)C1 34120,CCCC(C(=O)NCCCOCCNC(C1CCc2nnnn2C1)=O)S(N)(=O)=O 34121,N1(C(C(F)=CCC)=O)CCCC(NC(=O)COCC2CCCO2)C1C 34122,N1(C(c2nc(F)ccc2Cl)=O)CC(C2(N=c3[nH]nc(-c4ccccc4)o3)CC2)C1 34123,C1(C(=O)NCC(C)CN(C)C(c2ncsc2C2CC2)=O)COC2(CCC2)C1 34124,C(=O)(C(CNC(=O)Cn1cccc1)CC(C)C)NC1CC(OC)C1(C)C 34125,N1(C(c2c(C)noc2C)=O)CCCC(F)(C(=O)NCc2cncnc2)C1 34126,N1(C(c2c[nH]c3nccc-3c2)=O)CC2OCCN(C(=O)Cc3cc[nH]n3)C2C1 34127,C1(NC(CCCC2CN(C(c3c(C)sc(O)n3)=O)C2)=O)(CO)CC2CCC1C2 34128,CC(C1OCCc2ccccc21)N(C(=O)CCc1cncc(F)c1)C 34129,N1(C(C2C(NC(C3CCC(C)O3)=O)CC=CC2)=O)CC(=O)NC(C)(C)C1 34130,c1(C(=O)NCC(CC)N(C)C(c2nn[nH]c2Cl)=O)ccnn1C(F)F 34131,N1(C(C(C(C)(C)C)SC)=O)CCCC(C2CN(C(=O)CN3CCOCC3)C2)C1 34132,N1(C(c2c(CC)nn(C)c2)=O)CC2CC1CN(C(c1nocc1Cl)=O)C2 34133,Nc1cc(Cl)cc(Cl)c1C(=O)NC(CNC(c1cncnc1)=O)C1CCC1 34134,C(CC(C)C(=O)N1CCC(CCNC(=O)Cc2cccc(SC)c2)C1)=CCC 34135,CC1CN(C(C2CCCN2C=O)=O)CC1NC(C1(N(C)C)CCC1)=O 34136,CC1OCCC1(C)C(N1CCC(C(=O)NCC(C2CC(C)(C)C2)O)CC1)=O 34137,C1(NC(=O)NC(c2csc(-c3ncccc3F)n2)C)CCN(CC(F)(F)F)C1=O 34138,C1(CN(C)C(c2cc(C(N)=O)cn2C)=O)CC(F)CN1C(C1(S(N)(=O)=O)CC1)=O 34139,c1(CC(C)C)ccc(C(=O)N(C(C)CCNC(=O)CSc2nc[nH]n2)CC)s1 34140,c1(C(=O)NC(C(C(C)C)NC(c2cccc(OC)c2)=O)C)cc2sccc2s1 34141,c1(NCc2c(Br)ccc(OC)n2)[nH]c(=NCc2c(C)coc2C)nc2sccc12 34142,c1(C(N(C(c2ccccc2)CNC(c2onc(C)n2)=O)C)=O)ccc(O)nn1 34143,c1(C(=O)NC2C(NC(C(CC)CC3CCCC3)=O)CCC2)ncc2ccccn12 34144,C1N=C2C=CN=C(N2)Nc2cnccc21.N1(C(C)=O)CCN(C(C)C)CC1 34145,c1(CN(C(C2CCCN(C(c3coc(C)n3)=O)C2)=O)CC)ccc(O)cc1 34146,N1(CCS(C)(=O)=O)CCCN(C(=O)Nc2ccc(CO)c(C(F)(F)F)c2)CC1 34147,c1(OC)cc(NC(c2ccn(C)c2)c2nnnn2C2CCCC2)sn1 34148,N1(C(CC(C)(C)O)=O)CC2(CC(C(=O)Nc3ccc(F)c(F)c3)CO2)C1 34149,c1(CC(=O)NC(C)CCCCNC(c2cc(C(N)=O)[nH]n2)=O)cccc(F)c1O 34150,C(=O)(CC(C)CC(F)(F)F)NCc1cc2cc(Cl)ccn2n1.CC1CN2CC1C2=O 34151,C1(CCC(=O)N(C2CCOC2)C)CCCN(C(c2cccc(F)c2)=O)C1 34152,N1(C(c2c(C)cccn2)=O)CC(C)CN(C(c2ccc(F)c(N)c2F)=O)C(C)C1 34153,N1(C(c2cc(COC)sc2)=O)CCCC(C)(NC(=O)CN2CCOC2=O)C1 34154,c1(C(N2CC(N(C(C(C)OCC=C)=O)C)C3(C2)CC3)=O)ccc(S(N)(=O)=O)cc1 34155,C(=O)(C(C)(C)CC(=O)OCC)N1CC(NC(COCCC=C)=O)C(O)C1 34156,C1(C(=O)OC)CN(C(=O)C(=O)NCc2ccc(Cl)c(F)c2F)CCC12OCCO2 34157,C1(CC(=O)OCC)CN(C(=O)C=CC2CCCN2)CCC1C 34158,C(C(CC(=O)NCC1(CF)CC1)NC(=O)C(C)(C)CSC)OC 34159,C(=O)(CCCCN(C(=O)C=Cc1nccs1)C)NC(CC)(C)C#N 34160,N1(C(C2N(C(C)C)CCC2)=O)CCCC(C)(C(=O)NC(C)(C)C(O)CO)C1 34161,c1(CC(=O)N(C2CCCN(C(=O)Cc3cccnc3)CC2)CC)c(F)cncc1Cl 34162,C1(C(=O)NCC(C)NC(CCCN(C(=O)OCC)C)=O)CCc2nc(C)cn2C1 34163,C(=O)(C(C(CC)CC)NC(=O)C(c1cnn(C(C)C)c1C)=O)N(CCC)CCC 34164,c1(C(=O)NC2C(NC(C=CCOC)=O)C2)cccc2oc(C)cc12 34165,c1(C(=O)NC2(CNC(c3c(C)ocn3)=O)CCC2)cnc2c(c1)CCOC2 34166,C1(NC(CCNC(c2c(C)ccnc2C)=O)=O)CC(C2CCCC2)C1 34167,C1(C(=O)NCC#CCNC(C(CC)C2CCOCC2)=O)(OC)CCC(C)(C)C1 34168,C1(CCOC)(NC(=O)CCCc2nc(C)cs2)CCN(C(=O)C=Cc2c[nH]cn2)C1 34169,c1(C(=O)NC(C(C)(C)OC)C)ccc(CNC(=O)Cn2cc(C#N)cn2)nc1 34170,c1(C(=O)NC(CSCC)CO)cnc(CNC(c2ccnn2C(C)C)=O)nc1 34171,N1(C(C(C)=C(C)OC)=O)CC2OCCN(C(C3CCC(F)(F)C3O)=O)C2C1 34172,C(c1cccc(C)c1)=CC(N1CC(C(C(=O)N(C2(CC)CC2)C)O)C1)=O 34173,N1(C(c2cc(COC)no2)=O)CCN(C(C2CCC(=O)O2)=O)CC2(CC2)C1 34174,C1(NC(c2cc(CC)c(Cl)cc2)=O)CCN(c2nccc(C)n2)CC(C)(C)C1 34175,N1(C(C2C(OC)CCCC2)=O)CC(C(=O)NC2(C(C)O)CC2)C(F)(F)C1 34176,c1(C(N(CCNC(C2(F)CCC(C)CC2)=O)CC)=O)nn(C)c(C)c1[N+](=O)[O-].C1CC1 34177,N1(C(c2nc(CC)oc2)=O)CCC(CC)C1CNC(C1CCS1(=O)=O)=O 34178,N1(C(c2cc(OCC)no2)=O)CCCOC(CNC(C2CCOC2C(C)C)=O)C1 34179,N1(C(C(C=C)C2CCOCC2)=O)CCN(C(c2cnc(CC3CC3)s2)=O)CC1CO 34180,n1(CC(=O)NCCC2CC(NC(C3(C)C(C)OCC3)=O)C2)nc2c(n1)CCCC2 34181,c1(NC(C(C)SC2CCCO2)=O)cccc(C(F)(F)F)c1F 34182,CCCCC(C)(F)C(=O)NCC(C)N(C(=O)CN1CCOCC1)C 34183,N1(C(C2(C)COC2)=O)CCC2C(NC(=O)CCSCC(N)=O)C2CC1 34184,N1(C(COCCC=C)=O)CC2CCC(CNC(=O)C(CCC)OC)CC12 34185,C1(NC(c2ccc(SC(C)C)cc2)=O)CC2CC1CN2C(=O)CN(C)CCO 34186,c1(NC(=O)OC)ccc(C(=O)N(CC(O)CNC(=O)CC2(CO)CC2)C)c(F)c1 34187,N1(C(CC2C(CC)C2(F)F)=O)CC2(CCCC2NC(c2sccc2CC#N)=O)C1 34188,c1(C(=O)NCCN(CC(CC)NC(=O)C2CC2)CC)cc(CC)cc(F)c1 34189,C(=O)(C1CCCn2ccnc21)Nc1c(-c2ccc(OC)cc2OC)cccn1 34190,c1(CC(=O)NCC(CC)NC(=O)COc2cn[nH]c2)csc(C(C)(C)C)n1 34191,CCCCC(CC)(c1nnnn1CC1CCOCC1)NCc1n[nH]c(C)n1 34192,c1(NC2(c3n(CCOCC)nnn3)CCOC(CC)C2)ccn2ccnc2n1 34193,c1(C(=O)NC2(CCOC)CCN(C(c3cnn(C)c3)=O)C2)cc(C)cnc1F 34194,c1(C(N2C(C(C)C)C(NC(c3ccc(CO)cn3)=O)CC2)=O)ccc(=N)[nH]c1Cl 34195,N1(C(=O)Nc2ccccc2)CCN(Cc2cnc(-c3ccccn3)nc2)C2CC12 34196,C1(CNC(CC2CC(SC)C2)=O)CCCCC1NC(c1nnccc1C)=O 34197,N1(C(C2(CC=C)CCCCC2)=O)CC2CC(CNC(C3C=CCCC3)=O)C2C1 34198,c1(C(c2n(CCCC)nnn2)NC(c2ncccc2C)C)nn(C)nc1Br 34199,C1(CNC(c2n(CC)nc(C)c2)=O)CCCCN(C(C23CCCC2C3)=O)C1 34200,c1(CC(=O)NC2C(NC(C(c3ccccc3)NC(C)=O)=O)COC2)ccncc1C 34201,C1(C(N2CCN(C(CNC(C3CCC(C#C)C3)=O)=O)CC2)=O)CCCCN1N=O 34202,CC(C)CCCCCCC(=O)N1CCC2CCCC12CNC(=O)C(C)(C)C(N)=O 34203,c1(NC(C2CCCO2)COC)ccc(S(=O)(=O)NCc2ccnn2C)c(Cl)c1 34204,C=CC(F)(F)C(=O)NC(C1CCN(C(c2ccc(C(F)F)cn2)=O)CC1)CO 34205,Cc1cc(Cl)cc(C)c1OCC(=O)NC(C)CCCNC(c1noc(N(C)C)n1)=O 34206,CCC(C)CCC(=O)NCC(CC)(CC)NC(C12CC(C)(C1)OC2C)=O 34207,C(=O)(NNC(=O)C(O)C1CCCC1)NC1C(C(Cc2c(C)cccc2C)O)C1 34208,C(=O)(C(CCNC(C1CN(C(C)C)C1)=O)OC)N1CC(=CC)C1 34209,CCCCC(C)(c1nnnn1C1CCC(CCC2CC2)C1)Nc1nccn1C1CCC1.S 34210,c1(NC(C2(C(=O)NC3CC3C(=O)OC)C(=C)CC2)=O)ccncc1CSC.C(=O)OC 34211,N1(C(CSC)=O)CCN(CCCC2CCCN(C(=O)C(C)CF)C2)CC1 34212,CCC(CNC(=O)C(=O)Nc1cc(Cl)ccc1C(C)=O)CC(F)F 34213,C1(C(=O)NCC(C=C)(C)C)CN(C(=O)CCc2ccnn2C)CC1F 34214,N1(C(Cc2c(C)cccc2C)=O)CC(C)(C)CCC1CNC(=O)C(O)C(C)C 34215,c1(CC)noc(C2CC2C(=O)NC(c2cc(-c3ccccc3)[nH]n2)(C)C)n1 34216,CN1CCOCC(NC(C2CCCN(C(=O)CNc3cnccn3)C2)=O)C1 34217,c1(C(=O)NCC2CC(NC(C3C(C)N(C)CC3)=O)C2)cncc2n[nH]cc12 34218,C1(C(=O)NCCC(C)N(C(C(C)S(N)(=O)=O)=O)C)CCc2nncn2C1 34219,C1(C)(C(=O)NCCOCCC=C)CCN(C(=O)CCc2cc(Cl)no2)C1 34220,C1(OC)C2CCN(C(c3cc(C(F)F)cs3)C(=O)NC3CCCC3)C2C1(C)C 34221,C1(OC(C)=O)CCN(C(C2CC(NC(c3ccns3)=O)C2)=O)C1 34222,C1(NC(c2cc(C)c(Br)o2)=O)(CO)CCCN(C(c2nocc2C2CC2)=O)C1 34223,c1(C(C)NC(C(n2cc(C(C)NC)nn2)C)=O)cccc(C#N)c1 34224,C12(C(=O)OC(C)C(N)=O)CCN(C1)S(=O)(=O)C2 34225,c1(OC)cc(C)c(C(N2CCC(C)(CNC(C3CCC(=O)N3)=O)C2)=O)c(C)c1 34226,C1(F)(C(N(CCCNC(C2(OC)CCC(C)C2)=O)C2CC2)=O)CC2(CCC2)C1 34227,Cc1ccc(C(=O)NCC=CCNC(=O)CC2CC2C2CC2)c(C2CC2)n1 34228,N1(C(C2C(CCOC)C2)=O)CCC(C)(C)C1CC(N1CC(S(C)=O)C1)=O 34229,c1(C(=O)NCCCN(C(=O)CC2(C(F)(F)F)CC2)CC)cc(F)c(F)c(O)c1F 34230,c1(C(=O)NC(C(=O)N(CC#C)CC)C2CCCO2)c[nH]c(=NC)s1 34231,C1(C(C)NC(CC2(N(C(COCCCC)=O)C)CC2)=O)CCOC1 34232,Cc1c(Cl)ccc(C(C)NC(C2(NC(=O)OC(C)(C)C)CCSC2)=O)c1F 34233,C(CC(O)C(=O)NCc1nc(C#N)cs1)SC 34234,N1(C(C(C(C)C)C)=O)CCC(CNC(=O)Cc2c(Br)cnn2C)C(C)C1 34235,c1(C(C)C)c(C(=O)N(CCCOCCNC(=O)CC2CCCCO2)C)cnn1C 34236,C(=O)(C(CC(C)(C)C)OC)N(C(C(N1CCN(C(C#C)C)CC1)=O)C)CC=C 34237,C(=O)(C1=Cc2ccccc2C1O)N1CCC(CN(C(C(C)CC(F)F)=O)C)CC1 34238,c1(CCC)cc(C(=O)NC(C)(C)C(C)NC(c2cccnc2F)=O)nn1C 34239,N1(C(C(C(=C)C)(C)C)=O)CCC(C2CN(C(C3(c4ccnn4C)CC3)=O)C2)CC1 34240,c1(C(=O)NCCCOCCC(=O)NC(C#C)CC2CC2)cnc(O)c(C)c1 34241,N1(CC(=O)Nc2c(C)cccc2)CCCN(CC(=O)Nc2ccnn2C)CC1 34242,N1(C(c2cc(OC)n(C)n2)=O)CCN(C(C2CCNC2=O)=O)C(C2CCCC2)C1 34243,Cc1ccc(N2CCCC3(NC(C4CCCC(F)(F)C4)=O)CC3C2)c([N+](=O)[O-])c1 34244,c1(C(=O)NCC(CO)NC(c2n(CC)ncc2)=O)c(F)cc(C)cc1F 34245,CC(C)CC(F)(F)C(=O)N1CC(O)(C2CCCN2C(=O)Cc2c[nH]ccc2=O)C1 34246,Cc1cnn(C)c1C(=O)N(C)CC1(CNC(C2COCC(C)O2)=O)CC1 34247,c1(C(N(C2CCN(C(c3cc(C)ns3)=O)C2)CC2CC2)=O)nc(=O)n(C)[nH]1 34248,N1(c2cc(OC)ncn2)CCC(NC(c2ccccc2N(C)C)=O)C1(C)C 34249,c1(C(N(CC(=O)NC(C)C(O)C(C)C)CCC)=O)ncnc(O)c1F 34250,Cc1ccc(O)c(C(=O)NCCC(C)(C)NC(c2cc(Br)cs2)=O)n1 34251,C1(NC(c2nccc(SC)n2)=O)CN(C(=O)CC2COCCO2)CCC1C 34252,C1(CNC(CSCCN(C)C)=O)CCC(OC)C1.C1(C)CCOCC1.C1(=O)CN1 34253,CC(C)CCCCCC(=O)NCC1(C(N)=O)CN(C(C2CC(C)N(C)C2)=O)C1 34254,c1(C(=O)NCCCN(C(=O)CC2(CO)CCOCC2)C2CC2)ccc2cnoc2c1 34255,CC(CN(C)C)CCC(=O)N1CCCC(C(=O)NC2(CO)CC3CCCC23)CC1 34256,C(N=c1nc(SC)[nH]s1)C1(O)CN(C(C(CC)OCC)=O)C1 34257,c1(C(N(CCN(C(c2cc(C)nnc2O)=O)C)C)=O)c(Cl)ccc2c[nH]nc12 34258,c1(C(C)C)cc(C(=O)NCC(O)CNC(=O)C(F)=C2CCCC2)ccc1Br 34259,C1(CC(=O)N(CC)Cc2cnn(C)c2)COCCN1C(=O)C(=O)NOC 34260,c1(C(=O)NCC2CN(C(c3ccc(C)cn3)=O)C2)n[nH]c2ccc(Br)cc12 34261,c1(C(N2CCC(C)(NC(c3cncc(C)c3)=O)C2)=O)cc(C)cnc1F 34262,C12(C(=O)NCCNC(C(CC)(C)O)=O)CCC(C)(C(=O)O1)C2(C)C 34263,C12(CNC(C3(C=C)CC3)=O)CCC1CN(C(c1cc(CC)n(C)n1)=O)C2 34264,c1(C(=O)NC(C2(O)CN(C(=O)Cc3cncs3)C2)C)cc([N+](=O)[O-])n(C)n1 34265,CC1(C)CC(C(=O)NC2CCCC(O)C2O)CCN1C(=O)CC1CCCC2CC12 34266,N1(C(C2C=CCN(C(CCOCC(C)C)=O)C2)=O)CC2CCCC2(CO)C1 34267,CCC(CC(=O)NC12CC1CN(C(c1cocc1C)=O)C2)c1ccccc1 34268,c1(NC(C)CCNC(C2CCOC3(CCC3)C2)=O)cc(=O)n2ccccc2n1 34269,N1(C(CSCCOC)=O)CC(NC(C2CCCN(CCOC)C2)=O)CC1(C)C 34270,Cc1cccc2nc(C(=O)NC(C)CNC(=O)C=Cc3nccs3)cn12 34271,N1(C(c2cnc(C(C)OCC)s2)=O)CCCC(CCNC(=O)C(C)(C)OC)CC1 34272,C1(C2CCN(C)CC2)(C(=O)NC(C(C)NC(C=Cc2cccc(C)c2)=O)C)CC1 34273,C#CCCCCC(=O)NC(C1CCCN1C(=O)C(N)=O)C 34274,Cc1cc(OCC(=O)NC2CC(C)(NC(=O)C(F)C3CC3)C2)ccc1F 34275,c1(OC(CNC(C(=O)NC(c2cccc(C)c2)C)=O)C)cc(C)ccc1C(N)=O 34276,Cc1noc(C)c1COCCC(=O)NC1(C(F)F)CCN(C(=O)CN(C)C)C1 34277,C1(CC(=O)NCCC2CC(NC(CCc3ncc(C)[nH]3)=O)C2)CCC2(CC2)C1 34278,N1(C(CCC#C)=O)CC(C(=O)NC(CO)C2(O)CC2)CCC1C 34279,C(=O)(CS(=O)(=O)CCOC(C)=O)N(CC(=O)OC1CN(C(C2CSCC2C)=O)C1)C 34280,c1(C(N2CCC(CNC(c3ccc(O)nc3Cl)=O)C2)=O)c(Br)ccc(Br)c1F 34281,C(C(C)(C(C)C)NC(=O)C(N)=O)NC(C(c1cccnc1)OC)=O 34282,CC1CC(C)(C)CCC1NCCCN(C1CCC(F)(F)CC1)C1CC1 34283,O=CN(C(CCCSCC(F)(F)F)C)CC(C)SC 34284,c1(OC)cc([N+](=O)[O-])ccc1CN1CC=CC1C(=O)Nc1nc(C#N)cs1 34285,c1(SC)ccc(OCC(N2CCC(N(C(=O)Cc3nc(=N)[nH][nH]3)C)C2)=O)cc1 34286,C12(NCCn3cncc3C(=O)NCCNC(C=CC)=O)CCCCC1C2 34287,c1(C(N2CCC(C)(NC(=O)C(O)C3CCCC3)C2)=O)csc2c(O)ccnc12 34288,N1(C(C(CC)C(C)C)=O)CC2CC(O)C1C2NC(=O)C=Cc1cscn1 34289,c1(CC2(C(C)NC=O)CC2)ccc(F)cc1F.C1(N)CC(C)(C)C1Oc1ccccc1 34290,N1(C(C2(CC)CCCC2)=O)CCC(C#C)(C(=O)NC2CC2C2CCCCC2)CC1 34291,C1(NC(c2nc(C)sc2)=O)COCCN(C(=O)CC2CCC(F)(F)CC2)C1 34292,N1(C(c2cn(CC)nc2C)=O)CCC(F)(CNC(=O)Cc2nnc(O)s2)CC1 34293,N1(C(C2(C)N(C(CN(C(=O)OC)C)=O)CC=C2)=O)CCC2(CC1)CC2 34294,C1(F)(CNC(c2n[nH]c3c2CCC3)=O)CCN(C(C2CC3CC2CC3O)=O)CC1 34295,Cn1nc(C(F)(F)F)c(CN2CCC(F)(C(=O)NCCCCCO)CC2)c1Cl 34296,CC(CN(C)C)C(=O)NCC1CCN1C(c1sccc1Cl)=O 34297,C#Cc1cn(C)nc1C(N1CCCC(CCNC(=O)COCCC)CC1)=O 34298,c1(OCC(=O)NCCN(C(=O)CC2CCC(=O)O2)C2CC2)ccc(Br)cn1 34299,c1(N2CCCC(NCC(=O)OC)C2)cc(Cl)nc(-c2ccccn2)n1 34300,N1(C(C(CC)(C)C#N)=O)CCC(C2CCOCC2)(CNC(c2ncoc2C)=O)C1 34301,c1(C(=O)NC(C2CN(C(=O)C3=COCC3)CCO2)C)cc(Cl)cc(Br)c1 34302,c1(N(c2ncnc(SC)c2F)C(C2CNCC2C#N)=O)ncnc2c(C)csc12 34303,Cn1cc(C(C(=O)NCC(CO)C2CC2)NC(=O)C(O)C2CCCC2)nn1 34304,c1(N2CCN(C(=O)NC(C3CCOC3)C#C)C2)ccc(F)cc1NC 34305,C1(C(N2CC(C(C)NC(=O)CN3CCC3)OCC2)=O)CC2(CCCC2)C1 34306,C1(F)(CNC(c2ccn(C3CCCCC3)n2)=O)CN(C(C2CC2Br)=O)C1 34307,N1(C(CNC(C=C(C)C(F)F)=O)=O)CCN(C(C2COCC2(C)C)=O)CC1 34308,c1(CNC(C2(OC)CNC2)C)ncc(C(F)(F)F)[nH]1 34309,c1(SCC(=O)NCCNC(C2CC2F)=O)nnc(-c2ccc(Cl)cc2)n1C1CC1 34310,c1(C(=O)NC(CC)CCOC)ccc2c(c1)CCN2C(=O)OC(C)(C)C 34311,N1(C(CCOCC#C)=O)CCC(C(=O)NCC(O)COCC)C12CC2 34312,C1(CN2C(C)CCC2C)CC2CC1CN2C(=O)C(=O)Cc1ccccc1 34313,CCCC(C(=O)N1CCC(CNC(=O)CCc2cn(C)nn2)C12CCC2)C(C)C 34314,C1(CNC(C2(Cl)C(C)(C)C2)=O)CC(F)(F)CN1C(=O)COc1ccc(Cl)cc1F 34315,C(=O)(C1=CCN(C(=O)Cn2ncnn2)C1)NCC(COC)(O)CO 34316,CC1CN(C(=O)CC(C)N(C)C)CC1NC(=O)CSCC1CCCO1 34317,N1(C(C(C)OCCC(C)C)=O)CCC2(CCC(NC(=O)C(F)CC3CC3)CC2)C1 34318,C1(NC(c2cc(C)c(F)nc2)=O)CCC(F)(F)C(C)(C)C1 34319,CC1C(NC(=O)C=CC2CCOCC2)CCCN1C(C1CC2(CCC2O)C1)=O 34320,C(=O)(C(C(C)(C)C)NC(=O)CNC(CSCC)=O)C1C(CN)CCCC1.C(C)=O 34321,C(=O)(CC(C)(C)C1CCCCC1)NC1(C(=O)OCCNC(CCOCC)=O)CC1 34322,c1(C(N2CC3C(NC(=O)CC(C4CC4)C4CC4)(CC3)C2)=O)cn2c(n1)CCCC2 34323,C1(NC(CCC=C=C)=O)CCC2CCN(C(c3ccc(F)c(C)c3Cl)=O)C1C2 34324,c1(C(=O)NCCCCNC(C2(C#N)CCC2)=O)cc(Br)ccc1F 34325,c1(OCC)ccc(Cl)c(NC(=O)C(CC(C)C)Nc2nccc(C#N)n2)n1 34326,C(CNC(=O)CN1CCOC1=O)(CCNC(=O)C(C1CCCCC1)N(C)C)OC 34327,CC(O)C(F)(F)C(=O)NC1CCC1NC(c1cc([N+](=O)[O-])n[nH]1)=O 34328,N(C(=NCC1=CCCCC1)NCCC1(C#N)CCC1)CC1N(CC)CCC1 34329,C(=O)(C(C)(C)C(C)O)NC(CC(C)NC(COCc1c(C)ncs1)=O)C 34330,N1(C(C(C)OCCC=C)=O)CC(NC(c2nocc2C(C)(C)C)=O)CC1(C)C 34331,N1(C(C(C)C2CC2)=O)CCN(C(=O)CN(C(c2ccco2)=O)C2CC2)CC1 34332,N1(C(CNC(c2c(CCC)n[nH]c2)=O)=O)CC(N(C)C)C(C)C1 34333,Cc1ncc(C(=O)NC(C)(C)C(=O)NCCC2CCCCO2)cc1C#N 34334,C1(CC(=O)NCC(C2CC2)NC(C2CC3(CC(=C)C3)C2)=O)NC(=O)CN(C)C1=O 34335,c1(C(=O)NCC2(CNC(c3ccc(NC)c(F)c3)=O)CC2)nn(C)cc1[N+](=O)[O-] 34336,C1(CN(C)C(C2CC(C#N)C2)=O)CCCN(C(=O)C(O)CF)C1 34337,N1(CN(N2C(c3ccccc3)CC(C)(C)C2)C)CCC(S(=O)(=O)C(F)F)C1 34338,C(=O)(CCC(C)OC(=O)CCc1c(N)cnn1C)OC(C)C 34339,c1(NC(C2OCCCN(CC#CC)C2)=O)ccc(N=Nc2ccccc2)cc1 34340,C1(C(=O)Nc2ccn3cncc3c2)CN2CC3CC2(CO1)C3 34341,n1(CCC(=O)N(CCn2cc(-c3ccncc3)nn2)CC)cnccc1=O 34342,N1(C(c2cc(OC)cc(C)c2)C(=O)NC(CC)C)CC(C)c2ccccc21 34343,C1(O)(CC(N2CC(NC(C3(C(=O)OCC)CC34CC4)=O)C2)=O)CCCCC1 34344,c1(CNC2(c3n(CCCSC)nnn3)CSC(C)C2)cnc2ncccn12 34345,N1(C(C2CCN(CC)C2)=O)CCCC(N(C(c2cc(F)ccc2F)=O)CC)C1C 34346,[N-]=[N+]=NC1CCC2(C(=O)NC(CNC(=O)Cn3cnnn3)CO)CC12 34347,N1(C(C2ON=C(C)C2)=O)CCCC(C)(CNC(c2c(C)noc2C(F)(F)F)=O)C1 34348,C1(CC(=O)NC(C2CCN(C(C3CC(N(C)C)C3)=O)CC2)(C)C)CCOC(C)(C)C1 34349,c1(C)nnc(O)cc1O.C1(NCC)CC(C(=O)NOc2nnnn2C)C1(COC)CC 34350,C1(C)(C(N(CCC)CCNC(=O)CCC2CC2CC)=O)CCCC1C(=O)OC 34351,c1(OCC(=O)N(C)CC2CCC(NC(=O)CC3CCCC3)C2)cccnc1 34352,C=CC(C)(CCOC)C(=O)NCCN(C(=O)C1=COCCO1)C 34353,c1(C(=O)NC(C)C(CO)NC(C2CC3CCC(C2)O3)=O)cccc2c1ncn2C 34354,C(C(O)CC(=O)NCC1(CC2CC2)CCC1)NC(=O)CCc1ncccn1 34355,C1(N(C(CC(C)CF)=O)C)CCC2(CC1)CCN(C(c1ccc(F)cc1O)=O)C2 34356,c1(NC(C=CC(C)NC(c2c(C)noc2)=O)=O)ccccc1C(C)C 34357,C1(NC(C2CCCO2)=O)CCN(C(C2(C3CCC3)CC2)=O)C12CCC2 34358,CC1(C)NC(=O)CC1C(N1CCC(CCC(=O)NC2CCS(=O)CC2)CC1)=O 34359,CC(C)CC(CNC(=O)CC1CCC(=O)C1)C(=O)NCCN=S(C)(C)=O 34360,CC(C)CC(C(=O)NC(C)C(CO)NC(=O)C(N1CCN(C)CC1)(C)C)C(N)=O 34361,C1(N(C(COCC=C)=O)C)CC2CCC(C1)N2C(C1(C(F)F)CCOCC1)=O 34362,C(=O)(CC(C)(C)C(F)(F)F)NCCOC1CN(C(C(CC)(O)c2ccccc2)=O)C1 34363,c1(CC)ccc(C(N2CCN(C(=O)Cc3cnc(Cl)cc3C)CC2)=O)c(C)n1 34364,C1(CNC(CCCN(C)C)=O)CN(C(=O)CCN2CCNC(=O)C2)CC(C)(C)O1 34365,c1(C(=O)NCCC2C(C)CN(C(C3CCCCO3)=O)C2)cc(Br)c(F)cc1N 34366,CCCN(NC(=O)Cn1cc(C2CCN(C)C2)nn1)C(=O)OCC 34367,C1(CCC#C)CCCN1C(=O)C(C1CCN(C(C2CC(=O)C2)=O)C1)C 34368,N1(C(C2CCC(C(C)(C)C)CC2)=O)CCCCCC1CNC(C1CCCSC1)=O 34369,c1(CN(C(C2CCC2NC(C2CCCSC2)=O)=O)CC)ccccn1 34370,CC1(CCO)CCN1C(=O)C(c1cccs1)NC(C1C=CCS1)=O 34371,Cn1ncc2ccc(CN3CCC(O)(C(=O)Nc4cc(C#N)ccc4Br)C3)cc12 34372,c1(C(=O)NCC2CCC(CNC(C(C)SCCCC)=O)CC2)cc(N)cnc1C 34373,C1(NC(c2coc(C3CCC3)n2)=O)COC2(C1)CN(C(c1cc[nH]n1)=O)C2 34374,C1(C(=O)NCC2CCCN(C(c3cncc(Cl)c3)=O)C2)CC1C1CCCC1 34375,N1(C(c2cc(C)sc2)=O)CCCC(NC(c2n[nH]cc2Br)=O)C(F)C1 34376,C(=O)(C#CC1(C)COC1)NCC1CN(C(Cn2ccc(C)cc2=O)=O)CC1O 34377,N1(C(C(=O)NCCSC2CC2)=O)CCC(NC(=O)CCn2cccnc2=O)C(CO)CC1 34378,C1(NC(CCC2(C)CN(C(C(C)=CCC)=O)C2)=O)C(O)C2CCOC12 34379,c1(OC)cc(OC)cc(C(N2CC(O)CC2C(N2CC3CC3C2C#N)=O)=O)c1 34380,C12(CNC(c3cc(CC)n(C)n3)=O)CC(CO1)N(C(=O)C(C)CO)C2 34381,C(=O)(CCCC(C)CC)N1C(C(N2CCCCC(CC)C2)=O)(CC)CCC1 34382,c1(C(N2CCC(O)(C(C)NC(=O)CC3CC(F)C3)C2)=O)n[nH]c2c1CCC2 34383,c1(C(=O)NC(C)CCNC(C2CC3CC3C2)=O)cncc2n[nH]cc12 34384,C=Cn1nccc1C(=O)N(C1CC(C(=O)NC2(C(=O)OCC)CC2)C1)C 34385,C1(C#CC(=O)N2CC=C(CNC(=O)C(n3cc(Cl)cn3)C)CC2)(CC)COC1 34386,C1(C2CC2)(NC(CCNC(c2nn(C)c(O)c2)=O)=O)CCOC1 34387,c1(OC)cc(NCC(C2CC2)N(C(=O)C(C)(C)C(F)F)C)ccc1[N+](=O)[O-] 34388,CCC(CC)(CC)C(=O)NCC(CNC(=O)CCc1cn(C)cn1)C(F)(F)F 34389,N1(C(C(C)O)=O)CCC(n2cc(NC(=O)CSCCC(F)(F)F)nn2)CC1 34390,C1(OCc2cn(C(C)C)nn2)CCCN(C(=O)CC2CCCC(O)C2)C1 34391,C=CC1CN(C(c2ncsc2C)=O)CC1NC(=O)CC12CCCC1C2 34392,C1(NC(Cc2c(C)ccnc2)=O)CC2(C1)CC(CNC(=O)C(c1ccnn1C)O)C2 34393,CC1(C2CC2C(N2CC(F)(c3nn[nH]n3)C2)=O)COC1.N12CCC(C(O)C1)C2=O 34394,n1(CC(=O)NCC(N(C)C(C2COCCO2)=O)C2CC2)cc(CO)nn1 34395,C(=O)(CC(C)(C)CN(C)C)NC(CC(C)C)CNC(C1(N(C)C)CCCSC1)=O 34396,C(c1cccnc1)=C(C)C(=O)NC1CCCN(C(C2(C)CCCOC2)=O)C1 34397,Cc1nn2cc(CC(=O)N(C(C)CN(C(=O)Cc3ccccc3F)C)C)nc2s1 34398,N1(C(C2OCCN(C)C2)=O)CCC2(CC1)CC(NC(c1nccn1C)=O)CCO2 34399,CC1C(NC(=O)C(CCN(C)C)NC(=O)Cc2ncccc2F)CCCN1C 34400,n1(S(C)(=O)=O)cc(CN2CCC2C(=O)NCC(O)CNC(N)=O)cn1 34401,C1(CC)CCC(C(N2CCC2CC(=O)NCCC2(CO)CC2)=O)CC1 34402,C(=O)(C1=Cc2ccccc2C1C)NC(C)CCCNC(=O)C1=C(Cl)CC1 34403,Cc1ccc(C(N2CC=CC(NC(c3ccccc3C(C)O)=O)C2)=O)cc1F 34404,Cc1ccc(Cl)cc1CN1CCOC(CNC(=O)C(C(C)C)c2cccnc2)C1 34405,N1(C(c2cc(C)ncn2)=O)CCC(CO)C(NC(c2csc(C(F)(F)F)c2)=O)C1 34406,C(=O)(C1=CS(=O)(=O)CCC1)N1CCC(N(C(=O)C(C)n2cccn2)CC)CC1 34407,c1(C(=O)OCC)cc(Cl)c(NC(=O)Cc2c(F)cc(F)cc2F)c(Cl)c1 34408,c1(CC(=O)NCC2CC(OC)CN2C(C2CC(C)C2)=O)ccc(F)c(F)c1 34409,N1(C(C(C)NCC2CCc3c(nnn3C)C2)C)CCSc2ccccc2C1 34410,C1(C(=O)NCC2N(C(C3(CCCC)CC3)=O)CC2)CCC(F)C1 34411,N1(C(c2cc(Br)no2)C(=O)NCC(C)C)CCN(C)c2ccccc21 34412,c1(OCc2scc(C(N3CCC(C)(CCO)C3)=O)n2)cnc2ccccc2c1 34413,C1(n2cc(COCC(N)=O)nn2)CCCN(C(=O)CC2COCCOC2)C1 34414,N1(C(Cc2cn(CC)nc2)=O)CCCC(C)C1CNC(=O)Cc1c(C)cnn1C 34415,c1(C(=O)NC2(CNC(=O)CCF)CCC2)cc(Cl)c2c(c1)OCCCO2 34416,N#Cc1ccnc(N2CCC3(CC3C(=O)N(CCCCO)CCO)C2)n1 34417,c1(C(N(C2CN(C(=O)CCc3ccc(N)cn3)C2)C)=O)cccc2c1C(=O)NC2=O 34418,C=CCC(CNC(C1C2CCCC12)=O)C(=O)N1C2CCC1CC2 34419,c1(CC(N2CC(NC(C=CS(C)=O)=O)CC2(C)C)=O)ccc(Br)cc1C#N 34420,CCCCC(C(=O)NCCCCCNC(c1ccnc2ccsc12)=O)C(C)C 34421,NS(=O)(=O)CC(=O)NCC(C1CCCC1)NC(=O)C(F)CC1CCCC1 34422,C(=O)(CC(O)CCCCC)N1CCC(=C)CC1C(=O)NCc1cc(C2CC2)on1 34423,C(C)(CNC(c1cnc(C)s1)=O)(CO)NC(CSCCCC)=O 34424,Cc1cc2c(C(N3CCCC(CCNC(=O)C(C)C#N)C3)=O)cccc2o1 34425,C1(NC(Cc2c(C)ccs2)=O)CCCN(C(c2ccccc2C(F)(F)F)=O)C1C 34426,C1(NC(C2N(CC3CC3)CC2)=O)CCSC12CN(C(C1CCN(CC)CC1)=O)C2 34427,c1(C(=O)NCC2C=CC(NC(c3ccnn(C)c3=O)=O)C2)ccc([N+](=O)[O-])cc1 34428,N1(C(Cc2c(C)ccs2)=O)CCC2CN(C(=O)COC3CCCC3)CCC12 34429,Cc1cc(NC(C2CN(C(=O)C(c3cncnc3)C)CC2(F)F)=O)c(C)cc1O 34430,C1(NC(c2cccc(COC)c2)=O)CC2(C1)CN(C(C1(C)CCCCO1)=O)C2 34431,N1(C(=O)NCCOC(C)C)CCc2c(ccc(NC(c3ccccn3)=O)c2O)C1 34432,c1(C(=O)NCCCC(C)NC(C2CN3CCC2CC3)=O)nn(C)c2c1CCCC2 34433,c1(CN(C)Cc2cc(C3CC3)n(C)n2)cn2cc(Cl)ccc2n1 34434,C(=O)(CC(F)(F)CC)NC(CCC)CNC(C1(C(=O)OCC)CCC1)=O 34435,Cc1cnc(N)c(C(N2CC(F)CC2CN(C)C(C2CCC3(CCC3)O2)=O)=O)c1 34436,Cc1nn2cc(C(=O)NCC(CC(C)C)NC(C3COC(=O)N3C)=O)nc2s1 34437,C#Cc1cccc(C(=O)NC2(C)CCN(C(c3cn(CCSC)nn3)=O)C2)c1Cl 34438,N1(C(=O)CC2CC2)CC2CCCC(C1)N2C(c1cccc2c1NCC2)=O 34439,CC1CCN(C(c2cn3c(n2)CCC3)=O)CC1NC(=O)Cc1ccccc1Cl 34440,N1(C(C(CC)n2cncn2)=O)CC2CCC1CN2CCCc1cccnc1 34441,c1(C(=O)NCCCCCNC(c2nc(C(C)OC)sc2)=O)cc(C2CC2)ncn1 34442,C(=O)(C#CC1CCCCO1)NC1CN(C(c2cc(SC)c(F)cc2)=O)C(C)(C)C1 34443,N1(C(CNC(CC(C)C)=O)=O)CC2CCCN(Cc3cccc(F)c3Cl)C2C1 34444,c1(COCCC(=O)N(C2CCN(C(C3CC3C)=O)CC2)CC)ccc(F)cc1 34445,C(=O)(C(C)(C)CCC#N)NCC1(F)CC(NC(c2c(C)nco2)=O)C1 34446,CCC(O)C(F)(F)C(=O)NC1CC1NC(C1CCC1)=O 34447,Cc1ocnc1CC(=O)N(CCCCCNC(=O)CC(C)n1cccc1)C 34448,C(CCCC(C)NC(=O)C(C1(C)CC1)NC(=O)CCCC1CCCO1)OC 34449,C(CCCC(=O)N1CCCC1CN(CC(=O)Nc1nc[nH]n1)C)NC(CC)=O 34450,c1(OC)cccc(S(=O)(=O)N2CC3C(NC(=O)CCc4nc(C)no4)C3C2)c1 34451,C1(NC(C)=O)CCCCC12CCN(C(c1cc3c(Cl)cccn3n1)=O)C2 34452,c1(NC(COC)=O)ccc(C(=O)NCC2CCC(NC(=O)CCSC)C2)cc1 34453,c1(C(C(C(=O)OC)C)NC(=O)Nc2ccc(OC)nc2)cc(C)ccc1OC 34454,n1(CC(=O)OC)cnc(C)c1C(=O)NCCCCNC(=O)C(C)Cn1cccn1 34455,N1(C(c2c(C(C)NC(C3CC(F)C3)=O)noc2)=O)CCC2CC12 34456,C1(C(=O)NCCOC2CN(C(CC3(C=C)CC3)=O)C2)CCS(=O)(=O)C(C)C1 34457,N1(C(C23CC(OC)C2C3)=O)CC(NC(=O)CCCc2nc(C)cs2)C(O)C1 34458,CC(=O)CCN=C(NCc1cccc(Cl)c1F)NCc1ccc(C)cc1C 34459,N1(Cc2c(OC)cccn2)C2CCCC1CC(NC(c1ccc(C)cn1)=O)C2 34460,C1(C)(CNC(NC(C#C)C2CC2)=NCC2CC2)NC(=O)NC1=O 34461,CC(C)(CCNC(C1CCC1C(C)(C)C)=O)NC(=O)OC(C)(C)C 34462,Cc1cc(NC(N2CCC(C)C2CO)=O)ccc1OC(F)(F)F 34463,C(C(C)(C)CCNC(C1(CF)CCOCC1)=O)NC(CC(C)n1ccnc1)=O 34464,C1(N(CC(C)NC(=O)CCOCC(F)F)C)CCCNC1 34465,N1(C(C)=O)CC(O)CC1C(=O)NC1CCC1NC(c1nn(C)nc1Br)=O 34466,c1(C(N2C(C)CC2C(=O)NC2CCCCC2)=O)ccn2cncc2c1 34467,c1(C(=O)NC2CCN(C(C(CC)F)=O)C2(C)C)ccc2nc(O)oc2c1 34468,N1(C(C(=O)NCCCC(=O)OCC)C2CC2C2OCCO2)CCOC(C(N)=O)C1 34469,C1(C(=O)NCC2CC(NC(C3CN(S(CC)(=O)=O)C3)=O)C2)CCC(F)(F)CC1 34470,CC(C)CC(F)C(=O)NC1CCCC1NC(=O)Cc1nn(C)cc1Br 34471,Cn1cnc(C(N2CS(=O)(=O)CC2C(=O)NC=O)=O)cc1=O 34472,C12(NC(c3ccc(O)nc3)=O)CCCC1N(C(c1ccc3nccn3c1)=O)CC2 34473,N1(C(c2c(C)nc[nH]2)=O)CCOC(C(C)NC(=O)C(c2ccccc2)O)C1 34474,CC1CN(C(C2CCCN2C)=O)CCN1C(c1cc(Cl)ns1)=O 34475,Cc1c(C(N2CCC2C2CCCCC2)C(=O)NCCC2CC2)oc2ccccc12 34476,C(=O)(C(CCSC)NC(=O)CNC(N)=O)NC12CC(OC)C1C2 34477,c1(Cn2cc(CN(C(C(C)OCC=C)=O)CC)nn2)ccc2[nH]ncc2c1 34478,C1(NC(CC2CC(=C)C2)=O)CC2CCC1(NC(=O)CN1CC3CC3C1)C2 34479,Cn1ncc(=NC(=O)C2CC23CCN(Cc2ccc(C(=O)O)s2)C3)[nH]1 34480,c1(C(=O)NC2CCCC(NC(C3CC(F)C3)=O)C2)c(F)c(F)c(F)c(F)c1F 34481,N1(C(C2CC(C)CN2C(c2cn(C)cn2)=O)=O)CCC2(CCSC2)C1 34482,Cc1cnc2cc(C(N3CCCC3C(C)NC(=O)CC(F)(F)F)=O)ccn12 34483,N1(C(C2(COC)CCCC2)=O)CCC(C2CC2)(NC(=O)C(O)C2CCCC2)C1 34484,C1(C2(O)CCOC2)(C(N2CCC(CN(C)C(c3ccc(C4CC4)o3)=O)C2)=O)CC1 34485,C1(C(=O)NCC23N(C(CCC=C)=O)CC(C2)C3)CCc2nc(C(F)(F)F)[nH]c2C1 34486,C1(C(N(CC(C)C)C2CC2)=O)CC2CN(C(=O)C3=COCC3)CC2C1 34487,C1(NC(Cc2c(C)noc2Cl)=O)CC2CCC1N2C(=O)C=Cc1cn(C)nn1 34488,C=CCC(CC(C)C)C(=O)NC1CCN(C(=O)CC2CCSC2)C1C 34489,N1(C(C(CC)F)=O)CCN(C(=O)CSc2cccs2)C2COCC12 34490,CC(CC(=O)N1CCC(C(=O)NCC(C)(C)N2CCCC2)O1)N(C)C 34491,C1(NC(CCN(C(C)=O)C)=O)CCN(C(=O)CC2CC3(COC3)C2)C1C 34492,C1(NC(C2(SC)CC2)=O)CCCCC1NC(=O)CCc1cncnc1 34493,c1(CC)oc2ccccc2c1C(N1CC(CNC(=O)C(C)CSC)C(F)(F)C1)=O 34494,CC(Cc1cnc[nH]1)N=c1[nH]c(=NC(C)c2cc[nH]n2)[nH]c2ncn(C)c12 34495,Cc1nc(CC(=O)NC(C2(O)CN(C(C3(NC(N)=O)CC3)=O)C2)C)co1 34496,C(=O)(CCCCBr)N1CC(C)(C(=O)NC(C(C)C)COC(C)(C)C)C1 34497,c1(OCC(=O)NC(C2CCCN2C(c2nn(C)cc2CO)=O)C)cccc(F)c1 34498,CCCC(C)CC(=O)NCC1(O)CCCN(C(=O)CCc2nc(CCC)no2)C1 34499,CN1CCCOC1CC(=O)N(CC)CC1CN(C(=O)CCc2ccncc2)CCO1 34500,c1(NC(C(=O)NCCNC2CC2(F)F)=O)cccc2c1CNC2=O 34501,Cc1sc(Cl)nc1C(N1CCCCC1C(C)NC(c1cc(C(C)C)n(C)n1)=O)=O 34502,c1(C(=O)OCC)cc(=O)n(C(N2C(C)(CN)CCCC2)=O)cn1 34503,C1(CC(=O)OCCCC2(CC=CCC(=O)OC)CC2)CCC(C)C1 34504,c1(C(=O)NCCCCCN(C(=O)CC2CC2(C)C)C)cnn2c(Cl)cccc12 34505,Cc1cc(C(=O)NC2CC2NC(=O)COCc2nccn2C)cc(C)c1Cl 34506,CC1CN(C(=O)CSS(C)(=O)=O)CC1NC(=O)CCCc1ccsc1 34507,n1(C(C)(C)C)cc(Cl)c(C(=O)NC2CCC2NC(C2CC(F)C2)=O)n1 34508,N1(C(c2n[nH]c(C)c2Cl)=O)CCCC(C)(CNC(=O)CC2CC(C)(C)CCO2)C1 34509,N1(C(c2cc(CCC)[nH]n2)=O)CCN(C(C2CCC(=O)N2)=O)CC1C(C)(C)C 34510,S(=O)(=O)(c1c[nH]c2nc(Br)ccc12)NCC1CCC(CC)C1 34511,C1(CNC(CCNC(=O)OCC)=O)CC2(CCC2)CN1C(C1CC1(Cl)Cl)=O 34512,C1(NC(CCC2N(C)CCC2)=O)CC=C(C(=O)Nc2ccc(C3CC3)nc2)C1 34513,O=S(=O)(c1ccncc1)NC1C2CCC1CC2 34514,CC(CS(C)(=O)=O)C(=O)N1CC2CC(NC(=O)CSc3cccnc3)C(C2)C1 34515,C1(NC(C(CC)C)=O)C2CC1(C)CN2C(c1nccn1C(C)C)=O 34516,CC(CCCc1ccccc1)C(=O)NCC1N(C(=O)CC2(C)CC2)CCC1(C)C 34517,Cc1cc(C(N2CCC(CC(=O)NC3(CN4CCCC4)CC3)C2)=O)sn1 34518,c1(CC(=O)NC2C(NC(C(CC)(C)OC)=O)CC2)ccc2scc(C)c2c1 34519,c1(CCC)nnc(S)n1CC(=O)N(C)CC1(NC(c2cc(C#N)cs2)=O)CC1 34520,CCCCC(C)(C)NC(=O)C(C1CN(C(C2CC3C=CC2O3)=O)C1)OC 34521,C=CCC(C)(C)C(=O)NCC(C1CCN(C(C2CCC(C(N)=O)C2)=O)CC1)O 34522,OC1COC2C(NC3CCCC4(C3)N=N4)COC12 34523,c1(C(CC(=O)NCCOCCN(C(=O)C(=O)C(C)(C)C)C)O)cc(Cl)cc(Cl)c1 34524,CC1CC2(CCO1)CC2C(=O)N(CCCCN(c1ccnn1CC1CCC1)C)C 34525,N#Cc1ccc(CCNC(=O)CC2CCN(C(=O)CCc3ccc[nH]3)C2)cc1 34526,C(c1ccc(F)cc1)=C(C)C(=O)NCC1CC(F)(CNC(C2(F)CCOC2)=O)C1 34527,N(C(=NCC(C)(C)CC#C)NCC(C(C)(C)C)SCC)C(C#C)CNS(C)(=O)=O 34528,c1(C(N2CCOCC2)CNC(Cn2cc(C(C)(C)SC)nn2)=O)ccc(Br)cc1 34529,N1(CC(N2CCC(OCC)C2)=O)CCN(CC(C)(C)C2CCCC2)CC1 34530,C1(CN(C(C(n2ccc(C(F)(F)F)n2)C)=O)C)CC(F)CN1C(c1ccco1)=O 34531,N1(C(COc2cccc(C)c2)=O)CCC(C)(C)C(NC(=O)CC2(CO)CC2)C1 34532,N1(C(C(C(C)NC(c2cccc(NC)n2)=O)C)=O)CCC(CO)C(O)C1 34533,CN(C)NC(=O)CCC(=O)N(CCC(=O)NC1COCCC1CO)CCCO 34534,C1(C(CN(CC=O)C)(C)O)CCCNC1.C(=O)(CN(C(C)=O)CC)NCCOC 34535,N1(C(C2CCOC2=O)C(=O)Nc2c(OC)scc2)CCOCC12CCC2 34536,C1(C(=O)NC(C2CCN(C(Cc3ncc(C)o3)=O)CC2)C)CCCC(C)(C)C1 34537,C(=O)(C1=NN(C(C)(C)C)C(=O)CC1)N1CCN(CC(C)CC(F)F)C(=O)C1 34538,c1(C(=O)NC2CC3(CN(C(C(COC)O)=O)C3)C2)cccc2c1ncn2C 34539,Cc1c[nH]c(C(=O)NCC2CC2NC(c2[nH]nnc2-c2ccnn2C)=O)c1 34540,Clc1ccc(I)c2c1CCN(CC1CCc3ncccc3N1)C2 34541,N1(C(C2CCC(COC)C2)=O)CCN(C(c2cncn2C)=O)CC(O)C1 34542,C(C(O)CS(=O)(=O)c1cccs1)CNC(Cc1c(OC)ccc(Cl)c1)=O 34543,n1(CC)nc(C)c2cc(C(N3CCC(NC(=O)CCC4CC4)C34CC4)=O)sc12 34544,C12(C(N3C4CN(C(C5C(CC)C5)=O)CC3CC4)=O)CCCCC1CCCC2 34545,C#CC1CC2CCC1N(C(C1(CC)CCN(C(=O)CC(F)(F)C(F)F)C1)=O)C2 34546,c1(C(C(=O)NCC2CN(C(=O)C(C)OCC3CCCO3)C2)SC)cccc(C)c1 34547,c1(C(N2CCC(CNC(Cc3cc(OC)ncc3)=O)C2)=O)cc[nH]c2nccc1-2 34548,c1(NC(N2CCC(O)(c3n(C)nnc3)C2)=O)nc(C(F)(F)F)ccc1Br 34549,n1(CC)cnc2c(N3CCC(CC#N)C3)[nH]c(=NCCCCCCOC)nc12 34550,c1(OC)nscc1C(C(=O)NC1CCCC1)N(c1occc1C)C 34551,C(CCOC1CC1)(C(=O)N(C(C)CC(N)=O)C)NC(C(C)C)=O 34552,C1(CS(=O)(=O)NCC(C)(C)CO)(CCOC)CCCC1 34553,CCC(CC)(C(=O)NCCOC(C)CC(C)C)NC(C1C2COCC12)=O 34554,c1(C(=O)N=c2cc(-c3ccccc3)o[nH]2)cc(Cl)cc2c1NCCC2 34555,C(=O)(C#CC1CCCCC1)NC12C(OC(c3ccc(Cl)c(F)c3)=O)C1CCC2 34556,c1(OCC)ccccc1C(=O)NC(C)CCCNC(c1cscc1SC)=O 34557,Cn1cc(C(N2CCC(O)(CNC(C3CCC(O)C3)=O)C2)=O)c2cc(F)ccc12 34558,Cc1cc(C(N2CCC(C)(C(=O)NCC3(C)CC4CCC3C4)CC2)=O)c(C)n1C 34559,C#CC1CCC(N(C(=O)C(=O)NCC(=O)NCC=C)CC2CC2)C1 34560,N1(C(CNC(N)=O)=O)CCOCC1C(=O)NC1COCC1CCO 34561,C(=O)(CCC(=O)NN(C)C)NC1(C)CC(NC(C(C2CCCC2)OC)=O)C1 34562,c1(C(N2C3(CNC(c4cccc(Br)c4)=O)CCC3CC2)=O)cccc2cccn12 34563,c1(C(=O)NCC(C(C)C)NC(C2(F)CC2)=O)ccc(SC(F)(F)F)nc1 34564,N1(C(CC2(C)CC2)=O)CC(NC(c2ccc(SC(F)(F)F)o2)=O)CC2(CC2)C1 34565,C1(NC(C=CSC)=O)C(C)CN(C(=O)CN2CCCNS2(=O)=O)CC1C 34566,c1(CC(C)NC(=O)C(N)=O)ccccc1CNC(=O)CC1(O)CCOC1 34567,N1(C(CC2C(C)(C)CCO2)=O)CC=C(CNC(=O)Cn2cnc(C(N)=O)n2)CC1 34568,C1(NC(CNC(=O)NC)=O)CN(C(c2cc(Cl)cn2-c2ccccc2)=O)CC1C 34569,CC(C)C(CC(=O)N(C1CC(CO)C1)C)NC(C1CC2CC(=O)C1O2)=O 34570,C(CCC(=O)c1ccccc1)OCCN(C(=O)C(=O)NC)C.CC(=O)N(C)CCO 34571,c1(C(N2C(CNC(C3C(C)=CCS3)=O)CC(O)C2)=O)cnn2c1CCC2 34572,CC1(CNC(=O)C=CC(N)=O)CC(F)(F)CN1C(C1CCC2(CC2)C1)=O 34573,C1(NC(Cc2nc(C)[nH]n2)=O)CNCCOC1 34574,C1(NC(c2cccc(=O)o2)=O)CN(C(=O)CCCC(F)(F)F)C2(CCOC2)C1 34575,c1(CC)nc(C(=O)NC2CCCC2NC(c2cc(Cl)c[nH]2)=O)c(C)o1 34576,C(C)(C(=O)N1CCN(C2(C)CCC(=O)NC2)CC1)(C(C)C)OC 34577,c1(C(N(CC(C)NC(C2CCCN(C(C)C)C2)=O)CC)=O)cc(Cl)ncc1F 34578,N1(C(CCNC(COC)=O)=O)CCOC(CNC(c2c[nH]nc2COC)=O)C1 34579,c1(C(N(C2CCN(C(C3CC34CC4)=O)CC2)CC#CC)=O)ncncc1Cl 34580,c1(C(N2CCC(NC(=O)CCC3CC3)C23CC3)=O)ccc2cnnc(O)c2c1 34581,C(CC(C(=O)NCc1cncs1)NC(=O)C=CC(F)F)=CC 34582,c1(C(N2CC(CNC(CCCc3cc(C)no3)=O)OCC2)=O)cnc(N)c(N)c1 34583,Cc1ccc(CNC2CC3(C2)CC(NC(=O)Cc2ccc(C#N)cc2)C3)c(O)c1 34584,N1(C(C=C(C)C2CC2)=O)C2COCC1CC(NC(=O)Cc1cnn(C)c1)C2 34585,c1(-c2c(C(=O)NC3C(CNC(C(C)CN(C)C)=O)C3)occ2)nnc(S)n1C 34586,C1(CC)CN(C(C2CC(=O)CS2)=O)CC1C(=O)NC1CCC(C)(CC)C1 34587,c1(NC(C(c2sccc2Br)N(C)Cc2cncc(F)c2)=O)ccccc1F 34588,C(=O)(C(O)C(C)(C)CC)N1CC(NC(CCC=CC)=O)C2(C1)CC2 34589,C1(CC)CN(C)C(=O)CN1C(=O)NCC1CCN(Cc2ccccc2)C1 34590,C1(CCC2N(C(=O)CSC(F)(F)F)CCC2)CCCCN1C(=O)CC1CCC1 34591,N1(C(C2C(NC(CCOC(C)=O)=O)CC2)=O)CCOC(C#N)C1 34592,c1(C(=O)NCc2occ(C(N(CC(CC)NC(C)=O)C)=O)c2)cc(O)nc(C)n1 34593,CN=S(C)(=O)c1cccc(C(=O)NC2CCN(C(=O)COC3CCC3)C23CC3)c1 34594,C#Cc1ccc(C(=O)N(CC(O)CN(C)C(c2cn(C3CC3)nc2C)=O)C)cn1 34595,Cc1ccc2nc(N3CCCC(C(C)NC(c4c(C)nn(C)c4C)=O)C3)sc2n1 34596,CC1(C)OCCOC1CC(=O)NCCOCCCNC(=O)CC1OCCCO1 34597,N1(CC(C)CC=CC(F)(F)F)C(=O)CN(C(C)C)C1=O 34598,C1(CCNC(C2C(C)C2)=O)CCCN(C(c2cocn2)=O)C1 34599,Cn1cnc(CCNc2cccc(OC3CCC3)c2)cc1=O 34600,c1(C(N2CCCC(C)C2CCNC(=O)CNC=O)=O)c(Cl)ccc(Br)c1N 34601,c1(CCCNC(c2cccc(-c3nn[nH]n3)c2)=O)cc(Cl)cc(Cl)c1 34602,C1(CC(=O)NCC(C)(C2CCC2)NC(c2cc[n+]([O-])cc2)=O)CCC(=O)CC1 34603,C1(C2CCN(C(C3(C)CC3C)=O)C2)(NC(c2n[nH]c(C)c2C(F)(F)F)=O)CC1 34604,c1(C(=O)NCC2(OC)CN(C(C3(CC)CCCCO3)=O)C2)ccc(C)cc1Cl 34605,c1(CN(CCC(=O)OCC)C(=O)NC)ccc(C)cc1OCCCCCC 34606,C(=O)(C(CCC(N)=O)NS(C)(=O)=O)NCCCn1cc(-c2n(C)ncc2)nn1 34607,N(C(=NCCC(=O)N1CCCC1)N1CCCC(F)(F)C1)CC(C)C(F)F 34608,C#CCCC(=O)NCC1CC(C(=O)NCCC(C)(C)N(C)C)C1 34609,c1(OC)ccc(S(=O)(=O)NC(C2(F)CCCN(C(=O)CSC)C2)=O)cn1 34610,C(CC(C(=O)N1CC(F)(CF)C1)NC(=O)CCCc1ccsc1)OC 34611,c1(CC(=O)NCCCNC(CC(c2cccc(OC)c2)C)=O)ccc(F)c(C)c1 34612,CC(C(=O)NCc1ccc(CNC(=O)C=CCN2CCCC2)cc1F)S(N)(=O)=O 34613,C12(CNC(=O)NCc3ccc([N+](=O)[O-])cc3C3CC3)CCOC1CS(=O)(=O)C2 34614,N1(C(C(CC#C)(C)C)=O)CC2CCC1C(CNC(c1ccn(C3CC3)n1)=O)C2 34615,N1(C(C=CC(=O)N(C)C)=O)CCCC(F)(C(=O)NC2C=CC(CO)C2)C1 34616,c1(C(N2CC(OC)(CNC(c3ccnnc3)=O)C2)=O)noc(CC)c1Br 34617,Cc1nc(O)nc(O)c1CC(N1CCCC(CNC(C2(C(N)=O)CCC2)=O)C1)=O 34618,c1(N(C)C)ncc(C(N2CC(C(C)(C)O)(CNC(c3cnc[nH]3)=O)C2)=O)s1 34619,N(C1CC2(CCC2)Oc2ccccc21)C(CSc1[nH]c(=N)sc1)=O 34620,C1(C(N2CC(CC)C2)=O)CN(C(=O)C(C)n2ccnn2)CC2(CCC2)C1 34621,c1(C(=O)NCCCNC(C(c2ccc(F)cc2)C)=O)nccc(C#N)c1F 34622,c1(C(N(C2CCCC2)CCNC(=O)CO)=O)c[nH]c2cccc(Br)c12 34623,c1(OCC)ccccc1C(N1CCCC1(C)c1cn(Cc2ncnn2C)nn1)=O 34624,CCCCCCCCC(F)C(=O)N1CCN(C(c2c(C)nsc2N)=O)CCC1C 34625,c1(CNc2cccc(OC(CCCCCC#N)=O)c2)ccc2c(O)nncc2c1 34626,C=CC(C)CC(=O)NCCOCCOCCN(C)C(C1CCCCO1)=O 34627,N1(C(c2cncn2C2CC2)=O)CCCC(F)(C(=O)NCC2=CCCOC2)C1 34628,C1(CC#C)CCCCN1C(C1CCN1C(=O)CC1CCOC1)=O 34629,N1(C(C(CC)(C)F)=O)CCC2(CC1)CN(C(C1CC3CCC3C1)=O)C2 34630,O=C(C1=CC(O)CCC1)NCC1CC1NC(c1cccc[n+]1[O-])=O 34631,C(c1ccccc1)=C(C(=O)NCC1C(NC(CCC=C)=O)CCC1)CC 34632,n1(CC)cccc1CCNC(c1nnnn1C1CCOC1)c1cnsc1 34633,c1(C(=O)NC(CCNC(C(C(C)O)N(C)C)=O)C)nnc2n1CCCCC2 34634,Cc1coc(C(C)(C)C)c1C(N1CC(N(C(=O)C(F)C2CCOC2)C)C1)=O 34635,c1(CN(C)C(=O)NCc2ccc(Cl)nc2)cc(Cl)c(F)c(Cl)c1 34636,N1(C(C2(C)N(C(c3c(C(C)C)noc3)=O)CCC2)=O)CCc2ncncc2C1 34637,C1(C(N(CC(C)NC(=O)CCc2cnc[nH]2)C)=O)CC2(C1)C(F)(F)C21CC1 34638,C(CO)(CCCCNC(C1(F)CCCCC1)=O)NC(C1(CC)CCC1)=O 34639,C(=O)(CC1=CCOCC1)NC1C(C)CN(C(c2cc(N(C)C)ccc2N)=O)C1 34640,C1(CN(C(c2c(OC)nsc2)=O)C)CCCN(C(C2CCCCN2C)=O)C1 34641,N(C1CCOc2ccc(Cl)cc21)C(c1c(Sc2ncc(C)s2)ccc(F)c1)=O 34642,N1(Cc2c(C)sc(Cl)c2)Cc2cncnc2C1 34643,C#Cc1ccc(CC(=O)NCC2(NC(c3coc(C(F)(F)F)c3)=O)CC2)cc1 34644,N1(C(C2CC(SC)C2)=O)CCN(C(=O)CC(C)F)CC1c1ccnn1C 34645,CC(C)S(=O)(=O)CCC(CNC(C)C(=O)Nc1ccc(Br)cc1Cl)C(F)(F)F 34646,CC(C)(Cc1cccc(Cl)c1)C(=O)N1CCC(C(C)(C)NC(=O)C2=CCCC2)C1 34647,c1(CCC)cc(C(=O)NC2CCC2CNC(c2ccnn2CC(C)C)=O)on1 34648,c1(SCC(=O)NCC(CNC(C2(CCC#C)CC2)=O)(C)C)ccc(Cl)cc1 34649,S(=O)(=O)(c1ccncc1)N(C(=O)Cc1cncnc1)CCOCC 34650,CC1c2c[nH]nc2CCC1C(N1CCC(CNC(=O)CC2=CCCC2)C1(C)C)=O 34651,N1(C(=O)OC(C)(C)C)CCN(Cc2cnc(OC(F)F)c(C)c2)CC1C#N 34652,c1(C(=O)NC(C)C(=O)NC(c2nc[nH]n2)CO)cc[nH]c2nccc1-2 34653,c1(C(=O)NC2C(NC(c3cc(C)nc(C)n3)=O)CCC2)ccc([N+](=O)[O-])n1C 34654,C1(CC(N2CCC(O)(CNC(c3ccc(CC)s3)=O)C2)=O)OCCCC1(C)C 34655,c1(C(=O)NCCNC(c2snnc2C2CCC2)=O)cccc2cnsc12 34656,C1(NCC(C)(C)OC(=O)NC(C(=O)NCCCOC)C)CC2C=CC1O2 34657,Cc1ccc(C(=O)NCC2CCN(C(C34CCC3C4)=O)C2)cc1 34658,c1(C(=O)NC2C3CC2N(C(c2cc4n(n2)CCO4)=O)C3)nccn2ccnc12 34659,N1(C(=O)CCN2CCCC2)CCC(C(N2CCCC(CN(C)C)C2)=O)CC1 34660,C1(C(N2CCN(COCC)CC2)=O)CCCC12OCCO2 34661,C1(NC(C(=O)N(C(C)COC)CC)=O)CCCCC1.C1CC(=O)O1 34662,N1(C(CNC(CC)=O)=O)CC(NC(=O)Cc2ccccc2C)CCC1C 34663,C1(C(N2CCCC2c2nccs2)C(=O)NCCOCC2CC2)C=CCCC1 34664,C(C(F)(F)CCC(=O)NCCNS(N)(=O)=O)n1cc(C=CC)nn1 34665,C(=O)(C(CCN(C)C)NC(=O)Cc1ccc(Cl)cc1)N1CC(C=C)C1 34666,c1(SCC(C(=O)NS(=O)(=O)C2(c3ccccc3)CC2)O)ccc(O)cc1 34667,C1(C(N2CC(C)C(NC(C3(C(C)(F)F)CC3)=O)C2)=O)CC1C1CCOCC1 34668,CCC(COC)C(=O)NC1CC(CCN(C(C=CC(=O)OC(C)=O)=O)C)C1 34669,c1(CCC)nc(C)c(C(=O)N(C2CCCC(NC(c3cn(C)c(O)n3)=O)C2)C)o1 34670,N1(C(C)C)CCCCC1C(=O)NCCC1(O)CN(C(C2CCCN2C)=O)C1 34671,C(=O)(C(C)CC(=C)C)N1CCC(N(CC#C)C(C2(CC(F)F)CCC2)=O)C1 34672,Cc1nc(O)nc(C)c1C(=O)N(CC(C)NC(C1COCCC1(F)F)=O)C 34673,C12(C(=O)NCC(C3CC3)NC(C(CN(C)C)(F)F)=O)CCCN(C1)S(=O)(=O)C2 34674,c1(C(=O)OC)ccc2ncc(C(N3CCCCCCC3c3ccccc3)=O)cc2c1 34675,c1(CNC(=O)NCC(=O)NC(CC)(C)CNC(C2CCCC2)=O)ncc[nH]c1=O 34676,N1(C(c2c(OC)nccc2)=O)CCCC(N(c2cnc(C#N)cn2)C)CC1 34677,c1(C(N(C2CCN(C(C3CCC3C)=O)C2)CC)=O)c2c(nn1C)CCC2 34678,c1(C(N2C3CN(C(=O)Cc4cn[nH]c4)C(C3)C2)=O)nc2cnccc2s1 34679,C(CC(C)(C)CCO)NC(C1N(C(C(C)OC(C)=O)=O)CCCC1)=O 34680,Cc1cncc(C(F)(F)F)c1.C12CCN(C1)C(=O)O2 34681,c1(C(=O)NCC23C(CN(C(C4(C)C(C)C4)=O)C2)CC3)ccnc2cc(Cl)ccc12 34682,CC1(C(=O)NC2CC2NC(=O)C(c2ccc(F)cc2)(F)F)CCC(O)CC1 34683,N1(C(C(C=C)O)=O)CCN(C(=O)COc2cc(Cl)cn2-c2ccccc2)CC1 34684,c1(C(N2CC(C=C)C(NC(=O)COc3cn[nH]c3)C2)=O)csc2ccc(F)cc12 34685,C(CCCCC(=O)NC1CCC(C(NC[Si](C)(C)C)=O)C1)OC 34686,Cn1ccc2sc(CN3CCCN(C(=O)CNS(C)(=O)=O)CC3)cc12 34687,C1(OC(C)(C)C)CC(CC(=O)OCc2ccc(C(F)F)cn2)C1(C)C.C1CCC1 34688,c1(NC(N=c2n(-c3c(OC)ccc(F)c3)[nH]nn2)=O)cccc2c1nc(O)n2C 34689,c1(C(N2CC(NC(C3CCN(C(CC)=O)C3)=O)C(F)C2)=O)c(N)sc(C)c1C 34690,CC1=NN(C)C(=O)C1CC(=O)NCC(C(C)(C)C)NC(=O)C(C)CC1CC1 34691,c12c(cc(C)cc1C)C(=O)N1CCN(CC1C)C(=O)c1cscc1-2.CN.OC 34692,C1(NC(c2c(C)nc(C)c(C)n2)=O)CCC2(CCCN2C(=O)CC2CSC2)CC1 34693,c1(CN2CC(NC(=O)OC(C)(C)C)C(c3ccnn3C)C2)cc(O)ccc1F 34694,CC1CN(C(C2CC2c2ccc(Br)cc2)=O)CCN1S(=O)(=O)c1cccs1 34695,C=CCN=C(NCS(=O)(=O)CC)NCCNC(C1CC(=O)N(c2ccccc2)C1)=O 34696,Cc1cccc2c(CC(=O)NCC3(C(=O)NC4(C)CCN(C(N)=O)C4)CC3)c[nH]c12 34697,c1(C(=O)NC2(CO)CN(C(C3CCC(OC)C3)=O)C2)cnc2ncnn2c1 34698,c1(C(=O)NCCCCNC(c2c(C)cc(CO)o2)=O)cc(C)c(O)c(N)c1 34699,CCC(CC)C(C)C(=O)N1CCC(C(=O)Nc2cn(C)nc2C(C)C)(CF)C1 34700,c1(C(N2CCC(C(C(=O)NC(CCC)C3CCC3)F)C2)=O)cc(OC)n(C)n1 34701,C1(C(=O)NCc2c(C)ccs2)C2CC3C(C2NC(=O)C(C)(C)C(C)O)C13 34702,c1(CN(C)CCNC(c2cccc(-c3ccncc3)n2)=O)nsc2c(Cl)cccc12 34703,N1(C(CCC2CC(CC(c3cc(C)sc3)O)C2)=O)CCCCC1C 34704,Cc1ccc(C(CNC(c2occc2C)=O)NC(c2scc(C)c2C)=O)cc1 34705,O=C1CCCCn2nc(C(N3CCOCC(CNC(C4CCOC4)=O)C3)=O)cc21 34706,C1(NC(CC2(C(=C)F)CCC2)=O)CN(C(=O)C(C)CC(F)F)C(C)(C)C1 34707,c1(CC)cnc(C)nc1N1CCC(N(C(C)=O)CC)C1.C1(=O)CO1.C(C)(C)(C)O 34708,C1(CC#C)CN(C(=O)C(Cc2ccoc2)NC(c2cc(Cl)cn2CC)=O)CCO1 34709,CC1CCC(C)(C(=O)NCC(=C2CN(C(C3CC4CCC3C4)=O)C2)F)CC1 34710,Cc1c(C)c(C)c(C(=O)NCC2CCCC2NC(=O)CCOC2CC2)c(C)c1C 34711,c1(C(=O)NCCC2N(C(CCCC#C)=O)CCC2)ccc(NC)c(C(C)C)c1 34712,c1(C(=O)NC(C(=O)NCc2ncc(C)[nH]2)C2CC2)cncc(C#N)c1 34713,Cc1ccc(CC(C(=O)O)NC(C2CCO2)=O)nc1 34714,c1(N2CCCC(CC3CCCN3NC(C3(C#C)CCC3)=O)C2)ncc(C#N)cc1F 34715,C1(N(C(=O)C(C)C(C)C)CC)CCN(C(=O)CC23COC(C)(C2)C3)CC1 34716,c1(C(N(C(CNC(C2(CC=C)CC2)=O)C)CC)=O)ccc(F)c2ccncc12 34717,c1(C(N2CC(C)C(NC(c3csc(O)n3)=O)CC2)=O)cncc2c(O)nccc12 34718,C(CCC(C(=O)NC(C1CC(=C)C1)C)N(C)Cc1cccc(C)n1)OC 34719,n1(CC(=O)NCCOC2CCN(C(=O)C=Cc3cc[nH]n3)C2)cnnc1O 34720,Cc1cc(C(=O)NCC(C)(C)OCC(=O)N(C)CC2(O)CCC2)ccc1O 34721,C1(CCC)CN(C(c2cc(F)ccc2F)=O)CCN1C(c1cc2n(c1)CCC2)=O 34722,C1(C(=O)N(CC(C)CN(C)C(c2ccnnc2)=O)C2CC2)CC(C)(c2ccccc2)C1 34723,C1(CCC)CCCCC1NC(c1csc(CNC(C2(CF)CCCCC2)=O)c1)=O 34724,CC1(C(N2CCCN(C(=O)CC3CCCC(F)(F)C3)CC2)=O)COCCC1(F)F 34725,c1(N)ccc2c(n1)CCCC2=O.CC1(CO)CCN(C(C2CCC(=O)N2C(C)C)=O)CC1 34726,c1(CC(=O)NCC(CO)NC(c2coc(C3CC3)n2)=O)cnc(C2CCC2)[nH]1 34727,C(=O)(C1=C(Cl)CCCC1)NCC1(COC)CCCN1C(C1CC12CCC2)=O 34728,c1(C(N2CCC(COC)(NC(C3(CF)CC3)=O)C2)=O)cc(Cl)cc(C(F)(F)F)n1 34729,N1(C(C(C(C)C)C2CCC2)=O)CCC(C)(NC(c2nnc(O)nc2O)=O)CC1 34730,c1(OC)c(Cl)ccnc1NC(C1CN(Cc2ccc(F)c(F)c2)CC1O)=O 34731,N1(C(C2CC(O)(CC#C)C2)=O)CCC(COC)(NC(C2CN(C)CCO2)=O)CC1 34732,C(CC(C)(C)Cc1cn(C2CC2)nn1)N(C)CC1CCCN(CC#N)C1 34733,N1(C(=O)NC(C)C(=O)NC2CCC2)CCN(C2CC2)C(C)C1 34734,N1(C(CCN(CC)CC)=O)CCN(C(=O)C=C(C)C(C)C)CC(C)C1.C(C(=O)OC)NC 34735,C1(OC)CC(C(=O)NCC(C)CNC(=O)C(C)OC(C)(C)C)N(S(C)(=O)=O)C1 34736,N1(C(C2(C)CNC(=O)C2)=O)CCCN(CCNC(=O)C=Cc2ccsc2)CC1 34737,CN1CCC(F)C(NC(=O)CCOC2CN(C(=O)C3=CCCOCC3)C2)C1 34738,C=CCCCC(C(=O)NCc1cccc(Br)c1)OC(C1CN(CC)C(C)CO1)=O 34739,N1(c2nnc(C(CC)O)n2CCC(N2CCCCC2)=O)CC2CCCCC2C1 34740,Cc1cc(F)ccc1CC(=O)NC(CNC(=O)CC1CCCC(=O)N1)CC(C)C 34741,C(C(O)CNC(=O)C(F)C1CCC1)N(C)C(C1CC(CCO)C1)=O 34742,c1(C(N2C(C(N(C(CC(=O)NCC(=O)OC)C)C)=O)CC2C)=O)c[n+]([O-])c(C)cn1 34743,C1(CC(=O)NCCNC(C(CCOC)c2ccccc2)=O)CC2(CCCC2)CO1 34744,c1(NC(Cn2c(C)cnc2)=O)cccc(CNC(c2cncc(N)n2)=O)c1 34745,N1(C(COC)=O)C2CCC1CC(O)(CNC(=O)C(C)OC1CCCC1)C2 34746,Cc1cc(C(=O)NC2CCN(C(C3CC4(CC4)C3)=O)CC(O)C2)cc(C)c1N 34747,N1(C(c2nccc(C)c2N)=O)CCOC2CN(C(=O)CC3CCC(O)C3)CC12 34748,c1(C(N2CC(C(C)C)N(C(C3CC(C)(F)C3)=O)CC2)=O)coc(S(C)(=O)=O)c1 34749,CCCCCC(C)CC(=O)NC1CCCC1NC(C1CC2(C1)OCCO2)=O 34750,C(CNC(c1cncs1)=O)(C(C)C(C)C)NC(c1c(C)cn(C)n1)=O 34751,C=CC1(C(=O)NC2CN(C(=O)Cc3ccn(C4CCCCC4)n3)C2)CCCCC1 34752,C1(NC(C(n2ccc(C3CC3)n2)C)=O)C2CC1CN(C(=O)CC1CCCO1)C2 34753,CC(C(C)(C)CN(C)C)CC1(N2CCOCC2)CC1.c12cn(nn1)C1CN(C1)C2=O 34754,C123CC1CN(C2)C(=O)Cn1cc(nn1)C3.C1(CCC)CCCC1NC(=O)C1CC1 34755,Cc1cccc(CCNC(=O)CC2CCCOC2)n1.ONC(=O)Cn1cnnn1 34756,c1(CNC(CCN(C(C(CSC)OC)=O)C)=O)ncc2ccccn12 34757,C12(CC(=O)NCCCNC(C3(C)CC(C#N)C3)=O)CC3CC(C1)CC(Cl)(C3)C2 34758,C(=O)(C(C)(C)C(F)F)NC1(CF)CCN(C(c2cn(CCOC)nn2)=O)C1 34759,C1(CNC(c2ocnc2C2CCC2)=O)CN(C(C2CNC(=O)C2)=O)CCO1 34760,c1(C(N2C(CNC(C3C(C)C3C)=O)C=CC2)=O)cn(C)nc1-c1nccs1 34761,CC(CC(=O)NCC(O)CNC(C1(F)CCCC1)=O)NC(=O)NC1CCCC1 34762,c1(C(=O)NCC(CNC(c2ccc(C(C)C)nc2)=O)(C)O)cc(CO)ccc1Cl 34763,N1(C(C(CCC)OC)=O)CCC(CO)(NC(=O)CCOc2ccc(F)cc2)CC1 34764,c1(CC)n[nH]cc1C(=O)NC1CCC(CCC(=O)NCc2ccco2)C1 34765,N1(C(CCCCC#C)=O)CC(C(=O)NCCC2NC(=O)NC2=O)CCC1(C)C 34766,C(CC1CCCC1)(C(=O)Nn1cnnc1)NC(CS(CC)=O)=O 34767,C(=O)(C1=C(C#N)CCC1)N1CCC(C(=O)NC(CCC)CC)C1CC 34768,c1(C(N(CCNC(c2c(C)noc2)=O)C)=O)cccc(CCNS(C)(=O)=O)c1 34769,C1(C(=O)NC(C2CCN(C)C2)C)(CO)CN(C(C2CCN(S(C)(=O)=O)C2)=O)C1 34770,c1(N(C2CCNCC2)CCCc2c(Br)cccc2)ncnc2c1CCCC2 34771,Cc1cc(C(=O)NCCC2CCCN(C(=O)Cc3cnc[nH]3)CC2)cc(F)c1C 34772,C#Cc1ccccc1CC(=O)N(CCN(C)C(C1SCCC1C)=O)C(C)C 34773,N1(C(C(=CC2CCCC2)C)=O)CC2(CC(NC(=O)C=CC=C(Cl)Cl)CO2)C1 34774,C1(C(N2C(CCN(C(=O)C#CC3CCC3)C)CCCC2)=O)CC2(CCC2=O)C1 34775,CCC(CC(=O)NCCCOCC(N1CC=CC1CN(C)C)=O)SC 34776,Cc1ccccc1CC(=O)NC(C(C(C)C)NC(=O)C=NOC)c1ccccc1 34777,CC(C)S(=O)(=O)C(C)C(=O)N1CC(O)(CCNC(=O)CCCCNC(N)=O)C1 34778,c1(C(=O)NCCCCNC(=O)C(c2ccccc2)F)cn(C2COC2)nn1 34779,c1(OC)cc(Cl)ncc1C(=O)Nc1c[nH]nc1C(=O)Nc1cc(I)ncn1 34780,CC1CC2CN(C(c3cccnc3O)=O)CC2N1C(=O)CCCC1CCCC1 34781,C1(CC(=O)NCCCCNC(C(Cc2ccccc2)OC)=O)CCC(=O)N1C 34782,N1(C(Cc2cc(C)on2)=O)CCCC(C)(CNC(=O)C(C2CCOCC2)C)C1 34783,c1(C(N(C)CC2CCCCN2C(=O)C=CC2CCCC2)=O)ccc2ccnn2c1 34784,CCC(F)(F)CC(=O)NCC(C)CN(C(=O)Cc1ccncc1Cl)C 34785,c1(C(=O)NC2CCCC(C(=O)Nc3cncs3)CC2)cccn2nccc12 34786,C1(n2cc(CC(C=C)O)nn2)CCN(C(=O)CN2CCC(C)C2)CC1 34787,C(=O)(C(C)(C)C(F)(F)F)N1CCC(CNc2c(Cl)ccc(OC)n2)C1 34788,c1(C(=O)NCCOC2CN(C(C3CC34CCCOC4)=O)C2)cn2cccnc2n1 34789,CCC(C)(C#N)C(=O)N1CC(NC(C2CC(n3cnnc3)C2)=O)C(C)(C)C1 34790,c1(SC)ccc(C(=O)NCCC2CCCCN2C(=O)C(Cl)=CCl)c(Cl)c1 34791,CCC(C)CCC(O)CC(=O)NC1(C)CN(C(=O)Cc2csc(COC)n2)C1 34792,N1(C(C(C)Sc2ccccc2)=O)CC(CNC(c2cnnc(O)c2)=O)CC1(C)C 34793,C1(N(C(c2c(C)cc(C#N)cn2)=O)C)CCCCC1S(C)(=O)=O 34794,c1(COC)ccc(C(=O)NC(C)CNC(C2(C(F)(F)F)COC2)=O)o1 34795,N1(C(c2cc(SC)oc2)=O)CCC2CN(C(c3[nH]cc(C)c3C)=O)C2C1 34796,Cc1nn(C)c(C)c1C(C)C(=O)NCC1CN(C(C2C3CCCCCC23)=O)C1 34797,Cc1nc(=NCCOCCNC(c2nn(-c3cnn(C)c3)nc2C)=O)[nH]cc1Br 34798,N1(C(CN(CCSC)C(C)C)=O)CCC1CC(=O)Nc1cnsc1 34799,c1(C(N(C)CCNC(=O)COc2nc(O)nc(O)n2)=O)ccc2[nH]ccc2c1F 34800,C(C(C)(C)CCC=C)N(CCCCCC=C)CC(C)CC 34801,C1(NCC(N2CCOCC2)=O)CC2(CCN(Cc3cnc4ccccn34)CC2)C1 34802,N(C1CN(C(=O)C(F)=C2CCC2)Cc2ccccc21)C(c1c(C)ccnn1)=O 34803,C1(N(C(c2cnoc2C2CC2)=O)CCSc2ccccc2)Cc2ccccc2C1 34804,O=C1CCN(C(C2C3CCC(C3)C2C(F)F)=O)c2ccccc21 34805,C1(C2CCN(C(=O)CC(C)CN(C)C)C2)(NC(CCSCC(C)C)=O)CC1 34806,C=CC(C)(CC)C(=O)NCCC(F)(F)Cn1cc(C2CC23CC3)nn1 34807,C(=O)(C1=NOC(C)(C)C1)N1CC(C#C)(C(N2CCC(OCC(N)=O)C2)=O)C1 34808,c1(C(=O)NCCCNCCC2CCC(C#N)C2)cc(F)cc([N+](=O)[O-])c1 34809,C1(C2CCN(C(c3c(C)cc(C)oc3=O)=O)CC2)(NC(CCCOC)=O)CCC1 34810,Cc1cc(C#N)nc(=NCC23CC(NC(=O)Cc4sccc4C)(CO2)C3)[nH]1 34811,c1(C(=O)NCC(CC)NC(c2ccc([N+](=O)[O-])s2)=O)cnc2c(c1)c(C)nn2C 34812,C1(C(N2CCC(C(C(N3CCCC(=C)C3)=O)F)C2)=O)CCCC1C1CC1 34813,Cc1[nH]c(C(=O)NC2CC2)c(C)c1C(N1CCC(Oc2cccc(F)c2)C1)=O 34814,C(=O)(CC(C)(C)OC)N(CCCNC(c1csc(-c2cn[nH]c2)n1)=O)CC 34815,C(=O)(C(C1CCCO1)NC(=O)CCc1ccsc1)N(C(COC)C)C 34816,Cc1cc(=O)n(CCC(=O)N2CC(OCCNC(=O)CC(C)F)C2)cn1 34817,CCCC(CNC(C1CCC2(CCC2)C1)=O)C(=O)N1CCCCC1CF 34818,c1(CN(C2C=CC(C=O)C2)C(=O)CSC)ccccc1.c1(C2C(CO)C2)cccs1 34819,C1(CNC(C(C#C)(C)C)=O)CN(C(=O)CCn2ccnc2)CC(C)(C)O1 34820,CCCC(C)CCCC(=O)Nc1cnc(Br)c(OCC)c1 34821,C1(N(C)C)(C(=O)NCC2CCC(NC(=O)Cc3sccc3Cl)C2)CCCOC1 34822,C(CC)(CCC(=O)N(C1CN(C)C1)C)NC(c1c(CC)ncnc1)=O 34823,c1(C(=O)NC2CC(CCNC(=O)CCOC(=O)NC3CC3)C2)occ2c1CCCC2 34824,c1(CC)noc(CC)c1CC(N1CC(NC(C2CCCCNC2)=O)C(O)C1)=O 34825,C1(NC(c2c(CC)ocn2)=O)CCC2CC1CN2c1snc(C)c1C#N 34826,Cc1nc(C(C)C)nc(N2CCCC(NC(c3ccnn3C(F)F)=O)C2C)c1F 34827,C1(NC(C(C2CC2)SC)=O)CCCC1NC(=O)Cn1ccc(Br)n1 34828,CC(C)CC(F)(F)C(=O)N1C2CCC1CC(NC(=O)COC1CCCCC1)C2 34829,C#CCC(C)(C(=O)N(C)CC1CCCS1)NC(c1cc(C#N)cs1)=O 34830,C1(C(N2C(C)CC2)=O)CCc2ncnc(C)c2C1.C1(N2CC(=O)N2)CCCC1.CC 34831,CCCCCCC(C)(CC)C(=O)NC1(C)CCCN(c2ncc(Cl)cn2)C1 34832,C(C(=O)N1CCC(C)C1)(C(C)C)N.C1(C(=O)OC)CC1C(=O)NCCOC(C)=O 34833,CC1=C(C(=O)N2CCC3(NC(c4cscc4C(F)(F)F)=O)CCCC23)CCCO1 34834,CC1C(NC(=O)C(C2CCOCC2)=O)CCCN1C(c1cn(C(F)F)cn1)=O 34835,C(=O)(CC1c2ccccc2C(=O)N1C)N1CC2C(NC(CSCC)=O)(CC2)C1 34836,Cc1ccc(C(F)(F)C(=O)NC2CC(C)N(C(=O)CC3(C)OCCO3)C2)cc1 34837,S(=O)(=O)(c1ccc(=NCCS(=O)(=O)N(C)C)[nH]c1)N(CCCC(C=C)(C)C)C 34838,c1(C(=O)NCC(CC=C)NC(=O)Cc2cnc[nH]2)cc(Cl)cc(Cl)c1Cl 34839,Cc1cc(C(N2CC(C)CCC2CNC(c2cn(C(C)C)nn2)=O)=O)c(C)nc1C 34840,C(C)(C(O)C(=O)NC1(CO)CN(Cc2ccc(C(=O)O)cn2)C1)OC 34841,C(=O)(C1=CCCC1C)N1CC2(C(C(=O)N(C(C)C3CC3)CC)C2)C1 34842,C12(C(=O)NC(C)C(=O)NC3CC3)COC(C1)C(NC(C1CC3(CC3)CO1)=O)C2 34843,CC1CCN(C(=O)C(F)(F)C(F)F)CCN1C(c1ccn2ccccc12)=O 34844,CC1CN(C(c2c[nH]c(C(N)=O)c2)=O)CC1NC(=O)CC12COCC(C1)C2 34845,C12(COC)CC(Nc3cccnc3SC(F)(F)F)(CN1C(=O)OC(C)(C)C)C2 34846,C12(CC(=O)NC(CNC(C#C)=O)C(C)(C)C)CC3CC(C1)CC(O)(C3)C2 34847,CCCC(C(=O)O)N(C1CCN(c2cccnc2)CC1)Cc1ccccc1 34848,c1(C(=O)NCCC(C)NC(=O)CCC2CCC(=O)NC2)c2c(nn1C)CCSC2 34849,c1(N(CC(O)CNC(=O)C=CC2CCCO2)C)cc(C2CC2)nc(Cl)n1 34850,c1(C(=O)NC(C(C)NC(CN(C(=O)OC)C)=O)C)cnc(CC(C)C)[nH]1 34851,C1(NC(CSCCOC)=O)CN(C(C23CC2CN(C(C)=O)C3)=O)C2(CCC2)C1 34852,Cc1cnc[nH]c1=NCCCCNC(C1CCCN(CCCO)C1)=O 34853,c1(N2C(C)CCN(C(=O)C(C)Cc3ccc(Cl)cc3)CC2)ncnc2sccc12 34854,C1(C(=O)NC(CCCCC)C)CN(C(C2(O)CCOCC2)=O)CC12CC2 34855,c1(CCC(=O)N(c2cccc(CCC)n2)C2CC3CC2CN3)ccc(F)c(F)c1 34856,N1(C(C2C(CN(C)C)C2)=O)CC2(C1)C(NC(=O)C=CCO)CCS2(=O)=O 34857,C=CCC(C)(C)CC(=O)NC1CCCC1NC(=O)C=C(C)C1CC1 34858,CCC(O)(CC(=O)NC1CC(O)CN(C(C2(O)CCOC2)=O)C1)c1ccccc1 34859,c1(OC)cc(Cl)cc(N)c1C(=O)N(CCO)CCc1scnc1C 34860,C1(C(N(C)Cc2ccns2)=O)CCC(C2CC2)N1C(c1ccc(C#N)s1)=O 34861,c1(C(N2CCC(C#N)CC2)C(=O)NCc2ccc(Cl)s2)ccc2ccccc2n1 34862,CCCCCC(O)C(=O)N(C)Cc1cn(-c2ccc(C#N)cc2)nn1 34863,C1(CCN(C(=O)CSC(F)(F)F)C)CCCCN1C(=O)CN1CCC(F)(F)C1 34864,c1(C(N2CCC(CCNC(C(C)CC(F)F)=O)C2)=O)cccc2c1CC(=O)N2C 34865,C1(N(C(CC(=O)NCC#C)=O)C)CCN(C(=O)C(C)CSC)CC1 34866,N1(C(CC2CN(C)C2)=O)CC2CC2(C(=O)N(C2CCCC(O)C2)C)C1 34867,c1(C(C)C)ccc(C(=O)Nc2cccc(NC(=O)CCC3CNC(=O)N3)c2)cn1 34868,Cc1oc(-c2ccccc2F)nc1C(=O)NCC(O)CN(C)C(c1cncs1)=O 34869,C(=O)(NNC(=O)Cc1ccccc1C(F)F)CCCCCC 34870,Cc1c(C(=O)NC2CCC23CN(C(=O)CC2CC24CC4)C3)cnc2c(Cl)cccc12 34871,N(C1CCCc2c1cnn2Cc1ccccc1)C(c1cc(C)c(O)c(C)c1)C 34872,C(=O)(C1CCc2ccccc21)NC1C(CNC(c2cnsn2)=O)COC1 34873,C(C(=O)N=c1cc(C2CC2)n(C)[nH]1)C1CN(C(CCC=C(C)C)=O)C(C)C1 34874,C1(NC(C2CCC(NC(CCC3C(C)C3)=O)C2)=O)CC2CC1CC21CC1 34875,C(CC(C)C(=O)NCC(O)CNC(c1ccnc(NC(=O)NC2CC2)c1)=O)=CC 34876,C(=O)(CC(C(F)(F)F)N1CCOCC1)N1CCC(F)(CN(C)C)C1 34877,O(NC(=O)COc1ccn(C)n1)CCO.C1(OC)CN(C(=O)C(C)SCCC(C)C)C1 34878,c1(C(N2C(CC(=O)Nc3c(C#N)ccs3)CCC2)=O)cccnc1[N+](=O)[O-] 34879,N1(C(C(=Cc2ccccc2)C)=O)CC2(CCC2)CC1C(N1CCC(C(C)C)C1)=O 34880,c1(NC(C2C(NC(c3nccc(Cl)c3F)=O)CCC2)=O)ncnc2cc(Br)sc12 34881,CCCC(C)CCCC(=O)NCC1CN(C(c2cc(Cl)ns2)=O)CC1(C)C 34882,CC1CN(C(=O)C(c2ccn(C)n2)C)CC(C)CN1C(C1CC12CC(O)C2)=O 34883,Cc1cc(C=CC(N2CC(NC(C3CC3(Cl)Cl)=O)C(C)(C)C2)=O)c[nH]c1=N 34884,C(CN=C(NCC1CC12CC(OC)C2)NC1CCN(C2CC2)CC1)OCC(=C)C 34885,c1(OC)ccc2ccccc2c1NC(C1CNCCN1Cc1csc(C)n1)=O 34886,C(C(=O)NCCSC1CC1)(C(C)CCC=C(C)C)N1CCC(OC)(CO)C1 34887,N12CCN(C(=O)C1)C1CCCN(C1)C(=O)CNCC(OC)C2=O.OC 34888,C12(C(=O)NCCNC(c3cccnc3)=O)CCC(O1)c1ccccc12 34889,C1(NC(C2C(C=C)C2)=O)CN(C(c2cc(C)n(CCN(C)C)n2)=O)CCC1CO 34890,N1(Cc2nc(-c3ccc(CC)cc3)on2)CCC(CC(N)=O)C(F)(F)C1 34891,c1(CC)cc(C(=O)NCC(C)CNC(c2cncc(N)n2)=O)cc(O)n1 34892,CCC(C)C(=O)C(=O)NC1COCCC1C(=O)N(CCC(N)=O)CC 34893,N1(C(CNC(C2C(C)C2)=O)=O)CCC(C(=O)NC2CCC2)(C(C)C)C1 34894,c1(C(=O)NCC2CN(C(c3c(COC)scc3)=O)C(C)C2)c(Cl)ccnc1C 34895,S(=O)(=O)(c1c[nH]c(=NCCC2CC2C2CC2)cc1C)N1CCC(N(CC)CC)CC1 34896,C12(C(=O)NC3C(OC)CN(C(C(CC=C)C)=O)C3)CC3(F)CC(F)(C1)CC(F)(C2)C3 34897,Cc1cc(C(N2CC(C(=O)N(CC(N3CCCCC3)C)C)C2)=O)cc(C(F)F)c1 34898,c1(C(C)NC(C2CCCOC2)C2CC2)c(F)cc(Cl)cc1Cl 34899,Cc1c(C2(C(=O)N(C(C)CN(C(=O)CSC3CC3)C)C)CC2)cccc1F 34900,c1(NC(C2(C)CN(C(=O)Cn3ccnc3)C2)=O)ccc(F)cc1I 34901,c1(Cn2cc(C(C)NC(C(C)CCN(C)C)=O)nn2)csc2ccccc12 34902,c1(C(=O)NC2CCCN(Cc3c(Cl)c(C)n(C)n3)CC2)cncc2c1CCCC2 34903,N(C(=NCCCF)NCC(C)(C)OC(F)F)C(C#C)Cc1ccccc1 34904,Cc1ccc2c(c1)C(=O)N(CC(=O)NCC1COCCN1C(=O)CN(C)C)C2=O 34905,N1(C(C2CC(=C)C2)=O)CC=C(C(=O)Nc2cccc(C#N)c2)C1 34906,n1(CCOC(C)C)nc(Cc2ccccc2Br)nc1-c1cncn1C1CC1 34907,N1(C(C(CCC)O)=O)CC(CNc2ncc([N+](=O)[O-])cn2)OC(C)(C)C1 34908,N1(C(c2ccc(CCC)cc2)=O)CCCC(C)(NC(C2CCC3CC2CO3)=O)C1 34909,CCCCC(O)CC(=O)N1CCC(C)C1C(=O)N(CCO)CC 34910,C1(NC(CC2CC(C)(C)OC2=O)=O)CN(C(c2ncccc2Cl)=O)C2(CCC2)C1 34911,Cc1noc(CN(C)C(=O)NCc2ccn(CC(F)(F)F)n2)n1 34912,C(CN=c1[nH]c(=NCCC2CC=CCC2)c2ncccc2[nH]1)N1CCC(C)CC1 34913,C(CCCC(=O)N1CC(O)CC1CN(C)C)NC(c1c(NC)scn1)=O 34914,C1(C(N2CC3C(CNC(C(CCC)C)=O)(C3)C2)=O)CC(C(C)C)=NO1 34915,C1(C(N(CC(C)(C)NC(COCCCC(C)C)=O)C)=O)CCCCC1(F)F 34916,N1(CC)CCC(CC(=O)NC2(CNC(c3nc(C)no3)=O)CCC2)C1 34917,N1(C(c2c(C)cc[nH]2)=O)CCC(C(C)(O)CNC(c2nocc2Br)=O)CC1 34918,c1(OC)nccc(C(N2CC(NC(c3nc(C)ncc3Br)=O)C(F)C2)=O)c1F 34919,CC1(C)OC2(CN=c3ccc(-c4nn[nH]n4)c[nH]3)CC1(C(N1CCSC1)=O)C2 34920,N1(C(C(=O)NC(CC)(C)C)C2CC2)CCC(CC2CC2)C(C(N)=O)C1 34921,C(=O)(CC(C)C(=O)OC)NC1(CNC(c2cc(CC)ncc2)=O)CCCO1 34922,c1(NC(c2nnnn2Cc2ccco2)(C)CC2CCOC2)ccccc1I 34923,c1(OC)cc(C(=O)NC2CC(NC(=O)C(OC)OC)C2)cc(C)c1 34924,C1(CNC(CCc2onc(C)n2)=O)CC(O)CN1C(c1cc(C(N)=O)cs1)=O 34925,C1(C)(C(=O)NCc2cn(CCN(C)C)nc2)CCCN1C(c1cnc(Cl)s1)=O 34926,c1(C(=O)NCC2C3CN(C(C4C(OCC)C4)=O)CC32)c(F)cc(F)cc1Cl 34927,N1(C(C(CSC)(C)C)=O)CCC(CNC(C2CCCC(C(F)(F)F)C2)=O)C(O)C1 34928,c1(CC(=O)NCC(CNC(C(C)SCCCC)=O)C)ccc(-n2ccnn2)cc1 34929,c1(C(=O)NCC2C3CCCC2N(c2ncnc(Cl)c2F)C3)cc2ccccc2o1 34930,CC1CCC=C1C(=O)N1CCC(C)(C)C1CC(=O)NOCCCF 34931,c1(-c2ccn(C)n2)cccc(C(=O)NCC2CCCN2Cc2ccsc2Br)c1O 34932,O=C(O)CCC(F)(F)C(=O)N1CC2CC1CN2Cc1ccc(F)cc1 34933,c1(NCCCN(C(=O)C(C)N2CCCC2)CC(C)C)cc(Cl)cc(Cl)c1 34934,N1(C(CCOCCC)=O)CCCC2CN(C(c3cncc(NCC)c3)=O)CCC12 34935,C=CCC(C)C(=O)N(C1CCCN(C(=O)C=C(CCC)CCC)C1)CCF 34936,C1(CNC(CC(=C)C)=O)CC(F)(F)CN1C(=O)CC(C)(C)COCc1ccccc1 34937,C1(C(=O)NCCOC2CCCC2)COCCN(C(C2(O)CCCC2)=O)C1 34938,C1(C(=O)NCC2N(C(c3c(OC)nsc3)=O)C3C(C2)C3)Cc2ccccc2S1 34939,C1(CN(C(C(C2CCCC2)NC(C(C)=C(C)C)=O)=O)C)C(C)(C)C1(C)C 34940,CC(C(=O)N1CCC(O)(C(C)CNC(=O)C(C)(C)CO)C1)C(F)F 34941,C(=O)(C(F)(F)C(C)O)N(c1cc(F)cc(Cl)c1)CCNC(Cc1c(C)ncs1)=O 34942,c1(-n2cc(C(CC)O)nn2)ccc(C(F)(F)F)cn1 34943,C=C=C(C)CC(=O)NC1(CC=C)CCN(C(c2cnn(C(C)CC)c2C)=O)C1 34944,C(CC(C)(C)C(=O)N(CC(N1CCOCC1)=O)C)NC(C=CC=CC)=O 34945,c1(OC(=O)NC2(C)CCN(C(CCCC(C)C)=O)CC2)cc(Cl)c(Cl)cc1C#N 34946,N1(C(CC2COC(=O)O2)=O)CC2CC(NC(=O)Cn3cc(CO)nn3)CC2C1 34947,c1(OC(C)C)ccc(CNC(c2ccnn2-c2c(F)cccc2F)=O)c(O)c1 34948,C1(C(N2C3CC(NC(=O)CC4CCC(F)(F)CC4)(C3)C2)=O)CCCCCC1(F)F 34949,N1(C(C2CC(C)SCC2)=O)CCN(C(=O)Cn2cccc2)CC1CO 34950,c1(NCc2cccc(OCCOC)c2)[nH]c(=NCC2CC2C)nc2ncn(C)c12 34951,c1(OCCCC)c(C(=O)N(CC(=O)O)Cc2cnc(C)nc2C)cccc1Br 34952,C(C)(CC(=O)NC1(CC(=O)NCC(C)(O)C2CC2)CCCC1)=C(C)C 34953,Cn1cncc1C1CC1NC(=O)CC1(C)CCN1C(=O)CSCC(F)F 34954,C1(OC)(CNC(C2CC=CCC2NC(=O)CCN=[N+]=[N-])=O)CCC(C)C1 34955,N1(C(CCOC(C)=O)=O)CCC(CN(C(=O)C(C(C)C)n2cncn2)C)CC1 34956,CN1N=CC(CC(=O)N(CC(CO)(CO)NC(=O)CC2CCCC(O)C2)C)C1=O 34957,CCC(CC)CCCC(=O)N1CCC2CN(C(c3nnn4ccccc34)=O)C2C1 34958,N1(C(c2cc(C(F)(F)F)cc(F)c2)=O)CCC(C)(CNC(C(C)C(F)F)=O)CC1 34959,Cc1ccc(CCCC(=O)NC2CCCC2CNC(=O)Cc2cncn2C)s1 34960,C1(C)(CNC(c2c(N(C)C)ccs2)=O)CCC(NC(C2CCS(=O)(=O)N2)=O)C1 34961,N1(C(c2c(C)noc2)=O)CCN(C(=O)CCn2cccn2)CC1CO 34962,C(=O)(C1=CS(=O)(=O)CCC1)NC1CN(C(C(C2CC2)OCC)=O)CC1(C)C 34963,CCC(C)CC(C)C(=O)N1CCC(F)(CNC(=O)CC2(CO)CC2)CC1 34964,c1(CC(=O)Nc2ccc3c(c2)OCCO3)noc2ccc(Cl)cc12 34965,N1(C(C2C(CCOC)C2)=O)CCCC1(C)C(=O)NCCC1(COC)CCC1 34966,C1(CNC(C2(C)CC2(F)F)=O)(CNC(C2(C)CCSCC2)=O)CC12CCC2 34967,c1(C(=O)NCCCN(C(=O)Cc2cc(C)ns2)CC)ccn(O)c(=O)c1 34968,C1(C)(C(=O)NC2CCC(NC(c3ccc(CC)[nH]3)=O)C2)CCC(C)(C)CC1 34969,C(=O)(C(CO)C(C)(C)C)NCc1c(C(=O)NCC(C(=O)NC)(C)C)occ1 34970,C1(NC(c2c(CC)n[nH]c2)=O)CCCN(C(=O)C(C2CCC(=O)N2)C)CC1 34971,c1(C(C(N2CC(n3cc(CSC)nn3)C2)=O)O)ccc(Br)cc1 34972,O=C(CCCC1CCC1)NC(c1ncccn1)C(N1CC(O)(c2nn[nH]n2)C1)=O 34973,c1(SCC(=O)NC2CCOC2)c[nH]c(C(=O)NC2CC2NC(C2CCCO2)=O)c1 34974,N1(C(c2ccc(C)cn2)=O)CC(C2CCCCN(C(c3nccnc3C)=O)C2)C1 34975,c1(C(=O)NCCC2CC(NC(c3cn(CCC)nc3C)=O)C2)nnc(O)cc1O 34976,N1(C(c2c(OC)ccc(Br)c2)=O)CC2(CN(C(=O)CCN3CCOCC3)CCO2)C1 34977,C(=O)(CCCCC(=O)NC1CN(C(=O)CSc2nnnn2C)CC(C)(C)C1)NC 34978,N1(C(C(C2CCCCC2)NC(C(C)SC2CCCC2)=O)=O)CCC2(CC(F)C2)C1 34979,N1(C(C2C3(CC(OCC)C3)C2)=O)CCC(O)(C(=O)NC)CC1 34980,CC(C)CCCOCC(=O)NCC(C)N(C(=O)CC1CCN(C)C1)C 34981,N1(C(c2cc(C)sn2)=O)C2CCC1CC(NC(c1nnccc1C)=O)C2 34982,C12(C(=O)NC3(CC)CCOC3)CC(CNC(CCOCC)=O)(C1)OC2C 34983,O=C(CCCCO)NCC(N1CC(O)(CNC(=O)CCc2cnn[nH]2)C1)=O 34984,c1(CC)oc2ccccc2c1C(=O)NCC(CCOC)NC(C1CC2CC1CO2)=O 34985,c1(OC)ccc2cccnc2c1CNc1cc(NC2CC2CC(C)C)ncn1 34986,c1(NC(CN(CCOC)Cc2ccc(Cl)s2)=O)nc2c(s1)CCCC2C(=O)OC 34987,CCCCCCC(C)C(=O)NCCC1CC(F)(F)CN1C(=O)C(F)C1CCC1 34988,C12(C(=O)NCC(=O)NC(C=C)C3CCC3)COCC1C2 34989,N1(C(=O)NC(c2ccncc2Cl)C)CCCCC1c1cccnc1 34990,C1(COC)COCC1NC(C1C(NC(=O)COc2cccnc2)C1(C)C)=O 34991,CN=c1ccc(C(=O)NCC2CCN(C(=O)C(C)(C)c3cscc3Cl)CC2)c[nH]1 34992,c1(OC)cc(C(C)C(N2CCCC(C)(NC(=O)CCCC3CC3)C2)=O)ccc1C 34993,C(=O)(C1=NOC(C)C1)NC1(CO)CN(C(CC(c2cccs2)NC(=O)OC)=O)C1 34994,N1(C(c2cccc(Cl)c2)=O)CC(C2CCCN(C(C3CCCCS3)=O)C2)C1 34995,c1(C(=O)NC(Cn2c(CC)ncc2)C)ccc(Br)cc1N=[N+]=[N-] 34996,c1(C(N2CC(C)(c3cn(C4C=CCCC4)nn3)C2)=O)ccc(C(O)CF)cc1 34997,C1(F)(C(NOCC2(C)CC2)=O)CN(C(c2cccnc2)=O)C1 34998,N1(C(C(C)SCCCC)=O)CC(NC(c2ncc(F)cc2C)=O)CCC(O)C1 34999,N1(C(c2c(C)nsc2)=O)CCCC2(NC(=O)CSC(C)(C)C)CCCC12 35000,N1(C(Cc2n[nH]c(=NC)s2)=O)CC=C(CNC(c2cc(OC)ccc2F)=O)CC1 35001,N1(C(COCC=C)=O)CC2CCC(C1CO)N2C(c1ccc2c(n1)CCC2)=O 35002,c1(CC)nc(C2CC2)[nH]c1C(=O)NC1CN(C(=O)CC2C=CCCC2)CC1O 35003,[N-]=[N+]=NCC(C(=O)NC1(C2CC2)CCC1)NC(C1CSC1)=O 35004,C12(NC(c3c(C)cccn3)=O)CCN(C(=O)COCc3ncnn3C)CCC1C2 35005,C#CCCC(C(=O)NCC(C)C#N)NC(=O)CCCCCN(C)C 35006,n1(CC)ccnc1C(=O)NCCc1n[nH]cc1C(=O)N(CCCn1ccnc1)C 35007,C1(NC(CC(C(C)C)C)=O)CCCC12CCN(C(=O)C(C)CS(C)(=O)=O)CC2 35008,c1(OC)ccc(Br)c(-c2cc(C(N3CC(=O)NCC3C(=O)N(C)C)=O)no2)c1 35009,C1(C(=O)NCc2cn(CCNC(C(C)N(C)C)=O)nn2)CC2CCC2C1 35010,c1(C(N2CC(C(C=O)O)C2)=O)c[nH]nc1[N+](=O)[O-].CC1CCCC1C(N1CCC1)=O 35011,C1(C)(C(=O)NCCC2(C(N(C3CC(OCC)C3)C)=O)CCC2)CC2CC2C1 35012,N1(C(C=C(CC)CC)=O)CC2(CC2)CC1CNC(=O)C(C)OCC(F)(F)F 35013,C(=O)(C(C)(C)CCOC)NC1CCCC(NC(C2(COC)CC(=C)C2)=O)C1 35014,Cn1ccc(C(N2CC(NC(=O)CCC(=O)N(C)C)CC2CO)=O)cc1=O 35015,C1(C(=O)NCCC2CCN(C(CC3C(C)C3)=O)CC2)CCOC2(CCOCC2)C1 35016,CC1(C)CC(O)(CC(N2CC(CNC(=O)CCC3CCOC3)C(C)(C)C2)=O)CO1 35017,C1(C(=O)NCc2cc(C(=O)N(C)CC3CCN(C)C3)n[nH]2)(OC)CCC(C)C1 35018,Cc1cc(F)c(C(N2CC3CN(Cc4cncc(C)n4)C3C2)=O)c(F)c1 35019,Cn1nc(C(=O)NC2CCCC2NC(C2CCC3CC23)=O)c2c1CCC(C)(C)C2 35020,N1(C(C(CC)C)=O)CC2CCC(C(=O)NCCc3ncn(C)n3)(C2)C1 35021,Cc1nccc(C(=O)NCC2(NC(=O)CNC(C3CCCCC3)=O)CCOC2)c1O 35022,N1(C(Cc2ccc(C)o2)=O)C2CCC1CC(CNC(=O)C(C)CCO)C2 35023,c1(Cn2cnc(NC(CC(c3c(C)n[nH]c3C)C)=O)n2)c(F)cccc1Cl 35024,S(C1CCc2c(F)cc(F)cc21)N1CCC(c2cccc(C)c2)(F)C1.CC(=O)O 35025,C1(OCC)CC2(CCC(C(N3CC4CCN(C(c5cnsn5)=O)C4C3)=O)CC2)C1 35026,C(CC(C(=O)N1CCC(OCC2CC2)C1)NC(c1cc[nH]c1CCC)=O)=CC 35027,CCCCCC(C)CC(=O)NC(CN(C(=O)CN1C(=O)C(C)C(C)C1=O)C)CC 35028,CCC(C)C(O)C(C)C(=O)N1CCC(N=[N+]=[N-])(C(N2CCC3CCCC23C)=O)C1 35029,CCC(C)(C)C(C)CC(=O)NC1(CNC(=O)C=Cc2cc(Cl)ccc2Cl)CCC1 35030,C1(CNC(C2CCC(CC)O2)=O)CC(NC(c2cnc[nH]2)=O)CC1O 35031,N1(C(C2C(C)(C)CO2)=O)CC2CN(C(c3cccc4c3COC4)=O)CC2C1 35032,N1(C(CC(COC)C)=O)CCCCC(CNC(=O)C=C2CCC(C)(C)CC2)C1 35033,N1(C(CCC(=O)NC)=O)CC(NC(=O)C(C)OC)CCC1C 35034,CCCCCCC(F)C(=O)NCC12COC(CNC(=O)CC(C)F)(C1)C2 35035,c1(C(=O)NCC2N(C)CCN(C(c3ccsc3)=O)C2)cnn2ccn(C)c12 35036,C=CCCCCC(=O)N1CCC(OCC(=O)NC(CCF)C(=O)OC)C1 35037,C=CCC(CC)C(=O)NC1CCCCC1C(N1CC(O)(COC)C1)=O 35038,c1(C(N2CCN(S(=O)(=O)C3CC3)C3CC23)=O)cc(C(F)(F)F)ccc1F 35039,Cn1nnc2c(NC3C(C)C(O)C3)ncnc12.c1(C)ccc(F)cn1 35040,CC1CCN(CCCOCCCCCCCNC(c2[nH]ccc2C2CC2)=O)CC1 35041,CCC(CCCC(=O)N1CCCCC1C)NC(=O)C(C)(C)c1ccno1 35042,Cc1nn(C)c(C)c1CCCNC1CC1Nc1nccc(Oc2ccccc2)n1 35043,N(C(=NCC1CCSC1)NCC(F)F)CC(CC)Oc1ccc(C)cc1 35044,CC(C)CC(CNC(=O)C1=CCCCO1)C(=O)NC(C1(O)CCCC1)(C)C 35045,S(=O)(=O)(c1cc(C(=O)NCC(C)N(C(=O)Cc2cn3ccsc3n2)C)co1)NC 35046,c1(-c2cccnc2)ccc(C(=O)NCC2(O)CC(NC(C(F)OC)=O)C2)c(C)c1 35047,C1(C(N(CCN(C(C(C(=O)OC)(C)CC)=O)C)C)=O)CCc2ncnc(C)c2C1 35048,C1(C(=O)NCCOCCC(=O)N(CCC#C)CCO)C(C)(C)C1(F)F.CCOC 35049,C(C)(C)(CC(=O)N1CCSCC1CO)N(C(C1(C(=O)OCC)CC1)=O)C 35050,CC1CCC(CNC(=O)Cc2cc[nH]c2)N(C(=O)CN2CCC(CO)CC2)C1 35051,Cc1cccc(-c2cccc(NC(C3CC(C)N(c4ncns4)C3)=O)c2)c1 35052,c1(C(=O)OC)cc(C(=O)NCc2ccc(CNC(C3OCCO3)=O)cc2)n(C)n1 35053,C12(C(=O)NC3CN(C(COCc4onc(C)n4)=O)C(C)C3)CCCN(CCC1)C2 35054,c1(C(N2C3(CN(C(C4CC4Cl)=O)C3)CC2)=O)ccc(Cl)c(F)c1F 35055,c1(OCC(=O)NC2CC2CNC(=O)CSCCC(F)(F)F)ccc(Br)cc1 35056,C1(CC(NCP(OCC)(C)=O)=O)CN(C(c2ccnc(COC)c2)=O)CC12CC2 35057,N1(C(Cc2cc(C)ncc2)=O)CC2CN(Cc3ccc(Cl)cc3F)C2C1 35058,N1(C(C(CO)N(C)C)=O)CCC2(C1)CN(C(=O)CS(=O)(=O)C(C)(C)C)CCO2 35059,N1(C(C2C=C(C)CS2)=O)CC2CC1C2NC(c1cccc(C2(C)CC2)c1)=O 35060,c1(NC(CNC(c2cc(C)nc(C)c2)=O)C2CC2)cc(C(C)C)n2ncnc2n1 35061,N1(Cc2c(OC)cco2)CCCC(NC(c2cnc(Cl)cc2I)=O)CC1 35062,C(=O)(C(C)(C)CC(F)F)NCc1c(C(=O)NCC(C#C)OC)con1 35063,c1(SC)ccccn1.c1(N2CCC(=O)N(C)C3CCN(C3)C2=O)ccccn1 35064,C(=O)(C(O)C(F)(F)F)N1CCC(CC2N(C(=O)CSC(F)F)CCC2)CC1 35065,c1(N2C(CNC(c3c(CC)nns3)=O)CCC2)ncnc2cccc([N+](=O)[O-])c12 35066,c1(C(N2C(CNC(CSCC)=O)CC(C)CC2)=O)n[nH]c2cc(C)ccc12 35067,N1(C(C2(COC)CCC2)=O)CC2CCC1C2NC(=O)CCc1ccc(Cl)cc1 35068,C1(C(=O)OCC)CN(C(=O)C(C)N(C)C(c2occc2C)=O)C(C)(C)C1 35069,C1(NC(CCC(C)O)=O)CN(C(c2cnc(N)c(N)c2)=O)CC12CCC2 35070,C(C1OCc2ccccc21)N(C(c1ccn(C(CC)CC)n1)=O)C(C)C 35071,C1(NC(CCCCN(C(C)=O)C)=O)CC2(C1)CN(C(=O)CC1C(CO)C1(C)C)C2 35072,C1(C)(CCCC)CCC(NC(C2CC3CC2N(C(C2CC(OC)C2)=O)C3)=O)CC1 35073,C1(NC(C2C(C)CCS2)=O)CCC(NC(=O)C(C)(C)c2ccc(Cl)s2)CC1 35074,c1(NC(C2(C)CCN(Cc3c(O)cccc3O)C2)=O)cccc2sccc12 35075,N1(C(C(C)=CC2CC2)=O)CCCC(NC(=O)Cc2csc(S)n2)C(F)C1 35076,N1(C(C(C(CC)C)O)=O)CCCC2(C1)CN(C(c1nc(O)[nH]c(=O)n1)=O)CCO2 35077,c12cc[nH]c1C(=O)NC2.C1(O)(OCC)CC(CNC(=O)CNC(=O)CSC)C1 35078,C(c1cccc(O)c1)=CC(N1CC2C(C1)N2C=O)=O.c1(SCO)cccnc1C(F)(F)F 35079,c1(CC(=O)Cc2cn(CC3CCO3)nn2)sccc1Cl.N12CCCC1C2=O 35080,N1(C(C(c2ccc(Cl)s2)C)=O)CCC(NC(=O)Cc2ccc(O)c(Cl)c2)CC1C 35081,Cc1cc(C)n(CC(=O)N(C)CC2COCCN2C(=O)C(C2CCCCC2)O)n1 35082,c1(CCN=C(NCC(=O)NC2CCCO2)NC2CCCCC2C)ccc(S(N)(=O)=O)cc1 35083,c1(C(N2CC3(CN(C(c4ccc(C)s4)=O)C3)C2)=O)cc(N)cc(C)c1F 35084,c1(-c2onc(CCCOc3ccc(Br)cc3)n2)cccc2ncsc12 35085,CCC(C(=O)NC1CC(N(C(=O)COCc2nccs2)C)C1)C(F)(F)F 35086,CN1CCN(C(C2CC(O)CN2C(=O)C(F)C(C)(F)F)=O)CC12CCC2 35087,N1(S(CCOC)(=O)=O)CCC2CN(C(c3cn4cccnc4n3)=O)CC12 35088,C1(NC(C(c2ccc(F)cc2)OC)=O)CC12CC(NC(c1ccncc1F)=O)C2 35089,c1(SC(C)C)nnc(NC(=O)CC2CNC2)s1.C1(C2CCN2C(=O)N)CCOCC1 35090,C(=O)(C(CC(N)=O)NC1CCCC1)NC1C(CC)N(C(=O)OC(C)(C)C)CC1 35091,c1(OCC)ccc(C(c2nnnn2C)NC(CCO)CC(C)C)cc1OCC 35092,C1N=C2C=C(N=CN2)NCC12CC=CC2.CC(C(C)(C)C)=C1CCSCC1 35093,C(=O)(CCCCNC(N)=O)NCC1(F)CC(NC(CC2(C=C)CC2)=O)C1 35094,CCCC(C(O)C(=O)NCC1CCC=CO1)NC(c1n[nH]c2c1CCC2)=O 35095,N1(C(c2nc(C(C)C)sc2)=O)CC(NC(C2(C(F)(F)F)CC2)=O)CC1C 35096,N1(C(C(CC)C#N)=O)CC(O)(C2CCN(C(=O)Cc3cn4ccsc4n3)CC2)C1 35097,CC(C)(C(=O)NCC1CC(NC(=O)Cc2ccno2)C1)C(F)(F)F 35098,N1(C(C2N(C(C3CC(=O)NC3)=O)CC2)=O)CCOCC(CO)C1 35099,c1(NC(C2CC(n3cc(CNC4C(C)CCCC4)nn3)C2)=O)cc2sccc2s1 35100,C(C)(C)(CCCC(=O)NC(C(C)C)C1CC1)NC(c1ccc(OC)cc1)=O 35101,c1(NC(C2C3CN(C(C4CCC(C)CO4)=O)CC32)=O)nc2cc(F)ccc2s1 35102,C12CCCCCCN1C(=O)NCCC2.c1(CN(C)C)c(O)cccc1Br 35103,N1(C(c2onc3ccccc23)=O)CC2CC(C1)N(NC(=O)Cc1ccccc1)C2 35104,C1(C(=O)NCc2nocc2C(=O)NCc2cccc(F)c2)CCCCC1O 35105,C12(CC(=O)Nc3ncc(C(C)=O)s3)CCC1CN(C(c1cc3occc3[nH]1)=O)C2 35106,C12(NC(C3CNC(=O)N3)=O)CCC(C1)N(C(=O)CCCCNC(=O)C1CC1)C2 35107,c1(SCCC(=O)NCCNC(C(C)NC(=O)OC)=O)ccccn1 35108,C(CC(=O)N1CCC(NC(c2nc(Br)sc2C)=O)C1)(C(F)(F)F)OC 35109,Cc1cc(C(=O)NCCN(C(=O)C(c2ccc(Cl)cc2)C)C)c(C)nn1 35110,C1(C(=O)NC(CCCCNC(C2(C(=O)NC)CC2)=O)C)COc2cc(O)ccc2C1 35111,N1(CC(=O)NC(C)CN(C(=O)CCc2cscc2Br)C)CCCCCC1 35112,N1(C(c2c(C)nc(CCC)o2)=O)CCC(NC(=O)C(C)NC(=O)NC)C(CC)C1 35113,c1(C(=O)NC(C(C)C)CCNC(=O)C(C)SC(F)(F)F)ccccc1[N+](=O)[O-] 35114,Cc1cc(Br)ccc1C(C)NCC1CC2CC2N1C(=O)OC(C)(C)C 35115,c1(NC)ccc(C(N2CCCC2(C)CNC(c2cnc(Cl)cc2N)=O)=O)c(F)c1 35116,c1(C(N2C3CN(C(=O)Cc4c(F)cccc4F)CC32)=O)cccc2c1OCO2 35117,c1(C(=O)NCC(CC)NC(C2CC(N(C)CC)C2)=O)cc(C#N)cs1 35118,c1(OC)cc(CNC(=O)C(c2cn(C)nn2)NC(=O)C=C(C)C(C)(C)C)[nH]n1 35119,c1(OC)ccc(S(=O)(=O)Nc2n[nH]c(-n3nc(C)cc3C)n2)cc1 35120,C12(CNC(C(n3ncc(C)c3)C)=O)CCC(CN(C(c3cnnc(C)c3)=O)C1)C2 35121,C1(C(N(CCCOCCNC(COCC#C)=O)C)=O)COc2cc(O)ccc2C1 35122,CC1CNc2c(-c3nc(CCC4CC4)nn3CCc3cccs3)cnn2C1 35123,C1(N(C2CCOC2C)C(c2cccc(OC(C)=O)c2)=O)CCNCC12CC2 35124,C(C1CN(C(=O)CCN(c2ccncc2)C)CC1C(=O)N(C)CCO)=CC 35125,c1(OCC(=O)NCC(CC)(C)OC(=O)C(n2nccc2C)C)ccccc1F 35126,N1(c2c(C(C)=O)cccn2)CCC(NC(=O)C(C)n2cnnn2)C(O)C1 35127,Cn1nc(C(N2CCOC(CCCNC(=O)COCC3CCCC3)C2)=O)cc1Cl 35128,c1(CCC)cc(CNC(C2CC(OC)C(n3ccnn3)C2)=O)n(C)n1 35129,C1(CC#C)(C(=O)N(C)CC2CCOCC2)CCN(C(=O)CCc2conc2C)C1 35130,C1(CN(C(C=Cc2c(C)ccs2)=O)C)CN(C(c2ns[nH]c2=O)=O)CC12CC2 35131,N1(C(c2c(CC)ncs2)=O)C(CNC(c2cc(C(F)F)on2)=O)CC2CC12 35132,C(=O)(C1CCCc2cn(C(C)(C)C)nc21)NCCCCOc1cc(C)cc(C)c1 35133,c1(OC)ccc(C(C)=CC(=O)NC2CCC2NC(c2csc(CO)n2)=O)cc1 35134,CC(C)C(C(=O)NC1CN(C)CCN(C)C1)C(C)NC(C1CC=CC1)=O 35135,c1(C(=O)NCC2CCCCN(C(C(CCCC)C)=O)C2)csc2cccc(F)c12 35136,C1(NC(CCC(=O)NC)=O)(CNC(c2cccnc2F)=O)CCCCC1C 35137,N1(C(C2CCCSC2)=O)CCCCC2(CCN(C(C3CC3C(F)(F)F)=O)C2)C1 35138,c1(C(=O)NC2C(CNC(=O)Cn3cnnc3O)C2)cc2ccc(Cl)c(F)c2[nH]1 35139,c1(CN(C(C2N(C(C)C)CCC2)=O)CCOCc2cn[nH]c2)ccc(Cl)cc1 35140,Cc1ccc(S(=O)(=O)N)cc1C.C(Cc1ccncn1)(C(=O)O)CC(=O)NC 35141,C1(CNC(c2cnn(C)n2)=O)C(C2CC2)CCN1c1ncnc(Cl)c1C(C)(C)O 35142,CC1(C)C(CC(=O)NCC2COCCO2)CCN1C(C1CCCCCC1)=O 35143,C(C(C(=O)NCC)N(C)C(C1CC(NC)C1)=O)O.C1(C(=O)OC)(CSC)CC1 35144,N1(C(C2N(CC)CCCC2)=O)CC2CCN(C(c3ccnn(C)c3=O)=O)C2C1 35145,c1(C(N(CCOC)CCNC(C2CCCCS2)=O)=O)ccc(C(=O)C2CC2)cc1 35146,c1(C(=O)NCC2(O)CN(C(C3(C(C)C)CNC(=O)C3)=O)C2)nn(C)c(Cl)c1Cl 35147,c1(NCC2CN(C(C3(C=C)CCC3)=O)CC2C)ncnc2c1nnn2C 35148,CON(CCC(=O)NCCc1ncc[nH]1)C(=O)C1=CCCC1C 35149,N1(C(c2cn(C(C)C)nn2)=O)CCOC(C(=O)NCCCC2CCC3CC23)C1 35150,c1(C(N2C(C)CCC(NC(c3cn(CC=C)nn3)=O)C2)=O)cnc(O)n(C)c1=O 35151,O=C(C1=CCCSC1)NC1CCN(C(=O)C(O)CCn2cncn2)CC1 35152,C12(C(=O)NC(CN(C(=O)C(C)C3CCC3)CC)C)CC3CC(C1)CC(F)(C3)C2 35153,Cc1c(C(=O)N(C)CCC2CCCCN2C(=O)C#CC2CC2)cccc1CO 35154,c1(C(=O)NC(CCCC)CNC(c2ccco2)=O)cccc(OC)c1OC 35155,C(CC(=O)NCC(C1CCCC1)NC(C1CC1OC(C)(C)C)=O)N(C)C 35156,c1(C(=O)NCCC(=C)CNC(c2cc(Br)c(C)o2)=O)cccc(C(C)C)n1 35157,c1(NC(=O)NC(c2ccc(C#N)s2)C)cn(CCO)nc1C1CC1 35158,C12(NC(c3c(C)cncc3)=O)CC(CNC(C3C=CCC3)=O)(C1)OC2C 35159,C(=O)(C1=NOC2COCC12)N1C(C)CN(C(C(C)=NOCC#N)=O)C(C)C1 35160,Cc1ccc(NNC(=O)CNC(C2CCC(C(F)(F)F)CC2)=O)cn1 35161,N1(C(c2ccc(NC(C)=O)nc2)=O)C2CCC1CN(C(=O)COC1(C)CCC1)C2 35162,c1(C(N2C(CN(C(=O)COC)CC)CCC2)=O)ccc(F)c2ccncc12 35163,C=CC(C)(O)CC(=O)NC1C2CC(NC(=O)CCc3nc(=N)[nH][nH]3)CC12 35164,C1(CC(N)=O)CCCCN1C(=O)C(N1CCC(CCS)CC1)=O.n1(CCO)cncn1 35165,c1(C(=O)NC(CNC(C2(C)CCC(C)C2)=O)C)cnn2ccccc12 35166,C1(C(N(CC(CCC)C)C)=O)CC12CCN(C(c1n[nH]c(=N)[nH]1)=O)C2 35167,c1(C(=O)NCC2CCCN(C(c3ncncc3Br)=O)C2)cncc2c[nH]nc12 35168,N1(Cc2cn(CC(C)NC(c3ccc(=N)[nH]n3)=O)nn2)CCCS1(=O)=O 35169,CC1(F)CCC(C(=O)NC2CCCC2NC(c2ccc([N+](=O)[O-])o2)=O)CC1 35170,CC1(C)CCC(c2ccccc2)N(C2CCSC2)C1 35171,c1(C(=O)NCC2N(C(CN(S(CC)(=O)=O)C)=O)CC(O)C2)cccc(F)c1C 35172,CC(C)(C)C(O)C(=O)NCC1CN(C(c2ccnc(CC(N)=O)n2)=O)CC1(C)C 35173,Cn1nc(C(=O)NC2CCC(NC(c3coc(CC4CC4)n3)=O)C2)cc1C#N 35174,N1(C(C2(CC)CC2)=O)Cc2cccc(CNC(=O)Cc3cn[nH]c3)c2C1 35175,c1(OC)ccc(S(=O)(=O)N2CC3CC2CN3C(c2ccc(Br)c(F)c2)=O)cn1 35176,N#Cc1ccc(CNC(=O)Cc2ccccc2CC(N)=O)nc1 35177,CC(CCCNC(c1ncsc1-c1ccccn1)=O)NC(c1ccco1)=O 35178,Cc1nc2cc(C(N3CC(NC(C4CNC(=O)N4)=O)C3)=O)ccc2n(C)c1=O 35179,CSC1=C(C(=O)NCC2(CNC(=O)C(CO)NC(=O)C(C)C)CCC2)CCCC1 35180,C1(C(=O)N(CCNC(c2c[nH]cc2C2CC2)=O)C2CC2)(COC)CC1(F)F 35181,C1(NC(N2CC=C(C(=O)OC)CC2)=O)CCN(C)C2(CCCC2)C1 35182,C1(NC(C(CC)NS(CCC)(=O)=O)=O)CCN(C(=O)CC2(CSC)CC2)C1C 35183,c1(C(=O)OC)c(OCC)cc(NC(=O)NC2CN(C(=O)C3CC3)C2)cc1I 35184,CCCCS(=O)(=O)N(C(C)C(=O)NCC12CC1CN(C(=O)CSC)C2)C 35185,C1(C(N2CC(C=O)C2)=O)C2CCC(=O)C12.C1(OCCSCC)CN(CC)C1 35186,c1(CC)onc(C)c1C(=O)N(CC(=O)O)CCNC1CN(CC(C)O)C1 35187,C12(C(=O)NCC(C)(C)CNC(C3(c4cccs4)CCCC3)=O)CC=CC(C1)OC2 35188,C=Cn1nccc1C(N1CCCCC1CN(C(c1cncnc1C)=O)CC)=O 35189,c12ccccc1S2.O=C(O)CC(C)C1CCCCC1.c12nc(cs1)CC(=O)N2 35190,Cc1ncncc1C(=O)NCCn1cc(CNC(C2CC2(F)Cl)=O)nn1 35191,N1(CCNC(c2c(C)occ2)=O)CCC(NC(c2c[nH]c(=S)cn2)=O)CC1 35192,C1(NC(C(C)C2(O)CCC2)=O)CCCCCC1NC(c1cc(F)cc(Cl)c1)=O 35193,CC1CC(C(=O)N(C)CCOCCN(C(=O)CSc2nc[nH]n2)C)=NO1 35194,C(CCNC(=O)CO)(C(C)(C)C)N(C(CN(C)CCO)=O)C.N12CC(C1)OCC2=O 35195,C1(CC(=O)NC(Cc2cc(C)[nH]n2)C)C2CCCC2N1C(c1cnc(O)o1)=O 35196,CC1(CNC(=O)C=Cc2ccco2)CN(C(=O)CCN2CCC(F)C2)CCO1 35197,C(=O)(C#CC(C)(C)CNC(C1(C)CC1(F)F)=O)NC1C(C)COC1 35198,CCCN=c1[nH]c2c(c(=NC(C)c3ccc(Cl)nc3)[nH]1)CSC2 35199,c1(C(=O)NC2C(NC(=O)Cc3ccnnc3O)CCCC2)ccc([N+](=O)[O-])o1 35200,N1(C(C2C(C(=O)OC)COC2)=O)CCN(C(c2cc(=O)c(OC)c[nH]2)=O)CC(O)C1 35201,N1(C(C)=O)CCC2(CC1)CC(Sc1nnnn1C1CC1)CO2.C1(=O)CN1C1CC1 35202,CCC(CC(=O)NCCCCc1cnc[nH]1)NC(=O)CN(C(=O)C(C)C)C 35203,C(=O)(C(C(C)OC(C)(C)C)N(C)C)NCCCC1N(C(CCC=CC)=O)CCC1 35204,C(C(C)(CSC)CO)NCc1nnnn1C.c1(CC)cnc(CC(C)C)[nH]1 35205,c1(C2C(CNC(C(N3C(CC)CC3)=O)=O)C2)ccc(Cl)cc1Cl 35206,C1(C(N2CCC(CNC(CCC(=C)C)=O)C23CC3)=O)COc2cc(F)ccc2C1 35207,N1(C(c2cc(OCC)cc(F)c2)=O)CC2(CC(NC(=O)Cc3ccsc3)CO2)C1 35208,c1(C(N2CCC(N(S(CC(=O)OC)(=O)=O)CCO)CC2)=O)ccc2nccn2c1 35209,C1(CN)CC(C(F)(F)F)CN(C(c2ccc(Br)o2)C(=O)NCc2ccccc2)C1 35210,c1(C(=O)NCCC2(O)CN(C(C(COC)O)=O)C2)cccc2c1CNC2=O 35211,c1(NC2CCN(C(CC3C(=O)NC(=O)N3)=O)C2)ncnc2c1CCC2 35212,CC1C2C(CCN2C(=O)CN(C)C2CC2)CN1C(=O)CN1CCCCCC1=O 35213,c1(C(N2CC(C=C)(CC(=O)NCCOC3CCOC3)C2)=O)ccc([N+](=O)[O-])[nH]1 35214,C1(C(N(CC(C)NC(=O)CC2(c3cccc(F)c3)CC2)C)=O)CCCC(=O)N1C 35215,C(=O)(C1=CC2CCCCC12)NC1C(SC)CN(C(c2n[nH]c(C)c2Cl)=O)C1 35216,c1(NC(C2N(C(C3CN(C)C3)=O)CCC2O)=O)ccc(C(=O)N(C)C)c(F)c1 35217,N1(C(Cc2c(C)nc(C)s2)=O)CC2CCC(C1)N2C(C1(Br)CC1)=O 35218,C1(C(=O)NC2(C(=O)NC3CCCN(C(=O)OC)C3)CCCC2)CCC12CCOCC2 35219,C(=O)(C1CCCn2cnnc21)NCC(C)(Cn1cccn1)NC(CC(C)C)=O 35220,C(=O)(C1CCCc2sccc21)NCC(CNC(c1c(CC)cccc1CC)=O)C 35221,N1(C(CC=C)=O)CC(C)(C)CC1CC(=O)NC(C)C(O)C(F)F 35222,N1(C(CC2C(=O)NC(=N)S2)=O)CC(NC(c2coc(O)n2)=O)C2(CCOCC2)C1 35223,C1(C(N2C(CC(=O)N(C3CCOC3)CC)CCC2)=O)CCCS1(=O)=O 35224,C1(N(C)C(C2(C)CC3CC3C2)=O)CCCN(Cc2ccc(CN(C)C)cc2)CC1 35225,c1(NC(C2SCCN(Cc3c(Br)cn(C)n3)C2)=O)n[nH]c2c1CS(=O)(=O)C2 35226,N1(C(c2ncc(CC)s2)=O)CC(CCNC(c2cncnc2)=O)OC(C)C1 35227,C(C(C(F)(F)F)N1CCN(C(=O)CCc2ccsc2)CC1)NC(COCC#C)=O 35228,c1(C(=O)NC(CNC(=O)CCF)C2CCC2)coc(Cl)c1.c1(C)ccc(Cl)s1 35229,C1(CCNC(C2(C)C(C(=O)OC)CC2)=O)CCN(C(C2OCCC2(C)C)=O)CC1 35230,c1(C(=O)NCCC(C)NC(c2ccc(Cl)o2)=O)oc2ccccc2c1CS(C)=O 35231,C(=O)(CCCCCNC(C12C=CC(CC1)C2)=O)NCc1c(C)cc(C)s1 35232,C1(C(=O)NCC(C(C)C)NC(c2cn3c(n2)SCC3)=O)CCC(S(C)(=O)=O)CC1 35233,C1(=O)C(F)CC2CN(C2)C(=O)O1.C(=O)(C(Cc1cccnc1)NC(C)(C)C)OC 35234,c1(NC(=O)C(C)OC2CCCC2)cccc(C(N(CC(C)O)CCO)=O)c1 35235,C(=O)(CC(O)C(C)(C)C)NC1CCC(NC(CC2ON=C(C)C2)=O)CC1 35236,CCCCC(C(=O)NCC=C(C)C)NC(=O)CCC(N)=O 35237,c1(N(C(c2ccn(C)c2)C(=O)NCCSC)C)nnc(C2CC2)n1C 35238,c1(C(N2CCCC(CC(=O)Nc3nccc(C)c3)C2)=O)cc(Br)cnc1O 35239,c1(C(=O)NC2CN(C(C3(O)CCOC3)=O)CC2O)cc(F)cc(Cl)c1 35240,N1(C(C(C2CCCC2)SC)=O)CCN(CCN(C(=O)C=C(C)C2CC2)C)CC1 35241,c1(C(N2CCCCC(NC(=O)Cc3cn[nH]c3)CC2)=O)cccc2nsnc12 35242,C(=O)(C1=C(Cl)CCC1)NCc1c(C(=O)NC(C)C(C)CO)nco1 35243,c1(C(=O)NCc2n(CC)nnn2)ccc2c(c1)COCO2 35244,CCCC(C)(O)CC(=O)N1C2CCC(C2)C1C(=O)NCCCc1ccccc1 35245,N1(C(C(C)(C)C(N)=O)=O)CCOCC2(COCCN2C(=O)C2=CC3CCCC23)C1 35246,c1(CC)ccc(C(=O)NC2CCC(NC(C3(F)CCC3)=O)C2)[nH]1 35247,C(C(CC(C)(C)C(=O)OC)Oc1ccc(Oc2cc(C)cc(C)c2)cc1)OC 35248,C12(CNC(C(C(C)C)C)=O)CCC(CN(C(=O)CCc3nccs3)C1)C2 35249,Cc1[nH]c(C#N)cc1C(=O)NCC1C(C)CCCN1C(C1CCCC1O)=O 35250,C1(S(N)(=O)=O)(C(=O)NCC2(O)CN(C(C3N(C(C(N)=O)=O)CCC3)=O)C2)CCCC1 35251,c1(OC)cnc(F)cc1C(=O)NC(CNC(=O)C=Cc1cccnc1)CO 35252,Cc1cccc(C(N2CC(CC(C)NC(=O)COC3(C)CCC3)C2)=O)c1Cl 35253,C(=O)(C1=NOC2(CCC2)C1)N1CCC(NC(c2cc(OC)nn2C)=O)C1 35254,N1(C(C(C)n2cnnn2)=O)CCN(C(=O)C#CC2CC2)C(CC(F)F)C1 35255,c1(C(N(CC(CC)NC(c2ccc(F)nc2)=O)C)=O)cncc2cccnc12 35256,C1(C(=O)NCC2(NC(c3cc[nH]c3)=O)CCC2)CC12CCSCC2 35257,C(=O)(C(O)C(C)OC)N(C1CCN(C(C2(CF)CCC2)=O)CC1)CCC 35258,c1(CNC(C2CC2C(=O)NCc2ncc[nH]2)=O)ccc(S(=O)(=O)N2CCCC2)o1 35259,C#CC1(O)CN(C(c2ncoc2CNC(C2CC3(CCC3)C2)=O)=O)C1 35260,C1(CC)C(C(=O)N(CCC(=O)N(C)CC2CCCCO2)CCO)CCN1C 35261,c1(OC)ccc(C(N2CCC(C3CCCN3C(=O)Cc3nc(CO)cs3)C2)=O)o1 35262,c1(CC)nn[nH]c1C(=O)NCCC1(NC(=O)C(COC)OC)CC1 35263,c1(NC(CN2CCN(C)CC2)=O)ccc([N+](=O)[O-])cn1.C12CC13CCN(C3)C2=O 35264,C(=O)(CCCS(C)(=O)=O)N1CCC(=CCNC(C(c2cnn(C)c2)OC)=O)CC1 35265,C(=O)(C1=NNC(=O)C1)NC(CC)(C)CCNC(c1cccn1C1CCCC1)=O 35266,c1(C(=O)NC(C(C)O)C(=O)NCC(C)(C)CCO)ccc(C#N)cc1 35267,c1(C(=O)NC2CCC(CCNC(C(C(C)C)O)=O)C2)cncc2sccc12 35268,c1(C2C(F)(F)C2)nccc(=NC(CC2CCC2)c2ccccc2)[nH]1.c1(S)ccccc1 35269,CC1(C)CCC(CNC(C2CCCO2)=O)(NC(=O)C(O)C(C)(C)C)CC1 35270,C(=O)(CCC(C)(C)F)NCC(CCNC(C1N(C(CC(C)C)=O)CCCC1)=O)O 35271,C1(CNC(=O)CC2CCC2)CCN(C(=O)CSc2ccsc2[N+](=O)[O-])C12CCC2 35272,c1(CC(=O)NC(C2CCCN(C(=O)CC3CC3)C2)C)ccc(F)c(F)c1 35273,C1(C(N2CCC(NC(C(CC)=CC)=O)C(C)C2)=O)CCCC2CCCN12 35274,CC1(C)CCCC(CC(N2CCCC2CCCNC(=O)CCCC#N)=O)O1 35275,CC(C)(CCC(=O)NCCC1(O)CCCC1)NC(C1CCC(CO)O1)=O 35276,C(CCC(C)C(=O)N1CCCC1C(C)NC(c1cc(F)cs1)=O)OC 35277,N1(C(CN(C(=O)OCC)C)=O)CCC(C)C(NC(=O)CSC)C1 35278,N1(CC)C(=O)CCC1CC(=O)NC1(CN2CCN(C(c3cc[nH]n3)=O)CC2)CC1 35279,C1(C)(CCC(=O)NCCCN(C(C)C)C(C2CC(F)(F)C2)=O)CCC(=O)N1 35280,n1(CC(=O)NC2(C)CC(NC(C3(CC)CCNC3=O)=O)C2)c([N+](=O)[O-])cnc1C 35281,O=C(CCC(=O)N1CC(NC(c2ccccc2CO)=O)C(O)C1)Nc1cccs1 35282,C12(CC(=O)NC3C(NC(COCCC)=O)COCC3)CC3CC(CC(C3)C1)C2 35283,Cn1cc(Cn2cc(-c3cnn(CC(=O)O)c3)nn2)nn1.C12CCN1C2=O 35284,c1(C(=O)NC2CC(O)(CNC(=O)CC3CCCS3(=O)=O)C2)cc2c(s1)CCC2 35285,CC(C)S(=O)(=O)CCCN1CC=CC(NC(c2coc(Cn3cccn3)c2)=O)C1 35286,C(=O)(CC(C)(C)N(C)C(C1CCC(CC)CC1)=O)NC(CC)C(C)C 35287,C=CC1CN(C(=O)Cn2cc(C3CCC3)nn2)CC1NC(c1cc(C)c(C)[nH]1)=O 35288,N1(C(C(C2CCOCC2)OCC)=O)CCC2C1CCCN2C(c1cnc(O)s1)=O 35289,C=C(Cl)CC(C(=O)NOCC(=O)NCC)NC(C1C2CC3C(C2)C13)=O 35290,C1(C(=O)NCC(C#C)CC)(C(C)C)CCN(C(c2cocc2C)=O)C1 35291,Cc1ccc2n[nH]cc2c1-c1cnc(CN(C)Cc2ccccc2)s1 35292,N1(C(C2C(C(=O)OC)C2)=O)CC2CCC(N=c3ccc(OC)c(OC)[nH]3)CC2C1 35293,C1(NC(=O)CC2COCCCO2)CCN(C(c2cc3ccsc3s2)=O)CC12CCC2 35294,C(=O)(CC(C)CNC(=O)C(C)Cn1cccn1)NC1(C(=O)OCC)CCC1 35295,c1(CC(=O)NC(C)CCNC(=O)C(C)C2CCCO2)ccc2nonc2c1 35296,C1(CNC(CP(C)(C)=O)=O)CC2CC(C1)CN(C(=O)COCC(F)(F)F)C2 35297,C1(C(=O)NC(C)CCOC)(CC)CCCN(C(c2cc(CO)nn2C)=O)C1 35298,c1(C(=O)NC2C(NC(c3c(C)nc(COC)s3)=O)C2)cc([N+](=O)[O-])c(C)cc1C 35299,c1(C(=O)OC)ccc(C(=O)NC2CCC(NC(=O)CS(N)(=O)=O)CC2)nc1 35300,c1(CCC(=O)NC(CC)CNC(=O)CC2CCC(F)(F)CO2)nc2ccccc2o1 35301,C(C1CCOC1)=CC(=O)N(N(CC(=O)NCCCCSC)CCCN(C)C)CC 35302,N1(C(C2OCCN(CC)C2)=O)C2CCC(C2)C1CNC(c1sccc1F)=O 35303,N1(C(C)=O)CC2(COC(CNC(c3cnn(CC(F)(F)F)n3)=O)C2)C1 35304,N1(C(C=C(CCC)C)=O)CCCC(NC(c2c[nH]c(=NC)o2)=O)C1C 35305,CCC(CC(C)C)C(=O)NCC1(O)CN(C(=O)Cc2ccn(CC(F)(F)F)n2)C1 35306,O=C1CCc2cccc(C(=O)NC3CCCC3CNC(c3coc(Cl)c3)=O)c21 35307,C1(C)(NC(C2CN(C(C=CC=CCC)=O)CC(C)O2)=O)CCC(=O)NC1=O 35308,C1(CC#C)CCN(C(=O)CCC2CCN(C(c3ncn(C)n3)=O)C2)C1 35309,c1(C(C)C(=O)N(CCC(=O)N(CC(O)CF)C)C(C)C)ccn(C)c1 35310,C12CC3CC1CC3NC(C)(C)C(=O)N2.c1(NC(C(=O)OC)=O)ccccn1 35311,N1(C(C(c2cccs2)NC(C(CC2CC2)NC(=O)COC)=O)=O)CCC(O)CC1 35312,C=C1CCN(C(c2ccn(C)c2)=O)C(C(=O)NC2(CO)CCCCC2)C1 35313,C1(CC)CN(C(=O)C=Cc2cccnc2)CCN1C(=O)COCC(=O)NC 35314,N1(CCC)CC(C(=O)NCCN(C(C2CCN(CC)C2)=O)CCN(C)C)CC1=O 35315,c1(C(=O)NCC(CN(C(C(CNC)O)=O)CC)(C)C)cncc(N(C)C)n1 35316,N1(CCC(=O)NC2CCCCC2NC(=O)CCc2cnoc2)CCC(O)CC1 35317,N1(C(C(C)=CC2CC2)=O)CCCC(C)C1CCNC(=O)C(F)F 35318,CC1CS(=O)CCN1C(=O)CCC1CCCN1C(=O)C=Cc1ccnn1C 35319,C12(C(N(C)Cc3ccco3)=O)COCC1CN(C(c1cc3ncccn3n1)=O)C2 35320,C(COCC(F)F)(C(=O)N(C1CC1)Cc1cccnc1)NC(=O)C=CC1CCC1 35321,c1(CN2CCCC(N(C(c3cn(C4CCOC4)cn3)=O)CC)C2)ccc(C)nn1 35322,Cc1ncc(C#N)cc1NC(C1(O)CCN(C(=O)Cc2cc[nH]n2)C1)=O 35323,N1(C(CCC(=C)Cl)=O)CCC2CN(C(C3(C)CCCNC3=O)=O)CC2CC1 35324,C1(COC)CN(C(C2CC(F)(CO)C2)=O)CCN1C(=O)CC1CN2CCN1CC2 35325,C(=O)(CC(C)CNC(=O)C(Cl)Cl)NCCc1ccn(CC)n1 35326,C(CC(C)C(=O)N(CCC(C)NC(C1(C(F)(F)F)CCC1)=O)C)=CC 35327,CC(C)CCC(F)C(=O)NC1(CCC(=O)N(C)Cc2ccsc2)CCCC1 35328,c1(OC)ncnc(C(=O)NCC2CCN(C(=O)Cc3csnc3C)CC2C)c1F 35329,N1(C(C(=O)NCC=C)CC2CCC(C)(C)CC2)CCCC2OCCC2C1 35330,CCC(Cc1cccc(C)c1)C(=O)NCC1CCCN(C(=O)Cc2cncs2)C1 35331,CCCC(CC)C(=O)NCC(O)CCNC(c1cc(=O)c(Br)c[nH]1)=O 35332,N1(C(CC2CC(=O)OC2)=O)CC=CC(C(=O)NC2CC(CO)C3CC23)C1 35333,CC(CC(F)F)C(=O)N1CCC(CNC(c2cccc(CO)n2)=O)C1 35334,CC1(C2CC2)CCCN1C(=O)NCCCC1CCC(O)C1 35335,C1(C(=O)OC)CN(C(=O)CCC(=O)NCC(F)(F)F)CCO1.C12CC(C1)C(=O)N2 35336,C(CCS(C)(=O)=O)(C1CC1)NC(c1nnnn1Cc1cnn2c1CCC2)C 35337,CCCC(CC(=O)N1CCCC(CCO)C1)NC(=O)CCCOC(C)(C)C 35338,N1(C(c2c(C)[nH]cc2)=O)CCCCC(C(=O)NCCc2ccnc(O)c2)C1 35339,c1(C(N2CC3CN(C(CCc4scc(C)n4)=O)C3C2)=O)ccc2ncnn2c1 35340,C(C)(CCCNC(=O)CCSCC(C)C)NC(C1(NC(C)=O)CCC1)=O 35341,C(=O)(NNc1cccc2ccsc12)C1N(C(=O)OC(C)(C)C)C2(CO1)CCC2 35342,N1(C(c2cc(C)[nH]n2)=O)CC2CCCCN2C1CNC(=O)CC12CC(C1)C2 35343,c1(C(c2n(CCC)nnn2)NCC=C(C)C)cc(OC)ccc1F 35344,c1(C(N2CCCC(CNC(c3on(C)c(=O)c3)=O)CC2)=O)c(F)ccc(F)c1N 35345,N#CC1(C(N2CCN(C(C3(S(N)(=O)=O)CCC3)=O)CC2)=O)CC2CC2C1 35346,N1(C(CNC(=O)NC)=O)CCN(C(=O)CCCN(C)C)CC1C(F)F 35347,Cc1cc2[nH]c(C(=O)NC3CC(C)CN(C(C4CC5COCC5C4)=O)C3)cc2s1 35348,CC(=O)CCCCC(=O)NC(C(=O)N(C)CC1(O)CCCC1)C(C)(C)O 35349,C1(C(N2CCC(C(C)OC)CC2)=O)CC2CCC1N2C(c1csc(C)c1)=O 35350,CN=c1[nH]c(=NCCCOC)[nH]c(=NC2CCOC3(CCC3)C2)[nH]1 35351,c1(C(N(CCCCN(C(CCn2c(C)ncc2)=O)C)C)=O)ccc(F)c(Cl)c1F 35352,c1(C(=O)Nc2c(C(N3CCC(C)C3)=O)cc(OCC)nc2)cc2ccccc2s1 35353,N1(C(C(C)n2cccn2)=O)CCCCCC1C(N1CC(CO)C(O)C1)=O 35354,c1(C(N2CCC(CNC(C(COC)N(C)C)=O)C2)=O)c[nH]c2ccc(O)cc12 35355,N1(C(C2=CCC(NC(C=CC=CCC)=O)C2)=O)CC2(CCC2)C12CCC2 35356,C1(CNC(CC2C(C)CCO2)=O)CCCN(C(C2(c3ccc(Cl)cc3)CC2)=O)C1 35357,N1(C(CCCOC)=O)CCC(C)(CCNC(=O)C(C(C)C)NS(N)(=O)=O)C1 35358,C(=O)(C(C)C(O)CC(C)C)NCC1N(C(Cc2c(F)ccc(C)c2)=O)CCC1 35359,c1(OC)ccc(CC(=O)NCCC(O)CNC(C2CNC(=O)N2)=O)cc1O 35360,C=CCC(CNC(C1(C)CC(=C)C1)=O)NC(c1csc(C(C)OC)n1)=O 35361,C=C(Cl)CC(C(=O)NC(c1ncc(C)o1)C)NC(=O)Cc1ccn(CC)n1 35362,C1(NC(C2(CC(C)C)CC2)=O)C2CC3CN(C(c4cc(Br)n[nH]4)=O)C1C3C2 35363,Cc1ccc(C(=O)NCC(C)(CO)NC(=O)CC2CCCCO2)c(O)n1 35364,c1(CO)c(CNCC(O)CN2CCCCC2)ccc(Cl)c1Cl 35365,c1(OCC)cc(C(N2CCC(=CCNC(=O)CCC3(C)CC3)CC2)=O)cc(F)c1 35366,Cc1ccc(Cl)c(C(=O)NCC(C2CCC2)NC(=O)Cc2ccc(F)cn2)c1N 35367,N1(C(C(CSC)OC)=O)CCC(NC(=O)Cc2nc3ccccc3s2)C(C)(C)C1 35368,C1(NC(C2C(C)CCN2C(=O)C(C)CCN(C)C)=O)(CO)CC2CCCC12 35369,CCCCCC(O)CC(=O)NCC1CC2(CC2)CN1C(=O)C(O)CC1CC1 35370,N1(CCCNC(c2nc(C(C)(C)C)oc2)=O)CCCN(C(C2CC2(F)Cl)=O)CC1 35371,CC1CC(NC(c2ccc(O)c(Cl)n2)=O)CN(C(=O)CSC2CC2)C1 35372,n1(CC(N2CCN(CC(=O)NO)CC2)=O)ccc2ccc(F)cc12 35373,Cc1nc([N+](=O)[O-])cn1CCC(=O)OC(F)(F)F.C(CC1CC1)CN 35374,C1(CN=C(NC(CC)CC)NCC(C)(C)C)COC2(CCC2)CO1 35375,c1(C(=O)NC2C(NC(C(C)(C)OC(C)C)=O)C2)ccc(Cl)c(F)c1O 35376,O(C1CCCc2ccccc21)CC(=O)N(C(C)C)Cc1n[nH]c2c1CCCC2 35377,C(=O)(C(O)C(C)C1CCCCC1)N1CC(NC(Cc2c(OCC)cccc2)=O)C1 35378,N1(C(Cn2cc(C(CC)O)nn2)=O)CC2C(CO)C3CCC2(C1)O3 35379,c1(N(CCNCC)C)ccc(C)c(F)c1F.N12CCCC1C2 35380,C1(NC(CCC2(C)N(C(CCc3c(C)noc3)=O)CCC2)=O)(CO)CC2CCCC12 35381,c1(C(=O)NCC(C)CNC(C23CC(C)(C2)C3)=O)cc2c(o1)CCCNC2=O 35382,C1(CNC(c2c[nH]c(=N)o2)=O)CCC2(CCC2)C1NC(=O)CCCc1cccs1 35383,N1(C(=O)NCc2ccc(-n3ccc(C)n3)nc2)CC(CC(C)CO)c2ccccc21 35384,Cc1cn2cccc(C(N3CC(C4(NC(=O)Cc5sccc5C)CC4)C3)=O)c2n1 35385,C1(C(=O)NCCOC(C)=O)(CC)CCCCCN1C(CC1CCOC1)C(=O)NC 35386,n1(CC#C)cccc1C(=O)NCCCNC(=O)C(C)OCc1ccccc1 35387,C1(NC(C2C=CCN(C(CCNC(COC)=O)=O)C2)=O)CC2CCCC(C1)C2 35388,N1(C(C(CC=C)OC)=O)CCC(C)N(C(=O)CC2(CSC)CC2)CC1 35389,CN1CCN(C(=O)CCc2cc(F)ccc2Br)C(CNC(=O)C2=CCC2)C1 35390,c1(N(C)C)ccc([N+](=O)[O-])cc1CN1CCCC1C(N1CCN2CCC1CC2)=O 35391,c1(C(N(C)CC2CCCCN2C(=O)CCC(N)=O)=O)ccccc1P(C)(C)=O 35392,N1(C(C(C)=C2CC2)=O)CCC(C(=O)NCC(C)(C)C(C)C)C1C 35393,N(C(=NCCC(=O)NC)NCC1Cc2ccccc21)C(C=C)C 35394,CCCCCCCCOCC(=O)NCC1C2CN(CC3COCCN3C)CC12 35395,n1(CCC)ccc2ccc(CC(N3CCC4OCCN(C)C4C3)=O)cc12 35396,Cc1ccc(Cl)cc1C(=O)NCC(O)CN(C(=O)CN1CCC(C)C1)C 35397,CC1CN(C(C2CC(O)(CNC(C3(C)CCC3)=O)C2)=O)CC(C)(C)C1 35398,CC1(NC(C23CC(CN2C(C2(CCN=[N+]=[N-])CC2)=O)C3)=O)CCOC1=O 35399,C1(CNC(Cc2ccc(C)o2)=O)CN(C(C2CC2C)=O)C(C)(C)C1 35400,C1(NC(C(C)=CC)=O)CN(C(=O)C(c2ccncc2C)C)Cc2ccnn2C1 35401,c1(C(N2CCC(C(N(CCC(=O)OC)C)=O)C2)=O)ncc(F)cc1F 35402,C(N=c1nc(N2CCCC(CSC)C2)cc(C)[nH]1)C1(OCC)CCC1 35403,N1(C(c2scc(OC)c2OC)=O)CCN(C(C2(CSC)CC2)=O)CC2(CC2)C1 35404,c1(C(=O)NC(CCNC(Cc2c(C)n[nH]c2C)=O)C)cc2c(cnn2C)nc1C 35405,C1(C(=O)NCC(C#C)OC)CN(C(=O)C(=O)NC(C)CC)CC(C)O1 35406,N1(Cc2c(OC)cc(C)cc2)CC(NC(C2COC(C)C2)=O)CC(C)(C)C1 35407,C=Cc1cnc(NC(C2CCN(c3cnccn3)CC2F)=O)nc1 35408,N1(C(CCCNC=O)=O)CC(NC(=O)COc2cccc(C)c2F)CCC1C 35409,c1(C(N(C(CC(=O)OCC)c2ccccc2)CCC)=O)ccc(COC)o1 35410,c1(C(=O)N(Cc2c(C(=O)NCC(C(CC)C)C)con2)C(I)CC)ccnc(C)c1N 35411,c1(C(N(C)CC2N(C(CCCCCC=C)=O)CCC2)=O)cc(N)c(F)c(F)c1Cl 35412,c1(CC(N2CC(COC)(NC(C3CCC(C)C3)=O)C2)=O)cncc(Br)c1 35413,C(c1cn(CCCNC(C2CCN(c3ccc(Cl)cn3)CC2)=O)nn1)=CC(C)C 35414,C1(C(N2CCCN(C(C(C)CCN(C)C)=O)CC2)=O)CCC(F)(F)CC1(C)C 35415,C12(C(N3CCC(NC(c4cc(C)cc(O)c4)=O)C3)=O)CCC(C)(CC1)OC2 35416,N1(C(C=C(CCC)C)=O)CCC2CCN(C(c3cnc4ccc(C)cn34)=O)C2C1 35417,C1(C(N2CC(C(N)=O)C2)=O)CC(F)CN(C(c2cncc(C(F)(F)F)c2)=O)C1 35418,Cc1ccc2sc(C(N3CCN(C(=O)C(C)C4CCOC4)CCC3C)=O)cc2c1 35419,N1(C(c2c(C)nc(C)o2)=O)CC2CCCC(C1)N2C(=O)C(C)n1ccnc1 35420,c1(CC(N2C(CNC(C3CC(C(F)F)C3)=O)CCCC2)=O)cnc2ncccn12 35421,C(=O)(CCC(=O)NCC1CN(C(c2ccn(CC)n2)=O)C1)Nc1nnc(CC)s1 35422,C12(C(N(CCN(C(C3CC3(C)C(C)C)=O)CC)CC)=O)CC(C)(C1)OC2(C)C 35423,CC1(C)CC(CC(=O)Nc2ccnc(C3CNC3)c2)C(=O)O1 35424,C1(NC(=O)CC2=CCCC2)CCCC2CN(C(=O)Cc3ccc(O)c(F)c3)CC12 35425,C1(Nc2ccc(CC)nc2)CC2c3ccccc3C1c1ccccc12 35426,Cn1nnc(CC(N2CC(=C(F)CNC(c3cc(F)c[nH]3)=O)C2)=O)n1 35427,N1(C(c2c(C)ocn2)=O)CCC2CC(C(=O)N(C3CCC(C)CC3)CCO)C2C1 35428,CC(C)CC(C(=O)NCc1noc(C(N)=O)n1)OC1CCCC1 35429,C1(C(=O)NCCCCC(C)NC(=O)C(C)Cc2ccco2)(CC)CCNC1=O 35430,C1(NC(c2cccc(F)c2OCCF)=O)CN(C(=O)COC(F)F)CCC1CO 35431,c1(C(CC)C)nc(C2CCC(=O)N2C)n(-c2nc(C)nn2C)n1 35432,N1(C(CCCCOCCC=C)=O)CCN(C(=O)Cc2ccnc(C)c2)C(C)C1C 35433,C1(F)(NC(CCC(C)N(C)C)=O)CCCN(c2nnc(-c3ccccc3Cl)s2)C1 35434,N1(C(c2onc(CC)n2)=O)CC2(CCN(C(=O)Cc3cccs3)CC2)C1 35435,c1(C(=O)NCC(N(C(C2(OC)CCSC2)=O)C)C2CC2)cc(Cl)c(Cl)s1 35436,c1(OC(Cc2ccc(-c3cccc(C)c3)cc2)=O)ccc(F)c(Cl)c1F 35437,N1(C(C(C(C)C)SC)=O)CCOC2(CCN(C(c3nnc(O)nc3O)=O)CC2)C1 35438,C1(C(=O)NCC(CC=C)NC(c2cc(CCC)oc2C)=O)CC2C=CC1C2 35439,CC(C(=O)NC(C(=O)N(C)CC1(CO)CCC1)c1cccs1)OC1CCCC1 35440,C(=O)(CCCC(C)(C)C)N1CCC(CN(C(=O)Cc2cn3ccsc3n2)C)C1 35441,Cc1cc(O)nnc1C(=O)NCC(C)NC(=O)C(C)(C)c1ccccn1 35442,c1(CC)c(NC2(C)CCCN(C(=O)CC(C)C3CCCCC3)C2)nc(C)nc1Cl 35443,N1(C(C2C(Cl)(C(=O)OC)C2)=O)CCC(C2(NC(=O)Cc3oc(C)nc3C)CC2)C1 35444,[N-]=[N+]=NCCCC(=O)NCC1(O)CC(CNC(=O)CCc2csc(=N)[nH]2)C1 35445,c1(C=O)cc2c(C(=O)NCCCN(C(N)CC)CC)cccc2n1C 35446,C12CCCN1CCC2.C1(COC)CCCN1C(=O)C(O)Cn1cncn1 35447,N1(C(C(CC)OCC)=O)CCC2(CCCN2C(C2CC2c2ccccc2)=O)CC1 35448,n1(CC)nc(C)cc1C(=O)NCC1CC1NC(=O)C(C)(C)n1ccc(C2CC2)n1 35449,C1(CC)CCN(C(c2ccc(SC)s2)=O)C1C(=O)Nc1cnn(C)c1SC 35450,N1(C(C2C(C)(C(F)(F)F)C2)=O)CCC(CNc2ncncc2Cl)C(O)C1 35451,N1(C(c2c(C)nc(C)o2)=O)CC2(COC(CNC(c3ccns3)=O)C2)C1 35452,N1(C(c2cnn(CC)n2)=O)CCC2CN(C(c3ccoc3C)=O)CCC2C1 35453,C(=O)(CC(CCC)NC(=O)CSCC)NC1CC(C=C)C1 35454,C=CCC(C)C(=O)N(C(C)CNC(C1(C(=O)OCC)CC=CC1)=O)C 35455,CC(C)(C(=O)NC1CC12CCC2)C(O)C1CC1 35456,CC1(C)C2CC(C(=O)NC3CC4(C3)CC4C(=O)NCc3cccnc3)CC12 35457,C1(NC(C(C)OCCCCCC)=O)C=CCN(C(C2CC23CCC3)=O)C1 35458,Cc1cc(C)c(C=CC(=O)NC2(CO)CN(C(c3cc(CO)[nH]n3)=O)C2)cc1C 35459,C(=O)(C1=CCC(C)(C)CC1)N(C(C(=O)NC1CCCN(CC)C1)C)C 35460,N1(CCC2CC(NC(=O)OC(C)(C)C)C2)CC2CCC2C1.C1CO1 35461,c1(C(=O)NCC(CCC)NC(C2CCOCC23CCC3)=O)ccc2c(c1)SCCN2 35462,c1(N(CCN(C(c2cc(CC)on2)=O)C)CC)ccc(S(=O)(=O)NC)cc1 35463,CCC(CC)CCCC(=O)N1CC2(CCCC2)C1C(=O)NC(C)Cn1ccnc1 35464,N1(C(c2scc(CNC(C(C=CC)O)=O)c2)=O)CCc2c(cnn2C)C1 35465,CC(=O)CCN=C(NCC1COC(=O)O1)NCC1CN(S(C)(=O)=O)C1 35466,C12(C(N(C3CCN(C(C4OCCC4C(F)(F)F)=O)CC3)CC)=O)CCC(CC1)O2 35467,C(N=c1nc(C(=O)OC)c(Cl)c[nH]1)C1CCC(NC(C(CCC)(C)O)=O)C1 35468,c1(OC)cc(C(=O)NC(CNC(C2CCCC23CC3)=O)C2CC2)c(F)cc1N 35469,C(=O)(C(C)C(O)CC)NCCCCCCN(C(C(C=C)OC)=O)C 35470,C1(c2n(C)ccn2)CCN(C(=O)NCC2CC(OC3CC3)C2)C12CC2 35471,c1(C(=O)NC2CN(C(c3c(COC)ccs3)=O)C3C2C3)cc2sccc2[nH]1 35472,c1(C(=O)NCCNC(C2N(C(C)=O)CCOC2)=O)c([N+](=O)[O-])cnn1CCO 35473,C1(CNC(c2c(CC)noc2)=O)CN(C(C2CC3CC3C2)=O)CCC1C 35474,Cc1cc(C(N2CCOC(C(C)NC(C3CCCCO3)=O)C2)=O)cc(C)c1F 35475,C1(NC(C2(OCC)CCCC2)=O)COC2CN(C(=O)Cc3ccnnc3O)CC12 35476,C1(CNC(c2cn(C)nc2C2CC2)=O)CCC12CN(C(=O)CN1CCOC1=O)C2 35477,c1(C(=O)NC2C(NC(c3nncc(OC)c3)=O)CCCC2)cc(C)c(Cl)cn1 35478,S(=O)(=O)(CCC(=O)NCC1CC(NC(=O)CN2CCC2C)CCO1)NC 35479,C1(C(=O)NCC2(CSC3CCSC3)CCC2)CCC(n2cc(C)nn2)C1 35480,N1(C(c2c(C)coc2)=O)CCC2(CC1)CN(Cc1csc3nccn13)CCO2 35481,c1(C(=O)NCCCNC(c2occ(S(N)(=O)=O)c2)=O)ccc2c(c1)C(=O)CCO2 35482,C1(C(=O)NCc2cn(C(C)C)nc2)(CNC(=O)Cc2ccc[nH]2)CC(C)(C)C1 35483,CC1CC(CNC(=NCCN2CCCCC2)NCCCc2ccsc2)CC(C)O1 35484,N#Cc1ccncc1NC(C1CCC(NCc2ccc(Br)c(C(=O)O)c2)CC1)=O 35485,C1(CC=C)(NC(c2ccoc2)=O)CCCN(C(c2[nH]c(O)nc2C)=O)C1 35486,C(C(C(=O)NCCN(C(=O)C(C)(C)n1ccnn1)C)C(C)(C)C)OCC=C 35487,C1(=O)CCCC(=O)NCCCCN1CC.c1(C(=O)NC(C)C)ccc(CO)cn1 35488,Cc1c(C(F)(F)F)n[nH]c1C(=O)NCCCNC(=O)Cn1cc(Cl)cn1 35489,C(=O)(CCCCCC#N)N1C(CNC(c2cc(C)n(C3CC3)c2C)=O)CC(F)C1 35490,c1(C(=O)NCCCC(C)NC(c2ccncc2Cl)=O)cccn(C)c1=O 35491,c1(C(N2CC(NC(C3(COC)CC3)=O)C(C3CC3)C2)=O)oc2ccccc2c1C 35492,c1(CNCC2N(CC(C)C)CCC2)n[nH]c2cc(F)ccc12 35493,c1(N2CC3CN(C)CC3C2)nc2c(c(=NC3CCCc4cnn(C)c43)[nH]1)CCC2 35494,CCC(CCC(=O)NCC(C)(C)C(=O)NCCOC)NC(C)(C)C(N)=O 35495,C1(CC(C)NC(C=C(COC)C)=O)CCN(C(=O)C(N2CCCCCC2)C)CC1 35496,c1(C(=O)NC(C(=O)NCc2c(C)ccs2)(C)C2CCC2)ccc(C#N)n1C 35497,C1(CNC(C(CO)N(C)C)=O)CN(C(c2nnc(S)n2C)=O)CC1(C)C 35498,c1(C(=O)Nc2cc(OC)ncc2)[nH]c(C)c(NC(c2cccc(N(C)C)n2)=O)c1C 35499,c1(C(=O)NCCCC(C)NC(c2cc(CC3CC3)on2)=O)cc[nH]c(=N)c1 35500,N1(C(C(CN=[N+]=[N-])NC(=O)CCCn2ccnn2)=O)CC2CCC(O)C2C1 35501,n1(CCOc2c(OC)cc(C(C)NCC3CCO3)cc2)cnc2ccccc12 35502,c1(C(=O)OCC)ncc(NC(c2cccnc2)C2CCCO2)nc1N 35503,c1(OC)nccc(C(=O)NCc2occc2C(=O)NC(c2ccccc2)C)n1 35504,C1(F)(CNC(CCSCCCC)=O)CCCN(C(=O)C(CCC)OC)CC1 35505,c1(C(N2CCC(N(C(c3cncn3C)=O)CC)C2)=O)cccc2ccnn12 35506,c1(NCCNC(c2c(NC)nccc2)=O)ccc(C(=O)OC)c(C)c1 35507,C1(COC)(CNC(C2CC(N(C)C)C2)=O)CN(C(=O)C(n2ccc(C)n2)C)C1 35508,N1(C(C(C2CCCN(C(c3c(C)noc3)=O)C2)C)=O)CCCC(C)(C)CC1 35509,c1(CC(N2C(C)CC(NC(CC(CC)C3CC3)=O)C2)=O)ccc(O)c(C)c1 35510,C(=O)(CCCCCNC(C1CC1C(C)C)=O)OCC.c12ccc(Br)c(c1)CS2 35511,c1(C(=O)NCC2CCC(NC(CCSCCCC)=O)CC2)cccc2occc12 35512,NC(=O)C1CN(C(C2CC3(C2)CC3(F)F)=O)c2ccccc21 35513,C(C)(CCC(=O)N1CCN(C2CCN(C(=O)C=C3CCC3)CC2)CC1)OC 35514,c1(C(=O)NC2C(O)CCN2C(=O)COc2ccc(Br)cc2)cc(Br)c(Cl)nc1 35515,C1(C(=O)NC(C)C)CCCCCC1NC(C1CC1(F)F)=O 35516,C(C)(C)(CC(=O)NCCC1CN(C(=O)CCC2CCC(=O)C2)CCO1)SC 35517,c1(C(=O)NC(C)(C)CCNC(C2CCCCC2C(N)=O)=O)cc(N)ccc1Cl 35518,N1(C(CCc2cn(C)nc2)=O)CCC(NC=O)C(C)(C)C1.C(CC(=O)NC)NC1CC1 35519,C1(C)CCN(c2cnccn2)C1.N#CC1CC1C(=O)NC.C12CC(C1)NC2=O 35520,c1(CNC(C2CCCOC2)C)cc[n+]([O-])cc1 35521,N1(CC(=O)NCC(C(C)C)NC(=O)CC2CCCCN2C)CCC(=O)NC1=O 35522,c1(NC(C2C3CN(C(CCCC=C)=O)CC32)=O)cc(CC)cc(N)c1 35523,C(=O)(CC(C(C)C)NC(C1CN(NC(C)=O)CCO1)=O)Nc1n(CC)cnc1 35524,C1(C(=O)NC2C(NC(C=CC(=O)OCC)=O)CC2)CC(=O)N(c2cnn(C)c2)C1 35525,C1(C)(C(=O)NC(c2cccnc2F)C)CCCN(C(=O)CC2COCC(C)O2)C1 35526,C(=O)(C(C)(C)CC(C)(C)C)N1CCN(C(COCCCC)=O)C(CCO)C1 35527,C1(N(C(=O)CN2CCSCC2)C)CCCC(NC(=O)C=CC2CCCC2)C1 35528,N1(C(C2(Oc3ccc(C)o3)CCC2)=O)CCCN(C(C2CCC2)=O)CC1 35529,C12(C(N3CC(NC(=O)Cc4cnccc4Cl)C(O)C3)=O)CCCC1C2(F)F 35530,N(C(=NCCCF)NCCc1cnccn1)CC1(c2ccc(OC)cc2)CCC1 35531,Cc1nc(NC(C2CC(C)CN2Cc2cnn(C)c2C)=O)cc(Cl)n1 35532,C1(CNC(C(CC=C)(C)C)=O)CC2CCC(C1)N2C(=O)CC1CC(C)C1 35533,Cc1nnc(N2CC(C(F)(F)F)CC(C)C2)c(C#N)c1C.C(=O)C(C)CC(C)(C)C 35534,c1(CN(C)C)ccc(C(=O)NC2COCC2CNC(=O)CN2CCNC2=O)o1 35535,C1(C(=O)NCC(C2CC2)SC)CCC2(CC2)N1C(C1CCC(C)(C)OC1)=O 35536,CC1=CC(NC(=O)CCN(CCO)C(C2CCC(=C3CCC3)CC2)=O)CCC1 35537,CC1CC2CN(C(=O)CCCCNC(=O)CCNC(=O)CCC(CF)CF)CCN2C1 35538,N1(C(C2ON=C(C)C2)=O)CC2(CNC(C3CC3C3CC3C)=O)CC1CO2 35539,N#Cc1ccc(C(=O)NCC2(C(N)=O)CN(C(c3cccc(F)c3)=O)C2)o1 35540,C(=O)(CCC1CCc2ccccc21)OCc1c(N(C)C)cc(C(F)F)nn1 35541,C1(NC(c2n(C)nc(Cl)c2)=O)CCN(C(=O)C=CC2CCCCCC2)CC1F 35542,c1(NC(C2CSCCN2C(c2cccc(CO)c2F)=O)=O)cccc2c[nH]nc12 35543,n1(CCOC)cnc(C(=O)NCC2CC(NC(=O)C(CC3CCC3)SC)C2)c1 35544,N1(C(c2cc(CC)on2)=O)CCCN(C(=O)C(N2CCN(C)CC2)C)C(C)C1 35545,C(=O)(CC1=CCOCC1)N1CCC(C(C)(C)NC(=O)Cc2cccc(C#N)c2)C1 35546,C(N=c1cc(C)nc(C2CC2)[nH]1)C1OCCN(C(C(C(CC)C)OC)=O)C1 35547,Cc1ccc2cc(C(N3CCCC(NC(c4sc(C)cc4Cl)=O)C3)=O)ccc2n1 35548,CCC(C)CCC(=O)NC1CC2(NC(c3cccc(N(C)C)c3)=O)COC1C2 35549,C1(c2n(C)cnc2)CCN(C(c2sccc2CNC(c2ccccn2)=O)=O)CC1 35550,c1(C(=O)NCC(CC)(C)NC(=O)Cn2cccc2)cccc(C2CC2)n1 35551,c1(CCC(=O)NC2CC(CCNC(C(C)=CC)=O)C2)ccc2ncccc2c1 35552,N1(C(C2CCOCC2)C(=O)NCC)CC2CC1(C(=O)OC(C)(C)C)C2.C1CCC1 35553,c1(C(C(=O)NCCC)N(c2ccccc2)CC2CCOCC2)ccc(CC)cc1 35554,C1(CCC)(C(=O)NCC(C)N(C(=O)CCOCC(C)C)C)CCNC1=O 35555,N1(C(CSCCCC)=O)CC2ON=C(CNC(c3cccc4c3OCO4)=O)C2C1 35556,CCCC(C)CC(=O)NCCC(C(C)C)NC(=O)CCSc1cc(F)ccc1F 35557,c1(C(=O)NC(C2N(C(CCCC(=C)C)=O)CCC2)C)ccc2cc[nH]c2n1 35558,c1(Nc2ccccc2OC)ncc(C(F)(F)F)cc1Cl.Fc1ccccc1CCS 35559,C1(CNC(C(C)C2CCCC2)=O)CCC(NC(C2(C(C3CC3)N(C)C)CC2)=O)CC1 35560,n1(CCC(=O)NCC(CC)NC(=O)CCNC(C2CCCO2)=O)cnc(=N)[nH]1 35561,CN(C)NC(=O)CCC(=O)NC1(CCNC(c2ncn(C(C)C)n2)=O)CCC1 35562,N1(C(c2c(C)ocn2)=O)CCC2(CC1)CCN(C(C1CN3CCN1C(C)C3)=O)C2 35563,C#CCCCCCC(=O)NC1(CCOC)CCN(C(=O)C(c2ccccc2)F)C1 35564,C1(NC(COCCC)=O)(CF)CCN(C(c2sc(C(C)C)nc2C)=O)C1 35565,N#Cc1cccc(C(=O)NC2CCN(c3ncnc4n[nH]cc34)CC2)c1Cl 35566,c1(C(=O)NCCC(C)NC(c2c(CC)nns2)=O)ccc(C#N)n1C 35567,N1(C(C(=O)NCCC)CC2CCC(F)(F)CC2)CCCC2CN(C)CCC12 35568,C1(NC(=O)CCc2nncs2)CC12CCC(NC(=O)CCc1ccoc1)CC2 35569,C(C(C(=O)N(C)CC1CCCCN1C(C1CCOC(=O)CC1)=O)C(F)(F)F)OC 35570,Cc1ccc(C=CC(=O)NCCCNC(c2c(-c3cccs3)noc2C)=O)cn1 35571,c1(OC)ncc(C(=O)NCC(Cc2ccccc2)NC(C2CCCO2)=O)s1 35572,C(=O)(C(C)(C)CN(C(=O)Cc1ccsn1)C)NCCS(CC)=O 35573,N1(C(C2N(C(C)C)CCC2)=O)Cc2ccccc2C(NC(c2nncs2)=O)C1 35574,CC1(C(N2CC3CC(NC(c4cnnc(O)c4)=O)C2C3)=O)CCC(O)CC1 35575,c1(OCC(=O)NC(c2nocc2C(N2CCC(CC3CC3)C2)=O)C)cccnc1 35576,c1(C(=O)NC(C)CCCCNc2ncc(C#N)cc2F)cnc2c(c1)ncn2C 35577,c1(NC(C(CC2CCOCC2)NC(C)=O)=O)cccc2nc(O)nc(O)c12 35578,CC(C)CC(CNC(=O)CC1CCCCOC1)C(=O)NCC1(C)COCCO1 35579,C1(C(=O)NCC2CCN(C(c3c(C)nn[nH]3)=O)CC2)Cc2nn[nH]c2C(C)C1 35580,N1(C(C2(C)CCC2)=O)CC2COCCC2(NC(=O)CC2CCNC2=O)C1 35581,C1(C(N(CCCC)C2CC2)=O)CCN(C(=O)CC2CCCCN2C)O1 35582,C1(NC(C2CCCN(C(N)=O)C2)=O)CN(C(=O)CC2CCCCO2)CC2(CC2)C1 35583,c1(C(=O)NCC(=C2CN(C(Cc3n(C)ncc3)=O)C2)F)cnc2[nH]cnc2c1 35584,Cc1c(C(=O)NC(C2CCCCC2)CNC(=O)CC(C)c2ccccc2)ncn1C 35585,CC(C)C(CC(=O)NCc1ccc(C#N)cn1)OCC(=O)NCc1nc[nH]n1 35586,N1(C(C(CCC)OC)=O)CCC2(CC1)CC2C(=O)NC(c1cncnc1)C 35587,CN1CCC(C)(C(=O)NCC2CCN(C(=O)Cc3cn[nH]c3)CC2O)CC1 35588,c1(C(=O)NCCN(CCOC)C(C2CC(=C3CCC3)C2)=O)c(C)n[nH]c1C 35589,C(C(C(=O)N1CCOC2CC12)C(C)(C)C)NC(COC(CC)C)=O 35590,c1(C(=O)NC(CC)C(F)(F)F)ccc2c(-c3csc(=NCC)[nH]3)nn(C)c2c1 35591,N1(C(CC2CC(=O)C2)=O)CC=CC(NC(C23CSCC2C3)=O)C1 35592,C1(NC(c2[nH]c(=N)sc2)=O)CC2CC1N(C(c1cccc(C(F)(F)F)c1)=O)C2 35593,Cn1cc(C(N2CC(NC(=O)CCOC3CC3)C(C3CC3)C2)=O)c(=O)n(C)c1=O 35594,C#CC1CN(C(=O)CCC2CCCCN2C(c2cc(Cl)no2)=O)CCO1 35595,C1(C(=O)NC2CC(C(C(=O)NC(C#C)CC3CC3)F)C2)Cc2ccccc2C1 35596,C(=O)(C(C)(C)F)N1CC(CN(C)C(C2CCCN2c2ccncn2)=O)C1 35597,N1(CCC2(NC(=O)CC3CC(Cc4cccs4)C3)CC2)CC1CN1CCC1.C1(C)CC1 35598,c1(SCC)ccc(NC(C2CCNC2)=O)cc1.C12CCN(C1)C(=O)N2C 35599,C12(C(=O)NC(C(C)F)C)CC(CCO1)N(C(C1CN(C)C(=O)N1)=O)C2 35600,CCC(C)(C)C(=O)N(C)CC1(C(=O)NC2(C3CCCO3)CC2)CC1 35601,c1(C(N2CC(N(C(C3(CC)CC3(F)F)=O)C)C2)=O)ccccc1S(C)(=O)=O 35602,CCCC(C(=O)NC1CN(C(=O)C(C(C)O)N(C)C)CC1C)NC(=O)C(C)(C)C 35603,c1(CC)[nH]nc2c1CN(N1CCC(C(=O)NCCC3CCCC3)CC1)CC2 35604,N1(C(Cn2nnc(C)n2)=O)CC=C(C(=O)N2CCC(OC3CC3)CC2)CC1 35605,C(=O)(CCCCC(F)(F)F)NC1CN(C(CC(C=C)C)=O)CC1C1CC1 35606,C(CC(C(C)(C)C)NC(c1c[nH]c(=N)c(C)c1)=O)N(C(C1C(CC)CCO1)=O)C 35607,CCCCCCC(c1nnnn1-c1ccc(F)cc1)NC(C)C(=O)NC(C)(C)C 35608,Cc1cnc(F)c(C(N2CCC(NC(c3cc(C(N)=O)ccn3)=O)C2C)=O)c1 35609,Cc1nnsc1C(=O)N(C1(CC(=O)NCC(C)N2CCC2)CC1)C 35610,CN1C(=O)OCC1C(N1CC2C(NC(=O)C=CC3CCOC3)C2C1)=O 35611,c1(C(N(CCCNC(C(C(=O)OC)OC)=O)CCO)=O)cc2n(n1)CC(F)C2 35612,C12(C(=O)OC)CC1CN(C(=O)CC(O)CNC(c1cc(C3CC3)[nH]n1)=O)C2 35613,c1(C(=O)NC2CCC(C)C2)coc2c1CN(C(=O)CC1CCOC1)C2 35614,C1(CC(N2CCCC(O)C2)C(=O)NC(c2cccs2)C)CCC(F)(F)CC1 35615,N1(C(CC2(OC)CCC2)=O)CCC(CCNC(=O)CCc2cc(C)[nH]n2)CC1C 35616,c1(C(=O)NCC(CC)N(C)C(c2cnsc2C)=O)n[nH]c(C)n1 35617,C(=O)(C1=CCCCCC1)NCCCN1CCN(C(c2cccc(N)n2)=O)CC1 35618,n1(C(CC)C)nccc1C(=O)N(C)CCOCCNC(=O)CC1COC(=O)N1 35619,CC1=C(C(=O)C(=O)CCCC(C)(F)F)COCC1.C1(O)(N)CCN(C(=O)C2CC2)CC1 35620,CCCC(C)CC(=O)NCC(O)CN(C(=O)COc1ccc(CC(N)=O)cc1)C 35621,N1(C(C=CC(=O)OCC)=O)CC2CC(NC(=O)Cc3cnco3)CC2C1 35622,C1(NC(c2ccnc(C3CC3)c2)=O)CN(C(c2cnsc2)=O)CC1F 35623,N1(C(C(C=C)(C)C)=O)C(C)CN(C(c2cc3ccccc3[nH]2)=O)CC1C 35624,Cc1ccc(S(N)(=O)=O)cc1C(=O)N(CC(O)CNC(c1ncccc1O)=O)C 35625,c1(C(=O)NC2(CC)CCN(C(C3(OC(C)=O)CC3)=O)C2)c[nH]cc(Cl)c1=O 35626,c1(N(C(=O)O)C2CC2)ccc(CN(C(C)(C)C)CCCO)cn1.c1(C)occc1Br 35627,N1(C(C(CC)(C)COC)=O)CC(NC(c2cnn3ccccc23)=O)C2(CCC2)C1 35628,C1(C(N(C(C2CCCC2)CO)C)=O)CCC(CNC(=O)C=CC2CCCC2)CC1 35629,CC(C)CCC(=O)N1CC(OC)CC1CCNC(c1cccnc1SC(F)F)=O 35630,C1(CNC(C(C)(COC)NC(CC2CC(OCC)C2)=O)=O)CC(C2CC2)=NO1 35631,CC#CCC(C(=O)N1CCC(OCCOC(C)=O)C1)NC(c1sccc1SCC)=O 35632,Cc1cc(F)cc(Br)c1C(=O)NC1CC2CCC1N2C(C1CCCN1C)=O 35633,c1(C(=O)NC(CC(F)F)C(=O)NCC(O)CCO)ccnc2cc[nH]c12 35634,c1(C(=O)NCC2CCC(C)N(C(c3cc[nH]n3)=O)C2)cccc([N+](=O)[O-])c1Cl 35635,c1(C(=O)OCC)c(C)c(C)cc2c1N(C(=O)NC(C)CC1CCCS1)CCC2 35636,C#CC1(C(=O)N(CC(=O)NC)CCC)CCN(C(c2cccc(C#N)c2)=O)C1 35637,c1(C(=O)NCCOCCCNC(c2cc(Cl)c[nH]2)=O)ccc([N+](=O)[O-])s1 35638,C1(S(C)(=O)=O)(C(c2nnnn2C)NC2C(CC)C2)CCCCC1 35639,c1(COC)nnc(N(CC(C)CNC(=O)CC2(C(F)(F)F)CC2)C)s1 35640,c1(C(=O)NC2CC(NC(C3CCCO3)=O)C2)c[nH]cc(F)c1=O 35641,CC1(C)CCC(C(N2CC3CC3(CNC(c3ccc(Cl)nc3)=O)C2)=O)O1 35642,N1(C(c2scc(C(C)=O)c2)=O)CC(O)CC1CNC(=O)CCOC1CCOCC1 35643,c1(NCC(C(C(C)C)O)(C)C)cc(S(=O)(=O)NCc2ncsn2)ccc1C#N 35644,CCC1=NOC(CC(=O)NCCC(O)C(=O)N2CCCC(CCF)C2)C1 35645,CC1(F)CN(C(c2c(Cl)ccnc2F)=O)CCN(C(c2c(F)ccnc2Cl)=O)C1 35646,c1(CC)ccc(C(N2CC(CO)(NC(=O)C=Cc3cncn3C)C2)=O)cc1CC 35647,N1(C(c2c(C)nccn2)=O)CC2CC(C(=O)NCCCCCC(C)C)C(C2)C1 35648,C1(C2N3CCCC(C)(C3)CCn3cc2nn3)CCCCN(C2CCC2)C1.COCC 35649,CCCCCCCCCC(=O)NC1COCCN(C(=O)CC2CCCCCO2)C1 35650,C(=O)(CCCCCNC(C1C(C)(C)C1(F)F)=O)NCc1nc(CC)sc1 35651,C12(C(=O)NCC(CN(C)C(C3CC4CC4C3)=O)O)CC(C)(C1)OC21CCC1 35652,C(=O)(C(CO)C(F)(F)F)N1CC(CCC)C(NC(C2CC(C)(C)CCO2)=O)C1 35653,C(=O)(C(F)C(F)(F)F)N(C)CCNC(C1CCC(Oc2ccncc2)C1)=O 35654,C1(C(N(CCCF)C)=O)CCCCN(C(C2(N(C)C)CC2)=O)C1 35655,CC1CC(=O)NC(C(=O)NCCOCCC(=O)NC2(C(N)=O)CCCCC2)C1 35656,c1(CCCCN(CC)Cc2nnnn2C)ccn(CC(F)(F)F)c(=O)c1 35657,c1(N2C(C(=O)OC)CN(C)CC2)ccc(S(=O)(=O)N2CCCCCC2)cc1 35658,c1(C(N(CC#C)CCO)=O)ccc(C#N)cc1Cl 35659,CCC(C)C(C(=O)N(CC(C)(C)C(=O)N(CC1=CCSC1)C)C)N(C)C 35660,Cc1cc(C)c(C(=O)N(C(C)CCNC(=O)COCCF)C)[nH]1 35661,C=C(CNC(C1CC1SCC)=O)CCNC(c1ccoc1C)=O 35662,CCCCCC(CC)C(=O)NC(CNC(c1nocc1C)=O)CO 35663,c1(C(N2CCC(NC(Cn3c(C)ncc3)=O)CC2C)=O)cc2cccn2cn1 35664,c1(C(=O)NC2C(NC(C(C)O)=O)COC2)cnc(C2CCC2)nc1O 35665,CCCC(C(=O)NC)NC(=O)CC1(CSC2CC(C)(C(=O)NC)C2)CC1 35666,N1(C(CCNC(=O)C=CCl)=O)C(CNC(=O)CC2(O)CCC2)CC2CCCC12 35667,c1(C(C)NC(CC2C(C(N3CCC(SC)C3)=O)C2)=O)nccc(C)n1 35668,C1(CCC)CCCCN1C(=O)CSCCNC(=O)CCc1ncc[nH]1 35669,N1(C(C=CS(C)=O)=O)CC(NC(=O)Cc2cccc3c2CCC3)C(C2CC2)C1 35670,C(C(C)C(C)C(=O)NCC1(C(=O)NC2CCC(=O)N(C)C2)CC1)OC 35671,C1(C(=O)NCCC(C)CCNC(=O)COC(F)(F)F)C(F)(F)C12CCC2 35672,CCC(Cc1ccccc1C)C(=O)N1CC(NC(c2csc(CO)n2)=O)C(C)C1 35673,C1(C(CNC(C2CC(=O)NC2)=O)O)CCN(C(c2ccc(Cl)cc2)=O)CC1 35674,c1(C(N2CC3(CC(NC(CCCCOC)=O)C3)C2)=O)cc(F)c(O)c(Cl)c1 35675,C1(CC=C)(NC(C2CCC(=O)N2C)=O)CCN(C(c2ocnc2C2CC2)=O)C1 35676,C1(C(=O)OC)(CC)CN(C(c2ccc(C(F)F)o2)=O)C1.N(CCC1CC1)OCC 35677,N1(C(C2N(C(CC(C)(C)C)=O)CC(O)C2)=O)CCC(N=[N+]=[N-])C1 35678,N1(C(C(C)=NOCC#N)=O)CC2CCCC2(C(=O)NC(C(C)C)C2CCC2)C1 35679,C(=O)(C(C)(C)CCCO)NC(C(C)(C)C)CNC(C1C2CNCC12)=O 35680,Cc1nocc1NC(=O)CNC(=O)CC1CC1CNC(c1ccc(F)s1)=O 35681,N1(C(CCCCC)=O)CCCC(NC(c2cnn3cc[nH]c23)=O)C1C 35682,C1(C(N(CCN(C(=O)CN2CCNC(=O)C2)CC)CC)=O)Cc2cc(Cl)ccc2O1 35683,N1(C(C(COC)NC(C2CCC(=O)C2)=O)=O)CC2(CNC(=O)C2)C1 35684,N1(C(c2c(CNC(C3C(C)CC(=O)CC3)=O)n[nH]c2)=O)CC2CCCC(C1)N2C 35685,c1(C(=O)NCC(CN(C(c2nc(CC)oc2)=O)C)C)ccc2c(c1)nc(O)n2C 35686,c1(OCC)cc(NC2CC(NC(c3ccc(C)c(F)c3)=O)C2)nc(OC)n1 35687,C1(C)(CNC(CN(C)C(N)=O)=O)CN(C(=O)CC2CCCC23CC3)CCO1 35688,C1(CNC(CCC(C)OC)=O)CN(C(c2nnn(C(C)C)c2C)=O)CC(C)(C)C1 35689,N1(C(CN2CC(C)(C)C2)=O)CC2CCN(C(c3nccc(Cl)c3O)=O)C(C2)C1 35690,c1(C(N2CC3C(NC(C(C)OCCC#C)=O)C3C2)=O)ccc(Cl)c(F)c1F 35691,c1(OC)cccc(C(=O)NC2CCC(NC(C3CC3c3cccs3)=O)C2)c1F 35692,N1(C(Cc2cc(C)nn2C)=O)CC(NC(=O)C=Cc2cnco2)CC(C)C1 35693,C1(C(=O)NCC2(n3cncn3)CC(=O)C2)C2CCC1(c1ccc(OC3CC3)cc1)C2 35694,c1(CC)ccc(C(=O)NCC(CO)NC(c2ccc(C)cc2C)=O)cc1C#N 35695,n1(CC)cncc1C(c1nnnn1C1COC1)NC(c1cc(C)on1)C 35696,c1(COC)c(C(=O)NCCC2(OC)CCSC2)oc2ccccc12 35697,c1(CN(C(=O)C(N2CCN(C3CCCN(C)C3)CC2)=O)C)c(F)cc(F)cc1Br 35698,CC1(C)CCC(Cn2cc(C3CCCO3)nn2)O1 35699,CC(C)(CC1CCOC1)C(=O)NCC1CCN1CC(O)COCC1CCOCC1 35700,N1(C(c2c(OC)scc2)=O)CCC(NC(=O)CC2(CO)CC2)CC1C 35701,C1(NC(C2(OCC)CCSCC2)=O)COCCN(C(c2csnc2Cl)=O)C1 35702,N1(C(=O)CCc2cc[nH]n2)CCC2(CCCN2C(c2ccccc2Cl)=O)C1 35703,O=C(CC1=CCCCC1)NC1COCCN(C(c2cc3n(c2)CCC3)=O)C1 35704,N(C1=NC2CCCCC2N1)CC(COc1ccc(COC)cc1)O 35705,C(C(C)(C)CN(C(=O)C(CC1CC1)NC(=O)CCOCC1CCC1)C)OC 35706,c1(C(=O)NC2CC(F)CN(C(C3CCCO3)=O)C2)nnn2c1CSCC2 35707,C(=O)(C(C)(F)C(C)(C)F)N1CC(C)C(n2cc(-c3ccc(C#N)nc3)nn2)C1 35708,C#CCC(CC(=O)NC(c1cccc(C)c1)C)NC(c1ccc(O)nc1)=O 35709,c1(NCc2cnn(C)n2)coc2c1C(O)CCC2.Cc1ccon1 35710,Cc1nn(CC(N2CCCC(C(C)NC(=O)Cn3nnc(=O)[nH]3)C2)=O)c(=O)o1 35711,C1(C(=O)NCC=CCC)CC2C=CC1N(C(=O)CCNC(=O)OC)C2 35712,N1(C(C2CCC(C)O2)=O)CC(CNC(c2cc3ccccc3o2)=O)OC(C)(C)C1 35713,C1(N(c2ccccc2)CC(=O)NCC2CC2)C2CN(C(=O)C(F)=C3CCC3)CC12 35714,N1(C(C(F)=CC)=O)CCC2(NC(c3cccc(C)c3C)=O)CCCCC12 35715,c1(C(N2CCCC(CC(=O)Nc3cnc(Cl)nc3)C2)=O)cnc2ccccn12 35716,N(C1CCc2cc(CNC(C3(O)CCCCC3)=O)ccc21)C(C(CCC#C)O)=O 35717,C(CC)(CCC(=O)NC(c1ccc(Br)cc1OC)c1nnnn1C(C)CC)NC 35718,c1(C(=O)NC2CC3CN(c4nc(SC)nc(C)c4)CC32)ccc2ncsc2c1 35719,C1(c2ccc(C)o2)CSCCCN1CCN1CC(C)OC(C)C1 35720,C1(C(=O)NC2COCCC2C(=O)N(CCC(N)=O)C(C)C)(OC)CCOCC1 35721,Cc1cc2cc(C(N3CCC(OCCNC(c4ccoc4)=O)C3)=O)[nH]c2cc1Cl 35722,C(CC)(CC(=O)NC(C)C(F)(F)F)NC(C1(CC#C)CCCC1)=O 35723,S(=O)(=O)(CC(=O)NCCC(C)NC(=O)Cc1nnc(C)o1)NCC 35724,Cc1cc(F)ccc1C(=O)NC1CCCN(Cc2scnc2C)C1 35725,Cc1cc(C(=O)N(CCCCN(C)C(c2ccc(CO)nc2)=O)C)c(Cl)cc1F 35726,N1(C(C2CN(C(=O)C=Cc3ccsc3)CC2F)=O)CC2(CO)CC2(CO)C1 35727,C(CC(=O)NCCC(COC)OC)(C(C)C)NC(C(CC)(C)C)=O 35728,CC(=O)n1ncc2ccc(-c3c[nH]c(=NCCN4CCOC4=O)s3)cc12 35729,c1(OCC)nccc(C(=O)NC2CC(CNC(c3cccnc3S)=O)C2)c1F 35730,c1(NC(C2C(NC(c3c(C(C)C)cccc3)=O)CCC2)=O)cccc2c1OCO2 35731,C(c1cnn(C)c1)=CC(=O)NCC(COC)NC(c1csnn1)=O 35732,c1(C(=O)NC2CC(C)N(C(c3cnc4[nH]ccc4n3)=O)C2)cccc2nn[nH]c12 35733,c1(C(=O)NCCN(C(CCC#C)=O)CCC)cc(Br)c(OC(C)C)s1 35734,CCCCN=C(NCC1(O)CCC1)NCC1CCCCN1S(C)(=O)=O 35735,CC1CN(C(=O)CCCc2cnn[nH]2)CCC1NC(=O)Cc1cncc(Br)c1 35736,C(=O)(CC(C)CNC(C1(CCNC(C)=O)CC1)=O)N(C(C)C)CC 35737,C1(NC(c2cc(CC)sn2)=O)C=CCN(C(c2nonc2N)=O)C1 35738,C(=O)(C(F)CCC(C)C)N1C(CC)(CC)CC(NC(c2ccn(COC)n2)=O)C1 35739,c1(NC(C)=O)ccc(F)c(C(N2CCCC2Cn2cc(C(C)(C)C(N)=O)nn2)=O)c1 35740,CCC(CC(=O)NCc1ncc(C(N2CCCC2(C)C(=O)OC)=O)cn1)C(C)(C)C 35741,CCC(C)(C)OCC(=O)N(CC(CC)NC(=O)Cc1ccsn1)C 35742,N1(C(c2c(C)nccn2)=O)CCN(C(=O)CC2(O)CCOC2)C(CC2CC2)C1 35743,C1(NC(c2cccc(C#N)c2)=O)CC2CC1CN(C(c1cnc[nH]1)=O)C2 35744,N1(C(C2(COC)CCCC2O)=O)CC2CCC1CN2C(=O)Cc1c(C)cccc1C 35745,C1(NC(c2cc(SC)c(C)o2)=O)(CNC(c2nccn2C)=O)CCCCC1C 35746,C1(C2CCN(C(=O)CCNS(C)(=O)=O)CC2)(NC(C2C(C)CCC2)=O)CC1 35747,CC1(CCNC(C2CC(CCO)C2)=O)CCN(C(C2(CO)CC(F)(F)C2)=O)C1 35748,Cc1ncc2n1CCC(C(=O)NC1(CF)CCN(C(c3ccncc3Cl)=O)C1)C2 35749,C#CCCCCCC(=O)N1CCC2CN(C(=O)C(C)OCC(C)C)CC12 35750,CCCCC(C)CCC(=O)N(CCCNC(C1CCC(OCCC)CC1)=O)CC 35751,c1(CNC2CCC(C(N(CC)CC)=O)CC2)sc2ccccc2c1Cl 35752,c1(OC)cccc(CN2C(=O)CN(CCC3CCCCO3)C2=O)c1Br 35753,c1(OCC)ccc(C(N2CCCC2CC(=O)NCC2CCC2)=O)cc1C 35754,C12(CNC(c3c(CC)cno3)=O)COCCN1CCN(C(C13CCC(CC1)O3)=O)C2 35755,CSC1=C(C(=O)NCC2(CCNC(=O)C(n3ccnc3C)C)CC2)CCCC1 35756,c1(CC)noc(C)c1C(=O)NC1CCCC(NC(c2ccn(CC(C)C)n2)=O)C1 35757,N1(C(Cc2cn(C)nc2)=O)CC(N(C)C(C2CC3CCC3C2)=O)C2(CC2)C1 35758,C1(C(=O)NCC23CN(C(CCN(C)CCO)=O)C(C2)CO3)CNc2ccnn2C1 35759,C1(CC)CCN(C(=O)OC(C)(C)C)C1NC(=O)NCCN1CC(C)(O)C1 35760,C1(NC(CSC)=O)CCCCC12CCN(C(C1CCC1c1nncn1C)=O)CC2 35761,c1(CCC(=O)NCC)ncccn1.O=C(O)C(O)C1(CC2CCCC2)CC1 35762,C1(CNC(C2(CC(=O)OC)CC2)=O)C2CCCC1N(C(c1[nH]cnc1C)=O)C2 35763,c12ncnc(C3CCCO3)c1-c1nc(C3CCC(F)(F)CC3)nn1-2.CCC 35764,CCCCCCCCC(CO)NCc1cc2nc(Br)sc2[nH]1 35765,N1(C(C2(CC=C)CC2)=O)CCC2(CC1)CC2(CO)CNC(=O)COC 35766,Cc1nc(C(=O)N(CC(C)NC(C2(C3CCCO3)CCC2)=O)C)c2ccccn12 35767,Cc1c(C(=O)NC2(C3CCCN(C(C4CCO4)=O)C3)CC2)oc2ccc(F)cc12 35768,c1(-c2ccc(NC(CSC(C)=O)=O)cn2)ccc2c(c1)OCCN2C 35769,C1(OC)CC(CNC(c2cccc(F)c2)=O)N(C(c2cnn(C3CC3)c2)=O)C1 35770,c1(CC)cc(C(=O)NC2CC(CC(=O)NCCCC(C)(F)F)C2)ncn1 35771,c1(C(=O)NC2C(NC(c3cc(C)nc(C)c3)=O)COC2)cc2nccn2c(O)n1 35772,C1(C(=O)NCC(CNC(C(n2c(C)nnn2)(C)C)=O)F)CCc2nc[nH]c2C1 35773,N1(C(C2C(C)CCO2)=O)CCCCC2(C1)CN(C(c1coc(CC3CC3)n1)=O)C2 35774,C1(NC(c2n(CCC)ncc2)=O)CCCCC12CCN(C(C1CC1CF)=O)C2 35775,CCCC(C(=O)NCC1(C)CCCN1C(=O)C(F)C(C)C)OCC 35776,C(C)(CCCC(C)C)(OCCN(CC1CC(=C)C1)Cc1cncs1)SC 35777,S(=O)(=O)(c1ccc(C(=O)O)cc1F)NC(c1n(CC)ncc1[N+](=O)[O-])=O 35778,CCCC(C)(O)CC(=O)N1CCC1C(=O)NCC.c1(C(=O)OC)cc(CC=O)ccc1Cl 35779,N1(C(C(C)=C2CC2)=O)C2CCC1C(C(=O)NC(c1ccns1)C)C2 35780,c1(C(=O)NCC2(S(N)(=O)=O)CC2)cc2ncc(-c3nn[nH]n3)cc2[nH]1 35781,N1(C(C2CC(=C)C2)=O)CCN(C(C2CCS(=O)(=O)CC2)=O)C2CC12 35782,N1(C(CSCCC)=O)CCC(C2CC(NC(c3nc4nc(C)ccn4n3)=O)C2)C1 35783,c1(C(=O)NCC(CN(C)C(c2ccnn2C(F)F)=O)O)coc2ccc(O)cc12 35784,CC(CCC1CC1)N=c1nc2sccc2c(NCCCCNC2CCCCC2)[nH]1 35785,Cc1[nH]nc(CNC(=O)C(c2cccs2)NC(=O)C=Cc2cncs2)c1C 35786,c1(CC)cc(C(N2CCC(CC(=O)N(CC(C)C#N)C)C2)=O)on1 35787,N1(C(c2cc(CC)n(C)n2)=O)CC2CC(NC(C3CC4CCC4C3)=O)C(C2)C1 35788,C1(COC)CN(C(=O)C(C)(C)n2cccn2)CCN1C(c1cc2n(c1)CCC2)=O 35789,c1(C(=O)NCCC2N(C(CSc3onc(C)n3)=O)CCC2)c(C)cccc1C 35790,Cc1c(C(=O)NCC(C)(C)OCCNC(=O)C(C)C(C)C)cnn1C(C)C 35791,Cc1ccc(C(N2CCCC(C)(NC(=O)Cc3csc(S)n3)C2)=O)c(Cl)c1 35792,C1(CNC(C2(CCC)CC2)=O)(NC(C2CC3C=CC2O3)=O)CC(F)(F)C1 35793,N1(C(c2ccc(C(=O)NC)o2)C(=O)NC2CC2)CCOC(c2nccs2)C1 35794,C(=O)(C1CCCn2cncc21)N(C1CCN(C(CSC2CCC(=O)N2)=O)CC1)C 35795,n1(CC(N2CCC(C3CCN(C(=O)CC4CC4)C3)C2)=O)ccc2ncc(Br)cc12 35796,N1(S(c2c(C)ccc(C(CC)=O)c2)(=O)=O)CCOC2(CCC(C)CC2)C1 35797,N1(C(C)C)CCCC1CNC(=O)CC1CCN(C(c2ccsn2)=O)C1 35798,C1(CC(=O)NC(C2CC2)C2CC2)COCCN1CC 35799,c1(C(=O)NC(C2CCN(C(c3c(C)cn(C)c3)=O)CC2)C)ccc(Cl)cc1F 35800,[N-]=[N+]=NCCCC(=O)N1CCN(C(=O)CN2CCOCC2=O)CC1C1CCCC1 35801,Cc1[nH]c(C)c(C(=O)NCC2CN(C(c3cn(C(F)F)cn3)=O)CC2C)c1C 35802,c1(CC)onc(C)c1C(N1CCCC(NC(=O)COCCCCC(C)C)C1)=O 35803,Cc1ncc(Cl)c(C(=O)NCCN(C(=O)C(c2cc(F)cc(F)c2)C)C)n1 35804,N1(C(C(C(CC)C)O)=O)CC(NC(C2OCC2(C)C)=O)CC(C)(C)C1 35805,c1(CC(C(=O)NC2(CNC(C(C=C=C)C)=O)CC2)O)ccc2sccc2c1 35806,c1(C(=O)NCC2N(C(C3CC(C)(C)O3)=O)CCN(C)C2)ncnc2c1ccn2C 35807,C1(CCC)(CO)CCN(C(=O)C(CNC(=O)C(CO)OC)CC2CCCC2)C1 35808,c1(C(N)=O)cc2c(N3CCC4(CCN(C(=O)COC5COC5)C4)C3)[nH]cnc-2n1 35809,c1(C(=O)NC(CNC(c2ccc(C)nc2O)=O)(C)CO)nccc2ccccc12 35810,C1(C(N2CCCC(=C)C2)=O)CC1C1CN(C(=O)CC2CCC(=O)NC2)C1 35811,Cc1cc(F)ccc1CC(=O)NCC1CC2(CC2)CN1C(=O)C(C)CF 35812,O=C(C#CC1CCCOC1)NC1CCCC2CN(C(c3cncs3)=O)CC12 35813,CC(C)=C=CC(=O)NC(C)CN(C)C(c1ccc(CN2CCCC2)cc1)=O 35814,C(C(C(=O)N1CC(C(N)=O)C2(CC2)C1)C(C)(C)C)NC(C(C)(C)Cl)=O 35815,C1(CNC(=O)Cn2cncn2)(NC(c2cc(Br)no2)=O)CCCC1 35816,C1(SC)CN(C(=O)CCN2CCCS2(=O)=O)CC1NC(=O)C#CC1CC1 35817,C1(NC(C2(CC=C)CC2)=O)CN(C(=O)CCCc2csc(C)n2)CC1F 35818,C1(NC(CN(CC(=O)NC(C)C)C)=O)CCCCN(C(=O)CC2CCOCC2)C1 35819,CC(CC(=O)NCCOC1CN(C(=O)CC2CC2)C1)C1CCCO1 35820,c12cc([N+](=O)[O-])c(Br)cc1O2.C(C(CC(=O)O)c1ccc(Cl)cc1Cl)(C1CC1)OC 35821,C#CCCCCCC(=O)NC(C)CN1CCN(C(=O)CC2CSCCS2)CC1 35822,Cc1nc(SCCC(=O)N(C2CCN(C)C2)C(=O)Cc2c[nH]nc2C)n[nH]1.CC 35823,c1(C(=O)NCCCCNC(C2CCCN(C(C)=O)C2)=O)cc(F)c(F)c(F)c1 35824,C1(C(=O)NC(CCC)Cc2ccccc2)CC2CC(=O)C1O2 35825,C1(C(C=O)C)CCCN(C(=O)C(F)(F)c2nccs2)C1.CC(C)NCCN(C)C 35826,C(=O)(CCCCC(C)(C)C)N1CCC(CNC(Cc2ncc(C)s2)=O)C1(C)C 35827,Cc1nc(C2CCCCC2)nc(O)c1CCC(=O)N1CC(NC(=O)CO)C1 35828,c1(CN2CCC(N(C(c3c(C=C)cccc3)=O)C)C2)c(Cl)ccc(F)c1F 35829,N1(C(c2c(Cc3n(CC#C)ccc3)n[nH]c2)=O)CCC(C)C1C(=O)NOCC 35830,C1(O)(NC(CCSCC)=O)CCCN(C(C2CCN(C(=O)OC)C2C2CC2)=O)CC1 35831,N1(C(CCCOC)=O)CCC(F)(CNC(C2CCOC2C)=O)CC1 35832,C1(NC(C=CC(=O)N(C)C)=O)CCCN(C(c2coc3c2COC3)=O)CC1 35833,n1(CC(=O)NC2C(CNC(=O)CCc3ccon3)CC2)ccccc1=O 35834,N1(C(CC(CC)OC)=O)C2CCC(C(=O)NCC34CC(C)(CCO3)C4)C1CC2 35835,N1(C(CCN(CCCCOC)C)=O)CC(F)(F)CC1CNC(=O)Cc1cc[nH]n1 35836,Cn1nc(C(=O)NCCC2CCC(NC(C3(CF)COC3)=O)C2)cc1Cl 35837,C1(C#N)(C(N2C(C)CN(C(CCC(C)OCC)=O)C(C)C2)=O)CC2CCC1CC2 35838,c1(OC)cc(C(=O)NCCN(C(=O)CCCc2cccc(Cl)c2)C2CC2)cc(Cl)n1 35839,C1(C(=O)NCC2(OC)CC2)CCCCC1NC(=O)C(C)(C)C1CC1 35840,C1(C(=O)NC2CCC(NC(Cc3ccn(C(C)C)n3)=O)C2)CC2(CCO2)C1 35841,Cc1cccc2c1CC(C(N1CCC(N(C)C(c3occc3Cl)=O)C1)=O)O2 35842,Cc1c(C(=O)NC2CCC(NC(=O)CC(O)C(C)C)CC2)cccc1F 35843,c1(C(N(C2CN(C(C=CC)=O)CC23CC3)C)=O)cnc2c(C)cccn12 35844,N1(Cn2c(C)ncc2)CCCC(C(=O)NCC2=CCCCC2)C1 35845,c1(SCCC(=O)NC2CCN(c3ncc(C(=O)OCC)s3)C2)ccc(Cl)cc1 35846,N1(C(C=C)=O)CCCC1C(=O)NC(c1cccnc1)c1ccccc1 35847,CN1CCC(C)(C(N2CCOCC2CNC(=O)CC2CCC2)=O)C1=O 35848,C1(CNC(c2c(CC)cccn2)=O)CN(c2cnc(F)cn2)CC2(CCC2)O1 35849,C(=O)(CS(=O)(=O)C1CC1)N1CCCC(CC2N(C(COC(CC)C)=O)CCC2)C1 35850,c1(CC)cc(C(=O)NCC2CCCN(C(=O)CC3CC(F)C3)C2)cc(O)n1 35851,N1(C(C2(COC)CCCO2)=O)CCCN(C(c2cnn(C3CC3)c2C)=O)CCC1 35852,C1(CNC(=O)Cc2ccc(Cl)s2)CN(C(C2CC3(CCCO3)C2)=O)CC12CCC2 35853,N1(C(CCC=CC)=O)CCOC(C)C1C(=O)NCCC(C)C(C)C 35854,[N-]=[N+]=NCCCCC(=O)N1CCC=C(C(=O)NC2CNC(=O)C23CC3)C1 35855,C1(C(c2n(CC(=C)C)nnn2)NCC2(OCC)CCCOC2)CC2(CCC2)C1 35856,n1(CC(=O)NCC(CNC(C(C2CCC2)OC)=O)OC)cc(COC)nn1 35857,N1(C(C(CCC)NC(c2cccc3cc[nH]c23)=O)=O)CCC2CCC(C1)S2 35858,C1(C(=O)NC(CCC)C(=O)NCCS(C)(=N)=O)CCCCC1(C)C 35859,Cc1ccnc2sc(CNC(=O)C(=O)NCC3CCOC(C(F)(F)F)C3)c(C)c12 35860,N1(C(C)C(=O)NCCN(C(c2ccc(C(=O)N(C)C)o2)=O)C2CC2)CCCCC1=O 35861,C1(NC(C2CC(=C)C2)=O)(COC)CCCN(C(c2ccc(F)c(Cl)c2)=O)C1 35862,c1(C(=O)NC23CC(NC(CC(C=C)C)=O)(C2)C3)cc(NC(C)=O)ccc1C 35863,C(=O)(C(C)CCC(C)(C)C)NC1(CO)CC(NC(C(c2ncc(F)cn2)C)=O)C1 35864,CC(O)C(C(=O)NCCOc1cccnc1)NC(C1(n2ccnn2)CC1)=O 35865,c1(NC2C(CC)CCC2)nccc(Sc2cccc(N3CCN(C)CC3)n2)n1 35866,N1(C(C=C(CCC)C)=O)CC(Nc2nnco2)C2CC2C1 35867,c1(C(N(CC)CC2(C(C)(F)F)CC2)=O)ccc(CNC(=O)Cn2cnnc2)o1 35868,N(C(=NCC1(C)CCN(C(=O)CC(C)C)C1)NC(C)C)C(C#C)CCC 35869,S(=O)(=O)(c1cccc(Cl)c1)CNC(C1CCCN(S(C2(CC=C)CC2)(=O)=O)C1)C 35870,Cc1ccc(C)c(OCc2ccc(C(N3CC(N4CCCS4(=O)=O)C3)=O)cc2)c1 35871,N1(C(c2c(CCC)occ2)=O)CC(C)(C)OCC1CNC(=O)C(C(C)C)SC 35872,C(=O)(C(F)C(C)C)NC(CN(C(Cc1ccn(CC)n1)=O)C)CC 35873,N1(C(C2CCC(CC)O2)=O)CC2CCC2(CNC(c2cccc[n+]2[O-])=O)C1 35874,c1(C(=O)OC)c[nH]c(C)cc1=NC(=O)NC(C1CCN(CC(N)=O)C1)=O 35875,N1(C(c2cc(F)c[nH]2)=O)CCCOC2(COC2)C1 35876,Cc1nn(C)c(NC(=O)OC(C)(C)C)c1CNC(C12CCC(CC1)O2)=O 35877,C(=O)(C(CCCC(=O)NCC)OC)N(CC(C)N(C(=O)OC(C)(C)C)C)C 35878,C(=O)(CC(C(F)F)NC(C1CC1(Cl)Cl)=O)N(CC)Cc1ncn(C)n1 35879,c1(CC)ccc(F)c2[nH]ccc12.O=C(C(=O)N)NCC1(CNC(C2CCC2)=O)CC1 35880,C(=O)(C(O)C(C)(C)C)NCC1(O)CN(C(C2(CC=C)CCC2)=O)C1 35881,Cc1cc(C2CCN(C(=O)NCC3CC34CCOC4)CC2)cc(C)c1 35882,C=CCC(C)(C)CC(=O)N(CCNC(c1c(C)coc1C(C)C)=O)CCOC 35883,N1(C(C2C(CCOC)C2)=O)CC2(CC(NC(=O)C=CCN(C)C)CO2)C1 35884,n1(CC)c(-c2cccs2)nnc1S.CCC(C)CNCc1nnnn1C(C)(C)CC 35885,C(c1c(Cl)nc2sccn12)=CC(N1CC(NC(C2CC3C=CC2O3)=O)C(O)C1)=O 35886,c1(CCNC(c2n(CCC)nnn2)c2cnc(C3CCCO3)s2)cccnc1C 35887,Cc1nc(O)nc(C)c1C(N1CC=C(CNC(=O)CCCN(C)C)CC1)=O 35888,Cc1ccc(F)cc1C(N1CCC(C(=O)N(C)CCn2cncn2)(C(C)C)C1)=O 35889,CCCN=C(NCC(C)(C)CC)NC1CCN(C(=O)OC)C(C)C1 35890,CC1CCN(C(=O)CCn2cccc2)CC1NC(c1ccnc(OC(F)F)c1)=O 35891,Cc1ccnc(C)c1C(=O)NCC1CC(C)N(C(=O)C=CCN(C)C)C1 35892,c1(-n2c(CCOC(F)F)nc(C(C)OC)n2)cccc2nc[nH]c12 35893,C12(NC(c3n(C=C)nnc3)=O)CCN(C(c3c(Cl)cnn3C)=O)CC1C2 35894,c1(C(N2CC(NC(C3CN(C)C(=O)C3)=O)C(O)CC2)=O)nccn2nccc12 35895,c1(C(=O)NC2CC3CN(C(c4c(N)cccc4F)=O)CC32)cnn2c1CCCC2 35896,C(CCCCC(=O)N1CCOCC(CNC(C2CC23CC3)=O)C1)OCC 35897,C1(NC(C=C(C)C(C)C)=O)CCCCCC1C(N1CCC(C)C1)=O 35898,C1(CC=C)(NC(=O)CC2CCCN2C)CCN(C(=O)CCC)C1.C(C(C)(C)C)C(=O)O 35899,C1(N(C(=O)C(F)Cc2ccccc2)C)CCCN(C(=O)OC(C)(C)C)CC1 35900,C1(C(=O)NC2CC2C2CCCN(C(C3CCCO3)=O)C2)CCCCC12OCCO2 35901,C1(NC(C2C(C)=CCS2)=O)CN(C(=O)C(c2cccnc2)C)CC1(C)C 35902,C12(CNC(=O)CSC(F)F)CCC(C1)N(C(C1CC(=C3CCC3)C1)=O)C2 35903,N1(C(C(C)c2cccs2)=O)CCC2(CCN(C(c3cnn(C)n3)=O)CC2)C1 35904,c1(SCC#C)cccc(C(=O)NCC(O)CN(C(=O)CCN2CCCC2)C)c1 35905,Cc1cc(C(N2CCC2(C)C(=O)Nc2cnc(Br)c(C)c2)=O)ccc1O 35906,CCCCC(F)C(=O)NCC1C(C(N2CCCC(N3CCC3)C2)=C(C)C)C1(C)C 35907,c1(C(=O)NC2CCCN(Cc3ccc[nH]3)CC2)cn2c(Cl)cccc2n1 35908,c1(N(C)C)cnc(C(N2CCC(NC(c3ccncc3C(F)(F)F)=O)C2)=O)nc1 35909,C1(NC(CCOC)=O)CC2CCC(C1)N2C(c1cnc(O)c2ccsc12)=O 35910,N1(C(Cn2c(C)nc([N+](=O)[O-])c2)=O)CCC2CCN(C(c3ccsn3)=O)CC2C1 35911,CC1C(NC(=O)C(c2ccc(Br)cn2)(C)C)CCN1C(c1cscn1)=O 35912,C=CC(C)(CC)C(=O)NCC(C)(C1CC1)NC(=O)CCc1nc(N(C)C)no1 35913,C(=O)(CCC(C)(C)NC(=O)CN1CCOCC1)NCCCCN(CC)CC 35914,N1(CC(=O)NC23CC(CNC(Cc4c(C)n[nH]c4)=O)(C2)C3)C(=O)C(C)C(C)C1=O 35915,c1(C(N2CC(C)N(C(C3CCN(S(N)(=O)=O)C3)=O)CC2)=O)nc2cnccc2s1 35916,c1(CC)nn(C)c(CC(=O)NC2CCCN(C(c3oc(C)cc3C)=O)C2C)c1Cl 35917,C12(NC(c3c(C)ccs3)=O)CCCN(C(C3(CS(C)(=O)=O)COC3)=O)CC1C2 35918,CCCCC(O)C(=O)NCC1(C)CCN(C(c2ncccc2C2CC2)=O)C1 35919,N1(C(CN(CCCNC(Cc2c(C)scc2)=O)C)=O)CCOC2CCCC12 35920,C(=O)(CN=c1[nH]c(C)cs1)N1CCC(CNC(c2c(OC)nsc2)=O)C1(C)C 35921,C1(COC)CC(C)(C)CN1C(CC)C(=O)NC1(C)CC1 35922,N1(C(CCCC(C(C)C)(C)C)=O)C2CCC1C(CNC(=O)CCC1CC1)C2 35923,C(CCCCNc1cc(C(=O)OC)no1)SCC 35924,c1(C(N(CCN(C(c2c(C)nn[nH]2)=O)C(C)C)C)=O)cc(Cl)ccc1F 35925,c1(C(N2C(CCNC(CCOCCN(C)C)=O)CCCC2)=O)nnc(O)cc1O 35926,N1(C(c2n[nH]c3c2CCC3)=O)CC2CC3CC2C1C3.C12CCCCCN1C2=O 35927,Cc1snnc1C(=O)NCCOC1CCN(C(c2cnn(-c3nccs3)c2)=O)C1 35928,C(=O)(C1CCCn2ccnc21)NCCCN(C(C(C#N)C1CC1)=O)C1CCCC1 35929,CCC(C)CCCC(=O)N1CC(O)(CN(C(=O)CCc2ccc(O)nn2)C)C1 35930,CC1Oc2ccc(C(N3CCC3CNC(C3(C)CCCS3)=O)=O)cc2NC1=O 35931,N1(C(C2C(C)(C)OCC2)=O)CCC2CN(C(c3ccnc4ccnn34)=O)CC12 35932,c1(C(=O)NC(c2ncoc2C2CN(C(C3(N=[N+]=[N-])CC3)=O)C2)C)ccnc(S)c1 35933,c1(OC)ccc(Cl)c(CC(=O)NC(C)C(C)(C)NC(C2CC(C3CC3)=NO2)=O)c1 35934,c1(C(=O)NCC2CC(NC(c3ncccc3F)=O)C2)cc2c(nc1O)CCCC2 35935,c1(OCC(=O)N(CC(C)NC(C)=O)C)ccc(F)c(Cl)c1.N12CCC(C1)C2=O 35936,c1(C(N)=O)ccc(S(=O)(=O)NC(C2CC(F)(F)C2)CO)cc1Cl 35937,N1(C(C=CCC)=O)CCC(CNC(=O)Cc2ccc3c(c2)OCO3)C(F)(F)CC1 35938,n1(CC)ncc(C(=O)NCC(n2cc(CNC(c3c[nH]c(=N)s3)=O)nn2)CC)n1 35939,CCC(C)CC(C(=O)NC(C)CC1CCC1)NC(=O)CCc1ncnn1C 35940,c1(C(=O)NCC2CN(C(c3ccccc3F)=O)C2)cc2ccsc2c(O)n1 35941,c1(OCC(=O)NCCC(C)N(C(c2cc(C)c(C)s2)=O)C)nn(C)cc1[N+](=O)[O-] 35942,N1(C(CCN(S(C)(=O)=O)C2CC2)=O)CCCC1Cn1cc(CCn2cncn2)nn1 35943,c1(CC(N2CCN(C)C(=O)C2)=O)ccc2n[nH]cc2c1.C1(=O)CC(C)O1.N(C)C 35944,C1(CC)CN(C(c2ccns2)=O)CCN1NC(c1cccn1C(C)C)=O 35945,c1(C(=O)NCCCCC(C)NC(c2cncc(C)c2)=O)cc(S(N)(=O)=O)oc1C 35946,C(=O)(CC(C)C(F)F)NCC(CC)(C)NC(c1nc[nH]c1C(C)(C)C)=O 35947,CC1C2CCC(C2)C1C(N1CC2(C)CC1(C(=O)N(C)CCC1CC1)C2)=O 35948,Cc1ccc(F)c(C(=O)NC2CC2NC(c2ncsc2S(N)(=O)=O)=O)c1F 35949,C1(NC(C)CC(=O)NCCc2ccc(F)cc2)CC(O)C12CC(F)(F)C2 35950,CC(CC(=O)OCC(=O)NCCC1CCN(Cc2ccco2)C1)c1ccsc1 35951,C=C(Cl)CCC(=O)N1CCC(C(F)CNC(c2cn(CCOC)cn2)=O)CC1 35952,C(=O)(C(F)(F)c1cccs1)N.C12(CCC1)C(=O)NCCC2C1CC1.CO 35953,O(C1CCCc2ccccc21)CC(=O)NCC1CN(C(=O)CCF)C2(CCC2)C1 35954,Fc1cc2cc(c1)C(C1CCCC1)NC2.c1(SC2CC2)nccc(C(F)(F)F)n1 35955,c1(OC)ccc(F)c(C(=O)NCC(CNC(=O)C(C)CC(N)=O)CO)n1 35956,C1(NC(C(C2CC2)OC)=O)CN(C(c2c(O)ncc3c2CCC3)=O)CC(C)(C)C1 35957,C(=O)(C(C)(O)C(F)(F)F)NC.c12ccc(cc1)C(=O)NC(C)C1CCCN(C1)C2 35958,c1(OCCC(N2CCC(C(=O)NCC3(n4ccnn4)CC3)C2)=O)ccccc1 35959,C1(NC(CCC(=O)NCCC)=O)CC2CN(C(=O)C=C3CCCOC3)CC12 35960,C1(C2(NC(C(C)OCC=C)=O)CC2)CCCCN1C(c1ccn(C)c1)=O 35961,c1(C(=O)NC(C2(CNC(C3C=CC(C(=O)OC)C3)=O)CC2)C)ccc(Cl)cn1 35962,CC(C)=C=CC(=O)NC(C(=O)NOCC1CCCC1)C1CC=CCC1 35963,C12(C(=O)NC3CC(C(C)NC(c4cnn(CC)n4)=O)C3)CCC(OC)(CC1)C2 35964,N1(C(C(COCC)C)=O)CC2CCC1C(CNC(c1cncc(NC)c1C)=O)C2 35965,N1(C(c2ccc(Cl)nc2)C(=O)NCc2ccc(Cl)cc2Cl)CCc2[nH]nc(O)c2C1 35966,c1(C(=O)NC(CN(C(c2ccn(C3CCC3)n2)=O)CC)C)nc(C)sc1C 35967,C1(C(N(CCC)CCNC(c2cnc(CC(C)(C)C)o2)=O)=O)C=NN(C)C1=O 35968,c1(C(=O)NCC(C)(C2CC2)NC(c2ccc[nH]2)=O)cccc(S(=O)(=O)CCO)c1 35969,C12(NC(CCc3n(C)cnc3)=O)CN(C(c3cccs3)=O)CC1CS(=O)(=O)C2 35970,Cc1cc(C)c(C(=O)NCC2(O)CC(NC(=O)Cn3cc(C(F)F)cn3)C2)o1 35971,C1(C=O)CN(C(=O)OC(C)(C)C)C(C)(C)C1.C(CCOC)CCN(C)C 35972,c1(C(=O)NC(CN(C(=O)CC2CCCC2)CC)C)cc(F)cc(Cl)c1 35973,CCC(C(=O)NC1CCC1C(=O)NC1CCOCC1F)C(F)(F)F 35974,C1(CCCNC(C2(C(=O)NC)CC2)=O)CN(C(c2nn(C)cc2SC)=O)CCO1 35975,N1(CCNC(CCCOC)=O)CCN(C(=O)CCCn2ccnn2)CC1 35976,C(C1CCN(C(=O)CCCN=[N+]=[N-])CC1)=CC(=O)NCc1nc(C(C)C)on1 35977,N12CCCC(C)(C1)C2=O.c1(NC(CCN(C)C)=O)cn(C)nc1C(N)=O 35978,C1(C(=O)NC2C(CNC(CN(C)C(=O)C3CC3)=O)CC2)Cc2ccccc2S1 35979,C1(C(N2CCC3(C(NC(c4cc(O)ccc4Cl)=O)C3)C2)=O)COC2COCC2O1 35980,Cn1cc2c(-c3cnccc3C(N3CCC4(C3)CC4(F)F)=O)cccc2n1 35981,c1(C(=O)NC2CC(CNC(C(CC3CCC3)NC(C)=O)=O)C2)c(F)cccc1Cl 35982,n1(CCC(=O)NC2C(C(=O)NCCC)C2)sc2ccccc2c1=O 35983,CN1CC2(CCN(S(=O)(=O)c3cccnc3NCCN=S(C)(C)=O)C2)CC1=O 35984,N1(C(CCCSC)=O)CCC2CN(C(C3(C)CC4CC4C3)=O)CC2C1 35985,C1(C(=O)NCC(=O)NCCC=C)C2CCC(C2)N1C(=O)C(C1CC1)C1CC1 35986,C1(NC(c2cnn(C3CC3)c2)=O)CC2CN(C(=O)C3=COCCO3)CC2C1 35987,N1(C(c2c(N)cn(C)n2)=O)CC(NC(=O)Cc2cc(Cl)n(C)n2)CC2(CC2)C1 35988,N1(C(CN(C(=O)OC)C)=O)CCC(NC(=O)CSc2nncs2)CC(C)(C)C1 35989,C1(CC)C(OC)C2CCCCCCC12.c12cn(nn1)CC(=O)NC2 35990,N1(C(c2cccc(OC(F)F)n2)=O)CC2CCC(C1)N2CC1CCCO1 35991,c1(C(N(CCCCNC(COCCC=C)=O)C)=O)cc(C#N)ccc1Br 35992,c1(SC)ccc([N+](=O)[O-])c(C(=O)NC2CC(CCNC(=O)CC(C)C(C)C)C2)c1 35993,C(=O)(CCC(=O)N1CCCCC1CNC(C1CN(C(C)C)C1)=O)N(C(C)C)C 35994,C1(NC(Cc2ccc(SC)cc2)=O)CCN(C(c2cccc(I)c2Br)=O)CC1F 35995,C1(C(C)NC(c2ccn(CC(F)(F)F)n2)=O)CCCCN1C(=O)Cc1nncn1C 35996,C1(NC(CSC(C)C)=O)CC2(CCN(C(c3csc(C4CC4)c3)=O)CC2)C1 35997,CN1C2CCC1CN(C(C1CNCCN1Cc1ccc(O)c(O)c1O)=O)C2 35998,Cc1cc(CNC(=O)CC2C=CC(NC(c3ncc[nH]3)=O)C2)n(C)n1 35999,C1(C(=O)NCc2ccc(C)c(C)c2)N(C(=O)CC=C(Cl)Cl)CC12CCCC2 36000,Cn1nc(CO)c2c1CN(C(c1ncc(I)cn1)=O)CC2 36001,C1(C(=O)NCC#C)C(CC)CCCN1C(=O)CC(C)C=C 36002,c1(CCC)ccc(C(=O)NC2CC(F)(CNC(C3(C)CCC(=O)N3)=O)C2)cc1 36003,c1(OC)cc(CC(N2CCC(C)(NC(c3ccnn3C(F)F)=O)C2)=O)cc(Cl)c1 36004,N1(C(CCCCOC)=O)CC2(CCCCN2C(C2(C)CC3CCC2O3)=O)C1 36005,N(C1CCCn2c(C)nnc21)C(N(C12CCC(CC1)C2)CC)=O 36006,Cc1ccc(C(=O)NC2CC(CNC(=O)CNC(c3cccs3)=O)C2(C)C)n1C 36007,Cc1ccc(S(=O)(=O)N(C)C)cc1NC(=O)C(N1CC(C)NC(C)C1)=O 36008,c1(C(C)N=c2ccnc(N(CC(=O)NC3CC3)C)[nH]2)nn(C)c2ccccc12 36009,C1(OCCNC(c2ccon2)=O)CCN(C(=O)CCC2CCCC2)C1 36010,C(=O)(CC(CNC(=O)CN1CCC(=O)CC1)C1CCC1)N(C1CCN(C)C1)CC 36011,C(=O)(CC(c1ccccc1)C1CCCC1)NCC(CO)NC(C(=O)NCC(F)F)=O 36012,c1(CCC(N2CCC(NC(C3(F)C(C)C3)=O)C23CC3)=O)ccc([N+](=O)[O-])cc1 36013,C(=O)(CCS(=O)(=O)c1ccccc1)NCCOCCOC.C(=O)(C(CO)OC)NCC 36014,CCCC(CC)CC(=O)NC1CN(C(=O)CNc2cccc(C#N)c2)CC1F 36015,C1(F)(C(N(CCC)CCNC(C2CC2C(F)(F)F)=O)=O)CC1C 36016,C(=O)(CCCC(=O)N1CCC1CNC(=O)C(C)Oc1ccc(O)cc1)NCCC 36017,C(=O)(CCCCN=[N+]=[N-])NC(CN(C(C1(C2(C)CC2)CC1)=O)CC)C 36018,Cc1cnc(CCNC(=O)CNC(C2CC2C(N)=O)=O)nc1 36019,N1(C(C2N(C(C=C(COCC)C)=O)CCOC2)=O)CC(C2CC2)(CC)C1 36020,N1(C(c2ccc(C)c(F)c2)=O)CCCCCC(NC(C2(C)CC2(F)F)=O)C1 36021,C#CCCC(C(=O)NC1(C(=O)OC)CC1)NC(c1cc(C)no1)=O 36022,N1(NC(c2ccc(C(=O)OC)c(I)c2)=O)Cc2nn(C)c(N)c2C1 36023,Nc1ncc([N+](=O)[O-])cc1C(=O)NC1(CF)CCN(C(C2CC2(F)F)=O)C1 36024,c1(C(N2C(CN(C)C(c3scc(Cl)c3Cl)=O)CCC2)=O)cccc(=O)n1C 36025,CCCC(C(=O)N(C(C)CNC(=O)CC1(OC)CCOCC1)C)c1ccccc1 36026,N1(C(CCC(=O)NC)=O)CCN(C(c2coc(C(C)=O)c2)=O)C(C)C1 36027,C1(C(=O)NC(C2N(C(c3c(Cl)ccc(NC)c3)=O)CCC2)=O)CCc2nccn2C1 36028,Cc1cc(C(N2CCC(NC(=O)Cc3scnc3C)C23CC3)=O)cc(N)c1 36029,C(=O)(C1CCCn2ccnc21)NC1(CNC(C2C(C)CC(=O)NC2)=O)CCC1 36030,N1(C(C)C)CC(NC(=O)CCCN(C(=O)CC2CSCCO2)C)C(C)C1 36031,c1(COC(C2CC2n2ncc(Br)n2)=O)cccc(-n2ccnc2O)c1 36032,C1(COC2CCN(C(CC=C)=O)C2)CCN(C(C2CC(F)C(=O)N2)=O)CC1 36033,CC1CC=C(C(=O)N2CCCC(CC(=O)NC3(CO)CCCCC3)C2)CC1 36034,c1(C(=O)OC)ccc(C(N2CC(CC(C)NC(c3c[nH]cc3C)=O)C2)=O)c(C)c1 36035,N1(C(C(c2ccc(C)o2)C)=O)CC2(CCCC2)C1C(N1C2CCC1(CO)CC2)=O 36036,C1(CCCC)CCN(C(c2cc(CCNC(=O)C(C)Cn3cccn3)on2)=O)C1 36037,C=CCC(F)(F)CN(C(=O)C(C1CCN(C(=O)Cc2cnoc2)CC1)C)C 36038,c1(C(=O)NC(C(C)NC(C2(CCOCC)CCC2)=O)C)cc2c(cc1Cl)CCCC2 36039,c1(NC(CNC(COc2cccc(OC)c2[N+](=O)[O-])=O)C)cn(C)c(=O)cc1C 36040,Cc1ccc2c(c1)CC(N(C)C(C13CC1CN(C(=O)OC(C)(C)C)C3)=O)C2 36041,C1(CCNC(C(C)(C)NC(COC)=O)=O)CN(C(c2nccnc2C)=O)CCO1 36042,N1(C(CC=C=C)=O)CC(C)OC2(CCN(C(c3c(C)nc(O)nc3S)=O)CC2)C1 36043,c1(COC)nc(C)c(C(=O)N(CCNC(c2nc(C3CC3)cs2)=O)C2CC2)s1 36044,C12(CNC(=O)CC3CC(F)C3)CCC(NC(C3CC4CCC4C3)=O)(CC1)CO2 36045,c12cnc3n1CCN(C3)C2=O.c1(C(=O)NCC2CCC(F)C2)cccc(=O)n1O 36046,C1(CNC(c2ccnc(CO)c2)=O)CC2CC2N1C(=O)COCC1CCOCC1 36047,C1(NC(C=Cc2cc(OC)ns2)=O)CCCN(C(c2cccc(F)c2F)=O)C1C 36048,c1(C(C)NC(C2CN(C)C2)=O)ccc(CNC(c2ccc(C#N)[nH]2)=O)cc1 36049,N1(C(c2cc(OC)cc(Cl)c2)=O)CCC2(CCCN(CCn3cccn3)C2)C1 36050,N1(C(COc2cccc(C#C)c2)=O)CC(C2CN(C(=O)C(C)(C)CCCO)C2)C1 36051,c1(CNC(c2cnns2)=O)cnn2c1CN(C(=O)CC1COC(=O)C1)CC2 36052,C1(C(=O)NCc2ccc(C(N(C3CCCC3)CCC#C)=O)s2)CC(C)(C)CN1C 36053,C(=O)(CCCCC#N)NCC(C)(CO)NC(=O)CCC1CCC(F)(F)C1 36054,C1(CNC(C(C#C)(C)C)=O)CCCC2(CCN(C(c3nc(C)oc3C)=O)CC2)O1 36055,c1(CC(=O)NCC(CN(CC(=O)N(C2CCCCC2)C)C)O)cc(F)ccc1O 36056,N1(C(C(CC=C)OC)=O)CC(C(=O)NCc2n[nH]cc2CC)C(C2CC2)C1 36057,n1(CCC)cccc1C(=O)N(C)CCN(C)C(c1cc(C2CCCCC2)on1)=O 36058,c1(C(C(=O)NC(CC(C)NC(CC(CC)OC)=O)C)(F)F)cccc(F)c1F 36059,c1(OC)ccc(F)c(C(=O)NCC2CC3(CC3)CN2C(=O)CC2CN(C)C2)c1 36060,C1(NC(C(CC)CC(C)C)=O)CCCC12CCN(C(=O)CC1CC(F)(F)C1)CC2 36061,N1(C(c2c(C)[nH]cc2)=O)CCC(CO)C(NC(=O)Cc2cn(C)cn2)C1 36062,C(=O)(C(O)CCNC(C1CC1(C)C(F)F)=O)NCc1nnn(CC)n1 36063,C=CC1CN(C(=O)CCS(C)(=O)=O)CC1NC(=O)C(C1CC1)SC 36064,C1(c2n(C)ncc2)CN(C(C2CCC(C(F)(F)F)N2)=O)CCO1 36065,C=Cc1ccc2c(c1)CN(c1nc(N(CCC(N)=O)C)nc3cc(C)ccc13)CC2 36066,N1(C(C2CSCCS2)=O)CC2CCN(C(C3(O)CCSCC3)=O)CC12 36067,N1(C(C(C)(C2CC2)OC)=O)CCN(C(C23CC2COC3(C)C)=O)CC(O)C1 36068,N1(C(C(c2ccccc2F)C)=O)CC(NC(c2c[nH]c(=O)cn2)=O)C(C)C1 36069,C(CCC(=O)OC)(C(=O)Nc1ccccc1)C(C1CC(OC)(OC)C1)=O 36070,CCCCCC(C)(C)C(=O)NCC(CO)NC(=O)Cn1cc([N+](=O)[O-])cn1 36071,C(CCCCCCCO)=CC(=O)NC1C=CC(CNC(=O)CCCCCC#N)C1 36072,C#CCC(CC(=O)NC1CC(CNC(=O)Cc2cc(C)no2)C1)c1ccccc1 36073,C(=O)(CC(C)C(C)C)NCC1(NC(c2cn(CCC=C)nn2)=O)CCOCC1 36074,c1(C(=O)NCC(N2CC=CC(NC(C=CC)=O)C2)=O)cc[nH]c2nccc1-2 36075,C(c1cccc(C)c1)=CC(=O)N(C1CN(C(=O)CNc2ccccc2Cl)CC1F)C 36076,C1(C(=O)Nc2cccc(NC(c3cnn(C)n3)=O)c2)CC2(C1)CC2(F)F 36077,C(=O)(C1CCc2nnc(C)n21)NCC(C)(C)NC(C(C)SC)=O 36078,c1(OCCNC(CC2C3CN(C(C)C)CC32)=O)ccccc1O.C1(C)CCC1 36079,C1(CNC(C2CC(=O)ON2)=O)C(C2CC2)CCN1C(C12CCC(F)(CC1)C2)=O 36080,C(CC(CC)C(=O)NC(c1cnn(C)c1)C(=O)NC(COCC)C(C)C)=CC 36081,Cc1ccc(-n2nnnc2CNC(=O)C(=O)Nc2cnn(CCCCN)c2)cc1 36082,CCCCC(CC(=O)NCC1=C(C)CCC1)NC(C1CC2(CC2)CO1)=O 36083,n1(CC(=O)N(C(CC)(C)C)C2CN(C(=O)Cc3cccs3)C2)nnc(C(C)(C)C)n1 36084,c1(C(=O)NC2CC3(CC(NC(C4C(C(=O)OC)C4)=O)C3)C2)ccnc2[nH]cnc12 36085,N1(C(c2onc(C(C)(C)C)n2)=O)CCCCC(NC(=O)CCCC2CCCO2)C1 36086,C(=O)(C1CCCc2ncc(C)n21)NCc1nnc(C(=O)OC)s1.C=O 36087,c1(OC)ccc(C(=O)C(=O)NC2CCC(NC(C3CC3(F)F)=O)C2)cc1OC 36088,CC1CCCC1(C(=O)NCC12CC(F)(C1)C2)NC(=O)C=CC1(C)COC1 36089,CCCC(C(=O)OC)C(=O)N1CCC(C)(C(=O)NC(c2cncnc2)C)C1 36090,C(C1CCOCC1)=CC(=O)NC1CC(NC(C2(C(N)=O)CCC2)=O)C1 36091,c1(N2C3CC(CNC(C4(OCC)CC4)=O)C2CC3)ncnc2sc(CC)cc12 36092,C=C=CC(C)C(=O)NC1(C)CC(NC(=O)CCc2nc(-c3ccoc3)no2)C1 36093,C(=O)(C(C)(C)CC#N)N(C1CC(NC(c2cn(C)nc2C2CCCO2)=O)C1)C 36094,N1(C(C(N2CCC(O)CC2)C)=O)CCCC(CC(=O)NCCn2cncn2)C1 36095,c1(C(=O)NC(C(C)NC(CNS(CC)(=O)=O)=O)C)cc2oc(C)c(C)c2[nH]1 36096,c1(OCC(=O)OC)ccccc1NC(C)Cc1cnc[nH]1 36097,C1(C(=O)NCC2OCCN(C(C3N(C(C)=O)CCC3)=O)C2)CCCC(=O)N1C 36098,c1(CN(C(CCNC(=O)NC)=O)C)nnc(CNC(C2CC2C(N)=O)=O)s1 36099,C1(C(=O)NC2CCC(NC(=O)Cc3ccccc3F)CC2)(COC)CCOCC1 36100,C=CC(CCC)CC(=O)NCC1CCN1C(c1cc(F)c(N)c(F)c1)=O 36101,N1(C(C2CCN(C)C2=O)=O)CC2CN(C(c3cnc4ccsc4c3)=O)CC2(C)C1 36102,C1(C(N(CCCNC(CNC(=O)CCN2CCCC2)=O)C2CC2)=O)CCCCC1O 36103,N1(C(CC(C)N(C)C)=O)CCCCC1SCC(=O)N(C(=O)CC(C)(C)C)C 36104,C1(CONC(c2cn(Cc3ccc(C)o3)nn2)=O)CC12CCCCC2.C1(C)C(=O)N1 36105,c1(C(=O)NCC(=C2CN(C(c3cc(C(C)C)no3)=O)C2)F)ccc([N+](=O)[O-])cn1 36106,CCC(CNC(C1(C(C)NC(=O)CCC2CCCC2)CC1)=O)CCO 36107,Cc1ccc(C(=O)NCC2(F)CCN(C(=O)CCCC3CC3C)CC2)c(O)n1 36108,N1(C(CC=C)=O)CC(C(=O)NCC2CCC(CO)O2)C(CCC)C1 36109,C(=O)(C(COC)CC(C)C)NCC(CC=C)NC(=O)C(C(C)C)c1cccnc1 36110,C12(C(=O)NCC3(C)OCCN(C(c4cc(C)oc4C)=O)C3)CCCCC1C2(F)F 36111,Cc1ncnc(N2CCC(CCNC(c3ccc(=O)n(CC4CC4)c3)=O)C2)c1F 36112,C1(NC(CC2(OC)CCC2)=O)CCCN(c2nc(-c3ccccc3Cl)ns2)C1 36113,c1(C(N2CCN(C(c3ncc(C)cc3F)=O)CC2)=O)c([N+](=O)[O-])ccc(Cl)c1Cl 36114,C(=O)(C1CCCc2sccc21)NCCC1CCN(C(C2(CC=C)CC2)=O)C1 36115,c1(C(N2CC(CNC(c3[nH]nnc3C3CC3)=O)C2)=O)cc2c(F)cc(F)cc2[nH]1 36116,c1(C(=O)NC2CC(CNC(C(CC)n3cncn3)=O)C2)cc(C)nc(O)n1 36117,C1(C(=O)NCC(CN(C(=O)C=Cc2cncn2C)CC)(C)C)CCCCN1C 36118,C(=O)(C1=CCCSC1)N(CC(C)NC(=O)CCC(=O)NC)CC 36119,CC1CCC(C)(C(=O)NC(C2(CNC(c3coc(N(C)C)n3)=O)CC2)C)CC1 36120,c1(C(=O)NC2(C)CC(NC(c3ccnc(C)n3)=O)C2)cc2nc(=O)ccn2[nH]1 36121,N1(C(c2sc(C)cc2C)C(=O)NCC)CCN(C)c2ccc(C)cc21 36122,CC1(C(=O)NC(CCN(C)C)C(=O)NC2C3CCCCC23)CCC(=O)NC1 36123,C1(C(=O)NC(C#C)C(C)OC)CC(C)CN(C(c2ccncc2F)=O)C1 36124,c1(CNC(NCCOC)=NCCc2cn3c(n2)SCC3)ccc(C#N)c(F)c1 36125,c1(C(=O)Nc2c(C(=O)OC)scc2)ccccc1N1CCNC1=O 36126,C=C=CC(C)C(=O)NC(CNC(c1cc(C)n(CC(F)(F)F)n1)=O)CC=C 36127,n1(CC(=O)NCC2CC(OC)CN2C(=O)CCn2cncn2)ccc(O)nc1=O 36128,C1(NC(c2cncc(OC)n2)=O)CN(C(c2cc(C)c(C)o2)=O)C(C)(C)C1 36129,C(=O)(C#CC(C)(C)C)NCCN1CCN(C(C(=O)NCNC(C=COC)=O)C)CC1 36130,CC1(CNC(=O)CC2CC(=O)NC2=O)CCCN(C(C2CC3(C2)CC32CC2)=O)C1 36131,c1(C(=O)NCCN(C)C(c2cncs2)=O)ccc(S(=O)(=O)NC2CC2)o1 36132,C1CCCCN1C.C1(C(C(=O)NCC)F)CCN(C(=O)Cc2csc(C)n2)C1 36133,Cc1cc2cc(F)cc(C(N3CCC4CCC34CNC(=O)CC3CC3)=O)c2[nH]1 36134,CC(C)CC(O)CC(=O)N1CC(C)C(C)(CNC(C2(C(C)C)CC2)=O)C1 36135,Cc1ccc(C(=O)NC2CCC(C)N(C(=O)Cc3ccns3)C2)cc1N 36136,Cc1ccc(CC(=O)NC2CC2CNC(C2C(C)(C)C2(F)F)=O)cn1 36137,C1(CNC(c2c(SC)cccc2)=O)(NC(C2CC(C)(C)CO2)=O)CCCCC1C 36138,N1(C(C)C)CC2C(C(=O)NCC(c3ccc(Cl)cc3)c3ccncc3)C2C1 36139,c1(NC(N(CC(CC)O)Cc2ccncc2)=O)c(C)nn(COC)c1C 36140,CC1CCCN(C(=O)CC2(C)CCN2C(=O)Cc2cn[nH]c2)CC1 36141,C1(OC)CCC2(CC1)NC(=O)CCN2C(C)C.C12CCC(CC1)C(=O)N2 36142,Cc1cc(C(=O)N(CC(C)C(=O)NCc2nn[nH]c2C2CC2)C)n(C)n1 36143,c1(OC)cc(C(N2CCC(N(C)C(c3sccc3C)=O)C2)=O)ccn1 36144,C1(CNC(CCC(=C)Cl)=O)CN(C(c2c(N)cc(Cl)cc2F)=O)CC2(CCC2)O1 36145,CCC1=C(C(=O)NCCN(C2CCCC2)C(C2CCCC(F)C2)=O)SCCO1 36146,Cc1cc(O)ncc1NC(C1CCC(C2CC2)N1C(c1nnn(C)c1N)=O)=O 36147,CC(C)C(CNC(C1CCC(N(C)C)C1)=O)C(=O)N1CCCC(C)C1 36148,C1(C(=O)NCCCCCN(C)C(c2cccc(Cl)c2)=O)CC(F)(F)C12CCC2 36149,N1(C(CC2N(C(C(C)OCCCC)=O)CCCC2)=O)CCN(C)CC1C.C(C)=O 36150,C1(CNC(c2n(C(C)C)ccn2)=O)CC(C)N(C(=O)CN2C(=O)CCC2=O)C1 36151,N1(C(CSCCN(CC)CC)=O)CC2CCC1C2CNC(c1[nH]cc(C)c1C)=O 36152,Cc1cc(CC(=O)NC2CN(C(C3CCCN(CC)C3)=O)CC23CC3)c(C)cn1 36153,C(=O)(C(CNC(C1CCC(=C)CC1)=O)CC(C)C)NCC(C)C 36154,C(=O)(C(CNC(c1cnn(C)c(=O)c1)=O)CC(C)C)NCc1c(C)nc(C)o1 36155,C1(CCCNC(=O)CC2CCC3CC23)CCN(C(=O)Cc2ccccc2F)CC1 36156,CC1CN(C(c2cc(CF)on2)=O)CC(C)C1NC(c1n[nH]c(CC2CC2)n1)=O 36157,N1(C(COCc2onc(C)n2)=O)CCCC(C(=O)NCc2ccccc2)C1 36158,C=C=CCC(C(=O)N1CCC(CCOCF)C1)NC(=O)OC(C)(C)C.C(C)(=O)O 36159,C1(NC(CCCC=C)=O)CC2CC1N(C(c1ccc(CS(C)=O)cc1)=O)C2 36160,N1(C(C(C(C)(C)C)n2cc(CC3(O)COC3)nn2)=O)C2CCC1CC(F)C2 36161,c1(NC2C(C)(C)OCC2)c(-c2ccccn2)nc2ccccn12 36162,C=CCC(CC)C(=O)NCC1=CCN(CC(O)COC(C)=O)CC1 36163,c1(C(N2CCN(C(c3cn(CC)nc3)=O)C(CO)C2)=O)cccn2c(O)nnc12 36164,CCC(C)(C)C(C)CC(=O)NC1CCC1CNC(=O)Cn1cnc(C#N)n1 36165,CCC(CCC(=O)N1CCC(C(C)(F)F)CC1)OC 36166,C(C(=O)NNC(=O)c1ccc(-c2cn(Cc3cccc(OC)c3)nn2)o1)OC 36167,C1(CC(=O)NC(CSC)C(=O)O)CC(NC(=O)CC2CCC=CCC2)C1(C)C 36168,C1(CC(=O)N(CCC)CCNC(=O)CN2CCS(=O)CC2)COC(C)(C)CO1 36169,C(=O)(C(F)CC(C)(C)NC(=O)CCCCCF)N1CCCC(C(C)C)CC1 36170,c1(C(=O)NCC(C)=CC(N2CCC(O)(C(F)F)C2)=O)cnc(F)cc1C 36171,C1(NC(C2N(C)CC(C)(C)C2)=O)C2CCC1CN(C(c1ccc(F)c(F)c1)=O)C2 36172,c1(OC)ccc2[nH]cc(C(=O)NC(C)CC(C)NC(=O)CSC3CC3)c2c1 36173,N1(C(C(C)OCC(C)C)=O)CCC2(CCC2)C(NC(=O)CSC2CC2)C1 36174,C#CC1CN(C(=O)Cc2ccc(Cl)s2)CCN1C(c1cc(C(C)(C)C)[nH]c1C)=O 36175,C#CC1(C(=O)NCCC(=C)CNC(=O)CN2CCC(OC)C2)CCCCC1 36176,Fc1cc(F)c2c(c1)C1=NC(CC(C)C(F)(F)F)C(=NCC3C=CCC3)N=C(N2)N1 36177,C(CCCC(C)(C)C)NCc1snc(OC)n1 36178,c1(C(N2C(CNC(=O)COC3CCOCC3)C=CC2)=O)ccc(O)nc1Cl 36179,C1(NC(COCCCC#C)=O)CC=C(C(=O)NC2CC3C=CC2CC3)C1 36180,N1(C(c2nc(C(C)=O)sc2)=O)CCC2(CC1)CCN(C(=O)C1=CC(O)CCC1)C2 36181,N1CCC2(CC1)NC(=O)CO2.CCCCCCCCCOc1ccc(N2CC3CC(C2)O3)c(C)c1 36182,c1(C(=O)NC(CCNC(c2c(CC)ncnc2)=O)C)ccc(C(C)(F)F)nc1C 36183,CN1CCN(C(c2cc(CNC(=O)CCc3ccsc3)[nH]n2)=O)CC1CO 36184,Cc1nc(NCC2CCC(NC(=O)C(CO)C(C)C)C2)c2cnn(C)c2n1 36185,N1(C(C(COC)OC)=O)CCc2sc(CNC(c3cc(F)c(C)cc3O)=O)nc2C1 36186,c1(CC)ncc(C(=O)NCC2CC(C)N(C(=O)CC3CCC=CCC3)C2)c(C)n1 36187,C1(C(N2CCCC2CF)=O)C(C2CC2)CCN1OCC.c12csc(c1)C(=O)NC2 36188,C(C)(C)(C(=O)NC1CCC1CNC(=O)CN1CCCC1C)SC 36189,C(C(=O)NNc1ccc(Br)cc1F)OC(C(CCC)CCc1ccccc1)=O 36190,N1(CCC)CCC(N=c2[nH]c(N3CC4COCC(C4)C3)nc(=NC)[nH]2)C1 36191,c1(C(=O)NC2CCN(C(C3CCNC(=O)C3)=O)CC2)ccnc2ncccc12 36192,C1(CC)CN(C(=O)C(C2CCC2)NC(c2ccnnc2C)=O)CCO1 36193,N1(C(Cc2cc(C)no2)=O)CCC2CCN(C(C3CC3C(F)F)=O)C2C1 36194,c1(CN(C(=O)CC2CC2c2cc[nH]c2)CCC)nccn1CCC(=O)O 36195,C#CCN(OC)C(=O)CC1(CNC(c2ccn(CCF)n2)=O)CC1 36196,CCC(O)C(C)(C)C(=O)NCC1CCN(C(=O)CSCCC(C)C)C1 36197,Cc1c(C(=O)NC2CC2CNC(C2COC(=O)N2)=O)[nH]c2c(C)cccc12 36198,C1(CC)CN(C(c2c(F)cccc2Cl)=O)CCN1C(c1cc(CN(C)C)c[nH]1)=O 36199,CC1(C)C(NC(C2COC(=O)C2)=O)CCN1C(=O)COC1CCCC1 36200,c1(CNC(C(CCC)CC)=O)ccc2c(c1)CN(C(C1CCN1S(C)(=O)=O)=O)C2 36201,C#Cc1cnn(CC(N2CCC(c3cc(C)[nH]n3)CC2)=O)c1 36202,C1(C(N(CC(C)(C)NC(C23CC(C4CCC4)(C2)C3)=O)C)=O)CCCC(F)C1 36203,N1(C(C(=O)N(C)C)=O)CC2CCCCC2(CNC(C2(C)CCCCNC2=O)=O)C1 36204,c1(NC(C(CC)(C)OC)c2nnnn2CCCF)ccc(C)c(S(C)(=O)=O)c1 36205,O=C1CCC(C(=O)N2CC3CC(C(=O)NC4CC(N5CCCC5)C4)C3C2)=NN1 36206,C(=O)(C(C)(C)CCCNC(c1cc2cccn2cn1)=O)N1C(C)(C(=O)OC)C=CC1 36207,C#Cc1ccc(C(N2CC(C)CC2C(=O)Nc2cnn(C)c2)=O)cc1C 36208,Cc1nc[nH]c2ncc(C(=O)NCCCC(C)NC(c3cc(C#N)cn3C)=O)c1-2 36209,C(C)(N=c1[nH]c(=NCC(CO)C2CCCC2)c2c(ncn2C)[nH]1)c1ncc(C)s1 36210,C1(C(=O)NC(CC)CNC(c2snnc2C)=O)CCN(S(=O)(=O)NC)CC1 36211,C(=O)(C1=CCCC1)NCCCC(C)NC(CN(C(=O)OCC)C)=O 36212,C1(CNC(c2c(OC)n(C)nc2)=O)C(C2CC2)CCN1C(c1nnn(C)n1)=O 36213,C1(C(=O)NC2(CNC(Cc3scc(C)n3)=O)CCOC2)CCc2c(cnn2C)C1 36214,n1(CC)ccnc1C=CC(=O)NCC1CCC(NC(C2(C(F)F)CCCO2)=O)C1 36215,C(CCCCNC(c1ccn(C2CCOCC2)n1)=O)N(C(C)C)C(c1cnns1)=O 36216,Cn1cc(C(=O)NC2CCCN(C(=O)CCc3ccncc3)C2)c(O)n1 36217,Nc1ccc(Cl)nc1C(N1CCCC(CNC(c2cccc(OC(F)F)n2)=O)C1)=O 36218,N1(C(C(CC)C)=O)CC(CNC(c2sccc2C)=O)OC(C)(C)C1 36219,Cc1cc(N2CCCC(NC(=O)C=Cc3cscn3)C2)ccc1[N+](=O)[O-] 36220,C(=O)(C#CC1CCCOC1)NCC(CCNC(C1CCC(N(C)C)CC1)=O)O 36221,N1(C(C(C)N(C)CC)=O)CCOC(C(N2CCCC(C)(C)C2)=O)CC1 36222,c1(C(N(CCC(C)NC(C2CC2[N+](=O)[O-])=O)C)=O)cncc(Cl)c1Cl 36223,C(N=c1[nH]c(=NC2CCCN(C3CC3)C2)c2ncccc2[nH]1)C1C(C)(C)SCC1 36224,c1(NC(C2CCCN2S(=O)(=O)C(F)(F)F)=O)cc(F)c(Nc2cc[nH]n2)cc1F 36225,Cc1sccc1C(=O)NCC1CCCN1C(=O)CSS(C)(=O)=O 36226,CC1CN(C(c2ccc3sccc3c2)=O)CC(C)CN1C(c1cscn1)=O 36227,N1(C(C(C)OCC)=O)CC(NC(=O)CCc2cnc(O)[nH]2)C2(CCOCC2)C1 36228,c1(OCC(=O)NC2CCC(NC(C(C(C)C)SC)=O)CC2)cc(C)ccc1F 36229,c1(C(N(C2CN(C(c3ccc(CC)nc3C)=O)C2)C)=O)cc2sc(NC)nc2s1 36230,c1(SC(C(=O)N(C2CCS(=O)(=O)C2)CC)C)cc(N(C)C)ccc1OC 36231,c1(SC)nc(N(C)CC2CCCN2C(=O)CCc2cccc(F)c2)cc(Cl)n1 36232,CCC(CC(C)C)C(=O)N1CCC1CC(=O)N(CC(F)F)CCO 36233,c1(CC(N2CC(C3CC3)C2CO)=O)c[nH]c2ccccc12 36234,C1(O)(CNC(C(C)(F)F)=O)CCCN(C(C23CCC(CF)(C2)OC3)=O)CC1 36235,c1(C(c2n(CC(=C)C)nnn2)NC(c2cccc(F)c2)C)cc(F)c(F)cc1F 36236,S(=O)(=O)(C1CCN(CC#Cc2cn(C)nn2)CC1)N1C(C)CCC1 36237,c1(OC)ccc(CN2CC3OCCC23)c(C)c1.c12ccc(s1)CC(=O)N2 36238,C1(c2nnc(C(C)NC(c3cc(C(C)C)[nH]n3)=O)s2)CCCN(C=O)C1.C1(SC)CC1 36239,N1(C(c2coc(CO)c2)=O)CCCN(C(=O)C2=C(Cl)CCC2)C(CO)C1 36240,c1(CC)cc(C(=O)NCCCC(=O)NC(CO)(CO)CO)c(C)o1 36241,Cc1cccc2c1OC(C(N1CC(N(C)C(c3ncoc3C)=O)C(C)(C)C1)=O)C2 36242,C1(O)(CN(C)C(c2ccc(CCN)cc2)=O)CCCN(C(c2nsnc2O)=O)C1 36243,N1(C(C(CC)OCC)=O)CCC(O)(C(C)CNC(=O)CCc2cnco2)C1 36244,c1(CNC(CCC)CCO)cc2ccc(C(=O)OC)cc2o1 36245,C1(C(=O)NC(c2nc(CC)sc2)C)CCC(n2cc(CC3(O)CCC3)nn2)CC1 36246,C1(C(N(C2CN(C(c3cc([N+](=O)[O-])cn3C)=O)C2)C)=O)CCCCC(C)(C)C1 36247,c1(-c2ccc(NC(C)=O)cc2)c(C)ccnc1F 36248,c1(OC)ccc(Cl)c(OC)c1C(=O)NCC1(C)CN(C(c2cc(C)nn2C)=O)C1 36249,N1(NS(=O)(=O)CF)CCCC1C=Cc1cccs1 36250,c1(NC(N(CC(=O)NCCC2CCCCO2)CCC)=O)cn(C2CCC2)nn1 36251,Cc1cncc(C(N2CCOC(CN(C)C(c3cc(Br)oc3C)=O)C2)=O)n1 36252,C1(C(N2CC3(CN(C(Cc4c(C)scc4)=O)C3)C2)=O)CCCC12NC(=O)NC2=O 36253,N1(C(CCOCC#C)=O)CCCN(C(C2CN(CC=C)C(=O)N2)=O)C(CO)C1 36254,C1(C(N(CCCNC)CC)=O)(NC(=O)CCCCC2CC2)CCCCC1 36255,C(CC(O)CC(=O)NC1CC2(C1)CC(NC(=O)CCc1nnc(C)n1C)C2)SC 36256,C1(CN2CCCC2C#N)CC2CCC1(COC)C2 36257,c1(C(=O)NC2CC3N(C(C(C)SC)=O)C(CC3)C2)csc2c(O)ccnc12 36258,C1(NC(CC2C(NC(Cc3c(C)nsc3)=O)CC2)=O)(CO)CC2CCCC12 36259,c1(C(C)(C)C(N(C(C)C)Cc2cccc(F)c2)=O)cc(F)c(Cl)cc1Cl 36260,C1(CC)(CO)CCN(C(C2CN(C(=O)CC(C)NC(=O)NCC)C2)=O)C1 36261,Cc1cc(C)c(C(N2CCOC(CCNC(=O)C(C)(F)F)C2)=O)c(O)n1 36262,C(c1ccc(Br)cc1)=CC(=O)NCCN(C(C1(C)C(C)OCC1)=O)C 36263,CC1(C)CN(C(=O)CC2CCC(=O)NC2)CCN(C(C2(c3ccno3)CC2)=O)C1 36264,c1(CSc2cccc(C(=O)OC(C3(CC)CCC3)=O)c2)ccc2ncccc2c1 36265,C#CCCCCC(=O)NC(C1CCOC1)CNC(C1(C(F)(F)F)CC(=C)C1)=O 36266,N1(C(CCS(C)=O)=O)CC2CCC(CNC(C3C4CCCCCCC34)=O)(C2)C1 36267,C1(OC)CC(NC(=O)C(C)Cn2ccnc2)CN(C(C2(n3nccn3)CC2)=O)C1 36268,c1(CC(=O)NC2CCCC(CNC(c3ccncc3O)=O)C2)cccnc1O 36269,c1(NCC2C(C)CN(C(c3ccc(=O)oc3)=O)CC2)c(F)cccc1[N+](=O)[O-] 36270,c1(SC)ccc(NC(C2CSCN2C(=O)CCCN2CCCC2)=O)o1 36271,N(C(=NCc1cc(C)cc(C)n1)N1CCc2ccc(Cl)cc2C1)C(CC)C 36272,Cc1cccc(C2CC2)c1CN1CCCC(c2ccno2)C1.c1(=O)c(=O)[nH]1 36273,N1(Cc2ccc(-c3c(OC)cccn3)s2)CC(F)(F)CC1CN1CCCCC1C 36274,Cc1c(C(N2CCCC2CN(C)C(C2(O)CC2)=O)=O)sc2cc(F)ccc12 36275,C12(OC)CCCC1N(C(=O)C(c1noc(-c3ccc(OC(F)F)cc3)n1)=O)CC2 36276,C1(CNC(C(=O)NCCC(N)=O)=O)CCN(C(c2coc(N(C)C)n2)=O)CC1O 36277,C1(NC(C2N(C(CNC(=O)OCC)=O)CCC2)=O)CCN(C(=O)CC)C12CCC2 36278,c1(C(N(C(CSC)Cc2ccc(F)cc2)C)=O)cc(P(C)(C)=O)ccc1Br 36279,Cc1cc(F)c(C(=O)NCC(O)CN(C(=O)Cc2c[nH]ccc2=O)C)cc1F 36280,Cc1cccc(-c2nc(C(C)N(C)C)nn2C2CCCCC2C)n1 36281,Cc1[nH]c(C)c(C(N2CCOC(CNC(=O)CC(C)C(F)F)C2)=O)c1C 36282,c1(C(=O)NC(C)CNC(c2cnn(CCO)c2)=O)cc(S(=O)(=O)N2CCC2)c[nH]1 36283,C1(CC(=O)NCc2c(C)cc(C)s2)CCCN(C(c2ccccc2)=O)CC1 36284,C(=O)(C(C(=O)N1CCCCC1CNC(=O)CCOC(F)F)C1CC1)OC(C)(C)C 36285,C1(CNC(=O)CCOCC(F)(F)F)CN(C(=O)COC2CC=CC2)CC12CC2 36286,C#CC1(O)CC(C(=O)NC2CCC(C(=O)NOCC(C)(C)C)CC2)C1 36287,N1(C(c2c(C(C)C)noc2)=O)CCN(C)CC1CNC(=O)Cn1nccc1N 36288,N1(C(COC)=O)CCC(CNC(=O)C(c2cncnc2)C)C(F)(F)C1 36289,c1(C(N(C2CCCC2)CCNC(C(C)OCC=C)=O)=O)cnc2[nH]cncc1-2 36290,C(C(C(C)(C)C)NC(=O)C(C)Oc1cccc(C(C)=O)c1)NC(CCSC)=O 36291,C1(CC)C(NC(=O)COCC(C)C)CCN1C(=O)C(C1CCC(=O)N1)C 36292,NC(=O)CCC(C(=O)O)NC(=O)CC(c1cccs1)n1cccc1 36293,c1(OCC(=O)NC(CC=C)CNC(C2CCCC2(F)F)=O)ccccc1C(F)F 36294,C1(C)(C(N(CCNC(C2CC3C(C2)C3(C)C)=O)CC)=O)C2CC3CC(C2)CC1C3 36295,C1(CN(C(C2CCN(CC)C2)=O)CCOC)CCN(C(C2CC(F)(F)C2)=O)CC1 36296,C(=O)(C(C)(CSC)OC(=O)Nc1ccccc1)NCCC(C1CCCC1)OC 36297,C1(NC(CC(=O)OC)=O)CN(C(c2ncc(Br)cn2)=O)CC1O 36298,c1(C(N2C3C(CNC(C4CC(C)(C)C4)=O)C(C3)C2)=O)ccc2ncc(=O)[nH]c2c1 36299,CCCC(C(=O)N1CCC1C(=O)N(CC(C)(O)C1CC1)C)OC 36300,CC1CCN(CC(=O)NCC2CCC(N(C)C(C3(C4CCC4)CC3)=O)CC2)CC1 36301,C(=O)(C(C(C)C)N1CCCC1)NCC1(C(=O)NCCCCCC)CC=CC1 36302,CC1CN(C(C2CCC(N(C)C)CC2)=O)CC1NC(c1nncs1)=O 36303,N1(C(C(C)n2ccnc2)=O)CCC2(CCC2)C(NC(=O)CCc2cnoc2)C1 36304,C1(O)(CC(N2CCC(NC(C(C)N(C(C)=O)C)=O)C2)=O)CCOCC1 36305,N1(C(C2(CC)CN(C(C(CCC)NC(C)=O)=O)C2)=O)CCC2(CCCN2C)C1 36306,c1(C(N2CCC(OCCNC(CS(CC)=O)=O)C2)=O)cc(C(=O)OC)cc(O)c1 36307,c1(C(N2CCC(NC(C3CC=C(C)CC3)=O)C(F)C2)=O)cc(S(C)(=O)=O)c(C)o1 36308,C1(C)(NC(C#CC(=O)N(C)C2CC2)=O)CCCC1(F)F 36309,N1(CC(=O)NC2CCC(CNC(C3(N(C)C)CCC3)=O)C2)C(=O)CC(C)(C)C1=O 36310,C1(CNC(=O)CCOC2CN(C(=O)C(O)CNCCCC)C2)CC2CCC2C1 36311,c1(C(N2CC(C)C(C(=O)NC3(C4CCCO4)CC3)C2)=O)cc2ncccc2[nH]1 36312,C(CC(O)C(F)(F)F)NC(C1N(C(c2cc(C(C)=O)[nH]n2)=O)CC1)=O 36313,Cc1nn2c(c1CNC(=O)Cc1ccsn1)CN(C(C1CCC(=O)C1)=O)CC2 36314,c1(C(=O)NC2CCC(NC(C(C)n3ccnn3)=O)CC2)nn(C)c2c1CCC2 36315,C1(C(=O)N)CCN(N2CCC2C(=O)OCC)CC1.C12(CCCCC1)C(=O)NCCS2.CSC.CC.C 36316,CC1=C(C)CC(C)(C(N2CC(O)(CNC(c3cc(F)c(O)c(F)c3)=O)C2)=O)CC1 36317,c1(C(=O)NCc2c(C(N(C(CCC)C)C)=O)scc2)cc(OC)n(C)n1 36318,C1(CC)COCCN(C(c2cc(CNC(=O)C(C)SC(C)C)on2)=O)C1 36319,C1(C)(C(=O)OC)CCN(C(CCc2ccc(C)c(N)c2)C(=O)NC2CCC2)CC1 36320,c1(C(=O)NCCC(CC)(C)NC(c2sccc2Cl)=O)c(O)cc(F)cc1F 36321,C(=O)(C(O)Cc1ccccc1)NCCCN(C(C1C(CC)C1)=O)C 36322,c1(-n2c(CCCC#C)nc(CC(C)(C)C)n2)ccc(S(=O)(=O)CC)cc1 36323,C1(NC(CC(C)(C)SC)=O)CN(C(C23CCC(N=[N+]=[N-])C2C3)=O)CC(C)(C)C1 36324,C1(NC(C(C2CCCOC2)OC)=O)CN(C(=O)C2=CCS(=O)(=O)C2)CC(C)(C)C1 36325,c1(N2CC(C)NC(=O)C2)[nH]c(=NC2CC2C2CCOCC2)nc2c1cnn2C 36326,Cc1ccc(C)c(C(=O)NC2CC(C)N(C(C3CC(O)(C(F)(F)F)C3)=O)C2)c1 36327,c1(CC(=O)NC(C)Cc2cnn(C(F)F)c2)ccc(F)cc1F 36328,C=CC(CC)CC(=O)NCCC1CC(NC(C2CSCC(=O)N2)=O)C1 36329,c1(OC)nc(C(=O)NCC(C)CNC(=O)CCC(=O)c2ccccc2)cc(O)n1 36330,N#Cc1c[nH]c(=NC(=O)C23CC2CN(c2ncc(F)c(C4CCC4)n2)C3)cc1Cl 36331,C(C(C)NC(=O)CCc1cc(C)n(C)n1)(C(C)C)NC(C1(C#C)CC1)=O 36332,C(=O)(C(CC(F)F)C1CCC1)NC1CC(CNC(=O)CCn2cncn2)CC1O 36333,C1(F)(CNC(CCC=C)=O)CCCN(C(=O)CC(N2CCCCC2=O)C)CC1 36334,c1(C(N(CCCCN(C(C(CSC)O)=O)C)C)=O)ccc2nnnn2c1 36335,N1(C(c2c(OC)cccc2)=O)CCC(C)C(CNC(=O)CCc2cccs2)C1 36336,CN1CCC(C(=O)N(CCNC(=O)C2=C(Cl)CCC2)CC2CC2)S1(=O)=O 36337,Cc1cc(C)n(CC(=O)NC(C(N2CCCCC2C(F)F)=O)C2CCC2)n1 36338,c1(CC)cc(F)c(F)cc1NNC(=O)NCCCCCS(C)(=O)=O 36339,c1(C(=O)NCC2N(C(c3cc(C)[nH]n3)=O)CC(C)(C)C2)ncnc2c1CCC2 36340,CN1C(=O)OC2CN(C(C3CCN(C(C4(C)CCCS4)=O)CC3(C)C)=O)CC12 36341,C1(NC(C2CCOC(C)C2)=O)CCCC(C(=O)CC2(SC)CCC2)C1 36342,c1(CC(=O)NC2CN(C(C(P(C)(C)=O)O)=O)CC23CC3)cc(Cl)cc2c1OCC2 36343,C(=O)(C(O)C(C)(C)C)N1CCC(n2cc(CNC(C3CC(C)OCC3)=O)nn2)C1 36344,Cn1cnc2cccc(C(=O)NCC(O)CNC(=O)C(C)(C)C(F)(F)F)c12 36345,c1(CC)c(C(N2CCN(C(c3coc(CO)c3)=O)CC2)=O)ccn1C 36346,C12(C)CC(CN1C(=O)C=CC(F)(F)F)N2.C(=O)(COC)NCCOC 36347,C(CCCCC(=O)N(C(C)C(=O)NCC1CC(O)CN1C)CC)OCC 36348,C(=O)(C(C(C)C)OC)NCC1C(NC(C(COC)C)=O)CCC1 36349,C1(NC(C(C)NC(C2CCCC2)=O)=O)CCN(C(=O)CC(C)(C)C2CC2)CC1F 36350,N(C1CCCc2ccoc21)C(C1N(C(=O)COC2CCC2)CCN(C)C1)=O 36351,C1(CNC(C2(CC)CC2)=O)CN(C(c2snnc2C2CC2)=O)CCC1(C)C 36352,C(C(C)C(C)C)OCCC(N1C(CNC(C(C)OCCCC)=O)CC1)=O 36353,N1(C(C)C)CCCN(C(C2CCC(C(C)C)N2C(=O)C2=CCOCC2)=O)CC1 36354,CC1=CCSC1C(=O)NCc1ccsc1C(=O)N(CC(C)O)CCF 36355,C(=O)(CC1=NNC(=O)C1)NCC1N(C(c2c(C)cc[nH]2)=O)CC=C1 36356,C1(O)(Cn2cc(CNC(C)=O)nn2)CCCN(C(=O)CCS(C)=O)C1 36357,c1(N2CCC(N(C)C(C3CCCC(NC(N)=O)C3)=O)C2)ccc([N+](=O)[O-])cc1C#N 36358,c1(C(=O)NCC=CCNC(c2ccc(CC)c(N)c2)=O)cccc2scnc12 36359,c1(C(=O)NC(CC=C)CNC(=O)C(CC)CCOC)cc2ncccc2s1 36360,C1(CNC(Cc2c(C)ccs2)=O)CN(C)CCN1C(c1cccc(=S)n1O)=O 36361,c1(C(N2CC(NC(C3C(=C)CC3)=O)C3(C2)CC3)=O)cc(Br)c(OC)cc1N 36362,c1(CC)cccc2[nH]c(C(N3CC(CNC(C4COCCO4)=O)C(O)C3)=O)cc12 36363,CC1=CCC(C(N2CC(O)(C(C)(C)CNC(=O)CC(C)(C)C)C2)=O)CC1 36364,c1(C(N2C3(C(N(C4CCCCC4)CCC)=O)CC(C2)C3)=O)cc2ccccn2n1 36365,C1(NC(C=C(COC)C)=O)CC(OC)CN(C(c2cccc(C(C)OC)n2)=O)C1 36366,c1(C(C)C)nccc(N2CC(NC(=O)Cc3ccccn3)C(C)C2)n1 36367,C1(CNC(C2COCC2O)=O)CCN(C(c2ccc(C3CC3)cc2)=O)C12CCC2 36368,c1(C(=O)NCCCN(C(c2cccc(CN(C)C)c2)=O)C)coc2ccccc12 36369,N1(C(C(CCO)N(C)C)=O)CCC(C=CC(=O)NC2CCSCC2)CC1 36370,N1(C(C2CC(C#C)(O)C2)=O)CC(NC(c2cnn(CC(F)(F)F)c2)=O)CC1(C)C 36371,C(=O)(C(CC)CC=CC)N1CC(CN(C(CC2CC(=C)C2)=O)C)OCC1 36372,C1(NC(=O)Cc2cccs2)CN(C(c2cccnc2-c2cccs2)=O)CC1F 36373,C1(CNC(c2ccsc2)=O)CN(C(=O)CC2CCC3(CCC3)O2)C2(CCC2)C1 36374,C1(C(C)(O)CNC(c2ocnc2C2CCC2)=O)CCCN(C(c2cc[nH]c2)=O)C1 36375,C(=O)(CCCCCCCCC)NCC(CNC(C1C(=C)CC1)=O)(C)C 36376,c1(C(=O)NCC2C3(CCN(C(CC4(C)CC4)=O)CC3)C2)cnc2ncnn2c1O 36377,CCC(C)CC(CO)NC(c1cncc(CNC(c2nocc2C)=O)c1)=O 36378,CCC(CC)C(C)C(=O)NC(C)(C(=O)NCC1=CCCCC1)C1CC1 36379,C1(O)(NCC=NC(=O)CSC(F)(F)F)CN(C(c2cn(C3CCC3)nn2)=O)C1 36380,C1(CC)CN(C(=O)Cn2ccccc2=O)CC1NC(c1ccc(Br)c(C)n1)=O 36381,C1(NC(CC(C)n2cccn2)=O)CC2(C1)CN(C(c1ccccn1)=O)C2 36382,CC1CCC(NC(=O)Cc2cnn(C(F)F)c2)CN1C(=O)Cc1ncc(Cl)s1 36383,C(CC)(C(C)(C)O)N.N12CC(C1)C2=O.C(C(=O)N1CCC1)N(C(=O)OCC)C1CC1 36384,C1(C(=O)NCCN(C2CC2)CC)CC2(CC2)CN1C(C1CCCC(=O)C1)=O 36385,N1(C(=O)NCc2cccc(Cn3cncn3)c2)CCCC2(C1)OCc1ccccc12 36386,CCC(C)(C)CC(=O)NCC1CN(C)CCN1C(c1cc(Cl)ccc1OC)=O 36387,C1(O)(C(=O)NC2(CNC(=O)Cc3cc(C)ns3)CC(OC)C2)CC2CCC1C2 36388,C#CCC(CC#C)NC(=O)C(CNC(=O)C=CC1CCOC1)N(C)C 36389,N1(C(C(C(C)NC(c2ccn(C(F)F)n2)=O)C)=O)CCC(F)(F)C(F)C1 36390,C1(NC(COC(CC)C)=O)CC(C(F)C(=O)N(C2CC2(C)C)C)C1 36391,C1(CC)(NC(=O)CC(c2ccc(SC)cc2)C)CCN(C(=O)C(C)(C)CO)CC1 36392,CC(CC(F)F)C(=O)NC1CCC(NC(=O)C(Cc2ccccc2)N(C)C)CC1 36393,N1(C(CCCCC)=O)CC2CCC(C1)C2CNC(C1CC2CC2C1)=O 36394,N1(C(CCCCOCC)=O)CCC(N(C(=O)C(C(C)C)SCC)C)C(C)C1 36395,C1(NC(CCC(=C)C)=O)CCc2nncn2CC1 36396,c1(C(N2CC(NC(C(CCC)(C)CC)=O)C(C)C2)=O)nnc2ccccc2n1 36397,CC1(C)OC(=O)CC1C(=O)NC1CCCN(C(c2cnn(C3CC3)c2Cl)=O)C1 36398,N1(C(C(CC2CN(C(C(CCSC)O)=O)C2)F)=O)CC2(C1)CC(C)(F)C2 36399,N1(C(CC)=O)CCC2(CC1)C(NC(=O)COc1ccccc1SC)CCS2(=O)=O 36400,C1(O)(CCNC(C(C=CC)O)=O)CCN(c2ccc(C(=O)OCC)nn2)C1 36401,CCCC(C(=O)N1CC(CNC(c2cocn2)=O)(COC)C1)C(C)C 36402,C1(NC(=O)CC2CCCCC2)CC(F)CN(C(=O)C(F)F)C1 36403,C1(OC2CN(C(c3c(CCC)nns3)=O)C2)CCN(C(c2ncoc2C)=O)CC1 36404,N(C(=NCCCNS(C)(=O)=O)N1CN(C)C(=O)C1C)CC(C)O 36405,C(CCN=c1cc(C)nc(C2CCC2)[nH]1)N1CCC(c2ccc(OC)nc2)C1 36406,C1(NC(c2cscc2C2CC2)=O)CC2CCC(C1)N2C(c1ccns1)=O 36407,N1(C(C(C)NC(C)=O)=O)CCC2(CC1)COC(CNC(c1c(Cl)n[nH]c1C)=O)C2 36408,Cc1c(Cl)ccc(C(=O)NC2CN(C(c3cccc(=O)n3C)=O)CC2CO)c1O 36409,C1(NC(COC2C(CC)CCCC2)=O)CCN(C(c2cc(O)cs2)=O)C(C)C1 36410,Cc1nc(N2CC3CC2(CNC(c2cnn4cc[nH]c24)=O)C3)c(C)c(O)n1 36411,C(=O)(C(C)(C(C)C)OC)NCC1(CO)CN(C(c2ccc(NC(=O)OC)s2)=O)C1 36412,Cc1nnccc1-c1noc(-c2cccnc2OC(C)C)n1 36413,c1(C(=O)OCC)nnc(COCC(c2nnc(C)o2)C)s1 36414,n1(CC(=O)NCC2CC2CNC(c2ccccc2)=O)nc(Cl)ccc1=O 36415,CC1CN(C(c2scnc2C(F)(F)F)=O)CCN1C(C1CC2(CCOC2)C1)=O 36416,c1(-c2cn(CN(CCCCCCCO)C)nn2)ccc(P(C)(C)=O)cc1 36417,c1(CNC(c2cccc(Sc3ccccc3)c2)C)cc(S(N)(=O)=O)cs1 36418,Cc1ccc2c(C(N3CC(CNC(C4CC5CCCCN5C4)=O)C3)=O)coc2c1 36419,c1(Cn2c(NC(=O)NC(C#C)C3CC3)ccn2)ccc(Br)cc1F 36420,CC1CCC(NC(C2(NC(N)=O)CC2)=O)CN1C(c1n[nH]c2c1COC2)=O 36421,C1(C(N(CCNC(c2cc(C3CCCC3)[nH]n2)=O)CC)=O)CCC(C(N)=O)CC1 36422,C1(NC(C2(SC)CC2)=O)COCCC1NC(c1coc(-c2cccc(Cl)c2)n1)=O 36423,c1(C(N(CCN(C(=O)CC2CCN(C)CC2)CC)CC)=O)ccnc(F)c1OC 36424,c1(CSC)cc(C(N2CCC(CNC(=O)CC3CCCO3)C2)=O)ccc1F 36425,Nc1ccc(F)c(C(=O)NC2CCC(NC(c3snc(O)c3Cl)=O)CC2)c1F 36426,N12CCCC(C)C1C(=O)C(C)SNCC2=O.C#CCOCCOCCOCCO 36427,C1(CCC(=O)N(C(C)C)CC2CCC2)CCN(C(C2(C3(C)CC3)CC2)=O)CC1 36428,c1(OC(C)C)ccccc1N(C(C)C(=O)OC(C)(C)C)C(c1cccc(Cl)c1)C 36429,C12(C(=O)NCC3(C)N(C(c4c(C)ccnc4)=O)CCC3)CCCN(CC1)C2 36430,Cc1cc(C(=O)NC(C)C(C)C)cc(C#N)c1.c12cc[nH]c1C(=O)N(C)C2 36431,N1(C(CSCC)C)CCCC(C(=O)NC(c2coc(CSC)c2)=O)C1 36432,N1(C(c2c(CC)ocn2)=O)CCCC(C)C1CNC(=O)Cn1nc(C)n(C)c1=O 36433,C1(OC)CC2(C1)CN(C(=O)C(O)CCNC(=O)Cc1cncs1)C2 36434,C(CN=C(NCc1cc(O)cc(O)c1)NCc1cc(C)ccn1)N(CC)CC 36435,c1(CC(=O)NC2(CC(=O)N(CC(C)Cc3cn[nH]c3)C3CC3)CCC2)cccn1C 36436,c1(C(N(C)CC23CCCC2OCC3)=O)c(Cl)nc2ccccn12.C12(CC1)C(=O)N2 36437,c1(C(=O)NCC2(CNC(C3CC4CC3C4)=O)CC2)cc(Br)ccn1 36438,C1(OC)CC(NC(c2cc(C)ns2)=O)CN(C(C2CCC(=O)N2C2CC2)=O)C1 36439,C1(C(=O)NC2CCC(NC(c3ccncc3O)=O)C2)CCCC1(F)F 36440,Cc1nn(C2CC2)cc1C(=O)NCC(C1CC1)NC(=O)CNc1ccccn1 36441,C1(C(=O)NCCC2(C(N(C)CC3CCCCO3)=O)CCCC2)CC(=O)NC1(C)C 36442,N12CC3CCN(CC13)C(=O)c1cc(on1)CC2=O.C1(N(C)C)CC(C(N)=O)C1 36443,c1(NC(CC2CN(S(CC(=O)OCC)(=O)=O)C2)=O)cc([N+](=O)[O-])ccc1Cl 36444,N1(C(Cc2nc(C)sc2)=O)CCCN(C(=O)Cc2cccc3nonc23)C(C)C1 36445,C(CCC(N)=O)(C(=O)NCCC1CN(C(=O)CCN2CCCCCC2)C1)N(C)C 36446,C(C(COC)C(C)C)NC(c1ccccc1C)c1n(CCSC)nnn1 36447,C(=O)(CCC(=O)NN(C)C)NC1CC(C)CN(C(c2ccoc2Br)=O)C1 36448,c1(CC)nc(C)c(C(N2CC(C(=O)NC(C)(CO)C3CC3)(CC)C2)=O)o1 36449,C1(C(=O)CC2(CC(=O)C(C)=O)CC2)CCCN(C(=O)C(=O)C2CC2)C1C.NC 36450,CC1(C)CCCC(CC(=O)NCC2COCCN(C(c3ccoc3Cl)=O)C2)C1 36451,c1(C(=O)NCC2C(NC(CC(=O)OCC)=O)COC2)c(F)cccc1[N+](=O)[O-] 36452,N1(C(CCN(C(c2cn(C(C)C)nn2)=O)CCO)=O)CCN(C)C(C)C1C 36453,c1(C(N2C(C(C)NC(c3[nH]cc(C(C)=O)c3)=O)CCC2)=O)cc(C)n(C)c(=O)c1 36454,C(=O)(C(C)(O)CC(C)C)NC(CC(=O)NCc1snc(CC)n1)C(C)C 36455,C(=O)(C#CC1CCCOC1)OCc1n(CCC(=O)OC)c2c(n1)cccc2 36456,C(CC(=O)NCC(c1cccnc1)O)(CC(C)C)NC(c1cccc(C)c1O)=O 36457,C1(C(=O)NC(C2CCCCC2)C#C)COCCN1C(c1ccnc(C)n1)=O 36458,CCCS(=O)(=O)c1ccccc1C(=O)NCCCCCNC(C1CC1(C)Br)=O 36459,Cc1nc(C(=O)NC2CC2CNC(=O)C=CC2CCCCCC2)c(C)n1C 36460,n1(CCOC)nccc1C(=O)NCC1(NC(C2CCC(C)C2)=O)CC1 36461,C1(C(c2n(CCSC)nnn2)NCCc2ccncc2)CC2CCC1CC2 36462,c1(OC)ccc(C)cc1CNCC(O)CNC1(C#N)CCCC1 36463,Cc1ccc(S(=O)(=O)NC2CCCC2C(N2CCOC(C)C2)=O)c(F)c1 36464,N1(Cc2ncc(CC)o2)CC2(C)CN(C(=O)CCC(C)OC)CC2(C)C1 36465,c1(CC(=O)NC2C(NC(c3c(=N)c(Cl)c[nH]n3)=O)CC2)ccc2c(c1)CCCS2 36466,C1(CC(=O)NCCC(C)(C)NC(CC(C)SC)=O)CCOC(C)(C)C1 36467,C1(CN(C(C(C)c2cncs2)=O)C)CCCCN1C(c1ccc(SC2CC2)o1)=O 36468,C1(C#CC(=O)NC(CNC(=O)C=Cc2ccccc2C)C(C)(C)C)(CC)COC1 36469,C12(CNC(c3n(C)nc(Br)c3)=O)CCC(C1)N(C(=O)C(C)(C)F)C2 36470,c1(CNC(C(C)O)(C)C2CCOCC2)ccc(Br)cc1OC(F)F.CC(=O)O 36471,N1(C(CC)=O)CCC(CC(F)(F)F)C(NC(=O)Cc2cc(C)nn2C)C1 36472,C(=O)(NNc1cc2ccccc2s1)c1cc(C)nc2c1cc(Br)cc2 36473,Cn1c(F)c(COC(C2CC2C(F)(F)F)=O)c(O)nc1=O 36474,CC(C)C(O)C(C)C(=O)NCCCC(CCCc1ccccc1)C(=O)OC(=O)CN 36475,c1(SC)ccc(C)c(C(=O)NC(C)CN(C)C(C2CC2C)=O)c1 36476,CC1CCc2nc(C(=O)NCC3CCCC3NC(=O)CC(C)(C)O)ccc2C1 36477,C1(NC(c2onc(-c3c(C)cccc3)n2)=O)(CNC(=O)C(F)F)CC2CCC1C2 36478,Cc1ccc(F)cc1CC(=O)NC(C)C(C)(C)NC(=O)CC1CC2(CCC2)CO1 36479,n1(C(C)C)ncc(C(=O)N(CC(C)CNC(C2CC3CCC2C3)=O)C)c1N 36480,c1(C(=O)NCCCN(C(CSS(C)(=O)=O)=O)C2CC2)cccc2ncsc12 36481,C(=O)(N=c1[nH]nc(C2CC2)s1)N(C)Cc1ccccc1SC(C)(C)C 36482,C1(COC)(NC(=O)C=CC(F)(F)F)CCN(C(=O)Cn2cnc(=N)[nH]2)CC1 36483,Cc1nc(F)ccc1-c1cn(C2CCN(C(=O)Nc3cccc(Cl)c3)C2(C)C)nn1 36484,CCC(N=c1ccnc(N2CCCC(N3CC(C)(C)C3)C2)[nH]1)C(C)C 36485,N1(C(CC=CC)=O)CC(NC(=O)C=Cc2ccoc2)CC(F)(F)C1 36486,CCCCCCCCC(C)C(=O)NC(C1CCN(C(C2(C)CCC(=O)C2)=O)C1)C 36487,N1(C(CNC(C)=O)=O)CC(=O)NCC1C(=O)NCC1(O)CCOC1 36488,N1(C(COC)=O)CCCC(C)(C)C1CNC(C1(Cc2ccc(F)cc2)CC1)=O 36489,c1(C(=O)OC(COC)=O)cn2nc(OC(COCC)CC(F)(F)F)ccc2n1 36490,C1(CNC(CCCN(C(C)=O)C)=O)CCCC(NC(c2nnnn2C2CC2)=O)C1 36491,c1(N2CC(CN(C(C(c3ccc(C)o3)C)=O)C)OCC2)ncnc2scc(C)c12 36492,c1(N2CCCC(CCNC(C3C(C)CC(C)O3)=O)CC2)ncc([N+](=O)[O-])c(=N)[nH]1 36493,C1(c2nnc(C(C)C)o2)COCCN1c1nnnn1CCOCC(C)C(F)(F)F 36494,N1(C(c2ccn(C)c2)=O)CCC(C(C)(O)CNC(=O)Cc2ccncc2F)CC1 36495,CC(C)(C)CC(F)C(=O)NC(C1CN(C(C2COCC(C3CC3)O2)=O)C1)(C)C 36496,C1(NC(c2ccc(OC)c(I)n2)=O)CCc2ncc(Br)n2C1 36497,c1(C(=O)NCC2(OC)CCN(C(=O)C(C)CF)C2)cc2c(=O)[nH]ccn2c1 36498,n1(C(C)C)cnc(C(=O)NC(CO)C(C)NC(C2CN(C3CCOC3)C2)=O)c1 36499,C(=O)(C(C(C)C)C(C)C)N(C1CCCN(C(C(CC)NC(C)=O)=O)C1)CCF 36500,Cc1cc(C(N2CCC(F)(CNC(C3CCCN3C3CC3)=O)C2)=O)nnc1C 36501,CN=c1[nH]cc(C(=O)N(CCN(C(=O)Cc2cnn(C(C)C)c2)C)C(C)C)s1 36502,C(c1ccc(F)nc1)=CC(=O)NCC1CCCN(C(c2cncc(Cl)c2Cl)=O)C1 36503,C1(N(CCC)C(C2CCC2)=O)CCN(C(=O)C=Cc2sccc2C)CC1 36504,c1(OC2CN(CC(c3ccc(CC)cc3)O)C2)ccc(Cl)cc1[N+](=O)[O-] 36505,C1(NC(c2c(C(=O)OCC)c[nH]c2)=O)CCN(C(C2CC(C)(C)CC=N2)=O)CC1 36506,N1(C(C2(C(=O)OC)CC2)=O)C2CCC1CN(C(C1(c3ccccc3)CC1)=O)C2 36507,C1(C2CCOCC2)(NC(C(C(CNC(c2nnn(CC)c2C)=O)C)F)=O)CC1 36508,C1(CNC(COCCOCC)=O)(OC)CCN(C(=O)C=Cc2ccsc2)CC1 36509,Cc1cc(C)c(C(=O)NCC(C)(C)CNC(c2cccc(C(N)=O)n2)=O)c(S)n1 36510,C(=O)(C1=CC2(CN(C(=O)Cn3cnnc3O)C2)OC1)N(C)CC1(CO)CCC1 36511,C1(CCC(=O)NC(CNC(CCC=CC)=O)C)CCCC(O)C1 36512,C(C(F)(F)C(=O)NC(C)CCC(=O)NC1C(OC)CC1O)OC 36513,C1(CNC(C(CC)CO)=O)CCN(C(c2cnn(C3CCCC3)c2)=O)C1(C)C 36514,c1(C(=O)NCC(C)CNC(c2cccc(I)c2)=O)ccc2cnccc2c1 36515,c1(C(CO)NCCCCCNC=O)cccc(OCF)c1.C(F)(F)(C(F)Cl)O 36516,c1(NC(C2(C)N(C(CC(C)O)=O)CC2)=O)cc(Cl)c(Br)cn1 36517,CCCC(C(=O)NCC1CCCCN(C(=O)CCN2CCOCC2)C1)S(N)(=O)=O 36518,Cc1noc(-c2ccccc2)c1C(=O)NC(=O)CN(C)C.c12sc(nc1C)s2 36519,N1(C(C2(NC(C)=O)CCCC2)=O)CCC(CO)(CNC(C2CC(C)(C)CO2)=O)C1 36520,c1(C(N2CC(O)(CNC(CN3CC(CC)C3)=O)C2)=O)sc(C)nc1C 36521,c1(NC(c2n(CCC)nnn2)C2CC2C2CC2)ccc(Cl)c(C(N)=O)c1 36522,c1(C(N2CC(CC)C(NC(=O)C=C3CC3)CC2)=O)c(C)ccc(OC(C)C)c1N 36523,c1(N(C)Cc2cnccn2)nc2c(c(=NCC3CCC=CCC3)[nH]1)COC2 36524,CCC(C)C(=O)NCC(=O)NC1CC(CNC(C2(C3CC3)CCCO2)=O)C1 36525,N1(C(c2c(C)snc2)=O)C2CCC1C(CNC(=O)CCc1nc(C3CC3)no1)C2 36526,CC1(NC(c2c[nH]nc2-c2ccn[nH]2)=O)CCN(C(=O)CC=C(Cl)Cl)C1 36527,C12CC(C)(C)C1CNC2=O.c1(SC)ccc(C(=O)NC23CC(C(F)(F)F)(C2)C3)s1 36528,N1(C(C(COCC)C)=O)CCC2CCCC12C(N1CCCCC(C)C1)=O 36529,C=C(Br)CC(C)(C)C(=O)N1CC(CNC(=O)C(C)NS(C)(=O)=O)C(C)C1 36530,C(=O)(C1=C(F)CN(C(=O)CC(C)N(C)C)CC1)Nc1ccc(C)c(CO)c1 36531,C(CC(COC)OC(=O)C(Cc1cnc[nH]1)NC(=O)OC(C)(C)C)OC 36532,N1(CC(=O)NCc2c(OC)cncc2)C(=O)NC(C)(c2ccc(F)cc2C)C1=O 36533,c1(C(N2C(C(=O)Nc3c[nH]nc3Cl)CC2)=O)ccc2c(c1)CCCO2 36534,c1(C(N2CCC(NC(CCc3c(C)nccc3)=O)C2)=O)ccc(C(F)F)c(Cl)c1 36535,c1(C(C(=O)NCC)OCOC)ccc(Br)c(OCCCC)c1F.C(CNCC)O 36536,C1(C(=O)NC(CCN(C(=O)C(=C2CCCCC2)F)C)(C)C)CC(C)(C)OC1(C)C 36537,C(=O)(C#CC1CCCCC1)N1CCCC(CCC(=O)NCC2(O)CCC(C)C2)C1 36538,C1(CC)CNC(=O)CN1C(=O)CC=CCNC(C1CC12CC2)=O 36539,C1(C(=O)NC2(CC)CCNC2=O)CC2C=CC1N(C(=O)CCOCC(C)C)C2 36540,c1(C(=O)NC2CCC(C)(CNC(=O)C(Cl)=CCl)C2)cccn2cncc12 36541,Cc1ccc([N+](=O)[O-])cc1C(N1CCC2CN(C(C3(C#N)CC=CC3)=O)CC12)=O 36542,c1(NC(=O)NC(CC(=O)OCC)Cc2ccc(Br)cc2)nccc(C)c1O 36543,CCCCC(F)F.C1(=O)C(CC)N1.C1(C)(C)CNC(=O)CO1 36544,C12(CCC(=O)NC(C3(NC(=O)CN4CCOCC4)CC3)C)CCCCC1C2 36545,C1(CCC(N2CCN(C(C=CCC)=O)C(C)C2)=O)CCc2ccccc2C1=O 36546,C(c1ccc(C)cc1C)=CC(=O)NC1CCCC(CNC(CN(C)CC)=O)C1 36547,Cc1cc(F)cc(C(N2CC(NC(c3cn(C)cn3)=O)C3CC23)=O)c1O 36548,C=CCC(Cc1ccccc1)C(=O)NCCCOc1c(F)cccc1F 36549,N1(C(CN(C(C)CC(C)C)CCC)=O)CCC(CNc2cnccn2)C12CCC2 36550,N1(C(C=Cc2cc(C)no2)=O)CC2CCC(N(C(=O)C3=CCCSC3)C)C2C1 36551,c1(C(=O)NC2CC3CC2N(C(=O)CCC(F)F)C3)nccc2[nH]ccc12 36552,C(CNC(C1CC=CC1)=O)(C(C)(C)C)NC(CCN(c1ccccc1)CC)=O 36553,C1(C(N(CCC)CC)=O)CCC(O)CN1C(c1cc(C(N)=O)[nH]n1)=O 36554,N(C(=NCc1nc(-c2ccco2)no1)N1CCC(C)(F)C1)C(C)C1CC1 36555,C1(OC)(CNC(c2n[nH]c(C)c2O)=O)CCN(C(c2cn(C(C)(C)C)nn2)=O)C1 36556,CC1CC2(CCN(C(=O)Cc3cncs3)CC2)CN1C(C1CC12CCCC2)=O 36557,c1(CCNS(NCCNC(=O)NC2CNC2)(=O)=O)cccnc1N1CCCC1 36558,N1(C(Cn2ccc(C)n2)=O)CC2CC(C1)CN(C(=O)CC1CCC(=O)C1)C2 36559,C12(C(=O)NCC3C4CN(C(CC(=C)Br)=O)CC43)CCC(C)(C1)OC2 36560,N1(C(CCc2cccs2)=O)CCC(CNC(C2(C)CC2)=O)C1.c12cnc(s1)[nH]c2=O 36561,C(CNC(c1nccn1C)=O)(C(=O)NC1(C)CC(N(C)C)C1)OC 36562,C1(C(=O)NC2CCC(CCNC(c3ccc(C(C)C)s3)=O)C2)CC(F)(F)C1(C)C 36563,C(=O)(CC(CNC(c1nn(C)cc1C)=O)C1CCC1)NC(C(=O)NCC)C 36564,C(=O)(C(C)(C)CCCF)NCC(C(=O)NCc1c(C)cc(O)cc1)CC1CC1 36565,N1(C(CCOCC(C)(C)C)=O)CCCC(F)(C(=O)NCC23CCCC2CCC3)C1 36566,C1(CNC(C2CC3(C2)CC3F)=O)COCCN1C(=O)Cn1cnnc1O 36567,CC1CN(CCc2cn(Cc3cc(Cl)no3)nn2)C12CCOCC2 36568,c1(OCC(=O)NCC2OCCN(C(c3c(C)nn(C)c3)=O)C2)cc(Cl)cc(Cl)c1 36569,CC(=O)C(C)(C)CC(=O)N(C1CCN(C(c2ccccc2[N+](=O)[O-])=O)C1)C 36570,C(C)(CCC(=O)N1CCCCC1C1(NC(c2ocnc2C(F)F)=O)CC1)SC 36571,N1(c2snc(SC)n2)CCC(NC(c2cn(C3CCOC3)cn2)=O)C(C)C1 36572,C1(C(C)C)CCC(C(=O)N(C)Cc2cn[nH]c2)N1C(c1cnnn1C)=O 36573,C1(CNC(CC(C)SC)=O)CN(C(c2ccc(Cl)c(C)c2N)=O)CC12CCC2 36574,C(=O)(CCCCCNC(C)=O)NCC1CC(NC(COCCC)=O)C1 36575,C(=O)(C(C)C(C)(C)C)NCCCN(C(=O)C=Cc1cccc(CO)c1)CC 36576,c1(C(N)=O)ccncc1NC(c1cc(CCC(=O)CC2CC3CC3C2)on1)=O.N 36577,c1(CC)ccc(F)c(C(=O)NCC2CC(F)CN2C(c2nnc(S)n2C)=O)c1F 36578,C1(CNC(c2c(C)cncc2C)=O)COC(C)(C)CN1C(c1cc(Cl)c[nH]1)=O 36579,N1(C(COCC(=C)C)=O)CC2CC1CN(C(c1cc(C3CCCC3)[nH]n1)=O)C2 36580,C1(NC(C(=Cc2ccccn2)C)=O)C2CCC1N(C(c1cc(C(C)C)no1)=O)C2 36581,C1(C(N(CCOC)C2CC2)=O)(NC(C2CC2(F)Cl)=O)CC1(C)C 36582,CCCC(C)CC(=O)NCC1CCCN1C(c1cn(C)cc(Br)c1=O)=O 36583,C(CCCCCC(=O)N1CC2(Cc3cn(CCO)nn3)CC2(C(F)(F)F)C1)SC 36584,c1(C(=O)NC2CC(CO)N(C(c3ncccc3F)=O)C2)ccc2c(c1)OCCO2 36585,Cc1c(NCCN2CCOCC2)nc[nH]c1=NCC1(C)CC1(Cl)Cl 36586,N1(C(CCSCC)=O)CCC(NC(=O)CC2(C)CCOCC2)C1C(C)(C)C 36587,c1(OC)ccc(CC(N2CCCN(C(C3CC4(C3)CC4F)=O)CC2)=O)c(C)c1 36588,C12(C)CCCN(C1)C(=O)OC(=O)C2.CC(C)C(C(=O)OC(C)(C)C)n1cncn1 36589,c1(NCCCCC(N)=O)[nH]c(=NCCCC2CCCCC2)nc2scnc12 36590,c1(C(=O)NC(CCC)CNC(c2cnc(C)s2)=O)c(OC)nsc1OC 36591,C#CCCCC(C)C(=O)N1CCOC(CC(=O)NC(c2n[nH]c(C)n2)C)C1 36592,C1(C(=O)NCCOCCN(C(=O)CC2CCN(C)C2=O)C)CC12CCOCC2 36593,CCS(=O)(=O)CCN=c1[nH]c(N2CC3CCCCC23)nc2c1CCC2 36594,Cc1ccc(CC(N2CCC2CNC(=O)CN(S(C)(=O)=O)C)=O)c(Cl)c1 36595,C1(O)(CN(C)Cc2ccc(CC(C)O)s2)CCN(C(=O)OC(C)(C)C)C1 36596,C(=O)(C=C1SCC(=O)N1C)NC1CCN(C(c2n(CCC)ccc2)=O)CC1O 36597,CC1CC(C(=O)NCCC2CN(C(C3CC3c3ccc(Br)nc3)=O)C2)=NO1 36598,C(=O)(C1=NOC2(CCC2)C1)NC(C1CN(C(=O)Cc2cn3ccccc3n2)C1)C 36599,c1(C(=O)NCCC(C)NC(C2CC23CC3)=O)c[nH]c2ccc(Cl)cc12 36600,N1(C(C(CSC)O)=O)CCC(NC(=O)COC2CCCCCC2)C(F)C1 36601,CC(CCCCNC(c1cnn(C2CCCC2)c1)=O)NC(C1CCCCC1O)=O 36602,c1(-n2c(C(N3CCC(N(C)Cc4sccc4Cl)C3)=O)ccc2)ccccc1Cl 36603,c1(SC(CNC(N)=O)C)nc(C)c(C(=O)N(C)NC(c2cc(C)ns2)=O)o1 36604,CC1=NOC(C)(C(=O)NC(CO)C(C)NC(=O)Cn2nc(C)cc2C(F)F)C1 36605,C(C1=NOC2CN(C(=O)C=CSC)CC12)NC(C=C(CC)CC)=O 36606,C(CCC(=O)NNC(=O)OCc1ccc(OC(F)F)cc1)c1cn(C)nc1 36607,C(c1c(C)noc1C)=CC(N1CCC(N(C(C2CCCN2C=O)=O)CC)C1)=O 36608,N1(C(CCSC)=O)CCN(C2CCN(C(C3CCN(S(C)(=O)=O)C3)=O)C2)CC1 36609,N1(C(c2ccc(NC)cn2)=O)CCCN(C(C2C3CCCCCCC23)=O)CCC1 36610,Cc1cnc(C(N2CCC(N(C(=O)CC3CCS(=O)(=O)CC3)C)C2)=O)cc1C 36611,N1(N(C)CC=CC=O)CC(C#N)(CCF)C1.C1(C=O)CCCC1F 36612,CC(C(CO)NC(C1(C)CC1(F)F)=O)NC(=O)Cc1n[nH]cc1Br 36613,C12(C(N(C)OC3CCCC3)=O)CC(C)(CN1C(c1cc(C(N)=O)co1)=O)C2 36614,Cc1ccc(CNC(c2nnnn2CC2CCOC2)(C)CC2CC2(Cl)Cl)c(F)c1 36615,c1(OC)ccc(C(=O)NC2CC3(CC3)CN2S(=O)(=O)C(Cl)(Cl)Cl)c([N+](=O)[O-])c1 36616,C1(CNC(CN(C(C)C)C)=O)CN(C)CCN1C(c1cnn(C2CC2)c1)=O 36617,N1(C(c2n(CCC)ccc2)=O)CC2CC(C1)CN(C(C1CC1C(C)(C)C)=O)C2 36618,CC(C)(CCCO)C(=O)N1CCCC(CCNC(c2c[nH]nc2[N+](=O)[O-])=O)C1 36619,C(=O)(C(CNC(C1(C)CC(F)(F)C1)=O)CC=C)N(CC#C)CCOC 36620,Cc1nc(Cl)ccc1CC(=O)NCC(O)CNC(=O)C(C)Cc1cnc[nH]1 36621,c1(C(N2CC(NC(CCCOCC)=O)C(OC)C2)=O)cccc2ccc(C)nc12 36622,N1(C(C(CCSC)N(C)C)=O)CC(NC(c2cnn(C)c2N)=O)CC12CCOC2 36623,C1(C(N2CC(O)(CCNC(=O)COCC(F)(F)F)C2)=O)CCC(C2CCC2)CC1 36624,N1(C(C(=O)N(CC)Cc2ccc(C(F)(F)F)cc2)=O)CCC(CC(F)CN)CC1 36625,C(=O)(CC(C)c1ccco1)N(CCCOC)CCO 36626,C=Cn1nccc1C(=O)NCC1CCC1NC(c1ccco1)C1CC1 36627,C1(NC(C(c2ccccc2)C)=O)CCCCN(Cc2ccncc2Cl)C1 36628,Nc1ccnc2c(C(=O)NC3CCN(C(C4CCOC(=O)CC4)=O)CC3)cnn12 36629,C1(OC)CCC(CC(=O)NC2CCN(C(c3ccn(C)c3)=O)C2C(C)C)CC1 36630,c1(CC(N2C(c3ccc(C)s3)CCC2)=O)ccc(S(=O)(=O)C(C)C)cc1 36631,c1(-c2nnc(C(=O)NCCSCCO)n2CC2CCCS2)cnc(N)c(Cl)n1 36632,N1(C(c2ccns2)=O)CCN(Cc2cccc(O)c2Cl)CC1CO 36633,C(C(C)(C)C(=O)NCC12CC(CNC(=O)CN(C3CCC3)C)(C1)C2)OC(C)C 36634,Cc1c(C(=O)NC(C2CCCN2C(=O)Cc2cn(C)nc2Cl)C)sc2nccn12 36635,c1(C(N2C(COC)CN(C(c3nc(Cl)ccc3N)=O)CC2)=O)cc(C)cc(C)c1O 36636,O(C=CC(=O)N1CCCC1CN(C(=O)CC1CCC(=O)N1)C(C)C)CC 36637,c1(C(=O)NC(C2(O)CCCCC2)C(=O)NCC(CC)CCO)ccc(C#N)cc1C 36638,C(=O)(CC1CCC(C)(C)c2ccccc21)NCCCNC(C(COC)O)=O 36639,CN(CCCC(=O)OCN1CCOCC1)N=O 36640,c1(CC(N2C(C=O)CC2)=O)ccc(C#N)cc1.C(=O)(C(C)(C)C)NCC1C(=C)CC1 36641,c12ccc(C)c(c1)C(C(=O)NC1COC1)N2C.C1(C(=O)OC)CCCCC1 36642,c12n[nH]cc1C(=O)NCC2.N1(C(COCC#C)=O)CCC(C(=O)OC)C1 36643,C(CC(C)C)(C(=O)N(C1CCSC1)C)ON(C(c1c(CC)nco1)=O)C 36644,C=CCC(C(=O)N(C(C)C(F)F)C)NC(C)=O.C1(=O)C(C)N1 36645,N1(C(C=C(C)C)=O)CC2(CCN2C(c2cc(-c3ccncc3)on2)=O)C1 36646,C1(C(N2CC(CNC(c3cccc(SC)c3)=O)C(C)C2)=O)CCC2(CCC2)CO1 36647,CCCC(CCNC(=O)C(C)(C1CCC1)NC(=O)C(CSC)OC)C1CC1 36648,Cc1cc(O)ccc1C(=O)NCC1CCCN(C(=O)CCC2CCCN2C)CC1 36649,Cc1nn(CCNc2ncncc2Cl)c(C)c1NC(=O)N(C)C 36650,CC(CC(F)F)C(=O)NCCC1CCCCN1C(=O)Cc1ccon1 36651,N1(C(C2CC(=O)NC(=O)N2)=O)CCC(CNC(=O)Cn2cc(Cl)cn2)C(F)(F)C1 36652,c1(CNC(C2C(CNC(=O)CC3CCCOC3)CCC2)=O)ccnc(O)c1 36653,Cc1nc(C2CCC2)sc1C(=O)NC1(C)CCN(C(=O)C(C)NCCC(C)C)C1 36654,C1(C(N(C(CNC(CN(C(=O)OC)C)=O)C)C)=O)CCc2nnn(C)c2C1 36655,N1(C(C2CC(=O)NC2)=O)CC2(C1)CN(Cc1cccc(C(F)(F)F)n1)C2 36656,N1(C(C(CC)NC(C)=O)=O)CCN(C(=O)Cc2nc([N+](=O)[O-])n[nH]2)C(C(C)C)C1 36657,c1(-n2c(C(C(C(C)C)OC)NCCCCn3ccnc3)nnn2)ccc(F)cc1 36658,C1(CN)CCN(C2(C(=O)C(=O)NCC3(C)CCCO3)CC2)CC1.C1(C)CCCC1 36659,C1(NC(c2nc(CC)oc2)=O)CC2CC1N(C(C1CCC(F)(F)CC1)=O)C2 36660,N1(C(C(C)(C)OC(C)=O)=O)CCC(C)(C)C(CNC(c2c(F)cccc2F)=O)C1 36661,N1(C(CC(CC)OC)=O)CC2CCC(C1)N2C(=O)CSCC(=O)OC 36662,N1(C(C2C(C(=O)NCC#C)C2)=O)CC=C(CCNC(=O)CC2CCOC2)CC1 36663,c1(C(N2CCC(O)(C(=O)NC3CC(F)C3)C2)=O)cccc2c1OCCC2 36664,C1(C(=O)NCC2N(C(CC3(CC)CCOCC3)=O)CC=C2)CCC(C)(C)CC1 36665,C1(CC(n2cc(C(C)(C)C3CC3)nn2)(C)C)CCN(C(=O)OC(C)(C)C)C1 36666,CC(C)CC(C)CC(=O)NC(c1ccccc1)CNC(c1nncn1C1CC1)=O 36667,N1(C(c2c(C)nc(CC)s2)=O)CC2(CCCCN(C(=O)C=C3CCC(C)C3)C2)C1 36668,C1(CNC(c2c(C)noc2N)=O)CCN(C(=O)CCCC2CCC2)C1(C)C 36669,c1(NCC(CN(C)C2CC2)(C)C)ccc(S(=O)(=O)NC2CCCC2C(F)F)cn1 36670,N1(C(CC2C3CN(C(C4C(C(=O)OC)C=C4)=O)CC32)=O)CCOCC12CC2 36671,c1(CO)cc(Cl)ccc1NC(c1nnnn1C1CCOCC1)C1CC1(Cl)Cl 36672,c1(-c2nc(C)c(C(=O)Nc3cc(F)c(Cl)cc3F)cc2)ccc2c(C)[nH]nc2c1 36673,c1(OC)cc(CC(=O)O)ccc1CN1CCC(N(CC(F)(F)F)C)C1 36674,C1(CN(C(=O)C=CC(C)CC)CC)CCC(NC(=O)Cc2ccn(C)c2)CC1 36675,C1(NC(c2cn(CCNC(=O)CCCn3ccnc3)nn2)=O)C=CCCCC1 36676,C1(NC(CSCCCC)=O)CC(OC)CN(C(c2cc(C)nc(C)c2)=O)C1 36677,c1(C(=O)NC(C)CNC(C2CCC23CCOCC3)=O)n[nH]c2cc(Cl)ccc12 36678,N1(C(CCCCCOC)=O)CC2CCCN(C(=O)CCC(C)(C)C)C(C2)C1 36679,C1(NC(c2cccc(C)n2)=O)CC2CC1N(C(=O)C(F)(F)CCn1ccnn1)C2 36680,C(=O)(C1=CCCSC1)N1CC2C(CC(N3CCC(C(=O)NC4CC4)CC3)=O)C2C1 36681,C1(NC(=O)OC(C)(C)C)CCC(C(C(=O)OC)NCc2csc(=N)[nH]2)O1 36682,C(=O)(C1CCCc2ncccc21)N1C2CC(CN(C(c3ccc(Cl)o3)=O)C2)C1 36683,c1(OCC)ncc(NC(=O)CC2CCCN(C(=O)C(C)C(C)C)C2)cn1 36684,CC(C)CC(F)(F)C(=O)NC1CN(C(c2nc(C(F)(F)F)cn2C)=O)CC2(CC2)C1 36685,C(=O)(CC(C)CC(=O)NCCC(C)NC(c1ncn2c1CCCC2)=O)OC 36686,N1(C(c2cc(C)sc2)=O)CCCC(NC(c2ccn(C)c2C2CCC2)=O)C1C 36687,N1(C(c2cn(C3CC3)cn2)=O)CCCC(F)(C(N2CCCCC2CO)=O)C1 36688,c1(C(N(C2CCN(C(c3c[nH]nc3SC)=O)C2)CC)=O)cn2ccc(C)cc2n1 36689,C1(NC(COCC)=O)CC(O)(CNC(=O)C=CC(C)C)C1.C1(C(=O)O)CCCC1 36690,C1(C(=O)NC(c2nccs2)C)CCCC12CCN(C(c1ccc[nH]1)=O)C2 36691,c1(C(=O)NC2(C)CCCN(C(C3(O)CC3)=O)C2)nc(Br)c2n1CCCC2 36692,N1(C(C(C)C)=O)CCN(C(=O)C(O)CCN(C)C)C(C2CC2)C1 36693,Cc1ccc(C(=O)N(C2CCCC2)CCNC(=O)C(C)(C)C(N)=O)c(C)c1Br 36694,c1(OC)ccc(CC(=O)NCC2CC2CNC(C2(CF)CC2(F)F)=O)c(F)c1N 36695,C(=O)(C(F)CC1CCN1C(=O)O)NC1C(OC)CC1.c1(NC(C)(C)C)ccccc1 36696,C12(CNC(=O)COc3ccon3)COCCN1C(=O)CN(C(C1CCOC1)=O)C2 36697,c1(C(N2CC(O)(CN(C)C(c3cccn3C)=O)C2)=O)cccc(F)c1F 36698,CC1CN(C(c2ccnc(O)c2)=O)CCC1CNC(=O)CC1CCC(O)C1 36699,N1(C(C(C)=C(CC)C)=O)CCC=CC1C(=O)NCCc1ccnn1C 36700,C1(NC(CCC#C)=O)CC2CC1CN(C(c1cc(C(C)(F)F)on1)=O)C2 36701,c1(NC(C2(NC(C(CC)OCC)=O)CCCC2C)=O)c(C)ccn(C)c1=O 36702,c1(C(N2CC3CCC2CN3C(C23CCC(CC2)C3)=O)=O)cc2oc(Br)cc2[nH]1 36703,CCC(C)CC(=O)N1CCC(CCC2CCN2C(=O)Cc2ccccc2Cl)CC1 36704,c1(COC)cc(Br)ccc1CNC(C1CC(F)CN1C(=O)CCc1cnn(C)c1)=O 36705,c1(CC(=O)NCC(CN(C(CC2(OC)CCC2)=O)CC)C)ccc(O)cc1 36706,c1(C(=O)NC2CCC(NC(=O)CCCF)C2)cc2scc(Br)c2[nH]1 36707,N1(C(C(CC)(C)OC)=O)CC2(CC(C(=O)NOC3CN(c4ncco4)C3)CO2)C1 36708,S(=O)(=O)(c1cnc(N(C)CC2CCCC2O)c(Cl)c1)NCCc1c(C)ncs1 36709,CC1(C)CN(c2ccccc2)CC1C(N1CCC(c2ccncc2)C1)=O.C(=O)O 36710,C(C(=O)NC(C)(CNC(=O)C=Cc1cn[nH]c1)CO)(C(C)(C)C)SC 36711,c1(CC)ncc(C(=O)NCC(C)CN(C(=O)C(C(C)C)NC=O)C)cn1 36712,C12(C(=O)NCCC3N(C)CCC3)C(NC(C3CC4C=CC3C4)=O)C3CC1C2C3 36713,c1(-c2cn(Cc3c(C)nsc3)nn2)cccc(C(=O)O)c1.N12CCC(C1)C2 36714,C1(CNC(Cc2cc(OC)ncc2)=O)CCN(C(C2CC(C)(O)C2)=O)C12CC2 36715,C12(CC)CCC(C(=O)NC3CCC(NC(C4(C)CC(F)C4)=O)C3)(CC1)CO2 36716,N(C(=NCC1CCOC1)N1Cc2ccccc2C1)Cc1cnc2n1CCCC2 36717,N1(C(c2c(N)ncc(C)c2)=O)CC2CC3CC2C1C3NC(c1nc(Cl)cs1)=O 36718,c1(C(C(=O)NCCCC(C)NC(CCCCC)=O)C)ccccc1C#N 36719,CC1CN(C(C2CC(F)CN2Cc2cnn(-c3ccc(Br)cc3)c2)=O)CC1O 36720,c1(NCC2CCCN(C(C3C(C)(C)C3n3cccn3)=O)C2)ncc(C#N)cc1F 36721,N1(C(c2sc(C(F)F)nc2Br)C(=O)NCCCC)CC2(CCC2)CC1CO 36722,C(C(C)(C)CN(C(=O)Cn1cnnn1)CC)NC(CSCC#C)=O 36723,C1(C(N(C)CCOCCCO)=O)CCN(C(C2(OC)CCCCC2)=O)CC1(C)C 36724,C1(NC(C2(C(=O)NCC3C(CC)CCC3)CCCO2)=O)CCC(C#N)CC1 36725,Cc1c[nH]nc1C(=O)N(CCC(C)NC(=O)C(Cc1ccccc1)N(C)C)C 36726,C1(OCC)CN(C(c2nccc(C)n2)=O)CC1CNC(c1ccc(SC)cc1)=O 36727,C(CCCC(=O)N1CCC(CNC(=O)Cc2ccccc2C)C(C)C1)(OC)OC 36728,N1(C(C(C)OC)=O)CCSCC1CCNC(c1cnc(C(C)O)s1)=O 36729,C(=O)(C1CCC(=O)c2cccn21)N1CCCC(NC(CNC(CC)=O)=O)C1 36730,c1(C(=O)NC2CN(C(CC(C(C)C)O)=O)CC23CCC3)nn(C)c2ccccc12 36731,c1(C(N2CCOC(C)(CNC(C3(SC)CC3)=O)C2)=O)cc2ncccc2[nH]1 36732,c1(SC)cc(C(=O)N(CCCCCNC(=O)CC(C)N2CCCC2=O)CCO)co1 36733,c1(C2CN(C(C(=O)NCCC3CCN(C(C)=O)C3)=O)C2)cccc(Cl)c1 36734,C1(C(N2CC(OCCC(=O)N(CC(N)=O)C)C2)=O)CC(C2CC2)=NO1.CC1CC1N 36735,C(=O)(CC(O)C(C)C)NCC(C1CCN(C(c2c(OC)noc2C)=O)CC1)(C)O 36736,N1(C(=O)OC)CC(C(=O)N(C)C)C1.C1(C)C(=O)N1C.C1(=O)CO1 36737,N1(C(C2(C=C)CC2)=O)C2CCC(C2)C1CNC(c1cc(OC)ccn1)=O 36738,C(=O)(CC(F)(F)F)NCC1CCC(C(=O)NC2(CC=C)CN(C(C)=O)C2)C1 36739,c1(C(N2C(C)CCC(NC(=O)CCCn3cccn3)C2)=O)ccc2cncn2c1 36740,Cc1c(N)cc(C(=O)NCC(C)NC(=O)C(c2cccc(Cl)c2)O)cc1[N+](=O)[O-] 36741,c1(C(N2C(CNC(c3n(CC)ncc3)=O)CC2)=O)cc(C2CC2)nc2ccnn12 36742,C1(NC(C=CCC)=O)C2CC3C(C2)C13C(N1CCOCC1)=O 36743,N1(C(c2n(CCC)ncc2)=O)CCOC(CNC(=O)CCCc2cccnc2)C1 36744,c1(CC(=O)NCCN(CC2CC(C)(C)O2)CC)cccc(Cl)c1Cl.C1(C)CC1 36745,Cc1cc(O)ccc1C(N1CC=CC(NC(=O)Cn2cccnc2=O)C1)=O 36746,c1(C(N(C2CC(NC(c3c(C)cc(Br)o3)=O)C2)C)=O)cc[nH]c2nccc1-2 36747,C(=O)(CCC(=O)NC1CC1NC(c1csnc1C1CCCC1)=O)OC 36748,c1(C(=O)NCC2OCCN(C(CSCCOC)=O)C2)cc(OC)c2c(c1)OCCO2 36749,C(=O)(C(C)(C)CCCNC(=O)C(c1cnn(C)c1)C)N1C(CC)CCOCC1 36750,C(C(C)(Cn1cccn1)NC(c1c[nH]nc1C1CCCO1)=O)NC(C1C(=C)C1)=O 36751,c1(C(N2CCC(NC(C(CCSC)OC)=O)C(F)C2)=O)cc2oc(C)c(C)c2[nH]1 36752,c1(CC(=O)OCC2(C)CCOC2)cccc(N)c1.c1(S)ccccc1O 36753,CC1CCN(C(=O)C(C2(O)CCC2)NC(=O)COCCCN=[N+]=[N-])CC(C)O1 36754,CCCC(C)(C)C(=O)NC1C=CC(C(N2CC(=O)NC(C(=O)OC)C2)=O)C1 36755,N1(C(c2nncc(OC)c2)=O)CC(F)(F)CC1(C)CNC(c1ccc(Cl)cn1)=O 36756,CC1(CNC(C2CCN(C(C3OCCCC3(C)C)=O)CC2)=O)NC(=O)NC1=O 36757,c1(C(C(=O)Nc2ncc(CSC3CCOC3)s2)N(CCC)C)ccc(C)cc1Cl 36758,C1(C)(CC)C=C(C(=O)N2CCOC(CC(=O)NCCOCC(C)(C)O)C2)C1 36759,C(=O)(C(CO)C(C)C)NC(C)CN(c1ncc(Br)c(O)n1)C 36760,C(=O)(C1CCc2c[nH]nc21)NCc1cn(CCC(=O)OC)nn1 36761,C1(NC(c2c(C)cn(C(C)C)c2)=O)CC(F)CN(C(c2nn(C)c(Cl)c2Cl)=O)C1 36762,C1(=CC(=O)NC(C2(NC(C3CC(n4ccnn4)C3)=O)CC2)C)CCC(C)C1 36763,C1(O)(CNC(C(C)N(C)C)=O)CC(NC(=O)CCc2cnn(C)c2)C1 36764,C1(O)(CN(C(C(C)CF)=O)C)CCN(C(C2CCCC2C(F)F)=O)CC1 36765,CC(=O)C(C)(C)CC(=O)N1CC=CC(NCC=CC(=O)NC(C)C)C1 36766,CCC(C)CCN=c1[nH]c(=NCC2CC23CCC3)c2ncccc2[nH]1 36767,CC1(C(=O)NCC2CCCC(NC(=O)C(=O)NCC(F)(F)F)C2)CCC2CC2C1 36768,c1(NCC(c2onc(CC)n2)OC)cccc2c1CCN(C(C)CO)CC2 36769,c1(C(=O)NC2CC(F)(CC3CC(C(=O)N)C3)C2)ccc(OC2CC2)nc1.C1(N)CC1 36770,C(=O)(C1=COCCC1)N(CCNC(CS(CC)=O)=O)CCc1ccccc1 36771,C1(C(N2CC(=CCC)C2)=O)CN(C(C2CC(N(C)C)C2)=O)CC1F 36772,Cc1cc(C2(C(=O)NC3CCCN(CCC4CC=CCC4)C3)CC2)cc(C)c1 36773,Cc1ccnc(C(=O)N(CCCC(=O)N(C)CCN2CCCC2)C)n1 36774,c12cnc(nc1)NC(C)C1(O)CN(C1)C2=O.C(C(F)(F)F)=CC=O.CO 36775,N1(C(C(CC)=CC)=O)CCCC(O)(CCCCNC(=O)C(C(C)C)NC(=O)NC)C1 36776,N1(C(c2c(C#N)ccs2)=O)CC(NC(c2ccncc2O)=O)CC12CCCOC2 36777,C(CN=C(NCC(C)C)N1CC(O)C(C)(C)C1)c1c(OC)ccnc1 36778,c1(C(=O)NC2(CCNC(CSCCC)=O)CCC2)scc(C)c1C 36779,CCCCC(O)C(=O)NCC(O)CO.C12(CCCC1)C(=O)N2C(C)C 36780,Cn1cc(-n2cnc(C(=O)NC3(C)CC(NC(C4CC4c4cccs4)=O)C3)c2)cn1 36781,C(=O)(C#CC1(C)CCCO1)N(CCC(=O)NCC(CC)C(C)C)C(C)C 36782,c1(C(=O)NC2CC(C)(NC(C3N(C)C(=O)CC3)=O)C2)cn(C)c(=O)nc1O 36783,c1(CCC)cc(OC)c(OC)c(OCC(C)(C)C(=O)N(C2COC2)C(C)C)c1 36784,C1(O)(CN(C(=O)C(=Cc2c[nH]cn2)F)C)CCN(C(C2CCCC2O)=O)C1 36785,N1(C(c2ccn(CCCC)n2)=O)CCC2(NC(=O)C=CC3CC3)CCCCC12 36786,c1(OC)ccc(F)c(CC(=O)NC2CCN(C(C3(C(=O)N(C)C)CCC3)=O)C2)c1 36787,C12CCC3(C1)CN(C3)C2.Cc1c(Br)c(CC(=O)OC(C)(C)C)nn1CC(F)(F)F 36788,c1(C(C)NCC(C(F)(F)F)N2CCN(c3nnc(C#N)s3)CC2)ccc(Cl)cc1Cl 36789,C=CCC(CC=C)C(=O)N1CCC(C(=O)N(CCCCC)C)(CC)C1 36790,C1(NC(C(C)(C)OC)=O)CCC(C)C(C)C1 36791,c1(C(=O)NCC2C(C)CCN(C(C3(CC=C)CCC3)=O)C2)cnc2c[nH]nc2c1 36792,N1(C(C=CC(CC)=CC)=O)CC(NC(c2nccnc2C)=O)CC1CO 36793,Cc1c(CNCC2(F)CC2)ncnc1N1CCC(OC2CCC2)CC1 36794,n1(CCC(=O)NCCCCCN(C(=O)CC2CC23CC3)C)ccc(O)nc1=O 36795,c1(C(N(C)CC2N(C(CCC#C)=O)CC(F)C2)=O)cncc(F)c1C 36796,c1(CCc2nn[nH]n2)ccc(OCC2C(C(C)C)OCC2)nc1Cl 36797,CCCC(C)(CC)C(=O)NCc1cccc(C(=O)NCC2CC23CCSCC3)c1 36798,C1(C(N(C2CN(C(C(c3cccnc3)C)=O)C2)C)=O)C(C)(C)C1(C)C 36799,C1(NC(CC(CCC)CCC)=O)CC2CN(C(=O)C(C)NC=O)CCN2C1=O 36800,CCC(CC)C(C)C(=O)NCC1CCN1C(=O)CCCOc1ccc(F)c(F)c1 36801,c1(C(C(C)N(C(c2cc(S(C)(=O)=O)n(C)n2)=O)C2CC2)O)ccc2ccccc2c1 36802,c1(CC(=O)NCCC2C(C)CCCC2)cc(Br)ccc1Cl 36803,Cc1cc(C(=O)NC(C)C(C)NC(=O)CCc2cc[nH]n2)cc(N)c1 36804,N1(C(=O)CCn2cncn2)CCC(C2CCCN2C(c2cnns2)=O)CC1 36805,c1(C(N2C(C(N(CC(C)OC)C(C)C)=O)CC2)=O)ncc(Cl)cc1Cl 36806,c1(OC)c(C(=O)NCCC(C)N(C)C(C2CC2CF)=O)cc(Cl)cc1Cl 36807,N1(C(c2cnc(CC)[nH]2)=O)CCC2CCCN(C(c3cn(C)nc3CC)=O)C2C1 36808,C1(NC(C=NOC)=O)C2CCN(C(=O)C(C)Cc3cccnc3)CC12 36809,C1(C(=O)NCC2N(C(c3nc(C)sc3)=O)CCCC2)CC2CC1C1C2C1(F)F 36810,C#CCC(CC(F)F)C(=O)N1C(C(=O)NCC2(O)CCCCC2)CCC1C1CC1 36811,c1(NC(C2CN(C(=O)Nc3ncccn3)C3CC23)=O)cc(OC(F)(F)F)ccc1F 36812,c1(C(=O)NCCCC2N(C(c3c(C(C)C)ncs3)=O)CCC2)cc2n(n1)CCC2 36813,c1(OC)ccc(Br)c(CC(=O)NCCC(C)(C)NC(=O)C2=CCCC2)c1 36814,c1(C(=O)NC(CC)C(=O)NCC(c2nncn2C)O)ccc(CO)nc1 36815,C1(CNC(C2C(CNC(CSC(C)(C)C)=O)OCC2)=O)CC(C2CCC2)C1 36816,C1(CC#C)(C(=O)OC(C)(C)C)CCCC1.C1(C)C(=O)N1C1CC1 36817,c1(NCC(C2CCOC2)C)ccc(Cn2cc(CN(N3CCCC3)C)nn2)o1 36818,c1(NC(CC(COC)NC(=O)C(O)CSC)=O)ccccc1N=[N+]=[N-] 36819,c1(C(Cc2onc(-c3nccc(C)c3)n2)(F)F)cc(Cl)ccc1Cl 36820,C1(N(C(=O)CCN2CCOC2=O)C)CCCC(NC(c2cc(Cl)n(C)n2)=O)C1 36821,c1(C(N2CC3CC2CN3C(c2nc3ccccc3o2)=O)=O)cccn2ncnc12 36822,CC1CCC(O)(c2noc(C(F)(F)F)n2)CC1.C12CCCN(C1)C2 36823,C1(C(=O)NCc2nc(C)on2)CCN(CC(O)C(C)(C)C)CC1 36824,c1(CC(=O)NC2(CC=CC(N3CCC(C)(OC)C3)=O)CCC2)c(C)nn(C)c1N 36825,CC(C)C(CC(=O)N1CCC(O)(C)C1)NC(=O)C(C)O 36826,CCC(CC(=O)NC(C(=O)NCC1(COC)CCC1)C(C)O)OC 36827,CC(C)C1=NOC(C(=O)NCC2CC3CCC2N3C(=O)C=CC2CCOCC2)C1 36828,CCC(C)C(O)C(=O)N1CCCN(Cc2[nH]c(-c3ccc(Cl)cc3)nc2C)CC1 36829,c1(C(=O)NC2C(CNC(C(C)NC=O)=O)C2)ncc(F)cn1 36830,c1(N(C)CCn2cc(Br)cn2)cc(S(=O)(=O)NC)ccc1Cl 36831,N1(C(CC2C=CC(NC(c3cc[n+]([O-])cc3)=O)C2)=O)CCn2c(cnc2C)C1 36832,CC1(C)CCCCCC1NC(=O)CC1CCCNC1=O 36833,Cc1ccc(I)c(C(=O)NC2CN(C(=O)Cc3ccc(F)cc3F)CC23CC3)c1 36834,C1(NC(C2C(C(C)C)CN(C(=O)CC3CSCCO3)C2)=O)CCNC(=O)CC1 36835,CP(C)(=O)C(O)C(=O)NCCC1CN(C(=O)CCC2CCCC2)C1 36836,CC1CN(C(=O)CCc2cccnc2F)CC(C)CN1C(=O)Cn1cnnc1 36837,C(C(C(=O)NOCCCCC1CC1)C(C)C)NC(C(CCC)C#N)=O 36838,N1(C(c2cc(OC)n[nH]2)=O)CC(C(=O)NCc2ccc(CN(C)C)o2)C2(CC2)C1 36839,C1(C(=O)NCCCCN2CCOC2=O)Cc2ccc(Br)cc2N1 36840,c1(C(N(CC(O)OC)Cc2ccccc2)C)nc2ccc(Cl)cc2[nH]1 36841,C=C(C)C(CC(=O)NCC1CCC1NC(=O)COCc1ccc(F)cc1F)OC 36842,C1(NC(C2CCCC(F)C2)=O)CCN(C(c2cnccn2)=O)CC12CCC2 36843,C1(NC(C=CCCC)=O)(COC)CCN(C(=O)CCC=C(C)C)C1 36844,c1(C(=O)NC2CC(NC(CCC=CC)=O)C23CCC3)cc2ccccn2n1 36845,C12C(CC)CCCN1C(=O)COC2=O.c1(C(=O)NC2(C)CCC2)ncsc1C(C)C 36846,C1(C(=O)NCCOC2CCN(C(C(C)(C)CC3CC3)=O)C2)CCCCC(=O)N1 36847,Cc1nn[nH]c1C(N1CCCC1C(=O)NCC1(C(O)C(C)C)CC1)=O 36848,c1(C(N(CC(CC)NC(=O)Cc2ccco2)CC)=O)c[nH]nc1-c1ccco1 36849,C12(C(=O)NC3CC(NC(C(CC)(C)O)=O)C3)CC3CC(C(=O)N1)C2C3 36850,c1(OC)c(C(=O)NCC2CCCN(C(=O)C(C)S(N)(=O)=O)C2)ccc(Cl)c1C 36851,N1(C(C2N(C(C(C)NC=O)=O)CC(F)C2)=O)CCOC(C)(C)C1 36852,c1(C(N(C)CC2CN(C(c3ccncn3)=O)C2)=O)cc(N)cc(O)n1 36853,C1(C(=O)NCCOCCNC(c2c(CC)scc2)=O)CC2CCCC2C1 36854,C(=O)(C(C)(C)C(C)(F)F)N1CC=C(CNC(CCn2c(=O)cc(C)nc2)=O)CC1 36855,N1(C(C(CC)COC)=O)CC2CCCC(C1)N2C(=O)C1=NOCC1 36856,C1(C(C(=O)CCC2CCCCO2)=O)(CC(=O)N(CCO)N)CC12CCC2.C1(C)CC1 36857,c1(C(=O)NCC(C)(CC2CCCCC2)NC(CNC(=O)NC)=O)cnccc1C 36858,C1(CC(=O)NC2(CC)CN(C(CCC#C)=O)C2)CCCC1O 36859,CC(C)CC(CNC(C1(C(F)(F)F)CC(F)(F)C1)=O)NC(c1ccccn1)=O 36860,C1(CC=CC)CCCN(C(=O)CC2CC2CNC(=O)C(C)OCC)C1 36861,C1(NC(C(c2scc(C)n2)C)=O)CC2(CCN(C(C3(CO)CCCCO3)=O)C2)C1 36862,N1(C(c2c(C)cns2)=O)CC(C(N2CC(O)CC2CO)=O)CC12CCC2 36863,c1(C(N2CCC(Br)C2)=O)cnn2c1CN(Cc1ccc(F)cn1)CC2 36864,C1(C(=O)NC23CC(NC(c4c(CC)c[nH]c4)=O)(C2)C3)CC(=O)NC(C)C1 36865,c1(C(NOCC(C)CC2CC2(F)F)=O)cc(OC(F)F)cc(Cl)c1 36866,CC1CN(C(=O)C(C)(F)F)CCN(C(C2CC3(C2)CC(C)(C)C3)=O)C1 36867,Cc1cc(F)ncc1CN(CCC(=O)NC1CCOCC1)CC1CC1 36868,N1(C(c2cc(CC)[nH]n2)=O)CC2CCC(C1)C2NC(c1cc(CSCC)on1)=O 36869,c1(C(N2CCC(CNC)C2)=O)c(I)cnc(Cl)c1F 36870,c1(CC)cc(C(=O)NCC2CC(CNC(=O)CN(c3ccccc3)C)CO2)on1 36871,c1(C2C(C(=O)NCCC3(CNC(=O)CN4CC(F)C4)CC3)C2)ccc(F)cc1F 36872,N1(C(c2[nH]nnc2C2CC2)=O)CC2(C=C(C(=O)NCCO)CO2)C1.N12CC(C1)C2 36873,c1(-c2cc(C)ncc2)ccn2cc(C(N3CC(O)C(F)C3)=O)nc2c1 36874,N1(C(COC)=O)CC2CCCN(C(c3ccc4oc(O)nc4n3)=O)C2C1 36875,Cc1ccc(OCC(=O)NC2CCC23CN(C(=O)CCC(F)F)C3)c(C)c1 36876,N1(C(CC(C)OC)=O)CCn2c(CNC(c3nnsc3SC)=O)nnc2C1 36877,Cc1cccc(C(=O)NC2CCC(C)(CNC(c3cc(C(F)(F)F)no3)=O)C2)n1 36878,c1(C(CC)CC)cc(C(=O)NC2CC(CNC(=O)CN3CSCC3=O)C2)on1 36879,C=CC(CC)CC(=O)NCC=CCNC(=O)C(c1cccc(Cl)c1)(F)F 36880,c1(C(=O)NSCCC)cc(N)ccc1F.C12CN(CC1C)CCc1cn2nn1.NCCC.S.SCCO 36881,c1(C(C(=O)NCCCCCN(C(C2CN(C)C2)=O)C)=O)c[nH]c2cc(F)ccc12 36882,c1(C(=O)NC(CNC(CC2(C=C)CC2)=O)CO)cc2ncccc2o1 36883,C1(NC(C(C=CCCC)O)=O)CCC(O)CN(C(c2c[nH]c(=O)s2)=O)C1 36884,c1(C(N2CC(NC(c3cnc(CC)s3)=O)C2)=O)cc(C(=O)OC)ccc1O 36885,N1(C(CCN(CC=C)C(C2CCCC(=O)N2C)=O)=O)CC2(NC(C)=O)CCC1CC2 36886,c1(C(=O)NC)cccc(C(C(=O)NCCC2NC(=O)NC2=O)OC)c1 36887,c1(C(N2C(C(=O)NCC3C(C(=O)OC)C3)COCC2)=O)cn2cc[nH]c(=O)c2n1 36888,n1(CCC2(C(N3CCOCC3)=O)CC2)cc(CCOCC2CC2)nn1 36889,C(=O)(C1=C(C)OCC1)NC(C1N(C(c2n(CC)nc(C)c2)=O)CCCC1)C 36890,c1(C(=O)NCC(=O)NC2C(CNC(=O)CCn3cncn3)C2)ccc(Cl)cc1Cl 36891,Cn1ccc(CCC(N2CC(CC(=O)N(C3CCC(CC4CC4)O3)C)(OC)C2)=O)n1 36892,c1(NC(=O)CC2COCCN2C(C2CC3CCCC3C2)=O)ccc2nc(O)[nH]c2c1 36893,c1(NC2CN(C(c3cnn(-c4ccccc4)n3)=O)C2)ccccc1SOCCO 36894,N1(C(C2N(C(C)=O)CSC2)=O)CCCCCC(NC(c2csc3cncn23)=O)C1 36895,c1(C(N(CCN(C(CN(CCC)C)=O)C(C)C)C)=O)cc(C)c(Cl)cc1C 36896,N1(C(CC2CC(OC)C2)=O)CCCC(C)C1CCNC(=O)CCC1CC(F)(F)C1 36897,C(=O)(CCCN=[N+]=[N-])NC1C(NC(c2nn(C(CC)C)c(C)c2)=O)COCC1 36898,N1(C(c2c(C(C)C)noc2)=O)CCC(C(C)(C)CNC(C2CCCC2C)=O)CC1 36899,c1(C(=O)NC(c2ccc(N(C)C)cc2)C)cnn2ccc(C#N)cc12 36900,N1(C(CNC(CCC)=O)=O)CC2CCCC(CNC(=O)C(=O)O)(C2)C1 36901,c1(CC)ccc(C)c(C(F)(F)F)c1.c12nc(n(C)n1)C2 36902,C1(NC(c2ccn(CC)n2)=O)CC2(C1)CC2NC(=O)CCc1ccc(C(F)F)o1 36903,c1(C(=O)NCC2(O)CC(NC(c3cn(CCO)nn3)=O)C2)cc(Cl)ccc1O 36904,C1(CC)(NC(C2CC3CC3C2)=O)CCCN(C(C2CC(=O)N(C3CN(C)C3)C2)=O)C1 36905,C1(C(N(CC(=O)OCCC)C)=O)CCC(CNC(C2(CO)C=CCC2)=O)C1 36906,c1(CC(C(=O)NC2CCC(NC(CCSCCC)=O)CC2)C)ccc(F)c(F)c1 36907,CCCCC(C)C(=O)N1CCC(CC(=O)NC(CC)C(C)CN(C)C)C1(C)C 36908,C1(CNC(CC2N(C)CCC2)=O)CC2(C1)CN(C(c1cc(CO)on1)=O)C2 36909,C(C(C)(C)CNC(c1nocc1Br)=O)N(C)C(C1C=CCCC1)=O 36910,C1(N(C(C(C2CC(C)(C)C2)OC)=O)C)C2CN(C(=O)CC(C)(F)F)CC12 36911,C(=O)(C1=CC2C=CC(C1)C2)NC(CCC)C(=O)NC1CCN1C 36912,c1(-c2nc(C(CCCCCC)C)on2)ccccc1[N+](=O)[O-].C1(=O)CCC(=O)O1 36913,c1(C(C)(F)F)ccccc1C(=O)NCC1CN(C(=O)CC2(O)CCC2)CC1O 36914,C(=O)(C1=CS(=O)CCC1)N1C(CNC(C=Cc2c(C)ccs2)=O)COCC1 36915,c1(OC)ccccc1CNC(=O)C(=O)NC(C1(Br)CC1)C 36916,c1(N(CC(=O)NCC(CCCC)NC(=O)CC(F)(F)F)C)ncnc2[nH]cnc12 36917,Cc1ccc2oc(C(=O)NC(CNC(C3CN4CCN3CC4)=O)C3CC3)cc2n1 36918,C(=O)(C(=O)C(C)(C)C)N1CCC(OC)(CNC(c2ccccc2SC)=O)C1 36919,CC(C)CC(C)(CNC(=O)CC1CC2C=CC1C2)NC(C1(C(N)=O)CC1)=O 36920,C1(CNC(C(CC)C)=O)CCCCN1C(=O)NCC(C)(C)n1cccn1 36921,c1(NC(C2CC(SCCO)C2)=O)cc(Br)cnc1N1CCCC1 36922,CCC(C)(C(=O)NCC1CC(OC)CN1C(=O)C=Cc1cccc(F)c1F)C(F)F 36923,C(=O)(C(CC)C(C)O)NCC(=C)CCNC(c1cnc(CC(C)C)s1)=O 36924,c1(C(=O)NC2CCC(N(C(Cn3ncc(C#C)c3)=O)C)C2)ccc(OC)nc1Cl 36925,N1CCC2CC12C(=O)NCCn1ncc(C(N)=O)c1.C12(CO)CCC(NC3CC3)C1C2 36926,N1(C(CC2CN(C(C)=O)C2)=O)C(CCC(=O)NC2(CO)CCC2)CC2CCCCC12 36927,c1(NC(C(C2CCCN(C(=O)CNC=O)C2)(C)C)=O)ccccc1F 36928,C1(NC(CCOCC#C)=O)CCC(CNC(=O)CC2CCCC2)C1 36929,C(=O)(C(O)P(C)(C)=O)N1CCC(NC(C(C)OC(C)(C)C)=O)C1 36930,C1(OC)CC(CNC(=O)CC2CCN(C)CC2)N(C(c2cnn(C(C)C)c2)=O)C1 36931,c1(C(N2CC(NC(c3cc(CC)nn3C)=O)C(C)C2)=O)nc(C)c(C)[nH]c1=O 36932,c1(CCC(=O)NCCN(CCC)C(C2CCC2(C)C)=O)nc(-c2cccs2)no1 36933,Cc1cc(C(=O)NC2(CNC(c3c[nH]c4nccc-4c3)=O)CCC2)c(C)cc1Cl 36934,CCC(C(=O)NC1CC1NC(=O)CCc1sccc1Br)c1ccccc1 36935,Cc1cnc(C(=O)NCC2C(C)CCN2C(c2cnn(C3CC3)c2)=O)cc1C 36936,c1(OC)ccc([N+](=O)[O-])cc1C(N1CCC12CN(c1ncccn1)C2)=O 36937,c1(C(=O)NC(CCN(C(C(CC)n2cncn2)=O)C)C)ccccc1C(C)=O 36938,N1(C(C(Br)=C(C)C)=O)CC(C)OC2(CCN(c3nc(Cl)ncc3C(N)=O)C2)C1 36939,CCCCC(C(=O)NC1CCN(C(C2CCCCS2)=O)C1C1CC1)N(C)C 36940,N1(C(C2C(OC)CCC2)=O)CC(C(=O)O)C2(C1)CN(CCCc1ccccc1)C2 36941,C1(CNC(C2CN(C(C)C)C(=O)C2)=O)C(C)CCCN1C(=O)C(C)(C)C1CCC1 36942,c1(N2C3CC(NC(CNC(=O)OCC)=O)CC2C3)ncc(F)c(C(=O)OC)n1 36943,C1(NC(c2ccnc(C)n2)=O)CN(C(C2CCCC(F)(F)C2)=O)CC1S(C)(=O)=O 36944,c1(SCC(=O)N(CCN(C(C(C2CCCCC2)NC(C)=O)=O)C)C)n[nH]c(O)n1 36945,Cn1nc(NCC2CC3CC(OC(F)F)C3C2)c(C(F)F)c1Cl 36946,C(=O)(C1=NOC2(CCN(C(=O)CC3(O)CCC3)C2)C1)N1CCN(C)CC1 36947,Cn1c(C(=O)NCCCNC(c2c(F)cccc2Br)=O)cc2c1CCOC2 36948,C(=O)(CCCCO)NCCC1CCN(C(C(C)SC)=O)C1 36949,n1(CCOC)nc(C2CCCC2)nc1-c1cc(OC)ccn1 36950,c1(C(CC)C)ccc(C(N2CCN(C(c3ccncc3)=O)CC2CO)=O)c(O)n1 36951,c1(C(=O)NC2CCCC(NC(C3CC(n4ccnn4)C3)=O)C2)cccc2ccsc12 36952,CC(CC(=O)OCCCCc1ccc([N+](=O)[O-])cc1)C(C)(C)C 36953,N1(C(C(CC)NC(N)=O)=O)CCCC(N(C)Cc2ccc(F)c(Cl)c2)CC1 36954,C1(NC(=O)OC(C)(C)C)CC(C(N2CCCC2c2ncno2)=O)CN(C(N)=O)C1 36955,C1(CC=C)(NC(=O)CC(C)(C)C)CCCN(C(=O)CSc2ccc(C)c(C)c2)C1 36956,CN1CCCC(C(=O)NCCC2(CNC(c3scnc3Cl)=O)CCCC2)C1 36957,Cn1c(Cl)nc2nc(Cl)nc(N3CC4C(CNC(C5COCCO5)=O)C4C3)c12 36958,CCC(C)(C)CC(=O)N1CCCC(CCNC(C2CCC3(CCC3)C2)=O)CC1 36959,C(C1=NOC2CN(C(=O)C=Cc3cncs3)CC12)N(C(=O)COC1CCC1)C1CC1 36960,Cn1ncc2c(NC3CC=CC3)[nH]c(=NCC34CCCC3C4(F)F)nc12 36961,C#Cc1cn(C)nc1C(N1CC2CC1CN2C(=O)CCCCNC(C)=O)=O 36962,c1(C(N2CC(C(C)NC(=O)CCc3cncs3)C(O)C2)=O)cc(F)cc(F)c1 36963,C(=O)(CCC(=O)N1CC(C(F)(F)F)CC1CN)NC 36964,C(=O)(CCC(=O)NC(COC(C)=O)CO)OCC.C12(O)CC(C1)NC2=O 36965,C1(NC(C2CCC3(CCC3)OC2)=O)CC2CCCC(C1)N2C(C1CSC1)=O 36966,C1(C(N2CC(C#N)(SC)C2)=O)(CC)CCCN1C(=O)C=CC1CCCN1C 36967,C(=O)(CC(CC)CC)NC(CCCC)CNC(c1ccn(CCF)n1)=O 36968,c1(C(=O)NCC2CC(OC)CN2C(=O)CC(C)F)cc(Cl)c2[nH]c(O)nc2c1 36969,N1(C(CC2(CC)CCC2)=O)CCC2CC2(C(N2CC(C#N)(CCF)C2)=O)CC1 36970,c1(C(C)(CNC(C2(O)COC2)=O)NC(Cc2cn(CC)nc2)=O)ccc(F)cc1 36971,c1(NC(CC(CC)C2CC2)=O)c([N+](=O)[O-])ccc(F)c1Cl 36972,c1(C(CC)C)nc(C)cc(=NCC2CCCN(C(c3cc(CO)oc3C)=O)C2)[nH]1 36973,C12(C(N3C4(CN(C(c5cnc[nH]5)=O)C4)CC3)=O)CC3CC(CC(C3)C1)C2 36974,c1(Cc2nc(C)c(-c3nc(-c4cnc(Cl)cc4Cl)no3)s2)ccc(C#N)cc1 36975,C1(C(N2CC(c3cc(C)on3)(O)C2)=O)C=CCNC1=O 36976,N1(C(c2cc(OC)ncn2)=O)CCC(CCNC(=O)COCC(C)C)CC1C 36977,c1(N2CCC(C(=O)NCC(C)NC(C(C(=O)OC)C)=O)C2=O)c(F)cccc1F 36978,C1(C(N2C(CC(=O)NCC=C(Cl)Cl)CC2)=O)CC2C(C1)C2(F)F 36979,c1(C(CCCOC)C)nc(C2CCCN(C)C2)nn1-c1ccc(F)cc1 36980,n1(C(CCC)C)ncc(C(=O)Nc2nccnc2-c2cnn(C)c2)c1C 36981,C1(Cn2cc(C(C)O)nn2)CC(CNS(C)(=O)=O)CN1C(=O)CC1(C)CCOC1 36982,C1(C(=O)NCC(C)NC2(c3ccccc3)CCC(=O)NC2)C2CC3C(C2=O)C13 36983,CCC(O)C(=O)N1CC(CCNC(C2CC(F)(CO)C2)=O)C1 36984,C12(C(=O)NC(CN(C(COCCC)=O)CC)C)CCC(C)(CC1)CC2 36985,C1(NC(c2c(C)onc2)=O)C2CC1N(C(C1(n3cccn3)CCC1)=O)C2 36986,c1(OC)ccccc1C(CNC(=O)CCF)NC(=O)C(c1cnccn1)C 36987,C#Cc1cncc(C(=O)NCC(C(C)(C)C)NC(=O)Cc2ccsc2Cl)c1 36988,N1(C(c2c(CC)nnc(C)c2)=O)CC2(COC(CNC(=O)C=NOC)C2)C1 36989,C(C)(CC)(CCNC(=O)C(C)Cc1cnn(C)c1)NC(C(C)=CC)=O 36990,N1(C(C)CC(=O)N2CC(NC(C3(C(N)=O)CCC3)=O)C2)C(=O)CCC1=O 36991,c1(OC)nc(C)ccc1C(N1CCCCC1CNC(C1(C)CC(O)CN1C)=O)=O 36992,C1(C(N(C2CC(SC)C2)C)=O)CCCCN(C(C2CCOC2(C)C)=O)C1 36993,C12CCN(C1)CC1CC(C1)C(=O)N2.C(CC(=O)NC(=O)C(C)C)=CC 36994,Cc1sncc1C(=O)N(C(C(=O)N(C1CC1)Cc1ccccc1)C1CC1)C 36995,C1(N(CC(C)C)C(c2c(CCC)n[nH]c2)=O)CCN(C(c2cscc2C#N)=O)CC1 36996,c1(CCN2CC(C3CC3C(=O)OC(C)(C)C)(C(=O)OCC)C2)ccc(C)c(F)c1 36997,c1(C(=O)NCC(C)N(C(=O)CO)CC)ccc(Br)c([N+](=O)[O-])c1 36998,C1(CC(N2CCCC(C(N3C(C)CC3CO)=O)C2)=O)OCCCC1(C)C 36999,Cc1cc(NC(=O)NC2CCN(C(N3CCOC3=O)C)C2)cc(C)c1Cl 37000,c1(C(=O)NCC2(CNC(C(CC)(C)C)=O)CCC2)cc(OC)c(OC)c([N+](=O)[O-])c1 37001,C1(C(=O)NCC2C=CC(NC(c3n(CC)ccc3)=O)C2)CCc2cnc(C)n2C1 37002,S(=O)(=O)(c1cc(Br)ccc1F)C1C(CCCCCC(N2CCCC3CCCCC23)=O)C1 37003,Cc1nnc(CCCNC(=O)Nc2csc(-c3ccc(F)cc3)n2)n1C 37004,CC1CCC1NC(=O)NCCC1CC1(F)F 37005,c1(C(N(C2CCCC2)CCCNC(C(SC)SC)=O)=O)ccc(C)c(F)c1F 37006,C(C)(C)(C(C)NC(=O)CC(C)C1CCCO1)NC(C)=O 37007,C1(C(=O)NC2(CC(=O)N(CC(C)C#N)C)CC2)CCNC(=O)C1 37008,CN1C(=O)OCC1C(=O)NC1CN(C(c2cn(CCc3ccccc3)cn2)=O)C1 37009,C1(NC(COCC(C)C)=O)CN(C(=O)CCc2cnco2)C2CCCC12 37010,C1(CCC(=O)NCCOc2ccccn2)CCCCC1NC(=O)CC(Cl)Cl 37011,N1(C(=O)NCc2ccnc(CCC(=O)OCC)n2)CCC(C2(O)CC2)CC1 37012,CCC(O)C(=O)N1CCCC1C(=O)NCCCc1cn[nH]c1 37013,CC1(C)CCC(O)(C(=O)NC2CCOC2(C)C)CC1 37014,c1(NC)nc(C)ccc1C(N1CCCC(NC(c2cc3sccc3[nH]2)=O)C1C)=O 37015,CCC(CN(C)C)CC(=O)NC1CN(C(c2cc(C)nc(O)n2)=O)CC12CC2 37016,C12(NC(C3C(=C)CC3)=O)CC1CN(C(=O)Cc1sc(C3CCC3)nc1C)C2 37017,CC1CN2CCN1C(C(=O)NC(C1CCN(C(=O)Cn3cccn3)C1)C)C2 37018,N1(C(c2cc(OC)cc(Br)c2)C(=O)NC2CC2)CCCC(C2(O)CCC2)C1 37019,Cc1ccnc(O)c1C(N1CC(O)(CNC(C2CC2C#N)=O)C1)=O 37020,CCC(C(=O)OC)C(=O)Nc1ccc(C(N2CC(CC)C2)=O)nc1 37021,c1(CC(=O)NCCN(C(c2ccc(COC)o2)=O)C2CC2)ccc(F)cc1C 37022,Cc1ccc2snc(C(=O)NCC3CC3CNC(=O)Cc3cnnn3C)c2c1 37023,C(=O)(CN=c1cc[nH]cc1)N(CCNC(=O)C1=C(C)OCCS1)CC 37024,N1(C(c2nn(C)c(Br)c2C)C(=O)NC(c2ccccc2)C)CCC2(CNC(=O)C2)C1 37025,N1(C(C(n2c(C)ncc2)C)=O)CCC(C(=O)NC2CC2(C)C)C1C 37026,C(=O)(C1=C(SC)CCCC1)NCC(C)CN(C)C(c1ccc(Br)o1)=O 37027,N1(C(C(CCC)SC)=O)CC(NC(c2cnc(N)c(Cl)c2)=O)CC12CCC2 37028,CC1(C)CN(C(C2(C#N)CCCOC2)=O)CCC1NC(=O)CCCN=[N+]=[N-] 37029,C#Cc1ccccc1CC(=O)NC(C)CNC(c1cc(C2CC2)on1)=O 37030,C1(NC(C(N2CCOCC2)C)=O)CC2(CCN(C(C3CN(C(N)=O)C3)=O)C2)C1 37031,c1(C(C)C)cccc(N(C(=O)C(c2cccc(F)c2)C)C)c1 37032,c1(N(CCC=CCCC)C)nc2cccnc2c(=NCc2nn(C)cc2C)[nH]1 37033,N1(C(c2occ(C)c2C)=O)CCCC12CCN(C(=O)CC1CSC1)CC2 37034,C1(C(=O)NC(COCC=C)C)(CC=C)CCN(C(=O)C(C)=CC2CC2)C1 37035,c1(OC)cc(C(=O)NC2CCC(NC(c3csc(C(C)=O)c3)=O)C2)ccn1 37036,N#Cc1ccc(C(=O)NCC(CC2CCCC2)C(=O)NCCC(F)F)o1 37037,C12(C(N(C(CC)CC)C)=O)CC(N(C(=O)C(F)C3CC3)CC)(C1)C2 37038,N1(C(C2(C)CCN(C(c3cc(C)c(C)[nH]3)=O)C2)=O)CC2C(C1)C2(C)C 37039,C1(C(N2C3C(NC(C(CCC)=CCC)=O)C(C3)C2)=O)CCC([N+](=O)[O-])CC1 37040,c1(C(=O)NC2CC(CNC(Cc3cc(C)on3)=O)C2)c(Br)nc2n1CCC2 37041,c1(C(N2CCOC(CC(=O)NCC3CC3C(F)(F)F)C2)=O)cc(OC)ccc1Br 37042,c1(N2CCSCC(C)C2)nc(=NCCOc2ccncc2)[nH]c2c1SCC2 37043,C(c1ccc(C)cc1)=CCNC1C(CC(C)=O)N(C(=O)OC(C)(C)C)CC1 37044,c1(NCc2ncsc2)cc2occc2[nH]1.NC(=NCC1CC=CCC1)NC1CC1 37045,c1(C(=O)NCC(C)(C(C)C)NC(C(C)OCCOC)=O)ccnc2ncsc12 37046,c1(SCC)cnccc1C(=O)NC(CNC(=O)Cc1nccn1C)CC 37047,c1(C(C)C(=O)N(C2CCCC2)Cc2ccc(Cl)cc2)ccc2c(c1)OCO2 37048,C1(OC)CC(C(=O)NCC(CNC(C2CCCS2(=O)=O)=O)OC)CC1OC 37049,C1(NC(C(C)=C2CCCC2)=O)CCC2CN(CCc3ccc(CO)cc3)CC2C1 37050,Cc1ncc(CC(N2CCC(NC(=O)C(C)NC=O)C(C)C2)=O)c(O)n1 37051,c1(C(=O)NCC2N(C(C=C(COC)C)=O)CC(F)(F)C2)cc2nc(=O)ccn2[nH]1 37052,N(C1CCCc2cc(OC)ccc21)C(c1n(CC(=C)C)nnn1)c1c[nH]nc1C 37053,Cn1cc(I)cc1C(N1CCCC1c1cccs1)C(=O)NCCOC 37054,C1(N(C(C(CCC)NC(C)=O)=O)CC)CCCCN(C(=O)C=CC(C)CC)C1 37055,C(=O)(C(C)(O)CCNC(=O)Cc1cccc(C#N)c1)NCCC(C(C)C)C 37056,C(C)(N=c1nc(N(CC(Cl)Cl)C)c2c([nH]1)CCC2)c1c(C)nc(C)s1 37057,C(=O)(CCC(C)(C)C)NC1CCCOC1.c1(N(C)C)ccc(C2CN2)cc1 37058,c1(C(=O)NCCCCNC(C(C)CC(F)F)=O)cnc2c(c1)c(O)nc(=O)n2C 37059,C1(OC)CC(C(=O)N(C)CCNC(=O)CC(F)F)N(C(=O)CCCC2CCCC2)C1 37060,CCC(CC(C)C)C(=O)NCC(O)CNC(c1ccc(Br)c(Cl)c1)=O 37061,c1(NC(C(=O)NC2C(OC)CCC2)=O)ccc(C(F)F)cn1 37062,C12(C(=O)NC3C=CCN(C(C4CCOCC4)=O)C3)CC1CCC2(F)F 37063,c1(CC(=O)OC(CCOC)c2cccs2)nccc(Cl)c1F.C(C)=O 37064,N(C1CCCc2n[nH]cc21)C(C(c1cn(C)nn1)NC(C(CCCC)O)=O)=O 37065,CCCCC(CCCC)C(=O)N1CC(NC(=O)C(C)(C)NC(=O)C(F)(F)F)C(C)C1 37066,C=CCN=c1nc(N2CCC3(C2)CN(C)C(=O)O3)c2ccccc2[nH]1 37067,Cc1c(C(=O)NCCCCCCNC(=O)CN2CCCC2=O)c(C(F)F)nn1C 37068,N1(C(c2cn(CC)nn2)=O)CCC(C)(C)C1CC(=O)NC(C(O)CO)C1CC1 37069,C1(CNC(C2C(CCC)C2)=O)C2CN(C(C3CCCN3CC(C)C)=O)CC12 37070,c1(OCC)cccc2[nH]cc(C(=O)NC(CO)C#N)c12.N12CCCC(C)(C1)C2=O 37071,c1(NC)ncccc1C(N1CCC(F)(C(N2CCC(CN(C)C)C2)=O)C1)=O 37072,C#CCC(C(=O)N1CC(O)CCO1)NC(=O)CC1C=CCCC1 37073,C1(NC(C2(C)CCC(=O)NC2)=O)CC1C1CCCN(C(=O)CCCC(F)(F)F)C1 37074,C1(NC(C(CC=C)(C)N(C)C)=O)CCOC2(CCN(C(=O)CC3(OC)CC3)CC2)C1 37075,CC1CN(C(C(=O)NCc2cc[nH]n2)C2CCCC2)CC(C2CC2)O1 37076,CCC(N=c1nc(N2CCc3ncnc(O)c3C2)c2c([nH]1)CCC2)c1cccs1 37077,N#Cc1ccc(CN2CCC(O)(C(=O)Nc3cc(Cl)ccc3I)C2)cn1 37078,N1(C(c2n(C)nnc2CNC(C2(Cl)CC2(F)F)=O)=O)CC12CCC1(CC1)CC2 37079,c1(C(N(C2CCCCN(C(CC)=O)C2)C)=O)ccc2c(c1)OCCO2 37080,N1(C(C2C(C)(C)C(=O)C2)=O)CC=C(CC(=O)NC2CCC23CCC3)CC1 37081,c1(CC(=O)N(CCNC(C(COC)OC)=O)C2CC2)ncn2c1CCCC2 37082,C(=O)(C(C)(C)CCCC(=O)N(CC(C)NC(=O)CCC1CC(C)(C)CO1)C)OC 37083,C(=O)(C1=CCCCO1)N(C1CCCN(C(C(CC)=CC)=O)C1)CCO 37084,C1(CCC)CCC(C(C(=O)Nc2ccccc2OCC)N(C)CCN(C)C)CC1 37085,CC1(C)CC(O)(C(=O)NC2CCCN(C(=O)CSc3ccccc3F)C2)C1 37086,Cc1cccc(C)c1CNC(C1CCCC1NC(c1ccncc1)=O)=O 37087,c1(C(=O)NCC(CO)NC(c2sccc2F)=O)cccn2nncc12 37088,N1(C(=O)C=C2CCCC2)CCCCC(C2CN(C(=O)CC3CCOCC3)C2)C1 37089,CCC(C)C(CC(=O)N(C(c1cccnc1)C(C)C)C)Sc1ccccn1 37090,N1(C(C=C(CC)C)=O)CC2CCC2(CNC(C2CC(CC(F)F)C2)=O)C1 37091,N1(C(c2ccc(CC(C)C)s2)=O)CC=C(CCNC(C2CC2(F)Cl)=O)CC1 37092,CCCCCC(=O)OC.C12CC(C1(C)C)C(=O)NCCC1(CC1)CNC(=O)C2 37093,CC(CNC(=O)OC(C)(C)C)C(C)(C)C 37094,C1(C(N2CCN(CC=C)CC2)=O)CNC(=O)CN1C(C1(CC2CC2)CCC1)=O 37095,C1(C(=O)NCCCN(C(c2cnn(C)c2Cl)=O)CC)CC2C=CC1C2 37096,C1(CNC(CC(=C)C)=O)(OC)CCS(=O)(=O)CC1 37097,C1(CC(C)(C)C)CN(C(c2scnc2C(F)F)=O)CC1NC(=O)C(F)n1cccn1 37098,N1(CC)CC(C(=O)NCCCNC(=O)CCc2ncc(C)[nH]2)c2ccccc21 37099,C(=O)(CC1=NN(C)C(=O)C1)N(CCCC(=O)NC1CC(O)C(F)C1)C 37100,C#Cc1ccc(Cl)c(C(N2CC(NC(=O)CC(F)F)C(CCC)C2)=O)c1 37101,N1(C(c2cc(CNC(CC(C)(C)OC)=O)[nH]n2)=O)CCCC2CC1C2(C)C 37102,CCCCCCC(N1CC(Cn2cc(C(CC)CC)nn2)C1)=O 37103,O=C(N=c1ncnc2[nH][nH]cc1-2)C1CC12CN(Cc1ccc(Br)c([N+](=O)[O-])c1)C2 37104,Cn1nc2ccccc2c1CN1CCCC1(C)C(=O)Nc1cnccn1 37105,N1(C(C(CC)C)=O)CCC2CN(C(=O)CCc3nc[nH]n3)CCC12 37106,C1(CCCNC(c2c(OCC)n[nH]c2)=O)CCN(C(=O)C(O)CN(C)C(C)=O)CC1 37107,C1(CNC(c2cc(CC)nn2C)=O)CC2(CCN(C(c3cnc(C)o3)=O)C2)CO1 37108,c1(CNC2C(C(=O)OC)COCC2)nc2ccccc2n1CC(F)F 37109,C1(COC)CCC(C)(C)CN1C(c1ccc(C#N)s1)C(=O)NC1CCC1 37110,CCCCC(C)C(=O)NCc1n[nH]cc1C(=O)Nc1conc1C 37111,c1(C(=O)OC)cc(C(=O)NCC(C)CNC(c2ccc(F)s2)=O)c(F)c(F)c1 37112,N1(C(C(=O)NCC)=O)CCC2CN(C(c3ncnc(OC)c3F)=O)CCC2C1 37113,C12(CNC(C3N(C)CCC3)=O)CC(CO1)N(C(C1CCN(CCO)C(=O)C1)=O)C2 37114,Cc1ccc(C(=O)NCC(CCNC(c2n[nH]c(C)c2O)=O)N(C)C)cc1 37115,N1(CC=C)CCCC(N=c2[nH]c(=NCC3CCSC(C)(C)C3)c3[nH]ccc3[nH]2)C1 37116,C(=O)(CC(C)CCC(=O)NCC(CC(C)C)NC(=O)C=Cc1cnc(C)s1)OC 37117,C(=O)(CCCC(C)(F)F)NCCN(C(=O)CCOCC1CCC1)CC 37118,CC1(C)CC(C(=O)N(CC(N)=O)CC2CC2)CN(C(=O)Cc2ccns2)C1 37119,C(c1cccc([N+](=O)[O-])c1)=C(C)C(=O)NC1CCC(NC(=O)C(C)(C)C(F)(F)F)C1 37120,Cc1nc(C(C)(C)C)ncc1NC(=O)CSCCNC(C)C 37121,C12(C(N(C(CN(C(C)=O)C)C)C)=O)CC(C)(CN1C(=O)C(F)C(F)(F)F)C2 37122,c1(C(N2C(C)CC(CNC(=O)CN3CCOCC3)C2)=O)cc2ccccc2cn1 37123,N1(C(CC(CC)C)C)CCCOC(CNC(=O)CNC(=O)C(F)(F)F)C1 37124,C1(C(N(CCC(=O)OCC)C)=O)CN(C(=O)CCc2ccco2)CC12CC2 37125,c1(C(N(C(C)CNC(C2(C)CC2(Cl)Cl)=O)C)=O)c[nH]c2ncccc12 37126,C1(C(=O)NCC=CCNC(c2c(C(N)=O)scc2)=O)CCn2cnnc2C1 37127,CC(C)C(CO)C(=O)N1CCC(NC(=O)Cn2nnc(-c3ccco3)n2)C1C 37128,C(=O)(C(C)CC(C)C)NCC1C(CC(=O)N(CCC#C)CC)C1 37129,C1(CSC)CCCC(NC(=O)CC2(NC(=O)CC3CC3C3CC3)CCC2)C1 37130,C(=O)(C(O)CC(F)(F)F)NC1CC(C)(CC)N(C(=O)COCC(F)F)C1 37131,c1(OC)cncnc1C(=O)NCC1(CC(=O)NCCCn2ncnn2)CC1 37132,Cc1nc(CNC(=O)C(CC2CC2)NC(=O)CCC2CC2(C)C)oc1C 37133,C1(NC(=O)C=CC2CCCC2)CC2CCC1(NC(C1(F)CCCCC1)=O)C2 37134,c1(N(CC=CC(=O)OCC)C)nccc(CCNC(=O)OC(C)(C)C)n1 37135,C1(NC(C(C)SC)=O)CC2(C1)CC(CNC(c1cc(C3CC3)nc(O)c1)=O)C2 37136,C1(CC2(C)CC(NC(=O)CNC(=O)CN3CC4CC4C3)C2)CCCCC1(F)F 37137,C1(CNC(CCOC(C)C)=O)CC2COCC2N1C(C1CC12CC2)=O 37138,C1(C(N2C(C)(C(=O)NC)CC2)=O)CCN(C(C2(CC3CC3)CCC2)=O)CC1(C)C 37139,C1(C)(C(N(C(C)Cc2ccco2)C)=O)CCCCC1(C)C 37140,C(CC(O)C(=O)NCC(C1CCC1)NC(c1ccc(-n2ccnc2)nc1)=O)SC 37141,C1(CNC(CN(CC(C)C)C(c2cnsc2)=O)=O)CC(C)(C)CCO1 37142,c1(C(=O)NC2(C)CC(NC(c3c(C)ncc(C)c3)=O)C2)ccc2nnn(C)c2c1 37143,c1(N2CCC(CC)CC2)cc(NC(c2ccc(C)cc2)CF)nc(C)n1 37144,C1(C(=O)NCC(CNC(C2CCOCC2)=O)OC)CCCCCC1(F)F 37145,C1(C)(C(=O)NCC2C(NC(C=CC=CC)=O)COC2)CC2CCC(C1)S2 37146,N1(C(c2ccc(Cl)cc2F)C(=O)NC(CC)(C)C)CC(C)OCC1(C)C 37147,N1(C(C2=CCCCC2C)=O)CCn2nc(CNC(=O)C3CC3)cc2C1 37148,C1(O)(CNC(C=CC(CC)=CC)=O)CCN(C(C2CNC(=O)C2)=O)C1 37149,c1(C(N(CC(C)NC(c2ccnc(C(C)(F)F)c2)=O)C)=O)cncc(Cl)c1Cl 37150,c1(CC(CO)N(CC(=O)O)C(C)C)ccc(C#N)cc1.C1(N(C)CC)CCCCC1 37151,c1(CC(N2CCC(CNC(Cc3cc(C(C)C)no3)=O)C2)=O)cc(F)cc(Cl)c1 37152,C1(OC)CCC(C(=O)NCC(C)CCn2cc(-c3c(C)cnn3C)nn2)CC1 37153,N1(C(C(=O)NCC)=O)CCC(O)(CCNC(=O)CC2(NC(C)=O)CC2)C1 37154,N1(C(C2CC(C#C)(O)C2)=O)CCCC(CC)(NC(=O)C(C)CC(F)F)C1 37155,c1(C(C2CC2)OC)nc(-c2oc(-c3ccccc3)nc2C)n(C2CCOC2C)n1 37156,CC1CN(C)CCC1NC(c1coc(C(C)NC(c2cncnc2)=O)n1)=O 37157,C1(NC(c2c(C)n[nH]c2)=O)CCC2(CC1)CCN(C(=O)C(=O)C(C)(C)C)C2 37158,N1(C(C)=O)CCC(C2CCCN(C(c3cc4c(s3)CN(C)CC4)=O)C2)CC1 37159,c1(C(=O)NC(C(=O)N2CCC(CC=C)C2)(C)CSC)cc(C)ncc1C 37160,N1(C(Cc2c(C)con2)=O)CCN(C(=O)Cc2ccccc2Br)C2CCC12 37161,C1(C(=O)NCCCSC)CCN(C(c2nc[nH]n2)=O)C1C 37162,Cc1ccc(F)c(C(N2CCC(F)CC2C(=O)NCC2CC(CN=[N+]=[N-])C2)=O)n1 37163,c1(C(=O)NCC(C2CCCC2)NC(Cc2cc(C)ncc2)=O)occ2c1CCC2 37164,CC1CN(C(C2(CCCF)CC2)=O)CCC1C(=O)NCCC1CCC(C)(C)C1 37165,C1(NC(Cn2ncc(C)c2)=O)CN(C(=O)COCC2CCCO2)CCC12CCC2 37166,C1(F)(CC)CCCN(C(c2csc(Cl)n2)C(=O)NCCC(=O)OCC)C1 37167,c1(C2CC(C(N(C)CC3CN(C(C(C)NC(CC)=O)=O)C3)=O)C2)ccccc1F 37168,C1(CNC(C(C)OCC=C)=O)C2CCCC1N(N1CC(C=O)C1)C2 37169,C1(C(=O)NCCOCC#C)CC(F)CCN1C(=O)CCC1CC1(C)C 37170,Cc1ccccc1-n1ccc(C(=O)Nc2ccc(C(=O)N(C)C)nc2)n1 37171,CCCCCCC(C)(CC)NCc1ccc(-c2nncnn2)cc1 37172,N1(C(c2cc(C(=O)OC)on2)=O)CCC(CCN(C)C(C2(CC)CC2)=O)CC1.C1CC1 37173,c1(CCC)cnnc(C(=O)NC2CN(C(c3cc[nH]c3)=O)CC2OC)c1 37174,c1(OC)cnncc1C(=O)NCC(O)CNC(C1(O)CCCCC1)=O 37175,C1(NC(=O)Cc2cscn2)CN(C(c2n[nH]c(O)n2)=O)C2(CCCCCC2)C1 37176,C(C1c2ccsc2CCN1C(=O)CSCCOC)NC(C1C(OC)(OC)CC1)=O 37177,C1(C(=O)Nc2cn(C)c(O)nc2=O)CCCC2CN(C(=O)OC(C)(C)C)CC12 37178,Cc1cc(C(=O)NC2CCCC2CNC(c2ccc(Cl)s2)=O)c2c(c1)CCO2 37179,[N-]=[N+]=NC1CCC(C(=O)NCC2(CNC(=O)CCCCN3CCCC3)CC2)C1 37180,CCCCCC(=O)N1CCC(C(=O)OCCCCOC)C1C 37181,C1(C(=O)NCC2CN(C(C)=O)C2)CC(F)(F)CN1C(C1CNC(=O)N1)=O 37182,c1(SC)ccc(C(=O)NC2(CNC(=O)C#CC3CC3)CCCCC2)cc1 37183,CCCCCC(O)C(=O)N1CCCC(CNC(=O)C(C)Sc2ncccn2)CC1 37184,c12nc(-c3cnn(Cc4cccnc4)c3)nn1C2.N1(CCOC(F)F)CCCCC1 37185,CCN=C(NCc1ccsc1)NC(C)CC 37186,c1(C(N(CCN(C(C2(O)CC2(C)C)=O)CC)CC)=O)scc(C)c1C 37187,C(=O)(C1=CCCCO1)N1CCC(OCCNC(C2CC(Cl)(Cl)C2)=O)C1 37188,CC#CCCC(=O)N1CC(NC(=O)Cc2ccnn2C(C)C)C(CC(C)(C)C)C1 37189,c1(C(=O)NCC2(OC)CCN(C(C3CC3CF)=O)C2)oc2ccccc2c1C 37190,N1(C(CCCC#C)=O)C2CCCC1CC(CNC(c1ccccc1C)=O)C2 37191,c1(C(C(=O)NC(CC)C2CC2)NC(=O)C(C2(C)CC2)SC)c(C)cccc1Br 37192,C12CCN(CC1)C2=O.C12(C(C)(C)N)COC(CF)(C1)C2 37193,c1(C(N2CCCN(C(C3(OC)CCSC3)=O)CC2)=O)cc2c(s1)C(C)(C)CCC2 37194,N1(C(C(CC)=O)=O)CC(NC(c2cnn(C(=O)OC)c2)=O)C2(CCOCC2)C1 37195,C1(CNC(=O)CC2CCC(O)C2)CC2CCCC2N1C(=O)CSc1ccccn1 37196,c1(OC(=O)CN(CC(NOC(C)C)=O)CC2CC2)ccc(F)c(Cl)c1 37197,C1(C2CCCN(C(c3cc4ccc(F)cc4s3)=O)C2)(NC(CC2C(C)C2)=O)CC1 37198,O=C(C1=CC2(CCOC2)C1)N1CCC(F)C(Nc2nccc(C(F)(F)F)n2)C1 37199,N1(CC(=O)NC2C(CNC(C(C)CC3CC3)=O)CC2)CCCNC1=O 37200,c1(CCC(N2C(C(=O)NCc3cc4sccc4s3)CC2)=O)cccc(Cl)c1Cl 37201,N1(C(C(=O)NCC)=O)CCC2CN(C(=O)COc3ccccc3C#N)CC12 37202,c1(C(=O)NCC2CN(C(Cc3scc(C)c3)=O)C2)cccc2cccnc12 37203,C1(C(=O)NC(CC(=O)NC)C2CC2)CC2(CC2)CN1C(=O)C(C)OCOC 37204,Cc1nc2c[nH]c(=NCC3CCCC3C)nc2s1 37205,C1(C(=O)OC)CCC(C2CCC2)CC1.C(=O)(CCN)N(CCCN(S(C)(=O)=O)C)C1CC1 37206,C1(C(=O)NC2(CC#N)CCC2)C=CCN1C(c1cccs1)=O 37207,c1(CC)cc(F)ccc1C(=O)NCCCN1CCC(NC(=O)CC(=O)OC)C1 37208,S(=O)(=O)(c1ccc(Cl)nc1)N1CC2(CC(C(=O)NCc3c(C)ncs3)C2)C1 37209,C1(C(=O)NCC(C2CCCC2)NC(C(N)=O)=O)(C(F)F)CC2(CC2)C1 37210,C1(N(C(CCn2ncc(C)c2)=O)C)CC2CC1N(C(=O)CNC(N)=O)C2 37211,Cc1cc(=O)oc(C)c1C(=O)NCC=CCNC(=O)C(=O)CC(=O)c1ccsc1 37212,c1(-c2ccc(NS(=O)(=O)Cc3ccncc3)cn2)cccc2ccccc12 37213,c1(CNC(C2(C(N(CC(C)OC)C)=O)C=CCC2)=O)cc2c(cc1Cl)NC(=O)C2 37214,c1(C(C(=O)NC2CC2)N(C2CC2)Cc2cc(F)ccc2F)nc2ccccc2s1 37215,N1(C(C(CC=C)CC)=O)CCC2(CCC2NC(c2nncn2CC)=O)CC1 37216,N1(C(C(CO)NS(C)(=O)=O)=O)CCCC(C2CCCN2C(c2cc(Cl)n[nH]2)=O)C1 37217,Cc1cc(F)c(O)c(C(N2CC(CO)C(C)C2)=O)c1F 37218,N1(C(C(C)OCC#C)=O)CCN(C(=O)CC2C(CC)C2(F)F)CC1 37219,C12(C(=O)NC3CC(C)(CNC(C=CC)=O)C3)CCCCC(=O)N1CCC2 37220,N1(C(Cc2nc(COC)sc2)=O)CCCN(C(=O)C(C2CCOCC2)O)CC1C 37221,S(=O)(=O)(c1cnccc1N1CCC(N(C)CC)(CC)CC1)N(C)CCF 37222,c1(C(N(C2CC3CCC(C2)N3CC2CC3CC3C2)C)=O)ccc([N+](=O)[O-])n1C 37223,Cc1ccc(C(=O)N(C)CCNC(C2CCOC2=O)=O)cc1OC(F)F 37224,C1(C(=O)NC)(C(=O)NC)CCCN1C(=O)CC(=O)OC 37225,c1(NC(N(C2CC(OCC)C2(CC)CC)C)=O)cnccc1[N+](=O)[O-] 37226,c1(C(=O)NC(c2nc(C)on2)C)ccnc(CNC(=O)CC2(O)CCOCC2)c1 37227,Cn1c(CC(=O)NCC(=O)NC2CC2F)nnc1S 37228,C(=O)(C(CCC1CC1)NC(=O)OC(C)(C)C)NC(C)CCC1CCCC1 37229,N1(C(CSCC)=O)CC(C(=O)NCc2cn(C3CCCCC3)nn2)OC(C)(C)C1 37230,N1(C(C(F)=CC)=O)CCCOC(CCNC(=O)CC2COC(C)(C)CO2)C1 37231,c1(C(=O)NCC(CO)NC(=O)CC2COCCO2)ccc(-c2nnc(S)o2)cc1 37232,C1(C(=O)NCCCC(C)NC(C(CNC(C)=O)(C)C)=O)CCC(C)=C(C)C1 37233,c1(OC)ccc2ccccc2c1C(=O)Nc1cc(-n2ccnc2)ccc1Cl 37234,C(CCCC(=O)NC(C1(C(=O)N(C)C(C)C2CC2)CC1)C)OCC 37235,CC(C)CC(CNC(=O)CC1CC2(CCC2)C1)NC(C1CCCCC2CC12)=O 37236,C(CCCCCC(=O)NOCC(F)(F)F)NC(Cc1nnc(C)o1)=O 37237,O=C(C1=CCCC1)NCC1CCCCN1C(=O)C=CC(c1ccccc1)=O 37238,N1(C(C2CC(=C)C2)=O)CC(NC(=O)Cc2cnc(C)[nH]2)C(c2cnn(C)c2C)C1 37239,C(N=c1nc(C)c([N+](=O)[O-])c[nH]1)C1C(C)CCN(C(C(C(CC)O)C)=O)C1 37240,c1(C(=O)NC(CC)CNC(C2CC3CCC2C3)=O)cnc2c(C)cccn12 37241,C1(N(C(C2CC(C)(C)OC(c3ccccc3)C2)=O)C2CC2)CCOC2(CCCCC2)C1 37242,c1(CNC(C2CCC(C)N2CC2(C)N=C(C)SC2)=O)cc(C#N)ccc1C 37243,c1(CCn2cc(C3CN(C(C4OCC(C)C4)=O)C3)nn2)cc(F)cc(F)c1 37244,Cc1cc(F)cc(Br)c1NC(C1CCN(C(c2cc(Cl)cc(I)c2)=O)CC1O)=O 37245,C1(=O)C(OC)CCO1.C(=O)(C(CC1CC1)OC(C1OCCC1C)=O)OCC 37246,N1(C(CCN(CC)CC)=O)CC2(CCC(CNC(C3CCCN3N=O)=O)O2)C1 37247,N1(C(CCN(C)C)=O)CC2CN(C(c3cc4cc[nH]c4cn3)=O)CC2C1 37248,C1(CSC2(C(=O)NCc3[nH]cc(C)c(=O)c3C)CC2)CN(CC)C2(CCOC2)C1 37249,c1(OC)ccc(CNCC(O)C(O)C2CCCC2)c(F)c1F 37250,C(=O)(C1=CCCC1(C)C)N1CCC(O)(CNC(CC2CCN(OC)CC2)=O)C1 37251,C1(CNC(C2(CN(C)C)CC2)=O)C(O)C(O)CN1C(=O)CSC(C)(C)C 37252,C1(C)(C(N(CCC)CCNC(=O)C(C)O)=O)Cc2ccccc2NC1=O 37253,c1(OC)cccc(S(=O)(=O)CC(=O)N2CCC(CC(=O)N(C)C3CC3)CC2)c1 37254,c1(CCC(N2CCC(NC(C3CC3(F)F)=O)C2)=O)ccc(F)c(NC(=O)OC)c1 37255,CC(C)CC(O)C(=O)N(C1CC(NC(=O)CCc2nc(C(C)(C)C)no2)C1)C 37256,N1(C(CCCCSC)=O)CCCC(C2CCN(C(=O)C3CC3)CC2)CCC1 37257,Cc1cn(C)nc1C(=O)NC(C)C(C)(C)NC(c1ncccc1Cl)=O 37258,N1(C(c2c(Cl)ccc(C)c2)=O)CCC(C2CC2)C1CNC(=O)C(N)=O 37259,C1(C(=O)NC(C2CC(CCNC(CC3(CC(=O)OC)CC3)=O)C2)=O)NC(=O)OC1(C)C 37260,N1(C(Cc2cc(C)on2)=O)CCC(NC(=O)CN(C2CCSC2)C)C(C)(C)C1 37261,C1(C(=O)NCC(c2cccs2)=O)(COC)CCN(C(C2CCC3(CC2)CC3)=O)CC1 37262,C1(CC(=O)OC(C)C(=O)NC(c2ccc(Br)cc2)C)CCCCCC1 37263,C1(NC(c2cnc3n2CCC3)C)CCC(O)(C(F)(F)F)CC1 37264,N(C1c2ccccc2CC1NC(C1CCOC1)=O)C(C=CS(CC)(=O)=O)=O 37265,CCCCCCCN=c1nc(N2CCC(CCO)(OC)C2)c2c([nH]1)COC2 37266,C12(NC(=O)Nc3cc(CN4CCOCC4)cc(F)c3)CCC(O)(CC1)CC2 37267,N1(C(CNC(CN(C)C)=O)=O)CC=CC(NC(C2CC3CCC2C3)=O)C1 37268,C(=O)(C#CC1(C)CCCO1)NC1C2CN(C(CCCCOC)=O)C(C2)CC1 37269,N1(C(c2cc(C)nc(O)c2)=O)C2CCC1CC(CNC(c1cn(C)nc1Cl)=O)C2 37270,N(C(=NCCCCl)N1CCC(OC(F)F)C1)C(CC)C 37271,C(=O)(CC(C(F)(F)F)C1CC1)N(C)CC1(NC(C(C=CCCC)O)=O)CC1 37272,C1(OC)CN(C(c2cncc(F)n2)=O)CC1NC(C1CC2CCC2C1)=O 37273,C1(OC)CCC2CN(C(C3(F)CCCN(C(=O)C(C)(C)CF)C3)=O)CC12 37274,CC1CN(C(c2cccc(C#N)n2)=O)CCN1C(C1CCCN1c1ccccc1)=O 37275,Cc1ccc(C(C)NC(=O)C(=O)NCCC2COCC2(C)C)cc1C 37276,N1(C(C(C2CCOCC2)C)=O)CCC(NC(C2CC(F)(CO)C2)=O)C(C)(C)C1 37277,C1(NC(c2cncc(OCC)c2)=O)CC2CCC1CN(C(=O)COCC(F)F)C2 37278,N1(C(C(N2CCSCC2)C)=O)CCCOC(CNC(=O)C=Cc2cccs2)C1 37279,Cc1sc(C(=O)NC2CCCC(NC(=O)CC(C)NC(N)=O)C2)nc1O 37280,c1(OC)c(C(=O)NCC2CCCN2C(c2ncccc2O)=O)c(C)nn1C 37281,c1(C(N2CC(CCNC(C3(OC)CC3)=O)(OC)C2)=O)cn2ccnc2s1 37282,Cc1cc(C(N2CC=C(CCNC(=O)CC(O)C3CC3)CC2)=O)c2n[nH]cc2c1 37283,C1(CNC(CC=C=C)=O)CCN(C(C2(C(C)C)CC2)=O)CC1(F)F 37284,C(N=c1cc(Cl)nc[nH]1)C1(C(N2CC3CCC2C(O)C3)=O)CC1 37285,CCCCC(O)C(=O)N1CCCC(NC(c2ccc(C(=O)OC)cn2)=O)CC1 37286,N1(C(C(c2ccc(C)o2)C)=O)CCC(C)N(C(=O)COc2cn[nH]c2)CC1 37287,C1(C(N(OC)C)=O)CCOCCN1C(C1CC1(F)Cl)=O 37288,C=CCC(CC)C(=O)N1CCN(C)C(CNC(C2CC3(CC3)C2)=O)C1 37289,CCC(C)C=CC(=O)NCC(C)=CC(=O)NCCN(C)C(=O)C1CC1 37290,c1(C(=O)NCC(c2ccc(C)cc2)NC(c2ncccc2O)=O)c[nH]c(C)cc1=O 37291,Cc1ccc2[nH]cc(CCNC(C3C=CCN3C(c3csc(CO)n3)=O)=O)c2c1 37292,c1(OCC)ccc2ccccc2c1NC(=O)NC1CCc2nc(C)sc2C1 37293,CCCCC(C(=O)OCc1cc(C)ccc1O)ON=C(C)C 37294,N1(C(=O)OC(C)(C)C)CCCC1C(=O)NC1CCCC1NC(C1(C)CC=CC1)=O 37295,CC(C)C1=NOC(C)(C(N2CCC(C)(CNC(=O)C=C(C3CC3)C3CC3)C2)=O)C1 37296,N1(C(c2cncc(C)c2)=O)CC(NC(=O)Cn2ncn(C)c2=O)C(F)(F)C1 37297,c1(C(C(N2CCC(CO)(NC(C3(O)CCC3)=O)CC2)=O)O)cccc([N+](=O)[O-])c1 37298,C(C)(N=c1[nH]c(=NCC2CC2)[nH]c2c1CCCCCC2)c1c(C)ncs1 37299,C1(NC(C2CCN(C)C2)=O)CC(F)CN(C(=O)COc2cccnc2)C1 37300,N1(C(C(C)(C)NC(=O)NCC)=O)CCCC(NC(=O)CC(C)C2CCCO2)C1C 37301,C(C(C(=O)NCCC1CC(=O)N(C)C1)C(C)(C)C)NC(C1CC(CC)C1)=O 37302,Cn1nnnc1C(c1ccc(C2CCCO2)s1)NC1CC1F 37303,c1(-c2occ(CC(N3CC(CNC(C(C4CC4)OC)=O)C3)=O)n2)ccc(Cl)cc1 37304,C1(C(=O)NC(C(=O)OC(C)C)C)CC(C)(C)CCN1C(=O)Cn1cnnn1 37305,C(=O)(CCCc1cncs1)NCC(CC)N(C(=O)CSc1nc[nH]n1)C 37306,CC1(C)CN(C(C2CC3(CCO2)CC3)=O)CC1NC(=O)C=Cc1cncs1 37307,c1(C(=O)NCC2N(C(C3C(C)C3)=O)CC(O)C2O)cnc2c(c1)CCOC2 37308,C1(CNC(CCCOC)=O)CC(C(F)(F)F)CN1C(C12CC(F)(C1)C2)=O 37309,c1(CC(=O)NCc2cn(C3CCN(C(C(CC)F)=O)C3)nn2)c(F)cccc1F 37310,Cc1nccc(=NCC2(CCNC(=O)C(C3CCC(=O)N3)C)CC2)[nH]1 37311,N1(C(c2c(OC)cccc2C)=O)CC(C)(CNC(C2CCCCS2)=O)CC1(C)C 37312,Cc1noc(C)c1S(=O)(=O)N(C1(C(=O)N=c2nc(C)[nH]s2)CCCC1)CCC1CC1 37313,Cc1sc(C(F)(F)F)nc1C(=O)N(CC(C)(C)NC(=O)CC1C=NN(C)C1=O)C 37314,c1(C(=O)NC2(C(N(C)Cc3ccnc(C)n3)=O)CC2)cc(O)nc(C)n1 37315,c1(C(N(CCC(=O)NC)C(=O)Nc2sccc2C)C)ccccc1Br 37316,CC(C(=O)N1CC(O)(CNC(C2CCC(=O)NC2)=O)C1)S(=O)(=O)C1CCOCC1 37317,C(C(C(C)(C)C)NC(C1(C(F)F)CC1)=O)NC(C=C(C)C(F)F)=O 37318,c1(C2C(C(N(CC=C)CCOC)=O)C2)cccnc1 37319,CCS(=O)(=O)CC(=O)N(CCNC(=O)C(=O)Nc1c(C)nn(C)c1C)CC1CC1 37320,CC1(CC(N2CCOC(CNC(=O)CNC(c3ccco3)=O)C2)=O)CCS(=O)(=O)N1 37321,O=C(C1=NOC2(CCC2)C1)NC12COC(CNC(c3ncncc3Cl)=O)(C1)C2 37322,c1(OC)ccc(CN2CCN(C(N)=O)CC2)c(Br)c1O 37323,c1(C(CNC(N)=O)N(C(=O)NC(c2ccccc2C)C)CCO)cc(F)cc(F)c1 37324,c1(N2CCC(NC(c3ccc(CCC=C)cc3)=O)C2(C)C)ccc([N+](=O)[O-])cn1 37325,C(=O)(CCCCCS(N)(=O)=O)NCC1CCCCN(C(CSc2nc(C)[nH]n2)=O)C1 37326,c1(NC(c2nc(C(=O)NC(C(CC)C)CO)sc2)=O)cc(C#N)ccc1N(C)C 37327,CCCC(C(=O)NCC1(O)CCCN(C(=O)C2=NOCC2)CC1)S(N)(=O)=O 37328,C(C(C)(C(=O)NC1CCC(CC(N2CCSC(C)C2)=O)C1)OC)OC 37329,c1(C(=O)NC(CCCNC(c2cnn(C(C)C)n2)=O)C)nccc(Cl)c1F 37330,c1(C(=O)NCC2C(NC(COCCC#C)=O)CCC2)cn2ccccc2n1 37331,c1(CCC(N2C(C3(C(=O)O)CC3)CC(OC)C2)=O)nc2c(O)nc(=O)n(C)c2[nH]1 37332,c1(CN2CC(NC(c3cocn3)=O)C(O)C2)nc2ccccc2o1 37333,N1(C(CC=C(C)C)=O)CCC2(CC1)CN(C(=O)C(C)n1ccnn1)C2 37334,C(CCCCCNC(=O)C(c1ccc(F)cc1)O)N(C)C(C1CCCOCC1)=O 37335,N1(C(CCC(C)=O)=O)CCC(O)C(C(=O)Nc2cc(C(F)(F)F)cc(F)c2)C1 37336,N1(C(C(CC)(C)OC)=O)C2CCC1CC(NC(C13CCC(N=[N+]=[N-])C1C3)=O)C2 37337,c1(-c2cn(C(CNC(C3(CC)COC3)=O)C)nn2)ncccc1C 37338,Cc1c(F)ccc(N)c1C(=O)NCC12CC(NC(=O)CC3CCCC3C)(C1)C2 37339,C=Cn1nccc1C(=O)NCCOCCCNC(C1CCCN(CC(F)F)C1)=O 37340,C(C(=O)NNC(=O)C(C)(C)CCCCNC(=O)C(C)=CC1CC1)=CC(CC)C 37341,c1(CC)cc(C)[nH]c(=NCC2(NC(=O)C3=CS(=O)(=O)CCC3)COC2)n1 37342,CN(CCc1cnn[nH]1)N1CCN(c2nc[nH]n2)CC1.C1C(=O)N1.C1C(=O)N1 37343,CC1CN(C(C2CC2CNC(C2(CO)CC2)=O)=O)CC2(CCC2)O1 37344,Cc1cnc(F)cc1C(N1CC(NC(=O)C(CC2CC2)c2ccccc2)C(O)C1)=O 37345,C1(CCC)CN(C(C2CCN(C(=O)C(C)C)CC2)=O)CCN1C(C(=O)CC(F)F)=O 37346,C1(NC(CNC(CCC)=O)=O)CC2C(CNC(=O)COC3CCOC3)C2C1 37347,CC1(C)CC(CO)CN1C(=O)CCc1nccs1 37348,c1(CC)c(C(=O)N(C)CC2CCCN2C(c2ccsn2)=O)cnn1C(C)(C)C 37349,C1(CNS(=O)(=O)CC2CCNC2)CCCCCC1 37350,N1(C(C(C=C)O)=O)CC2CCC1CN2C(c1[nH]c(C(C)=O)cc1CC)=O 37351,N(C1CCCc2cc(F)ccc21)C(c1cc2c(nc1)NC(=O)CO2)=O 37352,c1(C(CNC(C2CCCN(Cc3cccc(Br)n3)C2)=O)O)cccc(F)c1 37353,C1(CNC(c2c(C)scc2)=O)CCC(C)(C)CN1C(C1CN(C(C)C)C1)=O 37354,C1(NC2C(C(=O)NCC)CCCC2)CCC2CN(C(=O)C(F)F)CCC2C1 37355,c1(C(=O)NCC(C)CN(C(=O)C=CCN2CCCC2)C)ccc(C(F)F)cn1 37356,C1(C(N2C(CNC(c3c(CC)ocn3)=O)C(C)(C)CC2)=O)Oc2ccccc2C1C 37357,CCC(CCOC)C(=O)NCCCOCCN(C(=O)C(C)(C)N1CCCCC1)C 37358,CC1(C)CCCC(N2CCCC(Cc3ccc(C#N)cc3)C2)C1 37359,CCC(CC1CCCCC1)C(=O)NC1CC(NC(=O)C(C2CCOCC2)C)C1 37360,C1(NC(=O)C(C2CC2)C2CC2)CCC2CCN(C(=O)C(O)c3ccsc3)C1C2 37361,n1(C(C)C(N2CCC(CN(c3ncccn3)C)C2)=O)c(C2CCCCC2)nnc1S 37362,N1(C(Cc2c(C)nc[nH]2)=O)CC(NC(=O)Cc2cc[nH]c2)CC12CCCCCC2 37363,CCC(C)(CN)C(=O)NC1CCN(C(c2cc(-c3cc(F)ccc3F)on2)=O)C1 37364,C(=O)(C(CNC(c1cc(C#N)n(C)n1)=O)C(C)C)N1CCCC(CSC)C1 37365,C12(C(=O)NCCC3CN(C(C(CC)(CC)OC)=O)C3)CCCCC1C2(F)F 37366,CC1(C)CCCC(C(=O)NCCC2=CCN(C(c3ccc(C#N)[nH]3)=O)CC2)CC1 37367,c1(C(=O)NCC2(CCNC(C3CCCCO3)=O)CC2)cnc(O)c2ncccc12 37368,c1(C(=O)NC2C(CNC(CC3CCC(C)O3)=O)C2)ncccc1Cl 37369,CCCC(CCCNS(C)(=O)=O)NC(=O)CCCN.C1(=O)CN1.C(=O)(COCC)C(N)=O 37370,C(CS(=O)(=O)c1cccs1)NC(=NCC=C)NC(C)CNC(=O)OC(C)(C)C 37371,c1(C(N2C3CC(NC(C(CCC)OC)=O)C3CC2)=O)cccc2c1nnn2C 37372,N1(C(C2(CCC)CCC2)=O)CCC(OCC2CC2)C1 37373,C(C(C(F)(F)F)N1CCN(C(c2cn(CC)nn2)=O)CC1)NC(CC=CC=C)=O 37374,C=CCC(F)(F)C(=O)NC1CCCC(N(C)C(c2ncncc2N)=O)C1 37375,C(CCCCC(=O)N1CC2(NC(c3ccc(C)c(O)n3)=O)CCC1C2)OC 37376,C1(C(=O)OC)C(NCC(O)S(=O)(=O)CC(F)(F)F)C2(C)CCCCC12 37377,c1(C(=O)NCCOC2CN(C(C(C)NC(CC)=O)=O)C2)cc(C(F)(F)F)ns1 37378,c1(C2(CNC(=O)C3=CCCCO3)C(C(=O)OC)COC2)c(C)cc(O)nc1C 37379,CC1(C(NOCCCNC(=O)C(F)C2CCCC2)=O)CCCO1 37380,c1(C(=O)NC2CC(NC(C(N3CC(C)C3)C)=O)C2)ccc(CS(C)(=O)=O)o1 37381,C=CC1CCN(C(C2(CNC(=O)C(F)F)CC(=C)C2)=O)C1 37382,N1(C2C(C(=O)OCC3C(OC)CC3)C2)C(=O)c2ccccc2C1=O 37383,C1(NC(c2[nH]cc(C)c2)=O)CN(C(c2cncc(Br)c2C)=O)CC12CCC2 37384,C1(OC)CC(c2nc(C)no2)N(C(c2cccc(NC3CCC3)c2)=O)C1 37385,c1(OC)ccc(C(=O)NC2(CF)CN(C(C3CC34CC(C)(C)C4)=O)C2)c(Cl)n1 37386,c1(C(=O)NCC(C)NC(c2cccc(NCC#N)c2)=O)cc2c(cc1N)CCCC2 37387,c1(CC(N2CCC(NC(=O)CC3CC4CC3C4)C(F)C2)=O)cn2cc(F)ccc2n1 37388,c1(CC(=O)N(CCN(C(=O)C(C)CCOC)CCC)CC)ccc(OC)cc1C 37389,C1(C(=O)NCC2OCCCN(C(C3CC(=O)OC3)=O)C2)Cc2cncn2C(=O)N1 37390,C#Cc1ccc(CN(CCOC(=O)C2=CCOC2)C(C)=O)cc1 37391,C(=O)(C(C)(CC)CC)N(CC(CNC(C(CCC)=CCC)=O)O)C 37392,C(=O)(C(F)C(F)(F)F)NCCCC(CO)NC(C=CCN(CC)CC)=O 37393,Fc1cc(Br)cc(F)c1CSCc1cc(Cl)cnc1F 37394,CC1CN(C(=O)C(C)C2CCC2)CCN1C(c1cc[nH]c(=N)n1)=O 37395,C1(F)(CNC(CN(CCOC)C)=O)CCC(NC(=O)Cc2cc(Cl)n(C)n2)C1 37396,c1(C(C(=O)NCC(C)N(C)C(C2(F)CCCCC2)=O)C)cncc(F)c1 37397,C(=O)(C1CC(=O)c2ccccc21)NC1C(NC(CSc2c(C)cccc2)=O)C1 37398,N1(C(CCOCCOC)=O)CCCC(CCNC(=O)CC2CCC(=O)N2)C1 37399,c1(OC)ccc(CC(C)(C)C(=O)N(C)CCc2ccc(Cl)cc2Cl)cc1OC 37400,CC(C)CC(CNC(c1csc(F)c1)=O)C(=O)N1CCC(CC(C)C)C1 37401,N1(C(C(C)NC(=O)OC)=O)CC2(CCCN(C(=O)CC3COCCN3C)C2)C1 37402,C(=O)(CS(=O)(=O)C1CCCC1)NCCN(C(C(C)N(C)C)=O)C1CC1 37403,Cc1cc(S(N)(=O)=O)oc1C(=O)NCC1(NC(c2c(C)n[nH]c2C)=O)CC1 37404,N1(C(C=Cc2n(C)ncc2)=O)CCC2(CC1)CCN(C(c1cncnc1)=O)C2 37405,c1(C(N2C(CNC(C3C(=C)C3C(=O)OC)=O)CC2)=O)cc(C(C)C)cc(F)c1 37406,c1(C(N2CC(CNC(=O)COc3ccc(F)nc3)C2)=O)c(Cl)cncc1Cl 37407,C1(C(=O)NCC(C)N(C)C(C2(F)CC2)=O)CC(Cl)=C(C)CC1 37408,Cc1cc(C(=O)NCC(C2CC2)NC(c2cnsc2)=O)cc(Cl)c1 37409,C1(C(=O)NC2(C(=O)NCC)CC2)CN(C(c2cc(C3CC3)[nH]n2)=O)CC1(F)F 37410,C(=O)(C1=CC2C=CC1C2)NCC(CNC(=O)C(C)(C)c1cscn1)OC 37411,Cc1nccc(C(=O)NC(c2ccccc2)C(C)NC(=O)Cc2cnn(C)c2)c1O 37412,c1(OC)nccc(C(=O)NCC2(C(=O)NC3CCN(C)CC3)CCCCC2)n1 37413,c1(C(N(CC(CN(C(Cc2cc(OCC)no2)=O)C)O)C)=O)ccccc1OC 37414,CCC(C(=O)N1CC(C(=O)Nc2cn(C)nc2C(N)=O)OC(C)C1)C(C)O 37415,C1(C(N2CC(CC)(OC)C2)=O)CN(C(=O)CC(O)C2CCCC2)CC1(F)F 37416,c1(CC(=O)NCC(C2CCC2)NC(C(C)OCC=C)=O)ccc(Br)s1 37417,C1(CNC(C2N(CC)CCC2)=O)CN(C(C2CSC2)=O)CCC12CCC2 37418,c1(CC(=O)NCC(CC=C)NC(c2n[nH]cc2Cl)=O)cnc2ccccc2c1 37419,c1(OC)cc(C)c(F)cc1-c1cnc(C(=O)Nc2c(Cl)c(C)nn2C)cc1C 37420,c1(C(N2CC3(N(C(C(CCC)N)=O)CC3)C2)=O)ccc(C#N)cc1F 37421,Cc1nc(=N)[nH]c(C)c1C(=O)NCCC(C)NC(C1OC(C)CC1C)=O 37422,C1(C(=O)NC(c2cccnc2)C)C2C(CN1Cc1cc(F)c(Cl)cc1Cl)C2(C)C 37423,CC1=C(C)CN(C(C2(C)C=CCN2C(C2CC(C)C2)=O)=O)C1 37424,C(CN=c1[nH]c(=NC2CC3C(C2)C3(F)F)[nH]c2c1CCCC2)c1nn(C)c(O)c1 37425,N1(C(C2CC3(CC(=C)C3)C2)=O)CC2CCCC(C1)N2C(C1(C)CCC1C(=O)OC)=O 37426,c1(CC)cc(C)c(C(=O)NNC(=O)OCCOC(C)(C)C)o1 37427,C=CC1(CC(N2CC(OC)C(NC(=O)C(C)C#N)C2)=O)CCOCC1 37428,c1(OCC)nccc(C(=O)NC2CCCCN(C(C3(CF)CCC3)=O)C2)c1F 37429,c1(CC)cc(OC)ccc1C(N1CCC(C)(C(=O)NCc2ncc[nH]2)C1)=O 37430,C(=O)(CCCCCc1cccs1)NC1CCCN(C(c2nc(C)[nH]n2)C)C1 37431,c1(C(N2C(CNC(C(C)(C)NCc3cc[nH]n3)=O)CC(F)C2)=O)ccc(Cl)cc1 37432,c1(C(=O)NC2C=CC(CNC(c3ccc(O)nc3)=O)C2)ccc2nn[nH]c2n1 37433,c1(C(=O)NC(c2ccc(CNCCC3(C#C)CCCC3)s2)=O)ccc2ccoc2c1 37434,c1(OC)ccc(C(=O)NC2CCCC(NC(C3CCCCC3O)=O)C2)c(C)c1 37435,c1(-c2nc(C(CC)CC)nn2CCCN(C)C)ccc(Br)c(OC)c1 37436,N1(C(CC(=O)N(C)C)=O)CC2CS(=O)(=O)CC2(CNC(c2scnc2Cl)=O)C1 37437,O=C(CCN=c1[nH]c(=NCCF)[nH]c2c1COC2)N1CCOC1=O 37438,C(=O)(C1CCC(N)c2ccccc21)N(C)CC1CCCN(S(C)(=O)=O)C1 37439,C1(C(=O)NCCC2CC(NC(c3c(C)occ3)=O)C2)CCC2(CCC2)C1 37440,N1(C(CNC)=O)CCN(C(=O)CCc2ccccc2N)C2CC12.c1(S)cccnc1 37441,N1(C(C(=O)Nc2ccc(C)cc2Br)C)CCC(C2CC(O)C2)CC1 37442,CC(C)CCC(O)C(=O)N1CCOCC(NC(c2cc(CO)on2)=O)C1 37443,C1(OC)CCCC(CC(=O)NC2CCC(C(=O)NC3CC(Cl)(Cl)C3)CC2)C1 37444,CC1(C)CCC=C(C(=O)NCC#CCNC(C2CC23CCOCC3)=O)C1 37445,c1(CNC(C2N(C(C(c3ccn(C)n3)C)=O)CC3CC32)C2CC2)cccc(F)c1O 37446,N1(C(c2cncc(NC(CC)=O)c2)=O)CC2(CC(NC(=O)C(C)CCCOC)C2)C1 37447,c1(C(N2CC(F)(CNC(C3CCC(OC)C3)=O)C2)=O)nccc(C(F)(F)F)n1 37448,C(=O)(C#CC1CCOC1)NCCCCCN(C(c1nccc(OC)c1O)=O)C 37449,CCCCC(O)C(=O)N1CC(O)CC1C(=O)Nc1nc(F)ccc1C(=O)OC 37450,N1(C(CCc2ccc(C)cc2C)=O)CC2CC(NC(=O)CN(C)C3CC3)CC2C1 37451,c1(NC2C(OC)CCC2)[nH]c(=NCC2CC2C2(C)CCOCC2)nc2scnc12 37452,N1(C(c2ccc(NC)nc2)C(=O)NC(C)(C)CC)CCC2(COC(=O)N2)C1 37453,C1(C)(CNC(c2c(CNC(C3CCC(C)O3)=O)cnn2C)=O)CCCC1O 37454,N1(C(c2n(C=C)ncc2)=O)CCCC(N(C)C(C2CC3CC3C2C(=O)O)=O)CC1 37455,C#CCCCCCCC(=O)N(CCCCCC(=O)NCc1cnccc1C)C 37456,c1ccc(F)c(F)c1.N1(C(C(C)C2CCCC2)=O)CCCC(CCC)C1 37457,c1(CC)cccc(F)c1C(=O)NCCC1CC(NC(=O)CC2(C)CCCC2)C1 37458,Cn1c(C(N2CCC(Cn3cc(C4(C(N)=O)CC4)nn3)C2)=O)cc2cc(Br)cnc12 37459,c1(NC(C(=O)NCC(CC(C)C)C)=O)ccccc1S(C)(=O)=O 37460,N1(C(CC(=O)NCC)=O)CCCC(C2CN(C(c3cc(CC)c(CC)o3)=O)C2)C1 37461,c1(CNC(=O)NCC2(CC)COC(=O)C2)ccc(I)c(O)c1 37462,C12C3CCC1CN(C3)C2.c1(NC(C=C(CCC)CCC)=O)ncc(C)cc1Br 37463,C(CC(F)F)(C(=O)NOCC)NC(C(CCC)F)=O 37464,c1(OCC(C)C)cccc(C(N2CCCC(CCOC)C2)C(=O)NCC(C)C)c1 37465,N1(C(CCC2(C)CCCN2C(c2ccccc2Cl)=O)=O)CC(O)C2CCCCC12 37466,c12cc(ccc1C1CC1)CS2.Fc1cnccc1CN1CCCC1 37467,c1(C(=O)NCC2CCCC2NC(C2CCOC2)=O)c[nH]c2ccccc12 37468,C1(C(N(C2CC(NC(c3ccc(C)s3)=O)C2)C)=O)C2CC2C2CC12 37469,c1(OCCCOC)ccc(C(N2CC(C)(NC(c3cnc(S)[nH]3)=O)C2)=O)cc1 37470,c1(C(=O)NC(CC(C)NC(c2n(C=C)ncc2)=O)C)cc(Cl)c(N)c(Cl)c1 37471,C(=O)(CCCN=[N+]=[N-])NCC(C)NC(=O)CSCc1ccncc1 37472,Cc1cc(F)c(C(=O)NC2(C3CCCN3C(=O)C(=O)C(C)(C)C)CC2)cc1F 37473,n1(CCC)c(SCCOc2ccccc2F)nc2ccc(Br)cc2c1=O 37474,N1(C(C)(C)C)CCN(Cc2ccc(NC(c3ncon3)=O)o2)CC1 37475,O=C1OCc2cc(C(=O)NC3CCCC(CN=c4[nH]ccnc4Br)C3)ccc21 37476,N1(C(c2c(C)cn(C)c2)=O)CCN(C(=O)CCc2cccc(F)c2Br)C2CC12 37477,n1(C(c2cn(C3C(OC)CCC3)nn2)NC(=O)C(C)O)c(C(=O)O)nc2ccccc12 37478,c1(CC)ccc(NC(c2ccc(NCc3ncc(C)s3)cn2)=O)c(C)c1 37479,N1(C(C(C(CC)C)O)=O)CCC2(CC1)CN(C(=O)CN(C1CC1)CC)CC2CO 37480,c1(C(=O)NC2CC3(CN(C(C(CN(C)C)O)=O)C3)C2)cccc2ccccc12 37481,CS(=O)(=O)c1nccc(N2CCC2(C)C(=O)Nc2cc3ccccc3nc2Br)n1 37482,C1(C(=O)OC)CCC(C(=O)NC(C)(C)C(C)NC(=O)CCCN(C)C(C)=O)CC1 37483,Cc1ccc([N+](=O)[O-])c(CN=C(NCC(CO)C(C)C)NC(C)COC(C)C)c1 37484,c1(CC)c(C(N2CCC(C)C2C(=O)NCc2cnn(C(C)C)c2)=O)ccn1C 37485,c1(N2CCC(F)(C(=O)Nc3cc(OC)cc(Br)c3)C2)ncc2ccccc2n1 37486,N(C1CCCn2ccnc21)C(C1CCC(C)N1C(=O)Cn1cccc1)=O 37487,c1(C(=O)NC2C(CNC(C(CC)(C)CO)=O)CCC2)noc(C)c1[N+](=O)[O-] 37488,C1(NC(=O)OC(C)(C)C)CCC(n2cc(CN(C(c3cccnn3)=O)C)nn2)C1 37489,C(=O)(CCCC(=O)Nc1cnc(C(F)(F)F)cc1C(N1C(C(=O)OC)CC1)=O)OC 37490,CCC(O)CC(=O)N1CC(CNC(=O)C(C)Cc2cccc(F)c2)C(C)C1 37491,O=C1NC2(CO1)CC(C(N1CCC(NC(C3CCc4nccn4C3)=O)C1)=O)C2 37492,C1(NC(C(CCC)NC(=O)C(O)CC2CCCC2)=O)CC2(C1)CC(C)(C)C2 37493,S(=O)(=O)(c1ccc(N2CCC2=Cc2ccccc2)c(F)c1)N1CCSC(C)C1C 37494,C12(C(N(CCCN(C(=O)Cc3cnoc3)C)C)=O)CCCN(CCC1)C2 37495,C1(C(=O)NCc2nc(C(=O)NC3COC(C(F)F)C3)co2)(OC)CCC(C)C1 37496,c1(C(N2CC(F)CC(NC(=O)CC3(O)CCC3)C2)=O)c(Cl)ccc2ccccc12 37497,C(=O)(N=c1cc(Cl)cn[nH]1)c1c(F)ccc(CNC2CC3(CC(C(=O)O)C3)C2)c1 37498,Nc1cc(F)cnc1C(=O)NCCC1(NC(C2CCCNC2=O)=O)CCC1 37499,C(=O)(CC(CC#N)C1CCC1)c1cn(C(C)C)nn1.C1(=O)CN1C1CC1 37500,c1(OC)cc2c(cc1C(N1CCC(NC(=O)CCc3cccn3C)C1)=O)OCO2 37501,C1(n2cc(CNC(CC)=O)nn2)CCC(C(=O)NCCC(C)(C)OC)CC1 37502,CCC(C)(C)CCCC(=O)NC1CCC2CCN(C(=O)CCC(C)(C)F)C12 37503,C1(CC(=O)N(C2CCN(C(C3C(C)C3)=O)CC2)CCOC)COC2(CCC2)CO1 37504,c1(NC(c2cncc(NC(c3cnc(C)[nH]3)=O)c2)=O)cnn2ccncc12 37505,c1(C(=O)NCC2(NC(c3cnn(C4CC4)c3)=O)CC2)cnc(S)n1C1CC1 37506,c1(CC(=O)N(CCNC(=O)C(C(C)C)N(C)C)CC)cc(Cl)cc(Cl)c1 37507,C(C(C(C)C)NC(C12CC(CO1)C2)=O)NC(C=CC=CCC)=O 37508,c1(OC)cc(C)c(OCCNC(=O)Cn2cc(Cl)c(C)n2)c(C)c1 37509,c1(CNC(C=CC(CC)C)=O)nc(C(=O)N(CCCN=[N+]=[N-])CC)c(C)o1 37510,c1(CC)ccc2cc(NC(N3CCC(F)CC3)=O)ccc2c1 37511,CC(C)N=C(NC1CC(c2ccc(F)cc2)(C(C)C)C1)N1CCC(C(N)=O)CC1 37512,c1(Cc2nn(CCCCC)c(C3CC(C)=NO3)n2)ccc(O)cc1 37513,C(=O)(CCC(C)(C)OC)NCCC1CCN(C(C2C(CC)CCO2)=O)C1 37514,c1(C(N2CCN(C(CSCCN(C)C)=O)C3C2C3)=O)ccc2occc2c1 37515,N1(C(C2N(C(=O)C(Cl)Cl)CCC(=C)C2)=O)CCC2(CC1)CC(=O)N2.C1C(=O)N1 37516,Cc1cscc1C(N1CCC(C(C)NC(C2(C)CC2C)=O)C1)=O 37517,N1(C(Cc2c(C)occ2)=O)CCC2C(CCCN2C(=O)CN2CCC(C)(C)C2)C1 37518,c1(C(N(CCNC(c2ccc(C(=O)OC)s2)=O)C)=O)csc2nnsc12 37519,c1(OC)nc(N2CCCC(C)(NC(=O)CCCCCCBr)C2)nc2[nH]cnc12 37520,C1(C(N2CC(OCC(F)F)C2)=O)COCCN(C(c2cccc(O)n2)=O)C1 37521,C1(CNC(=O)CC)C2CN(C(C3C4CCCC34)=O)CC12.c1ncoc1-c1ccco1 37522,c1(CNC(C2CC(C)(C(C)(C)C)C2)=O)ccc(Br)cc1N1CCNCC1 37523,C1(NC(C=CCC)=O)CC12CCC(NC(c1ccc(C(F)F)o1)=O)CC2 37524,C1(NC(CN(CCC)C)=O)CCCC(NC(=O)C(C(C)CC)OCC)CC1 37525,C(C(C)(F)CNC(c1cccn1Cc1cccs1)=O)NC(CSC)=O 37526,C1(NCc2c(COC)ocn2)CS(=O)(=O)CC1NC(=O)Nc1cccc(Br)c1 37527,c1(C(N2CC(CNC(c3ccn(C4CC4)n3)=O)C2)=O)conc1C1CC1 37528,c1(C(=O)NCC(C2CC2)NC(C2CC(C)(F)C2)=O)cc(F)cc2cc[nH]c12 37529,O=C(C#CC1CCCC1)NC1CCCCC1NC(=O)CC12CCCN1CCC2 37530,N1(C(C(C)(C)C)=O)CCC2(CC1)CC(NC(=O)C(F)(F)C(O)C1CC1)C2 37531,C(C(O)C(C)(C)CO)CN(c1cccs1)C(N(CC(=O)OC(C)(C)C)C)=O 37532,n1(CCN(C(CN(C(C)=O)C(C)C)=O)C)cc(C2(NC(C)=O)CC2)nn1 37533,O=C(C1=CS(=O)CCC1)N1CC2=C(C1)CN(C(c1cn(C3CCCC3)nn1)=O)C2 37534,C(C#Cc1cn(-c2cccnc2)nn1)NC(c1c[nH]nc1C1CCC12CCC2)=O 37535,N1(C(C(CC)N2CCCC2)=O)CCN(C(=O)C(C)n2cccn2)CCC1C 37536,C(=O)(C(C)C(C)(C)C)NCCC1(OC)CN(C(c2n(CC)c(O)nc2)=O)C1 37537,N1(C(CC(CC)C)=O)CC2CCC1C1CN(C(c3c(N)cc(Cl)nc3Cl)=O)CC21 37538,C1(C)(NC(C(C(C)C)NC(c2sccc2C#N)=O)=O)CCC(=O)NC1=O 37539,C1(C(=O)NCC(C2CC2)SC)C2CC2CN1C(=O)Cc1cnccn1 37540,C1(NC(c2c(C)c(Br)ccc2F)=O)CCN(C(=O)C2=CCCS2)CC12CCC2 37541,c1(CCNC(N(CCO)Cc2cccc(OC)c2)=O)cc2[nH]ccc2s1 37542,C(C(=O)NC1CCN(CCC(F)(F)F)CC1)(C(C(C)C)OC)OC 37543,C1(C(N2C(C(C)(C)CNC(=O)Cn3cccn3)CCC2)=O)COC2COCC12 37544,C(=O)(CC(C)CC(C)(C)C)N1C(COC)CN(C(=O)C2=CCCCO2)CC1 37545,c1(C(=O)OC)cccc(CC#N)c1-c1nc(-c2cnc(C)[nH]2)no1 37546,Cc1cccc2c1OC(C(=O)NCC(F)CNC(=O)CSCCC(F)(F)F)C2 37547,Cn1c(C(=O)NC2CCC(C(=O)Nc3ccc(Br)nc3)OC2)cccc1=O 37548,c1(C(=O)NC2(C)C(NC(C(CC)C(F)(F)F)=O)CCC2)cccc2nn(C)nc12 37549,C(=O)(CCCC(C)(C)C)NCC(C(=O)NC(c1nc(CC)on1)C)(C)CC 37550,C1(C(=O)NCC(CN(C(=O)C(C)CC(F)F)CC)(C)C)CCOC(=O)CC1 37551,N1(C(C(CCC)N(C)C)=O)CCC(C)(c2cn(C3CCN(CC)CC3)nn2)CC1 37552,C1(C(=O)OC)CCC(O)CN1C(c1ccncc1C)C(=O)NCCC1CC1 37553,c1(C(=O)NCCCCCN(C(C(=Cc2ccco2)C)=O)C)nnc(S)n1C 37554,CC1(C)CC(C(=O)N2C(CNC(C3CCC(C(N4CCOCC4)=O)O3)=O)CC2)=NO1 37555,C1(COC)CC(CNC(=O)C(C2CCOCC2)O)N(C(=O)CCC2OCCO2)C1 37556,c1(C(=O)NC(C2CN(C(C=C(COC)C)=O)C2)C)cc(C(=O)O)ncn1 37557,CS(=O)(=O)c1ccc(F)c(C(=O)NCC2(NC(=O)CC3CC=CC3)CCOC2)c1 37558,CC(C)(CC1CCOCC1)C(=O)N1CCCC1c1cn(CCNC=O)nn1 37559,C1(S(N)(=O)=O)(C(N2CC(CC)C(NC(c3[nH]c(O)nc3C)=O)CC2)=O)CCCC1 37560,C=CCC(CC(C)C)C(=O)N1CC2C(NC(=O)C3=CCC(C)(C)CC3)C2C1 37561,c1(NC(C(=O)NCC2CCCSC2)=O)ccc(N2CCOCC2)cc1 37562,c1(C(=O)NCC2(Nc3ccc(CC)cn3)CCC2)c(Cl)cccc1[N+](=O)[O-] 37563,C(=O)(C1CSc2ccccc21)NC(C)CNC(=O)CC(C)(C)C(F)(F)F 37564,C(C)(N=c1[nH]c(=N)c2[nH]cc(Br)c2[nH]1)c1ccc(CC(=O)OC)cc1 37565,N1(Cc2c(C)nn(CCOC)c2C)CCOCC(C(=O)NC(C)CC2CCCC2)C1 37566,c1(C(=O)Nc2nscc2C(=O)NC2(C=CC)CC2)ccc2nc(O)n(C)c2c1 37567,CN1CC(C(=O)NCC2(F)C3CCCC23)c2ccccc2C1=O 37568,C(=O)(C(C)(C)c1ccns1)N(CCCCNC(C1C(C)C1)=O)C 37569,CN=c1nc(C(N2CCCC(CNC(=O)CSc3ccccn3)C2)=O)cc(C)[nH]1 37570,C1(CNC(C2(CC)CCCO2)=O)CCN(C(c2ccc(C)nc2N)=O)CC1(F)F 37571,Cc1oc(-c2ccccc2)cc1C(=O)NC1CCC1NC(=O)CC1(C(F)F)CC1 37572,C(C(CC(F)(F)F)NC(C1CCCN1N=O)=O)NC(=O)Cn1cnnc1O 37573,C1(NC(C(C)(CO)OC)=O)C2CC3C1C3C2C(=O)NC1CCN(C2CCC2)C1 37574,CC1CC(NC(=O)C=Cc2ccc(C(F)F)o2)CN1C(c1ccc(C#N)o1)=O 37575,c1(C(=O)NCCN(C)C(c2csc(C(C)(C)C)n2)=O)ccc(S(C)(=O)=O)o1 37576,C(=O)(CCC(CF)CF)N(CC1N(C(C2(SCC)CC2)=O)C2CCC1C2)C1CC1 37577,S(=O)(=O)(c1ccc(C)c(Cl)c1)N1CCN(Cc2ccc(C)cc2O)CC1 37578,c1(C(=O)NCC2C3CN(C(C(C(=O)NC)(C)C)=O)C2C3)ccc2nnc(S)n2c1 37579,C1(CNC(C(C)NC(C)=O)=O)CCN(C(C2CC2C(N)=O)=O)CC1C 37580,C1(NC(c2c(OC)c[nH]n2)=O)CCCC12CCN(C(c1cc(Cl)cnc1O)=O)C2 37581,Cc1nc(O)[nH]c1C(=O)NC1CC2(C1)CC2NC(=O)Cc1cc[nH]c(=N)c1 37582,N1(C(CC2C(C)=NOC2=O)=O)CC(NC(c2ccc([N+](=O)[O-])[nH]2)=O)C(C2CC2)C1 37583,C1(N(CCC)C(c2ncsc2CC)=O)CCN(C(C)C(=O)Nc2cccs2)C1 37584,N1(C(C=CCC)=O)CCC(CNC(C2C3C4CCC(C4)C23)=O)(OC)CC1 37585,c1(C2C(C(=O)NCC3CC(NC(CCSC)=O)C3)CC2)ccc(F)cc1 37586,C1(O)(CN2CC3(C(NC(=O)Cc4cscn4)CCS3)C2)CCC(F)(F)CC1 37587,c1(C(N(CC(C)NC(c2cccnn2)=O)C)=O)c[nH]c2cc(Br)ccc12 37588,c1(OCC)nc(C(=O)NCC(C2CC2)NC(C2CCCO2)=O)co1 37589,c1(C(N(CCCNC(C2CC2F)=O)CC)=O)cc2n(n1)CCN(C)C2 37590,c1(C(=O)NC2CC(C)(C)N(C(c3cccnc3)=O)C2)ccsc1S(C)(=O)=O 37591,c1(C(C(=O)Nc2ccccc2)N(C(C)C#N)C)cccc(Cl)c1Br 37592,N1(C(c2ccc(=N)[nH]c2)=O)C2CCC1(CNC(C1CCN(C3CC3)CC1)=O)CC2 37593,c1(CN2CC(NC(C3(F)CCCC=C3F)=O)C(F)C2)ccc2cc[nH]c2c1 37594,CCCC(C)CCCC(=O)NCCCOCCCNC(c1cn(CCO)nn1)=O 37595,Cc1ccc(C(N2CCC(C)C(NC(=O)CN(C)C(N)=O)C2)=O)cc1Br 37596,c1(NC(CC2CCN(C(CC3CCN(C)C3)=O)C2)=O)cc2c(F)cccc2[nH]1 37597,C1(C(N(C)CC2N(C(CN3CC(C)C3)=O)CCC2)=O)CCCN(C2CCC2)C1 37598,c1(C(N(CC(CC)NC(=O)CCCNC(C)=O)C)=O)nccn2cnnc12 37599,N1(C(c2cc(C)on2)=O)CCCCC1CNC(c1cnc(C(C)(C)CF)o1)=O 37600,C1(C(=O)NCCC2N(C(CCC(C)SC)=O)CCCC2)CCC(C)(O)CC1 37601,C1(C(N(CCOCCN(C(C(C#C)(C)C)=O)C)C)=O)COC2(CCC2)CO1 37602,C1(C(N2CCCCC2CO)=O)COC2(CCN(C(c3cncc(Cl)c3)=O)CC2)C1 37603,Cn1nc(-c2ccccc2)cc1C(=O)NC1CC(C)(NC(C2CC23CC3)=O)C1 37604,c1(CCC(=O)NC23CC(NC(C4(C(=O)OCC)CCCC4)=O)(C2)C3)cccc(C)c1 37605,CCC(C)(C)CC(C(=O)NCC1(C)CCS(=O)(=O)N1C)N1CCN(C(=O)CO)CC1 37606,c1(C(C(=O)NC(CC)C)N(C)C(C2(C)CC2)C)csnc1OC 37607,CC(C)CC(C(=O)N1CC2CC(NC(=O)CCC(C)(C)O)CC1C2)C(N)=O 37608,c1(SC)ncc(C(=O)NCC2(F)CN(C(C3CC(c4ncc[nH]4)C3)=O)C2)s1 37609,C(=O)(C1=C2CCCN=C2NN1)N1CC2C(NC(C3CC4CCC4C3)=O)CC(C2)C1 37610,C1(S(N)(=O)=O)(C(=O)NC(C)CCNC(c2cn(CCN(C)C)cn2)=O)CCC1 37611,C1(C(=O)NC2C=CCN(C(Cc3scc(C)n3)=O)C2)C(O)C(=O)N(C)C1C 37612,N1(C(CN(C)CC2CC(F)(F)C2)=O)CCC(N(C2CCCC2)C)CC1 37613,CCCCCC(C)CC(=O)NCC(C)(CC)C(=O)NCCC(O)CCC 37614,Cc1ccccc1C(C)C(=O)NC1CCC(NC(=O)CCC2CCCCN2C)C1 37615,C1(C(C)C)CCCN(C(=O)NCCCNCc2nccn2Cc2ccccc2)C1 37616,N12CCCC(O)(C1)OCCCC2=O.c1(CC(=O)NCCOC)nc(C)sc1C 37617,c1(C(CC(=O)NC2C(CNC(CC(=O)OCC)=O)C2)OC)ccc(Cl)cc1 37618,C1(C(C(=O)NCC(C2CC2)OC)C)CCN(C(c2csc(C#N)c2)=O)CC1 37619,C(=O)(CC(CNC(=O)C(C)OC)C1CCC1)NC(COCC)C.C(C)(C)S 37620,C=CCC(C)(C)CC(=O)N1CCC(NC(C2(c3oncc3C)CC2)=O)C(C)C1 37621,N1(C(C(C)N(CC)CC)=O)CCC2(CCC(N(C)C(C3CCCOC3)=O)CC2)C1 37622,C1(O)(CNC(c2c(COC)ncs2)=O)CCN(C(c2nnn3c2CCC3)=O)CC1 37623,C1(CNC(CC=CCCCCC)=O)C(C)CCN1C(c1cc(C)c(CC)o1)=O 37624,C(=O)(CCCC(=O)NCC(C)CNC(c1cc(C)nn1C)=O)NC 37625,Cc1cc(C(=O)NC2CN(C(=O)Cn3nc(Cl)ccc3=O)CC2O)ccc1Cl 37626,c1(C(=O)NC2CCC2CNC(C2CC2CF)=O)cc2cc[nH]c(=O)c2s1 37627,CC(C)(CCCNC(=O)Cc1nc[nH]n1)NC(=O)CC1CC(CF)C1 37628,c1(CC(=O)NCC2CC2NC(=O)CSC2CC2)c(F)cc(F)cc1F 37629,Cn1cncc(C(N2CC(N3CCN(C(=O)CN4CCCC4=O)CC3)C2)=O)c1=O 37630,CC1(C(N2CCSCC2)=O)CCCN(C(=O)CCc2cccs2)C1 37631,c1(C(N2CCC(NC(c3cccn(C4CC4)c3=O)=O)C2)=O)ccn2ncccc12 37632,c1(C(=O)NC(CCN(C(COCC(=O)NC)=O)C)C)cnc(Cl)s1 37633,C(C(=O)NCCC1(NC(C2CCCC(C)O2)=O)CC1)(C(C)C)OC 37634,C1(NC(c2cccc(Cl)c2)=O)CCC2CN(Cc3ncc(C(C)(C)C)o3)CC2C1 37635,C12(NC(c3cnn(C(C)C)c3Cl)=O)CCCC1N(C(=O)CSCC(N)=O)CC2 37636,C(=O)(CC(C)C(F)F)NC(CN(C(=O)C(C1CC1)SC)CC)C 37637,c1(-c2nc(-c3cc(Cl)ncc3)nn2CC2CCCOC2)cc(F)cc(F)c1 37638,O=C1C(Nc2nnc(C3CNC3)s2)CCN1c1ccccc1F 37639,N1(CC(=O)NC(CC)C)CCN(CCCCCc2ccc(Cl)cc2)CC1 37640,C1(C(N2C(C)(C(=O)OC(C)(C)C)CC2)=O)CC(F)(F)CCC1(C)C 37641,c1(CC(=O)NC2CCCN(c3ccnc(Br)n3)C2)cnn2c1CCCC2 37642,C(=O)(CC(C)(C)c1cccc(Br)c1)NC1C(CN(C(C2(C)CC2)=O)C2CC2)C1 37643,c1(OC)ccc(C(=O)NCC2CCN(C(=O)C(O)C3CCCC3)CC2C)c(Cl)c1 37644,C12(C(N3CCN(C(c4ccccn4)=O)CC3)=O)C3C4C1C1C2C3C41CO 37645,c1(C(=O)NC2(CCNC(C(c3ccc(Cl)s3)C)=O)CCC2)n[nH]c2c1COC2 37646,C1(CC=C)(NC(C2CCCC2O)=O)CN(C(C2CCCN2C)=O)C1 37647,CC(C)C(CCN(C(=O)C(C)C(F)F)C)NC(=O)C(c1ccc(Cl)cc1)=O 37648,c1(C(C(=O)NCCOC)N(C2CCC(F)(F)C2)C)ccc(F)c(Br)n1 37649,Cc1ccc(C(N2CCC2CNC(C2CCCC2C)=O)=O)c(N)c1C 37650,c1(C(=O)OC)ccnn1C(C)(C)NC(C1CC1C1CCCC1)=O 37651,N1(C(=O)CCC2CCCO2)CC2CCC(C1)N2C(=O)CC1CC2CC2C1 37652,N1(C(c2ccsc2)=O)CC2(C1)CN(Cc1ccnc(F)c1)CCO2 37653,C1(C(N2C(CN(C(CC(C=C)(C)O)=O)C)CC(F)C2)=O)C2CCC1(C)C2(C)C 37654,CC1C2C(CCN2C(C23CSCC2C3)=O)CN1C(=O)C=Cc1cc[nH]n1 37655,C1(CNC(c2nccc(C)c2)=O)CN(C)CCN1C(c1ccnnc1S)=O 37656,c1(C(=O)NCC(CCCC)NC(=O)CCC(F)F)cc([N+](=O)[O-])ccc1O 37657,C1(NC(c2c(O)cccc2O)=O)CCCC12CCN(C(C1CS(=O)(=O)C1)=O)CC2 37658,N1(C(c2nc(C)sc2)=O)CCN(C(=O)C(c2cc(F)cc(F)c2)C)C(C(C)C)C1 37659,c1(CC(=O)NCC(CNC(c2c(C)ncc(C)c2)=O)O)cc(Cl)cc2c1OCC2 37660,CS(=O)(=O)c1ccc(C(N2CCC(NC(=O)CO)C(CO)C2)=O)cc1Br 37661,c1(C(N2CC(CCn3cc(C4CCCO4)nn3)C2)=O)cnc(S)[nH]1 37662,C1(C(N2CC(CC(=O)NCc3nccc(OC)c3)OCC2)=O)CC(=O)OC1(C)C 37663,c1(C(=O)NC2CC3(C(NC(C(CC#C)C4CC4)=O)C3)C2)ccc(Cl)cc1F 37664,C(=O)(C(CNC(=O)CN1CC(C)(C)C1)C(C)(C)C)NCCc1c(C)ncs1 37665,CCCCCCn1nnnc1C(c1cnn[nH]1)NCc1ccc(CO)o1 37666,CC1CN(C(C2NC(=O)NC2=O)=O)CC(C)CN1c1nnc(-c2ccccc2)s1 37667,Cc1c(C(=O)NC(C)C(C)NC(c2c(Cl)ccc(Cl)c2O)=O)sc2ccccc12 37668,C(CC(=O)NCC1CN(C(=O)Cc2cccc(C(N)=O)c2)C1)(C(C)C)OCC 37669,Cc1cc(C(=O)NC23CC(NC(=O)C(C)OCCC(C)C)(C2)C3)cc(C)c1N 37670,N1(C(C(CC=C)N(C)C)=O)CCc2nc(CNC(c3ccc(O)nc3)=O)sc2C1 37671,c1(CC(=O)NCC2CN(C(C3(CC4CC4)CC3)=O)CC2O)cccnc1Br 37672,C(=O)(C(F)(CC)C(=O)OC)NCC(C)NC(c1c(CC)occ1C(F)(F)F)=O 37673,c1(C(N2CCC(C)(NC(C=C(COC)C)=O)CC2)=O)cc2c(s1)CN(C)CC2 37674,N1(C(Cc2ncc(C)[nH]2)=O)CC(CNC(=O)C(C)SC(C)C)CC1(C)C 37675,C1(NC(CCSC)=O)CN(C(=O)C(F)CC(C)C)CC2CC12 37676,N1(C(C2CC(C#C)(O)C2)=O)CCN(C(=O)Cn2ccc(C(F)F)n2)CC1C 37677,Cc1nc2cc(C(=O)NCCC(C)N(C)C(c3ccc(Cl)o3)=O)cnc2s1 37678,N1(C(CCC#C)=O)CCC(F)(F)C(C(=O)NC(C)(C)C#CCCC)C1 37679,c1(OC(C)C)ccc(Cl)cc1C(=O)N(CCC(C)NC(=O)CC1CC(=O)C1)C 37680,C1(NC(C2(COC)CC2)=O)CN(C(c2cc(C(N)=O)cc(F)c2)=O)CCC1(C)C 37681,N1(C(C2CC(C)NCC2)=O)CCCCC2(CCOCC2)C1 37682,C1(N(C(C2N(CC)CC2)=O)C)CCC(NC(C2(CN(C)C)CCCCC2)=O)CC1 37683,c1(CNC(C2CC(CC)C2)=O)cc(F)c(F)c(F)c1.C12CCC(CO1)NC2=O 37684,c1(C(N(C)NC(C2CN(CC3(CSC)CC3)C2)=O)=O)c(C)nc(C)n1O 37685,CC(CCC(=O)N1CC(F)(CNC(c2cnc(-c3ccco3)s2)=O)C1)NC(N)=O 37686,C1(CNC(Cc2cc(C(C)C)no2)=O)(CNC(=O)CC2CC23CC3)CC12CCC2 37687,c1(C(=O)NC2CC(NC(C(CC)n3ccnc3)=O)C2)n[nH]c(C)c1Cl 37688,Cc1cnn(C)c1CC(=O)NCCC(C)CCNC(c1ccnn1C1CC1(F)F)=O 37689,C1(C(N(CCC)CC2CC2)=O)CN(C(=O)CC(C)C(C)C)CCC1(C)C 37690,C1(C(=O)NC23CC(NC(c4cnc(CCC)s4)=O)(C2)C3)CCCCC1C1CC1 37691,N1(C(C2CCC(=O)NC2=O)=O)C2CCC1CN(C(C13CC(CN1C1CC1)C3)=O)C2 37692,c1(C(N2CCCN(C(C(=O)NCC)=O)CC2CO)=O)[nH]c2ccc(F)cc2c1C 37693,N1(C(c2c(SC(C)C)cccc2)=O)CCCC(NC(C23CCC2C3)=O)CC1 37694,N1(C(C2CCC(Oc3ccccc3)C2)=O)CCN(Cc2ccc(Cl)cc2)CC1 37695,c1(CCC(=O)NC(C(C)NC(CCN(C)CC)=O)CO)ccccc1[N+](=O)[O-] 37696,c1(C(=O)NC2C(NC(C=C(C)C3CC3)=O)CC2)cnc(OCC(F)F)cn1 37697,C1(NC(C(C)C(C)(F)F)=O)CN(C(=O)Cn2ccc(=N)[nH]2)CC2(CCC2)C1 37698,c1(NC2CCN(CC(C)(O)NC(=O)OC(C)(C)C)C2=O)cc(Cl)c(Cl)c(Cl)c1 37699,C(=O)(C(C)(C)C1CCCN1C(=O)CC1(C)CCC1)NCCN(CCCF)C 37700,C1(C)(C(=O)NC2CCN(C(Cc3c(C(C)C)con3)=O)C2)CC(C(F)(F)F)=NO1 37701,c1(OC)cc(C(N2CCC(CNC(C3(O)CC3(C)C)=O)C2)=O)cc([N+](=O)[O-])c1Cl 37702,C1(NC(COC)=O)CCN(C)C12CCCN(C(=O)Cn1cc(Cl)cn1)C2 37703,c1(CC)ccc(C=CC(=O)NCCC(C)N(C(=O)Cn2cncn2)C2CC2)o1 37704,N1(C(C2N(C(C)=O)CCC2)=O)CCCC(NC(=O)CCN2CCC2)C1.C(C)(C)(C1CC1)N 37705,C1(NC(COC(C(C)(C)C)(C)C)=O)CN(C(C2CCOC(=O)CC2)=O)C(C)(C)C1 37706,c1(C(=O)NC2CCN(C(CC3OCC(C)OC3)=O)CC2F)cccc2ccnn12 37707,c1(C(=O)NC2CN(C(CCCCC)=O)CC2C)ccc2c(c1)C(C)CO2 37708,C1(C(=O)NCC2(C(N3CCCC(F)C3)=O)CCCCC2)CC(F)C(=O)N1 37709,C1(C(=O)NC(c2cnn[nH]2)C)CCCN1NC(=O)c1c(Cl)cnn1C 37710,CCCC(C)(O)C(=O)NCCCC(C)NC(=O)Cc1cnc(C)o1 37711,C1(C(N(CCCN(C(=O)CCCc2ccc(F)cc2)C)C)=O)C2CCC(=O)C12 37712,C(CS(=O)(=O)C1CCOC1)C(C#N)C(=O)N.c1ccccc1F 37713,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NCC1(NC(Cc2ccc(CC)cc2)=O)CC1 37714,N1(C(c2c(CC)nns2)=O)CCN(C(=O)CC(C)CN(C)C)CC1CC(=O)NC 37715,c1(C(=O)NC2C3CN(C(c4ccnc(O)c4Br)=O)CC23)ccn2ncnc2c1 37716,C1(C(=O)NCC2(O)CN(C(c3ccc(CC)o3)=O)C2)CC(=O)N(CC(F)(F)F)C1 37717,N1(CCn2c(CC)nc(-c3n[nH]c(C)n3)n2)CC2(CCC2)OCC1CC(=O)OC 37718,C(C)(c1cccs1)=CC(=O)NCC(CC)NC(=O)C(c1cccnc1)C 37719,C(=O)(CC(F)(F)F)NCCN(C1CCC(N(C)C)C1)C(=O)COCC1CCOC1 37720,c1(CC(=O)NCCCN(C(=O)Cc2cnsc2)C)cccc2c1OC(F)(F)O2 37721,C1(NC(C(C(C)C)n2cnnc2)=O)CCN(C(=O)Cc2ccccn2)C12CCC2 37722,C1(C2CCC2)(C(=O)NCCC(CCNC(c2cccc(C)c2C)=O)C)CC1(F)F 37723,CC1CC(C(F)(F)F)CCN1C(C1(CNC(=O)Cn2ncnn2)CCC1)=O 37724,CCC(CC(=O)N1CCCC(CNC(C2(c3ccno3)CCC2)=O)C1)C(C)C 37725,N1(C(CC2CC(C)(C)CN2C(C2CC(O)C(F)C2)=O)=O)CCOCC(C)(O)C1 37726,N1(C(c2occ(C)c2C)=O)CCOC(C)(CNC(=O)CSCCC(C)C)C1 37727,C=CCCCCCCCCNC1(c2nnnn2C2CCC2)CCCC1CCF 37728,c1(CNC(C(=O)NC(C=C)CCc2ccccc2)=O)cn2cc(F)ccc2n1 37729,C(=O)(C(O)C(F)F)NC1CC(NC(CN(CCOC)C)=O)C1 37730,c1(C(=O)NCCC2CC(NC(c3cc(Cl)no3)=O)C2)sc(F)cc1Cl 37731,C1(CC(C)C)(C(=O)NCC(CO)NC(CCCSC)=O)CCCC1 37732,c1(C(=O)NCC2C(NC(C3CCCC3COCC)=O)CCC2)cccc(C#N)c1C 37733,C1(C(=O)NCC2CC2(Cl)Cl)(COC)CN(C(=O)CC2(O)CCC2)C1 37734,c1(CC(N2CC(NC(c3ccc(OC)s3)=O)C(F)CC2)=O)ccc2c(c1)CCC2 37735,c1(CN2CCN(C(c3ccc(CO)o3)=O)CC2)c(-c2ccccc2)cccc1O 37736,C12CN(C)CCCN1C2=O.c12cc([nH]n1)CNC2=O.c1(CC)cc(C2CC2)[nH]n1 37737,c1(NC(C2CCCC(C(N3CC(SCC)C3)=O)C2)=O)ncnc(C)c1C 37738,CC(C)(C)CC(O)C(=O)N1CCCC1CN(C(=O)CCC1CC2CCC1C2)C1CC1 37739,C(=O)(C1COc2ccccc21)NC(C)CC1CCN(C(=O)C(C)(C)N(C)C)CC1 37740,c1(C(=O)OC)nnn(CC(=O)NC(=O)C(C)NCC2CC2CSC2CCCCO2)c1C 37741,c1(C(N2CC(NC(C(CC)OC)=O)C2)=O)ccc(OC(C)(C)C)cn1 37742,Cc1ccc(C(N2CC=CC(NC(C3(C)CCCS3)=O)C2)=O)c(N)c1F 37743,CC1(CNC(=O)CCN2CCCCC2=O)CCCN(C(=O)Cn2cncn2)C1 37744,C(C)(CN=c1[nH]nc(SC)o1)Oc1c(COC)c(OC)ncn1 37745,n1(CCC)nc(C)c(Cl)c1C(c1nnnn1CCC)NCNC(C)CCC.OC 37746,C(C)(CC(C)C(F)F)NC(CCN(CC#C)C(c1cnc(CC)o1)=O)=O 37747,c1(CC(=O)N(C2CCCCN(C(=O)C(O)C3CC3)C2)C)ccc2occc2c1 37748,c1(Cn2c(C(N(C(CNC(CC(=O)OCC)=O)C)C)=O)ccc2)ccccc1Cl 37749,Cc1nc2sccn2c1C(N1CCC(NC(=O)CC2CC2(Cl)Cl)C12CC2)=O 37750,C1(CCNC(C=CC(=O)OCC)=O)CSCCN1C(=O)CS(=O)(=O)NC 37751,c1(C(=O)NCC(CC)(C)NC(=O)Cc2cccc(F)c2)ncc[nH]c1=O 37752,c1(C(=O)OCc2n(C)cnc2)ccc2c(c1)CCC(=O)N2CC1CCC1 37753,Cc1cc(C(N2CC(n3cc(C4(N(C)C)CC4)nn3)C2)=O)c2c(Br)cccc2n1 37754,C1(C(=O)NC2CC(OCCO)C2)CCC(CN(C(CN(CC)CC)=O)C)CC1 37755,C1(C(=O)NCCOCCCNC(C2CC(F)(CF)C2)=O)CC(=O)N(CCO)C1 37756,c1(NC(C2C(C(=O)Nc3cnc[nH]3)C2)=O)ccc(I)cc1[N+](=O)[O-] 37757,c1(OC)ccc(CN2CCSC(C(=O)NCc3ccc(C4CC4)cc3)C2)c(Cl)c1 37758,Cc1cc(CNC(C2C=CCCN2C(c2cc(C(C)C)on2)=O)=O)n(C)n1 37759,Cc1cc(C(N2CCOCC2C(N2CCOCC(O)C2)=O)=O)cnc1C 37760,c1(C(=O)NC2C(OCC)C2)c(C)nn(C2CC2)c1C.c12nc(C)c(s1)C(=O)NC2 37761,c1(C(=O)NCC(CNC(C=C(CSC)C)=O)(C)C)cn(C2CC2)c(C)cc1=O 37762,CC(C)(C)C(C(=O)NC12CCN(C(=O)CCOCC3CC3)CC1C2)N1CCCC1 37763,CC(C)(C)CC(=O)N1CCC1(C)C(=O)NCC=CCOc1ccc(Cl)cc1 37764,C(C)(C(=O)N1CC(NC(c2ccc(CN(C)C)nc2)=O)C2(CC2)C1)(C(C)C)OC 37765,C(=O)(CCC(=O)N1CC2C(NC(=O)C(C)(C)C3CC3)C2C1)N(CCC)CCC 37766,N1(C(C(C2CC2)OC)=O)CCC(C(=O)NCC(C)CCO)C1 37767,N1(C(CC(COC)C)=O)CC(C)(CNC(=O)CSS(C)(=O)=O)CC1(C)C 37768,CC(C)CCC(O)C(=O)NC(C)(CO)C(=O)N1CCC(n2ccnc2)C1 37769,S(=O)(=O)(c1ccc(NC(C2CCC2)C2CC2)c(Cl)c1)NCC(C)C1CCC1 37770,c1(C(=O)NCC2C(NC(C3(F)C(C)OCC3)=O)CCC2)ccc(=O)n(CCF)n1 37771,Cc1ccc(C(=O)N(CCCCCNC(=O)CC2(CO)CCCCC2)C)cc1C 37772,c1(C(=O)NC2(C)CN(C(=O)CCCn3c(O)nnc3O)C2)ccc2ccccc2n1 37773,CC(C)C(C)(C)C(=O)NC1CC(NC(c2c[nH]nc2[N+](=O)[O-])=O)CC1O 37774,c1(N(CC=C)CC2(CO)CC2)nnc(-c2cc(Br)c[nH]2)n1CC1CCOC1 37775,C(=O)(C(CC(C)C)OOC(C)=O)N1C(CN(C(=O)CCCC2CCC2)CC)CC1 37776,c1(C(=O)NCC(CCCC)NC(C2(CC#C)CC=CCC2)=O)cc(F)ccc1N 37777,c1(C(=O)Nc2cccc(C(N3CCC(N(C)C)CC3)=O)c2)cc(Cl)cc(Cl)n1 37778,Cc1cnc(N2CCN(C(=O)C(C)(C)C)CC2C(=O)Nc2cccc(C)n2)nc1C 37779,C(=O)(CC(CNC(=O)Nc1ccc(C(F)(F)F)o1)C(C)C)OCC 37780,c1(C(C)(C)C)nc(N2CCCC(CNC(C3CCCCC34CC4)=O)C2)cc(Cl)n1 37781,C(=O)(CN=c1cc[nH]cc1)N1CC(CC(N2Cc3c[nH]nc3C2)=O)OCC1 37782,N1(c2ncc(C(=O)OC)nc2)CCC2(CCCN(C(=O)CC3(O)CCOC3)C2)C1 37783,CCCCC(CNC(=O)COCCCOC)NC(=O)CC1CCS(=O)(=O)C1 37784,CCC(CN(C)C)CC(=O)N1CC2(C1)CN(C(=O)Cc1nc[nH]n1)C2 37785,c1(C(N2CCC(O)(CN(C)C(c3cncs3)=O)C2)=O)[nH]c2ccccc2c1Cl 37786,C=CC1(C(=O)NCC(O)C(C)(F)F)CCN(C(=O)C(F)C(CC)CC)CC1 37787,C12(C(N(C(c3ccccc3)CNC(c3nn[nH]c3Cl)=O)C)=O)CC1CCC2(F)F 37788,C1(CCC)CN(C(=O)Cc2ccnn2C)CC1C(=O)NCC(N1CCCC1)=O 37789,N(C(=NCC1CCC(=O)NC1)NC1CCCCC1C)CC12CC(CC)(OC1)C2 37790,c1(C(N(C)CC)=O)cccc(C(=O)NCC2CN(C(=O)C(C)CSC)CCO2)c1 37791,CCCCCC(C)NC(C1CCC(NC(=O)CCCC2CC2C)CC1)=O 37792,C(=O)(CC(F)(F)CS(C)(=O)=O)N1CCC(C(C)NC(c2n(CC)cnn2)=O)C1 37793,c1(CN2CC(NC(c3ccc(SC)cc3)=O)C(F)C2)cccc2nccnc12 37794,C(=O)(C1CC(=O)c2ccccc21)N1CCC(C)(NC(C=C(COC)C)=O)C1 37795,c1(C(=O)NC2C3CC(C3)C2Cc2ccccc2)cc2nccn2c(O)n1 37796,N1(C(CC2(C=C)CC2)=O)CCN(C(=O)C(F)(F)C(C)O)CC1C 37797,c1(C(C(=O)NCC2C(NC(c3c(C)n(C)nc3)=O)C2)(C)C)ccc(F)cc1F 37798,C1(C(=O)NCCCCNC(Cc2ccc(C)o2)=O)CCn2nncc2C1 37799,c1(C(=O)NC(C2(NC(C3(S(N)(=O)=O)CC3)=O)CC2)C)cc(C)n(CC(F)(F)F)n1 37800,CN1CCc2c(C(N3CCCC3C(=O)NC3CC3(F)F)=O)cccc21 37801,c1(C(=O)NC23COC(CNC(C4(CF)CC4(F)F)=O)(C2)C3)cn2c(n1)CCCC2 37802,N1(C(CCOC)=O)CCC(CO)C1.C1(C(=O)NCCOC)CCCSC1 37803,c1(CC)ccc(C(=O)NC(C)CNC(=O)CCC2CCOCC2)cc1S(C)(=O)=O 37804,c1(C(=O)NC(C2CCN(C(CSCC)=O)C2)C)cccc(Br)c1 37805,C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CC(F)(CNC(c2ccc(C=C)cc2)=O)C1 37806,c1(NC2CCCC(OCC)C2)cc(=NC2CCN(CP(C)(C)=O)C2)[nH]c(C(C)C)n1 37807,C(=O)(C(=NOC)c1ccco1)NC1CCCCN(C(C2C(C(=O)OC)C2)=O)C1 37808,N1(C(C=NOC)=O)CC2CC(NC(c3cc(O)ccc3Br)=O)C(C2)C1 37809,N1(C(C2(CC(C)C)CC2)=O)CCC(c2ccc(F)cc2)C(NC(=O)C(C)(F)F)C1 37810,c1(CC(=O)NCC(C2CC2)NC(C2(O)CCOC2)=O)c(F)cccc1F 37811,c1(C(=O)NC2CCCC(NC(C3CCOCC3O)=O)C2)ccc2c(c1)CCCS2 37812,c1(CC(N2CCCCC(NC(C3CCCS3)=O)C2)=O)cnc2cccnn12 37813,c1(CC)nc(C(=O)NC(C2(CNC(c3ncsc3C)=O)CC2)C)n[nH]1 37814,C1(CN(C)C(=O)NC2CON(C)C2=O)(NCC2CC2)CCCCC1 37815,c1(C(N2CC(NC(CCCC(C)=O)=O)CC2(C)C)=O)cc2ccc(F)cc2[nH]1 37816,N1(C(C2C(SC)=NC=CC2)=O)C(CNC(=O)CN2CC(=O)NC2=O)CC2CCCC12 37817,N1(C(c2cccc(C)n2)=O)CC(N=[N+]=[N-])CC1C(=O)N(CC(C)C(F)(F)F)C 37818,c1(C(=O)NCC2CCC(OC)(OC)CC2)nccc2ccc(Br)cc12 37819,Cc1cc(Cl)c(C(=O)NNC(=O)C2CCC3CC3C2)c(Cl)c1 37820,C(=O)(C(C)(C)CO)NC(C(C1(O)CN(CCc2n(C)ccn2)C1)F)=O 37821,CC(C(=O)NC1CCC(c2ccc(Cl)cc2)C1)C(=O)c1ccc(Cl)cc1 37822,C12(NC(C3(CF)CCC3)=O)CC1CN(C(CC1(CN(C)C)CCCC1)=O)C2 37823,N1(C(CC2CC(OC)C2)=O)CCCC(F)(CNC(=O)C(C)(C)c2ccccc2)C1 37824,c1(CCN=C(NCCC2(C)CC2)NCC2CC2)cnc2c(Cl)cnn2c1 37825,N1(C(CCCOC)=O)CCC(C)(C)C(C(=O)NC(C)(C)COC(C)C)C1 37826,Cc1cc(C(F)F)n(CC(N2CCCCC2CNC(=O)C(C)c2ncco2)=O)n1 37827,N1(C(CC2(C=C)CC2)=O)CCC2CCCC12CNC(c1ccnc(CC)c1)=O 37828,c1(C(N2CCC(O)(CNC(c3cc(CC)c(C)s3)=O)C2)=O)ccc(N)c(Cl)c1O 37829,C(CC(C(=O)NCC1(COC)CCC1)NC(=O)Cc1ccc(C)s1)OC 37830,c1(CNC(c2cnn(C)n2)=O)ncccc1C(N1CCC(C(N)=O)C1)=O 37831,CCCCCCCC(=O)N1CC(CC(=O)NCCCCN(C)C)C2(CC2)C1 37832,C1(CC)CCC(C(=O)NC(C)(C)CNC(c2ccc(C3CC3)o2)=O)CC1 37833,c1(CNCC2(C)CC2)c[nH]c2cc(C#N)ccc12.N12CCC(C(O)C1)C2=O 37834,C1(NC(CC(C=C)C)=O)CN(C(c2nccc(C)n2)=O)C2(CCCC2)C1 37835,C1(C)(CC)CC(C(=O)NC(Cc2cc[nH]n2)CO)CCO1 37836,C1(OC)CN(C(=O)Cn2nccn2)C(C)(CNC(c2ncc[nH]c2=O)=O)C1 37837,CC(C)(C)C(C(=O)NC1CN(C(C2(C#N)CCOC2)=O)C1)c1ccccc1 37838,C12(C3C(n4cc(C(=O)NCCCNC(=O)CCC5CC5(F)F)nn4)C3)CC(CO1)C2 37839,c1(C(=O)NCC2N(C(c3cccn(C)c3=O)=O)CCC2)cnn(C)c1S(C)(=O)=O 37840,N1(C(C(CC#C)O)=O)CC2CCC(C1)C(NC(C1CC3C=CC1C31CC1)=O)C2 37841,c1(C(=O)NCC(CC)NC(C2(CSC)CC(F)(F)C2)=O)cccnc1C(F)F 37842,c1(C(=O)NCCN2CCC(OC)CC2)nc2cc(Br)ccc2n1C 37843,C(C1CC1)(C1CC1)=CC(=O)NCCCN(C(c1cc(SC)oc1C)=O)CC 37844,C1(CNC(CSS(C)(=O)=O)=O)CCCCC1NC(c1ccnn1C(F)F)=O 37845,c1(SC)c(C)nn(C)c1NC(=O)NC1CC2CC(C(N)=O)CC12 37846,C=CC1CN(C(C2C(Oc3ccccc3)C2)=O)CC1NC(C1(C(=O)N(C)C)CC1)=O 37847,N1(C(c2cc(C)no2)=O)CCC(NC(c2cnc(C(N)=O)s2)=O)C(F)C1 37848,C(=O)(CCCCC(F)(F)F)NCC1C(NC(C=C2CCC(C)C2)=O)C1 37849,c1(C(=O)NCC(C)NC(C(CCCC=C)(C)C)=O)ccc2c(c1)NC(=O)CCC2 37850,N1(C(c2c(SC)cccn2)=O)CCC2CN(C(C3Cc4nccn4C3)=O)C2C1 37851,N1(C(C(C2(O)CCC2)NC(CCCCCC)=O)=O)CC(F)(F)CCC1C 37852,N1(C(CSCC(=C)C)=O)CCC(NC(c2cccc(OCCC)c2)=O)C2CC12 37853,c1(C(=O)NC2(C)CC(NC(c3cccnc3O)=O)C2)cc2c(s1)CCOC2 37854,N(C(=NCCN1CCOCC1)NCc1ccco1)CCC(C=C)(C)C 37855,C12(C(=O)NCCC3CCN(C(C4CC5(CSC5)C4)=O)C3)CCC(CC1=O)C2 37856,N1(C(CCCC2C(C)C2)=O)CCCN(C(c2cc(O)nn2C)=O)CC1C 37857,c1(NC2CCN(CC)CC2C)ccc2c(c1)CCN(C(=O)OC(C)(C)C)C2 37858,C12(C(N(CC(CC)NC(=O)CCc3cc(C)[nH]n3)C)=O)CCCN(CCC1)C2 37859,Cn1cc(C(=O)NCc2cn(C3CN(C(C4CC4(C)C(F)F)=O)C3)nn2)ncc1=O 37860,c1(CNC(=O)NC2CCC(C)(CC)C2)c(F)cc(Cl)cc1Cl 37861,c1(N2CCOCC(NC(C3(C)ON=C(C)C3)=O)C2)ncc(Br)cc1C#N 37862,C(=O)(C(F)CCC(C)(C)C)N1CCC(NC(c2c(COC)noc2)=O)C(O)C1 37863,Cc1cc(Cl)cc(C(=O)NC(CNC(=O)CCS(C)=O)CO)c1N 37864,c1(N(CCOC)CCNC(c2cn(-c3nc(C)cs3)nn2)=O)ncccc1Cl 37865,C1(CN(C)CC2CCC(c3ccccc3)O2)CCCCC1N1CCCC1=O 37866,CCC(C)C(C)CN=c1[nH]c(=NCCCc2nc(C)cs2)c2cc(Cl)ccc2[nH]1 37867,c1(C(=O)NC(C2(O)CCCCC2)C(=O)N(c2cn[nH]c2)CCO)cc([N+](=O)[O-])n[nH]1 37868,C1(OC)(CNC(c2c[nH]nc2-c2ccc(Br)cc2)c2nnnn2C)CCC(C)C1 37869,C1(C(N2C3C(CNC(c4csc(C(F)F)n4)=O)C(C3)C2)=O)CCC2(CCOC2)O1 37870,N1(C(=O)CC2CC3CC3C2)CCN(C(c2cnc(C3CCC3)o2)=O)C(CCO)C1 37871,c1(C(=O)NCC2(NC(C3COCC(C)O3)=O)CCCCC2)cc(C#N)ccc1O 37872,CCCCCC(O)CC(=O)N(CC)CC1CCCN(C(c2cc(=O)cc[nH]2)=O)C1 37873,CC(C)(C)C(C(F)F)NC(C1CCN(C(=O)CCN2CCCCC2)C12CC2)=O 37874,C1(NC(C(CC=CC)CC)=O)Cc2ccccc2C1NC(=O)CCc1cn[nH]c1 37875,CCCN=C(NCC(O)CN1CCN(C)CC1)NCCc1conc1SCC 37876,n1(CC(=O)NCc2scc(C(N3C(C(N(C)C)=O)C=CC3)=O)c2)ccccc1=O 37877,C(=O)(C1=CCCC1(C)C)NCCCCCN(C(C1(C=C)CCC1)=O)C 37878,N1(C(C(F)=CC)=O)CCC2CCN(C(=O)CC3CCCCN3C)C2C1 37879,N1(C(CC2(C)CC2(F)Cl)=O)CC2CCC(C1)N2C(c1cnn(C2CCC2)c1)=O 37880,N1(C(CSC(C)(C)C)=O)CCC2(C1)CN(C(=O)CC(F)(F)Br)CCO2 37881,Cc1nc(-c2scnc2C)n(CCNC(c2ccc(C(F)(F)F)cc2)=O)n1 37882,CC1COC(C)(C)CN1C(=O)NCCOc1cccnc1Br 37883,C1(C(C)C)CN(C(=O)C(C)(F)F)CCC1NC(=O)CN1CCCCCC1=O 37884,c1(NC(=O)Nc2cnc(C(F)F)s2)cccc(SCCC(F)F)c1 37885,c1(NCCCNC(C2CCCN(C)C2)=O)nc(-c2ccccn2)nc2sccc12 37886,C(=O)(C(O)C(C)(C)C)NC1CC(C)(NC(c2nc(CN3CCOCC3)cs2)=O)C1 37887,C#CCCC(O)C(=O)N1CCCN(C(=O)C(C(C)(C)C)NC(C)=O)CC1 37888,Cc1ccnc(F)c1NC(c1nc(C(=O)Nc2ccc(O)cc2Br)cs1)=O 37889,C12(C(CNC(c3cn(C(C)(C)C)nn3)=O)NC(C=CC(C)C)=O)CCC(CC1)C2 37890,O=C(C(CO)NC(=O)CC1(O)CCC1)NC1CCCCC1 37891,N1(CCc2c(C)cccc2)C2CCCC1CN(C(C1CCC(C)O1)=O)C2 37892,N#Cc1c(C(N2CC(CNC(=O)CCC3CCC(C(N)=O)O3)C2)=O)cccc1F 37893,N1(C(C2(OC)CC(C)C2)=O)CCC(C2(O)CN(C(c3nnn(C)c3N)=O)C2)CC1 37894,CCCCC(C)CCC(=O)N(CC(C)O)CCNC(c1cccc(C)c1N)=O 37895,c1(C(N2CCC(NC(C3(CC#C)CC3)=O)C(O)C2)=O)ccc2nc(C)[nH]c2c1 37896,Cc1c(C(N2CCCN(C(c3ccc[nH]3)=O)CC2)=O)sc2[nH]cnc(=S)c12 37897,C1(NC(C2C(OCC)C2C)=O)CCS(=O)(=O)C12CN(C(=O)Cn1cc(CO)nn1)C2 37898,C(C)(C(C(=O)NC1CC(O)C1SC)NC(C1OCCC1(C)C)=O)OC 37899,C1(C(N2C(C)C(NC(c3cscc3Br)=O)CC2)=O)CCn2nncc2C1 37900,N1(C(C2CC(C(C)C)C2)=O)CCCC2(NC(C3CCCOC3)=O)CCCC12 37901,Cc1nn(C)nc1C(=O)NCC1(CNC(c2cc(Cl)cs2)=O)CCCC1 37902,O=S(=O)(c1cnc(Cl)c(CC2CC2(Cl)Cl)c1)N1CCN(CC(F)F)CC1 37903,c1(OC)cccc(-c2cc(C(=O)OCCCn3cc(Cl)cn3)no2)c1 37904,Cc1[nH]c(CN2CC3CC2C3C(=O)Nc2ccc(Br)c(Cl)c2C)c(C)c1[N+](=O)[O-] 37905,CCC(C)CC(C)C(=O)NCC1CC2CCC1N(C(c1cnnc(Cl)c1)=O)C2 37906,C1(CNC(c2c[nH]c(=N)o2)=O)CCN(C(=O)C(F)C2CCC2)CC1(F)F 37907,N1(C(Cc2c(C)occ2)=O)CCC(CNC(=O)CC(C)(C)C)C1C 37908,N1(C(c2cc(OCCC#C)ncc2)=O)CCC(C)N(C(=O)C(O)C=CC)CC1 37909,C1(C(N2CCC3CN(C(C4=C(C)OCC4)=O)C3C2)=O)CC2CCC1CC2(F)F 37910,C(CC(C)C)(CC(C)C)(C1CCCCC1)NCc1nnnn1C.CCCCOCC=O 37911,C1(C(=O)NC(CC)C2CCC2)(NC(=O)Cc2cccs2)CSC1 37912,c1(CC)c(C(N2CCCC2C2CCCOC2)=O)cnn1C(C)(C)C 37913,c1(OC)cnc(C(=O)NC2(C)CC(NC(c3n[nH]cc3OC)=O)C2)c(F)c1 37914,C1(NC(c2ccc(N3CCC3)nc2)C)CCN(Cc2cnn(C)c2)C(C)C1 37915,C#Cc1ccc(C(=O)NC2C3CC2N(C(C2CCC(=O)N(C)C2)=O)C3)nc1 37916,C(=O)(CCCCc1cn(C2CCC(C(=O)OC(C)COC)C2)nn1)OCC 37917,C1(C(N2CC(NC(C=C(C)C3CC3)=O)C(CO)CC2)=O)CCc2nc[nH]c2C1 37918,c1(C(N2CCC(C(C)NC(=O)Cc3nc(C(F)(F)F)n[nH]3)C2)=O)cncc(Cl)c1 37919,c1(CC(N2C(C)(C(=O)NCC(C)OCC#C)CC2)=O)ccc(C)c(C)c1 37920,C(=O)(CCN(OC)C(=O)CCCCCNC(=O)CC1CCCC2CC12)OC 37921,c1(C(=O)NC2(C)CC(C(N(CC(C)SC)C)=O)C2)cccc(F)c1F 37922,c1(C(=O)NC2(CCNC(C(C)c3ccco3)=O)CCC2)cnc2sccc2c1 37923,C1(CNC(C2(COC)CCCO2)=O)CC(C)CN(C(=O)C(C)(C)SC)C1 37924,c1(C(=O)OC(C)(C)C)cc(C(=O)NCCCOCCOC2CCCCC2)no1 37925,C(CCC(C)(C)OC)NC(c1c(CC)csc1)=O.C1=CCNC1=O 37926,C(C)(CO)(C(=O)NCCC1CCC(=O)N1)NC(CC(C)F)=O 37927,C1(NC(c2n[nH]c(O)n2)=O)CC2CN(C(c3ccnnc3Cl)=O)CC12 37928,C(=O)(C(C)(C1CCC1)NC(=O)COCC1CCCO1)N(CCCO)C 37929,C(N=c1cc2c(c[nH]1)CCCC2)C1(NC(c2c(CCOC)ocn2)=O)COC1 37930,c1(C(=O)NC(C(C)(C)NC(C(CCSC)O)=O)C)ccc(C2=NOC(=O)C2)cc1 37931,CCCCC(N=c1ccn2ncc(S(=O)(=O)N(C)CCNC(C)=O)c2[nH]1)C(C)C 37932,c1(C(N2CC3CN(Cc4c(OC)nccc4)C3C2)=O)cc(C)c(Cl)cc1Cl 37933,C(=O)(C1CCCc2n[nH]cc21)NCC1(NC(=O)C(Cl)=CCl)CC(OC)C1 37934,c1(C(N(CCNC(Cc2c(C)scc2)=O)C2CC2)=O)cc2cccc(F)c2nc1O 37935,c1(CC(N2CC(NC(C3CC4(C3)CC4F)=O)C(O)C2)=O)cccc2c1SCCC2 37936,C1(NC(c2c(C)cncn2)=O)CC(F)CN(C(=O)C(c2cccc(F)c2)C)C1 37937,C=CCCCC(C)(C)C(=O)NC1CC(OCC(=O)NCC(C)(C)C(F)(F)F)C1 37938,Cn1ncc2c1CC(C(=O)NCC(O)CNC(=O)COCC(F)F)CC2 37939,N1(C(c2c(C)cc(SC)s2)=O)C(CNC(C2CC2(C)C)=O)CC2CCCC12 37940,c1(-n2c(C3CN4CCCC4CO3)nc(CCCOC)n2)nc2ccc(Cl)cc2[nH]1 37941,N1(C(C2N(C(C(C)C)=O)CCC2)=O)CCN(C(C2CCC2)=O)C2(CCC2)C1 37942,c1(CC(=O)NC(C)CNC(=O)CCc2ccccc2O)ccc(Cl)nc1F 37943,Cc1cnnc(C(=O)NC(CCCNC(c2ccc(F)cn2)=O)c2ccccc2)c1 37944,Cn1nc2c(c1NCC(F)(F)Oc1cc(C#N)ccc1C(=O)O)CCC2 37945,C1(CO)(CO)CC2(CC(F)C2)C1.N(C(=NCCC)NCC(C)(C)CC(F)F)SC 37946,CCCCC(F)C(=O)N1CCC1C(N1CCC(OC)C(F)C1)=O 37947,Cc1ccnc2c(C(=O)NCC(C)NC(C34CC(C)(C3)C4)=O)cnn12 37948,c1(OC)ccc2cc(C(=O)NC3CCCN(C(=O)CO)C3)sc2c1F 37949,Cn1cc2c(n1)CC(C(=O)NCCCNC(c1csc(-c3ncc[nH]3)n1)=O)CC2 37950,c1(N2CCC(n3ncc(C)c3)CC2)ncnc(N2CCC=CO2)c1C 37951,c1(C(=O)NCCN(CCCCCC)C(c2cccc(C)n2)=O)c(C)ncnc1C 37952,C(=O)(C1=NN2CCC(C)N=C2N1)NCCOCCOCCOCCC=C 37953,C1(C(=O)OC)CC2(CCN1C(=O)COc1ccccc1[N+](=O)[O-])CC2 37954,C1(C(N2CCC3(CC2)OCCO3)C(=O)NCCCSC)CC2OC(C)(C)OC2C1 37955,C(CC(=O)OCCOC)(C(C)C)Sc1n(CCCC)nc(-c2ccc(F)cc2)n1 37956,C1(NC(CNC2CC(C#N)C2)=O)CCn2nccc2C1 37957,N1(C(c2occ(C(=O)OC)c2)=O)CC2CC(N(C)C(C3(OC)CC3)=O)C1C2 37958,C1(C(=O)NCC(CNC(CCC(C)c2ccccc2)=O)(C)C)CCCCC1(F)F 37959,C1(NC(C2C(OC)CN(C(CN(CCC)C)=O)C2)=O)CCN(C)CC1(C)C 37960,Cc1nn(C)cc1CCNC(C1CN(C(=O)CC2(O)CCCC2)CC1C)=O 37961,N1(C(C(=Cc2ccco2)C)=O)CC2(CC2)CC1CC(N1CC(C)(O)C1)=O.c1(O)ccsc1 37962,C1(CCC)(NC(c2csnc2Cl)=O)CCN(C(c2cccc(O)n2)=O)CC1 37963,c1(-c2sc(C(N3CC(NC(C=C(C)C4CC4)=O)C3)=O)c(C)n2)c(C)nn(C)c1C 37964,c1(C(C)OC)ccc(-c2nc(-c3cnn(C)c3)nn2-c2c(C)noc2C)cc1 37965,C1(C(N(CCCNC(C(C(=O)OC)(C)F)=O)C)=O)CCc2nn[nH]c2C1 37966,c1(C(=O)NCC(CNC(CCN(C(CCC)C)C)=O)F)cc(O)cc(Cl)c1 37967,C1(C(=O)NC(c2cn(CC(F)(F)F)nn2)(C)C)COCC(=O)N1C(F)F 37968,C1(OC)(OCC(=O)NO)CN(CCC2CCC2)C1 37969,Cc1ccc(C(C)NC(C2CC=CCN2C(c2cnn(C)c2Cl)=O)=O)cc1 37970,c1(C(N2C(Cn3cc(CCCSCC)nn3)C=CC2)=O)ccc2nc(O)sc2c1 37971,C1(C)(C(=O)NCC=CCNC(Cc2c(C)noc2Cl)=O)CCCCC1C 37972,C(C(C)(C)F)(C1CCCCC1)N(CCNC(c1nnnn1C1(C)CC1)=O)CC 37973,c1(C(=O)NC2CCCC(N(C(CCC(=O)NC)=O)C)C2)oc2ccccc2c1C 37974,c1(C(=O)NC2C3CN(C(c4ccc(O)c(O)c4)=O)CC23)c(Br)cc(F)c(F)c1F 37975,CC(N=c1[nH]c2c(c(=NCCSC3CCOCC3)[nH]1)CCCCC2)c1ccco1 37976,CC1=NS(=O)(=O)NC=C1C(=O)NC1(CNC(C2(S(C)(=O)=O)CC2)=O)CC1 37977,C1(NC(c2c(C)noc2)=O)CC2CCC(C1C)N2c1ncccn1 37978,Cc1ccc2c(c1)CC(C(=O)NC1COCCN(C(=O)C(C)(C)O)C1)S2 37979,C(=O)(CCCCC1CC1)N(C(C)C)CCN(C(=O)C(O)c1ccco1)C(C)C 37980,c1(C(=O)NCC2C3CN(C(C(C)n4cccc4)=O)C2C3)cc([N+](=O)[O-])ccc1Cl 37981,Cc1cn2c(C(=O)NCC3CCCCN3C(=O)CCC(C)C)cnc2s1 37982,c1(C(=O)NCC2N(C(c3c(C)cncn3)=O)CC(F)C2)ccnc2ccccc12 37983,Cc1ccc(Br)c(C(=O)NC2CCC2CNC(C2(F)CC2)=O)c1 37984,N(C1CCc2sc(Br)cc21)C(=O)N(Cc1cccc(COCC)c1)CC 37985,C1(CCC)CCCCC1C(=O)NCC1(NC(c2cncc(CO)c2)=O)CCC1 37986,C1(CCC(=O)NC(C)CCC(C)(C)C)CCCN(C(c2nocc2C2CC2)=O)C1 37987,C1(C(=O)NC(C)(C)CC(=O)NCC2C3CCC(F)C23)CC2(CCC2O)C1 37988,C1(O)(CNC(CC(=O)N(C)C)=O)CCN(C(c2n[nH]cc2C(F)(F)F)=O)C1 37989,C1(NC(C2C(C(=O)OC)CC=CC2)=O)CN(c2nccc(C)n2)CC(F)(F)C1 37990,C1(CNC(CNC(CC)=O)=O)CN(C(=O)CCNC(=O)OC)CC(C)(C)C1 37991,S(=O)(=O)(c1cnn2ccc(=NC(C)c3nc(Cl)sc3Cl)[nH]c12)NCCC(CCC)O 37992,CCC(C(=O)N1CCSCC1CCNC(c1cncc(Cl)n1)=O)NC(C)=O 37993,N1(C(C(c2ccc(Cl)cc2)C)=O)CC(C)(C)CC1CNC(C1CC1F)=O 37994,N1(c2nnc(C(CC)CC)n2CCC(=O)OC(C)(C)C)CC2(CCSCC2)C1 37995,C1(C(N(C(C)CNC(C23CC(C#N)(C2)C3)=O)C)=O)CC(=O)C12CCC2 37996,N1(C(CCC#C)=O)C(C(=O)Nc2ncncc2I)CC2CCCCC12 37997,CC(C)(C)CCC(F)C(=O)N1CCCC(C2CCCCN2C(C2CSC2)=O)C1 37998,C1(CC)CCCC1CCOC(C)C.C12(C(=O)O)CN(C1)Cc1c[nH]nc1NC2=O 37999,C12(NC(C3N(C)CCOC3)=O)CCCC1CN(C(c1cc[nH]n1)=O)C2 38000,C1(CC(=O)O)CCCN(Cc2cn(CC3(n4ccnc4)CC3)nn2)C1 38001,C1(C(N2CC3CC(C2)O3)=O)CC2CC2N1C(C1CCNC(=O)C1)=O 38002,C1(CN(C(c2c(CC)cc[nH]2)=O)C)CCC(NC(C2CC=CCC2C)=O)CC1 38003,N1(CCC)CCCC(C(N2CCC(N(C(=O)C(F)OC)C)CC2)=O)C1 38004,C12=CN=C3C=CC=CN1N3C(=O)C(O)(CNC(C(COC)C)=O)CC(C)NC2=O 38005,c1(C(=O)NC2CC(CNC(CCc3cnn(C)n3)=O)C2)cccc(=O)o1 38006,c1(CNC(c2nn(CC)c(O)c2)=O)nnn(C)c1C(=O)NC1(c2cccs2)CC1 38007,C1(C(N2C(C)(C(NOC(C=C)C)=O)C=CC2)=O)CC2CC(=O)C1C2 38008,C(=O)(C(CO)NC(=O)COC(F)F)NC1C(C(C)(F)F)C1 38009,c1(CCC)cc(C(=O)NCC23CC(NC(c4cnc(C)s4)=O)(C2)C3)n[nH]1 38010,c1(C(=O)NCC(C)NC(=O)CC2CC=CCN2C)ccc2c(c1)CCC(C)(C)O2 38011,C1(CC)(NC(c2ccnc(C)n2)=O)CCN(C(=O)CCN2CCOC2=O)CC1 38012,CCCCC(CC)CC(=O)N(CC(C)(C)C(=O)NCCS(=O)CC)C 38013,C1(NC(=O)CN2C(=O)CCC2=O)CCCCN(C(C2CN3CCN2CC3)=O)C1 38014,Cn1nc(C(F)(F)F)c([N+](=O)[O-])c1NC1CCN(C(c2cc(Cl)no2)=O)C1 38015,c1(C(N(CCCNC(C)=O)CCO)=O)ccc2ccncc2c1 38016,N1(C(c2c(C)ccnc2)=O)CCCC(CO)(NC(=O)CCCC(C)O)C1 38017,c1(CN2CC=CC(C(N3CCC(C)(O)C3)=O)C2)c(F)ccc(Br)c1F 38018,N1(C(C)=O)CCCC(O)(C(=O)NC2CC(NC(=O)CC3CCN(C)CC3)C2)C1 38019,C(=O)(CCCN(C)N=O)NCC1(OC)CN(C(=O)CC2CCOCC2)C1 38020,C1(CC(=O)NCc2cc(C)ns2)CN(C(=O)COCC(F)(F)F)CCC1C 38021,c1(CSC)cccc(C(=O)NCC(C)(C)CNC(c2ocnc2C(F)F)=O)c1 38022,c1(C(=O)NCCC2CCN(C(C(C)C#N)=O)CC2)ccn2cncc2c1 38023,C1(F)(CNC(CN(C)C(N)=O)=O)CCCN(C(=O)C(F)Cc2ccccc2)CC1 38024,CC(C)(CC(F)(F)F)C(=O)NCC1CCC1NC(C1CCC(C(F)(F)F)O1)=O 38025,CC1(C)CCCN(C(c2ccc(N)c(F)c2)=O)C1CNC(=O)Cc1ccc(Cl)s1 38026,C1(NC(c2n(CC)ncc2Br)=O)CCCN(C(=O)CC2(OC)CCC2)CC1 38027,Cn1cc(C#CCNC(=O)C(C2CC2)NC(C2COC(=O)N2)=O)cn1 38028,CC1CCCCC1C(N1CCC(CNc2nccc(C(F)(F)F)n2)C1)=O 38029,c1(CNC(CSCC(C)=O)=O)ccc2c(c1)CN(C(c1cc(CO)ccn1)=O)C2 38030,C1(CC(=O)NC2CC(CSC)C2)CCCN(C(=O)NCCNC(CSCC)=O)CC1 38031,C1(CNCc2[nH]cc(C#C)c2)(NC)COc2ccccc2C1 38032,c1(CC)ccc2c(c1)C(CCNC(c1cc(C)nn1CC1CCC1)=O)C(=O)N2 38033,c1(N(C)C)ncccc1C#N.n12cc(cn1)CNC(=O)COCCOCC2 38034,CC1CN(C(=O)CNc2ccccn2)CCC1CNC(=O)C=Cc1cc[nH]c1 38035,c1(C(N2CCC(C)CC2CNC(=O)C(F)=C2CCC2)=O)cc2cc[nH]c(=O)c2s1 38036,c1(C(N2C(CNC(CN3CCCC(CC)C3)=O)CC2)=O)cc(S(N)(=O)=O)cnc1C 38037,C1(ONC(C2CCC(F)CC2)=O)(CC)CCCN1CCOC 38038,c1(N2CC(CNC(C3(CC#C)CCCC3)=O)OCCC2)ccc2c(n1)CCC2=O 38039,CCC(CC)C(C)C(=O)NCC(CC(=O)N(C)C(c1ccccn1)C)OC 38040,c1(CC)c(C(=O)NC2CCCC(NC(c3cscc3OC)=O)C2)ccn1C 38041,N1(C(CC(C=C)CC)=O)CCOC2(CCN(C(=O)Cc3ccco3)C2)C1 38042,C(=O)(C(F)(CNC(=O)C(C#N)C(C)C)C(C)C)NCC(C)(C)NC(C)=O 38043,C(=O)(C(O)C(O)c1ccccc1)N(CCCCNC(C(=O)N(C)C)=O)C 38044,N1(C(c2c(CC)occ2)=O)CCC(N(S(=O)(=O)Cc2ccc(F)cc2)CC)CC1 38045,C1(C(=O)NCCC2N(C)CCC2)COCCC1NC(=O)CP(C)(C)=O 38046,CCC(O)C(C)C(=O)N1CCN(C(C2CCCC2C(=O)OC)=O)CC1C1CC1 38047,c1(C(N2C(C)(CNC(=O)C=CC(N)=O)CCC2)=O)occ2c1CCOC2 38048,c1(NC(N2CC3C(c4onc(C)n4)(C3)C2)=O)cncc(F)c1I 38049,c1(SC)cccnc1C(=O)N(CCCNC(c1ccc(-c2cccs2)[nH]1)=O)C 38050,C=C(C)C1OCCC1CNC(=O)CC1CN(C(c2cccc(Br)c2F)=O)C1 38051,CCC(C(C)(C)O)NC(=O)C(C1CCN(C(c2ccc(O)cc2)=O)CC1)C 38052,c1(C(N2CC(NC(C3(n4cncn4)CC3)=O)C(O)C2)=O)nsc2ccccc12 38053,c1(SC)cc(C(N2CC3CC2CN3C(c2cn[nH]c2)=O)=O)cc(SC)c1 38054,C1(NC(C(CC)NC(N)=O)=O)CN(C(C2(CN(C)C)CCCC2)=O)CC1OCC 38055,C1(C(=O)NCC2CN(C(c3c(C)nn(CCO)c3C)=O)C2)CC2(C1)CC1(CC1)C2 38056,c1(C(=O)NC2(C(=O)NC)CCC2)coc2c1CN(C(=O)C=CCN1CCC1)C2 38057,c1(CN2CCC(C)(C(=O)NC(CC)CO)C2)cc2ccccc2s1 38058,N1(C(CNC(CNC(C(c2ccccc2)C)=O)=O)=O)CC2CCC(CO)(C2)C1 38059,c1(CNC(CCCOC(C)=O)=O)cncc(C(=O)NC2COC(C(C)C)C2)c1 38060,c1(C(=O)NC(C2CCN(C(=O)C(=C3CCCCC3)F)C2)C)cccc(C2CC2)c1 38061,C(=O)(CCCC1CCCC1)N(C(C)C(=O)NCCCOC1CCOCC1)CC 38062,c1(N2CCC(CCO)CC2)nc(N2CCC(n3cncn3)C2)c2ccsc2n1 38063,C(=O)(CC(C)C(C)C(C)C)NC1CN(C(c2c(C)nc3sccn32)=O)C1 38064,C1(C(N(CC)CC2(O)CCC2)=O)CN(C(C2SCCS2)=O)CCC1(C)C 38065,N1(C(=O)COCCF)CCC2CN(C(=O)CSCc3ccc(Cl)cc3)C2C1 38066,C1(C(=O)NCC2CCC(C3CC3)O2)CCN(C(=O)CCc2cncnc2)CC1 38067,N1(C(C(C)(C)C#N)=O)CCC(F)(F)C(CNC(C2(C)CNC(=O)C2)=O)C1 38068,N1(C(C=CC)=O)CCOC2(CCC(NC(C3CCCC(C(F)(F)F)C3)=O)CC2)C1 38069,c1(C(=O)NCC2N(C(CC(=O)NC)=O)CCN(C)C2)ccccc1N=S(C)(C)=O 38070,C1(C(=O)NCC(C)CNC(=O)CC(C)CC)CCc2nn[nH]c2C1 38071,CC(CC(=O)NCC1CCN1C(=O)CC1CCCC1)c1cnn(C)c1 38072,C(C(=O)NCCCCC(C)NC(C1(c2cccc(C)c2)CCC1)=O)(C(C)C)SC 38073,c1(CC(=O)NCC2N(C)CCN(C(c3cnsc3)=O)C2)ccn2cncc2c1 38074,CC1(C)CN(C(=O)OC(C)(C)C)C1CNC(=O)NC1C(Sc2ccccn2)C1 38075,C12(C(N(C)CCNC(=O)CC3COC(C)(C)C3)=O)CCC(=O)N1CCS2 38076,C1(C(=O)NCC2(COC)CCCN2C(=O)CN=S(C)(C)=O)COC2(CCC2)C1 38077,c1(C(N(CCNC(C(CC)CC(F)F)=O)C2CC2)=O)ccc2c(c1)CCCC2=O 38078,c12c(nnc3c1CCC3)N1CCC(C1)NC2.c1(OCC(=O)OC)ccccc1Cl 38079,N1(C(CC2CC(NC(C#CC)=O)C2)=O)CCC2(CCOC2)C1 38080,CC1(C)COC(C(N2CCC(C(C)(C)C(=O)NC(C3CCOC3)CO)C2)=O)C1 38081,C(=O)(C1CCc2cccc(=O)n21)NC1C(OC)CN(C(CCNC(=O)NC)=O)C1 38082,C(=O)(C(F)CC(C)(C)C)NCc1ccc(C(N(C)CC2(OC)CC2)=O)nc1 38083,c1(C(=O)OC(C)(C)C)cccc(CN(C)C)n1.C12(C)CCN1C2=O 38084,C(=O)(C(C(C)(C)C)OC(C)(C)C)N(C)CC1CCN(C(C2(C(N)=O)CCC2)=O)C1 38085,N1(C(C#CC2(C)CC2)=O)C2CCC1CC(NC(=O)CC1CCCCCC1(F)F)C2 38086,C(C1CCN(C(C2CCC3(CCC3)C2)=O)CC1)=CC(=O)NC(CCC=C)C 38087,N1(C(c2c(NC(N)=O)cccc2)=O)CC2(CCN(C(c3cc(CO)[nH]n3)=O)C2)C1 38088,c1(C(=O)NC(CC(C)NC(c2cc3n(n2)CC(F)C3)=O)C)cccn2nccc12 38089,C1(CNC(CCCc2ncc(C)o2)=O)CC(NC(=O)CNC=O)C12CCC2 38090,Cn1cc(C(=O)NCC(CO)NC(=O)C2=CCSC2)ncc1=O 38091,CCC(C)CCCCC(=O)NCC(C)N(C(c1ccc(OC(C)C)cn1)=O)CC 38092,C1(NC(C(CCC)CC2CCCC2)=O)COC2(C1)CN(C(c1cncs1)=O)C2 38093,Cc1cc(C(=O)NC2CC(NC(=O)C=Cc3ccco3)C2)c2c(c1)CCC2 38094,Cc1cc(F)ccc1C(N1CCC(C)(OCCNC(=O)C(O)C2CCC2)CC1)=O 38095,Cc1ccnc(O)c1C(=O)NC(CNC(c1ccnn1CC(F)F)=O)C1CC1 38096,C(=O)(C(CC)(CC)CC)NC.C1(=O)C(CC2CCCC2)CNC(=O)C(CC)N1 38097,C1(NC(=O)CN2C(=O)CNC2=O)CN(C(=O)CCc2nncs2)CC12CC2 38098,N1(C(C2N(CC)CCC2)=O)CCN(C(=O)C=C2CCOCC2)C2CS(=O)(=O)CC12 38099,c1(NC(C)=O)ccc(Cl)c(C(=O)NC2CC2NC(=O)COCc2ccncc2)c1 38100,C1(C(N(CC(C)NC(c2cccc(OC(F)(F)F)n2)=O)C)=O)CC=CCC1C 38101,c1(N2CCC(N(CC(=O)NC)C)CC2)nc(=NCC2CC2C)[nH]c2c1SCC2 38102,CCC(C(=O)NCC(C)CNC(=O)Cc1cccc(OC)c1F)C(F)(F)F 38103,C1(c2nccn2C)(OC)CCCN(CC2CCC(C#N)CC2)C1 38104,CC1(C)CC(CNC(C2CC3(CCO2)CC3)=O)CN1C(c1ccc(N)c(Cl)n1)=O 38105,CC(CN1CC(c2ccccc2)(NC(C2CCC3CC3CC2)=O)C1)CS(C)(=O)=O 38106,CCC(C(=O)NC(CO)C(=O)NCCCCO)n1ccnc1 38107,Cc1cc(O)c(C(N2CCCC(CNC(=O)C(n3nccc3C)C)C2)=O)cc1F 38108,c1(NC2CCC(NC(c3c(C)cc(F)c(Cl)c3)=O)CC2)ncccc1S(C)(=O)=O 38109,c1(C(=O)NC(CNC(=O)CC2CC(F)C2)C2CC2)c[nH]nc1Cl 38110,C1(NC(Cc2cncc(C)c2)=O)CC(F)CN(C(=O)Cn2cccc(C)c2=O)C1 38111,C#CCC(C)(C(=O)NC(CCO)C1CCCC1)NC(c1ncnc(C)c1C)=O 38112,N1(C(C(CC#CC)C)=O)CC2(CCC2)C1c1ccncc1 38113,C1(NC(C2N(C)C(=O)NC2)=O)CCN(C(C2CN3CCC2CC3)=O)CC1O 38114,c1(C(=O)NCCOC2CN(C(c3nn(CC)c(C)c3)=O)C2)sc(C)c(C)c1C 38115,c1(C(=O)NC2(C)CN(C(C3(C)CCCS3(=O)=O)=O)C2)ccc(F)c(C(F)F)c1 38116,C=CC1OCCCC1C(N1CCC(N(C(=O)CCSCC)C)CC1)=O 38117,N1(C(C2C(C3C(C)C3)C2)=O)CCC(O)(CN(C)C(c2cn3ccsc3n2)=O)CC1 38118,C12(NC(CC3(NC(C)=O)CC3)=O)CCCC1CN(C(=O)Cc1c(C)cccc1Cl)C2 38119,c1(C(=O)NC2(CN(C(=O)C(O)CCS(C)=O)C)CC2)nnc(O)c2ccccc12 38120,c1(C(=O)NC(C(=O)NC(CC)CCCO)c2ccoc2)c[nH]c(C)cc1=O 38121,Cc1cc(F)sc1C(=O)NC1CCCC1CNC(c1cnc(O)o1)=O 38122,N1(C(Cc2nnc(C)o2)=O)CCC2CC1CN(C(=O)CC1CC1)C2 38123,N1(C(C(OC)OC)=O)C2CCC1CC(NC(C1CCNC(=O)C1)=O)C2 38124,CC1CCN(C(=O)C2=CCCC2)CCN1C(c1noc2c1CCCC2)=O 38125,n1(CCC(=O)NC(C)CN(C)C(C2(C)CC2C)=O)c(C)nc2ccccc2c1=O 38126,Cc1ccc(C(=O)NC2CCC(NC(c3cnn4c3CCCC4)=O)C2)c(C)c1Br 38127,c1(CC(=O)NC2CCC(CCNC(CN(C)S(N)(=O)=O)=O)C2)ccc(O)nc1 38128,Cc1oc2ccccc2c1C(N1CCN(C(=O)CCC2CCCOC2)C(C)C1)=O 38129,C1(C(N2CCC(O)(Cn3cc(C4CCCC4O)nn3)C2)=O)CCCC2(CCC2)O1 38130,N1(C(c2ncccc2F)C(=O)NC)CCC2CCCN(C(=O)OC(C)(C)C)C2C1 38131,N1(C(C(C)NC(=O)OC)=O)CCOCC(F)(CNC(C2(C3(O)CCC3)CC2)=O)C1 38132,C(=O)(C(F)C(=O)N(CCCCCNC(C1CCCC(OC)C1)=O)C)OCC 38133,CCCC(C)(CCC)C(=O)NC1CC(NC(=O)CN(CC)CC)CC1O 38134,C1(N=[N+]=[N-])(C(=O)NCC(CCC)(C)C)CCN(C(c2cnc(S)nc2)=O)C1 38135,c1(S)ccc2c(c1)OCO2.C1(NC(=O)OC(C)(C)C)CC(CNC(=O)O)C12CCC2 38136,c1(CC(N2CC(OCCNC(C(CSC)O)=O)C2)=O)ccc(Cl)cc1C 38137,N1(C(Cc2cn(C(C)C)nc2)=O)CC2CCC1C1CN(C(=O)CC3CC3)CC21 38138,c1(C(CC)C(=O)N(CCCN2CCCC2)C)ccc2c(c1)OCO2 38139,Cc1coc(C(C)(C)C)c1C(=O)NC1CCC(NC(=O)CS(N)(=O)=O)C1 38140,C1(C#CC(=O)NCCC(C)NC(=O)CC2CCCN2C)(CC)CC1 38141,CC(C(C)(C)C(=O)NCCn1cccnc1=O)NC(c1cnc2n1CCC2)=O 38142,C1(C(=O)NCC(CC)(F)CC)CCCN1NC(=O)C(C)C1CC1 38143,C1(C#N)(C(N2CC(C(C)NC(C(C)c3cc[nH]n3)=O)C2)=O)CC=CC1 38144,C(C(F)(F)C(F)(F)F)OCC(=O)N(CCCN(C(=O)CC1CSC1)C)C 38145,C=CC(C)(CC)C(=O)NC1(CCCNC2C(c3ccccc3)(C(=O)OC)C2)CC1 38146,n1(CC)ccc2cc(OCCc3ncnc(NC(=O)OC)c3C)ccc12 38147,c1(CNC(CCC#C)=O)cccnc1CNC(=O)CCc1ccnn1C 38148,C#CC(C)(C)C(=O)NC(CNC(c1ccc(C(F)(F)C(F)(F)F)s1)=O)C1CC1 38149,n1(CCOC)nnnc1C(c1cnc(C2CCC2)s1)NCc1noc(C(N)=O)n1 38150,C1(C(=O)NC(C)CC(=O)NCCc2cccc(F)c2)CC(C2CC2)=NO1 38151,c1(C(=O)OCC(C(C)C)O)nc(Br)sc1Br 38152,c1(C(=O)NCC(CC)NC(C2(C3CC3)CCCO2)=O)[nH]c2ccc(C)cc2c1C 38153,C#Cc1ccc(OCC(=O)NCC(CO)NC(c2ccc(Cl)cn2)=O)cc1 38154,C1(CNC(COC(C)C)=O)CCCC12CCN(C(=O)C=CI)CC2 38155,C1(OC)CN(C(=O)CN2CSCCSC2)CC1NC(c1cn(C)cn1)=O 38156,N1(C(c2c(C)csc2)=O)CCCCC1CNC(c1ccc(-c2ccco2)s1)=O 38157,N1(C(CC(C)C)=O)CC(NC(=O)C(CC(C)C)NC(N)=O)C(C)(C)C1 38158,Cc1n[nH]cc1C(C(=O)NC(C)C)N(C)CCC1CCCCC1 38159,C1(CNC(CC=C)=O)(CO)CCCN(C(C2CCCO2)=O)C1 38160,C1(CN(CC(CN(C(n2ccc(CC)n2)=O)C)O)C)C2CCCCCC12 38161,N1(C(c2c(C)nn(C(C)C)c2Cl)=O)CC2CC(C1)CN(C(C1CC(C)(C)O1)=O)C2 38162,C1(NC(c2cnn(COC)c2C)=O)CC2CC(C1)N(C(c1ccnnc1O)=O)C2 38163,N1(C(=O)NC2(C)C(C)OCC2)CCN(S(=O)(=O)N2CCCC2)CC1 38164,C1(C(N(CC(O)CNC(=O)CC2(CO)CC2)C)=O)CCC=CCCC1 38165,C1(CCC)C(O)C(O)CCN1C(=O)NCc1ncc(OC(C)(C)C)cn1 38166,CC1(C)CC(CC(=O)NCC2(F)CCC(NC(c3c[nH]nc3F)=O)C2)CCO1 38167,c1(N(CCC)C(=O)OC2CCCC(C)C2)n[nH]c2ccc(OC)cc12 38168,Cc1ccc(C(N2CC3CC(NC(c4ccc[nH]4)=O)C2C3)=O)c(O)c1Br 38169,c1(C(=O)NCC(CC)Oc2ccc(OC)cc2)nc(C(F)(F)F)oc1C 38170,c1(C(=O)NCC2C3CN(C(c4ccc(NC)cc4)=O)CC32)c(C)oc(C)c1Br 38171,c1(C(=O)NCCCCNC(c2c(SC)cccc2F)=O)ncnc2ccsc12 38172,n1(CC)nnc2cc(C(=O)Nc3ccc(C(C)(C)O)cc3C(C)=O)ccc12 38173,C(CCCCC(=O)N1CC(NC(=O)CSC(C)(C)C)CCC1C)=CC 38174,CCCC(C(=O)N1CCCC(CCNC(=O)C(C)(C)COC(C)C)C1)N(C)C 38175,C1(=O)C(C2(OC)CC2)N1.C(CC#N)N(CCCC)CC 38176,N#Cc1n[nH]c(=NC2CCCC23CN(C(C2CCCC(F)(F)CC2)=O)C3)s1 38177,CC1CC(C(=O)O)CCN1C(=O)NCCCc1ccc(F)cc1 38178,C1(C(N2CCC(OC)C2C(C)C)=O)COC2(C1)CN(C(c1cccc(F)c1)=O)C2 38179,C(=O)(C(C)CCCC(C)C)N(C(CN(C(C(=Cc1cn[nH]c1)C)=O)C)C)C 38180,N1(C(CSC2C(=O)OCC2)=O)CC23CCCC2(C1)CN(C(C12CCCC1C2)=O)C3 38181,C1(CNC(c2cc(C(C)=O)c(C)cc2)=O)CCN(C(=O)C(C)S(N)(=O)=O)C12CCC2 38182,N(C1COc2ccccc21)C(C(C(C)(C)C)NC(C(C)C(F)F)=O)=O 38183,C12(C(=O)NC(C)(C(=O)NC3CC(CCO)C3)C3CC3)CCC(C1)C2(C)C 38184,c1(NC(C2SCCN(Cc3c(C)nc(C)c(C)n3)C2)=O)cn2cc(Br)ncc2n1 38185,CC1CN2CCN1C(C(N1CC3(CC(NC(c4cc[nH]c4)=O)C3)C1)=O)C2 38186,CC1(C)CCN(C(=O)CC2(C#N)CC2)CC1C(=O)NCC1CC(O)C(O)C1 38187,C1(CNC(C2C(C)CCC2)=O)CCCN(C(=O)CC(C)(C)O)CC1 38188,C1(C(=O)NC(C2COC2)C)(CC)CN(C(=O)CSC2CCCC2)C1 38189,N1(CC)C(=O)CCC1CC(=O)NC1CCCC(CNC(=O)Cn2cnc(=N)[nH]2)C1 38190,C1(C(=O)N(C2CC2)CC2N(C(c3nn[nH]c3Cl)=O)CCCC2)(CO)CCOCC1 38191,N1(C(CC)C(F)F)CCS(=O)C(C)(C)CC1 38192,c1(C(=O)NC2C(C)CN(C(c3ccnnc3O)=O)C2)nc(Cl)ccc1F 38193,C(C(C)C(=O)NOCCCCC1CC1)N(C(c1cnn(C(C)C)n1)=O)C 38194,C1(CC)(CNC(=O)C(c2ccccc2)F)CCN(C(C2CC23CC3)=O)CC1 38195,C(=O)(NNC(=O)Cc1ccccc1Br)C1CC(C)N1 38196,C(=O)(C(C)C1=CCCC1)N1C2C(CNC(CS(CCC)(=O)=O)=O)C(C2)C1C(=O)OC 38197,Cc1nc(C(C(=O)NC2(C)CC2)N(C(c2ccc(F)cc2)CF)C)sc1C 38198,c1(C(C(=O)NC2CCC(CNC(c3n(C)cnc3)=O)C2)O)ccc(F)cc1 38199,CC1CN(C)CC(C(N2CCCN(C(=O)CN3C(=O)C(=O)N(C)C3=O)CC2)=O)O1 38200,C1(OC)CC(CNC(=O)CCc2cncs2)N(C(=O)CC(C)(C2CCC2)N(C)C)C1 38201,c1(C(=O)NCCNC(Cc2cnc(C)o2)=O)ccccc1NCc1ccccc1 38202,C1(C(=O)NC)(C(=O)NC2CCOC2)CCCCC1.c12cn(nn1)CCNC2=O 38203,c1(CC(=O)NC(C2CCCCC2)C(=O)NCC(C(C)O)O)ccccc1F 38204,C(=O)(C(C)C(O)CC)NCC1CCC(C(=O)NC2(CC=C)CCCCC2)CC1 38205,c1(C(=O)NC(c2cn(C)nn2)C(=O)NCCCC2(C)CC2)ccc(O)nc1 38206,C(C1=CCN(C(=O)Cc2ccsc2)CC1)NC(c1cn(C2CCC2O)nn1)=O 38207,C1(C(N2CCCN(C(CCSc3n(C)nnn3)=O)CC2)=O)CC2CCCCCC12 38208,C1(NC(c2cc(CCC)ncc2)=O)CCN(C(c2sccc2F)=O)CC1C(N)=O 38209,CC1(C)CC(=O)N(CC(=O)NC2C=CCN(C(c3cccc(F)n3)=O)C2)C1=O 38210,c1(CC)cccc(C(N2CCC(C(=O)N(c3ccc(C)cc3)C)C2C)=O)c1 38211,C=CC1CN(C(=O)Cc2cnns2)CC1NC(=O)CCC1CC1 38212,c1(C(N(C2CCCCC2NC(C2(C)COC2)=O)C)=O)ccc2c(c1)OC(C)(C)C2 38213,N1(C(C=CC)=O)CC2CCC2(CNC(c2cc(-c3ccccc3)[nH]n2)=O)C1 38214,C(=O)(C(O)C(F)(F)F)NC1C(N2CCN(C(Cc3cc(C)sc3)=O)CC2)CCC1 38215,C1(NC(c2c(CC)cco2)=O)CCN(C(C2(C)CCCN2C)=O)CC1O 38216,Cc1c(N2CCN(C(=O)CN(C)C)CC2)cccc1Cl 38217,C1(C)(C(=O)NCc2c(C(=O)NCC(=O)NCC(C)C)cco2)CCOC1C 38218,c1(C(N(CC(C)(C)CNC(C2(CC)CC2(F)F)=O)CC)=O)cc(C)c(C)c(C)c1 38219,C1(NC(C(C)(F)F)=O)CN(C(c2ccc(C(F)(F)F)cn2)=O)C2(CCOCC2)C1 38220,C1(NC(C(CC=C)CNC(=O)C=C(C)C(F)F)=O)CC2CC1CC21CC1 38221,C1(C(N2CC(c3ccc(OC)c(F)c3)OCC2)=O)CCc2n[nH]cc2C1 38222,N1(C(c2ccc(CC)cn2)C(=O)NC(C)C)CCC(C2CCOC2)C1 38223,c1(C(N(CCNC(c2ncc[nH]2)=O)CC)=O)cc2c(ccn2C)[nH]1 38224,C1(C(C)(C)C)CCN(CC(O)COc2ccc(Cl)c(F)c2)C1(C)C 38225,c1(C(=O)NCCNC(c2c(CC)nc(C)nc2)=O)cnc2ncccc2c1 38226,C12CCN(CC1)C(=O)CCCOC2C.c1(CCOC)noc(-c2cccs2)n1 38227,N1(C(c2c(SC)cccn2)=O)CCN(C(=O)CCC2CCCC(O)C2)CC1CF 38228,N1(C(C(CC)=CC)=O)CCC(CNC(=O)CCc2ccc(OC)c(Cl)c2)C(C)C1 38229,c1(CN2CC(C(=O)Nc3cnc(I)cn3)OCC2)ccc(Br)nc1Br 38230,c1(C(N(C2CCN(C(c3n[nH]cc3C)=O)C2)CC)=O)n[nH]c(C)c1O 38231,c1(C(=O)NC(CNC(C(C)S(N)(=O)=O)=O)(C)C)cccc2c1nc(O)n2C 38232,N1(C(c2ncn(CC)c2)=O)C2CCC1CC(CNC(=O)C(=Cc1cscn1)F)C2 38233,CCCCCC(O)CC(=O)NC(CC1CCCC1)C(=O)Nc1cncc(C#N)c1 38234,C1(CNC(C=CCC)=O)CN(C(=O)CC2CC(SC3CC3)C2)C2CCCC2O1 38235,N1(C(c2c(C)nc(N(C)C)s2)=O)CCCC12CCCN(C(=O)C(O)C1CC1)C2 38236,c1(OC)ccc(OC)c(C(N2CCC(C)(CNC(C3(C)CC(F)C3)=O)C2)=O)n1 38237,Cc1ccc(C(N2CCOC(C(=O)NCCCN(C)C3CC3)C2)=O)cc1Br 38238,c1(C(N2CCC(N(C(=O)C(O)CC(N)=O)C)C2)=O)cccc(S(=O)(=O)C2CC2)c1 38239,c1(CC)ncoc1C(=O)NC(C)CN(C)C(c1cnoc1-c1ccoc1)=O 38240,C1(CNC(c2nc(CCC)oc2)=O)C(O)C(O)CN1C(C1CCCCS1(=O)=O)=O 38241,C1(C(=O)NCC2CCC(O)CC2)CCN(C(=O)CNc2nccs2)CC1F 38242,c1(C(=O)NC(C)C(CO)NC(=O)CCCC2CCOCC2)cccc(F)c1F 38243,C1(C(=O)NC(C#C)(C)C)(NC(=O)C(C)=CC(C)(C)C)CCN(C)C1 38244,C(=O)(CC(c1cccs1)C1CC1)NC(CN(C(C(=O)NCC)=O)C)CC 38245,CC1(CNC(c2cc3cn[nH]c3cn2)=O)COCCN(C(C2CCCCS2)=O)C1 38246,Cc1cccc(C)c1CC(=O)NC1CC2(C1)CC(NC(C1(F)C3CCCC13)=O)C2 38247,c1(C(=O)Nc2cc(O)n[nH]2)cnc2n[nH]c(-c3cccnc3C(F)F)c2c1 38248,N1(C(C(CC#C)C)=O)CC2CCC2(CNC(c2ccc(NS(C)(=O)=O)nc2)=O)C1 38249,c1(NCC2C(C)(C)CCCO2)ncc(S(=O)(=O)NC(c2nccs2)CO)cc1Cl 38250,Cc1c(C(=O)NC2CC3CCC2N3c2cc(OC3CC3)ncn2)cncc1Cl 38251,C=CCC(CC(=O)NCc1ncoc1CC)NC(=O)C(CCC)N(C)C 38252,C1(C(=O)OCC)CN(C(=O)CN2CCC2c2cccc(Br)c2)C(C)(C)C1 38253,c1(NC(C)(C)C)cccc(S(=O)(=O)NC2(C)CCC(=O)NC2=O)c1 38254,c1(C(N2CCN(C(C(C(CC)C)O)=O)C(C(C)C)C2)=O)cc(C)c2[nH]nnc2c1 38255,c1(C(=O)NC(CNC(=O)CNC(c2ccoc2Br)=O)C2CC2)ccc2nn[nH]c2c1 38256,C1(CC(=O)NC2C(OC)CCC2)CCCCN1C(=O)CC1COCC(C)O1 38257,N1(C(C2C3CN(C(CC4(C)CCCC4O)=O)CC32)=O)CCn2cncc2C1 38258,c1(C(=O)NC2CCCN(C(Cc3cccc(OC)n3)=O)C2)ccc2c(c1)CCN2 38259,C1(NC(C(C)N2CCCC2)=O)CC2CCC1CN2C(=O)CCCCN(C)C 38260,C1(CC(=O)NCC(CO)C2CCC2)C2CCCC2N1C(=O)CC1CC2(CCC2)C1 38261,C1(NC(CCCC=C)=O)CCC2(CC1)CC2NC(c1c(C2CCC2)cnn1C)=O 38262,n1(CC(N2CCC(NC(=O)CSCC(=O)NC3CCOC3)C2)=O)cc(Cl)cn1 38263,C1(C(N2CC(CNC(C(c3cncnc3)C)=O)C2)=O)CC(=O)N(C2CCCC2)C1 38264,C=C(C)CCC(C)NC(=O)CN(C)C(c1cc(OC)ncn1)=O 38265,CC1COCc2cc(C(=O)NC3CC(CCNC(c4cnco4)=O)C3)nn2C1 38266,CCN=c1ccc(C(=O)NCC2(F)CCCN(C(c3ccc(SC)o3)=O)C2)c[nH]1 38267,c1(C(=O)NCCCn2cc(C(C)(C)C)nn2)ccc(CO)cc1F 38268,c1(C(N2CCC(CNC(C(C=C)O)=O)CC2C)=O)c[nH]c2c(F)cccc12 38269,O=C(NNCCCC(F)(F)F)C1=CCCCNC1 38270,N1(C(Cc2ncc(C)s2)=O)CC2CC(NC(c3cn(C)nc3C(F)(F)F)=O)C2C1 38271,CC1=C(C(=O)N2CCC(C)(NC(C3CC4CC4C3)=O)C2)CCCO1 38272,c1(C(N(C(C2CCOCC2)C)C)=O)ccc(CNC(C2CC3(CC3)CO2)=O)cn1 38273,c1(CC)oc(C(=O)NCCC2CN(C(=O)CCC(C)OC)C2)cc1C(=O)OC 38274,c1(C(=O)NC2(CCOC)CCN(C(c3cnncc3O)=O)C2)c[nH]cc(C)c1=O 38275,Cc1cc(F)ccc1-n1cc(O)c(C(=O)OCC2C=CCC2)n1 38276,c1(C(=O)NCCC2N(C(C(CC=C)C)=O)CCSC2)ccc(Br)cc1Cl 38277,CC1CCC(C)(NC(=O)COC(C2CNCC23CCOC3)=O)C1(C)C 38278,c1(CNC(C2CCC3(CN(C(CCC(C)C)=O)C3)O2)=O)ccc2ncccc2c1 38279,c1(C(=O)NC2C(CNC(c3c[nH]c(=N)o3)=O)C2)cn2cc(Cl)cnc2n1 38280,C1(C(N(C(C=C)C2CC2)C)=O)OCCC1CNC(=O)Cn1nnnc1C 38281,C12(C(=O)NC3CCCC(N(C(C(CC#C)C)=O)C)C3)CCOC(C)(C1)C2 38282,CN=c1[nH]cc(C(=O)NC2CCOCC2C(=O)NCc2cc(Cl)ccn2)s1 38283,C(C)(CNC(c1csc(C(C)(C)C)n1)=O)(C(C)C)NC(c1c(C)occ1)=O 38284,N1(C(=O)NCc2nc(C(=O)OCC)on2)CC(C2CCC2)CCC1C 38285,C(=O)(CC(O)(c1ccccc1)n1cccn1)N(CC(C)NC(C1CC(=O)C1)=O)C 38286,c1(C(=O)NCC2CC3CCC2N3C(C2CC23CC3)=O)coc2c1CCCC2 38287,C1(C(N2C(CNC(C3CC4(CCC4)C3)=O)CC3CC32)=O)CCc2nc(O)[nH]c2C1 38288,C1(CC(=O)NCCCCCNC(C(CSC)OC)=O)CCCCC12CC2 38289,c1(C(=O)NC2CC(CNC(C3CC4CC4C3)=O)C2)cccc2ccnn12 38290,N1(C(CC2CCN(C)CC2)=O)CCC(NC(=O)C=CC2CCC2)CC(C)(C)C1 38291,N1(C(C=CC(C)(C)C)=O)CC2CC1CN2C(c1[nH]ccc1-c1ccccc1)=O 38292,c1(C(=O)NC2(C)CCC(NC(=O)C(N)=O)CC2)coc(C#Cc2ccccc2)c1 38293,c1(CC(=O)NC(c2cccc(OC)c2)CC)cnc([N+](=O)[O-])c(C)c1 38294,O=C(CC(C(F)F)c1cccc(F)c1)NCC1CC1CNC(=O)CO 38295,N1(C(c2cc(OC)ncc2)=O)CCCN(C(c2cnc(C3CC3)o2)=O)CC1C 38296,C1(NC(c2c(C)ocn2)=O)C2CC3C1C3C2C(=O)N(C(C)C)CC1CCC1 38297,N1(C(CCC(=C)Cl)=O)CCCCC(CNC(C2CCCN(CC(C)C)C2)=O)CC1 38298,C(C(C)CC(=O)N(C(C)CN(C(=O)Cn1nc(C(F)(F)F)cc1C)C)C)OC 38299,C1(CCC(C)NC(c2nnc(SC3CCOC3)s2)=O)CCCN1C 38300,C(=O)(CC(O)CNC(=O)CCC1CC1(F)F)N(C)CC1CCCC1 38301,C(CC(=O)NCC1(F)CCN(C)C1)(C(F)(F)F)NC(C1(OC)CCOC1)=O 38302,c1(C(C)NC(c2nc(C(=O)NC(C(=O)OC)C3(C)CC3)[nH]n2)C)c[nH]ccc1=O 38303,CCCC(C)(O)CC(=O)NCC1(C)CN(C(=O)Cc2nc(C)c(C)s2)CC1C 38304,N1(C(C(C)C#N)=O)CCOC(C)(CNC(c2ncccc2-c2ccccn2)=O)C1 38305,C1(C(=O)NC2C(c3cn(C)nc3)C2)N(C(=O)CC2CCC=CCC2)CCC1(C)C 38306,C(=O)(C(CCC)NC1COC(C(F)F)C1)OCC=C 38307,Cc1ccc(C(N2CCC3CN(C(C4CCCCC4F)=O)CC23)=O)cc1C#N 38308,CC(CN(C)C)N=c1[nH]c(N2CC(CO)C(C)(C)C2)nc2c(F)cccc12 38309,Cc1nc(O)ccc1C(N1CC2CC2C1C(=O)NC(C)Cc1cnccn1)=O 38310,C(CNC(c1cc(Br)no1)=O)(C(C)(C)C)NC(c1ccc(C(=O)OC)s1)=O 38311,N1(C(c2cnc(-c3ccccc3)o2)C(=O)NCC=C)CC(=O)N2CCCCC2C1 38312,C(=O)(CCCCO)N1C(C2(C(=O)NCC3CCC(F)(F)C3)CC2)CCC1 38313,C=C(C)CC(C(=O)NC(C)C(=O)N(CC(C)O)CC1CC1)OC 38314,C1(CNC(c2c(C)[nH]c(C)c2C)=O)(NC(=O)C(C)CN(C)C)CCC(C)(C)CC1 38315,CC(=O)CCCC(=O)N1C2CCC(C2)C1C(=O)Nc1cn(C)nc1C#N 38316,c1(OC)ccc2oc(C(=O)NC3CCCCC3NC(=O)C=C(C)Cl)cc2c1 38317,C1(N(C(C(CC)O)=O)C)C2CN(C(=O)CCCNC(=O)OC)CC12 38318,c1(C(=O)NC(C2CCCN2C(=O)CCc2cccs2)C)cc(C(F)(F)F)n[nH]1 38319,c1(C(=O)NC2C(CNC(CSCC(C)C)=O)CCC2)nnc(O)cc1O 38320,Cc1cc(=O)n(C)cc1NC(C1CC12CC(NC(=O)C(C)CN(C)C)C2)=O 38321,C(=O)(C(C)C(O)C(C)C)NC(C(N1CCCC(C)(CC)C1)=O)(C)CO 38322,C1(C(N2CC=CC2Cn2cc(CCN3CCOCC3)nn2)=O)C2COCC12 38323,C1(C(=O)NC(c2cc(F)ccc2OC)CC)CC2(CCC(N)CC2)C1 38324,c1(OC)cc(C(N2CCC(O)(C(C)NC(=O)CCC3(C)CC3)C2)=O)cc(F)n1 38325,S(=O)(=O)(c1ccc(N2CCC3CCCC3C2)cc1Cl)NC1CC2N(C)C(CC2)C1 38326,c1(OC)ccc(C)c(CNC(c2cccc(N3CCCCC3=O)c2)=O)n1 38327,Cc1nc2ccc(C(=O)N(C)CC3CCCCN3C(c3occc3Cl)=O)cn2n1 38328,C12(CNC(C(C)NC(=O)NC)=O)CC1CN(C(=O)C=Cc1c[nH]nc1C)C2 38329,c1(C(=O)NC2CC(C)(NC(c3c(Cl)cnn3C3CC3)=O)C2)cncc(F)c1Cl 38330,N1(C(C2CCCOC2)=O)CCC(N(CCO)C(C2(C(F)F)CCC2)=O)CC1 38331,CC1(C2CC2)CCN(C(=O)CC2CCCCN2C(=O)C#CC2CCOC2)C1 38332,C1(C(=O)NCC(CC)(CC)OC)C=CCN(C(C2(C)CC3CC3C2)=O)C1 38333,N1(C(C(=O)NC(C(CC)C)=O)CCO)CCc2sccc2C1 38334,N1(CC(N2CC(C3N(C(C(CC)CC)=O)CCC3)(O)C2)=O)C(=O)CN(C)C1=O 38335,C1(C(=O)NCC(C)N(C(=O)Cc2ccnn2C)CC)CC(O)CN1C 38336,Cc1c(C(N2C3CCC2C(NC(C24CC(F)(C2)C4)=O)C3)=O)cnc2ccccc12 38337,S(=O)(=O)(C1CC2CCC1O2)N1CCC(N(C2CCCC2)C)C1 38338,c1(C(=O)NC(CNC(CC(CCC)C)=O)C(C)(C)C)ccc(C)c([N+](=O)[O-])c1 38339,C(CCCCNC(=O)CNC(=O)NC1CC1)NC(C(C1CCOCC1)OC)=O 38340,C1(NC(c2cc([N+](=O)[O-])n[nH]2)=O)CCN(C(=O)COCC2CC2)CC1F 38341,N1(C(c2ccc(NC)cn2)=O)CCC(O)(CNC(c2cc(Cl)ccn2)=O)CC1 38342,C1(NC(C(C)SCC)=O)CCCN(C(C23CC(CC)(C2)C3)=O)C1 38343,N1(C(C2CCC(OC)C2)=O)C(C(=O)NCCCC2CCC2)CCC1C1CC1 38344,CC1CN(C(=O)CCN(C)C(c2ncccn2)=O)CC1(F)F 38345,c1(C(N(C(CNC(C2N(CC)CC2)=O)C)CC)=O)cn(CC)nn1 38346,N1(C(C2(C)C(C(=O)OC)C2)=O)CCOC(CNC(=O)CCSC(F)(F)F)C1 38347,c1(C(=O)NCCOCCN(C(C(CCC)OCC)=O)C)c(N)ccc(C)c1F 38348,C1(=C(CNC(c2cc(CCC)on2)=O)F)CCN(C(=O)C(C)(COC)OC)CC1 38349,C=CC1CCCCN1C(=O)COC(C1CCN(C=O)CC1)=O.C(C)(C)(C)OCCS 38350,N1(C(CCC2CCN(C(C3N(CCC)CCC3)=O)C2)=O)CCC(O)CC(C)C1 38351,C(C(C)(C)C(=O)NOCc1ccc(F)cc1)N(C(CC1CCC(C)O1)=O)C 38352,N1(C(C(=O)N(C(C)C)CC)=O)CCCC(N(CC(C)C)C)CC1 38353,N1(C(c2c(CC)c(F)ccc2)=O)CCC2(CCN(C(C3CN(C)C3)=O)CC2)C1 38354,N1(C(COCC(=O)NC)=O)CCN(C(=O)CC2(C(F)(F)F)CCC2)CCC1C 38355,CCC(CC(=O)N1CCC(C#N)(c2ccc(F)cc2)CC1)CC(C)C 38356,N1(C(C(CC2CC2)OC)=O)CCN(C(=O)Cc2cnn(C)c2C)CC(C)C1 38357,c1(C(=O)NC(c2cn(C)cn2)C(=O)NC(CC=C)C)cccc2c[nH]nc12 38358,Cc1csc2c(C(N3CC=CC3CNC(C3CCC4(CCC4)O3)=O)=O)ncnc12 38359,N1(C(CCOCC)=O)C2CCC1CC(O)(CNC(=O)C(F)Cc1ccccn1)C2 38360,C1(CNC(c2nc(C)sc2)=O)CCC2CN(C(=O)CC(C)C)CCC2C1 38361,C1(C(C)C)C(=O)N1.C1(CNCCC2(NC(C=CC)=O)CCCC2)CCCCC1F 38362,Cc1cc(NC(c2nc(Nc3ncc(F)c(C)n3)cn2C)=O)cc(C#N)c1 38363,c1(CC(=O)NC2C3CCN(C(c4nc(C)oc4)=O)C32)c(C)cccc1C 38364,C1(C2CC2)(COC(c2ccc(-c3ccncc3)o2)=O)OCCO1 38365,C1(CCC)(CNC(c2[nH]ccc2COC)=O)CCN(C(C2CN3CCC2C3)=O)C1 38366,c1(C(=O)NCCC2N(C(C34CC(C)C3C4)=O)CCC2)cccc(CC2CCC2)c1 38367,c1(C(=O)NC(CCNC(C2CCC(C(=O)OC)C2)=O)(C)C)nc(C)sc1Br 38368,S(=O)(=O)(c1ccsc1)N1C(C)(C(=O)NCC2COCCO2)CCC1 38369,C1(C(N(C(C)CC(=O)NCC(O)(C2CC2)C2CC2)C)=O)CC12CCOC2 38370,CC(CCCCNC(C1(N(C)C)CCOCC1)=O)NC(C12COCC1C2)=O 38371,C1(NC(c2nnnn2CCOC)(CC)C2CC2)CCC2(CC1)CSC2.C1CCOC1 38372,c1(C(=O)NC2C(NC(C(N(C)C)C3CC3)=O)CC2)ccc2cccc(Cl)c2n1 38373,c1(N(CCCN)C(c2coc(-c3ccccn3)n2)=O)nccc(C)n1.CC 38374,Cc1nc(C=CC(N2CC(NC(=O)CC3CCCCCO3)C(F)C2)=O)[nH]c1C 38375,C(=O)(CCCC(C)=O)NCC(CNC(C)=O)OC.c12cnc(o1)[nH]c2=O 38376,CC(C(=O)N1CCOCC(CNC(=O)CNC(C2CCOCC2)=O)C1)S(C)(=O)=O 38377,C1(C(N2CC(OC)(CNC(C3(C)CC3(C)C)=O)C2)=O)CN2CCN1C(C)C2 38378,c1(N2CC(C)(C)C(CO)C2)nc(NCCN2CCOCC2)c2ncsc2n1 38379,CC1CCN(C(C2(F)CC=CC2)=O)CC1NC(=O)CCc1ccc(F)cc1 38380,c1(C(=O)NC2(C3CCCCN3C(=O)C(F)=CCCF)CC2)cc(Cl)c(F)c(Cl)c1 38381,c1(C(=O)NCC(C)(CNC(=O)C(C)(C)N(C)C)OC)c(C)oc(C)c1C 38382,C1(CNC(C(C(C)C)N(C)C)=O)C2CCCC1N(C(=O)CSC(F)(F)F)C2 38383,c1(NCC)ncnc2sc(C(N3CCC(CNC(C4CC(O)C4)=O)C3)=O)c(C)c12 38384,N1(C(C(C(C)(C)C)OC)=O)CCC(C2(NC(c3scc4c3OCCO4)=O)CC2)C1 38385,c1(CC)ncc(C(=O)NC2CC(NC(c3c[nH]nc3C(=O)OC)=O)C2)[nH]1 38386,C1(c2nnnn2CCC2CC2)(NCC(n2cc(Cl)cn2)C)CC2(C1)CC(F)(F)C2 38387,Cc1cc(=NCC2(O)CC3CCC2C3)[nH]c(CCN(C)C(c2ccccc2)C2CC2)n1 38388,CCC(CC(=O)N(CCNC(c1c(C)nnn1CC)=O)C1CC1)C(C)(C)C 38389,C1(CCCCNC(=O)CC2COCCO2)CCN(C(=O)CC2C=CCC2)CC1 38390,c12c(cnn1C)-c1cn(nn1)CC(=O)N2.C1(C(C)(C)OC)CCN(C(C)=O)CC1 38391,N1(C(c2cc(C)c(C)nc2C)=O)CC(CO)C2(CCN(C(=O)CC(C)F)CC2)C1 38392,C1(NC(c2c(C)onc2CO)=O)CC2CC1N(C(=O)C(=CC1CCCCC1)F)C2 38393,C1(NC(C=CCOC)=O)(CO)CN(C(=O)CCCSC(C)(C)C)C1 38394,c1(NC(c2c(C)nco2)=O)cccc(NC(=O)C=C(Cl)Cl)c1 38395,N1(c2c(C)nc(N3CCc4c(Br)cccc4C3)o2)Cc2cc(Br)ccc2C2CC1C2 38396,c1(CCC(=O)N(CCC)CCNC(C2CC3CC2C3)=O)ccc2c(c1)CCCO2 38397,c1(N(C2CC2)CC)nc(C(=O)OC(=O)C(C)OC)cs1 38398,CC1(C)Cc2cccc(NC(=O)C(N3CC=CC3NCCO)=O)c2O1 38399,N1(C(C(CC)(C)O)=O)CC2(CC2)CC1C(=O)Nc1ncc(Br)nc1C 38400,C#CCC(C(=O)N1CCC1c1cn(CC2(n3ccnc3C)CC2)nn1)OC(C)=O 38401,N1(C(=O)OC(C)(C)C)CC2C(NC(=O)Cc3ccc(Cl)cn3)C2C1 38402,C=CC(O)(C(=O)N1CCCCCC(NC(c2sc(C)cc2Cl)=O)C1)C(F)(F)F 38403,C1(C(=O)NCC(CC=C)NC(=O)CSCC(=O)OC)CCC(CC(F)(F)F)CC1 38404,C1(CC(=O)NCc2ccn(CC)n2)CN(C(=O)CCc2nc(C)no2)CCO1 38405,Cc1cccc(C(CNC(c2ncncc2C)=O)NC(c2cn[nH]c2)=O)c1 38406,C1(C(=O)NC(c2ccccn2)C)CCN(C(c2ccc(=O)n(C)c2)=O)C(C)(C)C1 38407,C(C(C)(CC(C)C)NC(=O)CCC1CCCO1)NC(c1sn(CCC)c(=O)c1)=O 38408,CCC(C)CCCC(=O)NCCCCC1CN(C(=O)CCC2OCCO2)C1 38409,c1(OCC)nc(Cl)ccc1C(=O)NCC(CC)NC(C1(O)CC(C)(C)C1)=O 38410,N1(CC(C)Oc2ccc(Br)cc2)CCCCC1c1ccsc1 38411,c1(C(N2CC(NC(CC3(C)CC3)=O)C2)=O)ccc(-n2cnnc2)cc1 38412,N1(C(CCC2CCCC(=O)N2)=O)CCCN(C(C23CSC(C2)C3)=O)CC1 38413,c1(C(=O)NCCN(CCOC)C(C2CC=CCC2)=O)csc(O)n1 38414,C1(C(=O)NC(CC#C)CC)CCCCN1C(=O)Cc1cc(C)on1 38415,Cc1csc2ncc(C(=O)NC34CCCC3N(C(=O)COCCC(C)C)CC4)n12 38416,C1(C(=O)NC2CC(NC(c3cc(Cl)cc(Cl)c3)=O)C2)CCN2CCCC2C1 38417,n1(NC(C(Cn2cncn2)NC(C(N2CCNC2=O)C)=O)=O)ccc(C2CC2)n1 38418,Cc1ccc(C)c(CC(=O)NC2CCN(C(=O)CC3(C)OCCO3)C(CO)C2)c1 38419,c1(CN2CC(C(N3CCC(Br)C3)=O)SCC2)c(O)cccc1O 38420,C1(NC(Cc2c(C)ccs2)=O)CCC(CNC(=O)C(N2CCOCC2=O)C)CC1 38421,C1(C)(C(=O)NCCCCN(C)C(C2CC2c2ccccc2)=O)CC(C2CC2)=NO1 38422,CC1CCN(C(=O)Cc2cnns2)CC1NC(=O)C=CC1CCCCC1 38423,c1(C(=O)NC2CCN(C(=O)Cn3ccc(O)nc3=O)C2)ccc2nccn2c1 38424,Cc1c(Cl)cc(C(C)NC(=O)C(=O)NCC(c2ccc(Br)s2)O)cc1I 38425,C(CC(C)(C)C)(C(=O)N1CCC(CF)(NC(=O)CSC(F)(F)F)C1)OC 38426,C1(C(=O)NC2(CNC(Cc3nc(C)c(C)s3)=O)CCCCC2)COCCC1(F)F 38427,C(=O)(C1=COCCC1)NC1CCC(CNC(C(CCOC)OC)=O)C1 38428,Cc1ccc(CN2CCC(CCNC(=O)C(C)CCO)C2)cc1 38429,c1(N2CC(CC)(NC(=O)CC3COCC3O)C2)ncnc2[nH]c3ccccc3c12 38430,c1(NC)cccc(OC)c1C(N1CC(CCO)(NC(C2CC(Cl)(Cl)C2)=O)C1)=O 38431,C1(CN(C)C(c2ccns2)=O)CCCN1C(=O)CCCc1nccs1 38432,Cc1nn(C(C)C)c(C)c1C(N1CC2CN(C(=O)CCC3CC3)C2C1)=O 38433,C12(C(=O)NC(C3CCN(C(=O)C(c4ccccc4)O)C3)C)CCC(N=[N+]=[N-])C1C2 38434,N1(C(C(C=CCCC)O)=O)CC(CNC(C2CC23CC(O)C3)=O)C(C(F)(F)F)C1 38435,c1(SC)cccnc1C(=O)NC(CNC(c1ccn(C(F)F)n1)=O)C1CC1 38436,Fc1cc(C2CC2CN(C(=O)CCc2cncs2)C2CC2)ccc1Br 38437,CCCCC(O)C(=O)NCC(CC(C)C)NC(c1cnn(CCOCC)c1)=O 38438,c1(C(=O)NCC2CCCC2NC(=O)C=C2CCCCC2)cccc(C#CCO)c1 38439,c1(OC)cc(C(=O)NCC2(NC(C3CCN(C)C3C)=O)CCOC2)ncn1 38440,C1(C)(NC(c2c(SCC)cccn2)=O)CCCN(C(=O)Cc2cccnc2)C1 38441,C(C(C)(O)CC(=O)N(C(C)C(=O)N(C)Cc1cncs1)C1CC1)OCC 38442,C(=O)(C(CCC)C(=O)OC(C)C)OCCOCCC=C 38443,CCCC(C#N)C(=O)NCC(CNC(=O)C(CSC)OC)OC 38444,N1(C(c2c(C)c(N)cnc2)=O)CC2CCCC2(NC(=O)Cc2cccnc2Cl)C1 38445,N1(CC)CCC(CN(C(=O)C(c2cnn(C)c2)NC(c2sncc2C)=O)C)C1 38446,C12CC(C1(C)C)C(=O)N2C(=O)C=C(C)C1CC1.N1(CCOC)CCCNC1=O 38447,c1(NC2CCCC(NC(C3CCOC3)=O)C2)ncnc2ccc(O)cc12 38448,c1(NC(C2CC(=C)CN2C(c2ccc(Br)s2)=O)=O)cc(F)cnc1C#N 38449,C=CCCCCCCC(=O)NCC(C)NC(c1c(N)cc(F)cc1F)=O 38450,c1(N(C)C)ccc(C(=O)NC(CCCNC(c2ccncn2)=O)c2ccccc2)s1 38451,c1(NC(=O)C(C2CCCO2)c2cccs2)cc(Cl)cc([N+](=O)[O-])c1O 38452,CC1CC2(CCN(C(=O)CC3CCCCO3)CC2)CN1C(c1nn[nH]c1Cl)=O 38453,c1(C(N2CCC(O)(CNc3cc(OCC)ncn3)C2)=O)cc2cccc(Cl)c2o1 38454,c1(C(N(CCC)CCNC(C2CCC2C)=O)=O)coc2ccc(OC)cc12 38455,C(C(=O)NN1CCSCC1)(C12CC3CC1C2C3)c1ccccc1.CC(C)(C)O 38456,c1(CC)c(OC)cccc1C(=O)NC(CNC(C1COCCC1(F)F)=O)C(C)C 38457,N1(CC(=O)N(CCCCCNC(=O)C2CC2)C2(CC)CCC2)CC2CCC1C2 38458,N1(C(C(CC)F)=O)CCC2(CCCN(C(=O)COc3ccc(Cl)nc3)C2)CC1 38459,N1(C(C(C2CC2)SC)=O)CC2(CCCC2CC(=O)NCCCC2CCOC2)C1 38460,N1(C(c2c(C)cc(N)cn2)=O)CC2COCC2(C(=O)NCc2ncc[nH]c2=O)C1 38461,c1(OC)cc(OC)c(C(N2CCN(Cc3cccnc3Br)C3CC23)=O)cc1Br 38462,CCC(CC(F)F)C(=O)NCC1CCCCN(C(=O)CC2CCCNC2=O)C1 38463,CCCCC(C(=O)N(C1CC(NCC)C1)C)NC(c1ccoc1COC)=O 38464,Cc1ccc(Cl)c(O)c1C(=O)NCCCCC(C)NC(C1CC(C)CCO1)=O 38465,N1(C(=O)CC2=CCCC2)CCC2C(CCCN2C(c2cnc(-c3ccco3)s2)=O)C1 38466,c1(C(N(C)CC2(NC(C3CC(C(C)(C)C)=NO3)=O)CC2)=O)ccc2n[nH]cc2n1 38467,C(c1cn(C)nn1)=CC(=O)NC(C(=O)NC(CC)Cn1cncn1)C1CCCO1 38468,c1(C(=O)NC2CCN(Cc3c(C)ccs3)CC2)cc(F)cc(Cl)c1 38469,c1(C(N2CCC(N(C(=O)CNC(C3CC3C)=O)C)C2)=O)ccnc(O)c1 38470,C12(OC)CCCCC(C(=O)NCC(C3CC3)NC(=O)CCn3ccccc3=O)(C1)C2 38471,C1(C)(NC(C=C(C)C(C)C)=O)CCN(C(=O)C(C(C)C)n2cnnc2)CC1 38472,c1(OC(CCCc2c(C)ccs2)=O)cc(Br)c(F)cc1F.c1(N)cccc(C=O)n1 38473,C12(C(=O)NC3C(C)CCN(Cc4nnc(COC)s4)C3)CCCC(=O)N1CCC2 38474,c1(CN2C(C3CCN(C(C(CC=C)C)=O)CC3)CCC2)ccc(C)c2cccnc12 38475,N1(C(CC2C(C)(C)C2)=O)CCC(NC(c2cc(N)c(O)c(F)c2)=O)C(F)(F)CC1 38476,C1(F)(C(=O)NC2CC(CNC(C=CC(C)(C)C)=O)C2)CCCOC1 38477,CN1CCC2CN(C(C3CCN(Cc4ccc(N(C)C)cc4)CC3O)=O)CC2C1 38478,N1(C(CNC(C(CC)C)=O)=O)CC=C(C(=O)NC(CO)C2CC2)C1 38479,Cc1nc(Cl)[nH]c(=NCC2CC(CNC(=O)CC3CCCCO3)CO2)c1Cl 38480,C1(NC(C(c2n(C)cnc2)O)=O)CC2(CCC(NC(C3OCCCO3)=O)CC2)C1 38481,c1(C(=O)NC(CN(C(c2c(C)snn2)=O)C)C)csc2cc(Cl)cnc12 38482,C=C(C)CC(C)C(=O)NCCOC1CCN(C(=O)C(C)N2CC(C)C2)CC1 38483,c1(CC)cc(C(N2CCC(NC(c3cc(O)ncn3)=O)C2)=O)ccn1 38484,Cc1cc([N+](=O)[O-])c(Cl)cc1S(=O)(=O)NC.C1(C(=O)O)(OC)CC2(C1)CC2(F)F 38485,n1(CCC)cc(Cl)c(C(=O)NCC23CC2CN(C(=O)Cc2conc2C)C3)n1 38486,c1(COC)nccc(=NC2CCC3CN(C(c4n[nH]c(C)c4C)=O)CC23)[nH]1 38487,Cc1nnc2n1CC(C(=O)NC(C1CN(C(=O)CC3CCC3(C)C)C1)C)C2 38488,C(=O)(CCCCN(C)C(C)C)N1CC(F)(CNC(C(C=C)O)=O)C1 38489,C(=O)(C(C)(C)S(C)(=O)=O)NC1C(CNC(c2ccc(OC)c(O)c2)=O)CCC1 38490,N(C1CCCn2cnnc21)C(CC(C)NC(C(=C1CCCCC1)C)=O)=O 38491,c1(CNC(C)=O)cc(Cl)cnc1OCCN1CCC(c2ccccc2)C1C 38492,c1(OC)ccc(CN(C2CCOC(c3ccncc3)C2)CC(C)C)cc1 38493,N1(CC2CCN(C(c3cc(OC)cc(F)c3)C(=O)NC)C2)CC2CCC(OC)C2C1 38494,C(=O)(C1Cc2ccccc21)NC(C1CCCCC1)CNC(c1c(CC)ocn1)=O 38495,N1(C(C(C)SCC)=O)CCC(CNC(c2cnnc(C3CC3)c2)=O)C(F)(F)CC1 38496,C1(C)(c2cn(CC=CCOCCOC)nn2)CCCN(C(C2(C#N)CC2C)=O)C1 38497,C1(CNC(CCCN(C(C)=O)C)=O)CCCN(C(=O)C(N2CCCC(O)C2)C)C1 38498,C(=O)(CCCCC(C)(C)C)N1CC(NC(c2c(CC)onc2)=O)(CF)C1 38499,c1(OC)cc(NC(=O)CS(C)(=O)=O)c(-c2sc(N3CCCC3)nc2C)cn1 38500,N1(C(CCC#CC)=O)CCCC(NC(=O)Cc2c(O)ncnc2O)C(F)C1 38501,C1CCCCCC(C(=O)N(C(C)C)C)N2CC3C1C3C2.C(CC1CC1)N.C(C)C 38502,C(=O)(C1=C(C)OCCS1)N1CCCC(CN(C(CCC=CC)=O)C)C1 38503,N1(C(CCOCCOCC)=O)CCC(C)(N(C)C(c2cnccn2)=O)C1 38504,N1(C(CC2C(CC)C2)=O)CC(C(=O)NCC(=O)NOC)CCC1(C)C 38505,N1(C(C2C3CC4C(C3)C24)=O)CCC(C2CCCN(C(=O)NC3CC3)CC2)CC1 38506,N1(C(Cc2c(C)cnn2C)=O)CC2(CC(NC(=O)C(C)CF)c3nccn32)C1 38507,C(=O)(C#CC(C)(C)C)N1CC(OC)C(NC(c2ccccc2SC(C)C)=O)C1 38508,c1(CC)nn(C)c(CC)c1C(=O)N(CC(C)NC(=O)Cn1nnnc1C(C)C)C 38509,N#Cc1c[nH]c(=NC(=O)NC(c2cccc(F)c2)C(=O)NOC2CCOC2)cc1Cl 38510,C(N=c1[nH]ccn2nnnc12)C1CC(NC(c2onc(C)c2C(C)C)=O)C1 38511,c1(C(N2C(CC(N3CCN(CC(C)C)CC3)=O)CCCC2)=O)cccc2ccnn12 38512,C1(C2CCCN(C(c3ccn4ncccc34)=O)C2)(NC(c2n(C)cnc2)=O)CC1 38513,C12(CNC(CC(CC)C)=O)CCCC1N(C(=O)Cc1c(OC)cccc1F)CC2 38514,N1(C(C(CC)OCC)=O)CCCC(C2CN(C(c3cccc4[nH]ncc34)=O)C2)C1 38515,C1(C)(C(=O)NC2CCN(C(COCc3cc(OC)ncc3)=O)C2)CCS(=O)(=O)N1 38516,c1(CC)conc1CC(=O)NCCC1(O)CN(C(c2n[nH]cc2Cl)=O)C1 38517,C1(C(=O)NCCNC(CC)=O)C=CCCN1C(=O)CC1CCC1 38518,N1(C(Cc2c(OC)cccc2Cl)=O)CCC2(CCC2)C(NC(=O)CC(C)F)C1 38519,N1(C(CCCc2nnc(C)n2C)=O)CCCC(NC(=O)CC2CCCCC2)C1C 38520,c1(C(C)C(=O)NC2CC2c2cccc(NS(C)(=O)=O)c2)ccc2c(c1)OCO2 38521,c1(N(C)C)nc2cc(C(=O)NC3CC(NC(=O)COC4CC4)C3)ccc2o1 38522,C1(CCOC)CN(C(c2cccc(F)c2Cl)=O)CCN1C(C12CC3CC1C2C3)=O 38523,N1(C(C(c2cc(C)oc2C)C)=O)CCC2CCN(C(c3cnn(C)c3)=O)C2C1 38524,c1(CC)ccc(C(=O)NC2(CC)CN(C(C3CC[Si](C)(C)C3)=O)C2)cc1 38525,N1(C(C(C(C)O)N(C)C)=O)CCOCC(C)(CNC(c2coc(CO)c2)=O)C1 38526,c1(C(CNC(c2ccc(OCCOC)nc2)=O)C(F)F)ccc2cc[nH]c2c1 38527,C(C)(CNC(C1(C(C)(C)C)CCCCC1)=O)(C(C)C)NC(Cc1nnc(C)o1)=O 38528,C(=O)(C(C)(C)CCCNC(=O)C(F)C1CCOC1)NC(C)Cn1cnnc1 38529,N1(C(C2CN(C(C(CC)(C)COC)=O)CC2CC)=O)CCOC2C(O)CC12 38530,CC(CO)CN=c1[nH]c(N2CCC(C(C)CO)CC2)nc2c1CCCC2 38531,C(=O)(CCCCC(C)C)NC1CCC(C)(CNC(c2nccc(OC)c2)=O)CC1 38532,C1(C(N(C(CNC(C2N(CC#C)CCC2)=O)C)C)=O)CCc2nncn2C1 38533,C(=O)(C1=NN(C)C(=O)CC1)NC1CCN(C(CC)=O)C(C2CC2)C1 38534,c1(C(=O)NCC(CNC(=O)C(C)c2cc[nH]n2)OC)cccc2ccncc12 38535,C(Cn1cncn1)(C(=O)N(C)C(C1CCOCC1)C)NC(C=CC)=O 38536,N1(C(c2nccc(OCc3nc(C)on3)n2)=O)CCCN(CC2CC(O)C2)CC1 38537,C1(C(=O)NCC2CC(NC(CCc3cc(C)on3)=O)C2)OC(C)(C)OC1(C)C 38538,N1(C(=O)Nc2nccc(F)c2F)CCC(C(F)(F)F)C(Cc2ccc(C#N)[nH]2)C1 38539,c1(C(=O)NCC2(C)CCN(C(C(C)C3CCC3)=O)C2)ccc(N)c(F)c1F 38540,C1(C)(C(=O)NCC(CNC(c2c(CC)[nH]cc2)=O)(C)F)Cc2ccccc2C1 38541,C1(C)(C(=O)NCC(CCNC)OC)CCN(C(C2(O)CC(F)(F)C2)=O)CC1 38542,Cc1cn2cc(C(=O)NC(c3ccc(F)cc3)CNC(=O)CC#N)cc(Cl)c2n1 38543,C1(C(=O)NCCn2cncn2)C2CN(Cc3ccc(-c4ccccc4)o3)CC12 38544,c1(C(=O)NC(CNC(c2ccc(C)cn2)=O)(C)C(C)C)cc(C2CC2)n(C)c1C 38545,Cc1nnc(NC(c2ccc(F)cc2)CO)n1CC(F)(F)F 38546,C(=O)(CC1OCCc2ccccc21)NCCNC(CNC(CCCCC(=O)NC)=O)=O 38547,O(NC(=O)C(F)C1CC1N(C(=O)OC(C)(C)C)CC)CCOC(C)(C)C 38548,N1(C(C2(C)C(C)OCC2)=O)C2CCC(C(=O)NC3CCCCCC3F)C1CC2 38549,c1(OC)c[nH]c(C(=O)NC(C2CCN(C(C3CCC4(CC4)C3)=O)CC2)C)cc1=O 38550,c1(SC(c2cc(Br)ccc2O)C)ccc(F)cc1F.C12CCN(CC1)C(=O)N2 38551,C(CC(O)C(=O)NC1CCCC1NC(C1(C2CCCCO2)CC1)=O)N(C)C 38552,c1(C(=O)Nc2ncc[nH]2)cc2ccc(-c3ccc4c(c3)CNC4=O)nc2[nH]1 38553,N1(C(C(CN(C)C)O)=O)CCCC(CO)(NC(C2CCC(F)(F)CC2)=O)C1 38554,c1(OC)cccc(C(O)C(N2CC(NC(c3nc(C)nn3C)=O)C(C)C2)=O)c1 38555,C1(CC(=O)NCCN(C)C(c2ncc(F)cc2N)=O)CCCC(F)(F)C1 38556,CC1(C)CN(C(=O)CCCCC2CCCC2)CC1NC(c1cnn(C(F)F)c1)=O 38557,C(=O)(N=c1[nH][nH]c(C)c1Cl)C1C(F)(F)CCN(C(c2cc(C)c(N)cn2)=O)C1 38558,c1(NC(=O)NC2CC(OCC)C2(C)C)ccc(OCC2COC2)cc1.c1ccoc1 38559,C1(c2nnnn2CCCF)(Nc2cccc(SC)n2)CCCC(F)(F)CC1 38560,C(=O)(CC(=O)NCCCC(C)NC(c1[nH]nnc1Br)=O)NCC#C 38561,N1(C(c2ccc(C#C)o2)=O)CC2CCC1CC2NC(c1cc(C(N)=O)[nH]n1)=O 38562,C1(CNC(Cc2cc(C)nn2C)=O)CCCCCN1C(C1CCC(C)(C)CC1)=O 38563,c1(C(N2CCC(F)(C(=O)NCCOCCF)C2)=O)ccnnc1O 38564,c1(NCC)ccc(CN(C(C(=O)NC)C2CC2(Br)Br)CCC2CCOCC2)cc1 38565,CC1CCN(C(C2CCCCC2O)=O)CC1CNC(C1(c2cccs2)CC1)=O 38566,C1(NC(C2(CC=C)CCC2)=O)CC2(CCCN(C(=O)C=C(C)C(C)(C)C)C2)C1 38567,C1(C(N2CC(C(CC)CC)C2)=O)(NC(c2ccn(CCF)n2)=O)CCSC1 38568,Cc1ccc2c(c1)C(C(=O)N1C3CCC1(CNC(C1CC1F)=O)CC3)CC2 38569,C1(C(N(CCOC)CCNC(=O)C=CC2CCC2)=O)CC(C2CCCC2)C1 38570,C1(C(N(CCCNC(c2ncoc2C2CC2)=O)C2CC2)=O)CCCC(O)C1 38571,C(=O)(CCS(C)(=O)=O)NCC1(C(=O)NC2CCCC(C)C2C)CC(=C)C1 38572,N1(C(CC(C)CNC(=O)C=Cc2cc[nH]c2)=O)CCC2CN(C)CC2C1 38573,N1(C(c2n(C(C)C)ncc2)=O)CCCOC(CNC(=O)CC2CC3CCC2C3)C1 38574,C1(C(N2C(C3CCN(C(C4CCCN4C4CC4)=O)C3)CCC2)=O)CC(=O)N(O)C1 38575,c1(C(=O)OC)n[nH]c2cc(-c3cncn3C)ccc12.N12CCC(CF)(CC1)C2=O 38576,CC1(C)NC(=O)C2(CCN(C(=O)NCCc3cc(-c4ccccc4)no3)CC2)O1 38577,C(=O)(CCC(C)CN(C)C)N1CCC(O)(C(C)NC(C(CC=C)C)=O)C1 38578,N1(C(CCOCC(C)C)=O)CCC(C)N(C(c2cc3c(s2)CCOC3)=O)CC1 38579,CC1(c2cn(CCCCCC3CC3)nn2)CCCC(F)(F)C1 38580,c1(COC)ccc(NC(N2CCN(C(C3(Cn4cccn4)CC3)=O)CC2)=O)cc1 38581,n1(CC)cc(NC(=O)C(C)(C2CCC2)NC(c2cncc(C#N)c2)=O)ccc1=O 38582,C(C(=O)NNC(=O)N(C)CCCC=CCN)=C(C)C.c1(O)cccnc1F 38583,Cn1ncc(C(=O)NC(CNC(c2csc(=N)[nH]2)=O)C2CCC2)c1S(N)(=O)=O 38584,c1(OC)cccc(C)c1C(N1CC2C(C(N3CCC(C#N)C3)=O)C2C1)=O 38585,Cc1c(Cl)ccc(C(N2CCC23CN(C(=O)Cn2cnnc2)C3)=O)c1Cl 38586,C(=O)(CCC(C)(C)[N+](=O)[O-])NCC(C)CNC(=O)CSCc1ccccn1 38587,O=C1Nc2ccc(C(N3CC4(C3)CN(C(=O)CC3CCC3C3CC3)C4)=O)cc2CO1 38588,N1(C(C(CC)OC)=O)CCN(C(=O)C(O)Cc2[nH]cnc2C)C(CCO)C1 38589,C1(C(=O)NCCC)(CC)CCC(c2nnnn2C(C)CC)(OC)CC1 38590,C(CCCCC(=O)N1CCC(C)(C)C1C(=O)N(C)C(C)C)SC.C1(C)CO1 38591,CCC(O)C(F)(F)C(=O)N1CCC(NC(c2coc(C(C)(C)C)n2)=O)CC(O)C1 38592,N1(C(C(n2ccc(C)n2)C)=O)CC(C)(C)OCC1CNC(C12CCC(C1)C2)=O 38593,Cc1ncc2ccc(C(N3CCC(NC(c4csc(C5CC5)n4)=O)C3)=O)cn12 38594,C1(SCC)COCCN(C(=O)COCn2nnc(C(=O)Nc3ccsn3)c2N)C1 38595,CCCC(C(=O)Nc1cnccc1NC(C)C)NC(=O)OC(C)(C)C 38596,N1(C(=O)Cn2ncccc2=O)CC2CCN(C(=O)CCc3ccncc3)C2C1 38597,C1(C(=O)NC(CC)CN(C(=O)CCCOCCOC)C)OCCC1(C)C 38598,n1(CCN(CC)Cc2coc(C(C)C)n2)cc(CN(C)C(C)=O)nn1 38599,c1(C2(C(=O)NCCC(C)(C)N(C)C(C3COCCO3)=O)CCC2)c(F)cccc1F 38600,CCC(CCCC(=O)NCC(C1CCC1CO)=O)NC(=O)Cn1ccc(=O)cc1 38601,c1(CSc2scc(CN3CC(C(=O)OC(C)C)C3C(=O)O)n2)nnc2n1CCC2 38602,C1(COC)(N)CN(C(=O)C(C)=C2CC2)C1.C1(=O)CC1=O.C(C=CCO)N 38603,c1(C(=O)NCC2C(CNC(Cn3c(C)nnn3)=O)C2)ccc(NC=O)cc1 38604,C(=O)(CCCS(C)(=O)=O)NCC(C)NC(c1ccc(F)c(N2CC(C)(C)C2=O)c1)=O 38605,Cc1noc(C)c1C(=O)NCCC(C)NC(=O)C(C)OCC1CCCCO1 38606,N1(C(Cn2nnc(C)n2)=O)CCC2(CCCCC2NC(C2CCC(=O)N2C)=O)C1 38607,O=C(NN1CCCC1C(N1CC2(C=CCO2)C1)=O)C(C)C 38608,C1(NC(c2ccnc3[nH]nnc23)=O)CC2(CCN(C(=O)C=CBr)C2)C1 38609,C(=O)(CC(C)CC(C)(C)C)N(C1CC(OCC(=O)N(C(C)C)C2CC2)C1)C1CCCC1 38610,N1(CC(=O)NCc2onc(COC(C)C)n2)CC2C=CC1C2.N1(C)CC1 38611,Cc1ccc(F)cc1CC(=O)NCC1(C)CCCN(C(C2C3(CC3)C23CC3)=O)C1 38612,c1(CC)ccc(C(N2CC(NC(c3ccc(CN(C)C)[nH]3)=O)CC2C)=O)cn1 38613,C1(CCOC)(NC(=O)Cn2nnc(F)c2C)CCN(C(=O)C=CSC)CC1 38614,c1(CNC(=O)CN2CCCC2C)nc(C)c(C(=O)NCCCC(C)(C)OC)s1 38615,c1(C(N2CC(C)(CC(N3CC4CCCC4C3)=O)C2)=O)ccc2c(n1)NC(=O)CC2 38616,c1(C(C)NC(C2CC(CNC(c3occc3C3CC3)=O)C2)=O)cccc(C#N)c1 38617,CCC(O)(CC(=O)N1CC(NC(=O)Cc2ccc(Cl)cc2C)C1)c1ccccc1 38618,C(CC(CNC(=O)COC1CC=CC1)NC(C1CCCN1C(C)C)=O)OC 38619,C(=O)(C(C)C(O)CC)NCCN(CCC)C(c1cc(C2CC2)[nH]n1)=O 38620,C1(C(NC=C(C)C)=O)CC2CCC1N(C(=O)Nc1cc3cc[nH]c3cn1)C2 38621,C1(CC(=O)NCC2(F)CC(NC(Cn3ncc(C)c3)=O)C2)CCCC(C)C1 38622,C(=O)(C(F)(F)C(C)(C)O)NCC12OCC(CNC(C(C)NC(CC)=O)=O)(C1)C2 38623,C1(CNC(COC2CCN(C(C3C(OCC)C3)=O)C2)=O)CCC(C)CC1 38624,C1(C#N)(C(=O)NC(CC)CNC(C2CC(=O)N2)=O)CC12CCCC2 38625,C1(NC(c2c(C)n(C)cc2)=O)CC2CC1N(C(c1nc(Cl)sc1Cl)=O)C2 38626,CC1CCC(NC(=O)CCC2CC2)CN1C(c1cc(-c2ccccc2)[nH]n1)=O 38627,c1(C(=O)NCCCCNC(C2C(C#N)C2)=O)cccc2sncc12 38628,c1(C(=O)NC2CCN(C(C(c3cscn3)N(C)C)=O)C2)cn(C)c(=O)cn1 38629,n1(C(C(=O)NC(CC)CNC(c2cnccc2C)=O)C)cnc2ccccc12 38630,Cc1nc2cc(C(=O)NC(CNC(C3CCCC(=O)N3C)=O)C(C)C)cnc2[nH]1 38631,C1(C(=O)NCc2c(C)occ2)CCC(C(C)C)N1C(C1CCCCCC1)=O 38632,CC1CC(C(=O)NC2CC(CCNC(=O)CN3CC=CC3)C2)CCC1=O 38633,Cc1ccc(C=CC(=O)NCC2(CNC(C3CCS(=O)CC3)=O)CCC2)cc1C 38634,CCCC(C)CC(=O)N1CCC(C(C)CNC(C2(CF)CC2)=O)CC1 38635,c1(C(N2CC(NC(C3(SC)CCC3)=O)C(C)C2)=O)ccc(F)c(SC)c1 38636,C(=O)(CC(F)F)NCCC1CC(NC(C2C(CC)C2)=O)C1 38637,N1(C(C(CC)C)=O)CC2(CC(NC(=O)C(=O)Nc3c(C)cccc3C)C2)C1 38638,c1(NCC(CC(=O)NC)O)nc(N2CCOC(C3CC3)CC2)cc(C)n1 38639,c1(C(c2ccccc2)CNC(c2ccc(C(=O)O)nc2)=O)cc(Cl)cc(Cl)c1 38640,c1(CNC(C(C2CCCN(C(C3CCN(C)C3)=O)C2)C)=O)cc(F)ccc1F 38641,C(=O)(C1=CCCCC1C)NCC1N(C)CCN(C(c2cc(C)on2)=O)C1 38642,C1(NC(C(COCC)OC2COC2)=O)(COC)CCN(C(=O)CCOC)CC1 38643,C1(C(=O)NC(CCN(CC)CC)C)COCCC1NC(C1CN(C)CCO1)=O 38644,C1(C(=O)NOCc2nc[nH]n2)CCOCCN1C(=O)C=Cc1nccs1 38645,c1(CNC(c2n(C(CC)C)nnn2)c2cc(C(N)=O)no2)ccc(Cl)cc1 38646,C(C(COC)CC(=O)N1CC(n2cc(NC(=O)CC(C)(C)O)nn2)C1)OC 38647,C(CC(F)F)(C(=O)NC1CC2C(C1)C2(F)F)N(C(COc1cc(C)on1)=O)C 38648,c1(C(=O)NCC(CC=C)NC(=O)C=C(C)c2ccco2)cc(C)cc([N+](=O)[O-])c1 38649,Cc1cc(C(N2CCC(C)(CNC(c3ccn(C(C)(C)C)c3)=O)C2)=O)cc(C)c1 38650,c1(OCC(=O)NC(C)C(C)NC(c2ccncc2)=O)ccc(C(F)(F)F)cc1 38651,C1(CCNC(CC(=C)I)=O)CN(C(=O)C(F)(F)F)CC(C)O1 38652,c1(C2(C(N3CCCC3C#N)=O)CC2)cc(NC(c2ccccc2)=O)ccc1OC 38653,c1(C(N2C(C)CC(NC(c3cncc(COC)c3)=O)C2)=O)ccc(N)c(Cl)c1O 38654,c1(N2CC(C(C)NC(=O)CC3CC3C)OCC2)cc(-n2cncn2)ncn1 38655,c1(C(C)=O)ccc(CC)nc1N1CC(CC(C)NC(C2CC(=O)N(C)C2)=O)C1 38656,c1(-c2cc(NCc3c(C)c4c(s3)cccc4)ncc2)ccc2c(c1)OC(C)(C)O2 38657,C1(CC)CN(C(C2CC3CC3C2)=O)CCN1C(C)=O.c12ccnc(Cl)c1NC2=O 38658,C(C(F)(C(=O)NCc1coc(C)n1)C(C)C)NC(C(CC#C)O)=O 38659,c1(CC)cc(CC(=O)NC2CCN(C(=O)Cc3sccc3Br)C2)n(C)n1 38660,Cc1cccc(C2c3cncc(c3)N2)c1.c1(-c2nnnn2C(C)C)cnc(Cl)n1C 38661,C(C(=O)NC1C2CCC1(c1cscn1)C2)(C(C)O)NC(C)=O.C12(CC1)C(=O)N(C)C2 38662,C(=O)(C(C(C)C)NCc1c(C)scc1)NC(c1ccccc1)c1ccccc1 38663,c1(CNC(C2(CC=C)CC2)=O)conc1NC(=O)CC1CCCN1C.C(CCOC)O 38664,Cc1c(C(=O)NC2CC(C)N(C(C34CCC(C3)C4)=O)C2)noc1C1CC1 38665,Cc1c(NC(c2cnn(C)c2)C(=O)OC(C)(C)C)cccc1Cl 38666,N1(C(C2(OC)CCCOC2)=O)CCC(C)N(C(=O)C(=Cc2cn(C)cn2)F)CC1 38667,C1(N(C(C2C(CCC)C2)=O)CCC)CCN(C(C2CC2Br)=O)CC1 38668,N1(C(C(=O)NC(C)CCn2cncn2)=O)CC(F)(CO)C1 38669,C(=O)(C(CCC1CC1)NC(C1CC(CC(C)(C)C)C1)=O)OC(C)(C)C 38670,CN1C(=O)CSC1=CC(=O)NCC(C)(C1CC1)NC(=O)Cc1cnccn1 38671,N1(C(C=CC=CC)=O)CCC2CN(C(c3cc(C4CCCO4)c[nH]3)=O)CC2C1 38672,Cc1cc(C(=O)N(CC(C)CNC(=O)C(C)Cc2ccc(F)cc2)C)ccc1N 38673,N1(C(c2ccc(CC)cc2O)=O)CCC(O)(C2CCN(C(=O)CC(C)O)CC2)C1 38674,C(C(C(=O)N(CC(=O)NC(C)C)C)C(C)C)NC(C1(CC=C)CCC1)=O 38675,Cc1ccc(C(N2CCN(C(=O)CC3=NNC(=O)C3)C3CC23)=O)c(F)c1F 38676,S(=O)(=O)(CCC(=O)NC1CCN(C(=O)C(C)(C2CC2)OC)CC1F)OC 38677,CC1CN(C(=O)CN2CCN(C(C3CC3c3ccco3)=O)CC2)CC(C)(C)O1 38678,Cc1cnc(C(N2CCC(c3nccs3)C2)C(=O)NC(=O)CC(C)(C)C)c(C)c1 38679,c1(C(=O)NC)cn(CC(=O)NCCCC(C)NC(=O)C(C)n2cncn2)nn1 38680,c1(CCC(N2CC(CC(C)NC(c3ccc(C(F)F)s3)=O)C2)=O)ccccc1O 38681,c1(C(CNC(c2nnnn2C(C)C)(C2CCCO2)C)OC)ccc(OCF)cc1 38682,c1(C(=O)NC2CC(NC(c3n(C(C)C)ncc3F)=O)C2)cnc2ccsc2c1 38683,c1(OCCC(C)C)ccc(C(=O)NCC(O)CNC(C2CCCN2C=O)=O)cc1 38684,c1(OC)ccc(C=CC(N2CCC(NC(C3CC34CC4)=O)CC2)=O)cc1Cl 38685,n1(C(C)(C)C)cc(N)c(CN(C(=O)CC2CCC(C(F)(F)F)O2)C2CC2)n1 38686,N1(C(C(COC(C)C)NC(Cc2c(C)nsc2)=O)=O)CCC2(CC2)C1 38687,C(=O)(CC(C)F)C(=O)C(F)C1CC(NC)C1.C=CCCCNCC(=O)OC 38688,c1(CNC2CC(C(C#N)OC)C2)cccc2c1CCC2 38689,c1(C(=O)NC2(CCOC)CCN(C(=O)C(C)=C(C)C)CC2)scc2c1CCCC2 38690,C1(CC=C)OCCC1(c1nnnn1CC(=C)C)NCCSc1ccncc1.C1(C)CC1 38691,c1(C(N2CCN(C(=O)CC(F)F)C3CC23)=O)cc2ncc(Br)cc2o1 38692,Cc1[nH]c(=N)[nH]c(=NCC2CCN(CC(C)C)CC2)c1Cl 38693,N1(C(c2c(C)n(C)nn2)=O)C2CCC(C2)C1C(=O)NC1CC(C(F)(F)F)C1 38694,C(=O)(CCCCC(=O)OC)N1C(CCCNC(C(CC)C(C)O)=O)CCCC1 38695,C1(COC)(CNC(=O)C(C)CF)CN(C(=O)C(C)(C)F)C1 38696,C(=O)(CCC(CF)CF)NC(C(=O)N1CCCC(CC(=O)OCC)C1)CC(C)C 38697,N(C(=NCC1CCCC(F)(F)CC1)N1CCN(c2ccccn2)CC1)CC1C(C)C1 38698,N1(C(c2c(F)ccc(C)c2)=O)CCCN(C(c2nc(C)ncc2Cl)=O)CC1C 38699,c1(C(=O)NCCCC(C)NC(C2CC3CCC2C3)=O)cc2sccc2s1 38700,N1(C(C(C(C)C)O)=O)CCC2CN(C(=O)C(c3cccn3C)=O)C(C)C12 38701,N1(C(C(CC)F)=O)CC(NC(c2ccc(C#N)c(C)c2)=O)CC12CCCC2 38702,CCCS(=O)(=O)C(C)C(=O)NC(C)(C)CN(C(=O)C=Cc1ncco1)C 38703,c1(C(=O)NC2(C(=O)NC(C(CC)C)CN(C)C)CC(F)C2)c[nH]c2ccccc12 38704,CC(c1ccco1)=CC(=O)NC1CCC(NC(=O)CC(F)F)C1 38705,C=C(C)CC(C(=O)NCCn1ccccc1=O)NC(=O)C=CC(C)CC 38706,Cn1ncc(CNC(c2c[nH]c(C#N)c2)=O)c1C(=O)NCCc1cc[nH]n1 38707,c1(CN(C(c2ccoc2C(=O)O)C(=O)NCc2cccs2)C)ccc(C#N)s1 38708,C1(CCOC)(NC(c2ccc(Br)o2)=O)CCN(C(c2cccc(CC#N)c2)=O)C1 38709,c1(C(c2cn(CCCC(=O)O)nn2)N(C(C2CCC(C)O2)=O)C)cc(=O)cc[nH]1 38710,Cc1ncc(Cl)cc1NC(c1c(C)[nH]c(C(=O)NCC2CC(F)(F)C2)c1C)=O 38711,c1(C(N2CCC(CF)C2)C(=O)OC)cccc(S(N)(=O)=O)c1 38712,C=CCCCCCC(=O)NC(C)(CC)CCNC(N1C(CC)COCC1)=O 38713,N1(C(C(C)C)=O)CC2(CCN(C(=O)Cc3ccn(C(C)C)n3)C2)C1 38714,c12ccc(cc1)C(N1CCN(C(=O)C(C)C)CC1)C(=O)N2.C1(COC)CCOC1 38715,N1(C(C(CC)CC)=O)CCC(C2CCN(C(=O)C3CCCc4nncn43)C2)C1 38716,C(c1ccc(F)c(Cl)c1)=CC(N1CCCCC(CNC(C(C)OC)=O)C1)=O 38717,c1(CNC(c2c(SC)csc2)=O)ccc(CNC(=O)Cc2cc(C)cs2)cc1 38718,CSC1=C(C(=O)NC2CCN(CC(O)Cn3cccn3)C2)CCCC1 38719,CC(C)(C)C(C)(O)CNC(=O)CNC(=O)Cc1csnn1 38720,c1(CC)nonc1C(=O)NC(C)(CNC(c1ccnnc1)=O)CO 38721,CC1(C(=O)NC2CCCC2(C)C)C=CCN1C(c1cc(C(F)F)[nH]n1)=O 38722,N1(C(c2ccc(CNC(CC(C)CN(C)C)=O)o2)=O)CC(CO)C(C)(C)C1 38723,c1(OC)c(F)ccc(F)c1C(N1CC(c2ocnc2CNC(=O)CCF)C1)=O 38724,C=CC1(C(N2CCC(C3CCCN3C(c3cc(COC)on3)=O)C2)=O)CCC1 38725,C(=O)(CC1=CSC2=NCCN12)NCC1(NC(C(C)(C)N(C)C)=O)CCOCC1 38726,c1(C(=O)NC(CC(C)NC(=O)C=CC=C(Cl)Cl)C)cc2n(n1)CC1(CC1)C2 38727,Cc1cc(Cl)cc2cc(C(=O)Nc3cnn(-c4ccccc4)n3)[nH]c12 38728,C1(NC(C(C)(CO)OC)=O)CN(C(c2cc(Cl)c(C)cn2)=O)C(C)(C)C1 38729,C1(C(=O)NCC2(CNC(C3CCCCS3)=O)CC23CCC3)CC=CCC1CO 38730,c1(CCSCCC(N)C2CCC2)c(F)cccc1Cl 38731,CC1CC(NC(C2CC3CCC2O3)=O)CN(C(c2cccc(CCO)c2)=O)C1 38732,c1(OC)cccc(C(N2CCC(C(=O)NCC3(Br)CCC3)CC2)=O)c1O 38733,C1(CC)CCCN(C(=O)C(CC2CC2)NC(=O)CCc2ncnn2C)CC1 38734,CC1(C)C2CCC1(C(N1CCC(NC(=O)Cn3cccnc3=O)C(CO)C1)=O)C2 38735,N1(C(C(C)(C)CC2CC2)=O)CCC(NC(=O)CC2CC=CCN2C)C(F)C1 38736,N1(C(c2cncc(CC)c2)=O)CC2CCCC2(NC(=O)Cc2ccn(CC)n2)C1 38737,c1(C(=O)OC)cc(=NCC(O)CNC(C2COC(C)C2)=O)[nH]c(Cl)n1 38738,c1(C(=O)NC(COC)COC)cccnc1NC(c1nccc(C(F)(F)F)n1)C 38739,Cc1cccc2c1CC(C(=O)NC1CCN(C(C3CC(Cl)(Cl)C3)=O)C1)N2 38740,c1(CC)ncccc1C(=O)NC(c1ccccc1)CN(C)C(C1CCC(C)C1)=O 38741,C(c1cncnc1O)=CC(=O)NCC1N(C(C2(C)C(C)(C)C2)=O)CCOC1 38742,c1(OC)ccc(N)c(C(=O)NC2CC(CNC(=O)C(C)C3CCC3)C(O)C2)c1 38743,Cn1c(C(=O)NC2CN(C(C3(C4CC4)CCC3)=O)C2)c(Cl)c2ccccc12 38744,C(=O)(C#CC1CC1)NCC1CC(C(N(CC(C)(C)O)C)=O)C1 38745,O=C1CCC2(CN(Cc3cc(Cl)ccc3Cl)C2)N1 38746,N1(C(c2[nH]ccc(=N)n2)=O)CC2CC1CC2CNC(C1(C(=O)N(C)C)CC1)=O 38747,CCC(C)CCC(=O)N1CCCOC(c2cccs2)C1.C1(=O)C(CC2CCCC2)N1 38748,CC(CC(N)=O)NC(C1C(C)CN1C(c1cnn(C2CC2)c1)=O)=O 38749,CN1CCCCC1CC(N1CCOCC1CCNC(c1ccc(F)cc1)=O)=O 38750,c1(C(=O)Nc2ccc(C(N(C(C)(C)C)CC)=O)nc2)cncc(C#N)c1 38751,CCC(CC)CC(=O)N1CCN(C(C2CCOC(C)C2)=O)CC1 38752,C12(NC(C(C=C)O)=O)COC(CNC(=O)CN3CCCNC3=O)(C1)C2 38753,N1(C(CCOC)=O)CCC2C(CCN2C(c2cnc(F)cc2C)=O)C1 38754,N#Cc1csc(C(=O)NC2(CCNC(C3CCN(C4CCSC4)CC3)=O)CC2)c1 38755,C1(CC=C)(NC(c2cncc(OC)n2)=O)CCCN(C(=O)C(O)P(C)(C)=O)C1 38756,c1(NC(C2C(CC)CN(C(=O)Cn3cccc3)C2)=O)cc(CO)ccc1C 38757,C1(NC(C2C(C=C)OCC2)=O)CC2(CCN(C(=O)C=C(C)COC)C2)C1 38758,N1(C(c2cncs2)=O)CC(NC(C2CC2c2cncc(F)c2)=O)CC(O)C1 38759,C(=O)(C(F)(F)CCn1cccn1)NCC(CNC(c1c(N)nccc1)=O)O 38760,c1(N(C)C)ccc(Br)c(SC(CNC(=O)OC(C)(C)C)C2CC2)c1 38761,c1(CC)ncc(C(=O)NCC2CN(C(=O)Nc3ccccc3Cl)CCO2)cn1 38762,c1(C(C(=O)NC2CCOC2)N(C2COC2)CC)snc(OC)c1F 38763,N1(C(CCNC(C)=O)=O)CCCC2(C1)CN(C(=O)C=C1CCOCC1)C2 38764,C1(F)(CNC(C(CN(C)C)N(C)C)=O)CCC(NC(c2cc[nH]n2)=O)C1 38765,Cc1nn2c(c1CNC(=O)C(O)C1CC1)CN(C(C1CC(=O)NC(=O)C1)=O)CC2 38766,c1(C(=O)OC)cc(C(=O)NCCN(C(C2CCCC2O)=O)C(C)C)cs1 38767,CCC(C(=O)NCCC1(C)CCN(C(=O)COc2ccsn2)CC1)C(F)(F)F 38768,N1(C(C2CN(C(C(CSC)C)=O)CC2F)=O)CCCOCC1C 38769,c1(N2CCC(CC)C2)cc(=NCc2nc(=N)n(C)[nH]2)[nH]c(C(C)C)n1 38770,C1(C(=O)NCC(CC2CC2)C(=O)N2CCC(n3ccnc3)C2)CCCC1C1CC1 38771,N1(C(CSc2nc(C)[nH]n2)=O)CC2CN(C(c3nccn3C)=O)CC2C1 38772,Cc1cc(C(=O)C(N2CCC(NC(c3nc(Cl)oc3C)=O)CC2)=O)ccn1 38773,N1(C(c2c(Cl)cnc(CC)n2)=O)CCC(C2CCN(C(C3CC3F)=O)CC2)C1 38774,N1(c2n(CCC#N)c(NCC3CC3)nn2)CC2CS(=N)(=O)CC2C1 38775,C1(OC)CCCCC1.C12CCC(C1)CC(=O)OCC(=O)NCC(C)N2C(C)=O 38776,C1(C(N(C)CC2(CNC(C3CC(n4ccnn4)C3)=O)CC2)=O)Cc2nccn2C1 38777,c1(NC(c2ncc(-c3cccc(OC)c3C(F)(F)F)nc2)=O)ccc(Br)c(F)c1F 38778,C1(CCC)CN(C(c2cccc(OC3CC3)c2)=O)CCN1C(=O)C(F)=C(C)C 38779,N1(C(C2(C)C(C)C2)=O)CC2CCN(C(=O)CCc3ccc(C(F)(F)F)cc3)C2C1 38780,C1(NC(c2c(C)cc(N)cn2)=O)CC2CCC1C(NC(C1CN(C)CCO1)=O)C2 38781,c1(C(=O)NCC(CC)NC(C2CCCN2N=O)=O)cc(C)n(NC(N)=O)c1C 38782,C1(O)(CC(=O)NCCOCCCNC(CC2C(=O)NC(=N)S2)=O)CCCCCC1 38783,C12CN(C(C)(C)C1)C(=O)CONC2=O.c1(OC)cnn(C)c1 38784,c1(C(N2CC=CC(NC(C3C(C)COCC3)=O)C2)=O)ccc2cc[nH]c2n1 38785,C1(NC(c2c(OC)cncc2)=O)CCC(C)N(C(C2(OC(C)=O)CC2)=O)C1 38786,CC1=CC(Cn2cc(C34CC(CN3C(c3cnoc3)=O)C4)nn2)=C(C)S1=O 38787,C1(C(=O)NC(CC=CC)C(=O)NCC2(CCC)CC2)CCC2CC1CO2 38788,C(=O)(N=c1ccn(-c2ccc(F)cn2)[nH]1)CC(C)C.C1CC1 38789,Cc1cc(C(N2CCN(C(C34CSC(C3)C4)=O)CC2)=O)c(N)c(F)c1 38790,C1(C(=O)NC2CCN(C(C3CCN(C4COC4)C3)=O)C2)CCCCC12CCC2 38791,n1(CC(N2CCN(C(c3c(C)cno3)=O)CC2CCO)=O)ncc2ncccc12 38792,Cc1ncc2n1CCC(C(=O)NCCNC(=O)Cc1cncc(F)c1)C2 38793,C1(O)(CNC(C(C(C)C)C)=O)CCCN(C(C2CCC3CC2CO3)=O)C1 38794,N1(C(CCC(=O)OC)=O)CC2(CC(NC(C3CCSC(C)C3)=O)CO2)C1 38795,O=S(=O)(c1ccc(Br)cc1Cl)NC(c1ccc(F)cc1)CN1CCC1 38796,c1(C(N2CCC(NC(Cn3ccc(C)n3)=O)C2)=O)ccc(C(=O)O)c(C)c1 38797,N1(C(C=C(C)Cl)=O)CCC2(CC1)CN(C(=O)Cc1cnn(C)c1)CC2CO 38798,C1(CC(N2C(C(C)NC(C=CC(C)C)=O)CCC2)=O)CC=CCN1C 38799,C1(NC(c2nn[nH]c2Cl)=O)CC2(CCN(C(=O)Cn3cccc3)C2)C1 38800,C(=O)(C1=CC2(CCOC2)C1)N(C1CCN(C(c2ccoc2)=O)C1)C 38801,CCCC(C)(O)C(=O)NCC1CN(C(=O)C(F)(F)COC)CC1(F)CO 38802,N1(C(CC2ON=C(C)C2)=O)CCCCC1C(N1CCN(C(=O)C(C)C)CC1)=O 38803,C1(C)(C(N(CCNC(c2ccc(C(C)=O)nn2)=O)CC)=O)CC(C)OC(C)C1 38804,c1(C(=O)NCC2N(C(=O)COCC(F)F)CCC2(C)C)cnc2n1CCOC2 38805,c1(OCCc2nc(-c3ccnn(C)c3=O)on2)nc(F)ccc1Br 38806,C#CCCC(O)C(=O)NCc1ccccc1-n1cc(C2CC2C(=O)O)nn1 38807,N1(C(C=CCCC)=O)CCCC(O)(CCNC(=O)C(O)C(C)CC)C1 38808,C(C)(C(C)NC(c1ncoc1CNC(=O)C=Cc1cocn1)=O)(C1CC1)OC 38809,c1(CC)nn(C)cc1C(=O)NC(C1CCCN(C(=O)C(C)OC)C1)C 38810,C1(C(=O)NC(C(=O)OCC)(C)C)CC2C=CC1N(C(=O)CC1(CC)CCC1)C2 38811,C1(NC(C(=O)NCC2CC2)=O)CN(C(C2CC2(Cl)Cl)=O)CCC1C(F)(F)F 38812,CCC(C#N)C(=O)NC1CCCC(CNC(c2ccc(OCC(C)C)nc2)=O)C1 38813,Cc1cn2c(n1)CC(C(=O)NC1CCN(C(c3cnn(C)n3)=O)CC1O)C2 38814,C1(C2CCC2)(C(=O)NCC2CCCCN(C(CCC=C)=O)C2)CC1(F)F 38815,C1(C)(CNC(C2N(C(COC(CC)CC)=O)C(C)CC2)=O)CCC(=O)NC1 38816,n1(CCC)cc(C(=O)NC2CCCC2CNC(c2ccc(NC)cc2)=O)c(C)n1 38817,N1(C(=O)NCc2n(C(C)C)nc(C3CC3)c2)CC(C)CCC1C1CCCCC1 38818,c1(C(N2CC(O)(CCNC(C3CC3(F)Cl)=O)C2)=O)ccc(SC(F)(F)F)nc1 38819,C1(C(N2C(C(NOCC=CC)=O)CC(O)C2)=O)CC2C(C1)C2(C)C 38820,N1(c2snc(C)n2)CC2CC(NC(C3(Br)CC3)=O)C2C1 38821,N1(C(C2(C)CC(C)(C)C2)=O)CCC(C2(NC(C3(C4CCC4)CC3(F)F)=O)CC2)C1 38822,c1(C(N(CC(CC)NC(=O)CSC2CC2)C)=O)cccc2oncc12 38823,O=C1CCCc2cc(C(N3CC(NC(c4cc(F)c(I)c(F)c4)=O)C3)=O)ccc21 38824,c1(C(=O)NC(c2ccc(Cl)cc2)CC(=O)OC)ccc(S(C)(=O)=O)c(F)c1 38825,c1(C(N2CCCC(CN(C)C(c3nncs3)=O)C2)=O)ccc2nn[nH]c2c1 38826,C1(NC(c2ncc(CC)s2)=O)CC2CCC(C1)N2C(C1(O)CCC1)=O 38827,S(=O)(=O)(c1cccnc1NCc1ccc(C)s1)NC(CC)CS(C)(=O)=O 38828,CCCC(CC(=O)NCC1CCC(C)CC1)NC(c1sc(C)nc1C)=O 38829,C1(C)(CNC(c2c(C)cns2)=O)CCCN(C(c2ccc(C(C)C)cc2F)=O)C1 38830,c1(C(=O)NCC(C)(C2CCC2)NC(CS(=O)(=O)NC)=O)cccc(C#CCO)c1 38831,C=C(C)C(C)(C)C(=O)NC(C1CCN(C(C2CSC3(C)CCC(=O)N23)=O)CC1)C 38832,C1(CC)CCN(C(=O)C(OC)SC)C(C(=O)N(C)CC2(O)CCC2)C1 38833,Cc1ccc(-n2ncc(C(=O)N(C)C(c3cccnc3)C3CC3)n2)cc1 38834,N1(C(C(CC2CCC2)NC(C2CCO2)=O)=O)CCCCC1CCO 38835,N1(c2n(C)nc(Cl)c2)CCC2(CC1)CC2C(=O)NC1(c2ccccn2)CC1 38836,C(C)(C)(C(C)CC(=O)N(C)C(c1nccs1)C)NC(C(C)SCCCC)=O 38837,C1(NC(c2[nH]cc3c2CCCC3)=O)C2CCCC1CC(C(=O)O)C2 38838,C(=O)(CC(C)F)N(CCCNC(C1C(=C)C1)=O)CC1CCCC1 38839,C1(NC(c2ccc(C#C)cn2)=O)C2CCCN(C(=O)CC(F)(F)F)C2C1(C)C 38840,C1(C(=O)NCC(C2CCCC2)NC(C(C2CCC2)OCC)=O)CCC(C)(C)CC1 38841,C(=O)(n1cnc2cccnc12)N1CCN(C)C(C(F)(F)C(F)(F)F)C1 38842,C(=O)(CCCC(CC)CC)N1CCN(C(C(COCC)C)=O)C(C)C1 38843,C(=O)(C1=CCN(C(=O)CC(C)(C)COC)CC1)N1CCCC(CC=CC)C1 38844,c1(C(N(CCCN(C)C(C2CCCC(O)C2)=O)C)=O)nccc2[nH]ccc12 38845,C(C)(C(C(=O)NCC(n1cccn1)C)C(C)C)NC(Cn1c(C)ncc1)=O 38846,C(=O)(CC(C)(C)N(C)C)N(CCCCN(C(C(C)c1cc[nH]n1)=O)C)C 38847,N1(C(Cn2cc(C(=O)OC)nn2)=O)CC(NC(=O)C=CS(C)=O)C(F)C1 38848,CC1CCC(C(=O)NCCCN(C(C2(C#N)CC2)=O)Cc2cccnc2)O1 38849,c1(C(=O)NCC(CNC(c2ccn(C)n2)=O)OC)ccc(C(C)C)c(F)c1 38850,N1(C(CN2CCCC(C)(CC(=O)OC)C2)=O)CC2COCC(C1)C2C#N 38851,c1(CC(=O)Nc2cccnc2-c2cccc(Br)c2)ccc(Cl)cn1.C12CN(C1)C2=O 38852,c1(C(=O)NCc2cn(CC3(CCO)CC3)nn2)onc2ccccc12 38853,N1(C(c2cc(CC)on2)=O)Cc2cccn2CC(C(N2CCC23CCCC3)=O)C1 38854,c1(OC(CC)C)cc(C(N2CCCC(CNC(=O)CC3CCC(=O)O3)C2)=O)ccn1 38855,CCC(F)(F)CC(=O)N1CCC(F)CC1C(N1CCC(C(C)(C)O)C1)=O 38856,C1(NCCC(=O)Nc2c(OC)cc(-n3cncn3)cc2)CCN2CCCCC12 38857,N1(C(=O)NCc2c(C(=O)OC)scc2)CCCOC(CC(=O)C(C)CC(N)=O)C1 38858,C(C)(C)(CCCCC(=O)NCCC1CN(C(C2CCO2)=O)C1)OC 38859,CC(C)(CS(C)(=O)=O)C(=O)NCCC1CSCCN1C(=O)CN1CCCC1 38860,C(C(C)(C)C(=O)NCCC1CCC(C)O1)NC(C=CCCC)=O 38861,CC(C)(CCF)C(=O)NC1C=CCN(C(c2cc(CCO)on2)=O)C1 38862,C1(CNC(C(C)=CC(=O)NCCO)=O)CCCC1C(N1CC=CC1)=O 38863,N1(C(C23C(C)(C)OCC2C3)=O)CCCC2(C1)CN(C(c1ncc(F)cc1F)=O)C2 38864,c1(N(C(C)C)C)ccc(C(N2CC3CC2C3CNC(c2ccc[nH]2)=O)=O)cc1 38865,c1(N2CCC(CNCC3(C)CC=CCC3)C2)ccccc1C#N 38866,c1(C(N2CC3C(NC(C=Cc4n(CC)ccn4)=O)(C3)C2)=O)cc2[nH]ccc2s1 38867,c1(OC)ccc2[nH]c(=NCc3nn(C)nc3Br)[nH]c(=NC3CCCC3C3CC3)c2c1 38868,c1(C(C)C(N2CCC(N(C)C(C3(C)CCCO3)=O)CC2)=O)ccc(Cl)c(Cl)c1 38869,c1(C(=O)NC2C(C)C(F)(F)C2)cc(C#N)ccc1N 38870,C#Cc1ccc(OCC(=O)NCCC2(NC(C3CCN(C)S3(=O)=O)=O)CC2)cc1 38871,c1(C(=O)NCC(C(C)C(C)C)NC(C(C)=C2CC2)=O)cc(=O)c2ccccc2[nH]1 38872,c1(C(=O)NC2C=CC(CNC(C(C)(C3CC3)OC)=O)C2)nc(Cl)oc1C 38873,N1(C(c2n(C=C)ncc2)=O)CCOCC(C)(CNC(c2ccc(C)cc2CC)=O)C1 38874,CCCC(CCC)=CC(=O)NC(C)CC(C)NC(=O)CCc1nccn1C 38875,c1(CN(c2nnc(C(CC)(C)C)s2)C=O)ccc2nc(O)n(C3CCCC3)c2c1 38876,c12cc(co1)C(=O)NC2.C1(OC)(CNC(C2CC2C(=O)OC)=O)CCCC1 38877,C1(NC(CC(CC)C)=O)CC12CCN(C(c1cc([N+](=O)[O-])c[nH]1)=O)CC2 38878,N#Cc1c(NCC2CCN(C(c3coc(C(F)F)c3)=O)C2)cccc1F 38879,c1(CN2CCC(CC(=O)NC3CCCC(CC)C3)C2)cc(C(=O)OC)ccc1O 38880,C(=O)(C(C(C)(C)C)N(C)C)NCC1C(CC(=O)NC(C)CN2CCCC2)C1 38881,C12(C)CCN1C(=O)COCC(C)NC(=O)C2.C(CCN=[N+]=[N-])OCC1CC1 38882,Cc1cnc(Cl)c(CNc2cnc(F)cc2C(=O)NCc2nccn2C)c1 38883,C1(COCCOC)CCN(C(=O)CNC(C2CC2C)=O)C(C)C1.C1C(=O)N1 38884,C(=O)(CS(C)(=O)=O)NCC1(NC(C)C(C)n2cccn2)CC(=C)C1 38885,N1(C(c2n(CCC)ccc2)=O)CCCN(C(=O)C(F)CC2CCCCC2)CC1 38886,n1(CC(=O)NC(CC(C)NC(COCc2cc(C)on2)=O)C)nc(C)c(O)c1C 38887,c1(C(c2cccs2)NC(C2(C(C)C)CC2)C)nnnn1C1COC1 38888,c1(C(C=CC)=O)ccc(Oc2cncc(C=Cc3cc(O)n[nH]3)c2)c([N+](=O)[O-])c1 38889,C(=O)(CCC(=O)NCC1C2CN(C(C3CCC(F)CC3)=O)CC12)NC 38890,C1(CN(C(=O)C2=CCC2)C)CCCCN1C(c1c[nH]c(-c2ccc(F)cc2)c1)=O 38891,c1(C(N2C(C(=O)NC3CCOC(C4CC4)C3)CC2)=O)ccnc(S)c1 38892,c1(C(=O)NC(CNC(c2nc(OCC)sn2)=O)(C)C)ccc(OC)c2ccsc12 38893,c1(C(C)C(=O)N2CC(CCNC(=O)C(C)C(F)(F)F)C2)cccc(C#N)c1 38894,C1(C(=O)NCC(C(C)(C)C)NC(c2cc(OC)nn2C)=O)CCCCC1C1CC1 38895,N1(C(CCCC2C(C)C2)=O)CCC(C2CC2)C1C(N1CC(C#N)C1)=O 38896,c1(CC(=O)NCCCNC(c2c(C)n(C3CC3)nc2)=O)cn2cccc(C)c2n1 38897,N1(C(=O)NC(c2ccn(CC(C)C)n2)C)CC2CCC2(C)C1 38898,C(=O)(C(=O)N=c1cc(C)[nH][nH]1)Nc1c(OC)ccc(CC)c1 38899,C(C)(N=c1nc2c(ncn2C)c(NCC(C)(C)c2cccs2)[nH]1)C1C(C)C1 38900,c1(C(=O)NC2(C)N(c3nc(OC)c(F)cn3)CCC2)cc(O)ccc1[N+](=O)[O-] 38901,c1(C(=O)NC2CCN(C(c3c(C)nc(COC)s3)=O)CC2)cc2n(n1)CCOC2 38902,C(CCC(=O)N1C(CNC(c2ccc(Cl)[nH]2)=O)CC2CC12)(c1ccccc1)OC 38903,c1(C(=O)NCC=CCNC(=O)CC2CCCC2(F)F)ccc(C(F)(F)F)nc1O 38904,c1(C(=O)NCC(=C)CCNC(=O)C(c2ccccc2)NC(C)=O)ccc(C)c(O)c1 38905,C(=O)(C(C)(C)CCCO)NCC1CC2CN(C(c3cn(CC=C)nc3)=O)CC21 38906,C1(C(=O)NCc2c(C)noc2)CN(C(=O)CCC(=O)C2CC2)CC12CC2 38907,C(=O)(C1=CC2CCC=CCCC12)NCC1C(C)CCN(C(C2(O)COC2)=O)C1 38908,CCC(CC)C(=O)N1CCCCC1C(=O)N(CCN1CCCC1=O)CC 38909,C(C(=O)NC1CCN(C(c2c(Cl)cnn2C)=O)C1)(C(C)(C)C)OC 38910,Cc1ccnc(C)c1NC(C12CCC1CN(C(=O)Cc1c(C)nn(C)c1C)C2)=O 38911,C1(C(=O)NCCc2cnn[nH]2)(NC(=O)C(c2ccccc2)F)CCOCC1 38912,CC1CN(C(C2CCS(=O)(=O)N2)=O)CCN1C(c1cccnc1-c1ccco1)=O 38913,c1(CC(=O)NC(CNC(=O)C=CC2CCC2)C2CCC2)nc([N+](=O)[O-])n[nH]1 38914,C1(=O)CCCCCCCN1.C1(OC)CC(NC(=O)Cn2cc(CO)nn2)C1(C)C 38915,N1(C(C2=CC=C(CNC(C)=O)S2(CC)c2cnn(C)c2)=O)CC2CC1CCC2O 38916,CC(C)CN=C(NCc1nnnn1C(C)C)NCc1ccn(C)c1 38917,Cc1cnc(C(N2CC3C(C(=O)NCC(C)C(C)(F)F)C3C2)=O)c(C)c1 38918,Cc1scc(C(N2CC(NC(C3(n4cccn4)CCC3)=O)C(O)C2)=O)c1N 38919,c1(CNC(=O)N)ccc(C2CC2)cc1.C1(SCCC)CC(C)C1 38920,C1(C(N(C)CC2CCN(CC)C2)=O)CC2CCC1N2C(C1COC(=O)N1C)=O 38921,CC(C)C(C(=O)N1CC2CC1(CNC(C1CCC1)=O)C2)NC(=O)OC(C)(C)C 38922,C1(NC(C(CCC)OC)=O)CC2CN(C(c3cn(C)c(=O)n3C)=O)CC2C1 38923,Cc1cnc(C#N)c(-c2cn(-c3c(OCC(C)O)cccc3F)nn2)c1 38924,CC1C(NC(C2COCCN2C)=O)CCCN1C(c1[nH]ncc1C#N)=O 38925,N1(C(C2(CC#C)CC2)=O)CCN(C2CCCN(C(c3c[nH]ccc3=O)=O)C2)CC1 38926,CC1(C(=O)NCC2CN(C(=O)Cn3cc(C(F)(F)F)cn3)CC2O)CC=CCO1 38927,c1(C(C)C)ccc(C(=O)NCC2CCN2C(=O)CCN2CCCC2)cc1 38928,C1(C)(C(=O)NCC(c2nccc(C)c2)(F)F)CC(C2CC2)=NO1 38929,c1(SC)ncccc1NC(=O)CCC1CCCN(C)C1 38930,C1(NC(C=CCCC)=O)CCN(C(C(=O)NCCC#N)C2CCC2C(=O)OC)C1 38931,c1(C(=O)NCC2(C)CCN(C(C3CCC3(F)F)=O)C2)c(F)ccc(Cl)c1N 38932,c1(C(=O)NCCCN(C(C(C)SC)=O)CC2CC2)cc(O)c2[nH]c(C)nc2c1 38933,C1(O)(c2ccccc2)CCCN(C(=O)C=CCOC(C2(C(N)=O)CCC2)=O)C1.C=O 38934,c1(C(C(N2CCC(C(F)F)(CNC(C)=O)C2)=O)C)ccccc1S(N)(=O)=O 38935,C1(NC(CCCC(=O)OC)=O)C2CC(CN(C(=O)CC3CCCO3)C2)C1CO 38936,C1(NC(C2(CC)CC2(F)F)=O)CCCCC1CNC(=O)Cc1cn(C)c(C)n1 38937,c1(CNC(c2cnc(C)[nH]2)=O)cc2n(n1)CCN(C(C13CCCN1CCC3)=O)C2 38938,N1(C(C2C=C(C)CS2)=O)C2CCC1CC(C(=O)NC(C)C(C)F)C2 38939,C1(CNC(C2ON=C(CC)C2)=O)CC2CCC1N2C(c1cc(C)ccc1C)=O 38940,N1(C(c2ncn(CC)c2)=O)CCC2(CCN(C(=O)Cc3cnn(C(C)C)c3)C2)C1 38941,C1(OC(C)C(=O)NCC(C)(C)CNC(=O)COCCO)CCCCCC1 38942,c1(C(N2CCC(NC(c3c(C)onc3C3CC3)=O)C2C)=O)ccc([N+](=O)[O-])[nH]1 38943,C1(C(=O)NCC(C)(CO)NC(c2c(C(F)(F)F)ncn2O)=O)CC(=O)OC1(C)C 38944,c1(C(C)N(C)C)cn(CCN2CCC(c3ccco3)C2)nn1 38945,C1(C(N2C(C)CC(NC(c3snc(Cl)c3Cl)=O)CC2)=O)Cc2nccnc2C1 38946,CC1=NNC(=O)C1CC(N1CCCCC1CNC(C1(c2ncco2)CC1)=O)=O 38947,CS(=O)(=O)c1ccnc(N2CC3CC(NC(c4cnc5[nH]cncc4-5)=O)C3C2)n1 38948,C(=O)(CC(CC=C)NC(=O)C=C(C)COC)NC1CCC(C#C)C1 38949,CC1CCN(C(=O)C(=O)NCC2CCCN(C(=O)CC3CCCOC3)C2)CC1 38950,c1(-c2n(-c3c(C)cccc3)nc(CCCCOC(C)(C)C)n2)n[nH]c2c1CCC2 38951,n1(CC2(O)CN(C(N3CC(OC)C(OC(C)(C)C)C3)=O)C2)ccc([N+](=O)[O-])n1 38952,c1(C(N(CC)CC)=O)cccc(CNC(C2CC=CCO2)=O)c1 38953,C(=O)(CCS(=O)(=O)N(C)C)NCCOC1CN(C(c2ccc(OC)o2)=O)C1 38954,C1(C(=O)NC(COC)CC(=O)NC2CCN(C3CC3)C2=O)CC2CC1CC2O 38955,C1(CNC(Cn2c(C)cc(C)n2)=O)(NC(C2CCOC2)=O)CC2CCC1CC2 38956,Cn1cc2c(C(=O)NC3CCCC3C(=O)NCCC3=CCOCC3)cccc2n1 38957,CC(C)CC(CC(C)C)NC(=O)CCCC(C)NC(=O)Cc1ccc[nH]1 38958,C12(CNC(C3(C)CCCC3(F)F)=O)CC(NC(C3CC3F)=O)(C1)C(C)(C)O2 38959,Cc1cc(C(N2CC(CC(F)C(=O)NC3COCC3CO)C2)=O)sn1 38960,c1(C(=O)NCC2C(C)CCN(C(COC)=O)C2)cc(=O)c2cc(OC)ccc2[nH]1 38961,c1(C(=O)NCC2C(NC(CCC#C)=O)CCC2)ccnc(C(=O)OCC)c1 38962,c1(CSCC(C(C)(C)C)OC)nc2ccccc2o1 38963,C1(C(N(CC(CO)(CO)NC(CCC#C)=O)C)=O)CNC(=O)CC12CCC2 38964,N1(CCC(=O)NCC(CC)(C)NC(c2cnc(C(C)O)s2)=O)CCCCC1=O 38965,C12(CNC(C(CCCC)O)=O)CCCC1CN(C(=O)CCC1CC(C)(C)CO1)C2 38966,C1(N(C(C=CC(=O)NC(CN(C)C)(C)CO)=O)C)CCCN(C(=O)N(C)C)C1 38967,C1(C(=O)OC)CS(=O)(=O)CCN1C(C1CC=CCC1c1ccccc1)=O 38968,Cc1cnc(N)c(C(=O)NCC2CCC(NC(c3nc(Cl)sc3C(C)C)=O)C2)c1 38969,N1(C(c2nocc2C(=O)NC)C)CCN(C)CC1.c1(C(=O)N)cc(CO)[nH]n1 38970,C1(COC)CC1C1CCCC1.c12ccc(N)c(c1)CC1N(CCC1)C2 38971,Cc1cccc(C2CC2C(=O)NC(C)(C)CNC(c2ncccc2N)=O)c1Br 38972,Cc1nc(C)c(C(=O)N(CCC(C)(C)C)C2CC2)s1 38973,c1(C(=O)NC(COC)C)nc(CNC(=O)C(c2cc(OC)no2)C)oc1C 38974,C1(C(C2(C)CN(C(=O)C=Cc3cnc(C(C)(C)C)s3)C2)=O)CCC(N=[N+]=[N-])C1 38975,S(=O)(=O)(c1cccc(Br)c1)NCC(=O)OCc1c(F)ccc(Cl)c1F 38976,CC1C(NC(=O)C=CC=C(Cl)Cl)C(C)CCN1C(C1CC12CC2)=O 38977,Cc1nc2ccc(-c3cncc(NS(C)(=O)=O)c3)cc2n1C 38978,N1(C(c2nc(C)[nH]n2)=O)CCC2CCC(C1)N2C(C1CC2(CSC2)C1)=O 38979,c1(C(N2CC(CCC)N(C(=O)CCSC3CCCC3)CC2)=O)cc(O)cc(C#N)c1 38980,Cc1ccncc1C(=O)NC1(CCCC(=O)NCC2(C)CC(C)(C)C2)CCC1 38981,N1(C(CCOCC)=O)CC2C(CN(C)C(C3(CF)CC(F)(F)C3)=O)C2C1 38982,N1(C(C(C(CC)C)C)=O)CCC2CN(C(=O)C(CO)C(C)C)CC2CC1 38983,c1(C(=O)NCC2CN(C(CCCCSC)=O)C3C2C3)cc2cc(Cl)ccc2[nH]1 38984,C1(CNC(C(=O)NC2CC2)=O)CN(C(=O)CCC2OCCO2)CC12CCOCC2 38985,C(=O)(C(CC(F)F)C1CCC1)N1CC=CC(NC(CC2N(C)C(=O)CC2)=O)C1 38986,O=C1NC(=O)C(C2CC(C(=O)NCCCN3CCCC3)C2)N1 38987,N1(C(c2c(OC)c(Cl)sc2)=O)CC2ON=C(CNC(=O)COC(C)=O)C2C1 38988,C1(N(S(C)(=O)=O)CC)CON2CCC(C2)C(CSC)NC1=O.C(C)(C)(C)NC 38989,C12(C(=O)NCC3C(C)CCN(C(=O)COCCN(C)C)C3)CC(C)(C1)OC2(C)C 38990,C1(C2CCN(C(=O)CC3CSCCS3)C2)(NC(C2C=CC=CC=C2)=O)CC1 38991,Cc1scc(C(=O)NCC2(O)CN(C(=O)CCc3ccon3)C2)c1C 38992,c1(C(=O)NC2C(NC(C3CCCC(C)(C)C3)=O)COC2)nc2cc(O)ccc2[nH]1 38993,CC1CCC(CCNC(C2(C)CC2)=O)CC1.C1(C(=O)N)C2CC(=O)CC12 38994,N1(C(CC(CC)C2CCC2)=O)CCC(C(=O)N(CCCN(C)C)C)C(C)(C)C1 38995,Cc1ccc(C=CC(N2CCOC(CNC(=O)CCn3ccnc3)C2)=O)o1 38996,C1(S(=O)(=O)N2CCN(C(=O)CCC=O)CC2)(C(C)C(=O)OC)CC1.C#CC 38997,c1(C(=O)OC)sc(Br)cc1NC(c1coc(C(F)F)n1)=O.C12(CCC1)CC(=O)N2 38998,C1(NC(C(=O)Nc2c(C)cn(C)n2)=O)CC(OC(F)F)C12CCC2 38999,N1(C(C(CC)CC)=O)CCC2(CC1)CN(C(C1CCCC13CC3)=O)CC(C)O2 39000,C1(OCC)CC(NC(C2COCC(C)O2)=O)C12CCC2 39001,C1(C(N2CC=CC(C(N(CCC)C)=O)C2)=O)CC(C)(C)CN1C 39002,c1(OCC=C)c(C(=O)N(C)CCN(C)C(C2CC(F)C(=O)N2)=O)cccc1C 39003,C1(CC(=O)N(CCCC#C)C)CC(NC(=O)CCCCSC)C1(C)C 39004,C1(CC)CCCC(N=c2[nH]c(=NC3CC(N4CCC4)C3)[nH]c3c2COC3)C1 39005,N1(C(=O)CC2CC(F)(F)C2)CCC2CCN(C(C3CC4CC3C4)=O)C2C1 39006,CCCCC(CNC(c1cc(C2CC2)on1)=O)NC(=O)CC1(C#N)CC1 39007,C1(C(=O)NCCCN(C(C)C)C(c2ccc(F)o2)=O)CC1C1CC(F)(F)C1 39008,c1(C(N2CC(n3cc(CNC(CC4C(C)CCO4)=O)nn3)C2)=O)cc(O)ncn1 39009,N1(C(c2ccc(C(C)C)c(Cl)c2)=O)CCN(C(c2cnncc2O)=O)C2(CC2)C1 39010,c1(OC)ccc(Cl)c(CC(=O)NC2CC(CCNC(=O)CCc3cc[nH]n3)C2)c1 39011,Cc1cc(=NCCCS(=O)(=O)C(F)F)[nH]c(NCc2cccc(C)c2F)n1 39012,N1(C(CS(N)(=O)=O)=O)CCC2CCCN(C(=O)Cc3cccc4[nH]ncc34)C2C1 39013,C1(C(=O)NCCN(C(C(N2CCOCC2)C)=O)C2CCCC2)CC(F)(CF)C1 39014,C(=O)(C(C)(C)S(C)(=O)=O)NC12CCC(CNC(C3(CC)CCCCO3)=O)(OC1)C2 39015,C(=O)(CCCC(CC)NC(c1cnn(C(F)F)c1)=O)N(CC(=O)OC)C1CC1 39016,c1(OC)noc(C2CC2)c1C(=O)NCCC1CCCN1C(=O)CC1(O)CCOC1 39017,c1(CC)cc(C(=O)NC2CCCN(C(=O)C(C)n3cncn3)CC2)ccc1OC 39018,CCC(C)CCCCC(=O)N1C2CCC1CC(N(C(=O)CC1CC1)C)C2 39019,N1(C(C2CCCN(C(C3(C)ON=C(C)C3)=O)C2)=O)CCC2(CC1)CSC2 39020,c1(C(N2CCC(C)(NC(CNC(C)=O)=O)C2)=O)nn(C)c(C)c1N 39021,CC1COC(CC(N2CCOCC2CN(C)C(c2cnccc2Cl)=O)=O)CO1 39022,C(=O)(CC1=Cc2ccccc2C1)NCC(CC)(C)NC(=O)CCCc1cc[nH]n1 39023,Cc1nc2cc(C(N3CCCN(C(C4CCCN(C(C)C)C4)=O)CC3)=O)[nH]c2s1 39024,C1(NC(c2c(C)c(Br)ccn2)=O)CCCC2CN(C(=O)CSC(C)C)CC12 39025,C1(NC(C(C2CNC2)OC)=O)COCCN1C(=O)C(CO)OC 39026,C1(NC(c2n(CC=C)ccn2)=O)C(C)(C)C(NC(=O)C(C)O)C1(C)C 39027,N1(C(C=CCN(C)C)=O)CCC2(CCCN2C(=O)Cc2ncc(F)cn2)C1 39028,c1(C(N2CCCC2CCC#N)C(=O)NC(CC)C)cnc(C2CCC2)s1 39029,C1(CCC(=O)NC2CCN(C(CC3C(C)CCO3)=O)C2)CCCN(C)C1 39030,CC1(C)CC(NC(=O)CC2C=CS(=O)(=O)C2)CN1C(=O)CCCn1cncn1 39031,N1(C(C23CCC(CC2F)C3)=O)CC2(C1)CN(CC(F)F)C2 39032,c1(-c2cn(CCC(=O)NC(c3ccccc3)CC)nn2)cc[nH]c(=N)c1 39033,c1(C(=O)NC2CC(NC(C=Cc3nnc(C(C)C)o3)=O)C2)nnc(O)cc1O 39034,C(=O)(CS(=O)(=O)c1ccccc1Cl)NC1CCC(F)(CNC(C(CC#C)O)=O)C1 39035,c1(C(N2CC(CCC)N(C(c3cncs3)=O)CC2)=O)ccc(Cl)c(F)c1O 39036,CC1(C)CN(C(=O)C=C2CCCCC2)CC1C(=O)NCc1ccccc1Cl 39037,C1(C(N(CC(C)CNC(c2sc(Cl)cc2Cl)=O)C)=O)CCCC1C1CC1 39038,C1(CNC(C2CN(CC(C)C)C2)=O)CCC(C)CN1C(c1ccc(C2CC2)o1)=O 39039,c1(C(=O)NC2CCC(NC(C(C)OCCN(C)C)=O)C2)cnc(SC2CC2)nc1O 39040,C(CCN=c1nc2scnc2c(NC(C2CC(F)(F)C2)C)[nH]1)OC(C)C 39041,C(=O)(C(CC(C)C)NC(C1CCCC1)=O)NCCN(C(C1C(C(=O)OC)C1)=O)C 39042,C(CC(c1cccs1)NC1CC1(C)OC(=O)OC(C)(C)C)NC 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39060,N12CCN(CC1)CC2=O.C1(NC(C(CC)c2ccccc2)=O)CCN(C(N)=O)CC1 39061,c1(C(=O)NCC#CCNC(CC2C(C)CCC2)=O)cnc(C(F)(F)F)c(F)c1 39062,N1(C(c2c(C(C)C)cnn2C)=O)CCCC2(C1)CN(C(=O)CC1=CCCCC1)C2 39063,C1(CNC(CCOCC)=O)(COC)CCN(C(C2C(C)CC2C)=O)CC1 39064,C1(C(=O)NC(C(C)NC(C2CC3CC3C2)=O)CO)CC(C)(C)CO1 39065,N#Cc1cccc(N2CCC2)c1.c1(Sc2ccc(Cl)cc2)nnc2n1C2 39066,C1(CNC(CC(C)SC)=O)C=CCN(C(=O)CC2CCC=CCC2)C1 39067,C1(C(C(=O)NC(C2CSC2)C)C)CCN(C(=O)COC2CCCC2)C1 39068,CC(C)(CCNC(=O)C(C)(C)c1ccsc1)NC(=O)CNS(C)(=O)=O 39069,CC1CC(NC(=O)CN(C2CCCC2)C)CCN1C(=O)C=Cc1ccc(F)cc1 39070,C1(NC(C23CC2CN(C(N2CCCC(C(=O)OC)C2)=O)C3)=O)CC(C2CC2)=NO1 39071,c1(C(=O)NCCOC(C)=O)ccc2c(-c3c(C#N)cccc3[N+](=O)[O-])n[nH]c2c1 39072,C(C(C)(C)C(=O)NCCC1CCCN(C(=O)CCc2ccccc2C)C1)SC 39073,n1(CC(=O)NC(C(C)NC(C2=C(C)CCCC2)=O)(C)C)ccc2ccc(C)cc12 39074,C1(CNC(c2c(C)snc2)=O)CC2(CCC2)CN1C(=O)Cc1cncnc1 39075,C(=O)(C1=COCCO1)NCC(CN(C(c1ccc(C2CCC2)cn1)=O)CC)(C)C 39076,c1(C(=O)NC2CN(C(CC(C)N(C)C)=O)CC2O)nccc2ccncc12 39077,N1(C(C(C)OCCOC)=O)CCN(C)C(C(=O)NC2CC(CC)(CO)C2)C1 39078,C1(CC=C)(C(=O)N(CCCCCC2CC2)C(C)C)CCCN1C(=O)C(C)C(F)F 39079,Nc1cncc(C(=O)NC2CCCCC2CNC(c2cc(Br)no2)=O)c1 39080,S(=O)(=O)(c1cccc(Cl)c1)NC(CC)C(N1CCN(C(=O)CN(C)C)CC1C)=O 39081,N1(C(C(C(C)C)OC)=O)CC2(NC(=O)C(CO)NC(N)=O)CCC1CC2 39082,CC1CCCN1CC(=O)N(CC(=O)NC(c1cccnc1)CO)C1CCC1 39083,N1(C(C2(CC)CC2)=O)CCN(C(=O)C(c2ccc(C(F)(F)F)nn2)C)C(C2CC2)C1 39084,C1(C(=O)NCCN(C(=O)COc2ccc(Cl)c(F)c2)CC)CCOC(=O)CC1 39085,N1(C(C(C=C=C)C)=O)CCCC(CC)(NC(c2cc(Cl)ccc2Cl)=O)C1 39086,C1(OCC(N2CCC(N(C(c3cc(C)no3)=O)CC)C2)=O)CCC(F)(F)CC1.OC 39087,C1(C)(OC)CCCN(c2cc(N(C)C)nc(CNc3ccsc3C(N)=O)n2)C1 39088,CC1(C#CC(=O)NC(C2(Cc3cnc(C4CC4)o3)CCC2)=O)CC1 39089,c1(N(C2CCC23CCNCC3)C(Cc2nc(C)sc2)=O)ncc2c(Br)cccc2n1 39090,c1(C(N2CC(O)(CCNC(CNS(CCC)(=O)=O)=O)C2)=O)ccc(CC#N)cc1 39091,c1(C=O)cccc(F)c1.c1(C(=O)NC(c2nc[nH]n2)C)ccc(C(C)(F)F)cc1 39092,C(=O)(C(C(C)(C)C)SC)NCC1(OC)CCN(C(=O)COCCC2CCCC2)C1 39093,C(=O)(CS(=O)(=O)CCO)N1CCC(C)(C(C)NC(COCC(C)C)=O)CC1 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39112,n1(C(C)C)ncc(C(N2CCC(CF)(NC(=O)CC3CCCC(=O)N3)C2)=O)c1Cl 39113,N=c1ccn(CC(=O)NCCNC(=O)Cc2cnn(CC3CCCC3)c2)[nH]1 39114,c1(CC)cc(C#N)ccc1C(N1CC(Cn2c(C)ccc2C)C1)=O 39115,c1(C(=O)NCC(CCOC)NC(=O)CCCC(N)=O)ccc(F)c(OC(F)(F)F)c1 39116,N1(C(CC2(CC=C)CCCC2)=O)CCCN(C(=O)Cn2nnc(=O)[nH]2)CC1 39117,C1(CNC(CCCOCCOC)=O)CCCN(C(c2ccc(F)c(N)c2)=O)CC1 39118,c1(C(N2CC(C)(C)C2Cn2cc(CCCNCCCO)nn2)=O)cnn2ccsc12 39119,N1(C(C(CN(C(CCCOC(C)C)=O)C)C)=O)CC(C)OC(C)(C)C1 39120,N1CCC(Nc2nc(CC)cc(CC)n2)CC(O)C1.C(=O)C#CC1CC1 39121,C(=O)(NNc1c(C#N)cc(CCC(=O)O)cc1[N+](=O)[O-])Nc1ccc(SC)cc1 39122,CC1CCCC(N2CCN(C(c3ccoc3)=O)CC2)C1 39123,c1(N(CCCNC(c2cccc(OC)c2C)=O)C2CC2)nc2ccccc2o1 39124,c1(C(=O)NCC2N(C(C3N(C(C(C)=CC)=O)CSC3)=O)CC2)ccc(N(C)C)cn1 39125,Cc1noc(C)c1CC(=O)NCCNC1CCCC(C(=O)NC(C2CCC2)=O)C1 39126,c1(CN(C)C(C23CC(C2)C3)=O)cnn2c1CN(C(=O)Cc1cnnn1C)CC2 39127,C(=O)(C(O)C(F)(F)F)NCC1(CCCNC(C(COC)(C)OC)=O)CCCC1 39128,C(=O)(C1=CCC(C)(C)CC1)N1C(CNC(c2cc(C(C)=O)sc2)=O)CCC(C)C1 39129,c1(C(N2C(C(N3CC4C(C(=O)O)C4C3)=O)C3CCC2C3)=O)ccc2c(c1)CCC2 39130,C1(C(=O)NCC(CC)NC(=O)C(c2ccc(F)cc2)(C)C)CCCCN1N=O 39131,C(=O)(C(Cn1ccnn1)NC(c1cc(C2CC2)[nH]n1)=O)NC(CCOCC)C 39132,c1(C2CCN(C(=O)NCC(C(CC)O)(C)C)CC2)csc2cc(C)ccc12 39133,c1(C(N2CC(NC(C(C)Sc3ccncc3)=O)(CO)C2)=O)ccc([N+](=O)[O-])o1 39134,C1(O)(CC(N2CC(CNC(C(C=C)(C)C)=O)C(C(F)(F)F)C2)=O)CCN(C)CC1 39135,C1(C(=O)NCC(C(C)C)(C)NC(=O)CC2CC3(CC3)CO2)CC2(C1)CC1(CCC1)C2 39136,C(c1cccnc1)=CC(=O)N(CCNC(CN(CCC#C)C)=O)C 39137,C=C(C)CC(C(=O)N(Cc1ccccc1)OC)NC(C1CC2(CC2)CO1)=O 39138,N1(C(c2ccc(OC)cc2O)=O)CCC(C)C(NC(=O)CSCC(N)=O)C1C 39139,N1(C(C(CCCNC(c2cc(C)c(C)s2)=O)O)=O)CCC12CCCCC2 39140,CCCCCCC(F)C(=O)N1CCC(C)(CNC(c2ccc(O)c(N)n2)=O)C1 39141,c1(C(=O)NC2CC(CCNC(C3(C=C)CC3)=O)C2)cccc(C(N)=O)c1N 39142,Cc1scc(C(=O)NC2CCCCC2CNC(c2cn(C)cn2)=O)c1N 39143,n1(CC)nc(C)cc1C(=O)NC(C)CC1CN(C(=O)COCCN2CCOCC2)C1 39144,c1(C(CNC(c2ccc[nH]2)=O)NC(c2c(COC)nn(C)c2)=O)c(C)cccc1C 39145,c1(NC(c2nc(C)oc2)=O)nc2c(s1)CC(O)CC2 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39180,N1(C(CC2(N(C(CCC3C(C)C3)=O)C)CC2)=O)CCC2(CC1)CC2 39181,C1(C(=O)OCC)C=CC(C(=O)NC2CC(NC(=O)CCN3CCOC3=O)C2)C1 39182,C1(C(N2C(COC)CC2)=O)CCC(C)(C)N(C(C2CCCCO2)=O)C1 39183,c1(C(N(CCC(C)NC(=O)CC(C)c2cccnc2)C)=O)ncncc1Cl 39184,CCCCS(=O)(=O)NC(C)C(N1CCC(CNC(C2CCCCC2C)=O)CC1)=O 39185,c1(OCC=C)ccc(Cl)nc1C(N1CCC(C(C)CNC(=O)CCOC)CC1)=O 39186,N1(CCNC(C2(C)COC2)=O)CCN(C(=O)CCC(F)F)CC1 39187,N1(C(C2(CC=C)CCC2)=O)CCC2(C1)CN(C(=O)CN(C)C(=O)C1CC1)CCO2 39188,C1(CCC)CN(C(c2cccnc2)=O)CC1C(=O)NOC1CCOC1 39189,C1(NC(C2C(CC)CCCC2)=O)CC(N=c2[nH]c(CC(C)C)nc(=N)[nH]2)C1 39190,N1(C(c2ccc(CN(CCC)C)o2)=O)CC=C(CCNC(=O)C(C)CSC)CC1 39191,C(=O)(C(CC)CCSC)NCCN(C(c1cc(CCC)n(C)n1)=O)CCOCCO 39192,n1(CC)ccc(C(N2CCC(CNC(=O)CCc3cncs3)C23CC3)=O)cc1=O 39193,CCCCC(C(=O)N=c1ccn(C2CCOCC2)[nH]1)c1ccco1 39194,C1(C#N)(C(=O)NCC(CNC(c2ccc(NC)cc2)=O)F)CCS(=O)(=O)CC1 39195,CCC(C)CC(C(=O)N(CC(N)=O)C)NC(=O)CCCCSC 39196,C1(NC(=O)C(F)CC2CN(C(C3CC(=C4CCC4)C3)=O)C2)CC12CCCCCC2 39197,C1(CC(=O)NCC(C)(C)OCCNC(CC(=O)NCC)=O)CCCCC1C 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39252,C(C(C)(C)C(c1nnnn1C(C)C(=O)OC)NCc1sccc1C)OCC 39253,c1(CCC(=O)NC2C(NC(CCCNC(C)=O)=O)CCC2)cccc(F)c1F 39254,c1(OC)ccc(C(N2CCCC23CN(C(=O)OC(C)(C)C)C3)=O)n2nccc12 39255,CC(C(=O)NCC1CN(C(=O)CCn2cc([N+](=O)[O-])cn2)CCO1)C(C)(C)C 39256,Cc1ccc(F)cc1NC(=O)C(C)N(C(=O)Cc1cc(Cl)cs1)C 39257,C(CCS(N)(=O)=O)n1cc(CO)nn1.c1(OC(C)C(=O)NC(CO)C(=O)O)ccccc1 39258,c1(C(N2C(CN(C(C3CCC34CCC4)=O)CC)CCC2)=O)c[nH]ccc1=N 39259,c1(C(=O)NC2C(C)(COC)C2)cnn(CCNC(=O)CC=C(C)C)c1 39260,c1(C(N(C(C)C)CCN(C(=O)COc2ccccc2Cl)C)=O)n[nH]c2c1CCC2 39261,O=C(CCc1ccc(CNC(C2C3CCC(=O)C23)=O)cc1)CCCO 39262,C1(CNC(C2C(C)C2)=O)CCC12CCN(C(=O)COCc1ncnn1C)CC2 39263,CCC(CCC(=O)N1CC=C(C)CC1)NC(=O)CCNC(=O)NC 39264,N(C(=NCCC(=O)NC1CCSC1)NCCSC)CC(CC)(C)C 39265,c1(CNC(=O)NCC#CCOC)cn(C2CCCCC2C(F)(F)F)nc1C 39266,CCC(C)(C(=O)NC(C1CCN(C(=O)C(C)(C)c2ccccn2)CC1)C)OC 39267,C1(C(=O)NC(CC)C(C)(C)C)CCN(C(=O)CN2CCOCC2=O)O1 39268,C1(OC)CC(NC(c2cc(C)oc2C(F)(F)F)=O)CN(C(C2(C#N)CC2(C)C)=O)C1 39269,c1(OC)ccc(Cl)cc1C(N1CCC(CCNC(C2(C)CCN(C)CC2)=O)C1)=O 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39288,c1(CC)cc(=NC(=O)C2CC=C(C)CCN2C(c2cccc(=O)n2C)=O)[nH]n1C 39289,C(=O)(C(CC)CC(F)F)NCC(CCOC)NC(c1n(C=C)ncc1)=O 39290,CN=c1[nH]cc(C(=O)N(C2(C(=O)N(CCCF)C(C)C)CC2)CCO)s1 39291,N1(C(C#CC)=O)CC(C(=O)NC2(CN(C)C)CCC2)CC(C)C1 39292,CCCCC(O)C(=O)NCCc1cc(C(N2CCCC(C)C2CO)=O)no1 39293,C1(CNC(=O)Cc2cccc(C(=O)NC(C)C)c2)C2CCCC1NC2 39294,C1(CC(=O)NC(CCCNC(C(CC)C2CCC2)=O)C)NC(=O)NC1=O 39295,c1(C(=O)NCCC2CCCN(C(=O)COC(F)(F)F)C2)ccnc2ccccc12 39296,C1(NC(C2CC(=C)C2)=O)CCN(C(=O)Cc2nc(Br)sc2C)CC1C 39297,N1(CCCOC)CCCC1C1CCCCN1C(C1CCc2ncncc2C1)=O 39298,c1(C(N2C3(CNC(CS(=O)(=O)NC)=O)CC(C2)C3)=O)c[nH]c2cc(N)ccc12 39299,N1(C(C)=O)CC(F)CC1C(N1CCC(CN(C(=O)Cc2ccon2)C)C1)=O 39300,N1(C2CCN(C(C)C)C2=O)CC2CN(C(=O)CCCN=[N+]=[N-])CC2C1 39301,N1(C(c2c(C)c[nH]n2)=O)CCCC2CN(C(=O)Cc3ccc(C#N)cc3)CC12 39302,Cc1cc2ccccc2cc1C(=O)NCC(O)CNC(c1cc(Cl)ccc1N)=O 39303,Cc1nc(CNC(c2nnsc2N)=O)oc1C(=O)NCCOCC(F)F 39304,CC1Cc2c(Br)ccc(Br)c2CN1C(c1cc(F)ccc1-c1cnn(C)c1)=O 39305,c1(NC(c2ccc(C)cc2)C2CC2)n[nH]c2c1CCCCC2 39306,Cc1cccc2c1CCN(CC(C1C3CCOC3C1(C)C)=O)C2 39307,Cc1ccc(C#N)c(N(C)CCN(C(=O)CNC(C2CCCC2O)=O)C)n1 39308,S(=O)(=O)(c1ncc(F)cn1)N1C(CS(C(C)C(C)(C)C)=O)CCC1 39309,c1(C(C)C)noc(C(c2nnnn2C2CCCC2)NCc2cnn(C)n2)n1 39310,C(C)(C)(C(C)NC(=O)C(C1(O)CCC1)NC(=O)CCCC1CCC1)OC 39311,C1(Cn2c(-c3cc[nH]n3)nc(-c3cnccc3)n2)CCC12CC(F)(F)C2 39312,c1(OC)c(C(N2CCC(CO)(CNC(=O)CC(C)OC)C2)=O)csc1C 39313,N1(C(CSCC(N)=O)=O)CCC(O)(CNC(C2CC(=O)N(C3CC3)C2)=O)C1 39314,c1(NC(c2ccc(-c3c(OCC(C)C)ncnc3)cc2)=O)cc(C#N)ccc1Br 39315,Cc1ccc2nc(N3CC4CC3(CNC(=O)CC3C=CS(=O)(=O)C3)C4)sc2n1 39316,Cc1cc(C(F)(F)F)c2cc(C(=O)NC(C)CCN(C)C)oc2n1 39317,CCC(CC)C(O)CNC(=O)CC1CN(C(=O)CCc2ccco2)CC1C 39318,N1(C(C=CSC)=O)CC(N(C)C(c2cccc(-c3ccco3)c2)=O)C(C)(C)C1 39319,N1(C(c2cnc(CCC)s2)=O)CCC(C2CCCN(C(C3(C)CC3(F)F)=O)C2)C1 39320,CON(C)C1CN(C(C2CCN(C(c3ccc(C)o3)=O)CC2C)=O)C1 39321,c1(CCC(=O)N(C)C)nc(=NCc2cc(F)ccc2Cl)[nH]c2c1COCC2 39322,Cn1nnc(C(n2nnnc2C(C)COC)(C)C)n1.c1(CNC2CC2)cnccn1 39323,C1(C(=O)NC)CCCN(C(C2CC3CCC2O3)C(=O)NCCCF)C1 39324,C1(SC)CCC(N=c2nc(N(C)CC3CCSCC3)c3c([nH]2)CSC3)CC1 39325,C(=O)(C(F)(F)C(O)C1CC1)N1CCC(NC(C(C(C)C)NC(N)=O)=O)CC1 39326,c1(C(OC)OC)ccc(C(N2CCC(NC(=O)Cc3nccn3C)C2)=O)o1 39327,c1(OC)cc(N)ccc1OCC(N)=O.C1C(C(C)C)NC(=O)N1.c1(C)cocc1C 39328,N1(C(=O)OC(C)(C)C)CCN(C(c2cccc3oncc23)=O)CCCC1CCO 39329,CC1CC(=O)CCC1C(N1CCOC(C(=O)N(CC(=O)NC(C)(C)C)C)C1)=O 39330,N(C)S(N)(=O)=O.C1(N(CC(=O)OCN)C)CC(NC(=O)Cc2ccco2)C1 39331,C(=O)(C(O)CC(F)(F)F)N(CC(C)NC(C(CC)NC(c1ccccc1)=O)=O)C 39332,CC(CS(C)(=O)=O)C(=O)NC1CCC(NC(=O)C(C)(C)CC#N)CC1 39333,C1(C(N(CC#C)CC)=O)(CC)CCN(C(c2ccc(CC)s2)=O)C1 39334,CC1(C(N2CC(NC(C3CCC(CC4CC4)CC3)=O)C2)=O)Cc2ccccc2N1 39335,c1(CC(=O)N(CC(C)O)CCNC(C=COCC)=O)n[nH]c(=NC)s1 39336,CN1CCn2ncc(C(N3CC(NC(=O)C4=COCCC4)CC4(CC4)C3)=O)c2C1 39337,c1(C(N(CC(C)NC(C2(C)COC2)=O)C)=O)cc(F)c(Br)cc1O 39338,c1(C(N2CCC(NC(C(CC#C)(C)C)=O)CC2C)=O)cc2c(C)[nH]nc2s1 39339,c1(C(N2CC(CNC(CCSC)=O)C2)=O)ccncc1Cl 39340,C(=O)(C(O)CC(F)(F)F)NCCC1CCC(NC(C2CC3(CC(OC)C3)C2)=O)C1 39341,C1(CN(C)C(=O)NC2CC3(CSC)COC2C3)COC(C)(C)CO1 39342,C1(C)(NC(C)=O)CCN(C(=O)C(=O)N)CC1.c1(C=O)cnn(C(F)F)c1 39343,c1(CC)nc(=N)[nH]cc1C(N1CC(F)CC1CN(C)C(c1ccoc1)=O)=O 39344,C1(NC(c2c(C)con2)=O)CC2(C(=O)NC3CC(O)(CO)C3)COC1C2 39345,C12(C(=O)NC3C(SC)CN(C(C4CCCC(C)(C)C4)=O)C3)CC=CCN1CCC2 39346,C1(C(=O)NC2CCN(C(c3nccc(SC)n3)=O)CC2F)Cc2ccccc2C1 39347,C1(C(=O)NC(C2OCCN(C(CC(=C)C)=O)C2)C)CCCCC12OCCO2 39348,Cc1ccn2nc(C(N3CC4CCC3C(NC(c3nncs3)=O)C4)=O)nc2n1 39349,c1(CCC)cc(C(N2CC(CNC(c3cccc(=O)o3)=O)C(O)C2)=O)sc1C 39350,C(=O)(CC(C)(C)CC(=O)N(C)C)NC(CC)Cc1cccc(Br)c1 39351,c1(C(N(CCCN(C(c2ccc(OC)c(F)c2)=O)C)C)=O)c(C)cc(Cl)nc1Cl 39352,c1(OC)c(F)cc(C(=O)NCC2CCN(C(=O)CCCSC)CC2)cc1F 39353,N1(C(CCCN(C)C)=O)CCC2CCCC12CNC(c1cc(Cl)ccc1F)=O 39354,C(=O)(N=c1nc[nH]n2cccc12)C1SCCN(C(c2ccc(C#N)cc2F)=O)C1 39355,C(=O)(C(F)C(C)(C)O)NC1CC(C(C)NC(c2cncc(CC)c2)=O)C1 39356,C(=O)(C1CCCc2n[nH]cc21)N1C2C(NC(c3cccnc3)=O)(CCC2)CC1 39357,C1(CNC(CS(CC)=O)=O)(NC(=O)C(C)Oc2ccccn2)CCC(C)(C)CC1 39358,C1(C(=O)NC2(C)CN(C(c3n(CCCC)ncc3)=O)C2)CCCC(C)(C)CC1 39359,c1(C(=O)NCC2N(C(C(CC#C)C3CC3)=O)CC(OC)C2)c(O)nnc2c1CCC2 39360,C(=O)(NNc1cc(C(F)(F)F)ccc1F)C1CNC(=O)N1 39361,N1(C(c2ccc[nH]2)=O)CCC(N2CCN(c3ccc(F)cn3)CC2)CC1 39362,N1(C(C(C)OCCN(C)C)=O)CC2CC(NC(=O)CCC(C)(C)O)CC2C1 39363,CC1=CC(C)CN(C(=O)CC2CCC(NC(=O)Cc3cccnc3O)CC2)C1 39364,C(C)(C(C(=O)N1CCC(O)C1C)C(C)C)NC(c1c(C)c(O)ccc1)=O 39365,Cc1ncc([N+](=O)[O-])n1CC(N1CCN(C(=O)C(C)OCCN(C)C)C(C)C1)=O 39366,N1(C(c2cc(C)no2)=O)CCCCC(C2CN(C(c3coc4c3COC4)=O)C2)C1 39367,C1(C#N)(CC#N)CCN(C(=O)CC(Cc2cccs2)NC(=O)C(F)F)C1 39368,C1(C(=O)NCCN2CCCC2CCO)CCCC12CCN(C(=O)CO)CC2.C1(C)CC1 39369,N1(C(C2CN(CC(C)C)C(=O)C2)=O)CCCCCC(S(C)(=O)=O)C1 39370,N1(Cc2nn(C)c(C(F)F)c2)CCOCC1C1CCCO1 39371,c1(C(N(C2CCCN(C(C=COCC)=O)CC2)CC)=O)cc2c(nn1)CCOC2 39372,c1(CC)cc(C(=O)NCC(O)CN(C(=O)Cn2ccnc2)C)ncn1 39373,C1(C(N2CC(CCNC(CN(C(C)C)C)=O)OCC2)=O)CC2(C1)CC2(F)F 39374,C1(C(=O)NC(C)C(CO)NC(=O)Cn2cccnc2=O)C2CN(C)CC12 39375,C=CC(CCC)CC(=O)N(CCNC(C1CCN(c2nc(C)cs2)CC1)=O)CC 39376,C(=O)(CC(F)(F)CC(=O)NC(C1CCN(C(=O)CC2(C)CCCO2)C1)(C)C)OC 39377,C1(N(C(COC)=O)CCC)(NC(=O)C(C2CCOC2)OC)CCOCC1 39378,C1(CC(N2CC(OCCC)C2)=O)CCCCN1C(C1CC1C(C)C)=O 39379,N1(C(CC(C)N(C)C)=O)CC2(CC(C(=O)NOCC(=C)Cl)CO2)C1 39380,N1(C(CC(CNC(=O)Cc2csc(C)c2)OC)=O)CCN2CC(C)CC2C1 39381,Cc1cc(C(F)(F)C(=O)NC2CC(CNC(c3cc[nH]c3C3CC3)=O)C2)cs1 39382,c1(C(=O)NC(C)CCCNC(C2(C)CC2Br)=O)ccc2ccnc(O)c2n1 39383,CCC(CC)C(C(=O)N1CC(OC)C(NC(=O)CCCC2CCC2)C1)OC 39384,CCC(O)C(F)(F)C(=O)NCC(=C1CN(c2nc(Cl)ncc2C2CC2)C1)F 39385,C1(CC)(NC(=O)C=Cc2cncn2C)CCCCCC1.N12CC(COC)(C1)C2=O 39386,n1(C(C)(C)C)ccc(C(=O)NCCC2CCC(NC(=O)C=CCO)C2)n1 39387,Cc1nc(O)nc(C)c1C(=O)NCCC(C)CCNC(=O)CN1C(=O)CCC1=O 39388,C1(CC)CN(C(=O)Cn2cc(Cl)c(C)n2)CC1NC(C1CCO1)=O 39389,C(C)(N=c1[nH]c(=NCc2ccc(N)cn2)[nH]c2c1COC2)c1c(OC)nsc1 39390,C(C)(C)(CC(=O)NCC1=NOCC1)N(C(CC1(CC)CCC1)=O)C 39391,C1(NCC(F)(F)F)CCN(c2nccc(OCCNC(CC(=O)OC)=O)n2)CC1 39392,c1(C(=O)NC(CN(C(c2c[nH]c3nccc-3c2)=O)CC)C)sc2cncn2c1C 39393,c1(C(=O)NCC2(NC(CCCOC)=O)CCCCC2C)cnc2c(c1)COCC2 39394,N1(C(c2scc(CSCC)c2)=O)CCC(C(F)(F)F)C(O)CC1 39395,c1(C(C)(C)C(=O)NCC2CCN(C(C34COCC3C4)=O)CC2)c(F)cncc1Cl 39396,N1(C(=O)CSc2cccs2)CCC2CN(C(c3cc(CO)[nH]n3)=O)CCC2C1 39397,c1(N2CCC(N(C(c3onc4ccccc34)=O)CC)C2)ncn(C)c(=O)c1Br 39398,c1(C(=O)OC)cccc(N(C)C(=O)NCCCC2CCCCC2)c1 39399,C1(C(=O)NCC(=O)OCC=C)CCN(C(=O)C(CC)SC)CCO1 39400,C1(CNC(c2n(C)cnc2)=O)CCCN(C(=O)CSc2ncccn2)CC1 39401,C(CCCCC(=O)NC1(CNC(=O)C(C2COC(C)(C)C2)OC)CCCC1)=CC 39402,C(=O)(CCCC(=O)NC1CC1)N(CCC(=O)NC(C(=O)NCC)C)C1CC1 39403,C1(C)(C(N(C)CC(C)C(=O)NCc2cccc(CSCC)c2)=O)CCCS1(=O)=O 39404,C1(C(=O)NCC2(C)CCCN(C(CC3(C)OCCO3)=O)C2)OCCOC12CCC2 39405,c1(OCC)ccc(C(N2CCN(C(=O)N(C)CCOC3CCOCO3)CC2)=O)cc1 39406,Cc1cc(C)c(C(N2CC(NC(C34CC(C(C)(C)C)(C3)C4)=O)C(O)C2)=O)o1 39407,c1(C(=O)NCC2(F)CCCN(C(c3c(SC)snn3)=O)C2)ccc2[nH]ccc2n1 39408,N(C1CCc2cc(F)ccc21)CCn1nnnc1C(c1coc(C)n1)SC 39409,N1(C(C(CC)O)=O)CCN(C(=O)Cc2cncc(F)c2)C(CC(F)F)C1 39410,Cc1cc(C(=O)NCC2(n3cc(Br)cn3)CC2)ccc1I 39411,CCCC(C(=O)NC1CC(CCC(N2CCC(C)(C)CC2)=O)C1)C(C)C 39412,c1(C(=O)NC2C(NC(=O)Cc3ccncc3Cl)C2)ccn2cccnc12 39413,N1(C(C=CC(c2ccc(C)cc2)=O)=O)CC(NC(C2(F)CC2)=O)CC(C)(C)C1 39414,C(C(C)CC(=O)N1CCC(C(C)C)(CO)C1)NC(C(OCC)OCC)=O 39415,c1(OCC(=O)NCCCN(C(C(CC=C)C)=O)C)ccc(F)cc1F 39416,Cn1c(I)cc2c(N3CC(F)(C(=O)Nc4cnnc(Cl)c4)C3)ncnc12 39417,N1(C(c2cccc(NC)n2)=O)CCCC12CCN(C(=O)CN1CCC(C)C1)CC2 39418,C1(OCC)CCN(C(=NCC2CC2)NCC2CC(F)(F)CO2)CC1C 39419,C12(C(=O)NCCCOCCCNC(c3c(C)nc(C4CC4)[nH]3)=O)COC(CCO1)C2 39420,c1(CC(=O)NC2CCN(C(C=Cc3cn(C)nc3)=O)C2C(C)C)cc(F)cc(Cl)c1 39421,CC1CC(CCNC(c2cnn(C)n2)=O)CCN1C(=O)CCNC(=O)C=CCl 39422,c1(OC)cc(C(=O)NC(C2CN(C(C3C4CC5C(C4)C35)=O)CCO2)C)ccn1 39423,N1(C(C(CC)O)=O)CC(C2CN(C(c3ccc(C)c(O)n3)=O)C2)C1 39424,C1(CC)(CNC(=O)C(c2cncnc2)C)CN(C(C2(N)CC2)=O)C1.C(C)(=O)O 39425,C(=O)(C(C)(O)CCc1ccccc1)NCC(CO)NC(CCCN(C)C)=O 39426,c1(CC(C(=O)NCc2c(COC)ocn2)N)ccc(Br)cc1Cl 39427,C1(NC(CCC#C)=O)CC(CNC(c2csc(-c3ccncc3)n2)=O)C(O)C1 39428,N1(C(C2C(C)C2)=O)CCC(F)(F)C(CN)C1.c1(CSCC)ccc(Cl)cc1OCCO 39429,N1(C(c2ccc(C)nn2)=O)CCCC(NCCNC(c2ccsc2C#N)=O)CC1 39430,C1(C(=O)NC2CCC(N(C(CN(C3CCC3)C)=O)C)CC2)CCC2CC2CC1 39431,c1(OC)ccc(C(C(=O)NCCCC(C)(C)NC(c2oncc2C)=O)OC)cc1 39432,C1(CC(=O)N(C2CN(C3COC3)C2)C)CCCCN(C(C2(n3cccn3)CC2)=O)C1 39433,c1(C(=O)NCC(C)NC(C(=O)NCC)=O)cc(C(C)OCC)on1 39434,N1(C(C(C2CCN(C(C3(C4CC4)CC3)=O)C2)C)=O)CCC2CN(C)CC2C1 39435,c1(CC)ncc(Cl)c(C(=O)NC2(C)CCCN(C(=O)CC3CCCC34CC4)C2)n1 39436,Cc1nc2nc[nH]n2c(=O)c1CC(N1CCN(C(=O)C(C)CO)CC1C1CC1)=O 39437,C1(NC(C(C2CC2)NC(C)=O)=O)CC2CC1N(C(C1(C(F)F)CCCO1)=O)C2 39438,CC(CCCCNC(C1CC1(C)C)=O)NC(=O)Cc1ccc(CO)cc1 39439,C(=O)(C(CCSC)NC(C)=O)NC(CNC(C(C)NC(CC)=O)=O)C(C)C 39440,c1(OC)ccc(-c2cn(C3CCN(C(C4(N(C)C)CC4)=O)CC3)nn2)cc1F 39441,CC1(C(=O)NCC2COCCN2C(C2COCCN2C=O)=O)CCCNC1=O 39442,N1(C(CC(=O)NCC#C)=O)CCC(C)C(N(C)C(C2CN(C(N)=O)C2)=O)C1 39443,C1(CNC(c2nnn(CC)c2C)=O)CN(C(c2nn(C)cc2N)=O)CCC1C 39444,C1(O)(CNC(C=C(CCN(C)C)Cl)=O)CN(C(c2csc(C(=O)N(C)C)n2)=O)C1 39445,C(C1CN(C(=O)Cc2ccc(C)cc2)CC1C(=O)NCC(C)(F)C(C)(C)F)=CC 39446,N1(C(Cc2cccc(C)c2)=O)CCC2CCC12CNC(=O)C=Cc1cncs1 39447,C1(CNC(C(C)O)=O)CN(C(=O)CCCc2ccccc2)C(C)(C)C1 39448,CC1CCCc2ncc(C(N3CCCC(C)(NC(=O)C4=C(Cl)CCC4)C3)=O)n21 39449,CCCCCCC(C(=O)NCC1CN(C(c2scnc2Cl)=O)CC1O)NC(C)=O 39450,C12=CC(=NCC(C)(C(C)(C)C)NC(=O)N1)NC(C1CC1)=N2.CCCC(C)OCC 39451,C1(=O)CCN1.C(CC(=O)NCCOC)N(CC)CC.C(C)(C)(C)OC.C1CC1 39452,N1(C(CCC=CC)=O)CCc2ccccc2C1CNC(=O)CCC1(C)CC1 39453,C1(=O)C(CC(C)C)CNC(C)CN1C.c1(C(C)OCC)nc(COC)cs1 39454,C1(OC)C2CCC(C2)C1C(N1CCC(CO)C(C)C1)=O.c12nc(co1)C(=O)NC2 39455,c1(OC2CCNC2=O)cc(C)ccc1C(N)=O.C(CC(=O)O)N.CC(=O)NC1CC1 39456,CCC(C)(CCC(C)C)C(=O)N(CCCN(C)C(c1n[nH]c2c1CC1CC21)=O)C 39457,Cc1cn2c(n1)CC(C(=O)NCCC1CCCN1C(c1ccncc1Cl)=O)CC2 39458,c1(C(=O)NC(CC(C)NC(COC(CC)C)=O)C)c(C)ccnc1O 39459,C1(C)(C(=O)OC)CN(C(C2CCC2)=O)C1.C1(N(C)C)(CN)CC1 39460,C(=O)(C(=O)CCC(C)C)N1CCCCC(C(N2CC(C)C=C(C)C2)=O)C1 39461,c1(C(=O)NCC2CCN(c3c(F)cnc(OC)n3)CC2C)cccc2c1CCC2 39462,N1(C(=O)CCCC2CCOCC2)CCC2(CCCN2C(=O)CCOC2CC2)C1 39463,c1(C(C)C(=O)NCC2CCC(F)C2)cccc([N+](=O)[O-])c1.C12CN(C1)C2=O 39464,C1(C)(CNC(Cc2c(C)occ2)=O)CC(F)(F)CN1C(c1ccc(C)nn1)=O 39465,C1(C2(O)CN(C(=O)CCC(F)(F)F)C2)(CNC(c2ccn3c2CCCC3)=O)CC1 39466,Cc1nc(=NN2CCC(N3CCCC3)CC2)n(-c2cccc(F)c2F)[nH]1 39467,c1(CC(=O)NC2CCN(C(=O)CC3CCC3)CC2F)ccc2ccccc2c1 39468,c1(N)n[nH]cc1[N+](=O)[O-].C12CCC(CC1)CC(=O)NC(=O)C1C(C1)C(=O)N2.CO 39469,C12(NC(CNC(C)=O)=O)CCCC1N(C(=O)C1=NOC(C3(O)COC3)C1)CC2 39470,c1(NC(C(=O)NCC2C(NC(c3c(C)scn3)=O)CC2)=O)ccc(Cl)cc1 39471,C(=O)(C(C)(C)C(C)NC(=O)C(C)COC)N(C(CC#C)C)C 39472,c1(C(=O)NC23C(CN(C(C4(F)C(C)C4)=O)C2)C3)nccc2ccccc12 39473,C1(N(C)C(C2CNC(=O)C2)=O)CCCN(C(c2ccnc(O)c2)=O)CC1 39474,C1(C(C)C)(C(N2CCCCC2)=O)CCN(CC=CC2CCCC2)C1 39475,Cc1cc(Cl)ncc1NC(C1CC2CC2N1C(c1sc(Br)nc1C)=O)=O 39476,C#CC1COCCN1C(c1ccc(OC)c(F)c1)C(=O)NCCOCC 39477,CCCCCCC(F)C(=O)NC1CC2CCC(C1)N2C(c1ccc(Cl)o1)=O 39478,NC(=O)CCCC(=O)OCCSCCOC(C1NC(=O)CC1C(F)(F)F)=O 39479,CN1CC2(CN(C(c3c[nH]nc3CNC(C3CC34CC4)=O)=O)C2)C1 39480,C1(C(=O)NC2C(NC(Cc3cccc(C)c3)=O)COCC2)CC2CCC1CC2 39481,C=Cn1nccc1C(=O)NC(CNC(c1cn(-c2ccncc2)nc1C)=O)CO 39482,c1(OC)ccc(C(O)C(N2CCC(NC(c3nc(C(C)(F)F)cs3)=O)C2)=O)cc1 39483,C1(C(=O)NC2C(C(N)=O)COC2)CCCCO1.c12coc(n1)CNC2=O 39484,C1(C(=O)NCC(C(C)C)NC(C2CCN(C(N)=O)CC2)=O)C2CCN1CC2 39485,Cc1cccc(NC(=O)CC2(C)CCN2C(c2cnn3c2OCC3)=O)c1C 39486,C1(C)CCCN(NC)C1C.C1(C=O)CC2(C1)CC2(F)F 39487,C12(NC(C3CC4CCC3O4)=O)CCC1CN(C(=O)Cn1nc(O)ccc1=O)C2 39488,C1(C(N2CC(O)(CCC)C2)=O)(NC(=O)C(C)NC(C)=O)CCCC1C 39489,CC1(C)CCCC(CC(=O)N(CCNC(=O)CC2CC=CCC2)C2CC2)C1 39490,C(=O)(C(CN(C)C)C(C)C)N1CC(O)(CC(=O)NC(CC)C)C1 39491,c1(C(C(=O)NCC(CNC(c2c(CC)con2)=O)(C)C)(C)C)ccc(O)cc1 39492,N1(C(=O)OC(C)(C)C)CCC(C2CC2)(NC(N2CCC3(CCCO3)C2)=O)C1 39493,N1(C(c2c(NC)scn2)=O)C2CCC(C(=O)NC3CCCC(C)CC3)C1CC2 39494,c1(C(=O)NC2(C)CN(C(C=Cc3cn(C)nn3)=O)C2)cc(F)c(Br)c(Cl)c1 39495,Cc1cncc(CC(=O)N(C(C)CN(C(=O)CC2CCCC(=O)C2)C)C)c1 39496,C1(CC(=O)NCC(CNC(C(COCC)C)=O)F)CCCCC1(C)C 39497,c1(C(N2CC(C(C)NC(CN(CCOC)C)=O)C2)=O)ccnc2[nH]nnc12 39498,C12(C(=O)NC(c3ccccc3)CNC(CN(C)C(N)=O)=O)CC(C)(C1)OC2(C)C 39499,N1(C(c2c(C(=O)OC)nccc2)=O)CC2CC1CCN2C(C1(F)CCOC1)=O 39500,C1(NC(CCC2CCN(C(c3ccc(C(C)C)o3)=O)C2)=O)CNC(=O)C1(C)C 39501,C1(C(N2CCCC(CNC(=O)COCC3CC3)CC2)=O)CCc2ncsc2C1 39502,C1(F)(CNC(c2scnc2Cl)=O)COCCN(C(C2OCCCO2)=O)C1 39503,CCCC(C)(O)CC(=O)N1CC(NC(c2cccc(CF)c2)=O)C(C(F)F)C1 39504,c1(OC(C)C)ccc(C(=O)NCCCCCCNC(=O)CN2CCC2C)cn1 39505,c1(C(=O)NCC2CCCOC2)cn2cc(-c3ccncc3F)ccc2n1 39506,CC(O)C(F)(F)C(=O)NCCC(C)(C)CNC(=O)CCOCc1ccncc1 39507,N1(S(C(C)C)(=O)=O)CCN(C(=O)NC(c2ccccc2-n2ccnc2)C)CC1 39508,C12(NC(=O)C(F)CC3CC3)CC1CN(C(C1(c3ccno3)CCC1)=O)C2 39509,C1(C(N(C(c2ccccc2)C)C)=O)CCC1(F)F 39510,N1(C(Cc2cc(C(C)C)no2)=O)CCC(NC(=O)C(F)C(C)(F)F)C(CO)CC1 39511,C=CCC(F)(F)C(=O)NCC(O)C(=O)NC1CC2CCC(C1)O2 39512,C(=O)(C(F)CC(C)(C)NC(C1CC(=O)CC12CCC2)=O)NCC(=O)OCC=C 39513,C(=O)(C(F)CC(C)(C)NC(=O)CC1CCN(C)CC1)NCCC(C(C)C)C 39514,c1(CC)c[nH]c(C)cc1=NC1CCc2nccnc2C1 39515,c1(OC)ccc(CCNC(=O)Cc2cc(Cl)ccc2Cl)c(F)c1F 39516,CCC(CC(=O)N1CC2CC(NC(c3ccc(C)c(F)c3)=O)C(C2)C1)C(C)(C)C 39517,O=C(CCCCC(F)F)NCCC1CSCCN1C(=O)C(O)Cc1cnc[nH]1 39518,C1(NC(C2(CCOC)CC2)=O)CCN(C(=O)CCc2ccccc2C)CC1F 39519,N1(C(C(CCF)NC(C=NOC)=O)=O)CCC12CC(C(N)=O)C2 39520,c1(SCCC)cc(Cl)nc(NC(=O)C(N2CCCC(OC)C2C(=O)OC)=O)n1 39521,C(CNC(=O)CC1(C)CCOC1)(CCNC(=O)Cc1[nH]cnc1C)OC 39522,C1(NC(c2ccc(C)n2C)=O)CCC12CN(C(=O)CN1CCOCC1)C2 39523,N1(c2cccc(OC)c2)CCN(CC(=O)Nc2ccc(SC)cc2)CC1=O 39524,C(c1cncc(O)c1)=CC(=O)NCC1N(C)CCN(C(=O)CCC=CBr)C1 39525,C(=O)(CN1C(=O)Cc2ccccc21)NC(CCCCNC(c1c(C)con1)=O)C 39526,c1(C(N(C(C)C(=O)NC(C)Cc2ccncc2)CC)=O)cc[nH]c1NC 39527,CCCC(O)(CCC)CC(=O)N1CCN(c2cc(OCCN(C)C)ccn2)CC1 39528,CC1CCN(C(=O)CSc2ccccn2)CC1CNC(=O)CSc1n[nH]c(=N)s1 39529,C1(NC(C)=O)C2CC3C(C2)C13CCC(C)NC=O.C(CC(C(=O)O)SC)SC 39530,C1(NC(CN(CC(C)C)C(C2CNC(=O)CC2C)=O)=O)CCc2nncn2C1 39531,N1(C(c2sc(C)c(Br)n2)=O)CCC(NC(c2cc3n(n2)CCO3)=O)C(C)C1 39532,CC(C(C(=O)C(NC(C1CC(O)C1)=O)C1CC1)Nc1ccoc1)NC(=O)COCCF 39533,N1(C(C(C=C)(C)C)=O)CC2(C1)C(NC(=O)C1Cc3ccc(F)cc31)CCS2(=O)=O 39534,C1(CC(C(=O)NC2CN(CC)C2)C)CCCN(C(c2ccc(SC)s2)=O)C1 39535,C1(CS)CCCN(Cc2ccccc2)C1.c1(C(C(=O)N)C2CNC2)ccccc1 39536,c1(SC)ncc(C(=O)NCC(C)(F)CNC(=O)CN(C)CC2CC2)s1 39537,c1(C(=O)NCC2N(C(C3C(C(C)(C)C)C3)=O)CCC2)cnc2ncnn2c1O 39538,C(C1=CCN(C(C2CCCN2Cc2nnn(C)n2)=O)CC1)NC(C(C=C)(C)C)=O 39539,C(CCCCC(=O)N1CCC(C(=O)NCC2CC2(Cl)Cl)C1(C)C)OC 39540,Cc1ncc(C=CC(N2CC=CC(NC(C3(C)CCCOC3)=O)C2)=O)s1 39541,c1(C(C(=O)NC2CC(NC(c3cn(CC=C)nn3)=O)C2)(C)OC)ccccc1F 39542,C1(CCC)CCCCC1NC(=O)NCC12CC(COCCC(C)C)(CO1)C2 39543,Cc1[nH]c2ccccc2c1C(N1CCCCC(CNC(c2cnns2)=O)C1)=O 39544,C1(NC(c2ccc(OC)nc2)=O)CC1C1CCN(C(=O)C2=CCC(C)CC2)CC1 39545,N1(C(c2cc(C)c(C)s2)C(=O)NC2CCOC2)CCC(C)(N2CCOCC2)CC1 39546,C1(CNC(CCC(=O)OC)=O)COC(C)(C)CN1C(C1CC2CCC(C1)N2C)=O 39547,N1(C(c2nnn(C)c2C(F)F)=O)CCC2CCN(C(c3cccc(Cl)c3)=O)CC12 39548,c1(C(N2CC(NC(C(C(C)C)O)=O)C(C)C2)=O)nc(C(F)(F)F)n2ccncc12 39549,N1(C(CC(C)C)=O)CCC2(CCCCN(C(C3CN4CCN3CC4C)=O)C2)C1 39550,N1(C(C2(CCC)CC2)=O)CC(C)(C)C(NC(=O)CC(C)(C)COC)C(C)(C)C1 39551,C12(CNC(c3cc4sccc4s3)=O)CN(C(c3cnco3)=O)CC1(C(F)(F)F)C2 39552,C12CN(C(c3cn(C(C)C)cn3)=O)CC1NC2=O.N1(C(CC)=O)CCC(CO)C1 39553,c1(OC)cnccc1C(=O)NCCC1CCCCN1C(c1cc(C(C)=O)c[nH]1)=O 39554,c1(CNCc2nc(C3CCC(C)C3(C)C)on2)c2ccccc2nn1C 39555,C#Cc1cc(F)c(C(N2CC3CC3(NC(C3COC3)=O)C2)=O)cc1F 39556,O=C1COc2cc(C(N3C4CCC3CN(C(C3CCC5CC35)=O)C4)=O)ncc2N1 39557,N1(C(C2(NC(CC(C=C)CCC)=O)CC(F)(F)C2)=O)CCC2(CCC2)C(O)C1 39558,C1(C(=O)NC(COCC)C(=O)NCCN(C)CCO)CCC(F)CC1 39559,c1(C(=O)NCC(CCC)C(=O)N(CCC(F)(F)F)C)ncn2ccccc12 39560,CC(C)CCCC(C)C(=O)N1CCC(CCNC(c2cc3occc3[nH]2)=O)C1 39561,C1(CNC(c2c(C)occ2C(F)(F)F)=O)CC(F)(F)CN1C(c1c[nH]c(=N)s1)=O 39562,c1(CC)nc(C(=O)NCc2ccnc(C(=O)NC3(CO)CCC(O)C3)c2)c(C)o1 39563,c1(C(=O)NCCC(C)N(C(=O)CNc2ccccn2)C)occc1C1CC1 39564,C1(C)(N(C)CC)CCN(C(=O)CC2CCN(Cc3cccc(I)c3)C2)C1 39565,C1(C(N2C(CCNC(Cc3c(C)cnn3C)=O)CSCC2)=O)Cc2cscc2C1 39566,C1(N(CC(C)C)C(=O)COC2CCCC2)CCN(C(C2CC(F)C2)=O)C1 39567,C(c1cc(C)cc(C)c1)=CC(=O)NC1CCN(C(C2(CC=C)CC2)=O)C1 39568,N1(C(CC2(OCC)CCC2)=O)CCCCC(C(=O)NCCCCC(C)(C)C)C1 39569,Cc1ccc(C(N2CCCC2CCC(=O)N(CC(C)C)C2CC2)=O)nc1 39570,c1(C(=O)N2CC2)ccccc1C(C)=O 39571,c1(C(=O)NC(C)CCNC(C2(N(C)C)CC2)=O)ccn(C(C)(C)C)c1 39572,c1(C(C)NC(CC(OC)OC)C2CC2)cnn(C)c1N(C)C 39573,C(C)(CCCCNC(c1snc(O)c1Cl)=O)NC(C1OCC(C)C1)=O 39574,Brc1ccc(C23CCC2CNC3)cc1 39575,N1(c2cc(C)nc(C(C)C)n2)CCC(C)C(NC(C2CC=CCC2)=O)C1C 39576,C1(O)(CNC(C)=O)CCCN(C(=O)CC(O)C(C)C)C1 39577,c1(CCC(=O)NC(CC)CN(C(=O)C(C2CCCC2)OC)CC)cncc(C)c1 39578,CCCCCS(=O)(=O)CC(=O)NCC1(OC)CN(C(C2OCCC2C)=O)C1 39579,c1(SC)c(CC(=O)OCCc2ccc3c(c2)OCO3)cc(C)cc1Br 39580,c1(C(=O)NCC(CO)NC(c2cn(C3CCOCC3)nn2)=O)ccc(Cl)nc1O 39581,c1(CCNC(C2N(C(CS(C)(=O)=O)=O)CCC(O)C2)=O)ccc(S(=O)(=O)F)cc1 39582,C(C1=CCN(C)CC1)NC(C1CC(C)N1C(=O)CC1C(C)(C)C1(C)C)=O 39583,N1(C(c2c(Cl)cn(CC)n2)=O)CCC(C)C(CNC(=O)C#CC(C)(C)O)C1 39584,N1(C(C(CC)OC)=O)CC(O)CC1C(=O)NCC(F)F 39585,c1(C(N(C2CCCC(NC(=O)CC(F)F)C2)C)=O)ccc(P(C)(C)=O)s1 39586,c1(CCNC(=NC)NCC2(C3CC3)CC2)ccc2c(c1)OCCO2 39587,n1(CC(=O)NCC(C)N(C(C2CCCN2CC)=O)CC)ccc(C)cc1=O 39588,c1(OC)ccccc1C(=O)NC(c1cccnc1OC)C(=O)N(C)Cc1cncs1 39589,C(=O)(C1=C(C#N)CCC1)NCC1CC(C)(C)CN1C(=O)COC(F)F 39590,C1(C(c2cn(C3CCN(C(c4ncon4)=O)C3)nn2)=O)CCc2nncn2CC1 39591,Cc1ccncc1C1CC1C(=O)NCC1CCC1NC(=O)CC1CSCCO1 39592,C1(C(N(C(C=C)C)C)=O)CC12CC(NC(c1c[nH]nc1C(F)F)=O)C2 39593,CC(C)CC(C(=O)NC1CC2C1CCN2C(C1CN2CCC1CC2)=O)C(N)=O 39594,c1(OC)cccc(C(=O)NCC2CCC2NC(=O)C(c2ccccc2Cl)OC)c1 39595,C1(CNC(CSc2n(C)ccn2)=O)CCCCN1CC(=O)Nc1cnsn1 39596,N1(C(C2NC(=O)OCC2)=O)C2CCC1(CNC(c1ccnn1CCF)=O)CC2 39597,c1(NC2(C#N)CC2)nnnn1C(=O)CCCc1cccnc1.CCCF 39598,N1(C(c2cnc3ccccc3c2)=O)CCC2CN(c3ncns3)CC2CC1 39599,Cc1ccc(F)c(O)c1C(=O)NC1CCCCN(C(=O)CCc2cscn2)C1 39600,N1(C(CCCCOC)=O)CCC(C)(C)C(NC(=O)C(C(C)CC)NS(C)(=O)=O)C1 39601,C1(NC(CC(C)=C(C)C)=O)CCCC(NC(c2c[nH]nc2-c2ccccn2)=O)C1 39602,C1(C(C)(C)NC(=O)CC2CCOC2=O)CCCN1NC(C=C(CC)CC)=O 39603,Cc1cc(C(=O)NCC(C)CCCO)ccc1[N+](=O)[O-] 39604,c1(OCCC(=O)NC(C(C)NC(=O)C(C2CCCCC2)O)CO)cccc(F)c1 39605,C1(CNC(CC(C)(C)n2cc(CC3COC3)nn2)=O)CCCCCC(=O)N1 39606,C1(CC(N2CC(CCO)(NC(CCCC#C)=O)C2)=O)NC(=O)CN(C)C1=O 39607,C1(C(=O)OC(C2(C(=O)NCCC(O)CNCC)CC2)=O)CC2CCC1O2 39608,C(CCCCC(=O)N(C)CCN(C)C(c1c(C)ccn1C)=O)=CC 39609,C(=O)(C(C)(C)CCC#N)N1CCCC(CN(C(C2CCCC(C)CC2)=O)CC)C1 39610,C(C)(CCCC(=O)N1CCOCC1C1CC1)NC(COCCCC(C)C)=O 39611,Cc1cncc(CCC(N2CC(NC(=O)C=CCCC(C)C)CC2C)=O)n1 39612,c1(CC(=O)OC)cc(Cl)c(NC(=O)C(=O)NN2C(C)CCC2C)cc1F 39613,C=CCCCCCC(=O)NCC1CCCN1C(C1CC(C)(C)CCO1)=O 39614,Cc1ccc2ccccc2c1CNC(N1CCCN(Cc2ccccc2)CC1)=O 39615,N1(C(C2CCC2)=O)CCCC2C1CCN2C(c1sccc1F)=O 39616,N1(C(C(CC=C)NC(C)=O)=O)CCC(C(=O)NCc2nccs2)C1(C)C 39617,C1(F)(C(=O)NC(C2C(C)C(=O)C(=O)OCC2)(CC)CN)C(C)(C)C1(C)C 39618,CC1CCCC(OCC(=O)NC2CC(c3ccccc3)(NC(=O)COC(F)F)C2)C1 39619,c1(C(=O)NS(CCC(C)(C)C)(=O)=O)cc2cc(F)ccc2cn1 39620,C12(CC)CN(C(=O)C3=CCC3)C(CNC(c3ccnn3CC(F)(F)F)=O)(C1)C2 39621,CC1OC(C)CN(C(=O)C(=O)NCC2CCC3(CCCN3)O2)C1C 39622,Cc1cc(=NC(C)CNC(=O)C(C)Sc2ccccc2F)[nH]c(C)n1 39623,C(=O)(C(F)CC(C)(C)C)N1C(CC(=O)NC(C(=O)NC)C2CCC2)CCC1 39624,c1(C(N2C(CNC(CCc3onc(C)n3)=O)CC2)=O)cc(Cl)nn1C 39625,C(=O)(C1=NN(C)C(=O)CC1)NCCC1N(C(Cn2nnc(C)n2)=O)CCOC1 39626,c1(OC)c(-c2noc(C3C(=O)N(C)CCN3C)n2)ccc(I)c1F 39627,N1(C(C(C)S(=O)N(C)C)=O)CCCCC1(C)c1cn(CCc2cccc(F)c2)nn1 39628,Cc1cc(C(=O)NC(C)(C)CNC(C2CN(C3CCOC3)C2)=O)ns1 39629,Cc1cncc(C(=O)NCC(F)CNC(=O)C(C2CCCN(C)C2)(C)C)c1 39630,O=C(NN1CCCC1C(=O)NCCc1nc[nH]n1)C1(C(=O)O)CC1 39631,N1(C(C)C)CCCCC1C(=O)NC1CC(N(C)C(C2COCC2(C)C)=O)C1 39632,c1(CC)cc(C(N2CCN(C3CCC3)CC2)C(=O)NC(C)C(=O)OC)nn1C 39633,C#CC(CC1CCOC1)NC(=O)CCC 39634,c1(CC)cc(C(C)(C)C)nc(N(C)CC2(CNC(=O)C(F)=C(C)C)CC2)n1 39635,C1(C(=O)NCCCNC(C(C)c2ccco2)=O)CSc2ccccc2O1 39636,N1(C(c2cnn(CCC)c2C)=O)CC(N(C)C(c2nnc(S)n2C)=O)C(C)(C)C1 39637,C(=O)(C(F)(F)C(F)F)NC(C(=O)NCC(C)Cc1cccs1)C1(O)CCC1 39638,C(=O)(C(F)CC(C)(C)NC(c1ccc(F)cc1C)=O)NC(C#C)CC1CCC1 39639,CN1CCN(C(c2cnn[nH]2)=O)C(CNC(C2CCOC(C)(C)C2)=O)C1 39640,C1(C(N(CC(CC)NC(c2ccc(CO)cc2)=O)C)=O)CCCCC1CF 39641,C(CCC(=O)NC1CC(CNC(=O)CNC2(C)CCCC2)CO1)SC 39642,c1(C(=O)N)cc(C(F)(F)F)ccc1O.c1(OC)cc(SC2(CO)CC2)ccn1 39643,c1(NC2CC3(CC(Nc4cc(C#N)ncn4)C3)C2)ccnn2ccnc12 39644,C=C(Br)CCC(=O)N(C)CC1CCCCN1C(c1cnc(NC)cn1)=O 39645,c1(CC)[nH]nc(C(=O)NC2CC(C(=O)N(C)OCc3ccccc3)C2)c1C 39646,N1(C(C2N(C(C3CCC4(CCC4)O3)=O)CC(O)C2)=O)CCC2(C=CCO2)CC1 39647,c1(C(CCO)N(C=O)CCc2ccccc2)c(F)cccc1F 39648,c1(CC(=O)NC(CCCNC(c2c(C)n[nH]c2C)=O)(C)C)ccc(Cl)cc1Cl 39649,n1(CC(=O)NC2(C3CN(C(C(COC(C)=O)O)=O)C3)CC2)ncc2ccccc12 39650,C1(CCC)CN(C(N2CC3CCC2C3)=O)CC1(C)C.c12nsc(n1)N1CC2C1 39651,N1(C(c2cc(C)n(CCO)n2)=O)CC(CNC(c2n[nH]cc2Cl)=O)OC(C)(C)C1 39652,NS(=O)(=O)C1(C(N2CCCC2CNC(C2CC3CCC2C3)=O)=O)CCCC1 39653,c1(NC(c2c(F)cc(C#C)cc2F)=O)cc2oc(=O)sc2cc1O 39654,Cc1cccc(C(=O)NCC2CC(C)N(C(c3c(F)cccc3F)=O)C2)c1C 39655,c1(C(=O)NC2CCC(NC(CC(c3c(C)n[nH]c3C)C)=O)C2)cnc(N)c(N)c1 39656,C(=O)(C(C)(C)CS(C)(=O)=O)N(CCC1N(C(C(COC)COC)=O)CCCC1)C 39657,n1(CCSCC(=O)NC2CN(C(C(c3cccnc3)C)=O)C2)cc(C2CC2)nn1 39658,Cc1ccn2c(C(=O)NC3CC(NC(C4CCCCC4(F)F)=O)C3)c(C)nc2c1 39659,c1(C(=O)NCC2(O)CN(C(c3cn(CCOC)nc3)=O)C2)cccc(Cl)c1Cl 39660,c1(CNC(C(=O)NCc2ccc(OC)c(OC)c2)=O)cc2c(s1)CCOC2 39661,C1(C(=O)NC(CC(=O)OC)C2CC2)C=CCCN1C(=O)CC(O)CN(C)C 39662,C1(N(C(C2(C#C)CCCC2)=O)C)CC2CC1N(C(=O)C(C)=C1CC1)C2 39663,C(CN=C(NCc1ccc(F)cc1Br)NCC12CC(C1)C(C)O2)SC 39664,C1(c2n(C)cnc2)CN(C(=O)CSC(F)(F)F)CC1NC(=O)CSC1CC1 39665,Cc1nc(O)ccc1C(N1CCCCC(n2cc(CNCC3(F)CC3)nn2)C1)=O 39666,Cc1cc(NC(C2C=CCCN2S(=O)(=O)C(F)(F)F)=O)ccc1Br 39667,N1(C(C2N(C(C(C=C)(F)F)=O)CC3(CC3)C2)=O)CC2(CC(CO)CO2)C1 39668,N#Cc1ccc(C(=O)NC2CCCN(C(=O)CCNC(C3CCC3)=O)C2)s1 39669,C1(C(=O)NC(CCNC(C2(OCC)CCCCC2)=O)C)CCCCC(=O)C1 39670,c1(C(=O)NCC(CC)NC(C2(CO)CCCC2)=O)ccc(N2CCC(C)CC2)nc1 39671,c1(COCC=CC(=O)NCC2CC2N)ccncc1.O=CC=CCl.C1CC(=O)N1 39672,Cc1cccc(C)c1CNC1(c2nnnn2CC(F)F)CC(NCC2CC2)C1 39673,C(C1CCN(C(C2CCCC(C)(C)C2)=O)CC1)=CC(=O)NC1C(C(C)C)CCC1 39674,N1(C(C(C2CCC2)OC)=O)CC(NC(c2cc(Cl)c(F)cc2F)=O)C(N=[N+]=[N-])C1 39675,N1(C(CCCNC(C)=O)=O)CCCC(C(=O)NCCN(C)C)(CO)C1 39676,c1(C(=O)NCC2(NC(C3CCN(C)CC3)=O)CCOCC2)cc(F)ccc1N 39677,N1(C(C(C=CC)O)=O)CCC(c2n[nH]cc2C(N2CCCC(N)C2)=O)CC1 39678,C(=O)(CCC(C)(C)O)NC(C1CN(C(=O)C2=CCCCC2)C1)C 39679,c1(OC)ccc(F)cc1CNC(=O)N(C)CCNC1COCCC1c1ccccc1 39680,N1(C(c2cncc(N)c2)=O)CCN(C(c2cc3c[nH]nc3s2)=O)C2CC12 39681,C(=O)(C(=O)CC(C)CC)NCC(CN(C(=O)CC1CCCC(C)O1)CC)(C)C 39682,c1(C(=O)NC2CCC(N(C(c3c(CC)nns3)=O)C)CC2)cc2c[nH]cnc-2n1 39683,n1(CC)c(=O)oc2ccc(NC(N3CCCC(C(=O)OCC)C3)=O)cc12 39684,Cc1cc(CNC(=O)CC2(C)CCN2C(c2ccc(Cl)s2)=O)c(C)s1 39685,C(=O)(C1=NNC(=O)CC1)N1C(CNC(c2c(Cl)nc(OC)s2)=O)C(C)CC1 39686,S(=O)(=O)(c1[nH]c(=NC(C)Cn2cccn2)ccc1Br)N(CCCCCC=C)C 39687,c1(C(N2C(CNC(C(C)(C)Br)=O)CCC2)=O)cccc2cc[nH]c12 39688,CCC(C)(C#N)C(=O)NCC1CCN(C(c2cnc3sccn23)=O)C12CC2 39689,C(CCC(c1ccccc1)NC(C1CC(SC)C1)=O)NC(C=CCC)=O 39690,c1(C(C)C)c(NC(C2(CNC(C3CC3CC(C)C)=O)CC23CCC3)=O)cnn1C 39691,C1(C2CCOCC2)(C(=O)NC(C)CN2CCN(C(=O)CN(C)C(N)=O)CC2)CC1 39692,C1(C(=O)NCCOCCCNC(C2C(C)=NN(C)C2=O)=O)CCc2nnnn2C1 39693,C(=O)(CC(C(=C)C)OC)N1C(CC=C)(C(=O)NC2CCN(C(C)=O)C2)CCC1 39694,c1(N(C2CC(OCCC(=O)OCC=C)C2)C)cc2nnc(C)n2cn1.C1(C)(O)CCC1 39695,C1(NC(C2N(C(C)=O)CCC2)=O)CC2(C1)CN(C(=O)CC1C(=O)N(C)N=C1C)C2 39696,C(=O)(C(F)C(=O)NCc1ccc(C(=O)NCC2(F)CCC2)cn1)OCC 39697,Cc1ccc(CNC(C2(CCNC(=O)CN3CC=CC3)CCC2)=O)cn1.C(=O)(C)N 39698,N1(C(CCOCC)=O)CCC2(CO)CN(C(C3CC(N4CCCC4)C3)=O)CC2C1 39699,C1(C(=O)NC2CN(C(COCCCC)=O)CC2(C)C)CC12CCCCCC2 39700,C(=O)(CCCCC(F)F)NCC1N(C(c2c(NC3CC3)ccc(N)c2)=O)C2C(C1)C2 39701,n1(CC)cc(Br)cc1C(=O)NCC1CC1NC(C1(C(=O)NC)CC1)=O 39702,C1(CCOC)CCCCC1NC(c1ncnn1C(C)C)c1nnnn1C1COC1 39703,C=C=CCC(=O)NOCC(N1CCCC(C)C1)=O 39704,Cc1cc(C(=O)Nc2cnc(OC3CCOC3)s2)c(O)c(Br)c1 39705,c1(NCC)cccnc1C(=O)N(CC(C)NC(=O)CC1(N2CCCC2)CC1)C 39706,c1(NC(C(=O)NCC2C(CCC)CCC2)=O)ccc2nc(N(C)C)[nH]c2c1 39707,C1(NC(Cc2c(C)scc2)=O)CCCC(NC(=O)C=CBr)C1 39708,c1(C(=O)NC2CC(C)(NC(=O)CCC3CCOC3)C2)cc(N)c(F)cn1 39709,C(=O)(CC(F)(F)F)N1C(C(C(=O)NCCN(CCC)CC)(C)C)CCC1 39710,CC1=C(C(=O)N(C)CC2CCCN2C(C2OCCC2C(C)C)=O)CCO1 39711,C1(N(C(C(n2c(C)ncc2)C)=O)CCO)CCCN(C(=O)CC2COCC2O)CC1 39712,N1(C(CC(=O)OC)=O)CCOC2CN(C(c3n[nH]c4cc(C)ccc34)=O)CC12 39713,C1(NC(c2n[nH]c(C)c2O)=O)CN(C(=O)CC(C)(C)c2ccccc2)CCC1C 39714,N1(C(C(=O)Nc2cccc(Cc3c(F)cccc3F)c2)=O)CCc2[nH]ccc2C1 39715,C(=O)(C(CCCCCO)N1CC2CC(=O)NC2C1)NC(C)(C)C 39716,c1(OC)ncc(CC(N2CC(CNC(=O)C=CC3CCOC3)C(O)C2)=O)cc1F 39717,c1(C(N2CCCC2Cc2cc(O)ccc2O)=O)nc2ccccc2s1 39718,N1(C(c2c(C)nc(C)s2)=O)CCN2CCOCC2(CNC(=O)Cc2cc[nH]n2)C1 39719,c1(C(=O)NCC(CC)(CC)NC(=O)C(F)CC(C)C)snc2ccccc12 39720,C1(CC)CN(C(=O)CCc2ccc(F)cc2)CCN1C(C1CCCC(C#N)C1)=O 39721,c1(CC(=O)NCC(c2ccc(F)cc2)C)cccc(F)c1NCC(C)(O)CCO 39722,Cn1cnc2[nH]c(C(N3CCN(C(=O)CC4=CCCC4)C4CC34)=O)cc12 39723,N1(C(C2(C)C=CCCC2)=O)CC2CC1CC2CNC(=O)CCc1ccc(Cl)nc1 39724,N1(c2cc(CC)ncn2)CCCC12CCN(C(c1cccc3c1ncn3C)=O)C2 39725,C1(C(N2CC(CCC)C(NC(=O)CC3C=CCC3)C2)=O)Cc2cscc2C1 39726,N1(C(CC2(COC)CC2)=O)Cc2ccccc2C(NC(c2ccc(C)nc2)=O)C1 39727,C(c1ccccc1F)=CCC(=O)NCCN(C(=O)CC1CCOC1)C 39728,C1(C(=O)OCC)CCN(C(C2CC=CCC2)C(=O)NC2CC2)C1 39729,CC1CCC(=CC(=O)NC(C)CNC(=O)C(C)N2CC(C)C2)CC1 39730,C1(C(N2CCOC(CCNC(c3cccc(Cl)c3)=O)C2)=O)(CSC)CCOCC1 39731,N1(C(c2nc(CC(C)C)sc2)=O)CC2(C1)CN(C(=O)CC1(C)CC1(F)Cl)C2 39732,C1(C(N(CCCN(C)C(C2(CO)CC(C)(C)C2)=O)C)=O)CCC2(CCC2)OC1 39733,CCC(C)C(O)C(C)C(=O)NCCn1cc(C(=O)NCC2(SC)CCC2)nn1 39734,C1(NC(c2ncn(C(C)C)c2)=O)CN(C(C2(O)CCOC2)=O)CC1C 39735,N1(C(C(C=CCCC)O)=O)CC(NC(=O)Cc2c(C)ncn2C)CC12CCCCC2 39736,CC(CCC(=O)NCC1CCN1C(c1cnc(OCF)s1)=O)c1ccccc1 39737,c1(OC)c(C(=O)NC2CN(C(c3c(N)cccc3Cl)=O)C2)oc2ccccc12 39738,C1(CC)C(C(=O)NCc2ccc(C)cc2)CCN1C(=O)C(C)O 39739,N1(C(C2C=C(C)CS2)=O)CCC(C2CC2)C1CNC(c1cnc(C)s1)=O 39740,c1(OC)ccc(C#N)cc1NC(c1nc(N(C)C)no1)c1nnnn1C 39741,N1(C(c2sc(CC)c(C)c2)=O)CCC2CN(C(c3[nH]c(O)nc3C)=O)C2C1 39742,c1(C(=O)NCc2cncc(NC(=O)COC3CCOC3)c2)nc[nH]c2nccc1-2 39743,c1(C(C)(C)NC(c2ccncc2)CF)ccnc(Cl)c1F 39744,C(=O)(C1=CCC(F)(F)CC1)N.N1(C(c2c(NCC)cccn2)=O)CC(N)C(CO)C1 39745,C(CC1=CCOCC1)NC(C(CC)N(C)C(c1cn(C)c(=O)cn1)=O)=O 39746,c1cc(CNC(C2(CNC(C3(CSC)CC3)=O)CC2)=O)cs1.C(C)(=O)N.C.C 39747,N1(C(C2CCC(=O)C2)=O)CCCN(C(c2cc(Cl)ccc2Cl)=O)CCC1 39748,N(C(=NCCCSc1ncccn1)NCC(c1cccc(Br)c1)O)C(C)C 39749,C1(CNC(=O)NCC(C(C)C)(F)F)CCC2(CCOCC2)C1 39750,Cc1ccc(C(=O)NCC(C(C)(C)C)NC(C2CCOC2)=O)c(C)c1 39751,N1(C(Cc2scc(C)c2)=O)CC(C)CN(C(=O)CN2CCCCC2)C(C)C1 39752,C(C)(C)(CC(=O)N(C)Cc1cn(C)nn1)NC(C(C)SC)=O 39753,c1(C(=O)NCC#CCNC(C2(C)CCC2)=O)cc2cc(Cl)ccc2o1 39754,C(=O)(CC(C)C(C)(C)NC(c1cc(=O)cc[nH]1)=O)N1CCC(C)(CSC)C1 39755,c1(C(=O)NCC2C3CN(C(C4(C)CC=CCC4)=O)CC32)csc2cccnc12 39756,c1(C(=O)NC(C2CCN(C(c3csc(C)c3N)=O)CC2)C)ccn2nnnc2c1 39757,c1(C(=O)NC2CCN(C(C(COC)(C)OC)=O)CC2CO)cn2cnnc2cn1 39758,C1(NC(c2cnn(C(C)C)c2F)=O)CCN(C(=O)C(C)Cc2cnc[nH]2)C1(C)C 39759,CCC(C(=O)NC(CNC(=O)CNS(N)(=O)=O)CC(C)C)C(C)(C)CC 39760,C(=O)(CCC(C)(F)F)N(CC(CC)NC(c1c(Cl)cnn1C)=O)CC 39761,CC1Cc2ccccc2N1C(C1CN(C(c2ccncn2)=O)CCC12CCC2)=O 39762,CC(C)(CC(=O)NC1CCC(CNC(C2CCCC3C2C3(F)F)=O)C1)C(F)F 39763,C1(C#N)(C(=O)NCC2CCC(NC(c3scc(C)c3Cl)=O)CC2)CC12CCCC2 39764,C1(C(=O)NCc2cn(CC)nn2)CCC(C)(C)N(C(C2CCCCN2C)=O)C1 39765,c1(CC(=O)NCC2(F)CN(C(=O)C3CC3)C2)cc(Cl)sc1Cl 39766,CC(Cl)(Cl)C(=O)N1CCC(CCNC(C2CCC(C(=O)OC)O2)=O)C1 39767,N1(C(CC2(CC)CCC2)=O)CCN(C(c2csc(C3CC3)n2)=O)CC1C(F)F 39768,C1(OC)(CNC(C2C3CN(C)CC23)=O)CCN(C(c2c[nH]c(C#N)c2)=O)C1 39769,C#CCCC(C(=O)NCC(C)(O)CC)NC(=O)C=C1CCC(C)CC1 39770,C1(C(=O)NCC(CC)N(C)C)CC(=O)CN1C(c1cccn1C1CC1)=O 39771,c1(NC(CC2CCCN(C(c3c(C)scn3)=O)C2)=O)ccc(C#N)c(Cl)c1 39772,C(=O)(C(F)C(F)(F)F)NCCCOCCNC(C(C)Cc1cccnc1)=O 39773,C1(C(N2CC(C(N)=O)(CNC(C3CC(C#N)C3)=O)C2)=O)C2(CC2)C12CC2 39774,N1(C(C(C(COC)C)C)=O)CCCC2(NC(C3CCCCC3C)=O)CCCC12 39775,O=C(C1=C(Cl)CCOC1)NC1CCC12CN(C(=O)C(Cl)=CCl)C2 39776,c1(CC=C)ccccc1C(N1CC(C(C)NC(C2CCOC2=O)=O)C1)=O 39777,N1(C(C2CCN(CCOCc3cscn3)CC2)=O)CCC(F)(CNCC2CC2)C1 39778,N1(C(Cc2c(C)scc2)=O)CC2CN(C(=O)C(=O)NC(C)C)CCC2(CO)C1 39779,C(=O)(C1=NOC(C)(C)C1)N1CC(NC(c2cnc(C(C)C)s2)=O)C(C)CC1 39780,C12(NC(=O)CNCc3nn[nH]n3)CCCCC1CN(C(=O)C(F)(F)F)C2 39781,C(=O)(C(C)S(N)(=O)=O)NCCC1CC(OC)CN1C(C1CCC(C(N)=O)CC1)=O 39782,C1(C#CC(=O)NC2CN(C(C3(CCOC)CC3)=O)CC2OC)(CC)CC1 39783,C(CC)(C(=O)NC1CCCC1NC(C1(C(F)F)CCCC1)=O)=CCCC 39784,O=C(CC1=CCCCC1)N1CCC2C(C(N3CCC(n4cnnn4)C3)=O)C2C1 39785,Cc1ccc(C(=O)C(=O)NC2CCC2CNC(C2CCCCC2)=O)cc1 39786,N1(C(c2ccc(C)s2)=O)CC2CCCCC2(NC(c2occ(C)c2C)=O)C1 39787,C1(O)(CNC(c2cc(-c3ccco3)no2)=O)CCCN(C(C2SCCS2)=O)CC1 39788,C(=O)(C(F)(CNC(=O)C=CC(F)F)C(C)C)N1CC(CC)N(C)CC1 39789,N1(C(CC2(COC)CC2)=O)CC2CN(C(c3ccc4nccn4c3)=O)CC(C1)O2 39790,N1(C(c2cccs2)C)CC2CC1CN2C(c1nc(Cl)sc1Cl)=O 39791,C12CC13CCN(CC3)C(=O)C(OC)C1CN(C1)C2=O.n1(COC)cc(OC)cn1 39792,C1(CNC(C2(C)ON=C(C)C2)=O)Cc2ccccc2CN1C(=O)Cc1ccns1 39793,N1(C(c2c(C)nn[nH]2)=O)CC2CN(C(C3CCCC3S(C)(=O)=O)=O)CC2C1 39794,Cc1ccnc(O)c1C(=O)NCCC1(CNC(C2(C(N)=O)CC2)=O)CC1 39795,c1(OC)ccc(SCC2CCN(C(=O)C(=O)NCc3scnc3Cl)C2)cc1 39796,C1(NC(c2c(COC)ccs2)=O)CC(C)N(C(=O)CCNC(=O)C=CCl)C1 39797,C12(C(=O)NCC3N(C(C4CC(F)C4)=O)CC(O)C3)CC3CC(CC(C3)C1)C2 39798,c1(CC)noc(C(=O)NCC(C2(O)CCN(C(c3cnco3)=O)C2)C)c1C 39799,C1(C)(C(N2CC(O)(CN(C(=O)CNC(c3cscn3)=O)C)C2)=O)C=CCCC1 39800,C(=O)(CCCNC(C1CCC1)=O)NC(CN(C(C1(C#C)CC1)=O)C)(C)C 39801,c1(C(=O)NCC2(CC)CCCC2)c[nH]nc1CCNC(=O)Cc1ccoc1 39802,C1(NC(=O)CCCC2CC2)CCCC12CN(C(C1(c3cccs3)CCOCC1)=O)C2 39803,C1(C)(CNC(C(C)OCCC(C)C)=O)CCCN1C(c1cccc(CCO)c1)=O 39804,Cc1noc(C)c1CN1CC2CC2(CNC(C2(CN(C)C)CC2)=O)C1 39805,Cc1ccc(C(N2CCCN(C(=O)C3=CCC3)C(C)C2)=O)c2c1NCCC2 39806,C(C)(CN=c1nc(C)[nH]s1)NC(=O)NCC(Cn1ncc(C)c1)C.C(C)(C)(C)O 39807,C1(C(=O)NC2(C(=O)NCC(O)CC3CCC3)CCN(C)C2)CCC2(CCC2)O1 39808,C1(C(N2CCC(CC)O2)=O)CC2CCC(C1)N2C(c1cc(F)cc(Br)c1F)=O 39809,N1(C(c2nc(CSCC)sc2)=O)CC(NC(=O)CCC(F)F)CC1C 39810,C(C(O)C(=O)N1CC(O)(C2CCCN2C(=O)CCc2nc(=N)[nH][nH]2)C1)SC 39811,N(C(=NCC(C)(C)F)N1CCN(C(C)=O)C(C)C1)CCSC(CC)C 39812,N1(C(C=CC(=O)OCC)=O)CC(CO)C2(C1)CN(C(=O)CC(C)(C)CC(C)=O)C2 39813,N1(C(C(C=CCCC)O)=O)CC(NC(c2cc(C)c(C)[nH]2)=O)C(C)(C)C1 39814,N1(C(C(C2CCC2)OC)=O)CCC2CN(C(=O)Cc3cc[nH]n3)C(C)C12 39815,N1(C(CC(=C)Br)=O)CCC2(CCCN(C(=O)CCSC3CCCC3)C2)CC1 39816,C1(C=O)CC(C(=O)O)N(C(C2CC3CCC2O3)=O)C1.c1(COC)ncc(Cl)cn1 39817,Cc1c(C(c2cccc(Cl)c2C)N(c2nc3sccc3s2)C2CC2)cc(Br)cc1F 39818,S(=O)(=O)(c1cccs1)NC(CNC(CNC(C1(C)CCC1)=O)=O)C1CCC1 39819,c1(CN(CC)CC)cccnc1NC(=O)C(=O)NCc1nocc1C(C)C 39820,Cc1ccc(C(=O)NC2CCC(CNC(c3ccn(C4CC4)c3C)=O)C2)nc1O 39821,c1(C(C(=O)NCC(CN(C)C(C2(C)CC(C)(C)C2)=O)O)F)ccc(F)cc1 39822,N1(C(=O)NC2CCN(C(C)=O)CC2)CC2CCN(C(=O)Cc3cnccn3)C2C1 39823,C1(CNC(C(CC)(C)C)=O)CN(CCCc2ccc(Cl)cc2)CCC1(F)F 39824,N1(C(C2(C#N)CCC2)=O)CC2CC(NC(c3nccc4n[nH]cc34)=O)C(C2)C1 39825,c1(C(N(CCOCCN(C(C(CCC)OCC)=O)C)C)=O)cc(OC)ccc1C 39826,C1(P(C)(C)=O)(C(N2CC(OC)(CNC(C3(OC)CCOC3)=O)C2)=O)CC1 39827,c1(OC)ccc(C(=O)NCC(C)NC(C2CCCCN2C(C)=O)=O)c(O)c1 39828,C1(C(N2CC(CC)(CC)C2)=O)CCN(C(c2cc(C3CC3)no2)=O)C(C)(C)C1 39829,C(CCCCCNC(c1c(C(=O)OC)c[nH]n1)=O)NC(=O)CCS(C)=O 39830,O=C1NCC2CN(Cc3ccccc3)CC12.c12ccccc1C(=O)NOC2 39831,c1(NC(C(CCSC)NC(=O)Cc2cc[nH]n2)=O)cnc2[nH]cnc2c1 39832,Cc1ccc([N+](=O)[O-])c(C)c1C(N1CCC1CNC(c1cnc(C2CC2)s1)=O)=O 39833,N1(C(c2c(CC)ocn2)=O)CC(NC(C2(c3ccno3)CC2)=O)C(O)C1 39834,C12(NC(CC)=O)CCOCC1CN(C(c1ccccc1S(=O)(=O)NC)=O)C2 39835,c1(NC(C2CC(O)CN2Cc2ccc(I)o2)=O)cccc(CO)c1 39836,C1(C(=O)NC2CC(C)(CO)C2)C2CCC(C2)C1NC(C1CCCCS1)=O 39837,c1(OC(C)C)ccc(C=CC(N2CCN(Cc3cncnc3)C3CC23)=O)cc1 39838,Cc1ccccc1N1CCC(NC(c2cccnc2)C(c2ccccc2)C)CC1 39839,c1(CC(C)NC(c2ccc(C)s2)=O)ccc(CNC(C2CCC(F)(F)C2)=O)cc1 39840,C1(NC(c2c(C)[nH]nc2Cl)=O)CN(C(=O)CCCC(C)SCC(N)=O)CC1(C)C 39841,CC(CC(=O)N1CCC(F)(C(N2CCCCCCCC2)=O)CC1)C(F)(F)F 39842,c1(C(=O)NCC(CNC(C2(CC(C)C)CC2)=O)C)ccc(Br)cc1O 39843,c1(C(=O)NC(C)CCCNC(c2csc(=N)[nH]2)=O)nccn2nccc12 39844,N1(C(c2c3cccc(C)c3[nH]n2)=O)CC(C)(C)OC2(CCCOC2)C1 39845,C12(C(N)=O)C3C4C1C1C2C3C41C(=O)NCC12CC1CN(C(=O)CSC(F)(F)F)C2 39846,C1(N(C(COCC#C)=O)C)CN(C(C2CCCCN2S(C)(=O)=O)=O)CC1(C)C 39847,O=S(=O)(c1ccc(NCC2CCCC(O)C2)cc1Br)NC1CC(C)(C)C1 39848,CCCC(CC(C)C)C(=O)N1CCCC1CN(C(=O)CCC(=O)NCC)C1CC1 39849,C(=O)(CCC(C)(F)F)NC1C(OC)CN(C(=O)CC2CCCCC2)C1 39850,N1(C(C(C)C2CCC2)=O)CC(C2CN(C(=O)C(CO)NC(=O)OC(C)(C)C)C2)C1 39851,CCCCCC(C)(CC)C(=O)NCCC1CCCCN1c1ccnc2ncnn12 39852,c1(C(=O)NC2C(C(=O)Nc3scc(C(C)C)n3)C2)ccc(F)c(Cl)c1 39853,N1(C(C2(CC#C)CCN(C(C3COCCO3)=O)C2)=O)CC2(CC(F)C2)C1 39854,c1(C(N2CCC(O)(C(N3CC(CC#C)OCC3)=O)CC2)=O)cnc2cc[nH]c2c1 39855,N1(C(CNC(C2CCN(CC(=O)NC3CC3)CC2)=O)=O)CCCC2(CC(O)C2)C1 39856,N1(C(c2ccc(F)c(C)c2F)C(=O)NCC(F)F)CC2CCN(C)C(=O)C2C1 39857,c1(C(=O)NCC2(F)CCC(NC(C(CCOC)C)=O)C2)cc(OC)c(O)c(N)c1 39858,N1(C(CCC(=O)c2cccs2)=O)CCC2CN(C(C3CC3C(F)(F)F)=O)CC2C1 39859,S(=O)(=O)(c1ccc(NCC2(C(C)C)CCOC2)c(Cl)c1)N1C(C)CC2(CCC2)C1 39860,C1(CNC(c2[nH]cc(COC)c2)=O)C(C)CCCN1C(C1CCCN1C=O)=O 39861,CCC(C)CCC(=O)N1CCOCC1C(=O)NC(C)CSC(F)F 39862,c1(CC(=O)NC2CC3(NC(=O)C4=CCSC4)COC2C3)c[nH]c2ccncc12 39863,C1(NC(c2cc(COC)oc2C)=O)(CO)CCN(C(=O)C(C)CC(F)F)CC1 39864,c1(CCC(=O)N(C2CCCN(C(C3CN(C(=O)N(C)C)C3)=O)C2)C)cccnc1F 39865,N1(C(c2nc(CCC)oc2)=O)C(CNC(=O)C(C)(C)CO)CC2CCCC12 39866,N1(C(=O)OC)CCC(CNC(C2COCC2NC(=O)CC2CC=CC2)=O)C1 39867,C(C)(C1CCCc2ccccc21)NC(c1ccc(Cl)cc1F)C 39868,c1(N2CC3C(NC(c4c(F)ccc(C)c4F)=O)C3C2)ncnc2sc(C)nc12 39869,C1(C(=O)NCc2cc(CC)no2)C2CCN(C(C3COC(=O)N3C)=O)CC12 39870,CCCCC(C(=O)N(C1CCN(C(C2(S(C)(=O)=O)CCC2)=O)CC1)C)NC(C)=O 39871,c1(CC(=O)NC(CN(C(CN(CCOC)C)=O)C)C)ccc(Br)c(F)c1 39872,c1(C(C(N2CCCC(N(C(CC(=C)C)=O)CCO)C2)=O)C)c[nH]c2ccccc12 39873,C(CC(C)C)(C(=O)N1CCCC(CCCNC(c2c(C)noc2C)=O)C1)OC 39874,n1(CCOC)cccc(C(=O)NC2CC2CNC(=O)C(O)CN2CCCC2)c1=O 39875,C=C(C)C(O)CC(=O)N(C(C)CN(C)C(c1cnn(C2CCCC2)c1)=O)C 39876,C12(CC(=O)NCc3cccc(C)n3)CCC1CN(C(C1CCCCNC1=O)=O)C2 39877,CC(C#N)CCC(=O)N1CCC2C(NC(=O)C(C)(C)Cc3ccccc3)CC12 39878,C(C(C)C)(C(O)C(=O)N1CCCCCC1C(=O)N(C(C)CC1CC1)C)OC 39879,C(=O)(C#CC1CCCOC1)N1CC2(C1)C(O)C=C2.c1(C=O)ccnc(C)c1.CCNCC 39880,N1(C(CCC)=O)CCC(CF)(NC(C2CC(F)C2)=O)C1 39881,C1(NC(c2ccc(C)nc2)=O)CN(C(c2ccc(C(N)=O)[nH]2)=O)CCC1C 39882,C=CCC(C)(C(F)F)NC(=O)C(CC(C)C)N(C(=O)CC1CC(OC)C1)C 39883,Cc1nc(C)c(CCC(=O)NC(C2CN(C(=O)COC3CC=CC3)C2)C)c(O)n1 39884,CCCC(C(=O)NCCCCCN1CCN(C(C2COC(=O)C2)=O)CC1)N(C)C 39885,C1(CNC(c2cc(C)on2)=O)(CO)CCN(C(=O)CC2CCCC2C)CC1 39886,C1(C(N2CCC(CN(C)C(c3cc(Cl)nc(=N)[nH]3)=O)CC2)=O)CCOCC1(C)C 39887,C(=O)(C(F)CC(C)(C)C)N1C(C(=O)NCCc2c(C)nccn2)CC1 39888,c1(C(=O)NCCCN(C(C(C)C2CCCC2)=O)C)cc(F)cc(S(N)(=O)=O)c1 39889,C(CCC(C)CC(=O)N1CC(O)(CCNC(C2CCCOC2)=O)C1)=C(C)C 39890,N1(C(c2cc(C)c(=N)[nH]c2)=O)C2CCC(C(=O)NC3(CC(C)C)CC3)C1CC2 39891,C1(CC(=O)NCCC2(OC)CCC2)CN(C(C2CC(=C)C2)=O)CCC1C 39892,c1(CN(C)CC2CN(C(c3c(OC)cccn3)=O)C2)cc(Br)cnc1C 39893,N1(C(CC2C(C)(C)C2)=O)CCCCC12CN(C(C1SC3C=CC1CC3)=O)C2 39894,C1(CC(=O)NCc2ncoc2C2CCCO2)CCC(=O)N1 39895,C12(CSC)CCN(C1)C2=O.C1(CCC)CCCN1C(C)=O.C12(CC1)CC(=O)NC2 39896,C1(C(=O)NC(COC)COC)CN(C(c2c(C)cccc2Cl)=O)C(C)(C)C1 39897,CS(=O)(=O)c1cc(C(N2CCOC(CCNC(=O)CCC3CC3)C2)=O)ccc1Br 39898,C1(CCOC)(NC(c2n(C)cnc2)=O)CCN(C(=O)C=C2CCCCC2)C1 39899,Cc1cc(Cl)c(C(N2CC(C)(C)C2Cn2cc(C3CCCCO3)nn2)=O)s1 39900,C1(C(N(CC(N2CCCCC2)=O)C(C2CC(C(C)C)C2)=O)=O)CCS(=O)(=O)C1 39901,C(=O)(C1=NOC(C)C1)NCCN(C(C1C(C=C)OCC1)=O)C 39902,C1(NC(CC(=O)OC)=O)CC(O)CN(C(=O)Cc2ccc(OC(F)(F)F)cc2)C1 39903,C(CCCCC(=O)N1CC2CC1(C=O)C2)SC.C(C)(=O)NC1CC1C(C)C 39904,c1(C(N2CC(C)C(CNC(=O)C3=CCOC3)C2)=O)cc2oc(Br)cc2[nH]1 39905,c1(CC(=O)NC2(COC)CN(C(c3cc(C#N)c[nH]3)=O)C2)cnccc1Cl 39906,C(=O)(C(CC)n1nccc1C)N(CC(=O)OCC)C(C)=O 39907,C1(CC)CCCN(C(=O)CC2COCCO2)C1C(=O)NCC1CC(=O)N(C)C1=O 39908,c1(CC(=O)N(CC(CC)NC(c2ccc(F)cc2F)=O)C)csc2sc(C)cc12 39909,O=S(=O)(c1cccnc1NC(C1CCCC1)CO)NCc1cc(C(F)F)on1 39910,c1(C(=O)NC2C(C)N(C(=O)CCc3cnoc3)CC2)nccc2[nH]ccc12 39911,Cc1c(C(N2CCN(C(=O)C(C)CO)CC2c2ccncc2)=O)cccc1C#N 39912,C(C(CC(C)C)C(=O)NC1CC(CCNC(=O)C(C2CCCC2)SC)C1)OC 39913,C(C(C)(F)F)N(C(C=CC(C)NC(C1(C(N)=O)CC1)=O)=O)C 39914,N1(C(CC)=O)CC2CCC(C3C(N(C(=O)OC(C)(C)C)C)CCSC3)(C2)C1 39915,c1(C(C(=O)NCC2CC(NC(C(=O)NCC)=O)C2)C)ccc(C(F)(F)F)cc1 39916,N1(Cc2ccc(-c3c(OCCC)c(Cl)ccc3)s2)CCSC2CCNCCC12 39917,C1(CC(=O)NCC(C)(C)OCCN(C(c2c(C)coc2)=O)CC2CC2)C2CC2C2CC12 39918,N1(C(c2cccc(CC)c2)=O)CCC2(CC1)CC2NC(C1(C)CC(C)=NO1)=O 39919,N1(CC#C)CCCC2(CCN2C(=O)CC(c2cccs2)NC(C)=O)C1 39920,CC1OC2(CO)CC1(C(N1CC3CC3(CNC(=O)Cn3ccccc3=O)C1)=O)C2 39921,C1(COC)(CO)CCCN(C(C2CC2F)=O)C1.C12(CCCC1)C(=O)N2 39922,c1(CC)nc[nH]c1C(N1CCCC1CN(C(=O)CC1CCSCC1)C)=O 39923,C1(C)(C(=O)OC)CCC1(C)C(=O)NCC(O)CNC(c1ccc(F)s1)=O 39924,c1(C(=O)NCCCN(C(C2CCCC(OC)C2)=O)CCO)cc(Cl)ccc1N 39925,C1(C(=O)NC2C=CC(C(N3CC=CC3CF)=O)C2)Cc2nccn2C1 39926,N1(C(C=Cc2cc(OC)ns2)=O)CC2CC(C1)N(C(=O)CCC(C)(C)F)C2 39927,C1(NC(C2COc3ccccc3O2)=O)CC(N=c2[nH]c3cccc(F)c3o2)C1 39928,C1(CNC(c2cccc[n+]2[O-])=O)CN(C(=O)C(O)CC2CC2)CCCO1 39929,c1(C2C(C(=O)NCCN(C(=O)Cc3cnn(C(C)C)c3)CC)C2)ccccc1Cl 39930,C1(CC)CN(C(=O)CCCC#N)CCC1NC(=O)C=C1CCCCC1(C)C 39931,c1(C(N2C(CNC(C3C(C=C)CC3)=O)CC(C)(C)C2)=O)ccc(Cl)c(N)c1Cl 39932,N1(C(c2c(C)nsc2C)=O)CC(NC(=O)C(C)Sc2ccccn2)CC2(CC2)C1 39933,C(C)(CCC(=O)NCc1cc(C(=O)N(CC(C)(C)N(C)C)C)n[nH]1)OC 39934,c1(C(=O)NCC2(F)CN(C(CNC(=O)OC)=O)C2)ccc(C)cc1C 39935,C1(C(=O)NC(C)C(=O)NCCF)CN(C(C2(CO)CCCC2O)=O)CC1(F)F 39936,c1(C(N(C(CNC(CC(C)OC)=O)C2CC2)C)=O)cnc2ncnn2c1C(C)C 39937,N(C1CCc2cc(CNC(=O)CNC(N)=O)ccc21)C(CC(CC)OC)=O 39938,C1(C(=O)NCCc2nc(C)[nH]n2)(CNC(=O)C(C)C)CC12CCC2 39939,c1(C(N(CCOCCCN(C(C(CC=C)C)=O)C)C)=O)c(C)cc(C)nc1O 39940,CCC(C(=O)N(C)CCOCCO)N(C(=O)CNN(C)C)C.c1(C)cnc(C)s1.OC 39941,N1(C(C(C(=O)OCC)(C)C)=O)CC2C3CCC(C2C1)N(C(C1CC1F)=O)C3 39942,C(C(C(=O)N1CCN(C(C)C)C(=O)C1)C(C)(C)C)NC(CCC=C)=O 39943,CN(C1CCCS(=O)(=O)c2ccccc21)C(C1COCCC12CCC2)=O 39944,c1(C(N)=O)cc(C(=O)NCC2OCCC2C(=O)NCC2(F)CCOC2)n[nH]1 39945,Cc1cc(CNC2CC(O)(c3cccnc3)C2)c2c(c1)CCC2 39946,c1(NC)cccnc1C(N1CC(C(N)=O)(CNC(=O)CCc2ccncn2)C1)=O 39947,C=C(C)CC(C(=O)NCC1CC(F)(F)CO1)NC(=O)Cc1cn[nH]c1 39948,N12CCC(C1C)C(=O)NCC=CC2=O.n1(CC)nnnc1C(C)C 39949,c1(SC(C)C)nnnn1CC(=O)NC(C)(CNC(=O)CC(C)N(C)C)CC 39950,Cn1cncc1C(c1nnnn1Cc1cccs1)NCCC(=O)NO 39951,c1(C(N2C(CNC(C3C(C#N)C3)=O)CCCCC2)=O)noc2c(F)cccc12 39952,O=C(N=c1[nH]c(Cl)ncc1O)C1CN(S(=O)(=O)c2cn[nH]c2)CCC1O 39953,C1(N=[N+]=[N-])(C(=O)NC(C(C(=O)OC)C)C)CCN(C(C2CC(CF)C2)=O)C1 39954,N1(C(CC(C)N2CCCC2=O)=O)CCC(C(F)F)(CNC(C2(Cl)CC2)=O)C1 39955,c1(C(=O)NCC(CO)NC(c2ccc(N(C)C)nn2)=O)cnc2n1CCC2 39956,C#CC1CCN(C(=O)C(CCC=C)NC(C2CC(C)(C)C2)=O)CC1 39957,c1(C(=O)NC2CCN(C(CC(C)C(F)(F)F)=O)C2C)c(N)c(F)cc(F)c1F 39958,CCC(Cc1ccccc1)C(=O)NC(C)C(C)NC(c1cc(C(F)(F)F)no1)=O 39959,S(=O)(=O)(c1cc(C(F)(F)F)c(Cl)cc1Cl)N1C(C(=O)CC2CCC2)CCC1 39960,Cc1cc(C(=O)N(C(C)C(C)S(C)(=O)=O)C)ccc1N1CCC(O)CC1 39961,C=C(C)C(C)(C)C(=O)NCC1(CNC(c2ccnc(C3CC3)n2)=O)CCOCC1 39962,c1(C(N2CCC(O)(C(C)CNC(=O)C(O)C3CCC3)C2)=O)ncc2ccccn12 39963,C(=O)(N=c1[nH]n(C)cc1I)C1CC(c2cn(C)nc2)CN1C(C)(C)C 39964,N1(C(C)=O)CCC(CC(=O)NC2(CF)CN(C(C3SCC=C3C)=O)C2)C1 39965,c1(C(=O)NCC2CCCC(NC(CCC)=O)C2)cc(C)c(C)c2ncccc12 39966,N1(c2snc(C(C)C)n2)CCCOC(CNC(c2n[nH]c(C3CC3)c2Cl)=O)C1 39967,N1(C(CCNC(COC)=O)=O)CCC(C(=O)Nc2cnnn2C)C1 39968,S(=O)(=O)(c1cnc(NC(C2CCCO2)C)c(Cl)c1)NCCc1cccc(C)c1C 39969,n1(CCCC)nc(C)c(C(=O)NCCC(C)NC(=O)CC(CC)OC)c1Cl 39970,C1(Cl)(C(=O)OCC)CC12CCN(Cc1cn(Cc3cnn(C)c3Br)nn1)CC2 39971,CCC(O)C(C)C(=O)N1CC(CCn2cc(-c3ccc(C)cc3C)nn2)C1 39972,C(=O)(C(C)(C)C(C)C)NCC(C#C)OC.C1(=O)C(C)(C)CCN1 39973,C(C(CNC(=O)CCC1CC1(C)C)NC(=O)C=CC(C)=C(C)C)OC 39974,CC1(C)C(NC(c2cc3ccsc3[nH]2)=O)CCN1C(C1CCNC1=O)=O 39975,C=CC(C)C(C)C(=O)N(CC(CO)(CO)NC(c1cc(C(F)F)no1)=O)C 39976,N1(C(CNC(CC)=O)=O)CC2CCC1C1CN(C(=O)Cc3ccsc3)CC21 39977,C(=O)(CCN(OC)C(=O)C(C)(O)COC)NCCN(CC#C)C(C)=O 39978,C1(S(C)(=O)=O)(C(=O)NCC2C(NC(CSC)=O)CC2)CC(O)C1 39979,C1(NC(C2Cc3n(cc(C)n3)C2)=O)CC2CCC(C1F)N2C(C1(C)CC1(F)F)=O 39980,N1(C(c2occ(C)c2)=O)CCC(N=[N+]=[N-])(C(N2CCC(C(F)F)CC2)=O)C1 39981,C(=O)(C(O)CC(N)=O)NCC1CC(OC)CN1C(=O)CCCNC(=O)C1CC1 39982,c1(N(CC(=O)NC(C)CS)C(C)=O)cccc(O)c1F.C1(OCC#C)CCCCC1 39983,C1(C(=O)NCC2CC(c3ncccn3)C2)CCCCC1Cc1ccccc1 39984,N1(C(CCOc2ccc(C)cc2)=O)CCN(C(C2CCCCN2C)=O)CC1C 39985,c1(C(=O)NCC2CCCC(C)C2)cccc(S(C)=O)c1 39986,c1(C(=O)NCCN(C(c2c(OC)c[nH]n2)=O)C)ccc2c(c1)NC(=O)CCC2 39987,c1(C(=O)NC(C(C)NC(c2c(CCC)nco2)=O)C)cc2cccc(C)n2n1 39988,CC1CN(C(C)C(=O)N(CC(=O)NC(C(N)=O)C2CCCC2)C2CC2)C1 39989,C1(NC(=O)Cc2ccccc2)CC(O)CN(C(c2cccc(I)c2F)=O)C1 39990,C(C(CC(C)C)NC(=O)NC(=O)CN1OC(C)CC1=O)NC(C1CC(SC)C1)=O 39991,C(=O)(CCC[N+](=O)[O-])NCCOC1CN(C(C2(COC)CCOCC2)=O)C1 39992,c12cc(Br)c(c(Br)c1)NC(=O)C2.C1(COC(C)=O)CCCN1c1ccccc1 39993,c1(C(c2ccccc2)SC)cc(C(=O)Nc2cccc(OC)c2Cl)c(C)nc1O 39994,C1(CC)CN(C(=O)C=C(C)c2cccs2)CC1NC(C1(CC2CC2)CC1)=O 39995,c1(C(N2C(C(C)(C)NC(c3ccccc3CO)=O)CCC2)=O)cc(N)cnc1Br 39996,CC(O)(Cn1cc(Br)cn1)C(=O)N1CCC(CC(N2CCSCC2)=O)C1 39997,N1(Cc2cc(C)c(I)cc2C)CCC2CCCNC2C1 39998,C1(C(=O)NC(C)C(C)(C)C)CN(C(C2CC(c3ccccc3)C2)=O)CCC1(C)C 39999,c1(C(c2n(CCOCC)nnn2)NC2CC(COC)C2)cc(Cl)cc(C)c1CC 40000,c1(C(=O)OCC)cccc(C(=O)NC2(F)CN(C(C3CC3C)=O)C2)c1 40001,C1(NC(COCCCOC)=O)CC12CCN(C(c1cncc(NC(C)C)c1)=O)C2 40002,N1(C(c2c(C(C)=O)cccc2)=O)CCC(F)C(NC(C2CCC(=O)C2)=O)C1 40003,c1(NC(C2(F)CN(C(c3c(CC)cccc3)=O)C2)=O)cc([N+](=O)[O-])ccc1I 40004,CC1OC2(C(=O)NCC=CCNC(c3ccc(Cl)cc3F)=O)CCC1C2 40005,C12(C(=O)NCC3(SC)CC3)COC(C1)C(NC(c1ccnn1C(C)C)=O)C2 40006,c1(C(N2CC(O)(C(C)NC(c3ccc(C4CC4)o3)=O)C2)=O)cc2c(s1)CCCC2 40007,C(=O)(C(CCC(N)=O)n1cc(C2C3COCC23)nn1)NC(CCC)C 40008,n1(C(C)C)nccc1Cc1nc(-c2ccc(C3CCCO3)[nH]2)no1 40009,C1(C2CCCN(C(=O)Cc3ccc4n[nH]cc4c3)C2)(NC(C=CSC)=O)CC1 40010,C1(C(N2CCN(C(C3CCC(C)CC3)=O)C3(C2)CC3)=O)CC2(CCOCC2)CO1 40011,C1(CNC(=O)Nc2cccc(OC)c2)CC2(CN1C(=O)OC(C)(C)C)CC2(F)F 40012,N1(C(c2c(CC)occ2C)=O)CCN(C(C2(C)CC2F)=O)C2(CCC2)C1 40013,c1(CC(=O)NC(CCNC(CCCOCC)=O)C)cccc(Br)c1 40014,C1(C(C)(C)NC(=O)OC(C)(C)C)CCCC1O.C12(CC1)C(COC)N2 40015,C(=O)(C(O)CC[S+](C)C)NCC1(F)CCN(C(CC2(CSC)CC2)=O)C1 40016,c1(OC)nccc(C(=O)NC2CCN(C(=O)C(C)(C)Br)CC2F)c1Cl 40017,[N-]=[N+]=NCCC(=O)NCCC(F)Cn1cc(C2CC2OC(=N)O)nn1 40018,C(=O)(C(F)C(CC)CC)N1C(CNC(COCCCC)=O)CC(OC)C1 40019,N1(C(=O)CCCC2CCC2)CC2(CCCCN2C(=O)CCN2CCOC2=O)C1 40020,Cc1ncc(C#N)cc1NC(C1(F)CCN(C(=O)C=Cc2cscn2)CC1)=O 40021,C(CN=c1ccnc(N2CCN(C3CCOC3)CC2)[nH]1)N1C(=O)NC(C)(C)C1=O 40022,c1(C(=O)NC(CCNC(Cc2ccn(CC)n2)=O)C)cc(C)cc(O)c1 40023,c1(C(N2CC(NC(=O)C(O)C(F)F)CC(C)(C)C2)=O)c[nH]c2ccncc2c1=O 40024,C1(N)CN(C(=O)C(C)(C)C(=O)C(C(C)CC2CC2)=O)CCC1O.C(C)(C)(C)C=O 40025,CC(C)C(C)CC(=O)N1CCC(CC(F)C(=O)NOC(C)C)CC1 40026,c1(C(=O)NCC23N(C(C4COC(=O)O4)=O)CC(C2)C3)c[nH]nc1[N+](=O)[O-] 40027,N1(C(C(C(C)C)O)=O)CC=C(CCNC(c2cc(F)c(C(F)F)c(F)c2)=O)CC1 40028,c1(C(N2CC3CC(NC(CSc4n(C)cnn4)=O)C3C2)=O)ccc([N+](=O)[O-])cn1 40029,C1(C(N(C(CCNC(c2c(C)ncnc2)=O)C)C)=O)COc2ccc(F)cc2C1 40030,c1(NC(C(N2C(C)CC(CO)CC2)C(C)C2CCC2)=O)ncc([N+](=O)[O-])cc1Cl 40031,O=C1CN(CC(=O)NCC2C3CN(Cc4csc(-c5ccco5)n4)CC23)C(=O)N1 40032,c1(C(=O)NCC2C=CC(NC(C(CC)SC)=O)C2)c(Cl)ccc2c1OCO2 40033,c1(CN2C(CCNC(=O)CC3(CC(=O)OC)CC3)CCCC2)cccn2cnnc12 40034,C12(C(=O)NCc3ccnc(C)n3)CCC1CN(C(C1CCCC1F)=O)C2 40035,C(=O)(CC(C(C)OC)NC(C1CC1CN(C)C)=O)N(C(CC)CO)C 40036,C(C(=O)N(C)CCN1CCCC1)(c1ccoc1)NC(C(C)SC(C)C)=O 40037,c1(C(N(C(C)CCNC(=O)CC2CCC(F)(F)C2)C)=O)cccc2c1CCC2=O 40038,C(C(COC)C(=O)N1CC(C(O)C(=O)NCC2(OC)CCC(C)C2)C1)OC 40039,C#Cc1c[nH]nc1C(=O)NCC=CCNC(c1ccnnc1C)=O 40040,C1(NC(C2(COC)CCCC2)=O)COCCN(C(=O)Cn2cc[n+](C)c2)C1 40041,C(=O)(C1=CCCCO1)NC(C(C)OC)C(=O)NCC1CC(=O)NC(C)C1 40042,C1(CNC(c2cnc(CCC)s2)=O)(OC)CCN(C(=O)CCc2ncco2)C1 40043,c1(C(=O)NC2CCC(NC(c3ccnn3CC(F)F)=O)C2)cnc(O)c(Cl)c1 40044,c1(OC)ccc(Cl)cc1CC(=O)NCC(C)(CC(C)C)NC(C1CC=CCC1)=O 40045,N1(C(c2nc(CNC(C(C)C3CCCC3)=O)oc2)=O)CC(C2CCCCC2)C1 40046,C12(C(N(C3CCCN(C(c4c(CC)c[nH]n4)=O)CC3)C)=O)CC3CC(CC1C3)C2 40047,C12(NC(C(=O)NC(c3ccc(F)cc3Cl)C)=O)CCC(CN)(C1)OC2 40048,C(CCC)(C(=O)NC1CC(NC(c2ccc(C(C)=O)cc2)=O)CC1O)=CCC 40049,C1(C(=O)NC2CC(NC(CC(C=C)(C)C)=O)C2)COc2ccc(OC)cc2C1 40050,Cc1ccc(=O)n(CC(=O)NCCc2ccc(OCC(C)C)cc2)c1 40051,C1(C(=O)NCCC(C)NC(=O)C(c2ccc(F)cc2)(F)F)CCCCN1C 40052,C1(C(=O)NC(CC)C(=O)NC)CNC(=O)CN1C(=O)C1=COCCC1 40053,c1(COC)nc(NC2CN(C(c3ccn(C)n3)=O)CCC2CO)cc(O)n1 40054,Cc1nn(C)c(NC(=O)CC(P(C)(C)=O)c2ccccc2)c1C=O 40055,c1(C(=O)Nc2ccnc(N3CCOC(C(F)(F)F)C3)c2)cc2c(cc1O)CCCC2 40056,CC(C)CC(O)C(=O)NC1CCCC1(C)CNC(=O)CC1CCC(C)(C)CO1 40057,C(=O)(C1CCCn2ccnc21)NCCN(C(CCC(C)(C)C#N)=O)C1CC1 40058,N1(C(C=CCNC(C2CC(C)(O)C2)=O)=O)CCc2ncccc2C1 40059,C1(c2nn[nH]n2)(CN(CCC(C)C)CC)C=CCN1C(=O)COCCCN=[N+]=[N-] 40060,C(c1ccc(F)c(F)c1)=C(C)C(=O)NC1CN(C(c2nc(Cl)c(Cl)s2)=O)CC1C 40061,c1(C(=O)NC2CN(c3nc(OC)c(C)cn3)CC2C)ccc2ncsc2c1Br 40062,Nc1ccc(C(=O)NCC(C2CC2)NC(c2ncccn2)=O)nc1N 40063,N1(C(c2n[nH]c(CC)c2C)=O)CC(C(=O)NCCC2CC2C)OC(C)C1 40064,C12(CC)CC1CN(C(C1CCC=CC1NC(=O)CCC1CCOCC1)=O)C2 40065,c1(C(=O)NCC(C)N(C(=O)C(=O)NC2CC2)C)ccc2nnc(O)n2c1 40066,c1(C(=O)NCc2c(C(N(CCCCCC)C)=O)nco2)cccc(=O)o1 40067,c1(C(N2CC(C)N(C(C3CCN3C3CCCC3)=O)CC2)=O)cccc([N+](=O)[O-])c1 40068,Cc1ccc(C(F)(F)F)cc1C(C)C(=O)NCC(C1(C)OCCO1)N 40069,O=C(C(O)C(O)c1ccc(O)cc1)OCc1noc(-c2ccco2)n1 40070,Cc1ncsc1C=CC(=O)N(CC(C)(C)NC(C1CCN(C(C)C)C1)=O)C 40071,c1(CNC(C2(C(N3CC(c4ccccc4)C3)=O)CCCC2)=O)ncccc1N.CSC 40072,C1(C(=O)NCC2C(CNC(CC=CC)=O)C2)CCc2ncsc2C1 40073,c1(C(=O)NC2C(NC(c3cccn4cnnc34)=O)CC2)cnc2[nH]ccc2n1 40074,Cn1nc(C2CC2)nc1CC(=O)N(C1CCCCC1)CC.C(=O)(C(=O)C1CCCC1)N 40075,N1(C(c2c(C(=O)OC)[nH]cc2)=O)CCC(NC(c2cc(=O)on2C)=O)CC1C 40076,C1(C(=O)NCC(=O)NCC2COC3(CNC3)C2)CCCC12CCN(O)C2 40077,c1(NCCC2CC(NC(C3CCCN(C(=O)OC)C3)=O)C2)ccc2n[nH]cc2c1 40078,c1(C(N(CCC2CCCNC2)CCn2ncc(C)c2)=O)cccc(P(C)(C)=O)c1 40079,c1(C(N2CC(CNC(C3(O)CCSC3)=O)C2)=O)ccc(S(=O)(=O)NC2CC2)cc1 40080,Cc1ccsc1-c1cn(CC2(C3CCC3)NC(=O)N2)nn1 40081,CCCC(CC(C)C)C(=O)NCC1(CN(C)C(c2cc(N)ccn2)=O)CC1 40082,NS(=O)(=O)C1CN(C(=O)NC2CCOC2c2ccc(Cl)c(F)c2)C2(CCC2)C1 40083,c1(CC(=O)NCc2nc(CNC(C(C)(C)C3CCC3)=O)sc2)ccc2c(c1)CC2 40084,c1(C(=O)NC2C(CNC(C(CCC)OCC)=O)CCC2)cn(C)c(C)cc1=O 40085,CC1(C)C(CC(=O)NCCC2C=CCC2)CCN1C(=O)CCCC1CCC1 40086,Cc1nc(COC)ncc1C(=O)NCCCN(CCO)C(c1ccco1)=O 40087,CC(CNC(C1COCCC1C)=O)C(F)C(=O)NC1(CC2CCC2)CC1 40088,n1(CC(C)C)c(SCC2NCCC2C2CC2)nc2sc3c(c2c1=O)CCC3 40089,C=CCC(F)(F)C(=O)NCC(C)CC(=O)N(C(C)CN(C)C)C 40090,N1(C(CN(S(C)(=O)=O)C)=O)CCCN(C(C2CC2F)=O)C(c2ccccc2)C1 40091,CC(C)C(O)C(F)(F)C(=O)NC1CCC(CNC(=O)Cc2ccc(Cl)s2)C1 40092,c1(C(=O)NC(CNC(C2C(=C)CC2)=O)CCOC)c(C)cc(C)oc1=O 40093,C1(NC(CCOCCCNC(C(C)c2cccs2)=O)=O)CC2(C1)CC(C)(C)C2 40094,C1(CCNC(C)=O)CCN(CCNC(c2cc(C)c(C)s2)C)CC1 40095,CCCCCC(C)CC(=O)NCCC(O)CNC(c1ncoc1C1CC1)=O 40096,CC(C)CC(C(=O)N(C)CC1(CO)CC1)NC(C1CCC(=O)N(C)C1)=O 40097,C(CCSC1CC1CSC)(C(=O)NCc1cn(CCCc2nncs2)nn1)N(C)C 40098,C1(C(N(CC)CC2CCC2)=O)CCC(O)CN1C(=O)CCCC(C)C 40099,C1(C(N2C(CC(=O)NC)COCC2)=O)CC2OCCC2N(C(=O)CCCCCl)C1 40100,C(=O)(C1OCCn2ccnc21)NC(C(C)C)CNC(c1coc2c1CCCC2)=O 40101,Cc1nn(CC(=O)N(C2CN(C(C3(C)CCC3)=O)C2)C)c(C)c1Br 40102,CCCC(CCC)C(=O)N1CCN(C(c2cc(SC)cc(Br)c2)=O)CC1 40103,Cc1nc(N2CC3CN(C(c4cc(Cl)c(Br)c(Cl)c4)=O)C3C2)c2c(n1)CCC2 40104,Cc1cc2sc(CC3=NOC(C(=O)NC4CCC4)C3)cc2s1 40105,C(=O)(C(C)(C)C(C)(F)F)N1CCC(N(CCOC)C(C2CC2C2CC2C)=O)CC1 40106,N1(C(CCOCCC)=O)CCC(CN2CCN(C(c3cscc3C)=O)CC2)CC1 40107,c1(C2(CNC(COC)C3CC3)CC2)nnc2n1CCNC2=O 40108,N1(C(C(CCCNC(C(C(=O)OC)OC)=O)O)=O)CC2(CNC(=O)OC2)C1 40109,C1(NC(C(CC)CNC(c2coc(CO)c2)=O)=O)(CC)CCCN(C(C)=O)C1 40110,c1(C(=O)NCCC2CC(NC(C3CC3Cl)=O)C2)cc2c[nH]cnc-2n1 40111,Cc1ccc(F)c(C(N2CCCC(C)(CNC(c3c[nH]c(C#N)c3)=O)C2)=O)c1F 40112,O=C1CCC2(CNC(c3cccc(-c4nnco4)c3)=O)CC3(CC3)CN12 40113,C1(OC)CN(C(C2(C)C=CCN2C(c2nnsc2C)=O)=O)CCO1 40114,N1(C(c2cc(C)ncc2)=O)CC(C(=O)NCC2CC(=O)N(C)C2)CC(F)C1 40115,c1(C(N(C2CCCN(C(c3csnc3Cl)=O)C2)CCO)=O)ccc2[nH]ccc2c1 40116,c1(-n2nnc(C(=O)OC(c3cccc(Br)c3)CCC)c2C)c(F)cccc1F 40117,n1(C(C)C)ncc(C(N2CCCC(OCCNC(=O)CCF)C2)=O)c1C1CC1 40118,N1(C(C2(COC)C=CCC2)=O)CCCC(C2CN(C(c3scc(C)c3Cl)=O)C2)C1 40119,N1(C(c2c(C)[nH]cc2)=O)CCC2CC2(C(=O)Nc2cc(O)ccc2F)CC1 40120,CC(CCNC(=O)C=Cc1ccco1)CCNC(C1COCCN1C)=O 40121,c1(C(N2CC(C(C)NC(c3c(C)scc3)=O)C2)=O)cnc2ccccn12 40122,C1(NC2(CC(=O)N(CC(=O)OC(C)(C)C)C)CCC2)CCCCCC1 40123,c1(C(N2C3C(CNC(C4C(C)CC4)=O)C(CCC3)C2)=O)nc2n(c1Cl)CCCC2 40124,N1(C(C(CCC)OCC)=O)CCc2nc(CNC(=O)Cc3cnc[nH]3)sc2C1 40125,C=C(C)CCCC(=O)N(CCNC(c1cnnc(O)c1)=O)Cc1cccc(Cl)c1 40126,c1(C(=O)NCCCC#N)ccc(C2CCC23CCC3)cc1 40127,C12(CC(=O)N(c3ccc(CO)cc3)C)CCC1CN(C(c1ccncc1N)=O)C2 40128,C(=O)(C(C#N)CC)N(CC(=O)NC1CCN(CC)C1)CCOCCO 40129,C12(CC)CC3CCC(C1)N3C(=O)N2.c1(C(=O)OC(C)(C)C)cccc2cncn12 40130,c1(N2CCC(NC(C3C(CCC(C)C)CCC3)=O)C2)cc(F)ccc1F 40131,CC(C)(C)CC(C)(C)C(=O)N1CCC(C(=O)NCCC(F)F)C1 40132,C1(O)(C(=O)NC2C(OCC)COCC2)CC(C)(C)C1.c1(N2C(=O)C2)cncc(Cl)n1 40133,N1(C(C2CN(C)C(=O)C2)=O)CC(NC(=O)COc2ccccc2)CC(F)C1 40134,c1(C(N(CCNC(c2cc(C)n(C)n2)=O)C)=O)ccc2ccccc2c1 40135,c1(NC(C)=O)ccc(C(=O)NC23CC2CN(C(=O)C(O)C(F)F)C3)cc1 40136,CCC(C)C(O)CC(=O)NCC(C)(C)OCCNC(c1cnc2ccccn12)=O 40137,C1(NCc2cn(CCC(=O)N(C3CCN(CC)CC3)C)nn2)CCCC(C)(C)C1 40138,c1(CC(=O)N(C)CC2(NC(c3nocc3Cl)=O)CC2)ccc(Cl)c(Cl)c1 40139,N1(C(CC(CC)C2CCC2)=O)CCC(CC(=O)NCC2CNC(=O)O2)C1(C)C 40140,c1(C(=O)NCC(C2CCCC2)NC(CC=C(C)C)=O)csc(-c2ncc[nH]2)n1 40141,Cn1ccc2sc(C(=O)NC3COCC3NC(c3cc4n(n3)CC(F)C4)=O)cc12 40142,N1(C(=O)Cn2cccc2)CC2CCC(C1)N2CCOCC1CCCO1 40143,c1(C(C(=O)NC2CCCC2)N(CC(C)C)CCCO)cnc2n1CCC2 40144,N1(C(c2c(C)c[nH]n2)=O)CC2=C(C1)CN(C(c1cnc(C(F)F)c(C)c1)=O)C2 40145,c12cc(F)c(C(F)(F)F)cc1N2.CCC(F)(F)C(=O)N1CCCC1.C1C(=O)N1 40146,c1(CNC(C2N(C(COCCCCC)=O)CCOCC2)=O)ccc2nccn2c1 40147,c1(NC(CCC2(NC(C3CCCC(=O)O3)=O)CCCC2)=O)cccc2c[nH]nc12 40148,C(=O)(C1=CCC(C)(C)CC1)NCC1(F)CCCN(C(CSCC=C)=O)C1 40149,c1(O)cc(C(F)(F)F)c(C)c([N+](=O)[O-])c1.C(=O)(CN)OCCNC(=O)OC 40150,C1(NC(C2(CCC)CC2)=O)CCCCN(C(=O)CCOCC2CCCO2)C1 40151,CC(C)C(CC(=O)N(C1CCSCC1)C)NC(=O)CCc1cn[nH]c1 40152,C(=O)(CN1C(=O)CCc2ccccc21)NCC1C(NC(CC2CN(C)C2)=O)CC1 40153,c1(CCNC(=O)NC(CC(CC)C)C)ccc(Br)cc1F 40154,CC1(C)COCCC1CNC1CC1C.C(=O)(CCCCCF)NC(=O)C1CC1 40155,C1(C(N(CCN(CCC)C)CCOC)=O)CCC1C(=O)OCC 40156,N1(C(Cc2c(C)cnn2C)=O)CCN(C(=O)COc2ccsn2)CC(O)C1 40157,C(=O)(C(C)C(C)NC(c1cc(C2CC2)no1)=O)NCCOCCCC#C 40158,c1(C(N2C(C)CC(CNC(c3snc(Cl)c3Cl)=O)C2)=O)ccnc2ncnn12 40159,N1(C(C(C)(C)F)=O)CCC2(CCN(Cc3cc(Sc4ccc(F)cc4)on3)C2)C1 40160,N1(C(C2C(C)(C)CCN(C(=O)CCC3CCCC3)C2)=O)CCC2(CCCCO2)C1 40161,c1(NC(CC2CCC(N)C2)=O)cccc(N2CCOCC2)c1 40162,Cc1ncc(C(=O)NC(C)(CO)C(=O)NC2CC2CCOC)c(C)n1 40163,C1(NC(C(C)n2cccc2)=O)CC(C)N(C(c2ccc(C(F)F)nc2)=O)C1 40164,N1(C(COCCOC)=O)CCN(C)C(CNC(C2CN(C)CCO2)=O)C1 40165,C1(NC(C2(C)COC2)=O)CCC2(CC1)CCN(C(=O)CC1CCCC1(F)F)CC2 40166,C1(NC(=O)C(CC(F)F)N2CCOCC2)CCN(C(=O)C(Cl)=CCl)CCC1(F)F 40167,Cc1csc(C(F)(F)C(=O)NC(C)C(C)NC(C2CCCC2)=O)n1 40168,c1(CN2CCN(C(C(c3ccccn3)C)=O)CC2C)ccc2c(c1)C(=O)NC2 40169,c1(-c2cn(CC)nn2)nc(C(C)C2CC2)nn1C1CCCOC1C 40170,N1(CC(N2C(C)CC(CC(N3CC(NCCOC)C3)=O)C2)=O)CCNC(=O)C1 40171,c1(N2CCCC(NC(C3C(CC)OCC3)=O)CC2)cc2ncnn2cn1 40172,c1(C(=O)NCCCN(C(C2C(C=C)C2)=O)CC)ccc2c(c1)OCC2 40173,Cc1no[nH]c1=NC(=O)C1(C)CCN(C(C2CC2c2ccccc2)=O)C1 40174,c1(C(=O)NCCC2N(C(CSC)=O)CCSC2)ccc2c(Br)nn(C)c2c1 40175,N1(C(C(C=C)OC)=O)CC(CC(=O)NCC(C)(O)CCC)C2(CC2)C1 40176,CN1CCN(C(C2N(C(=O)Cn3ncnn3)CCCC2(C)C)=O)CC(O)C1 40177,C1(C(N(C(CC)CC(=O)Nc2cccc(OC)c2)C)=O)CCC(N=[N+]=[N-])C1 40178,c1(NC(C(CC)SC)=O)ccc(F)c(NC(=O)CCC(=O)c2cccs2)c1 40179,c1(CC(C)C(=O)Nc2nc(-c3ccc(Cl)s3)cs2)ccc(F)c(F)c1 40180,CCCCC(C(=O)NC(C)CNC(=O)OCC)NC(=O)C#CC1CCC1 40181,N1(CC)CCN(CCC(=O)NC(C)(C)C(C)NC(=O)CC2CCN(C)C2=O)CC1 40182,CC1CCC=C1C(=O)N(C)CC1(CNC(=O)C(C)Oc2ccc(Cl)cc2Cl)CC1 40183,c1(OCC(=O)N(CC(C)O)CCNC(C(C)(C)OCC)=O)ccc(Cl)cc1 40184,C1(CC)CN(C(=O)CCc2c(C)n[nH]c2C)CCN1C(c1cc(Cl)ccc1F)=O 40185,Cc1[nH]c2ccccc2c1C(=O)NC1(CF)CCN(Cc2nn(C)cc2Br)C1 40186,C=CC1CN(C(=O)C(CN(C)C)NC(=O)CCSCC)CCO1 40187,c1(NC(=O)CC2CCCN2C(c2cc(OC(C)C)ncc2)=O)cc(F)cnc1Cl 40188,C1(=O)CCCCCN1.c1(CNC(=O)NCC(CC)OCCN)ccc(OC)cc1 40189,C(=O)(N=c1nn[nH]n1CCC(C)C)NC(c1ccc(Cl)cc1)CCC 40190,C(=O)(C(C)(C)C(=O)NCC#N)N1CCC(N(C(=O)C(F)CC2CC2)CCC)CC1 40191,C12(COC)COC(C(N3CCCCC3CNC(=O)Cc3ccccc3C)=O)(C1)C2 40192,c1(CC(C)C)cc(NCC(C)(C2CC2)NC(C2CCC(CO)CC2)=O)ncn1 40193,C(C(=O)N1CCCC1C1(NC(C2CCCC(C)(C)C2)=O)CC1)(C(C)(C)C)SC 40194,c1(C(=O)NCc2cn(CCNC(C3C(C)C3(F)F)=O)nc2)csc(Cl)c1Cl 40195,c1(OCC#C)ccc(Br)c(C(=O)OCc2nnc(-c3cccc(N)c3)o2)c1F 40196,C1(C(N(C(C)CN(C)C)C)=O)N(C(c2cnnc(O)c2)=O)CCCC1(C)C 40197,c1(C(N(CC(CNC(Cc2c(C)noc2)=O)O)C)=O)cncc(-n2cccn2)n1 40198,N1(C(=O)Nc2cc(CO)ccc2F)CCC2CCCN(Cc3ccncc3)C2C1 40199,C1(C(N(CC(=O)NCC(CCOC)O)C2CCC2)=O)CCCC(O)C1 40200,C(CCCCCCC(=O)NC(CNC(=O)CC(C)C(C)C)C1CC1)SC 40201,c1(OC)ncc(C(=O)NC2CN(C(=O)COCC3CCCO3)C2)nc1C 40202,CC(O)(CCc1nc(-c2ccc(-c3ccccc3)cc2)nn1CC1CC1)C(F)(F)F 40203,c1(OCCNC(C2CC2(C)C)=O)ccc(C#N)cc1.N1(C(C(C)N)=O)CCCC1 40204,N1(C(CCOC(C)=O)=O)CC(C2CC2C(=O)N(C2CCOCC2C)C)C1 40205,N1(C(CC)=O)CCN(C(c2cnc(C(C)Br)s2)=O)CC1C 40206,C1(NC(Cn2c(C)c(Cl)cn2)=O)CC2CCC1N2C(c1cnn(C(C)C)c1)=O 40207,CC1=C(C(=O)NC2CCC(NC(c3cn(C)nc3Cl)=O)C2)C=C2CCCN=C2N1 40208,CCCCCCOC(C)C(=O)NCC(CC)NC(c1ccnn1C1CCCC1)=O 40209,C1(C)(C(=O)NCC2CCN(C(COCC)=O)C2)CNC(=O)C1 40210,N1(C(C2(CC)CCCC2)=O)CCC(O)(CN(C(=O)CC2CCN(C)C2=O)C)CC1 40211,N1(C(C2(C(C)C)CCN(C(=O)C=CC(C)(C)SC)C2)=O)CCCCC(OC)C1 40212,C1(C2CCN(C(C3CC(C)C3)=O)CC2)(NC(C(CCCC)C(=O)OC)=O)CCC1 40213,C(c1ccc(SC(C)CCNC(=O)C(CC)n2ccnc2)cc1)=C(CC)CC 40214,C1(C(=O)OC)CC=CCN1C(=O)COC(C1CC2CCCC12)=O 40215,C1(CNC(C(CC#C)C2CC2)=O)(NC(c2nccnc2C)=O)CC2CCC1CC2 40216,C1(CCCNC(C2(SC)CC2)=O)CCCCN1C(C1CC12CCC2)=O 40217,n1(CCC)cccc1C(=O)NCC1OCCC1C(=O)NCC(O)COC(C)C 40218,C(C(C)C(=O)NCC(C1CC1)NC(c1ccn(CCF)n1)=O)SC 40219,N1(C(c2c(CC)ccs2)=O)CC(CNC(c2nsnc2O)=O)C1(C)C 40220,C1(C#N)(C(=O)NCc2cn(C3CN(C(CCC=CC)=O)C3)nn2)CC2CC2C1 40221,Cc1[nH][nH]c(=N)c1C(=O)N(CCCCCCNC(c1coc(C(F)(F)F)c1)=O)C 40222,C1(CC(=O)N(CC)CC2CCCN2C(C2CC=CC2)=O)CCC(C)(C)O1 40223,CC1CN(C(=O)C(c2ccsc2)N(C)C)CCC1NC(=O)C(C)(C)C1(O)CCOC1 40224,C=CCCCC(C(=O)Nc1cccc(NC=O)c1)NC(=O)CCC(=O)CC 40225,n1(CC(=O)NC2C(NC(C(F)=CCC)=O)CC2)cc(Cl)c(C)n1 40226,N1(C(c2ccc(C)c(F)c2)=O)CCN(C(c2cncc(F)c2)=O)CC2(CC2)C1 40227,C(c1cnn(C)c1)=CC(=O)NC(C=CC(=O)N(C1C(C)CCC1)C)(C)C 40228,C1(C(N(CC(=O)NCC(C)OCCO)CCOC)=O)CC1 40229,C1(C(N(C(CC)C)C2CCC2)=O)COCCN(C(C2(C#N)CC2)=O)C1 40230,C(CCCCC(=O)NC1CC2(C1)CC(NC(c1cc(CO)oc1C)=O)C2)SC 40231,N1(C(c2ccc(OC)o2)=O)C2CCCC1CN(C(=O)CCS(N)(=O)=O)CC2 40232,C#CC1(C(=O)N(CCCN(C(=O)C(CCC2CC2)OC)C)C)CC(=O)C1 40233,CCCC(C(O)C(=O)NCC)NC(=O)CN(C)C(=O)OCCC1COCC1O 40234,N1(C(CCCCC)=O)CC(C(=O)NOCC(=O)OC(C)(C)C)C(C)CC1C 40235,C(=O)(CCCCC#N)NC1CCCN(C(C(CC#C)O)=O)C1 40236,N1(C(C2(CC=C)CC=CC2)=O)CC2(CCC2NC(=O)CSS(C)(=O)=O)C1 40237,C1(C(=O)OCC)CN(C(C2CC(C)N2Cc2ccc(C)o2)=O)CC1C 40238,C1(CNC(C(N2C(=O)CCC2=O)CC)=O)CC(C)(C)CN1C(=O)CCOC1CC1 40239,C1(NC(c2c(SCC=C)cccc2)=O)CC(C)CN(C(c2n[nH]cc2OC)=O)C1 40240,C(CCCC(=O)NC(c1ccc(C)s1)C)NC(c1cc(OC)n[nH]1)=O 40241,C1C(C)(C)C(=O)N1.C(CC(C)(C)OC)NC(C1CC(COC)C1)=O 40242,Cc1nc(C(C)C)ccc1C(=O)NCC1CCCC(NC(=O)CNS(N)(=O)=O)C1 40243,N1(C(COCCCC)=O)CCC(C)(C)C(NC(=O)CCN(CC(F)(F)F)C)C1 40244,C1(C(N2CC(CCc3cn(CC)nn3)C2)=O)COC2(COC2)C1 40245,C1(CNC(c2ncn(CC)c2)=O)CC(C)N(C(C2CCC(=O)N2C)=O)C1 40246,Cc1ccccc1Cn1cc(C2CCCN2C(c2c(Br)noc2C)=O)nn1 40247,C(CC(=O)Nc1cc(COCC)no1)NC(=O)N.C(CN(C)C)OC 40248,c1(NC2CCCC2C(N2CC(O)(CC(=O)Nc3ccccn3)C2)=O)ccccn1 40249,c1(OC)ccc2cc(C(=O)NC3CCN(C(=O)CCC4CC4(C)C)CC3)[nH]c2c1 40250,C1(NC(Cc2nc(=N)[nH][nH]2)=O)CCC2CCN(C(c3csc(Cl)n3)=O)C12 40251,c12cccnc1C(=O)N1CCC(F)(C1)c1cn(nn1)C(CC(N)=O)O2.C(=O)O 40252,N1(C(C=Cc2c(C)coc2C)=O)CCC(C)(C)C(CNC(=O)COC2CC2)C1 40253,C1(C2CCOCC2)(C(N2CC3C(NC(C(C(=O)OCC)C4CC4)=O)(C3)C2)=O)CC1 40254,c1(C(=O)NC(c2ccccc2)C(C)NC(C2CCNC2=O)=O)cc(Cl)ncc1N 40255,C1(NC(=O)Cc2cccnc2O)C2CC3CN(C(C4C5CCCCC45)=O)C1C3C2 40256,N1(C(CCNC(C2(C(=O)OCC)CCC2)=O)=O)CCC2(CO)CCCC12 40257,C1(C2C(C)(Br)C2)CCN(C(=O)CC2CC(F)CN2CCCCN(C)C)CC1 40258,c1(C(=O)NC(CCOC)CNC(=O)CC(C)CF)ccc(S(N)(=O)=O)c(F)c1 40259,C(=O)(C1=CCCSC1)NC1(CNC(=O)COCCCF)CCOCC1 40260,N1(C(c2cc(C(CC)CC)no2)=O)CC(NC(c2cnsn2)=O)CC(F)(F)C1 40261,C12(C(=O)NCC#CCNC(CC(CC)C3CCC3)=O)CCCC1CC(=O)C2 40262,CC1(C)CCC(CNC(=O)C(C2CCCCC2)F)N(C(=O)CN2CCSCC2)C1 40263,c1(C(N2CC(C)C(NC(c3cc[nH]n3)=O)C2)=O)cccc(C(N)=O)c1N 40264,N1(C(C(CC)(CC)CC)=O)CC2CCN(C(=O)C=C(C)c3cnn(C)c3)CC2C1 40265,N1(C(c2n[nH]c(C)c2O)=O)CCC(CNC(=O)C(c2ccc(F)cc2)C)C12CC2 40266,C1(C(=O)NC(C)C(C2CCCCC2)NC(c2csc(Cl)n2)=O)(OC)CS(=O)(=O)C1 40267,C1(C(N(C)CC2CCC(CNC(=O)COC3CCOC3)CC2)=O)CCCCC1(F)F 40268,c1(C(=O)Nc2snc(C(=O)OC)n2)cc(C#N)ccc1F.C12(O)CN(C1)N2C 40269,C1(NC(CC(C)(C)F)=O)C2CCN(C(=O)COc3ccccc3C#N)CC12 40270,CCC(C)(CCC(C)C)C(=O)NC1CC(CC(N2CCC(O)C(O)C2)=O)C1 40271,c1(-c2cc(C)[nH]c2C)csc(=Nc2cccc(Cl)n2)n1CCC1CCSC1 40272,C=CCCC(c1nnnn1C1CC1)NCc1cc(C2CCCC2)no1 40273,C=CC1CN(C(c2cnn(C3CC3)c2)=O)CC1NC(C1(C)CCCS1(=O)=O)=O 40274,C=CCC(CC(=O)N(CC(O)CC)C)NC(=O)C(C)COCOC 40275,c1(COC(C2COC(C3CC3)C2)=O)nc2cc(Cl)cnc2[nH]1 40276,C(=O)(C(C)(C)C1=CCN(C(=O)CC2CCCC2C)C1)NC1CC(SC)C1 40277,CC(O)C(C)(C)C(=O)NCC1CCCCN1C(c1cc(Br)cs1)=O 40278,c1(OC)ncc(C(=O)NCC2(O)CCN(C(c3n[nH]cc3C)=O)C2)c(C)n1 40279,c1(N2CCCC(N(C)C(C3CCCNS3(=O)=O)=O)CC2)ncc2ccsc2n1 40280,C12(C(=O)NCCC3CCCC3)COCC1CN(C(=O)CCc1csnn1)C2 40281,C(=O)(CC(C)CC(C)C)NCC1(C(=O)NCCC(CCC)O)CCCCC1 40282,c1(C(=O)NC2CC(N(C(=O)COCCO)C)C2)c(F)ccc2nc[nH]c12 40283,c1(CC(=O)NCCN(c2ccc(F)cc2)CC)ccc(F)c(C(F)(F)F)c1 40284,N1(C(CCCCN(C)C)=O)CC2(CCCC2)C1C(N1CCC2(CC(F)C2)C1)=O 40285,Cc1cn2cc(CC(=O)NCC(C)CNC(=O)CC(C)CF)nc2s1 40286,c1(CSCC(=O)NC(c2ccccc2)CNC(C(C)O)=O)nccc(C(F)F)n1 40287,n1(CCN(C)CCNC(=O)C(F)(F)C2(O)CCC2)cc(CS(=O)(=O)C2CC2)nn1 40288,C1(NC(c2snnc2C2CC2)=O)CCCC1CNC(=O)CCSC1CCCC1 40289,c1(C(=O)NCCCNC(=O)COc2ccsc2)ccc(SC2CCC2)s1 40290,CC1=C(C(=O)N2CCC(O)(C(C)NC(=O)C(C)N(C)C)C2)CCO1 40291,Cc1ccc([N+](=O)[O-])cc1C(N1CCC(F)(F)C(NCc2cnn(C)c2C)C1)=O 40292,N1(C(CC(C)C2CC2)=O)CCC2(C=C(C(=O)N(C)C)C2)C1.C12CN(C1)C2(C)C 40293,C1(NC(=O)CCOCCCNC(C2CCCC(CN)C2)=O)C2CCC(F)(F)C12 40294,c1(CC)sc(C(=O)NCC2(C(C)(C)O)CN(C(c3cc[nH]c(=N)c3)=O)C2)cc1C 40295,C(CCCC(=O)N1CC(C(=O)NC2CC(CCF)C2)OC(C)C1)(OC)OC 40296,CCCCC(CC)C(=O)N1CC(C(=O)NCCN2CCC2)CC1(C)C 40297,C1(C(N(CC(CNC(c2ccn(CCCC)n2)=O)(C)C)C)=O)C2CCC(=O)C12 40298,c1(C(N(CC2N(C(CCCC#CC)=O)CCOC2)CC)=O)cnc2[nH]nnc2c1 40299,C(=O)(C1CCCn2ccnc21)NC1CCN(C(COC)=O)CCC1(F)F 40300,c1(NC)ccc(C(=O)NCC2CCN2C(=O)Cc2cnc(C(F)(F)F)s2)c(C)c1 40301,CC1(NC(c2ccc(F)cn2)=O)CCN(C(=O)CC=C(Cl)Cl)C1 40302,Cc1occc1C(=O)NC(C1CCCN1C(c1cc(C(F)F)on1)=O)(C)C 40303,C#Cc1cncc(NC(=O)NCC(=O)NCCc2ccc(Br)cc2)c1 40304,c1(C(C2C(C(=O)NC(=O)OC)C2)=O)[nH]c(C)c(C(N2CC(CC)C2)=O)c1C 40305,C(=O)(C(CNC(C1CCCC1CNC(c1cnn(CCO)c1)=O)=O)OC)NC 40306,Cc1c(C(N2CC3CN(C(=O)COC4CC4)CC(C2)O3)=O)nc2sccn12 40307,C1(C(=O)NCC(CNC(Cc2c(C)ncnc2C)=O)C)OCC2CCCCC12 40308,CCC(CC(=O)NC1CCC(C)(NC(=O)Cc2cnns2)CC1)CC(C)C 40309,c1(C(N2CCC(N(C(C3(c4cc(C)no4)CC3)=O)CCO)C2)=O)ccc(F)c(Cl)c1 40310,CCCCC(CC)C(=O)NC1CC(CO)N(C(=O)CN2CCCC2)C1 40311,C(=O)(C1=CC2(CN(C(=O)C(O)CN3CCCC3)C2)OC1)NCC(COC)(C)CO 40312,c1(C(=O)OC)ccc2ncn(C)c(=O)c2c1.C12CN(CC13CCC3)C2 40313,CCCCCC(C(=O)NC1CCC(NC(=O)Cc2cn(C)nc2Cl)CC1)C(C)C 40314,c1(C(=O)NCC(C)CN(C(COC)=O)CC(N)=O)oc2ccccc2c1CS(C)=O 40315,c1(C2CCC(C(=O)NCCNC(CCC=CC)=O)C2)ccc(F)c(F)c1 40316,C1(C(N(C2CCN(C(=O)C=C(Cl)Cl)CC2)CC)=O)C2CCC1(c1ccccc1)C2 40317,N1(C(C)=O)CCCC1(C)C(N1CCOCC1)=O.C12CCC(CC1)C(=O)NC2 40318,C1(CC(=O)NCCN(C(c2cncc(C)n2)=O)C)CCCCC1(C)C 40319,C(C(F)(F)C(N)=O)NC(C1(CC)CN(C(=O)CN2CCOCC2)C1)=O 40320,Nc1cc2c(cc1C(=O)NC1CCC(NC(C3CC3(Cl)Cl)=O)CC1)CCC2 40321,C(=O)(CCCC(F)(F)CO)N1CC(C(C)NC(C23CCC(CC2)CC3)=O)C1 40322,C1(F)(CNC(C(C)OCCC#C)=O)CCN(C(=O)C=Cc2cn(C)cn2)CC1 40323,c12ccc(cc1S(C)(=O)=O)CN1CCN2CC1.CN=c1[nH]nc(C)s1.OC 40324,Cc1nc(C=CC(=O)N(C2CCCN(C(C3CCCS3(=O)=O)=O)C2)C)cs1 40325,c1(CC)ccc(C(N2CC(CNC(C3(C)CC=CC3)=O)C3(CC3)C2)=O)cc1C#N 40326,N12CCC(C1)N(C)C(C)C2=O.C(C(F)(F)F)NC(=O)C(N1CCCC1)C1CC1 40327,c1(NC(N)=O)ccc(Cl)c(C(=O)NCCN(C(C2CC2Cl)=O)C2CC2)c1 40328,c1(C(N2CC(C(=O)Nc3ccc(O)nc3)SCC2)=O)cn2ccc(Cl)cc2n1 40329,c1(OC)cc([N+](=O)[O-])c(OC)cc1NC(=O)OCC(=O)CCC(C)C 40330,C1(O)(CNC(C2(C#C)CN(C(=O)CC3CCCN(C)C3)C2)=O)CC2CCC1O2 40331,N1(C(Cc2ccc(CC)s2)=O)CCCN(C(c2cc(C)ncn2)=O)CC1C(C)C 40332,C(=O)(CCCCc1ccc(Cl)cc1)NCC(CN(C(Cc1cc(C)sc1)=O)C)O 40333,C(CC1(C#N)CC1)(C(=O)NOCCC(C)O)NC(c1c(CC)csc1)=O 40334,Cc1cc(N2Cc3ncsc3C2)nc(=NCCCc2nnnn2C)[nH]1 40335,N1(C(c2c(C)nco2)=O)CCC2(CC(NC(=O)C(F)(F)c3ccncc3)CO2)C1 40336,c1(C(=O)NC(CCOC(C)C)(C)C)nnc(S)n1C.C1(=O)CCC(C)N1 40337,C#CCCCCC(=O)N1CCCC(C)(NC(=O)C(CCC)OCC)C1 40338,C1(NC(CC=C)=O)COCCC1NC(=O)CCCCN1CCOCC1 40339,N1(C(C2(SC)CC2)=O)CC2CC(NC(=O)CC3CC(=O)NC(=O)C3)CC1C2 40340,c1(CC)cc(C(=O)N(C)CC2COCCN2C(=O)CCC2CCC2)ccc1Cl 40341,Cc1cc(F)c(C(N2CCC(C)(CNC(=O)C=Cc3cncs3)C2)=O)c(F)c1 40342,Cc1cc(C(N2CC(N(C)C(c3ccc(CC(C)(C)O)s3)=O)C2)=O)cnc1C 40343,CC1CN(C(=O)CCNC(C2CCC2)=O)CC1NC(=O)CC1OCCO1 40344,CC1CC(C(N2CC3(CC(CNC(c4cccc(Br)c4)=O)C3)C2)=O)CC(C)C1 40345,N1(C(C(c2cnn(C)c2)C)=O)CCC(C2(NC(=O)Cc3cc(Cl)n(C)n3)CC2)C1 40346,C1(N(C(C(C)OCC(C)C)=O)C)CCC(Nc2cnn(C)c2C(F)(F)F)CC1 40347,c1(C(=O)NC(CC(C)NC(CCN(C)CC)=O)C)cccc(Cl)c1C 40348,N(C)(S(=O)(=O)N(C)C)CC(=O)NC1CC(n2cc(C(=O)NCC(C)O)nn2)C1 40349,C12CCC(C)(C1)Cc1c(con1)C(=O)N1CC(C(C)C)(C1)CNC2=O.CCC1CC1 40350,C=C(C)CC(C(=O)C1CCNC(=O)C=CC(C)NCC1)OC.C(CO)S 40351,C1(C#N)(C(=O)OCC(c2n(C)ccn2)=O)C(C#N)C1(C)C 40352,N1(C(C(CC)OC)=O)CCOC(C(C)NC(c2cn(C)nc2C(C)C)=O)C1 40353,c1(OCC(=O)NCC(C2CC2)NC(C2N(C(CC)=O)CSC2)=O)ccc(C)cc1 40354,N1(C(c2cc(SC)oc2C)=O)CCCN(C(=O)Cn2ccc(O)nc2=O)C(C)C1 40355,c1(C(N2CCN(C(=O)NC(C)C)CC2C(F)F)=O)cc(F)c(N)cc1F.C(C)(=O)OC 40356,c1(OC)cc(NC(c2cccc(N3CCNC(=O)C3)c2)=O)ccc1O 40357,N1(C(c2c(CC)cccn2)=O)CCCC12CCN(C(C1CC=CCC1)=O)C2 40358,c1(NC(C(C(C)C)N(CC(=O)Nc2ccc(Br)cc2)C)=O)cc(F)ccc1Cl 40359,c1(C(=O)NCC(CC)NC(=O)C(C)(C)C(N)=O)ccc([N+](=O)[O-])cc1 40360,N1(C(c2c(COC)cc[nH]2)=O)CC(CNC(=O)C=C2CCC(C)C2)CC1(C)C 40361,Cc1nc(C(=O)NC2(CNC(C3(C)CC=CCO3)=O)CC2)ccc1C#N 40362,Cc1occ(-c2ccccc2)c1CCCNC1(C(F)F)CCCC1 40363,CCCC(C(=O)N1CCC1Cn1cc(-c2cnn(C(C)C)c2)nn1)OC 40364,C1(NC(C2CCC(CNC(C(C)(F)c3ccon3)=O)O2)=O)CCOC(C(N)=O)C1 40365,C1(=O)C=CCN(C)C(=O)CN1C(C)C.C=CCNC(C)=O 40366,N1(C(CC2(F)CCN(S(CC3(CN)CCC3)(=O)=O)CC2)=O)CCC2(CCCC2)C1 40367,C1(C(N(C(C)CNC(=O)C2CC2)C)=O)(NC(=O)OC(C)(C)C)CC=CC1 40368,c1(SCCC(=O)NCC(CO)NC(c2cocn2)=O)nnnn1-c1ccccc1 40369,C1(C(=O)NCC2N(C(COCCCC)=O)CCCCC2)CNC(=O)CC1(C)C 40370,N1(C(c2c(C)cns2)=O)CCOCCC1C(=O)NC(c1cncs1)C 40371,C1(OC)CC2(C1)CC2C(N1CCCC1CCC(=O)NC(c1ccc(C)cn1)=O)=O 40372,C(=O)(C(C)(C)CC(C)C)N(C)CC1N(C(C(=O)NCC)=O)CCC1 40373,c1(C(=O)NCC(C(C(C)C)C)NC(c2ccc(Cl)s2)=O)noc2c1CCCC2 40374,CC1(C)CCC(C(N2CC=CC2CNC(c2ccon2)=O)=O)C1 40375,N1(C(c2ccccn2)=O)CCC(NC(C2(C(c3ccccc3)=O)CC2)=O)C1C(C)C 40376,C1(NC(c2c(CC)onc2)=O)CCCN(C(c2nc(Br)c[nH]2)=O)C1C 40377,C1(O)(CCNC(c2c(C)csc2)=O)CCN(C(c2ccc(F)cc2Br)=O)CC1 40378,c1(C(N2CC(CNC(CCC3CC(C)C3)=O)OCC2)=O)ccc(F)c(Cl)c1N 40379,Cc1c(Br)csc1C(N1CC(CC(C)NC(=O)C(C)C2CCC2)C1)=O 40380,C(C(=O)N1CC(O)CO1)NC(c1ccncc1O)=O.CC1(C)CC(=O)N1 40381,C1(C(N2CC(NC(C(COC)OC)=O)C(C(F)F)C2)=O)CCC(C)(O)CC1 40382,C1(CNC(C2CCCC(NC(CC(C)F)=O)C2)=O)CC12CCOCC2 40383,C1(C)(C(=O)NCCOCCC(N2CC(C(CC)CC)C2)=O)CCC(=O)N1 40384,C(=O)(C(C)CC(C)(C)C)NC1(CC=C)CCN(C(c2cnn3ccncc23)=O)C1 40385,c12ncc(cc1Cl)S(=O)(=O)N2CC1CCCO1.C1(CNC(=O)CC2CC2)CC(Cl)(Cl)C1 40386,CCCCCCC(C)C(=O)N1CCSCC1CCNC(C1CCCCN1N=O)=O 40387,N1(CN2CC(NC(=O)CSc3ccncc3)C2)CCCCCCC1=O 40388,C(=O)(C1=CCOCC1)N1C(CC=C)(CNC(CN2CCOCC2)=O)CCC1 40389,Cc1cc(N2CCC(C)(C(=O)NCC(c3cccc(O)c3)O)C2)ncn1 40390,C(c1ccncn1)=CC(=O)NC(CNC(C1(CC=C)CCC1)=O)(C)C 40391,Cc1cccc([N+](=O)[O-])c1C(=O)N(C1CN(C(=O)CC2OCCOC2(C)C)C1)C 40392,c1(C(=O)NCC(CNC(C2CCN(C)C2)=O)(C)O)c[nH]c2cccc(Cl)c12 40393,C(=O)(CS(=O)C(F)(F)F)NC1CCN(C(C(C(=O)OC(C)(C)C)OC)=O)CC1O 40394,CC1CCc2ncc(C(N3CCC(CNC(=O)C(N)=O)C34CCC4)=O)n2C1 40395,N1(CC(=O)N(C(C)CNC(=O)C(C)NS(C)(=O)=O)C)CCCNS1(=O)=O 40396,N1(C(c2ncn(CCOCCOC)c2)=O)CCC(C(=O)OCC)(C(C)C)C1 40397,C12(NC(C=C(C)Cl)=O)CC(NC(c3cncs3)=O)(C1)C2 40398,N1(C(C(C)NC(=O)OC)=O)CC(C(N2CCCC(F)CC2)=O)OC(C)C1 40399,N1(C(c2c(N)nccc2)=O)CCC=C(CNC(c2sccc2CO)=O)C1 40400,CCCCC(C)C(=O)N1CC(C(=O)N(CC)CC2CCOC2)C(F)C1 40401,c1(C(N2CC(C#N)C(N(C)C)C2)=O)cc(-c2ccccc2C#N)c2[nH]ccc2c1 40402,C[Si]1(C)CCN(C(=O)CC2(NC(=O)CC3CCCSC3)CCCCC2)C1 40403,c1(C(=O)NC(CNC(=O)CN2C(=O)CCC2=O)C2CC2)cc(C2CC2)nc(O)c1 40404,c1(NC(N2C(C(CC)O)CCC2)=O)ccc2c(c1F)CCC2 40405,c1(C(=O)NCC(CNC(C(CC)(C)OC)=O)CO)ccnc2ncccc12 40406,c1(C(N2CCC(CNC(C(C(=C)C)(C)O)=O)CC2)=O)ccc2c(C)nn(C)c2n1 40407,N1(C(c2c(OCC)cccc2)=O)CC2CN(C(c3ccc(O)cc3OC)=O)CC12 40408,c1(N2CCN(C(=O)OCC)CC2)cc(C)c(S(=O)(=O)NC(C)C(C)SC2CC2)cn1 40409,C12(NC(=O)Cc3ccccc3Cl)CCN(C(=O)CCN3CCOCC3)CCC1C2 40410,Cc1ccc(CN(c2nnc(CC3CCC(F)(F)C3)n2C2CC2)C)cn1 40411,c1(C(N2CC3CCN(C(C)=O)CC3C2)=O)cnc2c(c1)OCC(=O)N2 40412,N1(C(C(Cc2c(C)nc[nH]2)O)=O)C(C)C2CC1C2NC(c1cccnc1O)=O 40413,N1(C(COCC#C)=O)CCC(NC(=O)CCc2ccc[nH]2)C1C1CC1 40414,c1(OC)cc(N)ccc1C(=O)NC(C)C(C)NC(C1CCC1c1nc[nH]n1)=O 40415,C1(N(C(C(C(C)(C)C)=O)=O)C2CC2)(C(=O)Nc2cc(F)ccc2O)CCC(C)(C)C1 40416,C(N=c1ccc([N+](=O)[O-])c[nH]1)C1C(OCC)CCC1 40417,c1(C(=O)NC(C)CNC(=O)C(C)(C)COC2CCC2)cccc2nsnc12 40418,c1(OC)cc(F)c(C(=O)NC2COCC2NC(C2(OC)CCOC2)=O)c(F)c1 40419,c1(C(=O)NCC2C(NC(c3cc(C#N)sc3)=O)C2)cc(S(N)(=O)=O)ccn1 40420,N#Cc1cc(C(=O)NC2CN(C(c3c(Cl)ccc(F)c3F)=O)C2)c(N)nc1O 40421,C1(Nc2nc(C)nc(C(C)C)c2)CCC2CN(c3ncccn3)CCC2C1 40422,c12nccnc1C(=O)N2.Cc1ccc(-c2cnn(CC(=O)Nc3cnc[nH]3)c2)o1 40423,CC1CCCCC1(CNC(c1ccc(O)c(O)c1)=O)NC(c1c[nH]ccc1=O)=O 40424,Cc1cccc(S(C)=O)c1NC(c1coc(S(C)(=O)=O)c1)=O 40425,C1(CNC(c2scc(C)c2)=O)CC(NC(C2CN(C(N)=O)C2)=O)C12CCC2 40426,C(=O)(C(O)CCNC(C1COCC(C)O1)=O)NC(c1nnc(C)s1)C 40427,C1(CNC(C=CCN(C)CC)=O)N(C(=O)CC(O)C(C)C)CCCC1(C)C 40428,C(=O)(CCCN(C(=O)C(C)CN(C)C)C)N(C(C(=O)NC)C1CC1)C1CC1 40429,c1(CC)nc(C)[nH]c1C(=O)NC1CC(CN(CC(=O)NC)C)C1 40430,CC1(NC(=O)COC2CCOC2)CCCN(C(c2c(Cl)nsc2Cl)=O)C1 40431,c1(C(N2CC(OCC(=O)NCC3CC3C3CCCO3)C2)=O)ccc(Cl)s1 40432,C1(C(C)C)N(C(c2cncn2C)=O)CC12CCN(C(C1(C#N)CC1)=O)CC2 40433,N1(c2cc(NCc3cnc(C)s3)nc(C(C)C)n2)CCCCNC(=O)CC1 40434,CC(C)(C)C(CC(=O)NC1CC(O)(CNC(=O)CN2CSCCSC2)C1)C(F)F 40435,c1(C(=O)NCC2(NC(C3CC34CC4)=O)CCC2)ccc(C2CC2(F)F)cc1 40436,CN1CCOCC1C(=O)NCC1(C(N2CC=CC2CF)=O)CC1 40437,Cc1c(C(=O)NC(C)CNC(=O)CCc2ccon2)ccn1C 40438,c1(C(=O)NCCOC(F)F)cc(S(=O)(=O)N)c[nH]1.N1(CC2CCOC2)CCCCC1 40439,C(=O)(C1=NOC2(CCN(S(=O)(=O)CC3CCCC3)C2)C1)NCc1cccc(C#N)n1 40440,N1(C(CCSCC)=O)CCC2(CCCCN(C(c3coc(COCC)n3)=O)C2)C1 40441,C12(C(N(CCNC(C(COC)(C)OC)=O)C3CC3)=O)CCCC(C1)C(=O)NC2 40442,Cc1cc(OCCC(N2CC(C)C2c2ccccc2)=O)no1 40443,c1(N2CC(NC(C3C(C)(Br)C3)=O)(CO)C2)ncncc1Br 40444,N1(C(C2C(C)(C)CO2)=O)CCCCC1C1CCN(C(=O)CCCC2CCC2)CC1 40445,N1(C(C(=O)NCCOC)=O)CCCC(CN(C)C(c2scc(C)c2OC)=O)C1 40446,N1(C(C(C2CCN(C(=O)C(N3CCOCC3)C)C2)C)=O)CCC(O)C(C)C1 40447,CC1C(NC(C23CCC(F)(CC2)C3)=O)CCCN1C(=O)COc1cnn(C)c1 40448,Cc1sc(C)c(C(N2CC3(CC(NC(=O)C(C)CC(F)F)CO3)C2)=O)c1C#N 40449,C1(C(N2CC(F)(C(=O)NC3CN(C4CCC4)C3)C2)=O)CC2CCC2C1 40450,CC(c1ccccc1)=CC(=O)NCC1CCC1NC(C1CC12CC2)=O 40451,N1(C(C(C)CC(F)(F)F)=O)CCCC2(NC(=O)CN3CCC3)CCCC12 40452,C1(CC(=O)NCC(C(C)C)(C)C)C2CCC(C2)N1C(=O)CCCn1cncn1 40453,c1(C(=O)NC(C2CCCCC2)CNC(C(COC)O)=O)c(OC)ccnc1F 40454,N1(C(CN(C2CC2)CC)=O)CCN(C)CC1CNC(=O)Cc1n[nH]c(C)n1 40455,c1(C(N(CCCNC(=O)Cn2cc(C3CCOC3)cn2)CC)=O)ccc(O)nn1 40456,N1(C(C=CC=CCC)=O)CCC2(NC(=O)COc3cccc(C)c3F)CCCC12 40457,Cc1ccsc1C(=O)N(CCC(=O)NC(C)(C)CO)C 40458,C(=O)(CCCS(=O)(=O)N1CCCC1)NCC=CCNC(COCCC#C)=O 40459,c1(OC)cccc(Cl)c1C(=O)NC1CCN(C(C2(C(C)C)CC2)=O)C(C)C1 40460,c1(C(N(CC(CNC(CC2(OCC)CCC2)=O)(C)C)C)=O)ccnc(OC)c1 40461,N1(C(=O)C2=NOCC2)CC2CCCC1CN(C(c1ccc3nc(O)[nH]c3c1)=O)C2 40462,C(=O)(CCCC(C)(C)C)NC(CC(C)C)C(N)=O.c12ncccc1C(=O)N2 40463,N1(C(C(C)S(N)(=O)=O)=O)CCC2(CCCC2NC(=O)CCc2cc(Cl)no2)CC1 40464,C(CCCC(=O)NCC1(O)CN(C(c2cn(C(C)(C)C)nc2C)=O)C1)NC(C)=O 40465,N1(C(C2(OC)CC2)=O)CCC(C(=O)Nc2cnc(N(C)C)nc2)=C(F)C1 40466,O=C(C1=CC2CCCC12)NCC1CC(NC(c2ncnc(O)c2Br)=O)C1 40467,CCC(C)C(O)C(=O)NCC(CO)NC(c1ccc(F)c(C(F)(F)F)c1)=O 40468,CCC(C(=O)OC)C(=O)NC(CCCc1ccccc1)C(=O)N1CC2CC2C1 40469,C#CC1(C(=O)NCCN2CCOC(C)C2)CCN(C(=O)CC2CSC2)C1 40470,c1(-n2c(C(CC3CC3)NCC3(C(C)(C)C)CC3)nnn2)ccc(F)c(Cl)c1 40471,c1(OC)cnc(F)c(C(=O)NCC2C3CN(C(=O)Cn4ccnn4)CC23)c1 40472,Cc1[nH][nH]c2ncnc(=NC(=O)C3CC3C(=O)Nc3ccc4c(n3)OCCO4)c1-2 40473,C12CCN(CC1(C)C)C(=O)COC2=O.CCC(C)(C)OCCNC(C1CCC1)=O 40474,c1(N(CC#CC)C)ncnc2c1ncn2C(CC(C)C)NC(N)=O 40475,c1(C(N(C2CCCN(C(CC(C)F)=O)C2)C)=O)ccc2oc(S)nc2c1 40476,C1(C(=O)NCC2(OC)CCC2)CCCN(C(=O)C(C)OCC(C)C)C1C 40477,C1(C(N(CCCCN(C(C2CCC(C(=O)OCC)C2)=O)C)C)=O)CCCCC1C 40478,N1(C(CS(CCC)=O)=O)CCC2(CCOCC2)C(NC(c2cnn(C)c2F)=O)C1 40479,N1(C(CC=C=C)=O)CCC(NC(c2ccn(-c3ccccc3)n2)=O)C1C(C)C 40480,c1(C(N2CC(NC(=O)Nc3cc(C(CC)C)no3)C2)=O)cc(OC)ccc1F 40481,c1(CNC(C)=O)cc(C(=O)N(CC(N)=O)C)on1.C12(CC1)C(=O)N2C(C)C 40482,c1(C(=O)NCC(CC)N(C(=O)C(c2cnn(C)c2)C)C)cccc(F)c1OC 40483,C(=O)(C1=CC2CCC=CCCC12)N1CC(N(C)C(c2cn(C)c(=O)n2C)=O)C1 40484,C1(NC(=O)CS(=O)(=O)NC2CC2)CN(C(=O)C=C(Cl)Cl)CC2(CCC2)C1 40485,N1(C(c2cc(CNC(c3c(C)ocn3)=O)nn2C)=O)CC2(CC2)CC1CO 40486,C=C(F)C1(CC(=O)N(CCC(=O)NCCc2ncn(C)n2)CC)CCC1 40487,c1(C(N(CCC)CCNC(=O)C=CBr)=O)cccc2c1OC(F)(F)O2 40488,O=C(N=c1[nH]ccc2cc(Cl)ccc12)C12CC1CN(Cc1c(Cl)cc(F)cc1Cl)C2 40489,C(=O)(C1=C(C)CCOC1)NCC(CNC(C1(C)COCCO1)=O)OC 40490,C1(C(N2CCC(C)CC2)=O)CCCN1NC(=O)CC(C)CN(C)C 40491,N1(C(c2ccc(CSC(F)F)o2)=O)CCN(C(=O)CCF)C2CCCCC2C1 40492,c1(CNC(=O)NCc2n[nH]c(=N)s2)cc2n(n1)CCC2 40493,c1(N(C(c2ccc(CNC(c3ncn(C(C)C)c3)=O)o2)=O)C)cccc(F)c1 40494,C1(OC)CN(C(=O)CCN(CC(F)(F)F)C)CC1NC(=O)Cc1cccn1C 40495,Cc1ncnc(C)c1CC(=O)NCC(O)CNC(C1(C)COC1)=O 40496,CC1CCN(C(=O)C=CC=C(Cl)Cl)CCN1C(C1CC(=O)NC(=O)C1)=O 40497,C1(C)(CC)CCN(C(C2(CNC(=O)C(C)O)CCC2)=O)CC1 40498,C1(C(N2C(CCNC(=O)Cc3ncc(Cl)s3)COCC2)=O)CC2CCC(C1)C2 40499,C1(CNC(c2c(C)c[nH]n2)=O)CN(C(c2ccc(F)cn2)=O)CC1C(F)(F)F 40500,Cc1cnnc(O)c1C(=O)NC1CC(CCC(=O)NCC(N2CCOCC2)C)C1 40501,C#CC1CC2(CC2)CN1C(=O)C(C1CC=CCC1)NC(C1CC2CCC2C1)=O 40502,c1(OCC)nn(C)cc1NC(c1cnn(CCNC(=O)C=Cc2cncn2C)c1)=O 40503,C(=O)(C(Cc1cnc[nH]1)NC(=O)COC1CC=CC1)N(C(C(C)SC)C)C 40504,c1(OC)cccc2c1OCCC2NC(c1c(Br)cc(Br)cc1Br)=O 40505,N1(C(c2c(C)cncn2)=O)CCC(O)C(NC(=O)CCOCCN(C)C)C1 40506,N1(C(C(C)OC)=O)CC2=C(C1)CN(C(C1CN3CC4CC3(CO1)C4)=O)C2 40507,C(=O)(C1=NNC(C(F)(F)F)C1)NC1CC(NC(=O)CC2(O)CCC2)C1 40508,C1(N(C(C(CC)O)=O)CC2CC2)CCN(C(=O)C=Cc2sccc2C)CC1 40509,c1(C(=O)NCC2N(C(C(C)S(N)(=O)=O)=O)CC3(CC3)C2)coc2ccc(O)cc12 40510,N1(C(c2c(C)cno2)=O)CCCC(N(CCO)C(c2c(C)ccn2C)=O)C1 40511,N1(CC(C)F)CC(C)CCC(C)(C)C1 40512,CN1CC2(CCN(C(NC3c4ccccc4C(=O)N3C)=O)CC2)c2ccccc21 40513,N1(C(C2CC(CCC)C2)=O)C(C(=O)NCc2cnn(C)c2OC)CC2CC12 40514,CC1(C)CN(C(C2CC3CCCCC23)=O)CC(CNC(=O)CC2CC2)O1 40515,c1(NC2CC(F)(CNC(c3cn(COC)nc3)=O)C2)ncc2c(ncn2C)n1 40516,C1(CCOC)SC(=Nc2ccccc2-c2ccccc2O)N(CCC#N)C1=O 40517,N1(C(c2cn(C(C)C)nc2)=O)CCC(C)(CNC(c2[nH]nnc2C2CC2)=O)CC1 40518,CC1(C(=O)NCC2COCC2NC(c2cc(-c3ccco3)c[nH]2)=O)CCOCC1 40519,c1(C(N(CCCCCCNC(C(F)=CC)=O)C)=O)cc(=O)n(C)cc1Br 40520,CCC(CC(=O)N(C(C)C(=O)NC1(CC)CCCCC1)CC)OC 40521,C1(C(=O)NCc2ccc(CCC(=O)OC)cc2)CCc2nc(O)nc(O)c2C1 40522,C1(CC(=O)NC(CN(C(COCC(=C)C)=O)C)(C)C)CCC(=O)N1CC 40523,C(C)(C)(C(=O)N1CCCCO1)C1CCN(C(c2ccn(COC)n2)=O)C1 40524,Cc1ccsc1CN(C(C1CCN(C(C2SCCS2)=O)C1)=O)C 40525,C=CCC(C)(C)CC(=O)NCC(CCC)C(=O)NCC(C)(O)C(=O)OC 40526,C1(CNC(C(C)Sc2nncn2C)=O)CCCCN1C(=O)Nc1ccccc1F 40527,N1(C(C2C(OC)CCC2)=O)CCC2(CCCN2C(=O)C2=CCCC2)C1 40528,c1(C(NNC(c2cc(OC)c(OC)c(Br)c2)=O)=O)cc(F)c(C#N)cc1F 40529,N1(C(c2cccc(C)c2)C)CC2CCC1CN2C(c1nccc(C(F)(F)F)n1)=O 40530,C1(C(N(C(C)C(C)(C)O)C)=O)CCC2CCC1N2C(C1CCCC(O)C1)=O 40531,CCC(O)C(F)(F)C(=O)N1CC2C(C1)N2C(=O)C(c1ccccc1)F 40532,C(=O)(CCC(F)(F)Cn1cc(Cc2cc(C)on2)nn1)N(C1CCC(=O)N(C)C1)CC 40533,N1(C(Cc2c(OC)nccc2)=O)CCC(C)(C)C1CNC(=O)COCC(C)(C)C 40534,c1(OC)cc(Cl)c(C(N2CCCN(C(C)=O)CC2)C(=O)NC2COC2)cc1OC 40535,c1(N(S(N)(=O)=O)CC)ccc(Cl)cc1.n12nnnc1COC(=O)C2.c1(OC)ccccc1 40536,C1(NC(CN(CC(C)C)C(c2ncn(CC)c2)=O)=O)CCC(C)(C)C1 40537,C(=O)(C=C1SCC(=O)N1C)N1C2CC(N(C(C3C(OC)CCC3)=O)C)CC1CC2 40538,CCC(C)(C)C(=O)NC(c1nc(C(=O)Nc2ccc(C(N)=O)o2)co1)C 40539,c1(N(C(C)=O)C)ccc(CC(=O)NC2C3CN(C(=O)C(F)=C(C)C)CC23)cc1 40540,C1(C(=O)NCC(CC)C#N)CC12CCN(C(=O)CN(CC)CC)C2 40541,Cn1nnc(C(c2nnnn2Cc2ccco2)NCCCC2(C)CC2)n1 40542,C1(C(=O)NCC2CN(C(CC(=C)C)=O)CC2C(F)(F)F)Cc2nccn2C1 40543,n1(CC)c(C(=O)NCCC(F)Cn2cc(C3(C)CCCC3O)nn2)cnc1O 40544,c1(C(N(CC(CNC(CCC(=C)C)=O)O)C)=O)cnc2c(cnn2C(C)C)c1 40545,N1(C(c2nc(C)n(C)n2)=O)CC(NC(c2cccnc2N(C)C)=O)C2(CCC2)C1 40546,c1(NC(c2c(NCc3ccc(OC)nc3Br)ccs2)=O)cccc2cn(C)nc12 40547,C1(CC=C)(NC(=O)Cc2c[nH]nc2C)CCN(C(=O)C(C)(C)COC(C)(C)C)C1 40548,S(=O)(=O)(c1ccc(=NCc2nccc(=N)[nH]2)[nH]c1)NC1(CO)C(C)CCCC1 40549,c1(NC(N)=O)ccc(C(=O)NC2(C)CC(NC(N)=O)C2)cc1.C1CCC(=O)N1 40550,CC1(NC(C2CCOCO2)=O)CN(C)C1.C(C)(C)(C)ON 40551,C(C1CCCN1C(c1cc(C)sc1N)=O)=CC(=O)NC1(CC)CCOC1 40552,c1(OC)ccc(F)cc1CN1CCCC1CNC(=O)C(=O)N.C1(C)COC2CC1C2 40553,C#Cc1cncc(C(=O)NC2CCCCC2CNC(=O)C(F)C(C)(F)F)c1 40554,C1(C(N2C(COC)CCCC2)=O)CN(C(=O)C(C)c2cc[nH]n2)CC1(C)C 40555,c1(C2c3ccc(o3)C(=O)N2CC2CCCO2)cc(C)ccc1F.n1(CC)cc(C2CC2)nn1 40556,CN1CCN(C(C2CCC(=O)C2)=O)C(C(=O)N(C2CCN(C)C2=O)C)C1 40557,N1(C(CC(CC)C)=O)CCCCCC(NC(C2OC(C)CC2C)=O)C1 40558,c1(C(=O)NCC2C(C)CCN(C(c3c(C)snn3)=O)C2)cc2c(s1)CCSC2 40559,Cc1cc(F)c(Cl)cc1C(=O)NCC(F)CNC(=O)CC(O)C(C)C 40560,C1(C(=O)Nc2ccsc2)C2CN(C(c3cc[nH]c3)=O)CC12 40561,C(=O)(CC1=CCCCC1)NCC1CCCN(C(CCCOC(C)=O)=O)C1 40562,c1(C2C(OCCOC(C=Cc3n(CC)ncc3)=O)C2)ccc(Cl)c(Cl)c1 40563,CCC(C(C)O)NC(=O)C=CCC1(NC(c2c[nH]c(C(N)=O)c2)=O)CCC1 40564,C1(CC(=O)N(C(C)CNC(=O)C=CC2CCCCCC2)CC)CCC(F)(F)CO1 40565,c1(CC)cc(C(=O)NC(C)C(=O)NCC(C)N(C)C(C)C)n[nH]1 40566,C=CCC(CC(=O)N1CCCC(N(C)C)CC1)NC(c1ccc(C)c(C)c1)=O 40567,C(CCN(C(=O)CC1(OC)CCC1)CC)(C(C)C)NC(C(CC)n1cncn1)=O 40568,c1(C(=O)NCCN(C(=O)COCCCF)CC)cnc(C(C)C)o1 40569,CC(C)CC(C)(C)C(=O)NCC(C)(CO)NC(=O)COC1CCC(C)CC1 40570,Cc1nn(C)c(C)c1CNC(=O)C(C(C)O)NC(=O)OC(C)(C)C 40571,C(=O)(C1=CCCS1)NC(C1CCN(C(c2csc(C(N)=O)n2)=O)C1)C 40572,c1(C(C(=O)O)NC(C2(C)CS(=O)(=O)C2)=O)cccc(Cl)c1Cl 40573,C(C(C)NC(c1ccn(C(F)F)n1)=O)(C(C)C)NC(c1c(OC)csc1)=O 40574,C(=O)(C(C)C(O)C(C)C)N1CCC(C(C)NC(C(Br)=C(C)C)=O)CC1 40575,C1(C(=O)NCC(C)N(C)C(c2cc(C3CCCCC3)[nH]n2)=O)CC=CCC1 40576,C1(C)(CC(=O)NCCSCC#C)CCN(C(C2(O)CCCC2)=O)C1 40577,c1(C(=O)NCC(CO)NC(CC(C=C)CCC)=O)ccc(=O)n2c1CCC2 40578,c1(C(=O)NCC2CCN(C(=O)Cc3ccnc(Br)c3)C2)cc2n(n1)CCO2 40579,CCC(CCC(=O)NCCOCCNC(=O)CCOCC(F)F)OC.C(C)C 40580,C(=O)(C(C)(F)C(C)(C)F)NCCCC1(NC(CCc2cccc(OC)c2)=O)CC1 40581,C1(NC(C(CSC)C)=O)CC2CCC1N2C(=O)Cn1nc(O)ccc1=O 40582,c1(CN(CCOCC)C)cc2c(cc1O)CCCC2 40583,C(Cn1cccn1)(C(=O)N(CCC(=O)NC(C)=O)CCC)NC(CCOCC#C)=O 40584,N1(C(C=CC)=O)CCC(C(F)(F)F)CC1CNC(=O)C(c1ccc(CC)cc1)O 40585,C1(NC(=O)CSc2cccc(F)c2)CC(O)CN(C(c2ccc[n+]([O-])c2)=O)C1 40586,C1(CNC(C2(CCC)CCC2)=O)C2CCCC1N(C(=O)C(C)(C)F)C2 40587,CC1=C(C)CC(C(=O)NCCCC(N2CC(C(C)C)CC(C)C2)=O)CC1 40588,c1(C(C2(C)CCCC2NC(=O)O)C(C)(C)C)ccccc1O.OC(F)(F)F 40589,C1(NC(c2ccc(OC)nc2C)=O)CCN(C(=O)CC(C)N(C)C)CC1(C)C 40590,C=CC(C)(CCOC)C(=O)NC1CCC(C)N(CC(=O)NC2CC(F)(F)C2(C)C)C1 40591,C1(C(N2CC(C)C(n3cc(C(C4CC4)N(C)C)nn3)C2)=O)COc2ccccc2O1 40592,CC1(C(=O)NCC2CC2NC(c2ncoc2C2CC2)=O)CC2(CCC2)C1 40593,C1(C(=O)NCCN(C)C(c2cnns2)=O)C2Cc3c(Cl)cccc3C12 40594,c1(Nc2n(CC)c(CCc3cc(C)nn3C)nn2)nc2c(F)cccc2o1 40595,C1(CNC(CCOCCCNC(c2cc(C)sn2)=O)=O)CC2(C1)CC(O)C2 40596,c1(C(N2CCC(CC(C)NC(C(C(C)C)F)=O)CC2)=O)cccn2nccc12 40597,c1(C2(NC(CC=C)=O)CN(C(=O)C(=Cc3cn[nH]c3)C)C2)ccc(Br)cc1 40598,c1(CN2CCC(=CC(=O)N(C3CCCCC3)C(C)C)CC2)cccc2c1CCC2 40599,N1(C(C2C(NC(=O)COc3ccc(F)cc3)CCCC2)=O)CCN2CCC1CC2 40600,C(=O)(C(C)(O)C(C)C)NCC#CCNC(c1c(C)[nH]nc1C(F)(F)F)=O 40601,C1(CC)CC(NC(c2cnn(CC3CCCCC3)c2)=O)CCN1 40602,C12(CN(C(C)=O)CC)CC1CN(C(C1CCCN(C(c3ccc(Cl)s3)=O)C1)=O)C2 40603,C1(C2CCC(=O)NC2)(C(=O)OCCc2c(C)nc(C)s2)CCC1 40604,C1(N(C(c2cc(C)sc2)=O)C)CN(C(c2n[nH]c(C)c2C)=O)CC1F 40605,C1(CC)(NC(c2cc(C(N)=O)[nH]n2)=O)CCN(C(C2(c3ccccc3)CC2)=O)CC1 40606,c1(C(N2CC(CC=C)(NC(C3CC3F)=O)C2)=O)ccc2[nH]c(=N)[nH]c2c1 40607,Cc1ncc(C(=O)NC(C(=O)N(CCC#N)C)c2nccs2)s1 40608,C1(C(N2CC=CC(NC(C3CCC(C)(CC)O3)=O)C2)=O)CCC(F)(F)C1O 40609,c1(C(=O)NC(C)CNC(=O)CSCC2CCCCO2)ccc(Br)cc1Cl 40610,CC#CCCC(=O)N1CCC(N2CCN(C(c3c(Br)cnn3C)=O)CC2)CC1 40611,N1(C(C(C)COc2ccccc2)=O)CCC2CC1CN(C(C1(Cl)CC1)=O)C2 40612,c1(C(=O)NCC(CNC(c2c(CCC)n[nH]c2)=O)O)ccnc2c1CCC2 40613,c1(-n2cc(C(C)NC(c3cc(Br)c(Br)[nH]3)=O)nn2)cccc(OCCF)c1 40614,C1(C)(C(=O)NCC(CC=C)NC(=O)COc2cc(C)on2)CCCCNC1=O 40615,C(C)(C)(CCCNC(=O)C(C1CCCCC1)NC(c1coc(CC2CC2)n1)=O)OC 40616,N1(C2CN(C(C3CC(NC(c4cnn(CCO)c4)=O)C3)=O)C2)CC2CCC1C(O)C2 40617,CC(CC(F)(F)F)C(=O)N(CCNC(=O)CN1CCCCCC1)CC1CC1 40618,c1(C(=O)N(CC(C)NC(CCNC(C)=O)=O)C(C)C)c(Br)ccc2n[nH]cc12 40619,C1(=O)CC(C)NC(=O)OCCCN1.C1(F)(CC)CC1C(=O)C1CC1.C(CC(C)C)N 40620,C1(CCC)CC(C(=O)NOCC(=O)NCC2(C)CCOCC2)=NO1 40621,O=C(C1=CS(=O)CCC1)NC1CCCN(C(c2cn(C3CCC3)nn2)=O)C1 40622,C1(NC(c2cc(C)sn2)=O)CCC2(CC1)CCN(C(C1CCC(F)C1)=O)CC2 40623,C(=O)(CCC(=O)NC1CCC(F)(CNC(c2ccsc2C(F)F)=O)C1)NC 40624,C1(n2cccn2)(C(N(CC(C)N(C(=O)Cc2ccns2)C)C)=O)CCCC1 40625,c1(NC)snc(C)c1C(N1CC(CNC(c2cn(CC(N)=O)nn2)=O)C(O)C1)=O 40626,C1(NC(Cc2cccc(C(C)C)c2)=O)CN(C(=O)C(C)n2cncn2)CC1(C)C 40627,CC1CN(C(c2cc(Cl)ccn2)=O)CC(C)N1C(c1cnn2ccncc12)=O 40628,C1(NC(C2C(CC)CCN2C(=O)CN2CCC(=O)CC2)=O)CCCCCC1C 40629,c1(C(C(=O)NCCC)N(C)CCc2ccco2)cc2n(n1)CC(C)(C)CO2 40630,C1(CNC(c2n(C3CC(F)(F)C3)nnn2)C2(n3cccn3)CC2)C(F)(F)C12CC2 40631,C1(Cc2cc(CC)no2)CC(C)(C)CCC1N(C(=O)Cc1csnn1)CC 40632,C1(NC(C2N(CC)CC2)=O)CCC2CN(C(=O)Cc3ccc(O)nc3)CC2C1 40633,c1(C(=O)NCCC(C)NC(c2cc(C)nnc2O)=O)c2c(nn1C)CCC2 40634,C=C(F)C1(CC(=O)N(CCCNC(=O)C=C(CC)CC)C2CC2)CCC1 40635,CC1(C)COCC(NC(=O)C(C)(C2CC2)NC(=O)CCc2nc(=N)[nH][nH]2)C1 40636,C1(CC)(OC)CCN(C(=O)C(CO)NC(C2SCC=C2C)=O)CC1 40637,c1(C(c2n(CC=C)nnn2)NCC2(OCC)CCOC2)cc(C)nnc1C 40638,C1(NC(c2scc(OC)c2)=O)CC2CN(C(C3CC(F)(F)C3)=O)CCN2C1=O 40639,N1(C(C(CC)C#N)=O)CC2CC(N(C)C(c3ncc[nH]c3=O)=O)C1C2 40640,C1(C(=O)NCC(CNC(CN2CCN(CC)CC2)=O)CO)CCC2CC2CC1 40641,C(C(C)C(=O)NCC1CCC(NC(c2c[nH]nc2C2CCOCC2)=O)C1)OCC 40642,C#Cc1cn(C)nc1C(=O)NCCC1CC(NC(=O)C2=COCCO2)C1 40643,Cc1nc(CN=C(NCC(C)(C)C)NC2CCCN(c3ncccn3)C2)c(C)o1 40644,CC(C)C(CCN(C(=O)CC1CCOC1C)C)NC(C1(N(C)C)CCCCC1)=O 40645,N1(C(C(CCC)OCC)=O)CC(CNC(c2cn(C)nc2CC)=O)OC2(CCC2)C1 40646,CC(C)(C)C1=CCN(C(C2CCN(C(c3cc[nH]n3)=O)C2)=O)CC1 40647,c1(CC)n[nH]c(CC)c1CC(=O)N(C1CC(NC(C2(C(F)(F)F)CC2)=O)C1)C 40648,N1(C(CCCCC#C)=O)CCN(C(=O)CCCC(F)(F)F)CC(CO)C1 40649,C1(NC(C(CNC(C2(COC)CC(=O)C2)=O)C)=O)C(O)C2CCOC12 40650,C(=O)(C1=CCC12CCOCC2)NC(CC)(CC)CCC(=O)Nc1ccsc1 40651,c1(OC)ccc(C(N2CCC(N(C)C(c3cc(F)ccc3N)=O)C2)=O)c(F)c1Cl 40652,c1(CC)c(OC(C)C(=O)N(C2CN(C(=O)CNC(C)=O)C2)C)ccn1C 40653,C1(C(=O)NC(CC(C)NC(C(CC)C)=O)C)CCN(C(=O)OCC(C)C)CC1 40654,c1(CC(=O)N(CC(CC)NC(=O)C(C)CN2CCCCC2)CC)ccc(C)s1 40655,N1(C(C2CCN(C(C)=O)C2)=O)CCCC2(NC(C3COCCN3C)=O)CCCC12 40656,c1(C(=O)NCCCN(C(=O)CN2C(C)CCC2C)C)cc2occc2s1 40657,C(C)(C)(CN=c1nc(N2CCSCC(C)C2)c2c(ncn2CC)[nH]1)N(C)CC 40658,CC(Cc1ccccn1)C(=O)NNC(=O)c1ccc(-n2nncc2I)cc1 40659,c1(C(C(=O)NCC(C)NC(=O)C(C)c2cncs2)(C)C)ccc(C#N)cc1 40660,C(=O)(CCCC(F)(F)F)NC1CCC(CC(=O)NC2CC(C)OC2=O)C1 40661,N1(C(c2cc(N)c(Cl)cc2)=O)C2CCC1CN(C(c1cn(C3CCC3)nn1)=O)C2 40662,n1(CCNC(=O)NC(c2ccc(F)cc2)C(=O)OC)c(=O)oc2ccccc12 40663,N1(N2C(C(C)C)COCC2)CC2CN(C(c3c(Cl)cncc3Cl)=O)CC2C1 40664,c1(CC)ncc(C(=O)NCC(F)CNC(c2cc(-c3cnn(C)c3)[nH]n2)=O)[nH]1 40665,c1(C(N2CC(O)(CN(C)C(c3nsnc3O)=O)C2)=O)ccc(Cl)c2c1OCCO2 40666,c1(C(=O)NCCN(C(C2CN(C)C(=O)N2)=O)C)cccc(C#CCO)c1 40667,N1(C(c2c(C)nsc2)=O)CCSCC1CCNC(=O)CC1NC(=O)NC1=O 40668,CC1CC(NC(C2CC3(C2)CC(C(N)=O)C3)=O)CCN1CCC1CCCCC1 40669,C1(CNC(=O)C=CC2CC2)CC2COCC2N1C(=O)Cn1ccc([N+](=O)[O-])n1 40670,N1(C(C2(CC)CCN(C(c3n(CCC)ccc3)=O)C2)=O)CCC(C2(C)CC2)C1 40671,CCCCCCC(C)(c1nnnn1C(C)CC)NC1CCn2cncc2C1 40672,C(CN(C)C(C1CN(C)C(=O)N1)=O)(CO)(CO)NC(C(CC)NC(N)=O)=O 40673,c1(C(N2CCC(OC(C(=O)OC)C)CC2)=O)noc2c1COCC2 40674,C#Cc1cccc(C(N2CCC3(NC(c4nn(C)cc4C)=O)CC3C2)=O)c1 40675,C1(C)(C(=O)NC(C2CN(C(c3cccs3)=O)C2)C)COC(=O)N1 40676,C1(NC(c2occ(C)c2)=O)CCC(C)N(Cc2ccc(F)cc2Cl)C1 40677,C=C(C)C1CCC(C)=CC1CC(=O)NC12CC(NC(=O)CCS(C)(=O)=O)(C1)C2 40678,Cc1cc(C#N)cc(C(=O)NCC(C2CC2)NC(=O)C(O)C(C)(C)C)n1 40679,c1(C(C)C)cc(CNC(=O)C(C)N(C(c2cc(CO)on2)=O)C2CC2)no1 40680,n1(CC(=O)NCC(C)CSC2CCOCC2)cc(C2CCC2)nn1 40681,C1(C(=O)NCC2(CC)CCC(=O)N2)CCCCCCN1C(C1COC(=O)N1)=O 40682,C1(NC(c2cnc(C)nc2O)=O)COC2(C1)CN(C(=O)CCC(C)CN(C)C)C2 40683,c1(CC(=O)NCC(=O)NC(c2nc[nH]n2)CC)ccncc1Br 40684,C(=O)(C1=NNC(C(F)(F)F)C1)NC(C1CN(C(=O)C(C)(C)O)C1)C 40685,c1(C(N(CC(C)CNC(c2csc(Cl)c2)=O)C)=O)ccc(F)c(Br)c1 40686,N1(C(CC(C)(F)F)=O)CCC(NC(c2cnnn2-c2ccccc2)=O)C(CO)C1 40687,C(CSC)(C(C)C)N(C(CC1CN(C(C2CC2C)=O)C1)=O)CC.CCOC 40688,N1(C(C2C(C(C)NC(c3cccc(C)n3)=O)C2)=O)C2CCC1CC(C)C2 40689,C1(C(=O)NC2(c3cn(CCC)nn3)CCC2)CCc2ncc(C)n2C1 40690,CN1CCC(C)(C(=O)NC2CC(CO)N(C(C3COCC3C(N)=O)=O)C2)C1 40691,C(C(CN=c1cc(C(N2CCS(=O)(=O)CC2)C)nc[nH]1)OC)OC 40692,C1(C(=O)NCCC2CCN(C(C(C(C)O)(F)F)=O)C2)CC2COCC(C1)C2(F)F 40693,C1(CNC(Cc2ccn(C(C)C)n2)=O)CC(C)(C)CN1C(C1CC(C)C1)=O 40694,C1(NC(c2ccc(C)s2)=O)CN(C(=O)CC2CC=CCN2C)CC1C 40695,N1(C(COc2cn(C)nc2)=O)CCCC(CC)CC1.C1(C)(NC(=O)CC(N)=O)CCCC1 40696,Cc1cc(C(=O)NC2CCN(C(C3CCCC3)=O)CC2CO)cc2c1NCCC2 40697,c1(C(N2CCC(CCNC(=O)CCCC3CCC3)C2)=O)cc([N+](=O)[O-])n[nH]1 40698,c1(C(=O)NCC2C(NC(Cc3n(C)ncc3)=O)CCCC2)n[nH]c2c1CCC2 40699,c1(CC(=O)NCC2CC(CNC(=O)CN3CCCC3)CC2O)ccnnc1O 40700,CC1CCOC(C(=O)NCc2cccc(-n3cc(CCC#N)nn3)c2)C1 40701,CCC(C(=O)NC(C1CCN(Cc2nnc(-c3ccco3)o2)CC1)C)C(C)C 40702,N1(CC(=O)NC(CC)(C)C)CCCc2cc(C)cc(F)c21 40703,c1(CC(=O)NCCCN(C(CCC2CCN(C)C2)=O)C2CC2)cccc(Cl)c1 40704,C1(C(=O)NCCC(=O)NC(C)CO)(OC)CCC(C)(C)C1 40705,C1(CNC(=O)NC2(OCCO)CCCC2)CCCCC1CC(F)(F)F 40706,c1(C(=O)OC)nn(C)nc1C(=O)N(C)CC1CCN(C(=O)CN2CCCC2)C1 40707,C(=O)(C1=NN(CC)C(=O)CC1)NCCC1N(C(c2nc(CC)oc2)=O)CCCC1 40708,c1(CSCCNC(c2nc(C)c(C)o2)c2n(CCOC)nnn2)ccccc1C 40709,C1(NC(c2cccc(C(=O)NCC3(CC)CC3)n2)=O)CCC12CCCC2 40710,N1(C(CCCC=C)=O)CCCC(O)(CNC(C2ON=C(C)C2C)=O)C1 40711,c1(C(=O)NCC2N(C(C(C)(C)NC)=O)CCC2)cc(C(=O)OC)ccc1Cl 40712,Cc1ccc(C)c(C(N2CC(CNC(c3cccc[n+]3[O-])=O)C3(CC3)C2)=O)c1C 40713,c1(C(N(C)NCc2onc(CC)n2)=O)ccc(-n2cc(COC)nn2)cc1 40714,C1(C(=O)NC(C2CCCN(C(=O)CCC3CC3)C2)C)(NC(C)=O)CCCCC1 40715,C(=O)(CCCC(C)(C)C)NCC(CN(C(Cc1c(C(C)C)con1)=O)C)C 40716,Cc1ccc2cc(C(N3CCC(C(C)NC(C4CCCC4F)=O)CC3)=O)cn2c1 40717,c1(C(N2CCN(C)CC2CNC(=O)CCCCO)=O)cnc2n1CCOC2 40718,C1(CC=C)(C(=O)NCC(c2cscn2)N(C)C)CCCN1C(=O)CCN1CCCC1 40719,C(C(CC(F)(F)F)NC(=O)CC(C)COC)NC(c1ccc(NC(CC)=O)cc1)=O 40720,c1(C(=O)NCC2(C)N(C(c3nn(CC)c(O)c3)=O)CCC2)cc2scnc2[nH]1 40721,CN1CCN(C(=O)COC2CCCC2(F)F)C(C(=O)Nc2cc(O)n(C)n2)C1 40722,c1(C(=O)NCC=C)oc(CNC(C2(Cl)CC2)=O)nc1C 40723,N1(C(C2CC3(CC(=C)C3)C2)=O)CC2(CCN(C(=O)C=Cc3cccnc3)CC2)C1 40724,N1(CCN(CC)CC)CCC2(CCN(C(=O)Cc3cncn3C)C2)C1 40725,C#CC1(C(=O)N(C)CCN2CCCC2)CN(C(c2cc(Cl)c[nH]2)=O)C1 40726,N1(C(CN(c2ccccc2)C)=O)CCOC(c2cccc(Cl)c2)C1.CCN(C)C 40727,c1(C(=O)NC(CNC(=O)CCC2CCC2)C2CC2)cccc(F)c1 40728,N1(C(C(C)=CC)=O)CC2CC(C1)C2NC(=O)CC1CCN1CC 40729,CC1CC2CC(C(=O)NCCC3CCCN(C(=O)C4=COCCO4)C3)(C2)O1 40730,c1(C(C)NCC2(NC(=O)OC(C)(C)C)CCCCC2)ccc(Cl)c(F)c1 40731,N1(C(C2C(C(=O)OC)CC2)=O)CCC(C(=O)NC(c2nc(C)no2)C)C12CC2 40732,C1(NC(CCCC2(C(=O)OC)CC2)=O)CCOC(c2ccccc2Cl)C1 40733,n1(CC(=O)NC2CN(C(CC3(OC)CCCCC3)=O)CC2C)cc(F)ccc1=O 40734,CC1OC2(C(=O)N(CCCOCCNC(=O)CC(C)C3CC3)C)CCC1CC2 40735,N1(S(CCC)(=O)=O)CC2CN(C(=O)CCc3ccc(C)c(F)c3)CC12 40736,CCCC(CCC)CC(=O)N1CCN(C(=O)CSCCOC)C(CS(C)(=O)=O)C1 40737,C1(C(=O)NC(CNC(C(C(C)C)NC(=O)C(C)(C)C)=O)(C)C)CCC(F)(F)CO1 40738,C(=O)(C(C)(C#N)CC)NCC1C(NC(c2c(CC)nn(C)c2)=O)CCCC1 40739,N1(C(c2cc(C)c(Cl)cn2)=O)CCCC(C2CCN(C(=O)CCCC#N)C2)C1 40740,C(c1cncnc1O)=CC(=O)NCC1(C)CC(NC(Cc2nn(C)c(Cl)c2)=O)C1 40741,CC(C1CCCCC1)=CC(N1CCC(N(C)C(c2ccnc(C)c2N)=O)C1)=O 40742,NC(=O)CCCCC(=O)NCC1CCCN1C(c1ccc(O)cc1Cl)=O 40743,CCC(C(=O)OC)C(=O)NCC1CCC(C(N2CCC(C(=O)NC)CC2)=O)O1 40744,c1(C(N2CCC(NC(C(C(C)C)OCC)=O)C2)=O)cnc(C)nc1C1CC1 40745,N1(C(CC(C)F)=O)CCC(CNC(=O)CNS(C)(=O)=O)C(F)(F)CC1 40746,N1(CC(=O)NC23CC(NC(CC=C=C)=O)(C2)C3)CCCC(C(F)(F)F)C1=O 40747,CC(C)(C)CCCCC(=O)NCc1nc(C(=O)N2CC(O)CCO2)co1 40748,C(C)(C)(C(=O)NCCCN(C(=O)CC1(C)CCCC1)C1CC1)N(C)C 40749,N1(C(C(C)NCc2cn(C3C=CCCC3)nn2)=O)CCCC(C)C1 40750,CCCC(C)(C)C(=O)N1CC(C(=O)Nc2ccc(Cl)cc2C(F)(F)F)CC(C)C1 40751,O=C(C1CNc2ccccc21)N1CCN(Cc2ccc(Cl)c(Cl)c2)C(=O)C1 40752,C=CCC(CC=C)C(=O)NCCN1C2N(C1=O)C(CC)CCC2 40753,CS(=O)(=O)c1coc(C(=O)NCC2CC3CCC(C2)N3C(=O)C2=CCCS2)c1 40754,Cc1c(C(=O)NCCCOCCCNC(=O)CC2CCC(O)C2)ncn1C 40755,Cc1nc(Cl)[nH]c(=NC(C)CC(C)NC(=O)C(CO)NC(N)=O)c1[N+](=O)[O-] 40756,CCCCC(CNC(=O)C1=CCCC1)NC(=O)CCc1cnc(C2(C)CC2)o1 40757,C12C3CC4C(C3NC1=O)C24.C(=O)(C(C)(O)CC)SCC.C12CN(C1)C2=O 40758,N1(C(C(CC#C)C2(N)CC2)=O)CCN(C(=O)C(C)(F)F)CC1c1ncc[nH]1 40759,c1(C(=O)NC(CC)CN(C)C(c2n[nH]c(C)n2)=O)cc2c(cc1O)CCC2 40760,C1(CNC(c2c(CC)non2)=O)CCN(C(=O)CC23CCCC2C3)CC1 40761,c1(C(N2CCC(C)(NC(C(C)OCCOC)=O)CC2)=O)ccc2occc2n1 40762,CN1CC(C(=O)NCC(C)(C)CN(C(=O)C=C2CCCC2)C)C(C(F)(F)F)C1 40763,c1(C(=O)NCCN(C(=O)CC2C=CCC2)CCC)c[nH]c(C)c(Cl)c1=O 40764,c1(CN2CC(c3c(F)cccn3)(O)C2)cc(C(F)(F)F)ccc1F 40765,c1(CNC(N(CCOC)Cc2nn[nH]n2)=O)cn2c(n1)CCCC2 40766,c1(CC(=O)NC(C2C(C)C2C)=O)nnnn1C1CC1.CC1C(=O)SCCCN1 40767,c1(CC)ccc2occ(C(N3CCC(C)(CNC(c4cc[nH]c4C)=O)C3)=O)c2c1 40768,c1(C(N(C)CC2CCCN(C(=O)Cn3cnnc3)C2)=O)cc(Br)c([N+](=O)[O-])[nH]1 40769,C1(C(=O)NC2(CC=C)CC2)CCCC(N=c2[nH]c(Cl)nc3ncn(C)c23)C1 40770,C(C1c2ccccc2CN1C(c1ncoc1C)=O)NC(CCC(CC)C)=O 40771,c1(C(N2CC(O)(CCNC(c3n(CC=C)ccc3)=O)C2)=O)c(C)cc(Cl)cc1N 40772,CC(C)(C)C(C)(O)C(=O)N1CC(C(C)(C)O)(CNC(C2CCCC2)=O)C1 40773,N1(C(CNC(C)=O)=O)CC(NC(=O)C(C2CC2)OC)CC2(CCC2)C1.C(C)(C)(C)S 40774,c1(C(=O)Nc2nnc(N3CCCC(CC)C3)n2C)cc(Cl)ncc1N 40775,CC1(C)CCC(C(=O)NC2(CNC(C3(CCF)CC3)=O)CCOC2)C1 40776,C1(Nc2c(C(=O)NC)c(Cl)ccc2)CC(C)CN(C(=O)C(=O)NCCN(C)C)C1 40777,CCN=C(NCCOC)NCC1CCOC1.C12CCCC1NC2 40778,C1(CC(=O)NCCN(C(C(CCC)C)=O)CCCN(C)C)COC(C)(C)CO1 40779,C(=O)(CC1OCCc2ccccc21)NC1CC(NC(C2(C)CCC(O)CC2)=O)C1 40780,C123CCC(N=C4N=C1NS4)(CO2)C3.Cc1cc(C(=O)NCC2CC2)nn1CCO 40781,C12(C(N3CCN(C(c4c(C)onc4C4CC4)=O)CC3)=O)CCC(CC1)C(C)O2 40782,C12CCC(=O)N(C1)C(=O)NCCN2CC.C1(C(=O)OC)CCCC(C)(C)O1 40783,CCC(C)CC(C(=O)NC1CN(CC)CC1C)NC(=O)Cn1cccc1 40784,N1(Cc2cc(C)ns2)CCC2(CCN(C(C3CC4(C3)CC4F)=O)CC2)C1 40785,C1(F)(CNC(CC2(COC)CC2)=O)CC(NC(=O)C(C)(C)C2CCCCO2)C1 40786,c1(C(N2CC(C(C)NC(Cc3c(C)noc3)=O)OCC2)=O)ccn2nncc2c1 40787,N1(C(CCCCN(C(CC=C)C)CC)C)CCN(C(c2ccccn2)C)C(=O)C1 40788,c1(C(N2CC3(C(NC(c4ccc(F)s4)=O)CC3)C2)=O)coc2ccccc12 40789,c1(C(N2CCC(C)(CNC(CN3C(C)CC3)=O)C2)=O)cnc2[nH]cnc2c1 40790,CC(CNC(=O)CNC(=O)CNC(C1CC2CC2C1)=O)S(C)(=O)=O 40791,c1(C(=O)NCCOCCN(C(CC(COC)(C)C)=O)C)cc(N)c2ncccc2c1 40792,c1(C(C(=O)NCCN(C(CC(C)(C)O)=O)CC2CC2)(F)F)ccc(F)cc1F 40793,C(CCC(C)C)NC(=O)O.C(=O)(C(O)C(F)F)NC(CCCCCC)=O 40794,N1(CC(CC)C2CCOCC2)CCC2C(C1)NC(=O)N2c1ccccc1C(=O)O 40795,C=CCCC(C1CC1)NC(=O)C(CNC(=O)C=NOC)N(C)C 40796,C1(NC(C2CCC(C)O2)=O)CCOCC1C(=O)NCCCCc1ncc[nH]1 40797,CC(C)CC(O)C(=O)NC1(C(=O)NCC(O)CNC(N)=O)CC(F)(F)C1 40798,c1(SC)ccc(CCC(=O)NCC(C)NC(C2CCN2C(C)(C)C)=O)cc1 40799,C(=O)(C1=NN(C)C(=O)CC1)N1C(C)CCC(NC(c2csc(C(C)=O)c2)=O)C1 40800,N1(C(C2OCCC(C)C2)=O)CC(C2(NC(=O)C(C)Cc3ccccc3F)CC2)C1 40801,CC1CN(C(=O)C(C)n2ccnn2)CCC1NC(=O)CSc1n[nH]c(O)n1 40802,c1(C(N2CCC(N(C(=O)CCP(C)(C)=O)C)C2)=O)ccc2cnsc2c1 40803,CC(C)C(O)C(F)(F)C(=O)NC1CN(C(c2onc3ccccc23)=O)CC1C 40804,c1(C(=O)NCc2ncn(-c3cccc(F)c3)n2)n[nH]c2c1CCSC2 40805,CC#CC1CN(C(C2CCN(C(c3cn[nH]c3)=O)CC2)=O)C1 40806,N1(C(COCCC#C)=O)CCC(C=C)(CC(=O)NOC(c2noc(C)n2)C)CC1 40807,Cc1cc(C)n(CCCNCc2ccccc2-c2ccc(F)cc2)n1 40808,C(c1cc(Cl)ccc1Cl)=CC(=O)NCCCNC(CCc1ccc(C)s1)=O 40809,C1(C(N2CCC(CCCNC(C(CSC)O)=O)CC2)=O)CCc2ccccc2C1 40810,N1(C(C2(O)CCN(Cc3n[nH]cc3Cl)C2)=O)CCc2cccc(O)c21 40811,CCCC(CNC(=O)CCOC(C)(C)C)NC1CC(N(C)C)C1 40812,c1(C(N2C(C(=O)NCC(CC(C)C)OC)C=CC2)=O)cc(C)nc(O)c1 40813,C1(NC(c2cc(OC)c(F)cc2)=O)CCN(C(C2CC2(Cl)Cl)=O)CCC1CO 40814,Cc1c(C(N2CC(CCNC(=O)CC3CCCC3)C2)=O)cnn1CC(F)F 40815,N(C1c2ccccc2CC12CCNCC2)CC1N(C(N)=O)CCC1 40816,N1(C(COC(C)C)=O)CC(NC(=O)CC2(C)CC2)C2CC12 40817,N1(C(CC2CN(C)C2)=O)Cc2ccccc2CC1CNC(C1CC2C=CC1C2)=O 40818,N1(C(c2cnc(C)[nH]2)=O)CCOCC(C)(CNC(=O)C(C)NC(C2CCC2)=O)C1 40819,CC1(C)C=C(C(=O)N2CCN(C3CCCN(c4ccncn4)C3)C(=O)C2)C1 40820,N1(C(C2C(C)C2C)=O)CC2CC(C1)N2C(=O)CN1CCNC(=O)C1 40821,N1(C(C(CC#C)C2CC2)=O)CCC2CN(C(c3cc4sc(C)cc4s3)=O)CC12 40822,c1(NC(C(=O)NCCC2N(C(CC(CC)OC)=O)CCC2)=O)cc(Cl)cc(Cl)c1 40823,CC(C)(CS(N)(=O)=O)C(=O)NCC1CN(C(C2(O)CCOC2)=O)CC12CC2 40824,CN1CCC(C(=O)NCC(=O)NC2(C)CCCO2)S1(=O)=O 40825,C1(C(N2CC(c3c(CNC(c4cnc(COC)s4)=O)nco3)C2)=O)CC2CCC1O2 40826,CC(c1cccnc1)=CC(N1CC(N(C)C(c2cccnn2)=O)C(F)C1)=O 40827,Cc1cc(NC(=O)C#CCNC(C2COCCC2C)=O)cc(CO)c1 40828,CCC(CC(=O)N1CCN(CC2CN(C(=O)CCNC(=O)CO)C2)CC1)OC 40829,Cc1cccc(F)c1CNC(=O)C(C1CCCO1)NC(=O)CC1CC=CCN1C 40830,c1(NC(CC2(NC(c3ccc(C)cn3)=O)CCCCC2)=O)ccc2occc2c1 40831,c1(C(=O)NCC(CC)(CC)NC(C2C(C=C)CC2)=O)c[nH]c2c(OC)nccc12 40832,C(=O)(CC(C)CC(C)C)NC(CC=CC)C(=O)N(C)Cc1cccnc1O 40833,c1(C(C(=O)NCC(CN(C(=O)CSCC(N)=O)C)O)(C)C)cccc(C(F)(F)F)n1 40834,C#CC#CC(C)(C)NC(=O)C(c1cccs1)NC(=O)CC1CC2CCC1C2 40835,O=C(C1=Cc2ccccc2C1)NCC1CCCC1NC(c1ccccn1)=O 40836,c1(OCC(=O)N(CC)CC2CCCN(C(=O)CC3(O)CC3)C2)cc(Cl)ccc1Cl 40837,C1(CCOC)CCN(C(=O)C(CCOCCO)NC(=O)CC2CCC2)C1 40838,c1(C(=O)OCC(CC)C)cccnc1-c1ccccc1 40839,CC1CCCC(C)C1NC(=O)CCOCCCNC(c1ccc(CF)cc1)=O 40840,c1(CN(c2ccncc2)CC=C)[nH]cnc1C 40841,C=CC(CC)C(=O)NC1CCCCC1CNC(=O)CN(c1nc(C)cs1)C 40842,C(CC(C)C(=O)NCCOCCNC(=O)CC(O)(c1ccccc1)C1CC1)OC 40843,c1(C(=O)NCCCCC(C)NC(=O)C(F)(F)C(F)F)cnc2c[nH]nc2c1 40844,CC1(CCC(=O)NC2(CCO)CCCCC2)CCCN1C(c1ccoc1)=O 40845,N1(C(CC2(C#N)CCCCC2)=O)CCC2(CCC2)C(NC(=O)CCNC(N)=O)C1 40846,C1(CNC(c2nnc(C(C)C)s2)=O)CN(C(c2ccc(O)nn2)=O)CC1C 40847,Cc1nc(C(=O)NC2CCCC(NC(C3CCC(=O)NC3)=O)C2)c2ccccn12 40848,N1(C(CN(CC#C)C=O)=O)CCCC(CN(c2cn(C)nc2C(F)F)C)CC1 40849,N1(C(=O)NCc2ccccc2)CCC2(CC1)CC(O)C2.C12(C=CCCC1)C(=O)O2 40850,C=Cn1nncc1C(=O)NCCCCCNC(c1c(Br)nnn1C)=O 40851,C(=O)(CC(CC(C)C)NC(c1ncccc1CC)=O)N(C(C=C)C)C 40852,C(C)(CC(=O)NC(C)(C)CN(C)C(c1cn(C2CCCC2O)nn1)=O)=C(C)C 40853,C(=O)(C(CCC1OCCO1)NC(c1nnnn1CCOC)C1COCCO1)OCC 40854,c1(C(=O)NC2C(NC(CCN(S(C)(=O)=O)C)=O)CC2)cccc(N)c1 40855,c1(C(N2CC(CCCCNC(C3(C#C)CC(=O)C3)=O)C2)=O)cccc(F)c1F 40856,C123C4C5C1C1C2C4C51CN(O)C1CCN(C1)C(=O)C3=O.c1(CC)ccc(Cl)cc1 40857,Cc1cc(C#N)c[nH]c1=NC1CN(C(C2CCCC2N(C)C)=O)Cc2ccccc21 40858,c1(C(=O)NCC2C(NC(CC(CC)CC)=O)CCC2)cc(Cl)cc2ccccc12 40859,c1(C(=O)NC(C2CCN(C(C3CCC(=O)N3C)=O)C2)C)ccc2nc(O)[nH]c2n1 40860,Cc1[nH]nc2ccc(C(N3CC4(C)CN(C(=O)C(=O)N(C)C)CC4(C)C3)=O)cc12 40861,S(=O)(=O)(c1cccnc1NCC1CCC(C)(C)N1)NC1(CC)CCCOC1 40862,C1(c2onc(CC)n2)(C(=O)OC)CCN(C(c2cc(C)[nH]n2)=O)CC1.CCCOC 40863,C1(C)(C(N(CCC2CN(C)C2)C)=O)CN(C(=O)CCN2CCOCC2)C1 40864,c1(C(C(=O)NCC(C(C)C)NC(C(CC)C)=O)(C)C)cccc(F)c1 40865,c1(OC(COCC)C)nccnc1C(=O)OC1CCN(CC(C)C)C1 40866,C1(CC)CN(C(c2cnn(C)c2CC(C)C)=O)CCN1C(=O)CS(=O)(=O)N(C)C 40867,c1(CC)oc(C)cc1C(=O)NCCC(C)N(C(=O)Cc1cc(C)cs1)C 40868,CC(C)CC(O)C(=O)NC1CCCN(C(c2cccc(C3CC3(F)F)c2)=O)C1 40869,N1(C(c2ccc(C)c(Br)c2O)=O)CCC2CN(C(C3CC3(C)C)=O)CC2CC1 40870,C1(N(C(C(c2cncnc2)C)=O)C)CCCN(C(=O)CCc2cnn[nH]2)C1 40871,N1(C(C2C(NC(=O)CC3CSCCO3)COC2)=O)CCC2(CC1)CC(O)C2 40872,c1(OC)ccccc1OCCCN(C)C(=O)NCCNC(C)=O 40873,c1(C(N2CC(C(=O)NCc3c[nH]c(=N)o3)C2)=O)cc(CN(C)C)on1 40874,C1(NC(c2n(CC)ncc2)=O)CC2(CCN(C(C3CC(N4CC(O)C4)C3)=O)C2)C1 40875,C(=O)(C1=C=CCCC1C)N1CCC(CNC(c2c(C)sc(Cl)n2)=O)C(O)C1 40876,c1(C(N2C(CN(C(=O)C(O)C3CCC3)C)CCC2)=O)ccc(CC=CCO)nc1 40877,Cc1ccc(OCCCC(N2CC(NC(=O)C(C)NC=O)C(C)C2)=O)cc1 40878,N1(c2ncc(C)c(O)n2)CC(CNC(=O)CCCn2cncn2)OC(C)(C)C1 40879,N1(C(=O)COCC2CCCO2)CCC2C(C1)CN2C(c1cc(C(F)(F)F)c[nH]1)=O 40880,c1(OC)nccc(C(C)NC(=O)NC2(C(C3CC3)N(C)C)CCC2)n1 40881,N1(C(CCC#C)=O)CCCC1(C)C 40882,c1(CNC(C(CC)OCC)=O)nnn(C)c1C(N1CCC(F)(C(=O)OC)C1)=O 40883,Cc1cc(F)c(CC(N2CCC(NC(=O)CNS(=O)(=O)N(C)C)C(C)C2)=O)cc1F 40884,C1(C#N)(C(=O)NC(C)CC(C)NC(c2conc2C(C)(C)C)=O)CCN(C)C1 40885,CCC(C)CCCCC(=O)NC1C2CN(C(=O)C=CC(C)(C)NS(C)(=O)=O)CC12 40886,c1(C(=O)NCC2CC(NC(C3=CCC(C)CC3)=O)C2)cccc2nc(O)oc12 40887,C1(CC(=O)N(C(CC#C)C)C)CN(C(=O)CC2CCC(=O)C2)CC12CC2 40888,c1(CCC)ncc(C(N2CC(C(=O)N(C)CCC3CN(C)C3)(CC)C2)=O)s1 40889,c1(C(=O)NC(C2CCCN(C(c3n(CC)ncc3)=O)C2)C)cc2n(c1)CCSC2 40890,c1(C(N2CC(CNC(C3(c4cc[nH]n4)CC3)=O)C(O)C2)=O)ccn2c1CCCC2 40891,c1(C(N2CC(CC(C)NC(c3c(CCC)[nH]cc3)=O)C2)=O)cnc(O)n1CC 40892,c1(C(=O)NCC(COCC)(C)C)ccnnc1C.C12(CCC1)C(=O)N2 40893,C=C(CNC(=O)C(CCC1CC1)NC(C1CC(=O)CS1)=O)C(F)(F)F 40894,Cc1ccccc1C1(C(=O)NCC2CC(NC(c3n[nH]cc3Cl)=O)C2)CC1 40895,C1(CNC(COCCC=C)=O)CN(C)CCN1C(c1cc(C2CC2)nc(O)c1)=O 40896,N1(C(C2(F)CN(C(c3cc(C)no3)=O)C2)=O)CC2CCC2(C)C1 40897,c1(C(=O)NCC2C3CN(C(CC(=O)NC4CC4)=O)CC32)ccc2scnc2c1 40898,N#Cc1ccc(SCC(=O)NCC2(O)CN(C(N)=O)C2)cc1 40899,c1(C(=O)NCC2(F)CC(CNC(=O)CC3CCC4CC34)C2)cccn2nncc12 40900,Cc1[nH]c(C#N)cc1C(N1CCC(N(C)C(c2coc(C(F)(F)F)n2)=O)C1)=O 40901,C1(CC)CN(C(C2CCC3(C2)N=N3)=O)CCC1Nc1nc(C)cc(C)n1 40902,C(CN=c1[nH]c(C)cc(=NCc2ncc(Br)cn2)[nH]1)c1ccc(OC)cc1 40903,c1(C(N(C2CCN(C(=O)CCCOC(C)C)CC2)CCC)=O)cn(C)c(=O)n1C 40904,c1(CCCNC(=O)CCC(F)Cl)cccc2c1OCCC2 40905,c1(C(N2CCC(CCNC(C(CCCC)CC)=O)C2)=O)cnc2cccc(C)n12 40906,c1(C(=O)NCCCCNC(C(C)(C)OC(C)=O)=O)snc(Cl)c1Cl 40907,C1(NC(c2c(CC)c(C)sc2)=O)CCCN(C(c2ccc(=N)[nH]c2)=O)CC1 40908,C(=O)(N=c1[nH]nc(-c2ccc(OC)cc2)s1)N1C(CC(C(=O)OC)F)CC1 40909,C1(O)(CNC(c2c(CNC(C=NOC)=O)ccs2)=O)CCCC1C 40910,O=C(CCCn1cncn1)NCCCc1cn(C2CCCC2O)nn1 40911,C(CC1=CCCCCC1)NC(c1c(C)cc(CNC(=O)Cc2cnsc2)o1)=O 40912,C1(NC(C2(CCOCC3CC3)CC2)=O)CCN(c2ccc(Br)cc2)C1=O 40913,Cc1nc(C(=O)NCC2(C)CCC(NC(=O)CCC(=O)N(C)C)C2)c(C)n1C 40914,C1(C(C(F)F)OC)(CSC)CC(C)(C)C1.C12CC(CO1)CNC(=O)NC2 40915,CC1(C(=O)NC2CCC(CC(=O)NC3CCOCC3F)C2)CC2C=CC1C2 40916,C#CC1CCCCN1C(=O)C(F)CC1CN(C(c2cc(C(C)=O)[nH]n2)=O)C1 40917,C1(CCC)(N(C(=O)C(C)SC(F)(F)F)CC2C=CCC2)CCCNC1.Cc1ncco1 40918,C1(NC(=O)C#CCNC(=O)CCC2CCC(=O)C2)CCN2CCCCC12 40919,C(CCC(C)NC(c1cscc1OCC)=O)NC(CN(S(CC)(=O)=O)C)=O 40920,N1(C(COC2(C)CN(C(C(C)CC(N)=O)=O)C2)=O)CCC2(CC1)CN(C)C2 40921,N1(C(COC)=O)CCN(C(=O)CNC(c2cccs2)=O)C(C)CC1C 40922,c1(NC(CC2CC(=C)C2)=O)cc(Cl)ccc1CNC(=O)CC1CCOC(CC)C1 40923,c1(C(=O)NCCCCC2CN(C(c3cnc(S)nc3)=O)C2)c[nH]c2ncccc12 40924,c1(NC(CC2N(C(Cc3nc(C)sc3)=O)CCC2)=O)ccc(C(N)=O)cn1 40925,C1(NC(C2C(C=C)C2)=O)CCCN(C(c2cnnn2C)=O)C1 40926,CC(C)(C)C(CCc1ccccc1)C(=O)NC1(C)CCCN(C(=O)C=CI)C1 40927,Cc1cc(C)cc(C=CC(=O)NCC(CNC(C2C(C#N)C2(C)C)=O)CO)c1 40928,C(=O)(C1=CCCC1(C)C)N(C)CCOCCN(C)C(c1nonc1N)=O 40929,c1(C(N2CCC(NC(CN(C)C)=O)C2(C)C)=O)cnc2ncc(Br)cc2c1 40930,N1(C(C2CN(CC(C)C)C(=O)C2)=O)CC(NC(=O)COc2ccon2)CCC1C 40931,CC(C)(C)C(CO)C(=O)N1CCC(N(CCO)C(C2CCn3ncnc3C2)=O)C1 40932,N1(C(c2c(C)ccn2C)=O)CCC2(CC1)CN(C(=O)C1=CCCCC1C)C2 40933,c1(-c2cnc(N3CCN(C(C(C)Cc4cnc[nH]4)=O)CC3)s2)cc(Cl)ccc1Cl 40934,c1(C(N(CC#C)C)=O)cc(CNC(C2(Cl)CC2)=O)no1 40935,CCC(C)CC(=O)C(=O)NCC(C(=O)N(C1CCC1)CCN(C)C)C(C)C 40936,C(c1ccccc1C)=CC(=O)NC1(C(=O)NCC(CC)O)CCSC1 40937,N1(C(C2(CC=C)CC2)=O)CC(C(=O)NC(C)CC(C)(C)CO)CCC1(C)C 40938,c1(C(=O)NCC2C(C(=O)NCC3CC(O)C(O)C3)C2(C)C)ccc([N+](=O)[O-])[nH]1 40939,C1(C(=O)NCC#CCNC(c2c(OC(C)C)cccc2)=O)CCCC1S(C)(=O)=O 40940,c1(CN(C)C(c2cnn(CCNC(c3cnccn3)=O)c2)=O)ccccc1Cl 40941,CC1CCN(C(=O)CC2CCC2)CC1CNC(=O)CNC(=O)NC1CC1 40942,N1(C(C(CC)=O)=O)CCC(O)(c2cn(C(c3ccccc3F)C)nn2)CC1 40943,c1(OCC)oc(C)nc1C(N1CCN(C(=O)CC2CCC(C)(C)O2)CC1)=O 40944,C1(NC(COCC#C)=O)CCOC(C(=O)N(C)Cc2cccn2CC)C1 40945,N1(C(c2c(Cl)cn(CCC)n2)=O)CCCC(N=c2nn[nH]n2C)C1 40946,c1(C(=O)NCC2C(NC(C3CCCN(C)C3)=O)COC2)cc2sccc2[nH]1 40947,CC(CSC(F)(F)F)C(=O)NCC1CCN(C(=O)CCOC2CCC2)C1 40948,CC(C(=O)NC1(C)CN(C(=O)C(c2cncn2C)O)C1)C(=O)N1CCOCC1 40949,C(=O)(C1Cc2ccc(Cl)cc21)NC1C(C)N(C(C2CC3CCC2O3)=O)CC1 40950,c1(CCC(=O)NC(C(=O)N(CC(C)C#N)C)C2(O)CCC2)cn(C)nn1 40951,C1(C(N2C3C(NC(=O)CSC4CC4)CC(CC3)C2)=O)CC2CCC1CC2(F)F 40952,N1(C(CC2C=NN(C)C2=O)=O)CC(O)(C2(CNC(c3ccc(CO)o3)=O)CC2)C1 40953,C1(CC(=O)NCCCOCCNC(=O)Cc2cnc[nH]2)CCC2CC12 40954,c1(C(N(C2CC(NC(CC3C(C)COCC3)=O)C2)C)=O)cc(C(=O)O)ccc1N 40955,Cc1ccc2c(c1)CCC2C(=O)NCC(O)CCNC(=O)CCOCC(C)C 40956,C(CC(C)C)(C(=O)N(CC(=O)NNC(=O)C1CCCC1)c1ccco1)NC(C)=O 40957,c1(C(=O)NCC(CC(=O)NCC(C(C)(C)C)OC)(C)C)ccc2nccn2c1 40958,C1(CC=C)(C(=O)NCc2ccccc2OC)CCCN1C(=O)C(C)C1CCC1 40959,c1(CC(=O)N(C2CN(C(=O)COC(C)=O)CC2F)CC)nc(C)sc1Br 40960,c1(C(=O)NCC2C(CNC(CC(=O)NCC)=O)C2)cc(-n2ccnc2)nn1C 40961,n1(CCCC)ncc(C(=O)NC2(CO)CCN(C(c3cnc(S)n3C)=O)C2)c1C 40962,C=CC1(C(=O)NC(c2cccc(O)c2)C)CCN(C(c2[nH]ccc(=O)c2C)=O)C1 40963,c1(OC)nc(C)ncc1C(=O)NCC(C)NC(C1CCC2CC2CC1)=O 40964,C1(CNC(C=CC(C)C)=O)C2CCC1CN(C(C1CCC(F)(F)C1)=O)C2 40965,C1(OC)CCCCC1CC(=O)NCC1CCN(C(c2cncnc2C(C)C)=O)C1 40966,N1(C(Cc2c(C)nc(SCC)s2)=O)CC2(CCCC2)OCC1CO 40967,Cc1cc(F)cc(C(=O)NC(Cc2cnc[nH]2)C(=O)O)c1Br 40968,C1(NC(c2n(CC)nnc2)=O)CN(C(c2ccc(C)cn2)=O)CC1N=[N+]=[N-] 40969,C(=O)(CC(C)CC(C)C)N1C(CNC(c2n(C(CC)CC)ncc2)=O)CC1 40970,C1(NC(C23C(C)(C)OCC2C3)=O)CCCC12CN(C(c1ccc(O)nn1)=O)C2 40971,CN1CC(O)CC1(C)C(=O)NCC(N1CCN(C(=O)COC(F)F)CC1)(C)C 40972,CCCC(CC1CCCC1)C(=O)NC(C)(CNC(C1CC(F)(CO)C1)=O)CO 40973,Cc1ocnc1C(=O)NC(C)(C)CN(C)C(C1CCCC1c1ccccc1)=O 40974,C1(NC(CC(C=C)CC)=O)CCSC12CN(C(=O)C(CC(C)C)N(C)C)C2 40975,C1(CC(=O)N(CCOC(C)=O)C)CCN(C(c2c(C)noc2C(F)F)=O)CC1 40976,CC1C(C(=O)NCC2CC3(CCC3O)C2)CCCN1C(c1ncncc1Cl)=O 40977,C#Cc1cnc(NC(C2CCN(C(=O)Nc3ccc(F)c(Br)c3)C2)=O)cn1 40978,C1(C(=O)NCC(C)N(C(C2(C3CC3)CCCO2)=O)CC)COC(C)(C)CO1 40979,Cn1ncc2nc(O)c(C(N3CCOC(CCNC(C4C=CCC4)=O)C3)=O)cc12 40980,C1(NC(COCCCC)=O)CCN(C(c2cccnc2SCCC(C)C)=O)CC1 40981,C(CN=c1[nH]c2c(c(=NC3CCCc4occc43)[nH]1)SCC2)C1CCN(CC)C1 40982,C(CC(C)(C)C(=O)NCCC(C)CCNC(c1cncc(N(C)C)c1)=O)SC 40983,Cc1[nH]nc(C(=O)N(C(C)C(=O)N(CC(c2ncccn2)C)C)C(C)C)c1C 40984,Cc1ncnc(C(=O)NCc2ccc(CNC(=O)C(C)C(C)C)c(F)c2)c1C 40985,c1(C(=O)NCC(CNC(C2CCN(CC(C)C)C2)=O)CO)cccc2ccnn12 40986,N1(C(c2cccs2)=O)CCC2(C(=O)NCCCC(F)(F)F)COCCC12 40987,N1(C(CCC2CCC(=O)C2)=O)CCCC(F)(C(N2CCC(CCO)CC2)=O)C1 40988,N1(C(C2CCCCS2)=O)CCOC2(CCC(N=c3[nH]c4ccc(F)cc4s3)CC2)C1 40989,C1(C(=O)NCCC2(O)CCN(C(C(C)(C)OC(C)C)=O)C2)CCCCC12CCC2 40990,N1(C(C(c2ccc(Cl)s2)C)=O)CCN(C(=O)COCC(C)(C)C)C(CC2CC2)C1 40991,C12CC3CC1N(C3)C(=O)CN(C)CC1C(CC1)C(=O)N2C.S(C)(=O)(=O)N 40992,C1(N(CC(=O)NC(C)CCCCCC=O)CCC)CCc2ccccc2C1.OC 40993,C(CN=c1[nH]c(=NCCN2CCCC(C)C2)[nH]c2c1COC2)(C1CCCC1)SC 40994,CC1CNC(=O)CN1C(C1(NC(c2coc(C(N)=O)c2)=O)CC(F)(F)C1)=O 40995,C1(C(=O)NCC2N(CC)CCCC2)CCN(C(=O)CCCCCSCC)C(C)C1 40996,C1(C(=O)NC2CCN(C(CCOC)=O)C2C(C)(C)C)CN(C)C(=O)CCO1 40997,C1(SC)CN(C(C2CCC(=O)N2)=O)CC1NC(c1ccnc(Cl)c1)=O 40998,C(=O)(C1CCc2nnc(C)n21)NCC1(F)CC(NC(C2(OC)CCOC2)=O)C1 40999,Cc1ccnc(O)c1C(=O)NCCC1C(C)CCCN1C(=O)CSCC(F)F 41000,C12CCCN1C2=O.n1(CC2N(C(=O)NC)CC2)cc(C(c2ccccc2)O)nn1 41001,c1(CC)ccc(C(=O)C(=O)NC23CC(CNC(c4ncsc4C)=O)(C2)C3)s1 41002,Cc1coc(C)c1C=CC(=O)N(C1CN(C(C2CCC(C3CC3)C2)=O)C1)C 41003,C1(OCC#C)CCCN(C(C2CCC(CNC(=O)C(C)O)C2)=O)C1 41004,Cn1nccc1CC(N1CSCC1C(=O)NOC1CCOC1)=O 41005,c1(C(N2CC(CCOC)(NC(=O)C(=O)N(C)C)C2)=O)cc(N)c(C)cc1C 41006,CCC(C)C(C(=O)NC1CCCC1CNC(=O)CCCOC)N(C)C 41007,CN1CCC(C(N2CCN(C(=O)C=Cc3cn(C)cn3)C(CCO)C2)=O)CC1=O 41008,C1(NC(C(C)=CC)=O)COC2C(NC(c3cnn(C)c3C(C)C)=O)COC12 41009,Cc1c(C(=O)NC2CCN(C(c3ccc(CO)[nH]3)=O)CC2)cnn1C1CCCC1 41010,CCCC(C)(C)CC(=O)NCC1CCN(C(C2C3CCC(=O)C23)=O)C1(C)C 41011,c1(C(=O)NCCN(CCC(=O)NCC(C)O)CC)c(O)nnc(C)c1C 41012,CC1(C)CCC(CNC(=O)C(=O)NC2CCCNC2=O)O1 41013,c1(C(=O)NCC(N(C(C(CC)(C)O)=O)C)C2CC2)cc(Br)ccc1C1CC1 41014,C(=O)(CC1=CCCCC1)NCCC(C(=O)NCC(CC)O)(C)C 41015,c1(C2CC(C(N3CCC(C(=O)O)CC3)=O)(C(=O)O)C2)cc(Cl)c(O)c(Cl)c1 41016,CC1C(NC(=O)Cc2csc(Cl)c2)CCN1C(=O)CCc1ccc[nH]1 41017,c1(CC)ncc(C(N2CCC(CN(C)C(c3ncccn3)=O)CC2)=O)c(C)n1 41018,C1(CNC(CC=C(C)C)=O)CC2(CCN(C(=O)C(C#N)C(C)C)CC2)CO1 41019,C(=O)(C(COC)NC(=O)CCc1nc[nH]n1)N(CC(=O)N(CC)CC)C1CC1 41020,N1(C(c2cc(CC)[nH]n2)=O)CCC(C)(NC(=O)CCCOC(C)(C)C)C1 41021,c1(OCC)ccc(Br)cc1S(=O)(=O)NCc1ccc(C2CCCCC2)cn1 41022,c1(N(C)CCO)nnc(-c2ccccc2Br)n1CCCN1CCC(C(F)F)C1 41023,C1(C(=O)NC)CCN(C(=O)C(O)C(C)(C)C)O1 41024,C(=O)(CCCC(=O)OC(C)(C)C)NCCC(C)CCNC(C1CC(=O)N(O)C1)=O 41025,C(=O)(C1=C(Cl)CC1)NCCCCC1CN(C(C(C)CC2CCC2)=O)C1 41026,C1(C(=O)NCCC(C)(C)NC(=O)C=C(Cl)Cl)CC(C(C)(C)C)=NO1 41027,c1(N(C)C(C(C)N=c2[nH]nc(C#N)s2)=O)cnc2[nH]c(C(F)(F)F)nc2c1 41028,C1(C(C)C)N(C(=O)N(c2ccncc2Br)C)CC12CCC2 41029,c1(NC(COCCC(NOCCC(C)O)=O)=O)ccc(F)cc1O 41030,CC1CC(=O)NC1C(=O)NCC=CCNC(=O)CCOc1cccc(C(N)=O)c1 41031,c1(C(=O)NCC2CCN(C(C3ON=C(C)C3)=O)CC2O)cc(F)c(F)cc1O 41032,c1(OC)cc(C(=O)NCC2(OC)CN(C(c3ccnc(Cl)c3OC)=O)C2)cc(C)n1 41033,C12(C(=O)NCC(CNC(CCCOC(C)C)=O)F)CC3CC(F)(C1)CC(F)(C3)C2 41034,C(=O)(C1=C(C)OCC1)N1C(C(N(CC(CC)C)C)=O)(COC)C=CC1 41035,CC1CCCC(CN2CCN(CC(=O)NC3CCN(Cc4cccs4)C3)CC2)C1 41036,N1(C(C(C2CC2)OC)=O)CC(O)(CNC(C2(CO)CCC2)=O)C1 41037,c1(CC)n[nH]c(CC)c1CC(=O)NN1CCCC(c2cn(C3CCCC3O)nn2)C1 41038,Cn1ncc([N+](=O)[O-])c1C(=O)NC1CC2(C1)CC2NC(=O)Cc1ccnnc1O 41039,C1(CC(=O)N(C)CCOCCNC(c2ccc(Br)cn2)=O)COCC(C)(C)O1 41040,C1(C(=O)OC)CCCC(F)C1.c12cn(nn1)C1COCC1C(=O)NOCC2(C)C 41041,Cc1cccc2nc(C(N3CC4CCC3CN4C(C3(Br)CC3)=O)=O)cn12 41042,C1(NC(c2c(C)c[nH]c2)=O)CC(C(=O)NCC(C)(C)F)C1(C)C 41043,C1(CC(=O)N(C2CCCC2)CCNC(CC(C)N(C)C)=O)CCNC(=O)C1 41044,N1(C(c2c(C)con2)=O)CC2COCC2(C(=O)NC(C)CC2CCC2)C1 41045,C(=O)(CCCCCS(N)(=O)=O)NCCC1CCC(NC(C=CC=CCC)=O)C1 41046,c1(C(=O)NC2CC(CNC(C(CC)SC)=O)C2)oc2c(C)ccc(C)c2c1C 41047,C(CC(O)C(=O)N(c1cccc(F)c1)C)NC(C1C(CCOC)C1)=O 41048,CCCCC(CNC(=O)NC(C)C)NC(C1CCNCC1C)=O 41049,C1(C(=O)NC2CC3CN(c4nnc(C#N)s4)CC32)CC2(CCCCC2)CO1 41050,c1(N(C)C)ccc(CCC(=O)NC2CC(C(=O)Nc3ccc(F)cc3)C2)cn1 41051,N1(C(c2nn(CC)c(=O)cc2)=O)CCOC2CCN(C(C3(O)CCCC3)=O)CC12 41052,N1(C(C2(C)CCCCC2)=O)CC2(CNC(=O)C=C3CCCCC3)CC1CO2 41053,CC1C(=O)CCC1CC(=O)NC1(CCNC(c2coc(C3CC3)n2)=O)CCC1 41054,N1(C(C=C(C)NCC(F)(F)F)=O)CC(F)(c2ccccc2)C1 41055,C1(CNC(CC2(CC(=O)OC)CCCC2)=O)CC(F)CN1C(c1cc(F)c[nH]1)=O 41056,C1(NC(Cc2cn(CC)nn2)=O)CC2(C1)CC2NC(C1CCCN1CC(C)=O)=O 41057,C1(NC(c2ccc(C(F)(F)F)cn2)=O)CC(CNC(C2CC(O)C2)=O)C(O)C1 41058,c1(C(=O)NCC2CC(OC)CN2C(C2C(C)C2C)=O)c[nH]c2c(C#N)cccc12 41059,Cc1cc(=NC(=O)c2cc3cc(C(=O)NC4CCC(F)(F)C4)ccc3[nH]2)[nH]n1C 41060,N1(C(C(C)=C(CC)C)=O)CCN(C(C2CCN(CCC)CC2)=O)C(C(C)C)C1 41061,c1(C(=O)NCC(O)CNC(=O)C2=COCCO2)cc(F)ccc1-n1cccn1 41062,Nc1cc(C(=O)NCC(CO)NC(=O)CC2CC3CC3C2)cc(C(F)(F)F)c1 41063,CCC1=C(C(=O)N2CCCCC2C2(NC(=O)CCCSC)CC2)CCCO1 41064,C(C(CC1CC1)C(=O)Nc1cscc1C1CC1)NC(C(C)CC1CC1)=O 41065,C12(NC(Cc3onc(CC)n3)=O)CCC(C(=O)NC(C)C(C)(C)OC(C)C)(CC1)C2 41066,N1(C(C(C)=C(CC)C)=O)CC2(NC(=O)CCc3cccc(Cl)c3)CC1C2 41067,Cn1ccc2ccc(C(N3CCC4(CCCC4NC(=O)C=C4CCC4)C3)=O)cc12 41068,c1(N)cnc(Cl)c(Br)c1.n1(C)nnnc1C1(CCOC)CCCC1 41069,C1(NC(C2C(C)(C(C)C)C2)=O)CCC2CN(C(C3CC(O)C3)=O)CC2C1 41070,N1(C(C(C(C)C)S)=O)CCCC2(C1)CN(C(=O)C(c1ccccn1)C)CCO2 41071,C(=O)(C(C)(C)CC(=O)OC)N1CC(OC)(CNC(C2CC3CC2CO3)=O)C1 41072,CC(=O)CCCCCCC(=O)NC1(CNC(=O)C(C)NS(C)(=O)=O)CCCC1 41073,c12cccc(c1)COC(=O)N1C(CC1)C(=O)N2.Cn1nncc1CN1CCCC1 41074,CC1(C)C(C(N2CC=CC2(C)CO)=O)CCN1C(c1coc(C(F)F)c1)=O 41075,N=c1[nH]c2c(s1)CCCC2C(=O)NC1COCCN(C(=O)C2=COCCO2)C1 41076,c1(CC)ccc(C(=O)NC2(CC(N3C(C(=O)OC)CC3C)=O)CCC2)nc1 41077,C1(NC(C(C)NC(=O)OC)=O)CC=C(C(=O)Nc2cnc(C(C)C)nc2)C1 41078,C1(C(=O)NCCOCCNC(=O)Cc2ccnc(Cl)c2)CCCC2(CCC2)O1 41079,CC1CN(C(c2cn(CCNC(C3CNC(=O)N3)=O)cn2)=O)CCO1 41080,C1(CC(C)Nc2cn(C)nc2Br)CCCN(C(=O)NC2CCC2)C1 41081,c1(C(N2CCC(O)(CN(C)C(C3(C)COC3)=O)CC2)=O)cc2n(n1)CCOC2 41082,Cn1cc2cccc(NC(C3CCC4(CN(C(=O)C(N)=O)C4)O3)=O)c2n1 41083,n1(CCCOC)cc(-c2noc(C3CCCN3C(N)=O)n2)cn1 41084,C(=O)(C(C)(C)CC(C)C)NCC1(NC(c2c(Cl)ccc(OC(C)=O)n2)=O)CCC1 41085,c1(C(=O)NCCNC(=O)CSC2CCOC2=O)cnc2ncnn2c1O 41086,N1(CCC(N2CC(C(C)NC(=O)CCc3nc(=N)[nH][nH]3)C2)=O)CCN(C)CC1 41087,C1(C)(C(=O)NCCCCN(C(=O)C(O)C2CC2)C)CCCO1 41088,N1(c2c(OC)cncn2)CCC(C2CC2)(CNC(c2csc(CO)n2)=O)C1 41089,C1(OC)CCC2(C(=O)NC(C)(C)C(C)NC(c3ccn(C)c3)=O)CC12 41090,N1(C(c2cccc(OC(C)C)c2)=O)CCN(C(=O)CC2CCCC2)C(C#N)C1 41091,N1(C(C2CCC(C)O2)=O)CC2(CCC(CNC(c3cccc[n+]3[O-])=O)O2)C1 41092,N1(C(CC(CC)C)=O)CC2CC(NC(c3[nH]c(=N)sc3COC)=O)CC1C2 41093,c1(NC(C(=O)NC(c2ccc(OC)cc2)CC#N)=O)cc(C)ccc1C 41094,c1(C(=O)NCC2CN(C(C(C(C)C)OC)=O)C(C)C2)cncc2c(O)nccc12 41095,C1(C(=O)NCCOCC(F)F)CCCN(C(=O)C(C2CCCCCC2)O)CC1 41096,N1(C(CS(N)(=O)=O)=O)CCC(S(=O)(=O)CN2CCCC2=O)CC12CC2 41097,C1(O)(C(C)NC(C(CCC)O)=O)CCN(C(c2cc(C)sc2C)=O)CC1 41098,c1(C(N2CC(C)(C(=O)OC)OCC2)=O)ccc2ccccc2n1 41099,N(C(=NCCN(C)C)NCC1CC(C2CCC2)C1)Cc1c(OC)ccc(Cl)c1 41100,c1(C(=O)NCC2(OC)CN(C(=O)Cc3ncc(Cl)s3)C2)cccc2c1NCC2 41101,C1(C(N2CC(C#C)(O)C2)=O)CCC(C)(C)N(C(=O)CN2C(=O)CNC2=O)C1 41102,CC1CCN(C(c2sccc2C2CC2)=O)C(CNC(c2cc(N)cc(F)c2)=O)C1 41103,C(CCC(=O)NCc1nocc1C(=O)NC1CCCSC1)OC(C)=O 41104,c1(C(=O)NCC2N(C(CCCCOC(C)C)=O)CCCC2)nc2c(s1)COCC2 41105,c1(CCC=C)ccc(C(N2CC(CCO)(C(=O)NCC3CNC(=O)C3)C2)=O)cc1 41106,C(=O)(C1=CC2CCCCCC12)N(CCNC(CS(C(C)(C)C)(=O)=O)=O)CC1CC1 41107,c1(C(=O)OC)sc(NC(C23CC(C)(C2)OC3C)=O)c(C(=O)OCCOC)c1C 41108,Cc1cccc(OCC(=O)N(CC(C)(C)NC(C23CC2COC3(C)C)=O)C)c1F 41109,N1(C(=O)Nc2cnn(-c3cccc(C)c3)c2C)CCN(C(=O)OC(C)(C)C)CC(O)C1 41110,c1(NC(=O)CC2CCN(C(c3ccc(I)c(O)c3)=O)C2)ncc(I)nc1Cl 41111,C1(C(=O)NC2CC(NC(CN3CCC(C)CC3)=O)C2)SC2C=CC1CC2 41112,N1(C(C)C)CCOC(C)(C(F)(F)F)C1.n1(CC(=O)N)cc(CCO)nn1 41113,C(=O)(N=c1cc[nH]c2cc[nH]c12)c1c[nH]c2ccc(-c3c(OC)cccc3)cc21 41114,c1(NC(C2C(Br)(C(=O)OCC)C2)=O)cc(Br)cc(F)c1O 41115,C12(NC(C(CSC)C)=O)CC1CN(C(=O)Cc1ccnn1C)C2 41116,N1(C(c2ccc(CC)nc2)=O)CCN(C(=O)C=CCF)CC1c1ccnn1C 41117,C(CCC(=O)N1CCCC1C1(C(=O)NC2(CC3CC3)CC2)CC1)N(C)C 41118,CCC(CCC(=O)NC1CCC(CCOC)C1)NC(c1cncn(C)c1=O)=O 41119,C(c1cc2ccccc2o1)=CC(N1CC(CCNC(C(C=C)(C)C)=O)C(C)C1)=O 41120,C(CCCC(CO)NC(C1(N2CCCC2)CC1)=O)NC(CC(CC)C1CC1)=O 41121,CCCCCC(F)C(=O)N(C)CCN(C(=O)Cc1cn(C2CC2)cn1)C(C)C 41122,C=CCC(C)(C)C(=O)N1CCCOC(CNC(C2CC2C(C)O)=O)C1 41123,C1(C(=O)NCCC(C)NC(CCN(CCC)C)=O)CCCSC1 41124,c1(CCC)sc(C(=O)NC(C)CCN(C)C(c2nnsc2C)=O)cc1Br 41125,C1(NC(c2ncn(CC)c2)=O)CC(NC(=O)CC2CCC3CC23)C(O)C1 41126,CC1(C(=O)NCc2cc(Br)cs2)CC(NC(=O)Cc2ccoc2)C1 41127,C1(C)(CNC(C2(C)CCN(C(C)=O)C2)=O)COCCN(C(=O)Cc2cc[nH]c2)C1 41128,C(CC1CC1)(C(=O)NC(c1ccccc1)CCCNC(=O)CC1(C)CC1)OC 41129,C1(C(=O)NCC(C2(c3cc(C)c(O)nn3)CC2)NC=O)CCc2ncsc2C1.C1CC1 41130,C(=O)(CS(=O)CCC(F)(F)F)NCCc1c(CNC(CCC(N)=O)=O)nco1 41131,C(c1ccc(F)c(Cl)c1)=CC(=O)NC(C1(O)CN(C(c2ccccn2)=O)C1)C 41132,O(NC(=O)CC(CC)NC(=O)CC(=O)OCC)CC(=O)OC(C)(C)C 41133,c1(CNCC(=O)NCCOCCOCC(C)(OC)OC)ccc(S(N)(=O)=O)cc1 41134,CC1CN(C(=O)CCSc2ccc(F)cc2)CCCN1C(=O)CC#N 41135,c1(C(=O)NC(CC)CN(C)C(c2ccsc2S(N)(=O)=O)=O)cnn2cccnc12 41136,C1(CC)NC(=O)N(CCOC(=O)CCCSC)C1=O 41137,C12(CNC(C3N(C)CCCC3)=O)CCC(CC1)CN2C(c1cc(Cl)cnn1)=O 41138,C(=O)(C1=C(Cl)CCOC1)NC1C(CNC(c2nc(CCOCC)oc2)=O)CCC1 41139,CC(C)C(C(=O)NC1(CC=CC(=O)NCC23CC(F)(C2)C3)CCC1)N(C)C 41140,C1(C(N(CCCC)CC(N)=O)=O)OCCC1NC(c1cc(C)ns1)=O 41141,C1(C(=O)NCCn2c(C)cnn2)CCN(C(=O)CCc2cccn2C)C1C 41142,N1(C(c2cn(C)nc2C(F)(F)F)=O)CC2CCC1C2NC(=O)Cc1cnccn1 41143,C1(C(=O)NCCCc2cc[nH]n2)CC2CC1CN(C(=O)Cn1cnnc1)C2 41144,C=CCCC(C(=O)NCc1ccnc(OC)n1)NC(c1cnc(OC)nc1)=O 41145,C1(CNC(C2(C)CCN(C)C2)=O)CN(C(C2CC(C#N)C2)=O)CCC12CCC2 41146,CC1(C)CC(NC(=O)C=CBr)CCN(C(c2ccnc(F)c2Cl)=O)C1 41147,C1(C(=O)NCCN(OC)C)CC2(CC(NC(=O)CC(C)(C)C)C2)C1 41148,C(=O)(C1c2ccccc2C2CC1C2)N(C)CC1(CNC(CC=CCC)=O)CC1 41149,N1(C(c2ccc3c(c2)CCC3)C(=O)NC(C)C)CC(CO)CC(C)(C)C1 41150,CC1(C(=O)NC(CNC(=O)CCCc2cc[nH]n2)C2CC2)CCC(=O)N1 41151,CC1(OC(F)F)CCN(C(=O)NC)CC1.C1(C)(C(=O)O)CCCOC1 41152,c1(C(N2CCCC(n3cc(C(C)(C)N(C)C)nn3)C2)=O)cc(O)nc(Cl)c1 41153,C=CCC(CNC(C1CCSCC1)=O)NC(=O)C(C1CC1)SC 41154,C1(NC(CC2C(C)CCC2)=O)CN(C(c2ccnc(OCCOC)c2)=O)CC1C 41155,C(=O)(N1CC(n2cc(C3(C)CCCCO3)nn2)CO1)c1n(CC)ccn1 41156,c1(C(=O)NC2(C)CN(C(c3ccc(COC)o3)=O)C2)cccc(C2CC2)c1C 41157,N1(c2snc(C(=O)OC)n2)CCC(C)(C)C(CNC(C2(C)CC2)=O)C1 41158,CC1(C)Cc2cccc(S(=O)(=O)NCCn3ccc(O)nc3=O)c2O1 41159,C1(O)(C(C)NC(=O)CCOC2CC2)CCN(C(C2CC2c2nccn2C)=O)C1 41160,CN(CC1=NOC2C3CCC(C3)C12)NCc1ccc(OC(F)F)cc1OC(F)F 41161,c1(C(C(=O)NC(C)C(CO)NC(c2c[nH]c(C(N)=O)c2)=O)(C)F)ccccc1F 41162,N1(Cc2c3ccc(OC)cc3[nH]c2)CCC(N=c2[nH]cnc3cc(I)sc23)C1 41163,c1(C(=O)NC(C(=O)N(C(C2CCCC2)C)CC)C2CCCC2)ccccn1 41164,C(=O)(C1=CC2(CCOC2)C1)N1CC(CNC(CC=C)=O)OCC1 41165,c1(C(N2CC(F)(CN(C(C3(c4ccccc4)CC3)=O)C3CC3)C2)=O)ncccc1F 41166,C1(CNC(CC2(C)CC2(F)Cl)=O)CCC(CNC(C2(F)CCCCC2)=O)CC1 41167,c1(CC)cc(Cl)ccc1C(=O)NC1CC(O)(CNC(=O)C(C(C)C)[SH](=O)=O)C1 41168,C(c1ccc(OC)cc1OC(C)C)=CC(=O)N(CCNC(C(COC)OC)=O)C 41169,C(=O)(C(CC(C)C)SC(F)(F)F)N1CCC(C(C)NC(c2c(CC)occ2)=O)CC1 41170,Cc1cc(C(=O)NC2CN(C(=O)CC3CCCN3C)CC2F)c(O)nn1 41171,N1(C(C2N(CCC(C)C)CCC2)=O)CC2CC(O)C1C2NC(c1cccnc1)=O 41172,C1(OCC)CCC(C(N2CC(C(C)CC)C2)=O)CC1.C1(C)(C(=O)N)CC1C(=O)O 41173,C12(CNC(CCOCC)=O)CCC(C1)N(C(c1ccc(C(F)F)nc1O)=O)C2 41174,N1(C(C(C)NC(C)=O)=O)CC2OCCN(C(c3ccc(C(=O)N(C)C)cn3)=O)C2C1 41175,c1(CN2CCN(C(c3n(C)nc(C)c3F)=O)C(C(C)C)C2)ccc2c(c1)CCO2 41176,c1(CC#N)ccc(CN2CCCC2C(N2CCN(c3ccncn3)CC2)=O)cc1 41177,C1(C)(NC(C2CCC(CNC(CCCOC)=O)O2)=O)C=CCCC1 41178,N1(C(CC(=O)NCC)=O)CCC=C(CNC(=O)C(C)CC2CCC2)C1 41179,N1(C(CCC)=O)CC2CCCCN2CC1CNC(=O)CCc1cnoc1 41180,C1(C(=O)NCC(C)NC(c2nccnc2N)=O)COc2ccc(Cl)cc2C1 41181,C1(CNC(CN(C(C)=O)C)=O)CCC(C)(C)CN1C(C1CCOC1)=O 41182,C(C)(C(=O)NC1COCCN(C(=O)Cc2ccc(Cl)cc2)C1)(C(C)C)OC 41183,N1(C(c2cc(C)ncc2)=O)CCN(C(=O)CC2CC(=O)NC2=O)C(CS(C)(=O)=O)C1 41184,c1(NC2(CNC(=O)NCc3ccc[nH]3)CCC2)ncc2cc(Br)cnc2n1 41185,c1(C(=O)NCCCC(c2ccccc2)NC(C(CC=C)C)=O)c(F)cccc1F 41186,c1(N(C(=O)C(C)(C)OCC(F)F)C)ccc(S(C)(=O)=O)cc1 41187,N1(C(CC(C(C)C)NC(C2CCSCC2)=O)=O)CC2(C1)CC(C)(O)C2 41188,CC(CCC(=O)NCCc1cccnc1)NC(C1(C)CCCS1)=O 41189,N1(C(CN(C(=O)OCC)C)=O)CC(OC)CC(NC(=O)CC2CCC(C)CC2)C1 41190,C(=O)(CCCCCc1ccc(O)cc1)NCC1(F)CC(NC(C(C=C=C)C)=O)C1 41191,c1(C(=O)NCCC2(OC)CN(C(=O)COCCF)C2)ccc(F)c(C#N)c1 41192,C1(Cl)(C(N2CC(CNC(=O)COC3CCCC3)C2)=O)CC12CCOCC2 41193,CC(C(C)C(=O)N1CC=CC(NC(C23CCCCN2CCC3)=O)C1)S(C)(=O)=O 41194,O=C1Nc2ccc(C(N3CCCC3(C)CNC(=O)CC3CC(F)C3)=O)cc2CO1 41195,C(CCN=c1[nH]c(N2CCOCC3(CCC3)C2)nc2ccccc12)SC 41196,CN1CCN2CC1C(=O)N1CCC(CC1)C2=O.C(C)(C)(C)NC(C1CC1CF)=O 41197,c1(C(N(C)CC2(NC(=O)C(C)(O)C3CCOC3)CC2)=O)cnc(O)n(C)c1=O 41198,c1(C(=O)NCCC(CNC(c2nn(C)c(O)c2)=O)O)cc(F)c(C(=O)O)cc1N 41199,C1(CC(=O)NC(C(=O)NCC2(C=C)CCC2)Cc2cc[nH]n2)CCCNC1=O 41200,c1(C(N2CC3C(CNC(c4cn(CC)nn4)=O)(C3)C2)=O)ncc(F)cc1F 41201,N1(C(c2cnn(C)c2Cl)=O)CC2=C(C1)CN(C(=O)CP(C)(C)=O)C2 41202,C1(NC(c2c(C)nc(C)o2)=O)CCN(C(=O)Cc2cc[nH]n2)C12CCC2 41203,C1(CC)CC(NC(=O)CNC(=O)OC(C)(C)C)CN(C(=O)CC2(C)CCCO2)C1 41204,C1(NC(CC=C)=O)CC2CCCC(C1)N2C(C1CN(C2CCN(C(C)=O)C2)C1)=O 41205,N1(C(Cc2c(C)cc(OC)c(OC)c2)=O)CCN(C(=O)C(N)=O)CC(CO)C1 41206,Cc1cc(C(=O)NCC(CNC(C2(CC(C)C)CCC2)=O)S(C)(=O)=O)ccc1O 41207,c1(OC)cc(F)ccc1C(=O)NCC(CNC(c1nccnc1C(N)=O)=O)CO 41208,c1(C(N2CCC(NC(C(C=CC)O)=O)C2(C)C)=O)c(N)cc(F)cc1Cl 41209,C1(CC(=O)NCCCOCCNC(Cc2cn(CC)nn2)=O)CCCCC1F 41210,c1(C(N2CC(CC)C(OC)CC2)=O)ccc2cnn(CCOC)c2c1 41211,C(=O)(C1CC(=O)Nc2ncccc21)N1CCCC(c2cc(COC)on2)C1 41212,N1(C(Cc2c(C)cccn2)=O)CCOC(C)(CNC(C2CCC(F)(F)CC2)=O)C1 41213,N1(C(c2c(CC)c[nH]n2)=O)CCN(C(=O)C(C(C)O)N(C)C)C2(CC2)C1 41214,c1(OC)cccc(Br)c1C(=O)NC12CC1CN(C(=O)C(=O)NCC(F)F)C2 41215,CC1C(=O)CCCN1C(=O)CNCc1ccc(NS(C)(=O)=O)cc1 41216,C=C1CC(CC(=O)N(CC(C)(C)NC(=O)Cc2ccsn2)C)C1 41217,CC1=CCC(C(N2CCC(OCCNC(C3(C)SCCCS3)=O)CC2)=O)CC1 41218,Cc1cc(C(=O)NCC2CCCC2NC(=O)C=Cc2cc[nH]n2)c(F)cc1N 41219,c1(C(N(C(COCC)C)C)=O)ccc2c(c1)C(=O)CCN2C.C12(CC1)C(=O)N2 41220,c1(Cc2nccc(N3CCC(OC(C)C)C3C)n2)ccccc1I 41221,CCC(C)C(O)C(=O)N1CCCC1C1CCN(C(c2c[nH]c(=NC)s2)=O)CC1 41222,c12ccccc1OCC2.c1(CNC(=O)NC(C)CC#N)cccnc1 41223,c1(C(N2CCC(CNC(C(C)SCC)=O)C2)=O)[nH]c2c(c1C)C(=O)CC(C)(C)C2 41224,CC(C)CC(C(=O)NCCN(C)C(c1ccc(NCC(C)(C)C)cc1)=O)C(N)=O 41225,CCCC(C(=O)NCCC1(NC(=O)C(C)NC(=O)C(C)(C)C)CCCC1)OCC 41226,Cc1c(Cl)ccc(CC(=O)NC(C)(C)C(O)C(F)F)c1Cl 41227,N1(C(CC2C(C)OCC2)=O)CCC2CN(C(c3cccc(CC4CC4)n3)=O)C2C1 41228,CCCC(CN(C)C)OCC.n12cc(nn1)C(C1CC1)NC(=O)C2.C1CN1 41229,C(=O)(CC(F)(F)C(F)F)NC(CC#C)(C)C(=O)NCCN1CCCCC1 41230,C12(C(N)=O)CC(NC(C3(O)CCOC3)=O)(C1)C2.C1(=O)C=CC(=O)N1C1CC1 41231,C1(NC(CN(CCC)C)=O)CC2CC1CN(C(c1cc(C#N)cc(C)n1)=O)C2 41232,C1(CN2CCCC(NC(COc3cc(C)cc(C)c3)=O)C2)CC2(CCC2)C(=O)O1 41233,c1(C(C)C(N2CC=CC(NC(=O)CC(C)(C)C3CC3)C2)=O)cc(F)cc(F)c1 41234,C1(NC(=O)COc2cccc(C(F)(F)F)c2)CC2CCC1N(C(C1CC(O)C1)=O)C2 41235,C12(C(=O)NC(CCNC(C(C=C=C)C)=O)C)CC3CC(CC1C3)C2 41236,CC(CC(=O)NCc1ncccc1CNC(=O)C=CCOCC(F)(F)F)C(F)F 41237,C(=O)(CC(O)CNC(=O)C(CC)OCC)N1CC(CCC=C)C1 41238,CC1CC(C(N2CCC(C)C2CNC(c2ccon2)=O)=O)CCO1 41239,C1(C(=O)NCC2(C(=O)NCCCC3CCC3)CC(=C)C2)CCC(C)=C(C)C1 41240,C12(CNC(=O)CC3CNC(=O)C3)CC1CN(C(C13CC(C1)C(C(F)(F)F)O3)=O)C2 41241,N1(C(c2cc(C)nnc2)=O)CCN(C(=O)C(C)OCC2CC2)C(C(F)F)C1 41242,C=Cc1ccc(-c2csc(NC(c3cc(CC)no3)=O)c2)cc1 41243,C1(NC(CN(C)C(N)=O)=O)CCC(N(C)C(c2cnc(-c3cnn(C)c3)s2)=O)C1 41244,c1(CN(C(C)C(=O)NC2(CCNC(C3CS(=O)C3)=O)CC2)C)ccccc1 41245,S(=O)(=O)(c1ccc(N(C2CCCCCC2)C)c(F)c1)N(C)CC1CCCC1O 41246,C(=O)(C1=NOC2(CCCN(C(=O)C(O)Cc3cccc(Cl)c3)C2)C1)NCCOC 41247,Cc1cccc(NC(C2OCCC2NC(c2cnsc2C)=O)=O)c1C 41248,C(=O)(C1CCc2ccc(Cl)nc21)NCCC1CN(C(C(CCC)OC)=O)C1 41249,c1(CNC(C2C(=C)CC2)=O)cccc2c1CCN(C(C1(CC(=O)OC)CC1)=O)C2 41250,c1(OC)cc(Br)ccc1C(=O)N(CC(C)NC(c1cc(F)ccc1C)=O)C 41251,CCCCC(CNC(c1c(C2CCC2)noc1C)=O)NC(=O)C(C)OCC1CC1 41252,Cc1cc(=NCCC(=O)NOC)[nH]c(NC2CC=CCC2C(F)(F)F)n1 41253,c1(C(=O)NC2C(C)CN(C(=O)C(C3CC(F)(F)C3)O)C2)cc(N)cc(F)c1 41254,N1(C(C(C)C2CC(NC(C3(c4ccccc4)CC3)=O)C2)=O)CCCCC1CN(C)C 41255,C#Cc1ccc(F)c(C(=O)NCC2CC3COCC3N2C(=O)C(C)C)c1 41256,CCC(CCN(C)C(C1C=CCC1)=O)C(=O)OC 41257,C1(C(N2CCC(NC(CCc3nc(C)sc3)=O)C2C)=O)CCc2nc[nH]c2C1 41258,c1(NC(c2n(C(C(=O)OC)C)nnn2)C2CC=CC2)cccc(S(C)=O)c1 41259,N1(C(c2cc(C)c(F)nc2)=O)CCc2ccccc2C1CNC(c1ccsc1)=O 41260,C(=O)(C#CC1(C)CCCO1)NC(C)CCCNC(c1coc(C2CCCC2)n1)=O 41261,CC1(C)CCN(C(C2CCC(F)C2)=O)CC1CNC(c1cc(C2CC2)on1)=O 41262,c1(C(N(CC(C)O)CC)=O)c(CNC(=O)CN(C)C(C)=O)nnn1C 41263,c1(C(=O)NC(CC)(C)CNC(=O)COCC2CCOC2)ccc(CO)c(Cl)c1 41264,N1(C(C(C)(c2ccccc2)N(C)C)=O)CCC2(CCC(=O)NC2)C1 41265,Cc1ccc(F)c(C(N2CC(N(C)C(C3CC(C)(C)C3C(F)(F)F)=O)C2)=O)c1F 41266,C(=O)(C1=NCC2CCCCC12)N1C(CNC(c2scc(C)c2C)=O)CC(OC)C1 41267,C1(CC)CCN(C(=O)C(CC)NC(c2ccc(CC3CCCCC3)o2)=O)CC1 41268,C#CC1(NC2CCn3nccc3C2)CC2(CCCC2)C1 41269,c1(O)ccc(Cl)c(F)c1.C1(OC(C(=O)NC2(Cn3cc(C)nn3)CC2)F)CCCCC1 41270,Cc1ncc2n1CCNC2.C1(C2CC2)(C(=O)N)CC(=O)C1.C1(=O)CC2(CC2)N1 41271,C(=O)(CC(C)(C)CC(F)F)N1CCCCC(NC(c2c(C)cc(C)nc2O)=O)C1 41272,C1(C(=O)NCC2N(C(c3c(C)nc(C4CCC4)o3)=O)CCC2)CCN(C)S1(=O)=O 41273,N1(C(CC(=O)NCC)=O)CCCC(C2CC2NC(c2ccccc2O)=O)C1 41274,CN1CC=C(CC(=O)N2CCC(O)(CNC(C3Cc4ccncc4C3)=O)C2)CC1 41275,C12(C(=O)NC3C(OC)CN(C(=O)CCS(C)=O)C3)CCC(CO)(CC1)CC2 41276,N1(C(C2(CCOCC)CCCC2)=O)CCN(C(C2CCC23CCC3)=O)CC1C 41277,C(CCCCC(C)C)NC(CN(CCOC)C(C1CCCC(F)C1)=O)=O 41278,Cc1cc(C)c(C(=O)NC(C)CN2CCN(C(=O)C(F)(F)CC3CC3)CC2)o1 41279,C1(N(C(CC(C)(F)F)=O)C)CC2CCC(C1)N2C(C1(O)CCOC1(C)C)=O 41280,C1(NC(c2c(CNC(CCC3CC(C)C3)=O)ocn2)=O)CCC(C#N)CC1 41281,Cc1ccc(F)c(CC(N2CC(CNC(c3nncn3C)=O)C3(CC3)C2)=O)c1 41282,N1(C(C(N2CC(C)C2)C)=O)CCC(n2cc(CNC(=O)Cn3cnnn3)nn2)C1 41283,C1(NC(c2ccc(C(=O)O)cc2C2CC2)=O)CC2(CCOCC2)CCO1 41284,CC(N=[N+]=[N-])C(=O)NC(C(=O)NCCC1COCCOC1)C1CCCC1 41285,CCCCCCC(F)C(=O)NC(C)CN(C(c1nc2ncccn2n1)=O)CC 41286,C1(CC(=O)NCCC(C)N(C)C(c2csc(Br)c2)=O)COC(C)(C)C1 41287,CCC(CNC(c1cn(C)nc1OC)=O)(CC)NC(=O)C(C)C(=O)OC 41288,Cc1ncc(C(=O)NOC(CC(C)C)C(=O)NCCSC2CCOC2)c(=N)[nH]1 41289,C12(CNC(C=CC(=O)N(C)C)=O)CC1CN(C(=O)CCCCc1cnc[nH]1)C2 41290,c1(C(N2C(N(N3CCC=C(F)C3)C)CSC2)=O)cccc2cc[nH]c12.C=O 41291,C1(CNC(CC2(C=C)CC2)=O)CC(OC)CN1C(C1CCC(=O)N1)=O 41292,c1(NC(c2c(CCC)occ2)=O)cccc(NC(=O)C(C(=O)OC)OC)c1 41293,N1(C(C(CC#C)(C)C)=O)CC2CCC(CNC(=O)Cc3nc(C4CC4)cs3)(C2)C1 41294,C1(NC(CC(CN(C)C)O)=O)CN(C(=O)COCc2ccncc2)CC12CCC2 41295,CC1C(C(=O)N2CCC(C)(C)C2C(=O)Nc2cc(Cl)cnc2O)=NOC1C 41296,C1(C(=O)NC(CCCNC(C(CC)c2ccccc2)=O)C)CC12CCCCCC2 41297,C(=O)(CCCCC(N)=O)N(C(C)CNC(=O)Cc1csc(-c2ccccc2)n1)C 41298,c1cccc(C(C)NC(C(=O)NC(C)C)=O)c1.S(C)(=O)(=O)NC(C1CC1)C1CC1 41299,Cc1cc(N)c(Br)cc1C(N1CCC(C)C1CNC(=O)COC1(C)CCC1)=O 41300,C(=O)(CC(CCCC)NC(=O)CC(=O)OC)NC(CCC=C)C(=O)OC 41301,CC1(NC(=O)CCCNC(C2(C(F)(F)F)CC2)=O)CCCOC1 41302,N1(C(C=CC)=O)CCC(NC(c2cccn(C)c2=O)=O)C(c2ccccc2)CC1 41303,c1(CC)nc(C)c(C(=O)NCCC(NC(C2CCOC2(C)C)=O)OC)o1 41304,CCCCC(O)CCC(=O)NCC1CC(NC(C2(C)CCC(=O)NC2)=O)C1 41305,N1(CC)CCN(C(C23CC(CO)(CN2C(c2nc(O)sc2C)=O)C3)=O)C(C)C1 41306,N1(C(C=CCC)=O)CC(C)N(C(c2cc(CC(C)C)c[nH]2)=O)CC1C 41307,C1(CC(=O)NCc2ccccc2)CN(CC2COCCN2CCO)C2(CCC2)CO1 41308,N1(C(CC(C)C)=O)CCC2COC(CNC(=O)C(c3ccc(Cl)s3)=O)C2C1 41309,N1(C(COC(CC)C)=O)CCCC1C(=O)N(CC(C)CO)C 41310,C(=O)(C(O)CC(C)(C)C)NC1C(C)N(C(=O)CSCCN(C)C)CCC1 41311,N1(C(c2ccc(C(C)=O)s2)=O)CC2CC(NC(c3oncc3C)=O)CC1C2 41312,c1(CC)ccc(NC(=O)CCOCCCNC(=O)CCOC)c(C)n1 41313,C(=O)(C(C)(O)Cn1ccccc1=O)NC(CNC(c1ccc(OC)s1)=O)C(C)C 41314,C=C(Br)CC(C)(C)C(=O)N1CC(CNC(C2CC2c2noc(C)n2)=O)C1 41315,C1(O)(C(N(C)Cc2c(C)cccc2)=O)CCN(C(c2ccn(CCF)n2)=O)CC1 41316,C1(C(N(CC(CC)(C)NC(C)=O)C)=O)C=CCCN1C(C1CC1Cl)=O 41317,N(S(=O)(=O)N1CCOC(C(C)CC)C1)(CC#C)C(C)C 41318,n1(-c2n(C(C)CO)ccn2)cnc2c(N3CC4COCC4(CO)C3)ncnc12 41319,Cn1cc(S(N)(=O)=O)c(C(N2CC(NC(=O)CC3COCC4(CCC4)O3)C2)=O)n1 41320,c1(C(=O)NCC2COCCN2C(=O)C(O)C2CC2)nc[nH]c2nccc1-2 41321,C1(C(=O)O)COc2c(C(=O)NC(Cc3ccccc3Br)CO)cnn2C1 41322,C1(CN2C(C(=O)O)CC(CC)C2)CC2CC(=O)C1C2 41323,C1(C(=O)NCc2c(C)nns2)CSCCN1C(c1cn(C)nc1C)=O 41324,CC1CC(NC(=O)COc2ccccc2)CN1C(c1cc(F)c[nH]1)=O 41325,c1(C(N(C(CNC(c2cnc(C)n2C)=O)C)C)=O)cnc2ccc(F)cn12 41326,c1(Oc2c(NCc3c(Br)cc(C)c(C)n3)cccc2)cc(Cl)cc(Cl)c1[N+](=O)[O-] 41327,C(=O)(CCCCN(C)C(C)C)N(CCC(=O)NCCCCN1CCC1)C(C)C 41328,CC1=CCC(C(=O)NC2CC(C)(NC(=O)CC(C)(C)O)C2)CC1 41329,c1(CN(C(CC(C)C)=O)CCc2ccccn2)c(Br)cnn1CC(=O)O 41330,c12ccnc(c1)C(=O)NC2.C1(CNC(C2(OC)CCOC2)=O)CCOC(C)C1 41331,C(C)(CN=c1ccnc(NCc2nnc(O)n2C)[nH]1)(C1CC1)OC 41332,Cn1ccc(=NC(=O)C2CC(O)CN2C(c2ccc(C(F)(F)F)cc2)=O)[nH]1 41333,C1(C(=O)NCC(=O)NCC(C(=O)OC)CC2CC2)C2CCC(C2)C1C 41334,c1(OC)ccc(F)c(F)c1C(N1CCN(C(c2cc(C(N)=O)no2)=O)CC1C)=O 41335,C(=O)(CCCCC(N)=O)N1CCC(C(CC)OCC)CC1.c12cnc(nc1)NC2 41336,Cn1cc(C(=O)NCC(CO)NC(C2CCC3(CCCC3)C2)=O)c(=O)[nH]c1=O 41337,c1(C(=O)OCC2(C(=O)OC)COC2)nnc2n1CCCC2C(F)(F)F 41338,C(=O)(C(C)(O)COC)N1CC(C(N2CCC=C(Cl)C2)=O)(COC)C1 41339,CCCCC(O)CCC(=O)NCC(C)(CC)NC(C1CCCCN1N=O)=O 41340,C1(C)(NCC(CN(C(C)C)Cc2nccn2C)O)CC2CCC(C1)S2 41341,Cc1cc(C(F)(F)F)ccc1NC(c1cc(O)cs1)=O 41342,C(=O)(CC1=CCN(C)CC1)N1C(CNC(C2(C(=O)OCC)CCC2)=O)COCC1 41343,C1(C#N)(CC(=O)NCC2CN(C(c3ccn(CCC)n3)=O)C(C)C2)CCCCC1 41344,C1(NC(=O)C=CC=C(Cl)Cl)CC2C(NC(c3ccc(Br)s3)=O)C2C1 41345,C12(CNC(C3CC(OC)C3)=O)CC(CO1)N(C(c1cnn(C)c1C1CC1)=O)C2 41346,C1(CNC(=O)COC2CC2)COCCN1C(=O)CCCn1c(O)nnc1O 41347,CCCC(CCC)C(=O)N1CCC(C(C)C(=O)N(C)Cc2cccnn2)C1 41348,c1(NCCNC(c2c(Cl)cnc(CCC)n2)=O)cc(CN2CCCC2)nc(C)n1 41349,C1(O)(CN(C(=O)CC2(O)CCC2)C)CN(C(C2CC2(c2ccsc2)C)=O)C1 41350,C1(CC=C)(NC(=O)C(C)(F)F)CC2CCC(C1)N2c1ncc2sccc2n1 41351,C1(CC)(CNC(=O)C(CO)NC(N)=O)CN(C(c2ccc(C(C)=O)[nH]2)=O)C1 41352,c1(OC)cc(CNC(c2ccccn2)C)ccc1S(C)(=O)=O.C1C(=O)S1 41353,c1(SC)ccsc1C(=O)NCCN(C(=O)C(C)SC1CCOCC1)C 41354,c1(OCC(=O)NCCN(C(=O)C(CN(C)C)N(C)C)CCC)cccc(F)c1F 41355,C=CC1CCCCN1C(=O)C(C12CCC(CC1)C2)NC(=O)CC(C)(C)CN(C)C 41356,c1(CNC(C2CC3(CSC3)C2)=O)ccc(CNC(C2(C(=O)OC)CCCC2)=O)nc1 41357,c1(C(N2CCC(CNC(CC=C=C)=O)C(C)(C)C2)=O)cccc2c1CC(=O)N2C 41358,C12(NC(=O)CC3CC(=O)C3)CCCC1N(C(c1cnc(Cl)s1)=O)CCC2 41359,c1(C(=O)NC2CN(C(Cc3c(C)cco3)=O)C2)cnn(CC(F)F)c1C 41360,n1(CCOC)cc(C(=O)NCC2COC(CNC(c3nn[nH]c3Cl)=O)C2)c(C)n1 41361,S(=O)(=O)(c1c(Cl)ccc(C)c1F)NCC(COCC)O 41362,CC1(F)CC2(CN(C(C3(C)CCN(C(c4cc5n(n4)CCO5)=O)C3)=O)C2)C1 41363,C1(C(N(CCCCN(C(C(c2cccc(F)c2)C)=O)C)C)=O)CC(=O)CCO1 41364,CCC(CC(=O)NCC(CC)(CC)NC(c1ccc(CC(N)=O)cc1)=O)C1CC1 41365,CC1CC(NC(C2(CCOc3cccc(N)c3)CC(F)(F)C2)=O)CCO1 41366,C#CCC(C)C(=O)NCC(C)(C)CN(C(=O)C(c1ccc(C)o1)C)CC 41367,C1(CC(=O)NCC2ON=C(C)C2)CCC(NC(C2CS(=O)(=O)C2)=O)CC1 41368,CC(CCCc1ccccc1)C(=O)N1CC(NC(=O)CCn2cnnn2)C1 41369,c1(CC(=O)N(C2CCN(C(=O)C=C3CCN(C)C3)C2)CC)cccnc1.NCC 41370,CCC(C(=O)NC1CCN(C(c2oc(C)nc2C)=O)CC1O)C(F)(F)F 41371,CC1(C)CCN(CCNC(=O)C(c2ccoc2)NC(=O)CSC2CC2)C1 41372,c1(NC(C(C2CN(C(C)=O)C2)O)=O)cc2c(s1)CCC(C)(C)C2 41373,c1(CC)ccc(N)c(C(=O)NCCN(C(=O)C=Cc2cc(Br)cs2)C)c1 41374,Cc1ccc(F)c(N)c1C(=O)NCCC(N)=O.C12(F)CC(C1)NC(=O)C(=O)NC2 41375,C(=O)(C1=CCC2CCC1N2C(C1(C#N)CC2CC2C1)=O)N1CC(C=C)OCC1 41376,c1(CC)nnc2c(C(N3CCCC(CO)(NC(C4CC4F)=O)C3)=O)cccn12 41377,C(=O)(C(C)(C)C(C)O)NCC1(OC)CN(C(c2c(Cl)c(CC)nn2C)=O)C1 41378,c1(N2CCC(N(C(C(CCC)OC)=O)C)C2)ncnc(N(C)C)c1[N+](=O)[O-] 41379,C1(CC=C)(NC(=O)CN2CCOCC2=O)CCCN(C(=O)C(C)=CCC)C1 41380,N1(C(c2c[nH]nc2C2CC2)=O)Cc2ccccc2OC2(C1)CN(C(=O)CCF)C2 41381,C(=O)(CCCCNC(=O)NC)NCC(c1ccccc1)NC(C(C=C)O)=O 41382,c1(C(N2CC3N(C(C(C4CC4)SC)=O)CC(C3)C2)=O)cn2cccc(F)c2n1 41383,C12(NC(=O)CN3CCCC3=O)CCC(NC(C)=O)(CO1)C2.N12CC(C1)C2=O 41384,n1(CC)cc(NC(C2CN(C(=O)C(C)(CO)OC)CC23CC3)=O)ccc1=O 41385,N1(C(COC2CCCC(C)C2)=O)CC2CC(C1)C2NC(=O)Cn1nccn1 41386,c1(C(=O)NCC2CCC(CNC(C3CCC(C)(CC)O3)=O)CC2)ccc(C)c(O)c1 41387,CCC(C)C(O)C(=O)NC1CCCCC1NC(=O)CC(c1ccc(F)cc1)C 41388,N1(C(C2C(C)(C)C2CN=[N+]=[N-])=O)CCCCCC(NC(c2ccc(O)cc2)=O)C1 41389,N1(C(C(C)CO)=O)CCC2(CCN(C(=O)Cc3cc(C4CC4)nn3C)C2)C1 41390,c1(C(=O)NCC(O)CNC(=O)CC(=O)OC(C)(C)C)c(C(=O)NC)cnn1C 41391,CC12CC(CC(=O)NC3CCOC3Cc3ccc(F)cc3)(CO1)C2 41392,N1(C(c2c(Cl)ccc(OC)c2)=O)CC2CCC1C(CNC(C1CCOC1)=O)C2 41393,c1(C(N2CCC(N(C(C(CC)O)=O)CC)C2)=O)cc(F)c(Cl)c([N+](=O)[O-])c1 41394,c1(-c2cc(C(N(CCCNC(C(C)=C(C)C)=O)C(C)C)=O)no2)ccc(Cl)cc1 41395,CC1(CNC(=O)COC2CCOC2)CCCN(C(=O)CSC2CCCC2)C1 41396,c1(CC(N2C(C(N3CCCOCC3)=O)CC(=C)C2)=O)cccc(Cl)c1F 41397,CC1(CNC(c2ncn3c2CCC3)=O)CN(C(c2cccc(Cl)c2Cl)=O)CCO1 41398,C1CCCC(C)(O)CC1.Cc1nnc(C(CN)N(C)C)o1 41399,c1(C2C(C)C2)ccc(C(=O)NCC2(NC3CCC3)CCCCCC2)c(F)c1 41400,N1(C(C=C(C)c2cccs2)=O)CCCC1C1CCCN1C(=O)C(F)=CCCF 41401,c1(C(C(=O)NCCCSC)N(CCOCC=C)C)csc(Cl)c1 41402,C(c1ccc(C(N)=O)cc1)=CC(=O)NCC(C)N(C(C(C)OCC)=O)C 41403,C1(C(N(C)Cc2ccsc2)=O)CCN(C(=O)CCOC2CCC2)O1 41404,Cc1[nH]c(C)c(C(=O)NC2CC(F)CN(C(C3CC4C=CC3C4)=O)C2)c1C 41405,CN1CC(NC(c2occc2CNC(C2C3CCCC23)=O)=O)C(F)(F)C1 41406,C12(C(=O)OC3CCC(C)(C)CC3)C3C4C1C1C2C3C41C#N 41407,N(C(=NCCOc1ccc(Cl)cn1)NCC1N(CC)CC1)CC1CCC(=O)N1 41408,N1(C(CC2N(C(CCOC)=O)CCOC2)=O)CC2C(C1)C2(F)F 41409,C1(C(=O)NCc2ncc(C)[nH]2)CN(C(=O)OC(C)(C)C)CC(C)O1.C(C(=O)NC)O 41410,c1(C(=O)NC2C(CC)CN(C(c3cc(C(=O)OC)on3)=O)C2)nc(C)ccc1C 41411,C1(NC(=O)COc2cccnc2)CN(C(c2ccc(Cl)cc2)=O)CC1F 41412,C1(OC)(CNC(c2cncc(SC)c2)=O)CCN(C(C2(c3cccs3)CC2)=O)C1 41413,C1(C#N)(C(=O)NCCc2c(C(=O)NCC3(O)CCN(C)C3)c[nH]n2)CCOCC1 41414,c1(CC(N2CCC(CN(C)C(c3ccco3)=O)C2)=O)cc(Cl)ccc1Cl 41415,c1(C(N)=O)cc(CC(=O)NCC2(O)CN(C(C3(n4nccn4)CC3)=O)C2)on1 41416,c1(CC)c(C(=O)NC2COCC2NC(c2c[nH]nc2C(F)(F)F)=O)cccc1C 41417,CCCC(C)CC(=O)NCC1CCCN(C(c2cc(CC)ccc2C)=O)C1 41418,CCCC(C)C(=O)N1CCCC(N(C(=O)C(C)OCCN(C)C)CCO)C1 41419,c1(OC)ccc(C)c(OC)c1C(=O)N(CC(C)CNC(=O)CCOC)C 41420,C12(COC(C3CC(=O)NC3)=O)CCN(CC1)CC2 41421,C1(C(N(C2CSC2)C)=O)C(CNC(=O)CC2CC=CCC2)C1(C)C 41422,c1(CC)[nH]nc(C(=O)N(CCCN(C)C)CCNC(=O)C(O)CC2CC2)c1Cl 41423,C=CCC(C)C(=O)NC1CC(NC(c2sccc2CO)=O)C1 41424,N1(C(C(CC)N(C)C)=O)CCC2(C=C(C(=O)N3CCCN(C)CC3)C2)C1 41425,C12(C(=O)NCC(C)(C)NC(=O)CC3(C(F)(F)F)CC3)CC3CC1C2C3O 41426,C(=O)(C(CC(C)C)NC1(C(C)(C)O)CCC1)NCC(COC)O 41427,C1(C)(COC)CC(NC(=O)CCc2csnn2)CN1C(C1CCCC1)=O 41428,N1(C(COCC#C)=O)CC2CCC1CN2C(C1CCS(=O)(=O)CC1)=O 41429,c1(C(=O)NC2CC(F)(CNC(C3CCC(C)S3)=O)C2)ccc(-n2cncn2)c(N)c1 41430,N1(C(C(CC)=CC)=O)CCCC12CCN(C(C1CCN(C3CC3)C1=O)=O)C2 41431,CN1N=C(CC(=O)N2C3CCCC2CC(Nc2ncncc2I)C3)CC1=O 41432,N1(C(C2(CC)CC2(F)F)=O)CCC(CNC(=O)CC2(C)CCOC2)(OC)C1 41433,N1(Cc2cn(CCCOC)nn2)CCN(C(C2(OC(=N)O)CCC2)=O)CC1 41434,CCCCCCC(F)C(=O)Nc1c(C)cccc1C.C12CC3CC1CN3C(=O)C2 41435,C(CN=C(NCCc1ccco1)N(C)CCn1ncc(O)nc1=O)c1cnc(C)s1 41436,c1(OCC)c(-c2ccccc2)c(C)nn1C.C12CCCN(C1)C(=O)C(=O)N2C 41437,c1(NC(CCCNCC(C(C)C)OCCC)=O)c([N+](=O)[O-])c(C)nn1C(C)C 41438,CC1(C)CCCC(CC(N2CC(CNC(c3cncc(N)c3)=O)C2)=O)O1 41439,CC1CC(C(=O)NC2CCC(CNC(C3(C)CCCCCC3)=O)C2)CC(C)C1 41440,C(CO)(CC(C)(C)C)NC(C(CC=C)NC(c1ccc(F)cn1)=O)=O 41441,CC1CN(C(c2c[nH]c(=N)o2)=O)CC1CNC(c1cnn(C)c1CC(F)(F)F)=O 41442,c1(CCSCC=C)nc(-c2ccc(OC(C)C)cn2)nn1CCCO 41443,Cn1c(C(=O)NC2CN(C(=O)CCC3CCCCO3)CCC2F)cc(Cl)c1Cl 41444,N1(C(CC=C)=O)CCOCC(C(=O)NC(C2CC(F)(F)C2)CC)C1 41445,c12ccc(C(C)=O)c(c1)NC2=O.c1(CNC(=O)OCC)cccc(CO)c1 41446,CC(C)CC(O)C(C)C(=O)NC(CC1CC1)C(N1CCCC(C=C)C1)=O 41447,C1(C(N2CCN(CCCNC(=O)CCOCC(F)F)CC2)=O)C2CCCCCC12 41448,N1(C(Cc2nn(C)c(Cl)c2)=O)CCC2CN(C(=O)C(O)Cc3[nH]cnc3C)CC12 41449,Cn1ncnc1C(C(N1CCCC1CF)=O)NC(=O)NCc1ccccc1 41450,CC#CCC(C(=O)NCC#CC1CC1)NC(C1CN2CCC1CC2)=O 41451,N1(C(CCCCC)=O)CC2(C1)SCCC2NC(c1ccccc1OC)=O 41452,c1(SCc2ccccc2N2CCCCC2)nc(C(C)C)nc(=N)[nH]1 41453,c1(C(=O)NC(c2c(C(=O)NCCCC=CC)con2)C)cc(CC)oc1C 41454,N1(C(COCc2cc(C)no2)=O)CC(NC(c2ccc(=O)oc2)=O)C(O)C1 41455,C1(O)(CCNC(C2CC2c2cccs2)=O)CCN(C(c2nc(Cl)cs2)=O)C1 41456,C1(NC(C=COCC)=O)CS(=O)(=O)CC1NC(c1cnsc1)=O 41457,C1(C(=O)NC(C(=O)NCC)C)CCN(C(C2CC(=O)N(C)C2)=O)C1C 41458,C(CN=c1nc(-c2ccccc2C2CC2)[nH]s1)CNC(CN1CC(C)(OC)C1)=O 41459,C1(N(C(=O)COc2cn[nH]c2)C)CCCCN(C(=O)C=Cc2cccc(O)c2)C1 41460,c1(C(=O)OC)cccc(C(N2CCCC2CNC(=O)CCN2CCOCC2)=O)n1 41461,N1(C(C(CC(=C)C)OC)=O)CCC2CN(C(=O)C(N3C(=O)CCC3=O)C)C(C)C12 41462,CCC(C)(CNC(=O)CCc1ccccc1I)C(N)=O 41463,c1(C(=O)NC2CC(C)N(C(c3ccc(Cl)o3)=O)C2)cncc2sccc12 41464,C1(C(=O)NC2C=CC(CNC(=O)CCCC3CCCO3)C2)CC2C=CC1O2 41465,C(=O)(C(C(=O)NCC1CCN1C(c1cc(O)n(CC)n1)=O)C(C)C)OCC 41466,C(=O)(CC(C)C(=O)NCCC(C)NC(=O)CN1CCCCS1(=O)=O)OC 41467,Cn1c(C(N2C3CN(C(c4ccc(Br)s4)=O)CC23)=O)cc2ccccc12 41468,Cc1ccc2oc(C(=O)NC3C4CCN(C(C5(C)CCCOCC5)=O)C34)cc2n1 41469,c1(C(=O)NCc2nc(CNC(c3ccc(C)s3)=O)sc2)ccn2nncc2c1 41470,c1(CC(=O)NCC(CN(C(C(C)SC)=O)C)C)cncc(C)c1 41471,c1(CCCOC(C)C(=O)NCC(C2CCCCC2)=O)cn(C)c2ccccc12 41472,C1(F)(CNC(C2N(CCC)CCC2)=O)CCN(C(c2nc(O)c(C)s2)=O)C1 41473,CC(=O)CCCC(=O)NC1C2CN(C(c3cc(C)c(C)s3)=O)CC12 41474,C(=O)(C(F)(F)CCC=C)N1CCC(OCC#C)CC1.C1(=O)C(CCC2CCC2)N1 41475,CC(C(=O)Nc1ccc2nncn2n1)N1C(=O)COc2ccccc21 41476,CC(C)(C)CC(O)C(=O)N(CCC(N1CCCCCC1)=O)CCO 41477,c1(C(=O)NCC(CNC(C(C)OC)=O)C)cn(-c2ccc(F)cc2)nc1C 41478,CCC(CC(=O)N(CCC(C)NC(=O)COC1(C(F)(F)F)COC1)C)OC 41479,c1(CCC(=O)NCC2N(C(C3(CC)CC3)=O)CCCC2)n[nH]c2ccccc12 41480,C1(C)(C(=O)NC(C(=O)N(CCC(O)CO)C)CCN(C)C)CCC(=O)NC1 41481,N1(C(C(C)OCCOCC)=O)CC(NC(c2sccc2F)=O)C2CCCCC12 41482,C1(C(C)C)(C(=O)NC2CSC(C)C2)CCN(C(=O)C=CC2CCCCC2)C1 41483,C(=O)(CC(C)(F)F)N(CC(C)O)CCNC(C1C(C)C1C)=O 41484,C=CCCCC(C(=O)N1CCC(c2cnco2)C1)NC(c1cn(C)cn1)=O 41485,N1(C(CCc2[nH]c(=N)sc2)=O)CCC2(NC(c3ncccc3Cl)=O)CCCC12 41486,c1(NC(C(CC=CC)NC(=O)Cc2nc(=N)[nH][nH]2)=O)cc(C)ccc1CC 41487,c1(CC)cccc2c1CNC(NC(c1csc(CSC3CCCO3)n1)=O)C2 41488,CCC(C)CCNC(C1CCN1C(=O)COCC(=O)NC)=O 41489,C1(O)(C(C)NC(CN(C2CC2)CC)=O)CCN(C(c2cc(C)n(C(C)C)n2)=O)C1 41490,n1(CC(=O)NC2CCCC(NC(Cc3c(C)nc[nH]3)=O)C2)cc2ccccc2n1 41491,C(=O)(C(F)CC(C)C)NCC(CC)NC(c1ccc(-c2ccccc2F)n1C)=O 41492,C1(C(=O)NCC(CNC(CN(c2ccccc2)CC)=O)C)CCCN(CC(F)F)C1 41493,N1(C(c2c(Br)c(C)n(C)n2)=O)C2CCC1CN(C(c1c(C#N)ncn1C)=O)C2 41494,Cc1nn(C)c(Cl)c1CN1CCOCC(CNC(=O)COCCC(C)C)C1 41495,CCC(C(=O)N1CCC(OCCNC(c2csc(CO)n2)=O)C1)C(C)(C)CC 41496,c1(C(=O)NC(CC)CNC(c2ncccc2Cl)=O)cc(Cl)sc1S(N)(=O)=O 41497,c1(C(=O)NCCN(C(C(CC)(CC)OC)=O)C(C)C)nccc2nn[nH]c12 41498,Cc1nc(CNC(=O)NC2CCN(c3ccnc(C)n3)CC2)sc1C 41499,CCN=C(NCc1ccc(-n2ccnn2)cc1)NCC1(COC)CCOCC1 41500,CC(O)(C(=O)NCc1n[nH]cc1C(=O)NC12CC(C1)C2)C1CCCC1 41501,C1(NC(Cc2c(OC)cccc2)=O)CCSC12CN(C(C1CCCOC1)=O)C2 41502,C1(OCC)COCCC1C(=O)NCC(=C1CN(C(C2(N(C)C)CCC2)=O)C1)F 41503,CCCCC(COC)N=c1[nH]c(=NCC(N)CC)[nH]c2cc(C)ccc12 41504,CC(C)CC(CNC(C1COC(=O)O1)=O)NC(=O)CN1CCSCC1 41505,C12(CNC(C=CCN(C)C)=O)CCC1CN(C(C1CC(O)CN1C)=O)C2 41506,CS(=O)(=O)C1CCCN(C(c2nc(O)nc(O)c2F)=O)C1 41507,N1(C(C(C)OCC)=O)CCCC(O)(CNC(c2c(Cl)c(C)nn2C)=O)C1 41508,Cc1c[nH]cc(C(=O)NC2CC(F)(CNC(c3cnnn3C)=O)C2)c1=O 41509,c1(N2CCC(NC(Cc3c(C)nccc3)=O)C(F)C2)ncccc1[N+](=O)[O-] 41510,C(=O)(C(C)(C)C(N)=O)NCCOCCCN(C(=O)C(C)(C)N1CCCCC1)C 41511,N1(C(C=C(CC)CC)=O)CCC(O)(CN(C(=O)Cc2cnn(C)c2)C)C1 41512,c1(C(N2CCC(C(=O)Nc3c(C)cccc3F)C2)=O)ccc(O)c(C#N)c1 41513,c1(C(=O)NC2COC3(C2)CN(C(=O)COC2CCCC2)C3)cc2cc(F)ccc2s1 41514,CC1(C(=O)NC(CCO)c2ccco2)CCCN1C(c1ccsc1)=O 41515,CC1CCCC=C1C(=O)N(C(C)CNC(c1cc2ncccc2[nH]1)=O)C 41516,C(=O)(CCCC(C)(F)F)NC(C1OCCN(C(c2c(C)csc2)=O)C1)C 41517,C1(NC(C(CC2CC2)NC(C2CC2Cl)=O)=O)CC2CCCC2C1 41518,N1(C(CN(C(C)C)C)=O)CCOC2CN(C(c3ccsc3C(F)F)=O)CC12 41519,C1(CC(=O)NCc2cc(C)[nH]c2)COCCN1C(C1(C(=O)O)CC1)=O 41520,Cc1ncc2n1CC(C(=O)N(C)CCN(C)C(C1CC3(CCCC3)CO1)=O)CC2 41521,N1(C(C(C)OCCC=C)=O)CC(C)(C)CC1CNC(=O)C(C)(C)C1CC1 41522,N1(C(=O)NCc2snc(C)n2)CCC2(CC1)CC(C)NC2=O 41523,N1(C(C2(N(C(CSCC#C)=O)C)CC2)=O)CC(O)(CO)C1 41524,N1(C(C)=O)CCCC(CN2CCCC(CCC(=O)NCCc3ccccn3)C2)C1 41525,N1(C(C(CC)SC)=O)C2CCC1CN(C(=O)C(C)Sc1ccccn1)C2 41526,CC(C)CCC(C)NC(C1(NC(=O)Cn2cc(C3CC3)nn2)CCCCC1)=O 41527,C1(CC(N2CC3C(CC)(C3)C2)=O)CN(C(C2CN(C3CCC3)C2)=O)CCC1C 41528,C1(CNC(CCNC(C(C=C)O)=O)=O)CCN(C(=O)CC2CCCCO2)C12CC2 41529,C(=O)(C(C)(CC(C)C)NC(c1cc(C(C)C)c(N)cc1F)=O)OC 41530,N1(C(C)C(N)=O)CCC(C2CCCN(C(c3cnc(C4CCC4)o3)=O)C2)C1 41531,c1(C(N2C(C(=O)NC3CC3CCF)COCC2)=O)ccc(F)cc1 41532,c1(C(N2CC3C(CNC(c4cnc(CCC)s4)=O)C3C2)=O)cc2nc[nH]c2cn1 41533,C1(C(=O)NCC2(C(=O)O)C(C=C)C2)OC(c2ccccc2)CC1C 41534,C1(CC)CN(C(C2COCCOC2)=O)CCN1C(C12CCCC1(C(N)=O)C2)=O 41535,c1(C(=O)NC(CN(C(C(CCCC)N(C)C)=O)C)C)oc2ccccc2c1CO 41536,c1(CC(=O)NCCC(=C)CNC(=O)C(O)C(C)(C)C)ccc(Cl)c(OC)c1 41537,C1(C(=O)NC2CC(C)(NC(Cc3ccc(C)nc3)=O)C2)CCCCNC1=O 41538,c1(C(=O)NC2(CN(C(C(CC)CC3CCCC3)=O)C)CC2)cc2cccnn2n1 41539,N1(C(c2nc(C(C)=O)sc2)=O)CCN(C(C2(c3ccc(Cl)cc3)CC2)=O)CC1C 41540,N1(C(CC(C)F)=O)CC2CCOC2(CNC(c2cc(=O)cc(Cl)[nH]2)=O)C1 41541,C1(NC(c2cc3occc3s2)=O)CC2CN(C(C3CCCCC3)=O)CC2C1 41542,c1(C2CCN(C(c3c(C(C)(C)C)c[nH]c3)=O)C2)ccc(C(F)(F)F)cc1 41543,CN1CCC(F)(C(=O)NCCCCCCNC(c2cccc(O)n2)=O)CC1 41544,CCC(C)(CNC(C1(F)CCN(C(c2ccc(CO)cn2)=O)C1)=O)C(N)=O 41545,C(=O)(C(C)C(CC)CC)N1CCCC(NC(CN(C2CC2)CC)=O)C1C(C)C 41546,c1(C(C)(C)C(N)=O)ccc(NC(C2CC2c2cncc(Br)c2)=O)cc1 41547,C(=O)(C1=CC(O)C(NC(=O)C=C(C2CC2)C2CC2)C1)Nc1cc(C)sc1 41548,C(=O)(CC(F)(F)CS(C)(=O)=O)NC1CC(F)(CNC(c2c(C)ncc(Cl)c2)=O)C1 41549,C(CCC(=O)NCc1nocc1C(=O)N(C1CCOC1)CCO)N(C(C)C)C 41550,c1(OC)ccnc(C(C(=O)NC2(C)CC2)N(C2CCCCC2C)C)c1C 41551,N1(C(C2N(CCC)CCC2)=O)CCC(CC(=O)NC(CC2CC2)C(=O)NC)C1(C)C 41552,c1(OC)cc(O)ccc1CC(C(=O)OC(C)(C)C)Nc1nccnc1C(=O)O 41553,C1(C(N(C2CCCN(C(c3sc(C)nc3C)=O)C2)CC)=O)CC2(CCC2)CO1 41554,Cc1cccc(C(CNC(=O)C(C)c2cccs2)NC(C2CC=CC2)=O)c1 41555,c1(C(N2CC(C(=O)NC3(C(C)(F)F)CC3)(CF)C2)=O)ccncc1N=[N+]=[N-] 41556,c1(C(C)C)nc2ccc(F)cn2c1C(=O)Nc1ncn(Cc2cnc[nH]2)n1 41557,C1(C(=O)NCC(C)(C2CCC2)NC(C2C=CCS2)=O)CCn2nccc2C1 41558,C1(C(=O)NC(CC2CCC2)CO)CCN1C(C1CCO1)=O 41559,C1(CNC(C2C(C(=O)OC)C2)=O)CCCC(CNC(c2nc(N(C)C)no2)=O)C1 41560,C(=O)(CCCC(=O)NC1(CCNC(C2CCN(CC)C2)=O)CCC1)OCC 41561,C1(NC(C2(CC#C)CCC2)=O)CCCC(NC(c2cc(C)n(C)c2)=O)C1 41562,Cc1nc2cc(C(=O)NCC3CC(NC(=O)C(=O)N=S(C)(C)=O)C3)ccc2n1C 41563,c1(C(=O)NC2(CF)CCN(C(CCCCCN(C)C)=O)C2)ccc(F)c(F)c1F 41564,C1(C(C)C)CCC(C(=O)NC(C)CCN(C)C(C23COCC(C2)C3)=O)CC1 41565,C1(C(=O)N(C(C)C(=O)OCCO)C)CN(Cc2cc(Br)c(Br)o2)CCS1 41566,c1(OCC=C)ccc([N+](=O)[O-])c(C(=O)NC2CC2NC(=O)C#CC(C)(C)O)c1 41567,Cc1nn(CCCNC(N2CCC(n3ccnc3)C2)=O)c(=O)c(C#N)c1C 41568,C1(N(C(C(C(C)C)NC(Cc2cn(CC)nc2)=O)=O)C)CCOC(C)(C)C1 41569,C1(C(N2CC(CNC(CC(C)F)=O)C2)=O)CC(C2CC2)=NO1 41570,C(C(=O)NC12CC(NC(c3csc(Cl)c3)=O)(C1)C2)(C(C)(C)C)NC(C)=O 41571,c1(C(=O)NCC2C(C)CCN2C(=O)C(F)=CCCF)cnn2c1OCC2 41572,CCC(CC)CC(=O)NCC1CCN(Cc2ccc(OC)nc2Cl)C1 41573,N1(C(C(CC)C)=O)CCCC(OC(C2N(C(c3ccccc3)=O)CCC2)=O)C1 41574,N1(C(CN(C(=O)CC2CCCC2C)C(C)C)=O)Cc2ncsc2C1 41575,C=CCCCCCC(=O)NCC1CCCCN1C(=O)Cc1ccc(C(F)F)cc1 41576,C1(C(=O)NCCC(C)N(CCC)C)COCCN(C(=O)OC(C)(C)C)C1 41577,N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CC2C(NC(c3ccc(C#N)o3)=O)C2C1 41578,n1(CCNC(CC)=O)nccc1C(=O)N(CCNC(=O)C(C)=C(C)C)CC 41579,c1(CC(=O)NC(CC=C)CNC(c2ccc(Cl)cn2)=O)cccc([N+](=O)[O-])c1C 41580,CC1(C)Cc2occc2CN1C(c1ccc(Cl)cc1I)C(=O)NC1CCOC1 41581,c1(CC(=O)NCC2C(NC(C3C(C(C)=O)C3(C)C)=O)C2)ccc(S(N)(=O)=O)cc1 41582,C1(C(=O)NC(C(C(C)C)NC(CN(C2CC2)CC)=O)C)CC2(C1)CC21CCC1 41583,c1(CCC(=O)NCC2(O)CCN(C(CCOC(C)=O)=O)C2)c(F)ccc(Cl)c1F 41584,C1(C(=O)OC)CCCC(C(=O)OC)CC1.c12cn(nn1)CCN(C(C)(C)C)C2 41585,C(CC(O)CNC(=O)CNC(=O)CN(C)C(C)C)OC 41586,C(=O)(C(C)N(OC)C(=O)C=CCNC(C(=O)OC)C)N(C)C(=O)C1CC1 41587,N1(C(CCn2c(C)cc(C)n2)=O)CC(C)(C)CC1CNC(c1cc(Cl)ns1)=O 41588,N1(C(c2ccc(CO)s2)=O)CCC(O)(CC(C)C)C1.C=CCC1CNC(=O)C(=O)N1 41589,c1(CC(CC)SCCC2CC2)cc(-c2ccccc2)n[nH]1 41590,C(=O)(CS(=O)(=O)CCC(F)(F)F)N1C(C(C)NC(c2c(C)occ2)=O)CCCC1 41591,Cc1nc(C)c(C(N2CSCC2C(=O)NC(C2CCC2)C)=O)o1 41592,C1(c2cccs2)(C(N2C(CNC(c3c(CC)nn[nH]3)=O)CCC2)=O)CCOCC1 41593,Cc1ncncc1C(=O)NC1CCCC1CNC(=O)C(C1CC(F)(F)C1)O 41594,C1(C(CC(=O)O)c2ccccc2)CCCN(C(C2CC2(F)F)=O)C1 41595,C#Cc1ccc(C(=O)NCC2(NC(C3CN4CCC3CC4)=O)CC2)c(F)c1 41596,C(=O)(C(CCc1cccc(F)c1)N1CC2CCC2C1)NCCCSC 41597,N1(C(C2(NC(C=Cc3ccc(C)o3)=O)CC(F)C2)=O)CC(C)OC2(CCC2)C1 41598,N1(C(c2c(CNC(C=C3CCC(C)CC3)=O)ocn2)=O)CC(C)C(O)C(C)C1 41599,CC1(NC(=O)CSC2CCOC2=O)CCN(C(=O)CSCC(F)(F)F)CC1 41600,CC1CC(CO)CN(C(=O)C(CO)NC(c2ncccc2Cl)=O)C1 41601,C(=O)(C(C)CC(N)=O)N1CCC(CCN(C(CCCCC)=O)CC(C)C)CC1 41602,CCN=c1ccc(C(c2c(Cl)ccc(C(=O)OCC)c2)N2CCOCC2)c[nH]1 41603,c1(NC(=O)NC(C)CC(C)(C)O)ccc2cnccc2c1 41604,CC1CN(C)CCN1C(=O)C(Cc1cnc[nH]1)NC(c1cncs1)=O 41605,c1(C(N(CC(=O)NCCC(C)OCCC)CCC)=O)coc(CSC)c1 41606,Cc1nn(C)c2ccc(C(=O)NCC3CN(C(=O)Cc4ccco4)CC3O)cc12 41607,c1(C(N(CCCCN(C(C(CC)O)=O)C)C)=O)c(C)sc(C)c1C#N 41608,c1(C(N(CCCNC(C(c2cccnc2)OC)=O)C2CC2)=O)cnn2ccccc12 41609,c1(C(N(CCCCNC(c2ccc(C(N)=O)cc2)=O)C)=O)cccc2c1NCC2 41610,N1(C(c2ccc(CCC)cc2)=O)CC(C)(C)OC2(C1)CN(C(C1(O)CCC1)=O)C2 41611,Cc1cncc(CC(=O)NCCC2CCCN2C(C2COCCO2)=O)c1 41612,N1(C(C(C)NC(CC)(C)C)=O)CC2(NC(c3ncncc3C)=O)CC1C2 41613,CC(C)CC(CNC(C1Cc2nccn2C1)=O)C(=O)NCCC(C)C(F)F 41614,C(=O)(C(CNC(=O)Cc1ccccc1F)(CC)CC)NCCCC 41615,CCC(C)C(C)CNC(=O)CC1CCC(NC(c2cc(C)nn2C2CC2)=O)CC1 41616,C(=O)(C#CC1CC1)NCC#CCNC(c1nc(CS(C)(=O)=O)oc1)=O 41617,C1(NC(CCc2ccn(C)c2)=O)CC12CC(NC(C1CC1C(F)(F)F)=O)C2 41618,N1(C(C=C(C)C(C)C)=O)CCC(C)C1CNC(c1cn(CC(F)(F)F)nn1)=O 41619,C1(NC(C2C(C(C)C)C2)=O)CN(C(=O)C(F)(F)OC(C)=O)CC1O.c1ccccc1 41620,C1(CCNC(CC=C=C)=O)CC(OC(C)=O)CN1C(C1CCCSC1)=O 41621,c1(OC)cccc2c(C(=O)NCC(O)CCNC(=O)C=C(C)C(C)(C)C)c[nH]c12 41622,c1(C(=O)OC)cc(CNC(C2CCN2C(C)=O)=O)no1.n12cc(nn1)CNC2 41623,C1(NC(c2c(CC)nccn2)=O)CN(C(C2C(C)C2C)=O)CC1N=[N+]=[N-] 41624,N1(C(c2cc(C)ns2)=O)CCCC(NC(C2(O)CC(C)(C)C2)=O)C1C 41625,C(=O)(C(F)(F)C(F)F)N1C(CN(C(C(c2ccc(C)cc2)(F)F)=O)C)CCCC1 41626,c1(OC(C(=O)NCCC(C)N(C(=O)CSC2C(C(=O)OC)C2)C)C)ccccc1 41627,c1(C(=O)NCCCC(C)NC(=O)C2=NNC(=O)C2)cc2cc(Cl)cnc2o1 41628,N1(C(c2c(C)nc[nH]2)=O)CCC2(CC1)CCN(C(c1cnco1)=O)C2 41629,C1(C(=O)NCc2nn[nH]n2)(CO)CC2C=CC1C2.C12CCN(CC1)C(=O)N2 41630,CC1OC2(CNC(C3CC3F)=O)CC1(NC(c1nccc(F)c1Cl)=O)C2 41631,N1(C(COCC=C)=O)CC2CN(Cc3ccc(CC(=O)O)c(I)n3)CC2C1 41632,N1(C(C(CC)NC(N)=O)=O)CC(CNC(C2CC(F)(F)C2)=O)C2CCCCC12 41633,C1(NC(CC2C(C)OC(C)C2)=O)CCC2CN(C(C3CCCC(=O)N3)=O)CC2C1 41634,CC1=NOC(CNC(c2csc(C)c2)=O)C1.C12(CC(O)C1)C(=O)N2 41635,Cc1csc(C(N2CCCC2CNC(c2ocnc2C2CCC2)=O)=O)c1 41636,c1(C(N2CCN(S(C)(=O)=O)CC2)C(=O)NC(CC)(C)C)noc2c(Cl)cccc12 41637,C(CN=c1[nH]c(=NCc2cccc(C(F)F)c2)[nH]c2c1COCC2)C(=O)CCF.N 41638,C(=O)(C(C#N)(CC)CC)NCCC1(OC)CN(C(C2CC(C(C)C)=NO2)=O)C1 41639,C1(NC(C=CC(C)NC(=O)C(C)C2CCCC2)=O)CC(N(C)CCO)C1 41640,CC1CCCC(C)CN1C(=O)Nc1ccccc1C(N)=O 41641,C(=O)(C#CC1CCOC1)N1CC(CNC(CCc2cc(C)cc(C)c2)=O)C1 41642,C1(CC(=O)NCC=C(Cl)Cl)CC(F)CN1C(=O)C=CC1CCCC1 41643,Cc1ccc2occ(C(N3CCC(NC(=O)C4=CC5CC=CCC45)CC3)=O)c2c1 41644,Cc1nc(C)c(C(=O)N(C2CCN(C(c3cc(-c4ccccc4)cs3)=O)C2)C)s1 41645,C(=O)(C(C(C)(C)C)C1CCCC1)NCC.C(=O)(C(C)S(C)(=O)=O)N(CCCCCC)C 41646,N1(C(C(c2cnn(C)c2)OC)=O)CCCC(O)(CCNC(=O)CC(F)(F)Cl)C1 41647,O=C(N=c1[nH]oc2cccnc12)C1CCN(Cc2cnc(Cl)c(Cl)c2)CC1O 41648,Cc1c(Cl)ccnc1C(N1CCCCC1CNC(C1(S(N)(=O)=O)CC1)=O)=O 41649,N1(C(C=CCC)=O)CCCC(N(C)C(C2(c3ccc(F)cc3)CCC2)=O)C1 41650,C1(N(CCCCC)CCC(=O)NC)CCN(C(=O)C(F)C(C)C)CC1 41651,Cc1cccnc1CCNC(C1CCCN1C(C1CCCCC1C)=O)=O 41652,C1(NC(c2cccc(OC)c2)=O)CS(=O)(=O)C2CN(C(C3CC3C(F)F)=O)CC12 41653,c1(C(=O)NCCC(C)NC(=O)CCC2CC2(Cl)Cl)cc2c([N+](=O)[O-])cccc2s1 41654,C1(C(=O)OCC)CCCN(C(=O)COC2CCN(C(=O)COC)C2)C1 41655,C(=O)(CCCCC(=O)c1ccc(C)cc1)NC1(C)CCCN(C(C(C)OC)=O)C1 41656,C#CC1CCCCN1C(C1CN(C(=O)CCC(=O)N(C)C(C)C)CC1CC)=O 41657,c1(CNC(C(=O)NCCN(C2CCCC2)C)=O)ccnn1CC(F)F 41658,CCCCCCCC(=O)NC(CCCOC)C(=O)NCc1cn(CC)cn1 41659,CCCCC(C)CCC(=O)N1C(C(=O)NOCCOCCOC)CCC1C1CC1 41660,c1(C2C(C(N(CCCCNC(C(C)OCC=C)=O)CC)=O)C2)cnn(CCO)c1 41661,N1(C(C=CC=CCC)=O)CC2CC(C(N3CCSCC3C3CC3)=O)CC2C1 41662,C1(CNC(N(c2ccc(F)c(Br)c2)CC)=O)CCC2(CC1)NC(=O)N(C)C2=O 41663,c1(SC)ccc(C(=O)NC2CC(N(C(=O)Cn3cc(C4CCC4)nn3)C)C2)o1 41664,c1(C(=O)NC(C2CCCN(C(=O)CC(F)F)C2)C)ccc(F)c(C2(C)CC2)c1 41665,C(c1ccc(Cl)s1)=CC(N1CCC(CC2CCN(C(CSCC)=O)CC2)CC1)=O 41666,N1(C(=O)NCCn2c(C(=O)OC)ccn2)CC2CC(O)C(O)CC2C1 41667,N1(C(CC(C)n2ccnc2)=O)CCC(C)(NC(C2CCC=CO2)=O)CC1 41668,CC(F)(F)C(C)(C)C(=O)N1CC(C(N2CCCC(CO)C2)=O)C(C2CC2)C1 41669,c1(C(C)(C)OC)ccc(C(=O)NC2CC(C)(CNC(=O)CSC(F)(F)F)C2)cc1 41670,N1(C(CC(c2ccc(O)cc2)C)=O)CCC2(CC1)CN(C(c1ccns1)=O)C2 41671,C(=O)(C(C)COC)NC(CC)(C)C.C(C=O)=C=CCC(C)(C)C 41672,N1(C(CSc2cc(C)c(Br)cc2C)=O)CCN(S(N)(=O)=O)CC12CCCCC2 41673,N1(C(CC2(NC(Cn3nnc(C)n3)=O)CC2)=O)CCOC(C)C1 41674,C12CCCCCCN1C2=O.C1(CCCNC(=O)C(N2CC=CCC2)=O)CCCOC1 41675,c1(C(=O)NCCCCCCNC(c2ccc(O)cn2)=O)ncnc(O)c1Cl 41676,C#CCC(C)(C)C(=O)NCc1cc(C(=O)NC2CCCC2CN(C)C)cs1 41677,C1(C(=O)OC)CCC(CN(C(CC2CCCC2)C(=O)NCCC(N)=O)C)O1 41678,N1(C(COCCNC(CCCCOCC)=O)=O)CC(C(F)(F)F)OC(CC)C1 41679,c1(Cc2nc(-c3sc(C)c(Br)c3)on2)nsc2cc(Br)ccc12 41680,C12(C(=O)NC(c3ncccn3)C)CCC1CN(C(C1CCNC(=O)C1)=O)C2 41681,Cc1cccc(C(C)C(=O)N2CC(NC(=O)C=CCOCC(F)(F)F)C2)c1 41682,c1(C(=O)NCCC(=C)CNC(c2ccc(C3CC3)nc2C)=O)ccnc(C)c1O 41683,N1(C(C=CCN(C)CC)=O)CC2CC(NC(=O)CC(C)(C)C3CC3)C1C2 41684,c1(C(N2CCCN(CCNC(C(CC)C#N)=O)CC2)=O)cccc2c1CCCN2 41685,CC1CN(C(c2ccc(CO)s2)=O)CC1(C)C(=O)NC1CCN(C)C1=O 41686,Cc1scc(C(=O)NCC(O)CNC(c2csc(CC(F)F)n2)=O)c1C 41687,C1(C(=O)NCCN(C(=O)C=NOC)CC)CC12CCC(C)(C)CC2 41688,CC1(C(F)(F)F)CCN(Cc2cn(C3CC4(C(N5CCCC5)=O)C3C4)nn2)CCO1 41689,N1(C(C(COCC)C)=O)CCC(CNC(=O)Cc2n[nH]c(=N)s2)(COC)CC1 41690,C(=O)(CCCCC(N)=O)N1CCC(Cc2cn(CC(=O)OC(C)(C)C)nn2)C1 41691,CCCC(CC)C(C(=O)NCC(=O)OCC)N(C1CCN(C)C(=O)C1)C 41692,N1(C(CCC(C)N(C)C)=O)CCC2(C=C(C(=O)NC(CCO)c3ccco3)C2)C1 41693,C#Cc1cnc(C(=O)NCCCCCCNC(c2ccccc2CC)=O)c(C)c1 41694,N1(C(C2C=CCN(C(c3ccc(F)c(F)c3)=O)C2)=O)CC2C3CCC(C3)C12 41695,C1(C(=O)OCC)(CNC(=O)COC(=O)N)CC(O)C1.C1(COC)CCOC1 41696,N1(C(C(C(C)C)C)=O)CC2CN(C(=O)C(C)SC(F)(F)F)CC(C1)O2 41697,Cc1cc(C(N2CCCC(NC(=O)C(C)(C)NS(C)(=O)=O)CC2)=O)c(F)cc1F 41698,CCC(C)CC(=O)C(=O)NC(CC(=O)N(C)CC1CC1(F)F)C(C)C 41699,N1(C(c2c(SC)csc2)=O)CCOC(C)(CNC(c2cc3sccc3s2)=O)C1 41700,C(CCCC(C)(C)C)NC(=NC)NCC1CCCCO1 41701,Cc1cnnc(O)c1C(=O)NCc1nc(CNC(c2conc2C)=O)cs1 41702,Nc1cc(C(=O)NCC2CCN(C(C34CCCN3CCC4)=O)CC2)cc(O)c1Cl 41703,C1(NC(c2c(Cl)cn(CCC)n2)=O)CCN(C(=O)CC(F)(F)Cl)CC1C 41704,c1(C(C)(C)C(=O)NCC2(O)CN(C(=O)CC3CC3(C)C)C2)ccc(O)cc1 41705,Cc1cc(-n2nc(C3CCC3)nc2CC2CCOC(C)C2)cc(Br)c1 41706,c1(C(C(=O)NC(CNC(c2c(CC)con2)=O)C)(C)C)ccc(F)cc1F 41707,c1(CN2C(C(N3C(C)CCC3CO)=O)CC3CC32)cc(F)c(Cl)c(F)c1 41708,CC(C)CC(O)C(=O)NC1CC2CCC1(NC(=O)CSCCC(F)(F)F)C2 41709,C1(NC(COC2(C)CCC2)=O)CCCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1 41710,C1(C(=O)NCC2C(C)CC2)CCN(C(C2CCCCS2)=O)C1 41711,N1(C(CN(C(=O)OC(C)(C)C)CC)=O)CCC2CN(C(c3ccc(C)nn3)=O)CC2C1 41712,C(=O)(C(F)C(C)CNC(=O)CN1CCNC1=O)Nc1cnc(COC)nc1 41713,C12(COC)CCC(C(=O)NC3COCC3NC(c3cnsc3C)=O)(CC1)CO2 41714,c1(C(=O)OC)c[nH]c(=NC2CN(C(=O)COC3CCCCC3)CC2C)cn1 41715,c1(C(=O)NC2CC=CC(n3cc(C4CC5CCC4C5)nn3)C2)ccc(Br)cc1 41716,N1(C(CC(=O)NCC)=O)CC2CC(C=O)CC2C1.N1CCC1 41717,C(C(C(=O)OC)NC(C1CSCN1C(=O)CN1CCC1C)=O)N(C)C1CC1 41718,N1(C(c2ccc(C(=O)OC)cc2Cl)=O)CC2CCCC(NC(C3CC3F)=O)C2C1 41719,CC(C)C#CC(=O)N(C1CCCCC1)CCNC(=O)C(n1ccc(Br)n1)C 41720,C1(C(=O)NC(C2CC(N(C)C)C2)C)CCCC12CCC2.C12CC(C1)NC(=O)C2 41721,C1(NC(C2N(CC)CC2)=O)CCC(O)CN(C(c2cn(C)nc2OC)=O)C1 41722,N1(C(C(=O)NCC)=O)CCCC2CN(C(c3ncc(Br)cc3C)=O)CC12 41723,C1(C)(C(N2CCC(C(C(=O)N(C(CC)C)CCO)(C)C)C2)=O)CCCCO1 41724,N1(C(c2c(C)sc(C(F)(F)F)n2)=O)CCCN(C(=O)CC2CCC2)C(C)C1 41725,C1(C(=O)NCCCCC2CN(C(c3ccc(C)s3)=O)C2)CC(CO)CC1O 41726,N1(C(c2cn(C)nn2)=O)CC2C(C(=O)N(C3CCCC3)Cc3ccccc3)C2C1 41727,c1(C(=O)NCC2(OC)CN(C(=O)COCC(C)(C)C)C2)cc2scnc2[nH]1 41728,C(=O)(C1CCc2cccnc21)NC1(C)CC(c2ccccc2)C1 41729,CC(C)CC(F)C(=O)NC1COCC1CNC(c1coc(Br)n1)=O 41730,N1(C(CC(C)N(C)C)=O)CC(C(=O)Nc2ccccc2C2CCC2)CC2(CC2)C1 41731,CC(C)CCCC(=O)N1CCN(C(=O)C=CCO)CC1CO 41732,C1(CNC(C(C)(C)OCC)=O)CC(C)N(C(c2cccc(-n3cncn3)n2)=O)C1 41733,c1(OC)ccc(OC2CCCN(C(=O)NCC(C)OC)C2C)c2ccccc12 41734,N1(C(C2N(CC)CCCC2)=O)CC2(CCN(C(C3(CC)CCCCC3)=O)CC2)C1 41735,C1(CC(=O)N(C(CNC(c2cc[nH]n2)=O)Cc2ccccc2)C)CCC=CCC1 41736,C1(CNC(c2cc(OCC)n[nH]2)=O)CC2(CC2)CN1C(=O)CC1CC(C)C1 41737,N1(C(=O)Nc2cnc(CCC)s2)CCC(C(F)(F)F)C(O)C1 41738,C(C(=O)NC(C(=O)NCC(=O)NCCO)c1ccco1)(C(C)C)OC 41739,c1(C(N(C2CCN(C(=O)C=Cc3nccs3)C2)C)=O)ccc2cnnc(O)c2c1 41740,c1(CNC(c2c3c(nn2C)CCC3)C)cc2c(O)cccc2s1 41741,C#CC(C)(C)C(=O)NCC(C1CCOC1)NC(=O)COc1cccc(C(C)=O)c1 41742,c1(C(=O)NC2CC(C)(NC(CC(C)(C)OC)=O)C2)ccc(S(=O)(=O)N(C)C)o1 41743,n1(CC=C)cc(C(=O)N(C2CCCC2)CCNC(=O)CSCCC(F)(F)F)nn1 41744,c1(C(N(C)Cc2ccc(CNC(C3C(C)C3C)=O)cc2)=O)cn2c(n1)CCC(C)C2 41745,c1(CNC(CCC=C(C)C)=O)cccc(NC(=O)C(O)Cc2cnc[nH]2)c1 41746,C1(NC(C=COCC)=O)CCC2CCN(C(=O)CC(C)C3CC3)C1C2 41747,N1(C(c2cnc(C)s2)=O)CC(NC(C2(C)COC2)=O)CC(O)C1 41748,c1(C(=O)NC(CNC(CCc2n(C)ccc2)=O)C2CC2)coc2ccccc12 41749,N1(C(c2nc(C)n(C)c2C)=O)CC2CCCC(NC(=O)CC3(O)CCCC3)C2C1 41750,C12(C(=O)NC3CCC(NC(c4cc(C)no4)=O)CC3)CC(C)(C1)OC2(C)C 41751,c1(OC)ccc(OCCC(=O)N2CC(C(C)NC(=O)CC=CC(C)(C)C)C2)cc1 41752,CC(C)(C#N)CC(=O)N1CCC(C)(C)C1CC(N1CCNC(=O)C1)=O 41753,c1(C(N2CC(F)CC(NC(C3CC(C4CC4)C3)=O)C2)=O)cc2cc(Cl)ccc2o1 41754,C(=O)(C(CC(C)C)NC(C)=O)N(CCOC)CCNC(=O)Cc1sc(O)nc1O 41755,N1(C(c2cc(C)nc(C)c2)=O)CCOC2(C1)CN(C(=O)C(C)OC1CCOC1)C2 41756,N1(C(C(CCC)C)=O)CCC2(C1)CN(C(C1CCCN1c1cnccn1)=O)C2 41757,C1(C(N(CC(C(C)C)C)C)=O)C(C)OCCN1C(c1c[nH]c(=O)cn1)=O 41758,C1(CC(=O)N(C2CC(C(=O)N)C2)C)(CC2C(C)CCO2)CCCCC1.N(C)C 41759,c1(CC)nccnc1C(N1CCN(CCNC(=O)C(C)CC2CCC2)CC1)=O 41760,C1(COC(C)C(=O)NCCCN(C(=O)CNC2CCOC2)C2CC2)CCCCO1 41761,c1(C(N2C(CNC(c3c(COC)cc[nH]3)=O)CC2)=O)cccc2nc[nH]c12 41762,C(=O)(CC(C)(C)C(=O)N1CCCN(C(C2CNC(=O)CC2C)=O)CC1)OC 41763,c1(CC(=O)NCC2CCCC2NC(=O)CNC(c2cccs2)=O)cncc(F)c1 41764,c1(OC)c(CN2CCCC(NC(c3cc(Cl)c(O)cc3F)=O)C2)cc(Cl)cc1Cl 41765,N1(C(C2CC(NC(c3c(CC)ncs3)=O)C(O)C2)=O)CCS(=O)C(C)C1 41766,C1(NC(C2C(C=C)OCC2)=O)CC(F)CN(C(c2ccc(Cl)cc2OCC)=O)C1 41767,C1(NC(CC(C)c2ccco2)=O)CN(C(C2CC3(C2)CC32CC2)=O)CCC1(C)C 41768,N1(C(CC2OCCN(C(c3c(C)ccnn3)=O)C2)=O)CC(O)CC(C)(C)C1 41769,C1(NC(c2c(C)cc(N(C)C(=O)N(C)C)cc2)=O)C2Cc3ccc(Br)cc3C12 41770,c1(NC(CCC(=C)C)Cc2ccccc2)ncc(C(N)=O)cc1Cl 41771,c1(C(=O)NC(C2CCCN2C(=O)CNC(N)=O)(C)C)coc2c1C(=O)NCCC2 41772,N1(C(C(=CC2CCCC2)C)=O)CCC(NC(c2sccc2F)=O)C(CO)C1 41773,c1(CC(=O)Nc2cccc(OC(F)(F)F)c2)ccc(Br)c(Oc2ccccc2)c1 41774,C1(CCC)CN(C(C23CCN(CC2)C3)=O)CC1C(N1CC(N(C)C)C1)=O 41775,N(C1CN(C(C2CC3(CC3)CO2)=O)CCc2ccccc21)C(C(C)(C)C#N)=O 41776,Cc1nc(=NCC2(C)CCN(C(C3CC3(C)C)=O)C2)[nH]cc1[N+](=O)[O-] 41777,CC(CC(=O)NCCC1CC(C(=O)NCc2nc(=O)o[nH]2)C1)CC(C)(C)C 41778,C1(NC(C(C)OC)=O)COCCN(C(=O)C(C)N(C)C)C1 41779,N1(C(C2N(C(C)=O)CCCC2)=O)CC(NC(c2scnc2Cl)=O)C2CCCCC12 41780,c1(C(=O)NCC(C)(C)CNC(=O)C=Cc2cnc[nH]2)ccc2nc(O)sc2c1 41781,C(C)(CNC(=O)COC(C)C)(C(C)C)NC(C=C(CC)C)=O.c12ccc(cc1)s2 41782,N#CC1(CC(=O)NC(C)(CNC(c2cc(F)ccc2F)=O)C2CC2)CCCCC1 41783,CC(C)CC(C)CN=c1[nH]c(N2CCC(C3CCCC3)C2)nc2c1CSC2 41784,C(=O)(CCC(C)(C)[N+](=O)[O-])N(CCC(C)C(F)F)C.C1(=O)C(C)(C)CN1 41785,CC1COC(C(F)(F)F)N1C(C1(C)CCN1Cc1[nH]cnc1-c1cccnc1)=O 41786,N1(C(=O)OC(C)(C)C)CCN(Cc2cn(C3C=CCCC3)nn2)C(C(N)=O)C1 41787,C1(C(N2C(CNC(C3C(C)=C3)=O)CN(C)CC2)=O)CCc2nncn2C1 41788,C1(NC(C2C(C)(C)C2)=O)CCCN(C(c2cc(Cl)nnc2Cl)=O)CC1 41789,Cc1ccc2c(c1)CC(C(=O)NC(C)(C)CCCCNC(c1[nH]nnc1C)=O)O2 41790,Cc1c(C(=O)NCC(C)(C)CNC(=O)C(C)NC=O)ccc(Br)c1F 41791,C1(C(=O)NCCC=C)CCCCN(C(=O)C(C)(C)C2CCCC2)C1 41792,N1(C(Cc2nnc(C)o2)=O)C2CCC1CC(CNC(C1CC13CC3)=O)C2 41793,N1(C(C(C(C)C)NC=O)=O)CC2(CCN(C(C3CC3(C)Br)=O)CC2)C1 41794,c1(C(N(CCNC(c2c(CC)c[nH]c2)=O)CCOC)=O)cccc(Cl)c1OC 41795,C1(C(N2CC(CCNC(c3c(C)nc(CC)s3)=O)OCC2)=O)CS(=O)(=O)CCO1 41796,N1(C(c2c3c(ccc2)C(=O)NC3)=O)CCC2(CCN(C(c3cnc(O)s3)=O)C2)C1 41797,c1(CC(N2C(CCNC(COCC(C)C)=O)CCC2)=O)cnc2c(=O)[nH]ccn12 41798,C=CCC(CC)C(=O)NCC1(NC(=O)Cc2sc(O)nc2O)CC1 41799,Cc1ccc(C(=O)NC2CC(C(=O)NCC(C)C(C)(F)F)C2(C)C)c(O)c1 41800,c1(C(C(=O)NC2CCC(CNC(C(C)O)=O)C2)=O)ccc(NC=O)cc1 41801,c1(CN(c2cc3ccccc3[nH]2)C)ccc2nccn2c1 41802,N1(C(CCC(=O)NCCC)=O)CCN(C(=O)C2=CCSC2)C(C2CC2)C1 41803,N1(CC)OCC(NC(c2coc(C(F)F)c2)=O)C1=O.C1(=O)C=CCCCN1 41804,N1(C(COCC(=O)NC)=O)CC(C)(C)OCC1CNC(C1CCCC(F)(F)C1)=O 41805,N1(C(C(C)CN(C)C)=O)CCN(C(C2(n3cncn3)CC2)=O)CC1CCN(C)C 41806,C1(C(=O)NCC2CC2CNC(c2coc(C)n2)=O)(OC)CCCOC1 41807,Cc1cn2c(n1)CCC(C(=O)NNC(c1nnc3ncccn13)=O)C2 41808,O=C(CS(=O)(=O)CCO)NCC1CCCC1NC(C1CS(=O)(=O)C1)=O 41809,N1(C(C2C(NC(c3ccnc(C(C)(C)C)n3)=O)C2)=O)CC(F)(F)C(F)(F)C1 41810,c1(OC)ncc(C(=O)NC2C3CC2N(C(C2CCCCC2F)=O)C3)c(C)n1 41811,CC(C)CC(C)CC(=O)N1CCC=C(CNC(c2cn(C(C)C)cn2)=O)C1 41812,N1(C(CCc2c(C)noc2C)=O)CC2(C1)CN(C(=O)C(C)(F)F)CCO2 41813,CC(C)(CC(=O)N1CC(N2CCN(C(C3(C#N)CC34CCC4)=O)CC2)C1)CC(F)F 41814,c1(OC)cc(N2CCC3CCC(C2)N3C(C2CCCO2)=O)ccc1[N+](=O)[O-] 41815,C(=O)(C1=CCC(F)(F)CC1)NC1CCC(NC(C(CCC)(C)O)=O)CC1 41816,N1(C(c2cnc(C(C)(C)C)nc2)C(=O)NCC)CCn2c(cnc2C(F)F)C1 41817,c1(OC(=O)NC2C(NC(CC)=O)C2)ncc(C)cc1C 41818,c1(CCN(c2nccc(N(C)CC(N3CCCC3)C3CC3)n2)C)cccc(Cl)c1 41819,C=CC(C)(CC)C(=O)NCC1(C)CCN(C(C2(Sc3ccccc3)CC2)=O)C1 41820,N1(C(C(CC)Oc2ccccc2)=O)CCC(NC(=O)C(C)(C)c2cnsc2)CC1 41821,C1(C#N)(C(=O)NC2CC(C(C)NC(C3(OC)CC3)=O)C2)CC1C(F)(F)F 41822,C(=O)(C1=C(C)CCOC1)NC(C(=O)NCC(C)OCC#C)C1CC1 41823,c1(C(=O)NCC(C)(C)NC(=O)CCc2ccsc2)cc(F)c2ccccc2c1 41824,CC1(C)CC(N=c2ccnc(N(CCO)CC3CCN(S(C)(=O)=O)CC3)[nH]2)CO1 41825,N1(C(COC(c2nccn2C)C)=O)CCC(C(C)NC(c2ccns2)=O)CC1 41826,C1(CN(C(C2N(CC)CC2)=O)C)C2CN(C(=O)CNC(=O)CCCCO)CC12 41827,c1(C2(c3nc(C4CN(C(c5ccccc5)=O)C4)on3)CC2)ccc(Cl)cc1 41828,CC(C)(CCCNC(=O)C#CC1CCCC1)C(=O)NC1CC(=O)N(C2CC2)C1 41829,c1(C(N2C(C)(CC(=O)NC3(C#C)CC3)CC2)=O)cc(C#N)[nH]c1C 41830,c1(N2CCCC(NC(C)=O)C2)nc2c(c(=NCc3ccc(Br)s3)[nH]1)COC2 41831,C1(O)(CC(=O)N(CC(C)(C)CNC(=O)CCN(S(C)(=O)=O)C)C)CCCOC1 41832,c1(CN(C(=O)C(=O)NC2CC2)CCOC)c(C)nn(C)c1C 41833,N1(C(=O)NC(CC)C(=O)NC)CCCC2CN(C(=O)Nc3ccccc3)CCC12 41834,c12cccc(c1)NC(=O)NC2.N1(C(C)=O)CC(C(c2cnsc2)C2CC2)C1 41835,c1(NC(C2N(C(C)C)C(=O)CCC2)=O)ccnc2cc[nH]c12 41836,c1(C(=O)NC(CNC(Cc2c(C)nccc2)=O)CC(C)C)ccc(S(C)(=O)=O)s1 41837,CC1(C)CC(NC(=O)C=CI)CN(C(=O)C(F)n2ccnc2)C1 41838,N12CC3CC(CC1C3)NC(=O)C2=O.c1(C(=O)NC2(C3CCCO3)CC2)ccccc1 41839,C(CC(C(C)(C)C)NC(c1ccccn1)=O)N(C(=O)CCC(=O)c1ccc[nH]1)C 41840,c1(CCCCNC2C(NC(=O)OC(C)(C)C)CC2)nnnn1CC1CCCO1 41841,C#CCC(CC#C)C(=O)N(C1CN(C(c2ccc(S(C)(=O)=O)o2)=O)CC1(C)C)C 41842,C1(NC(c2c(F)cncc2Br)=O)CC2(C1)CN(C(c1cnoc1)=O)C2 41843,n1(CC(=O)NCC2(CN(C(=O)CC(C)(C)C)C)CC2)cccc(N)c1=O 41844,CC1(C)CN(C(=O)CC(O)C2CCCC2)C1C1CCN(C(=O)C(O)C2CC2)CC1 41845,N1(C(C2CCCN(C(C)=O)C2)=O)C2CCC1CC(C(=O)NC1CC1C(N)=O)C2 41846,c1(OC)ncc(Cl)cc1C(N1CC(CNC(C2CCC(C)(O)CC2)=O)C(C)C1)=O 41847,O=C(O)CC(Br)C1CN(C(=O)CC2C=CCCC2)C1 41848,c12cc(ccn1)N2.n1(CC)nnnc1C(C)(COC(C)(C)C)NCC1CCOC1 41849,CC1CN(C(c2ccnc(O)c2F)=O)CCC1NC(=O)C=CI 41850,c1(C(N2CC(CC=C)(NC(c3ccnnc3C)=O)C2)=O)nnc(O)cc1O 41851,c1(CN(C2COC3(CCNCC3)C2)C(C(C)CC(N)=O)=O)ccc(C#N)cc1F 41852,c1(C(N(C(C)(C)C)CCN)=O)cnc2c(-c3cncnc3)cccc2c1 41853,C1(C(=O)NCC2(C)CCN(C(C(C)N(C)C)=O)C2)CCC=CCCC1 41854,CCC(C)(CNC(C1CC(F)(CO)C1)=O)NC(c1c[nH]nc1-c1ccoc1)=O 41855,c1(C(=O)NC(C(=O)N(CCCC)CC)CO)cnncc1OC 41856,c1(C(=O)NC(CC)CN(C)C(c2ccc(N)cc2Cl)=O)cc(P(C)(C)=O)ccn1 41857,Nc1ccc(CCC(=O)NCCOC2CCN(C(=O)CCC3CC3)CC2)cc1F 41858,Cc1n[nH]cc1CN(C(C(=O)NC1CCCC1CC(F)(F)F)c1cccs1)C 41859,CC(C)(CN=c1nc(N2CCCC(C(C)(C)C(N)=O)C2)c2c([nH]1)CCC2)C(N)=O 41860,C1(CC(=O)NCC(C)(C)OCCNC(C2CC(CC(C)(C)C)C2)=O)CS(=O)(=O)C1 41861,C1(OC)CCn2cc(C(=O)NC3CCCC(CSc4ccccc4)C3)nc2C1 41862,C1(C(N2CCCC(N(C(=O)COCC3(F)CC3)C)C2)=O)CCOCC12CCC2 41863,C(=O)(CC(C(F)F)n1ccnc1)NC(C(=O)NC(c1ccccc1Br)C)CO 41864,CCCS(=O)(=O)CC(=O)N1CC(NC(c2cc(N(C)C)ccc2F)=O)CC(F)C1 41865,Cc1cccc(C)c1C(=O)NCC(=O)NCC1COCCN1C(=O)CSC1CC1 41866,C1(C(=O)NCc2ccc(O)c(Cl)c2)CN(C(C2CCOC2)=O)CCC1(F)F 41867,N1(C(C(CCOC)C)=O)CC(C)OC2(CCN(C(=O)C3=CCCSC3)CC2)C1 41868,c1(C(N2CC(CC)N(C(=O)C(F)(F)C(C)(C)O)CC2)=O)ccc2c(c1)CNC2=O 41869,c1(CCNC(COCCOCCOCC)=O)cnn(CCO)c1C1CC1 41870,CC(C(F)F)=CC(=O)N(C)CCC1(C)CC1 41871,N1(C(Cc2ccc(C)s2)=O)CCC(NC(c2cnoc2-c2cccs2)=O)C(F)C1 41872,c1(C(=O)OC(C)(C)C)ccc2c(c1)CCN2C(=O)O.C(C(=O)O)N(C)CCO 41873,C12(C(=O)NC(CC)COC)C(NC(c3cccc(C)c3F)=O)C3CC1C2C3 41874,C1(CC(=O)N(CC(O)CN(C)C(c2coc(CO)c2)=O)C)CCCC12CC2 41875,c1(N(C)C)nccc(C(N2CC(CCNC(C3CCC(C(N)=O)C3)=O)C2)=O)n1 41876,CC1C(NC(=O)C#CC2CCCC2)C(C)CCN1C(=O)CNC(N1CCCC1)=O 41877,N1(CC(=O)NCC2OCC(CNC(c3ccc(OC)s3)=O)C2)CCC(F)CC1 41878,C1(O)(CNC(c2c(C)cns2)=O)CCN(C(C2CCCC(O)C2)=O)C1 41879,C1(C2CCN(C(C3C(CC)(CC)C3)=O)C2)CCCCN1C(C1CCCC1(C)C)=O 41880,C1(C(N2CCC(O)(CNC(C3CC4(C3)CC4F)=O)C2)=O)Cc2cncn2C(=O)N1 41881,C(=O)(C#CC1(CC)COC1)NC(CC=C)C(=O)NCC(C)(C)n1cccn1 41882,C(=O)(C(CCC)N(C)C)N(CC1(C(=O)NC(CC#C)CC)CC1)CC 41883,C1(NC(CCOC)=O)CCN(C(c2cnc(S)nc2)=O)CCC1(F)F 41884,c1(C(=O)NC(CC)CNC(=O)C=Cc2ncco2)cnc(O)n1CC 41885,C1(C)(C(=O)NC(CNC(c2c(C)cccc2C)=O)CO)CC(C(C)C)=NO1 41886,CC1(CNC(c2cc[n+]([O-])cc2)=O)CCC(NC(C2(c3ccno3)CC2)=O)C1 41887,N1(C(c2ccc(NC(C)=O)s2)=O)CCC(CNC(=O)CCN2CCC2)CC1 41888,C1(C(N(C)CC2CCN(C(=O)CC#N)C2)=O)C2CCC1(c1cncs1)C2 41889,C1(CC(=O)NCCC(F)(F)F)CCCC(NC(=O)C(F)=CC2CC2)C1 41890,CCC(CC(=O)NC1CCC(CO)C1)NC(c1cccnc1O)=O 41891,C(CNC(c1cnn(CCF)c1)=O)(CC(F)(F)F)NC(C(CCC)NC(C)=O)=O 41892,c1(C(CC)NCCc2c[nH]c(=NC)s2)ccc(F)c(Oc2ccccc2)c1 41893,C1(F)(CNC(c2nc(OCC)sn2)=O)CCCN(C(C2CN(C)C2)=O)C1 41894,c1(C(N(CCNC(c2cc(C#N)ccc2N)=O)CC)=O)ccc2ccccc2n1 41895,C12(C(N(CC(C)(C)C)CCO)=O)CC(NC(=O)OC(C)(C)C)(C1)C2 41896,C1(NC(=O)C2CC2)(CCCCN(C(C(C)OC(C)(C)C)=O)C)CCCCC1 41897,c1(OCCN(C)C)cncc(C(=O)NC2CCN(C(c3ccco3)=O)C2)c1.OC 41898,N1(C(C=CCOC)=O)CC(NC(=O)COc2cc(C)on2)CC(C)C1 41899,c1(C(=O)OCC)c(-c2cn(CC(C)NC(=O)C(C#N)CC)nn2)cnn1C 41900,C12(CNC(=O)C=Cc3nccs3)CC(CN1C(=O)COc1ccon1)C2 41901,CC1(C)CCC(C(N2CCC2CC2CC2)=O)CN1C(=O)CN1CCCCC1=O 41902,C1(CNC(C(C)=CC2CC2)=O)C(C)CCCN1C(c1cccnc1)=O 41903,C=C(C)C1OCCC1CC(=O)NC1CC(NC(C2(C)CC(C)C2)=O)C1 41904,N1(C(CN(C)C2CC2)=O)CCC(CNC(c2csc(Cl)c2)=O)C1(C)C 41905,C1(F)(C(N(C2CCN(C(c3cnc(C(N)=O)s3)=O)CC2)CC#C)=O)CCOCC1 41906,C1(COC)(NC(C2CC2C)=O)CCN(C(c2ccnc(-n3cncn3)c2)=O)C1 41907,c1(C(=O)NC2(C)CC(NC(C(C)NC(=O)NC)=O)C2)nn(C)cc1C 41908,C(c1ccc(F)c(F)c1)=CC(=O)NC(C1CCCCN1C(=O)C1=CCCSC1)C 41909,Cn1cncc1CN1CCCC1CNC(C1CC(=O)NCN1)=O 41910,C1(C(=O)NCc2scc(C)c2)C=CCCN1C(c1ns[nH]c1=O)=O 41911,c1(CNC(c2c(C(C)NC(C(CSC)OC)=O)noc2)=O)ccnc(F)c1F 41912,c1(CNC(C(CSC)C)=O)cc(C(=O)NCCc2noc(=O)n2C)ccn1 41913,N1(C(C2C(OC)CCC2)=O)CCC(C)(NC(=O)C(N2CCN(C)CC2)C)C1 41914,Cc1c(F)cc(CNC2CC(C(=O)Nc3cnn(-c4ccncc4)c3)C2)cc1Br 41915,c1(C(N2CCC(N(C(=O)C#CC3(C)CC3)CC)C2)=O)nn2c(c1Br)CCC2 41916,CCC(C)(C(=O)Nc1cccc(C(N2C(CO)CC2CO)=O)c1)OC 41917,C1(CCC2N(C(C=C)=O)CCC2)CCCCN1C(=O)COC(=O)CO 41918,C(=O)(C(C)(C)CF)NCC(CCOC)NC(C1(N2CCCC2)CCC1)=O 41919,Cn1ncn(NC(=O)CC2CCN(C(c3ccc(Cl)cc3)=O)CCO2)c1=S 41920,C(=O)(CC(C)C(F)(F)F)N(CCNC(C1C2CCC1(c1ccccn1)C2)=O)CC 41921,Cc1ccoc1C(=O)NC1CCC(CC(=O)NCC2CC=CCC2)C1 41922,c1(CC(=O)NCC(CC=C)NC(C2(OC)CCSC2)=O)cnn(C)c1C 41923,CC1(C)CN(C(=O)C(=O)N(C2CCCC2)CCCSC(F)F)CCS1(=O)=O 41924,c1(C(C)C(=O)N(C)C)nc2cc(-c3nc(C4CCC4)nn3C3CCSC3)ccc2o1 41925,CC(C)C(C(C)NC(=O)C=CCF)NC(c1cc(C2(C)CC2)on1)=O 41926,O=C1CC(C(=O)NCC2(C3CC3)CCCO2)N(C(=O)C(C2CCCCC2)=O)C1 41927,c1(C(C(C)NC(C2(CC3CC3)CC=CC2)=O)NC(C2C(=C)C2)=O)ccc(CC)cc1 41928,C1(COC)CC(CNC(=O)C=Cc2ccsc2)CN1C(c1ccn(C)c1)=O 41929,C1(NC(C2(C(N)=O)CC2)=O)CN(C(=O)COC2CC2)C2(CCC2)C1 41930,O=S(=O)(c1cccc(=NC2C=CCCC2)[nH]1)NCCCc1ccc(OC(F)F)cc1 41931,c1(CCC(=O)N(CC(C)O)CCNC(=O)CP(C)(C)=O)ccc(Cl)cc1F 41932,c1(CC(N2CC(C(C)NC(C(CCC)(C)C)=O)C2)=O)coc2cc(Cl)ccc12 41933,C=CC(C)CC(=O)N(C1(C(=O)NCc2ccc(Cl)cn2)CCC1)C1CC1 41934,C12(CNC(c3cccc[n+]3[O-])=O)CCCC(CN1C(C1CCCCC1)=O)C2 41935,C(C(CC(C)C)C(=O)N1CC2(CC(C)CO2)C1)NC(C1C(OCC)CC1)=O 41936,N1(C(CSCC#C)=O)CC(C2CC2C(N2CC(N3CCCC3)C2)=O)C1 41937,c1(C(=O)NC2(C)CCN(C(C(CCC)N(C)C)=O)C2)c[nH]c2ncccc12 41938,c1(C(=O)NC(CNC(CC(C=C)c2ccccc2)=O)C)cc([N+](=O)[O-])oc1C 41939,C1(N(C(C2C(C=C)C2)=O)C(c2snnc2C)=O)CCN(C(C)=O)CC1 41940,c1(CC)cncc(C(N2CCC(NC(=O)C(F)=C3CCCC3)CC2)=O)c1C 41941,C1(NC(C(C)NS(CCC)(=O)=O)=O)CC(NC(=O)CCC2(NC(C)=O)CC2)CC1O 41942,C1(CC=C)(NC(c2cc(Cl)cnc2O)=O)CCCN(C(=O)CSCCC(C)C)C1 41943,c1(C(=O)NCC2N(C(CN(C)CC)=O)CCCC2(C)C)ccc2nsnc2c1 41944,N1(C(CC(=O)NCCC)=O)CCC(OCC)C1C(=O)N(CCOC)CC 41945,C(=O)(C#CC1CC1)N1CCC(C(C)N(NS(N)(=O)=O)C(=O)Cc2ccccc2)C1 41946,C1(CNC(C2CC3CC3C2)=O)CC2(CCOCC2)CN1C(c1coc(O)n1)=O 41947,N1(C(c2c(OC)scc2)=O)CC(NC(=O)Cn2ccnn2)C2(CC2)C1 41948,c1(C(=O)NCC2CN(C(c3c(OC)n[nH]c3)=O)C(C)C2)nccc2[nH]ccc12 41949,c1(C(N2CCCC(NC(c3c(CC)onc3C)=O)C2)=O)c(C)nn2cccnc12 41950,Cc1ccc(Cl)c(C(N2CC(N(C(=O)Cc3cnc[nH]3)C)C(F)C2)=O)c1 41951,c1(C(=O)NC(C2CCN(C(C3CC(C)(C(=O)OC)C3)=O)C2)(C)C)cnn(C)c1C 41952,c1(CC)ccccc1C(=O)NC(CCF)C(=O)N(CCC1CC1)CC 41953,C1(C(=O)NCCCC2(NC(=O)CNC(=O)Cn3cncn3)CC2)CN2CCN1CC2 41954,C1(CNC(C=CC=CCC)=O)CCCCCN1C(=O)CC(C)(C)CNC(C)=O 41955,C(=O)(CCCCCCC(C)C)NCCN(C(=O)CCNCC)CC(C)O 41956,C=CC1(C(=O)NC(c2ccccc2F)(C)CNC(C2CC(C)C2)=O)CCCCC1 41957,CCCCC(O)C(=O)NC1COCCN(C(C2CCCCN2C)=O)C1 41958,C1(NC(=O)CCCn2c(O)nnc2O)COCCN(C(c2ccsc2CO)=O)C1 41959,c1(C(=O)NCC2(OC)CN(c3nnc(C)s3)C2)ccc2cccnc2n1 41960,N1(c2nc(OCC)c(Cl)cn2)CCC2(NC(c3nsnc3O)=O)CCCCCC12 41961,Cc1ccc(C(=O)NCCCCCC(=O)NCCC2CCCOC2)nc1C 41962,N1(C(C=C(CC)C)=O)CCN(C(C2(C(C)(F)F)CC2)=O)CC12CC2 41963,O=C1NCc2ccc(NS(=O)(=O)c3ccccc3C3CNC3)cc21 41964,c1(C(=O)NCC2CC(NC(c3cc(C)ns3)=O)C2)coc2c(F)c(Cl)ccc12 41965,N1(C(CC2C(C)CN(C(=O)CN3CCNC(=O)C3)C2)=O)CCC2CCCC12 41966,C(=O)(C1=CCCCC1C)N1CCC(F)(C(N2CCOCC(C)C2)=O)C1 41967,c1(C(N2C(CNC(Cc3cc(C)[nH]n3)=O)CC(F)C2)=O)c(F)c(F)cc(F)c1F 41968,C(C(CC=C)C(=O)NCC1=CCCCC1)NC(CSCC=C)=O 41969,c1(C(c2nn[nH]n2)N(C(C(=O)NC(CC)C2CC2)=O)c2ccsc2)ccccc1 41970,C1(C(N2CCN(S(C)(=O)=O)CC2)=O)C2CCC(C2)C1NC(C1CCCCC1)=O 41971,c1(CC(=O)N(C2CCN(C(c3cocc3C(N)=O)=O)CC2)C)ccccc1Cl 41972,CC1CCCCC1C(=O)N(C(CNC(C1(C)CC(F)C1)=O)C1CC1)C 41973,Cc1nc(CNC(=O)C(C2(O)CCC2)NC(=O)Cc2cn(C)nn2)cc(O)n1 41974,c1(CC)ncccc1C(=O)NC1CC(CNC(=O)COCC2CCC2)C1(C)C 41975,N1(C(C(=O)NC(c2cccc(C)n2)C)=O)CCC(F)(F)C2(CC1)NC(=O)NC2=O 41976,c1(CC(=O)NC2CCC(C(N3CCC(CF)C3)=O)CC2)ccnnc1O 41977,c1(C(=O)NCCN(C(c2n(C=C)nnc2)=O)C(C)C)cc(Cl)cc(C)c1C 41978,c1(CC)ccc2occ(-c3nc(CCN4CCOCC4)nn3C3CC3)c2c1 41979,N1(C(c2c(C)csc2)=O)CC(NC(c2cc(C(C)(C)C)no2)=O)CCC(O)C1 41980,CC1(C(N2CCN(C3CN(C(=O)C(O)C4CC4)C3)CC2)=O)CC=CCC1 41981,Cc1c(C(N2CCC(NC(c3ccc(N)cc3)=O)C2)=O)c(=O)n(C)c(=O)n1C 41982,C1(OC)CN(C(=O)CC(O)CNC(C2CC23CCCCC3)=O)CC12CC2 41983,N1(C(c2c(CC)nn[nH]2)=O)CC(CNC(=O)Cc2c[nH]nc2O)CCC1C 41984,N1(C(c2nc(C)[nH]n2)=O)CC2(CC2)CC1CNC(c1cc2sccc2s1)=O 41985,C1(NC(CCc2ncc(C)[nH]2)=O)CCN(C(C2CC3C=CC2CC3)=O)CC(O)C1 41986,c1(C(N2C(CNC(C(C(C)(C)C)O)=O)C3CCC2C3)=O)sc2ncccc2c1N 41987,CC1(C)CNc2ccc(C(=O)NCC(F)CO)cc21 41988,C1(OC)CCCC(NCC(=O)Nc2cccc(I)c2)C1 41989,C1(NC(CCc2cc(C)on2)=O)CCOC(CNC(=O)Cc2ccc(Cl)cn2)C1 41990,CC(C)C(C(=O)NCC(C)CN(C)C(C1CN(C)C1)=O)C1CCC1 41991,C1(NC(Cn2c(C)ncc2)=O)CS(=O)(=O)CC1NC(C1(C(N)=O)CC1)=O 41992,c1(C(=O)NC2CN(C(C3(CC)CCCCO3)=O)CC2F)cncc(C)c1Cl 41993,C(=O)(CC(C)(O)C(F)(F)F)NCC1(F)CCC(CNC(CN(CCC)C)=O)C1 41994,N1(C(c2cc(C)nc(O)c2)=O)CC2CCC(C1CO)N2C(c1ccccc1Cl)=O 41995,C(=O)(C1CC(=O)Nc2ccccc21)NCC1C(NC(CN(C)C2CC2)=O)C1 41996,C1(C(=O)NCCCCN(C(CCCCCC#C)=O)C)CCc2ccc(F)cc2O1 41997,C(N=c1[nH]c(=NCC(C)C#N)[nH]c2cc[nH]c12)c1c(CC)nsc1 41998,c1(OC)c(NC(=O)C=C2CCN(Cc3c(Cl)ccnc3Br)CC2)cccc1C#N 41999,C1(C)(C(=O)NC(C)CCCNC(c2n[nH]cc2Cl)=O)CC(C(C)(C)C)=NO1 42000,C(c1ccccc1F)=CCC(=O)NC1CN(C(C2(CCCC)CCC2)=O)CC1O 42001,CCC(C)(C)C(=O)C(=O)N1CC(C(=O)NCC2(CO)CC2)C(F)(F)C1 42002,c1(C(N2CC(N(C(CCSC)=O)C)C(C)CC2)=O)cnc2onc(C(C)C)c2c1 42003,c1(C(=O)OC)ccc2c(c1)CCC(NC(c1cc(Br)nn1C)=O)C(=O)N2 42004,C1(SCC)CCC(C(N2CC(C(N3CCCCC3)C(=O)NCC(C)C)C2)=O)CC1 42005,N1(C(C2(C(=O)OC)CCCC2)=O)CC(C2(NC(C3(F)CCC3)=O)CC2)C1 42006,CON1CCC(C(=O)NC2CC(c3cn(-c4ccc(Cl)cn4)nn3)C2)CC1 42007,C1(CNC(CSC)=O)(CNC(C2CNC(=O)O2)=O)CCOCC1 42008,C1(NC(c2cc(CCC)oc2C)=O)CCN(C(=O)CNC(=O)C(F)(F)F)CC1F 42009,Cc1c(C(=O)NCCN(C(=O)CC2CC(O)C2(C)C)CC2CC2)cnn1C(C)(C)C 42010,N1(C(=O)NC(C2(C#N)CCC2)C)CCCc2ccc(F)cc21 42011,C12CC(C)C1NC2=O.C(C(C)(C)CN(C(=O)C(C)OCC(C)C)C)NC(=O)OC 42012,N1(C(c2nc(CC)sc2)=O)CCC(C2CCCN(C(C3(O)CCOC3)=O)C2)CC1 42013,C(=O)(C(C)C(C)(C)C)N(C(C)CN(C)C(c1cn(C)nc1C(F)(F)F)=O)C 42014,N1(CC(=O)NC(CNC(c2cc(C(C)=O)on2)=O)C)CCCCC1=O 42015,Cc1cn2c(C(=O)NCC(C)CNC(=O)COc3cccc(C)c3F)cnc2s1 42016,c1(C(=O)NCCC(C)N(c2nc(SC)nc(O)c2)C)cc2cc(C)ccc2cn1 42017,c1(NC(C(C2CN(C(=O)CCC3(C#N)CCC3)C2)OC)=O)cnc2ncnn2c1 42018,C12CC(CCO1)NC2=O.S(C(F)(F)F)CC(=O)Nc1nn[nH]n1 42019,N1(C(CNC(=O)NC2CC3(C2)CC32CCC2)=O)CCCc2ccccc21 42020,Cc1cc(CNC(C2CC(NC(C3(N(C)C)CCC3)=O)CCO2)=O)ncn1 42021,C1(C(N2CC(C(O)C(=O)NC(C)CC(F)(F)F)C2)=O)(CC)CNC(=O)C1 42022,c1(OC)ccc(C(C)NCCC2CC(F)(F)C2(F)F)c(OC)c1 42023,C(c1cc(C)cc(C)c1)=CC(=O)NCC(CCOC)NC(C1CC1[N+](=O)[O-])=O 42024,CC(C)C(CN(C)C)C(=O)NC(C)(CNC(=O)CCC=CC=CC(C)(C)C)C1CC1 42025,N1(C(c2cccc(CCC)c2)=O)CCC(F)C(NC(C2CC2CF)=O)C1 42026,CCCC(O)CC(=O)NC(CNC(C1CCCS1)=O)(CC)CC 42027,c1(CC)ccc(NC(C2C3CS(=O)(=O)CC23)=O)c(C)c1 42028,CC(C)CCCCC(=O)NC1(C(=O)NCC2(Cl)CC2(F)F)CCCC1 42029,Nc1c(Cl)cc(C(=O)NC2CC(NC(=O)CC3CCC4(CCC4)O3)C2)cc1[N+](=O)[O-] 42030,N1(C(CC2(OC)CC2)=O)CCC(C(C)NC(=O)C(c2ccc(F)cc2)(C)C)CC1 42031,Cc1nc(C)c(F)c(=NCC(C(C)(C)C)NC(c2cccc3c2C(=O)NC3)=O)[nH]1 42032,c1(C(=O)NCC(n2cc(C(=O)O)nn2)C)csc(CNS(C)(=O)=O)n1 42033,C1(NC(CC2(CN(C)C)CC2)=O)CC(NC(=O)C(C)(C)CC2CCC2)C12CCC2 42034,n1(CC(N2CCC(C(C)NC(CCCC#CC)=O)C2)=O)cc([N+](=O)[O-])c(C)n1 42035,CN1CCOC(CSc2ccccc2)C1.N12CCOC(C1)C1CN(C1)C2=O 42036,N1(C(COCCC=C)=O)CC2CCC(NC(c3c(Cl)ccnc3F)=O)CC2C1 42037,c1(CCC(=O)NC(CNC(C2(CSC)CC2)=O)C)cnn(C)c1 42038,C12(C(=O)NCC3(C(C)NC(c4cnc(S)n4C)=O)CC3)CCCN(C1)S(=O)(=O)C2 42039,C(=O)(C(C1CCC1)NC(=O)C=CC(F)F)NCCCOC 42040,n1(CC)cc(Cl)c(C(N2CCC(CNC(C3CCC(=O)O3)=O)C2)=O)n1 42041,C1(CNC(=O)C(F)=C2CCC2)CC(NC(=O)CCc2ncc[nH]2)C12CCC2 42042,C(CCCCCCCO)=CC(=O)NCC(CNC(C1(CCCC)CC1)=O)(C)O 42043,CC1C(NC(C2CCCC2)=O)CC2CCC1N2C(c1ccc(C(F)F)o1)=O 42044,c1(C(=O)NC(CCC)CNC(=O)C(C)(F)c2ccon2)cc(C)c(C)o1 42045,c1(OC)cc(F)c(F)cc1-n1nc(CO)nc1C1CCCCN1C(C)=O 42046,C(CC(C)C)(C(=O)NCCC1(CO)CC1)N(C(C(ON=C(C)C)C)=O)C 42047,N1(C(COC(C)(C)C)=O)CCc2ccc(C(=O)NC3C(=O)NCC3(C)C)nc2C1 42048,c12cccc(n1)NC2.C1(C(=O)NC(=O)CC2(C(N)=O)CC2)CCC(CO)CC1 42049,C1(NC(c2c(C)nsc2C)=O)CC12CCN(C(c1cnn3ccn(C)c13)=O)CC2 42050,N1(C(CC2CCCN(C(C(CC)(C)COC)=O)C2)=O)CC(C)N(C)C(C)C1 42051,C(C(C)(C(=O)N(CC(C)(C)CO)C)NC(c1cc(=N)[nH][nH]1)=O)SC 42052,C1(C(=O)NC(C)CCCO)CCCC(NC(=O)Cn2ccnc2)CC1 42053,N1(C(c2ccc(CC)s2)=O)CC2CC3CC2C1C3NC(C1COCCC1(F)F)=O 42054,c1(NC(CC(CC#C)N)=O)cc2c(cc1Cl)NC(=O)C2 42055,N1(C(C2CC(C)(C#N)C2)=O)CC2CCCC2(CNC(c2ccsc2Cl)=O)C1 42056,CCC(O)C(F)(F)C(=O)N1CC(CCNC(=O)C(CC)c2ccccc2)(OC)C1 42057,c1(C(N(CC(C)NC(=O)CCCn2cncn2)CC)=O)c(C)cccc1C 42058,C1(O)(CNC(CC(CC)(F)F)=O)CCCN(C(c2ccc(Cl)cc2)=O)CC1 42059,N1(C(CC2(C)CC2)=O)C2CCC1CC(CNC(=O)CCCC1CCCC(=O)N1)C2 42060,C(CNC(C1(Cl)CC1(F)F)=O)(CC(=O)NCc1cnn(C)c1O)OC 42061,C1(CC(N)=O)(NC(C2CCOC2)=O)CCN(C(=O)CNC2CCCC23CC3)CC1 42062,CCCC(C)(C)CC(=O)N1CCC(N(C(=O)CCOCC2CCCO2)C)C(C)C1 42063,CCCCC(CC)CC(=O)N(C1CC(NC(c2csnn2)=O)C1)C 42064,CC1C(C)N(C(=O)C=Cc2cocn2)CCN1C(=O)C=Cc1ccco1 42065,N1(C(c2c(C)cnnc2)=O)CC(NC(=O)CC2NC(=O)NC2=O)C(C)(C)C1 42066,C1(CC(=O)NC(C(C)NC(CC2C(CC)C2)=O)CO)(CO)CCCCC1 42067,Nc1ccc(C(=O)NCC2CC2NC(=O)Cn2ccc(O)nc2=O)cc1Cl 42068,c1(OC)ccc(Br)c(C(N2CCC(CN(C)C(c3ccc(F)cc3)=O)CC2)=O)n1 42069,CCC(CC)C(=O)NC(Cc1ccncc1)C(N1CCCC(O)C1)=O 42070,C12(CNC(C=C3CCC(C)C3)=O)CC1CN(C(=O)COCC1CCCC1)C2 42071,C12(C(N3CC(NC(c4c(C)noc4)=O)C(C)C3)=O)CCC(C(F)(F)F)(CC1)CC2 42072,c1(C(=O)NCC(C2CCC2)NC(CN2CCC(C)C2)=O)ccc2cc[nH]c2c1 42073,C(c1sc(Cl)nc1Cl)=CC(=O)NC1(COC)CCN(C(C23CCCC2C3)=O)C1 42074,N1(C(C2C(C#C)C2)=O)CCC(NC(c2c[nH]cc(Cl)c2=O)=O)C(C)(C)C1 42075,c1(C(=O)NC2(CNC(c3n(CC)ccc3)=O)CCC2)ccc2c(c1)COC2(C)C 42076,CC(C)C(CCN(C(=O)CCc1cncc(O)c1)C)NC(C1CC2CCC1O2)=O 42077,Cc1cc(C(=O)NCC=CCNC(c2ccc(SC(C)C)cc2)=O)nc(O)n1 42078,C12(NCC(C)CC3CC3)CCCN(C1)n1nnnc12.C(CC(F)(F)F)SCC 42079,c1(NC(=O)CC2CC(NCc3cc(Br)cnc3F)C2)cc2ccccc2cc1O 42080,c1(CC2(OC)CC2)ncccc1NC(=O)CNC(=O)C(F)(F)F.c12ccsc1C2 42081,C1(NC(c2n(CC)ccc2)=O)CCCN(C(=O)CCc2n[nH]c(=N)s2)CC1 42082,CC(CC(=O)NCC1(CN(C)C(c2sc(=N)[nH]c2C2CC2)=O)CC1)C(F)F 42083,C1(C(C(=O)NCC(C)(C2CC2)NC(=O)CC2(OC)CC2)OC)CCOCC1 42084,C(C(=O)C(C)(CC)CC)N1C(CS(=O)(=O)NCC)CCC1 42085,N1(C(c2c(COC)con2)=O)CCC2CN(C(C3(C(=O)OC)CC3)=O)CC2CC1 42086,C(CN=c1[nH]c(=NCc2ccc(S(C)(=O)=O)o2)[nH]c2c1CSC2)c1n(C)cnc1 42087,c1(C(=O)NC(CNC(C2C(C(=O)OCC)C2)=O)CC(C)C)cnc(SC)[nH]c1=N 42088,c1(C(N2CC(CC=C)(NC(=O)Cc3nnc(C)s3)C2)=O)cnnc(C2CC2)c1 42089,N1(C(C(CC)OCC)=O)CCN(C2CCN(C(=O)C=Cc3ccco3)CC2)CC1 42090,c1(C(N(CCNC(C2C(C#C)C2)=O)CCC)=O)cc(Br)c(Cl)cc1OC 42091,Cc1ccnc(C)c1C=O.c1(CC(N2CC(OCCC(=O)NC)C2)=O)cnn(CCF)c1 42092,c1(C(=O)NC2C=CCN(C(C(C)OCCC=C)=O)C2)nc2c(s1)COCC2 42093,c1(CNC(C2CC(C(C)NC(=O)C(F)C3CCC3)C2)=O)cnc(O)nc1O 42094,C(=O)(NNC(=O)C(N)C1CCCC1)NCCCCc1ccc(C)cc1 42095,N1(C(C2CC(C(C)C)C2)=O)CCCC(CCO)CC1.c12cn(nn1)C2 42096,c1(CNC(C2CC(CCC)C2)=O)cn(C2CCN(C(c3cnc(Cl)s3)=O)C2)nn1 42097,C(=O)(C(C)S(C)(=O)=O)N1C(C2CCCN(C(c3c(C)noc3C)=O)C2)CCCC1 42098,C1(C(N2CC(NC(C3C(C)CC3)=O)C(F)C2)=O)CC2(CCCO2)C1 42099,c1(C(=O)NCCC2(C)CCN(C(COC(C)=O)=O)C2)n[nH]c2ccccc12 42100,CCS(=O)(=O)C=CC(=O)NCC1CCN(C(=O)C(C)c2cccs2)CC1C 42101,C1(NC(c2cc(CC)on2)=O)CC2(C1)CC2NC(=O)C(O)C(C)C 42102,C(=O)(C(CC(F)F)c1ccccc1)OC(=O)OC1CC(=O)N(c2ccc(F)cc2)C1 42103,Cn1cc(OCC(N2CC(C)(NC(=O)CCc3cscn3)C2)=O)cn1 42104,CS(=O)(=O)C1CN(C(=O)C(CC2CCC2)NC(=O)CC2CCCSC2)C1 42105,c1(CN(CCC)C)ccc(C(N2CCCC(N(C(=O)C=CBr)C)C2)=O)cc1 42106,c1(OC)cnc(C(N2CC3C(CNC(=O)C=Cc4ccc(Cl)s4)C3C2)=O)c(F)c1 42107,c1(NC(c2scc(-c3c(OCCCC)scc3)c2)=O)cc2cn[nH]c2cc1OC 42108,c1(C(N2C(CNC(c3c(OC)ccs3)=O)CC2)=O)cc(C(F)(F)F)cc(O)c1 42109,C(C1CN(C(=O)CN2CC3CC3C2)CC1C(=O)NC1C2CCCCCC12)=CC 42110,c1(C(=O)NCC2CC(COC)CN2C(=O)Cc2cnsc2)cccn(C)c1=O 42111,CCCCCCCC(F)C(=O)N(CC(C)NC(=O)CC1(OC)CCCC1)CC 42112,N1(C(C=C(C)C(F)F)=O)CC(NC(c2n[nH]c3c2CCC3)=O)CC12CCCCC2 42113,C1(=CC(=O)CCN(C(CC2C(C(=O)OC)C2)=O)C)CCOCC1.C1CCN1 42114,N1(C(c2cc(COC)sc2)=O)CCCC1(C)CNC(=O)C#CC1CC1 42115,C1(C2CCCCC2)(C(=O)NC(CC(C)NC(c2cc(OC)no2)=O)C)CC1 42116,N1(CC(C)(C)NC(=O)OC(C)(C)C)CCC(NC(=O)CC2CCCO2)CC1 42117,c1(C(=O)NCCOCC(N2C(C=C)CC2)=O)cnn(C)c1C 42118,C1(OCC(=O)NC(C2CCCN2C(=O)C=Cc2c[nH]cn2)C)CC(F)(F)C1 42119,N1(C(C2(OCC)CC2)=O)CC2CCC(C1)N(C(=O)CCCN1CCOCC1)C2 42120,c1(CC(=O)NCC(CNC(=O)C=CC2CCCC2)OC)ccccc1SC 42121,Cc1c(-c2cn(CCCC(=O)N(CC(N)=O)C)nn2)c(=O)oc2ccc(O)cc12 42122,C(=O)(CCCCCCN=[N+]=[N-])NC1C(C)CN(C(=O)Cc2csnn2)CC1 42123,N1(C(C2C(O)CCN2C(c2cccc(O)c2)=O)=O)CCC2(CCCC2)C1 42124,c1(CNC(C(=O)NCc2c(C)cccc2)=O)ccc2c(c1)CC(C)O2 42125,c1(-c2cccc(C(=O)NC3CN(CC4CC(=O)NCC4)C3)c2)ncnc2[nH]cnc12 42126,N(C(=NCCN1CCOCC1)NCC1CCC(C)C1)CCC(=O)NC 42127,C#CC1(NC(=O)C(O)CCNC(c2cccc(=O)o2)=O)CCOC1 42128,N1(C(C(C=C)(C)O)=O)CCN(C(=O)C(n2nccc2C)C)CC(C)(C)C1 42129,C1(CNC(c2scc(C(C)=O)c2)=O)CCCN(C(=O)C(=O)NCCC(N)=O)C1 42130,CC(C)(C)C(CNC(=O)C=CC1CCC1)C(=O)NCCCCCCF 42131,c1(C(=O)NCC2(OCC)CCN(C(CCC)=O)CC2)coc2cc(F)ccc12 42132,C(=O)(C1=CC2(CN(C(c3cccs3)=O)C2)OC1)N1CCN(CC=C)CC1 42133,CCC(O)C(=O)N1CCC(N(C)C(c2cc(-c3ccc(Cl)s3)on2)=O)C1 42134,Cc1ccc(F)cc1C(N1CC2(CNC(C3CCC(C)(C)C3)=O)CC1CO2)=O 42135,C1(NC(C2C(NC(C(CC)(C)C)=O)COCC2)=O)CCCOC12CCC2 42136,C1(CNC(=O)C(F)(F)Cl)CC1N=c1[nH]c(-c2ccccc2)nc2ccccc12 42137,c1(NC(c2nnc3ncccn23)C)nccc(=NCCCN(C2CCC2)C)[nH]1 42138,C1(C(N2CCC(N(C(CCCC)=O)CC3CCCO3)CC2)=O)CN(C)CC(C)O1 42139,CN1CC(O)CC1(C)C(=O)NCC1CCCCN1C(C1CCCCC1)=O 42140,C1(C(=O)NCC(C2CC2)NC(C(C)(C)C2CC2)=O)CCC2(CC1)CNC(=O)C2 42141,C1(CCC(=O)NCC#CCOC)CCCCN1C(=O)CCOCCOC(C)C 42142,C1(NC(c2cnco2)=O)Cc2ccccc2N(C(c2cocn2)=O)C1 42143,c1(C(=O)NCC2CCCN(C(CC3C(C)(C)C3)=O)CC2)cc(O)cc(F)c1F 42144,N1(C(C(C)OCOC)=O)CCC(C(=O)N(C)Cc2cnnn2C)C(C)(C)C1 42145,N1(C(=O)Nc2cc(F)cc(OC)c2OC)CCc2cccc(Br)c2C1 42146,C1(NC(C2=NNC(=O)C2)=O)CCCCN(C(C2(F)CCOCC2)=O)CC1 42147,C1(OCC(C)C)CCCN(C(=O)CC2CCCC(C(=O)O)C2)C1 42148,c1(C(N2C(CC(=O)Nc3cncc(C)c3)COCC2)=O)n[nH]c2ccc(F)cc12 42149,c1(C(N(CCCc2cn(CC3CCCCN3C)nn2)C)=O)ccc(Br)c(Cl)c1 42150,c1(CC)nn(C)cc1C(=O)NC(C)(C)CC(=O)NCC(O)C(F)(F)F 42151,CCC(C)(CCC(C)C)C(=O)NCCC1CC(NC(C2CCNC(=O)C2)=O)C1 42152,c1(C(=O)NC2CC(CNC(C3C(CC)OCC3)=O)C2)cc(C)cc2c[nH]nc12 42153,C1(NC(c2n(C(C)C)ncc2)=O)C2CCC1CN(C(c1ccc(F)cc1Br)=O)C2 42154,c1(C(N2CCC3(CCN(C(CCC=C=C)=O)C3)C2)=O)ccc2c(c1)C(=O)NC2=O 42155,Cc1cc(C(N2CCCC2CCNC(=O)CS(=O)(=O)N(C)C)=O)nc(O)n1 42156,CC(CC(=O)NC1CCCC1NC(C1(CF)CC1)=O)n1cc(Br)cn1 42157,O=C(COc1ccc(-c2ccc(CO)cc2)cn1)NNc1ccc(Br)cn1 42158,Cc1ccc(OCC(N2CCC(NC(C34CC(CSC)(CO3)C4)=O)C2)=O)c(C)c1 42159,Cc1cc2[nH]c(C(N3CC4(CC(NC(c5snc(Cl)c5Cl)=O)CO4)C3)=O)cc2s1 42160,c1(N2CC(NC(C=C(C)Cl)=O)CC3(C2)CC3)nc2cc(F)ccc2o1 42161,c1(C(OC)OC)ccc(C(=O)NCC2(O)CCCSC2)cc1 42162,CCCC(CC)C(=O)NC1CCOC1C1CCN(C(c2cc(C3CC3)on2)=O)CC1 42163,C(=O)(C(F)C(F)(F)F)NC(CC)CNC(=O)COCc1ccncc1 42164,CC1(C)CC(NC(=O)C(C)(O)Cc2ccccc2)CCN(Cc2sccc2Br)C1 42165,Cc1nc(C(=O)NCC2(C)CCN(C(=O)Cc3cnc(C)s3)C2)c2ccnc-2[nH]1 42166,c1(N2CCN(C(=O)Nc3cccc(F)c3)C3C2C3)ncnc2sccc12 42167,C1(NC(C(COC)OC)=O)CN(C(c2ccccc2OC(F)(F)F)=O)CCC1O 42168,C12(CC(=O)NCC3(F)CC(CNC(c4ncccn4)=O)C3)CCC(CC1)OC2 42169,c1(C(=O)NC2CC(CNC(C(CCC)C)=O)C2)ccc2nc(O)cn2c1 42170,c1(C(=O)NCC(C)(C(C)C)NC(C=CSC)=O)cc2c(cn1)COCC2 42171,c1(OC)cc(OC)c(CN2CC3CC(CF)C3C2)c(OC)c1 42172,C1(C(=O)NC(C)CNC(c2cn(C)nc2-c2cccs2)=O)CCOC(=O)CC1 42173,CC(C(=O)NCC1(F)CN(C(c2ccc(SC(F)(F)F)s2)=O)C1)S(N)(=O)=O 42174,c1(C(N2CC(OCC)(CNC(=O)CCC3CC3(F)F)C2)=O)cccc2c1COC2 42175,N1(C(CC2CC(=O)C2)=O)C2CCCC1CC(NC(C13CSC(C1)C3)=O)C2 42176,c1(C(N2CCC(OC3CCC3)C2)C(=O)NCCCOC)nccc(Br)c1C 42177,C1(NC(N(CC(c2ccccc2)C)C)=O)CC(C)(C)C12CC2 42178,CCCCC(O)CC(=O)N1CCCC(NC(=O)Cc2c(F)cccc2F)C1 42179,C1(CNC(CCC#C)=O)CC(F)(F)CN1C(=O)C=Cc1scnc1C 42180,Cn1oc(C(=O)NCCC2CCN(C(=O)COCC3CCC3)C2)cc1=O 42181,N1(C(Cn2c(C)cc(C)n2)=O)CC(C)N(C(c2nnn3c2CSCC3)=O)CC1C 42182,C(=O)(C#CC1CCCCC1)NC(CC=C)CC(=O)NC1CC(CO)C12CCC2 42183,C1(C(=O)NCc2c(C(=O)NC(C3CCCO3)CC)nco2)(CC)CCCC1O 42184,n1(C(C)(C)C)ccc(C(=O)NC2(CNC(=O)CCC3CCC(=O)N3)CCC2)n1 42185,Cc1ccc(C(=O)NC2(C(=O)NCc3cc(O)ns3)CCCC2C)c(O)n1 42186,C1(C(=O)NC(CC=C)CC)CCN(C(C2CC(=O)C2)=O)C12CC2 42187,NS(=O)(=O)C1CN(C(=O)NC2CC(C#N)C2)C2(CCC2)C1 42188,CC1CC2CN(C(c3cnc4[nH]cncc3-4)=O)CC2N1C(=O)Cn1cnnc1O 42189,C1(C)(C(=O)NC(C#C)C2CCC2)CCN(C(=O)CC2CCC=CCC2)C1 42190,c1(NC(C)=O)cccc(Cl)c1NC(C1CCCN1Cc1csc(C)n1)=O 42191,c1(CC(=O)NC2CCN(Cc3cn(C(CC)(C)C)nn3)C2)c(F)cc(Br)cc1F 42192,c1(C(=O)NCC(C2CC2)NC(=O)Cc2cnns2)ccc2c(O)nnc(O)c2c1 42193,C(CC(=O)NCCCN1CC=CC1)(C(F)F)NC(C(CC)OC)=O 42194,c1(CC)cccc(C(F)(F)F)c1S(=O)(=O)NC1(C2CCCO2)CCOCC1 42195,C1(N(C(=O)Cc2ccnn2C)CC#C)CCN(C(=O)C=CCN(CC)CC)CC1 42196,C(=O)(CCCC(F)(F)CO)NCCOCCCNC(C1C(C)OC(=O)N1)=O 42197,CCC(CNC(=O)C(C)NC(C1(OC)CC1)=O)(CC)OC 42198,c1(CSC)cc(C(=O)NC2CC23CCN(C(=O)CC2CCCCO2)C3)ccc1F 42199,C(C1c2ccsc2CCN1C(C1CCSCC1)=O)NC(C1C(OCC)C1)=O 42200,c1(OC)ccc(CN2CCN(C(=O)CCc3ccc(C)nc3)C(CO)C2)nc1Cl 42201,c1(CC(=O)NCC2(CNC(c3cnoc3C3CC3)=O)CC2)cccc2ccoc12 42202,C1(CC(=O)NC2CC=C(C)CC2)N(C(c2csc(C)c2)=O)CCC1(C)C 42203,N1(C(c2c(C)n[nH]c2)=O)Cc2cccc(CNC(c3cc(F)ccc3Cl)=O)c2C1 42204,Cc1c(C(N2CCC(CC(=O)NOCCC(F)(F)F)C2)=O)occc1=O 42205,C(=O)(C(c1cccs1)NC(=O)C(C)N1CC(C)C1)NCC(=O)OCC 42206,N1(CC(C)C)CCCC(C(=O)NCC(C)(CO)NC(c2cccc(CO)c2)=O)C1 42207,C1(NC(C2C(C)CCN2C(C2C3CCCC23)=O)=O)CC2(C1)CC(C)(C)C2 42208,C(C(F)(F)CCC(=O)NC(CN(C)C)CC1CC1)n1cc(-c2nc(C)oc2C)nn1 42209,c1(C(=O)NCC(C)NC(c2c(CC)ncs2)=O)cc[n+]([O-])cc1 42210,N1(C(c2cnn(CC)c2Br)=O)CCC(NC(=O)Cn2ccc(C)n2)CC1C 42211,C12(C(=O)NCCOCC=C)COCC1CN(C(=O)COC(C)=O)C2 42212,C(CCCCCNC(=O)CC12CCCC1C2)NC(CCCSC)=O 42213,c1(C(N(CCC)CCNC(C2CC2C)=O)=O)snnc1-c1ccccc1 42214,C(=O)(C(C)(C)C(C)C)NCCN(CCC)C(c1sc(C2CCOC2)nc1C)=O 42215,c1(C(N(CCNC(=O)C(C)C(F)F)CC)=O)cnn2c(N)cc(C)nc12 42216,C1(C(=O)Oc2cccc(COC)c2)CC1C1CCN(C(=O)NCC)C1 42217,C1(=O)C(O)CCCC2C(CC2O)N1.c1(-c2cn(CCOC)nn2)cnn(C)c1N 42218,N1(Cc2cc(C)sc2C)CC(C)C(CN)C(C)C1 42219,N1(C(c2n(C)nc(C3CCC3)c2)=O)CCCC(CNC(c2c[nH]c(=N)s2)=O)CC1 42220,c1(-c2nnc(N(CCCC)C)n2CC(C)OC)cc(Cl)ccc1OCC 42221,Cc1cc(NC(C2CSCCN2C(c2ccc([N+](=O)[O-])cc2)=O)=O)c(C)cc1Cl 42222,N1(C(CCC#C)=O)CCCN(C(=O)C(O)Cc2ccccc2)CC1CO 42223,C(=O)(C1=CC2(CCOC2)C1)N(C1CN(C(c2c(C)nc(O)cc2)=O)CC1(C)C)C 42224,C(=O)(C1=CCCOCC1)N1CCCC(CC)(NC(=O)Cc2c(C)cccc2F)C1 42225,c1(-c2nc(CS(CC)(=O)=O)nn2C)cc(C)cc(F)c1 42226,C=CC1(CC(=O)N(CCO)CC2CC2)CN(C(=O)C(C)(C)n2cncn2)C1 42227,C1(CC)CN(C(c2cc(Cl)cnc2C)=O)CCN1C(c1ccc(C)o1)=O 42228,Cn1nc(CO)cc1CC(=O)Nc1cccc(NC(c2cc(C3CC3)no2)=O)c1 42229,CC(CC1CCCC1)C(=O)NCC1OCCC1C(=O)NC(C)C(=O)OC(C)C 42230,N1(C(C(N(C(=O)CCCC2CCCO2)C)C2CC2)=O)CCC12CCCC2 42231,N1(C(c2n(C)nc(O)c2)=O)CCC2(CCC2)C(NC(C2(CO)CCOCC2)=O)C1 42232,C1(OC(c2scc(C(=O)OC)n2)=O)Cc2ccccc2C1C#N 42233,Cc1cc(C)c2cc(C(N3CC(NC(c4ncccn4)=O)CC3(C)C)=O)sc2n1 42234,C=CC(C)(CCOC)C(=O)N(CCCNC(=O)C(C)C(=O)OC)C(C)C 42235,c1(OC)cc(F)c(C(=O)NCC2CC(C)N(C(C3CC(CF)C3)=O)C2)cc1N 42236,C1(C)(C(N2CCCC(N(C(=O)CSC(C)C)CC)C2)=O)CCC(C)C1(C)C 42237,c1(C(=O)NCC(CCC)NC(=O)Cc2ncc(Cl)s2)nccc(C)c1N 42238,C1(C(N(C2CCCC(C)(C)C2)C)=O)CC(C)CN(C(c2cc[nH]c2)=O)C1 42239,O=C1CC2CC(C(N3CCC3CNC(=O)CCC3CCOCC3)=O)C1O2 42240,Cc1nc(O)nc(O)c1CC(N1CCN(c2ccc(C#N)nn2)CC(O)C1)=O 42241,c1(CC)cc(C)c(C(=O)N(C2CN(C(=O)Cn3cc(CO)nn3)C2)C)o1 42242,Cc1nocc1CC(=O)NCC1(C2CCCN2C(=O)COCC2CCC2)CC1 42243,C1(NC(CCOCCOC)=O)CC2CCC1N2C(=O)CC1CCCCC1(C)C 42244,C(=O)(C(C(C)(C)C)n1ccnn1)NC1(CCCNC(C2(CCCC)CC2)=O)CC1 42245,C1(NC(C(C)=C(C)C)=O)CCN(C(=O)CCOCC2CC2)CC12CCC2 42246,S(=O)(=O)(c1cccnc1C(=O)NCC1CCC(CO)O1)N(CCCS(N)(=O)=O)C 42247,c1(CC)ccc(F)c(C(=O)NCC2CN(C(=O)CC3CCCC3)CCCO2)c1F 42248,C=CC1(C(=O)NCCOCC(C)(C)O)CCN(C(c2ccc(F)s2)=O)C1 42249,C(CC1=CCN(C(C23CCC(O)(CC2)CC3)=O)CC1)NC(C1(C)CC1(F)Cl)=O 42250,C1(C(=O)NCC2(F)CC(CNC(COCC=C)=O)C2)Cc2ccc(F)cc2O1 42251,C1(C)(CC(=O)NC)CCC(=O)N1.N1(CC(=O)N(C(C)CN)CC)CCC(OC)CC1 42252,c1(C(N(CCN(C(c2nnn(C)n2)=O)CC)CC)=O)cc([N+](=O)[O-])n[nH]1 42253,C1(C(=O)NCC2CC(OC)CN2C(=O)C(=O)NC(C)C)C2CCC1(C)C2(C)C 42254,c1(C(N2CC(CCC)C(NC(=O)C(F)n3ccnc3)C2)=O)cc(C)cc(C)c1 42255,N1(C(CN(S(C)(=O)=O)C)=O)CC2CC(NC(C3(CC#N)COC3)=O)C(C2)C1 42256,N1(C(CCC=CCC=C)=O)CCOCC1C(N1CCCC(COC)C1)=O 42257,CCC(C)(C)C(=O)NCC1CC(NC(c2ccn(C)n2)=O)CC1O 42258,c1(C(N2CCCC(Cn3cc(C(CC)(C)O)nn3)C2)=O)c(C)[nH]c2ncccc12 42259,C1(C(=O)NCC(C=C)O)CC2CC1CN(C(=O)CCn1ccnn1)C2 42260,CC1CN(C(c2csc(F)c2)=O)C(C)CN1C(c1ccnn1CC(F)F)=O 42261,CCCC(CNC(=O)C=CC(C)CC)C(=O)N1CC(N2CC(O)C2)C1 42262,C1(CNC(c2c(OC)noc2C)=O)CC(C)CN(C(=O)CN2CCNC2=O)C1 42263,N1(CC(=O)NC(C(=O)N(CCC(=O)OC)C(C)C)(C)C)CCC(F)CC1 42264,CCC(C)(C)CCNC(=O)CCC1CCCN1C(=O)C=CCOC1CC1 42265,CN1CCCC(C(=O)N(CCCNC(C2CSCCS2)=O)CCO)C1 42266,C(=O)(CCCCCCCSC)NC1C(NC(c2cccc(CC)n2)=O)CCC1 42267,N1(C(C(C)NC(=O)NC)=O)CCC2(CC1)CC(C)N(C(=O)CC1(COC)CC1)C2 42268,c1(COCC(=O)NC2(C)CC(NC(C3CCCCO3)=O)C2)cccc(C(N)=O)c1 42269,N1(C(c2c(=O)ccn(C)c2)=O)CC2CCC(C1)C2CNC(c1c[nH]c(C#N)c1)=O 42270,c1(NC(=O)Nc2ncn(C)n2)cc(F)ccc1C(N1CCC(CO)C1)=O 42271,N1(C(C=CCOCCOC)=O)CC(C)(C(=O)NC2CCCO2)C1 42272,c1(C(=O)NCC2C(NC(Cc3c(C)ncs3)=O)C2)ccn2ccccc12 42273,C1(C2(O)CN(C(C3CC=CC(O)C3)=O)C2)(CNC(C2CN(C)C(=O)C2)=O)CC1 42274,C#Cc1cccc(CC(N2CCC(OCC(=O)NC3CC4(CC4)C3)C2)=O)c1 42275,N1(C(c2c(C)nc(O)cc2)=O)CC2(C(=O)NC(C)C(F)F)CC1CCO2 42276,C1(C(N(C2CC(OC)C2)C)=O)CC2CC2N1C(=O)CCc1cn[nH]c1 42277,N1(CCC)CCC(C(=O)NC2CCC(CC(=O)N(C3CCOC3C)C(C)C)C2)C1 42278,CC#CCCC(=O)N1CCCCC1CCCNC(=O)C(O)Cc1ccc(F)cc1 42279,C(=O)(C(C)C(O)CCCC)N(CCNC(c1cccc(C#C)c1F)=O)CC 42280,n1(CCCNC(c2cccc3c2CNC3)=O)cnc2ccccc2c1=O 42281,Cc1ccc(C(=O)NC2CC3CN(C(=O)CN4CCCC4)C2C3)nc1Cl 42282,C(CC(C)C)(C(=O)N(C)CC1CCCN1Cc1cncn1C)NC(C)=O 42283,C1(C(=O)OC)C(F)(F)C12CC(C(=O)NC(C)(CNC(c1cc[nH]n1)=O)CO)C2 42284,c1(C(N(CC(CC)NC(c2n[nH]c(C)c2Cl)=O)CC)=O)ccc2nncn2c1 42285,c1(NC(C2N(C(c3c(CCC)nco3)=O)CCC2)=O)c(C)cc(C)cc1C 42286,C12CCCN(C1)C(=O)c1cnnn12.c1(CC)cscc1OC 42287,S(=O)(=O)(c1ccc(C#N)cc1Cl)Nc1c(F)ccc(OC)c1 42288,C(=O)(C(CC)C(=O)NCC=CCNC1(CNC(c2ccnn2C2CC2)=O)CC1)OC 42289,c1(NC(N2CC(CC)(OC)C2)=O)nn(C)c(C)c1S(N)(=O)=O 42290,C1(C(=O)NCC2C(C)(C)COC2)CCC2(CC2)N1C(c1cc(C2CC2)no1)=O 42291,N1(C(=O)COC2CC2)CCC2(CCN(C(c3cc(Cl)c[nH]3)=O)C2)C1 42292,n1(CC)c(C(=O)NC2CN(C(C)C)C2)cnc1O.N12CC(C)C1C2=O 42293,C1(C(=O)NCC2CCN2C(c2csc(Cl)n2)=O)CC1C1CCC1 42294,c1(NC(CCC)CC)cc(=NC2CCCN(S(=O)(=O)N(C)C)C2)[nH]c(COC)n1 42295,N1(C(C(F)=CCC)=O)CCC(C)C(NC(=O)CCC2(C#N)CCC2)C1 42296,C(=O)(C#CC1CCCO1)N1CC(NC(c2ccc(OC)s2)=O)C(SC)C1 42297,Cc1ncn(C)c(=O)c1C(=O)NCCN(C(=O)CN(C1CCC1)C)C(C)C 42298,C(=O)(C(CC(C)(C)C)OC)NC1(CC=C)CCC1.C1(=O)CCC2(CCC2)N1 42299,N1(C(C(C)C(F)F)=O)CC(NC(=O)CN2CCCNC2=O)C(S(C)(=O)=O)C1 42300,Cc1nn(C)cc1Cc1noc(C2C3CC(=O)CC23)n1 42301,c1(C(=O)NC2(CC)CN(C(CSCC)=O)C2)cc(NC)nc(Cl)c1 42302,c1(CNC(C(CNC(=O)CC2CCCN2C)OC)=O)cnccc1Cl 42303,CCC(C)C(C)C(=O)N1CC(CF)(NC(c2n[nH]cc2Cl)=O)C1 42304,C(=O)(C(CN(C)C)NC(=O)CC1CCCN1C)NCCC1(OCC)CCC1 42305,C1(C(N2CC(NC(Cn3ccc(C)n3)=O)C(C)C2)=O)CC(C)(C)OC(C)(C)C1 42306,Cc1cnccc1C(C)C(=O)NCC(C)(O)CNC(=O)CCc1cccnc1 42307,CCN=C(NCc1ncc(Cl)n1C)N1CCOC(CF)C1 42308,C1(NC(c2on(C)c(=O)c2)=O)CCN(C(=O)COC2CCCCC2)CC1F 42309,C(=O)(C(CCNC(N)=O)OC)N1CCC(N(CCC)C(c2ccc(F)s2)=O)C1 42310,c1(C(=O)NCC(CC)N(C(=O)CC(C)SC)C)cccc2c(C#N)c[nH]c12 42311,N1(C(COC)=O)CCC2CN(S(=O)(=O)c3cnc(OC)s3)CC2C1 42312,c1(CN2CCCC(CN(S(=O)(=O)CC3CCCC3)C)C2)c[nH]c2cccnc12 42313,C#Cc1c[nH]nc1C(=O)NC(C)CC1CN(C(c2cnc(C3CC3)s2)=O)C1 42314,C=C(Br)CN=C(NCc1ccc(SC)cc1)NC(C)C 42315,c1(CN(C)C)cccc(-c2cnc(NC(=O)NCCc3nccn3C)[nH]2)c1 42316,C1(CC(=O)OCC(=O)Nc2csnc2C)(COC)CCOCC1 42317,c1(C(N2CCC(OCCNC(C3OCCN(C)C3)=O)C2)=O)nc[nH]c2ncnc1-2 42318,CC(=O)CCCCCCC(=O)N1CCN(C(C2CC3CC3C2)=O)CCC1C 42319,CC12CCC(C(N3C4CCC3C(=O)NC4)=O)(CC1)NC2 42320,N1(C(C)C)C(=O)CCC1C(=O)NCC(C)(C1CCC1)NC(=O)CC1CCCCO1 42321,C1(CC)CN(C(c2ccccc2SC)=O)CCN1C(c1cc2[nH]ccc2s1)=O 42322,C1(NC(=O)C=Cc2ccsc2)CC2C1CCN2C(=O)Cc1csc(C(F)(F)F)n1 42323,N1(C(C(CC)N(C)C)=O)CC2(CCN(C(=O)Cn3ncnn3)CC2)C2COCC12 42324,C1(C)(C(N2CCC(NCc3snc(CC)n3)C2)=O)CCC(O)CC1 42325,C1(NC(CN(S(C)(=O)=O)C)=O)CN(C(C2CC23CCSCC3)=O)CC1C1CC1 42326,Cc1nsc(C)c1C(=O)NCc1cc(C(N2CCCCC2CC(N)=O)=O)nn1C 42327,C(c1cc(F)cc(F)c1)=CC(N1CCN(C(C2CC2F)=O)C(CC2CC2)C1)=O 42328,CN1CC(CNC(c2ccc(CNC(=O)CNC=O)o2)=O)CC1=O 42329,C1(C)(CC)C=C(C(=O)Nc2csc(-c3cnc[nH]3)n2)C1 42330,c1(C(N(CCOCCCNC(C(C2CCC2)SC)=O)C)=O)cc2ccnn2cn1 42331,c1(OC)cc(CN(C(C(=O)NC2(C)CC2)C2CCOC2)C2CC2)cc(F)c1OC 42332,N1(C(C(CC2CC2)OC)=O)CCCCC1C1(NC(=O)CCC(C)SC)CC1 42333,N1(C(c2n(CC)nnc2)=O)CCC2(CCC2NC(c2cccc(F)c2C)=O)CC1 42334,C1(C(N(C(CCNC(C2(NC(C)=O)CCCC2)=O)C)C)=O)CCS(=O)(=O)C1 42335,C=C=CC(C)C(=O)NCCOCCOCCNC(C1(C#N)CC(C)C1)=O 42336,N1(CC(=O)NCC(CC)NC(C2CC2c2nccs2)=O)CCCCCC1=O 42337,c1(C2(C)CC(NC(C(c3ccccc3F)OC)=O)C2)cccc(Cl)c1 42338,c1(SCCNC(NCc2n(C)cnn2)=NCC2CCCCO2)c(F)cccc1F 42339,C1(CC)CCCCC1OCC(=O)NCCC1CCN(C(=O)C=C2CCC2)C1 42340,C12(C(=O)NCC(CC(=O)OC)O)CCCC1CCN2C(=O)C(C)C(C)(C)C 42341,c1(SCC(N2C(C)C(NC(C3CN(C)C3)=O)CC2)=O)ccc(C#N)cc1 42342,C1(C(=O)NC(C(=O)NC2CCOCC2)c2ccoc2)Cc2nccn2C1 42343,n1(Cc2cc(C)c(OC(F)F)cc2)nc(C(F)F)c2c1CCC2 42344,c12cc(Br)c(cc1O)CN2C(c1cc2cccn2cn1)=O.C(C(C)OC)OC 42345,C1(NC(c2cccc(C#C)c2)=O)CN(C(=O)C(C)SC(F)(F)F)CC12CCC2 42346,c1(C(=O)NCC(CNC(c2nc(OC)c(F)cn2)=O)C)c(F)cc(N)cc1F 42347,N1(C(C(C(CNC(C2(CC)CCC2)=O)C)F)=O)CC(O)(C2CCC2)C1 42348,N1(C(c2c(OC)scc2)=O)CCC(C(=O)Nc2ccc(C)nc2)C1(C)C 42349,C=C1CN2C(=O)CCC2(C(N2CC(C)(NC(=O)CC(C)n3cccn3)C2)=O)C1 42350,Cc1cccc2c(C(N3CC4CC4(NC(c4c(Cl)cnn4C)=O)C3)=O)cccc12 42351,N1(C(c2c(C)cnn2C)=O)CC2(CC(CC(=O)NCC(C)(O)CO)C2)C1 42352,c1(CC(=O)N(C)CC2N(C(CC(=C=C)C)=O)CC(F)C2)cc(C)ccc1F 42353,c1(C(=O)NC(C2CCCCC2)CNC(C(CC)(C)CO)=O)onc2ccccc12 42354,N1(C(CC(=O)OC)=O)CCC(CCC(=O)NCc2nccn2C(C)C)CC1 42355,C1(OC)CCCC(CF)C1.C12CC(NC(=O)OC(C)(C)C)(C1)C(=O)N2 42356,CCCC1Cc2c([nH]c(=N)s2)NC(C)C2(O)CCN(C1=O)CC2.C(C)(=O)NC 42357,CC12CCN(CC1)CC2NC(c1cc(CNC(c2c(F)cncc2F)=O)[nH]n1)=O 42358,C1(S(C)(=O)=O)(C(N2CCN(C(c3c(C)ccc(C)n3)=O)C(CO)C2)=O)CC(O)C1 42359,N1(CC)CCCC(CC(=O)NCCOCCCNC(c2cnc(C)[nH]2)=O)C1.C=C 42360,N1(C(C=CC=CC)=O)CCC2CC12C(=O)N(CC)Cc1cnn[nH]1 42361,c1(C(N2CCC(Cc3ccc(I)cc3)CC2)C(=O)NCC)cccc(C(F)F)c1 42362,N1(C(C2N(C(N)=O)CC2)=O)CCC(C)(CCOCC)C1.c12ccc(cc1)[nH]c2=O 42363,C1(N(CC(=O)OC(C)(C)C)C)CCCN(C(=O)CNC(c2cccnc2)=O)CC1 42364,C(=O)(CC(C(F)F)c1ccccc1F)NC(CNC(C=C(CC)CC)=O)C1CC1 42365,c1(COC)nc(N2CCCC(NC(C3(O)CCC(C)C3)=O)CC2)cc(Cl)n1 42366,N1(C(C(F)=CC)=O)CC(C)CCC1CNC(C1CC(OC)C1)=O 42367,c1(C(=O)NC(CC=C)CNC(c2c(Cl)sc(Cl)c2C)=O)cccc2nonc12 42368,c1(C(N(CC(CNC(C2(OC)CCSC2)=O)O)C)=O)ccc(C)c2cccnc12 42369,c1(CCC(N2CC(OC)(CNC(C34CC(CO3)C4)=O)C2)=O)cccc(F)c1Cl 42370,c1(C(=O)NCC(C)(C)NC(C(C(=O)OCC)F)=O)ccc2c(c1)COCCN2 42371,C=CC1(C(N2CC(C(=O)NCc3coc(C)c3)C(F)(F)C2)=O)CCCCC1 42372,COn1cnc(C)c1C(=O)NCC(C)NC(c1sc(Br)cc1C)=O 42373,C1(CC(=O)N(CC(=O)NC(C)CN(C)C)C)(NC(C)=O)CC1 42374,c1(C(=O)NC(CC)(CNC(C2(CO)CC2(F)F)=O)CC)cnc2c[nH]nc2c1 42375,Cc1nc(C(C)C)sc1C(=O)N(C)CCN(C(=O)COc1ccsc1)C(C)C 42376,c1(C(=O)NC(CN(C(=O)C(O)Cn2cncn2)CC)C)csc(COC)n1 42377,N1(C(c2nc(C)c(C)s2)=O)C2CCC1CC(n1cc(C34CCC(F)(CC3)C4)nn1)C2 42378,C1(C(N(CC(CC)NC(C2CCCOC2)=O)CC)=O)CCOC1C(C)C 42379,Cc1ncc(C(N2CCC(C(C)(C)C)(CNC(=O)C#CC(C)(C)C)C2)=O)cc1N 42380,Cc1cc(C(=O)NC2CC(O)CN(C(=O)COc3cccnc3)C2)c(F)cc1N 42381,c1(C(N2C(CNC(C(C3CC3)OCC)=O)C=CC2)=O)cc(F)c(C)cc1N 42382,C12(C(=O)N)CCCC1CN(C(=O)C1CC1)C2.N1(C(=O)NCC(=O)NC)CCOCC1 42383,n1(C(C)C)nc2c(c1C(N1CCCC(C(N3CCCCC3)=O)C1)=O)CCC2 42384,C(C(=O)N(C(C)CN(C(=O)Cc1ccc(F)cc1)C)C)(C(C)C)NC(C)=O 42385,C(=O)(C(C)(C)CC(C)C)NCCOCCCNC(C(CC)(O)c1ccccc1)=O 42386,N1(C(C=COCC)=O)CCC(CCCOC)(C(=O)N(C)CCn2cnnc2)CC1 42387,CC1(NC(C2CCC(P(C)(C)=O)C2)=O)CCCc2ccccc21 42388,c1(-c2cc(C(=O)NC)n[nH]2)ccc(C(=O)NCCCC2CCC(=O)CC2)cc1 42389,Cc1cc(O)cc(=O)n1CC(=O)NCC1CC(NC(=O)CCC2CCC(=O)N2)C1 42390,C(CC(=O)NCC1CCOC1(C)C)(CC(C)C)NC(C1C(CCC)C1)=O 42391,CCC(CC(=O)NCC(C(C)C)NC(=O)C(CO)C(C)(C)C)CC(C)C 42392,C1(OC)(OC)CC(C)(NC(CN(c2ccccc2C)C2CC(F)(F)C2)=O)C1 42393,N1(C(CN2CCN(C)CC2)=O)CCC2CN(C(=O)C(C)(C)c3sccc3Cl)CC12 42394,c1(CCNC(C(C=C)(C)C)c2nnnn2C(C)C)cccc2oc(C)nc12 42395,Cc1ccccc1COCC(=O)NC1C2CC1N(C(C1(C)CC(C)C1)=O)C2 42396,N1(C(C2(OC)CCC2)=O)CCC2C(CCN2C(c2cc(C)ncc2Cl)=O)C1 42397,Cc1cc(C(N2CC(C(=O)NCCSC(F)F)CCC2C)=O)nnc1C 42398,Cc1c(C(N2CCOCC(CNC(=O)COCCN(C)C)C2)=O)cccc1F 42399,c1(C(=O)OC)cc(NC2CCCN(Cc3ccccc3)C2)cc(F)c1F 42400,N1(C(c2cc(C(C)C)no2)=O)CCCC(NC(=O)C(O)CC2CCCCC2)CC1 42401,C(=O)(N=S1(=O)CCCC1C)NC(c1cc(N(C)C)ccc1O)C 42402,c1(CN2CC3C(C(=O)Nc4cc(N5CCC5)ccn4)C3C2)ccc2ncnn2c1 42403,CCCCC(CNC(=O)C(CC)OC1CCCC1)NC(C1CC(F)C(=O)N1)=O 42404,c1(C(=O)NC2C(CNC(c3cc(O)ccc3Cl)=O)CC2)ccn2cccc2c1 42405,N(C1CN(C(=O)C(C)c2ncco2)Cc2ccccc21)C(c1c(C)nc[nH]1)=O 42406,C1(NC(C2CC(C#N)C2)=O)CCCC(C(N2CCSCC2C2CC2)=O)CC1 42407,N1(C(CCC(=C)Cl)=O)CCC2(CC1)CC2CNC(c1cnc(OC)s1)=O 42408,C1(N(C(=O)C(F)F)CC#C)CCN(C(C2(C(C)(F)F)CC2)=O)CC1 42409,N(C1CN(C(C2(C)CC=CC2)=O)Cc2ccccc21)C(c1cc(C)[nH]n1)=O 42410,C1(c2cn(CCNC(c3ccncc3F)=O)nn2)CC2CCC1O2 42411,c1(C(=O)NC(CC)(C)C(=O)NC(CCOC)C(C)(C)C)cc(C)cc2nc[nH]c12 42412,c1(NCC2(CNC(C(C)SCCOCCOC)=O)CCC2)c(C)cccc1F 42413,CC1CN(C(=O)Cc2n[nH]cc2Br)CCC1NC(=O)CSCC(N)=O 42414,C1(C(N(C(C)C2CC2)C)=O)CCCN(C(c2ccncc2SC2CC2)=O)C1 42415,CC1CC(C)(C(=O)N(CCCCN(C)C(c2csc(Cl)c2)=O)C)CC(C)O1 42416,CC(C)(C(=O)NC12CC1CN(C(=O)CCOc1cc(Cl)cc(Cl)c1)C2)C(F)F 42417,c1(CNC(C2(C)CC(NC(CCc3nc(C)sc3)=O)C2)=O)ccnnc1O 42418,c1(OC)ccc(C(N2CCC(CNC(=O)CC(C)OC)(OC)C2)=O)cc1F 42419,c1(NC(CCOCC)=O)cccc(NC(c2snnc2C(C)C)=O)c1 42420,N1(C(CC(C)(C)OC)=O)C2CCC1CN(C(c1cnoc1C)=O)CC2 42421,C1(CNC(CC2CC(=C)C2)=O)CC(NC(c2coc(SC)c2)=O)C1(C)C 42422,C(=O)(C(C)CC(N)=O)N1CCCC(NC(c2c(C)c(C(F)(F)F)[nH]n2)=O)C1 42423,N1(C(C(C)C2CCOC2)=O)CC2CC1CC2CNC(=O)C(C)(C)c1cnn(C)c1 42424,c1(C(=O)NCC23OCC(NC(C=Cc4ccc(C)o4)=O)(C2)C3)cc(F)cnc1O 42425,N1(C(CC2C(C)=NNC2=O)=O)CC2CCOC2(CNC(=O)CCC2OCCO2)C1 42426,c1(OC)cc(C)nc(N(C)CCC2CCN(C(=O)CC(C)N(C)C)CC2)n1 42427,C1(C(C)C)C(NC(=O)CSc2cccc(F)c2)CCN1C(=O)CC(F)F 42428,C1(c2n(CCC)nnn2)(NCCCC2CCOC2)CCC2(CCOCC2)C1 42429,Cc1cccc2cc(C(=O)NC3(CNC(C45CCC4C5)=O)CCOCC3)nn12 42430,c1(C(=O)NC(C(C)C)CNC(c2nn(C)cc2Cl)=O)n[nH]c2c1CCCCC2 42431,c1(OCC)ccccc1C(N1CCC(C)(C(=O)NCc2ccnc(Cl)c2)C1)=O 42432,CC(=O)CCCC(=O)NC1(C2CCCCN2C(=O)CCc2cccnc2)CC1 42433,c1(OCC(=O)NCCN(C(=O)CN2CCC2C)C(C)C)ccc2c(c1)CCC2 42434,CCC(C)C(O)C(=O)NCC1(CNC(=O)C(C)(O)C(C)C)CC1 42435,C1(N(C)C(=O)OC2CCOCC2)CCN(C2CCN(C(C3CC4CC4C3)=O)C2)CC1 42436,C(=O)(CS(=O)(=O)CC(C)C)NC1C(OC)CN(C(=O)C(C)Sc2ccc(C)n2C)C1 42437,N1(C(c2c(C)n(C3CC3)nc2)=O)CC2CCC(C1)N2C(c1cnn2c1OCC2)=O 42438,C1(C)(C(N(c2ccn(C)n2)CC)=O)CCN(C(=O)CCc2ccc[nH]2)C1 42439,c1(C(=O)NCC(C)NC(C2(C)CNC(=O)C2)=O)ccc2c(Br)nn(C)c2c1 42440,C#CC1(O)CCN(C(C)C(=O)N(CC(C)NC(C2C3C4CCC(C4)C23)=O)C)CC1 42441,C1(CNC(CCc2cc(C)no2)=O)N(C(c2csnc2C)=O)CCC1(C)C 42442,C1(NC(Cn2cc(CC(NOC)=O)nn2)=O)C(=O)OCC1(C)C 42443,C(C)(C)(CC(C)NC(C1(NC(=O)C(=Cc2ccco2)C)CCCC1C)=O)OC 42444,C1(C(N2C(CNC(C(CC)(C)COC)=O)CC3(CC3)C2)=O)CCc2ncccc2C1 42445,CCC(C)(OC)C1CC(C)(C)CNC(=O)CCN(CC(C)(C)C)C1=O 42446,c1(CNC(C(=O)NC(c2cc(C)ccn2)CC)=O)ccc(N2CCOCC2)cc1 42447,N1(C(c2n(CCC)ccc2)=O)CCC2(C=C(C(=O)NOCC(=O)OCC)C2)C1 42448,C(C(=O)N=c1ccn(C(F)F)[nH]1)(c1cn(C)nn1)NC(C1CS(=O)C1)=O 42449,Cc1cnn(CC(N2CC(NC(=O)CC3CCC(C(F)(F)F)O3)C2)=O)c1 42450,C#Cc1cncc(C(N2CCN(C(=O)C(C)(CC)CO)CC2CC(=O)NC)=O)c1 42451,N1(C(COCCC=C)=O)CCN(C(CNC(=O)C(F)C(C)C)C(F)F)CC1 42452,N1(C(Cc2nc(CC)sc2)=O)CCCC(C)C1.C(CC)(C(=O)OC)NC(C(C)(C)C)=O 42453,c1(Cc2onc(C(=O)NC3C(C)=NNC3=O)n2)cc2c(nc1N)CCC2 42454,c1(NC(c2n(CCC)nnn2)CCCSC)ccc2c(c1)C(C)(C)CO2 42455,Cc1ccc2oc(C(=O)NCCN(CC(C)O)C(c3ccsn3)=O)c(C)c2c1 42456,C1(NC(c2cn(C)nn2)=O)CCOC12CCN(C(C1CC(SC3CC3)C1)=O)CC2 42457,C1(NC(c2nccn3ccnc23)=O)CCC12CCN(C(c1cnccn1)=O)CC2 42458,CC(C)(C)CC(=O)NCC(c1ccccc1)NC(c1ccc(C(C)(C)C)s1)=O 42459,C(=O)(CC(C)CCC=C(C)C)NCC1CC(NC(c2cncc(OC)n2)=O)C1 42460,N1(C(c2ncc(OC)cn2)=O)CCC(C2CC2)C1CNC(=O)C=C1CCCC1 42461,c1(NC(=O)CC2(O)CN(C(c3ccns3)=O)C2)ccc(Cl)c(Br)c1 42462,Cc1ccc(S(=O)(=O)N2CCCC2OCc2ccc(O)c(C)c2O)c(C)c1 42463,c1(N(C(C2(Cl)C(C(=O)N(CC(COCC)C)CC)C2)=O)C)cccc2nccn12 42464,C1(NC(C=C(C)Cl)=O)COC2C(NC(c3cnccc3Br)=O)COC12 42465,c1(SC2COCCN2C)ccc(F)cc1.C12CCCN1C(=O)C1(CC1)CN(C)C2 42466,C(=O)(CC(C)CCCCC)NC1CC(C2CCN(C(CSSC)=O)CC2)OCC1 42467,CN1CC2(CCN(C(c3csc(-c4ccc(O)cc4Br)n3)=O)C2)OCC1=O 42468,N1(CC(N2CCC(C(=O)NCCC(=O)OCC)C2)=O)CCCCC1C 42469,c1(N2CCSCC(C)C2)nc(N2CCOC(C(C)(C)C)C2)nc2c1CCOC2 42470,C1(C(=O)NC2CCOC23CCOC3)CC1N=c1[nH]c(C2CC2)nc2c1CCC2 42471,CCC(CC(=O)N1CCC2C(C(N3CCOC(CC4CC4)C3)=O)C2C1)C(C)C 42472,C1(C(=O)NCC(C)(C(C)C)NC(Cc2c(C)noc2C)=O)C(O)C(=O)N(C)C1C 42473,c1(C(N2CC(NC(C3C(C)(C(F)(F)F)C3)=O)C2)=O)c(C(F)F)nc2sccn12 42474,N1(C(=O)Cc2ccsc2)CC2=C(C1)CN(C(C1CC1c1ccccc1OC(F)F)=O)C2 42475,Cc1ccc2[nH]cc(C#N)c(=NCc3nnnn3C3CCC(=O)NC3=O)c2c1 42476,Cc1c(F)cc(C(N2CC3CN(Cc4ccc(O)c(I)c4)C3C2)=O)cc1Br 42477,c1(N2CC(NC(C3(F)CCS(=O)(=O)C3)=O)C2)ncnc2sc3c(c12)CCCCC3 42478,Cc1n[nH]c(C)c1C(C)C(=O)NCC(F)CNC(=O)CCC(F)F 42479,S(=O)(=O)(CCC1CCc2ccccc21)N1C(C)CC2(CCC2)C1 42480,C(c1ccc(Cl)c(Cl)c1)=CC(=O)N(CCCNC(c1cnnn1C)=O)C 42481,C12(CNC(=O)OC(C)(C)C)CC(CO1)N(c1ncccn1)C2 42482,CC(CN(C)C)CCC(=O)N(CC(C)(C)NC(=O)Cc1csnn1)C 42483,CC1(C)CN(C(c2ccsc2Cl)=O)CCC1NC(=O)CCCc1cncs1 42484,C1(C)(CNC(Cc2c(CN(C)C)con2)=O)CCCN(C(c2ccnnc2)=O)C1 42485,CCCCC#CC(C)(C)NC(c1ccc(OC)cc1Cl)c1nnnn1CCCF 42486,c1(SCC(=O)NCC2C(NC(CCc3nc(C)sc3)=O)C2)ccc(Cl)cc1 42487,C1(C(=O)NC2CCCC(NC(c3cc(Cl)no3)=O)C2)CCc2ccccc2C1 42488,N1(C(=O)NCC2CC(C)(C)SCC2)CCC(=C(Br)Br)CC1 42489,Cc1cccc2[nH]c(C(N3CCC(NC(=O)CCCc4cccs4)C3C)=O)cc12 42490,C(=O)(C(C)(F)C(F)(F)F)N1CCC(CCCNC(C2(C)CN(C)C(=O)C2)=O)CC1 42491,N1(C(COC)=O)CCCC(N(C(=O)CCc2nnc(C3CCCC3)o2)C)CC1 42492,C(c1nc2ccccc2s1)=CC(=O)Nc1ccc(Br)c(OC(F)(F)F)c1 42493,CC1(F)CC(C(=O)NC(C(=O)NCc2nncn2C2CC2)c2ccco2)C1 42494,N1(C(CS(=O)(=O)N(CC)CC)=O)CC(OC)CC(NC(c2cc[nH]n2)=O)C1 42495,c1(NCCCCCCSC)[nH]c(=NC2CCC(C(F)(F)F)CC2)nc2sccc12 42496,N1(C(CCOCC(C)C)=O)CCN(C(=O)CN2CCOCC2)CC1CCN(C)C 42497,C(=O)(C(C(C)C)C(C)C)NC12C(NC(CN(C(=O)OC)C)=O)C3CC1C2C3 42498,C1(CC(=O)NCC(C)OCC)CCN(C(c2ccn(CCOC)n2)=O)CC1 42499,c1(OC)ccc(CN2CCC(C(=O)NC(c3c(Cl)cccc3Cl)C)C2)c(F)c1F 42500,C(CC1=CCCCCC1)NC(=O)CC1CCN(C(C2COC(=O)N2)=O)C1 42501,O=C(C(F)(F)Cc1cnn[nH]1)N1CSCCSC1.C12CCC(C1)n1cc(nn1)C2 42502,c1(C(=O)NC(CC=C)CNC(=O)CC(C)C)ccn2cnc(C)c2c1 42503,C(=O)(CCCCCn1cc(-c2cnn(CCC#N)c2)nn1)N(C(C)(C)C)CC 42504,C(=O)(C1=CCN(C(c2csc(CO)n2)=O)CC1)NC1(CC)CCCC1 42505,N1(CCC)CCCCC1C(=O)NC1CCC1NC(c1ccn(C2CC2)n1)=O 42506,C1(C(=O)NCC2(NC(C(CC(C)C)O)=O)CCC2)COc2cc(Cl)ccc2C1 42507,N1(C(C(C=C)(C)CC)=O)CCC2(CCCN2C(C2CC(F)(F)C2)=O)C1 42508,c1(C(=O)NC(CNC(C(C)OCC=C)=O)CC(C)C)cnc2n1CCS2 42509,c1(C(N(CCNC(C=CC(=O)N(C)C)=O)CC2(O)CCCC2)=O)ccccc1 42510,C1(C(=O)NC(C(C)NC(c2cnc(C)[nH]2)=O)C)CC2CCC1CC2 42511,C12(C(N3CC(CNC(C=C(C)C)=O)C(C(F)(F)F)C3)=O)CCN(CC1)S(=O)(=O)C2 42512,CC(C)(CC1CC1)C(=O)N1CCC(O)(C(C)CNC(c2ccc(CF)cc2)=O)C1 42513,n1(CC#C)cnnc1C(=O)NCC1(NC(C2(C3CC3)CCCO2)=O)CC1.C 42514,c1(-n2c(CC(CCC)O)nc(CCCSC(C)C)n2)ccc2c(c1)OCCO2 42515,N1(C(CCCCC)=O)CCC=C(C=O)C1.c1nc(CC)no1 42516,c1(CNC2(c3n(CCCOC)nnn3)CCN(C)C2C)cccc2c1nnn2C 42517,C(=O)(C1=C(Cl)CCOC1)N1CCCC(C(=O)OC)C1.C1CC12CCOC2 42518,c1(N2CCCC(C)CC2)nc(NC2CCC3C(CC2)C3(F)F)c2ccsc2n1 42519,C1(C(=O)NCCC(C)NC(C2CCC3CC2C3(C)C)=O)CCC2CCCCC2C1 42520,c1(OC)ccc(C(N2CCN(C(=O)C=CC3CCC3)CC2CO)=O)c(OC)c1 42521,S(=O)(=O)(CCC(=O)N(C1CN(C(c2ccc(C(=O)N(C)C)cc2F)=O)C1)C)NC 42522,C1(NC(c2c(C)nns2)=O)CC(CO)N(C(=O)C(C2CCCCCC2)C)C1 42523,C(=O)(C(C)(C)C(=O)NC(C)CCC(=O)NCC1(CS(C)(=O)=O)CC1)NC 42524,C1(C(=O)NC2CN(C(C(=O)NCCOCCCC)=O)C(C)C2)CCCC(=O)N1C 42525,C1(NC(c2cc(Cl)sc2Cl)=O)CC2CC1N(C(c1ncsc1C1CC1)=O)C2 42526,CC(C)C(C(=O)NC(CC(N1CCOCC1)C)=O)OC(=O)C1CC1 42527,N1(C(=O)CC2CCCOC2)CCC(S(=O)(=O)N2CCCC2)CC1 42528,N1(C(C(C)NC(C)=O)=O)CC(NC(=O)CC2CCCC2)C2(CCC2)C1 42529,c1(C(=O)OCC)c(C)coc1Cn1cc(C(C)NC(c2sccc2F)=O)nn1 42530,c1(OCC=CC(=O)NC2(CCCNC(CSCCCC)=O)CC2)cnn(C)c1 42531,c1(C(C(=O)NC(CC)(C)C)Nc2cc(-c3cccc(Cl)c3)on2)ccc(Cl)cc1 42532,N1(C(=O)CC2CC=CCC2)CC2(CCN(C(c3nnn4c3CSCC4)=O)CC2)C1 42533,C1(NC(c2cc3cscc3s2)=O)(CO)CCCN(C(C2CC(=O)NC(=O)N2)=O)C1 42534,Cc1nncc(C(=O)NC(CCN(C)C)C(=O)NCCCC2CCC2)c1C 42535,N1(C(C2ON=C(CC)C2)=O)CCN(C(c2ccc3c(c2)CC3)=O)C(CO)C1 42536,C1(NC(C2(SC)CC2)=O)COC2(CCN(C(c3ccc4ccccc4c3)=O)C2)C1 42537,c1(CC(N2CCC(c3nnc(C4CCCO4)o3)CC2)=O)ccc(Br)c(Cl)c1 42538,C1(C(N2C(C3(O)CN(C(C4=CC(C)C4)=O)C3)CCC2)=O)CCc2nn[nH]c2C1 42539,C1(C)(COC)CC(NC(c2c(C)cnn2C)=O)CN1C(c1scnc1Cl)=O 42540,C1(NC(c2c(C)cn(C)n2)=O)CN(C(C2CC2c2ccccc2)=O)CC12CCC2 42541,CCCCCCCC(=O)NCCCC1CN(C(=O)CC2CC(=O)NC2=O)CCO1 42542,Cc1cocc1C(=O)N(CC(O)CNC1(CNc2ncccn2)CCCC1)C 42543,c1(OC)ccc(C=CC(=O)NCC(C)(C)CNC(=O)CCCS(N)(=O)=O)cc1O 42544,N1(C(C2CCC(=C)CC2)=O)C2CCC1C(C(=O)Nc1ccc(F)c(CC)c1)C2 42545,C1(CCC(=O)NC(CNC(=O)Cn2ncc(Br)n2)CO)CC2CCC1C2 42546,c1(CCC(N2CCC(CO)C2)=O)ccc2ccccc2n1.C123COC(C1)(C2)C3 42547,C(C(C)CN(C(=O)CCNC(=O)C=CCl)C)NC(C1C(C(=O)OC)C1)=O 42548,C1(NC(=O)COc2ncccn2)CCCCC1Nc1cnco1 42549,c1(NC(C(CNC(c2c(CC)n(C)nc2)=O)OC)=O)nccc2[nH]ccc12 42550,c1(NCC(CSC)C)cc(=NCC2CS(=O)(=O)CC23CCC3)[nH]cn1 42551,C1(C(=O)Nc2ccc(SCC)cc2)CCC(C)(C)N1C(=O)C(F)CC 42552,C(=O)(C(C(C)(C)Oc1ncccn1)N1CCC(OC(C)(C)C)C1)NCCOC 42553,c1(C(=O)NC(CC(=O)NCCCN(C)C)CC2CC2)ccc(F)cc1F 42554,CCCCCCC(C)CC(=O)N(CCNC(c1nocc1Cl)=O)CC 42555,c1(C(=O)NC2CN(C(c3cccc(OC)c3)=O)C(CO)C2)cccc2nn[nH]c12 42556,N1(C(CNC(=O)OCC)=O)CCC2C(C1)CN2C(=O)C(F)n1cccn1 42557,c1(C(=O)OC)cc(C(=O)NCC(C)CNC(=O)CC2CC2(Cl)Cl)n2c1CCCC2 42558,C(C1=CCN(C(=O)C(O)C2CCC2)CC1)NC(c1cccs1)=O 42559,c1(C(CC)O)cn(CCCNC(c2coc(C(C)C)n2)=O)nn1 42560,CC1(C)CC(O)CN(C(c2c[nH]nc2CNC(C2CCCN2C2CC2)=O)=O)C1 42561,CCC(C)(C)C(O)C(=O)N1CC(CNC(c2cn3c(n2)CCC3)=O)C(C(F)(F)F)C1 42562,c1(N2CCC(CNC(C(C(C)C)(C)O)=O)CC2)ncc([N+](=O)[O-])cc1C(N)=O 42563,c1(C(=O)NCC(C)NC(=O)C#CC2CCCCO2)cc2c(cc1Cl)NC(=O)C2 42564,c1(CC)cc(=NC(=O)C2CCN(C(=O)C(CC3CC3)OC)C23CCC3)[nH]n1C 42565,c1(NC2N(S(CCOCC)(=O)=O)CCCC2)ccc(CN2CCCS2(=O)=O)cc1 42566,Cc1n[nH]c(C)c1CC(N1CC2C(CNC(=O)C(C)(C)C)C2C1)=O 42567,C1(C(C(=O)NC2CC2NC(=O)CNC(C)=O)OC)CC(F)(F)C1 42568,Cn1ncc2cc(CN3CC4(CC4C(=O)Nc4cc(Cl)c(Cl)cc4Br)C3)ccc12 42569,CC1CCC(CNC(C2CC=CC2)=O)CN1C(=O)COC1(C)CCCC1 42570,c1(C(CCNC(=O)NC(c2nc(C(F)(F)F)cs2)C)O)cccc(Cl)c1 42571,c1(C(=O)NCCCC(=O)OC)ncc(Cl)cc1NC(c1cc(C2CC2)on1)=O 42572,C1(NC(C2(OC)CCC2)=O)CCN(C(C2CC(CSC)C2)=O)CC(C)(C)C1 42573,C12(NC(C(CC#C)CC#C)=O)CCCC1(F)CN(C(=O)C(C)COCC)C2 42574,Cc1nnc2c(C(=O)N(CCCNC(c3ccncc3N=[N+]=[N-])=O)C)cccn12 42575,c1(CN(CCCc2nnnn2C2(C)CC2)CC)cccc(C(F)(F)F)c1.SC 42576,n1(CC)cc(CC(=O)NCC2(NC(=O)CCCn3cc(C)cn3)CC2)nn1 42577,C1(COC)COCCN1C(=O)CC(C1CC1)NC(=O)CCc1nncs1 42578,C(=O)(C1=CC2CC(C1)CC2O)NC(CN(C(Cn1nc(C)oc1=O)=O)C)C 42579,S(=O)(=O)(c1ccc(F)cc1Cl)NCC(N1CCOCC2(COC2)C1)=O 42580,C1(C2CC2)(CNC(CCC)=O)CCN(C(=O)CCN2CCCCC2C)C1 42581,c1(OCC)ccc(C(C)NC(=O)CCC2(C)CC2)cc1F 42582,CC(CC(F)(F)F)C(=O)NC1CCN(C(=O)CCc2ccc(N)c(F)c2)C12CC2 42583,c1(NC(=O)Nc2ccc(C(F)C(F)(F)F)nc2)cnc(Br)nc1 42584,CCCC(C)(CCC)C(=O)N1CCC(CNC(=O)CSC(F)F)(OC)C1 42585,c1(NCCCCC#CC)cc(=NCC(C(C)C)c2ccnn2C)[nH]c(C(C)C)n1 42586,C1(NC(=O)Nc2ccc(C(=O)NCC(C)N(C(=O)CC#N)C)s2)CCN(C)CC1 42587,c1(C(N(C2CCN(C(c3c(C)ccnc3)=O)CC2C)C)=O)ccc2[nH]ccc2n1 42588,CCC(CC1CCCC1)C(=O)N1CC(NC(=O)CCOCC(F)F)C(C)C1 42589,Cc1nc(CCCC(=O)N(CC(C)NC(c2csc(C3CC3)n2)=O)C)cs1 42590,n1(CCNC(NC(C)C)=NCC2(C)CC2(Cl)Cl)ncc2c1CCCC2 42591,N1(C(COCCCOC)=O)CCC2(CCCN2C(=O)CCn2cccc2)CC1 42592,C1(C(=O)NCc2occ(C(=O)NCCn3c(C)cc(C)n3)n2)CC2CCCC2C1 42593,N1(C(c2n(C)cnc2)=O)CCc2sc(CNC(=O)CCc3cnc(O)[nH]3)nc2C1 42594,c1(C(=O)NC2(CNC(C(C3CC3)OC)=O)CC(F)(F)C2)cc2occc2[nH]1 42595,C1(CNC(CC2CC(=C)C2)=O)CCCC1NC(=O)C(CN(C)C)c1ccccc1 42596,CC1CN(C(c2nnn(C(C)(C)C)n2)=O)CC(CCNC(c2cn(C)cn2)=O)O1 42597,C1(OC)CC(C)CN(CCCCCO)C1.C(CCC1CNC1)S 42598,c1(C(=O)NCC(CC(=O)N(CC(=C)C)C)OC)cnn2c1OCC2 42599,C1(NC(c2c(C)cn(C)c2)=O)(CO)CCCN(C(=O)CC(C)n2ccnc2)C1 42600,N1(C(C(C2CCCC2)OC)=O)CC(NC(c2cc(CC3CC3)on2)=O)C(F)C1 42601,c1(C(=O)NC2C(NC(c3ccc(OC4CC4(F)F)cc3)=O)C2)ccc[n+]([O-])c1 42602,C1(CN(C)C)CN(C(=O)CN2CCC(N3CCC3)CC2)c2ccccc2O1 42603,c1(C(N2CCC3(C(NC(COCC)=O)C3)C2)=O)scc2c1OCCO2 42604,C(=O)(CC(C(C)C)NC(C1CCC2(CCC2)O1)=O)NCC(C)CCO 42605,Cc1cnn(C)c1CC(=O)NC1C2CN(C(=O)CS)CC12.c1(CC(N)=O)ccccc1 42606,C1(C(C)C)C(NC(=O)CNC(=O)CC(C)(C)C)CCN1C(=O)CC1CC(C)C1 42607,C1(CC(=O)NCC(=O)NCCC(C)C)CC(C)(C)CN1C(c1cc[n+]([O-])cc1)=O 42608,c1(OC)c[nH]c(C(=O)NCC(C(C)(C)C)NC(=O)C=C2CCC2)cc1=O 42609,CCC(C)C(O)C(C)C(=O)N1CC(NC(=O)CCCCCC(C)C)C(O)C1 42610,N1(C(C(C)Cc2ccc(F)cc2)=O)CC(CO)CC(C)C1 42611,CC12CC1CN(C(=O)C(N1CCN(c3cnccn3)CC1)=O)C2 42612,c1(C(=O)NCC(C)NC(C(CC)Sc2ccccc2)=O)ccc(SC(F)(F)F)cc1 42613,N1(C(C(CC)OCC)=O)CCC(CC(=O)N(C)CCF)C1(C)C 42614,C1(O)(CNC(=NCC=C)NCCCc2nc(C)cs2)CCC2(CC1)OCCO2 42615,O=C(C1Cc2ccccc21)N1CCC2(CCCN2C(C2CC(F)(F)CS2)=O)C1 42616,C=C=CCCC(=O)NCCCOCCCc1ccccc1.C(=O)(CCC1CC1(C)C)N 42617,C(C(=O)N1C(CNC(c2cc(C(C)C)[nH]n2)=O)CC2CC12)(C(C)C)SCC 42618,c1(CC(=O)NCCC(CNC(=O)Cc2cnoc2)O)nnc(S)nc1O 42619,S(=O)(=O)(c1ccnn1C1CCOC1)N1CCN(C(=O)Nc2ccsc2)CC1 42620,C(C(O)CS(C)(=O)=O)NC(=O)NCc1sc(C)c(-c2ccccc2)n1 42621,C(=O)(CC(C)(C)CCC)NCC(CC=C)C(=O)NC1COCC1F 42622,C(=O)(CCCC(C)=O)N1CC(NC(C(C)=CC)=O)C(c2nccn2C)C1 42623,C1(C(=O)NCCCN(C(c2cc(O)nn2C)=O)CC)OCCOC12CCC2 42624,N1(C(C(C)(C)NC(=O)OC)=O)CCC(CNC(c2cc(CO)n(C)n2)=O)CC1 42625,C1(C(=O)NC(CC)CNC(C2CC(F)(CC)C2)=O)COCCN1CC 42626,C=CC(C)CC(=O)N1CC(C(=O)NC2CC=C(C)CC2)(COC)C1 42627,O=C(C1=CCN(C(=O)C(F)OC(F)(F)F)CC1)NC1CC1C1CC1 42628,C(=O)(C(F)(F)C=Cc1ccccc1)N(C)CCNC(C1C2COCC12)=O 42629,c1(C(N(CCN(C(C2(C(=O)OCC)CC2)=O)C)CCOC)=O)sccc1F 42630,C1(C(=O)NC2C(C)CCN(C(C=CCC)=O)C2C)CCc2nc(O)[nH]c2C1 42631,c1(C(=O)NC2CC(CNC(=O)CC3CCCCC3O)C2)ncc(F)cc1F 42632,C1(CNC(Cc2c(CC)cccc2)=O)CCCCC1N=c1cc(Cl)nc(C)[nH]1 42633,C(=O)(C(F)(F)C(F)(F)OC(F)(F)F)N1CCN(C(C)=O)C(c2nccn2C)C1 42634,C1(CC(=O)N(C2CCN(C(C)C(=O)NC)C2)CC)CCN(CCC(C)C)C1 42635,c1(C(N2CC(C3(Nc4c(C#N)nccn4)CC3)C2)=O)cc2cc(Cl)cnc2[nH]1 42636,C(CCCC(=O)NCC1CCCCN1C(c1cccc(F)c1SC)=O)(OC)OC 42637,N1(C(=O)CN)CC2CC3CC2C1C3.CC(C)(C)C1C(=O)N1CC(F)(F)CO 42638,c1(CC(=O)NCCC2CCN(C(=O)CNc3cccnc3)C2)c(O)ncnc1O 42639,N1(C(CSCC#C)=O)CCN(C(=O)Cc2ccc(F)cc2)C(c2nccn2C)C1 42640,c1(SC(C(CC)O)c2ccccc2)cc(-c2ccccc2)n(C(C)(C)C)n1 42641,Cc1cc(C(N2CC3CC3(CNC(C3CC34CCC4)=O)C2)=O)cnc1C 42642,Cc1ccc(C(=O)NCC2COC(CNC(=O)Cc3ccsc3C)C2)cc1CO 42643,Cn1nc(C(=O)N(CCNC(C2(Cl)CC2(C)C)=O)CC2CC2)c(Br)n1 42644,c1(C(=O)NCCNC(c2c(COC)cc[nH]2)=O)ccc2c(c1)NC(=O)CCN2C 42645,C1(C)(CC(=O)NC2CN(C(CC3CCCN(C)C3)=O)C2)CCS(=O)(=O)N1 42646,C(=O)(C(C)(C)C(=O)N(C1CC(C)OCC1)C)N(C)C(C)C.c1(C(=O)N)ccc(CO)cc1 42647,Cn1nnc2cc(C(N3CC(NC(C4C=CCCC4)=O)CC(F)C3)=O)sc12 42648,CCCC(CCC)CCCC(=O)N(C)CCNC(c1cc2c(cn1)CCCC2)=O 42649,CC(C)CCCC(=O)NCC(O)CNC(c1cnc(C2CCCC2)[nH]c1=N)=O 42650,c1(C(=O)NC(C2CCOC2)CC)cc2c(-c3ccc(F)nc3C)cncc2s1 42651,CCS(=O)CC(=O)NC1CCC1NC(=O)CCc1cscn1 42652,C1(CC(=O)NC(=O)Nc2ccc(F)cc2)CCCN(C(c2cnn(C3CC3)n2)=O)C1 42653,Cn1cc(Br)c(CC(=O)NCC2C=CC(NC(=O)C(c3ccccc3)O)C2)n1 42654,c1(C(N2CCC(CC(=O)NCc3ccc(C)o3)C2)=O)nc2ccccc2[nH]1 42655,N1(CC)CCC(NC(=O)CCN(C(C2(C(C)(C)C)CCC2)=O)C(C)C)CC1 42656,N1(C(c2cc(OCC)ncc2)=O)CCCC(NC(=O)Cc2cncnc2)C(F)C1 42657,C1(NC(C(F)F)CCC2Cc3ccccc3C2)Cc2cncn2C(=O)N1 42658,C#Cc1c[nH]nc1C(=O)NC1CN(C(c2csnc2C2CC2)=O)CC1O 42659,c1(C(=O)NCC2(F)CC(NC(c3c(C(C)C)n(C)nc3)=O)C2)cc2ccsc2s1 42660,N1(C(CN2CCC(C)(O)C2)=O)CC2CC(NC(=O)CN3CCNC(=O)C3)C(C2)C1 42661,C1(N(C(CC(=O)NC2CC(NC(C(C(C)C)F)=O)C2)=O)C)CC(C)CC(C)(C)C1 42662,C(=O)(CC(=O)NC1COCC1CNC(=O)C(c1cncnc1)C)OCC 42663,C(=O)(C(CCCOC)NC(=O)C=Cc1ccn(C)c1)NC(C#C)CCCC 42664,c1(CC(=O)NC(C)(C)Cc2csc(Br)c2)ccnc2ccc(O)cc12 42665,C1(C(=O)NCC2(COC)CCC2)CCN(C(c2cc(C)[nH]n2)=O)C1C 42666,C1(C(N2CCOC(CCO)C2)=O)CC(F)(F)CN1C(c1cc(C2CC2)ccn1)=O 42667,c1(C(=O)NC2C(NC(C(CC#C)(C)CC)=O)CC2)ccc2ccccc2c1 42668,c1(OC)cc(C(=O)NC2CCC2NC(C2CC(C)(O)C2)=O)ccc1O 42669,C#CCCC(C(=O)N(C1CCCC(O)C1)C)NC(=O)Cc1ccco1 42670,C(C(=O)N1CC(NC(=O)C(C)(C)C#N)C(c2ccnn2C)C1)(C(C)C)SCC 42671,CCC(C(=O)N1CC(C(=O)OC)C1)NC(=O)CCCN1CCCCC1.C1CCC1 42672,C=CC(C)(CC)C(=O)NC1CC(CNC(c2ccc(C(C)=O)c(C)c2)=O)C1(C)C 42673,c1(C(=O)NCC2N(C(C(COC)OC)=O)CC2)n[nH]c2ccc(OC)nc12 42674,C1(CC=C)(NC(c2ccnn2C)=O)CN(C(c2cc(C(C)(C)C)c[nH]2)=O)C1 42675,N1(C(C=C2CCC(C)CC2)=O)CC2=C(C1)CN(C(C1CC1(F)F)=O)C2 42676,c1(C(=O)NCC2(O)CC(NC(CCS(C)=O)=O)C2)c(F)cccc1Cl 42677,c1(CCC)ccc(N)c(C(=O)N(CC(O)CN(C)C(c2csnc2Cl)=O)C)c1 42678,C(=O)(C(C)C(O)C(C)CC)N1CCC(C(=O)NCC(C#C)OC)C12CC2 42679,n1(CC(=O)NCC2CC(F)(CNC(C3CC(=C)C3)=O)C2)cc(C#N)cn1 42680,C1(O)(CNC(C(C=CC)O)=O)CCN(C(=O)Cc2ccccc2C)C1 42681,N1(C(CC=CC=C)=O)CC2CN(C(=O)C(C)(C)c3cscn3)CCC2(CO)C1 42682,c1(C(=O)NCC(C)C2CC2)ccn(CCNC(=O)CSCC(F)F)c1.CS 42683,N1(C(CC2(OC)CC2)=O)CC(n2cc(CC3C(C)C3(F)F)nn2)C(C)C1 42684,N1(C(Cc2c(C)nsc2)=O)CCN(C(c2ccn3nnnc3c2)=O)C2CCC12 42685,CC(C)S(=O)(=O)CC(=O)N(CC(C)NC(=O)C(=O)N(C)C)C 42686,N1(C(c2c(C)nsc2)=O)CCN(C(c2cnn(CC(F)F)n2)=O)CC(CO)C1 42687,CC(C)C(C)CC(=O)N1CC(N(C(=O)CCc2cc(Br)ccc2F)C)C1 42688,N1(C(CC2C(C)(C)CCO2)=O)CCC2CN(C(=O)C=CC=C(Cl)Cl)CC2C1 42689,Cc1cc(C(=O)NCC(CC(C)C)NC(C2CCC(F)CC2)=O)cnn1 42690,c1(N(C)C)ccc(C(=O)NC2(CCNC(C3(CO)CCCCC3)=O)CCC2)nc1 42691,c1(C(N(CC(=O)OC(CCC)CCC)C)=O)nn(C)c(C)c1-c1nn[nH]n1 42692,N1(C(c2cnn(C(C)C)c2F)C(=O)NCC)CC(C(C)C)c2ccccc21 42693,C1(C(=O)NCC(CC(C)C)NC(C2C=CCS2)=O)CC(C2CCCC2)C1 42694,C1(C)(CC(=O)NCCCC2(NC(C(C)Sc3nncn3C)=O)CC2)CC(F)(F)C1 42695,C1(CC)CCCCC1C(N1CCC2CC12C(=O)N(C)Cc1ccccc1C)=O 42696,C1(CC(N2CCCC(C)(C)CC2)=O)CCc2ccccc2N1 42697,N1(C(c2scc(C)n2)C(=O)NC2CCCC2)CCC(C)(C)C(c2ccccc2)C1 42698,N1(C(c2cc(C(C)C)[nH]n2)=O)CCC(C)C(CNC(c2ccncc2F)=O)C1 42699,c1(SCCNC(C2C(C(C)C)CN2C(=O)OC(C)(C)C)=O)ccc(Cl)cc1Br 42700,CCCCCCC(CC)(CC)C(=O)NC(COC)CNC(=O)CN(C)CCOC 42701,C1(CCOCC(=O)NCC2CC(C(C)(C)C)C2)CCC(F)(F)CC1 42702,C(C)(C(C)S(C)(=O)=O)N(C(C(=O)NC1CN(CCC)C(=O)C1)=O)C 42703,N1(C(=O)OC(C)(C)C)CCCC1C(C)(C)CO.c12cnc(o1)oc2=O 42704,c1(C(=O)NCc2c(C)nn[nH]2)n[nH]c2c1CN(C(=O)C(C)S(N)(=O)=O)C2 42705,c1(CC(=O)NCC23CCC2C3)ccc2ncccc2c1.N12CCCC(C1)CC2=O 42706,C1(O)(C(=O)NC(C2CCCN(C(=O)CCCC(C)(C)C)C2)C)CCCC(C)CC1 42707,c1(CCC(=O)OC(C2CC(C)(OC(F)F)C2)=O)cncc(F)c1 42708,c1(C(=O)NC2(C)CC(NC(C3(C)CCN(C)C3)=O)C2)cccc2nc(O)[nH]c12 42709,c1(OCC)cc(C)[nH]c(=NCC2CC3CCC2N(C(c2csc(CO)n2)=O)C3)n1 42710,N1(C(c2ccc(CC)nc2)=O)CCCC(O)(CNC(c2cc(C3CC3)on2)=O)C1 42711,c1(C(=O)NC(C(=O)NCCc2ccc(C)s2)C2CC2)cnc(C)c(C)c1 42712,c1(C(=O)NC2CC(CNC(c3cccc4ncnn34)=O)C2)ccc(O)c(F)c1F 42713,c1(CC)ccc(C(=O)NCC2CC2CNC(C2CC(=O)NC(=O)C2)=O)c(C)n1 42714,N1(C(CCC(=O)OC)=O)Cc2ccnn2CC(NC(c2cscc2Cl)=O)C1 42715,c12ccc(cc1)CNC2=O.C12CCC(C1)OC2=O.n1(CC2CC2)cncn1 42716,C(C(C)C(=O)NC1COCC1NC(c1cc(C(N)=O)c[nH]1)=O)OCC 42717,C1(C(C(=O)NCCN(C)C(C2(C)CCCN2C)=O)(C)C)CCC(O)CC1 42718,c1(C(CC)C(=O)N(CC(O)CN(C(=O)C(C)=CCOC)C)C)ccc(F)cc1 42719,C12(CCNC(c3c(C)con3)=O)CCC1CN(C(=O)CCOCC1CC1)C2 42720,Cc1cc(C(N2CC(NC(c3ccncc3Cl)=O)C2)=O)c(Cl)cc1Cl 42721,c1(-c2cc(C(N3CCC(=CCC)C3)=O)sc2)cncc(N2CCOCC2)c1 42722,c1(CC(N2CC(C(C)CO)C2)=O)ccc2c(c1)CCCN2C 42723,c1(C(N(CCC)C)=O)ccc2nc(S)oc2c1.n1(CC(=O)N)nc(C)cc1C(=O)OC 42724,N1(C(c2cn(CC)nc2)=O)CCC2(CCC(CNC(c3csnn3)=O)OC2)CC1 42725,Nc1c(C(=O)NCCNC(=O)C(O)Cc2ccccc2Cl)cccc1F 42726,c1(C(=O)NCC(N(C(=O)Cn2cccn2)C)C2CC2)ccccc1C1(C#N)CC1 42727,c1(C(=O)NCCCC(C)NC(COCCC)=O)cc(Cl)c(F)cc1F 42728,c1(NC(=O)CC)ccc(C)cc1.N1(C(CCNS(C)(=O)=O)=O)CC(C)(CCOC)C1 42729,C1(N(C)C)CCOC(C(N2CC(O)(c3cn(Cc4ccno4)nn3)C2)=O)C1 42730,C(C(=O)NC1CCC1CNC(C12CCC(CC1)CC2)=O)(C(C)(C)C)SC 42731,c1(CCCC)nc(C(=O)NC2CCCCC2n2cc(CCN(C)C)nn2)c(Cl)[nH]1 42732,c1(SC)cc(C(=O)NCC2C(C)CCCN2C(=O)CC(=O)NC2CC2)ccc1F 42733,CC(C)(CC1CCOC1)C(=O)N(C1CCN(C(=O)CCc2cnoc2)CC1)CCO 42734,CCC(C(=O)N1CC2C(NC(=O)Cc3scnc3-c3cccs3)C2C1)C(C)(F)F 42735,C(CCC(F)(F)F)N(C(C1N(C(Cc2c(C)con2)=O)CC1)=O)C 42736,c1(C(N(CCCCCC)CCNC(=O)C(O)C2CC2)=O)ccc2nonc2c1 42737,CC(C)CC(C)(CNC(=O)C(C)(C)c1cnn[nH]1)NC(c1cc(C(F)F)on1)=O 42738,c1(C(N2C(CNC(CCC=CCC=C)=O)C=CC2)=O)cnc2ccnn2c1C 42739,Cc1ccc2oc(C(=O)NC3CC(C)N(C(c4cc(CCO)on4)=O)C3)cc2n1 42740,CC(C1CC1)=CC(=O)NC1CC(NC(=O)C=C)C1.C1(C(=O)N)(C(N)=O)CC1 42741,c1(CC(=O)NC23CC(C(=O)NCC4CCCSC4)(C2)C3)ccccc1F 42742,C1(N(C(C(CNC(c2nc(C(C)C)oc2)=O)O)=O)C)CCCC1(C)O 42743,Cc1cc(Cl)cc(C(=O)NCCCCNC(c2n[nH]c3c2CSCC3)=O)c1C 42744,CN1CC(C(=O)NCC2CCN2C(C2(C)CC(O)CN2C)=O)CCC1=O 42745,c1(OCC)cccnc1C(N1CC(O)(CCNC(c2cccc(F)c2)=O)C1)=O 42746,N1(C(C2(C)CC2Br)=O)CCCC(C2CC2NC(c2cnn(CCC#N)c2)=O)C1 42747,c1(OC(C)C)cccc(C(N2CCC(=CCNC(C3SCCC3C)=O)CC2)=O)n1 42748,Cn1nc2c(c1CN1CCC(O)C1C(=O)Nc1ccc(I)cc1F)CCCC2 42749,C(=O)(C(C)CC(F)(F)F)NC(c1occ(C(N(CC(C)C#N)CC)=O)n1)C 42750,C(=O)(CCn1ccnc1)NCC1(CC(=O)N(CC(C)O)CCC#N)CC1 42751,c1(C(=O)CC)ccc(N2CCC2)cc1.C12(N)CC(C1)NC2.c1(CC2CC2)ccccc1 42752,c1(-c2n(-c3c(C)cccc3C)nc(C(C)C3CC3)n2)sc2cccc(F)c2c1C 42753,c1(C(N2CC(NC(=O)C(F)(F)CC3CC3)CC(C)C2)=O)nc2cccnc2s1 42754,CCCCC(CNC(C1CCCN1C)=O)NC(c1snc(Cl)c1Cl)=O 42755,N1(Cc2cn(C3C(CC)C3)nn2)CCC(Cn2nc(C)cc2C)CC1 42756,c1(C(C)=O)ccc(C(=O)NC2CCN(C(=O)CCNC(=O)C=CCl)C2)nc1 42757,N1(C(C2C(C)C2)=O)CCCC(CCNC(=O)CCN(C)CCO)CC1 42758,C(=O)(CC(COC)COC)N1CCCC(N(C(=O)CC2CCNC(=O)C2)CC)C1 42759,c1(C(N2CC(N(C)C(c3nnco3)=O)C2)=O)ccc2c(c1)NC(=O)CO2 42760,c1(OCC(N)=O)ccc(C(=O)NCC(C)NC(=O)C=CSc2ccccc2)cc1 42761,c1(C(=O)NC2(C(=O)NCc3ncccc3F)CC(CO)C2)ccc(O)cn1 42762,C1(NC(c2c(CC)c[nH]c2)=O)CCN(C(=O)CSc2cccc(F)c2)CC1(C)C 42763,C(=O)(C1=CS(=O)(=O)CCC1)NC1CCN(C(Cc2n(CC)nnc2C)=O)C1 42764,c1(CC(=O)NC(CCC)CNC(C2CCC(=O)NC2)=O)nc(C)cc(C)n1 42765,N1(C(C(C)Oc2ccccc2CN2C(=O)CNC2=O)=O)Cc2ccc(Cl)cc2C1 42766,Cn1cc(C(=O)NC2CC2CNC(c2ccc(-n3cncn3)cn2)=O)n(C)c1=O 42767,N1(C(C=CSC)=O)CCN(C(c2cc(C(C)C)n(C)c2C)=O)C(C)C1C 42768,c1(-c2cn(CC(CNC(CC(CCCC)O)=O)(F)F)nn2)ccc(S(N)(=O)=O)cc1Cl 42769,c1(C(=O)NC(C2CCCC2)CNC(C(CC#C)C)=O)cncc(C)c1Cl 42770,C(=O)(CCCCCF)N1C(CCC(=O)NCC(C(=O)NC)C)CCC1 42771,c1(C(=O)Cc2cn(C3CN(C(c4n(C)cc(F)c4)=O)C3)nn2)nc(Br)cnc1N 42772,C(=O)(C(C)(C)C(O)C(C)C)NC1CCN(C(c2cc(OC)c(Br)nc2)=O)C1C 42773,C1(C)(C(=O)NCCC(C)CCNC(=O)CCCc2ccccn2)CC2CCC1C2 42774,C1(C(N2C(CNC(c3c(C)scn3)=O)CCCC2)=O)COC2COCC12 42775,c1(C(N2CCC(C)(NC(c3nc(C)c(C)[nH]3)=O)C2)=O)ccc2[nH]c(=N)[nH]c2c1 42776,CCCN=C(NCc1ncc(Br)s1)NCC1(CC)CCCC1 42777,c1(C(CC)C)cc(C(=O)NC(C)(CNC(C2(C3CCCO3)CC2)=O)C2CC2)on1 42778,C(=O)(C(C#N)C(C)(C)C)N1C(CC(C(=O)CCCSC)=O)C2CCC1C2.CCO 42779,C(=O)(C1=CS(=O)(=O)CCC1)Nc1c(C(N2C(C#N)C3CC3C2)=O)scc1 42780,N1(C(c2cc(C)[nH]c2)=O)CC(NC(C2(Cc3cnn[nH]3)CCC2)=O)C(C)C1 42781,c1(-c2c(CN3CCC(O)CC3C(N)=O)cccc2)ccc(Br)cc1C(=O)NC 42782,C(C)(C(F)(F)C(F)(F)F)=CC(=O)NC(CCNC(C(C)NC(CO)=O)=O)C(C)C 42783,N1(C(C2C(C)(Br)C2)=O)C(CNC(=O)Cn2cnnn2)CC2COCC12 42784,C1(C(=O)Nc2c(CC=C)cccc2)CCC(C)(C)N(C(C2C3CC(=O)CC23)=O)C1 42785,c1(OC)cc(C=CC(=O)NCc2ccc(CNC(C3CCNC3=O)=O)cc2)sn1 42786,Cc1ccncc1C(=O)NCCC1(CNC(c2cn(C)nc2C)=O)CCCC1 42787,c1(C(N2CCCC(NC(C(C3CCC3)OC)=O)C2C)=O)ccc(C)cc1[N+](=O)[O-] 42788,C(C(=O)NCC(C)(CO)NC(C1CN(C2CCC2)C1)=O)(C(C)C)OC(C)C 42789,N1(C(C(CC=C)C)=O)CCCCC(NC(c2cc(-c3ccc(C)cc3)no2)=O)C1 42790,c1(C(=O)NCC2C(C)CCN2C(C2(C(=O)N(C)C)CC2)=O)cc2ncccc2o1 42791,c1(C2C(N3CC(CC(=O)OC)(C(F)F)C3)C2)cccc(OC)c1 42792,c1(C(=O)OCC2OCCN(C)C2=O)cnn2c1NCCC2 42793,c1(OC)cc(C)ncc1NC(=O)Cc1cccc(CN2CCN(C)CC2)n1 42794,c1(CNC(=O)NCC2CCN(C(=O)OC)CC2)ccc2cccnc2c1 42795,CC1CC(CNC(c2cccnc2)=O)CN1C(=O)CCCC1CCCC1 42796,CC1Cn2nc(C(=O)NC3COC3)cc2CN1C(=O)OC(C)(C)C 42797,C#CC1CN(C(=O)C(C)N(C(=O)CCc2ccoc2)CCOC)CCO1 42798,N1(C(C(C)Cc2ccco2)=O)CC(NC(c2cncc(F)c2)=O)CC12CCCC2 42799,C1(NC(c2ccc(C)nc2)=O)CC2(CCC(NC(C3C(C)CC3C)=O)CC2)C1 42800,N1(C(CC(C)(C)OC)=O)CCCC(C)(NC(c2ccc(O)cc2C(F)F)=O)C1 42801,N1(C(=O)C(O)CCCNC(C23CC2CNC3=O)=O)CCc2occc2C1 42802,Cc1ccc(O)c(CNC(C2CCOC2CNC(c2cn(C)c(=O)n2C)=O)=O)n1 42803,Cc1ccc(C2(C(=O)NC3CCCCC3CNC(c3cc[nH]n3)=O)CCC2)cc1 42804,N1(C(CC2CN(C(C(C)NC(C)=O)=O)C(C)(C)C2)=O)CC2(C1)CC(C)(C)C2 42805,CC1(C(=O)NCCCNC(=O)Cc2ccc(O)cc2Cl)CCC12CCC2 42806,Cc1ccc(CC(=O)NC2CC(CNC(=O)C(C)CN(C)C)C(O)C2)c(Cl)n1 42807,C=CCC(CC=C)C(=O)N1CC(O)CC1(C)C(=O)NCCCCC(C)(C)C 42808,Cc1cnc(C(N2CC(C(O)C(=O)NCCN3CCC(C)C3)C2)=O)cn1 42809,c1(C(CCOC)NCCC(F)(F)CO)c(C)cc(C)cc1O 42810,c1(CCC(=O)N(C2CCN(CCCO)CC2)CC2CC2)ncccc1Br 42811,C1(C(N2C(C)C(NC(c3ccc(CCO)cc3)=O)CC2)=O)CCCC(F)(F)C1 42812,c1(CCC(=O)NCC2CCCN(C(c3cccnc3Br)=O)C2)ccc(F)cc1 42813,c1(OC)cnccc1C(N1CCC(CN(C)C(C2CC(OC)C(OC)C2)=O)C1)=O 42814,CCCCC(O)C(C)C(=O)N1CC(O)(C(F)C(N2CCCCCCC2C)=O)C1 42815,C1(OC)CC(NC(c2ccnnc2C)=O)CN(C(=O)Cn2c(C)ccc2C)C1 42816,C1(CCC)CN(C(=O)C(O)C(F)(F)F)CCN1C(=O)C(c1ccccc1OC)F 42817,c1(C(=O)OC)cnc(C(=O)N(c2c(OC)ccc(Cl)c2)C2CCC2)c(N)c1 42818,C1(C(=O)NC(c2cccc(F)c2)C)CC(F)CN(C(c2ccc(O)c(I)c2)=O)C1 42819,N1(C(C(CCC)N(C)C)=O)CCCC2(NC(c3ccoc3Cl)=O)CC2C1 42820,c1(C(=O)NCC2(C)CN(CCc3ccncc3)C2)cccc(C(=O)NC)c1 42821,C(C(=O)N=S(C)(=O)N(C)C)N(CC(CC)(C)O)C(=O)OC(C)C 42822,c1(OC)cc(NC(=O)C(=O)NS(=O)(=O)CCSC)ccc1N1CCOCC1 42823,C1(N(C(=O)CCCOC(C)C)CCC)CCN(C(=O)CCC2CCCCO2)CC1 42824,N1(C(CCCCSC)=O)CC(C)C(C)(CNC(=O)C(C2CC(F)(F)C2)OC)C1 42825,C#CC1CC2(CC2)CN1C(=O)CCC(C)NC(C1CC2CC2C1)=O 42826,c1(OC)ccc(CC(N)C(=O)NCCO)c(OC)c1.c12cccc(c1)OC2 42827,N1(C(C2(C)CCN(C(c3cc(C)on3)=O)CC2)=O)CC(C#N)C2(CCC2)C1 42828,N1(C(CC(C)F)=O)CCCN(C(=O)Cc2ccc(Cl)cc2Cl)C(CO)C1 42829,c1(OC)ccc(F)c(-c2ccc(C3(C(=O)Nc4cc(Br)cc(I)c4)CCC3)cc2)c1 42830,C1(C(=O)NC(C=CC(=O)NC(C(C)F)C)C)OCC2CCCC12 42831,C1(C(N)=O)(NC(CN(C(C=C2CCC(C)CC2)=O)C2CC2)=O)CCC(C)CC1 42832,N1(C(C(C)(C)OC)=O)C2CCC1C(CNC(c1nccnc1C(N)=O)=O)C2 42833,CC1=C(C(=O)NC2CCCC2C(=O)Nc2ccc(Br)nc2)CCO1 42834,c1(CC(=O)NC(CC)CCCNc2ncncc2I)c(C)nn(C)c1C 42835,c1(NC(C2CC3CC3N2C(c2n[nH]c3c2CCCC3)=O)=O)nc(Br)c(Br)cc1Br 42836,C1(NC(C(CCC)N(C)C)=O)CN(C(=O)CNC(C)=O)Cc2nccn2C1 42837,C(=O)(CC(C=C)CC)N(CC(Cc1cnc[nH]1)NC(CCOCC#C)=O)CC 42838,N1(C(C2C(C=C)C2)=O)CC(NC(c2sc(Cl)c(Cl)c2C)=O)C(C)(C)C1 42839,C1(OC)CC2CC(C(=O)NCCCC(C)NC(=O)CC3CC(=O)C3)CC12 42840,C1(NC(=O)CCC=CBr)C2CCC1N(C(c1ccc(CF)cc1)=O)C2 42841,c1(C(c2nnnn2-c2ccc(F)cc2)NC(C)CC#N)cnc2[nH]cnc2c1 42842,C1(CC(N2CC(O)(CCNC(C(COC)OC)=O)C2)=O)COCC2(CCC2)O1 42843,CCCCC(O)C(=O)NCC(C)NC(=O)CCC1CCCC1 42844,N1(C(C2C(CC)C2)=O)CC(O)(CNC(C2(c3cncnc3)CCCC2)=O)C1 42845,c1(CNC(c2n(CCC)nnn2)c2occc2C)cc(Br)cc(Cl)c1F 42846,C(=O)(C1=CCCCC1C)N1CCC2C(C(=O)NCC=CCOC)C2C1 42847,C(=O)(CCCC(=O)NCC(C)(C)C)NC1(C)CCN(C(c2cncnn2)C)CC1 42848,C1(NC(c2cc(Cl)ccn2)=O)COC2(C1)CN(C(=O)CCCc1cnccn1)C2 42849,c1(CC(=O)NCC(C)CN(C(=O)C(C(C)(C)C)N(C)C)C)cc(F)c(N)cc1F 42850,N(C1CS(=O)(=O)Cc2ccccc21)C(CO)CCC1CC1 42851,C1(NC(CSCC=C)=O)CC2CC(NC(C3CCC4CC34)=O)C1C2 42852,C1(P(C)(C)=O)(C(N2C(CCNC(C(n3c(C)ncc3)C)=O)CCC2)=O)CC1 42853,C1(CNC(C2CCC(OC)C2)=O)CC2(CC2)CN1C(c1cc(Cl)c[nH]1)=O 42854,C(C)(CN=c1nc2scnc2c(NC2COc3cc(Br)ccc32)[nH]1)OCC=C 42855,C(C(O)C(F)(F)F)NC(C1C2CC1N(C(=O)CC1CCCCC1)C2)=O 42856,C1(NC(C=CCCSC)=O)CCN(C(C2COCCN2C)=O)C1(C)C 42857,CC(C)CC(C(=O)N1CCCC(NC(=O)CN(C)C(N)=O)C1)Nc1ccccc1 42858,C1(C(=O)NC2C3CC(NC(C(C)c4cccs4)=O)CC32)CC2CC(=O)C1O2 42859,C1(C(C)NC(=O)CSC(C)(C)C)CCCN(C(=O)CCCn2cccn2)C1 42860,C1(C(=O)NCC(CNC(=O)CCCOc2cccnc2)F)(COC)CC=CCC1 42861,Cc1ncc(C(=O)NC2CC(OCC(=O)N(CC(C)(C)C)C(C)C)C2)c(=N)[nH]1 42862,Cc1noc(C)c1CSC(C)C(=O)NC1CCCN(C(c2cc(O)nn2C)=O)C1 42863,c1ccc(C2CCCC2CCNCC2(c3cc[nH]n3)CC2)cc1 42864,CC1CC(C(N2CC(O)(CNC(=O)CSCC(F)F)C2)=O)CN1C 42865,c1(NC(C)=O)ncc(S(=O)(=O)N2CCCC(c3ccc(C(F)(F)F)cc3)C2)s1 42866,Cc1ccc(SCCC(=O)NCC2(F)CCC(CNC(C3CC3(F)F)=O)C2)cc1 42867,c1(C(=O)NCC2CCC3CC23)ccccc1Cl.C12CC(C1)CCNC2=O 42868,C1(CC)CC2(CCCC2)CN1C(=O)CC(C)=C(C)C 42869,C(C(CC(C)C)C(=O)NC12CC1CN(C(c1ccnc(C3CC3)c1)=O)C2)OC 42870,CC1(C)C(=O)CC1C(N1CC(C(=O)NCCC(O)C2CCC2)C1)=O 42871,C1(CC)(NC(=O)CCCn2cncn2)CCN(C(=O)CC2CCC3CC23)CC1 42872,C(C(CC(C)C)NC(c1ccc(F)cn1)=O)NC(CC1(CSC)CC1)=O 42873,C(C)(CC(C)NC(c1sccc1COC)=O)NC(COC(C)C)=O 42874,N1(C(CCCCC(=O)OC)=O)CCN(C(C2CC(=O)N2)=O)CC(C)(F)C1 42875,CC1CCN(C(=O)Cn2cnnn2)C(NC(=O)C(C)(C)OCC(=O)OC(C)(C)C)C1 42876,C1(C(N(C2CCN(C(c3ocnc3C)=O)C2)CC)=O)C2C(=O)OCC12Br 42877,c1(C(=O)NCCN(C(=O)C=CS(C)=O)C)cc2cc(F)ccc2o1 42878,c1(C(=O)NC(CCCCNC(c2nccc(C)n2)=O)C)cc2cccnc2s1 42879,C(=O)(C(=O)C(F)(F)F)N(CC)CC1CCN(C(=O)CCN2CCOCC2)CC1 42880,C#Cc1cc(C(=O)NCC2CN(C(C3(C)CCCS3)=O)C2)ccc1C 42881,c1(C(=O)NCC23C(CN(C(C(C)=O)=O)C2)C3)cc(Cl)cc(Cl)c1O 42882,CCCC(CC)CC(=O)NCc1cccc(NC(c2c(N)cc(F)cc2F)=O)c1 42883,C1(NC(Cc2c(C)n[nH]c2)=O)COC2C(NC(=O)CCCC(F)F)COC12 42884,c1(C(N(C)CC2(COC)CCC2)=O)cc(C)nc2c1c(C)nn2C 42885,c1(NC(c2snc(CC)n2)=O)nc(Cl)cc2cc(Br)ccc12 42886,Cc1cc(C#N)nc(=NCCC2CCN(C(=O)CNC(=O)CCC3CCCC3)C2)[nH]1 42887,N1(C(=O)OC(C)(C)C)CCC(CO)(NCCN2CCCCS2(=O)=O)CC1C 42888,Cc1nc(C(N2CC3(NC(=O)CC4CCC(C)(C)O4)CC2C3)=O)n(C)n1 42889,N1(CCC=C)CCC2(CC1)CC2N(Cc1ccc(C(=O)NC(C)C)nc1)CC 42890,C12(NC(c3cc(=NCC)[nH]cc3)=O)CCOCC1CN(C(=O)CN1CCCC1)C2 42891,C1(C(N2C(C)CC(NC(C3CCC(=O)C3)=O)CC2)=O)CCc2n[nH]cc2C1 42892,c1(CC(=O)NC2C(CNC(C(CC)F)=O)C2)ccc(Cl)cc1Cl 42893,O=c1cc(N2CCC(CC(F)(F)F)C2)ccn1Cc1ccnc(Cl)c1 42894,Cc1ccc2c(c1)CN=C(NCC1(C)COCCO1)NS2(=O)=O 42895,C1(NC(C(C(=O)OC)C)=O)CN(Cc2cc(C)ccc2Cl)CCC1(F)F 42896,c1(CCC(=O)NCC(C)CN(C)C(C2CC3C=CC2O3)=O)ccc(C#N)cc1F 42897,c1(C(=O)OC)cc(NC(=O)NCCCC(c2cnn(C)c2)C2CC2)c(Br)cc1C 42898,C12(C(N3CC(OC)C(NC(=O)C(F)(F)C(C)O)C3)=O)CCCN1CCC2 42899,N1(C(c2n(CCC)ncc2)=O)CCC(C(=O)NCC(C)C)C1(C)C 42900,N1(C(CCCCC#C)=O)C(CNC(c2cnc(CC(C)C)[nH]2)=O)CC2CCCC12 42901,CCCCC(CNC(=O)C(C)NC(=O)NC)NC(c1cocc1C)=O 42902,CCCC(C#N)C(=O)NCC1OCCC1C(=O)NCC(C1CCCC1)OC 42903,c1(C(N2C(CCNC(CCP(C)(C)=O)=O)CSCC2)=O)ccc(N)c(Cl)c1O 42904,CC(N=c1[nH]c(=NC2CCOC3(CCSCC3)C2)c2ncnn2[nH]1)c1ncc(CO)s1 42905,C(=O)(C1CCCc2nc[nH]c21)N1CC(NC(Cc2ccc(C)o2)=O)C(C)C1 42906,Cc1nc(C(C)C)nc(O)c1C(N1CCOC(F)(C(F)(F)F)C1)=O 42907,N1(C(CCCC(=C)C)=O)CC2COCCC2(NC(=O)CC2SC(=N)NC2=O)C1 42908,Cc1cc(C#N)cnc1C(=O)NC1CC(NC(=O)CC2CCC2)C1 42909,C1(N(C(C(c2cccnc2)NC(C=CCCC)=O)=O)C)CCC(C)(C)CC1 42910,CC(C)CC(C(=O)NC(C)CNC(c1ccncc1Cl)=O)N1CCCCC1=O 42911,c1(CC(=O)NCC2(C)N(C(C3CCN(CC)CC3)=O)CCC2)cccc(F)c1F 42912,c1(C(CNC(c2ncn(C)n2)=O)NC(CC2CC(OCC)C2)=O)ccc(F)cc1 42913,C1(N(C(=O)CCc2ncco2)CC)CCCN(C(C2(C3CCCO3)CC2)=O)CC1 42914,c1(CC)n[nH]c(CC)c1CC(N1CC(C)(NC(C2CC2C)=O)C1)=O 42915,Cc1ccc(C(N2CCN(C3CCC(NC(c4ccsc4C)=O)C3)CC2)=O)cn1 42916,CC(C)S(=O)(=O)CC(=O)NC1CCCCCN(C(C2CCC(C)C2)=O)C1 42917,C(=O)(C(C)(C)C(C)C)NC1C(CC)N(C(c2nc(Cl)sc2C)=O)CC1 42918,CCC(CNC(=O)Cc1ccc(C(C)C)cc1)(CC)NC(=O)C=Cc1scnc1C 42919,c1(C(N2C(CNC(CNc3cc(OC)ncc3)=O)CC2)=O)noc2c1COCC2 42920,N1(C(CC(C)C)=O)CCC(NC(c2cc(-c3cccnc3)[nH]n2)=O)C(C)C1 42921,N1(C(c2c(CC)c[nH]n2)=O)CCC2(NC(c3c(F)cccc3Br)=O)CC2C1 42922,C12CCC3(CN(C3)C1=O)O2.Cc1cc(C(=O)NCCNC(c2cccnc2)=O)c[nH]1 42923,C1(CC(=O)NC2CC(F)(F)CC2NC(C2SCCCS2)=O)CN2CCC1CC2 42924,N1(C(Cc2c(C)cccc2Br)=O)CC2(CCN(C(C3COC(C)C3)=O)C2)C1 42925,c1(CC(C(=O)NCC2CNC(=O)O2)NC(C(C)n2cnnn2)=O)cnn(C)c1O 42926,c1(C(N(CC(CNC(C2CCC(C#C)CC2)=O)C)C)=O)cnn2c1CC(F)(F)C2 42927,Cc1cccc(COCC(=O)NCCCC2CCN(C(=O)C=CC(C)C)CC2)c1 42928,N1(C(C(C)(CO)NC(C)=O)=O)CCN(C)C(CNC(c2ccco2)=O)C1 42929,N1(C(CCCCCOCC)=O)CCC(NC(=O)COCC2CCC2)C(F)(F)CC1 42930,CC1=C(C)CC(C(=O)NCCCN(C(=O)CC(C)NC(=O)OC(C)(C)C)C)CC1 42931,CCCC(O)C(CO)NC(=O)C(CN(C)C)NC(c1nc(C2CC2)no1)=O 42932,N1(C(c2n(C)ncc2)=O)CC(C(N2CCCC3C(O)CC23)=O)CCC1(C)C 42933,C1(C(N2CC(NC(C3CC(C)OC3=O)=O)C2)=O)(CC)CC(C)(C)C1 42934,N1(C(C(C)N2CCC2)=O)CCC(CNC(C2NC(=O)C3CCC23)=O)C(F)(F)CC1 42935,C(=O)(CC(O)CCCC)N1CC(CNC(CC=C)=O)C(c2cnn(C)c2)C1 42936,Cc1cc(CCC(=O)NCCC(O)CNC(C2(C)CCN(C)C2=O)=O)cc(C)c1 42937,C#Cc1cncc(C(=O)NCCC2CC(F)(F)CN2C(c2nocc2Cl)=O)c1 42938,CC1CN(C(C2(NC(c3occc3Cl)=O)CC2C)=O)CCN1C1CC1 42939,C(CC(C)CC)(C(=O)N1C2CCC1CN(C)C2)NC(C1C(C(=C)C)OCC1)=O 42940,n1(CC(N2CCC(CNC(C(C(C)C)OC)=O)CC2C)=O)cc([N+](=O)[O-])nc1C 42941,N(C1CC(C)n2ccnc21)C(CC1CCC(NC(C2(C=C)CCC2)=O)CC1)=O 42942,N1(C(c2ncn(-c3c(N)nc(Br)cc3)n2)=O)CCC2(C1)CN(CC(F)(F)F)C2 42943,CC(C)N(O)C(=O)C(=O)N1C(CNC(c2cc(CCO)on2)=O)CC2CCCC12 42944,N1(C(C(c2n(C)cnc2)=O)=O)CCC(C)(C)C(C(=O)NCC2CCC(F)(F)C2)C1 42945,c1(C(=O)NC(C(C)C)CCNC(=O)C(C)(C)C)nnc2n1CCCC2 42946,C1(NC(Cc2ccc(CC)cc2)=O)CN(C(=O)Cn2cnnc2)C2(CCOC2)C1 42947,C1(CNC(c2cc(F)c(O)c(F)c2)=O)CC2(CCN(C(=O)CC(F)(F)F)CC2)C1 42948,CCC(C)(C)CCCC(=O)NC(CO)C(C)NC(c1cn(C)c(=O)cn1)=O 42949,CC(C)(CC(=O)N1CC(C)(NC(=O)CCCC#N)C1)CC(F)(F)F 42950,c1(C(=O)NCC(CO)NC(=O)CCc2cnccn2)cc(Cl)c2c(c1)OCO2 42951,C(=O)(C(F)(CNC(C1(C#N)CCCC1)=O)C(C)C)NCC(CC1CC1)OC 42952,c1(C(N2CC(C)OC(c3ccc(F)cc3)C2)=O)cc(Br)cc(F)c1N 42953,N1(C(Cc2cc(C)[nH]n2)=O)CC(C)(C(=O)N(CC2=CCSC2)C)CC1(C)C 42954,C(=O)(CC(C)(C)C(F)F)N(CC(C)(C)CNC(=O)Cc1ccon1)C 42955,C1(CCC)(NC(=O)CN(CC(C)(C)C)C)CCCN(C(C2CCSCC2)=O)C1 42956,c1(NC(C2CN(C(c3c(C)nc[nH]3)=O)C2)=O)cnn2ccccc12 42957,C1(C(=O)NC(CCNC(c2[nH]cc(C)c2)=O)C)COCCN1CC(F)(F)F 42958,N1(CC(C)(C)C)CCC(F)(F)C(C(F)(F)F)C1.C1(=O)CC(=O)N1CCO 42959,N1(C(c2c(C)cnn2C)=O)CC(C)N(C(c2cc(C#N)c[nH]2)=O)C(C)C1 42960,C(CCC(C(=O)NCC(CO)C(C)(C)C)NC(=O)CC1CN(C(C)=O)C1)OC 42961,N1(C(CSCC=C)=O)CCC(C)(NC(=O)CCC2CCCN(C)C2)CC1 42962,C1(NC(CCCCSC)=O)CCC2(CC1)CC2NC(=O)C(=O)N(C)C 42963,CC1CCN(C(=O)Cn2ncnn2)CC1NC(c1cnc(N)c(Br)c1)=O 42964,N1(C(c2c[nH]c(=N)s2)=O)CCC(C(=O)NC2CN(C3CCC3)C2)C12CC2 42965,C1(C(=O)NCC2CCC2)(CNC(C2CCCS2)=O)CCCC1.C1COC1 42966,C(=O)(C(CCSC)NC(c1nnsc1N)=O)N1CCC(CC=C)C1 42967,c1(C(=O)NC(c2ccccc2)CNC(C2CC(=C)C2)=O)ccn(O)c(=O)c1 42968,CC1CN(C(C2(O)CCCCCC2)=O)CCC1CNC(C1CC2CCC1CC2)=O 42969,c1(C(C(=O)NC2(C)CC2)N(C(c2ccccc2)C(=O)NC)C)c(SC)cccc1F 42970,C12(CC(=O)NCC(CC=C)(F)F)CCC1CN(C(=O)CC1(C#N)CC1)C2 42971,c1(C(N2CCC3CN(C(C4ON=C(C)C4)=O)C3C2)=O)cnc2sc(C)cn2c1=O 42972,c1(CC(=O)NC2CN(Cc3cnc(Cl)nc3)CC2F)cc(F)c(F)cc1F 42973,C1(NC(C=C(C)C)=O)CC2CC1CN(C(c1ccccc1C1CC1(F)F)=O)C2 42974,C1(N(C)C(C2(C(N)=O)CCC2)=O)CCC(NC(c2c[nH]nc2C2CC2)=O)C1 42975,c1(-c2c(NC(C3CCC(C)(C)O3)=O)nccc2)ccc(Br)nc1F 42976,C1(C(=O)OC)Cc2c([nH]c3ccccc23)CN1CCCN(C)Cc1ccoc1Br 42977,c1(CC)cc(F)ccc1C(=O)N(CC(C)(C)CNC(c1ccc(NC)nc1)=O)C 42978,c1(SCC(=O)NC2COCCN(C(CC(=O)OC)=O)C2)ccc2c(c1)CCC2 42979,N1(C(c2cccc(COC)n2)=O)CCN(C(=O)C(F)C2CCOC2)C2(CCC2)C1 42980,N1(C(C(CC)(O)c2ccccc2)=O)CCCN(C(=O)Cc2ccn(C)n2)CC1 42981,C1(C(=O)NC(CC2CCN(C(C(C)N3CCC3)=O)CC2)C)CN(C)CCN(C)C1 42982,N1(C(c2cncs2)=O)CC(CNC(c2cc(-c3ccccc3)on2)=O)C2CC12 42983,N1(C(CCNC(=O)NC)=O)CCCCC(NC(C2(O)CCC2)=O)CC1 42984,c1(C(=O)NCCN(C(C2C(C(=O)OC)C2)=O)C)nnn2c1CSCC2 42985,C(CCCCC(=O)NC(C)CCC(=O)N(C)C(c1ccccc1)C)=CC 42986,C(C)(CCCN=c1nc(C(C)C)c2ncccc2[nH]1)N1CCC(=C)CC1 42987,C=CC(C)C(C)C(=O)NCC1(NC(=O)CC2CS(=O)(=O)C2)CCCC1 42988,c1(C(C2(CC)CC2)NCc2n(CC)nnn2)cc(Br)cc2c1OCC2 42989,CC1CN(C(c2ccc(CC#N)o2)=O)CCCN1C(C1(CC#N)CCCC1)=O 42990,c1(CN2CC3(OCC(C(=O)NCC4(F)CC4)C3)C2)nccc2[nH]ccc12 42991,C#Cc1cc(C(=O)NC2C3CC(NC(C45CSCC4C5)=O)CC23)ccc1C 42992,c1(C(=O)NC2CN(C(C(COC)(F)F)=O)C2)cn2c(n1)CC(C)CC2.C1CCCC1 42993,C(=O)(N=c1cc[nH]c(C)c1F)C1C(c2c3nc(C)[nH]c3ncn2)CCCC1 42994,c1(OC)cnc(N2CCN(C(=O)C(=O)Nc3cc(CCN(C)C)[nH]n3)CC2)nc1 42995,N1(C(c2n(CC=C)ccc2)=O)CC(NC(=O)C(O)Cc2[nH]cnc2C)CCC1C 42996,C(c1c(N)cnn1C)=CC(N1CC(C)C(CNC(c2ccc(F)cn2)=O)C1)=O 42997,c1(C(=O)NCC(CN(C)C(c2ccc(N)c(F)c2)=O)(C)C)nn(C)c2c1CCC2 42998,Cc1oc(C(=O)N(C2CN(C(C3C(C)C3(F)F)=O)CC2O)C)cc1S(N)(=O)=O 42999,CC(C)C(C)CC(N1CC(CCCC(=O)OC(C)(C)C)C1)=O 43000,c1(NC(CC)CNC(c2csc3cncn23)=O)ccc([N+](=O)[O-])cc1[N+](=O)[O-] 43001,CC(C)CC(O)C(C)C(=O)N(C)Cc1ccc2ccccc2c1 43002,N1(C(C2C(C(C)C)OCC2)=O)CCC(CNC(C2CCN(C3COC3)C2)=O)CC1 43003,c1(CC)cccnc1C(=O)NCCC1(O)CCN(C(=O)C(C)OCCC(C)C)C1 43004,c1(C(N2CCN(C(c3c(C)ccnc3O)=O)CC2C)=O)cccc(C#N)c1Br 43005,O=S1(=O)CCCC(NC(c2nnnn2C2CCCCC2)CC2(CO)CC2)C1 43006,c1(-n2cc(CC(N3C(C(=O)O)CCC3)=O)nn2)nnc(O)nc1O 43007,c1(OC)cc(C(=O)N(C2CN(C(C3(C)CCCS3)=O)C2)C)sc1S(N)(=O)=O 43008,C(CNC(=O)CCc1nnc(S)n1C)(CC(F)(F)F)NC(C(C)SCCCC)=O 43009,c1(CNC2C(C(=O)Nc3cc(OCC)n[nH]3)C2)c(F)cc(Br)c(F)c1F 43010,CCC(C)C(O)CC(=O)N1CC(F)CC1C(=O)NC1CN(S(C)(=O)=O)C1 43011,c1(C(=O)NC2CCN(C(CCCCOCCC)=O)C2)c(C)nn2cc[nH]c(=O)c12 43012,S(=O)(=O)(c1cccc(=NC(C)c2ccc(Br)cc2)[nH]1)C1C(OC)CS(=O)(=O)C1 43013,CCCN(OC)C(=O)CC1CCN1C(c1cn(CCC2CC2)nn1)=O 43014,C1(OC)CN2CC1OCc1c(cccc1)C2=O.C1(CNC(C)=O)CCOCC1 43015,N1(C(C2(C(F)(F)F)C(C)C2)=O)CCc2cc(C(=O)Oc3ccccc3)ccc2C1 43016,C1(C(=O)NC(C2CCN(C(=O)CCc3cccnc3)CC2)C)CCCCC(=O)C1 43017,CC(C)C(C(=O)N(C)CCNC(=O)C(c1ccc(F)cc1)O)NS(C)(=O)=O 43018,C1(N(C(=O)C(C)n2cncn2)CC)CCCN(C(=O)CCn2c(C)csc2=O)C1 43019,CCCC(C)CC(=O)NCCOCCCNC(=O)CC=C(Cl)Cl 43020,CC1CC(NC(c2ccc(Cl)nc2O)=O)c2nccn21 43021,N1(C(CNC(=O)OC)=O)CCC2CCCC12C(=O)Nc1cncnc1 43022,CC(C)C(C(C)NC(=O)CCSC(F)(F)F)NC(C12CCN(CC1)C2)=O 43023,C12(CNC(CCc3c(C)nn(C)c3)=O)CCC1CN(C(=O)CN1CCCC1=O)C2 43024,C(=O)(C(F)C(C)C(F)(F)F)NCC12CCC(CNC(CC=C)=O)(CC1)CO2 43025,Cc1cncc(CC(=O)NC2CC(NC(c3cn(-c4nccs4)cn3)=O)C2)c1 43026,c1(OCC2(OC)CCOC2)cc(CC(=O)OC(C)C)cc(Br)c1 43027,c1(C(=O)NC(CN(C)C)C(=O)NCC#CC(F)(F)F)ccc(C#N)n1C 43028,C1(NC(C(c2ccccc2)OC)=O)C=CCN(C(c2cc(C)ccn2)=O)C1 43029,Cc1ncc(C(=O)NCC(C)CNC(=O)Cn2c(C)c(C)sc2=O)c(C2CC2)n1 43030,c1(C(=O)NCC2N(C(C(CCOC)OC)=O)CC(OC)C2)scc2c1CCCC2 43031,Cn1cc(-c2nc(C(=O)N(CCn3cnc(C(F)(F)F)c3)C3CC3)cs2)cn1 43032,C1(C(=O)NCC#CCCO)(CC)CCN(C(=O)C(C2(O)CCCC2)F)CC1 43033,C1(NC(c2c(CC)ncnc2)=O)CN(C(=O)CCc2cccc(F)c2)C2CCCC12 43034,C1(c2n(CCSC)nnn2)(NCC2CC2(C)C)CCOCCC1C 43035,N=c1ccc(C(N2CCCC(NC(=O)COc3ccc(Cl)nc3)C2)=O)c(Cl)[nH]1 43036,c1(CNC(C(=O)Nc2c(C)cn(C)c2)=O)ccc(C(F)F)c(Cl)c1 43037,C1(CN(C2CC(C)CCO2)CC)CCCN(C(=O)CCCc2cncs2)C1 43038,CC1CC(O)CCN(C(=O)CC(C2CC2)NC(c2cnn[nH]2)=O)C1 43039,C1(C(=O)NC2(C(COC)O)CC2)CC(C)(C)CN1C(=O)C(n1ccc(C)n1)C 43040,c1(NC)cc(C(N2CC(NC(C3CC(O)CN3C(N)=O)=O)C(C)C2)=O)cc(Cl)n1 43041,C1(C(CCC)C)CCCCN1N1CCC(CCO)(C(=O)OCC)CC1 43042,N12CCC13CC(O)CCC3C1=CC=CC=CC(CCOC)NC1CNC(=O)C2=O 43043,c1(C(=O)NC2C(C#N)CN(S(=O)(=O)C(F)(F)F)C2)ccc2cccc(C(F)F)c2n1 43044,C1(C(=O)N(C(C)CO)C)(NC(CNC(CC(C)C)=O)=O)CCN(C)C1 43045,Nc1ccc(C(=O)NCCCOCCNC(=O)C=C(Cl)Cl)cc1OC1CC1 43046,c1(C(=O)NC(CN(C(C(C)OC2CCCCC2)=O)C)C)cccn2cnnc12 43047,c1(C(C(=O)NCC(CNC(c2ccc(OC)s2)=O)F)(C)C)ccc(=O)n(C)c1 43048,C(=O)(CC(C)C(F)(F)F)NCCCC(C)NC(C(C(C)C)C)=O 43049,C1(C(=O)NCC2CCCOC2)COCCC12CN(C(c1cc(C(F)F)no1)=O)C2 43050,FCCCN=C(NCC1(c2ccc(F)cc2)CCC1)NC1CC1C(F)F 43051,C(=O)(CCC(=O)N1CC=CC1CNC(=O)C(O)CC1CCCC1)NC 43052,C1(C(=O)OCC)(CCOCCN(C(=O)C(C)n2cnnn2)CC)CCOC1 43053,N1(C(CCOC)=O)CCN(C(c2cc(N)ccc2O)=O)C2CCC12 43054,c1(NC(c2n(CCCF)nnn2)c2cnc(-c3cccs3)o2)cc2n(c1)CCCC2 43055,c1(N(C(C2C3(C(=O)OC)CCCCC32)=O)C2CC2)nc2ccc(C)cc2s1 43056,C1(C(=O)NCCCN(C(C(c2ccccc2F)OC)=O)C)NC(=O)OC1C 43057,N1(C(C(C)C#N)=O)CCC2(CC1)C(NC(C13C4CC(CC14)C3(F)F)=O)CS2(=O)=O 43058,Cc1cc(C(=O)NC2CC2NC(=O)C(C2CCCCC2)C)cnc1C 43059,c1(C23CC(C2)C3)ccc(F)c(F)c1.N12CC=CC1CN(C(C1CCCN1C)=O)C(C)C2=O 43060,Cc1cc(C)c(C(=O)N(CCC(C)NC(=O)C=C2CCSCC2)C)c(=O)o1 43061,c1(CN(C(C2N(CC)CC2)=O)C)cnn2c1CN(C(=O)COC1CCOC1)CC2 43062,c1(CC(C(=O)NC(CN(C)C(c2ccncc2O)=O)(C)C)O)cccc(Cl)c1 43063,N1(C(C(=C)C)=O)CC12CN(C(c1ccc(NCc3ccncc3)cc1)=O)C2 43064,c1(C(N2CC(NC(=O)Cc3cc[nH]n3)C(F)C2)=O)cccc([N+](=O)[O-])c1Cl 43065,N1(C(C(CC(C)C)N(C)C(C2COCC2(C)C)=O)=O)CCc2cnccc2C1 43066,c1(CC2CCCN(CC(=O)NC(CC=C)C(=O)O)C2)c(F)ccc(Cl)c1F 43067,C(CS(=O)(=O)CC(=O)N1CC2(C1)CN(C(=O)CCCCC(C)C)C2)OC 43068,c1(N(C)CCC2CCCN(C(C3CCS(=O)(=O)CC3)=O)C2)ccc2ocnc2c1 43069,N1(C(CC=C)=O)Cc2[nH]nc(C(=O)NCC(COC)C(C)C)c2C1 43070,N1(C(c2c(C)n[nH]c2C)=O)CCCC1C1CCCN1C(c1csc(C#N)c1)=O 43071,Cc1c(C(C)(C)NC(c2ccc(C#N)cn2)=O)cc(F)cc1[N+](=O)[O-] 43072,N1(C(c2c(CC)csc2)=O)CCC2(CCN(C(=O)COC)C2)C1 43073,C(=O)(C(C)(C)CC(C)(C)C)NC1CC(C)N(C(C2CCSC(C)C2)=O)C1 43074,Cc1cc(C(=O)NC2C3CC2CN(C(=O)C(C)C(C)C)C3)c(N)c(C)c1 43075,c1(C(=O)NCC2CN(C(=O)C(C3CC3)C3CC3)CC23CC3)ccc2ocnc2n1 43076,CC(C)CC(C)(O)C(=O)NCCC1CCCN(C(c2ccc(Cl)cc2F)=O)CC1 43077,C1(C(=O)NCC2(C)CSC2)CNC(=O)CN1C(=O)CN1CC2CC2C1 43078,c1(NC(CC(C)N(C(C(CCOC)C)=O)C)=O)ccc2nccn2c1 43079,C1(CCCC)CN(C(=O)Cc2cnn(C)c2C)CCN1C(C1COCCO1)=O 43080,C1(OC(C2CC3CC2CO3)=O)CCOC2(CCCCC2)C1 43081,C(CCC(C)(C)C(=O)NCc1nonc1C)NC(C(=Cc1ccco1)C)=O 43082,C=CCC(CC(=O)Nc1cnc(Cl)cc1C)NC(=O)CCC1OCCO1 43083,c1(C(N2C(CN(C(=O)CC#N)C)CCC2)=O)cnn2c1CCC2 43084,N1(C(CC(C)(C)O)=O)CCCC2CN(C(=O)CC3CCC(=O)CC3)CC12 43085,C1(N(C(=O)CCCCCF)C)CN(C(=O)C(C)(C)CC#N)CC1(C)C 43086,C#CCC(CC(=O)N(C)Cc1nnc(C)o1)NC(=O)CNC(=O)CC(C)C 43087,c1(C(=O)NC)cncc(N(c2cccnn2)C)n1 43088,C(C(C)C(C)C(=O)NCC1(CCCNC(=O)Cc2ccnc(F)c2F)CC1)OC 43089,c1(CCC(=O)NCC(C)CNC(c2ccc(C#N)s2)=O)n[nH]c2ccccc12 43090,N1(C(c2ccc(C(=O)OC)o2)=O)CCCC1(C)CC(=O)Nc1ccsc1 43091,C(=O)(C1CCCc2nccn21)CCNC(C1CN(C(c2nccc(N)c2)=O)C1)=O 43092,Cc1sc(Cl)nc1C(N1CC(NC(c2cc(C(N)=O)c[nH]2)=O)CC1C)=O 43093,C1(C(=O)NCC(=O)OCCC)N(C(=O)C(C)SC(C)C)CCC1(C)C 43094,Cc1ncnc(C)c1C(=O)NCC1CC(F)CN1C(C1CC1(C)C(F)F)=O 43095,N1(C(C(C)CS(C)(=O)=O)=O)CCN(C(=O)CC(=O)Nn2cncn2)C2(CCC2)C1 43096,N1(C(C=C(CC)CC)=O)CCC(O)(CCNC(=O)C(c2csc(C)n2)=O)CC1 43097,C(c1cncc(C)c1)=CC(=O)NC(CC)CNC(=O)CSCc1cscn1 43098,c1(C(C(=O)N(CC(F)Cl)C)N(C)C)ccc(OC(F)(F)F)cc1 43099,CCCC(CCCS(C)(=O)=O)C(=O)N(CCCCN(C)C(C1CCO1)=O)C 43100,c1(C(N2CCC(NC(C3(C)CCC(C)CC3)=O)C(O)C2)=O)c(F)cc(Cl)cc1F 43101,c1(CC(N2C(C(=O)Nc3cncc(OC)c3)CC3CC32)=O)cc(Cl)ccc1Cl 43102,c1(C(C)=O)cc(C(=O)N(C2CCN(C(=O)Cn3cc(Cl)cn3)C2)C)cs1 43103,C1(C(N2C(CC#C)CCCC2)=O)CN(C(=O)CCc2cnn[nH]2)CCN1C 43104,c1(C(=O)NC2CCN(C(C3COC(=O)O3)=O)CC2O)cnc2c(c1)C(=O)CCC2 43105,C1(O)(CN(C(C2(CCC=C)CC2)=O)C)CCN(C(=O)CCS(C)=O)C1 43106,N1(C(CC(C(C)C)OCC)=O)CCN(C(c2c(C)cccc2Cl)=O)CC(C)(C)C1 43107,C(=O)(CCC(C)(F)F)NCC(C)C(=O)NCCN1CC(C)(O)C1 43108,N1(C(C(C=C)(C)CC)=O)CC(C2CN(C(c3[nH]c(=N)sc3CC)=O)C2)C1 43109,c1(N2C3C(NC(=O)CC4CCOC4)(CCC3)CC2)ncnc2[nH]ccc12 43110,N1(C(Cn2ncc(C)c2)=O)CCCCC1c1cn(CCN2CCC2CO)nn1 43111,C(CC)(CCCC(=O)NCc1cc(C#N)cs1)NC(C1(CC#C)CC1)=O 43112,C(CCC(N)=O)(C(=O)N1CCC(C(=O)NCCN=S(C)(C)=O)C1)N(C)C 43113,CCCCC(CC)C(=O)NC(C)(C)CN(C(=O)C(=O)Nc1ccc(F)cc1)C 43114,C1(C)(CNC(CCN(CC=C)C(c2cc(N)cc(F)c2)=O)=O)CCCCC1O 43115,C(CCC(C)C(=O)NCC1(F)CC(CNC(=O)COC(C)=O)C1)OC 43116,C(=O)(C1Cc2ccccc21)N1CCCC(N(C(CC2(COC)CC2)=O)CCF)C1 43117,c1(C(N2C(CNC(=O)C(=O)NC3CC3)C=CC2)=O)cc2cc(F)ccc2s1 43118,c1(C(=O)NCC2CC2CNC(c2n[nH]cc2C2CCC2)=O)csc(Cl)n1 43119,Cc1nc(N2CC3C(NC(c4cc(C(F)(F)F)n(C(C)C)n4)=O)C3C2)[nH]c(=N)n1 43120,c1(C(=O)N)cccc(CO)c1.C(CC)(C(=O)N1CCCC1Cn1cncn1)OCC 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43173,N(C(=NCCC(C)=O)NC(C1(O)CCOCC1)C)Cc1cnn(CC)n1 43174,CCC(O)(C(=O)N(CC(O)CNC(=O)CN(C)C1CC1)C)c1ccccc1 43175,C1(COC)CC(CNC(=O)COC2CCCC2)N(C(C2CCC(F)C2)=O)C1 43176,C1(C#N)(C(N(C2CC(NC(C(C)Sc3ccc(C)cc3)=O)C2)C)=O)CC2CC2C1 43177,CC(C)(CCl)C(=O)N(C1CC2CC1CN2)Cc1cccnc1 43178,C12(CCOCC1)CS(=O)(=O)N2.c1(CN(CCOC)C)ccc(C(F)F)cn1 43179,N1(C(c2ccn(CC)c(=O)c2)=O)CCCC2CN(C(C3(c4cccs4)CC3)=O)CC12 43180,c1(OC(=O)CCCNC(c2ccc(Cl)cc2)=O)cccc2c(I)n[nH]c12 43181,Cc1ccc(NC(C2CCN2C(C2CCCO2)=O)=O)cc1C 43182,C1(C(NOCC(=O)NC(CCOC)C(N)=O)=O)CCC(=O)C(C)C1 43183,C12(C(=O)NC(CN(C(C=C(C)C(C)C)=O)C)(CO)CO)CC3CC1C2C3(F)F 43184,Cc1cc(C(F)F)nn1CC(N1CC2C(NC(C3COC(=O)O3)=O)C2C1)=O 43185,C1(C(N2CCC(N(C(=O)Cn3cc(Cl)cn3)C)C2)=O)(OC)CCCOC1 43186,c1(C(N2C3CCC(NC(c4cc5sccc5s4)=O)(C3)C2)=O)nnn2c1CCCC2 43187,Cc1cc(NC(C2CC(F)CN(C(c3cc(Cl)cnc3Br)=O)C2)=O)cnc1C#N 43188,Cc1c[nH]c(C(=O)NCC2CCC2C(=O)NCC2CNC(=O)C2)c1 43189,Cc1cccc(OCC(=O)N(C(C)CNC(C2(S(C)(=O)=O)CC2)=O)C)c1F 43190,Cc1c(NCC(C2CCCCCC2)(C)C)ncnc1N1CCOC(C2CC2)CC1 43191,C12(NC(CCC(=C)Br)=O)CCC(C1)N(C(C1CC(C3CC3)=NO1)=O)C2 43192,N1(C(C=Cc2ccc(SCC)o2)=O)CCCC2C1CCN2C(=O)CN(C)C(N)=O 43193,c1(OCC)ccccc1C(=O)N(C1CCN(C(=O)C(C)c2cccs2)CC1)C 43194,CC(C)(CC(F)C(=O)N1CCC(n2nccn2)CC1)NC(=O)CSCC(F)F 43195,C1(C(=O)NCC2CN(C(CN(C3CC3)CC)=O)CC2C)CN2CCCC2CO1 43196,CC(N=c1[nH]c(=NCC(CO)C(F)(F)F)c2c(ncn2C)[nH]1)c1nncs1 43197,c1(OC)cc(CC(N2CC3CC(NC(=O)CCC(N)=O)C2C3)=O)cc(OC)c1O 43198,C1(CNC(=O)Cn2cnnn2)CCN(C(c2cnn(C(F)(F)F)c2)=O)C12CC2 43199,c1(NC(C(N2C(C)CC(NC(C3(CCOC)CC3)=O)C2)=O)=O)ccc(C)c(C)c1 43200,CCCC(C(=O)N1CC(C(=O)NCC2CCC2C)C1)OC 43201,Cc1cc(C(=O)NCCN2CCC(NC(=O)CC3CCCOC3)CC2)nn1C 43202,C1(C(N(CCNC(c2c(C)snc2)=O)C)=O)CNC(=O)CC12CCOC2 43203,c1(OC)ccccc1C1CC1C(=O)N(CC(C)(C)NC(c1nn(C)cc1C)=O)C 43204,N1(C(C2CCCCN(C(c3ccc(C)n3C)=O)C2)=O)CCOC2CN(C)CC12 43205,n1(CC)nc(C(=O)N(CCCC(=O)NCC(C2CCCC2)C)C)c(C)n1 43206,c1(C(=O)NCC23C(CN(C(C(CC)SC)=O)C2)C3)ccc(F)c(C(F)(F)F)c1 43207,C1(CC)(CNC(c2cc(CNC(=O)C(C3(O)CCCC3)F)on2)=O)CC1(F)F 43208,c1(OC)cc2[nH]ncc2cc1C(N1CCC1(C)C(=O)Nc1cc(Br)nc(Br)c1)=O 43209,C1(C(COc2cn(CC)nc2)=O)CC2CCC1N2C(=O)NC1CN(C)C(=O)N1 43210,C1(c2c(C)nccc2)CN(C(=NCCC2CCC2)NCc2ccnn2C)CCO1 43211,n1(CC)cc(C(N2CCC(CN(C)C(c3cscn3)=O)CC2)=O)cc(Cl)c1=O 43212,C1(N(C(C(CCC)OC)=O)C)CC2CCC(C1)N2C(=O)CN1CCC(CO)CC1 43213,C1(CNC(C(C)OCCCC)=O)CC2(CC(NC(=O)CS(=O)(=O)N(C)C)C2)C1 43214,c1(Cc2nc(-c3cc(F)ncc3Cl)on2)ccc2c(c1)COC2 43215,N1(C(C2CCN(CC(C)C)CC2)=O)CC(NC(=O)Cc2cnns2)CC12CCC2 43216,Cc1cc(C(=O)N(CCC(C(C)C)NC(c2snnc2C(C)C)=O)C)cnc1O 43217,c1(C(=O)NC(CC)CCc2ccco2)cncc2cnccc12 43218,c1(C(C(N2CCCC(CN(C(=O)Cc3ccccc3)C)C2)=O)O)cccc(F)c1F 43219,C12(CC(=O)NCCCCNC(c3nccc(N(C)C)c3)=O)CCCCC1C2(F)F 43220,C1(C(=O)Nc2cccc(N3CCC(NC)CC3)c2)Cc2ccccc2CO1 43221,N1(C(C(C)C(C)S(C)(=O)=O)=O)CCCC(C2(NC3CCCC3(F)F)CC2)C1 43222,c1(OC)cccc(CN(C(=O)C(=O)N(C)CC2CCC3CC23)C)c1 43223,Cc1cn(C)nc1C(N1CCCCC1CC(N1CCCC1(C)C1CCC1)=O)=O 43224,CCCC(CCCNC(C1C2(CC2)C12CC2)=O)NC(C1CCNC(=O)C1)=O 43225,C(=O)(C(C)(C)CNC(=O)Cn1ccnn1)N1CC(OC)C1 43226,Cn1cnc2sc(C(=O)NCC(C3CC3)NC(C3CSCC(=O)N3)=O)cc12 43227,N1(C(CSCC#C)=O)CCN(C)C(CNC(C2(c3ccccc3)CC(O)C2)=O)C1 43228,c1(N(C(c2cccc(C)c2O)=O)CCN2C(=O)CSC2=O)ccc2c[nH]nc2c1 43229,C1(NC(C=CCCC(C)C)=O)CCCN(C(c2cnn(C3CC3)c2)=O)CC1 43230,c1(C(=O)NC2CCN(C(=O)CCn3ccnn3)C2C2CC2)cc2ccsc2s1 43231,c1(C(=O)NC23CC(C2)N(C(C2(C(F)(F)F)CCOCC2)=O)C3)ccc(O)nc1Cl 43232,CC(C)(CN=c1[nH]c(=NCc2ccc(F)cc2Br)[nH]c2ccccc12)C1CCC1 43233,N1(C(c2c(C)cn(C)n2)=O)CC(NC(C2COCC(C)O2)=O)C2(CCCC2)C1 43234,Cc1cc2c(C(=O)NC3CCCCC3N(C)C(c3cc[nH]n3)=O)nccn2n1 43235,C1(NC(C2CN(C)C(=O)CC2)=O)CCC2CN(C(=O)CSCC(F)(F)F)CC2C1 43236,CCCCC(C)CCC(=O)N1C2CC3CC1CC(C2)O3 43237,N1(C(C(C)C(F)F)=O)CC(CNC(C2(c3cccc(C#N)c3)CC2)=O)CC1(C)C 43238,N1(C(C2(C=C)CC2)=O)CC(NC(c2cc(C(F)F)cc(F)c2)=O)CC2(CCC2)C1 43239,c1(C(=O)NCCCCCN(C)C(c2ccc(Cl)cn2)=O)cc2n(c1)CCOC2 43240,c1(-c2cc(NC(N3CCCC(C(=O)OCC)C3)=O)[nH]n2)ccc(F)c(C)c1 43241,C(=O)(C1=C(F)CN(C(=O)C(=C2CCCCC2)F)CC1)N1CC(OCC(N)=O)C1 43242,C1(C(=O)OCC)CC2(CCN(C(c3c(C(F)(F)F)cccc3O)=O)CC2)C1 43243,n1(C(C)C)cc(C(N2CCC3(CC3C(N3CCCC(C#N)C3)=O)C2)=O)ccc1=O 43244,c1(C(=O)NC2CCCC(NC(C3CC3F)=O)C2)cnc2[nH]ccc2n1 43245,Cc1cnc(S(C)(=O)=O)nc1N1CCC2(C(N3CC(CO)C(O)C3)=O)CC2C1 43246,N1(CCC)CCC(C(=O)NC2CN(C(=O)OC(C)(C)C)C2)C(O)C1 43247,CC1Cn2nc(C(=O)NCC(CC(F)(F)F)NC(=O)C(=O)N(C)C)cc2C(=O)N1 43248,c1(CC(=O)N(C)CC2COCCN2C(=O)CC2(C)CCC2)ccc(F)cc1Cl 43249,C(=O)(CCCN(CC)C(c1ncc(C)cc1C)=O)N1C(C#C)CCC1 43250,c1(N(C)C)ncnc(NC(C2COCCN2C(=O)OC(C)(C)C)=O)n1 43251,c1(-n2c(-c3c(CC)nc(C)[nH]3)nc(-c3ccccn3)n2)ncc(Br)cc1C 43252,C(N=c1[nH]c(=NCCc2nccc(O)n2)c2[nH]ccc2[nH]1)c1c(C#N)cccc1 43253,C(CCSC)(C(=O)NC(C1CCCCC1)CNC(=O)C(C)N1CCCC1)OC 43254,CC(C)CC(O)CC(=O)N(CCC(=O)NCCn1ccc(=O)cc1)C1CC1 43255,c1(CNC(c2cc(CCC)on2)=O)cccc(C)c1.c12occc1C(=O)N(C)C2 43256,c1(OCC)cc(NC(c2cnc(Cl)cc2NC(C2CC2C2CC2)=O)=O)ccc1O 43257,c1(OC)ccccc1NC(=O)C(C1CN(C(=O)CC2(OC)CCC2)C1)OC 43258,C1(c2nc(CSC3CCSC3)no2)(CC)CCC(=O)NC1 43259,N1(C(c2nc(C)oc2C)=O)CCOC2CCN(C(C3CCC(F)CC3)=O)CC12 43260,N1(C(CCOCC#C)=O)C2CCC1CN(C(=O)Cc1ccccc1CC)C2 43261,C1CCc2ccnn2C1.Cc1cc(C(=O)N2CC(n3cc(C(C)C)nn3)CO2)cnc1Cl 43262,C1(C(N(CC(=O)NC)CC)=O)CC12CCN(C(=O)Cc1ccc(C)nc1)CC2 43263,C1(NC(=O)CC(Cc2ccccc2)CO)CCCC2CCCCC12 43264,C(=O)(CCCC(F)F)N1CC(N2CCN(C(CCSc3ncc(CC)s3)=O)CC2)C1 43265,N1(C(c2ccc(F)cc2)=O)CC2ON=C(CNC(C34CCC(CC3)OC4)=O)C2C1 43266,N(C(=NCC)NCCN(C1CCS(=O)(=O)C1)C)CC(CC)N(C)C 43267,Cn1ncc2c(C(=O)NC3CN(C(=O)Cn4cc(Cl)cn4)CCC3F)ccnc12 43268,CC1(C)CC(C(N2CCCCC2CCNC(=O)CC2COC(=O)C2)=O)CO1 43269,CC12CN(C(=O)C3=COCC3)C(C(=O)NC(c3cscn3)CO)(C1)C2 43270,N1(C(c2c(C)n(C3CC3)cc2)=O)CCOCCC1C(F)(F)F 43271,C1(C(N2C3CN(C(C(CC(C)C)O)=O)C(C3)C2)=O)CCn2nncc2C1 43272,C12(NC(C(C(C)C)NC=O)=O)CCN(C(c3cc([N+](=O)[O-])n[nH]3)=O)CCC1C2 43273,Cc1cccc(NCCC(N2CC(CNC(c3cccnc3S)=O)C(C)C2)=O)c1 43274,C(C(S(C)(=O)=O)C1CC1)NC(c1ncccc1F)c1n(CCCOC)nnn1 43275,C1(C)(C(=O)NC2CC(C)N(C(c3ccon3)=O)C2)CCC(C)(C)CC1 43276,CCC(C)CC(C)C(=O)N1CCC(C)(NC(c2cc(=O)c(OC)cn2C)=O)CC1 43277,N1(C(CSCC(C)C)=O)CCCC1SCCNC(C(C)=CCC)=O 43278,N1(C(c2c(OC)nccc2)=O)CCCC(C2CCN(CCO)C2)C1.C(CCCCCl)S 43279,N1(C(C(C)SC)=O)CCC(NC(=O)COc2ccc(F)cc2F)C(F)(F)CC1 43280,C1(NC(c2n[nH]c(CC)c2Cl)=O)CCN(C(=O)C(C)OC2CCCC2)CC1C 43281,Cc1cccc(O)c1C(N1CCCC(Nc2nnc(C3CC3)o2)CC1)=O 43282,N1(C(C2CN(C(COC(CC)CC)=O)CC2O)=O)CCN(C)C(CC)C1 43283,N1(C(CSc2c(C)n[nH]c2C)=O)CCC(NC(=O)CN2CCCNC2=O)CC1C 43284,N1(c2ncc(C#N)nc2)CCC(CNC(c2cnc(C3CC3)s2)=O)C(F)(F)CC1 43285,N1(C(c2n(CC#C)ccc2)=O)CCC2CN(C(=O)CCC)CCC2C1 43286,CC1CCC(NC(C2CCC2)=O)CN1C(C1CC(=C(F)F)C1)=O 43287,CC1(C2CC2)CCCN1C(=O)Cn1cc(I)nn1 43288,c1(C(N2CC(NC(c3cc(C)sn3)=O)C(F)C2)=O)cc(F)c(C)cc1F 43289,C(=O)(CCCCC(N)=O)N1CCCC(C)(CNC(=O)CCc2nc[nH]n2)C1 43290,c1(-c2cn(CC(C)NC(C(COC)(C)OC)=O)nn2)c(C)cc(Cl)cc1N 43291,C(=O)(C(C)(F)C(F)(F)F)NCC1CCN(C(C=Cc2ccc(C)cc2)=O)C1(C)C 43292,C1(C)(CNC(C(CC)SC)=O)CN(C(C2(CO)CC(F)(F)C2)=O)CCO1 43293,C1(C(=O)NC(CC=C)CNC(=O)Cc2ccc(C)o2)CCOC(C)(CC)C1 43294,C1(CC(=O)N(C2CCN(C(=O)C(C)NS(C)(=O)=O)CC2)CC)CCCC2(CC2)C1 43295,C12(NC(CCC(N)=O)=O)CC(CNC(C3CCS(=O)(=O)C3(C)C)=O)(C1)OC2(C)C 43296,CCCCCC(C(=O)N1CCC(CF)(NC(=O)CCc2cn[nH]c2)C1)C(C)C 43297,C(=O)(C(CCC(=O)OCC)N1CCCC(c2ccn(C)n2)C1)NCCC 43298,c1(C(=O)NCCCC(C)NC(C2CN(C)C2)=O)nc(Cl)sc1Cl 43299,CC1(C)CCCC(CNC(C2CCC(NC(C3(C#N)CCCO3)=O)CC2)=O)O1 43300,CC(C(C)(C)C(=O)NCCC(=O)NC(C)(C)C)NC(c1cc(Cl)ns1)=O 43301,C12(NC(CC=CC=C)=O)CCC(CN(C(C3(NC(N)=O)CC3)=O)C1)C2 43302,CN1CCN(C(C2CCOC2CNC(=O)C(F)C(C)(F)F)=O)CC1C1CC1 43303,C1(NC(C2(C(C)C)COC2)=O)CC(NC(=O)CC2(N(C)C)COC2)CC1O 43304,C1(N(C(C(C)(F)F)=O)CCO)CCN(C(c2ccn(-c3ccccc3Cl)n2)=O)CC1 43305,Cc1nc(C)c(CC(=O)NCCCN(C2CCCC2)C(c2ccc[nH]2)=O)[nH]1 43306,CC1CC(Cc2ccccc2)CCN1CC(=O)OCC1CCOC1 43307,C=C(CN)CCNC(=O)COCCCNC(CCNC(C)=O)=O.O(C(F)(F)F)C(=O)C 43308,c1(C(=O)NCC2(CNC(C=CCOC)=O)CC2)cn(C)c2nc(C)ccc2c1=O 43309,C1(NC(C=C(CCC)C)=O)C(C)CCN(C(c2ncc(C(C)=O)s2)=O)C1C 43310,C1(C)(C(=O)NCC2N(C)C(=O)CC2)CCCN(C(c2cccc(Cl)c2F)=O)C1 43311,C(CC1CCCO1)(C(=O)NC(c1cscn1)CO)NC(=O)CCn1cncn1 43312,c1(C(N2CC(C)(C)C(CNC(=O)CCC#N)C2)=O)ccc2cncn2c1 43313,C1(NC(C(CC)SC(F)(F)F)=O)(NC(=O)CSC)CCCC1C 43314,C1(C(N2CCCC(F)(C(=O)NCCc3nc(C)sc3)C2)=O)CC(=O)CC12CCC2 43315,N1(C(C)=O)CC(O)CC1C(N1CCC(C(C)NC(=O)Cn2nc(C)oc2=O)C1)=O 43316,c1(OCCOC)ncccc1C(=O)NCCC(C)NC(=O)CC1CCC(C)(C)C1 43317,N1(C(COCC)=O)CC2CC1C2CNC(=O)C(C1CCC1)OC 43318,c1(OCC(N2CCC(N(C(=O)C(O)CC3CC3)CC)CC2)=O)cc(C)cc(C)c1 43319,C(=O)(CC(C)(C)N(C(=O)CN1CC2CC2C1)C)N(CC(C)C)CC(N)=O 43320,C1(CNC(C(C)SC)=O)CN(C(c2ccc(C(F)(F)F)cc2N)=O)CC1(F)F 43321,C1(CCNC(C(c2cscn2)OCC)=O)CCCN1C(=O)CC1CC(SC)C1 43322,c1(C(=O)NCC2N(C(C(N3CCCC3)C)=O)CCCCC2)cc2ncccc2o1 43323,C1(NC(N(CCCn2cc(C3CCCCC3O)nn2)C)=O)CCCC(C)(C)O1 43324,C(=O)(C(CO)C(F)(F)F)NC1C=CCC(C(N(C(CC)CC)CC(C)C)=O)C1 43325,N1(C(c2c(C)nsc2)=O)CC(C)CN(C(=O)COC2CCC2)CC1C 43326,c1(N2CCCC(=C)C2)nc(=NCC2CCC3(CCCC3)C2)[nH]c2c1CC(C)CC2 43327,C12CC3(C1)CN(C3)C(=O)N2.S(S(C)(=O)=O)NC(C1CC1C(=O)N(CC#C)C)=O 43328,C1(NC(C2CC2CF)=O)COC2CN(C(C3(Cc4ccncc4)CCC3)=O)CC12 43329,O=C(N=c1ccn(Cc2ncccn2)[nH]1)C(=O)NC(c1ccc(F)cc1)CCO 43330,C1(NC(N(C(C2CCC2)C)CC)=O)(OC)CCC1 43331,C1(CNC(C(C)OC)=O)CN(C(c2ccc(-c3ccccn3)s2)=O)CC12CCC2 43332,c1(OC)ccc(C(=O)NC2CCC(NC(=O)CCC3CCOC3)CC2)nn1 43333,C12(C(N3CCC(CCC(=O)NCC4(C)CC4)C3)=O)CC(C)(CCO1)C2 43334,C(C(CNC(c1c(C)cnnc1O)=O)C(F)(F)F)NC(C(C#C)(C)C)=O 43335,c1(C(=O)NCC23N(C(c4c(C)ccs4)=O)CCC2C3)cn2cccnc2n1 43336,C12(NC(CCCC#C)=O)CCCCC1N(C(=O)Cc1ncccc1C)CC2 43337,Cc1cccnc1C(N1CC(OCCC(=O)NCCC[Si](C)(C)C)C1)=O 43338,C1(C(N2CC(NC(c3cccc(O)n3)=O)(CO)C2)=O)CCC2CCCCN12 43339,C(=O)(C(C)(C)CC1CCOC1)N1CC(N(C)C(C2CCCC2F)=O)C1 43340,N1(C(CSC)=O)CCC2CN(C(c3cc(-c4cccn4C)[nH]n3)=O)CCC12 43341,N1(C(C2(CC#C)CCCO2)=O)CCC(NC(=O)C(CCO)N(C)C)CC1 43342,CC(C)(CC(F)F)C(=O)N1C2CCC1CC(NC(c1ccc3cc[nH]c3n1)=O)C2 43343,CCC(CCCC(=O)NCC1(CCO)CCC1)NC(c1cc(OC)n(C)n1)=O 43344,c1(CC(=O)NC2C(CNC(c3c(OC)scc3)=O)CC2)nn(C)c2ccccc12 43345,C1(NC(C2CCCS2)=O)CN(Cc2nnc(C(F)F)o2)Cc2nccn2C1 43346,N1(C(CCC2CCN(C(C(C)C3CC3)=O)C2)=O)CCC(C)(CO)CC1 43347,N1(C(COCC=C)=O)CCC(NC(c2cc3n(n2)CCC3)=O)C(CC)C1 43348,O=C1CCC(CC(=O)NC(CNC(c2ccc(C3CCOC3)s2)=O)C2CCC2)O1 43349,C1(NC(c2cccc(-c3ccccc3)c2F)=O)CN(Cc2cnco2)CC1(F)F 43350,N1(C(C2(COC(C)C)CC2)=O)CC(C)(CNC(C2CCC(C)O2)=O)CC1(C)C 43351,c1(C(=O)NCCCCCCNC(C2C(CCC)C2)=O)c(Cl)cnc(OC)c1Cl 43352,C1(C)(CNC(C2(C#C)CCC2)=O)CCC(NC(C2CCN(C(C)C)CC2)=O)C1 43353,C1(NC(=O)COC2CCCOC2)CC12CCN(C(C1CC3CC(=O)C1C3)=O)CC2 43354,N1(C(C(C)=C2CC2)=O)CC(C)CN(C(c2nc[nH]c3nccc2-3)=O)C(C)C1 43355,c1(Nc2ccc(C(=O)OC)nc2I)c([N+](=O)[O-])cc(C(F)(F)F)cc1[N+](=O)[O-] 43356,n1(C(C)C)cc(C(=O)NC23CC(NC(=O)C(F)F)(C2)C3)cn1 43357,C(CCCC(F)(F)F)OC12C(CN(c3n(CC=C)c(CC)nn3)C1)CC2 43358,C1(CC)(Cc2ccccc2)CCN1C(=O)C(N1CCCCC1)C 43359,CCCC(O)C(=O)N1CCC(N(C(=O)CC(C)NC(N)=O)C(C)C)C1 43360,C(CN=c1[nH]c(N2CCN(C(C3CCCCC3)C)CC2)nc(=N)[nH]1)OCC(C)C 43361,CC(C)(C)CCCNC(=O)NCCS(N1CCCC(C(F)(F)F)C1)(=O)=O 43362,C1(C(C(=O)NCCC)NC(=O)Cc2cnsc2)CCS(=O)(=O)C1 43363,C(CCC(=O)N1CCCC(C(N)=O)C1)(C(C)C)NC(c1c(C)coc1)=O 43364,C12(N(C(C(C)SC)=O)C(=O)C=Cc3ccccc3C)CCC(C1)C(O)C2O 43365,C(=O)(CC(C)(C)CNC(=O)C(C)(C)CO)N(C)CC1CCCCC1O 43366,Cc1ccccc1CCCNC(=O)NC12CCCC1C2 43367,N1(C(COCCC)=O)CC(CNC(c2cc(C(N)=O)co2)=O)OC2CCCC12 43368,C1(C)(CNC(C2C=CC(NC(C(C)=CCC)=O)C2)=O)NC(=O)NC1=O 43369,c1(C(=O)NCCC(C)CCNC(=O)C(C)(C)O)ccnc2c1CC(=O)N2 43370,N1(C(c2c(C)occ2)=O)CCC(NC(c2cnc(N(C)C)cn2)=O)C(O)C1 43371,CC(C)C1C(=O)N1C.c1(CC(N2CC(C(C)N(C)C)C2)=O)cccnc1 43372,C1(C(=O)NCc2cnco2)(NC(=O)Cc2ccsc2)CCCCC1 43373,CC(C(=O)NCC=C1CCN(C(C2CC(C#N)C2)=O)C1)C(C)(C)c1ccccc1 43374,C(=O)(C(F)C(C)CNC(C1CN(C(N)=O)C1)=O)NCC(C(=O)NC)(C)C 43375,C(=O)(C1CCc2cccnc21)NC1(F)CN(C(C(C)NC(=O)OCC2CC2)=O)C1 43376,N1(C(C(C)SCC)=O)CC(CC(=O)Nc2cc(OCCN)cnn2)CC1C 43377,c1(NC(=O)OCCc2ccccn2)cccc(Cl)c1Br 43378,c1(NC(C2(C)CCCN2C(=O)CCS(C)(=O)=O)=O)cc(Br)cnc1O 43379,C1(C(=O)NC2CCC(NC(c3c(C(C)C)c[nH]c3)=O)C2)CCCN(C)C1 43380,Cn1c(C(N2CCC(C)(CNC(=O)C(O)C(C)(C)C)CC2)=O)c(Cl)c2ccccc12 43381,CCC(CC)C(=O)N1C(CNC(c2cc(CC(C)C)nn2C)=O)CC2CC12 43382,c1(C(=O)NC2(C)CC(NC(CCC=C=C)=O)C2)cc(C)ccc1NS(=O)(=O)CC 43383,Nc1cc2ccccc2cc1C(N1CC(CCNC(C2CC3CC3C2)=O)C1)=O 43384,C1(NC(CC(C=C)(C)O)=O)C2CC(CN(C(c3coc(SC)c3)=O)C2)C1CO 43385,C1(C(N(C2CCN(C(=O)CCCc3cnn[nH]3)C2)CCC)=O)CCN(CC)C1 43386,C(=O)(CS(C)(=O)=O)NC(C)(C)CC1CCC(NC(=O)CN2CCS(=O)CC2)O1 43387,C1(C(=O)NCC(CNC(CCCOCC)=O)C)CCCC12OCCO2 43388,N1(C(c2c(CCC)n(C)nc2)=O)CC(C)CN(C(c2ccncc2N)=O)C(C)C1 43389,c1(CNC2CC(C(=O)NCCC(F)(F)F)C2)ccc(F)c(F)c1Br 43390,C1(C(N(CC(C)(C)CO)C)=O)C(C2CC2)CCN1C(c1ncccc1Cl)=O 43391,Cc1nc(C)c(C(=O)NCC(N2CCC(N(C)C(c3cccc(F)n3)=O)C2)=O)[nH]1 43392,C1(NC(c2c(C)nn[nH]2)=O)CCCCCN(C(=O)CCC2CCCOC2)C1 43393,Cc1nnsc1C(=O)NCC(C)(Cn1cccn1)NC(C1CC1c1ccnn1C)=O 43394,c1(CN(C(=O)C(F)C2CC(NC(C3(C)CCC3)=O)C2)C)ncnn1C 43395,C1(CCNC(=O)C(C2CC2)OC)(OC)CN(C(C2(c3ccnn3C)CCC2)=O)C1 43396,c1(NCCc2n(C)ncn2)[nH]c(=NCCc2ncc[nH]2)nc2c1cnn2C 43397,Cc1c(C(=O)N(CCCCNC(=O)C(c2cccn2C)=O)C)noc1C1CC1 43398,CCCCC(C(=O)Nc1ccco1)N(C(C)CN(C(=O)COC1(C)CCC1)C)C 43399,c1(N(C(CC)C)C)cc(N(CCNC(n2cccn2)=O)C)nc(CO)n1 43400,Cc1oc(CO)cc1C(N1CCOCC1CC(=O)NCC1CCC(C)C1)=O 43401,c1(COCC(=O)NCC(CO)CNC(C(C)c2cncs2)=O)ccnn1C 43402,Cc1cc(C(=O)NC(C)(C(=O)NCCc2cc(C)ns2)C2CCC2)ccc1C#N 43403,c1(C(N(C2CCCN(C(c3cc(C)c(C)o3)=O)C2)C)=O)cccc(C=C(F)F)c1 43404,C1(C(=O)N(CC2(CC)CCOC2)C2CC2)C2C3CCC(C3)C12 43405,C1(CNC(C(C=C)(C)CC)=O)CN(C(C2OCCO2)=O)CCC1(F)F 43406,c1(C(=O)NC2CC2)ccc(=NCC2CC(NC(c3sc(C)c(C(C)C)n3)=O)C2)[nH]c1 43407,C1(NC(=O)Cc2ccc(O)nc2)CN(C(=O)C2=CCCSC2)C2(CCCOC2)C1 43408,N1(CC)CCN(C(C2CCN(C(c3cc[nH]c(=N)n3)=O)C23CC3)=O)CC1=O 43409,c1(-c2ccc(NC(C3N(C)CCC3)=O)cc2)cc(O)nc(O)n1 43410,Cc1ccnc(C(C)NC(=O)CCC2CCCN2C(=O)Cc2ncc(F)cn2)n1 43411,c1(C(=O)NCCCc2ccc(C(=O)OCC)[nH]2)ncc(C(F)(F)F)cc1O 43412,CC(C(=O)N1CCN(CCNC(C2CCN(C(=O)C(C)C)CC2)=O)CC1)C(F)F 43413,N1(C(C=C(C)C(F)F)=O)CC(NC(c2ccncc2C(F)(F)F)=O)CC(O)C1 43414,C1(C)(C(=O)NCCCCC(C)NC(c2c(CC)nccc2)=O)CCC12CCC2 43415,N1(C(=O)OC)CCC(C(=O)NC(C)CNC(c2cccn2C)=O)CC1 43416,c1(NC)cnc(C(N2CC(C(F)(F)F)C(CNC(c3cc(C)no3)=O)C2)=O)cn1 43417,Cn1c(C(=O)NC(C)(CNC(=O)CSS(C)(=O)=O)CO)cc2ccsc12 43418,C=CC(C)(C)CCCN(C(=O)CCC(C)NC(=O)C(C)C(O)CC)CC 43419,Cn1c(=O)n(CCC(N2CC3(C2)CN(C(=O)NCCCl)C3)=O)c2ccccc12 43420,c1(C(=O)OCC)cc(C(F)(F)F)no1.c12csc(n1)C(C)NS(=O)(=O)C2 43421,CC1(C(N2CC(S(C)=O)C2)=O)CCN(C(c2cc(C(F)F)[nH]n2)=O)C1 43422,Cc1ccccc1C1(C=O)CC1.C1(C(=O)NC)C2CC1N(C(=O)OC(C)(C)C)C2 43423,C12(C(=O)OC)CCC(C(N3CCC(C)C(NC(=O)C(C)SC)C3C)=O)(CC1)CC2 43424,N1(C(c2c(OCC)nccc2)=O)CCC2CCCC12CNC(=O)CCC(C)(F)F 43425,C1(NC(CC2(C)CCOC2)=O)CC2CC(NC(C3CCC4(CC3)CC4)=O)C1C2 43426,C1(C(C)C)C(=O)NCCN1C(C1C2CCC(C2)N1C(c1cc(C#N)c[nH]1)=O)=O 43427,n1(CCC)cc(C(=O)NCC(C)(C)NC(c2n[nH]cc2Br)=O)nn1 43428,N1(C(C=CCCC(C)C)=O)CCCC(NC(c2ccc(CC(C)(C)C)cc2)=O)C1 43429,c1(C(N2C(C3(NC(=O)C(O)Cn4cncn4)CC3)CCC2)=O)cc2sc(Cl)cc2s1 43430,N1(CC)CC(C(=O)NC2CC23CC(NC(=O)CC2(C(F)F)CC2)C3)CC1=O 43431,N1(c2snc(C(C)C)n2)CCN(C(C2CC2NC(=O)OC(C)(C)C)=O)CC1 43432,C1(C(=O)NC)CCN(C(=NCCCF)NCCc2nc3ccc(Cl)cc3[nH]2)C1 43433,c1(CC)cc(=NC(=O)Cc2csc(NC(=O)Nc3ccccc3)n2)[nH]n1C 43434,CN1CC(C)(C)CC1C(N1CC(NC(=O)C2=COCC2)C(O)C1)=O 43435,C1(C(=O)NCC(CC(=O)NC(C)C(C)C)OC)CC2(CCC2O)C1 43436,c1(CCNC(CC2(NC(Cc3cc(C)[nH]n3)=O)CCCC2)=O)c(C)noc1C 43437,N1(C(CC=C)=O)CC(NC(C2(COCC)CCCO2)=O)C(c2cnn(C)c2)C1 43438,C1(NC(Cc2c(CC)con2)=O)CCOCC1NC(c1ccc(CO)nc1)=O 43439,N1(C(C(C)C2CCC2)=O)Cc2ccccc2C(NC(c2cccc(C(F)F)n2)=O)C1 43440,CS(=O)(=O)CCC(=O)NCC12CCC(CC1)N2C(c1cncc(OC2CC2)c1)=O 43441,C1(CC(=O)NCCC2CN(C(=O)CCc3cccs3)C2)CC(F)(F)C1 43442,c1(C(=O)NCC2CN(C(CCC3C(C)(C)C3)=O)C(C)(C)C2)cccc2[nH]ccc12 43443,N1(C(c2ccc(F)nn2)=O)CCOC2(CCN(c3nccnc3F)CC2)C1 43444,CCCC(C)(O)CC(=O)N1CCCCC(CNC(=O)CCNC(C2CCC2)=O)C1 43445,c1(OC)cccc(C(=O)NCC(C)(C)CNC(C2CC3CCC2O3)=O)n1 43446,Cc1ncc(C)c(N2CCC(NC(C3CCCCC3O)=O)C(F)C2)n1 43447,c1(OC)ccc(Cl)c(F)c1C(=O)NC1CC1NC(c1occc1C)=O 43448,c1(OC)cc(C(=O)N(C2CCN(C(c3onc(C)c3C)=O)C2)C)cc(N)c1O 43449,c1(CC)nc(C(=O)N(C)CC2(NC(=O)CC3(CO)CC3)CC2)cs1 43450,Cc1occc1S(C)(=O)=NC(=O)CC1(C)CC1(C)Br 43451,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC1CN(C(C(C)(C(C)C)OC)=O)CC12CC2 43452,C(=O)(CC(C(F)(F)F)NC(c1ccc2ccoc2c1)=O)NC(CCC)C1CC1 43453,N1(C(COC2(C)CCC2)=O)CCC2(CCN(C(C3CCCC3)=O)C2)C1 43454,C1(C(=O)Nc2cncc(C)c2)CCC(C)N(C(=O)C(CO)N(C)C)C1 43455,C1(CC(=O)N(CCN(C)C)CCO)CCCCC1NC(=O)CC1(N(C)C)CC1 43456,N1(C(c2cn(C)nc2)=O)CCC(C(N2CC3CCC2CC3)=O)C1(C)C 43457,CN1CCC(C(N2CC(C3CCCCC3)C2)=O)(NC(C2CC3(CC3)CO2)=O)C1 43458,Cc1cc2sc(C(N3CC(C(N)=O)(CNC(=O)C(C)n4ccnc4)C3)=O)cc2s1 43459,N1(C(C2(C#C)CN(C(=O)C(O)CN3CCCC3)C2)=O)CCC(C2CCC2)C1 43460,c1(C(N(CC(C)NC(c2cnc(Cl)c(N)c2)=O)C)=O)cnc2ncc(Cl)cn12 43461,c1(CC)cccc(C(=O)NC(C)C(C)(C)NC(=O)C=CC2CCCCCC2)c1F 43462,c1(C(=O)NCCCCCN(C(CC2(CC)CC2)=O)C)c(C(C)C)cccc1F 43463,c1(C(=O)NC2C(C(N(C3(CC(=O)OC)CC3)C)=O)CCC2)cccc(=O)n1C 43464,CS(=O)(=O)C(CNC(=O)C(O)c1cnc[nH]1)CNC(=O)CC1CCCOCC1 43465,C1(NC(C2CCCN(CCC)C2)=O)C2CC1CN(C(=O)CCN1CCCC1=O)C2 43466,C(=O)(CC(C(C)(C)C)NC(=O)CN(C)C(C)=O)NC(c1ccnn1C)CC 43467,Cc1cncc(C(=O)N(C)CC2CCN(C(=O)Cn3ccc(=N)[nH]3)C2)c1 43468,C1(NC(C=CC)=O)CCc2cc(OC(C)(C)C)ccc2C1 43469,c1(C(N(C2CN(C(=O)C(C#N)CC3CC3)C2)C)=O)c(F)cccc1Cl 43470,N12CCN(C(C(=O)OC(C)(C)C)C1)C2=O.c1(CC(C)C)nc(-c2ccccc2)no1 43471,C(=O)(C(CNC(=O)C(C)c1cc[nH]n1)CC(C)C)Nc1cc(CC)c(C)nc1 43472,C(=O)(C(C)(C)C(C)NC(c1c[nH]c(C)cc1=O)=O)N(CC(CC)O)C1CC1 43473,c1(C(N(CCNC(C2(CC=C)CC2)=O)C)=O)cccc2ncnc(O)c12 43474,N1(C(CC2CCCC(NC(CCCCC=CC)=O)C2)=O)CC(C)CCCC1C 43475,C1(NC(=O)CC2CCCCO2)CCN(C(c2cnc3[nH]cncc2-3)=O)C12CCC2 43476,CS(C)(=O)=NC(=O)C(=O)NC1CN(C(C2CCCN2C(C2CCC2)=O)=O)C1 43477,c1(C(=O)NCC(C)N(C(C(C)=C2CC2)=O)C)ccc(-c2cc[nH]n2)cc1 43478,N1(c2nccc(OCC)n2)C2CCC1CC(F)(F)C(NC(=O)C(O)CN(C)C)C2 43479,CC1CC2(CCN(C(=O)CN3CSCCSC3)CC2)CN1C(C1CC12CCCC2)=O 43480,c1(OCC)ccc(O)cc1C(=O)NCC(C1CC1)NC(c1nnn(C)n1)=O 43481,N1(C(COC(C)=O)=O)CCCC12CCN(C(=O)Cn1cc3ccccc3n1)C2 43482,C1(CC)CN2CC1C2=O.c1(C(=O)NCC(C)(C)C)ccccc1F 43483,C1(CNC(CC(C=C)CC)=O)CCC(C)(C)CN1C(c1cccc(C2CC2)c1)=O 43484,CC(C)C(C(=O)NOCCC(C)C)=C1C(S(=O)(=O)NC)=COC=C1.C1CC1 43485,C1(C(=O)NC(c2cccc(OC(F)F)n2)C)CCc2nc[nH]c2C1 43486,C=C(C)CC(C(=O)NCC1C(C)C1(F)F)NC(=O)CSCC(N)=O 43487,C12(C(=O)OC(C(=O)NC(C)C)C)CCC(CC1)C2(C)C 43488,C1(C(NNC(c2c(C)coc2-c2ccccc2)=O)=O)Oc2ccccc2OC1(C)C 43489,c1(C(=O)NCC2CCN(C(C(C)O)=O)C2(C)C)ccc2cc(Cl)ccc2n1 43490,c1(C(=O)NCC(C2CCCN(C(C3CS(=O)(=O)C3)=O)C2)(C)O)cnc2sccn12 43491,c1(CC)cnc(Cl)[nH]c1=NC(CNC(c1ccc(C)c(Cl)c1)=O)c1ccccc1 43492,C1(CNC(C(CC)NC(N)=O)=O)CCCN(C(C2(CO)CCC2)=O)CC1 43493,C1(CNC(CCCc2ccc(C)s2)=O)CCN(C(C2CCC2CF)=O)CC1 43494,CC1C(C(=O)N(C(C)(C)CC(N2CC3C=CC2CC3)=O)C)=NOC1C 43495,c1(C(N(C2CCN(C(c3cnnc(Cl)c3)=O)C2)CC)=O)cnn2ccn(C)c12 43496,C#CCCC(O)CCNC(=O)CN(C(=O)C(C1CCC1)OC)CC 43497,N1(C(c2nccc(CC)c2)=O)CC2CCC2(NC(c2cnc(C3CC3)s2)=O)C1 43498,N1(C(c2cc(C)[nH]n2)=O)CC(F)(F)CC1CC(=O)NC1CC(C)CCC1O 43499,C1(C(=O)NC2(CNC(C3(CC#C)CCCC3)=O)CCCC2)CCOC(C)C1 43500,c1(CCN(C(c2occc2F)=O)C2CC2)cccc(F)n1 43501,C(=O)(C(O)CC(C)C)C1C(CCC(=O)OC)C1(C)C 43502,CCCC(CC)C(=O)N1CCN(C(c2ccc(F)c(F)c2)=O)C(C)C1 43503,C(N=c1[nH]c2c(c(=NC3CCc4cccc(OC(F)F)c43)[nH]1)SCC2)C1C(O)COC1 43504,C(CC(CC)C(=O)N1CC(NC(=O)C=Cc2cncc(F)c2)C2(CC2)C1)=CC 43505,Cc1ncc(C(N2CC(C(=O)NCCC3(CO)CC3)CC2(C)C)=O)cc1C#N 43506,c1(C(N2C(C)CCC(NC(C3C(C)(C(C)C)C3)=O)C2)=O)ccc2c(c1)COB2O 43507,c1(CC)csc(CC(=O)N(CCNC(c2cc(CF)on2)=O)C(C)C)n1 43508,c1(CC(C)NC(c2ccc(=O)n(C)c2)=O)cc(Cl)cc(Cl)c1 43509,c1(COC)ccc(C(=O)OCC=Cc2ccc(OC)cc2)nc1CC(C)C 43510,C1(NC(c2cc(OC(C)C)ns2)=O)CCN(CCCCCF)CC1C 43511,C(C(C)C)(C(O)C(=O)N(C)CC1CN(C(=O)COC(C)C)CCO1)OC 43512,C1(CC(=O)NCC(C)(C)CNC(C2(CCCF)CC2)=O)CC(C)(C)CO1 43513,C(C(C(C)(C)C)NC(c1cn(C2COC2)nn1)=O)NC(C(C)C1CC1)=O.S(C)(=O)(=O)N 43514,N1(C(CCC(=O)N(C)C)=O)CCC2(CC1)CC2(C)C(=O)NC(C)C(C)(C)C 43515,Cc1cc(C(=O)NCC2CC(NC(=O)CC3CCC(C)CC3)C2)cc(N)c1 43516,C1(NC(=O)CCCCc2cnn[nH]2)CC12CCN(C(=O)C=Cc1cncs1)C2 43517,C1(C(=O)NCCOCCOC)CCN(C(=O)C(C)CC(C)C)CC1F 43518,N1(C(c2cccc(C)c2C)=O)CC(C2CN(Cc3ccn(CC(C)C)n3)C2)C1 43519,c1(CC)c(C(=O)Nc2cccc(Cn3ccnc3)c2)cnn1C 43520,CC1(C)CC(CNC(=O)CCCc2cc[nH]n2)CN1C(c1ccc(Cl)c(N)c1)=O 43521,C1(C(N(C2CN(C(C3CCCCCC3)=O)C2)C)=O)CN(S(N)(=O)=O)C1 43522,C1(N(C)C(C2COCCC2NC(C2(F)CCCC2)=O)=O)CCCCC1(C)C 43523,c1(C(=O)NCC2(O)CCCN(C(C3N(C)CCC3)=O)C2)ccccc1P(C)(C)=O 43524,N1(C(C(CC)=CC)=O)CC(C)N(C(=O)Cn2cncn2)CC1C 43525,C1(CNC(C2CN(C3CCC3)C2)=O)CCC(F)(CNC(=O)C=CBr)CC1 43526,c1(C(=O)NCC(c2cccnc2)NC(C(C)N(C)C)=O)cccc(NC(N)=O)n1 43527,N1(C(C#CC(C)(C)C)=O)CCCN(C(c2cc3scnc3[nH]2)=O)CC1CO 43528,C1(C)(C(N2C(CN(C)C(C3CCCN3C)=O)CCC2)=O)CCOCC1 43529,C1(CNC(CCCC(=C)C)=O)CC2COCC2N1C(c1cccc(Cl)c1)=O 43530,c1(C(=O)NC(CNC(c2c[nH]c(=NC)o2)=O)C2CC2)ccc2nccnc2c1 43531,c1(CNC(=O)NCCSCC)ccc(OC)c(Cl)c1 43532,C1(CCC)CN(C(c2cc(C)[nH]n2)=O)CC1C(=O)NCCn1cncn1 43533,c1(OC)nccnc1C(=O)NCC(=O)NCC1(C(N2CCC(OC)C2)=O)CCCC1 43534,C#Cc1ccc(CCC(=O)N(CC(C)NC(=O)CN2CCOCC2)C)cc1 43535,N1(C(CC)=O)CC(C(=O)NC(CCC)C(=O)NC)C2(CCC2)C1 43536,c1(CNC(c2n(C(CC)C)nnn2)CCOC)ccc(C(=O)NOC)cc1 43537,C1(C2CCCN(C(=O)CC3CC3(Cl)Cl)C2)(NC(c2c(C)cc(O)nc2)=O)CC1 43538,C1(COCCN)CCCN1NC1(C)CCC1 43539,N1(C(c2n(C)cnc2)=O)CCCN(C(c2cccc3ccoc23)=O)C(CO)C1 43540,Cc1ccnc(C)c1C(N1CC2(CCN2C(c2ccnc(C(F)(F)F)c2)=O)C1)=O 43541,c1(C(C(=O)NCCC2N(C(C(F)=C(C)C)=O)CCSC2)C)c(C)nn(C)c1C 43542,O=C(C1=CCN(C(=O)C(F)OC(F)(F)F)C1)NC1CCCC1n1cccn1 43543,c1(COC)cc[nH]c1C(=O)N(C(CN(C)C)C(C)C)C.C12(CC1)C(=O)N2 43544,c1(CNC2CCC(NC(=O)CC3CCCCO3)C2)cc(F)cc([N+](=O)[O-])c1 43545,C#Cc1cncc(C(=O)NC2CCC2NC(=O)Cc2ccc(F)c(Cl)c2)c1 43546,c1(N2CC(C)CC(OC)C2)ccc(S(=O)(=O)NC2CCN(c3ccccc3)C2)cn1 43547,n1(CC(=O)NCC(C)(C)CNC(=O)C(C)(C)CF)ccc2cc(F)ccc12 43548,C(c1ccncc1C)=CC(=O)NC(CN(C(C(CCOC)OC)=O)C)(C)C 43549,c1(C(=O)NC(C(CO)NC(C(CC=CC)C)=O)C)cc2nc(OC)ccc2[nH]1 43550,Cc1ccc(C(=O)NCC2CC(F)(CNC(C3(C(C)(C)C)CCCC3)=O)C2)nc1 43551,c1(C(=O)NCC(CC)NC(CCOCC#C)=O)cc(Cl)c(OC)c(Cl)n1 43552,N1(C(C2C(C)(C)CC2)=O)CC2(CCOCC2)CC1CNC(=O)CCc1ncco1 43553,c1(C(=O)NC2CC(NC(C(C)CCC(C)(C)C)=O)C2)cc(=O)c2ccccc2o1 43554,C1(C(=O)NC2(C(N(CC#C)CC3CCCO3)=O)CC2)CC1C1(C)COC1 43555,c1(CC)cnccc1CN1CCCC1C=O.c1(C(C(=O)NCC)F)ccccc1 43556,C(=O)(CCCCC(F)F)NC1(C)CCCN(C(CCc2ccc(SC)cc2)=O)C1 43557,c1(CC(=O)N(CC(O)CN(C)C(C2CC2C(C)(F)F)=O)C)ccnn1C 43558,C(=O)(CCN=[N+]=[N-])NCC=C(C(=O)N(CC(CO)OC)C)C 43559,c1(C(=O)NCC(CNC(=O)CC2CCCC2O)CO)nccc2ccncc12 43560,N1(C(c2c(OC)c[nH]n2)=O)CCN2CCN(C(C3CCCC(=O)N3C)=O)CC2C1 43561,C=CCC(C)(C(=O)N1CCC(C)(NC(=O)CNc2cc(C)ncc2C)C1)N(C)C 43562,C(=O)(C(CC)Nc1ocnc1C)N(CCC(=O)NC1CC(=C)C1)C 43563,CCCCN=C(NCCC(=O)N1CCCC1)NCC(CC(C)C)OC 43564,C1(CC(=O)NC(C)CCCCc2ccccc2)CC2CCC(C1)C2 43565,C(=O)(C(C)S(C)(=O)=O)NC1C=CC(CNC(CSCCOC)=O)C1 43566,C1(CCNC(C(C)n2cnnn2)=O)CCCN(C(c2cnoc2)=O)CC1 43567,c1(C(=O)NCC2N(C(C(CC)OC)=O)CC2)cnc(N2CCOCC2)cn1 43568,C1(NC(C2CC3(CC(=C)C3)C2)=O)CN(C(=O)C(c2ccc(Cl)cc2)=O)CC2(CC2)C1 43569,C1(C(=O)NC2C(CNC(CC3CCC(C)C3)=O)C2)CC=CC(O)C1 43570,C(CNC(=O)C(C)(C)c1ccccc1)(CC(F)(F)F)NC(CCC(C)OCC)=O 43571,C(CCC(O)C(=O)NC)NC(c1c(CC)c[nH]c1)=O.N12CC3CC3(C1)C2 43572,c1(C(=O)NC(CC=C)CNC(c2cnc(C)n2C)=O)cc2ccc(F)cc2nc1O 43573,c1(CC)nc(CC(=O)NC2CCCN2C(=O)C(C)NC(=O)C(F)(F)F)cs1 43574,C1(CC)CCN(C(=O)C(C)=CC(C)(C)C)C1C(=O)NCCC1CC(COC)C1 43575,c1(CC)ccc(C(=O)NCCC2CCN(C(=O)NC3CC3)CC2)cc1 43576,c1(OC)ccc(CNC2CCC(C(=O)O)C2)c(O)c1 43577,CON(CC1CCCCC1)C(=O)C(F)(CNC(=O)CC(C)C)C(C)C 43578,N1(C(c2c(SC)cccn2)=O)CC(CNC(=O)COC(C)C)CC1(C)C 43579,Cc1cc2cc(C=CC(=O)NC3CCC(NC(=O)CCCF)C3)ccc2[nH]1 43580,O=C(C(F)C(F)(F)C(F)(F)F)NCC1(F)CN(C(c2cc(F)c(Cl)cc2F)=O)C1 43581,C1(NC(c2ccc(CNC(C3C(C)C3C)=O)cc2)=O)CCC(=O)NC1C 43582,c1(CC(=O)Nc2c(Nc3ccc(C(=O)OCC)cc3)occ2)c(C)cccc1C 43583,N1(C(CC)=O)CC2CCCN(C(C34COCC3C4)=O)C2C1 43584,C#CCCCC(C)C(=O)N1CCC1CC(=O)Nc1ncc(CC#C)s1 43585,C1(NC(c2n(CCC)nc(C)c2)=O)CC2CN(C(=O)CCC(C)(C)F)CC2C1 43586,S(=O)(=O)(c1cc(C)c(Br)cc1F)NC(CCC)C(=O)NC(C)C 43587,C1(NC(CCCCN(C(CCC2N(C)CCC2)=O)C)=O)CCCCCC1CO 43588,N1(C2C(C)OCC2)CCC(NC(=NCC2CC2)NCC2(C3CC3)CC2)CC1 43589,c1(C(=O)NC23CC(CNC(C(C)SC)=O)(OCC2)C3)ccn2cnnc2c1 43590,N(C(=NCCC(=O)N(C)C)NCC1CCOC(n2cncn2)C1)N(C(CC)C)C 43591,C(=O)(CCCCC(C)(C)OC)OC(CC(c1ccc(CCC)cc1)C)=O 43592,C(c1cc(F)cc(F)c1)=CC(=O)N(CC(CN(C(CCCOC)=O)C)O)C 43593,N1(C(c2ccn(CCC)n2)=O)CCC2(CCN(C(c3cc(N)ccc3C)=O)C2)C1 43594,c1(-n2cc(NC(N3CCNCC3)=O)nn2)c(C(=O)OC)nc2ncccn12 43595,c1(C(=O)NC(C)CCCNC(c2cc(C(N)=O)cs2)=O)ccc(C(F)(F)F)nn1 43596,N1(C(c2c(C)n(C)nn2)=O)CCC(NC(C2(n3cc(Br)cn3)CC2)=O)C(C)C1 43597,C(=O)(C(F)(F)CN)NCC(Cc1ccccc1)OCC 43598,C1(CNC(c2cncc(OC)c2)=O)CN(C(=O)C=Cc2cccn2C)CCC1C 43599,c1(NC(C(C2CCN(C(C3(C)CC(=C)C3)=O)C2)C)=O)ccc(F)cc1C 43600,c1(CNc2ccc(P(C)(C)=O)cc2)ccc2cc(Cl)ccc2c1 43601,C1(C(=O)NCC(c2cn[nH]c2)O)CCN(C(=O)Cn2ccnn2)C1C1CC1 43602,N1(C(C(C)NC(=O)NC)=O)CC(NC(c2cnn(C)c2SC)=O)C2(CC2)C1 43603,N1(C(CC2(N(C)C)CCC2)=O)CC(NC(=O)C(O)CC2CCCCC2)C2(CC2)C1 43604,C(=O)(CC(CNC(=O)C(n1ccc(C)n1)C)C1CCC1)NC(C#C)(C)C 43605,C=CCC(CNC(Cc1cc(C)c(C(F)(F)F)s1)C(=O)OC)CC(C)C 43606,Cc1ccc(O)cc1NC(=O)CCCCCNC(=O)C(F)C1CCCC1 43607,C=CCCCCCCCC(=O)NCCn1cc(C(=O)NC(C)CC#N)nn1 43608,C1(CNC(CSCC(=O)OC)=O)CN(C(=O)CC2CCCN(C)C2)CC1C 43609,c1(C(N2CC(CNC(C(F)=CCC)=O)C(F)(F)C2)=O)cccc2nc(Cl)cn12 43610,S(=O)(=O)(c1ccc(CCSc2cnc(OC)nc2)cc1)N1CCC(CC(=O)OC)C1 43611,N1(C(c2cnc(CC)o2)=O)C(CC(=O)NC2C=CCCC2)C2CCCC12 43612,c1(C(N2CCN(C(CCCOC(C)C)=O)CC2)=O)cccc([N+](=O)[O-])c1 43613,c1(CNC(C(=O)Nc2cccc(OC)c2)C)ccc2c(c1)ncn2C 43614,c1(C(CNC(=O)NCc2c(C)nc(CC)o2)(C)C)cccc(Br)c1F 43615,C1(O)(CN)CCN(CCC2(C)CCN(c3ncccn3)C2)C1 43616,C1(O)(C(=O)NCCc2c(C(N(C3CC3)CC)=O)c[nH]n2)CC(F)(F)C1 43617,N1(C(c2c(NC)cc(Cl)cc2)=O)CC(CNC(=O)C(C)C2CC2)OC2CCCC12 43618,N#Cc1c[nH]c(=NCCN=C(NCCC2(O)CCCCC2)NC2CCC2)cc1Cl 43619,CC1CCN(C2CCOC2)CC1.[nH]1c(-c2cnn(C)c2)nnc1C 43620,c1(C(=O)NC2(CNC(=O)CC3(C(F)F)CC3)CCOC2)cc(O)cc(Cl)c1 43621,c1(-n2c(COCC3CCOC3)nc(-c3cc(C)oc3)n2)nc2ccccc2n1C 43622,C1(CC(=O)NC(CC)CN(C)CCO)CCCC1NC(=O)C=Cc1cncs1 43623,CC1CN(C(c2cncn(C)c2=O)=O)CCC1NC(c1cc(C2CCC2)[nH]n1)=O 43624,c1(OCC)nccc(C)c1NC(=O)CCC(C)NC(C1CCCN1C=O)=O 43625,C1(C(=O)NC2CC(N(C(c3n(C(C)C)ccc3)=O)C)C2)Cc2ccccc2C1 43626,C(CC(C)C(=O)NCC(CC)NC(C1(C)CCCC1)=O)=CCC 43627,C1(NC(C2CC(CCC)C2)=O)CCC2(CC1)CCN(C(c1cccnc1O)=O)C2 43628,c1(C(=O)NCC2(COC)CN(C(C3COC(=O)N3)=O)C2)ccc(C)cc1C 43629,C(=O)(CC(C)C(F)F)N1CCCC(NC(c2nc(COC)oc2)=O)C1 43630,c1(CCC)cc(C(=O)NC2COCC2CNC(C2CC2COC)=O)n(C)n1 43631,c1(C(=O)NC2CC(C)N(C(=O)Cc3ccc(F)c(O)c3)C2)ccc2nn[nH]c2c1 43632,Cc1cccc2[nH]cc(C(=O)NCC3(O)CN(C(=O)CCC4CC4CC4CC4)C3)c12 43633,N1(C(CC=C(C)C)=O)CC2CC2(CNC(=O)C(C)N(C)C)C1 43634,c1(N(CCNC(COC)=O)C)nc(N2CC3CCC(C2)N3C)nc2ccccc12 43635,c1(C(N2CCC(C(=O)NCc3ccc[nH]3)CC2)=O)c(F)cc(Br)cc1Br 43636,C(CCO)(C(=O)N1OC2CC1C(O)C2O)NC(CCC1COC(C)(C)O1)=O 43637,n1(CC)cnc2c(NC3CCCN(C(=O)C(c4cccc(Cl)c4)O)C3)ncnc12 43638,C#CCCCC(C)C(=O)N1CC(COC)(NC(c2ccc(Cl)c(F)c2)=O)C1 43639,Cc1cc(C(N2CCC(CCNC(C3CCN(C)C3)=O)C2)=O)cnc1C(F)(F)F 43640,C12(CC(=O)NC3CCCC(NC(C4CCC4(F)F)=O)C3)COC(CF)(C1)C2 43641,Cc1cc(Cl)c(C(=O)NCCN(C(C2C(C)C2(F)F)=O)CC2CC2)s1 43642,CC(N=c1ccnc(C2CCCC2)[nH]1)c1cccc(C(C2CC2)OC(C)(C)C)c1 43643,CC1=NN(C)C(=O)C1CC(N1CC(CO)(NC(=O)CC2CN3CCN2CC3)C1)=O 43644,c1(C(=O)OCC(=O)N(C2CCNCC2)CCCC)cc(C)ccn1 43645,c1(C(N2CC(C)(NC(C3CC3c3cn[nH]c3)=O)C2)=O)cnc(C(F)F)nc1 43646,c1(C(N2CCC(COC)(NC(C3CC=CCC3)=O)C2)=O)ccc(OC)c(Cl)n1 43647,c1(C(CC2CC2)NC(N(CC(O)CO)C(C)C)=O)ccccc1C(F)(F)F 43648,n1(NCCC2C(C)CCN(C(=O)OC(C)(C)C)C2)c(O)nc2ccccc12 43649,C1(CNC(C2(OC)CCOC2)=O)CC(C)(C)CN1C(c1scnc1C1CC1)=O 43650,C(=O)(CCS(=O)(=O)Nc1ccccc1)NCC1C(NC(C2CC(SC)C2)=O)C1 43651,C1(NC2(COC(c3c(C)nc(-c4ccccc4Cl)s3)=O)CC2)CNC(=O)C12CC2 43652,C(CCCCC(=O)N(C)CCOCCNC(C1CCC(C2CC2)C1)=O)SC 43653,c1(OC)ccc(C)c(C(N2CC(OCCNC(=O)CN3CC=CC3)C2)=O)n1 43654,C(=O)(CCCCC(F)F)N1CCC(CNC(=O)C(c2cc(F)cc(F)c2)O)CC1 43655,CC1(C)C(NC(=O)NCC2(c3nn[nH]n3)CC2)CC1O 43656,Cc1cc(C(=O)NC(CO)C(=O)NCC2CCC(C(N)=O)CC2)c(O)nn1 43657,N1(C(C(C(C)C)N(C)CC)=O)CC2CCC1C(NC(=O)Cc1n[nH]c(C)n1)C2 43658,N1(C(c2c(C(C)C)onc2)=O)CCC2(CC(C(=O)NCCN(C)C)C2)C1 43659,C1(N(CCNC(c2cc[nH]n2)=O)C(c2cc(F)c[nH]2)=O)CCCCCC1 43660,C1(NC(CCc2n[nH]c(=N)s2)=O)CCCCCN(C(C23CCN(CC2)CC3)=O)C1 43661,c1(OC)c(C(=O)NCCNC(=O)C(CSC)OC)cc(Cl)cc1C 43662,N1(C(c2ccc(C)cc2)C(=O)NC(CC)(C)C)C2CCC1CC(F)C2 43663,c1(C(=O)N(C)C)cc(F)c(O)c(Cl)c1.CC1CC2CN12 43664,CC1CN(C(=O)COC2CCN(C(=O)C=CC3CCC3)C2)CC(C)(C)O1 43665,C12(NC(c3c(C)ncc(C)c3)=O)CC(CNC(C3CC3CF)=O)(C1)OC2(C)C 43666,c1(C(=O)NC2CC(CNC(CN3CC(C)C3)=O)C2)ccnc2c1cnn2C 43667,N1(C(C2(C)N(C(C(CC)N(CC)CC)=O)CCC2)=O)CC2CC(CC)C2C1 43668,N1(C(C(C)(C)CF)=O)CCC2OCCN(C(=O)COc3cc(F)cc(Cl)c3)C2C1 43669,C1(CNC(C2N(C(C)=O)CC(O)C2)=O)CC2CCC(C1)N2C(C1(C(C)=O)CC1)=O 43670,C1(N(C(c2n(CC)ncn2)=O)CCO)CCN(C(=O)C(C)(C)C2CC2)CC1 43671,c1(C(N(CC(C)(C)CNC(C2CC2C2CCCCO2)=O)C)=O)cc(C2CC2)nn1C 43672,C1(C(N(CC)CC2CCCCN2C(C2CC2CCOC)=O)=O)OCCOC1(C)C 43673,CS(=N)(=O)CCNC(=O)C(Cc1cc[nH]n1)NC(=O)CC1CC(=O)C1 43674,N1(C(c2c(OC)ccc(F)c2)=O)C2CCC1CN(C(=O)C=C(C)Cl)C2 43675,CC1CN(C(=O)CCc2ccsc2)CC(C)N1C(c1ccc(Cl)cc1N)=O 43676,C(=O)(C(CCC)OC)N1CCC(CC=C)C1.C12(CCC1)CC(=O)N2 43677,C#CCC(C(=O)NCCC(C)SC(F)F)NC(=O)CC1(OCC)CCC1 43678,C1(CSC)OCCCC1(C)C.C1C(=O)N(C)C2(CC2)CC(=O)N1CC#C 43679,C(=O)(C(O)C(F)(F)F)N1CC2(C(CNC(=O)OC(C)(C)C)C2)C1.c12cn(nn1)C2 43680,N1(C(COCCC)=O)CC2CC1CN2C(c1ccccc1Br)C 43681,C1(C(=O)NC(CNC(c2cc(C)n(C)c2)=O)C2CC2)CC(c2cccc(F)c2)=NO1 43682,c1(C(N2CCC(CN(C)C(C3CC3CF)=O)C2)=O)cccc2nccn12 43683,c1(SC)ccc(C(=O)NC2CC(C)(NC(c3ccccc3F)=O)C2)c(Cl)c1 43684,c1(C(=O)NC2(c3nn[nH]n3)CCCCCC2)ccc(N2CCOCC2)c([N+](=O)[O-])c1 43685,O(NC(=O)C(C)(C)S(C)(=O)=O)C(CC(C)C)C(=O)N1CCC(O)(C(C)C)C1 43686,n1(CC(=O)NC2CN(CCn3cc(C=O)nn3)C2)cnnc1O.C1(CC2CC2)CC1 43687,C(=O)(C1CCCn2cncc21)N1C2CC(NC(Cn3c(C)csc3=O)=O)C1CC2 43688,N1(c2ccnc(SC)n2)CCC(NC(=O)Cn2nc(C)oc2=O)C12CCCC2 43689,C1(NC(CCCOC)=O)CC12CCN(C(=O)CN1C(C)CCC1C)C2 43690,C(c1cccnc1)=C(C)C(=O)NC1C=CCCC1C(=O)NC12CC(C1)C2 43691,C1(NC(c2ccc[nH]2)=O)CN(C(C23CCC(CC2(F)F)C3)=O)Cc2nccn2C1 43692,CCCCCC(F)C(=O)N(CC(N1CC(O)CC1COC)=O)CC1CC1 43693,N1(C(C2(C(=O)OC)CC2)=O)CC(CNC(=O)Cn2ncccc2=O)CO1 43694,c1(C(N2CCC(CCNC(c3ccc(C)c(C)n3)=O)C2)=O)ccc2[nH]ccc2n1 43695,C1(F)(NC(CCN(CC(C)(C)C)CCO)=O)CCN(C(=O)CS(N)(=O)=O)C1 43696,CC(C)(C(=O)NCC(=O)NCC1(CO)CC1)c1ccns1 43697,Cc1nn(CC(N2CCC(C(C)CNC(c3cc(C#N)c[nH]3)=O)CC2)=O)cc1Cl 43698,N1(C(C2C(=C)C2)=O)CCC2(CC1)CN(C(=O)C(C)n1cccc1)CC2CO 43699,c1(C(N2CCC(CCNC(C3C(=C)C3)=O)CC2C)=O)ccc2nnc(O)n2c1 43700,C1(C(=O)NCC(CC(=O)N(CCOC2CC2(F)F)CC)C)CN(C)CCN1C 43701,C(=O)(C(CCC=C)NC(c1ccncc1OC)=O)NCCCCCC#C 43702,C(=O)(C(C1(C)CC1)NC(=O)CNC(=O)CN(C(=O)C(C)C)C1CC1)OCC 43703,CC1COC2=CN=C(NC3CC4(CCN(C(c5cccs5)=O)C4)C3)NC2=N1 43704,N1(C(CCC(C)(C)NC(c2ccsn2)=O)=O)CCC2(CCCC2)CC1 43705,C1(=O)C(CC(C)C)N1CC.C12(CCOCC1)C(F)(F)C(=O)O2.C1(NN(C)C)(C)CC1.OC 43706,C1(C(N2CC(C(=O)NCc3cc(C)n(C)n3)C(C)C2)=O)CN2CCN1CC2 43707,C(=O)(C(C)S(N)(=O)=O)N1C(C)(CNC(C(c2cn(CC)nc2)=O)=O)CCC1 43708,CCCC(C(=O)NC(C)(C)CNC(c1cccc(COC)c1)=O)S(N)(=O)=O 43709,c1(C(C)C)nnc2cc(NCC(C)NC(=O)C(C)Cc3ccncc3)ncn12 43710,C1(O)(CNC(COC)=O)CC2C=CC1C2.N12CCC(C1)OCCC2=O 43711,c1(C(C(=O)NC2(C)CC2)N(C2CCC(F)(F)C2)C)cccc(CC(F)(F)F)c1 43712,C=CC(CC)CC(=O)NCC1(C)CCCN(C(c2cc(C(=O)OC)ccn2)=O)C1 43713,c1(CNCC(O)CC(F)(F)F)c(O)ccc(F)c1F 43714,CCC(=O)CCC(=O)N1CCOCC(NC(=O)C(c2ccccc2F)OC)C1 43715,Cn1cncc(C(=O)NC2CCN(C(C3(c4cccs4)CCOCC3)=O)C2)c1=O 43716,C1(C(N2C(C(C(=O)NCC(CC(C)C)O)(C)C)CCC2)=O)CCN(C)C(=O)C1 43717,N1(CC(=O)NC2CC(C)N(C(c3coc(Cl)c3)=O)C2)CCc2sccc2C1 43718,C1(C)(NC(CCCNC(C)=O)=O)CCC(NC(C2(O)CCSCC2)=O)CC1 43719,C(=O)(C1CC(=O)c2ccccc21)N1CC(N(C(=O)C2=CCOC2)C)C(O)C1 43720,CN1CCC(NC(c2c(CNC(C3CCCCN3C)=O)cnn2C)=O)C(C#N)C1 43721,CCC(C)C(C(=O)N(C1CCN(C)CC1C)c1nc[nH]n1)N(C(=O)CC)C 43722,Cc1ccc(C)c2[nH]c(C(=O)NCC3CCN(C(C4CCS(=O)CC4)=O)C3)cc12 43723,c1(C(=O)NCCCCNC(=O)CCc2cncnc2)c(Cl)ccc2c1OCO2 43724,C12CCCN(C1)C2=O.C=CCC(CNC(=O)NC(=O)OC(C)(C)C)NC1(Br)CC1 43725,c1(C(=O)OC)ccc(CCCC2=CCN(CC3CC(OC)C(OC)C3)CC2)s1 43726,C1(C)(C(=O)OC)CC(C(=O)N(CC(O)CNC(c2coc(Cl)c2)=O)C)C1 43727,c1(C(N2CC(C(C)NC(C(CC)OC)=O)C2)=O)cnn(C)c1N 43728,C(CCCCCn1cc(C2CCNC23CC3)nn1)C(c1ccccc1)O 43729,C1(C(N(CCCN(C(c2n(CC)ncn2)=O)C)C)=O)CCN(C2CC2)C1=O 43730,C1(C)(COC)CC(NC(=O)C(c2cccnc2)c2cnc(C)o2)CCO1 43731,CCCCCC(F)C(=O)N(CC)CC1CCCCN1C(c1cncc(C)c1)=O 43732,c1(C(N2CC(CN(C)Cc3ccccc3)C2)=O)ccc2nc(O)oc2c1 43733,C1(C(=O)NCCN(C(=O)Cn2nnc(-c3cccs3)n2)CC)CCC(C)(C)CO1 43734,c1(C(=O)NC2C(CC)CN(C(c3cccnn3)=O)CC2)cccc2nccn12 43735,c1(C(=O)NC(CNC(C2(c3cccs3)CCCC2)=O)CO)ccnnc1 43736,c1(C(N(C(C)C)CCNC(C2(C)CC=CCO2)=O)=O)cc2ccc(O)cc2n1C 43737,C(=O)(C(F)(F)C(O)C(C)C)NCCC1=CCN(C(c2cccc(CC)c2)=O)CC1 43738,c1(C(=O)OCC)cnc(N2CCS(=O)C(C)C2)cc1C 43739,C1(NC(C=CC(C)C)=O)CC(NC(=O)Cc2ccccc2)CC1O 43740,N1(C(CNC(CCC(C)C)=O)=O)CCC2(NC(=O)CC(=O)N(C)C)CC2C1 43741,C1(C(=O)NC(C2CC=CCC2)CNC(=O)CSC2CC2)(COC)CC=CC1 43742,C1(CC)CC2CN1C(c1cccc(-c3ccco3)c1OC)N(C)C2=O 43743,N1(c2nnc(C)o2)CCC(C(C)NC(C2C3COCC23)=O)CC1 43744,c1(SCC(=O)Cc2ccc(Cl)cc2)cnc(Br)cn1 43745,CC(C(=O)NC1CC2CC(NC(=O)C=Cc3cncs3)C2C1)S(N)(=O)=O 43746,c1(C(=O)NC2CC3CC2CN3C(=O)CN2CCC2)n[nH]c2ccc(Cl)cc12 43747,Cc1cnc2cccc(C(N3CC(N(C)C(c4c(Cl)cnn4C)=O)C(O)C3)=O)n12 43748,C1(CCNC(C(C)Sc2ccccc2)=O)COCCN1C(C1CC(=O)N(C)C1)=O 43749,C(=O)(C(C)(CO)CO)NCc1ccc(C(=O)NC(c2ccc(Br)s2)C)cc1 43750,c1(N(C(CC(=O)NC(COCC)C)C)C)ccc2nccnc2n1 43751,C(CCO)(CC(C)C)NC(C(c1c(C)cccc1Br)NC(c1cc(C)[nH]c1)=O)=O 43752,Cc1ccc(C(=O)NCCCOCCNC(C2(C)COC2)=O)c2ccccc12 43753,C1(C(=O)NCC2CC(OC)C2(C)C)CCS(=O)(=O)C(C)(C)C1 43754,N1(C(CN(CCC#C)C)=O)CC(NC(C2CC(n3ccnn3)C2)=O)CCC1C 43755,N1(C(CC2CCC(C(=O)OC)C2)=O)CCC(O)(C(N2C3CCCC2CC3)=O)CC1 43756,c1(C(N2CCC(CNC(C=CC=CCC)=O)C(C)C2)=O)cc2c(cn1)CCCC2 43757,O=S(=O)(c1cnccc1N1CCCC(CCO)C1)N.C1(CN)(CO)CC1 43758,C1(F)(CNC(C(CC2CCC2)OC)=O)CCN(C(=O)CC2CC(=O)C2)C1 43759,C1(C(N2CCC(CCO)CC2)=O)COCCN1CC1CCCC1 43760,c1(C(N2CCN(C3CN(C(c4c(C)nc[nH]4)=O)C3)CC2)=O)cc(C)cc(Cl)c1N 43761,CC(CC(=O)NCC1CC2CCC2C1)C(C)(C)NC(=O)CCCn1cncn1 43762,c1(C(=O)NCC(C)(C)NC(=O)Cc2ccoc2)ccc(-c2ccccc2)s1 43763,N1(C(C2C(C)C2)=O)CCCC(NC(c2ccc(I)o2)=O)C1 43764,c1(C(N(C2CCN(C(c3cc4cccnn4c3)=O)C2)C)=O)ccc2nonc2c1 43765,c1(NC(=O)NCC2(CC)CC2)ccc(C(=O)OC)cc1Cl 43766,CC1(C)C(C(=O)NCC23CCC(NC(=O)C=CC(F)(F)F)(CO2)C3)CC1[N+](=O)[O-] 43767,Cn1cc(S(=O)(=O)CCN2CCN(C3CCS(=O)(=O)C3)CC2)cn1 43768,C(C(C)(C)C#CC(=O)N(CC(=O)N(C)C)C)NC(C1CCCC(C)CC1)=O 43769,C=C(C)C1OCCC1Cn1cc(COC)nn1.S1(=O)(=O)C(C)CN1 43770,C1(C#CC(=O)NCC2CC2CNC(=O)CCCCN(C)C)(CC)CC1 43771,C1(C(=O)NCC(S(C)(=O)=O)CNC(C2CCCCC2O)=O)OCC2COCCC12 43772,Cn1cncc(C(=O)NCC2(O)CC(Nc3ncccc3C#N)C2)c1=O 43773,C(=O)(C(F)C(=O)NCCCOCCNC(C1CCC(NC(C)=O)CC1)=O)OC 43774,N(C(=NCCOCC=C)N1CCC2(CCCCCC2)C1)CCS(CC#C)(=O)=O 43775,C1(NC(C2C(C(C)NC(=O)CCc3ccc[nH]3)C2)=O)CCCC(O)CC1 43776,c1(C(=O)NC2CN(C(C(C)OCCOCC)=O)C(CO)C2)n[nH]c(C)c1[N+](=O)[O-] 43777,c1(C(=O)NCCNC(CSC)=O)cnns1 43778,C(C(C(=O)NOCC(O)C(C)(C)C)N(C)C(N)=O)OC.C12(CC1)C(=O)N2 43779,C1(O)(C(C)COC(c2c(Br)ncn2C)=O)CCN(C(=O)OC(C)(C)C)C1 43780,Cc1cc(C(=O)NCC(C(C)(C)C)NC(=O)Cc2cccc[n+]2[O-])ccn1 43781,C(=O)(C1CCCc2c1ncn2C)N1CCCCC(NC(C=CSC)=O)CC1 43782,C1(CC(=O)NC2CN(C(C3CC(NC4CC4)C3)=O)C2)C=CCCC1 43783,C1(C(N2CCCC(CN=[N+]=[N-])C2)C(=O)NC(C(=O)OC)C)CCCOCC1 43784,N1(C(C2(C(C)(C)OC)CCCC2)=O)CC(C)CN(C(=O)CCN(C)C)C(C)C1 43785,CC(C)(C#CC(=O)NC1CCC1(C)C)CNC(C1(C)CC(F)C1)=O 43786,Cn1c(CNC(CCC2CC2)C(=O)O)cc(C(=O)O)c1-c1ccccc1 43787,c1(C(N2CCN(C(c3ccn(COC)n3)=O)C3C2C3)=O)cn2c(C)cccc2n1 43788,C1(C(=O)NC2CC(CNC(CSC)=O)C2)CSc2ccccc2O1 43789,c1(CC(N2CCC(CNC(C(CC)(C)F)=O)C2)=O)ccc(Cl)cc1Cl 43790,c1(N2CC3CC(NC(C4=C(C)OCCS4)=O)C3C2)nc(Cl)nc(C(C)C)c1C#N 43791,N1(C(C(C)CC#N)=O)CC2CCC(c3ccccc3)(C2)C1 43792,C1(CC(=O)NCC2CCN(C(C3CC4(CSC4)C3)=O)C2)CC2CCC1C2 43793,Cc1cccc(C(=O)NCC2CCC2C(=O)NC(C)(C)CN(C)C(C)=O)c1 43794,CCC(CCC(=O)NCC(C)(C)C(F)F)NC(C1(CO)COC1)=O 43795,C1(CNC(C2(C)CC2(F)Cl)=O)C2CN(C(c3ccn(C4CCC4)n3)=O)CC12 43796,C=Cc1ccc(C(N2CCCC(NC(=O)C3=CC(C)(CC)C3)C2C)=O)cc1 43797,CC1(C)C2CC(C(=O)NCC3CC3NC(C3CC(=O)N(C(C)(C)C)C3)=O)CC12 43798,CCC(C)C(C(=O)NC(=O)OC)C(N1CCN(Cc2ncnn2C)CC1)=O.N(C)C1CC1 43799,c1(C(=O)NC(C(C)C)CNC(=O)C(N2CCOCC2)C)cc(N)c(O)c(F)c1 43800,CC(CNC(=O)CC1(O)CCC1)C(F)C(=O)NCCN1CCOCC1 43801,c1(C(=O)NCC(CC)NC(=O)Cn2ncccc2=O)ccnc(S)c1 43802,C1(CCNC(CCC=C)=O)CN(C(=O)C(CCC)OCC)CCCO1 43803,c1(C(=O)NCC2CN(C(c3c(C)coc3)=O)C(C)(C)C2)cc(P(C)(C)=O)cs1 43804,C(C(N=c1cnc(F)c[nH]1)C1CCC1)Nc1n(C)nnn1 43805,N1(C(C=C(C)C(F)F)=O)CCC(C2CC2)C1C(=O)NCC(CC1CC1)CO 43806,C(C(CC(C)C)C(=O)NC1CCCN(C(C2(OC)CCCC2)=O)CC1)OC 43807,CS(=O)C1(CNC(=O)CCN(C(=O)CC2CCCC(O)C2)C2CC2)CCC1 43808,c1(C2(C)CN(C(=O)NCCc3nccc(C(F)(F)F)n3)C2)ccccc1Br 43809,C1(C(N2CC(CC(C)NC(C(c3ccc(C)o3)C)=O)C2)=O)CCCC(=O)C1 43810,c1(C(C)NC(N(C2CC2)CC)=O)ncc(F)cc1F 43811,C1(C(=O)NCC2CC2NC(=O)C(F)CC2CCC2)(OC)CCSCC1 43812,CC(C)C(C)(CNC(=O)C=Cc1ccccn1)NC(c1nc(Cl)c(Cl)s1)=O 43813,c1(CC(=O)NC2CCN(C(CN(CCC#C)C)=O)C2)ccccc1CS(N)(=O)=O 43814,Cc1cc(C(N2CCC(NC(C3CC34CCCC4)=O)C(CO)C2)=O)ncc1CO 43815,C1(COC)CN(C(c2nccc(Br)c2C)=O)CCN1C(C1CC2C=CC1O2)=O 43816,c1(C(=O)NC2C(NC(c3c(C)cc(C(F)F)o3)=O)CC2)n[nH]c2c1COC2 43817,Cc1nc2ccccc2n1CC(=O)NC1CC(NC(c2ccns2)=O)C12CCC2 43818,C1(CC)NC(=O)N(C(c2nc(C)c(C)[nH]2)C)C1=O 43819,N(C(=NCC1(C)CCCC(=O)N1)N1CCc2ocnc2C1)C(CC)CC 43820,c1(C(C(=O)NC23CC(C2)C3)N(C(C2CCC2)C)C)cncc(Cl)c1 43821,CC1C(NC(=O)CCCC(N)=O)CCCN1C(C1CC1c1ccncc1)=O 43822,C1(C(N2CCC(Cl)CC2)=O)(CC)CCCN1C(c1ccccn1)=O 43823,N1(c2n(C3CC4CC(C(=O)C5=CCCCO5)C4C3)nnn2)CCn2nncc2C1 43824,c1(CC)cc(C(=O)NCC2CC(NC(C3CCN(C(=O)NC)C3)=O)C2)ccc1F 43825,N1(C(CCN(C(C(CC=C)CC)=O)C(C)C)=O)CC(C2CC2(F)F)C1 43826,C(CSC)(C(=O)NCC1(NC(=O)C=CCN2CCOCC2)CC1)OC 43827,NS(=O)(=O)c1ccc(C(=O)NCC2CCCCC2NC(=O)CC2NC(=O)NC2=O)o1 43828,Fc1cc2c(cc1F)CN(c1nc(N3CCSCCC3)c3ncccc3n1)CC2 43829,C12(C(=O)NCC(CNC(=O)C#CC(C)C)OC)CCC(F)(CC1)C2 43830,C(=O)(C(C)P(C)(C)=O)NCCN(CCCOC)C(c1ncccc1C(F)F)=O 43831,C1(CN(C(C2C(C(F)F)C2(C)C)=O)CC)CCCN(C(c2cn(C)c(C)n2)=O)C1 43832,Cn1nc(C(N2CC=C(C(=O)NCc3nc(=N)cc[nH]3)C2)=O)ccc1=O 43833,c1(C(N2CCCC(NC(C(CCSC)(C)C)=O)C2)=O)cc([N+](=O)[O-])cc(C)n1 43834,C(CC1=CCN(C(c2cnn(C)n2)=O)CC1)NC(C(c1ccccc1)NC(C)=O)=O 43835,C1(NC(c2cc(-n3nnnc3O)cc(F)c2)=O)CS(=O)(=O)CC1N1CCOCC1 43836,c1(C(=O)NCC2(F)CCC(NC(CC(CC)OC)=O)C2)c(C)nc(O)nc1C 43837,Cc1c(C(=O)NCCNC(C2OCCC2C(F)(F)F)=O)c(=O)oc2ccccc12 43838,Cc1cc(C#N)ccc1NC(=O)CC1(O)CN(C(c2ccc3nc[nH]c3c2)=O)C1 43839,c1(-n2cc(CNC(C3CC34CC4(F)F)=O)nn2)cc(F)cc(Cl)c1 43840,N1(C(C(C)(C)NS(C)(=O)=O)=O)CC(CNC(c2cnc(Cl)cc2N)=O)C(C)(C)C1 43841,C12(CNC(=O)CC3CC=CCC3)CCCC1N(C(=O)C=Cc1cccnc1)CC2 43842,C1(NC(c2cc(COC)no2)=O)CC1C1CCCN(c2nnc(C(N)=O)s2)C1 43843,N1(CC(=O)OC(C(c2ccc(CC)cc2)=O)C)C(=O)c2cccnc2C1=O 43844,N1(C(C2(C)CC2Br)=O)CC2(CCCC(CNC(C3CCCS3)=O)O2)C1 43845,C1(CC(=O)N(C(=O)CC(=O)NC2(NCC#C)CCC2)CC)CCOC(CC)C1 43846,C1(CCN(CC)CCCCc2ccn(C)c2)CCCCCC1.C1CC(=O)O1 43847,c1(C(=O)OCN(C(c2c(C)ccc(SC)c2)=O)C2CC2)ccc2c(c1)CCO2 43848,C1(CN(C)C(C2(N(C)C)CC2)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)CC1 43849,N1(C(C(=O)NCC(C)C)=O)CCCN(C(CC2(C)CC2)C(=O)N(C)C)CC1 43850,C1(CNC(C(C)=C(C)C)=O)CC(NC(c2cnn(C)c2N)=O)CC1O 43851,C1(CCC#C)CCCCN1C(=O)CCOCCN(C(=O)C(C)C1CCC1)C 43852,C1(NC(c2cn(CCC)nn2)=O)CCN(C(=O)C(c2ccc(F)cc2)CC)CC1 43853,C(=O)(C1Cc2ccccc21)N(C1CCN(C(C2CCCS2)=O)C1)C 43854,c1(C(c2n(CC)nnn2)NCC(C)OC)cccc(C(F)(F)F)c1.c12cc(ns1)C2 43855,CC(C)(C)C(CO)NC(=O)CCC1CCCN1C(=O)CC1(O)CCC1 43856,C1(=O)CCC(=O)N(CC)CC(C)N1.C1(C(=O)NC)CSCN1C(=O)OC 43857,c1(C(=O)NCC2N(C(C3C(C(C)O)C3)=O)CCCC2)cnn2c1CCC2 43858,C(=O)(C1=NN(C)C(=O)CC1)NCC(C)(CO)NC(c1cncc(C)n1)=O 43859,C(C(=O)N1OC2C=CC1CC2)(C1CC1)NC(c1ccc([N+](=O)[O-])[nH]1)=O 43860,c1(OC)ccc(CC(=O)NCCOCCNC(c2cc(Cl)c[nH]2)=O)nc1 43861,NC1C2CCC1N(C(=O)Nc1ccnc(OC(F)(F)F)c1)C2 43862,c1(C(N(C)CC2N(C(c3n[nH]c(C)c3Cl)=O)CCC2)C)ccc(S(C)(=O)=O)cc1 43863,c1(C(=O)NCC(C)(C)NC(c2c(CC)n(C)cc2)=O)oc2ccc(C)cc2c1C 43864,c1(C(N(C)CC2CCCN2C(c2ccc(N)c(Br)n2)=O)=O)n[nH]c2c1CC1CC21 43865,C(=O)(C(CCc1ccccc1)C(C)(C)C)N(CCC)CCNC(C1(C)CC1(C)C)=O 43866,c1(SCCC(=O)NCC(C)CNC(c2cn(CCF)nn2)=O)ccccc1 43867,c1(OC(C)C#N)ccc2cc(CNC(=O)NC3CC(OC(F)F)C3)[nH]c2c1 43868,C1(C(=O)OCC2(OCC)CC(C)C2)CCCCC1n1cccc1 43869,CC1=C(C)CC(C(=O)NCC2C(C)CCN2C(=O)Cc2csnn2)CC1 43870,O=C(C1=CCCCC1)NCCC(=O)NCCSc1cccnc1 43871,c1(CNC(C2C=CC(NC(C(CC)O)=O)C2)=O)cc(O)cc(F)c1 43872,C1(C)(NC(COCCCCOC)=O)CCC(NC(c2ccc(F)c(Cl)c2)=O)CC1 43873,C=CC(C)CC(=O)NC1CC(CNC(c2ccsc2-n2cnnn2)=O)C1 43874,CC(C)C(CNC(c1cnn2c1OCC2)=O)C(=O)NCCCc1cnccn1 43875,n1(OC(C)=O)nc(C)c(C(=O)NC2(C)CC(NC(CC3(C(=C)F)CCC3)=O)C2)c1Cl 43876,C1(NC(C2(CC)CCC2)=O)CCN(C(=O)C(C)(C)c2ccccc2)CC1CO 43877,c1(C(N2CCC(CC(=O)Nc3n[nH]c(O)n3)CC2)=O)cnn2c1CCC2 43878,C1(C(N(CC(=O)N(C(C(C)SC)C)C)CC(C)C)=O)CN(C)CC(C)O1 43879,N1(C(c2cc(C)sc2)=O)CCN(C2CCCN(C(=O)CCOC(C)C)C2)C(=O)C1 43880,C1(C(=O)NCc2cn(C(C)C)nc2)CCC2(CC2)N1C(C1CC(=C2CC2)C1)=O 43881,c1(OC)nn(C)cc1C(=O)NC1CCC(CNC(=O)C(C)n2ccnc2)CC1 43882,C(=O)(C(C)C(C)NC(c1c[nH]nc1C(C)C)=O)N(CCNC(C)=O)C 43883,N1(C(C(CC=C)OC)=O)CCC2(CCC(NC(=O)Cc3cccc(Cl)c3)CC2)C1 43884,c1(NC(C2(CC)CN(C(C(CC)CC)=O)C2)=O)ccc(F)cc1SC 43885,c1(OC)cccc(C(NCc2cn(C)nc2C(F)(F)F)CC2(F)CC2)c1.S.N 43886,c1(C(=O)NC(C)CCNC(=O)C(O)c2cnc[nH]2)ccc(Cl)o1 43887,c1(C(N(CCN(C(c2[nH]c(C)nc2C)=O)CC)CC)=O)cc(C)n(C(C)(C)C)n1 43888,N1(C(CC(C=C)C)=O)Cc2ccccc2C(NC(=O)Cc2ccc(O)nc2)C1 43889,c1(CC(N2CCC(O)(CCNC(CSCCOC)=O)C2)=O)cccc(C#N)c1 43890,c1(C(=O)OCc2ncn(CC)c2)ccc2nncn2c1 43891,c1(C(=O)NCC(C)N(C(CCC(C)c2ccccc2)=O)C)cnc2[nH]cnc2c1 43892,C(=O)(C1=C(Cl)CCOC1)N1C(CN(C(c2c(OC)cc(F)cc2)=O)C)CCC1 43893,C1(C(N2CC(COC)(NC(=O)Cc3cc(C(C)C)no3)C2)=O)CC=C(C)CC1 43894,N1(C(C(CCC)(C)C)=O)CCC2(CCN(C(=O)CC3CCC(=O)NC3=O)C2)C1 43895,N1(C(C(C2CCC2)OC)=O)CCC(C(=O)N2CC3CC3(CO)C2)=C(F)C1 43896,C(=O)(CC(C)CC(C)(C)C)N1CC(CNC(CC(CCC)CC)=O)C1 43897,C1(C(=O)NCC(CN(C(c2c(C)cc(C)o2)=O)C)O)CCC(C2CC2)CC1 43898,Cc1nc(C(C)C)ccc1C(=O)NCC(O)CCNC(c1cc(F)cc(F)c1)=O 43899,CC1CCCC1CC(=O)N(C)CC1CCCN1C(c1ccon1)=O 43900,Cc1cc(C2CC2)ccc1S(=O)(=O)NCCCCN 43901,C1(C)(C(=O)OC)CC(C(=O)NC2CC(NC(=O)CCC3(C)CC3(F)F)C2)C1 43902,N1(C(c2c(C)ocn2)=O)CCCC(CNC(=O)CCc2ccc(N(C)C)cc2)C1 43903,c1(C(=O)NCCNC(C2CCN(C(CC)=O)C2)=O)nnn(C2CCOC2)c1C 43904,c1(-c2ccc(NC3(C)CC3)cc2)ccc2c(n1)CCC2=O 43905,c1(C(N2C(C)CCC(NC(=O)CCCC#N)C2)=O)cc2c(cc1Cl)OCO2 43906,n1(CC(=O)NC2C(SC)CN(C(=O)C=CCO)C2)c(C)cc(C)nc1=O 43907,Cn1ncc2nc(Cl)nc(NC3CCOCC34CCC4)c12 43908,C1(O)(C(=O)NCC2C(N(C)C)CN(C(c3c(C)c(N)ccc3)=O)C2)CCCC(C)(C)C1 43909,Cn1nc(CC(=O)NCC2(C)CCCN2C(=O)COc2ccc(O)cc2)cc1Cl 43910,c1(C(=O)NCCSC)cc2cc(-c3cn(C)nc3C)ccc2oc1=O 43911,C1(NC(c2cccc(NC(C)=O)c2)=O)CC(C)CN(C(C2CCC(=O)O2)=O)C1 43912,C(=O)(C(C)C(=O)N1CCN(CCNC(=O)C(C)(C)C2CCCO2)CC1)OC 43913,c1(C(=O)NCC2N(C(C(COC)O)=O)CCOC2)c(Cl)cc(Cl)cc1Cl 43914,C1(C)(CC(=O)NC(CN2CCN(C(C(CC)=CC)=O)CC2)(C)C)C(C)(C)C1(C)C 43915,C1(C(N(C(C#C)C)CCO)=O)CCN(C2CCOC2C)CC1 43916,c1(C(=O)NC2C(NC(C(CC=C)NC(C)=O)=O)CCCC2)[nH]nc2ncccc12 43917,c1(C(N(C2CCCCN(C(C3C(CC)CCC3)=O)C2)C)=O)cccc2[nH]ccc12 43918,CC1(C)CC(=O)NC1CNCCS(=O)(=O)N1CCCC1 43919,c1(CCCC(=O)NCC(CC=C)NC(=O)CCNC(N)=O)ccc(Cl)c(OC)c1 43920,C1(NC(C2CC(O)(CC#C)C2)=O)CCCN(C(c2cccnc2CC)=O)C1C 43921,c1(C(=O)NCCC2CCN(C(=O)CCNC(=O)C3CC3)CC2)ncc(F)cc1C 43922,c1(C(NOCC(=O)OC)=O)cc(CNC(C2CNC(=O)C2)=O)cs1 43923,Cc1nc2ccc(C(=O)NC(c3cc(Cl)ccc3C(F)(F)F)C)cc2o1 43924,N1(C(c2ncc[nH]2)=O)CCC(C2CCCN(c3nccn4nnnc34)C2)CC1 43925,C#CC1CC(CC(=O)NCCOCCNC(NOC(=O)OCC)=O)C1.OC 43926,C#CC1(C(N2CC(C(C)(C)C#N)C2)=O)CN(C(c2cc(OC)ccn2)=O)C1 43927,c1(COC)ccncc1NC(C1COC(CNC(=O)Cn2cccn2)C1)=O 43928,N1(C(C2CCC(=C)CC2)=O)CCC2C1CCCN2C(=O)Cc1ccccc1OC 43929,c1(NC(C2CC(C)C(C)CC2)=O)cccc2c1CN(Cc1ccccc1)C2 43930,c1(N(C)C)ccc(C(=O)NCC2CCN(C(=O)CCn3cnc(=N)[nH]3)CC2)cc1 43931,CCN=c1ccc(C(=O)N(C)CCN(C)C(c2cc(CC)on2)=O)c[nH]1 43932,C1(C)(COC)CCN(N2CCC(C)(Oc3ccccc3)C2)C1 43933,C1(CC(=O)NCC2CCN(c3nnc(C(F)F)o3)C2)CCOC2(CCC2)C1 43934,C(=O)(C1CCc2nccn21)N(CCC1CCN(C(C2CC(C)(CC)C2)=O)CC1)C 43935,C1(N(C(C=NOC)=O)C2CC2)CN(C(c2ccc(C(F)(F)F)cc2Cl)=O)CC12CC2 43936,N1(C(C=C(C)C)=O)CC(NC(c2cc(C(C)(C)C)ccc2O)=O)C(C#N)C1 43937,C(c1cccc(CO)c1)=CC(=O)NCC(C)N(C(=O)Cc1c[nH]nc1O)C 43938,N1(C(c2c(CC)nns2)=O)CCC2OC(CNC(=O)CSc3nc[nH]n3)CC2C1 43939,c1(COC)noc(C(=O)NCC2CC2NC(=O)Cn2cnnn2)n1.N1(C=O)CCC1 43940,c1(C(=O)NC2C(CC=C)COC2)cc(CNC(C2CCC(F)CC2)=O)nn1C 43941,C1(C(=O)NC(c2scnc2C)C)CN(C(=O)Cc2cncnc2)CCO1 43942,c1(C(=O)NCCCNC(C(C)C2CC2)=O)ccnn1-c1cccnc1 43943,C(=O)(C1CCCc2nn[nH]c21)N(C)CC1(CNC(Cc2cnc(C)[nH]2)=O)CC1 43944,CC1CC(C)N(C(C)(C)C)CCN1C(=O)Oc1oc(S(N)(=O)=O)cc1C#N 43945,C(=O)(CCCCCCOC)N(C1CCCN(CCC(=O)OC)C1)CCC 43946,n1(C2CN(C(C(C3(C)CC3)N(C(C=CC(=O)OCC)=O)C3CC3)=O)C2)cc(C)cn1 43947,Cc1cc2ncnc(N3CCC4(CCN(C(c5conc5C)=O)C4)C3)c2[nH]1 43948,C12(C(=O)Nc3cc(N)c(C(N4CCCCC4)=O)cc3)CCCCC(=O)N1CCC2 43949,c1(OC)ccc(CN2CCC(C(N3CCOCC3C)=O)C(O)C2)c(Br)c1 43950,c1(C(=O)NC2C(CNC(=O)C3=CCCCC3)CC2)ccc2oc(=O)oc2c1 43951,C1(C(=O)Nc2nc(COc3cccc(F)c3)cs2)CCCC(F)(F)C1 43952,c1(C(=O)NC)ncnc(NC2(C)CCCN2CCSC2CCCCC2)c1C 43953,n1(CC=C)cc(C(=O)NCC2(NC(=O)CCn3cc(Br)cn3)CCC2)cn1 43954,N1(C(c2n(CC#C)cnn2)=O)CCC2CCN(C(=O)C(F)CCC(C)C)CC12 43955,CC(C)CC(F)C(=O)N1CC(CN(C)C)C(C)(C)C1.c1(C(C)N)ccc(O)cn1 43956,C=Cc1ccc(C(=O)NC(CCSC)C(=O)N2CCC(CC3CC3)C2)cc1 43957,c1(NC(C2C(C(=O)OC)C2)=O)sc2c(c1C(N1CCC(O)C(F)C1)=O)CCC2 43958,N1(C(C2C(C(=O)OCC)CC2)=O)CCCC1CC(=O)NC(C(C)C)C1CC1 43959,C1(C(=O)NC(CC=C)C(=O)NCCC)CC2(CCO1)CC2 43960,CC1CCN(C(c2ccn(-c3ccccc3)n2)=O)CC1N(C)C(c1cccs1)=O 43961,N1(C(C(C(C)C)N=[N+]=[N-])=O)CCn2ncc(CN(C(=O)C(O)CC3CC3)C)c2C1 43962,c1(C(=O)NCCCCC(C)NC(c2cocc2C(N)=O)=O)nnc(O)cc1O 43963,C1(CC)(NC(C2CCCN(C(c3ccc(COC)o3)=O)C2)=O)CCCCC1 43964,N1(C(c2n(CC)cnn2)=O)CCCC2(C1)CN(C(C1CC1F)=O)C2 43965,CCC(C)(CNC(=O)CSC(F)(F)F)NC(C1(CO)CCOC1)=O 43966,C(CCCCC(=O)NCC1CCCC1NC(c1ccc(C(C)C)cn1)=O)=CC 43967,C12(NC(C(CC)OC)=O)CCCC1N(C(=O)Cc1ccc(OC)cc1)CCC2 43968,c1(C(=O)NCCCN(C(=O)CCOCC(F)F)C)ccc(-c2nc[nH]n2)nc1 43969,C1(F)(CNC(c2cnns2)=O)CN(C(C2CCCN2Cc2ccsc2)=O)C1.C(=O)(N)O 43970,N1(C(C)C(=O)N(C2CCN(C(=O)CSC(F)F)C2)C)CCC(O)CC1 43971,c1(C(N2CCC(C)(C(=O)NC(CC)C3CC3)C2)=O)c(C)nn(C)c1C 43972,c1(NC(=O)OC(C)(C)C)ccc2c(c1)C(NCC1CC(C(F)(F)F)CO1)CCO2 43973,c1(C(N2C(CNC(CCSCCCC)=O)COCC2)=O)ccc2c(n1)CCOC2 43974,C(=O)(CC(C(F)F)C(C)(C)C)NCC1CC(OC)CN1C(=O)CN1CCOCC1 43975,N1(C(Cc2scc(C)c2)=O)CCC(F)(C(N2CC(CC(F)(F)F)C2)=O)C1.C(C(C)C)CC 43976,C1(CNC(C2(OC)CCCC2)=O)CC(NC(c2cncn2C)=O)CC1O 43977,C1(C(=O)N(CCCCCNC(c2conc2C(C)(C)C)=O)C)(OC)CS(=O)(=O)C1 43978,N1(C(c2c(Cl)ccc(C)c2)=O)CCCC12CCCN(C(c1ccc(=N)[nH]c1)=O)C2 43979,C(=O)(C(C(C)(C)C)NC(C1(C)CC(=O)N(C)C1)=O)N(CCOCC#C)C 43980,C(=O)(C(CC(C)C)C(C)C)NCC1CN(C(CCN(CC)CC)=O)CC(C)C1 43981,c12ccoc1C(=O)NC(c1nncn1C)CCC(=O)N2.CCCC(=O)N 43982,C(=O)(C(O)CC[S+](C)C)NCCN(C(c1c(C)c(Br)cnc1)=O)C 43983,N1(CCNC2CCN(C(=O)OC(C)(C)C)CC2)C(=O)C2C3C=CC(O3)C2C1=O 43984,C1(NC(=O)C=C(Cl)Cl)CCCC12CN(C(c1cn(C3CC3)nn1)=O)C2 43985,O(N(C)C(=O)CNCCC(=O)NC(C)C=C(C)C)CC 43986,CCC(C)(O)C(=O)N(C1(C(=O)NCn2cccn2)CC1)C.N12CCN(CC1)CC2 43987,c1(OC(C(N2CCC(CCCC(=O)OC)CC2)=O)=O)nc2ccccc2n1C 43988,N=c1nc(N2CC(CO)C(O)C2)[nH]c(=NCC2CCCCN2C)[nH]1 43989,c1(C(=O)OCC)cc(F)c(C(=O)NC(C(C)NC(=O)C=C(C)C)C(C)C)cc1F 43990,C1(NC(=O)Cc2cscn2)CC2CN(C(C3(CCO)CC3)=O)CCN2C1=O 43991,C1(C(=O)NC2C(NC(Cn3ccc(C)n3)=O)COC2)CCC(O)CN1C 43992,c1(CC(=O)NCC2N(C(CCC(C)SC)=O)CCCCC2)ccc2occc2c1 43993,C1(NC(C(C)(C)Br)=O)CCOC12CCN(C(c1cc3ccccc3[nH]1)=O)CC2 43994,C12(NC(C(C(C)C)C)=O)CCCCCC1N(C(=O)CCNC(=O)C(C)(C)C)CC2 43995,c1(C(N(CC(C)N(C(CC(=O)NCC#C)=O)C)C)=O)cc(C)c(Br)o1 43996,N1(C(C(C=C)(C)CC)=O)CC(C)(C)C(NC(C2CC=C(C)CC2)=O)C(C)(C)C1 43997,CCC(CC(=O)N1CCC(OCCCNC(=O)CC2CCOC2C)CC1)C1CC1 43998,N1(C(C2(N(C)C)CCC2)=O)CC(NC(CN(CCOC)C)=O)CC1C 43999,C(=O)(CCCC(=O)N1CCC(C)C1CNC(=O)C(C)(C)N1CCOCC1)OC 44000,c1(C(=O)NC2CCC(NC(CC3N(CC)CCC3)=O)C2)c(C)cn(C)c1CC(C)C 44001,C(=O)(C1=CCC(C)CC1)NCCC(C)NC(C1(C(C)C)COC1)=O 44002,C(=O)(CCCCC(F)(F)F)N(CC1N(C(C(CC)C(C)(F)F)=O)CC(F)C1)CC 44003,N1(C(C(CC)(C)C#N)=O)CC2CN(C(=O)C(C)c3ccsc3)CC2C1 44004,CC12CCC(C(=O)NC3CCC(NC(C4(C5CCC5)CCC4)=O)C3)(CO1)C2 44005,N1(C(C2=C(C)OCCC2)=O)CC2(CCCCN2C(c2cc3c[nH]cnc-3n2)=O)C1 44006,Cc1nccnc1C(=O)N(CC(C)(C)C(=O)NCC(C)(C)N(C)C)C 44007,C(C)(N=c1[nH]nc(C2CC2)o1)C1CCN(C(c2ccc(SCCC)cc2)=O)C1 44008,CN1CCOc2cc(CN3CCC(N(C)C(c4cc5sccn5c4)=O)C3)ccc21 44009,C1(CC)Cc2c(Br)cccc2CN1NC(=O)Nc1ncc(C)n1C 44010,c1(C(=O)NCCCCN(C)C(C2CCCO2)=O)cn2ccnc2s1 44011,N1(C(C(CCSC)(C)C)=O)CCC2(CCCN2C(c2ncc(Cl)cc2Cl)=O)C1 44012,N1(C(c2cc(Cl)ccn2)C(=O)NCC=C)CCOC2(CCSC2)C1 44013,C1(C(=O)NC(c2ncc(C)[nH]2)CC)CCN(C(C2CC23CCCC3)=O)CC1C 44014,C(=O)(C#CC(C)(C)O)N1C(CNC(C2CCCN(C(C)C)C2)=O)CC(COC)C1 44015,c1(CC(N2CC3C(NC(CC(C)CN(C)C)=O)C3C2)=O)ccn2cncc2c1 44016,N1(C(C(CC)NC(N)=O)=O)CC2(CCN(C(=O)C=C3CCC(C)C3)CC2)C1 44017,c1(OCC)ncc(C(=O)NC2CCC(NC(C3CC3Cl)=O)CC2)cn1 44018,N(C(=NCCC1CCc2ccccc21)NCC1CCC1)CCCC(F)(F)F 44019,c1(C(=O)NCC2C3CN(C(CC)=O)CC32)cc([N+](=O)[O-])ccn1 44020,c1(OC)cc(O)c(C(N2CCN(C(C3CCCC3(F)F)=O)C(C)C2)=O)cc1OC 44021,N1(CC)CCCC(C(=O)N(CC)CC2(CNC(C3CCCO3)=O)CC23CCC3)C1 44022,C1(C(N2CCOC(C)(CNC(=O)CSC)C2)=O)(COC)CCCNS1(=O)=O 44023,N1(C(c2cn(CC)nc2)=O)CCCC2(CC(NC(=O)CC3CCCC3C)C2)C1 44024,c1(C(C)NC(C2CC2CF)=O)ccc(CNC(C2(C)CCOC2)=O)cc1 44025,N1(C(CN(CCC)C)=O)CCC(C(N2CC(N(C)OC)C2)=O)C1(C)C 44026,N1(C(c2c(C)c[nH]n2)=O)CC2CCCC2(NC(c2occ3c2CCC3)=O)C1 44027,C1(NC(c2ccc(OC)nc2)=O)CCN(C(c2ccc(F)nc2F)=O)CC1F 44028,CC(C)C(C)C(CNC(c1cc(O)n(C)n1)=O)NC(=O)Cc1cnn(C(F)F)c1 44029,N1(C(C(CC)(C)C)=O)CC23CCCC2(C1)CN(C(c1cnc(OC)nc1)=O)C3 44030,C(=O)(C(CC(C)(C)C)NC(=O)Cc1ccc(O)nc1)N1CCC(C(C)C#N)CC1 44031,N1(C(c2ccc(CCC=C)cc2)=O)CC2CC(NC(c3snc(C)c3N)=O)C1C2 44032,Cc1nc2ccc(C(=O)N(C3CN(C(c4cc(C5CC5)ncn4)=O)C3)C)cn2n1 44033,c1(NCCCOC(c2ncc(CC)s2)c2nnnn2C(C)C)ccc(Cl)cc1F 44034,Cc1ccccc1C(=O)N(C1CCCC(N(C(=O)Cc2ccsn2)C)C1)C 44035,C(=O)(CC(C(=O)N(C)CCN(C(=O)CCN1CCN(C)CC1)C)N(C)C)OC 44036,c1(OC)cc(N)c(Cl)cc1C(N1CC(N(C)C(C23COCC2C3)=O)C2(CC2)C1)=O 44037,c1(C(=O)NC(CNC(C2(CCC)CCC2)=O)C)cc(C)c(Br)c(C)c1 44038,N1(C(C(CC)NC(C)=O)=O)CC(CNC(C2CCC(=O)N(C)C2)=O)CC(C)C1 44039,Cc1c(C(=O)NCC2(NC(=O)CC3CCCC(=O)N3)CCC2)nn2c1CCCC2 44040,c1(C(N2CCC(C(C)(C)NC(C(C=C)O)=O)C2)=O)cc2nc(C)[nH]c2cc1F 44041,C(C(O)C(=O)N(C1CCN(C(C)C)C1)C)NC(C(C)C1(O)CCC1)=O 44042,c1(C(N2CC(CNC(COCCOC)=O)C(C)(C)C2)=O)cc2cc(Cl)ccn2n1 44043,N1(C(Cc2cccs2)=O)CCC(NC(C2C(C(=O)OC)C2)=O)C(C)(C)C1.C(CC)O 44044,c1(C(N(CCCNC(c2c(C)snn2)=O)C2CC2)=O)cncc(N)c1 44045,Cc1cccc(Br)c1-n1cc(C(C)NC(=O)C(=O)OC(=N)O)nn1.CCO 44046,c1(C(N(C(CN(C(c2cc(CC)no2)=O)C)C)C)=O)cn(C)c(=O)c2cncn12 44047,c1(NC(C2C(NC(CN3CCC(C)C3)=O)COC2)=O)cncc(C2CC2)c1 44048,O(C=CC(=O)N(CCC(C)NC(=O)CC1CC(C)(C)C1)C)CC 44049,CC(C)C(C(=O)N(C1CCCN(C(=O)CCCNC(N)=O)C1)C)C1CCC1 44050,C(C)(CCC(=O)N(CC(O)CNC(=O)CSc1nncs1)C)NC(C)=O 44051,c1(C(N2C(c3c(OC)cc(Cl)cc3)CCC2)C(=O)OC)cn2cc(F)ccc2n1 44052,C1(NC(c2cnc(OCC)s2)=O)C2CCN(C(=O)CSc3nncn3C)CCC12 44053,c1(C(N(C2CCCN(C(c3cnsn3)=O)CC2)CC)=O)ccc2c(c1)CCNC2=O 44054,N1(C(C(C)NC(C)=O)=O)CC(O)(CN(C(=O)CC2COCC2O)C)C1 44055,c1(OCC(=O)NCCC2(OC)CN(C(C3COC(C)C3)=O)C2)ccc(O)cc1 44056,c1(NC(C(=O)NCC(CC=C)NC(=O)C(C)(C)SC)C)ccc(C(F)(F)F)cn1 44057,N1(C(c2c(CNC(CNC(C(N)=O)=O)=O)occ2)=O)CCC(O)(CO)C1 44058,C1(CNC(c2c(OC)nsc2OC)=O)CCC(C)N(C(=O)CCC(=O)N(C)C)C1 44059,N1(C(C(C(C)C)NC(N)=O)=O)CC2(CNC(=O)C=Cc3ccn(C)c3)CC1CO2 44060,C1(C(N2CC(O)CC(O)C2)=O)CCN(C(=O)C2(OCF)CCOC2)O1 44061,CC1COc2c(C(=O)NC3C4CC3N(C(c3cc(=O)cc(Cl)[nH]3)=O)C4)cccc21 44062,C1(C)(C(=O)NC(CCC)CO)CN(C(C2(C)CCC2)=O)CC1C 44063,c1(C(N2CCCC(NC(=O)CNC(C3CCCC3)=O)C2)=O)cc(C)c(C)nc1C 44064,Cc1nc2cccc(C(N3CCC4C3CCCN4C(=O)Cc3ccno3)=O)c2s1 44065,C1(NC(CCOC)=O)CC2CCC1CC2NC(C1(C)CC=C(C)CC1)=O 44066,CC1(CC(=O)NCC2CCN(C(=O)C(O)COCc3ccccc3)C2)CCOC1 44067,CC(C)(CO)CCCNC(C1(C=C)CCN(C(=O)CCP(C)(C)=O)C1)=O 44068,C12(C(=O)NC(C3OCCN(C(CSCC)=O)C3)C)CCC(CC1)OC2 44069,C1(CNC(C(c2ccc(Cl)cc2)(C)O)=O)CN(C(C2CC(F)C(=O)N2)=O)CCO1 44070,C(=O)(C1=NOC(C(C)(C)C)C1)NCC(CN(C(c1ccc(C(C)C)cn1)=O)C)C 44071,CCCCCC(CC)C(=O)NCC1CC2(CC(NC(C3(CC)CCNC3=O)=O)C2)C1 44072,Cc1cc(C(=O)NCC(C2CCCC2)NC(=O)C(C)(C)OC)n(C)n1 44073,c1(C(N2CCC(N(C(=O)C(C)(O)CC)CC)C2)=O)ccccc1S(=O)(=O)C(F)F 44074,C(c1cc[nH]n1)=CC(=O)NCC1CCC(NC(C2CCC(=O)N2)=O)C1 44075,Nc1cccc(F)c1C(=O)NC1CCCC1NC(C1(c2ccc(Cl)cc2)CC1)=O 44076,C(=O)(CCCC(C)(C)C)N1CC(NCCN(CCC)CCC)C(COC(C)C)C1 44077,CC(C(C(=O)NC1CC1)N1CCCN(c2cccc(F)c2F)CC1)C(C)(C)C 44078,c1(-n2c(C(N3CCC4(CC3)CC4)=O)cnn2)cc(Cl)ccc1Cl 44079,C1(C(=O)NCCOCCNC(C2CS(=O)C2)=O)CCCC1CC1CCC1 44080,N1(C(C(C(C)(C)C)NC=O)=O)CCC2(CC1)CC2CNC(c1cc(N)ccn1)=O 44081,C1(C(=O)NC2C(CNC(=O)CCC3CCCCO3)CCC2)CC2OC1C1CC21 44082,C(=O)(C1COc2ccc(Cl)cc21)NCCN(C(C1CCC1CF)=O)CC 44083,N1(C(CCC=C)=O)CCC2(CCCCN(C(=O)C(C)N(C)C)C2)C1 44084,C1(CNC(C=CC)=O)CN(C(c2ncc(Br)cn2)=O)CCC1OC 44085,c1(CNC(C2(C)CN(C(=O)CC3CC4CCC3C4)C2)=O)cnc(CO)nc1 44086,n1(CC)cc(Cl)c(C(=O)N(C(C)CCNC(=O)Cc2ncc(C)s2)C)n1 44087,N1(C(C)CN(C)C)CCCC(C)(C(N2CCOCC2CC2CC2)=O)C1.N(C)C 44088,c1(C(=O)OC)cncc(NC(C2CCCCC2F)=O)n1 44089,c1(C(=O)NCCCC(C)NC(C2(C)CC(C)C2)=O)cccc2c1COCCN2 44090,C(C(C)C)(C(O)C(=O)NCc1c(C)nsc1Br)OC 44091,N1(C(C2CCCN(C(C)C)C2)=O)CCCC2CN(C(=O)CCC3CC3(F)F)CC12 44092,c1(C(N2CC(CNC(C3(CCCC)CCC3)=O)C(C)C2)=O)cc2c([nH]1)CCCC2 44093,O(N(C)C(=O)CN=c1[nH]c(=NC)[nH]c(=NC(C)CCSC)[nH]1)CC 44094,C=CCCCC(C(=O)NC1CCC(C(N)=O)C1)NC(=O)CC1(OC)CCC1 44095,[N-]=[N+]=NCCCCCCC(=O)NCC1CN(C(=O)CC23CCCC2C3)C1 44096,C1(C)(C(=O)NC(C)CNC(=O)C(C)CSC(F)(F)F)CCCCO1 44097,c1(OC)ccc2cc(C(=O)NC3CN(C(C4CCC(F)(F)CC4)=O)C3)[nH]c2c1 44098,c1(C(N2CCC(NC(CCCC#CC)=O)C2C)=O)cccc2c1OCC2C 44099,c1(OC2CC(C(=O)Nc3ncc(C4CC4)o3)C2)ccc(F)cc1 44100,C(=O)(C1=C(Cl)CCCC1)NC1CN(C(Cc2c(C)scc2)=O)CC(F)C1 44101,C1(C(=O)NC2CCC(C(=O)NCCCNC(=O)NC)C2)CCN(C)C1=O 44102,Cc1sc(Br)cc1S(=O)(=O)NC(c1c(F)cccc1F)C 44103,C(=O)(C(C)(O)C(C)(C)C)N1CCC(CC(C)NC(=O)Cc2nccn2C)CC1 44104,CC(CC(=O)NCCCN(C(=O)CC1CNC(=O)O1)C1CC1)n1ccnc1 44105,C(=O)(C(O)C(F)(F)F)N(CCOCCN(C(=O)C(O)C(C)(C)C)C)C.C=O 44106,c1(CCC(C)(C)NC(=O)C(=O)NCC2CC2C2CCC2)ccc(O)cc1 44107,CN1CCOCC1CC(=O)NCc1ocnc1Cn1cc(C2CCCC2O)nn1 44108,C12(CC)COC(C(=O)NC3CC(NC(c4c(C)coc4C4CC4)=O)CC3O)(C1)C2 44109,C1(CC(=O)NCC(CC)NC(C2CCC(C)(C)OC2)=O)CCS(=O)(=O)CC1 44110,C1(NC(c2ncn(C)n2)=O)COCCN(C(=O)Cc2cccc(Br)c2F)C1 44111,N1(C(C(F)OC)=O)CC(C(=O)N(C)Cc2cc(C)on2)CC(C)C1 44112,C#CCC(C)(C)CNC(=O)C(CNC(=O)C1=CCSC1)OC 44113,c1(OCCC(=O)NCCC2CCCN2C(=O)CC2COCC2O)ccc(F)cc1 44114,N1(C(C(N2CCSCC2)C)=O)CC2CCN(C(=O)Cc3cccc(N)c3)C2C1 44115,C1(C(=O)NCC2C(NC(c3cnc(C(=O)OC)s3)=O)C2)Cc2ccncc2C1 44116,C(=O)(CC(C)CF)N(CCCNC(C)=O)CCNC(COCCOCC#C)=O 44117,C(=O)(N=c1c(Br)c[nH]cc1I)C1CCC(NC(c2ccc(F)c(F)c2O)=O)CC1 44118,C(N=c1[nH]c(=NCCC=CBr)[nH]c2c1CCCCCC2)C1(C)CCC(=O)N1 44119,c1(CC(=O)NCC2(O)CN(C(c3c[nH]nc3C3CCCO3)=O)C2)ccccc1 44120,N1(C(C2(C)CCC(=O)N2)=O)CCC2CCC(C1)N2C(C1CCC2CC1CO2)=O 44121,O=C1CCc2c(C(N3CC4CCCC4(c4ccc(Br)cc4)C3)=O)n[nH]c2C1 44122,c1(C(N2CCC(N3CCCC3=O)C2)=O)ccnn1Cc1cn(CC2CCCC2)nn1 44123,C1(CNC(=O)C(O)Cc2cnc[nH]2)CCCCN(C(c2ccsc2Cl)=O)C1 44124,C1(CNC(c2cocc2Br)=O)CCN(CCOCCOCCO)CC1O 44125,C1(NC(=O)Cn2ccnn2)CN(C(c2cc3cncn3c(O)n2)=O)CC2CCCC12 44126,C(=O)(C(CCC1CCC1)NC(c1c[nH]c(=S)cn1)=O)NC(CCC)COC 44127,C1(NC(c2ccn3nccc3c2)=O)CN(C(=O)CC2CC2(Cl)Cl)CC2(CC2)C1 44128,C(=O)(CC1(O)CCOc2ccccc21)N1CC(C)C(NC(C2CC23CCC3)=O)C1 44129,c1(C(C)C)cc(C(N2CCC(F)(C(=O)Nc3cc(C(C)(C)C)n[nH]3)C2)=O)n(C)n1 44130,c1(OC)cc(C)c(C(N2CC=CC(NC(=O)Cc3ccn(C)n3)C2)=O)cc1Cl 44131,N1(C(C2OCCN(C(Cc3cn(CC)nc3)=O)C2)=O)CCCC(F)(F)CC1 44132,N1(C(C(C(C)OC)O)=O)CC2CCCC(C1)N2C(c1ccsc1Cl)=O 44133,c1(CC)cc(OCC(O)CNC(=O)C(CC)c2ccccc2)cc(C)c1 44134,N1(C(C(Cc2ccco2)NC(c2cc(C(C)=O)[nH]n2)=O)=O)CC(CO)CC1C 44135,N1(C(C(C)(F)F)=O)CCCC(NC(c2cc(C(C)(C)C)n[nH]2)=O)C(F)C1 44136,C(C(=O)NN1CCCc2ccnn21)(C(C)OC)NC(C(CC)N(C)C)=O 44137,c1(C(=O)NCC2OCC(CNC(=O)C(Cl)=CCl)C2)cnn2ncccc12 44138,N#CC1CCCC(C(=O)NC2CC3CC2N(C(=O)CS(=O)(=O)NC2CC2)C3)C1 44139,C12(NC(C3C4CCN(C(=O)CN5CCCCC5=O)CC43)=O)CCC(O)(CC1)CC2 44140,c1(C(N2CCCCC(CNC(C(CC=C)C)=O)CC2)=O)c(F)cc(C#N)cc1F 44141,C1(C(=O)NC2(CC#C)CC2)CC(C)CN1C(=O)Cc1ccco1 44142,C1(CC(=O)N(C)CC2(CNC(=O)Cc3nncn3C)CC2)CCC2(CC1)CC2 44143,C12(CNC(C(C(C)C)C)=O)CCC(NC(c3ncc(F)cc3N)=O)(CC1)CO2 44144,Cc1ccc(O)cc1NC(C1CCC2(CC2)N1C(c1ccon1)=O)=O 44145,CN1CCN(C(=O)CC2(O)CCCCC2)CC1C(=O)NCc1cncnc1 44146,Nc1cc([N+](=O)[O-])ccc1C(N1CC(NC(=O)Cc2cncs2)C2(CCC2)C1)=O 44147,c1(C(=O)NCC(C)(C2CCC2)NC(C2CC2F)=O)cc(Cc2ccccc2)c[nH]1 44148,C(=O)(C1=CS(=O)(=O)CCC1)NCC(C1CC1)NC(C1CC2(CC(C(=O)OC)C2)C1)=O 44149,c1(CCn2c(-c3cnn(C4CCC4)c3C)nc(C(C)OC)n2)ccc(F)c(Cl)c1 44150,C1(CNC(Cc2ccc(C)s2)=O)CN(C(=O)CC(C)c2ccco2)CC1(F)F 44151,C=C1CC2CCCC(C1)N2C(C1CC(NC(c2ccc(C)cc2F)=O)CCO1)=O 44152,c12cnc(C(F)F)nc1N1CCC(C(O)C1)NC2=O.N1(CC)CCCCC1CO 44153,c1(NCC(N)=O)[nH]c(=NCC2CC=CCC2)nc2scnc12 44154,Cc1ccc(N2CCOC(CNCC3CCN3C(=O)OC(C)(C)C)C2)nc1Br 44155,C#CCC(CC(=O)NCC1CC(NC(c2cnc(C)nc2)=O)C1)c1ccccc1 44156,c1(C(N(C2CN(C(N3CCCC(N(S(C)(=O)=O)C)C3)=O)C2)C)=O)cccnc1N 44157,CCC(C)(COC)C(=O)NC(CNC(=O)C1=COCCC1)C1CCC1 44158,C12(CC)CN(C(=O)Cn3cnnn3)C(CNC(C3CCS(=O)(=O)N3)=O)(C1)C2 44159,C(=O)(C1COc2ccc(Cl)cc21)NC1C(NC(C=Cc2n(C)ccc2)=O)CCC1 44160,c1(Cn2cc(CS(CC)(=O)=O)nn2)cccc(C)c1Br.C1C(O)CC(=O)N1 44161,O=C(C1=CCC(NC(C2CCCOCC2)=O)C1)NCCC12CCCC1C2 44162,N1(C(C2CCN(C(C(C)NC(C)=O)=O)C(C)(C)C2)=O)CCc2n[nH]cc2C1 44163,CC1CN(C(C2(CCN(C)C)CC2)=O)CCCN1C(=O)CC(C)C(F)F 44164,C1(CC)CN(C(CCC2CCC2)C(=O)NCc2ccco2)CC1O 44165,C(C(=O)NCC(O)CCNC(=O)CCCc1cccnc1)(C(C)O)NC(C)=O 44166,c1(C(=O)NC2CCCC(NC(CN3CC(C)C3)=O)C2)cnn(C)c1C#N 44167,C(=O)(CCCCCN(C)C)NC(C(C)C)CNC(=O)C(C#N)C1CC1 44168,CC1(C)C(CNC(=O)C(F)(F)CO)CCN1C(=O)C(O)Cc1cnc[nH]1 44169,Cc1nc(C(N2CC(NC(c3ncccc3Br)=O)C(O)C2)=O)n(C)n1 44170,CCC(C(=O)N(C(C)C(=O)NCC1CCCCO1)C1CC1)OC 44171,C(=O)(C(F)(F)C(C)(C)O)N1CC(NC(C(CSC)C)=O)C(C(F)(F)F)CC1 44172,C1(C(=O)NCC2CC(NC(C3(CO)CC3)=O)C2)CC(=O)N(Cc2ccccc2)C1 44173,CCC(C)CCC(=O)N1CCCC1CCC1CCN(C(C2CC2(F)F)=O)CC1 44174,Cc1cc2[nH]c(C(=O)NC3CCCC(CNc4ncnc5cc[nH]c45)C3)cc2s1 44175,C1(NC(C(C=C)C)=O)CN(C(c2cnn3c2OCC3)=O)C2CCCC12 44176,C(=O)(CCCCC(N)=O)N1CCC(CC=C)(NC(=O)CSCC2CCCCO2)C1 44177,C(=O)(C#CC1CCCOC1)NC1CC2CN(C(C3(C)CCN(C)CC3)=O)CC2C1 44178,C1(NC(C2CC(N(C)C)C2)=O)COCCC1NC(c1nc(Cl)sc1Cl)=O 44179,C(C1c2ccsc2CCN1C(=O)Cc1nc(=N)[nH][nH]1)NC(CCCCN(C)C)=O 44180,N1(C(c2ccc(CCCCC)o2)=O)CCN(C(=O)CCP(C)(C)=O)CC2(CC2)C1 44181,CC(C)C(C(=O)N1CCC(N(C(=O)CSCc2ccc(F)cc2)C)CC1)NC=O 44182,C1(CC)CCOC(=O)CC1.C12CN(CCO1)C(=O)c1ccc(cc1)NC2=O 44183,c1(C(=O)NC2CCN(C(Cc3cc(CC)no3)=O)C2(C)C)ccn2nccc2c1 44184,c1(C(CC)COC(N2CCCC(CC)C2)=O)ccc(Cl)c(F)c1 44185,C#CC1CCC(c2nnnn2CC2(C)CC2)(NC(c2ccc(F)cc2C)C)CC1 44186,O=C(C1=CCCN(C(c2cc(Cl)ncc2F)=O)C1)Nc1ccc(OCF)cc1 44187,CC1CC(NC(C2CC(O)C2)=O)CN(C(=O)C(C)(O)c2ccccn2)C1 44188,c1(C(N(C(C(=O)N(C(C(C)C)C)C)C)C)=O)ns[nH]c1=O 44189,c1(OC)ccc(C(=O)NCC(C(C)C)NC(c2c[nH]ccc2=N)=O)c(C)c1 44190,N1(C(c2cc(CC)n(CCO)n2)=O)CC(N=c2[nH]c3c(C)cc(C)cc3o2)C1 44191,C(=O)(CN=c1cc[nH]cc1)N1C(C(C)C)CN(C(=O)CC2CCC(C)(C)C2)CC1 44192,C1(CNC(C(CC)F)=O)CC2(CCN(C(=O)CCc3cc(Cl)no3)CC2)C1 44193,c1(C(=O)NCC23CCOCC2C3)cc2cccc(Br)c2[nH]1 44194,N1(C(C2(C(CC)=O)CC2)=O)CCN(CC(=O)NCC2CCN(C(C)=O)C2)CC1 44195,C1(NC(c2c(C)[nH]nc2C(F)F)=O)CN(C(c2cncnc2C)=O)CCC1CO 44196,C(C1=Nc2cccc(F)c2S(=O)(=O)N1)N(C)CCc1cccc(O)c1 44197,c12ccccc1C2.C1(C(C(=O)OCCCC2C(C)C2)C)CCCCC1 44198,c1(C(=O)NC2CC(N)C23CCCC3)nc(O)nc2ccccc12 44199,c1(C(=O)NCC2(NC(c3n(CC)ccc3)=O)CC2)ccc2cnccc2n1 44200,CC1=NNC(=O)C1CC(N1CCOC(CCNC(=O)C(C2CC2)C2CC2)C1)=O 44201,C1(CC(=O)NC(CC)(C)CNC(c2cn[nH]c2)=O)Cc2cccc(Cl)c2O1 44202,C1(NC(COCCOCCOC)=O)CN(C(=O)Cc2ccno2)C2(CCOC2)C1 44203,CCCC(O)C(CO)NC(=O)NC(Cc1ccccn1)CO 44204,c1(CC)ccc(OC)cc1C(N1CCCCC1CNC(C1CC(C)(C)CO1)=O)=O 44205,C12CCC(CC1)CNC(=O)C2N1CC(C(=O)NC)C1.C1(NC(N)=O)CCC2(CC2)C1 44206,C12(CNC(=O)Cc3ccon3)CCC(CNC(=O)CC3=CCOCC3)(CC1)OC2 44207,C(CC1c2ccccc2CCN1C(=O)C(C)NC(C)=O)NC(CCN(C)CC)=O 44208,C12(C(N3CCCC(CNC(Cc4ccc(OC)cc4)=O)C3)=O)CCC(C)(C1)OC2 44209,c1(NC(C2CCOC2)C)[nH]c(=NCCc2nocc2Br)nc2ncn(C)c12 44210,N1(C(C(=O)NCc2ncc(C)nc2)=O)CCOC2(CC1)CCS(=O)(=O)CC2 44211,C=C(C)c1ccccc1NC(=O)CCOC1CN(C(C2OC3CCC2C3)=O)C1 44212,C1(C(=O)NCCCCCCNC(c2cnccc2Br)=O)CCn2cncc2C1 44213,C1(C(N(C)C)=O)CCCN(C(=O)C(=O)NC2COCC2OC2CC2)C1 44214,c1(C(=O)NCC2CC(COC)CN2C(C2CCCC2C)=O)cc2cccnc2s1 44215,CC1(CNC(=O)CCN2CCOCC2)CCCN1C(=O)CC1(CO)CC1 44216,C1(C(C)NC(c2ocnc2C(F)F)=O)CN(C(c2csnn2)=O)CC12CC2 44217,c1(C(N(C2CCCC(NC(c3cccn(O)c3=O)=O)C2)C)=O)cc([N+](=O)[O-])n[nH]1 44218,c1(NC(C(CC)C)=O)ccc(Cl)nc1C(F)(F)F.C1C(F)C(=O)N2CC(C2)O1 44219,c1(OC)c(NC(c2ccc(NCc3cncnc3)nc2)=O)ccc(Cl)c1Cl 44220,c1(CC(=O)NC(CC(C)NC(CC(CCCC)O)=O)C)coc2ccc(C)cc12 44221,C=CCC(C)(C)CC(=O)N1CCN(C(C2CC2c2ccoc2C)=O)CC1CCO 44222,C12(NC(c3ncc(C)cn3)=O)CC(C)(C1)OC21CN(C(=O)CCC(C)C)C1 44223,c1(NC(C(C)C)CNC(C2CCCO2)=O)ncncc1I 44224,c1(C(N(CCOC)CCNC(=O)Cc2csc(C)n2)=O)cccc2c1OC(F)(F)O2 44225,N1(C(C(C)(C)C2CC2)=O)CC(NC(=O)Cc2cc(C3CC3)no2)CC(C(N)=O)C1 44226,C1(CCNC(c2nc(C)sc2)=O)CN(C(C2OCCC2(C)C)=O)CCS1(=O)=O 44227,C1(C)(CC(=O)NCC2(CCCC)CC2)CCN1C(C1CC1OC(C)=O)=O 44228,Cc1ccc2c(c1)C(C(=O)NCC1(NC(C3CCCCO3)=O)CC1)CC2 44229,C(C(O)C(=O)N(C)Cc1cn(CC2CC2)nn1)N(C)C.c12nnc(o1)C2C1CC1 44230,Cc1cc(C)c(C(=O)NC2CC2CNC(=O)Cc2ccc(C(N)=O)nc2)c(S)n1 44231,C1(NC(C(COC)(F)F)=O)CCC(C)N(C(c2ccc(-c3cccs3)[nH]2)=O)C1 44232,O(NC(=O)C(CNC(C1COCC1N(C)C)=O)NC(C)=O)CCCOCC 44233,N1(C(C#CC2(CC)CC2)=O)CC(C)(CNC(=O)C#CC2CC2)CC1(C)C 44234,c1(C(N2CCC(CC(=O)Nc3ccc4sncc4c3)C2)=O)c(O)cccc1[N+](=O)[O-] 44235,N1(C(CCCNC(C)=O)=O)CCN(C(=O)Cc2ccc(Br)cc2)C(C)C1 44236,n1(CCCC)nnnc1C1C2CC2CN1.c1(SCC)ccc(C(F)F)o1 44237,CCC(C(=O)N(CC(C)CNC(=O)CCOCC1CC1)C)n1nccc1C 44238,C=CCC(CNC(C1C2CCC(F)C12)=O)C(=O)NC1CCN(C(=O)CC)C1 44239,C1(CNC(c2n(CC=C)nnn2)C2CCOC2CC)COC(C)(C)O1 44240,C1(NC(=O)Cc2ccc(O)cn2)(CO)CCCN(C(c2ccc(O)nn2)=O)C1 44241,Cn1cc([N+](=O)[O-])c(C(=O)NCC2(F)CCN(C(=O)CN3CSCC3=O)C2)n1 44242,c1(CC)oc(C(N2CC(CC(=O)NCC(C)CC3CC3)C(C)C2)=O)cc1C 44243,n1(CCC(=O)N(C2CN(C(c3c(C)oc(C4CC4)n3)=O)C2)C)ccc(O)nc1=O 44244,C1(SC)CCCCN(c2nc(=N)nc(N3CCC(c4cn[nH]c4)CC3)[nH]2)C1 44245,C1(NC(c2cc(C)ncn2)=O)CC2(C1)CC(C(=O)NCC(C)S(N)(=O)=O)C2 44246,C(=O)(C1=CCCC1C)N1C(CNC(C2OCCC2C)=O)CC(COC)C1 44247,C1(C(C)C)(C(=O)NC(C2CN(C(=O)C(O)C(F)F)C2)C)CNC(=O)C1 44248,c1(OC)ccc(NC(C2CC3CC3N2C(=O)Cc2ccccc2OC)=O)cc1C 44249,C(CCN(C)C)(C(=O)N1CCOCC1C(F)F)NC(c1scc(C)c1)=O 44250,c1(CCC(=O)N(C2CCN(C(=O)Cn3nccc3C)C2)CCC)nc(O)n[nH]1 44251,c1(C(=O)NC(C2CCN(C(C3(CO)CCCC3)=O)C2)C)cnnn1C 44252,N1(C(CC=C(C)C)=O)CCC2(CC1)CN(C(C1CC3CC1CC3(F)F)=O)C2 44253,C(C(=O)N1CCC(O)(CNC(=O)C(O)CN(C)C)C1)(C(F)(F)F)OC(C)=O 44254,C1(Cn2c(-c3c(C)cccn3)nc(-c3ccc(Cl)cc3)n2)CC12CC=CCC2 44255,S(=O)(=O)(c1ccc(F)c(C(=O)NCCN(C)C(C2C=CCCC2)=O)c1)NC(C)=O 44256,C1(COC)(CNC(C2SCC=C2C)=O)CCN(C(C2(CO)CCCO2)=O)C1 44257,N1(C(C2(CC)CCCN2C(C2CCCN2C(C)C)=O)=O)CC(C)OC2(CCC2)C1 44258,N1(C(C=Cc2c(C)cncc2)=O)CC2(C1)SCCC2NC(=O)C=CCN(C)C 44259,N1(C(C(C)SC(C)C)=O)CCC(C=CC(=O)NCC2CC(C)CO2)CC1 44260,N1(C(C2CC(C)SCC2)=O)CCC2(CC1)CCN(C(c1cnc(N)c(Cl)c1)=O)C2 44261,c1(C(=O)NCCCC2CCCN2C(C2CC23CCC3)=O)nccc2nn[nH]c12 44262,C(=O)(CC(C)P(C)(C)=O)NCC(CCCC)NC(=O)CNC(c1ccncc1)=O 44263,Cc1cc(Cl)c(C(=O)NCC2(F)CCN(C(c3cnncc3O)=O)CC2)cc1C 44264,n1(C(C(N2C3CC(CNC(C=CC)=O)CC2CC3)=O)C)cnc2cc(C)ccc12 44265,C(=O)(C1=NN2CC(C)CN=C2N1)N(CCCNC(C(COC)C)=O)C 44266,c1(C(=O)NCC(CNC(C(N2C(CC)CCC2)=O)=O)O)ccc2c(c1)C(C)CO2 44267,n1(CC)nnc(C2CC2)n1.C12(CN(C(=O)CC(C)n3ccnc3)C1)CC(=O)N2 44268,CCCC(CC)C(=O)NC1(CC)CCCN(C(c2ccoc2)=O)C1 44269,c1(C(N2CC(=C(CNC(CCNS(CC)(=O)=O)=O)F)C2)=O)cc(C)ccc1F 44270,CCC(CC(=O)N(C(C)CCNC(C1(C(=O)NC)CC1)=O)C)CC(C)C 44271,CC12CCN(CC1)C2.c1(CN2CCCC(C)(O)C2)cc(C(F)(F)F)cc(F)c1 44272,C12(CNC(c3c(C)nn[nH]3)=O)CCC(CC1)N(C(c1ccc(F)c(F)c1C)=O)C2 44273,c1(COC)ccccc1NC(c1ccnc(C(=O)NOCCN(C)C)c1)=O 44274,Cc1cc(F)c(C(=O)NC2CC(C(N3CCC(O)CC(C)C3)=O)C2)cc1F 44275,Cc1c(C(=O)NCC2(CNC(C3CC(=O)OC3(C)C)=O)CCCC2)cncc1F 44276,c1(OC)cnc(C(=O)NCC(C)(C)OCC(=O)NCC(N)=O)cn1 44277,c1(C(=O)NC(CNC(Cc2ccn(CC)n2)=O)C(C)C)cc(F)c(C)cc1Cl 44278,CC1CCN(C(=O)CN2CC3CCC2C3)C(C)C1NC(=O)CCc1nc[nH]n1 44279,c1(CCC(=O)N(C)CC2N(C(C(C)C3CCC3)=O)CCOC2)nnc(S)nc1O 44280,C1(CO)CC2(CCOCC2)CN1Cc1cc(N)ccc1F 44281,c1(C(N2CC(CC(C)C)C2)=O)cc(CNC(c2cnco2)=O)on1 44282,c1(N2CC3CN(S(CCCC)(=O)=O)CC(C2)O3)ncnc2ccc(OC)cc12 44283,C1(CC(=O)NCC2CC(NC(C(=O)NC(C)C)=O)C2)(C(F)(F)F)CNC(=O)C1 44284,C1(NCCNC(N2CCCC(OC(C)(C)C)C2)=O)CCC2OCCC2C1 44285,N1CCc2[nH]nc(C(F)(F)F)c2C1.N1(CCC(=O)NCCC#CC)CCOCC1 44286,c1(C(=O)NC2CN(C(c3cc(SC)oc3)=O)C(C)CC2)ccc(P(C)(C)=O)cc1 44287,N1(Cc2nc(CCC)on2)CCCC1C1CCCCN1C(c1c(C)ncn1C)=O 44288,c1(C(=O)NCC2C(NC(C(C)SC(C)C)=O)C2)cc(C(F)(F)F)ncc1Cl 44289,C12(NC(c3cc(C)c(Cl)s3)=O)CCC1CN(C(C1CC(=O)N(C)C1)=O)C2 44290,N1(C(c2c(CC)csc2)=O)CC2CC(C(=O)NCCN3CCOC3=O)CC2C1 44291,c1(OCC)ccccc1CC(=O)NCC1(CC(C)O)CCNCC1 44292,CC1CCCC(Nn2cc(CC3CC3)nn2)C1C.C12CC3(CC(C3)OC1=O)C2.C(C)(C)(C)O 44293,C(c1cc(C)n(-c2ccc(OC)cc2)c1C)=NC(C(=O)NCCCC)CC(C)C 44294,C1(OC)CN(C(=NCCc2sccc2C)NCc2ccco2)CC1O 44295,O=C(C1=C(Cl)CCOC1)NCCC1CN(C(c2cc(C3CC3)no2)=O)CCCO1 44296,c1(CC(=O)NC(CNC(c2ccc(C3CC3)o2)=O)C2CCC2)ccc(F)cc1Cl 44297,N1(C(C(CC)N(C)C)=O)CC2C(NC(=O)CCc3cccnc3)CS(=O)(=O)C2C1 44298,C1(CC)(NC(=O)C=CSc2ccccc2)CCN(C(=O)C(C)c2ncco2)CC1 44299,c1(C(=O)OC)ccc(O)nc1NC(C)CC(C)NC(C1CCS(=O)(=O)C1)=O 44300,c1(NC(CNC(c2ccc(COC)s2)=O)C)ncc(Br)cc1C#N 44301,c1(CC(=O)NC(CC)CNC(=O)CCCc2nc(C3CC3)no2)c(C)n[nH]c1C 44302,C1(C(=O)NC(C)C(C)(C)NC(c2cnc(N)cn2)=O)CCCC2(CCCCC2)C1 44303,c1(NC(=O)Nc2c(C)cc(Br)cc2F)c(C#N)oc2ccccc12 44304,N1(C(c2cc(C)n(C)c2C)=O)CCC(NC(=O)CCC2CCCO2)CC(C)(C)C1 44305,C1(C(C)C)(C(=O)N(C)Cc2ncco2)CCCN1C(=O)CCN1CCCC1 44306,N1(C(CCC(=O)NCCCOC)=O)CC2CCCN(C(=O)C=CC=C(Cl)Cl)C2C1 44307,C1(C(=O)NC(C2CN(C(=O)CC3CCS(=O)(=O)C3)C2)C)CCCC1(F)F 44308,Cc1cnc2ccc(C(=O)NC3CCN(C(=O)CCS(C)(=O)=O)C3)cn12 44309,S(=O)(=O)(c1cnn(CC(F)F)c1)N1C(C(N2CCCC(C(N)=O)C2)=O)CC2CC21 44310,Cc1ncncc1C(N1CCC(N2CCN(C(C3CCCCN3C)=O)CC2)C1)=O 44311,c1(C(N2CC(CN(C(C3ON=C(C)C3)=O)C)OCC2)=O)cccc2ncc(C)n12 44312,N1(C(CC2CCC(=O)C2)=O)CC2(CCCC2NC(c2cccc(C3CC3)c2)=O)C1 44313,c1(C(=O)NCCCC(C)NC(c2ncc(OCC)nc2)=O)c[nH]c2nccc-2c1 44314,C1(CNC(C(C)CC2CC2)=O)COCCN(C(=O)CC2CCN(CCF)CC2)C1 44315,c1(C(=O)NC2C(CNC(c3ccc(C#C)cc3)=O)COC2)cc2cn[nH]c2cn1 44316,C12(CCC)CC(C(=O)N(C)CCN(C(C3CC=CCO3)=O)C(C)C)(C1)C2 44317,c1(CC)ncnc(CC)c1C(=O)NCCCN(C(=O)C(O)CC(N)=O)C 44318,CC(C(=O)NCC(c1ccccc1)N(C)C(c1cc(Cl)ccc1Cl)=O)P(C)(C)=O 44319,N1(C(c2scc(CC)n2)=O)C2CC1CN(Cc1ccc(F)cc1I)C2 44320,C1(C)(CC)CCN(C(C2CC2C2CN(C(C3(C)CCCN3C)=O)C2)=O)CC1 44321,N1(C(C(Cc2ccco2)NC(c2ccc(C(C)=O)[nH]2)=O)=O)C2CC=CC(C2)C1 44322,CC(C)C(C(=O)NCC1(O)CCC(C)C1)C(C)NC(C1CC(=O)NC(=O)N1)=O 44323,Cc1cnn(CC(N2CCC3CC3(NC(=O)COC3(C)CCCC3)CC2)=O)c(=O)c1 44324,c1(C(=O)NCC2CCN(C(c3c(C)nn(C)c3C)=O)C2)cnn2cccc(C)c12 44325,c1(C(=O)NC2CCC(CCNC(=O)CC(F)F)C2)ccc(O)cc1F 44326,C(C)(C(=O)NCCOC1CCC1)N(C(C1CC1(C)C(C)C)=O)C 44327,c1(CCC)cc(C(N2CCC(CNC(=O)CC3(C)CCCC3)CC2)=O)cc(O)n1 44328,C1(NC(c2c(CNC(C3CC(O)(CC#C)C3)=O)occ2)=O)CCC(C)(C)C1 44329,N1(C(c2ccc(CC)cn2)=O)CCCCC(CCC(=O)N(CCCO)CCO)C1 44330,Cc1ncn(C)c(=O)c1C(=O)NCC1C(C)CCN1C(=O)CCCn1cccn1 44331,C1(CNC(COCCCCC)=O)CN(C(C2(COC)CC2)=O)CCO1 44332,c1(C(N2C(C)(CC(=O)N(C3CCOC3)C)CC2)=O)cnc(=N)[nH]c1 44333,CCC(C)C(C(=O)NOCc1nc[nH]n1)NC(c1ncc(F)cc1N)=O 44334,C1(CC#C)(NC(=O)C(COC)NC(=O)CC(=O)NCC2CC2)CCCC1 44335,C12(CC)CC(CNC(C)CC(C)(C)c3ccccc3)(CO1)C2 44336,C1(C(=O)NCC2CC(NC(=O)CC3CCCC34CC4)C2)CC2(C1)CC1(CC1)C2 44337,N1(C(c2ccc(OC(F)F)cc2)C(=O)NCCCC)CC(C)C(F)(F)C1 44338,c1(OCC)cc(C(=O)N(C)CC2CCCC(NC(C3(CO)CC3)=O)C2)ccc1Cl 44339,Cc1cncc(C(=O)NCCOCCCN(C)C(C2CCC(N(C)C)CC2)=O)c1 44340,C(CN=c1cc(NCCc2cc[nH]n2)nc[nH]1)(c1cccc(Cl)c1)N(C)C 44341,c1(CNC(C2(CC)COC2)=O)ccnc(C(N2CCC(O)(CN(C)C)C2)=O)c1 44342,C1(C(N(CCN(C)C(c2cccnc2)=O)C)=O)CCCC2CCCN12 44343,c1(-c2nc(-c3n(C4CCN(C)CC4)ccn3)on2)cn(C)ccc1=O 44344,N1(C(COC)=O)CCC(C2(O)CN(C(C3CCCS(=O)(=O)C3)=O)C2)CC1 44345,CC1CN(C(c2coc(C(F)F)c2)=O)CCN(C(C2CCCCC2F)=O)C1 44346,c1(CC(=O)NCC2CCCN2C(C2CC3CC2C2CC32)=O)ccc2nonc2c1 44347,C1(NC(c2cnn(CCC)c2C)=O)CC(C)CN(C(=O)CC2CCCC2(F)F)C1 44348,N1(C(c2cc(CC)cc(F)c2)=O)CCC2(CC1)CC2NC(C1(F)CC=CCC1)=O 44349,c12ccc(Cl)cc1C(=O)N(CC)C2.C1(O)(NC(=O)OC(C)(C)C)CCCC1 44350,C(=O)(CCS(=O)(=O)CC(C)C)NCC(C1(O)CCN(C(C2(CF)CCC2)=O)C1)C 44351,Cc1cccc(C(N2CCC(CCNC(C3CCS(=O)(=O)C3)=O)C2)=O)c1Cl 44352,c1(C(=O)NC2(CNC(CCCS(C)=O)=O)CC2(F)F)cccc2c1OCCO2 44353,C1(O)(CNC(C2CCC2O)=O)CN(C(C2CC(=C3CCC3)C2)=O)C1 44354,c1(C(=O)NCc2c(CC)noc2C)coc2c1CN(C(c1ccc(C)s1)=O)C2 44355,C1(c2cn(CC(CNC(c3cnc(C)nc3)=O)OC)nn2)CCC(F)(F)CC1 44356,N1(C(c2cccc(OC)n2)=O)CCc2ccc(C(=O)NCCCC(C)C)nc2C1 44357,CCC(CC)CCCC(=O)N1CC2CC1C2CNC(c1cc2c([nH]1)CCCC2)=O 44358,c1(C(c2nn(CCOCC)c(C)c2Br)(F)F)cc(F)cc(F)c1 44359,C(=O)(C(CCOCCO)NC(=O)CC1CCOC1=O)NCCOCC 44360,c1(C(=O)NC2C3CN(C(CSCCCC)=O)CC32)ncc([N+](=O)[O-])cc1C 44361,N1(C(c2c(C)cccn2)=O)CCC(NC(=O)CSC(F)(F)F)C2(CCC2)C1 44362,CC1C(NC(c2ccc(OCC(N)=O)cc2)=O)CCN1C(c1cc(F)n[nH]1)=O 44363,c1(C(N2CCC(C(=O)Nc3cncc(SC)c3)C2)=O)cc(Cl)ncc1I 44364,c1(C(=O)NCC2CCCCN(C(C3(C(F)F)CCC3)=O)C2)ccc2nccn2c1 44365,c1(SC)nc(C)c(CCC(=O)NCC2CCN(C(=O)C=C(Cl)Cl)C2)c(O)n1 44366,c1(C(N2CCC(O)(CNC(c3cc(CC)c(C)s3)=O)C2)=O)cc2ncccc2o1 44367,C(=O)(CCS(=O)(=O)NC(C)=O)N(C1CN(C(C2N(CCC#C)CCC2)=O)C1)C 44368,C(=O)(C(C)(F)C(C)(C)F)N1CC(C)C(CC(=O)NCC2CCC(=O)O2)C1 44369,C12CCN(CC1)C2c1nnnn1-c1ccsc1.C(C(O)COC)OCCOC 44370,N1(C(CC2N(C(CC3C(C)C(=O)CC3)=O)CC3(CC3)C2)=O)CCC2(CCCC2)C1 44371,C1(CNC(c2cc3occc3s2)=O)CC2(CO1)CN(c1nnc(CO)s1)C2 44372,C(=O)(C(C)(C)C(F)F)N1C(C2(N(C(CC(C)C3CCCCC3)=O)CC)CC2)CCC1 44373,CCC(C)(CNC(c1nc(C)n(C)n1)=O)C(=O)NCc1cccc(C)n1 44374,C1(N(C(=O)CSc2nncn2C2CC2)C)CCCN(C(=O)CC2CCC2(C)C)C1 44375,C1(C(=O)NC(CCC)CCCNC(c2ccc(CO)s2)=O)CC(C(C)(C)C)=NO1 44376,C1(NC(C(c2cnn(C)c2)NC(CSCCCC)=O)=O)COC(C)(C)C1 44377,N1(C(CNS(CC)(=O)=O)=O)CCN(C(=O)Cc2ccc(C)cn2)CC1C(C)(C)C 44378,C12(C(=O)NC3CC(N(C(C4C(C=C)C4)=O)C)C3)C3CC(CC13)C2(F)F 44379,Cc1nccc(Cl)c1C(=O)NCC1COCC1NC(C12CCC(CO)(CC1)C2)=O 44380,c1(C(N2CCC(NC(C3CC4CC3C4)=O)C2)=O)ccc(F)c(Cl)c1F 44381,CC1CC(NC(=O)CN2CCCNC2=O)CCN1C(C1(F)CCCCC1)=O 44382,CC1(C)OCC(CC(C)C(=O)Nc2cccc(C(N3CCCC3)=O)c2)O1 44383,N1(C(CCc2cc(C)on2)=O)CCC(NC(c2ncc(N)cc2Cl)=O)C(C)(C)C1 44384,N1(C(c2cc(CC)no2)=O)CCC=CC1C(=O)NC(c1cnccn1)C 44385,C(=O)(C1=CCC2CCC1N2C(=O)C(C#N)C(C)(C)C)NCC(C)CCO 44386,N1(S(c2occ(C(C)=O)c2)(=O)=O)CC(C)OC2(CCCCC2)C1 44387,C(=O)(CCCN(C)N=O)NCC(CC)(C)NC(=O)CCCc1ccccc1F 44388,Cc1cc(Br)c(F)cc1NC(c1cncc(C(C)(F)F)c1)=O 44389,c1(OCC(=O)NC(C)CC2CCC(=O)N2)ccc(Cc2ccccc2F)cc1 44390,C1(N(CC(F)(F)F)C=O)OC(C)CC1C.C(CNC(=O)C(C)C1CCCC1)(C)OC 44391,C#CCCCCC(=O)NC(C)(C)CN(C)C(c1nc(OC)cc(C(F)(F)F)n1)=O 44392,C(C#CC(=O)N(CCCCO)CC)NC(C1C(=C)C1)=O 44393,CC12CC(C(N3CCC(NC(C4CC4(C)Br)=O)C(F)C3)=O)(C1)C(C)(C)O2 44394,C(=O)(C(O)C(C)CC)NCC(C1CC1)NC(C=CC(=O)OCCCC)=O 44395,C(=O)(C1=NN(C)C(=O)CC1)N1CC(NCCc2cc(CC)no2)(CO)C1 44396,C1(C(N2CCC(C(C)NC(CC(=O)NCC)=O)C2)=O)CN2CCC1(C)CC2 44397,C(=O)(C1=NOC(C)C1C)NC1CN(C(CN(CCOC)C)=O)CC1(F)F 44398,C1(NC(C2C(OC(C)=O)C2)=O)CCC(C)N(C(C2CC(C)(C)C2)=O)C1 44399,C(=O)(C#CC(C)(C)C)N1CCC(C(N(c2ncccc2C(F)(F)F)C)=O)CC1 44400,C(C)(CC)(CCNC(c1cccc(C(N)=O)n1)=O)NC(CSCC#C)=O 44401,c1(CC(N2CCC(CCNC(COC(CC)C)=O)C2)=O)ccccc1F 44402,O(NC(=O)C(F)(F)C(C)(C)O)C(CC(C)C)C(N1CC2CC=CC1C2)=O 44403,C(N=c1[nH]c2cc(COC)ccc2o1)C1(CCC)CCN(C(=O)OC(C)(C)C)C1 44404,c1(CCC(N2CC(CC)N(C(=O)C(C)=CC3CC3)CC2)=O)cccc2oc(C)nc12 44405,N1(C(C(CCC)C)=O)CCN(C(=O)CC(C)Cc2cccc(F)c2)C(C(C)C)C1 44406,Cc1cc(Cl)ncc1-n1cc(C2CCCCN2C(=O)C(C)CO)nn1 44407,C(=O)(C#CC(C)(C)C)N1CCC(COC)(NC(=O)C(C)c2ccsc2)C1 44408,CCC(C)(C)CCCC(=O)N(CCCOCCNC(C1OCC2CCCC12)=O)C 44409,c1(C(=O)NCC2C(NC(c3c[nH]cc3Br)=O)CCC2)cc2nn[nH]c2cc1F 44410,N=c1[nH]c(=NCC23CC2COC32CCC2)[nH]c(=NCc2ccc3ccccc3c2)[nH]1 44411,N#Cc1cc(-c2cn(CCNC(c3ccc(OC(F)F)cc3F)=O)nn2)cc(F)c1 44412,C1(C(C)C)CN(C(C2(C3CCCO3)CC2)=O)CCN1C(=O)C=Cc1cnc[nH]1 44413,C12CCN(CC1(C)C)c1nnc(C3CC3)n1C2c1ccsc1S(C)(=O)=O.C1(C)CC1 44414,c1(OCC)ccc(C(=O)NCC(C)CN(C(=O)COCCCF)C)cc1C 44415,C1(C(C)(C)C)C(C(=O)N2CCCC2c2cc(F)ccc2F)=C(O)CCCC1 44416,C(C)(C(C(=O)NCc1cc(O)ns1)NC(c1nonc1C)=O)OC 44417,c1(C(N2CCN(C(C3C(=C)CC3)=O)C(C)C2)=O)cccc2nc(O)[nH]c12 44418,c1(C(=O)NC2C(CNC(CCCOC)=O)COC2)nccnc1C(N)=O 44419,C(=O)(C(=O)C(F)(F)F)N1CCC(C)C1c1cccnc1 44420,N(C1CCCc2n[nH]cc21)C(C1CC(CNC(COC(C)C)=O)OC1)=O 44421,c1(COC)ccnc(C(N2CCC(NC(=O)Cc3ccnc(Br)c3)C2)=O)c1 44422,c1(C(=O)NC(C)CC2CN(C(c3cnc[nH]3)=O)C2)cncc(N=[N+]=[N-])c1 44423,c1(CC)cc(NC(=O)C(CNC(c2cnc(C)s2)=O)N(C)C)cc(O)c1 44424,C1(C(CNC(c2scc(C(C)=O)c2)=O)(C)O)CCN(C(=O)C(F)OC(F)(F)F)CC1 44425,C(=O)(C1Cc2ccccc21)N1CCC(C)(NC(c2c(C)nc(CC)s2)=O)CC1 44426,c1(SC)ccc(C(=O)NC2CC2CNC(C2CC(C)(O)C2)=O)cc1 44427,C1(C(N2CC(C)(CCO)C2)=O)CCCN(C(=O)C(F)OC(F)(F)F)CC1 44428,c1(C(=O)N)ccc(N(C)CC)cc1.N1(C(CCOCC#C)=O)CCCC1CCCCC 44429,CC1(C)OCC2CC12C(=O)NOCCN(C1CS(=O)(=O)CC1O)c1ccccc1 44430,C1(CNC(C)=O)CCCCN1C(=O)NCC12CC(C(C)C)(CO1)C2 44431,C1(C)(NC(CC(C)c2cccnc2)=O)CCCN(C(c2cnc(O)n2C)=O)C1 44432,C(=O)(C(C)(C)CC(C)C)NCC1(OC)CCN(C(C2CCC=CO2)=O)CC1 44433,n1(CC)nccc1C=CC(=O)OCC1CCC(=O)NC1 44434,c1(OC)c(C(=O)NCC2(F)CC(CNC(=O)C3=CCCC3C)C2)cc(Cl)cc1Cl 44435,Cc1nc(C)c(C(N2CCC(C)(CCNC(c3scnc3Cl)=O)C2)=O)[nH]1 44436,N1(C(C(C(C)C)OCC)=O)CCN(C(C2CC(C)CCO2)=O)CC1CC(F)F 44437,Cc1cc(C(N2CC=CC(NC(C3(N(C)C)CC3)=O)C2)=O)c2c(c1)CCC2 44438,C12(C(N3C(C4(NC(Cc5c(C)ccs5)=O)CC4)CCC3)=O)CCC(CC1)OC2 44439,N1(C(c2cc(-c3cccnc3)no2)C(=O)NCC)CCC(CCC(C)C)CC1 44440,C1(=O)C2=CC(O)C(C2)N1.c1(C(N(C(C#C)(C)C)C2CC2)=O)cnn(C2CC2)c1 44441,C(=O)(C1Cc2ccc(F)cc21)N1CC(C)(C)C(NC(c2ccc(O)nn2)=O)CC1 44442,N1(C(C(CCC)O)=O)C2CCCC1CC(NC(c1coc3cccc(O)c13)=O)C2 44443,C1(NC(c2cccc(OC)n2)=O)CCCCN(c2cc(-n3ccnc3)ncn2)C1 44444,n1(CC(=O)NC2(C)CC(NC(c3n[nH]cc3Cl)=O)C2)ccc2ccc(F)cc12 44445,S(=O)(=O)(CC(C)C)NC(C1CN(CC(=Cc2cccs2)C)C1)=O 44446,C12(NC(c3ccc(CC)nc3)=O)CC(CNC(=O)Cc3[nH]cnc3C)(C1)OC2C 44447,CN1CC(O)CC1(C)C(=O)NCCCN1CCC(NC(=O)CC2C=CCC2)C1 44448,N1(C(C2(C)CCCCO2)=O)CCN(C(=O)CNC(c2ccncc2)=O)C(CO)C1 44449,c1(C(=O)NC2CC(NC(c3ccc(O)nc3)=O)C2)ccc2c(c1)C(=O)OC2 44450,N1(C(C(C)(C2(C)CC2)OC)=O)CC2C(N(C(=O)C(O)c3ccsc3)C)C2C1 44451,C1(CC)CCN(C(=O)CC2(O)CCC2)C(C(N2CCNC(=O)C2C)=O)C1 44452,CC(C)(C)C(CO)C(=O)NC1COCCN(C(C2CC2C#N)=O)C1 44453,C(C(CNC(=O)CC1CCCN1C)S(C)(=O)=O)NC(C(C=C)(C)O)=O 44454,C1(NC(CCC=CC)=O)CCN(C(c2ccc(F)cc2Br)=O)C12CCC2 44455,C#Cc1ccccc1NC(=O)C(CCC=C)NC(=O)CCCC(=C)C 44456,C(CCCCC(=O)N(C)CC1OCCC1(C)C)NC(C1CC(C(C)C)C1)=O 44457,Cc1cc(C(N2CC(N(C)C(C3CCC3(F)F)=O)C(C)(C)C2)=O)ncc1C(F)F 44458,N1(C(C2CC(C)N2C(c2cn(C)c(=O)n2C)=O)=O)CC(C)(CO)CC1(C)C 44459,C1(O)(C(C(=O)NCC#CC)F)CN(C(=O)C=NOC)C1 44460,C1(CNC(CCC(C)SC)=O)CCN(C(c2cn3ccsc3n2)=O)CC1O 44461,N1(C(C=Cc2cn(C)nc2)=O)CCCC2(C1)CN(C(=O)Cc1ccsc1Cl)C2 44462,C(=O)(CC(C)(C)CNC(c1sccc1C#N)=O)NCC(C)(C)C(F)F 44463,C(CC(=O)NCc1ccc(F)nc1C)(C(C)(C)C)NC(C(C)N(C(C)=O)C)=O 44464,Cc1cc(S(N)(=O)=O)oc1C(N1CCN(C(=O)COC2CCCOC2)C(C)C1)=O 44465,CC1CC(C)(C)CCC1Nc1cccc(SC(=O)OC(C)(C)C)c1.C1C(=O)N1 44466,C(=O)(C(C)(O)C1CCC1)NCC(C)CNC(C1(Br)CC1)=O 44467,N1(C(CC2(CC)CCC2)=O)CCCCC1CNC(C1CC(C)(O)C1)=O 44468,C1(C(=O)NC2CC(OC(F)F)C2)CCC2(CCCC2)C1 44469,CC1(C(=O)NCC#CC(=O)NCCCC2CCOC2)CCC(=O)C1 44470,N1(C(COc2cc(C)c(F)cc2)=O)CC2CCN(C(c3csnn3)=O)CC2C1 44471,C1(N(C(c2cc(C)n(C3CC3)n2)=O)C)CN(C(=O)C(C)c2cccs2)CC12CC2 44472,C1(=O)C(C(C)(C)C)n2cc(nn2)C(C(C)C)N1.C1(OCC)C(C(=O)O)C2CCCC12 44473,c1(C(N(CCNC(=O)C=CC(C)(C)C)CC)=O)cc(Cl)ccc1N 44474,C1(CNC(c2cc(Cl)ccc2OC(F)F)=O)CCCCN(C(C2COC(=O)N2)=O)C1 44475,c1(C(N2CC(NC(C3(SCC)CC(O)C3)=O)C2)=O)cc(S(N)(=O)=O)sc1Cl 44476,C1(C(=O)NC2(COC)CN(C(C3CCCC(F)C3)=O)C2)CC2(CSC2)C1 44477,N1(C(C=CC(C)(C)SC)=O)CCCC12CCN(C(C1CCN(CC(C)C)C1)=O)C2 44478,N1(C(C2CC(OC)C2)=O)CCN(C(c2ccc(SC)s2)=O)C(C)CC1C 44479,C=C(C)CCCC(=O)NC1(CNC(c2cc(F)ccc2OC)=O)CCCCCC1 44480,Cc1cc([N+](=O)[O-])cc(C(=O)NC2CN(C(=O)C=Cc3ccoc3)CCC2F)c1Cl 44481,C(=O)(C1=CCCSC1)N1CCC(CC#C)(C(=O)NC(COC)CO)C1 44482,c1(C(N(CCCN(C(c2c(C)ccs2)=O)C)C)=O)coc(C#N)c1 44483,C(=O)(C#CC(C)(C)CNC(c1cnn(CC)n1)=O)NC(C#C)CC1CC1 44484,c1(CNC(N2CCC(c3ccc(OCC)cc3)CC2)=O)ccc(OC)nc1C 44485,C(=O)(C(C)(C=C)CC)NCc1occ(C(=O)NCC(CC=C)OC)n1 44486,c1(N(CCNC(C2CC(C)N(C(=O)OC(C)(C)C)C2)=O)C)ncc(Cl)cc1F 44487,C=C1COc2c(C(=O)N(CCC(C)NC(C3(Br)CC3)=O)C)cnn2C1 44488,C1(C(=O)NCC(CNC(COCC(C)C)=O)O)CCCCCN1C 44489,CC1COc2cc(NC(=O)CCN3CCCCC(CN)C3=O)ccc21 44490,C1(NC(C2CC(OC)(OC)C2)=O)CCCN(C(=O)C(CC)n2ccnc2)CC1 44491,C1(CCOC)(NC(C2C=CC=CC=C2)=O)CCN(C(=O)CCc2cncnc2)C1 44492,c1(CC(N2C(C(C)NC(C3(C)CCCC3)=O)CCC2)=O)ccc(Br)c2cccnc12 44493,C1(CC#C)(C(=O)NCC(O)CNC(c2conc2C2CCCC2)=O)CCCCO1 44494,Cc1cc(=NC(C)c2cccs2)[nH]c(=NCCOC2CCCC2)[nH]1 44495,c1(CC(=O)NCCC(CNC(C=C(C)C(F)F)=O)O)csc2c(F)cccc12 44496,c1(OC)cccc(C(=O)NCC2(F)CCN(C(=O)CC3C=CCC3)C2)c1F 44497,N1(C(C(CC(=O)OC)(C)C)=O)CCCC12CCCN(C(=O)C(O)C(C)C)CC2 44498,c1(OC(CC)C)cc(CN2CCC(C(=O)N(C)C(C)C)CC2)ccc1OC 44499,C(=O)(C1CCCc2nncn21)NC(C)CCNC(c1cnc(O)c(Br)c1)=O 44500,Cc1c(CC(=O)NC(C)(C)CNC(=O)C=Cc2cnccn2)ccc(Cl)c1Cl 44501,Cc1noc(CCCCNC(=O)CN2CCOCC2)n1 44502,Cn1cc(C(=O)NC2CCC2C(=O)NC2CCC2(C)C)nn1 44503,C1(CCOC(C)(C)C)(c2n(CCOCC)nnn2)CN1.c1(CC)scnc1C 44504,C1(CC(=O)NCCCN(CCCN(C(c2ccncc2)=O)C2CC2)C)CC2CC1C2 44505,N12CCCN(CC1)C(=O)CC1CC(C1)C2=O.c1(SC)snnc1N(C)C 44506,c1(OC)cc(CC(N2CC(N(C(=O)C(C)C(C)C)C)C(O)C2)=O)ccc1Cl 44507,Cc1cnc2nc(C(=O)NC3(C)CCN(C(c4cc(C)nnc4O)=O)C3)nn2c1 44508,Cc1cc(C)nc(-n2nccc2C(N2CCC(C(N3CCOCC3)C3CC3)C2)=O)n1 44509,C=CC1CN(C(C2CC3(CCC3)C2)=O)CC1NC(c1cn(CC)nc1C)=O 44510,C1(C(N(CC(C)C#N)C)=O)CCN(C(=O)Nc2ccco2)CC1 44511,n1(CC)cc([N+](=O)[O-])c(C(=O)NCCCCN(C(=O)Cc2cc(C)sc2C)C)n1 44512,C1(NC(C(C)SCC)=O)CN(C(c2cnn(C3CCC3)c2C)=O)CCC1F 44513,C#CCC(C)(C(=O)NC(c1nn(C)cc1O)C)NC(=O)C(C)=CC 44514,c1(N2CC(CNC(C3(C(N)=O)C(C)(C)C3)=O)C2)nnccc1C#N 44515,Cc1ccc(C(F)CCOC(C)(C)C)cc1C.C12CCN(CC1)C(=O)C(=O)N2C 44516,CN1C(=O)NCC1C(=O)NCCOCCNC(C1OC2CCC1C2)=O 44517,N1(C(c2cc(CC)on2)=O)CCN(C(=O)C(=CC2CCCCC2)F)C(C)C1 44518,C1(C)(CCNC(C2CCC(C)O2)=O)CCN(C(c2cnccc2Cl)=O)CC1 44519,c1(N2CCN(C(Cn3c(C)ccc3C)=O)CC2)c(Br)cccc1[N+](=O)[O-] 44520,C(CCO)(CC(C)C)NC(c1cnc(CNC(C2CC(C(=O)OC)C2)=O)nc1)=O 44521,C12CCC(CC1)CNC2=O.c1(CC(=O)N(C)CC2CCCCS2)csc(Cl)c1 44522,C(CCS(=O)(=O)c1ccccc1)N(CC(=O)NC1CCCC(C(F)(F)F)C1)CC 44523,c1(CCN2C(C)C(NC(=O)CC3CCC=CO3)CCC2)cc2ccccc2o1 44524,CCC1=C(C(=O)N2CCCCCC(NC(c3ccc(O)nc3)=O)C2)CCCO1 44525,C1(C(N2CC(F)(CNC(c3c(C(C)C)ccs3)=O)C2)=O)CCCC2(CCC2)O1 44526,C#CCCCC(C)C(=O)N1CCCC1(C(F)(F)F)CNC(=O)C=CCN(C)CC 44527,C(C(C)(F)C(C)(C)F)ONC(C1(C)CCCC1NC(c1ncnc(O)c1F)=O)=O 44528,C1(=O)CC(Cc2ccccc2)N1.C1(CC(=O)OC)CSCCN1S(=O)(=O)C1CC1 44529,c1(N(C)C)cc(CNC(=O)C(c2ccc(Cl)c(F)c2)F)cc(Br)c1 44530,c1(C(N2C(C)C(NC(c3csc4cncn34)=O)CCC2)=O)cccc2oncc12 44531,S(=O)(=O)(c1ccc(C#N)cc1OC)NCc1c(OC)nccc1 44532,Cc1cc(C(=O)N(CC(O)CN(C(=O)C(C(C)C)n2ccc(C)c2)C)C)n(C)n1 44533,N1(C(CCNC(CC(c2cccc(F)c2)O)=O)=O)CC2CCCC1C2CO 44534,Cc1ccc(F)c(N)c1C(N1CCN(C(=O)CC2CC3(CCC3)CO2)C(C)C1)=O 44535,C(C(=O)N1CC(O)CC1CC(=O)NC1CC(CO)C2CC12)(C(C)C)SCC 44536,N1(C(CNC(=O)CC(F)(F)F)=O)C2CCC1CN(C(=O)CC(F)(F)F)C2 44537,N1(C(C(C2CCC(=O)N2)C)=O)CCN(C(c2ccc(CO)c(Cl)c2)=O)CC1CO 44538,N1(c2nnc(C(C)C)o2)CC2(CCC2)CC1CNC(c1ccc(F)c(Cl)n1)=O 44539,C(C(CO)C(F)(F)F)NC(=O)CSCC(=O)Nc1sccc1SC(F)F 44540,N1(C(CN(c2ccccc2)C)=O)CCOCC1CCNC(C1CC1C1CC1)=O 44541,N1(C(Cc2c(C)cco2)=O)CCCC(C)C1CCNC(c1cocn1)=O 44542,N1(C(CC)=O)CCC(CC)C1CNC(c1cnc(S)n1C)=O 44543,Cc1c(C(=O)NCC(C)CN(C)C(C2OCCC2C(C)C)=O)cncc1N 44544,C12(C(=O)NCC3(O)CN(C(=O)CCc4csnn4)C3)CCCCC1CCC2 44545,c1(C(=O)NC(CN(C(=O)C(C)CC2CCCC2)CC)C)cccnc1C 44546,C(=O)(C1CCCc2c[nH]nc21)NC1C(CNC(CSCC(C)C)=O)COC1 44547,C1(NC(CCNC(=O)CO)=O)C=CCN(C(=O)Cc2ccc(OCC#N)cc2)C1 44548,N1(C(CC(=O)OCC)=O)CC(NC(c2ccc(C(C)C)o2)=O)CC2(CCC2)C1 44549,C1(NC(c2c(C)nn[nH]2)=O)CN(C(=O)CCSC(F)(F)F)CCC1F 44550,Cc1nnc2n1CCC(C(=O)NC(C1CCN(C(C3CSCCS3)=O)C1)C)C2 44551,Cc1ccc(C(C)C)cc1C(=O)NCC1CCN(C(c2coc(C3CC3)n2)=O)C1 44552,C1(CNC(c2c(SC)cccc2)=O)CC(C)(C)CN1C(c1cc(C#N)oc1C)=O 44553,C1(CC(=O)NC(C)(CCNC(=O)NCCc2ccccc2)C2CC2)CCCCC1 44554,C#CC1CN(C(c2sc(Br)cc2C)C(=O)NC2COC2)CC1O 44555,CC1CN(C(=O)C=Cc2cccnc2)CC(C)N(C(c2cscn2)=O)C1 44556,N1(C(C(CCC)F)=O)CCC=C(C(=O)NC2CCCC(O)CC2)C1 44557,c1(C(N2CC3C(CNC(C4CC(=O)OC4)=O)C3C2)=O)ccc2nnn(O)c2c1 44558,CC1(CNC(C2CNC(=O)C2)=O)CCCN1C(c1ccc(C#N)o1)=O 44559,c1(NC(N(C2CS(=O)(=O)C2(C)C)C)=O)ncc(S(C)(=O)=O)cc1Cl 44560,C(C(=O)N(C1CCN(C(=O)CC2(CSC)CC2)C1)CC)(C(C)C)OCC 44561,C=CCC(F)(F)C(=O)N1CCCC1C(=O)NCc1nc(C(N)=O)no1 44562,Cc1cc(C(c2nnnn2C2(C)CC2)NC2CCC(F)(F)CC2)cc(C)c1Br 44563,N1(Cc2c(C)nncc2)CC2CC1CN2C(=O)C(=O)Nc1ccccc1 44564,C1(C(=O)NC2(C)CC(C(=O)OC)C2)CCN(C(C2CCCC(C)O2)=O)CC1C 44565,c1(C(N2CCN(C(C(CC=CC)C)=O)CC2C2CCC2)=O)ccc(C#N)cc1C 44566,O=C(C1=CC2CC=CCC12)NCC#CCNC(C1(O)CC(F)(F)C1)=O 44567,C1(F)(CNC(CSSC)=O)CCCN(C(c2cccc(C(N)=O)c2)=O)C1 44568,C1(CC(C(=O)OCC)NC(=O)C(c2ccc(F)cc2)N)CCC(F)(F)CC1 44569,c1(CN2C3CCN(C(c4c(C#N)cc(Cl)cc4)=O)C3CC2)cc2cc[nH]c2cn1 44570,CC1CCC(NC(c2ccc(Cl)c(C(F)F)c2)=O)CN1C(c1cnnn1C)=O 44571,N1(C(C(C)=C(CC)C)=O)CCCCC2(CCN(C(c3ccn(CC)c3C)=O)C2)C1 44572,C1(C(=O)NCCCCCNC(C(C)OCCOCC)=O)CC2CC1CC2(F)F 44573,N1(c2cc(NC3(C)CC4CCC3CC4)ncn2)C2CCC1c1ncccc12 44574,c1(-c2c(OC)cc(C(=O)Oc3cc(Cl)ccc3I)nc2)c(C)cc(Br)cc1C 44575,N1(C(CCSCCC)=O)C2CCC(C(=O)Nc3conc3C)C1CC2 44576,N(C(=NCCc1nccs1)NC1CC1)C(C1CCS(=O)(=O)CC1)C 44577,C1(NC(COc2cc(C)on2)=O)CN(C(C2CCOC2)=O)CC1C(F)F 44578,CC1(C(=O)NC2CC(CCC(=O)NC(C(O)CO)C3CC3)C2)CCC(=O)N1 44579,CC(N=[N+]=[N-])C(=O)N1CC=CC1NC(C1C2CCCOC12)=O 44580,CC(C)(C)CCCCCC(=O)NCC1(O)CCN(C(=O)CCC2CCC(=O)N2)C1 44581,C1(NC(C2(CC)CCOC2)=O)CCC(C)N(C(c2cnn(C)c2C(F)(F)F)=O)C1 44582,C1(NC(C(c2ccccc2)C)=O)CCC(CCNC(=O)C=CSc2nc[nH]n2)C1 44583,C1(OC)CCN(C(C2CC2C(C)NC(C2(C)CSC2)=O)=O)C1C 44584,C1(O)(CC)CCCN(C(=O)Nc2nc(C)cc(O)n2)C1 44585,c1(OC)c(C(=O)NC2CN(C(=O)C(C)C#N)C2)csc1C 44586,C(=O)(CC1=NN(C)C(=O)C1)N1CCC2(C(NC(C(CSC)OC)=O)C2)C1 44587,c1(N2CC(N(C(c3cn(CCC)nn3)=O)CC)C2)ncc2cccnc2n1 44588,N1(C2(C)CCC2)CCC(NC(=NCC2CC2CF)NC2CCCCC2)CC1 44589,N#CC1(C(=O)NCC2CCN(C(=O)C3=CCCS3)C2)CC12CCCC2 44590,c1(OCC(=O)OC)ccc(S(=O)(=O)NC(C)(C)CCC(=O)O)cc1OC 44591,n1(CC(N2CC(N(C)C(c3cncs3)=O)C2)=O)cc(Br)c(C(F)(F)F)n1 44592,CC(C)(C)CC(CO)NC(=O)CC(C1CC1)NC(C1CC(C2CC2)C1)=O 44593,c1(C(N2CCC(c3ccccc3F)C2)=O)ccc(-n2ccnc2)cc1[N+](=O)[O-] 44594,C1(N(C(C(CC)n2cccn2)=O)CCO)CCCN(C(c2ccc(Cl)cn2)=O)C1 44595,Cc1ccc(S(C)(=O)=O)cc1C(=O)NCCCCC(C)NC(C1(F)CCC1)=O 44596,c1(ONC(c2cc(CNC(C3CN(C)C3)=O)sc2)=O)nccc(Cl)c1Cl 44597,O=C(CCS(=O)(=O)Cc1ccccn1)NCCNC(C1CCCOC(C(F)F)C1)=O 44598,N1(CC)CCCC1C(=O)NCCCN(C)C(c1cc(C(=O)OC)co1)=O 44599,c1(C(=O)NCC2CC(NC(CC3CCC(C)C3)=O)C2)csc(=NC2CC2)[nH]1 44600,c1(OC)cc(OC)cc(C(=O)NC(CNC(=O)CC2CC23CC3)CCOC)c1 44601,C1(C(=O)NCC#CCC)CN(C(C2CCCN2C=O)=O)CCN1C 44602,N1(C(Cc2ccc(OCC=C)cc2)=O)CCC(NC(c2cc(C)ns2)=O)C(F)C1 44603,S(=O)(=O)(c1ccc2[nH]c(=NCC(C)(C)C(F)F)sc2c1)NCc1c(OC)cn(C)n1 44604,c1(C(=O)NCCN(C(=O)C(c2cccc(F)c2)O)C)ccc(O)c(Br)c1 44605,n1(CC)c(C(=O)NC(C)C(C)NC(c2ccoc2C)=O)nc2ccccc12 44606,N1(c2nc(C)cc(OC)n2)CC2CN(Cc3ccc(N4CCCC4)s3)CC2C1 44607,c1(C(C(=O)OCc2cc(-c3ccccc3)[nH]n2)C2CC2)ccccc1F 44608,C1(CNC(CCc2nnc(C(C)C)o2)=O)CCCC(NC(c2cscc2C)=O)C1 44609,c1(C(=O)NCCCN(C2CCCC2)C(C2CC(=C)C2)=O)cc([N+](=O)[O-])sn1 44610,C#CCC(C)(C(=O)NC1CC(OCC)C1)N(C(=O)C(C)SCC)C1CC1 44611,c1(NC(=O)CCc2ccoc2)cccc(CC(F)(F)F)c1.CCC1CNC(=O)N1 44612,N1(C(C(C(COC)C)C)=O)CCCC2(C1)CN(C(=O)CNc1cccc(F)c1)C2 44613,c1(CC(N2CCC(CN(C(c3cn(CC)nc3C)=O)C)C2)=O)ccc(C)cc1C 44614,c1(C(N2CCCC(CNC(CC(C)SC)=O)C2)=O)cnn2c1S(=O)(=O)NCC2 44615,c1(C(N2CCCC(CCNC(c3cc(C)n(CO)n3)=O)C2)=O)cccc(N)c1C 44616,N1(C(c2n(C)nc(O)c2)=O)CCC(C(N2CC3CC(O)CC2C3)=O)CC1(C)C 44617,C1(CNC2CCC(CC(C)OCCC(C)C)CC2)CC2CCC(C1)N2 44618,N(C)(S(=O)(=O)N1CCC(CCOC)C1)CCCC(C)C 44619,N1(C(C(=O)NC(C(=O)OC)C)c2cncs2)CCn2ncc(C(F)(F)F)c2C1.C1(C)CC1 44620,n12c3c(cc(cc3)c1=O)CC2.C1(C(N(CCNC)CCOC)=O)CCNC1=O 44621,C1(CNC(C(F)OC)=O)CN(C(c2cccnc2C)=O)C2CCCCC12 44622,C(=O)(CCCC(CC)NC(C1(CCC)CCC1)=O)NC(C#C)C(C)(C)C 44623,C(=O)(C(C)(C)C(=O)NCC(C1CCCCC1)NC(c1occc1C(C)C)=O)NC 44624,N1(C(C(C)NC=O)=O)CCCC1(C)CNC(C1CCCC2CC12)=O 44625,c1(C(N(C2CCC(NC(=O)CSC)CC2)CCCC)=O)cccc(S(N)(=O)=O)c1 44626,c1(C2C(OC(n3nnc(-c4cccs4)n3)=O)C2)ccc(Br)cc1 44627,N1(C(Cc2nn(C)c(Cl)c2)=O)CCC(C2CN(C(=O)CC(=O)NC3CC3)C2)CC1 44628,C1(CNC(C(C(=O)OCC)F)=O)N(C(c2ccc(F)c(CC)c2)=O)CCC1(C)C 44629,Cc1nc2nccc(C(N3CC(NC(=O)CC(O)CN(C)C)C4(CC4)C3)=O)n2n1 44630,N1(C(c2nc(C(=O)OCC)sc2)=O)CCCCC(CNC(C2CCCO2)=O)C1 44631,N1(C(c2ccn(C)c2)=O)CCC(CO)(CNC(C2CCCC23CC3)=O)CC1 44632,S(=O)(=O)(c1ccc(NCCCS(C)=O)c(C#N)c1)NC1CN(CC)C1 44633,c1(C(=O)NCCCN(C(C(C)=C2CCC2)=O)C2CCCC2)cccc(C(C)(C)C)c1 44634,C(CCCCCN=c1nc(-n2ccnc2)cc[nH]1)N(C)C(C12CCCCC1C2)=O 44635,c1(C(=O)NC(C(C(C)C)NC(=O)C=Cc2ncc[nH]2)C)cnn2cccnc12 44636,CCC(CC)C(C(=O)NCC(CCC)C(=O)NCC1CCCCN1C)OC 44637,CCC(C(=O)NC(C1(O)CN(C(c2cc(C)cs2)=O)C1)C)OC 44638,N1(C(C2C(=C)CC2)=O)CCC2(NC(=O)COc3ccccc3OC(C)C)CC2C1 44639,CCC(CNC(=O)C=CC(=O)N(C)C)(CC)NC(=O)C(C)Cc1ccccn1 44640,C(CCC(O)C(=O)N1CCCC(O)C1)NC(c1c(CC)ocn1)=O 44641,O=C(O)CC(C(=O)O)NC(=O)NCC12COC(CF)(C1)C2 44642,c1(C(=O)NC2CCCN(C(C=CC(C)C)=O)C2)ccc(C(F)(F)F)c([N+](=O)[O-])c1 44643,Cn1nnc(C(=O)NCCCC(C)(C)NC(C2CC3(CC3)C2)=O)c1C(F)F 44644,C(=O)(C1=CCCSC1)NCc1cncc(C(=O)NC(CCCC)CC)c1 44645,O=C1C2CC(C(=O)NCCCn3cnc4ccccc34)CC1CC(F)(F)C2 44646,Cc1cn2c(n1)CC(C(=O)NC(C)CC1CN(C(=O)CNC=O)C1)CC2 44647,n1(CC(=O)NC(C(C)NC(=O)C=Cc2ncc[nH]2)(C)C)ccc(O)nc1=O 44648,c1(-n2cc(C(=O)NCC3N(C(=O)OC(C)(C)C)CCC3)nn2)cnccc1C(=O)O 44649,C(=O)(CCCS(N)(=O)=O)N(CCCNC(c1ccc(-c2ccccn2)o1)=O)CC 44650,c1(C(=O)NCC(C(C)(C)C)NC(c2c(OC)cncc2)=O)n[nH]c2c1CCOC2 44651,Cn1nc(Br)cc1CCCCNC(=O)N(C1CCC(OCCO)CC1)CC1CC1 44652,C1(C(C(=O)NCc2ccc(C(C)O)cc2)O)CCC(C)(C)CC1.C(=O)(NC)O 44653,CC1CN(C(=O)CCc2cncnc2)CCC1NC(=O)C(F)=CC1CC1 44654,C(C)(CCC(=O)NCCCOCCOCCNC(c1ncccc1Cl)=O)OC 44655,C1(F)(CNC(c2n(C)ncc2)=O)CCCN(C(C2CC(=O)N(CC3CC3)C2)=O)C1 44656,N1(C(c2c(C)ccc(C)n2)=O)CCC2(CC1)CN(C(=O)CCCCC#N)C2 44657,N1(C(C(C)OCC=C)=O)CCCC(CNC(C2CC2C=C)=O)C1 44658,C1(CNC(CC2(OC)CCC2)=O)CN(C(=O)CC2(OC)CCC2)CC12CC2 44659,N1(C(CC2CC(C)(C)C2)=O)CCN(C(=O)CCCc2ccc(O)nn2)C2CC12 44660,N1(C(C(Cn2cncn2)SCC)=O)CCN(C)C(=O)C1.C1(C)C(=O)N1 44661,C(=O)(CCCC(F)(F)F)N1C(CNC(c2ccc(C(F)F)nc2)=O)CCCC1 44662,c1(CN2C(CC(=O)N(CCCC)CCCC)CCC2)nc(O)c2c(C)c(C)sc2n1 44663,C1(NC(C(CC=C)NC(C)=O)=O)CC2CCC1CN2C(=O)C(C)OCC(C)C 44664,C12(CNc3c(C)cnc(F)n3)CCC(CNC(=O)CCC(N)=O)(CC1)CO2 44665,N12CC(C3(CC3)C1)c1cn(nn1)-c1cccc(n1)C2=O.C1(Cl)(CC)CC2CCC1O2 44666,C1(CC)(NC(=O)CC2=CCCC2)CCCN(C(c2csc(S)n2)=O)C1 44667,C1(C(N(C(CC#C)C)C)=O)CCCN1C(C1CC1(C)C)=O 44668,C12(C(C)NC(C(COCC)NC(C3CC(F)(F)C3)=O)=O)CCC(CC1)C2 44669,C(=O)(CC(C(=O)N1CC(OC)C(NC(=O)Cn2cnc(C(N)=O)n2)C1)N(C)C)OC 44670,N1(C(=O)Nc2nc(=N)[nH][nH]2)CCNCC1c1cccc(Cl)c1 44671,c1(NC(C)=O)ccc(C(C)NC(=O)CCNc2ccc(C(C)(C)C)cc2)cc1 44672,N1(C(C(COC)(F)F)=O)CCCCC(NC(c2cnn(C)c2C)=O)C1 44673,N1(C(CN2CCN(C)CC2)=O)Cc2nccn2CC(NC(C2CCSCC2)=O)C1 44674,c1(CCCC(=O)OC(C)=O)ccc(Cl)cc1.C1(=O)CCCNCC2(CC2)C(C)N1 44675,C1(C(=O)Nc2ccc(CNC(C(C(=O)OC)OC)=O)cn2)CCC2(CC1)CC2 44676,N1(C(COCCOCC)=O)CCC(C(N2CC(C3(C)CC3)C2)=O)C1(C)C 44677,N1(C(Cc2c(C)nc(C)s2)=O)CCCC(NC(c2cnc(-c3ccco3)s2)=O)CC1 44678,C(CCC(=O)NOC(C)C)(CC(C)C)CCC.C(=O)(CSCC)N 44679,N1(C(c2ccc(CC)cc2)=O)CC(NC(=O)COCCSC)C2(CC2)C1 44680,C12(C(=O)NC(C)C(C)NC(c3ccc(O)nn3)=O)CCCN(CCC1)C2 44681,C(CC(C(=O)NCC1CCCC1O)NC(=O)C(C)CO)OC 44682,CCC(C)(CNC(=O)C(C)N(C)C)C(=O)NCC1CCCCO1 44683,O=C(C1=CCOC1)NCC1CN(C(=O)C(F)(F)Oc2ccc(F)cc2)CC1O 44684,C(=O)(CCCC(=O)C1CC1)NCCCNC(Cc1cc(C)sc1Cl)=O 44685,c1(SC)cccnc1C(N1CCC(NC(c2cnc(O)o2)=O)CC1)=O 44686,N1(C(C(CC=CCC)C)=O)CCC2(CCC2NC(c2ccnc(C)n2)=O)CC1 44687,N1(C(c2c(CC)n[nH]c2)=O)CCCCCCC1C.C12CCCC1C(=O)NC2 44688,C(CNC(=O)C(=O)C(C)C)(CC(=O)N(C(CO)C1CC1)C)OC 44689,CCC(C)C1C(=O)NC(C)CNC(=O)C2CC(=NO2)C(=O)N1.C(C)(=O)OC 44690,c1(NC(C(C)OC2CCCC(C)C2)C)cc2cc(Cl)ncc2o1 44691,CC(CC(=O)N1CC2CCC(O)C2C1)C1=CCCCC1.C12=CC=C(C=C1)C2 44692,c1(C2C(C(c3c(C)nsc3Br)Nc3n(CCC)nnn3)C2)ccccc1N(C)C 44693,C1(NCc2c(CC)cccc2)CCN(C(c2coc(Cl)n2)=O)CC1C 44694,c1(CC(=O)NCC2N(C(C(CC)F)=O)CC=C2)cc(C)cc(Br)c1 44695,CCC(O)C(C)(C)C(=O)NC1CC(NC(C2(COC)CCC2)=O)CC1O 44696,C(=O)(CS(=O)(=O)NC)NC.CCCC(O)CN1C(=O)C(C2(O)CCC2)NC1=O 44697,c1(C(=O)NC2C3CC2N(C(=O)C(F)OC(F)(F)F)C3)cc(F)ccc1F 44698,N1(C(C2(C)N(C(CCN(CCC)C)=O)CC2)=O)CCCC1CC(N)=O 44699,CC1CC(NC(=O)CCc2nccs2)CN1C(c1ccccc1O)=O 44700,N1(C(C2N(C(C3(C)CC(=C)C3)=O)CC(C)C2)=O)CCC(O)C(C)C1 44701,CC1(C(=O)NC(CNC(c2ccccn2)=O)CO)CCCOC1 44702,C1(NC(=O)CCc2cncs2)CC1C1CCCN(C(c2cc(Cl)cs2)=O)C1 44703,C1(C(=O)O)C(C(=O)NCCC(O)c2ccsc2)C1(F)F 44704,C1(CCNC(C(c2ccccc2)SC)=O)CCCN1C(C1CN(S(C)(=O)=O)C1)=O 44705,N1(C(C2CCN(C(C(N3CCOCC3)C)=O)C2)=O)CC(C)(C)CC1CC(=O)O 44706,N1(C(CCC2(C)N(C(c3ccc(OC)o3)=O)CCC2)=O)CCCNC(=O)CC1 44707,O=C(C1=NOC(CNC(c2c[nH]c(=O)cn2)=O)C1)NCCC1(CO)CC1 44708,N1(C(C2CCC2)=O)CC23CCCC2(C1)CN(C(C1CCC2CC2C1)=O)C3 44709,N1(C(C(CCOC)NC(=O)CCC(CF)CF)=O)CCCC2CNC(=O)C12 44710,C(CS(=O)(=O)CC(=O)NC(C)(C)CC=CC(=O)NCCCN(C)C(C)=O)OC 44711,CC(CC(C)(F)F)C(=O)NCCCN(C(=O)CCCc1nncn1C)CCO 44712,c1(N(C(C)=O)C)ccc(NS(=O)(=O)NC(=O)CCc2ncccn2)cc1 44713,C(=O)(C(C)CC1CC1)NCCCN(C(c1ncoc1C1CCC1)=O)CC 44714,C=CC(C)(C)CCCN=c1[nH]c(N(CC(Cl)(Cl)Cl)C)nc2c1CCC2 44715,C1(NC(c2c(CC)occ2)=O)COC2(CNC(c3ccc(Cl)c(O)c3)=O)CC1C2 44716,C1(N(C(=O)C(F)=C2CCC2)CC)CCN(C(=O)Cc2cnn(C(C)C)c2)C1 44717,Cc1ccc(C)c(C(N2CCC(CNC(=O)C=Cc3ccc(=N)[nH]c3)C2)=O)c1 44718,N1(C(c2c(C)cccn2)=O)CCCC(C2CC2NC(=O)CCC(F)F)C1 44719,N1(C(COCCCC)=O)CC(CNC(c2cnncc2OC)=O)OC2(CCC2)C1 44720,c1(C(=O)OC)cc(F)cc(F)c1NCc1cnc(C(F)(F)F)s1 44721,C1(CC=C)(NC(c2ccc(OC)nn2)=O)CCCN(C(c2nsnc2O)=O)C1 44722,C=C1CC(N=c2[nH]c(=NCC(=O)N3CC=CC3)[nH]c3cc[nH]c23)C1 44723,C#Cc1cc(C(N2CC(C)N(C(C3CC3C(N)=O)=O)CC2C)=O)cc(F)c1 44724,N1(C(c2cncc(C)n2)=O)CCC(NC(=O)CCc2ccnc(Cl)c2)C1(C)C 44725,C12(NC(=O)Cc3nc(F)c(F)cc3F)CCCN(C(c3cnsc3)=O)CC1C2 44726,C1(NC(CSCCOC)=O)CN(C(=O)C(c2cnc(O)nc2O)(F)F)CCC1C 44727,N1(C(C(CO)N(C)C)=O)C2CCCC1CC(NC(c1ccn3nccc3c1)=O)C2 44728,C(N(CC(C)C#N)N1CCCC(F)(F)C1)c1cnc(C)s1 44729,CCS(=O)(=O)c1ccc(S(=O)(=O)NC2(CO)CC(c3ccccc3)C2)cn1 44730,C1(CC)CN(C(c2cc(C)ncn2)=O)CC1C(=O)NC(CC1CC1)C1CC1 44731,CC(CC(=O)N1CCC(NC(=O)C=Cc2ccc(C(N)=O)o2)C(F)C1)C(C)(C)C 44732,c1(CC)ccc(C(N2CCCC2CCCNC(=O)C#CC2CC2)=O)c(C)c1 44733,C(C(C)(O)CC(=O)N1CC(F)(F)CC1C(N1CC2CC2C1)=O)OC 44734,c1(CC)cc(C(N2CCC(NC(c3cc(Cl)n[nH]3)=O)C(F)C2)=O)ccc1OC 44735,C(c1ccccc1F)=CCC(N1CC(CCO)(NC(c2cc(C#N)[nH]c2)=O)C1)=O 44736,C(=O)(C1OCCc2c(Br)cccc21)NCCCCN(C(C(CC)C)=O)C 44737,C(=O)(C#CC1CCCCC1)NCCCN(C(C1CCC(C)S1)=O)CC 44738,c1(CC)cc(C)nc(N2CC3CC(NC(C4(C5CCC5)CCC4)=O)C3C2)n1 44739,CCCCCCC(=O)N(C)CCc1[nH]c(-c2ccc(OCC)cc2)nc1C 44740,CC(=Cn1ccnn1)C(=O)N1CC2(CCN(C(=O)CC3CC4CC4C3)C2)C1C(C)C 44741,CCCCC(O)C(=O)N1CCC(CO)C(NC(=O)CCC2CCC2)C1 44742,C1(NC(C(c2ccc(C)cc2)C)C)CCN(C)C(C)C1 44743,c1(C(C)C)cc(S(=O)(=O)NC2CCCC2CCCC(=O)O)n(C)n1 44744,c1(C(N(CC(C)N(C(C(CCOC)C)=O)C)C)=O)cc(OC(C)C)ccc1Cl 44745,c1(OC)cc(C)ccc1OCC(=O)NC(CNC(c1cn(C)cn1)=O)C(C)(C)C 44746,c1(C(=O)NC2CN(C(CC(C=C)(C)C)=O)CC(C)C2)c(F)ccc2n[nH]cc12 44747,O=[SH](=O)c1c(Cl)cc(Br)cc1Cl.C1(S)CC(=O)N(CC2CCC2)C1 44748,Cn1nc([N+](=O)[O-])cc1C(=O)NC(C)(C)CNC(=O)C(c1cncn1C)O 44749,C1(CNC(c2c(C)cns2)=O)CC2(CCN(C(C3COCCN3C)=O)CC2)CO1 44750,C1(C(N2CCCC(N(C(c3c(CC)scc3)=O)C)C2)=O)CCc2ncncc2C1 44751,c1(C(N(CC(C)N(C(C(C)n2cnnn2)=O)C)C)=O)c(O)nnc2c1COCC2 44752,C12(NC(C=CC(CC)C)=O)CCC(C1)N(C(c1ccc(OC)nc1C)=O)C2 44753,C1(CNC(c2c(C)nns2)=O)CCCN(Cc2cnccc2C(F)(F)F)C1 44754,CCCN=C(NCC1CC1c1ccc(F)cc1)NCc1nc(C)cc(C)n1 44755,N#CC1CC12CCN(C(C1(F)CCN(C(C3CCNC3=O)=O)C1)=O)CC2 44756,C12(CNC(CCC(=O)NC)=O)CCC(CNC(C3CC3(C)C(C)C)=O)(CC1)OC2 44757,c1(COC)ccc(C(=O)NCCC(O)CNC(c2cccn2C2CC2)=O)cc1 44758,c1(CN(C(=O)C=CCN(C)C(C2CC2(C)C)=O)C)cnsc1 44759,N1(C(C(=C2CN3CCC2CC3)C)=O)C2CCC1C(NC(c1cc(Cl)cnc1C)=O)C2 44760,C(C)(C)(CCCC(=O)NC(c1ncc(C)o1)C)NC(C(CC)n1ccnc1)=O 44761,c1(C(C)NC(c2c(Br)cnn2C)c2n(CCOC)nnn2)ccc(F)cc1 44762,c1(OCC)nccc(C(=O)NCC2CC(OC)CN2C(c2cncs2)=O)c1F 44763,CC(C)C(O)C(F)(F)C(=O)NC(C1CN(C(=O)C(C)O)C1)C 44764,C1(NC(c2cn3ccsc3n2)=O)CN(C(=O)C(Cl)=CCl)C2(CCCC2)C1 44765,C(CC)(C(=O)NCC(C)(F)F)NC(C(F)=CCC)=O 44766,Cc1cc(=NC(=O)C(CNC(c2cncc(F)c2)=O)N(C)C)[nH]n1C 44767,C(C1=CCC2CC1C2(C)C)(c1nnnn1C)Nc1cccc(C(C)C)c1 44768,N1(C(CCc2c(C)noc2)=O)CCN(C(C23CC(CO)(C2)OC3C)=O)C(C2CC2)C1 44769,C1(CC)(NC(C2CCCCC2)=O)CCCN(C(C2CCS(=O)(=O)N2)=O)C1 44770,c1(C(=O)NC(CC=C)CNC(c2c(C)ncnc2O)=O)cnc2n1CCCC2C 44771,N12CC(C(F)(F)C1)C(=O)C2.c1(CC(C)C)ccccc1N(C)C 44772,c1(C(=O)NC2CCC(NC(C(CC)OC3CCCC3)=O)C2)ccccc1CC#N 44773,c1(C(C)=O)c(C)[nH]c(C(N2CCC(O)C(NC(=O)C=CBr)C2)=O)c1C 44774,c1(COC)ccccc1C(=O)NCCCN(C(=O)CCC(=O)OC)C(C)C 44775,c1(NCC2C(NC(c3ocnc3C(F)F)=O)CCCC2)ncc2cccnc2n1 44776,C1(NC(CC2(CNC(Cn3ncc(CC)c3)=O)CC2)=O)CCCC1N=[N+]=[N-] 44777,n1(CCC)ncc(C(N2CC3C(NC(c4n[nH]c(C5CC5)n4)=O)C3C2)=O)c1C 44778,c1(N(C2CC2)OC)cccc(NC(C2CCCCC2)C(=O)NC2C3CCCC23)c1 44779,N1(C(c2c(OC)cccc2C)=O)CC2CC3CC2C1C3NC(c1cocc1C)=O 44780,c1(OC(C(C)C)C(=O)NC2CCN(C(=O)CN(C)CCO)C2)ccc(F)cc1F 44781,N1(C(C)C)CCCC(C(N2CC(F)CC2CNC(=O)COc2ccccc2)=O)C1 44782,c1(CC(=O)NC2C(NC(C3(COCC)CCC3)=O)CCC2)ccc(Br)nc1 44783,c1(C(=O)NCC(CCNC(CCCOCC)=O)O)c(F)cc(O)cc1F 44784,CC(C)(C(=O)N1CC2CCC(NC(c3nc(Cl)cs3)=O)(C2)C1)S(C)(=O)=O 44785,c1(C(N2CCC(CNC(c3occc3C3CC3)=O)C2)=O)ccc2c(c1)OCCC2 44786,C1(CNC(c2cc(C)n(CCO)n2)=O)CN(C(=O)Cn2[nH]cnc2=N)CC12CC2 44787,CCC(F)(CNC(=O)CC1CCCCN1C(=O)C(C)CCOC(C)=O)CC 44788,N1(C(Cc2ccc(C)s2)=O)CCC(C)C1CNC(C1CCCN1C1CC1)=O 44789,Cn1cnc(C=CC(=O)OCC(=O)NC2(c3ccccc3)CCC2)c1.C1CC1 44790,C1(CC(=O)N(C)CC2CN(C(C3OCCO3)=O)C2)CCN(C)C1=O 44791,n1(CC)nccc1C=CC(N1CC(CNC(=O)Cn2ccccc2=O)C(C)C1)=O 44792,C(=O)(C1=COCCO1)NC1C(C2CCN(C(C(CC)=CC)=O)CC2)OCC1 44793,C1(CNC(c2cc(-c3ccoc3)[nH]n2)=O)CN(C(C2C3CCC2CC3)=O)CCO1 44794,c1(CC)c(C(N2CC(N(C(=O)C(C)(C)COCC(F)F)C)C(F)C2)=O)csc1C 44795,Cc1nc(C(C)C)ccc1C(=O)NC(C)(CNC(C1CCC(O)CC1)=O)C1CC1 44796,Cc1[nH]nc2ncc(C(=O)NC3CN(C(C4CCNC4=O)=O)CC3N=[N+]=[N-])cc12 44797,C1(C)(C(=O)NCC(CCOC)NC(c2nccc(N)c2Cl)=O)CCC(F)(F)C1 44798,c1(N(C(C)CNC(c2ccc(N(C)CCO)nc2)=O)C)c(F)c(F)c(F)c(F)c1F 44799,c1(C(CNC(C2CC=CCO2)=O)NC(C(C)(C)N(C)C)=O)ccccc1F 44800,c1(C(N(C)CC2(O)CCN(C(=O)CCNC(N)=O)C2)=O)oc2ccccc2c1Cl 44801,C1(C(=O)OCc2onc(CSC)n2)Cc2ccccc2CN1N=O 44802,c1(C(=O)NCC(C(C)C)NC(=O)C=CC=C(Cl)Cl)cccc(N)c1N 44803,N1(C(c2cc(COC)no2)=O)CC(NC(=O)C(O)C2CCC2)CC12CCOCC2 44804,Cn1nnc2c1C(C(=O)NCC1(CNC(c3c(Cl)nn(C)c3Cl)=O)CC1)CCC2 44805,N1(C(COC(CNC(C2CC(=O)NC2)=O)(C)C)=O)CCN2C(=O)NCC2C1 44806,c1(C(N(CCNC(C(C(C)C)CN(C)C)=O)C)=O)cccc2ncnn12 44807,C12(C(=O)NC3CCC(C)NC3=O)C3C4C1C1C2C3C41c1ccccc1 44808,c1(C(N(CCNC(CC2N(CC)C(=O)CC2)=O)CC2CC2)=O)ccc(CC)c(F)c1 44809,n1(CC)ncc2c1CC(Nc1nccc(N(C)Cc3ccc(Br)s3)n1)CC2 44810,C1(OCCOC)CC(N(C2CC(C#N)C2)C(=O)C(=O)Nc2ccccn2)C1(C)C 44811,N1(C(C(CC(C)C)OC)=O)CCC(C)(C)C(CNC(=O)C=CC2CC2)C1 44812,c1(C(=O)NCC2C(C)(C)CN(C(=O)C=Cc3cccs3)C2)cc2scc(Cl)c2[nH]1 44813,CC1OC2(C(N3CC=C(CNC(c4ccnn4C4CC4)=O)CC3)=O)CCC1CC2 44814,C(CCC(c1nnnn1C1CCC1)NC(C1(OC)CCCC1)C)OCC 44815,c1(CC)noc(C(=O)NCC(C2CCC2)NC(C2CC3C=CC2C3)=O)c1C 44816,C1(C2CCN(C(=O)CN3C(=O)CCC3=O)C2)(NC(=O)Cc2nccs2)CC1 44817,C(=O)(C(CO)NC(C1CC(=C2CCC2)C1)=O)N(CCC)CCC 44818,C(CC(F)(F)F)N.c1(C(=O)NC)cn(CCC(C(C2(CCO)CC2)=O)=O)nn1.CN 44819,N1(C(c2ccc(C(=O)OC)[nH]2)=O)CCN(C(=O)Cc2cc(C)ns2)CC(C)(C)C1 44820,CC(CC1CCCO1)C(=O)NCC1CCCN1C(c1cc(C(F)F)cs1)=O 44821,C1(SC)COC2(CCN(Cc3ccc(C)nc3Cl)CC2)C1.c12cc-1cc(F)c2 44822,c1(C(=O)NC(C2(O)CCC2)C)coc2c1CN(C(c1[nH]ccc1C1CC1)=O)C2 44823,C(c1ccccc1)=C(CC)C(=O)N(CCNC(=O)CCCCn1ccnn1)CC 44824,C1(CC(=O)NC2CCCCC2)CC(O)CN1C(=O)CC1CCC1 44825,N=c1[nH]c2c(s1)CCCC2NC(c1cc(F)c(C(F)F)c(F)c1)=O 44826,Cc1occc1C(=O)NCCc1cc(C(=O)NCC(C)(C)C#N)no1 44827,C(=O)(C(CCSC)NC(c1cccnn1)=O)NCC(=O)NCC=C 44828,O=C(C1=C(Cl)CCC1)NC1CN(C(c2cn(CC3CCCO3)nn2)=O)C1 44829,C1(CNC(C2N(C)C(=O)OC2)=O)CCOCCN1C(c1cc(F)ccc1N)=O 44830,C1(C(=O)NOC(c2ccccc2Cl)C)(CF)CCC(=O)CC1.C(=O)OCC 44831,N1(C(Cn2ncc(CC)c2)=O)CC(C)CC1CNC(=O)C(CO)OC 44832,c1(C(=O)NC(CC(C)NC(Cc2cc(C)no2)=O)C)ccc2ncc(=O)[nH]c2c1 44833,c1(C(N(CC(CO)NC(C2CC3CC3C2)=O)CC)=O)ccc(OC2CCC2)cc1 44834,c1(CC(=O)NC2CC(CNC(C(C)=CC=CC)=O)C2(C)C)ccc(F)c(C)c1 44835,CCCCC(C(=O)NCCCC(CO)NC(C1CCN1C)=O)NC(N)=O 44836,C(CC(O)CNC(C1CC(NC(=O)C(F)(F)F)C1)=O)OC 44837,c1(CN=c2cc(C)n(C3CC3)[nH]2)ccc2c(c1)ncn2C 44838,C1(C)(C(N(CCn2cc(CCCS(N)(=O)=O)nn2)CC)=O)COCC(C)(C)O1 44839,N1(C(C(CC)=CC)=O)CCC(NC(c2sc(C)cc2C)=O)C(CO)C1 44840,C1(CC(C)(C)C)C(=O)N1.CC(C)(C)CCC(=O)NCC(C)(C)CF 44841,Cc1nc(CC(N2CCC(OCC(=O)NCc3ccnnc3)C2)=O)n[nH]1 44842,C1(C(N2CC(NC(C3(C=C)CC3)=O)(COC)C2)=O)CC2CCC1CC2 44843,C1(O)(Cc2c(OC)scc2)CCN(C(c2ccc(-c3ccccc3I)s2)C)CC1 44844,C1(C(=O)NCC(=O)N(C2CC3CC3C2)C)(CO)CCCO1 44845,C(C)(CCCC(=O)N(CC1CCC1)CC1CCC1)NC(c1c(CC)cc[nH]1)=O 44846,Cc1ccc(CC(=O)Sc2cccc(N3CCC(C(C)(C)C)C3)n2)c(C)c1 44847,c1(C(N(CCC(C)NC(C(C)OCCC=C)=O)C)=O)ccc(C(C)C)s1 44848,C1(C2CCN(C(=O)CC3CCSCC3)C2)(NC(c2cc(C)sn2)=O)CC1 44849,C1(N(C(c2ccc(CC)[nH]2)=O)C)CCCC2CN(C(C3(F)CCCCC3)=O)CC12 44850,CN1CCC(F)(F)C(CNC(C2CC(NC(=O)CC34CSCC3C4)C2)=O)C1 44851,C1(C(N2C3C(CNC(C(C)(C)OCC)=O)C(C3)C2)=O)CCC(C)=C(C)C1 44852,CC(CCNC(=O)CCCCNC(=O)C(C)n1cccn1)CCO 44853,C=CCC(C(=O)NC(C)CCNC(c1cc2ncccc2s1)=O)C(C)C 44854,C1(NC(CC(C)CF)=O)CCCC12CCN(C(c1cnn[nH]1)=O)CC2 44855,N1(C(C=CC(CC)C)=O)CCC(O)(C(C)NC(C23CCC(OC)(CC2)C3)=O)CC1 44856,c1(NC(C2CN(C(=O)CCc3nccs3)CCN2)=O)nc2c(s1)COCC2 44857,CC1CN(C(=O)CCC2(C)CC2)CCC1NC(C1CCC2(CCC2)C1)=O 44858,Cc1ccc(C(=O)NC2(CNC(c3nnc(-c4ccc(Cl)cc4)o3)=O)CC2)cn1 44859,C(=O)(C#CC1CCCCC1)N1CCC(NC(C(C)N(CC(F)(F)F)C)=O)C(O)C1 44860,Cc1cc(C(=O)NCC2(NC(=O)C(C)NC(C3CCC3)=O)CC2)cc(F)c1C 44861,CC(C)CC(C)(CNC(C1(C#N)CC1(C)C)=O)NC(c1n[nH]cc1Br)=O 44862,N1(C(=O)Cc2cccc(C3CC3)c2)CCN(C(C2CCN(C3CC3)C2)=O)CC(O)C1 44863,C(=O)(CCCCC(C)C)NC1C2(CNC(c3cncc(C)n3)=O)CCC(C1)C2 44864,N1(C(c2c(NC)cncc2)=O)CCCC(C2CC2NC(=O)C(O)CC2CC2)C1 44865,c1(C(N(CCN(C(c2c(OC)oc(C)n2)=O)C)C(C)C)=O)cc(=N)[nH]c(Cl)n1 44866,C1(C(CNC(=O)CSc2cnccn2)O)CCN(C(C2CCNC2=O)=O)CC1 44867,c1(C(N(CC(CCNC(=O)OC(C)(C)C)F)CCC#N)=O)cccc2nn[nH]c12 44868,c1(OC)ccc(CN2CCC2(C)C(=O)Nc2cccc(C)c2C#N)c(Cl)c1OC 44869,c1(C(=O)NC23CC(NC(C(c4cccc(C)c4)O)=O)(C2)C3)cc(F)c(N)cc1F 44870,c1(-c2c(C(=O)OCC)ccc3c2OCO3)cc(OC)cc2[nH]ccc12 44871,C1(NC(C2CCC(C)(C)O2)=O)CC2CCC1CC2NC(=O)Cc1ccc(Cl)s1 44872,c1(C(N2CCC(F)(CNC(C=C(C)C3CC3)=O)CC2)=O)ccc2oc(O)nc2c1 44873,C=C(C)C1OCCC1CNC(C1CN(C(c2cnc(C)cn2)=O)CC1OC)=O 44874,c1(C(N2CC(C)(NC(CC(C)OC)=O)C2)=O)cc(Cl)cc(Cl)c1F 44875,C(C(C)(C(=O)N1CC(CC(=O)NCC(C)(C)C(C)O)C(O)C1)OC)OC 44876,c1(OC)ncnc(OC)c1CN1CC2CC2(C(=O)NCCc2cccc(C)c2)C1 44877,C1(NC(c2c(C)cccc2F)=O)CC1C1CCN(C(=O)Cc2csc(Cl)c2)CC1 44878,N1(C(C2C(C=C)C2)=O)CCOC(C)(CNC(c2ccc(NC(C)=O)c(F)c2)=O)C1 44879,C1(C(C)C)N(C(=O)N(C(c2ncc[nH]2)C2CC2)Cc2ccc(Br)cc2)CC12CCC2 44880,C(c1cn(C)c2ccccc12)=CC(=O)NC1C(C)CN(C(c2cnn[nH]2)=O)CC1 44881,C1(N(C(=O)Cc2cnoc2)CC)CCCN(C(=O)CC2CC(F)(F)C2)CC1 44882,N1(C(c2nc(Br)cs2)C(=O)NCCCSC)CCC(CCO)CC1 44883,C(=O)(CCCCC(N)=O)N1CCN(C(CCCCC2C(C)C2)=O)C(C)C1.CC(=O)N 44884,C1(S(C)(=O)=O)(C(N(CC(C)NC(=O)CS(N)(=O)=O)C)=O)CCCCC1 44885,O=C1OC2CCCC2C1C(=O)Nc1cc(-n2cnnn2)cc(Br)c1 44886,n1(CCC(=O)NCCOc2ccccc2)cc(CO)nn1.c1(C(CN)(F)F)ccccn1 44887,CCCCC(O)C(=O)NCCC(CC)(CC)NC(=O)CCc1scnc1C 44888,C1(CNC(CCC2CCN(C(C(C(=O)OCC)F)=O)CC2)=O)OC(=O)NC1(C)C 44889,CC(C)CCC=CC(=O)NC(C)C(=O)NCC(F)C1CCC1 44890,N1(C(C(C)OCC(F)(F)F)=O)CCC(N(CCO)C(c2cncc(N)c2)=O)CC1 44891,N1(C(C(C)O)=O)C2CCC1CN(C(=O)CCCCC(N)=O)C2 44892,N1(CCc2ccc(-c3cnccc3)cc2)CCC2(CC1)COC2 44893,Cc1cccc(Cl)c1OCC(=O)NC1CN(C(C2CC(C)(F)C2)=O)CC12CC2 44894,n1(NCc2ccsc2)cc(Cc2cc(Cl)cs2)nn1 44895,Cc1cc(F)ncc1C(N1CCN(C(=O)CCCCCF)CC1C)=O 44896,N1(C(c2c(C)snn2)=O)CC(C)N(C(=O)CSc2ccncc2)CC1C 44897,NS(=O)(=O)c1ccc(C(=O)NCCC2CSCCN2C(C2CNC(=O)C2)=O)s1 44898,c1(CNc2c(C(=O)NC(C(=O)OC(C)(C)C)CO)nccc2)cc(Cl)c(O)cc1F 44899,N(C(=S)N1CC(C)C(C)(C(=O)OC)C1)(CCOC)C1CC1 44900,CC1(C(N2CC(NC(=O)C(C)(O)C(F)(F)F)C2)=O)CCC(F)(F)CC1 44901,CC1(C)CCC(CC(=O)O)N(C(=O)CC(C(F)(F)F)c2ccc(Cl)cc2Cl)C1 44902,C1(NC(CC2(C=C)CC2)=O)CCC(C)N(C(C2(c3ccc(C(N)=O)cc3)CC2)=O)C1 44903,N1(CCC(C)C)CCCC1C1CCCCN1C(c1cccc2ncsc12)=O 44904,C(CC1CC1)(C(=O)NCCC1CCC(NC(C2(CC(C)C)CC2)=O)C1)OC 44905,c1(N2CCC(CC=C)(NC(c3cc(C4(C)CC4)n[nH]3)=O)C2)ncnc(Cl)c1CC 44906,C1(CNC(c2n(C)c(S)nc2)=O)CC2(CCN(C(C3CCC(F)CC3)=O)C2)CO1 44907,N1(C(CCN(CC(C)(C)C)C2CC2)=O)CC(CO)C2(CCNCC2)C1 44908,c1(NC(C2CCC2F)=O)cc(C(=O)O)c(Cl)cc1F 44909,C1(NC(C2C(C(=O)OC)C2)=O)CC2CC(Nc3ccnc(-c4ccccn4)n3)C1C2 44910,N1(C(c2c(C)cc(F)s2)=O)C2CCC1C(C(=O)Nc1nnc(O)cc1O)C2 44911,c1(C(=O)NC2CN(C(c3n(CC)nnc3)=O)C(CO)C2)ccc2nncn2c1 44912,C(=O)(C1=CS(=O)CCC1)N1CC=CC(NC(CCc2cn(C)nn2)=O)C1 44913,Cc1nn(C)c(N2CCCCC2)c1C(=O)NC1CCCN(c2ccccc2F)C1 44914,N1(n2c(N3CCC(c4nnc(C)s4)C3)nnn2)CC2(CCC2)C1c1ccncc1 44915,C1(CN(C(=O)CCc2cccc(O)n2)C)CN(C(=O)CC2CCC2)CC12CC2 44916,c1(CC(N2CCN(C(CS(C)(=O)=O)=O)CC2CF)=O)ccc(S(C)(=O)=O)cc1 44917,N1(C(CC2(NC(C)=O)CC2)=O)CCC2(CCCN2C(=O)CC2CCCC2C)C1 44918,c1(N2CC(C)(CNC(CCC=C)=O)OCC2)cc(C)c([N+](=O)[O-])cc1F 44919,C(CC(=O)NCCC1=CCOCC1)(C(C)C)NC(C(C)OCC(C)C)=O 44920,c1(C(=O)NCC2(CNC(C3CC34CCC4)=O)CC2)c(Cl)cccc1Br 44921,CCCC(C)CCCC(=O)NC1CCC(C)N(C(=O)C=Cc2ncc[nH]2)C1 44922,C(=O)(C#CC1CCCOC1)NCC1(O)CCN(C(c2ccc(C)n2C)=O)C1 44923,C1(c2ccc(C(=O)Nc3nccc4c(Br)c[nH]c34)o2)CC2(CO1)CC1(C2)OCCO1 44924,N1(C(c2cnoc2C)C(=O)NCCCC2(C)CC2)CC2CCC(C1)O2 44925,N1(C(C2(c3ncccc3F)CCC2)=O)CCCC2(CN(C(CCC)=O)CC)CC12 44926,S1(=O)(=O)c2cccc(c2)CC2CCN1CC2.N1(C(CSC)=O)CC(O)CC1CO 44927,C1(NC(c2cc(CCCCC)no2)=O)CCC(NC(C2CC3(CC3)CO2)=O)CC1 44928,N1(C(c2ccc(C#N)[nH]2)=O)CCC2(CCCN2C(=O)C(F)C(F)(F)F)C1 44929,CC1CN(C(c2cc(C#N)cs2)=O)CC1NC(c1cc(C#N)cs1)=O 44930,c1(CC(=O)NCC2(F)CC(NC(C3CC(F)C(=O)N3)=O)C2)ccc2sccc2c1 44931,c1(CC)nc(C(=O)NCCCCN(C(=O)CN2CCSCC2)C)cs1 44932,C1(c2cn(C(N3CCS(=O)(=O)CC3c3ccccc3)=O)nn2)CC2(CNC(=O)O2)C1 44933,S(=O)(=O)(CCC(F)(F)F)N1CC(CC)C(Nc2ncc(C#N)cc2Br)CC1 44934,N1(C(c2ncc(C)cn2)=O)CCN(C(c2nccc(Cl)c2C)=O)CC1C1CC1 44935,C1(CNC(=O)C2=C(Cl)CC2)C2CCCC1N(C(c1ccc(Cl)s1)=O)C2 44936,N1(C(c2[nH]cc(C#N)c2)=O)CC2(CCC2)CC1CNC(C1(NC=O)CC1)=O 44937,N1(C(CSc2c(C)n[nH]c2C)=O)CC2(CCC2)CC1CNC(C1(F)CCOC1)=O 44938,N1(Cc2c(OC)ccc(Br)n2)C2CCCC1CN(C(=O)NC(C)(C)C)CC2 44939,C(C(=O)N1CCCCC1CCC(N1CC(C)(COC)C1)=O)(C(C)C)SC 44940,C(C(CC)(CC)C(=O)NC(c1ccccc1)C)NC(C(CC=CC)C)=O 44941,c1(OCC)ccc([N+](=O)[O-])c(-c2ncccc2C(=O)Nc2ncccc2CC)c1 44942,N1(C(Cc2cnc(C)[nH]2)=O)CCCC2CN(C(=O)C(C)CS(C)(=O)=O)CCC12 44943,C(C(=O)N1CC(=O)NC(=O)C1)(C(C)(C)C)NC(C1C(OC(C)=O)C1)=O 44944,C(=O)(CCC(C)(C)NC(=O)CC1CCC(=O)C1)N(C)CCF 44945,c1(CC(=O)N(C2CCN(C(C3CCCN3S(C)(=O)=O)=O)C2)C)ncc(F)cc1F 44946,C(CC(C)C(=O)NCCSCC(=O)NCc1ncccc1Cl)=CC 44947,C1(CC)(NC(=O)C(Cn2cncn2)NC(=O)Cn2nnc(C)n2)CCCC1 44948,c1(OCCOC)ncc(NCC(O)CNC(=O)NC2CCCCNC2=O)cc1Cl 44949,C#Cc1cncc(CNC(=O)CC2(CNC(=O)C3=CCCC3C)CC2)c1 44950,C1(c2onc(-c3cccc(C)c3)n2)COCCN(CC(=O)NC2CCCC(C)C2)C1 44951,CC1(C)CC(CCNC(C2CCN(C(=O)CS(C)(=O)=O)CC2)=O)CO1 44952,CCCC(CCCNC(c1ccc(N(C)C(C)=O)cc1)=O)NC(=O)C(CC)C(C)C 44953,CCP1(=O)CCN(C(C)C(N2CCC(OCC(N)=O)C2)=O)CC1 44954,c1(C2CCN(C(=O)OCn3cnc(-c4ccccc4)n3)C2)cccc(Cl)c1 44955,N1(C(CC(=O)NCC)=O)CC2CN(C(=O)CC(C)C(C)C)CC2(C)C1 44956,C1(NC(c2c(C)nc(CC3CC3)o2)=O)CC(C)CN(C(C2(C)CCCS2)=O)C1 44957,C1(C(N2CC(C=C)C(NC(=O)C3=COCCC3)C2)=O)CC12CCCCCC2 44958,C1(NC(=O)Nc2c(Cl)ccc(C)c2)CCC(F)(CNC(=O)Nc2ccccc2)CC1 44959,c1(OC)ccnc(CNC(=O)NCC2CCOC2(C)C)c1 44960,C(=O)(C(C)C(O)C(C)CC)N1CC(C(=O)NCC(CC)N(C)C)C(C)(C)CC1 44961,N1(C(C(CCNC(=O)CC2OCCO2)OC)=O)CCOC(C)(C)C1C 44962,C1(NC(c2nc(C)oc2)=O)CCCCN(C(=O)COCC2CCCC2)CC1 44963,Cc1cc(F)cnc1C(=O)NCC1COCC1NC(c1[nH]ccc1C1CC1)=O 44964,N1(C(COC)=O)CCOC(CNC(=O)CNC(c2ccnc(N(C)C)c2)=O)C1 44965,C(C)(C(C)C(=O)C(CC(C)CC1CC1)=O)NC(c1cn(CC(C)C)nc1)=O 44966,CCCCCC(C)(C)CNC(=O)C(C(C)CC)N(C)C(C1COCCO1)=O 44967,C1(C(N2C(C)(CNC(C3N(C)CC4(CC4)C3)=O)CCC2)=O)CCC(C2CC2)CC1 44968,N1(C(CCC)=O)CC(=O)CC1C(=O)NCC(=O)N(C)O 44969,c1(C(CO)NC(C2C(CC(=O)OC)NCCC2)=O)ccc(F)c(Cl)c1 44970,CC1(CNC(=NCCCC2CCCCO2)NCc2cnco2)CCC(F)(F)CC1 44971,c1(C(N(CCNC(c2ccc(OC)s2)=O)C)=O)ccn2cccc2c1.C(CCOC)N 44972,C(=O)(C(C)(C)CN1CCCCC1)N1CC(NC2C(C#C)C2)C1 44973,c1(NC(C(=O)NC2CCN(CCCCCC)C2)=O)nn(C)c2c1CCC2 44974,c1(C(=O)NC2(CC=C)CN(C(=O)CC3CCC(C)O3)C2)cc(C)oc1COC 44975,N1(C(CC(CCC)(C)O)=O)CCC2C1CCCN2C(c1cn(C2COC2)nn1)=O 44976,c1(CN(C2CCCCCC2)CCNC(=O)C=C(C)c2ccco2)ccccc1Br 44977,CC(C(=O)NC1CCCCC1NC(=O)COc1cnn(C)c1)S(N)(=O)=O 44978,c1(C(N2C(C)CC(NC(C(C=C)(F)F)=O)C2)=O)cnc2scc(C)n2c1=O 44979,C(CN=[N+]=[N-])(C(=O)NCCCOC1CC1)NC(CCC(N)=O)=O 44980,c1(C(=O)NC(C)CNC(=O)C(c2ccc(C#N)cc2)O)cnn2cccc(Cl)c12 44981,C(CC(=O)CCO)n1cc(C(CCC)NC(=O)C=CC2COCCO2)nn1 44982,c1(C(=O)NC(CC)CN(C)C(C2CCN2CCCO)=O)ccc(C(F)(F)F)cc1 44983,c1(C(=O)NCCN(C(C2C(C)(COC)C2)=O)C)ccc(Br)c(F)c1 44984,N1(C(c2cn(C)n(C)c2=O)=O)CC2CCC1CC2NC(C1(C)CCOC1)=O 44985,CC1(C)CCCC1C1CCN(C(=O)C(N2CCOC3CC(C(=O)O)CC23)=O)C1 44986,CC(C(=O)NC(CNC(c1c(F)cncc1Cl)=O)C1CCC1)C(F)(F)C(F)F 44987,CCCCCCCCCCNC(C1CC1NC(=O)C=Cc1cccc(O)c1)=O 44988,CCCCC(CN=c1[nH]cncc1C#N)NC(=O)Cc1noc2ccccc12 44989,C1(NC(c2scc(OC)c2)=O)CN(C(C2CCOC2=O)=O)CC(F)(F)C1 44990,c1(C(N(C2(C)CCN(C(C=C(CCC)C)=O)C2)CC)=O)ccc(N)c(C)c1Cl 44991,CCCCC(O)CNC(=O)COC(C1CCCC1)(C)C 44992,c1(C(N2CCN(C(=O)Cn3cncn3)C(C(F)F)C2)=O)cncc2ncccc12 44993,C1(C(N2CC(C(C)O)OCC2)=O)C2CCN(C(C34CC3CNC4=O)=O)CC12 44994,N(C(=NCc1cnc(C)cn1)NCC1CCOC1)Cc1c(COC)cco1 44995,CN1CCN(S(=O)(=O)c2ccc(NCC3(c4cccc(Cl)c4)CC3)nc2)CC1(C)C 44996,c1(C(=O)NCCCOC(C=C)=O)cc(-c2cc(OC)c(C)cc2C)c2cc[nH]c2c1 44997,C1(NC(c2cccc(OCCOC)c2)=O)C(C)CN(C(C2CC2F)=O)CC1C 44998,c1(C(N2C(C(=O)NCCC(C)C)CC(F)C2)=O)ccc(Br)c(Cl)c1Cl 44999,Cn1cc(C(N)=O)cc1C(=O)NCC1CC(NC(=O)CC2COC(C)(C)C2)C1 45000,C1(NC(=O)CC23CCCN2CCC3)CN(C(=O)Cn2cncn2)CC1C1CC1 45001,N1(C(C(C)N(C(=O)Cc2cccc(C#N)c2)C2CC2)=O)CC2(CC(F)C2)C1 45002,C(=O)(CCC(C)(C)NC(C1CCC(O)C1)=O)NCC1CC(C)(O)C1 45003,N1(Cc2n(C(C)C)ncc2)CCC(F)(F)C(C(=O)Nc2ccc3nonc3c2)C1 45004,c1(NC)cc(C(N2CC(CCNC(c3cc(CO)on3)=O)C(C)C2)=O)ccc1F 45005,C1(O)(CNC(=O)CCCc2nccs2)CCCN(C(c2cocn2)=O)C1 45006,C#CCCC(O)C(=O)NC1(CCC)CCCN(C(=O)Cc2ccnc(O)c2)C1 45007,c1(CC)c(C(N2CCC(C)(CNC(=O)C(C)C3CC3)C2)=O)cnn1C(C)(C)C 45008,C(=O)(C(CC1(c2nc(O)n[nH]2)CC1)NC(C1(CNC(=O)CC)CC1)=O)OC 45009,CC1(C)CC(CC(=O)N(c2cccnc2)CCO)N(C(=O)Cc2cncnc2)C1 45010,c1(C(=O)NC2C(NC(C3C(C#N)CC3)=O)C2)ccc(C2CCCCC2)cc1 45011,c1(CC(=O)OC(C)C)ccc(N(CCCCNC(c2nc(=O)n(C)[nH]2)=O)C)nc1 45012,C(=O)(C(CNC(=O)CCCC1CCCC1)C(C)C)N(CC(C1CCC1)OC)C 45013,Cc1c(CC(N2CCC(CCCO)C2)=O)c(=O)oc2cc(N)ccc12 45014,Cc1cc(N2CCC3(NC(C4CC5(CC5)C4)=O)CCCC23)n2nc(C)cc2n1 45015,C=CC1CN(C(C23CCOC(C)(C2)C3)=O)CC1NC(c1csc(F)c1)=O 45016,CCC(CC(=O)NCC1CN(C(=O)CC(C)(F)F)CC1c1ccccc1)C(F)F 45017,c1(C(N2CC(C)(NC(C3C(C=C)CC3)=O)C2)=O)ccc(Br)c(Cl)c1 45018,C1(CNC(C2=CC(C)(C)C2)=O)CC2COCC2N1C(=O)COc1cccc(Cl)c1 45019,N1(C(C(=O)NCC(F)F)c2ccsc2)Cc2nccc(Cl)c2C1 45020,c1(CC(=O)NC(CCCNC(c2occ(C)c2)=O)C)c(C)n[nH]c1C 45021,c1(C(=O)NCC(C)NC(CCn2ncc(C)c2)=O)ccc(Cl)cn1 45022,c1(CC)ccc(C(=O)NCC(C)(C(C)C)NC(=O)CCc2cnc(O)[nH]2)cn1 45023,C1(C(N(C2CCN(C(=O)CCc3csc(=N)[nH]3)C2)CC)=O)CC(C)(C)CCO1 45024,C1(N(C)C(c2cocn2)=O)CCN(C(C2CCCC(O)C2)=O)CC1 45025,Cc1cc(-c2cn(CCNC(=O)CN3CCCC3C)nn2)ccc1F 45026,c1(CC(=O)N(C2CCCN(C(CCCC#C)=O)C2)CC)ccc(C)c(Cl)c1 45027,CC#CCC(C(=O)N1CCC1(C)CC)NC(c1cn[nH]c1)=O 45028,c1(C(=O)NC2CC(CNC(C(C)CC(N)=O)=O)OCC2)ccc2c(c1)CCC2 45029,C1(C)(CNC(C(C(C)C)NC(N)=O)=O)COCCN(C(=O)C2=CCCCO2)C1 45030,C1(C(=O)NC(CCSC)C(=O)NCC2CC23CC3(F)F)CC12CCCCC2 45031,c1(CC)cc(Br)ccc1C(N1CCCC(NC(c2oncc2C)=O)C1)=O 45032,CC(O)C(C)C(=O)N(CC(=O)NCC1CCCN1Cc1ccccc1)C 45033,c1(C(N(CCNC(C=CC)=O)Cc2cccc(C)c2)=O)nn2c(c1C)CCCC2 45034,Cc1cc(CC(N2CCC(c3nc(C(F)(F)F)cs3)CC2)=O)n(C)n1.C1C(=O)N1 45035,C1=C(F)C(=O)N(CCS)C2C1CCCC2.C(c1cccc(C(F)(F)F)c1)=C(C)C 45036,c12ncc(c(O)n1)C(=O)NC2C.N1(C(C2(CSC)CC2)=O)CC(=C)C1 45037,C=CC1CCCCN1C(C1CCCC1CNC(C1CC=C(C)CC1)=O)=O 45038,C(=O)(C(F)C(C)(C)O)NC1CC(N(C(c2c(NC(C)=O)c[nH]n2)=O)C)C1 45039,c1(NC(=O)NC2CC2c2ccc(Cl)cc2Cl)cc(O)c(Cl)cc1Br 45040,N1(CCN)CCS(=O)(=O)CC1.c1(C(=O)OCC)cc(C(=O)OCC)[nH]c1C 45041,c1(SC)ccc(C(=O)NCC(C2CCC2)NC(=O)COCCCF)cc1.C 45042,c1(NC(C2CSCCN2c2cc(OCCO)ncn2)=O)cc(CO)cc(C(F)(F)F)c1 45043,N1(C(C2N=C(C)SC2)=O)CCCOC(CNC(c2cc(C)n(C)c2C)=O)C1 45044,c1(C(=O)NCc2c(CN(C(CCCC)=O)C)cccc2)cc(C#N)c(N)cc1O 45045,C(=O)(C(C)CC(C)C)NC(c1cccc(C)c1)CNC(CSCC)=O 45046,c1(C(CNC(C(COC)C)=O)CC(=O)O)cc(F)cc(F)c1.C1(CC)C(=O)O1 45047,c1(C(=O)OC(C2CC(N(C(=O)CC#N)CC3CCOCC3)C2)C)nn[nH]c1Cl 45048,C#Cc1ccc(F)cc1C(=O)NC12CC(NC(c3cc4c(s3)CCSC4)=O)(C1)C2 45049,c1(C(=O)NCCN(C)C(C2(CS(C)(=O)=O)CC2)=O)cccc(CC2CC2)c1 45050,CC1CCC(C)C(C)C1NC(=O)N(C1CCCC(O)C1)CC(F)(F)F 45051,C1(CC=O)CCCCN1N1CCOCC1.CCC(C)C=CC(=O)OCC=O 45052,C(CC(C(=O)NCC1CCN(CCF)C1)NC(c1sccc1Cl)=O)N(C)C 45053,c1(C(N2CC(OCCNC(=O)C(F)CC3CCCC3)C2)=O)ccc2sncc2c1 45054,C12(C(N3CCC(CCCC)C3)=O)CCCC1CCN2C(=O)Cc1cncn1C 45055,c1(CCC(=O)N(CCCNC(C2CC3CCC23)=O)C)ccc2c(c1)NC(=O)CO2 45056,c1(C(N2CC(C)(C(=O)Nc3ccnc(F)c3)C2)=O)c(F)c(F)cc(F)c1F 45057,Cc1cc(C#N)ccc1NCc1csc(Cl)n1 45058,CC(C)(C(F)(F)F)OCC(=O)NCCOCCNC(C1(F)CC=CCC1)=O 45059,c1(C(N2CCC(NC(c3c(CC)non3)=O)(COC)CC2)=O)ccc(C)c(C)c1O 45060,N1(c2snc(CCC)n2)CC(CNC(C2CC23CCOC3)=O)OC2(CCC2)C1 45061,C1(C(=O)NC(CC(=O)NC)C)C2CN(C(c3ccc(C)s3)C(=O)O)CC12 45062,c1(C(C(=O)NCCC(C)NC(C2(C(F)F)CC2)=O)=O)cc(F)cc(Cl)c1 45063,C1(NC(C(C)SC)=O)CCCC1CNCCNc1nc(Cc2ccccc2)ns1 45064,Cc1noc(C(F)(F)F)c1C(=O)NCC(F)CNC(C1(C2CC2)CC1)=O 45065,c1(CCC(N2C(CNC(c3ccc(COC)[nH]3)=O)CC2)=O)ccc(SC)cc1 45066,c1(N2CC(CC)OCC2)cc(Br)ccc1S(=O)(=O)N(C(C)(C)COC)C 45067,C(=O)(C1COc2ccccc21)N1CC(CNC(c2cc(C)n(C)c2)=O)OCC1 45068,Cc1cc(C(=O)N(CCCCNC(=O)CCC(=O)c2ccncc2)C)c(C)s1 45069,N1(C(c2c(C)nn[nH]2)=O)CCN(C2CCCN(C(=O)C(C(C)C)N(C)C)C2)CC1 45070,C1(C(=O)NC(C#C)CCC)CC(=O)CN1C(=O)CC1CCC2CC12 45071,N1(C(C2C(COC)CC2)=O)CCC(NC(=O)CNc2noc(CCOC)n2)CC1 45072,n1(CC(=O)NC(c2c(CC)occ2)=O)ccc(=NC(=O)C2(C)CCOC2)nc1O 45073,N1(C(C2C(OC)CCCC2)=O)CCN(C(C2OCCCC2(C)C)=O)CC1CO 45074,C1(CC(=O)NCC2C=CCN2C(=O)C=CI)CC2(CCC2)C1 45075,c1(C(c2n(CC=C)nnn2)NCc2ccns2)ccc(C)cn1 45076,N1(C(C2C(CC)CN(C(=O)CCc3ccsc3)C2)=O)CCCC(N(C)C)CC1 45077,C1(C(=O)NCC(C)C(=O)NC2C=CC(C)(C)CC2)CCC(C)(O)CC1 45078,c1(CC)ccc(C(N2CC(C(=O)NCc3ccccc3CO)C2)=O)cc1 45079,CC(CS(C)(=O)=O)C(=O)NCCC(C)CCNC(=O)CCSCC(N)=O 45080,C(C(C)(C=O)OC)OC.C1=CCNC(=O)C1.C(C)(C)(CF)OC 45081,C(=O)(C1=C(Cl)CCOC1)NCC(C)(C)NC(C1(c2cccnc2Br)CC1)=O 45082,C(=O)(CS(=O)(=O)c1cccc2nsnc12)OCCCCCC#C 45083,c1(C(=O)NC2CCC2NC(C2(CC3CCC3)CC2)=O)cnc(Cl)o1 45084,c1(C(=O)OC)cc(Cl)c(OC)cc1C(F)F.c12noc(n1)CNC2 45085,C#CC(C(C)(C)C)NC(=O)C(C)(CSC)NC(C1SCC=C1C)=O 45086,c1(CC2(NS(=O)(=O)CC3CC3)CN(Cc3cn(C)nc3)C2)ccc(F)c(C(=O)O)c1 45087,c1(C(=O)NCC2(NC(C3(c4ccn(C)c4)CC3)=O)CC2)c(Cl)cncc1Br 45088,n1(CCCC)ncc(C(=O)NCC(O)CN(C)C(c2nnn(C)c2C)=O)c1CC 45089,N1(C(C)=O)CCCC1C(=O)NC(C)(C)CCNC(c1nsnc1O)=O 45090,C1(CNC(C(c2cnn(C)c2)C)=O)CCC(NC(=O)Cn2cncn2)CC1 45091,C(=O)(C1=CCCC1C)NC(CCOCC)C(=O)N1CC(NC(=O)CC)C1 45092,C1(C(N(C2CCC(NC(C(CC)=CCCC)=O)CC2)C)=O)CC(C)CC(C)(C)C1 45093,Cc1ncccc1C(N1CC=CC1CNC(C1C(F)(F)C12CC2)=O)=O 45094,c1(N(C)C)ccnc(CNC(C2(C)C=CCN2C(c2cnnn2C)=O)=O)c1 45095,c1(C(N(CCNC(c2ccc(C(C)(C)C)cc2)=O)CC)=O)cc(C)cc(C)c1 45096,c1(OC)cccc2c1OCCCC2NC(C1CCN(S(C)(=O)=O)C1)=O 45097,N1(C(=O)CCC2CCC2)CCC(C2CC2)C1C(N1CC(CO)C2(CCC2)C1)=O 45098,N1(C(CCCN(C(C)C)C)=O)CCCOC(CNC(C2CCNC2=O)=O)C1 45099,CC1(C(=O)NCC2CN(C(c3c[nH]c(=N)s3)=O)CC2C(F)(F)F)CCCNC1=O 45100,c1(CC(N2CCC(CCCCNC(C3=C(C)CC3)=O)CC2)=O)c(C)nn(C)c1C 45101,C1(C(N2C(C=C)CC2)=O)CC2CCC(C1)N2C(C1(F)CC1)=O 45102,C1(C(N2CCN(Cc3ccccn3)CC2)=O)CC(C)CC(C)C1.CO 45103,Cc1ccc(=O)n(CC(=O)N(CC(C)N(C(=O)C(F)(F)C(F)F)C)C)c1 45104,N#CC1CC(C(=O)NCC(O)CNC(C2(C(=O)NC=O)CC2)=O)C1 45105,C12(C(C3CC3)N)CC(CN(C(=O)C(n3ccnc3C)C)C1)C2.CCC(CC)C1CCC1 45106,CCCC(C)CC(=O)N1CCOC(CN(C(=O)CN(C2CC2)CC)C)C1 45107,N(C(=NCCC)NCC(C)C(C)C)Cc1cccc(COC)c1 45108,N1(C(C2CC(CC)(CC)C2)=O)CC(C(N2CCOCC(N(C)C)C2)=O)C(F)(F)C1 45109,N(C1CN(C(C2CC2F)=O)CCc2ccccc21)C(=O)Cc1cc(Cl)ccc1Cl 45110,C1(C(N2C(C)CC(CNC(c3cc(O)nn3C)=O)C2)=O)CCn2c(O)nnc2C1 45111,C12(CNC(c3c(CC)nc(=N)[nH]c3)=O)CCCC(CN1C(c1cnsc1)=O)C2 45112,c1(C(N2CCC(C)(C(N3CCCC(C#C)C3)=O)C2)=O)ccc(O)c(O)c1Cl 45113,c1(CC)onc(C)c1C(=O)Nc1cccc(C(=O)Nc2ccno2)c1.C(C=O)N 45114,c1(COC)nc(NCCC2CC2(Cl)Cl)cc(=NCCN2CCC2)[nH]1 45115,c1(C(=O)NCCCN(CCCNC(C2C(=C)C2)=O)C)ccc(C)c(S(N)(=O)=O)c1 45116,N1(C(CC(CC)SC)=O)CCC(C)(C)C(C(=O)N(C(C)CSC)C)C1 45117,c1(OC)ccccc1C(N1CC(N(C(=O)CCC(C)N(C)C)C)C(O)C1)=O 45118,Cc1[nH]c2c(C(N3CCC(CNC(=O)CC4CC4(Cl)Cl)C3)=O)cccc2c1C 45119,N1(C(C(C(C)(C)O)F)=O)CCC(C2(NC(c3cc(-c4ccoc4)[nH]n3)=O)CC2)C1 45120,c1(CN2C(C(=O)NCC(O)CO)CC(O)C2)cc(Br)ccc1F 45121,N1(c2c(OC)cnc(Cl)n2)CCCC(C2CC2NC(c2nccc(Cl)c2F)=O)C1 45122,c1(-c2cn(Cc3cn(C4CC(OC)C4)nc3)nn2)cc(C)cc(C)c1 45123,C1(O)(CN(C(CNS(CC)(=O)=O)=O)C)CCN(C(C2(C(N)=O)CCC2)=O)CC1 45124,N1(C(c2c(C)nc(C3CC3)s2)=O)CCN(C(c2cocn2)=O)C(C(C)C)C1 45125,Cc1cc(N2CC(C)(C)CC2CNC(c2csnc2Cl)=O)nc(C)n1 45126,c1(C(=O)NC2(C3CC3)CCN(C(C(CC)(C)C#N)=O)C2)cnc2ccncc2c1 45127,C(=O)(C(=O)C(C)(C)CC)NC(C(=O)N(C(C=C)C)C)C(C)C 45128,c1(C(=O)NC(C(C)NC(C2CC(=C)C2)=O)(C)C)cc(Cl)cc(F)c1N 45129,c1(C(=O)NCCN(CCC)C(C2CCCSC2C)=O)occ2c1CCC2 45130,C1(CCNC(CC2C(CNC(Cc3n(C)ccc3)=O)C2)=O)CCCC2CC12 45131,c1(C(N2C(C(=O)Nc3n(CC)c(O)nc3)CC3CC32)=O)cnc2c[nH]nc2c1 45132,C#CC1(NC(=O)CC2(NC(=O)C(C)CCCC)CCCCC2)CCCCC1 45133,N1(C(C=C(C)C(C)(C)C)=O)CC(C)N(C(=O)Cc2c(C)nc(C)nc2O)CC1C 45134,N1(C(CCCOCC)=O)CC(C)(CNC(=O)CC(C)c2ccccc2)CC1(C)C 45135,CC(C)CCC(F)C(=O)NCC(C)(CO)NC(C1CCC(C(N)=O)O1)=O 45136,c1(C(=O)NCC(CN(C)C(C2CCCC2)=O)O)ccc2cnnc(O)c2c1 45137,C(C1CCOCC1)=CC(=O)N(CC(C(=O)NCC1(COC)CCCO1)C)C 45138,c1(C(N2C(CN(C(CC=CC=C)=O)C)CC(F)C2)=O)cccc(OCCC)c1C 45139,c1(C(=O)NC(C)(CNC(=O)C(O)CN2CCCC2)CO)csc2nnsc12 45140,N1(C(CCCC=C)=O)CC(C)(C)CC1C(=O)N(CCc1nccn1C)CC 45141,N1(C(CCOC)C2CC2)CC(c2nnc(CNc3cc(C)ns3)o2)CC1(C)C 45142,c1(C(=O)NC(C)C(=O)NC(c2ccnn2C2CCC2)=O)oc2ccccc2c1Cl 45143,C1(F)(NC(C#CC(OCC)OCC)=O)CCCN(C(C2CCC=CCCC2)=O)C1 45144,C(CC(C(=O)NCCc1nncn1CC)NC(c1cnco1)=O)=CC 45145,C(=O)(CC(F)(F)C(F)F)NC1CCCC(C(=O)NC2CCC(OC)C2)CC1 45146,c1(OC)ccc(C(=O)NC2CCC2NC(C2CC2c2ccc(F)cc2)=O)c(F)n1 45147,Cc1ccc(F)c(C(=O)NC(C)CN(C(=O)C(C(C)C)n2ccnc2)C)c1 45148,C1(NC(C(C)OCC#C)=O)CN(C(=O)CCc2cccs2)CC2(CCC2)C1 45149,c1(C(=O)COCC=CC(=O)NC(CN)CO)ccnn1CCF.C(C)(C)(C)O 45150,CC1CC(CNC(=O)C(C(C)(C)C)NC(N)=O)CCN1C(=O)C(C)C1CC1 45151,C(N=c1nc(CNC(C2CC(=O)N2)=O)[nH]s1)C1(C2CCCC2)CC1 45152,c1(OC)ccc(F)c(C(=O)NCCCCCN(C(=O)CCc2nncs2)C(C)C)n1 45153,N1(C(C(CCSC)O)=O)CC=C(CC(=O)NC(C)CC(C)(C)OC)CC1 45154,CC1(C)CCC=C1C(=O)NC1CN(C(=O)CCC2CCCC(=O)N2)CC12CC2 45155,C(=O)(CC(CN(C)C)C(F)F)NC1CCN(C(CCc2cc(C)[nH]n2)=O)C12CC2 45156,N1(C(CC(C)(C)O)=O)CC2(C1)SCCC2NC(c1ccc(SC2CC2)cc1)=O 45157,C(=O)(C1=CC2(CCOC2)C1)N(CC(C)N(C)C(C1CN(C2CCCCC2)C1)=O)C 45158,C(=O)(C(C)CC(=O)OC)N(C1CCN(C(=O)CCN(C2CC2)CC)C1)CC#C 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45212,C1(C(F)F)(CNC(CN(C(COC)=O)C)=O)CCN(C(c2ccc(O)nc2)=O)C1 45213,C1(=O)C(C(C)(C)C)C(=O)NC(CC)C(=O)NC2(CCC2)CN1CC.C(N)(=O)OC 45214,c1(SCC)ccc(C(N2CC3CC2C3NC(=O)CSc2ccc(F)cc2)=O)cn1 45215,Cn1cc(C(=O)NCCC2CCN(C(=O)CCCC#N)C2)c(=O)c(Br)c1 45216,NS(=O)(=O)c1ccc(F)c(C(N2CC3CC2C3CNC(C2(C)CCCO2)=O)=O)c1 45217,CCC(C)CN=c1[nH]c2c(c(=NCc3nc4c(s3)CC(C)CC4)[nH]1)CCC2 45218,N1(C(C2CC3(CC3)CO2)=O)CCCN(C(=O)C(F)(F)CO)CCC1 45219,C(=O)(CC(Cc1ccccc1)CC)NCCC(=C)CNC(c1cnc(C)[nH]1)=O 45220,C(C(C)(CCO)NC(=O)C(C)C(C)NC(c1nnsc1N)=O)OC 45221,c1(C(CCC)NC(=O)NC(CCC(F)(F)C(F)(F)F)C(=O)O)ccc(F)c(F)c1 45222,N1(C(CC2CC(OC(C)(C)C)C2)=O)CC2CCC2(NC(=O)C(Cl)=CCl)C1 45223,N1(C(C2C(C(C)O)C2)=O)CCC(=CCNC(=O)CCc2ccccn2)CC1 45224,C1(C(N(C)CC(CC)C)=O)CN(C(C2(COC(C)=O)CCC2)=O)C1 45225,N1(C(CC(C)(C)C)=O)Cc2cccc(CNC(=O)CC3CCCCC(=O)N3)c2C1 45226,c1(C(=O)NC2CC(NC(C3C(C)CN(C)C3)=O)C2)cccc2c1ncn2C 45227,S(=O)(=O)(c1cccc(CCNC(=O)C(=O)NC2CCC2C2CC2)c1)NC(C)=O 45228,N1(C(CCC#C)=O)CCOC2(CCN(C(C34CCC(C3)C4(C)C)=O)C2)C1 45229,Cc1ccc2cc(C(N3CCC(CN(C(=O)Cc4cc(C)no4)C)C3)=O)cn2c1 45230,c1(C(N(CCCC(=O)NCC)C)=O)ncccc1NC(NC1=NCCS1)=O 45231,C1(C(C)C)CCC(n2cc(-c3cscc3C(N3CCC(C(=O)O)C3)=O)nn2)CC1 45232,N1(CCc2cc(OC(C)C)c(O)cc2)CCC12CCS(=O)(=O)CC2 45233,N1(CC(=O)NC2(CCNC(C(C)NS(C)(=O)=O)=O)CCC2)CCNC(=O)C1 45234,C(C)(N=c1ccnc(NCc2sc(=N)[nH]c2C)[nH]1)c1n(CC)ncn1 45235,Cn1ncc(C(N2CCC(O)(CNC(=O)CCn3cnnn3)C2)=O)cc1=O 45236,C1(OCC)CC2(C1)CC2C(=O)NCCNC(=O)C(C1CCC(=O)N1)C 45237,C1(C)(CC)CCCN(C(C2C3CC2N(C(C2CC(=C4CCC4)C2)=O)C3)=O)C1 45238,N1(C(C)=O)CC2OCCN(C(c3nc(-c4cccnc4)cs3)=O)C2C1 45239,CC1CCN(C(C(N2CC(NC(=O)CN3CCOCC3)C3CC23)=O)C(C)C)CC1 45240,C1(NC(c2n(CC)ccc2)=O)C2CC3C1C3C2C(=O)NCCCN1CCCCC1 45241,C(=O)(C1=C(Cl)CCC1)N1CC(CN(C(C(CC)(C)C)=O)C)OCC1 45242,c1(OC)cc(C)sc1C(=O)NC1CC(CCNC(C2CCC(C(N)=O)CC2)=O)C1 45243,c1(COC)cc(C(c2nnnn2CC2CC2)NC(c2ccccc2)CF)n(C)n1 45244,C1(C)(CC)C=C(C(=O)NCCCC(C)NC(=O)CN(S(C)(=O)=O)C)C1 45245,N1(CC(N2CCC(O)(COC)CC2)=O)C(=O)C(=O)N(C)C1=O 45246,Cn1nc2ccc(Br)cc2c1C1CCCN1Cc1cnc(C2CC2)s1 45247,c1(OC(C(=O)NC2C(NC(Cc3c(C)con3)=O)C2)C)ccc(F)c(F)c1 45248,CS(=O)(=O)c1ccsc1C(=O)NCC1(CNC(C2CCC(=O)N2C2CC2)=O)CC1 45249,N1(C(C#CC(C)C)=O)CC2(C1)CN(C(c1cccn3nnnc13)=O)CC2CO 45250,C(C(CC=C)C(=O)N1CC(N(C)C2CC2)C1)NC(Cn1ncc(C#C)c1)=O 45251,Cc1ccc(SC(C)(C)C2CC2)cc1.C12CCCN(C1)C(=O)c1cn2nn1 45252,c1(CC)conc1CC(=O)NC(C1CC(NC(c2cn(C)nn2)=O)C1)C 45253,C1(CC#C)(NC(=O)C(Cc2cnc[nH]2)NC(C2C3(CC3)C23CC3)=O)CCCCC1 45254,c1(C(=O)NC(C2CCCC2)CNC(=O)C(O)CC2CCOCC2)cc(Cl)ccn1 45255,N1(C(CCCCOCC)=O)CCC2C(CCCN2C(=O)CCC(C)(C)F)C1 45256,N1(CCNC(C(C)C)=O)C(=O)C(c2cc(Cl)cc(Cl)c2)N(C)C1=O 45257,c1(C(=O)NC(C)(C)CNC(=O)COC2CCCOC2)nncn1C1CC1 45258,C1(C(=O)NC(C(=O)NC)C(C)C)CCN(C(=O)CCc2ccoc2)O1 45259,N1(C(C(CC)NC(C)=O)=O)CCC(F)(F)C(NC(c2cc(Cl)ccc2Cl)=O)C1 45260,c1(C(N2C(C)C(NC(c3nscc3Br)=O)CC2)=O)cnc2c(cnn2C)c1 45261,C(=O)(N=c1ccn(CCCO)[nH]1)c1ccc(CCC(=O)NCCC2CC(O)C2)o1 45262,CCC(CC)CCCC(=O)N1CCCC(O)(CCNC(=O)C(C(C)C)OC)CC1 45263,C(=O)(CS(=O)(=O)CCO)N(CCCNC(c1cn(CC(N)=O)nn1)=O)C(C)C 45264,C1(C(N(CC(C)NC(c2ccoc2CC(=O)OC)=O)CC)=O)C2CCCC12 45265,N1(C(C=CC)=O)CCC(C2CC2)(CNC(=O)CC(C)P(C)(C)=O)C1 45266,C(CCCCC(=O)N1CCN(C(C2CCN(C)C2=O)=O)C(c2ncc[nH]2)C1)OC 45267,c1(C(N(CCCNC(C2CC(N(C)C)C2)=O)CC)=O)csc2c1CCC(C)C2 45268,C1(N(C(c2ccc(COC)o2)=O)CCO)CCCN(C(c2occc2C)=O)C1 45269,Cc1cc(-n2cncn2)ccc1C(=O)NC(C)CNC(c1sc(C)c(C)c1C)=O 45270,c1(CC(N2CC(N3CCN(C(C4C(C)OCC4)=O)CC3)C2)=O)ccc(F)c(F)c1 45271,c1(N(C)Cc2cn(CC)nc2)nc(N2C3CCC2COC3)nc2ncn(C)c12 45272,C1(C(=O)NC(CC=C)C(=O)NCC2(CC)CCC(=O)N2)CCC(O)CN1C 45273,c1(C(N2C(C(N(C)CCC3CCCC3)=O)CCC(O)C2)=O)ccc2[nH]ccc2c1 45274,C(=O)(C1CCCc2nncn21)N1C(C(C)NC(C(C)OCCC(C)C)=O)CCC1 45275,CCCC(C(=O)N1CC2CC2(NC(=O)C(CC)OC2CCCCC2)C1)C(C)C 45276,c1(C23CC(C(=O)NCC#CCN4CCOCC4)(C2)C3)nc2ccccc2s1 45277,c1(C(=O)NC2CC(CNC(c3coc(O)n3)=O)C2)csc2ccc(F)cc12 45278,C1(C(N(CC)CC)=O)C2CC1N(C(c1coc(C(F)F)c1)=O)C2 45279,C1(CC(=O)NCCN(C(Cc2n(C(C)C)cnn2)=O)C)CCCCN1C 45280,N1(CCN(C23CCC(C)(C2)OC3)C)CC2CCC(NC(C)=O)C2C1.CC=O 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45298,c1(CC)ccc(F)c(C(N2CCCC(C)(CNC(c3nnccc3C)=O)C2)=O)c1 45299,C1(NC(C2(CC)CC2(F)F)=O)CCN(C(=O)CC(=O)NCC(F)(F)F)CC(C)(C)C1 45300,c1(C(=O)NC2(CC=C)CCCN(C(=O)C3CC3)C2)ccc(S2(=O)=NCCC2)cc1 45301,CC1C(NC(=O)COc2cnn(C)c2)CCCN1C(=O)Cn1cncn1 45302,C1(C(=O)Nc2ccccc2-n2cc(C3CC3)nn2)CCc2ccccc2C1 45303,N1(C(CCC(c2ccc(CC)cc2)=O)=O)CCS(=O)C(C)C1C 45304,N1(CCNC(C(COC(C)C)N(C)C)=O)CCC(NC(=O)C=CCF)CC1 45305,N1(C(C=C(C)C)=O)CCCC(C2CC2NC(c2cn3ncccc3n2)=O)C1 45306,C(=O)(C1=CCCCC1P(C)(C)=O)NCCCCN(C)C(C1Cc2nccn2C1)=O 45307,c1(OC(C)(C)C(=O)NCCNC(=O)CCCOCc2ncc[nH]2)cccc(F)c1 45308,C1(N(C(CC(=O)NCC)=O)C)CN(C(=O)CCCC2CCCO2)CC12CC2 45309,c1(-c2cc(N3CCN(OC(C)C)CC3)ncc2)ccc2[nH]nc(CC3CC3)c2c1 45310,C1(NC(c2cnc(C)s2)=O)CC(C)N(c2ccnc(CO)n2)C1 45311,C1(CNC(C2CN(Cc3ccccc3)C2)=O)CCCN1C(=O)CC1CCCC1 45312,Cc1cc(C(=O)N(CC(C)NC(=O)Cc2cc[nH]c(=N)c2)C)c(C)cn1 45313,C1(C)(COC)CN(C(c2ccc(F)c(C)c2)C(=O)NCC(F)F)CCO1 45314,CC(CN(C)C)C(=O)N(CCCCNC(C1(C2CCCO2)CC1)=O)C 45315,N(C(=NCC1CC1(F)F)NCc1nc(C(F)(F)F)co1)Cc1ccccc1 45316,C1(CC)CN(C(=O)Cn2cc(C)cn2)CCC1CNC(=O)CNC=O 45317,CC1C(NC(=O)C=Cc2cn(C)nn2)CCN1C(=O)CC1OCCO1 45318,Cc1ccc(C(=O)NCC2CN(C(=O)C(O)CC(C)C)CC(C)(C)C2)c(F)c1F 45319,c1(NCCC(C)OC)nc(N2CCC(C(C)CO)CC2)nc2c1ncn2C(C)C 45320,C1(NC(=O)CC2NC(=O)NC2=O)CC12CCN(C(=O)C1=CCOCC1)C2 45321,C=Cc1cncc(C(=O)N(CC)CC2CCCCN2C(=O)CCC(N)=O)c1 45322,C(=O)(C(C(=O)OC)OC)N1C(C(C(=O)N(CCCC)CC)(C)C)CCC1 45323,C1(CC(=O)OCC)CCCN(C(=O)C(C)(C(=O)C=C(C)C(C)(C)C)C2(C)CC2)CC1 45324,c1(CNC(C2CC(NC(C3(COC)CCC3)=O)C2)=O)cc(-c2ccncc2)on1 45325,C=C(C)C1CN(C(=O)CC2CCCN(C(=O)Cc3cnns3)CC2)CCO1 45326,c1(NC(C2(CNC(C3CCC(=C)CC3)=O)CC2)=O)cc(Br)ncc1[N+](=O)[O-] 45327,N1(C(CC(C)CF)=O)CCN(C(c2cccn2Cc2cccs2)=O)C(C)C1 45328,CCC(O)(CC(=O)NC1CCC1CNC(=O)C=CCO)c1ccccc1 45329,C1(CC(=O)NC(=O)NCCOCCNC(c2ccc[nH]2)=O)CC(O)C12CCC2 45330,c1(-c2cn(C(C)C(=O)NC(C)CS(C)(=O)=O)nn2)cnn2c1NCC2 45331,C#CC1(C(N2CC(CNC(c3cocn3)=O)C2)=O)CCCC1 45332,C(CC(C)C)(C(=O)NCCC1(OC)CN(C(=O)C(C)NC(=O)OC)C1)OC 45333,c1(C(=O)NC2CC(CNC(CCOC(C)=O)=O)C2)ccn2nnnc2c1 45334,CN1CCC2CCCN(C(C3(N4CCOCC4)CCCC3)=O)C2C1 45335,C1(C(=O)NCC(CNC(C2=CC(C)(CC)C2)=O)(C)C)CC2CCC(C1)C2O 45336,CC1CN(C(=O)CC(C)c2ccccc2)CC1NC(=O)CC(F)(F)Cl 45337,c1(CCC(N2CC3CC3(CNC(C3C=CCCC3)=O)C2)=O)cccc(F)c1Cl 45338,O=C(C1=C(Cl)CCOC1)NCC1(NC(C23CSCC2C3)=O)CCOCC1 45339,N1(C(c2c(C)oc(C)c2C)=O)CCN(C(=O)Cc2csc3nccn23)C(C)C1C 45340,C(=O)(C1=CCC(F)(F)CC1)N1CC(CCNC(c2c(CC)cno2)=O)OC(C)C1 45341,CP(C)(=O)CCC(=O)NCC#CC(=O)N1CCC1C(=O)N(C)C 45342,C1(CC(=O)NCc2cccc(C)c2Cl)C2CCC1CN(Cc1ncc[nH]1)C2 45343,C1(OC)CN(C(c2conc2C(C)(C)C)=O)CC1NC(=O)C=CSc1nc[nH]n1 45344,c1(C(=O)NC(CC)CNC(=O)C(F)n2cccn2)cncnc1 45345,N#CC1(C(=O)NCc2csc(C(=O)NC(CC3CCC3)CO)c2)CCCC1 45346,C1(F)(CNC(=O)CCCN2CCCCC2)CCN(C(C2CCC(=O)N2)=O)CC1 45347,C#CCC(C)(CC)C(=O)N(CC(=O)Nc1nccn1CC)CC(C)C 45348,C1(CCNC(C(F)=CCC)=O)CN(C(=O)CCN2C(=O)CCC2=O)CC(C)O1 45349,c1(OC(C)(C)C)ccc(Cl)c(NC(=O)Cn2nc(C(F)(F)F)cc2C2CC2)c1 45350,N1(CCc2nc(C)sc2)CCCC(NC(=O)N(C)CC2COCCO2)C1 45351,N1(C(CP(C)(C)=O)=O)CCN(C(=O)CCCn2cncn2)CC1CC(F)F 45352,C(C)(CCC(=O)N1CCCC(C(C)NC(=O)NCCOC)C1)NC 45353,c1(C(=O)NCCCC(C)NC(=O)CNC=O)cnccc1C(F)(F)F 45354,c1(CNC(C(C2CC(F)(F)C2)OCC)=O)n[nH]c2c1CN(C(=O)C1=CCOC1)CC2 45355,N1(C(c2cc(OC)ns2)=O)CCC2(CCCN(C(=O)C=CC(=O)N(C)C)C2)C1 45356,c1(C(=O)NCC2(OC)CN(C(C3CC34CCOC4)=O)C2)ccc2c(c1)NCC2 45357,Cc1ccc2oc(C(N3CC(NC(c4cn(C)c(=O)n4C)=O)C(F)C3)=O)cc2n1 45358,C12(CNC(c3c(C)sc(O)n3)=O)CCC(CNC(=O)C(C)C3CCC3)(CC1)OC2 45359,Cc1cc(OCC(N2CCN(C(C3SCCS3)=O)CC2CO)=O)ccc1F 45360,CC(CCNC(C1(CCNC(=O)CCC2CCC(=O)C2)CCCC1)=O)C(C)(C)C 45361,Cc1cccc(Cl)c1S(=O)(=O)NC1CN(C(C2CCCC2C)=O)CC1O 45362,C1(C(=O)NC(CNC(C(C)SCC)=O)CC(C)C)COC2COCC12 45363,C1(C(=O)NC2CCN(C(C(C=CC)O)=O)C2CC)CCc2nnc(O)n2C1 45364,C1(C(=O)NC2CC(NC(C(CCC)NC(C)=O)=O)C2)CC2CCCC(C1)C2 45365,n1(CC)nc(C)cc1C(=O)NCC(O)CCNC(C1COC1)=O 45366,N1(C(C2CC(C(=O)OC)C2)=O)CC(NC(=O)C(C)(C)Oc2cccc(Cl)c2)C2CC12 45367,C1(C(N2CCOC(CC3CC3)C2)=O)CCOCCN1C(=O)CC1CC=CCC1 45368,C1(n2c(CSCC)nc(CCc3ccccc3)n2)CCC(F)(F)CC1 45369,N1(C(CC(CC)C)=O)CC(NC(C2CC3CCC2CC3)=O)CC(C)(C)C1 45370,c1(-c2scc(C(=O)NCCCCC#C)n2)cnn2c1CCCC2 45371,c1(C(N2CC(CC)(CO)C2)=O)n[nH]c2c1CN(C(C1C3CCCCC13)=O)C2 45372,CCC(C(=O)NCC1(F)CCC(CNC(c2csnc2C)=O)CC1)C(C)(F)F 45373,C12(C(N3CCC(N(CC#C)C(C4CCC(C)O4)=O)CC3)=O)CCC(N=[N+]=[N-])C1C2 45374,CCCCCC(O)C(=O)N1CC(O)(C(C)NC(=O)CN2C(=O)CNC2=O)C1 45375,CS(=O)(=O)c1ccsc1C(=O)NC1C2CC1N(C(C1(C#N)CC13CCC3)=O)C2 45376,C(=O)(C(O)C(C)(C)C)NCCn1cc(C(=O)NC(C#C)C2CC2)nn1 45377,C1(CN(C(=O)CN2CCOCC2=O)C)CCCN(C(C2CCCS2(=O)=O)=O)C1 45378,c1(CN(CCCNC(C23CCC(CC2)CC3)=O)CC)cc(Cl)ccc1Cl 45379,C(=O)(C1=COCCO1)N1CCC(CCCCCNC(C2CCCS2)=O)CC1 45380,c1(N(C=O)C(CC(C)C(=O)OC(C)(C)C)=O)cc(C2CC2)oc1C1CC1 45381,Cc1ccc(C)n1CC(=O)N(CCCN(C)C(c1c[nH]c(Br)c1)=O)C 45382,C1(CNC(C(C)Oc2ccc(F)cc2)=O)CCc2ncccc2C1.C1(=O)CN1 45383,C1(CN(C)Cc2nn(C)cc2Cl)CCc2cc(F)ccc2O1 45384,CCCC(C(=O)N1CCCC1(C)c1cn(CCCc2cnco2)nn1)OC 45385,N1(C(COCCC(C)C)=O)CC(NC(=O)C(c2cnn(C)c2)O)C(C2CC2)C1 45386,CC(C)(C)C(C)(C)C(=O)NC1CCCN(C(c2ccc(C(F)(F)F)[nH]2)=O)C1 45387,C1(C(=O)NCC(C2CC2)NC(c2c(CC)nc(C)nc2)=O)CC2CCCC(C1)C2 45388,c1(NCC2(Cc3ccccc3I)CC(OC)C2)nccc(OC)c1OC(C)C 45389,c1(CC)cncc(C(N2CC(CNC(=O)C(CC)NC(C)=O)C(C)C2)=O)n1 45390,C1(C(N2CC3(C(NC(c4c(C)ccs4)=O)CCC3)C2)=O)Cc2ccccc2CO1 45391,Cc1ccc(C=CC(N2CC=CC(C(=O)NCCCC3CCOC3C)C2)=O)cc1 45392,C(C1COC(C)(C)O1)=CC(=O)NC1CC(C)(NC(C(C=C=C)C)=O)C1 45393,c1(COC)cnc(NC(=O)CC2CCCN(Cc3csc(C)n3)C2)nc1C(=O)OC 45394,CCCC(CCC)=CC(=O)NC1CN(C(=O)Cc2ncccc2C)C2CC12 45395,Cc1ccccc1CSCC1CCCCN1C(=O)CC(C(F)F)c1ccccc1 45396,c1(C(=O)NCC2(CCC)CCN(C(C3CCN(C)C3)=O)C2)c[nH]nc1[N+](=O)[O-] 45397,N1(C(C(C)(C)SC)=O)CCC(NC(c2ccc(-n3ccc(C)n3)cc2)=O)C(C)C1 45398,c1(CC(N2CC(n3cc(CSC)nn3)(C(=O)NC)C2)=O)ccc(O)c(F)c1 45399,Cc1ccc2nc(C(N3CCC3CNC(=O)C(C)OCC(F)(F)F)=O)c(N)n2c1 45400,c1(OC(CC)C(=O)NCC2CC2NC(=O)CCc2cc[nH]n2)ccccc1C(N)=O 45401,C=C(C)CC(C(=O)NC(c1cncs1)C)NC(C1CC2CC(=O)C1O2)=O 45402,C(N=c1[nH]c(=NCC(C)(F)C(C)(C)F)c2ncccc2[nH]1)c1cc(C(C)C)sc1 45403,C12(C(=O)NCCC(O)C(F)F)CCC(CC1)N(C(C1(CO)CCCCC1)=O)C2 45404,C(C(C(=O)NCCSCCCO)NC(=O)CN(C)C1CC1)SC 45405,c1(CC(=O)NC2C3CN(C(c4c(C)cc[nH]4)=O)C2C3)ccc2c(c1)CC(C)O2 45406,C1(CNC(CCC(=O)NCCC)=O)CCC2(CC2)N1C(=O)CCC1(C)N=N1 45407,c1(C(=O)NC(CC=C)CNC(=O)C(c2ccc(F)cc2)O)c[nH]c2nccc-2c1 45408,c1(OCCOC)cnc(C(=O)NC(C)CNC(=O)Cc2scnc2C)cn1 45409,C(=O)(C1=CCN(C(c2cnc(C(C)C)o2)=O)CC1)N(C(CC(CC)C)C)C 45410,CCCC(CCCNC(C1(CC)CC1)=O)NC(c1cc(-c2ccco2)no1)=O 45411,c1(OCC(=O)N(CCCCN(C(=O)CN(c2ccncc2)C)C)C)cnn(C)c1 45412,C(=O)(CS(F)(F)(F)(F)F)NCC1(C)CCN(C(C(C)OC)=O)C1 45413,CN1CCC(NC(=O)CC(C)(C)C#N)C12CCCN(C(c1cscc1Cl)=O)C2 45414,Cc1c(C(=O)NC(C)(C)CNC(=O)CC2(O)COC(C)(C)C2)cc(N)cc1O 45415,C1(C(C)C)C(NC(C2CCO2)=O)CCN1C(C1CC2(CCC2)C1)=O 45416,Cc1ccnc2ccc(C(N3CCC(n4cc(CO)nn4)C3)=O)cc12 45417,c1(C(=O)NC2(C)CC(NC(=O)Cc3ccncc3)C2)ccc([N+](=O)[O-])cc1 45418,N1(C(c2ccc(CC=C)cc2)=O)CCN(Cc2nc(=N)[nH][nH]2)CC1C 45419,C1(NC(=O)NC(C(C)C)C(F)(F)F)CCN(C2CC2)CC1C#N 45420,C1(NC(CCC(C)OC)=O)CCN(C(=O)CCc2cc(C)cc(C)c2)CC1(C)C 45421,N1(C(CC(C)O)=O)CC2CCC(N(C(=O)CCc3cnn(C)c3)C)C2C1 45422,CC(C)C(=O)NNC(=O)C1CCN(C(=O)OC(C)(C)C)C1Cc1ccccc1 45423,CCC(C(=O)NC(CNC(c1cccc2c1CCO2)=O)CO)C(C)(C)CC 45424,c1(CC(=O)NCC2C3CN(C(CC4OCCN(C)C4)=O)C2C3)ccnc(Cl)c1F 45425,C1(NC(c2scc(CNC(COC3(C)CCC3)=O)c2)=O)CCCCC1C#N 45426,CCCCCCC(C)NC(=O)C(=O)Nc1cc(-c2ccco2)n(-c2ccccc2)n1 45427,N1(C(Cc2cc(C)on2)=O)CCC(CNC(c2c(CO)noc2C)=O)C(F)(F)C1 45428,Cc1c(C(=O)N(CCNC(C2(CO)COC2)=O)CC2CC2)sc2cccc(F)c12 45429,C=CCCCCC(=O)N(C1CN(C(=O)CN(C)C)CCC1C)C 45430,CS(=O)c1ccc(CC(N2CCC(NC(C3CC(C)(O)C3)=O)C2)=O)cc1 45431,N1(C(C2CC(NC(=O)CSC(F)F)C23CCC3)=O)CCc2nc(O)[nH]c2C1 45432,N1(C2CCN(C(C(C)(C)OC)=O)C2)CCN(C(C2(C(F)(F)F)SCCS2)=O)CC1 45433,c1(C(C(=O)NC(CC)CNC(C2CSCCS2)=O)(F)F)cccc(Cl)c1F 45434,C1(C(=O)NCC2C=CC(NC(C(C)c3ccsc3)=O)C2)CC2(C1)CC2(F)F 45435,C1(Cc2cn(CC(CCNC(CC(C)(C)C)=O)F)nn2)CCc2n[nH]cc2C1 45436,c1(SC)ccc(NC(c2c[nH]nc2CNC(c2cnc(C)nc2C)=O)=O)c(F)c1 45437,Cc1nccnc1C(N1CCC(CNC(=O)CC(C)CN(C)C)C1)=O 45438,N1(C(Cc2cccc(C)c2)=O)C2CC1CN(C(=O)Cc1scnc1C)C2 45439,C12(C(=O)NCC3CCN(C(=O)CCc4ccncc4)C3)CCC(CC1)OC2 45440,Cc1c(C(=O)Nc2ccc(OCC(F)(F)F)nc2)cc(I)cc1Cl 45441,C(CC1CCOCC1)N=c1[nH]c(N2CCCC3(CCNC3=O)C2)nc2cc[nH]c12 45442,CC1(C)COC(C(=O)NCC2CCCC(CNC(C3COCCOC3)=O)C2)C1 45443,C(=O)(C(C)(O)C1CC1)NCC(C)CN(C)C(c1n[nH]cc1Br)=O 45444,N1(C(c2ccc(C)cc2)C)C(=O)CN(CCc2ccc(F)cc2Cl)C1=O 45445,C1(F)(CN(C(=O)CSc2nccn2C)C)CCN(C(=O)C(c2cccnc2)O)C1 45446,n1(C(C)C)ncc(Cl)c1C(=O)NCCOCCNC(C1C(F)(F)C12CC2)=O 45447,N1(C(C(C)(C)C2CCCC2)=O)CC2C(C(=O)NC(C(N)=O)C3CCCC3)C2C1 45448,C1(CC(=O)NC)CN(C(C2CN(C)C2)=O)CCN1C(C1CC=CCO1)=O 45449,c1(CC(=O)N(CC(O)CO)C(=O)NCC(=O)OC)cc(Br)ccc1Cl 45450,c1(C(C)NC(=O)Nc2ccc(COCCOC)cc2)nc(C)ccc1F 45451,C(CC(=O)NNC(=O)c1cnn(CC(F)(F)F)c1C)n1ccc(C)n1 45452,C1(CNC(C(CC(C)C)C)=O)(NC(c2cn(CCO)nn2)=O)CC2CCC1CC2 45453,c1(NC(C2(CN(C(CS(CC)=O)=O)C)CC2)=O)cccc(F)c1O 45454,c1(C(=O)NC(CNC(C(F)=C(C)C)=O)C2CC2)ccc(F)c(OC(F)F)c1 45455,n1(CC)cnc2c(N3CCN(C(=O)C(C4CCC4)OCCOC)CC3)nc(Cl)nc12 45456,CCCCS(=O)(=O)CC(=O)NC1CN(C(=O)COc2c(Cl)cccc2Cl)CC1C 45457,C(=O)(C1CCc2c[nH]nc21)N1CCCC(C)(C(=O)NCC2(SCC)CC2)C1 45458,C1(CNC(C2(SC)CC2)=O)CCCCN(C(c2ccc(N)cc2Cl)=O)C1 45459,CN=c1[nH]cc(C(=O)NC(CC)C(N2CC3C(C(N)=O)C3C2)=O)o1 45460,c1(C(=O)NCC2CC(C)(C)CN2C(c2cnsc2)=O)cc2ccccc2[nH]1 45461,c1(-n2ncc(C(N3CC4C(NC(c5ccoc5)=O)(C4)C3)=O)c2)cc(F)ccc1F 45462,Cn1ccc(C(=O)NCC2CCN(C(C3(n4cc(Br)cn4)CC3)=O)C2)cc1=O 45463,C1(C(=O)NC(C)(C)CNC(=O)CC2SC(=N)NC2=O)CS(=O)(=O)CCO1 45464,c1(C(NOC(CC)CC)=O)cc(CNC(C2(C(=O)NC)CCC2)=O)ccn1 45465,Cc1ccc(CNC(C2CC2CNC(c2cc(C(F)F)no2)=O)=O)c(F)c1 45466,N1(C(c2ccc(C)cc2Cl)=O)CCCC(F)(CNC(=O)CC(O)C(C)C)CC1 45467,c1(CC(=O)NCc2n(C(=O)OCC)cnn2)c(C)n[nH]c1C.C1(=O)C(C)C2(CC2)C1 45468,N1(C(C(CCNC(C(CC=C)NC(C)=O)=O)O)=O)CCC12CN(C)C2 45469,c1(CC)ccnc(C(=O)NC(CNC(C2CC23CC(OC)C3)=O)CC(C)C)c1 45470,C1(CNC(C23OC(C)C(C2)C3)=O)(CO)CCN(C(=O)C(O)CC(N)=O)CC1 45471,N1(C(CCC(=C)Br)=O)CC2CC(C1)CN(C(=O)CCC(CC)OC)C2 45472,CCCC(C)(C)C(=O)N1CCCCC(CNC(=O)C(O)CCSC)C1 45473,C1(C(N2C(CNC(c3cnc(OCC)s3)=O)COCC2)=O)CCCCCN1C 45474,c1(OC(C)C)ccc(C(=O)NC2CCCCC2CNCc2ccnnc2O)nn1 45475,C12(C(=O)NC3C(NC(C(N(C)C)C4CC4)=O)CC3)CC3CC(F)(C1)CC(F)(C3)C2 45476,c1(-c2onc(C(c3cc(C)c(Br)cn3)c3cccc(C)c3)n2)ccc2cncn2c1 45477,C(C)(CC(=O)NC(c1nocc1C(=O)N(C)Cc1ccn(C)n1)C)SC 45478,Cn1ncc([N+](=O)[O-])c1C(=O)NCC(=C1CN(C(c2cc(Cl)cc(Cl)n2)=O)C1)F 45479,CC12CC(CC1C(=O)NCCCN(C(C1(O)CCOCC1)=O)CC1CCCC1)C2 45480,n1(CC(=O)NCC(C)(C)NC(C2(OC)CC2)=O)c(C)cc(O)cc1=O 45481,N1(c2ccc(C)nn2)CCC2(CCN(C(c3ccn4ccnc4c3)=O)CC2)CC1 45482,C(=O)(CCCS(N)(=O)=O)N1CC(NC(C2(C#C)CCC2)=O)C(C)C1 45483,c1(-c2nc(-c3cc(C)oc3C)nn2C2CCOC2)ccc2nsnc2c1 45484,Cc1cnc(C(C2CC2)NC(C2CS(=O)(=O)C2)=O)s1 45485,n1(CCOC)ccc(C(=O)NC(C)(CNC(c2cc(C)cs2)=O)C2CC2)n1 45486,C1(NC(C(C)NC(=O)NC)=O)CCN(C(=O)CC2CCC(C)CC2)C(C)C1 45487,C(C(C)CC(F)(F)F)NC(C1(C(C)C)N(C(c2ccc(CC)o2)=O)CC1)=O 45488,Cc1ccc(F)cc1CC(=O)NCC(O)CCNC(c1csc(C(C)(C)C)c1)=O 45489,C#CCC(CC)NC(=O)C(C)NC(C1(CO)CCCC1)=O 45490,C1(NC(CN2C(=O)NCCC2)=O)CCN(C(C2CC3C=CC2CC3)=O)C12CCC2 45491,C1(CN(C(C(n2c(C)ccn2)C)=O)C)CN(C(=O)CC2CC2(C)C)CC12CC2 45492,c1(C(N2CC3CCN(C(CC(=O)OC)=O)C3CC2)=O)cnc2c(C)cccc2c1 45493,S(=O)(=O)(c1cccnc1N1CCS(=O)CC1)NCC(c1ccccc1Cl)C 45494,N1(C(c2c(CC(C)C)onc2)=O)CCN(C(c2cc(N)c(Cl)cn2)=O)C2(CC2)C1 45495,N1(C(CC=CC=C)=O)CC(F)(F)CC1CNC(c1coc(Br)n1)=O 45496,C1(NC(C(c2cn(C)nc2)=O)=O)CCN(C(=O)C=Cc2cccc(F)c2)C12CC2 45497,C1(C(=O)NCc2c(CC)nco2)CNC(=O)CN1C(=O)C(F)C1CCC1 45498,CN1CC2(CC2)CC1C(=O)NC1CC(O)CN(C(=O)CC2CC3C=CC2C3)C1 45499,CCCCCCCCOCC(=O)NCCCN(C)C(C1CN(C(C)C)CCO1)=O 45500,c1(SC)cncc(C(=O)NCC=C2CCN(C(=O)CCn3cc(C)cn3)CC2)c1 45501,C#Cc1cc(NC(c2nnnn2C2CCOC2)C2(C)N=N2)ccc1C 45502,C1(NC(CCCOC(C)C)=O)CCC(CNC(c2csc(S)n2)=O)CC1 45503,c1(C(C(N2CCC(NC(C34CC(F)C3C4)=O)C2)=O)O)ccccc1Cl 45504,C1(C)(C(=O)NCCc2ccc(C)nc2)CN(C(c2ccsc2)=O)C(C)(C)C1 45505,N12CCC(CC)(CC1)NC(=O)C1CCCC1C2=O.C1(CC)CCCN(C)C1 45506,C1(OC)CN(C(=NCCCN(C)C(C)=O)Nc2ccc(OC)cc2)CC1O 45507,C1(C(=O)NC2C(NC(C3C(c4cn(C)nc4)C3)=O)CCC2)CCCCNC1=O 45508,Cc1ccccc1C1(C(=O)NC2COCC2NC(C23CCC2C3)=O)CCOCC1 45509,C12(C(=O)NCCN(C)C(c3cn(CCN4CC5CC5C4)cn3)=O)CCC(CC1)C2 45510,c1(C(N(C)Cc2cncc(C)c2)=O)nn(C)c(Cl)c1C(F)F.c12cccn1C2 45511,N1(C(CNS(CCCOC)(=O)=O)=O)CC2CC1CC2C(=O)Nc1cn[nH]c1 45512,C(C)(C)(C(F)(F)F)OCC(=O)NC1CN(C(c2c(-c3cn(CC)nc3)n[nH]c2)=O)C1 45513,N1(C(C=CC2C(C)C2(Cl)Cl)=O)CC2(CCN(C(c3cc(C(N)=O)no3)=O)C2)C1 45514,c1(OC)cc(NCC2CC(NC(C3CN(C)C(=O)N3)=O)C2)nc(OC)n1 45515,C=C1CCN(C(c2ccn(CCNC(=O)Cc3nocc3C)c2)=O)C1 45516,C12(C(=O)NS(=O)(=O)CC3CCCC(OC)C3)CN(CC)C(CNC)(C1)C2 45517,C1(NC(C=CC)=O)CCN(C(c2c(-c3ccccc3)cnn2C)=O)CC1F 45518,Cc1c(CNC(=O)CCC2CCCN2C(=O)C(C)(O)C2CC2)nnn1C 45519,Cc1nn(C)cc1CCNC(=O)C(C1(O)CN(C(C2CC2C(N)=O)=O)C1)F 45520,N1(C(C(C)C)=O)CC(O)CC1CCCNC(C1CC(=O)N(c2ccc(F)cc2)C1)=O 45521,C(=O)(C1=CCCCCC1)N1C(C)CC(CC(=O)NCC2COCCOC2)C1 45522,C1(NC(C(C2CCC2)OCC)=O)CCN(C(=O)CSC(C)C)CC12CCC2 45523,C(=O)(C1=C(C)OCCS1)N1CC(C(N2CCC(O)(CC)CC2)=O)OCC1 45524,N1(CC(C)NC(N2CCC(C=O)C2)=O)CCOCC1.C12CC(F)(C1)C2 45525,C1(OC)CC(NC(=O)CCCCCF)CN(C(c2cc(N)ccc2F)=O)C1 45526,N1(C(c2ccc(NC(C)CCN(C)C)cc2)=O)CCC2(CC1)C(C)(C)C2 45527,CC#CCCC(=O)NCC(C)(O)CNC(C1COCCN1CC(F)(F)F)=O 45528,N1(C(C2=NOC(C)C2)=O)C2CCC1CC(CC(C)NC(C1(C)CC=CC1)=O)C2 45529,c1(C(=O)NCCOCCOCC)cc(SC)[nH]n1.C12CC1NC2=O.CC 45530,C12(C(N(C)CC3CCN(C(=O)C(O)CF)C3)=O)CCC(C(F)(F)F)(CC1)CC2 45531,CON(CCO)C(=O)CNC1COCC1C(=O)NC1C2CCCC1CC2 45532,C12(NC(C(COC)C)=O)CC(C)(C1)OC21CN(C(C23CCCN(CC2)C3)=O)C1 45533,C1(C(=O)OC)CC2CCC(C1)C2NC(C1OCCC1C)=O 45534,c1(C(N2C3CCC(NC(C=C(CCC)CCC)=O)(C3)C2)=O)cccc2ccnn12 45535,c1(C(=O)NC(CC(C)NC(c2[nH]cc(C)c2)=O)C)onc2ccccc12 45536,c1(C(N2C(C(N3CCC(O)C3)=O)CC3CC32)=O)cccc(C(F)(F)F)c1F 45537,CC(C(=O)NCC1CN(C(=O)C(C)C2(O)CCC2)CCN1C)S(N)(=O)=O 45538,C12(NC(C(C)Cc3ccc(Cl)cc3)=O)CCC(C1)N(C(=O)C(F)=C1CCC1)C2 45539,O=C(C#CC1CCC1)NCC1(CNC(c2ccc(C(F)F)o2)=O)CCC1 45540,Cc1cc(Cl)c(C(=O)NCC(C)N(C)C(C2CC2c2ccn(C)n2)=O)c(Cl)c1 45541,Cc1cn2c(CC(=O)NC(c3ccc(F)cc3)CNC(c3ccsn3)=O)csc2n1 45542,C(CC1=CCN(C(c2n[nH]c(C)c2O)=O)CC1)NC(C1(CC)CCOCC1)=O 45543,C1(NC(CC2(C)CC2)=O)CCN(C(C2CC3(C2)CC3(F)F)=O)CC1F 45544,C#Cc1cc(C(N(C(CNC(=O)C(C)c2cccs2)C2CC2)C)=O)cc(F)c1 45545,N1(C(CCC=C(C)C)=O)CC(NC(C2(O)CCC2)=O)CC12CCOC2 45546,C(=O)(CC(C)C(C)(C)NC(c1ccnnc1)=O)N1CCC(C#C)(O)C1 45547,CCCCCCn1nnnc1C(C1OCCO1)Nc1cn(CC)cn1 45548,C1(OC(CC)CNC(=O)NC(Cc2cccs2)CC)CCOCC1 45549,c1(CC(C)NC(=O)CC23CCCC2C3)ccccc1Br.C1C(C)(C)CNC1=O 45550,c1(OC)ccnc(N(Cc2ccccc2C2CC2)CC2CCCCO2)c1 45551,C1(CNC(C2CNC(=O)N2)=O)CCCN(C(C2CC3CC3C2)=O)C1 45552,Cc1nc(CO)oc1C(=O)NCC(O)CNC(C1(C2CCCO2)CCOCC1)=O 45553,C(=O)(CCCC(C)(C)C)N1CC(C#C)(C(=O)NCC(F)Br)C1 45554,C1(CNC(c2cn(CC(C)C)nc2)=O)CC2CN(C(C3CC4CCC3O4)=O)CC12 45555,CC(C)(C(=O)N(O)Cc1cn(CC(=O)NCC2(S(C)(=O)=O)CCC2)nn1)C1CC1 45556,C1(C(=O)NCC2N(C(c3cscn3)=O)CCC2)(CC2CCCC2)CCCCC1 45557,O=C1CC2(CCN(C(=O)CC3CN(Cc4cccnc4O)CCO3)CC2)C(=O)N1 45558,C12(CNC(c3c(OCC)nccc3)=O)CCCC1N(C(=O)CSC1CC1)CCC2 45559,N1(C(C2CC(=C3CCC3)C2)=O)CCN(C(C2CCc3nccn3C2)=O)C2COCC12 45560,C12CC(C)N(C1)C2=O.c1(C2(CNC(C3(OC)CC3)=O)CC2)ccccc1F 45561,c1(C(=O)NCC2CCN2C(=O)COc2ccsc2)ccncc1F 45562,C123CC(C1)N(C2)C3=O.N1(C(=O)OC(C)(C)C)CCCCC1CCCN(C)CCO 45563,c1(N(CC(C)(C)CCC)C(=O)CC(=O)OC(C)(C)C)cn2cc(C)sc2n1.C(=O)OC 45564,Cc1ccc(C(N2CC3CCC(C2)N3Cc2c(F)ccnc2Cl)=O)c([N+](=O)[O-])c1 45565,c1(C(=O)NC2CCN(Cc3ccnc(C)n3)C2)cccc2nccnc12 45566,C1(C(=O)NC(C)CNC(C2(C(C)(F)F)CC2)=O)CC(OCC(F)(F)F)C1 45567,N1(C(CC=C=C)=O)CCC2C(CCCN2C(c2ccc3c(c2)CCOC3)=O)C1 45568,c1(C(=O)NCC2C3CN(C(C(C)OC)=O)C2C3)ccc(-n2cccc2)cc1O 45569,C1(C(=O)NCC2CN(C(c3cc(OC)n(C)n3)=O)C2)CCCC(C)(C)O1 45570,Cc1nn2ncccc2c1C(=O)NCCC(C)N(C(=O)CC(C)(C)CC(F)F)C 45571,CCC(CNC(=O)C(C)CSC)(CC)C(=O)NC1CC(C)N(C)CC1C 45572,Nc1nc(C(N2CC3CC(NC(c4cc(CCCO)on4)=O)C2C3)=O)ccc1O 45573,c1(CC)ccc(Cl)c(C(=O)NCC2(C(C)NC(C3CCCCC3(C)C)=O)CC2)c1 45574,C1(N(C(C2CC2(C)C)=O)CC)(CF)CCN(C(=O)C(C)C2CCOC2)C1 45575,Cc1c(C(N2CCOCC2CNC(=O)CCc2ccccc2)=O)ncn1C 45576,C(C(=O)NC1(CO)CC(F)C1)(C(C)(C)C)OC.c12nc(C)c(o1)c(=O)[nH]2 45577,Cc1ccc(CNc2ccc(C(=O)NCC3CNCCO3)nc2)c(Cl)c1Cl 45578,C=C(Br)CCC(=O)NC1CCC(CNC(=O)C=C(C)Cl)C1 45579,C1(C(N2CC(NC(c3c(CC)cc[nH]3)=O)C(C)C2)=O)CCC2CC2CC1 45580,C(=O)(C(=O)C(C)CC)NCC(CCOC)NC(CC(C=C)C)=O 45581,c1(C(=O)NCCC(=O)NC2CC2)ccoc1C(=O)NC1CC1c1cscn1 45582,C1(O)(CN(C(=O)CC2CC23CC3)C)CCN(C(=O)Cc2cccc(Cl)c2)C1 45583,C(=O)(CCC(=O)N1CCC(NC(=O)CCOc2ccccc2)C1C)OCC 45584,N1(C(Cc2ccc(C)s2)=O)CC(NC(c2cc(C(N)=O)n(C)n2)=O)CC(C)C1 45585,CC1CN(C(c2ccc(CN(C)C)o2)=O)CC1CNC(c1ccsc1C#N)=O 45586,CC1CC(C(N2CCC(NC(c3nsnc3O)=O)C(C)C2)=O)CC(C)O1 45587,S(=O)(=O)(CCC(=O)N1CCC(N(C(=O)C(O)C(C)(C)C)C)C1)NC 45588,N1(C(COC(CC)C)=O)CCC1C(=O)NCCC1(CO)CC1 45589,c1(NC(C2CC(NC(c3nc(CC)oc3C)=O)C(O)C2)=O)ccc(O)c(CC)c1 45590,N1(C(c2c(SC)cccc2)=O)CC2CCN(C(=O)C(F)n3cccn3)CC2C1 45591,Cc1ccc2c(N3CCSC4(CCC4)C3)nc(=NCC3CCC(C(N)=O)O3)[nH]c2c1 45592,c1(C(=O)NC2CCCC(NC(C3N(CC)CCC3)=O)C2)cc(C#N)oc1C 45593,CC1CCc2ncc(C(N3CC4CC(NC(=O)C(C)CC(N)=O)CC4C3)=O)n2C1 45594,N1(C(c2nc(N(C)C)oc2)=O)CCCC1(C)CNC(=O)CCS(C)=O 45595,C1(CNC(c2cccc(SCC#C)c2)=O)CCN(C(=O)C(C)C(F)F)C1(C)C 45596,C12(C(N(CCCNC(=O)C3=CCCSC3)C)=O)CC(C)(C1)OC2(C)C 45597,C1(CNC(c2c(COC)n[nH]c2)=O)CC(C)(C)CCC1NC(c1ocnc1C)=O 45598,C1(CCC)CCCC1C(=O)NC12CC(C(N3CCC3(C)C(=O)N(C)C)=O)(C1)C2 45599,Cc1ccc(CC(N2CC3CCC3(CNC(C3CCOC(=O)CC3)=O)C2)=O)c(C)c1 45600,CC1CN(C(=O)CC2CN(C)C2)CCN1C(c1coc(C2CCC2)n1)=O 45601,Cc1ccc(C(=O)N(C)CC2(O)CN(C(=O)C(C)N3CCCC3)C2)o1 45602,c1(C(N(CCCCN(C(C(c2ccnn2C)C)=O)C)C)=O)cc(O)nn1C 45603,C1(N(C(CSCC)=O)C)CCC2(CC1)CCN(C(=O)CC1CCCC(C)(C)O1)C2 45604,c1(C(N2CC(C(=O)OC)C2(C)C)=O)cc(F)cc2nc(S)[nH]c12 45605,c1(C(N2CC(NC(C3CCCN(C(=O)OC)C3)=O)C2)=O)ncc(Cl)cc1F 45606,N1(C(C(C2CCN(C(CC(COC)(C)O)=O)C2)F)=O)CC2(COCC(=O)N2)C1 45607,c1(C(C(=O)NCC(C)C)N(C)Cc2c(Br)cn(CC)n2)cccc2cnccc12 45608,C(=O)(CCCCC(C)(C)OC)NCC1(OC)CN(C(C2C(C(=O)OC)CC2)=O)C1 45609,n1(CCNC(C2C(C(=O)OCC)C2)=O)cc(Br)nn1 45610,c1(CNC(N2CC(C)(CC(c3ccccc3)O)C2)=O)ccc(Cl)cc1F 45611,c1(C(N(C2CCN(C(c3ccco3)=O)CC2)CC#C)=O)csc2c1CCCC2 45612,c1(SC)cc(C)ccc1C(=O)NCC(C(C)C)NC(=O)C(C)C(F)F 45613,N1(C(C2N(C(C)=O)CCOC2)=O)CCCN(C(c2ccc(Cl)o2)=O)CC1C 45614,n1(C2(C(=O)NCC3N(C(C(C)NC(C)(C)C)=O)CCC3)CC2)cc(C#N)cn1 45615,C1(NC(c2ccnc(S)c2)=O)CN(C(c2occc2Br)=O)C2(CCOC2)C1 45616,CN1CCOCC1CC(N1CCC(CCNC(=O)C(F)C2CC2)CC1)=O 45617,C1(NC(Cc2c(C)non2)=O)CC12CCC(NC(=O)CCC1(C)CC1)CC2 45618,C1(F)(CNC(=O)NC2C(c3cccc(OCC)c3)C2)CC2(CCC2)C1 45619,C(=O)(C(C)(C)C(F)F)N(C)CC1(O)CCN(C(=O)C=Cc2cccn2C)C1 45620,N1(C(=O)CCc2cc(Cl)sc2Cl)CCC2(CCCN2C(=O)CC2CC(F)C2)C1 45621,N12CCc3ccccc3C1CC(=O)NC(C)C2=O.C(C)(C)(C)OC(C)=O 45622,N1(C(CSCCOC)=O)CCC2CCN(C(=O)COCCCN(C)C)CC2C1 45623,CCCCC(O)C(=O)NCC1CCCN1C(c1csc(-c2coc(=N)[nH]2)n1)=O 45624,O=C(CN=c1cc[nH]cc1)NCC(O)CNC(c1csc(-c2ccco2)c1)=O 45625,n1(CC(=O)NCC(CC)NC(=O)Cc2ccn(C)n2)c(-c2cccs2)nnc1S 45626,C(=O)(C(C)C(F)(F)C(F)F)NC.C(=O)(C(C(=O)N(CCCN(C)CC)C)OC)OC 45627,Cc1ccc(C(=O)NC(C(N2CC(C(N)=O)C3(CC3)C2)=O)c2ccoc2)cc1F 45628,C1(NC(C2(CC)CN(C(=O)Cn3cc(C#N)cn3)C2)=O)CCCCC1(C)C 45629,CC1CCc2ccccc2C1NC(c1ccc(N2CCCC2=O)cc1)=O 45630,C1(OC)(CNC(c2nocc2C)=O)CCN(C(C2COCCC2C)=O)C1 45631,N1(C(c2c(N)cccn2)=O)CC2CC(NC(=O)CCSc3ccccc3F)C1C2 45632,Cc1ccnc(C(=O)NC2CC2CNC(c2ccc(Cn3cccc3)cc2)=O)c1 45633,c1(OCC)cccc(NC(C2(C)CC(C)=NO2)=O)c1 45634,C1(NC(Cc2c(C#C)cccc2)=O)CCN(C(=O)CC(C)SC)C12CCCC2 45635,c1(CC)ccc(CC(N2CC=CC(NC(=O)Cc3cnc[nH]3)C2)=O)cc1 45636,C1(CNC(C=C(C)C)=O)(NC(C2CNC(=O)N2)=O)CCC(F)(F)CC1 45637,c1(CC(=O)NCC2(COC)CCCN2C(=O)C=C2CCC2)ccc(Cl)nc1C 45638,CCC(CC)C(F)C(=O)NCC1CN(C(C2CC3(CCC3=O)C2)=O)CC1O 45639,c1(C(N(C(C)C(C)C)CC)=O)cc(C(F)F)cc(C)c1 45640,N1(C(c2c(CCC)nco2)=O)CCCC(C(=O)N(CC(O)CF)C)(CC)C1 45641,N1(CC(=O)NCC(C)C)CCCC1C1CCCCN1C(=O)CCN(S(C)(=O)=O)C 45642,N1(C(C(c2cccnc2)C)=O)CCCC(C)(NC(=O)CCn2ncn(C)c2=O)C1 45643,S(=O)(=O)(c1ccc(Br)cc1[N+](=O)[O-])NC(c1ccc(CSc2cccnc2)cc1)=O 45644,CCC(CC)(CCNC(=O)C(N1CCCCC1)C1CC1)NC(c1cnc(C)s1)=O 45645,C1(C(=O)OCC)CCc2cn(CCCC(F)(F)F)nc2C1.c12ccc(F)c(c1)CN2 45646,c1(C(N2CCCCC2C(C)C)C(=O)NCC)cccc2cc(CSC)sc12.C=O 45647,C1(NC(c2cc(CC)n(C)n2)=O)CC2CC1N(C(=O)CCOC1CCOCC1)C2 45648,C1(=O)C(CCSC)N(C)C2CCN1C2.C(=O)(C(=O)NCCOC)OCC 45649,C1(NC(c2c(C)nc(C(F)(F)F)o2)=O)CN(C(=O)C(O)C2CC2)C(C)(C)C1 45650,c1(C(N(CC(C)O)CCNC(c2c(C#C)cn(C)n2)=O)=O)cn2cc(C)sc2n1 45651,c1(SC)cccc(F)c1C(=O)NC1C2CC1N(C(=O)Cc1ccn(C(C)C)n1)C2 45652,c1(NC)cc(C(=O)NC2CCN(C(C3CC(C#N)C3)=O)CC2CO)cc(Cl)n1 45653,c1(N2C(CN(C)C(c3ccc(C(F)F)nc3)=O)CCC2)nc(Cl)nc2[nH]ccc12 45654,C1(Nc2n(C)cc(Nc3ncc(C(=O)OC)cn3)n2)CCC(C2CC2)C1 45655,c1(C(=O)NC2(CCNC(C=COCC)=O)CCOCC2)ccc2n[nH]cc2c1 45656,c1(CC(=O)NCCCNC(c2ccsc2Cl)=O)cc(Cl)ccc1O 45657,C(=O)(CCNC(C1CCC1)=O)N(C1CN(C(C2(N(C)C)CCC2)=O)C1)C 45658,N1(C(CC2(NC(C)=O)CCCCC2)=O)CCN(C)CC1CNC(C1CC=CC1)=O 45659,N1(C(c2cnc(OC)[nH]2)=O)CCCC2(NC(c3sc(C)cc3Br)=O)CC2C1 45660,C1(CCN(C)C(C2CCCO2)=O)CCN(C(C2C(Cl)(Cl)C23CC3)=O)CC1 45661,C1(N(C)C)CN(C(C2CCCN(C(N)=O)C2)=O)CCC1F 45662,Cc1ccc(C#N)cc1NC(C1CCN(C(C2CCOC2(C)C)=O)CC1(C)C)=O 45663,C(=O)(CC(C(F)F)N1CCOCC1)NC(C)CCNC(C1CC(O)C1)=O 45664,Cc1ccc(OC(F)F)c(NC(N2CCN(C(=O)CP(C)(C)=O)C3CC23)=O)c1 45665,c1(C(=O)NC(C)CCNC(=O)CCC2CNC(=O)N2)ccc2c(c1)[nH]c(=N)n2C 45666,c1(CC(=O)NC2C(NC(CC(=C=C)C)=O)CCC2)c[nH]c2c(F)cccc12 45667,N1(C(C(C(C)C)O)=O)CCc2nc[nH]c2C12CCN(C(c1cccc(N)c1)=O)C2 45668,CC1(C)C2CCC(C(=O)NC34CC3CN(C(C3(CC5CC5)CCC3)=O)C4)C1C2 45669,CC(C(=O)NCC1CCN1C(c1cccc(=O)o1)=O)C(F)F 45670,Cc1ccc2[nH]cc(CC3(NC(=O)NCC(N4CCC(O)C4)(C)C)CC3)c2c1 45671,C1(CC)CN(C(C2CC23CCOCC3)=O)CCC1(F)NC(=O)CC1CCCCC1 45672,c1(C(CNC(c2ccccn2)=O)NC2CCN(Cc3ccccc3)C2)ccccc1 45673,Cc1cc(F)cnc1C(=O)NCCCC(C)(C)NC(C1CC2CCC1C2)=O 45674,C1(OCC(=O)NCC(C)(F)CNC(C2(CO)CC2)=O)CCCCC1C 45675,c1(CC(=O)OC(CCC=C)C)cc(Cl)cc2ccccc12 45676,c1(OCC(=O)NCC(CN)F)ccc(F)c(F)c1.C(C(=O)NCCC(C)C)O 45677,c1(CC)cc(C(=O)NCC(F)CNC(c2cn(C)cc2C(F)(F)F)=O)oc1CC 45678,Cc1ncsc1C(=O)OCc1cocn1 45679,c1(C(=O)NCCC2CC(NC(CC3(C)CCC3)=O)C2)ccnc(-c2ccco2)c1 45680,C(C(=O)NNC(=O)C(C)(C)CCCCNC(=O)CSC1CC1)OCC=C 45681,C(=O)(CCCCN1CCCC1)NC(C(C)NC(c1ccc(=O)oc1)=O)(C)C 45682,C(=O)(C#CC1CCCOC1)N1CC(C)N(C(c2coc3ccc(F)cc23)=O)CC1 45683,C1(O)(C(C)NC(=O)CSC2(O)CCC2)CCCN(C(=O)CC2CCS(=O)(=O)C2)C1 45684,c1(C2(C(N3C(C4(C(=O)NC5CCCC5)CC4)CC3)=O)CC2)ccncc1 45685,C1(CC)OCCCC1C(=O)NCCN(C(c1cc(Cl)c[nH]1)=O)Cc1cccc(Cl)c1 45686,N1(C(CCN(C)C)=O)C2CCC1(Cn1cc(C3CC3C(=O)O)nn1)CC2.C(C)(C)(C)O 45687,C1(C(=O)NCCc2cc(C)nn2C)CCN(C(c2ccccn2)=O)CC1O 45688,N1(C(=O)CC2CCCCC2)CCCC(C2CN(C(c3cc(F)ccc3Cl)=O)C2)C1 45689,C(=O)(CC1OCCc2ccsc21)NC1(CCNC(=O)Cc2cncnc2)CCC1 45690,N1(C(C2(CC)COC2)=O)CC(C2CN(C(c3cccc(N(C)C)n3)=O)C2)C1 45691,C1(C2CC2)(CNC(C2C(OCC)C2)=O)CCN(C(=O)CN=S(C)(C)=O)C1 45692,C1(C(=O)NC(c2ncccn2)C2CC2)CC(=O)N(C2CCS(=O)(=O)C2)C1 45693,C12(C(N3CCN(C(C4CC(C)OC4)=O)CC3)=O)CCC(CC1)OC2 45694,C(=O)(C1CSc2ccccc21)NCc1c(OCC#C)nccc1 45695,N1(C(C(CNC(=O)C(c2ccc(F)cc2)(F)F)N(C)C)=O)CC2OCCOC2C1 45696,C=C(C)CCCC(=O)N1CCC(C(C)(C)NC(=O)C(CC)c2cccnc2)C1 45697,C12(C(=O)NCC(CC=C)NC(C3(C)CC4CCC3C4)=O)CC3CC(C(=O)N1)C2C3 45698,C=CCC(CNC(=O)C(C)C=C)C(=O)NCC(Cl)C(C)(F)F 45699,Cc1cccc([N+](=O)[O-])c1NC(C)CN(C)C(C1CC2(CSC2)C1)=O 45700,C=CCC(CC)C(=O)N1CCN(C(=O)COc2cccc(F)c2F)CC1COC 45701,N1(C(c2c(O)ccc(C)c2)=O)CCC(C(=O)NCC(c2cnc[nH]2)C)CC1(C)C 45702,C1(N(C(c2c(CC)ncs2)=O)C)CCN(C(=O)CC2(c3ccon3)CC2)CC1 45703,C1(NC(C(=O)N(C)C)=O)CN(C(=O)C#CC2CC2)C2(CCOC2)C1.C12(CC1)C(=O)C2 45704,C=C(Cl)CC(C(=O)NCc1cc(C)ccc1OC)NC(=O)CCCOC 45705,c1cccc(O)c1CNC(=O)NC12CC(NC(=O)OC)C1C2.C(C)(C)(C)OC 45706,c1(SC)nc(N2CC(OCC(N)=O)C2)cc(Cl)n1 45707,Cc1ccc(C)c(CC(N2CCC(CNC(=O)C=C3CCC3)C(C)C2)=O)c1 45708,C1(C(=O)NCC=CCNC(C(c2ccccc2F)C)=O)CCC2(CC1)CC(=O)C2 45709,c1(C(N(CCNC(c2c(CC)n(CC)nc2)=O)C(C)C)=O)cccc(C)c1F 45710,C(=O)(C(F)CC(C)(C)NC(C1(CO)CCCC1)=O)NC1CC(CCN(C)C)C1 45711,CC(CCNC(=O)Cc1cnc[nH]1)CCNC(C1CNC(=O)N1)=O 45712,CC1CC(NC(=O)CC2(C)CC2(Cl)Cl)CN1C(=O)CSCC(F)(F)F 45713,c1(CNC(C(CC)NC(c2occc2C(C)C)=O)=O)cnc(C)n1CC 45714,N1(C(C2(CCC)CCC2)=O)CC2CCCC2(NC(=O)C=C(Cl)Cl)C1 45715,N1(C(C2(CNC(CC3CC(=C)C3)=O)CC23CCC3)=O)CCCNC(=O)C1CC 45716,C1(CC)CCN(C(=NCCCCl)NCC(F)F)C1.c12cnc(C)c(c1)C(=O)N2 45717,c1(COC)ccc(C(=O)NCC(C2CCC2)NC(c2oncc2C)=O)cc1 45718,C1(NC(c2n(CC)ccc2)=O)CC2(C1)CC(NC(=O)CC(O)c1ccccc1)C2 45719,Nc1ccc(C(=O)NCCC2CCCN2C(=O)CN2CCS(=O)(=O)CC2)cc1Cl 45720,C=CC1(O)CCN(C(=O)C2=CCN(C(=O)Cc3ccns3)C2)C1 45721,c1(N(C(c2n(CCC)ccn2)C(=O)NC)C)cc(C)cc(O)c1 45722,N1(C(C(C)NC(C)=O)=O)CCOC(C(=O)NC(C)CC2CCC2)C1 45723,Cc1oc(C2CC2)nc1NS(=O)(=O)CC1CC1(F)F 45724,C(C(=O)NCC(C)C)(C(C)CC)NC(c1cc(CC)nn1C)=O 45725,C(C(C)C)(C(O)C(=O)N1CC(n2cc(COC(=N)O)nn2)CCC1(C)C)OC 45726,C#Cc1ccc(CNc2cccnc2C(=O)NC2(c3ccccc3F)CCC2)s1 45727,N1(C(c2cc(C)cc(O)c2)=O)CCC(C2(NC(c3cnnn3C)=O)CC2)CC1 45728,Cc1cncc(C(N2CCC(O)(C(C)CNC(=O)Cc3nocc3C)C2)=O)c1 45729,C1(N(CCNC(=O)C(O)CC)C(C)=O)CCCCC1.CCCC=O 45730,c1(CCNC(C(C2CC2)NC(CN(C)CC)=O)=O)cnc(C)cn1 45731,N1(C(C(CCC)OCC)=O)CC2CN(C(=O)CCc3cc(C)on3)CC2(C)C1 45732,c1(C(N(CCCCNC(c2ccsc2C(F)F)=O)C)=O)cc2c(nn1)CCCC2 45733,c1(C(N2C(CNC(CC3C(C)=NNC3=O)=O)C=CC2)=O)cc(C)ccc1F 45734,c1(NC(=O)C(F)CC2CNC2)cnccc1NC=O 45735,C1(C(C)NC(C(C)OCC#C)=O)CCCN1C(c1c[nH]nc1-c1cccnc1)=O 45736,N1(CC2CC(C(C)NC(c3cnc(C4CC4)o3)=O)C2)CCC(CC(=O)OCC)CC1 45737,c1(NCC2OCCN(C(=O)C=Cc3ccccn3)C2)ncnc2c(Cl)cc(Cl)cc12 45738,N(C(=NCc1ccccn1)N1CCC(Cc2ccsc2)C1)C(=O)Nc1ncccn1 45739,CC#CCCCCN=c1ccc2cc(S(=O)(=O)NC3CCOC(C)C3)ccc2[nH]1 45740,c1(SC)ccc([N+](=O)[O-])cc1C(N1CCC12CN(C(C1CCCNC1=O)=O)C2)=O 45741,C(=O)(C(C(C)(C)C)N1CCOC1=O)N(CCCCNC(C(C(C)O)N(C)C)=O)C 45742,N1(C(=O)C=CCN(C)C)CCCC(NC(c2n(CC)nc(C)c2)=O)CC1 45743,C1(C(C)C(N2CCCC2C2(NC(=O)CN3CCOC3=O)CC2)=O)CCN(C)CC1 45744,C#CCC(C)(C(=O)NCC1CC=C(C)CC1)NC(=O)CC1CCOC1(C)C 45745,C1(NC(c2occ(C)c2)=O)(CO)CCN(C(c2ccc(CC(C)(C)C)cc2)=O)C1 45746,N1(C(C2OCCN(C(C3(CC(C)C)CCC3)=O)CC2)=O)C2CCC1CN(C)CC2 45747,c1(C(=O)OC(CC)C(C)C)cn2c(n1)CCN(c1snc(CO)c1OC)CC2 45748,C(=O)(C#CC1CCOCC1)N(C(CCNC(C(CC(=O)OCC)C)=O)C)C 45749,c1(C(=O)NCC2C(NC(=O)Cc3cscn3)CC2)cc2ncccc2s1 45750,N1(C(C(C)NC(N)=O)=O)CC2(CC(NC(=O)C(C)(C)NS(C)(=O)=O)C2)C1 45751,CC(C)(C)C(CNC(=O)CCc1nccs1)C(=O)N1CCC(O)(C(F)F)C1 45752,C1(F)(CNC(C(C)=C(C)C)=O)CCCN(C(C2(C)CC(C)C2)=O)C1 45753,c1(C(N2CCC(O)(CNC(C(=CC3CCCCC3)C)=O)C2)=O)cc(=O)cc(Cl)[nH]1 45754,c1(C(=O)NCCn2cnc(C(=O)NCCc3cn[nH]c3)c2)c(O)cccc1Cl 45755,C(C(C)(C(=O)NC1=CN2CN=C2S1)NCCN(C(C)=O)C1CC1)OC 45756,C(c1ccccc1)=CCC(N1CCC(CCNC(C(COCC)C)=O)C1)=O 45757,N1(C(=O)CC2CNCCS2(=O)=O)Cc2c(ccc(F)c2Br)C1=O 45758,C(=O)(CCC(C(C)C)NC(c1c[nH]c(C)c1)=O)N1CCCC(OC)CC1 45759,N1(C(C)C)CC(C(=O)NCCCC2(C)CC2)CC1=O.c12ccccc1CNC2=O 45760,Cn1nccc1C=CC(=O)NC1CCCCC1NC(=O)CN1CCC(C(F)F)C1 45761,C=CCC(F)(F)C(=O)NCC1COC(C)(CNC(=O)C(C)Cc2cnco2)C1 45762,c1(-c2ccc(NC(N3CCC(c4ncc(C)cn4)CC3)=O)o2)ccc(Cl)c(F)c1 45763,Cc1ccc(CC(=O)NC2CC(CNC(=O)Cn3ccc([N+](=O)[O-])n3)C2)c(C)c1 45764,CC1(C)CC(NC(=O)CCSC(F)F)CN1C(=O)CSc1cccc(Cl)c1 45765,C1(C(=O)NCCCc2nc(C)[nH]n2)CCCC(NC(=O)C(F)CC2CCOC2)CC1 45766,N1(C(=O)CCOC2CCCC2)CCC(C(C)(C)C)(CNC(C23CC(F)C2C3)=O)C1 45767,CC1CC(NC(=O)C(=O)N(C)CCO)CN1c1nnc(C(F)(F)F)s1 45768,N1(C(C(CCCC)C)=O)CCCC2CN(C(=O)CCC3NC(=O)NC3=O)CCC12 45769,C1(C)(C(N(CCC(C)(C)C)C)=O)CCCN1C(=O)CCc1ncnn1C 45770,C1(SC)CC(=O)N(C2CC2)C1.C12(OC)CC(C1)C1(NC(=O)C=C(C)Cl)CN(C1)C2=O 45771,c1(C(=O)NCCC(=C)CNC(c2cc(C#N)oc2C)=O)c(C)ccc(C)c1C 45772,N1(C(c2cn(C(C)(C)C)nc2)=O)CCN(C(c2nnsc2N)=O)C(CO)C1 45773,N1(CCCCCN(C)C(=O)OC(C)(C)C)CCN(CC(=O)OCCCO)CC1 45774,Cc1ccc2nc(C)c(C(=O)N(C3CCN(C(C4CC(Cl)(Cl)C4)=O)C3)C)cc2c1 45775,C1(NC(c2ccc(O)c(C(N)=O)c2)=O)CCc2cnnn2C1.CC12CN(C1)C(=O)O2 45776,c1(OC)ccc(NC(c2nn(-c3ccccc3)c(=O)cc2OC)=O)cc1[N+](=O)[O-] 45777,CC#CCCCC(=O)N(C1CCCCN(C(c2cn(CCC(C)C)nn2)=O)C1)C 45778,C1(CNC(C(C=CC)O)=O)CC(C)CCN1C(c1ccc(CN2CCCC2)o1)=O 45779,c1(C(CC(=O)OC)NC(c2c[nH]cc2C)=O)cccc2ccccc12 45780,C1(N(c2cncnc2Cl)C(Cc2n(C)ncc2Br)=O)CCC2(CC1)CNC2 45781,N1(C(=O)COC(F)(F)F)CC2C(C(=O)NC(c3ccncc3)CO)C2C1 45782,c1(CC(C(=O)C(O)Cc2ccccc2)=O)ccnc(O)c1.C1(N)CC(N)C1 45783,C1(NC(c2c(OC)nsc2)=O)CCC12CN(C(c1cscc1F)=O)C2 45784,C12CCC(CC1)C(=O)N2.c1(OC)nc(CC(N2CCC(C(F)(F)F)C2)=O)cs1 45785,N1(C(c2cncc(COC)c2)C(=O)NC(CC)C)CCN(C=O)CC1 45786,c1(CC(=O)NC2CC2C(N2CCC(CF)CC2)=O)ccc2c(c1)CC2 45787,N1(C(C2(N(C)C)CCC2)=O)CCN(C(c2ccn3nccc3n2)=O)C2(CCC2)C1 45788,N1(C(C2(CCCC)CCC2)=O)CCC2(CCCN(C(=O)CNC(=O)OC)C2)C1 45789,C(=O)(C(C(C)C)NC(=O)Cn1nnc(C)n1)N(C(CCSC)C)C 45790,Cc1cc(CCC(=O)NCC(CNC(=O)CC2C=CCC2)CO)on1 45791,C1(CC(C)NC(c2cc(F)n[nH]2)=O)CCN(C(C2(C)CC=CC2)=O)CC1 45792,C1(N(C(C2CCC(C(C)C)CC2)=O)CC)(CC)CCCN(C(=O)C(C)C)C1 45793,Cc1ccc(F)c(CC(=O)NC2CCC(NC(=O)C(F)C3CCC3)C2)c1 45794,C1(C(=O)NC2CCC(c3ccccc3)C2)(NC(COC(C)(C)C)=O)CCCC1 45795,N1(C(C)=O)CCC2(CCOCC2)C(NC(c2coc3c2C(=O)NCCC3)=O)C1 45796,c1(CC)ccccc1C(CNC(=O)C(C)(C)OC)NC(C1CC(OC2COC2)C1)=O 45797,C1(C(N2CC(CC(C)NC(C3=C(C)OCC3)=O)C2)=O)CCc2nc(O)[nH]c2C1 45798,CCCC(C)CCCC(=O)N1CC2(CNC(=O)C(C)CCc3ccccc3)CC1CO2 45799,c1(C(=O)NC2(CN(C)C(c3ccc[nH]3)=O)CC2)ccnc(Cl)c1N 45800,C1(NC(C2CCCN(C)C2)=O)COC2(C1)CN(C(c1ncnc(O)c1F)=O)C2 45801,c1(C(N2CCC3CN(C(C4C(C=C)OCC4)=O)CC32)=O)cnc2ccccc2n1 45802,c1(OC)cc([N+](=O)[O-])ccc1-c1ccc(CN(C)C)cc1 45803,C(=O)(C1=CCC(NC(=O)CN2CC3CC3C2)C1)NC(C(C)(C)O)C1CC1 45804,CCC(Cc1ccccc1)C(=O)NCC(C)N(C(=O)Cc1nncn1CC)CC 45805,N1(C(C2(C)CCC2)=O)C(CNC(=O)C=CC2CCC2)CC2COCC12 45806,c1(-c2cn(CC)c(=O)cc2)ccc2ccc(C(=O)Nc3ccc(Br)nc3)nc2c1 45807,CC#CC1CCN(C(c2ccc(OCCC)cc2C)C(=O)NCCCC)C1 45808,CC(CN=c1[nH]c(=NC(C)c2nc(O)n[nH]2)[nH]c2cc[nH]c12)c1cnc[nH]1 45809,N1(C(C2(C)CC(F)C2)=O)CC(CO)C2(C1)CN(C(C1CCn3ncnc3C1)=O)C2 45810,C(=O)(C(C)CC(F)(F)F)NCC1CC(OC)CN1C(c1c[nH]cc1C)=O 45811,C(=O)(CS(=O)(=O)CC(=O)OC)N1C(CNC(C(C=C)CC)=O)C(C2CC2)CC1 45812,c1(C(=O)NC(CCCCNC(C)=O)C)cnc2c(C)cnn2c1 45813,C1(NC(c2c(OCC)con2)=O)COCCC1NC(=O)CCCN(C)C(C)=O 45814,C1(CC)(CC)CCN(c2nnc(C3CCOC3)n2CC2CCOC2)CCO1 45815,c1(NC(c2ccc(C(N)=O)cn2)=O)cccc2[nH]ncc12 45816,c1(C(=O)NCC2(NC(c3c(C)coc3)=O)CCC2)cccc(N(C)C)n1 45817,N1(C(=O)CC2CCCOC2)CC2(CCCCN2C(c2c[nH]nc2C2CCC2)=O)C1 45818,c1(NC(c2c(C)nccc2)C)[nH]c(=NCC2CC2(Cl)Cl)nc2scnc12 45819,C1(NC(c2nccc(C)n2)=O)CCC2CCN(C(=O)C=Cc3ccc(C)o3)C12 45820,c1(NC(c2nc(COc3ccccc3Cl)n(-c3cccnc3)n2)=O)ccc([N+](=O)[O-])o1 45821,N(C(=NCCC(C)(C)S(C)(=O)=O)NCc1ccc(OC)cc1)N1C(C)CC1 45822,N1(C(C=CCOC)=O)CC(CNC(c2cnc(C3CC3)nc2)=O)OC(C)(C)C1 45823,c1(OC(C)C(=O)N(CC(C)NC(=O)CC2CCCCC2)C)cccc(Br)c1 45824,CC1(C)CC(C(=O)NCCC2CC=CCC2)CN1C(c1cnsc1)=O 45825,c1(C(=O)NC(CCOC)CNC(C2(C)CC2C)=O)ccc(Cl)c(C(=O)OC)c1 45826,c1(C(=O)NCC(C)CN(c2ccnn2CC(F)F)C)cnc2ccccc2n1 45827,N1(C(CSCC)=O)CCSC(C(=O)NCCc2nc[nH]n2)C1 45828,C1(CC(=O)NC(C)CC2CCCC2CNC(=O)C=Cc2nccs2)CCN(C)C1=O 45829,C1(NC(c2ncn(CC)c2)=O)CCN(C(c2ncsc2C(F)(F)F)=O)CC1(C)C 45830,c1(C(N2C(CCC)CN(C(c3coc(C)c3)=O)CC2)=O)cc2n(n1)C(C)CCC2 45831,C1(C(=O)NCC2CN(C(C(c3ccc(Cl)nc3)(C)C)=O)C2)CCOC(=O)N1 45832,C1(c2n(CCOC)nnn2)(NCCNC(C)=O)CCCC1CC1CC1 45833,Cn1cnc2cc(C(=O)NCC3CCCN(c4nnc(CCO)s4)CC3)cnc12 45834,C1(NC(C(C)N2CCC2)=O)CN(C(=O)Cc2ccno2)C2(CCOCC2)C1 45835,c1(OC)ccc2c(c1)C(CC(C)C)NC1=NCCCN21 45836,CN1CC(O)CCC1C(N1CC2CC2(C(=O)NCC23CCCC2C3)C1)=O 45837,C1(C(=O)Nc2c(CC)n(-c3ccccc3)nc2)CNC2(CCOC2)C1 45838,N1(C(=O)C(O)c2ccsc2)CCC(F)(C(=O)NCc2cn(C3CC3)nn2)CC1 45839,C1(CNC(c2ccc(O)nc2)=O)CC2(CCN(C(C3(CF)CC3)=O)CC2)CO1 45840,Cn1cnc2sc(C(=O)NCC(O)CNC(=O)CC3(O)CCCCC3)cc12 45841,c1(C(=O)NC2CC(C(N3CCC(F)C(F)C3)=O)C2)cc2ccc(Cl)nc2[nH]1 45842,N1(C(C(=O)NC2CC2)c2ncco2)CCOCC1c1cccc(F)c1 45843,C1(N(C(=O)OCc2ccccc2)C2CC2)CCCC(N)C1 45844,C1(CC=C)(NC(c2ncoc2C2CCC2)=O)CN(C(=O)Cc2ccnn2C)C1 45845,C(=O)(C1=C(CC(F)(F)F)N(C2CC2C)C(=S)NC1c1ccc(C#N)cc1)OC 45846,CC1CCC(OCC(=O)NC2(CNC(=O)C=Cc3ccco3)CCC2)CC1 45847,C(=O)(C1=C(C)CCC1)N1CC(OC)C(NC(c2cc3c(s2)CCC3)=O)C1 45848,Cc1ccccc1N1CC(C(=O)N(CCCNC(=O)CC(C)F)CCO)CC1=O 45849,C=CCC(C(=O)NC(C)C(CO)NC(c1cnn(C)c1C(=O)OC)=O)C(C)(C)C 45850,CC1(C)CCN(C(c2cc(C3CC3)on2)=O)C1CC(=O)NCC1CCC=CO1 45851,c1(CN2C(C)CCC(NC(c3cc(C(C)=O)on3)=O)C2)ccc(P(C)(C)=O)o1 45852,CCC(=O)CCC(=O)N1C(C(=O)N(CCN(C)C)C(C)C)CCC12CC2 45853,CC(C)CC(O)CC(=O)NCCC1(O)CC2CCC1CC2 45854,O=C1C(=Cc2cc(Cl)cc(Cl)c2)Cc2ccc(C(=O)O)cc21 45855,C(=O)(CCC(=O)NCC1CC(O)CN1C(=O)CCOc1cccc(Cl)c1)OCC 45856,c1(C(N2CCC(NC(C3CCN(C)C3)=O)(CF)C2)=O)cc(Cl)cc(C(F)(F)F)n1 45857,c1(C(=O)NC2CC(CNC(C(CC)(C)CO)=O)C2)cc(F)c(F)cc1Br 45858,CC1(CNC(=O)C(CNC(c2cccc(CO)n2)=O)N(C)C)NC(=O)NC1=O 45859,c1(CCN(C2CC3(CNC3)C2)C(=O)Cc2ccncc2O)ccccc1[N+](=O)[O-] 45860,c1(C(=O)NCCN(C(C(C(C)c2ccccc2)O)=O)C2CC2)cc(C#N)ccc1F 45861,C(CC(C(C)(C)C)NC(c1sccc1C)=O)N(C(C(CC#C)C)=O)C 45862,C(CCC(C)(C)C(=O)NCC(C)CCCO)NC(c1c(C)ncnc1)=O 45863,CCCS(=O)(=O)C(C)C(=O)NCC1COCCN1C(C1CN2CCN1C(C)C2)=O 45864,C1(NC(CNC(c2c(C)occ2)=O)=O)CN(C(=O)CCCCCSC)C2(CCC2)C1 45865,N1(C(CNC(=O)OC)=O)CCC2(CCCN(C(=O)Cc3ccn(C)n3)C2)C1 45866,c1(C(N2CC3C(CNC(C4(COC)CCCC4)=O)(C3)C2)=O)ccc2nn[nH]c2c1 45867,c1(C(=O)NCC2C3CN(C(c4scnc4C(F)(F)F)=O)CC23)ccnc(Cl)c1Cl 45868,C1(CN(C(C2CCN(C(=O)Cc3cncc(C)c3)C2)=O)CC)CCCC2(CC2)C1 45869,N1(C(C(C(C)C)NC(C)=O)=O)CCC12CN(C(=O)C(C)NC(=O)C1CC1)C2 45870,C1(NC(c2cc3sccc3[nH]2)=O)CC2(NC(C3CC4(C3)CC4F)=O)COC1C2 45871,C12(C(N3CCC(C)(CNC(=O)C(Cl)=CCl)CC3)=O)CC(C)(C1)OC21COC1 45872,C(=O)(C1CCc2nccn21)N1CCN(C)CC1C(=O)NC1CCCCCC1CO 45873,C#Cc1cncc(C(=O)NC2CCCC(N(C)C(C34COC(CF)(C3)C4)=O)C2)c1 45874,C1(NC(CS(CC)=O)=O)CCC2(CCN(C(c3ccnn3C(C)(C)C)=O)CC2)C1 45875,c1(OCC2C3CCC(F)(F)C23)ccc(C(C)NC2CC2)c(OC)c1 45876,N1(C(C(C)NC(C2CCCC2)=O)=O)CC2(CCN(C(=O)CCCN(C)C)CC2)C1 45877,CC(C(=O)NO)NC(C1CC(C)N1C(=O)CCC1CCC(=O)C1)=O 45878,N1(C(c2ncc(OC)nc2)=O)C2CCC1CN(C(C1CCC3(CCC3)C1)=O)C2 45879,C1(CNC(CCCCSC)=O)CCC2(CN(C(c3cccc(C)c3C#N)=O)C2)O1 45880,C1(C(=O)OC)C=CCCN1C(=O)CCC1(C)CN(C(=O)CCOC(C)C)C1 45881,C1(C(=O)NCC(C)(CO)NC(c2ccc(C)cc2)=O)CCCC2(CCC2)O1 45882,N1(C(=O)C=Cc2ccc(C(F)(F)F)cc2)CCOC2(C1)CN(C(c1cc[nH]n1)=O)C2 45883,CC(=O)CCC(=O)N1CC=CC1C(=O)NC1CCCCC1F 45884,c1(CCC(=O)NCC2(OC)CN(C(C3N(CCC)CCC3)=O)C2)cccc(O)n1 45885,C1(C(N(CCOC)CCNC(=O)C(CO)N(C)C)=O)CC2(C1)CC2(F)F 45886,c1(C(N2CCC(C)(CC(=O)OCC)C2)=O)cccc2sc(C(F)(F)F)nc12 45887,C(CCCCC(=O)NCC1(O)CCN(C(c2scnc2CC)=O)C1)OCC 45888,C1(NC(C2(C(=O)OCC)CC2)=O)CCC(CNC(C2C=C(C)CS2)=O)C1 45889,C1(NC(C2C(C)C2)=O)CCC2(CCN(C(c3ccc4cc[nH]c4n3)=O)C2)C1 45890,C1(C(N2CCN(C(CC(=O)NCC)=O)C(C(F)F)C2)=O)CC2OC(C)(C)OC2C1 45891,C12(C(=O)NC3CC4(CN(C(c5c(CC)cns5)=O)C4)C3)C3C4C1C1C2C3C41C 45892,C1(NC(C(C)O)=O)CCCN(C(C2CC2c2cccc(Br)c2)=O)C1 45893,Cc1cc(CCC(=O)NCC2(CNC(=O)CCCC#N)CCCCC2)n(C)n1 45894,N1(C(C2(C)C(C)C2)=O)CCC(C2CC2)(CNC(c2ccc3[nH]ccc3n2)=O)C1 45895,C(=O)(C(F)CC(CC)CC)N1CC(C#C)(F)C1.C123CCN(CCC1C2)C3=O 45896,N1(C(=O)CSc2n[nH]c(O)n2)CCC2CC2(NC(C2CC(CC3CC3)C2)=O)CC1 45897,c1(OC)cc(Br)ccc1C(CO)NC(=O)NCc1oc(C)cc1C 45898,NC(=O)CC(C(=O)NCC1CC(F)(F)C1)NC(=O)C(=O)NC1CC1 45899,c1(C(N2CC(CNC(C3C(OCC)C3)=O)(OC)C2)=O)c(O)nnc2c1COCC2 45900,c1(C2(C(=O)NC(C3CCCCO3)C#C)CCCC2)ccccc1Cl 45901,C1(NC(C2CC(=C)C2)=O)C(C)CCN(C(c2cnn(CC)c2C)=O)C1C 45902,C(=O)(C1=NNC(=O)CC1)N(C1CCCN(C(C(CC)n2cccn2)=O)C1)CCO 45903,c1(C(=O)NCC2C(C(=O)Nc3cnc(OC)nc3)C2)coc2c1COC2 45904,C(=O)(CCCC(F)(F)CO)NC1CC2CN(C(Cc3cncc(C#N)c3)=O)C1C2 45905,c1(OC(C)C)ccc(CC(=O)N(C2CCC(CNC(=O)CC(C)C)CC2)C)cc1 45906,c1(C(C)NC(C(C)SC)=O)ccc(CNC(=O)CCOC2CCN(C)CC2)cc1 45907,c1(CC)nc(=NC2CCCC(NC(=O)CC3CCC4(CCOCC4)CO3)C2)s[nH]1 45908,Cc1cc([N+](=O)[O-])c(C)cc1C(N1CC2CN(C(=O)CSC(=N)N)CC12)=O 45909,C(C(CNC(C1(F)CCC1)=O)S(C)(=O)=O)NC(C(COC)C)=O 45910,N1(C(c2c(C)[nH]cc2)=O)C(C(=O)NC(c2ccco2)CN(C)C)CCC1C 45911,O=C(C1CCCc2cncn21)NC1CC2(CCN(C(c3ccsc3Cl)=O)C2)C1 45912,c1(C(N2CC(OC)C3(C2)CCC3)=O)cc2c(nc1O)CCCCC2 45913,C1(C(N(C2CC(NC(c3c(CC)csc3)=O)C2)C)=O)C(C)(C)C1(F)F 45914,c1(C(=O)NCC#CCNC(CC2CCCC(C)C2)=O)c(F)cc(Cl)c(F)c1F 45915,Cc1cnncc1C(N1CC(C(N2CCC(CO)C2)=O)C(F)C1)=O 45916,c1(N2CCC(N(C)C(c3ccc(O)nn3)=O)C2)nnccc1C#N 45917,C1(C(=O)NCCC(CNC(CN(C2CC2)CC)=O)O)CCCC(C)(C)O1 45918,c1(OC)ccc(C(N2CCCC2CC(C)O)C(=O)NCC2CCCO2)cc1Cl 45919,c1(-n2c(-c3cnc(F)c(C)c3)nc(C(C)OCC)n2)c(C)cc(C)cc1C 45920,c1(C(=O)Nc2ccc(NCc3nccc(C)c3)nc2)ccc2nc[nH]c2c1 45921,c1(C(N2CCCC(COC)C2)C(=O)NC2CC(C(=O)OC)C2)nc(C)ccc1F 45922,C(=O)(C1CCCn2nccc21)N(CC(C)(C)C)C(CNC(C=CCCC)=O)C 45923,c1(NC(c2ccc(C(=O)Nc3cscn3)nc2)=O)cnccc1C1CC1 45924,c1(C(=O)NC2CCC(CNC(C(C)n3ccnc3)=O)C2)ccc(F)cc1N 45925,n1(CC(=O)NCCCN(C(c2cn(CC)nn2)=O)C)ncccc1=O 45926,C#Cc1cnn(C)c1C(N1CCC(F)(CNC(c2cncn2C2CC2)=O)C1)=O 45927,CC1CC(NC(C2CC(=O)NC(=O)C2)=O)CCN1C(=O)CCCn1cccc1 45928,c1(C(N2CCC(O)(C(C)NC(c3c[nH]c(Br)c3)=O)C2)=O)ccc2nc[nH]c2n1 45929,c1(CC(C)C(=O)N2CCCC2CN(C)C(c2cc(F)c[nH]2)=O)ccc(F)cc1F 45930,C(=O)(CCC(C)NC(C1CC1OC(C)(C)C)=O)N(CCN1CCCC1)CC 45931,C1(NC(CCNC(N)=O)=O)CCCN(C(c2cncc(O)c2)=O)CC1F 45932,c1(C(CC)C(=O)NC23CC(NC(=O)CC4CS(=O)(=O)C4)(C2)C3)c(C)noc1C 45933,C12(NC(C3C(C)CC(C)O3)=O)CC3CC(CC(C(=O)Nc4ccccc4)(C3)C1)C2 45934,C1(C(=O)NC2C(N(C)C)CC2)C=CCN(C(=O)C2=CCCC2)C1 45935,c1(C(=O)Nc2ccc(Nc3cc(C#N)ncc3)cc2)ccc2ccnc(O)c2n1 45936,C1(NC(=O)COc2ccc(F)cn2)CCCCN(C(c2ncc(F)cn2)=O)C1 45937,N1(C(c2c(C)nco2)=O)CCC(NC(=O)C(C2CCCN(C)C2)(C)C)C1C(C)C 45938,c1(C(N(C(C(=O)OC)C2CCC2)CC(F)F)=O)ccc2[nH]cc(C=O)c2c1 45939,c1(C(=O)NC2CCN(c3nnc(C(C)(C)C)o3)C2)cc2c(=O)[nH]ccn2n1 45940,O=C1COc2ccc(C(N3C4CN(Cc5ccccc5[N+](=O)[O-])CC34)=O)cc2N1 45941,C1(CNC(CCN(C(=O)CC2NC(=O)NC2=O)CC)=O)(CO)CC12CCC2 45942,CCCC(C(=O)N1CCN(C(C23CCCN(CC2)C3)=O)CC1C(C)C)C(C)C 45943,N1(C(c2cn(CC)nc2)=O)CC(C)CCC1CNC(=O)C(CC)(CC)OC 45944,c1(NC(C(=O)NC(C2CCOCC2)CC)=O)ccc(-c2ccc(F)cc2F)cc1C 45945,CC1(C)CN(C(=O)COC2CC2)C1C1CCN(C(=O)C=CC=C(Cl)Cl)CC1 45946,C(=O)(CS(=O)(=O)Cc1ccccn1)NCC(=O)NCCS(CC)=O 45947,N1(C(C(C)C2CCCC2)=O)CC2(C1)SCCC2NC(c1ccccc1O)=O 45948,CC(CCCNC(c1csc(F)c1)=O)NC(=O)Cc1ccc(Br)s1 45949,NC(CNC(c1ccccn1)=O)C(=O)N(C1CC1)C(c1cccs1)C 45950,C1(CC)CCCN(C(C2CCCS2)=O)C1C(=O)N(C)CC1CCCS1 45951,C1(CC)CCCCN(C(C23CC(CO2)N(C(=O)CCc2cn(C)cn2)C3)=O)C1 45952,Cc1cccc(C(C)N(C)Cc2cc[nH]c2)c1C 45953,C=CCCC(C(=O)NC1(COC)CC(O)C1)NC(=O)C=Cc1cscn1 45954,c1(C(N2CCC(O)(C(C)NC(COCCC)=O)C2)=O)cc(=O)n2nccc2[nH]1 45955,C1(C(=O)NCC(COC(C)C)O)CC(C)CN1C(C1CCCC(=O)C1)=O 45956,C1(OCC)CCN(C(=O)OCc2c[nH]nc2C(F)F)C(C)C1 45957,N1(C(c2ccc(CSC)o2)=O)CCC(C)C(N(C(=O)Cc2ncoc2C)C)C1 45958,CC1(C)OC2(C(c3ccc(Br)cc3F)N3CCC(Cc4nn[nH]n4)CC3)CC1C2 45959,C(CC(C(=O)NC1CCCN(C(c2csc(C(F)F)n2)=O)C1)OC)OC 45960,CC1(C)OC(=O)NC1C(=O)NC(c1cccc(Cl)c1)CNC(=O)CCC(N)=O 45961,c1(OC)c(C(=O)NC2CC(NC(=O)C(=O)NC3CCCCC3)C2)sc2nccnc12 45962,C=C(C)CC(C(=O)NC12CC(NC(=O)CNC(C3CC3C)=O)(C1)C2)OC 45963,N1(C(c2ncc(C)nc2)=O)CCC2(CC2)CC1C(=O)NCC1CCc2nccn21 45964,N1(CCCNC(C2(CCC(=O)OC)CCCCC2)=O)CCSC(C)(C)C1 45965,C1(C(=O)NCC(C)(C)Nc2nc(C3CCCC3)ns2)CCc2c[nH]nc2C1 45966,C(=O)(C(CC(F)F)NC(c1nc(C)ccc1C)=O)NCc1cccc(OC)c1 45967,C1(C)(CCC(=O)NCCCc2cn(C)nc2)CCCN1C(=O)CC(Cl)Cl 45968,C=C(C)CC(C(=O)N(C1CC2(CCC2)C1)C)NC(C1CCC(C)(C)CC1)=O 45969,C1(NC(=O)NCCn2ncc(C(C)(F)F)c2)CCCC(C2CC2)O1 45970,C1(CC(=O)NCC(c2ccc(F)cc2)NC(CC=C)=O)CCS(=O)(=O)CC1 45971,C1(CC(=O)N(CC(=O)NCCSCCC=C)CCC)CCC(=O)C1 45972,C1(C(=O)NC2CC(NC(c3cn(C)nc3Cl)=O)C2)COC2(CCC2)CO1 45973,c1(CC)ccc2c(Cl)c(C(=O)N(CC(CC)NC(C3(O)CCC3)=O)C)sc2c1 45974,CN1CCCC(C)(C(=O)NCCSCC(=O)NC2CC(=O)N(O)C2)C1 45975,c1(C(=O)OCC(=O)Nc2cc(C(C)C)c(O)cc2)cc(F)c(F)c(O)c1F 45976,c1(C2(C(=O)NCCNC(C3C=CCN3)=O)CC2)cccnc1 45977,N1(C(CC#C)=O)CCC2CCC(C1)N2C(c1ccc(Cl)cc1Cl)=O 45978,C1(CCCC)CN(C(C2(C)CCNC2=O)=O)CCN1C(c1nnn(CC)c1N)=O 45979,C(=O)(C(CC(C)C)N(C)C)NC1CC(N(C)C(c2sccc2C(=O)OCC)=O)C1 45980,c1(CC)cc(O)ccc1NC(C1CN(C(=O)C(C)CCNC(C)=O)C1)=O 45981,C1(NC(c2cc(Br)c[nH]2)=O)(CO)CN(C(c2ccnn2CC(F)F)=O)C1 45982,N1(C(c2cc(OC)cc(F)c2)=O)CC(C)CN(C(c2oc(SC)cc2C)=O)CC1C 45983,CCCCCCCCC(C)CC(=O)N1CC(CO)(NC(=O)C=CCO)C1 45984,C1(CNC(c2cc(OCC)ncc2)=O)CC2CCC1N2C(C1(C(F)(F)F)CC1)=O 45985,N1(C(C2C(C)C2)=O)CC(NC(=O)CCc2cnccn2)C2(CCS(=O)(=O)CC2)C1 45986,N(C(=NCCCCl)NCc1nnc(SC)s1)CC(CC(C)C)OC 45987,Cc1c(C(C)NC(c2cn(C3(C(=O)NC(=O)O)CC3)nn2)C)cccc1Br 45988,C=CCC(C)(CC)C(=O)Nc1cc(-c2ccc(CC)[nH]2)ccc1F 45989,C1(C(=O)OC)(NC(C2CCCN2Cc2nccn2C)=O)CCOC1 45990,C1(CC(=O)N(CC(N2CC(O)(CC=C)C2)=O)CC2CC2)CCC(=O)NC1 45991,c1(NC(C2(C)CN(Cc3cncnc3)C2)=O)ccc(F)c(F)c1Br 45992,C1(NC(=O)C(F)=C2CCC2)CCN(C(C2CC(O)(C(F)(F)F)C2)=O)CC1CO 45993,C1(NC(C2CC(C)(C)OC2(C)C)=O)CCCCC12CCN(C(=O)C1CC1)CC2 45994,C1(C(C)NC(C(C)=CC)=O)CCCCN1C(=O)C(=Cc1ccccc1)C 45995,c1(NC(C23CC(NCc4ccc(OC)nc4)(C2)C3)=O)c(F)cc(I)cc1[N+](=O)[O-] 45996,C1(NC(=O)COCCF)CC(NC(c2ccc(CO)cc2)=O)C(O)C1 45997,C12(CNC(C3CCCN3C3CCCC3)=O)CC(NC(c3cc(F)n[nH]3)=O)(CO1)C2 45998,c1(OC)nc(C(=O)NCC2(F)CC(CNC(=O)Cc3nc(=N)[nH][nH]3)C2)sc1C 45999,N1(C(C2CCC(C)O2)=O)CCC2CC(CNC(C3(CO)CC3)=O)CCC2C1 46000,c1(C(C(=O)NCCCC)N(C)C(c2cccc(Br)c2)C)c2c(nn1C)CCSC2 46001,C1(C(N2CCC(CC=C)(C(=O)NC(CC)CC)C2)=O)CCC2(CC1)CC2 46002,CCCCC(C)(F)C(=O)NC1CC(C)(NC(=O)C=Cc2ccccc2)C1 46003,Cc1ccc(OC(C)C(N2CC(CNC(C3(C#N)CCCC3)=O)C(C)C2)=O)cc1 46004,c1(CCC(=O)NC2CN(C(C(CC)CO)=O)CC2SC)ncnc2[nH]cnc12 46005,CC(C)CC(C)CC(=O)NCc1cn(-c2cc(COC)ccn2)nn1 46006,c1(OCOC)ccccc1S(=O)(=O)NC1CN(c2cc(C)nc(C)n2)C1 46007,N1(C(=O)NCc2cc(N)c(Cl)nc2)CCc2c(C3CC3)cccc2C1 46008,C1(C)(CNC(c2n(C=C)ncc2)=O)CN(C(c2nc(O)nc(O)c2F)=O)C(C)(C)C1 46009,CC(C)(CS(N)(=O)=O)C(=O)NC1CC(F)(CNC(C23CCCN(CC2)C3)=O)C1 46010,CCCCCC(F)C(=O)N(C)CC1CCCCN1C(C1CC(C)(C)CCO1)=O 46011,c1(OCC(N2C(CNC(C(CC=C)C)=O)CC(O)C2)=O)ccccc1[N+](=O)[O-] 46012,Cc1ccc(C(C)C(=O)Nc2nc(-c3[nH]nnc3C)no2)cc1 46013,N1(C(CCOC)=O)CCC(O)(CCNC(c2cnc(-c3ccccc3)s2)=O)CC1 46014,C(=O)(CS(=O)C(F)(F)F)NCC(C)(C)NC(C12CCC(F)(CC1)C2)=O 46015,c1(C(N2CC3(C(C(=O)NCc4cccnc4)C3)C2)=O)cccc2c(Br)ccnc12 46016,CCCC(C#N)C(=O)NC1(CC)C(OC)CC1OCC(F)F 46017,N(C1COCc2ccccc21)C(=O)C(c1cccnc1)Sc1ccc(Cl)cc1 46018,C1(CCC(=O)N(CC)CC2CC2)CCCN(C(c2ccnc(O)c2)=O)C1 46019,c1(OC)cc(C(=O)NCC2CCC2NC(c2cscn2)=O)cc2c1OCC2 46020,N1(CCC(=O)NC(C)(CNC(=O)C=C(Cl)Cl)Cn2cccn2)CCC(O)CC1 46021,CC1(C(=O)NC2C3CC4C2C4C3C(=O)NC2CCC(O)CC2)CCC(=O)NC1 46022,c1(SC)cc(=NCC2(C)CCCN(C(c3ccc(F)cc3F)C)C2)[nH]c(CO)n1 46023,CC1CC(C2CN(C(=O)C(CC(F)F)N(C(=O)CCc3nc(O)n[nH]3)C)C2)=NO1 46024,N(C(=NCCNC(=O)C1CC1)N1CC(C)N(CC(F)(F)F)C(C)C1)C(C)C 46025,CC1(C)C(CNC(=O)Cc2ccnc(F)c2F)CCN1C(C1CSC1)=O 46026,Cc1cc(=NC2CCN(C(=O)Cn3nnc(-c4cccs4)n3)CC2)[nH]c(CO)n1 46027,Cn1nc(C(N2CCC(C(N3CC(N4CC(O)C4)C3)=O)(CF)C2)=O)cc1C1CC1 46028,c1(C(=O)NCCOCC(C2CCCC2)O)csc2c(Cl)cccc12 46029,N1(C(c2c(CC)c[nH]n2)=O)CCN(C(C2CC2c2cnn(C)c2)=O)CC1C(C)C 46030,c1(C(=O)NC2CC(NCc3c(OC)nccc3)C2)ccc2c[nH]nc2c1 46031,C1(N(C(Cc2cc(C)no2)=O)C)CN(C(C2CC3COCC3C2)=O)CC12CC2 46032,N1(C(C(CC=C)C)=O)CC2(C(=O)NC3CN(C)NC3=O)CCC1CC2 46033,C(CCC1CCC1)(C(=O)NCc1cccs1)NC(C(C)n1ccnc1)=O 46034,Cc1cc(C(=O)NCC2CCCC2C(=O)NC(c2ncc[nH]2)C)ccc1O 46035,Cc1nc[nH]c1CN(C(=O)CCCn1cc(C(C)O)nn1)C 46036,Cn1cc(C(O)C(=O)NCCC2CCN(C(=O)CCc3nc[nH]n3)C2)cn1 46037,c1(C(N2C(C3(O)CN(C(CC=CC=C)=O)C3)CCC2)=O)cnc(C)c(C)c1 46038,C(=O)(C1OC(=O)c2ccccc21)NC(CN(C(=O)C=Cc1ccoc1)CC)C 46039,N1(C(CCOCC#C)=O)CC23CCCCC2(C1)CN(C(=O)C=CC1CCOC1)C3 46040,C1(C(N2CC(NC(C3C4CS(=O)(=O)CC34)=O)C2)=O)CC2COCC(C1)C2 46041,c1(C(=O)NC2CCN(S(CCCC)(=O)=O)C2)cc(Br)c(O)c(Br)c1 46042,c1(C(N2CCN(c3c(OCC)cccn3)CC2)=O)cccc2cccc(C)c12 46043,N1(C(CC(C)(C)C)=O)CCCOC(CNC(c2cnnn2-c2c(F)cccc2F)=O)C1 46044,N1(C(C2N(C(C)(C)C)CC2)=O)CC=CC1(C)C(N1CC(C(C)(C)C#N)C1)=O 46045,C(CCN=C(NCc1ncc(Br)s1)NC(C1CC1)C1CC1)c1onc(C)n1 46046,c1(CC(=O)NC2(CC)CCN(C(c3cncn3C)=O)CC2)cnn2ccccc12 46047,C(=O)(C(C)(C)CS(C)(=O)=O)NC1C(C)CCN(C(c2ncnc3sccc23)=O)C1 46048,c1(C(=O)NCCN2CCN(C(C3C(OC)(OC)CC3)=O)CC2)c(C)cccc1Cl 46049,N1(CC(N2CCC(CC(=O)NC(C)C(C)NC(N)=O)C2)=O)CCC(N(C)C)CC1 46050,C1(N(C)C(c2cc3n(n2)CCO3)=O)CN(C(c2c(O)cccc2O)=O)CC1(C)C 46051,n1(CC)nnc(C)c1C(c1nnnn1C1CCN(C)CC1)NCCc1ccccc1 46052,Cc1ccc(CC(=O)NC23CC2CN(C(C2(C)CC(C)=NO2)=O)C3)c(Cl)c1 46053,c1(C(N(CCC(C)NC(c2cnc(C(C)(C)C)nc2)=O)C)=O)ccc(C#N)cc1 46054,C1(NC(C(C)(Cl)Cl)=O)COC2(CCN(C(=O)COc3ccc(C#N)cc3)C2)C1 46055,c1(NC(N2CCC(N3CCC(O)C3)C2)=O)ccnc2ccc(Cl)cc12 46056,c1(C(=O)NCC2N(C(CNC(=O)OC)=O)CC(O)C2)cc(N)ccc1F 46057,C1(C(N2CCC(CN(C)C(c3cnc(N(C)C)s3)=O)C2)=O)CC12CCCCC2 46058,c1(C(=O)NC2(C)CC(NC(C3N(C(C)=O)CCC3)=O)C2)c(C)nn(C2CC2)c1Cl 46059,c1(C(=O)NC2CCN(C(C3(CCC)CC3)=O)CC2CO)n[nH]c2c1CCSC2 46060,C1(C(=O)NCC(C)N(C(C=Cc2cncc(C)c2)=O)C)(N(C)C)CCC(F)(F)CC1 46061,C(=O)(CS(=O)C(F)(F)F)NCC(C(=O)NCC(CCOC)(C)C)C 46062,c1(CC)ccc(C(=O)N(C(C)CN(C)C(c2ccc(CN(C)C)[nH]2)=O)C)c(C)c1 46063,C1(NC(C(C)N(CCC)C(c2cc(C(F)F)[nH]n2)=O)=O)CC2(CCOC2)C1 46064,Cc1noc2ncc(C(=O)NC3(C)CCN(C(c4cccc(Cl)n4)=O)CC3)cc12 46065,Cn1cc(C(=O)C(=O)NCC2(CC(=O)NCCCOC3CCC3)CC2)cn1 46066,N1(C(C(C)C2CCCC2)=O)CC(O)(CN(C(=O)CCCN(C)C)C)C1 46067,N1(C(CCSCC)=O)CC2CCN(C(c3ccc(OC)c(N)c3)=O)CC2C1 46068,N1(Cc2c(OCC)cc(F)c(F)c2)CCC=C(c2cccnc2)C1 46069,c1(C(=O)NCCN(CCC)C(C2CCNC(=O)C2)=O)cc([N+](=O)[O-])c(Cl)cc1Cl 46070,CC1CCC(O)(C(=O)NCCC2CCC(NC(c3ccc(F)cc3Cl)=O)C2)CC1 46071,c1(OC)ccc2[nH]cc(CCN3C(=O)CCN(CC4=CCCOC4)C3=O)c2c1 46072,c1(NC(C(=O)NCC2CN(C)C(=O)C2)=O)cccc2c1C(=O)NC2 46073,C(=O)(CCCC(C)C)NCC(CCCC)NC(c1scc(CC(=O)NC)n1)=O 46074,c1(C(=O)NCC2C(NC(CCC(C)(C)OC)=O)CCC2)cccc2ccnn12 46075,C1(NC(c2cnc(N(C)C)o2)=O)CC2CN(C(=O)Cc3ccncc3Cl)CC12 46076,CC1=C(C)CC(C)(C(=O)NC(C2(CNC(C3CC(=O)N(C)C3)=O)CC2)C)CC1 46077,CC1CCc2c(C(=O)NC3CC(NCc4ccc(C(F)(F)F)c(Cl)c4)C3)n[nH]c21 46078,O=C(C1=CCCSC1)NCCC1CN(C(C23C=CC(CC2)C3)=O)C1 46079,c1(OC)cc(NCC(=O)OC2CCC2)ccc1Cl 46080,N1(C(CNC(CN(C)C)=O)=O)CCN(C(C2CC(C)(C)C2)=O)CC1C1CC1 46081,c1(OC(C)(C)C)cnc(C(ONC(=O)OC2CCCC2)=O)cn1 46082,c1(OCC)nc(C#N)cc(=NC(=O)CC2CCC(C(F)(F)F)O2)[nH]1 46083,c1(CCC#C)ccc(C(C)C(N2CCC(CN(C(=O)COC(F)F)C)C2)=O)cc1 46084,c1(C(=O)NCC2CCC(NC(C3(OC(C)C)CCC3)=O)C2)cnc2c(C)cccn12 46085,CC1(C)CCC(F)(F)CC1C(=O)NC12CCCC1N(C(=O)C(F)(F)CO)CCC2 46086,C1(CNC(C(C)NC(C)=O)=O)C2CC1N(C(c1csc(-c3cnccn3)n1)=O)C2 46087,C(C(C)(O)CC(=O)N1CCC1(C)CC(=O)NCC(C)(O)COC)OC 46088,N1(C(c2cc(CC)oc2C)=O)CCCC2(NC(c3cn[nH]c3)=O)CCCC12 46089,Cn1cc(C(=O)NC2CC(NC(=O)Cc3ccncc3)C2)c2ccccc12 46090,C(=O)(C(CC(C)(C)C)OC)NCCCC1OCCN(C(CNC(COC)=O)=O)C1 46091,c12cccc(c1F)CC1CC(C1)NC2=O.c1(CC)ocnc1C(=O)NCC1CCC1 46092,C1(NC(c2[nH]cc(COC)c2)=O)CCN(C(c2nc(C)c(C)s2)=O)CC1C(C)C 46093,Cc1cc(C(N2CCC(OCCNC(=O)Cn3cccc3)C2)=O)nn1C(C)C 46094,c1(C(N2C(C)(C(=O)NCCc3cnc(C)o3)CC(O)C2)=O)cc2ccccn2n1 46095,C1(C(=O)NC(CCCNC(C(CSC)OC)=O)(C)C)Cc2cc(Br)cnc2C1 46096,C1(C(N(C2CCN(C(C3CC34CCOC4)=O)CC2)C)=O)CC(O)CN1C 46097,C1(CNC(C(C)O)=O)CCC(F)(CNC(c2ncccn2)=O)CC1 46098,N1(C(C2(C)CCNC2=O)=O)CCCC(NC(=O)CSCc2ccccc2)CC1 46099,C1(CNC(c2[nH]cc(C(C)=O)c2)=O)CCN(C(c2cccc(=O)o2)=O)CC1C 46100,c1(C(N2CC(NC(c3cc(CCOC)on3)=O)C(F)C2)=O)nc(C)c(C)nc1C 46101,c1(C(=O)NCCCC(C)NC(=O)CC(C)C(F)(F)F)cnn2c1OCC(F)C2 46102,CCCCC(CN=c1[nH]nc(C(C)(C)C)o1)NC(=O)CC1C=CCC1 46103,c1(C(=O)NC2CN(C(C3CCC(COC)O3)=O)CC2C)cccc(Cl)c1O 46104,c1(CC(=O)N(CCCN(C(=O)C(F)C2CCC2)CC)CC)ncoc1C 46105,C(=O)(C1CCc2nccn21)N(CC(C)NC(C(n1c(C)ncc1)(C)C)=O)C 46106,Cc1[nH]c2ccc(Br)cc2c1CCNC(=O)Cn1cc(Br)c(=O)c(I)c1 46107,C=C(C)CC(C(=O)NC1(C(N2CC3C(CN(C)C)C3C2)=O)CCCCC1)OC 46108,Cc1cccc(F)c1C(=O)NC1CCC(NC(C2(F)CC=CC2)=O)C1 46109,C(C(C(=O)NC(Cc1ccco1)CO)N(C)C)NC(C(C1CCC1)OC)=O 46110,Cc1cnc(CNC(C2CN(C)CCN2C(=O)C(F)C(C)(F)F)=O)c(C)c1 46111,c1(C(=O)NC2CCS(=O)(=O)C2)n[nH]c2ccccc12.c12n[nH]cc1C(=O)N2 46112,C1(NC(CCSCCC)=O)CN(C(c2c(C)noc2CC)=O)CCC1CO 46113,N12CCC(C1)N(C(=O)CN1CC3CC3C1)CC2=O.c1(CSC)ncccn1 46114,C1(C(N2CCC(C(C)(C)O)C2)=O)(CNc2scnc2Cl)CCOCC1 46115,C1(CNC(c2n(CC)ccc2)=O)CN(C(C23CCC(CC2O)C3)=O)CCN1C 46116,C(=O)(CC(C(F)(F)F)N(C)C1CC1)NC(C)CCNC(=O)C1=CCCOC1 46117,C(=O)(CCCS(C)(=O)=O)N1CCCC(C)(NC(=O)CCn2cncn2)C1 46118,n1(CC)nc(C(C)C)cc1C(=O)NCCN(C(=O)CC(CC)=C(C)C)CC1CC1 46119,C1(CCOC)CCCCN1C(C1CN(C)NC1=O)=O 46120,c1(C(=O)NCC(CC=C)NC(c2cn(C3CC3)cn2)=O)cn(C)nc1Br 46121,C(=O)(C1=NOC(CC2(O)COC2)C1)NC1(CN(C(c2c(SC)csc2)=O)C)CC1 46122,c1(C(=O)NCCC2N(C(C(CC)SC)=O)CCC2)coc2c1CCCC2 46123,C(C(CC(C)C)NC(C1C(C)CCN1C(C)=O)=O)NC(c1cc(OCC)no1)=O 46124,CC(C(CO)NC(C1CCCS1)=O)NC(c1cc(Cl)ns1)=O 46125,c1(OCC)cc(C(=O)N(CC(CC)NC(=O)C(C)CC)C)ccc1C(F)F 46126,CCC(CC(=O)NC(C)CN(C(=O)COCC1(F)CC1)C1CC1)OC 46127,C1(C(=O)NCC2CCN(C(=O)CC34COCC(C3)C4)C2)C2CCCCCC12 46128,C1(C(C)NC(=O)C=CC(=O)NC2CC2)CCCCN1C(C1CC2CC1C2)=O 46129,c1(C(=O)NC(C)C(C)(C)NC(c2ccn(CCO)c(=O)c2)=O)cc(O)cc(O)n1 46130,CCCCC(CC(=O)N(C(CSC)CC)C)NC(=O)C=C1CCOCC1 46131,C(=O)(CC1COCc2ccccc21)NC(C1CN(C(=O)CCCF)CCO1)C 46132,C(=O)(CCCC(C)(C)C)N(C)CCNc1ncccn1.C12CCN(CC1)C2=O 46133,N1(C(CCC=CC)=O)CCCCC1CNC(c1cnc(C)s1)=O 46134,C(C)(C(C)(C)C(=O)NCCC1(SC)CCC1)NC(c1cn(CC=C)nc1)=O 46135,C1(CN(C(=O)C=C(C)C(F)F)CC)CCCCN1C(c1cn(C)nc1SC)=O 46136,C(C(C(C)(C)C)NC(c1cc(Cl)c(Cl)[nH]1)=O)NC(C=C1CCC(C)C1)=O 46137,N1(C(c2ncccc2F)C(=O)NCc2cccc(OCC)c2)CCOCC(C)C1 46138,C(=O)(C(F)C(C)(C)O)NC1C=CCN(C(COCc2ccc(C)cc2)=O)C1 46139,C1(CNC(C2N(CC)CC2)=O)CN(C(c2c(Cl)c(C)nn2C)=O)CCC1(F)F 46140,S(=O)(=O)(c1ccccn1)NCCNCC1COCC1C1CCN(C(COC)=O)CC1 46141,N1(C(C=CSC)=O)CC(C(F)(F)F)OC(CNC(c2cnc(C)cn2)=O)C1 46142,c1(CC)ncncc1C(=O)NCC(C1CCC1)N(C(C1CCN1S(C)(=O)=O)=O)CC 46143,C#Cc1ccccc1CN=C(NCC(F)F)NCC1(OCC)CCOC1 46144,N1(C(C2(CCOC)CC2)=O)CC=CC(NC(C23CCCC2(C(N)=O)C3)=O)C1 46145,C1(NC(Cc2cc(C)nn2C)=O)(CNC(C2C=CCS2)=O)CC2CCC1CC2 46146,CC(C)CCCC(=O)N(C1CCN(C(C2CC(C)CCC2C(C)C)=O)C1)CCO 46147,c1(CC(=O)NC(C)CCNC(=O)Cc2cccnc2F)c(F)cccc1F 46148,C(=O)(CCCS(C)(=O)=O)N1CC(CC)C(NC(c2cc(C(C)(F)F)on2)=O)CC1 46149,N1(C(c2sc(C)c(C)c2C)C(=O)NCCOC)CC2CCC(C1)C2O 46150,N1(C(c2cnc(C)o2)=O)CC(NC(=O)C(C)Cn2ccnc2)C2(CCCC2)C1 46151,NS(=O)(=O)c1ccc(C(=O)NCc2ccccc2C(=O)NO)cc1 46152,C1(C#N)(C(N(CCCNC(c2cn(C)cc(Br)c2=O)=O)C)=O)CC12CCCC2 46153,C1(C(=O)NCC2(COC)CN(C(c3nccnc3N)=O)C2)C2CC3C(C2)C13 46154,N1(C(C=CC=CCOC)=O)CC2CCN(C(C3(N4CCOCC4)CC3)=O)C2C1 46155,CCC(CC)(C(=O)NCC1(C)CCCC1NC(=O)CSCCC(C)C)OC 46156,C(N=c1[nH]nc(C(F)F)s1)C1(NC(c2cc(C(F)(F)F)on2)=O)CCCCC1 46157,c1nc2ccccc2n1CCN(C)C.C=C1CC2(C1)C(=O)NC2.C(=O)OC 46158,c1(C(=O)NCC2CCCN(C(C(C(=O)OCC)F)=O)C2)ccnc2nc(C)nn12 46159,CCCC(C)C(=O)N1CCC(N(C(=O)CCC#N)CC2CC2)C1 46160,CCCCCCC(=O)N1CCC(O)C(C(=O)NCc2csc(-c3cnc[nH]3)n2)C1 46161,C1(NC(c2ccc(C(C)=O)nc2)=O)(CO)CCCN(C(=O)Cc2ccsc2Cl)C1 46162,c1(C(=O)NC23CC(CNC(c4c(C#N)nc[nH]4)=O)(C2)C3)cc2cc(F)ccc2s1 46163,C1(C(=O)NC2CCCN(C(COCCCOC)=O)CC2)Cc2ccccc2S1 46164,c1(C(N2CC(O)(C(=O)NCC3(NC(CCC#C)=O)CC3)C2)=O)cccc(F)c1C 46165,c1(CC(=O)OC)nc(=NCCOCCN(C(=O)C(N2CCCCCC2)C)C)s[nH]1 46166,C(C)(C)(CN=c1[nH]c2cc(Br)ccc2o1)NC(Cc1c(C)noc1Cl)=O 46167,c1(CC(=O)NC2(CCCNC(C3C(C)(C)C3(C)C)=O)CC2)ccc(F)c(Cl)c1 46168,O=C(N=c1[nH]c2sc(-c3ccccc3)cc2s1)C1CC1NC(C1CCC1)=O 46169,CC(CNS(=O)(=O)c1c(F)cccc1F)C(=O)NNC(=O)C(F)(F)F 46170,C#Cc1cnc(C(N2CCC(C(=O)NCC3(C(F)(F)F)CC3)(CF)C2)=O)c(C)c1 46171,C#CC1(C(N2CCC(O)(C(C)NC(=O)CCCN3CCOCC3)C2)=O)CCCC1 46172,N1(C(=O)C=CC(F)(F)F)CCOC(C2CN(C(=O)C=Cc3ccco3)C2)C1 46173,C1(C(N2CCC(CCC)C2)=O)CSCCN1C(C1CCC(OC)CC1)=O 46174,C(=O)(C1=CNC2=NCCC2=C1)N1CCN(C(COCCOC)=O)CC1CO 46175,c1(N2CCCC(C)(CNC(c3n(CCC)ccc3)=O)C2)ncnn2cccc12 46176,C1(CC)CCC(C(=O)NC23CC(NC(c4cc(CC)on4)=O)(C2)C3)O1 46177,C(c1ccc(S(=O)(=O)NC)cc1)=CC(=O)NCCN(C(CC=CC)=O)CC(C)O 46178,Cc1nn(C)c(C(F)F)c1C(=O)NCCNC(C12CCCC1CCC2)=O 46179,CCCS(=O)(=O)N1CCCC1C(=O)NC1(CCCCNC(C2CCOC2C)=O)CC1 46180,C1(C(=O)NCCOCC(=O)NC)CCN(C(C2CCCC(C#N)C2)=O)CC1C 46181,c1(CC)ccc(F)c(NC(N2CCC(F)(c3ccccc3)C2)=O)c1Br 46182,N1(Cc2ccc(COC)s2)CCCCC(NC(c2cccc(=O)n2C)=O)C1 46183,N1(C(CCCNC(=O)OC)=O)CC2(C1)CN(C(=O)CC1CC(C)(C)CO1)C2 46184,C1(NC(CCc2cnc(C)s2)=O)C=CCN(C(C2C(C)(C)C2(F)F)=O)C1 46185,c1(CNC(C2C(O)CCN(C(CCC=C)=O)C2)=O)ccc2nc[nH]c2c1 46186,N1(C(c2cnc(C)n2C)=O)CCC2(NC(=O)Cc3cncnc3)CCCC12 46187,N1(C(C(C)CN2CCOCC2)=O)CCC(C)(CNC(C2(C3CC3)CC2)=O)CC1 46188,N1(NC(N(C)C)=O)C(=O)C2C3CCC(O3)C2C1=O.C123CC(CN1C2=O)C3 46189,C1(NC(=O)CCCC2CCOCC2)C2CC1N(C(C1CC(CC3CC3)C1)=O)C2 46190,C1(COC)(CNC(c2cc(O)nn2C)=O)CCN(C(C2CC(O)CN2C)=O)C1 46191,c1(C(=O)NC2CCCC(C#C)C2)coc2c1CN(C(=O)CC1CCC(=O)N1)C2 46192,C1(C(NC(c2c(CNC(c3c[nH]nc3C3CC3)=O)occ2)=O)C2CC2)CC12CCOC2 46193,C(=O)(C(C(C)(C)C)C1CC1)NC(CCCNC(CCc1c(OC)cccc1)=O)C 46194,C1(C(N(CCNC(=O)CC2COC3CC2C3)CC)=O)(OC)CCCCCCC1 46195,C1(N(C)C)CN(C(C2CC3CC3N2C(=O)CCCN2CCOCC2)=O)CCO1 46196,c1(C(=O)NCCCNC(c2c(F)ccc(CC)c2)=O)cc(S(N)(=O)=O)ccc1F 46197,Cn1ccnc1CC(N1CCC(OCC(=O)NC2COCC2N(C)C)C1)=O 46198,N1(C(CCc2ccc(C)o2)=O)CC(CNC(c2scc(C)c2Cl)=O)CC1C 46199,C1(NC(C2C3(CC(OCC)C3)C2)=O)CCN(C(c2ccncc2C)=O)C(C)C1 46200,C1(C(=O)NCC2(C(C(C)C)O)CC2)CCC=CCC1 46201,c1(C(N2CC=CC23CCC3)C(=O)Nc2cccc(OC)c2)cccc(C#N)c1 46202,c1(C(=O)NCC2CCN2C(c2cc[nH]c3nccc2-3)=O)cc(F)c(F)c(Cl)c1F 46203,c1(C(N(C2CN(C(C3CN(C(N)=O)C3)=O)CC23CC3)C)=O)n[nH]c2ccc(F)cc12 46204,C(N=c1[nH]c2cccc(F)c2s1)C1(C)CCN(C(c2cc3n(n2)CCCC3)=O)C1 46205,CCC(C)(C)CCCC(=O)NC1CN(C(=O)C(COC)N(C)C)CCC1(C)C 46206,CC1(CNC(c2ccc3ncc(Br)n3c2)=O)COCC2CCCN12 46207,C(c1ccc(OCC(=O)NC2CNCC23CCC3)c(OC)c1)=CC 46208,C1(c2cn(Cc3cnn(CC)c3)nn2)(C(=O)OCC)CCOC1 46209,C12(C(=O)NCCOCCCNC(C3CC(OC)C(O)C3)=O)CCC(CO)(CC1)C2 46210,N1(C(C(CSC)(C)NC(=O)COCC(F)(F)F)=O)CC2CCN(C)C2C1 46211,c1(NC(N2CCC(CNc3ncccc3Br)CC2)=O)ccc(-n2cnnn2)cc1 46212,C(C)(C)(CC(C)NC(=O)CCN(C(c1ccc(C)s1)=O)CC1CC1)OC 46213,c1(CC(N2C(C)CN(C(c3csc(O)n3)=O)C(C)C2)=O)ccc2c(c1)CCN2C 46214,C1(N(C)C(c2cnc(N(C)C)s2)=O)CCCN(C(C2(C#N)CCOC2)=O)CC1 46215,N1(C(COCCC=C)=O)CCC(CNC(c2cnc(CC)nc2O)=O)C(C)C1 46216,c1(CC(=O)NC2C(C)(C)CN(C(=O)C(F)F)CC2)ccc(O)c([N+](=O)[O-])c1 46217,C1(O)(NCCCCCNC(COCC(=O)NC)=O)CCN(C(C)=O)CC1 46218,N1(C(C(CCC)F)=O)CC2CC(C)N(C(c3ccnc(OC)n3)=O)C2C1 46219,c1(C(N2C(CNC(c3ccc(F)cn3)=O)CC3CC32)=O)cccc(Cl)c1Cl 46220,CCC(CC)(CO)C(=O)NCC(C)(F)CNC(c1ccc(N)cc1F)=O 46221,Cc1cc(C(N2CCN(C(=O)Cc3cnsc3)C3CC23)=O)c(C)nc1C 46222,C#CCC(C)(C)C(=O)NC1CCCCC1NC(=O)Cc1ccsc1C 46223,c1(CC)nn(C)c(CC)c1CNC(c1ccc(F)cc1)c1nnnn1C1CCCC1 46224,N(C(=NCC1CC(CC2CCCCC2C)C1)NCC(C)(C)C)C(C)C 46225,C1(Cn2cc(CS(C(C)C)=O)nn2)CCN(C(C2C3CN(C(N)=O)CC23)=O)CC1 46226,Cc1cc(=NCC2CCN2)[nH]cc1S(=O)(=O)NCC(O)CF 46227,c1(C(=O)NCC=C(C)C(C)C)ccc(Cc2ccccc2OC(C)C)cc1 46228,c1(SC)ncc(C)c(N2CCC(C(=O)Nc3c[nH]nc3C#N)C2)n1 46229,C(CCCC(=O)N1CC(C(=O)NC(c2ccccn2)C)CCC1C)(OC)OC 46230,Cc1cc(CNC23CC(C(=O)Nc4ccc(F)cc4Cl)(C2)C3)c(O)c(Br)c1 46231,C1(C(=O)NCC(C2CCC2)NC(=O)CC2CCCC2)CCN(C)S1(=O)=O 46232,C(=O)(CCC1=CCCCC1)NC(c1ccccc1)C(=O)NC1CN(C)CC1(F)F 46233,C1(N(S(c2c(C)onc2)(=O)=O)C)CCc2ccccc2C1 46234,C(=O)(C1=NOC(CNC(c2cncc(O)c2)=O)C1)NC(C#C)C1CCC1 46235,CC(C)(CC(F)(F)F)C(=O)NCC1CN(C(C2CCc3nccn3C2)=O)CC1O 46236,N1(C(C(=O)NCCc2cccc(C(F)(F)F)c2)=O)CCCC2(CCCNC2=O)C1 46237,N(C(=NCCn1cccn1)NC1CCS(=O)(=O)C1)C(COCC)CC 46238,N1(C(c2cc(C)no2)=O)CC(C)(C)CC1CNC(c1nccc(C)c1F)=O 46239,C1(NC(=O)CCOC2CCC2)CCN(C(C23CCC(C2)C3)=O)CC1O 46240,c1(C(=O)NCC2C(C)(C)N(C(=O)CC3CCCO3)CC2)cnn2cccnc12 46241,Cc1cccc2cc(C(N3CCCC3NCCOc3cccc(Br)c3)=O)cnc12 46242,CC#CCS(=O)(=O)c1cccc(C(=O)NCC=CCNC(=O)CCC(C)(C)OC)c1 46243,c1(NC(C2CSCCN2c2ccncn2)=O)cc(Br)cc2cn[nH]c12 46244,C12(NC(C(C3CN(C(=O)C#CC4CCC4)C3)OC)=O)CCC(CC1)C2(C)C 46245,C1(C(N(CC(C)O)CCNC(C2CC=CC2)=O)=O)CCOC(=O)N1 46246,C1(N(C(=O)C(C)C2CC2)CCNC(COCC(=C)C)=O)CC(C#N)C1 46247,Cc1c[nH]nc1C(=O)NC(CO)C(=O)N1CCCC1 46248,C(=O)(CCC1CCc2ccccc21)N1CCN(C(c2c(C)scc2)=O)CC1CF 46249,N1(CC)N=C(C(=O)N2CCCC2CCNC(=O)Cc2nnc(C)o2)CCC1=O 46250,C(=O)(C(CC1(C)CCOC1)N1CCC(C(=O)NC)C1)NCC(=C)C 46251,Cc1cc(C(=O)NC(C2CCCN2C(=O)C=CC2CCOC2)C)c(Cl)cc1Cl 46252,c1(C(=O)NC2C(NC(COCCOCC#C)=O)CCC2)cnn(C)c1C(F)(F)F 46253,CC(C)(C)S(=O)Cc1cccc(CNC(C2CCCCC2)=O)c1 46254,N#Cc1c[nH]c(-c2nnc(N3CCC(F)C3)n2CC(N2CCCC2=O)C2CC2)c1 46255,c1(C(=O)NCCCN(C(C(C)OCC=C)=O)CC)cccc2c1CNC2=O 46256,CCC1CN(C)c2ccccc2CN1C(=O)C(=O)Nc1cc(Cl)ccc1OC(F)F 46257,CCC(COC)C(=O)NCC(C)N(C(c1sc(C)nc1-c1ccccc1)=O)CC 46258,N1(c2nccc(Br)c2Br)CCC2CCCCC2C1 46259,CCC(C)CC(C(=O)Nc1cnc(SC)nc1)NC(=O)Cc1ccsn1 46260,c1(NC(C)C)ccc(C(N2CCC(C(C)NC(=O)CC3CCC(=O)N3)C2)=O)cn1 46261,CC(CCNC(=O)CCC1CCN(C(=O)Cc2cc[nH]n2)CC1)C(C)(C)C 46262,C1(NC(c2cc(OC)no2)=O)CC(CC(=O)Nc2c[nH]ccc2=O)C1(C)C 46263,c1(OCC)ccc(C(=O)NCCC2CN(C(C3(O)CC(C)(C)C3)=O)CC2C)cc1 46264,CC1CCOC(C(=O)NC(CC(F)(F)F)c2ccccc2)C1 46265,Cc1cc(C#N)cc(C)c1C(=O)NC1CCN(C(C2CCCC2)=O)CC1O 46266,c1(N(CC(N2CCCC2C(N2CCNC(=O)C2)=O)=O)C)ccc(F)cc1O 46267,c1(OC)ccc(C(=O)NCC(C(C)C)NC(=O)CC2C(C)C2(F)F)c(C)c1 46268,Cc1ccc(Br)c(NC(C2CCC(NC(c3cccc(C)c3O)=O)C2)=O)c1 46269,N1(C(C2CC2NCc2c[nH]nc2-c2ccccc2)=O)CCN2CCCCC2C1 46270,N1(C(c2cc(SC)oc2C)=O)CCC2(CCCN(C(=O)C(F)=C3CC3)C2)C1 46271,Cc1nn(C)c(C)c1C(N1CC(NC(=O)OCc2ccccc2)C(F)(F)C1)=O 46272,O=S(=O)(c1[nH]c(=NCC2C(F)(F)C23CCCC3)ccc1Br)NC1CC=CCC1 46273,Cc1cc(C(=O)NC2CC(NC(c3scnc3CCC(F)(F)F)=O)C2)no1 46274,C1(CN(C(=O)C(c2cccs2)NC(=O)C(=O)NC)CCC)CC1(C)C 46275,c1(C(N2CCC(CNC(C(CC3CC3)OC)=O)C2(C)C)=O)cccc2ccnn12 46276,c1(C(=O)NC2CC(C)(NC(=O)CC3CC3c3ccccc3)C2)ccc(F)cc1Cl 46277,N(C(=NCC#Cc1ccccc1)NC1CCCCC1)CC1(CO)CC(C)(C)OCC1 46278,O=C(N=c1cc[nH]cc1O)C1CCCN1Cc1ccc(-c2ccccc2)s1 46279,C1(C(=O)NC(CN(C)C)CO)(NC(=O)Cc2cnn(C)c2)CCN(C)C1 46280,N1(C(C(C(C)O)(C)C)=O)C2CCC1CN(C(=O)CC13CCCN1CCC3)CC2 46281,C1(C(N(C2(C(N3CC(CN4CCOCC4)C3)=O)CC2)C)=O)CCC2CC1CO2 46282,CC(C)(C(O)C(F)F)NC(C1CCCC1CNC(C1(n2cccc2)CC1)=O)=O 46283,Cc1cc(=O)oc(C)c1C(=O)NCC(CC(C)C)NC(C12COCC(C1)C2)=O 46284,CCCC(CCC)C(=O)NC1CC(CNC(c2cc(C)nnc2CC)=O)C1 46285,C#Cc1ccc(C(=O)NCC2CCCN(C(c3ccn(CC#N)n3)=O)CC2)cc1 46286,c1(C(C)NC(C(n2cc(-c3c(C)cccc3F)nn2)C)=O)ccc(S(C)=O)cc1 46287,C1(C(N2CCC(O)(CC)CC2)=O)CN(C(=O)Cc2cccc(F)c2)CCC1(C)C 46288,N1(CC(=O)NC(C(=O)N(CCCOCC)CC)C2CCCO2)CCC(=O)CC1 46289,Cc1nc(C)n(CCc2cn(CC(=O)N(C3CCC3C(F)(F)F)C3CC3)nn2)n1 46290,N1(C(c2ccn(CC)n2)=O)CC(OC)CC1CNC(c1sccc1Cl)=O 46291,N1(C(c2c(C)ccnc2O)=O)CCCCC(NC(c2cn(C)nn2)=O)CC1 46292,C(=O)(CC1CCOc2ccccc21)NCC(CNC(C(C=C)(F)F)=O)(C)OC 46293,N1(C(C(c2ccc(F)cc2)C)=O)CC2CC1C2NC(=O)CS(C)(=O)=O 46294,CCC(CC(=O)N1CCC(CN=c2nc(SC3CCCC3)[nH]s2)CC1)C(F)F 46295,C1(CC)(NC(=O)C(c2ccc(F)cc2)O)CCN(C(c2nnc(S)n2C)=O)CC1 46296,Cc1c(C(=O)NCC2CC2CNC(=O)C(F)(F)c2cncs2)cnn1CC(F)F 46297,c1(CN(C(C(=O)NC2CCCCC2)C2CCSC2)C)ccc(-c2ccccc2)o1 46298,N(C1CC2(CN(C(c3ccnn3C)=O)C2)n2ccnc21)C(CC(=O)NCC#C)=O 46299,C(=O)(CC(O)C(C)C)NC1CCC(CC(=O)NCc2cc(C)ncn2)CC1 46300,c1(SCC(N2CC(CNC(C3C(CC)OCC3)=O)C2)=O)ccc([N+](=O)[O-])cc1 46301,Nc1ccnc(C(N2CCC(F)(CNC(=O)CC3CSCCS3)C2)=O)c1Cl 46302,CCCCC(C(=O)NOC(C)CC)NC(c1nonc1N)=O 46303,c1(CC)n[nH]c(=NC(CCN(C)C(C2CCCN(C(C)C)C2)=O)C(C)C)o1 46304,N1(C(c2c(C)csc2)=O)C(C(N)=O)CCC1C 46305,C(=O)(C1CCCc2scnc21)NC1C(C)CN(C(c2csc(C(N)=O)c2)=O)C1 46306,c1(C(C)C)nccc(C(N2CC3C(CNC(=O)CN4CCCS4(=O)=O)C3C2)=O)n1 46307,c1(C(=O)NCC2C(C=C)CN(C(=O)COCCC)C2)cc(S(N)(=O)=O)c(C)s1 46308,c1(C(N2CCC(F)(C(=O)NCCn3cnnc3)C2)=O)cc(O)nc(C2CC2)n1 46309,N1(C(C=C(C)CNC(C2CCC(C)(C)C2)=O)=O)CC=C(CO)CC1 46310,CCC(C)CCCCC(=O)NCC(CC1CC1)C(=O)N1CC(C)C(F)C1 46311,C(CC(C)C(C)C)NC(C(CN(C)C)NC(Cc1scc(C)c1)=O)=O 46312,c1(C(N2CC(NC(c3cscn3)=O)C(F)C2)=O)cc2nc(Cl)ccc2o1 46313,N1(C(C2C(=C)C2)=O)CCn2c(CNC(C3C(Cl)(Cl)C34CC4)=O)nnc2C1 46314,C1(CNC(=O)CSc2ccncc2)CCN(C(c2c[nH]cc2Br)=O)CC1 46315,N1(C(C(C)N(C)C)=O)CCCN(C(c2cc(C(F)(F)F)ns2)=O)CC1C 46316,c1(C(=O)NCC2C(NC(c3nccc(C)n3)=O)C2)ccc2nc(O)[nH]c2c1F 46317,CCP(=O)(CC)c1ccccc1C(N1CC(C(C)NC(=O)CCC(N)=O)C1)=O 46318,C1(NC(C(C)C2CCCC2)=O)C2CCN(C(C3CCCO3)=O)CC12 46319,Cc1oc2ncnc(O)c2c1C(=O)NC1CCN(C(c2cc(Cl)no2)=O)CC1O 46320,n1(CC(=O)NCCCCCN2CCCC2)cc(C2CC2)nn1.c1(C)cnoc1 46321,c1(OC)cc(C(N2CC(O)CC2CNC(=O)Cc2c[nH]nc2C)=O)ccc1F 46322,C(C)(CC(C)N=c1c(C#N)c[nH]c2ccc(Cl)cc12)NC(Cc1cc(C)no1)=O 46323,n1(CC(N2CC(c3cnc(Br)s3)C2)=O)ccc(-c2ccccc2)n1 46324,c1(C(C)C)nc(N2CCCOC(CNC(=O)CCc3cscn3)C2)cc(Cl)n1 46325,N1(C2CCN(C(=O)CC3COCCO3)CC2)CCN(C(c2cnns2)=O)CC1=O 46326,C12CC3CC(C1)N(C3)Cc1cc(on1)CC(=O)N2.C1(CCC)(C(=O)OC)CC1 46327,C1(C=O)CN(Cc2ccco2)C2(CCOC2)C1.Cc1noc2ncccc12 46328,CC(C)CCCC(C)C(=O)CC(CN1C(C)CCC(N)C1)O.CC[Si](C)(C)C 46329,N1(C(=O)CCCn2cncn2)CC2CC2(C(=O)NC2CC23CCC3)C1 46330,C1(C(C)C)(C(=O)N(C2CCCCC2)CCO)CCCN1C(=O)CCC1CCCO1 46331,CCC(C)C(C)C(=O)NC(C)(CC)CCNC(c1cccc(=S)n1O)=O 46332,c1(C(=O)NC2(C)CN(C(=O)CCc3ccc(Cl)cc3Cl)C2)cc(O)cc(Cl)c1 46333,c1(C(=O)NC2C(CNC(CN(C(C(C)C)=O)C)=O)COC2)cnn2cccc(Cl)c12 46334,c1(C(N2C3C(NC(C(C)c4cncs4)=O)CC(C3)C2)=O)cccc2c1C(=O)CC2 46335,C(=O)(CC1=CCCCC1)NC(C(C(C)C)C)CNC(N1CCCC1)=O.C(C)(C)(C)O 46336,N1(C(Cc2c(C)nc[nH]2)=O)CCC2CCN(C(=O)CNC(N)=O)CC12 46337,c1(C(=O)NC2C(CNC(C=COCC)=O)COC2)cccnc1Cc1cc[nH]n1 46338,N1(c2nccc(SC)n2)C2CCC1CN(C(=O)C(C)Cn1ccc(C)n1)CC2 46339,n1(C(CC)C=O)c(=O)nc(O)c2c(C(=O)N(C)Cc3ccnc(F)c3)ncnc12 46340,C12(C(=O)NC(CCNC(C(C=C=C)C)=O)C)CC3CC1C2C3(F)F 46341,c1(C(N2C3CN(C(c4cc(Br)ccc4Cl)=O)CC32)=O)ccc([N+](=O)[O-])c(O)c1 46342,C1(CC(=O)NC(C(N)=O)CO)C2CCCC2N1C(=O)CN(C1CCCC1)C 46343,c1(C(=O)NC)ccc(C(=O)NCCCC(C)(C)NC(C2CCS(=O)(=O)N2)=O)cc1 46344,C1(NC(C(C2CCC2)OC)=O)CC(O)(CNC(C2CCCN2C(N)=O)=O)C1 46345,C(=O)(C1=CC2CCCC12)NC1(CNC(COC(C)=O)=O)CCCC1 46346,C(C(CCC(F)F)NC(=O)OC(C)(C)C)OC(C)(C)C.C12(CCOC1)CC(=O)N2 46347,C(=O)(CC(C)(C)C(=O)OCc1cn(-c2ccccc2)c2c1CCC2)OC(C)(C)C 46348,c1(NC(C2N(C(c3cccc(F)c3)C)CC2)=O)ccc(C2=NNC(=O)CC2)cc1 46349,C1(CC)(COC)CCN(C(C2(N(C)C(C3CCCO3)=O)CCCC2)=O)CC1 46350,CC(C)C(O)C(C)C(=O)NC1CCN(C(c2ccn3ccnc3n2)=O)C1C 46351,c1(C(N2C(C(C)NC(=O)Cc3ccno3)CCC2)=O)cc(Cl)ccc1Cl 46352,c1(C(=O)NCc2nc(CNC(CSCC=C)=O)sc2)cc(CS(C)(=O)=O)oc1C 46353,C(=O)(C1=CCN(C)CC1)N1CCC(NC(c2cc(CC)no2)=O)C(CC)C1 46354,c1(SCCNC(Cn2cc(CN3CCC(OC)CC3)nn2)=O)ccc(F)cc1F 46355,C1(CC)(CO)CCCN(C(=O)CC2CCN2C(c2ccc(O)cn2)=O)C1 46356,CCCC(C(=O)NC1COC2(C1)CN(C(c1cnn3ncccc13)=O)C2)C(C)C 46357,c1(C(=O)NC2CN(C(C(CCCC)c3ccccc3)=O)C2)cc(N)cc(O)c1C 46358,c1(C(=O)NC(C2CCCN(C(CCN(C)CC)=O)C2)C)ncc(Br)cc1F 46359,CCC(C)(CC)C(=O)N1CC(OC)C(NC(=O)CCc2ccnc(C)n2)C1 46360,c1(OC)ncc(C(=O)N(C2CCC(NC(c3cnc(C(C)(C)C)o3)=O)C2)C)s1 46361,c1(C(=O)NC2CC(O)(CNC(C(C)OCCC#C)=O)C2)cc(F)c(F)c(F)c1 46362,N1(C(C(C)(C)CF)=O)CC2CC(F)(F)CCC2(NC(c2cc(Cl)cnc2O)=O)C1 46363,c1(NC(=O)C(=O)N(C2CC(n3ccnn3)C2)C2CCSC2)ccccc1 46364,N1(C(CSCC=C)=O)CCN(C(=O)CCS(C)(=O)=O)C2CC12 46365,N1(C(Cn2c(C)cc(C)n2)=O)CC(C(N2CCCC(F)(F)C2)=O)C(F)(F)C1 46366,c1(C(=O)O)cc2cc(C(=O)Nc3ccc(C(F)(F)F)cc3F)sc2s1 46367,Cc1oc2c(F)c(F)c(F)c(F)c2c1C(=O)NC1CC1(C)C(F)F 46368,N1(Cc2nc(Br)oc2)CCc2sc(-c3cnn(C4CCCCC4)c3)cc2C1 46369,C1(CCCC)CN(C(=O)CCOC)CCN1C(=O)CCC1CC1 46370,c1(C(N(CCCC)CCCO)=O)ncccc1N(C)C 46371,C(=O)(C1CCCc2ncccc21)N1C(C)(C(=O)NC)CC(O)C1.C12CN(C1)C(=O)N2 46372,c1(C(=O)NCC2C3(CCN(C(C=C(C)C)=O)CC3)C2)c(C)nc2ncccn12 46373,CN1CC(C(=O)NCCN(C(C23CCCC2(C(N)=O)C3)=O)C2CC2)CC1=O 46374,N1(C(C2C(c3n(C)ncc3)C2)=O)CC2CC2(C(=O)NCC2CCCOC2C)C1 46375,CC1CCN(C(=O)Cc2ccccc2Br)C(C)C1NC(=O)CCF 46376,c1(CN2CCC(N(C(C(C)NC(CC)=O)=O)C)C2)ccccc1Cl 46377,c1(N2CCC(C(=O)Nc3nccnc3F)C2)ncnn2cc(Br)cc12 46378,C1(C)(CC(=O)N(CC(CNC(c2nccc(CC)c2)=O)O)C)CCS(=O)(=O)N1 46379,CCC1CC(=O)N1C.C(=O)(CCCN(CCC)C(C)C)NC(C)CCC 46380,N1(C(C2(CC=C)CCCN2C(=O)CC2CCCC3CC23)=O)CC2CCCC(C2)C1 46381,C1(C(O)=O)CCC2C(CCN2C(c2cc3ccccc3n2CC2CC2)=O)C1 46382,C1(NC(C(CN(C)C)NC(CSCC#C)=O)=O)CC=CC(O)C1 46383,c1(CC)nc[nH]c1C(=O)NC1(CNC(=O)COCCOCCO)CCOC1 46384,C1(C(=O)NC(C=C)C2CCC2)(CCNC(=O)CNc2ncccn2)CCOC1 46385,CC1C(C(=O)N2C3CCC2CC(C(=O)Nc2ccc(F)cc2)C3)=NOC1C 46386,c1(CC(C)C)cc(C(=O)NCC(C(C)C)NC(N)=O)cs1.C12CCCN1C(=O)C2 46387,c1(C(N2CCCCC(NC(C3C(C)C3)=O)CC2)=O)c(F)ccc2nc[nH]c12 46388,C1(CCCNC(C23CC(C)(C2)C3)=O)CN(C(C2CC2C2CC2)=O)CCO1 46389,N1(C(C2CCC(CC)CC2)=O)CC(CNC(c2cncn2C)=O)CC1(C)C 46390,N1(C(C)=O)CCOC(C(N2CCC(C(=O)NCc3ncsn3)CC2)=O)C1 46391,c1(C(N2CCC(C)(C(N)=O)C2)C(=O)[N+](CC)([O-])N(C)C)ccnc(S(C)(=O)=O)c1 46392,C1(CNC(C(C)OCC)=O)CCN(C(C23COC(CF)(C2)C3)=O)C1C 46393,Cc1cc(CCC(N2CCC(NC(C3CC(CF)C3)=O)C2)=O)n(C)n1 46394,N1(C(C(C(C)C)C)=O)CCC2(C(N3CCC(CN(C)C)CC3)=O)CCCC12 46395,C12(C)CCN(CC1)C2=O.C1(C(C)C)CCCN(c2ncc(I)cn2)C1 46396,C(=O)(N1CC2COCC2O1)C1OCCC(NC(=O)C=C2CCSCC2)C1 46397,c1(C(N(C2CCN(C(c3cccc(CC)n3)=O)C2)CC(F)F)=O)cnccc1C 46398,N1(C(CC=C=C)=O)CCCCCC1CNC(=O)CCC1CCC(=O)C1 46399,S(=O)(=O)(c1c[nH]c2cc(F)ccc12)Nc1ccc(C)c(OC(F)F)c1 46400,c1(C(=O)NCC(C(C)C)NC(c2[nH]nc(OC)c2Cl)=O)c(S(C)(=O)=O)cnn1C 46401,n1(CC(=O)NCC2N(C(CCCCC=C)=O)C3C(C2)C3)ncn2nccc2c1=O 46402,C(=O)(C(O)CCNC(=O)CN1CC2CC2C1)N(C(C)CNC(N)=O)C 46403,c1(C(N2CCC(C(CNC(C(C)(C)F)=O)O)CC2)=O)c[nH]cc(Cl)c1=O 46404,c1(C(C(=O)NC2COC2)N(C2C3CCCC23)CC)cc(C)nnc1C 46405,N1(C(=O)OC(C)(C)C)CC2CCCCC2(NC(N2CC3CCC(C2)C3(F)F)=O)C1 46406,c1(C(=O)NCC2CC(OC)CN2C(C2OCCO2)=O)cc2cc(Cl)cc(C)c2[nH]1 46407,c1(N(C(C(=O)NC2(C)CC2)c2cccs2)CCC)ccccc1 46408,N#Cc1ccccc1C1CCCCN1CCC(=O)OCCC(=O)NCC1CCC1.N.CC 46409,Cc1ccn(CC(=O)N(C(C)CNC(=O)COc2c(C)occc2=O)C)c(=O)c1 46410,N1(C(C(CC(=O)OC)(C)C)=O)CC2CCCCC2(NC(=O)C(C(C)C)SC)C1 46411,C(=O)(C(C)(CC)CO)NCC1C2CN(C(Cn3c(CCC)ncc3)=O)CC21 46412,C(CN=C(NCCc1cccc(F)c1)NC(c1nc(C(F)(F)F)cs1)C)SC 46413,N1(S(CCC(=O)OC)(=O)=O)CC2(CCCC2NC(c2cccc(OC)c2F)=O)C1 46414,CC(O)(C(=O)NCC1(NC(c2cnn(CC3CC3)c2)=O)CC1)C1CC1 46415,C1(NC(c2n[nH]c(C)c2Cl)=O)CCC2(CC1)CCN(C(c1ccc(CO)s1)=O)C2 46416,c1(C(=O)NCCC2(C(=O)NCCCCC)CCCC2)nc(=N)cc[nH]1 46417,c1(C(=O)NC(C)CN(C)C(c2ccc(-c3cccs3)[nH]2)=O)ncc(F)cc1N 46418,C1(NC(C2(F)C(C)C2)=O)CCC(F)(CNC(c2ccc(Cl)cn2)=O)C1 46419,c1(C(N2CC(NC(c3cc(CC)no3)=O)C(C)C2)=O)c(C)nc2sc(C)cn12 46420,O=C(C1CCc2ccccc21)NCCc1cc(F)cc(F)c1F 46421,C(CCCCCCCO)=CC(=O)NCC1CCN(C(C23CC(C)C2C3)=O)C1(C)C 46422,N1(C(C(C)c2cccs2)=O)CCC(O)CC1C(N1CCC(c2ccco2)C1)=O 46423,C1(C(=O)NCC2(NC(C(CCC)F)=O)CCC2)CN2CCC1CC2 46424,C(=O)(C(CNC(=O)CC1CC2C=CC1C2)CCC)NCC1CC(CCC)C1 46425,N1(C(CN(C(C(C)NC(=O)CC2C=CCC2)=O)C2CC2)=O)CC2CN(C)CC2(C)C1 46426,CC(CNC(=O)CCc1cscn1)(CO)NC(=O)CSC(F)(F)F 46427,c1(C(=O)NCC(CNC(C(CC)OC)=O)(C)O)cc(N)c(C)c([N+](=O)[O-])c1 46428,Cc1cc(Cl)c(C(N2CC(O)CC2CNC(=O)C(C)(O)C2CCC2)=O)cc1F 46429,c1(C(=O)Nc2c(C(=O)OC)nn(CC(F)(F)F)c2)c(C)cc(C)nc1Cl 46430,C=CCCCCC(=O)NC(C(=O)NC1CC12CCC2)c1cccs1 46431,Cc1cccc(SC(C)C(=O)NCC2CCC2NC(C23CC(C2)C(C)(C)O3)=O)c1 46432,N1(Cc2cccc(OC(C)C)c2)CCC(NC(C2CNC(=O)O2)=O)C(F)C1 46433,c1(NCc2onc(COC)n2)nc(=NCC#CCCO)[nH]c2c(C)nn(C)c12 46434,NC(=O)CCC(=O)NCC1CC(NC(=O)Cc2cccc(O)c2)CC1O 46435,c1(C(=O)NCCC2CCC(NC(C(COC)OC)=O)C2)cc2c(cc1N)OCO2 46436,C1(CN(C(=O)CC2C=CCCC2)C)CCCN1C(c1nocc1Br)=O 46437,CCCCC(CNC(C1(NC(=O)C(C)CC(=O)OC)CC(F)(F)C1)=O)CCC 46438,C(=O)(C1=Cc2ccccc2C1)NC1C2(CCN(C(CSCCOC)=O)C2)CCC1 46439,CCCCCS(=O)(=O)CC(=O)NCCCCCNC(=O)CC(CC)OC 46440,N1(C(CSCC#C)=O)CCCC2(CCCCC2NC(c2cnn[nH]2)=O)C1 46441,C1(NC(c2nc(C)oc2)=O)CC1C1CCN(C(=O)C(C)CC(C)(C)C)CC1 46442,C1(c2ncc(C)cn2)CCN(N(CC2CCCCC2)Cc2ccc(Cl)cc2)CC1 46443,C(=O)(CCCF)N1C(CC(=O)NCC2CC2Cl)CC1 46444,C1(C(=O)NCC#C)CC2C=CC1N(C(=O)CC(=O)NCC1CC1)C2 46445,CP(C)(=O)C1(O)CCN(C(C2CC=CCC2)C(=O)NCc2ccccc2Cl)CC1 46446,C1(NC(Cc2c(C)n[nH]c2C)=O)CC2CC1CN2C(c1ccc(O)c(F)c1)=O 46447,c1(C(CC)(C)NC(=O)CCn2cc(-c3cc[nH]n3)nn2)ccccc1Cl 46448,C(C(CNC(=O)C(F)C1CCC1)S(C)(=O)=O)NC(CCC)=O 46449,Cc1ccc(C)n1CC(N1CCCC1CCNC(c1cc(C(F)(F)F)cs1)=O)=O 46450,N1(C(c2c(C)n(C(C)(C)C)nc2)=O)CC2(CCN2C(C2(F)CCC(C)CC2)=O)C1 46451,c1(C(CNC(=O)COC2CC2)NC(c2coc(=O)[nH]2)=O)ccc2ccccc2c1 46452,C1(NC(C2COCCN(C(C3CC(OC)C3)=O)C2)=O)CC(C)N(C)CC1C 46453,c1(OC)cccc(C2CC(NC(=O)C(C)(C)C#N)C2)c1.C(=O)(C(F)C1CCC1)O 46454,N1(C(C(n2c(C)cc(C)n2)C)=O)CCC2C(C1)NC(=O)CN2C(=O)C(C)C 46455,C1(NC(C2CCCC(F)C2)=O)CCCC12CCN(C(c1cnnc(O)c1)=O)CC2 46456,C1(CCC)(NC(=O)CC2C=CCC2)CCCN(C(c2ccccc2CC)=O)C1 46457,c1(C(N2CC3CCN(C(CCC=C)=O)C3C2)=O)cc2nc[nH]c2cc1[N+](=O)[O-] 46458,C(=O)(C(C)(C)C(=O)N1CCCC(NC(=O)CC2(C#N)CCC2)C1)N(C)C 46459,C1(N(C(=O)Cn2cccn2)Cc2cc(Cl)ccc2F)CCC12CCNCC2 46460,CC1CCSCCN1C(c1[nH]ccc1CNC(C12CCC(CC1)CC2)=O)=O 46461,N1(C(C(CC)N(C)C(c2cc[nH]c2)=O)=O)CCCC(C(=O)OC)(CC)C1 46462,N1(C(C(C)OCOC)=O)CC(O)CC1CNC(=O)CCCn1ccnn1 46463,C(=O)(C(F)CC1CN(C(c2c[nH]c(=N)o2)=O)C1)NC(C1CCCO1)C 46464,c1(C(=O)NC(CNC(C=CCOCCOC)=O)CC)ncnc2sccc12 46465,Cc1cnc(Cl)[nH]c1=NC(=O)c1cnc2ccc(-c3ccnc(F)c3C)cn12 46466,c1(C(=O)NC2CC(CNC(C(C)(C)CF)=O)OCC2)cc(Cl)c2n[nH]cc2c1 46467,C(C(C)C)(C(O)C(=O)NCC1(O)CCCN(C(c2cnn3c2OCC3)=O)C1)OC 46468,C(CC(C)C(=O)NCC(c1ccccc1F)NC(C1CCC1(F)F)=O)=CCC 46469,CCC(C)(O)CCNC(=O)C(C(C)OC)NC(=O)CN1CCC(=O)CC1 46470,c1(N(CC(CNC(C(CC)NC(N)=O)=O)C)C)cc(Cl)nc(C(F)(F)F)n1 46471,C1(C(=O)NCCC(=O)OC)CN(C(c2ccc(Br)s2)=O)CC2(CCC2)C1 46472,CC(C(=O)NN(CCOCCCNC(c1ccsc1)=O)C)C(C)O.C(CO)O 46473,N1(C(c2csc(C)c2N)=O)CC(C)CN(C(c2sc([N+](=O)[O-])cc2Cl)=O)CC1C 46474,c1(SC(C)C(=O)NC2CCCCC2NC(=O)CCOCC2CC2)ccc(F)cc1 46475,C1(C(=O)NC2CCC(F)(F)C2)CC(F)(F)CN1S(=O)(=O)CCBr 46476,c1(C(=O)NCC2CC2NC(c2sc(Cl)cc2Cl)=O)cn2c(n1)CCC2 46477,Cc1nc2ccnn2c(C)c1C(=O)NCC1COCC1NC(=O)CCC(F)F 46478,N(C(=NCCc1cn(C)cn1)N1CCN(C(C)(C)C(N)=O)CC1)Cc1cc(C)no1 46479,c1(CC(N2C(C)CC(NC(c3cnc(=N)[nH]c3)=O)C2)=O)cnc2c(=O)[nH]ccn12 46480,N1(C(=O)C=CC(F)(F)F)CCOC2(CCCN(C(c3ccn(CCF)n3)=O)C2)C1 46481,C(C(C)(O)CCNC(=O)NC(C)Cc1ccc(C(F)(F)F)cc1)OC 46482,N1(C(C(CCOC)C)=O)CC(C2CC2)(C(=O)Nc2csnc2OC)C1 46483,CC(CCc1ccccc1F)C(=O)NCC1CCCN1C(c1c[nH]nc1Cl)=O 46484,N1(C(c2c(CCC)[nH]cc2)=O)CCC2(C=C(C(=O)NC(C)CCC(C)CC)C2)C1 46485,C1(C(N(CCCCNC(c2cc(COC)on2)=O)C)=O)CN(C)CCO1 46486,Cc1nn2c(c1C(=O)NC1CN(C(c3ncccc3N)=O)C3CC13)CCCC2 46487,N1(C(c2cnc(C(C)C)nc2)=O)CC(NC(c2ocnc2C2CC2)=O)C2(CC2)C1 46488,C1(C(N(C(C)CC(=O)NC(C)Cc2nncn2C)C)=O)CC(C)N(C)C1 46489,N1(C(c2cnc(C(C)C)[nH]2)=O)CC(CNC(=O)CCc2cscn2)C(O)C1 46490,c1(C(=O)NC(CCOC)C(=O)N(C2CCN(C)C2=O)C)cccc(F)c1C 46491,c1(OC)ncc(C(N2CC(CNC(C3CCC(C)O3)=O)C2)=O)cc1C 46492,c1(CC(C)C)occc1C(=O)NCC(C(C)C)CCN(C)C.C(=O)(COCCO)N 46493,C1(CNC(c2cnc(Cl)cn2)=O)CN(C(=O)CC2CCCCC2)CCC12CCC2 46494,N1(C(c2cnc(C(C)OC)s2)=O)CC2C(NC(=O)Cc3cscn3)C2C1 46495,c1(OC)cc(C(=O)NC2CCN(C(=O)C3=C(C)CCC3)C2(C)C)c(F)c(Cl)c1 46496,CC1(C)CN(C(C2CC(C(N)=O)C2)=O)CCC1NC(c1csc(C(N)=O)n1)=O 46497,C1(N(CC#C)C(c2nocc2Cl)=O)CCN(C(C2(O)CCC2)=O)CC1 46498,N#Cc1ccc(C(O)C(=O)NCC2CCC2c2ccccc2)cc1 46499,O=S(=O)(c1ccc(Br)cc1NC1CCCC1)N1CCn2cnnc2C1 46500,N1(N(C2(C)CCCCC2(C)C)C(C2(C=C)CCCC2)=O)CCCC(C2CC2)CC1 46501,c12snnc1CNC2c1ccnn1CCOCC.n1(CC(=C)C)nnnc1C1CC1 46502,c1(C(N(CCN(C(c2cccc(N)n2)=O)CC)CC)=O)ccc2nc(S)[nH]c2c1 46503,N1(C(CNC=O)=O)CCOC2CN(C(C3C4CC5C(C4)C35)=O)CC12 46504,CC1=C(C(=O)N2CC3(NC(c4cc(C#N)ccc4N)=O)CCC2C3)CCCC1 46505,N1(C(Cc2nc(C)sc2C)=O)CCCC(N(C)C(C2(C3CCCO3)CC2)=O)CC1 46506,N1(CC(=O)N(CC(O)CNC(=O)CCc2cn[nH]c2)C)CCC(C)(C)CC1 46507,C(=O)(C(C(C)C)N(C)C)N(C1CC(NCCC(=O)NC)C1)N(C)C 46508,N#CC1(C(=O)NC2CCCCCN(C(c3ccc[n+]([O-])c3)=O)C2)CC12CCOCC2 46509,c1(C(=O)Nc2n(CC)cnc2C(F)(F)F)c(OC)ncc(Br)c1C 46510,N1(C(CCc2c(C)ncs2)=O)CC=C(CCNC(=O)CCCNC(=O)C2CC2)CC1 46511,C(=O)(CC1COc2cc(O)ccc21)NC(CC(C)(C)C)CO 46512,C(=O)(C1=CCC(NC(=O)C(C)(C)C(=O)OCC)C1)NCCC(CCC)C 46513,c1(CC(C(=O)NC2COCOC2)N(C)Cc2cccc(Br)c2)ccc(Cl)cc1Cl 46514,CC1CCC(N(C(=O)C(C2CCCO2)Nc2nc(O)n[nH]2)C(=O)OC(C)(C)C)C1 46515,C1(C(=O)NCC2COCCN2C(c2csc(C3CC3)n2)=O)CN2CCCC2CO1 46516,C=CCC(C)(CC)C(=O)NCC1CCC1C(=O)Nc1ccc(C)cc1CO 46517,C1(CN(C(CC2(OC)CCC2)=O)C)CN(C(c2sc(CO)nc2C)=O)CC12CC2 46518,C12(CNC(Cc3cc(C)[nH]n3)=O)CC1CN(C(=O)C=CC(=O)NC1CC1)C2 46519,CCC(O)C(C)C(=O)NC1(CNC(=O)CCOCc2ccccc2)CCOCC1 46520,N1(C(C(=O)NC(c2nc(CCC(=O)OC)[nH]n2)C)=O)CCC(F)(C#N)C1 46521,CCCCC(CNC(C1CCC(CN2CCOCC2)O1)=O)NC(=O)CC1CCC1 46522,c1(CNc2sc3c(n2)C(C)(C)CC3)cc([N+](=O)[O-])cc2c1OC(F)(F)O2 46523,Cc1cc(C(=O)N(C(CNC(c2cccc(O)n2)=O)C2CC2)C)n2nccc2n1 46524,c1(C(N(C2CCCN(C(=O)Cc3nnc(O)s3)C2)C)=O)ccc(=O)n2c1CCC2 46525,Cc1cc(C(=O)NCCC2CC(NC(C3(OC)CCSC3)=O)C2)n2nccc2n1 46526,C(=O)(C(F)(F)C(F)(F)F)NC1C(CNC(C2=NOC(C(C)(C)C)C2)=O)CC1 46527,CC1CCCC(CNC(C2(NC(=O)Cn3cc(Br)cn3)CC2)=O)O1 46528,CC(C)C(O)CC(=O)N(CC(=O)NCc1ccc(C(C)C)cc1)C1CCC1 46529,C1(N(C(=O)CCc2cnn[nH]2)C)CCCN(C(=O)COC2CCC(=O)N2)CC1 46530,CC1CC(NC(=O)CCS(N)(=O)=O)CCN1C(C1CC2(C1)CC2(F)F)=O 46531,C(=O)(C(C)CCC)N1CC(OCCC(=O)NC(CCC=C)C)C1 46532,c1(CC)cc(C(N2CC(=C(F)CNC(=O)CC(C)c3ccccn3)C2)=O)oc1CC 46533,Cn1ncc2cc(C(N3CCN(C(=O)CCCC4CC4)C(CCO)C3)=O)cnc12 46534,C(=O)(C(C)CC(C)(C)C)NCC(C)(C1CCC1)NC(CCc1ccnc(C)n1)=O 46535,N1(C(C2C(=C)CC2)=O)CC2COCCC2(NC(c2nc(SC)ncc2N)=O)C1 46536,C1(C(=O)NCC(C2CCN(C(c3cnc[nH]c3=N)=O)CC2)(C)C)CCCCC12CC2 46537,c1(C(N2CC(NC(C=CCOCCOC)=O)C(O)C2)=O)cccc2cnsc12 46538,c1(C(=O)NCCCNC(CC2(C)CC(F)(F)C2)=O)cc2ccccc2[nH]c1=N 46539,c1(-c2n(CCS(CC)(=O)=O)nc(C(C)OC)n2)cc2ccccc2nc1OC 46540,C1(C(C)NC(C2(Br)CC2)=O)CCN(C(C2CCOC(=O)N2)=O)CC1 46541,C1(Cc2onc(CN3C(=O)COCC3)n2)CCC2(CCNC2)CC1 46542,c1(C(C(=O)NCCC#C)NCC(=O)NC(c2cccnc2)C)cn(C)cn1 46543,CCC(CC(=O)NCC1C(C(N2CCN(CC(C)O)CC2)=O)C1(C)C)C1CC1 46544,C1CCCC(=O)NC2CCOC2C(=O)NO1.CCCCC1(CC(=O)OC)CC1 46545,C1(CN(C(C)C)C(c2c(F)ccc(I)c2F)=O)CCC2(CCC2)CN1C 46546,C(=O)(CCCCCc1cccs1)NC12C(CN(C(Cc3cccc(OC)c3)=O)C1)C2 46547,C1(NC(c2cc(COC)no2)=O)CC2CN(C(=O)C(C)=C(C)C)CC12 46548,C(=O)(CC(O)C(C)C)NC1(CO)CN(C(c2ccc(CCCCOC)cc2)=O)C1 46549,O(P(=O)(OCCCl)C(F)C(=O)NCC(=O)NC1CC1F)OC(C)(C)C 46550,CCC(CN(C)C)CC(=O)N(C)CC1(O)CCN(C(c2cncn2C(C)C)=O)C1 46551,N1(C(CC2(CC=C)CCCC2)=O)CCC2CCN(C(C3C=CCC3)=O)C2C1 46552,c1(NC(C2CSCCN2Cc2scc(Br)c2Br)=O)ccc(O)cc1Br 46553,c1(C(N2C(C)CC(CNC(C3COCCO3)=O)C2)=O)ccc2c(c1)CCN2 46554,C1(C)(CNC(c2cnc(C)s2)=O)CCC(NC(c2coc(O)n2)=O)C1 46555,c1(C(=O)NCC2CCC(NC(c3cc[n+]([O-])cc3)=O)CC2)ccc2c(c1)COC2 46556,N1(C(c2nnn(C(C)(C)C)n2)=O)CCCC(C)(NC(=O)CC2CCC(=O)N2)C1 46557,c1(OC)ccc(CC(N2CCOCC2CCNC(C2CC(F)C2)=O)=O)cc1OC 46558,N1(C(CC(CC)CC)=O)CC2CCOCC2(NC(=O)CC(C)(C)CC(=O)OC)C1 46559,c1(N(C)CC2CCN(C(C3CC4CC3C3CC43)=O)C2)ncnc(Cl)c1F 46560,c1(C(c2nnnn2CCC2CC2)NC(c2nccn2C)CC)cc(Br)ccc1Cl 46561,C1(NC(C2(C(C)C)COC2)=O)CC(CNC(=O)C(C)CC2CC2)CC1O 46562,N1(C(CC(=C)Br)=O)CC(NC(=O)C(C)CC2CCC2)C(C(F)(F)F)C1 46563,C1(n2cc(C(C(C)(C)C)O)nn2)CN2CCCN1CC2 46564,N1(C(c2cccc(CC(C)C)c2)=O)CCOCC(CNC(=O)CC(O)C(C)C)C1 46565,C1(CC(N2CC3(OCCC(N)C3)C2)=O)CCC2(CCCC2)CC1 46566,CC1CCCC1(O)CC1(C)CN(C(=O)CCNC(=O)CN)C1 46567,c1(C(=O)NCC#CCNC(CN(CCC#C)C)=O)csc(O)n1 46568,Cc1ccc2[nH]c(C(=O)N(C)CC3CC4CC4C3)cc2c1Br 46569,c1(C(=O)NC2C(C)(C)N(C(=O)CN3CC=CC3)CC2)cc(P(C)(C)=O)cs1 46570,C12(CC)CCC(C(=O)NC3CCC(NC(=O)CCc4ccn(C)n4)CC3)(CO1)C2 46571,C1(C(=O)NC(C(N2CCC(c3ncc[nH]3)C2)=O)C2CCCC2)CC=CC(O)C1 46572,c1(-c2cn(C3CCC(C(N4CC5CCC4C5)=O)C3)nn2)ccc(CNC2CC2)cc1 46573,N1(C(C(C=C)(C)O)=O)CCC2(CCCN2C(C2CCC3(CCOCC3)O2)=O)CC1 46574,c1(C(=O)NCc2ncc(C)s2)ccc(-n2cc(-c3ccnn3C3CC3)nn2)cc1 46575,C(=O)(CC(C)C(C)(C)NC(c1cc(Cl)ns1)=O)N1CC(CC)N(C)CC1 46576,c1(C(=O)NC2C(NC(C3N(C)CCCC3)=O)CCCC2)cccc(=S)n1O 46577,c1(OC)cc(C(=O)NC(c2ncc[nH]2)C)cnc1-c1cncc(F)c1 46578,c1(C(=O)NC2CC(NC(C3=C(C)OCC3)=O)C23CCC3)cncc2nc(O)[nH]c12 46579,C1(N(C)C)CC2(NC(C)=O)COC1C2.c12cccc(c1)C(=O)NCc1cnoc1-2 46580,C(C(=O)N1CCC(NC(C2(Cc3cnn[nH]3)CCC2)=O)C1)(C(C)(C)C)NC(C)=O 46581,N(C1CCCc2c[nH]nc21)C(C(C(C)(C)O)NC(C=CC=CC)=O)=O 46582,C(C(C)(CC)C(=O)NC1CCC1C)NC(CC(CC)C1CC1)=O 46583,C12(NC(CCNC(N)=O)=O)CCCC1(F)CN(C(c1coc(CO)c1)=O)C2 46584,C(=O)(CCCCCN(C)C(C1CC(=O)C1)=O)NC(CC(=O)OC)C 46585,C(C(=O)N1CC2CC1C2NC(=O)CCOc1ccc(Cl)cc1Cl)(C(C)(C)C)SC 46586,O=C(CC(F)(F)F)NCC1CCCCC1NC(c1ccc(OCF)cn1)=O 46587,N1(C(C(C2CCC2)OC)=O)CCC12CN(C(=O)CCCSc1ccccc1)C2 46588,c1(C(N2CCCC(CN(C(C3C(C)C3)=O)C)C2)=O)ccc(F)c2occc12 46589,C(=O)(C1CCCc2ncccc21)N1CCC(CCCNC(C(C)SC(C)C)=O)CC1 46590,C(=O)(C(F)(F)C(C)O)NCC1CC(CNC(c2ccc(CC)[nH]2)=O)C1 46591,c1(C(=O)NCCNC(CC2COCC(C)O2)=O)coc2c1CCCC2 46592,C1(CNC(C(C)C2CCC2)=O)CC2CC2N1C(=O)C#CC(=O)N(C)C 46593,C1(CNC(CCCOCC)=O)CC(C)(C)CN1C(c1ccc(N(C)C)nc1)=O 46594,c1(C(=O)NC(C(C)C)CCNC(=O)CCCN(C)C)ccc2c(c1)C=CCC2 46595,C1(C)(C(=O)NC2(c3cn(CCC=C(C)C)nn3)CN(C(C)=O)C2)COCCO1 46596,c1(C(N2CCC(CNC(C3C(CCC)C3)=O)C2)=O)[nH]c(C)nc1C 46597,N1(C(c2c(OC)n[nH]c2)=O)CCC2(CC2C(=O)NCC(C)(C)CN=[N+]=[N-])C1 46598,C(=O)(C(C)CCCOC)NC1C(CC)CN(C(C2(n3ccnc3)CCCC2)=O)C1 46599,CP(C)(=O)C(O)C(=O)N1CC(NC(=O)CC2CCCC(=O)N2)CC(O)C1 46600,c1(CCNC(=O)CC2CCN(C(=O)CC3CCC3C(F)(F)F)C2)cccc(F)c1 46601,CC1(CN=c2ccn(CCC3CCOC3)[nH]2)CCCCCCC1=O 46602,c1(C(N2C(C)CC(NC(C3CC3(C)C)=O)CC2)=O)cc(F)c(O)c(F)c1 46603,c1(C(N2CC3C(C2)N3C(c2coc(Cl)n2)=O)=O)ccc2sccc2c1O 46604,C1(C(N(CCC(=O)NCC2CC(C)(C)CO2)CC)=O)CCN2CCCCC12 46605,C#CCCCC(c1nnnn1C1CC1)NCC.N12CCCC(C1)C2=O 46606,c1(C(=O)NC2CCN(C(c3cnc(-c4ccoc4)s3)=O)CC2)cnn2c1OCC2 46607,c1(C(N2CCc3nc[nH]c3C2)C(=O)NC(C)C)cc(F)c(Br)cc1F 46608,C1(CC)CCC(C)CN1C(C1CCN(C(c2cn(C(C)C)nn2)=O)C1C)=O 46609,CCC(CC(=O)N1CCCC1CNC(c1cc(C)nnc1O)=O)C(C)C 46610,c1(CN(C(CNC(C(=O)NC)C2COC2)=O)C)ccc(Br)cc1Cl 46611,c1(C(=O)NC2CCN(C(C(CC)SC)=O)CC2(C)C)cc2c(C)cccn2n1 46612,C1(NC(c2cc(C)ns2)=O)CN(C(=O)CCSc2ccccc2)CC1C 46613,C1(N(C(=O)CC2COC(=O)C2)C)CCN(C(c2cnc[nH]2)=O)CC1 46614,c1(C(N(CCNC(=O)CCC2CC2(C)C)CC)=O)cnc2n1CC(C)CC2 46615,N1(C(CCC#C)=O)CC2(CCOCC2)CC1CNC(c1cnc2sc(C)cn12)=O 46616,c1(COCC)ccccc1CC(C)C(=O)NCCCCCC(F)(F)F 46617,C1(C)(NC(CC2(C)N(C(c3ccc(SC)o3)=O)CC2)=O)CCCC1C 46618,C1(NC(C(CC)COC)=O)CN(C(c2cnc(OC)nc2)=O)CC1S(C)(=O)=O 46619,c1(CC)cn2c(C(N3CCOC(CC)CC3)C(=O)NC3COC3)cnc2s1 46620,C1(CC(=O)NC2(CC(=O)OC)CC2)CC(OC)CN1C(c1ccncc1CO)=O 46621,C1(NC(Cn2cc(CN(C)C)nn2)=O)COCCN(C(C2CCCCC2O)=O)C1 46622,N1(C(c2c(CC)scc2)=O)CCC(CNC(C2(Cl)CC2(F)F)=O)C(O)C1 46623,Cc1cc(C(N2CCN(C(c3coc(CC4CC4)c3)=O)CC2CO)=O)cc(C)n1 46624,CCCCC(C)CCC(=O)N1CC(C(C)(C)O)(CNC(=O)C(F)OC)C1 46625,C1(NC(c2cc(C)no2)=O)CN(C(=O)C(C)(C)N(C)C)CC1C1CC1 46626,N1(C(c2occ(C(N)=O)c2)=O)CCN(C(C2CCC(Cl)CC2)=O)C(CF)C1 46627,Cc1nc(CC(=O)NC(C)(C)CNC(=O)Cc2csc(Cl)c2)c(C)s1 46628,C#CC1(C)COCCN1C(=O)Nc1cnn(Cc2cccnc2)c1 46629,N1(C(c2c(C)cc(C(N)=O)s2)=O)CCCC2(CCCC2)CC1 46630,CN1CCCC(C(=O)NC(C2CCN(C(c3ccoc3)=O)CC2)(C)C)C1 46631,C1(CCC(=O)N(C)Cc2cn(CC(N3CCOCC3)C)nn2)CCCCN1C 46632,CC1=CC(C)C(c2cn(C(CC(C)C)C(=O)NCCc3csnn3)nn2)CC1 46633,C1(CC(N2CCC(CN(C(CCC(C)N(C)C)=O)C)CC2)=O)CC2(CCO1)CC2 46634,C1(CNCC(C)S(C)(=O)=O)CCC2(CCN(C(=O)OC(C)(C)C)CC2)CO1 46635,CC1CN(C(c2sccc2CNC(=O)CCc2ccoc2)=O)CCS1 46636,C1(O)(CNCc2cc(OC)ncc2)CCCN(C(c2cccc(C(=O)O)c2)=O)C1 46637,C1(OCCCOC)CCC(CC(=O)N(C)CCNC(C2CC(O)C2(C)C)=O)CC1 46638,c12cc([nH]n1)CNC2=O.C1(C(N(CCCN(C)C)CC=C)=O)C2CCCC12 46639,C1(C(N)=O)CC(C(=O)NCC(C)(C)CNC(=O)CCSc2ccccn2)=NO1 46640,c1(OC)cccc(C(=O)NC2CN(C(C3(C#N)CCCOC3)=O)CC2SC)c1C 46641,CC1(CC(=O)NC(CNC(C2CCOC2C(F)(F)F)=O)C2CCC2)OCCO1 46642,Cc1cccc(C(C)(C)C(N2CCN(C(C3CC3)=O)CC2)=O)c1.C1(N)COCC1(C)C 46643,C12(CONC(C3CC(C)(N(C)C)C3)=O)CC3CC1C2C3.C1(=O)C(F)CC2CN1C2 46644,N1(C(c2n(CC)ccc2)=O)CCOC2CN(C(=O)C(c3ccccc3F)C)CC12 46645,CCC(C)C(C(=O)N(C)Cc1nccn1CC)NC(C1CCC(F)(F)CC1)=O 46646,C(CCCNCN1CCCC1)OCC#C 46647,c1(C(=O)OCC)cnc(SC)[nH]c1=NCCCN(C(=O)CC(C)(F)F)C 46648,c1(C(=O)NC(CN(C(=O)C(C2CCOCC2)O)CC)C)cc(C(C)C)n(C)n1 46649,c1(C(N2C(C)(CNC(CC(C)F)=O)CC(F)(F)C2)=O)nc2c(s1)COCC2 46650,CN1CCc2cc(C(=O)NCCc3ocnc3CNC(=O)C=CS(C)=O)sc2C1 46651,CC(C)C#CC(=O)NCC1(C(N)=O)CN(C(C2CC(O)C(F)C2)=O)C1 46652,C1(C)(C(N2CCCC(NC(C(CCCC)F)=O)CC2)=O)CCC(C)=C(C)C1 46653,C12(CCNC(C(c3ccccc3F)C)=O)CCC(C1)N(C(c1nsnc1O)=O)C2 46654,C1(CC(C)NC(C2(CC#C)CCC2)=O)CCN(C(=O)CNC(C)=O)CC1 46655,C12(C(N3CC(CCC)C(NC(c4cn[nH]c4)=O)C3)=O)CCC(CC1)CC2 46656,C1(C(N(CC(CNC(C2(CSC)CC2)=O)O)C)=O)Cc2cc(C)ccc2S1(=O)=O 46657,c1(C(=O)NC(C)CCF)ccc(CNC(C2CC2F)=O)nc1 46658,C1(NC(CCSCCC)=O)CC(C)N(C(=O)C(=O)NCC(F)F)C1 46659,C12(NC(CCCC#C)=O)CCN(C(c3cnoc3C(C)C)=O)CCC1C2 46660,C(=O)(C1OC(=O)c2ccccc21)N1CC(NC(CCC)=O)C(C)(C)CC1 46661,CCCC(CNC(=O)C(CC)OC)C(=O)N(C1CCN(CC)C1)C 46662,c1(C(=O)NC(CC)CNC(=O)C(C)(C)C2CCCCO2)ccc(CO)cc1OC 46663,C(CC(Cc1ccccc1)NC(c1nn[nH]n1)C1CC1)OC 46664,C1(NC(C2N(CC)CC2)=O)CC2CCC(C1C)N2C(c1cnsn1)=O 46665,c1(CN(C)C)ocnc1C(=O)NCC(C)(C1CC1)NC(=O)Cn1cnnc1O 46666,N1(C(C(=C(C)C2CC2)F)=O)CCCC(N(C)C(c2scc(Br)c2Cl)=O)C1 46667,C1(C)(NC(c2c(C(C)NC(=O)C=C(C)C(C)(C)C)noc2)=O)CCCCC1(C)C 46668,S(=O)(=O)(c1sc(O)nc1O)NCC1N(C(C(C)=CCN)=O)CCC1 46669,C=C(C)CCCC(=O)Nc1cccc(NC(=O)COc2ccc(CC)cc2F)c1 46670,c1(N(C(COC)CC(C)C)C)cc(NCC(C)S(C)=O)nc(C)n1 46671,NC(=O)C(N)CCC(=O)NCC1CN(C(c2ccc(C3CC3)nc2)=O)CCO1 46672,CC1OC(=O)NC1C(=O)NCC(C)(C)CN(C(=O)C(c1cnccn1)C)C 46673,C1(C(=O)NC2(CNC(Cc3n(C)ncc3)=O)CCC2)CC2CCCCN2C1 46674,Cc1c(C(N2CC(NC(=O)C(C)Cn3ccnc3)C(O)C2)=O)ccn1CO 46675,C(c1ccc(OC(C)C(C)(F)F)c(OC)c1)=Cc1ccc(C)cc1 46676,CCC(C(=O)OC)C(=O)N1CCCCC1C(=O)NCCc1c(C)n[nH]c1C 46677,c1(CC(=O)NCC2(O)CN(C(c3c(C#C)c[nH]n3)=O)C2)ccc(Br)cc1C 46678,Cc1csc(C(C)C(C2CC2)C(N2CC(O)(Cc3cn(C)cn3)C2)=O)n1.O 46679,Cn1nc(I)cc1NC(=O)NCC1(C)CC(F)(F)C1 46680,c1(CCC)nc(C)c(C(N2CC(CNC(C3(C#N)CCC3)=O)CC2C)=O)o1 46681,C1(CC)CC(C)N(C(=O)C(=O)N(CCCc2nn[nH]n2)C)C(C)C1 46682,c1(C(N(C2CCC(NC(C3C(C(=O)OC)C3)=O)CC2)C)=O)cc(Cl)c(N)cc1F 46683,C#Cc1ccc(CN2CCCC(CNc3nccc(C#N)n3)C2)cc1 46684,N1(C(c2n(C)c(S)nn2)=O)CCCN(C(=O)CCc2ccc(N)cn2)CC1 46685,C1(CC(=O)NCCCCN(C)C(C2CCCN2CC(F)F)=O)CCC(=O)NC1=O 46686,N1(C(CN(C(C)C)C)=O)CCCC2CN(C(=O)CN3CCN(C(C)C)CC3)CCC12 46687,N1(C(c2c(CC)n(C)cn2)=O)CCC2CN(C(=O)C(C)(C)C)CCC2C1 46688,C(CC(C)C)(C(=O)OC)N(C(c1ncoc1C)C(=O)NCC=C)C 46689,n1(CC)nc(C(N2CC(NC(=O)CCc3ncccn3)CC2C)=O)cc1O 46690,N1(C(C2C(C)=CCS2)=O)CC2CC1C2CNC(=O)CCc1nncs1 46691,c1(CC)nn(C)c(CC)c1C(=O)NC(CNC(c1cc(C2CC2)[nH]n1)=O)CC 46692,Cc1nc2ccnn2cc1C(N1CC(NC(=O)C=CCF)C(C)C1)=O 46693,c1(C(=O)NC23CC(NCc4cc(Br)cs4)(C2)C3)cc(Cl)cnc1O 46694,c1(CNCc2scc(-c3c(OCC=C)cccc3)n2)cc(N)c(OC)cc1F 46695,c1(N(CC(C)NC(CCc2c(C)cccn2)=O)C)ncc2c(n1)CCCCC2 46696,N1(C(c2ccn(C)c2)=O)CCC(NC(=O)CC2CCCCC2O)CC(O)C1 46697,C1(NC(Cc2n(C)nnc2)=O)CN(C(=O)Cn2ncn(C)c2=O)CCC1CO 46698,c1(CNC(C(=O)NC2CN(c3ccc(OC)cc3)C(=O)C2)=O)nc2cccnc2s1 46699,C(=O)(C(O)CCCNC(=O)CC1CCOC1=O)N1CC(C(C)OC)C1 46700,S(=O)(=O)(c1cccc(Cl)c1Cl)N1CC2(CC(C(=O)Nc3cc(I)ncn3)C2)C1 46701,Cc1c(C(=O)NCC(C)NC(=O)CCC=CBr)ccn1C 46702,N1(C(CCC#C)=O)CCOC(CNC(C2(c3ccc(C)cc3)CC2)=O)C1 46703,c1(CC)ncc(C(=O)NCCOC2CCN(C(C3CC3(C)C(F)F)=O)C2)c(O)n1 46704,c1(C(=O)NC2CCN(C(C(F)=CC)=O)CC2(C)C)cc2c(nc1O)CCCC2O 46705,c1(NC(c2n(CC)nnn2)c2ccccc2)cc(SC)ccc1OCC 46706,N1(C(C2(CCCC)CCCC2)=O)C2CCC1C(CNC(c1cc(C)[nH]n1)=O)C2 46707,c1(C)cc(C(N2CCC2)=O)no1.C1(C(=O)CC)(N)CCC1.C(=O)NCC1CC1 46708,c1(CC(N2C(C(=O)Nc3c(C)noc3)C(C)CC2)=O)cccc(Cl)c1Cl 46709,CCCC(C(=O)NC(C)(C)C(=O)NCc1ncoc1C1CC1)OCC 46710,CCCCC(O)C(C)C(=O)N(CC(=O)NC1CC2C=CC1O2)C1CC1 46711,c1(C(N2CCCC(NC(=O)C#CC3CC3)C2)=O)cnc(-c2nccs2)nc1O 46712,N1(C(C2CCC(=C)CC2)=O)CCCC(C)(NC(C2CCC2(C)C(=O)O)=O)C1 46713,c1(C(=O)NC2(C(NOCCC#CC)=O)CC2(C)C)cnn2c1CCC2 46714,C=CCCC(=O)NCCC(C)N(C)C(c1occc1Cl)=O 46715,c1(OC)ccc(C2CCN(C(c3ccccc3)=O)C2)cc1.N12CCC(CC1)C2=O 46716,C(=O)(C(F)CC(C)(C)C)NCC1CC(NC(CC(CC)(O)c2ccccc2)=O)C1 46717,c1(C(=O)NCC(C)(C)OCCNC(C2CCCC2)=O)nc2c(s1)COCC2 46718,C1(C(=O)NCCCN(C(C(CC=CC)CC)=O)CC)CCC2(CC1)CNC(=O)C2 46719,c1(CN2CC3CN(C(c4c(C(C)C)cccc4)=O)CC32)c[nH]c2ncc(Br)nc12 46720,C1(C2CCC2)(CNC(CCC(C)(C)OC)=O)CCN(C(=O)OC(C)(C)C)CC1 46721,C1(CNC(C(C)NC(C)=O)=O)C2CN(C(c3ccccc3-n3ccnn3)=O)CC12 46722,C(C1CCOC1)=CC(C(=O)CCC)=O.C(C(CC)N)N(C(C=CCC)=O)C 46723,c1(C(=O)NCCNC(c2cc(OC)c(O)c(I)c2)=O)cc2n(c1)CCCC2 46724,CC(CC(=O)Nc1ccccc1OCC#N)(C(=O)O)C1CCOCC1 46725,CCCC(CCCNC(=O)Cc1nonc1C)NC(c1c(C)nn(CC)c1C)=O 46726,N(C(=NCC(C)Oc1ccc(F)c(Cl)c1)NCC)C(C#C)C 46727,c1(CC)nc(=NC)[nH]c(=NCCCC(C)(C)NC(=O)C=CCN(C)CC)[nH]1 46728,C(=O)(CCC(=O)C1CC1)N(C)NC(c1c(SCC2CC2c2cn[nH]c2)ccs1)=O 46729,C1(NC(c2snc(Cl)c2Cl)=O)COC2(C1)CN(C(c1onc3ccccc13)=O)C2 46730,C12(CNC(C(F)(F)CC3CC3C(N3CCC(OCC)C3)=O)=O)CC3CC1C2C3O 46731,C(CC(=O)N1CC2CC1CN2C(=O)CC(C)(C)C(F)F)(C(F)(F)F)OC 46732,c1(SC)cc(C(=O)NCC(c2ccccc2F)N(C)C)ccc1[N+](=O)[O-] 46733,C=CC(C)(CC)C(=O)N1CCCC1C(=O)NC1CCOC(C)(C)C1 46734,c1(NC(C)=O)cccc(C(=O)Nc2ccn(C3CCNC3)n2)c1 46735,c1(C(=O)OC)cc(C(=O)NCCC2CN(C(c3ccc(CO)nc3)=O)C2)c(C)o1 46736,N1(C(Cc2c(C)non2)=O)CC(C)(C)CC1CNC(C1CCC1(F)F)=O 46737,CCCCCCCCC(=O)NC(C)(C)CC=CC(=O)N(CC(C)CO)C 46738,C1(NC(CS(=O)(=O)NCC)=O)CCCC12CN(C(=O)C=Cc1ncc(C)[nH]1)C2 46739,C(=O)(C1=NNC(=O)CC1)N1C(C)CCC(NC(c2cc(CCC)c(C)s2)=O)C1 46740,C(=O)(C1=CCC(C)(C)CC1)NCC1CCC(CNC(c2ncn(CC)n2)=O)CC1 46741,c1(NC(C2N(C(c3cc(CC)[nH]n3)=O)CC(O)C2)=O)ncc(Br)nc1C#N 46742,C=C(C)C(CC(=O)NCCCN(C(=O)C(c1cc(F)cc(F)c1)O)C)OCC 46743,C(CCCO)N(C(=O)C=CCN(C(=O)C(N1CCC1)C1CC1)CC)C 46744,c1(CNC)ccc(O)cc1NCc1cc(OC)ncc1.C12CC1CN(C(C)=O)C2 46745,C#Cc1ccc(Br)c(C(=O)NCC2CN(C(c3cc(C)oc3C)=O)C3CC23)c1 46746,c1(OCC(=O)N(C(C)CNC(C2CC2Br)=O)C)cc(C(F)(F)F)ccc1O 46747,C1(C(=O)NC(=O)CCCc2nccs2)CCCCC1(F)F.c12ccccc1COC2 46748,C(=O)(C(C(=O)NC(C)(CNC(c1cnn(CCO)c1C)=O)C(C)C)OC)OC 46749,C(C(O)(C(F)(F)F)c1nccn1C)NC(C1(CNC(CC(=O)OCC)=O)CC1)=O 46750,C(=O)(C(F)C(F)(F)C(F)(F)F)N1CC2(CC(NC(=O)CC3CC34CC4)C2)C1 46751,C(=O)(C1OC(=O)c2ccccc21)NC1(CN(C)C(C2CCC=CO2)=O)CC1 46752,N1(C(c2cn(CCOC)nn2)=O)CCC(C)(NC(=O)C(C)n2cncn2)CC1 46753,N1(C(C(C)OCCN(C)C)=O)CCOC(CCCNC(=O)Cc2csc(Cl)c2)C1 46754,c1(C(C(=O)N(CCCN(C(Cc2c(C)cc(C)s2)=O)C)C)O)ccc(Cl)c(Cl)c1 46755,C1(=CCNC(C(C)CO)=O)CCN(C(=O)C(c2ccccc2)N(C)C2CC2)CC1 46756,C1(NC(C2CN(C(CC3(CSC)CC3)=O)CC2C)=O)CCN(C)CC1C 46757,CCC(CC)(CC)C(=O)NCCC(C)NC(=O)COc1c(C)cccc1C 46758,N1(C(C(C)OCC)=O)CCn2c(CNC(C3CC(CC)C3)=O)nnc2C1 46759,CC1CN(C(=O)C(C#N)C2CC2)CCCN1C(c1cn(C)[nH]c1=N)=O 46760,C(C1CCCc2cccnc21)NC(CC)C(C)(F)F 46761,c1(C(=O)OC)cc(CC)ccc1C.C12CCC(C1)OCCN2 46762,CCCC(C(O)C(=O)NC1CCN(C)C1=O)NC(=O)C(C)C(F)F 46763,N1(C(c2cncc(C)c2C)=O)CCN(C(C2CCCN2C(C)C)=O)CC(CO)C1 46764,c1(OC)cc(C)cnc1C(N1CCC(CO)(NC(c2ccoc2Cl)=O)C1)=O 46765,c1(CC)cccc(CS(=O)CC(=O)NCC2CCCCN2C)c1 46766,c1(CNC(C2(COC)CCCCC2)=O)ccc2c(c1)CN(C(=O)CCC(N)=O)C2 46767,c1(N(CCCC)C(=O)NCC(C)CCCO)nc(C)ccc1C 46768,CCC(C)C(C)C(=O)NC(C)CN1CCN(C(=O)CC(C)NC(=O)OC)CC1 46769,N1(C(c2cn(CCC)nn2)=O)CC2CC2(C(=O)NC2CCCN(CCC)C2)C1 46770,c1(C(=O)NC2CC(OC)CN(C(C(CCC)OC)=O)C2)nccn2ccnc12 46771,C1(N(C(CCOCCOC)=O)CCF)CCCN(C(=O)CC2(C#N)CCC2)C1 46772,N1(CC)CCCC(C(=O)NCC(O)CN(C)C(C2CCNC(=O)C2)=O)C1 46773,C(CN=[N+]=[N-])(C(=O)N1CCC(CCC)C1)NC(C(C=C)OC)=O 46774,C(CCO)(C(=O)N1CCCC(CNC(=O)CN(C)CCO)C1)N(C)C 46775,C1(NC(C(C)SCc2ccccc2)=O)CCCC(NC(c2ccnnc2O)=O)C1 46776,c1(C(N(C)CC2CCCN2C(C2CCCC2(C)C)=O)=O)cc2c(s1)CCC2 46777,c1(C(=O)NCC(CN(C(C(=O)NCCNC(C)=O)=O)C)C)ccnc(S)n1 46778,C1(C(N2CCOCC2)=O)Cc2nccnc2CN1C(=O)C1=NOC2(CCOC2)C1 46779,C(=O)(C(C)(C)CC(C)(C)C)NCCN(C(=O)Cc1csc(N2CCNC2=O)n1)C 46780,N12CCCCC1c1n[nH]cc1C2=O.n1(CCNC(CCOCC)=O)cc(CO)nn1 46781,C(=O)(C(CC(C)C)ONC(=O)CCC1CCOC1)NCCCC1(C)CC1 46782,C(=O)(C1OCCc2ccccc21)NC1CCCN(C(CCSCC(N)=O)=O)C1 46783,c1(C(=O)NCC2CC3(CC(NC(C(C)(C)O)=O)C3)C2)cc(P(C)(C)=O)ccc1O 46784,c1(C(=O)NCC(COC)C)occc1CNC(c1cncnc1)=O 46785,N1(C(=O)CCc2ccncn2)CCCC12CN(C(c1ccc(I)cc1Cl)=O)C2 46786,CC1(C)CCCC(O)(C(=O)NC(CNC(c2cc(C3(O)COC3)on2)=O)CO)C1 46787,c1(C(N2C(C)(C)CC(CNC(c3cnc[nH]3)=O)C2)=O)cc(Br)c2nccn2c1 46788,C(=O)(CCCC(=O)N1CC2CCOC2C1)NC(C)(C)C 46789,c1(SCCOCCNC(C(C)NC(C2OCCC2(C)C)=O)=O)ccc(F)c(F)c1 46790,c1(C(=O)NC2C(C)N(C(c3cccc(Cl)n3)=O)CC2)c(F)ccc(F)c1N 46791,C1(CNC(CC(C)(F)F)=O)C(C2CC2)CCN1C(c1ncc(Cl)c(N)c1Cl)=O 46792,c1(NC(C(=O)NC(C)C2CC2)=O)ccc(OCCN(C)C)cc1 46793,c1(C(=O)NCC(C)(CC)NC(C(CC)=CC)=O)cccc2c1ccn2C(C)C 46794,C1(C2CCN(C(c3ns[nH]c3=O)=O)C2)CCCCN1C(c1cscn1)=O 46795,CN(C1CN(C(=O)CCCC2CCOCC2)CCc2ccccc21)C(=O)C1CC1 46796,C(=O)(C(C)(C)CC(C)(C)C)NCCC1(CNC(c2nccc(C)n2)=O)CC1 46797,CCC(N=c1cc(NC(=O)CSCC2CCCCO2)nc(C(F)(F)F)[nH]1)C(C)C 46798,c1(N2CCN(C(C)CO)CC2)nc(N(C)CC2CCCO2)c2cnn(C)c2n1 46799,C(=O)(C(F)n1ccnc1)N(CCN(C(c1cnn[nH]1)=O)CC)CC 46800,C1(C(=O)NC2(C)CCN(C(Cc3cc(COC)on3)=O)C2)COCC2(CCC2)O1 46801,N1(C(C2(CCN=[N+]=[N-])CC2)=O)CC(=O)NCC1C(N1CCNC(=O)C1)=O 46802,c1(C(=O)NC(CC(C)NC(c2c(NC)cccc2)=O)C)c(F)cc(C)cc1Cl 46803,C(C)(C(C)C(=O)NCC1(C2CCC2)CC1)NC(C(C=C)C)=O 46804,c1(C(=O)NCC#CC)c[nH]nc1CCNC(C1CCN1C(C)(C)C)=O 46805,N1(CC)CC(NC(c2nc(C)c(C)s2)=O)C(C)C1.n12cc(nn1)CN1CC2C1 46806,C1(NC(CC(C=C)CC)=O)CCCCN(C(C2CC3(C2)CC2(CC2)C3)=O)CC1 46807,c1(NC(C2CC2Cl)=O)cccc(Oc2cccc(F)c2)c1 46808,Cc1cn2c(n1)C(C)N(c1nc3ccccc3nc1NC(c1cncs1)C)CC2 46809,c1(C(N2CCC(CN(C(C3CCN(C(C)=O)C3)=O)C3CC3)C2)=O)cnn2ccsc12 46810,N1(CC)CCCN(Cc2nc(Br)nn2CC)CCC1 46811,N1(C(CCCOCCOCC)=O)CCC(C)N(C(=O)C(C)SC2CC2)CC1 46812,C1(N)CCCC(C)CC1.C(=O)(C(C)(C)C)OCC(=O)NC1CC(CSC)C1 46813,c1(C(N2CCC(C)(CNC(CN3CC(CC)C3)=O)C2)=O)ncc(Br)cc1F 46814,n1(CCCOCCC2(C(N(C(C)(C)CC)CC)C)CCC2)cc(C#N)cn1 46815,c1(OC)cc(F)cc(C(=O)NC(C)(C)CNC(c2cn(C)nn2)=O)c1N 46816,c1(C(N(CC(CN(C(c2c(SC)cccn2)=O)C)O)C)=O)ccc(Cl)c(C)c1O 46817,N1(C(c2cc(OC)n[nH]2)=O)CC(NC(C2(CO)COC2)=O)CC12CCOC2 46818,CC(C(=O)N1CC(C(C)NC(=O)CSCc2ccccn2)C1)C(C)(C)C 46819,c1(N2CC(C(=C)C)OCC2)cccc(S(=O)(=O)NCC2CC23CCCCC3)n1 46820,C(CCCCNC(=O)C(C1CCOCC1)F)NC(=O)C=C1CCC1 46821,N1(C(C(=O)NCCCOC)C2CC2CC)CCOCC1(C)C(=O)OC 46822,Cn1nc2c(c1C(N1CCCC(CNC(C3CCSC3)=O)C1)=O)CS(=O)(=O)CC2 46823,c1(CC(N2C(Cn3cc(C4CCN(C)C4)nn3)CC2)=O)ccc2c(n1)OCCO2 46824,C(=O)(C(C(C)C)c1cccc(Cl)c1)NC1CC(NC(CCOCC(C)C)=O)C1 46825,c1(CC(=O)NCCCC(C)NC(=O)C=CC2CCCO2)c(F)cccc1Cl 46826,CC1CN(C(=O)CCCNc2ccnn2C2CCC2)CCN1C(=O)OC(C)(C)C 46827,C1(CNC(=O)NC(c2ccc([N+](=O)[O-])[nH]2)C)CC(C)(C)CCC1O 46828,C1(C(=O)NC)CCN(C(=O)Cc2cccnc2)C1.c12sccc1CNC2=O 46829,CC1CCCC1C(=O)NCCOC1CCN(C(=O)C(c2ccc(Cl)s2)=O)C1 46830,c1(C(N2CC(CC)C(NC(=O)C#CC3CCOC3)C2)=O)cc(OC)c(C)c(OC)c1 46831,C1(OCC)CCC(CC(=O)NCCCn2cc(CC3CCS(=O)(=O)C3)nn2)CC1 46832,C(=O)(C1Cc2c(Cl)cccc21)N1C2CN(C(=O)C3CC3(C3CC(S(N)(=O)=O)C3)CC)C(C2)C1 46833,c1(C(C)C)c[nH]nc1C(=O)N(CCNC(c1cnn(C(C)C)c1)=O)CC1CC1 46834,C(C)(C)(CC(=O)N(C1CCCC1)CCCNC(=O)Cc1cc(C)ns1)OC 46835,C1(NC(CC#N)=O)CCN(C(c2cnc3n2CCS3)=O)CC12CCC2 46836,c1(C(N2CC3CN(C(CN(C)CC)=O)CC3C2)=O)cc2c(F)ccc(F)c2[nH]1 46837,N#Cc1ccccc1CCC(=O)NCC=CCNC(c1cccc(Br)c1Cl)=O 46838,CC1(NC(c2cnn(C3CC3)n2)=O)CCN(C(C2(n3ccnc3)CCCC2)=O)C1 46839,c1(C(=O)NCC2CN(C(C3C(C(C)(C)C)C3)=O)CC23CC3)cc2cc[nH]c2cn1 46840,N1(C(C(=O)NCCC2(C)CC2)CC2CC2(Cl)Cl)CC2CCCCC12C 46841,C1(NC(CCN(CC#C)C(C2CCOCC2C(N)=O)=O)=O)CC(CO)C12CCC2 46842,N1(C(c2c(C)c(-c3ccccc3)on2)=O)CCC2C(NC(=O)CNC=O)C2CC1 46843,C1(Nc2nccc(C)c2[N+](=O)[O-])CC(NC(c2csc(Cl)c2)=O)C12CCOCC2 46844,N1(C(c2ncn(C)c(=O)c2)=O)CCC(CNC(=O)CC2COCCO2)C(F)(F)C1 46845,c1(C(N2C(c3nnc(CC)o3)C(C)(C)C2)=O)cc(OC)cc(Br)c1C 46846,CC(C)CCC(C(=O)NCc1ncn(C)n1)NC(C1CC2(CCCO2)C1)=O 46847,C12CCCC1CNCC(=O)N2.C1(C(C)N)CC1.C(C)(C)(C)OC(=O)N 46848,c1(C(=O)NCC2CC(C)N(C(c3cccc(CO)c3)=O)C2)ccc(Cl)c(C#N)c1 46849,c1(CC)cscc1C(=O)NC1CC1NC(=O)CCCNC(=O)NC1CCCC1 46850,c1(N2CCC(NC(C(CC)C)=O)C(F)C2)nc(C)nc(C)c1F 46851,c1(NC(C=CCOC)=O)c(F)cc(F)cc1Br 46852,C1(C(=O)Cn2cc(C(=O)O)nn2)(OCC(O)Cc2ccccc2)CCCCCC1 46853,CCC(CN1CCOCC1)N=c1[nH]c2c(c(=NCC=C(Cl)Cl)[nH]1)COC2 46854,Cn1c(C(=O)NCC2COCC2NC(c2c[nH]nc2C(F)F)=O)nnc1S 46855,N1(C(c2nc(NC(C)=O)sc2)=O)CC(C)(C)CCC1CNC(=O)C=C1CCC1 46856,C(=O)(CC1=CCCC1)N1CCC(CCNC(C=CC(C)(C)SC)=O)CC1 46857,c1(OC)ccc(CN2CCCC(C)(C(=O)N(C(C)COC(C)=O)C)C2)cc1C(C)C 46858,c1(C(N2CC(C)C(NC(c3cnc4ccccn34)=O)C2)=O)cc(F)c(F)c(F)c1 46859,C(=O)(CN=c1cc[nH]cc1)N1CC=C(C(=O)N2C(CC)CC(O)C2)C1 46860,c1(C(=O)NCCOCCCNC(c2n(C)ccn2)=O)cc2c(cc1O)CCCC2 46861,C1(c2n(C)ccn2)CN(C(=O)CC2CCC2)CC1NC(=O)CCC1CCOC1 46862,c1(C(=O)NC2CC(C(C)NC(C(COCC)(C)C)=O)C2)ccnc(O)c1Br 46863,CCCCCCCC(O)CC(=O)N1CCNC(C(=O)NCc2cccc(F)n2)C1 46864,C(=O)(C(C)(C)C(C)(C)O)NC(C)CC1CN(C(=O)COc2ccccc2)C1 46865,c1(C(=O)NC2CC(OCC(=O)N(CC(COC)C)C)C2)cccc2c1OCO2 46866,C12(CNC(c3c(CSC)cccn3)=O)CCC(CC1)N2C(C1CC=CCC1)=O 46867,c1(OC)ccc(F)cc1-c1cscc1C(=O)NCCCCCC(C)C 46868,C1(C)(CC)CC(NC(=O)CC2CCCCC2)CN1C(=O)CC1(OC)CCOCC1 46869,CC(CC(=O)N1CC=CC(NC(C2(C)CCC(=O)NC2)=O)C1)C(F)(F)F 46870,N1(C(C(C)C2CCCC2)=O)CCC2C(CCN2C(c2cccc3ccnn23)=O)C1 46871,CCC(CC(F)(F)F)N=c1[nH]c(=NCC2(CO)CCN(C)CC2)c2[nH]ccc2[nH]1 46872,C1(NC(CCCC)=O)CC2CCC(C1F)N2C(c1ccc2c(c1)CCN2)=O 46873,C(=O)(C1=CC2(CCOC2)C1)N1CCC(NC(C(COC)N(C)C)=O)C(F)C1 46874,C12(C(=O)NC(c3onc(C)n3)C)CC(CCO1)N(C(=O)C=Cc1ccsc1)C2 46875,c1(C(N(C2CN(C(=O)OC)C2)C)=O)ccc(C(C)C)cc1F 46876,N1(C(=O)NC(C2CCC3CC23)C)CCC(n2cccn2)(N(CCN=[N+]=[N-])C)CC1 46877,c1(CCNC(=O)Nc2ncn(-c3ccccc3)n2)cn2ccccc2n1 46878,N12CCN(CC1)C(=O)CC2=O.C(c1c[nH]cn1)=CC(N1CC(C(C)C)C1)=O 46879,c1(OC)cc(C(N2CCC(C)(NC(=O)CC3CCC3(C)C)C2)=O)ccc1F 46880,OC1CC(CCO)(N(c2ccccc2)C(Cc2ccccc2)C(=O)O)C1 46881,C=CC1(c2cn(CCCCO)nn2)COCCN1C(C1(CC(C)=O)CCCC1)=O 46882,C1(NC(C2CCC2)=O)COC2(C1)CN(CC1CCCS(=O)(=O)C1)C2 46883,c1(CC)sc(C(=O)NCC(C(C)C)NC(=O)CCCCN(C)C)cc1C 46884,C1(NC(c2ccc(Cl)nn2)=O)CCCN(c2ccccc2)C1 46885,C1(NC(c2cnsc2)=O)CCC2CN(C(C3CC3(F)F)=O)CCC2C1 46886,c1(OC)ccc(CCC(N2CC(CNC(C3CCCO3)=O)C(F)(F)C2)=O)cc1Cl 46887,C(CNC(C1C=CCCC1)=O)(CC(=O)NCc1n[nH]c(C)n1)OC 46888,N1(C(c2cnc(OC)s2)=O)CCC(NC(c2ccn3ccnc3n2)=O)C2(CC2)C1 46889,[N-]=[N+]=NCCCCCC(=O)NCC1CCC(CNC(C2(CCF)CCC2)=O)CC1 46890,CC1(C)CCC(C(=O)NCCC2COCCN2C(C23COC(CF)(C2)C3)=O)CC1 46891,CCC(C(=O)N(C)CCc1cn(-c2ccnc(C)c2)nn1)C(C)(C)CC 46892,C1(O)(CNC(C2(C#C)CCCCC2)=O)CCCN(C(C2(NC(C)=O)CC2)=O)CC1 46893,C(CC1=CCN(C(C2CCCS2(=O)=O)=O)CC1)NC(=O)CCC1CCC(=O)N1 46894,C(=O)(CCCC(=O)N(C)C)N(CCNC(CSc1nc(C)[nH]n1)=O)C(C)C 46895,CCC(C)(CCC(C)C)C(=O)NC1COCC1NC(c1cncc2nc[nH]c12)=O 46896,CC(O)CCCCCC(=O)N(C1CCCCN(S(C)(=O)=O)C1)CC1CC1 46897,C=C(C)CCCC(=O)N(C1CCN(C(c2ccncc2Br)=O)CC1)CCO 46898,CC(C)(C(=O)NC1CCSC12CN(C(c1cc(CO)on1)=O)C2)S(C)(=O)=O 46899,c1(C(N2CC(CNC(CN3CC(=O)NC3=O)=O)OCC2)=O)cnn2c1OCC2 46900,CC1=C(C(=O)N2CCN(C(c3cscn3)=O)C(CCO)C2)CCS1(=O)=O 46901,S(=O)(=O)(c1cn(C)c(C)n1)NCC(N1CC2(C(NC(C=NOC)=O)CC2)C1)=O 46902,Cc1c(C(=O)NC(C)(C)C(C)NC(=O)C(C)CC(F)F)nn(C)c1N 46903,N1(C(C(F)=CCC)=O)CCC12CN(C(=O)COc1c(C)cccc1Br)C2 46904,C(CCCCC(=O)N(C)CCC1CCCCC1)NC(C(C)CC1CCCC1)=O 46905,CC1COC2(C1)CN(C(=O)C(C1CC=CCC1)NC(c1nnc(S)n1C)=O)C2 46906,N1(C(COCCCCC)=O)CCCC1CNC(=O)CCSCC1CC1CF 46907,c1(CCC(=O)N(C2CCN(C(c3cc(C)c[nH]3)=O)CC2)CC)cc(F)ccc1F 46908,CC1(C(=O)NCC2(C(N3CCN(CC(N)=O)CC3)=O)CCCCC2)CCC2CC12 46909,C1(C(N2CC3C(CNC(c4ccc(=O)oc4)=O)(CC3)C2)=O)CN2CCCC2CO1 46910,c1(OC)cc(C)sc1C(=O)NC(C1CN(C(=O)CCCC2CCCC(=O)N2)C1)C 46911,C1(=O)CCCCCO1.c1(NC(C2CC(=O)CN2C(C)=O)=O)cc(O)nc(Cl)c1 46912,c1(OC)c(C(=O)NCC(O)CNC(c2cnc(C(C)O)s2)=O)csc1Cl 46913,c1(CC)c(C(N2CCOC(CNC(C3Cc4cscc4C3)=O)C2)=O)cccc1F 46914,C(=O)(C(C#N)C(C)(C)C)N1CCC(CC)(NC(=O)COCCN(C)C)C1 46915,C1(C(=O)NCC(C)N(C)C)(C(=O)OC(C)(C)C)CC=CC1.C12(CC1)C(=O)NC2 46916,C(c1ccc(F)cc1F)=CC(=O)NCC1(OC)CCN(C(C2CCC2)=O)C1 46917,C(=O)(C(O)c1ccco1)N(CCOCCCNC(C1C(C(C)O)C1)=O)C 46918,C1(NC(c2ccc(NC)nc2)=O)CCC(C)N(C(=O)CCSC)C1 46919,S(=O)(=O)(c1ccc2nc(C)oc2c1)Nc1c(C)cc(Br)cc1Cl 46920,C(=O)(C(O)C(F)(F)F)N1CC(O)(C(CNC(c2ccc(C#C)o2)=O)(C)C)C1 46921,C(CN=c1[nH]c(=NCc2cc(C)on2)c2sccc2[nH]1)C1C(C)=C1 46922,C(C(=O)N1CCCO1)NC(CC1CC(NC(=O)CCc2nncs2)C1)=O 46923,c1(CC(=O)NC2C(CNC(c3cc(OC)n[nH]3)=O)C2)cccc(C)c1Cl 46924,C(C)(N=c1[nH]c(=NCC(C)c2nccs2)c2ncccc2[nH]1)c1nc(C)[nH]n1 46925,C1(CCC)CC=CCN1C(C12CC(n3cc(CO)nn3)C1C2)=O.C1(=O)C(C)(F)CN1 46926,C1(NC(c2cnn(C(F)F)c2)=O)CC12CC(NC(=O)C(O)CC1CCCCC1)C2 46927,Cc1csc(=NCC(=O)N2CC3C(CNC(=O)CSC4CCCCO4)C3C2)[nH]1 46928,C1(NC(c2ccc(CC)[nH]2)=O)CCN(C(c2cc(CCC#N)oc2C)=O)CC1F 46929,c1(C(=O)NCC2CCCN2C(C=CC(C)(C)SC)=O)ccc(SC(C)C)cc1 46930,N1(C(CC(=O)OC)=O)CC2CC1C2NC(c1nscc1Br)=O 46931,C1(C(N(C2CC(OC)C2)C)=O)C2CCC1(c1cccnc1)C2 46932,N1(C(Cc2ccn(CC)n2)=O)CC2(CCC(CNC(=O)CC(C)n3cccn3)O2)C1 46933,CS(=O)CCCCNC(C1CCC(C)N1C(c1ccncc1O)=O)=O 46934,C#Cc1cnc(NCC(CNC(=O)C(c2ccccc2C)C)CO)nc1 46935,c1(C(=O)NCC2CN(C(C(C(C)C)F)=O)CC2C)ccc(C(N)=O)c(F)c1 46936,C(C1=CCN(C(c2ccnc(C(=O)OC(C)(C)C)c2)=O)CC1)NC(C(CC)F)=O 46937,C(C(C)C(F)C(=O)Nc1cccc(Cl)c1)NC(c1c(OC)nn(C)c1)=O 46938,Cc1ccnc(C(=O)NCC(C2CCCC2)NC(c2conc2C(C)C)=O)c1N 46939,C(CCC(O)C(=O)N(C(CC)CO)C)NC(CCN(CC)CC)=O 46940,C1(C(=O)NC2C(C(=O)NCCOC(C)C)COC2)CC2(CCCO2)C1 46941,N1(C(C(=O)NC(C)C)=O)CCC2(CC1)CC2NC(=O)CC(C)OC 46942,Cc1cc(C(N2CC(CCO)(NC(=O)C(C)SC(F)(F)F)C2)=O)cnc1C 46943,Cn1ccc2cc(C(=O)NC34CCN(C(=O)CCCC(F)(F)F)CC3C4)ccc12 46944,C1(N(C)C(C2CCC(=O)NC2)=O)(C(=O)NC2C=CCC2)CCOCC1 46945,c1(C(=O)NCC2CCC(NC(C3N(CC)CCC3)=O)C2)c(C)ccc(F)c1N 46946,C1(CC(=O)N(c2ccccc2)C2(C(=O)C3CC3)CC2)CCN(CC(F)F)C1 46947,CCCCCCCCC(C)CC(=O)NC1CCC1(C)C 46948,n1(C2CCN(C(=O)CC3CCOC3)C2)cnc2ccccc12.C1(N)CCOCC1 46949,C(=O)(C(C)P(C)(C)=O)N1CCC(N(C(CC(C)OC)=O)Cc2ccccc2)CC1 46950,c1(OC)cc(C)c(C(=O)NCC23CC2CN(C(=O)Cc2cnc(C4CC4)o2)C3)cn1 46951,C1(C(N2CC(CNC(C3(OCC)CCOCC3)=O)OCC2)=O)CC2C=CC1CC2 46952,N(C)(S(=O)(=O)N(C)C)CC(N1C(CN(C(c2ncn(C(C)C)n2)=O)C)CCC1)=O 46953,Cc1cccc(N)c1C(=O)NC1CC(NC(=O)CC2CCCC(C)C2)C1 46954,c1(OC)cc(C(=O)NC(C)CCCNC(=O)CCOc2ccccc2F)n(C)n1 46955,CC(C)CCCC(=O)NCC(CC(=O)N1C(CO)CC1C)C1CCC1 46956,C(=O)(CC(O)CC1CCCCC1)N(CC(C)NC(c1cc(Br)co1)=O)C 46957,Cc1cc(CS(=O)(=O)CC)ccn1.c1ccccc1F 46958,N1(Cc2ccc(OCC)cc2C(F)(F)F)CCCN(C(c2sccc2Br)=O)C(C)C1 46959,CCC1=NOC(C(=O)NC2CC(NC(C3(CC(=O)N(C)C)CCCC3)=O)C2)C1 46960,c1(C(N2CCCC3CNCCC23)=O)c[nH]c2ccc(F)cc2c1=O 46961,N1(C(c2c(OC)ncnc2C)=O)CCC(C)N(C(c2cc[nH]c2)=O)CC1 46962,Cc1ncc(C(N2CC(C(=O)NC(C)(C)CO)C3(CC3)C2)=O)cc1C#N 46963,C1(NC(c2cccc(C)c2)=O)CC2CC(NC(c3[nH]nc(N(C)C)c3Cl)=O)CC12 46964,C1(C(N(C2CCCCN(C(=O)Cc3ccc(Cl)s3)C2)C)=O)CC2CCCCCC12 46965,C=CCC(C)C(C)(c1nnnn1CCOC)NCCc1c(C)noc1C.C1(C)CC1 46966,CC1CCN(C(=O)CC2(Oc3ccon3)CC2)CC1NC(=O)CNS(=O)(=O)C1CC1 46967,C(C1=NOC2CN(C(c3cncnc3)=O)CC12)NC(c1cc(C)c(C)nc1O)=O 46968,c1(CC(N2CC(NC(C=C(C)C(C)C)=O)C(C)C2)=O)cn2ccsc2n1 46969,N1(C(CC=CCNC(c2csc(Cl)c2)=O)=O)CCCC2(CC2)C1 46970,C1(C(=O)NC2(C(=O)OCC)CC2)CCCC(NC(C2CC2CC)=O)CC1 46971,C#CC1(CNC(=O)C(C)NC(=O)C(CCC)OCC)CCCC1 46972,C1(C(=O)NCC2C3CN(C(C(n4ccc(C)n4)C)=O)CC32)CCN2CCOCC12 46973,c1(OCCC)cc(Cl)cnc1NCCC(C1CCCCO1)=O 46974,C(=O)(C(CC1CC1)NC(=O)CC(O)C1CCCC1)NC(c1nc(CO)n[nH]1)C 46975,CC1CC(C)(C(N2CCC(C(N3CCOC(C(N)=O)C3)=O)NC2=O)=O)CC(C)O1 46976,N1(C(C(=O)NC)=O)CC(C(=O)N(CCCOC2CC2)C)C(C2CC2)C1 46977,CCC(C(=O)N1CC2CC1C2CNC(c1cccc(F)c1C)=O)C(C)O 46978,c1(OC)ccc(CC(=O)N(CCNC(c2ncccc2O)=O)CC)cn1.C1CO1 46979,N1(C(c2cn(CC=C)nc2)=O)CCC(NC(=O)C(F)C(C)(F)F)CC1C 46980,N1(C(c2nncc(OC)c2)=O)CCC(N(C)C(C2SCCS2)=O)C(C)C1 46981,C1(C(=O)NCCN(C(C)C)C(c2nccc(N)c2Cl)=O)CCCC2(CCC2)O1 46982,N1(C(C(C)(C)NC(=O)OC)=O)CCC(NC(=O)C(C)(C)C)C(O)C1 46983,C1(CC(=O)NC2CC(CNC(CCCNC(C)=O)=O)C2)COCC(C)(C)O1 46984,N1(C(c2c(C)c(F)ccc2O)=O)CC2(C1)CN(C(C1(CN(C)C)CC1)=O)CCO2 46985,C(CN=c1[nH]c(=NC)[nH]c(=NCCCCOCC2CC2)[nH]1)N(CCCC)C 46986,N1(C(CC2(NC(C)=O)CC2)=O)CCOC(CN(C)C(c2cc(Cl)n(C)n2)=O)C1 46987,c1(OC)cccc(=NC(=O)Cc2nc(C(=O)Nc3cc(Br)c(C)cc3F)cs2)[nH]1 46988,c1(OC)ccc(OC)c(CCC(=O)OCC(C)(O)COCc2ccco2)c1 46989,C(N=c1[nH]c(N2CC=C(C)CC2)nc2ccccc12)c1ccc(C)cc1Br 46990,n1(CC)ncc2cc(NC(C3CCN(C(=O)Cc4ccc(Cl)cc4)C3)=O)ccc12 46991,CC1CC(C)(C(=O)N(C)CCOCCN(C)C(c2csc(O)n2)=O)C1 46992,CCCCCCCC(=O)N1CCCC1C(C)NC(c1c(Br)c(C)nn1C)=O 46993,C1(C(=O)NC2(COC)CCN(C(C3CC4CC4C3)=O)C2)CCC(=C(F)F)CC1 46994,C1(CC=C)(NC(C2CC2(F)F)=O)CC2CCC(C1)N2C(=O)CCc1c(C)noc1Cl 46995,C1(NC(CSCCC)=O)CCC2(CC1)CCN(C(=O)Nc1csc3cncn13)C2 46996,C(C(O)C(F)(F)F)N(C(CC1CC(NC(CNC(=O)NC)=O)C1)=O)CC 46997,c1(CCC(=O)NC2CC(C)N(C(=O)CC#N)C2)cc(F)ccc1Br 46998,N1(C(C2CCN(C)C2)=O)CC=CC(C(N2CCN(CC(N)=O)CC2)=O)C1 46999,C1(C(N(CC#C)CC#C)=O)CC2CC2N1C(C1CC=C(C)CC1)=O 47000,N1(C(CC2CCC(NC(CCC3CCN(C)CC3)=O)C2)=O)CCCC(F)CC1 47001,C(=O)(C1=NOC(C(C)(C)C)C1)N1C(CCN(C(=O)CSC(F)F)C)CCCC1 47002,N1(C(CCCC=C)=O)CCC(C2CC2)(CNC(=O)CC2C(C)(C)C2(C)C)C1 47003,C=C(C)CCCC(=O)NC12CC(NC(c3cc(C4CCOCC4)[nH]n3)=O)(C1)C2 47004,c1(C(=O)OC)ccc(COC(C2(CF)CC2)=O)c(F)c1.C(=O)OC 47005,N1(C(C(=O)NC)=O)CCCC(NC(N)=O)C1.C12(CC1)C(=O)NCCNC2=O 47006,c1(CCC)cc(C(=O)N(CC(C)CNC(=O)CC(CC)C2CC2)C)ccn1 47007,Cn1ncc(C(=O)NC2CCCCC2C(=O)NOCCc2ncccn2)c1Cl 47008,c1(C(C)C)nnc(SCCCCCN2CCOCC2)n1-c1ccc(F)cc1 47009,C1(C(=O)NCC(CNC(CC(C(C)=O)C)=O)O)CC(c2ccccc2)=NO1 47010,C1(NC(C=CC(C)(C)CC2C(CC(=O)OC)C2)=O)CNC2CC2C1 47011,c1(C(=O)NC2(O)CC(C(=O)NC3(CC(=O)OC)CCC3)C2)cc(C)oc1C 47012,c1(CC)nsc(N2CC(OCCNC(C3(CC)CC3(F)F)=O)C2)n1 47013,N1(C(CC)C)CC(CNC(=O)C(c2ccccc2)N(C)C)C(F)C1 47014,c1(C(=O)OC)coc(C=CC(=O)NC2CCC(N(C)C(c3snnc3C)=O)C2)c1 47015,C1(CN(C(=O)CC(C2CC2)C2CC2)C)CCCN1C(C1(c2n[nH]c(O)n2)CC1)=O 47016,C1(NC(CS(CCC)(=O)=O)=O)CCC2CCN(c3cncc(Cl)n3)C1C2 47017,c1(C(=O)NC(CNC(C2(SC)CC2)=O)C)ccc(-c2ccccc2)s1 47018,C1(n2cc(CC(C)(C)CN)nn2)CCC(NC(c2sccc2Cl)=O)CC1 47019,c1(C(N(CCCCNC(c2csc(-c3ccsc3)n2)=O)C)=O)cncc(F)c1 47020,C1(C(=O)NC(C2(O)CN(C(c3ccnnc3S)=O)C2)C)CCCC1(F)F 47021,CCN=c1[nH]cc(C(=O)N(CCCNC(C2CC2[N+](=O)[O-])=O)C)s1 47022,C1(CNC(C=C(C)C(C)(C)C)=O)CN(C(=O)Cn2cc(Br)cn2)C2CC12 47023,CC(C)(C#N)CC(=O)NC1CC(NC(C2CCC=CCC2)=O)C(O)C1 47024,c1(C(=O)O)cccc(-c2cn(C3CN(C(C4CC=CC(F)C4)=O)CC3O)nn2)c1 47025,C1(CC)CCOCCN1Cc1nc(Cl)cs1 47026,c1(OC)ccc(CN2CCC(=CC=CCNC(=O)OC(C)(C)C)CC2)c(F)c1F 47027,C1(CC)(CC)CC(NC(C2CCCOCC2)=O)CN1C(c1ccc(OC)cn1)=O 47028,N1(C(C(C)NC(=O)Cn2cnnn2)=O)CCCC(O)(CNC(C2(C)CC2)=O)C1 47029,c1(C(=O)NC(C)C(C)C(N2CCSCCC2C)=O)ccnc(O)c1F 47030,Cc1cc(C(N2CCN(CC3CC3)CC2)C(=O)NC2CC2)cc(F)c1 47031,C1(S(C)(=O)=O)(C(=O)NCC(C)(C)NC(C(C)CC(C)(C)C)=O)CCCCC1 47032,N(C1CC(C)(C)c2ccccc21)Cc1c(Br)cc(OC)c(OC)c1 47033,c1(C(N(CCCNC(CC2(C#N)CC2)=O)C2CC2)=O)cc(S(C)(=O)=O)cs1 47034,C(=O)(C(C(C)(C)O)NC(C1CC1(Cl)Cl)=O)N1CC(C)C(O)C1 47035,CCC1=C(C(=O)NCC(F)CNC(=O)CCCOC(C)(C)C)SCCO1 47036,C1(C(=O)NCCCN(C(c2ccc(=O)oc2)=O)CC)CCN(C2CC2)C1=O 47037,n1(CC(=O)N(C(CCC)C)CCOC)cc(C2COCC2O)nn1 47038,c1(C(C(=O)N(C(C2CN(C(Cn3nnc(C)n3)=O)C2)(C)C)CC)C)cc(C)oc1C 47039,c1(C(C(=O)NCC2(O)CN(C(=O)C(C3CCCCC3)O)C2)F)cncc(F)c1 47040,CCCC(C(=O)N1CC(F)CC1C(=O)N(C)CCc1cnccn1)OC 47041,c1(C(N2CCC(O)(CNC(c3ccnc(CO)c3)=O)C2)=O)noc2ncccc12 47042,c1(C(N(C(C(=O)NCC2(CCC)CC2)C)C)=O)cn(C(C)C)nn1 47043,c1(OC(C)C)ccc(C(=O)NC(c2ccccc2)(C)CNC(C2CCCO2)=O)cn1 47044,c1(CC(=O)NCC2C3CN(C(CC(n4ccc(C)n4)C)=O)CC32)ccc(F)cc1F 47045,CN1CCC(C)(NCC(CC(=O)N2CCCC(C3CCC(=O)N3)C2)NC=O)C1 47046,Cc1ccc(CN2CCC(C(C)NC(c3ccnn3C)=O)CC2)c(F)c1F 47047,C12(CNC(c3n(C(C)C)ncc3)=O)CC1CN(C(C1CCCC1C(F)F)=O)C2 47048,C1(OCCC)CCN(C(c2cc(CCNC(c3n[nH]cc3Cl)=O)on2)=O)CC1 47049,C#CC1(CNC(C2CN(C(c3nonc3N)=O)CCO2)=O)CCCC1 47050,Cc1ccc(C(F)F)cc1OCC(N1CCSCC1C(=O)NC1CC1)=O 47051,N1(C(C(C)OCC=C)=O)CCC(F)(F)C(Nc2ncc3c(n2)N=N3)C1 47052,C=C(C)CC(C(=O)NC1CCCCC1(C)C)NC(c1cncc(O)c1)=O 47053,c1(OC)noc(C2CC2)c1C(=O)NCC1(NC(C2(C#N)CC2C)=O)CC1 47054,CN1N=C(C(=O)NCCCCC2CN(C(=O)Cc3cccc(F)c3)C2)CCC1=O 47055,N1(C(C(C)CC2CCC2)=O)CCC(C(C)(C)C)(N(C(=O)CNC=O)C(C)C)C1 47056,C1(O)(C(C)NC(c2coc(C(C)(C)C)n2)=O)CCN(C(c2csc(Cl)c2)=O)C1 47057,C12(C(=O)NC(C3CCCCC3)CC)CC(CO1)N(C(c1ccc(Cl)cn1)=O)C2 47058,N1(C(CCOCCNC(c2ccnnc2O)=O)=O)CCc2ccccc21 47059,N1(c2ncnc(OC)c2OC)CCc2cc(C(N3CCS(=O)CC3)=O)ccc2C1 47060,C=C(C)c1cccc(NC(C2CCCN(C(=O)C(C(CC)CC)OC)C2)=O)c1 47061,c1(N(C)CC2CCCN(C(C(c3cccc(C)c3)O)=O)C2)ncc(C)c(SC)n1 47062,c1(C(=O)NC(CC=C)CNC(c2ccc(F)n2C)=O)ccc(OC)c(F)c1F 47063,Cc1c(C(=O)NCC(C)CNC(=O)C2=CCCC2C)c(O)nc2ccccc12 47064,CC1(NC(c2coc(Br)c2)=O)CCN(C(c2ccc(C3(C)CCO3)cc2)=O)CC1 47065,N1(C(c2c(C)nco2)=O)CC(C)(CNC(=O)CC2CCCC(=O)N2)CC1(C)C 47066,c1(C(N2C(C)CCC(C(=O)NC(c3nncs3)C)C2)=O)cccc2c1CCC2 47067,C12(NCc3ccc(C)s3)CCC(C(=O)NCCC(C)CCO)(CC1)CC2 47068,CC(C)CC(C)(CNC(c1cccc(O)c1)=O)NC(c1ccn(C2CC2)n1)=O 47069,N1(C(C(c2cccs2)NC(C2CCSCC2)=O)=O)C2CCCC1COC2 47070,CC(C)(C)CC(=O)N1CCC(C(C)(O)CC2CCCC2)CC1 47071,C=C=CCC(=O)NCC1COCC1NC(=O)CCc1cc(OC)no1 47072,c1(N(CC(C)N(C(Cc2nc(C)sc2C)=O)C)C)nc(Cl)ncc1Cl 47073,Cc1cc(-n2ccnc2)ccc1C(=O)NCCN(C(=O)C(F)C(F)(F)F)C(C)C 47074,C1(OC)CCCCCC1NC(=O)C(=O)NCCc1ccc(Cl)c(F)c1 47075,c1(C(=O)NCCCNC(=O)Cc2cnoc2)ccccc1SCCCO 47076,Cc1cc(=NCC2(CCCO)CCCC2)[nH]c(NC(c2cccnc2)C)n1 47077,CN1CCC(n2cc(C3CCN(C(=O)Cn4cc(I)cn4)C3)nn2)C1=O 47078,CC(CNc1ncc(C2CCCN2C(=O)OC(C)(C)C)s1)(CO)CO 47079,C1(CC(=O)N(C2CCN(C(c3ncsc3C)=O)C2)CC)CCCC2CC12 47080,N1(C(C2(C#C)CCCC2)=O)CCC2(CC1)CN(C(=O)C(O)CCn1cncn1)C2 47081,c1(OC)ccc(F)c(-c2cncnc2C(N2CC3(CCC3)C2C(C)C)=O)c1 47082,c1(C(=O)NCC2C(NC(CC3(CC)CCC3)=O)C2)cn(C2CCCC2)nn1 47083,c1(N2CCCC(NC(C)C)C2)cccc(S(=O)(=O)NCc2n[nH]c(=N)s2)n1 47084,C1(C)(CNC(c2c(CC)con2)=O)CN(C(=O)CC(C(F)(F)F)OC)C(C)(C)C1 47085,C1(NC(CC2C3CN(C(CCC#CC)=O)CC32)=O)CCN(C)CC1(C)C 47086,C1(C(=O)NCc2nc(C)nc(O)c2)CC2(CCN1C(=O)C(F)F)CC2 47087,c1(CC)cc(C(=O)NC(C2CCN(C(=O)COC(C)C)C2)(C)C)c(C)o1 47088,C1(C)(C(=O)NC)CCN(C(C2C3CC3CN2C(c2ccon2)=O)=O)CC1 47089,N1(C(C2CC3CCC2O3)=O)CCOC2(CCN(Cc3nc(C4CC4)no3)C2)C1 47090,CC(C)C(CN(C)C)N=c1nc(N2CC3CCC3C2)c2c([nH]1)CCS2 47091,Cc1nc(Cl)[nH]c(=NC2CC(C)(NC(C3CC3c3cccnc3)=O)C2)c1F 47092,Cn1nc(C(N2CCC(NC(c3ccncc3)=O)C23CCC3)=O)c2c1CCC2 47093,CC(CC(C(=O)N1C2CCC1CC(F)(F)C2)N1CCOCC1)CC(C)(C)C 47094,C1(C(=O)NCC(=C)CCNC(=O)C(C)OC)CC(=O)N(C2CCCCC2)C1 47095,C1(OC)CN(C(c2ccccc2Br)=O)CC1NC(C1CCN1C1CCCC1)=O 47096,c1(NC(C(N2CCCC(C(C)=O)CC2)=O)=O)csc2ccc(Br)cc12 47097,Cc1cnc(NC(C2CSCCN2Cc2c(C)cccc2Br)=O)c(Cl)c1 47098,c1(C(N(CCCNC(C(CCCCCC)C)=O)C)=O)cc2n(n1)CC(C)NC2=O 47099,C(C(CC1CC1)C(=O)NC(C)(C)C(C)O)NC(Cc1c(C)occ1)=O 47100,C(=O)(CC(C(F)F)NC(c1n[nH]c(O)n1)=O)NCCC(CC)(C)C 47101,Cc1cc(C(=O)NCCC2CN(C(C3COCC(C)O3)=O)CCO2)n(C(F)F)n1 47102,C1(C)(COC)CCCN(C(=O)C(O)C2CN(C(c3cncc(CO)c3)=O)C2)C1 47103,CCC(C(C)O)NC(c1cc(CNC(C2(COC)C=CCC2)=O)cs1)=O 47104,C1(NC(c2cn3ccsc3n2)=O)CN(C(=O)C(F)(F)C(O)C2CC2)CC1C1CC1 47105,Cc1c(CNC(=O)NCC2(F)CCCCC2)cccc1F 47106,CS(=O)c1cccc(NC(c2noc(C(F)(F)F)n2)C(=O)NC2COC2)c1 47107,C=CC1(C2(C(=O)NCCCCN(C(=O)CSc3cccs3)C)CCC2)CCC1 47108,C(c1ccc(F)cc1)=CC(=O)NCC12CCC1CCN2C(=O)CC1CS(=O)(=O)C1 47109,CC1CC(NC(c2cncc(O)c2)=O)CCN1C(c1cccnc1Cl)=O 47110,Cc1[nH]c(C#N)cc1C(=O)NCc1cc(C(N2CC=CC(O)C2)=O)no1 47111,N1(C(c2c(C)ncnc2)=O)CCC(F)(C(=O)NCCC(O)C(C)C)CC1 47112,c1(OC(C(N2CCC(C)CC2)C(C)C)=O)ccc2cnccc2c1 47113,C(C(C(C)C(C)C)NC(=O)Cc1ncn2c1CCC2)NC(C1CCC(=C)CC1)=O 47114,C#CCCCCCCC(=O)N1CCN(C(=O)CCCSC)C2CC12 47115,N1(C(c2c(C)scn2)=O)CCC2(CC(NC(c3c(C)ncnc3C)=O)C2)C1 47116,C(CC(O)C(=O)NCCCCC(C)NC(c1ccc(NC=O)cc1)=O)SC 47117,N1(C(C(CC)(C)CC)=O)CCC2(NC(=O)COCCCC(C)C)CCCC12 47118,Cc1nn(C)c(C)c1S(=O)(=O)NCCC(=O)NCC(C)(C)NC(C1CC1C#N)=O 47119,C(=O)(C(C(C)C)NC(C)=O)N(CCCNC(=O)Cn1cncn1)CC 47120,c1(C(=O)NCC(c2ccccc2)NC(C2CNC(=O)C2)=O)cc2cccnn2n1 47121,C1(CCNC2CC(c3ccccc3F)(C(=O)NCC)C2)CC2CCC1C2 47122,C1(C2(NC(C3CC3F)=O)CC2)CCCN1C(C1COCCO1)=O 47123,CC(C(=O)Nc1cccc(C2CCOCC2)c1)N1C(=O)Cc2ccccc21 47124,Cn1cnc2c1CCN(C(=O)CC(C)(C)C)C21CCN(c2nnc(C#N)s2)C1 47125,C1(C)(CC(=O)NC2(C#C)CC2)CCN(C(=O)C(F)OC(F)(F)F)C1 47126,Cc1cc(C(F)F)nn1CC(N1CC(NC(C2(F)CCOC2)=O)CC1C)=O 47127,C=Cc1ccc(C(=O)N(C2CCCCN(C(C3(C(C)C)COC3)=O)C2)C)cc1 47128,c1(C(=O)NCC2CCCN(C(C(C3CCC3)OC)=O)CC2)nc2ccccn2n1 47129,C1(NC(=O)OC(CC)C)CCCN(C2CC(=O)N(Cc3ccccc3)C2=O)CC1 47130,N1(C(C(CCSC)(C)C)=O)CC2CC(C1)CN(C(C1CC3CC(=O)C1C3)=O)C2 47131,C1(NC(=O)C=CC2CCOC2)CC2(C1)CC2C(=O)NC1CCOC1 47132,C(CC(O)CC(=O)N(C1CCC(NC(=O)C(C)(C)C2CC2)CC1)C)SC 47133,N1(C(Cc2c(C)nccc2)=O)CCC(O)(CNC(c2ccc([N+](=O)[O-])o2)=O)CC1 47134,c1(Cn2cc(CSC)nn2)cccc(C(=O)NC(C2CCOCC2)C)c1 47135,N1(CCn2c(C)cc(C)n2)CCCC(NC(=O)CN2CCCCC2=O)CC1 47136,C1(CNC(C2(C#C)CC2)=O)CC(O)CN1C(=O)C(F)C1CCC1 47137,c1(C(C)=O)cc(C(=O)NCC23CC(NC(c4ccoc4C)=O)(C2)C3)n(C)c1 47138,N1(C(C(C)(C)NC(=O)NCC)=O)CC2CN(C(=O)C(C)CO)CC2(C)C1 47139,C1(C(N(CCCNC(=O)CSCc2ccncc2)C)=O)CCC(=O)N2CCCC12 47140,C1(NC(C2C(=C)C2)=O)C2CC3C1C3C2C(N1CCCC(F)C1)=O 47141,C12CCC(O1)C(=O)NC2=O.C1(NC(=O)C=CCN2CCC2)CC=CCC1 47142,CCC(N)CCC(=O)N1CCC1(C(=O)OC(C)=O)C(C)C 47143,C1(CNC(CCNC(=O)CC(F)(F)F)=O)CCN(C(=O)Cc2cscn2)CC1O 47144,c1(C(=O)NCCC2CC(NC(c3ccn(CCF)n3)=O)C2)ccc(F)cn1 47145,C(=O)(C(F)C(F)(F)C(F)(F)F)N1CCC(NC(c2onc(C)n2)=O)C12CCCC2 47146,C1(C(N(CCCCCCF)C)=O)CN(C(C2C3CCC(F)(F)C23)=O)CC1(C)C 47147,c1(OC)ncc(C(=O)NCCC2(NC(=O)CC(C)c3cccnc3)CCCC2)s1 47148,N1(CC(=O)NCC(CC=C)NC(c2ccc(=N)[nH]c2)=O)CCC(C)CC1 47149,C1(CC(C)O)CCCCN1C(=O)NCCNCCCn1ccnn1 47150,CC12CC(C1)C(C(N1CC(O)CC1CNC(C1(CO)CCC1)=O)=O)CO2 47151,N1(CCCNC(C(C)(C)C2CCC2)=O)CCN(C(=O)CC(C2CC2)C2CC2)CC1 47152,C1(NC(c2noc(C)c2C)=O)CN(c2ncc(Oc3ccccc3)cn2)CCN1C 47153,c1(OCC(N2CC(OC)C(NC(=O)CCN3CCC3)C2)=O)ccccc1[N+](=O)[O-] 47154,CCCCC(O)C(C)C(=O)N1CC2CCC(C1)N2C(c1cnn(C(C)C)c1C)=O 47155,O=C(N1CC(O)CO1)C1CC12CCN(C(c1cnn(C3CC3)c1)=O)C2 47156,c1(NC(COC2(C)CN(C(c3cc(CCC)[nH]n3)=O)C2)=O)cncnc1O 47157,c1(C(c2nnnn2C2CCOC2)NC2C(OCC)C2)cc(C)ccc1Cl 47158,C=CCCC(C(=O)NOCCC)NC(C1CC=CCC1)=O 47159,C(=O)(C1CCCn2cnnc21)N1CCC(CCNC(C2CC3CC3C2)=O)C1 47160,S(=O)(=O)(C(Cl)(Cl)Cl)N(CCC#C)CCCC.C1(C(=O)N)CC1C 47161,N1(C(Cc2c(C)nn(C)c2)=O)CCC(C)C(CC(N2CCC(C3CC3)CC2)=O)C1 47162,N1(C(C(CSC)O)=O)CC2CC(C(=O)NC(C)(C)C)C(C2)C1.C1C(=O)N1C1CC1 47163,CCCCC(C)CCC(=O)NC1CCN(C(C23CCC(C2)C3(C)C)=O)CC1 47164,C12(C(N3CC(CC=C)(CNC(=O)Cc4nccn4C)C3)=O)CC(CF)(CO1)C2 47165,N1(C(c2cn(COC)nn2)=O)CC(NC(=O)CN2CCC(C)CC2)CC(C)(C)C1 47166,C1(C(=O)NCC2CC=CC2)CCCN(C(c2ccccn2)=O)C1 47167,C(CNC(=O)CCCc1ncco1)(CC(=O)N1CCC(C(N)=O)C1)OC 47168,C1(NC(c2c(CC)cccc2)=O)CC2CN(C(=O)CCc3cn(C)nn3)CC12 47169,Cc1sc(C)c(S(=O)(=O)NC2CN(C)CC2C(F)(F)F)c1Br 47170,N1(C(=O)CCCN2CCCC2)CCC(C(=O)NCCCCOC)(CO)C1 47171,Cc1cc(-c2nc(CC(F)(F)F)nn2CCCn2cncn2)nc2ccccc12 47172,N1(C(C)C)C(=O)CCC1C(=O)OCCC1(C)CC1(F)Cl 47173,C(=O)(C1CCc2c[nH]nc21)N1C(C)C(NC(c2cccnc2C(N)=O)=O)CCC1 47174,C(=O)(C(C(C)(C)C)NC(=O)C(C)O)N(CC#CC)C 47175,c1(-c2cccc(C(=O)NC3CC3c3ccc(Cl)cc3)c2)ccc2c(c1)OCO2 47176,C(C)(C(O)C(=O)NCC1CCC(NC(c2n[nH]cc2Br)=O)CC1)OC 47177,N1(C(C(C)SCC)=O)CC(C2(NC(=O)C(C)C(C)(C)C)CC2)C1 47178,CCCCC(O)C(=O)N1CC2C(C(=O)NCCCn3cccc3)C2C1 47179,C1(C(=O)NC(C)CN(C(=O)CN2CCNC(=O)C2)C)OC2CCC1CC2 47180,c1(C(=O)NCC2(CNC(c3sc(C)c(O)n3)=O)CC23CCC3)c(O)cccc1Cl 47181,c1(NCC(N(C)C(c2ccncc2F)=O)C2CC2)ncc2scc(Br)c2n1 47182,N1(C(c2ccc(OC)nc2)C(=O)NCCCF)CC2C3C=CC(CC3)C2C1 47183,N1(C(CC=CCC)=O)CCCOC(CNC(C2(C)CN(CC)C2)=O)C1 47184,C1(C(N(C2CC(C(=O)NCC(C)OC)C2)C(C)C)=O)CCCC(=O)N1C 47185,N1(C(N2C3CC(C(=O)OCC)C2CC3)=O)CC2COCC(C1)C2(F)F 47186,O(C1CCOc2cc(F)ccc21)CC(N)(CC(F)(F)F)C(F)(F)F 47187,c1(C(N)=O)ccnc(NCCC2CCCCN2C(=O)CSc2ccc(Cl)cc2)n1 47188,S(=O)(=O)(c1ccc([N+](=O)[O-])cc1Cl)NC.C(C)(C)(C)NC(C1CC1CNC(=O)O)C 47189,C(CCCCCC(=O)NC1CCN(C(=O)CC(O)C(C)C)C(C)C1)SC 47190,C1(CCC)(NC(=O)CCC2CCOC2)CCCN(C(=O)CCCc2cnn[nH]2)C1 47191,C1(C(N(C2CN(C(C3CCC(=O)O3)=O)CC2(C)C)C)=O)COC(C)(C)CO1 47192,C1(NC(C2CC2(F)F)=O)CCCN(Cc2cnn(-c3ccccc3)c2)C1 47193,Cc1cc(-c2cn(CC3CCCN3Cc3ccccc3O)nn2)cnc1C(=O)O 47194,N1(C(C=CC(=O)OC)NC(c2ccnn2C(C)C)=O)CCC2(CO)CC2C1 47195,N1(C(c2c(N)cccn2)=O)CC(O)CCC1C(=O)NCC1CN2CCC1C2 47196,c1(C(N2C(CNC(CCN(C(CCC)C)C)=O)CCC2)=O)ccc2nonc2c1 47197,CC(C)(O)C#CC(=O)NCc1cccnc1CNC(C1CCN(C2COC2)C1)=O 47198,CC(C)C(C(=O)N(CC(C)CNC(C12CC(CC(F)F)(C1)C2)=O)C)n1cnnc1 47199,CC1(C)COC(C(=O)NC(C)(CNC(=O)CCN2CCCC2)C2C(C)C2)CO1 47200,N1(C(C(C=C)(C)C)=O)C2CCC1CN(C(c1nc(C3CC3)ncc1Cl)=O)CC2 47201,C1(CNC(c2ccc(COC)s2)=O)CN(C(c2n[nH]cc2Br)=O)CCO1 47202,N1(C(C)=O)CCCC1C(N1CC(CCCCNC(=O)C(F)=C2CCC2)C1)=O 47203,N1(C(C2(CC=C)CC=CC2)=O)C2CCC1C(CNC(C1(C)CCCCCC1)=O)C2 47204,C1(CCC)CCCC1C(=O)NCCNC(C1CCO1)=O.C1(C)CN1 47205,C1(C(=O)NCCc2cn(C)nc2)CN(C(C2CC2c2cnc[nH]2)=O)CC1O 47206,C1(C(N(C2CCCC2)CC)=O)CCN(C(=O)CC2CCCC2OC)O1 47207,c1(OCC(=O)NC2C(CNC(=O)C=CCF)C2)cccc(Br)c1 47208,N1(C(C(C)(C)F)=O)CCC2(C(=O)NCC3CCCC3)CC2C1 47209,C(=O)(C(CC(F)F)N(C)C(c1ccc(C#N)cn1)=O)NCC(C1CCCC1)C 47210,N1(C(c2ncn(C(C)C)c2)=O)CCC2(C(=O)NCC3CCC(F)C3)CC2C1 47211,C#CC1(O)CC(C(N2CCC(N(C(=O)CC(C)(O)C3CC3)CC)CC2)=O)C1 47212,C1(CC)(NC(=O)CN2CC=CC2)CCN(C(C2CCC(=O)N(CCOC)C2)=O)CC1 47213,C(=O)(CCC(C)CN(C)C)NC(CCC)CNC(=O)CCC1CC(OC)C1 47214,Cc1conc1CNC(C1CCC(CNC(c2nccn2C)=O)O1)=O 47215,C#CCCCC(C)(C)C(=O)NC1CN(C(C2CC3CC2CC3O)=O)C2CCCC12 47216,C1(C)(C(NC(CC2CC(N(C)C)C2)=O)C)CCN(C(C2CC2(F)F)=O)CC1 47217,Cn1ncc(C(=O)NC2COCC2CNC(C2CCC(=O)NC2)=O)c1Cl 47218,C1(C(N2CCCC(c3n(CC)cnc3)C2)=O)Cc2c(C)cccc2O1 47219,C12(CNC(c3c(C)c[nH]n3)=O)CCC1CCN2C(=O)CC1=CCCC1 47220,c1(NCC(N2CCC(NC(C3CCCSC3)=O)C(O)C2)=O)ccccc1[N+](=O)[O-] 47221,c1(CC)ncoc1C(=O)N(CCCC(=O)NCC(c1ccccc1)F)C 47222,c1(C(C)Nc2sc(N3CCCC3)nc2Cl)cc(O)ccc1Br 47223,C1(CC#C)(C(=O)O)CCN(C(CCCC)C(=O)NCC2CCOC2)CC1 47224,C(=O)(CS(=O)(=O)C(C)(C)C)N1CCC(CNC(c2c(CC)n(C)cc2)=O)CC1C 47225,C(=O)(C(O)C(C)OC)NCC(C)(C1CC1)NC(c1cc(OCC)no1)=O 47226,C1(NC(C2CCCC3(CCC3)C2)=O)Cc2ccccc2N(C(=O)CC2CCC2)C1 47227,N1(C(=O)CC2CCOC2)CCN(CCNC(C2CC3CC3C2)=O)C2(CCC2)C1 47228,C(=O)(CCCC(F)(F)F)N1CC(C(=O)NCCCOCC2CCC2)CC(C)C1 47229,C(CCC(C)C)(C(=O)NCC1CC(C)C1)NC(C1CC=C(C)CC1)=O 47230,C1(C(N2CC(CC)C(CO)C2)=O)CC2CN(C(=O)OC(C)(C)C)CC2C1 47231,C1(CNC(CCC(=O)NC)=O)CCN(C(=O)CCSc2nnnn2C)C12CCC2 47232,c1(CNC(N2CCC(=CCc3nn[nH]n3)CC2)=O)n[nH]c2c1CCOC2 47233,c1(OC)cc(C=CC(=O)NCC2CC2NC(C2(c3cc[nH]n3)CCC2)=O)sn1 47234,C1(N(C2CC3CCC(C2)N3)CC(=O)OCC)CC12CCCCC2.C1C(=O)N1 47235,N(C1CCc2cccnc21)C(CCOCCNC(C1CN2CCC1C2)=O)=O 47236,C1(NC(C(C)NC(=O)Cn2cnnn2)=O)CCC(NC(c2scnc2C2CC2)=O)C1 47237,c1(C(N2C(C)CN(C(=O)CC#N)CC2)=O)cccc2c1CC(=O)N2C 47238,C1(C(=O)NC2C(NC(c3n(C)cc(C#N)c3)=O)CCC2)CCc2nccn2C1 47239,C(=O)(C(C)CC(C)C)N(CCCC(=O)N(CCC)CC)C(C)C 47240,c1(NC(c2c(CNC(C3(C)CC(F)C3)=O)cc[nH]2)=O)ccc2c(c1)CCC2 47241,c1(C(N(CC(C)CNC(=O)COCC2CCOC2)C)=O)cnn(C)c1F 47242,C=CC(C)(O)C(=O)N1CCC(CNC(c2ccc(CN(C)C)nc2)=O)(OC)C1 47243,C(=O)(C(F)(F)C(F)(F)C(F)(F)C(F)F)NCCC(=O)N(C1CC(C(N)=O)C1)C 47244,N1(C(c2c(C)nc(O)s2)=O)CCC2(CC(NC(c3ccnn3C3CC3)=O)CO2)C1 47245,C=C(C)C1OCCC1CNC(=O)CC1(NC(C2CCC(=O)O2)=O)CCC1 47246,C(CCC(C)CC(=O)NC1CC(CNC(=O)CC2CCC(C)(C)CO2)C1)=C(C)C 47247,c1(CC(C)C(=O)N2CCC(NC(=O)Cc3cccs3)C2)cccc(Cl)c1 47248,CC1CN(C(=O)C(C)Cc2cnn(C)c2)CC1NC(c1ncccc1C1CC1)=O 47249,N1(C(CC2C=CC(NC(c3c(C)cc(C)s3)=O)C2)=O)CC2(CCC(=O)O2)C1 47250,C#CCCCC(C)C(=O)N1CCC(C)(CNC(c2c(F)ccc(OC)c2F)=O)C1 47251,c1(C(C)C)ccc(C(=O)NCC(C)NC(=O)CCC2CCC(O)CC2)cn1 47252,c1(CN(C)C)ccc(C(=O)NCC2CCCCN2C(C2CC3CCC2O3)=O)cc1 47253,c1(OC)ccc(C(=O)NCC2(NC(c3c(N)cccc3Cl)=O)CC2)c2ccoc12 47254,N1(C(C2CC(NC)C2)=O)CC(CCNC(=O)CN2CCNC2=O)CCC1C 47255,C12(CNC(c3n[nH]cc3I)=O)CC1CN(c1ncc(I)cn1)C2 47256,Cc1c(C(=O)NCC(C2CCOC2)NC(=O)C(C)(C)NC(C)=O)nnn1C 47257,C(=O)(Nn1cccn1)C1(F)CN(NC(=O)Cc2ccccc2F)C1 47258,C(=O)(C(C#N)C(C)C)NCc1c(C(=O)NC(c2c(C)ccnc2)C)scc1 47259,c1(NC(C2N(C(C3COCC3C(N)=O)=O)CCC(=C)C2)=O)cnc2c(c1)CCC2 47260,Cc1ccc2c(C(N3CCC(CCNC(=O)CC(O)C(C)C)C3)=O)c[nH]c2c1 47261,c1(C(C(=O)NC2CN(c3ccccc3)C2)NC(C=C(C)C)=O)c(Br)cnn1C 47262,N1(C(C2(C#C)CCN(C(=O)C=CC3CCC3)C2)=O)CCCCC(C)(F)C1 47263,N1(C(c2ccc(C(C)=O)o2)=O)CCC(CNC(=O)CCC2CCOCC2)(OC)C1 47264,C1(C(N)=O)CC(C(=O)NCCCNC(=O)CSCC2CC2)=NO1 47265,N1(C(C(CNC(c2n(C)c(C#N)cc2)=O)CC2CC2)=O)CCC2(CCCCO2)C1 47266,N1(C(C(n2c(C)ncc2)C)=O)CC(C(=O)N(CCN=[N+]=[N-])C)C(C)C1 47267,C1(C(=O)NC2(C)CC(NC(C3CCC(C)CC3)=O)C2)CCn2c(O)nnc2C1 47268,Cn1nccc1CCC(=O)NC1CCCC1NC(c1coc(Cl)n1)=O 47269,Cc1cc(=O)n(C)cc1C(=O)N(C1CCCCC1NC(c1ccnc(O)c1)=O)C 47270,C1(NC(C(CC)C#N)=O)CC(O)(C2CCN(C(=O)CCc3csc(C)n3)CC2)C1 47271,N1(C(c2cc(COC)on2)C(=O)NCC(F)F)CC2CC2(CO)C1 47272,n1(CC(=O)Nc2c(F)cc(Br)cc2Br)ccc(=NC(=O)C2CC3CCC2O3)nc1O 47273,c1(C(N2CCC(NC(c3cc(C(F)(F)F)ccc3O)=O)C2)=O)cn2c(n1)CCC2 47274,C1(C(=O)OC)CCCC2CCCCC12.C12(C(=O)OCC)CN3C(C1)(C2)C3 47275,N1(C(C(CC#C)(C)C)=O)C2CCC1C1CC1(NC(C1CCC(=O)N1C)=O)C2 47276,c1(C(C(=O)NC23CN(C(C(C)O)=O)C(C2)C3)=O)cc(F)ccc1F 47277,c1(C(N2CC(CNC(=O)CC3CCOCC3)(OC)C2)=O)nc[nH]c2nccc1-2 47278,N(C(=NCc1ccccc1F)NC1CC(=O)N(CC(F)(F)F)C1)CC(CC)OC 47279,N1(C(CC(=O)OCC)=O)CC2(CCCC2)C1C(=O)NC(c1nccn1C)C 47280,C1(C2(NC(CN(C)C3CC3)=O)CC2)CCCCN1C(=O)CCn1ncn(C)c1=O 47281,S(=O)(=O)(c1cc(C)cnc1NCC(O)CF)NC(C(CC)C)C 47282,CC(C)C(CC(=O)N1CC(NC(C2CC2NC(=O)OC(C)(C)C)=O)C(C)C1)C(C)C 47283,C1(OC)CN(C(C2CCCN2C)=O)C(C)(CNC(c2cc(F)c[nH]2)=O)C1 47284,C(C)(C)(CC(=O)NCCCC(N1CCC(O)(C(C)C)C1)=O)OC 47285,C1(C(=O)NC(C)CN2CCN(C(c3ccon3)=O)CC2)CC12CCCCC2 47286,c1(C(=O)NCC2C(NC(C=C(COC)C)=O)CCCC2)cc(OC)cnc1F 47287,C1(CCOC)(NC(=O)C(N2CCNC2=O)C)CCN(C(C2CCC(O)C2)=O)C1 47288,c1(C(=O)NC(CNC(c2cnc(CC)s2)=O)C(C)C)cnn2ccnc(N)c12 47289,N1(C(c2ccc(C(C)C)nc2)=O)CC2=C(C1)CN(C(=O)Cc1cc[nH]n1)C2 47290,C1(C(=O)NC(CCC)C(=O)NC)CC2(CCC(F)(F)CC2)CO1 47291,C(=O)(C#CC1(CC)COC1)N1CC2CCC(NC(c3cc(OCC)no3)=O)C21 47292,c1(CC(=O)NC2(C3CN(C(C(C)(C)CF)=O)C3)CC2)c[nH]c2ccc(F)cc12 47293,C#CCCCC(=O)NCCN(C(=O)C=CCCC(CC)=CC)CCOC 47294,C1(NC(C2CCCOC2)=O)CC2(C1)CC(C(=O)NCC(O)C(F)F)C2 47295,CC1(F)CN(C(=O)C(C2CCCOC2)O)CCN(C(=O)CC(O)CCC2CC2)C1 47296,C(=O)(C1CCCn2cnnc21)NCCC1N(C(c2ncn(CC)n2)=O)CCSC1 47297,c1(CCC(=O)NC2CC(NC(C(C)CSC(F)(F)F)=O)C2)ccc(O)nn1 47298,Cc1ccc(N)c(C(N2CC(C)CCC2CNC(c2cc(C)c(C)s2)=O)=O)c1 47299,C(=O)(C(C)(C)C1=CCN(C(=O)CCCCC(C)CC)C1)NC(CC)C(=O)OC 47300,c1(CNC(c2onc(CC)n2)C)cccc(Br)c1O 47301,C1(CNC(C=CC=CC)=O)CN(C)CCN1C(C1CCCN1CC(C)C)=O 47302,N1(C(=O)NC2(c3ccccc3F)CC2(F)F)CCc2c(OC(F)(F)F)cccc2C1 47303,c1(C(N(C2CN(C(=O)C(O)c3ccco3)C2)C)=O)ccc(S(N)(=O)=O)s1 47304,c1(CNC(C(C2CCN(C(C(OC)OC)=O)C2)C)=O)cnn(C)c1O 47305,CCC(F)(C(=O)OC)C(=O)N1CCOC(C(C)NC(=O)Cc2cnoc2)C1 47306,CC(N=[N+]=[N-])C(=O)N1CCCC1CN(C(=O)C=CCN1CCCC1)C 47307,C1(NC(CCCSC)=O)CCCC12CCN(C(C1(Nc3ccccc3)CC1)=O)C2 47308,c1(SC)cn(C)nc1C(=O)NCC1C=CCN1C(c1sccc1C(C)=O)=O 47309,N1(C(C2OCCN(C)C2)=O)CCCCC(NC(=O)COC(C)(C)C(F)(F)F)C1 47310,C1(NC(CCC(N)=O)=O)CCN(C(C2CC(N3CCCC3)C2)=O)C(C2CC2)C1 47311,c1(C(=O)NC(CNC(CC(CC)C(C)C)=O)C)c(O)cnc2ccc(F)cc12 47312,CC(C)(O)C(F)(F)C(=O)NCC12CC(NC(=O)C(F)CC3CC3)(C1)C2 47313,N1(C(C(C)Cn2ccnc2)=O)CCC(CCN(C)C)(NC(=O)CNC=O)C1 47314,c1(C(=O)NC(COCCCCN(C(C(OC)C2CC2)=O)C)(C)C)ccc(CSC)o1 47315,N1(C(CC2(OC)CCC2)=O)C(C(=O)NC2CC(N3CCCC3)C2)CCC1C1CC1 47316,C(=O)(CC(=O)NCc1n[nH]cc1C(N1CCCC1CC(C)O)=O)OC 47317,C(=O)(C(CO)C(C)(C)C)NCC1CCN(S(C)(=O)=O)CC1.N12CCOCC(C1)C2=O 47318,Cc1cc([N+](=O)[O-])ccc1C(=O)NC1CCC1NC(=O)C(=O)NCC(F)(F)F 47319,Cc1ccc(C(=O)NCC2CCCCN(C(c3nccc(CO)n3)=O)C2)cc1Cl 47320,C1(C)(C(=O)NCC(Cc2ccccc2)N(C)C(c2cnsc2)=O)CC(=O)N(C)C1 47321,C1(C(N(CC(O)CN(C)C(C2(c3ccsc3)CC2)=O)C)=O)CCCN1CC(N)=O 47322,N1(CC)CCCCS(=O)(=O)CC1.c12cc(ccn1)CCC(=O)N2.c1(CN)ccccc1 47323,C1(CC)CCCCCN1C(c1sccc1Br)C(=O)Nc1ccccc1OC 47324,C1(N(C(C2(CC#C)CCCCO2)=O)C)CN(C(c2ccc(OC)s2)=O)CCC1C 47325,CC1CCCC=C1C(=O)N1CCCN(C(C2CS(=O)(=O)CCO2)=O)CCC1 47326,C(C)(C(C)(C)NC(c1cccn1C1CCCC1)=O)NC(C(C)n1cncn1)=O 47327,c1(CNC(CCN(C(C=C(CCC)C)=O)CC)=O)cc(O)ccc1C 47328,CCC(C(=O)N1CCC(C(=O)NCC(=O)OC(C)C)C1C(C)C)C(C)C 47329,N1(C(CS(CC)=O)=O)CCC2(OC)CCN(C(C3CC4(C3)CC(F)(F)C4)=O)CC2C1 47330,C(C(C)(C(=O)NCc1cccc(Cl)c1)NC(c1ccc(F)cc1)=O)SC 47331,C1(NC(C(CC)(F)F)=O)CN(C(=O)CCCCCNC(C)=O)CCC1O 47332,CC(C)(O)CCC(=O)NC1CCC(NC(=O)CN2CCNC(=O)C2)C1 47333,c1(C(=O)NCC2CN(C(C3C(C)C3C)=O)C2)n[nH]c(C2CC2)c1Cl 47334,C(CCN(C)C(C12CC(C)(C1)C2)=O)(C(C)(C)C)NC(C=CC=CCC)=O 47335,c1(C(=O)NCC2OCCC(NC(C(N)=O)=O)C2)ccc2c(c1)C(=O)CCCC2 47336,c1(NC(C2CCC(NC(=O)CCCCC3CC3)C2)=O)cnc2ccnn2c1 47337,C1(C(=O)NC(C#C)CC2CC2)CCCCCC1NC(C1(C)CNC(=O)N1)=O 47338,C(=O)(CCCCCCCC(=O)NCCNC(c1ccc2cn(C)nc2c1)=O)OC 47339,C(CN=c1[nH]c(=NC(C)C2CCC(F)(F)CC2)[nH]c2ccsc12)NS(CC)(=O)=O 47340,C1(NC(CCc2ccc(C)cc2)=O)CC12CCN(C(=O)CC1(C(F)F)CC1)C2 47341,C(C1=NOC2CN(C(=O)Cc3cnnn3C)CC12)NC(CSc1n(C)cnn1)=O 47342,C(=O)(CC(C)(O)C1CC1)N(C)CCNC(=O)Cc1cscn1 47343,Cc1[nH]c(C(=O)NCc2ncccn2)c(C)c1C(=O)NCc1cncn1C 47344,N1(C(c2cc(C)[nH]c2C)=O)CCCC(C)(NC(c2cn(C(C)(C)C)nc2C)=O)C1 47345,c1(C(N2CC(C)C(NC(c3cn(C)nc3Cl)=O)CC2)=O)c(N)cccc1[N+](=O)[O-] 47346,N1(C(=O)OC(C)(C)C)CCCCC(C)(C)C1.CC1(C)C2CC(C1)O2 47347,c1(C(=O)NCC2N(C(C(CC)(C)C)=O)CC2)c[nH]c2ccc(Cl)cc2c1=O 47348,n1(CC2(C(N(CC(=O)N(C)C)C)O)CC2)cc(C2(C3CC3)CC2)nn1 47349,C1(C(=O)NCC2COCCN(C(=O)COc3ccsn3)C2)CC12CCCCCC2 47350,c1(CC(N2CCC(N(C)C(c3c[nH]nc3F)=O)C2)=O)cncc(Br)c1 47351,C(=O)(C(C)(F)C(=O)NCCC(C)NC(c1cc(C)n(C(C)C)c1C)=O)OC 47352,Cc1ncnc(C)c1C(=O)NCC(F)CNC(=O)C(C)Cc1cccc(F)c1 47353,C(=O)(CC1=CCOCC1)NCC1CCC(C(N2C(CC)CCC2)=O)CC1 47354,CCC(C)C(O)CC(=O)N1CC2(C1)CN(C(c1c[nH]nc1Br)=O)C2 47355,Cc1ccn2c(C(N3CC4CC3C4NC(=O)CC(O)CN(C)C)=O)cnc2c1 47356,n1(CC)cc(Cl)c(C(N2CCC(O)(CN(C)C(C3(C)CSC3)=O)C2)=O)n1 47357,c1(C(N2C(CNC(CC3(OC)CCOCC3)=O)CCC2)=O)cnc2[nH]nnc2c1 47358,c1(C(=O)NCC(CNC(C(CC)C#N)=O)O)nc2ccc(Br)cn2c1F 47359,C1(C(C)C)(C(=O)Nc2cnsc2)CCN(C(c2ccncc2O)=O)C1 47360,C12(OC)CCCCC(C(=O)NCCCC(C)NC(=O)CC(C(C)C)C(C)C)(C1)C2 47361,c1(C(N2C(C(=O)Nc3cnccc3I)CC(C)C2)=O)ccc(Cl)c(C(F)(F)F)c1 47362,CCCC(C(=O)N1CC2CC1C2C(=O)NC(C)CCSC)OC 47363,C1(C(N(CCS(=O)(=O)NC)CC2CC2)=O)Oc2ccccc2OC1C 47364,N1(C(c2c(C)cc[nH]2)=O)CCC2(CCOCC2)C(CNC(=O)CC2CC23CC3)C1 47365,C1(CC(=O)NCC2(CO)CN(C(c3c(C)ncs3)=O)C2)CCCN(C)C1=O.CCCC 47366,c1(C(N(C2CN(C(=O)COCCCF)CC2F)C)=O)cccc(Cl)c1F 47367,c1(OC)cncc(C(N2CC(CNC(=O)CC3(C#N)CC3)CC2C)=O)n1 47368,C1(C(=O)NC)CCN(C(C2CCCCN2C(=O)C(C)N(C)C(C)=O)=O)CC1 47369,C1(NC(c2c(C)c[nH]c2)=O)CCCC2CN(C(c3nc4c([nH]3)CCCC4)=O)CC12 47370,N1(C(CCCC#C)=O)CCC2(NC(c3n[nH]cc3COC)=O)CCCCCC12 47371,c1(C(N(CC(CC)NC(c2cccn2Cc2ccncc2)=O)C)=O)cc(C)sn1 47372,c1(C(N(C)CCOCCNC(C2CCCN2S(C)(=O)=O)=O)=O)cc(Cl)n(C)n1 47373,c1(CC)ncc(NC(=O)C(C(C)C)NC(C2(OC)CCCCC2)=O)c(C)n1 47374,CC1CCC2CN1C2=O.C(C1=NOC2CCC12)NC(=O)CC(=O)N(C)C 47375,c1(C(N(CCN(C(C(C)C2CC2)=O)C)C)=O)cc(Cl)ncc1O 47376,C1(CC)CN(C(c2scc(C)c2Cl)=O)CCC1NC(=O)CCc1cccnc1Cl 47377,Cc1cc(Br)ccc1S(=O)(=O)N1CCSCC1C(N1C2COCC1C2)=O 47378,c1(C(=O)NCC(CNC(=O)CC2CC23CC3)O)c[nH]cc1-c1ccc(Cl)s1 47379,N1(C(C2C(C)=CCS2)=O)CCC(NC(C2CS(=O)(=O)C2)=O)C(C)(C)C1 47380,CC1(C)CC(NC(=O)CC2CN3CCC2CC3)CN1C(C1(C2CCC2)CCC1)=O 47381,C1(C2CC2)(NC(c2cc(C)c(O)nc2)=O)CCN(C(=O)C(C)(O)CC(C)C)C1 47382,N1(C(C2C(NC(C(C(C)C)C3CCC3)=O)COCC2)=O)CC(N(C)C)C2(CC2)C1 47383,C(C)(CC(=O)NC(C)CNC(C1(O)CCSC1)=O)=C(C)C 47384,C12(CC(=O)NC3CN(C(c4cn(C(C)C)nc4)=O)C3)CCC(CC1)CC2 47385,CON1CCC(NC(C2(NC(=O)CC3CC4CC4C3)CC(F)C2)=O)CC1 47386,C(=O)(C(C)(C)C(=O)NCCOC(C)(C)CNC(=O)C(c1ccccn1)O)NC 47387,c1(C(C)NC(=O)C(N2CCN(C(=O)CS(N)(=O)=O)CC2)=O)nc2ccccc2s1 47388,N1(C(C(C)CNC(=O)C(=O)NCCS(=O)CC(F)(F)F)=O)CCc2sccc2C1C 47389,C1(C(=O)NC(c2cccnc2O)C)CCCC(NC(=O)CC2CCOCC2)C1 47390,C1(CC(=O)N(C(C)CN(C(=O)CN2CCCC2=O)C)C)CC=CCN1C 47391,N1(C(C(C)Oc2cccc(Cl)c2)=O)CC2CCN(C(C3CC=CC3)=O)CCC2C1 47392,c1(CSCCOCCCC)cccc(C(=O)OC2CC3(CC3)CO2)c1 47393,c1(C(=O)OCC(=O)N(C2CCS(=O)(=O)C2)CCC)ccc(Br)cc1Cl 47394,N1(C(C(=O)NCCc2cccc(OC)c2)=O)CC2CC(C)C2C1 47395,c1(C(=O)NCCC(C)N(C(=O)CC2OCCC2(C)C)C)cc2c(F)cccc2s1 47396,C1(OC)(CNC(=O)Cc2ccc(F)cc2F)CCN(C(=O)CSSC)CC1 47397,CC(CC1CCCC1)C(=O)NC(C(=O)NCC1(O)CCOC1)C1CCCC1 47398,C(=O)(CC(C(C)(C)C)NC(c1ccc(CF)cc1)=O)NC(CCC)C(F)(F)F 47399,N1(C(C(CC)(C)C#N)=O)CCC=C(C(=O)NOCC(c2ccccc2)N(C)C)C1 47400,CC#CCC(C(=O)N(C1CCN(C)C1)C)NC(=O)CCC(C)(C)OC 47401,n1(CC)ccc(C(N2CC(NC(=O)Cn3ccnn3)CC2C)=O)cc1=O 47402,N1(C(C2OCCN(C)C2=O)=O)CCN(C(=O)CCc2nncs2)CC(CO)C1 47403,N1(C(COCCC)=O)CCC2CC2(C(=O)NCCC2CCN(C)C2)CC1 47404,CN1CC=C(CCNC(=O)C(C2CCCO2)NC(=O)CNC=O)CC1 47405,c1(CN(C(CCC)=O)C(C)(C)C)ccc2c(c1)OCCO2 47406,C1(C)(CC(=O)NCC2CN(C(CNC(C)=O)=O)C2)CCCO1 47407,C1(O)(C(=O)NC(CNC(c2n(C)nc(C)c2Cl)=O)C)CCCC(C)(C)CC1 47408,N1(C(CN(C(c2cc(COC)on2)=O)CC)=O)CCCC2(CC2)C1 47409,CC1CCCN(C(=O)C(N2CC(NC(=O)C=CCN3CCCC3)C(C)C2)=O)C1 47410,C1(CN(C)C(C2CC(C)(C)C2)=O)CCCN(C(C2C3CCC2CC3)=O)C1 47411,c1(CCC(N2CC(C)(CCC(=O)NC(CC)CC)C2)=O)ccc(N)cn1 47412,c1(CC(=O)N(C2CCN(CC#N)CC2)C)ccc(Cl)cc1.C1(C(=O)N)(CCO)CCCC1 47413,C1(C(F)(F)F)(C(=O)NCCCN(C(=O)C2=CCCS2)CC)CC=CCO1 47414,C1(CC(=O)NCC(CCNC(=O)CN2CCC2)O)CCCC(F)(F)C1 47415,C1(C)(CNC(C(CNC(c2ccn(CCC)n2)=O)O)=O)NC(=O)NC1=O 47416,c1(C(=O)NCC2N(CCC(C)C)CCCC2)ccc2cc(Br)ccc2n1 47417,CC1(CNC(c2cccc(O)n2)=O)CCCN1C(=O)CCc1cnc[nH]1 47418,S(=O)(=O)(c1cccnc1NCC1(CC#N)CC1)NCC(CCOC)(C)C 47419,C1(NC(CCN(CC#C)C(c2sc(=N)[nH]c2C)=O)=O)CC2C=CCC(C1)C2 47420,c12cccc(c1)C(=O)NC2.n1(CC(C)C)cc(CC2CCCO2)nn1 47421,c1(CC)ccc(C(=O)NC2CCC(CNC(=O)CCn3cnc(=N)[nH]3)C2)nc1 47422,C(=O)(C1CC(=O)Nc2ncccc21)NCCN(C)C(c1cnc(CC(C)(C)C)o1)=O 47423,C(=O)(C(C)(C)CCCF)NCCC1CC(NC(CCOc2c(C)cccc2C)=O)C1 47424,C(=O)(C1SCCc2ccccc21)N1CC2CCN(C(CN(C(=O)OC)C)=O)C2C1 47425,C1(CNC(Cn2c(N)cc(C)n2)=O)CN(C(c2ccc(SC)o2)=O)CC(C)(C)C1 47426,c1(NC(C)=O)cncc(C(N2CC(NC(c3cccnn3)=O)C(C)C2)=O)c1 47427,N1(C(C(c2ccn(C)c2)C)=O)CCCC1(C)CNC(=O)CCN(S(C)(=O)=O)C 47428,C1(C(=O)NC2CC(C)OCC2)CN(C(=O)C(CO)c2ccccc2)CCC1O 47429,C1(NC(c2cncc(CO)c2)=O)CC12CC(NC(c1cc(CO)ccn1)=O)C2 47430,c1(NC(C23C(CN(C(C(C)(C)OC)=O)C2)C3)=O)ncnc2c1ncn2CCO 47431,c1(NC(CC(c2ccccc2)OCCOCCOC)=O)cccc(CSC)c1 47432,N1(C(c2c(O)ccc(C)c2)=O)CC2(NC(C3CC3C)=O)CCC1CC2 47433,C(=O)(CC(O)CN(C)C)NCC(C)(C1CC1)NC(c1cc(C)[nH]n1)=O 47434,N1(C(C(=O)NC(C(CCC)C)=O)C2CC(C(=O)OC)C2)CCC(CO)(CO)CC1 47435,C1(C(CNC(Cc2n(C(C)C)cnn2)=O)(C)O)CCCN(C(c2csnn2)=O)C1 47436,C(=O)(CS(=O)(=O)C1CC1)NCC(C1CCN(C(COCC=C)=O)CC1)O 47437,O=C1OCCC12CCN(Cc1nnc(C(F)(F)F)o1)C2 47438,CC1(C(=O)NC2(CCF)CCC2)CCCN1C(C1CCOCC1)=O 47439,N1(C(C(CCC)O)=O)CCN(C(=O)CCc2cncnc2O)CC1CO 47440,C1(CNC(C(CC2CCC2)OC)=O)CN(C)CCN1C(=O)CC1CC1 47441,C(c1cccc(Cl)c1Cl)=CC(=O)NCCCCCCNC(=O)CC1CCOC1 47442,CONC(=O)C(=O)NCC1CCC(F)(CNC(=O)CCC(C)OC)C1 47443,C1(C(N2CCOCC2CO)=O)(CNC(CN(C)C(N)=O)=O)CC12CCC2 47444,N(C(=NCCCCN1CCOCC1)NCC(=O)NOC)CCOCCOC 47445,c1(C(=O)NC(CC)CCC(=O)N(CC(N2CCCC2)=O)C)ccc2c[nH]nc2c1 47446,n1(CC(=O)NC2CC3CC3N2C(=O)CSc2nn[nH]n2)cnc2ccccc12 47447,CCC1CC(=O)NCC(SC)N1.C(=O)(CC1CC1)C1(NC(CSC(C)C)=O)CC1 47448,C(=O)(C(CO)NC(N)=O)NCC(C)N(C(C1CCN(C2CCCCC2)C1)=O)CC 47449,c1(OC)cc(C(N2CCC(O)(C(C)NC(=O)C=Cc3ccco3)C2)=O)ncn1 47450,C(CC(CC)C(=O)N1CC(O)(CCNC(C2CCC23CCC3)=O)C1)=CC 47451,c1(C(=O)NC(C)CCNC(=O)CSC(F)(F)F)cnn(CC(F)(F)F)c1 47452,c1(NC2CN(C(=O)OC(C)C)C(=O)C2)c(C)nn2c1CN(C(=O)OC)CC2 47453,c1(NCCNC(N2CC[Si](CC)(CC)C2)=O)cnc(O)cc1O 47454,n1(CCCC)nc(NC(C2(CN(C(=O)C(OC)OC)C)CC2)=O)ccc1=O 47455,c12c(cnn1CC)NC2=O.c1(CC)ccccc1NC(=O)C(c1nncn1C)=O 47456,C1(CNC(C(CCCC)NC(N)=O)=O)CC2(CCC2)CN1C(=O)CCC(C)OC 47457,N1(C(C2CC(OC)C2)=O)CCCC(C)(CNC(=O)Cc2nn(C)cc2Cl)C1 47458,C1(C(=O)NCC=CCNC(C2CC(OCC)C2)=O)CC2CCC1NC2=O.OCC 47459,C1(F)(C(=O)NCC2C(NC(c3cccc(OCC(F)F)c3)=O)C2)CCOCC1 47460,Cc1nccnc1C(=O)NCCC(C)(C)NC(C1CC(F)(CF)C1)=O 47461,c1(C(N2CCC(NC(C3C(CC)C3)=O)C2)=O)cccc(OC)c1Cl 47462,c1(C(N(CCCNC(c2csc(Cl)n2)=O)CC)=O)ccc(CO)cc1 47463,C12(NC(c3n(CCSC)nnn3)c3ccno3)CCC(CO)(CC1)C2 47464,N1(C(c2c(OC)cns2)=O)CCC(F)(F)C(CNC(c2cc(Cl)c[nH]2)=O)C1 47465,S(=O)(=O)(c1ccc(F)cc1)Nc1ccc(NCC(N2CCOCC(O)C2)=O)nc1 47466,c1(OC)cc(F)c(C(=O)Nc2cccc(NC(C3CC4(CC4)C3)=O)c2)cc1F 47467,C#Cc1cccc(C(=O)NCC2(OC)CN(C(C3CCC(C)CC3)=O)C2)c1Cl 47468,N1(C(CCc2cccc(OC)c2)=O)CCC2CN(C(C3CCCS3)=O)CC12 47469,C1(CC(c2nnnn2CC2CCCCC2)(C)NC(C2CCOC2)(C)C)CC(F)(F)C1 47470,c1(NCC(=O)NCC=CCNC(c2c(C)ccnc2)=O)ccc2ccccc2c1 47471,CC1(C)CC(CC(N2CC(O)CC2CNC(C2CC=CCC2)=O)=O)CC(C)(C)O1 47472,c1(C(=O)NCC(CN(C(=O)CC(C)(C)OC)CC)(C)C)ccsc1C#N 47473,C1(CNC(C(C#C)(C)C)=O)CN(C(=O)C(C)=C2CCC2)CCC1C 47474,CC1(C)CC(CNC(=O)CN2CSCCSC2)N(C(c2ccnc(C#N)c2)=O)C1 47475,Cc1[nH]nc(C(N2CCCCC2CN(C)C(c2cc(C#N)on2)=O)=O)c1F 47476,N1(C(c2c(CC)n(C)cc2)=O)CC2CN(C(C34CC(F)C3C4)=O)CC2C1 47477,N1(C(c2c(C)nns2)=O)CC2(CCN2C(c2ncn(C)n2)=O)C1 47478,c1(C(C(=O)N(C(C)CNC(=O)CCc2cnn[nH]2)C)O)ccccc1C(F)(F)F 47479,C12CC(C1(C)C)SC2.Cc1nc(CCO[Si](C)(C)C)no1 47480,Cc1cc(CC(=O)NC2CCN(C(=O)Cc3cnn(C(C)(C)C)c3)CC2)nn1C 47481,N1(C(C(C)(Cl)Cl)=O)CCCCC(CNC(C23CCCCC2(C(=O)OC)C3)=O)C1 47482,N1(c2cc(C)nc(NCc3nccc(F)c3Cl)n2)CCc2nc(Br)sc2C1 47483,N1(C(CCC(=O)NC2CCn3nnnc3C2)=O)CCC2CN(C(C)=O)CC2C1 47484,c1(C(=O)NC2C(CC(=O)N(CCC(C)O)C)CCC2)ccc(N)cn1 47485,c1(C(N2C(SS(C)(=O)=O)CCCC2)=O)ccc(F)c(Cl)c1N 47486,C1(C2CCCCO2)(C(N(CCNC(c2ccn(CCC)n2)=O)CC)=O)CCCO1 47487,CCC(C)C(C(=O)NCC=CCNC(c1ccc(C2CCC2)nc1)=O)OC 47488,C=CC(O)(C(=O)NC1CCN(C(=O)C(=O)NCCOC)CC1O)C(F)(F)F 47489,c1(C(N(C)CC2N(C(Cc3c(C)noc3)=O)CCCC2)=O)cc2occc2n1C 47490,C(=O)(C(O)CC[S+](C)C)NC1C(NC(c2ncc(C)c(C)c2)=O)CCCC1 47491,CC1CCCCC1C(N1CC(C)CC1C(=O)NC1CCCN(C2CC2)C1)=O 47492,C1(C(=O)NCC(CNC(c2occ(C)c2)=O)F)CC2(C1)C(F)(F)C21CC1 47493,C=CCCCCCCC(=O)N1CC(C(=O)NCC2(O)CCC2(C)C)C2(CC2)C1 47494,c1(C(=O)NCC=CCNC(=O)CC23CCCC2C3)cc2cccnc2o1 47495,C1(NC(c2occ(C)c2)=O)CC=C(C(=O)NC2CC3(C2)CC(O)C3)C1 47496,CC1CCc2ncc(C(N3CC(C)N(C(=O)C4=CS(=O)CCC4)CC3C)=O)n2C1 47497,C1(NC(=O)Cc2cc[nH]c2)COC2(CCN(C(c3cnc4c(c3)CCC4)=O)C2)C1 47498,Cn1cc(Cl)cc1C(=O)NCC(O)CC(=O)NCC1(O)CCC1 47499,N1(C(C2C(C(C)(F)F)C2)=O)CCC2CN(C(c3ccc(Br)cc3)=O)CC12 47500,CCC(CC)(CN=c1cc(COC)nc(Cl)[nH]1)NC(=O)Cc1ccccc1NC 47501,N1(C(C23OCC(C)(C2)C3)=O)CCCC2(NC(c3csc(C4CC4)n3)=O)CC2C1 47502,c1(OC)ccc(C(=O)N(C2CCC2CC2COCCN2C(=O)NC)C)cc1OC 47503,c1(C(=O)NC2CC(NC(C=CCOC)=O)C2)cc2c(nc1O)CCCC2O 47504,C1(NC(C(CSC)C)=O)CCC2(CCN(C(c3ccoc3Cl)=O)C2)C1 47505,CN1CCC(N(C(c2csc(-c3ccccc3)n2)C(=O)NC2COC2)C)C1 47506,Cc1nc(O)[nH]c1C(=O)NCC(C)NC(C1(C#N)CC1C(F)(F)F)=O 47507,c1(OC)ccc(C(=O)NCC2(C(N)=O)CN(C(C3CC(=C4CC4)C3)=O)C2)c(Cl)n1 47508,CCCCCC(O)C(=O)N1CC2=C(C1)CN(C(c1ncc(Br)cc1N)=O)C2 47509,c1(C(=O)NCC(CCNC(c2c(C)cccc2O)=O)O)ccc2nnc(O)n2c1 47510,C#Cc1nccnc1NC(C1CCCC1NC(c1cnc(CC)cn1)=O)=O 47511,C(=O)(C(O)C(F)(F)F)NCCOCCCCC1CN(C(c2ccc(CSC)o2)=O)C1 47512,CC(C)CC(CNC(=O)C(C)(C1CC1)N(C(=O)CN1CCOCC1=O)C)N(C)C 47513,CC1CN2CCN1C(C(=O)NCCCCNC(=O)CCCSc1ccccc1)C2 47514,c1(OC)ccc2c(c1)CCN(C(=O)C(=O)NC1CCCCC1Oc1ccccc1)C2 47515,CCC(C)(O)C(=O)N1CCN(C(CNC(=O)C=CC2CCCCC2)C(F)F)CC1 47516,CC1(C)CC(CNC(=O)NCCOc2cccnc2)CC1(C)C 47517,C(=O)(C#CC1CC1)NC1CCN(C(CCN(C)CCO)=O)C1 47518,N1(C(CC2N(C)CCCC2)=O)CCN(C(C2CC2c2ccncc2)=O)C(CO)C1 47519,C(C(C)N=c1[nH]c(=N)[nH]c(=NCCc2cnn(C)c2)[nH]1)(C1CCOCC1)OC 47520,c1(C(N2CC(C)C(CNC(C3CC34CCCC4)=O)C2)=O)ccc(F)c2c1OCC2 47521,CC1(C(=O)NCC(C2CCCC2)NC(c2cc(Br)no2)=O)CC(F)C1 47522,N1(C(C(CSC)C)=O)CCC2(CCCN2C(c2cncc(NS(C)=O)c2)=O)CC1 47523,C1(NC(c2[nH]cc(C)c2)=O)CC(CNC(c2cn(C)nc2C(C)C)=O)C1(C)C 47524,C1(C(N(CCNC(c2cc(C)on2)=O)C)=O)CCn2nccc2C1 47525,Cn1ccc2cc(C(=O)NC3(CCNC(C4CC(F)(CO)C4)=O)CCC3)cnc12 47526,C1(NC(c2nc(CC)sc2)=O)CN(C(=O)Cc2cc[nH]c(=N)c2)CC2(CC2)C1 47527,N1(C(C(CC(=C)C)NC(=O)Cn2cc(C#N)cn2)=O)CC2(CC(CO)CO2)C1 47528,c1(C(=O)NCC(C)CNC(C23CCCN2CCC3)=O)ccc2c(c1)NC(=O)CC2 47529,c1(OC)ccc(C(N2CCCC2CN(C(=O)CC2CCCC2C)C)=O)cc1 47530,C1(NC(C(CCC)CNC(=O)C(C)(C)N2CCCC2)=O)CC(C2CCCC2)C1 47531,C1(C(=O)NC(CC=C)CNC(=O)COc2ccsn2)CC2(C1)OCCO2 47532,C12(CNC(c3cc4ccsc4s3)=O)CCCC1CCN2C(c1scnc1Cl)=O 47533,CC1(C(=O)NC2C=CC(CC(=O)NCCn3cncn3)C2)CCCOC1 47534,c1(OC)cc(C(=O)NC(CNC(=O)CC2OCCO2)C2CC2)c2ccccc2c1 47535,C1(c2nc(CCOC)nn2C2CCOC2C)CCN(c2ccc(Cl)cc2)S1(=O)=O 47536,C1(c2n(CC=C)nnn2)(NCCCC2(C)CC2)CCCN2CCCCC12 47537,c1(C(N2C(C)CC(NC(c3cc(CO)on3)=O)C2)=O)nccc2ncccc12 47538,c1(C(=O)NC(C(=O)NCCN2CCC3CC23)C2(C)CC2)c[nH]c2cccnc12 47539,c1(-c2c(CNC(c3ccc(OC)o3)=O)cccc2)cnc(C(F)(F)F)cc1OC 47540,C1(CNC(C2CCC(CC)O2)=O)CCCN(C(=O)Cc2cncnc2O)CC1 47541,c1(C(=O)NC(CC)CNC(=O)CC2CCCOC2)cccc(N)c1C 47542,C1(F)(CNC(C2(C(C)C)CCC2)=O)CCN(C(C2CC(F)(CO)C2)=O)C1 47543,N1(c2nc(C(C)C)nc(Cl)c2)CC23CCCC2(CN(C(C2CNC(=O)N2)=O)C3)C1 47544,C1(C#N)(C(N2CCCC(NC(Cc3n(C)cnc3)=O)CC2)=O)CC2CCC1CC2 47545,C12(CC(N3CC(n4cc(NC(CCC)=O)nn4)C3)=O)CC3CC(C1)CC(Br)(C3)C2 47546,C(=O)(C(C#N)C(C)C)N(CC(Cc1ccccc1)N(C(c1c(C)scn1)=O)C1CC1)C 47547,C1(C#N)(C(=O)NCC2(NC(C(CC=C)CC)=O)CC2)CC2CCC1CC2 47548,N1(C(C2(COC)CC2)=O)CCC(CN(C)C(c2cc(C(C)=O)[nH]n2)=O)CC1 47549,CC1CC(C)C(C(=O)NCC2CCC(Cc3n[nH]cc3COCOCC)CC2)O1 47550,N1(C(c2c(C#C)c[nH]n2)=O)CC(=O)NCC1C(=O)NC1CCCC12CC2 47551,S(=O)(=O)(c1c[nH]c2ccncc12)NCCN1CCCCC(C)C1 47552,N1(C(C(N2C(C)CC3(CC3)C2)=O)=O)CC2(CCN(C)CC2)C1.C1C(=O)N1 47553,CN1CCC2C(CCN2C(C23CCC2CN(C(=O)CC2CC=CC2)C3)=O)C1 47554,C(c1cc2ccccc2o1)=CC(=O)Nc1cc(C(F)(F)F)ccc1Br 47555,C(=O)(C(C)(C)S(C)(=O)=O)NC(C1CCCN(C(=O)COC(F)F)C1)C 47556,C1(NC(C2(C)CC2(F)F)=O)CCC(NC(=O)C(c2ccccc2)=O)CC1 47557,Cn1ccc2cccc(C(=O)NCC(O)CCNC(C3(C)CC3(F)F)=O)c12 47558,CCC(CC(=O)N1CC(F)CC1CO)N(C(=O)C=Cc1cn(C)cn1)C 47559,CC1CCCN(C(c2csc(C)c2N)=O)C1CNC(=O)CCCn1ccnn1 47560,c1(C(=O)OC)ccc(-c2ncnn2Cc2onc(C=O)n2)cc1.c1(C)cccs1 47561,c1(C(=O)NC2CC(NC(c3c(C)n(CC4CCC4)nn3)=O)C2)ccc(F)c(Cl)c1 47562,C(CC(C)CN=C(NC(C)C)N1CCC(NCC(F)(F)F)C1)OCC 47563,C(=O)(CC(C(F)(F)F)NC(c1sccc1CO)=O)NC(C1CCN(C)C1)C 47564,c1(C(C)C)oncc1C(=O)NCC1CCN(c2ccccc2)C1 47565,c1(NCCC2(NC(C)=O)CC2)cc(C2CCC2)[nH]n1 47566,CN1C(C)(C)C(Nc2cc(N3CCC(C(F)(F)F)C(CO)C3)ncn2)CS1(=O)=O 47567,N1(C(c2cc(C)n(C)n2)=O)CC2CCC1C(CNC(=O)C(C)(C)C(F)(F)F)C2 47568,C1(NC(c2cc(C(=O)OC)n[nH]2)=O)CC1C1CCCN(C(C2CCCCS2)=O)C1 47569,C1(NC(CN2CCC(CNC(C(C)C)=O)C2)=O)CC(=O)NC1=O 47570,C(=O)(CC(C)CNC(=O)OC(C)(C)C)NCC(C)NC(=O)Cc1cc[nH]c1 47571,c1(OC)ccc(CCNC(=O)C(=O)N(C(C)C)CC2(C)CCCC2)cc1C 47572,c1(-c2c(C)cc(C(=O)NCc3cc(Cl)nc(Cl)c3F)nc2)cnc2ccnn2c1 47573,C1(CNC(=O)CSCCC#N)CC(CNC(C2(C(=O)OC)CC2)=O)CO1 47574,N1(Cc2cn(C)nc2C2CCOCC2)CCCc2cc(C(=O)O)ccc21 47575,N1(C(c2c(C)n(C3CC3)cc2)=O)CC(NC(=O)C(C)(F)c2ccon2)C(C)(C)C1 47576,C(=O)(CCCCCF)N(C(C)C(=O)NC(C)(C)CCCO)CC 47577,C12(C(=O)NC(CCN(C)C)(C)C)CCC1CN(C(=O)Cc1ccsc1)C2 47578,C=CC(CC)CC(=O)NCC1CCC(C(=O)NC2(COC)CCC2)O1 47579,C(=O)(CS(=O)(=O)C1CC1)NCC1C(NC(C(C)Cc2ccncc2)=O)C1 47580,C(CN=c1nc2scnc2c(NC)[nH]1)C1(CO)COCC(C)N1C 47581,N1(C(C2(C=C)CCCC2)=O)CC(CO)C2(C1)CN(C(c1cnc(O)c(F)c1)=O)C2 47582,C1(NC(=O)C=C(Cl)Cl)CCCCCC1NC(C1CC2CCC(C1)C2)=O 47583,CCCCCC(C1CC1)NC(=O)CNC(c1ccc(C)nc1)=O 47584,c1(NC(C2N(C(C(C)O)=O)CC2)=O)nc(Cl)ccc1F 47585,CC(C)C(CCN(C)C(c1csc(C(F)(F)F)c1)=O)NC(=O)C(F)=CCCF 47586,CC(C)(C)CC(O)CC(=O)NC(CCF)C(=O)N(C1CC1)Cc1ccco1 47587,C1(C(NNC(C=Cc2c(C)cccc2)=O)=O)C2CCCCCCC12 47588,C(=O)(C(C)CCCOC)NCC(C)(C)OC 47589,C1(c2nnnn2CC2CCCO2)(NC2CC=CCC2)CCC2(CCO2)CC1 47590,N1(C(CC2CC(CC)C2)=O)CCOC2CN(C(=O)COC(C)=O)CC12 47591,CC1COCC(CONC(=O)C2(NC(c3ccsc3)=O)CC2)O1 47592,C(=O)(C1=CC2(CCOC2)C1)N(C1CCN(C(c2ccc(O)c(F)c2)=O)C1(C)C)C 47593,c1(C(=O)NCC#CCNC(c2c(CC)oc(C)c2)=O)onc2c1CCCC2 47594,CCC(C)CC(C)C(=O)N(C1CN(C(=O)C(CC)Oc2cccc(Cl)c2)C1)C 47595,C(CC(=O)NC1COCCN(C(C2(CF)CCOCC2)=O)C1)(C(N)=O)NC(C)=O 47596,c1(C(N2CCCN(C(C3C(=C)CC3)=O)CC2CO)=O)cc2c(C)ccc(C)c2[nH]1 47597,N1(C(CNC(CC)=O)=O)CCC(O)(CCNC(c2c[nH]nc2C)=O)CC1 47598,Cc1cc(C(=O)OCCC2CCC3CC23)ccc1-n1cnnn1 47599,c1(C(=O)NCC(CNC(C=CCC)=O)F)cccn2cc(C(F)(F)F)nc12 47600,CC1CN(c2nnnn2CCC2CCCCC2)CCCO1 47601,Cc1cccc(COCC(N2CCC2CNC(c2cn[nH]c2)=O)=O)c1 47602,C(=O)(CCCCC(=O)NC1CCC(CNC(c2ccn(CC(C)C)n2)=O)C1)NC 47603,N1(C(C=C2CCC(C)CC2)=O)CC(NC(c2ncc[nH]c2=O)=O)C(C2CC2)C1 47604,c1(C(N2C(CNC(=O)CC34COC(C)(C3)C4)CCC(C)C2)=O)cc2ncccn2n1 47605,c1(CC(=O)NC2CC3(CN(C(C=C)=O)C3)OC2)c[nH]c2ccc(Br)cc12 47606,N1(Cc2c(C)nc(C)c(C)n2)CCCc2ncc(F)cc21 47607,C=CCC(C)(C)CCN(C(C)C)Cc1ccc(OC)cc1 47608,C12(C(N3CCN(C(c4c(C)occ4)=O)C(C(F)F)C3)=O)CC1COC21CCC1 47609,C1(NC(C2CCCC(F)(F)C2)=O)CC2CC(NC(=O)CCCc3cnn[nH]3)C1C2 47610,C12(NC(=O)OC(C)(C)C)CCCN(C(=O)C(Cc3cccnc3)C3CCCC3)C1C2 47611,C1(NC(C(C)=O)=O)CN(C(=O)CCC(C)(C)C#N)C2(CCOC2)C1 47612,C1(C=O)(CC)CCCC1.N1(N(C(C)C(=O)N)CCC)CCC(CCN(C)C)C1 47613,CC(c1cccnc1)=CC(=O)NCC1(CO)CCCO1 47614,C(=O)(C1=Cc2ccccc2C1)N1CC(C)(C)C1C1CCN(C(=O)CC2CC2)CC1 47615,C(=O)(CC1=CCCCC1)NC1(C)CCCN(C(c2cncc3nc[nH]c23)=O)C1 47616,C1(C(=O)NC(C)C(CO)NC(C2CCC2c2nncn2C)=O)CC12CCCCC2 47617,CC1(C(=O)Nc2ccc(Br)cc2Cl)CCCN(Cc2cnc(Br)s2)C1 47618,C(=O)(C1=NOC(C)(C)C1)N1CC(C#C)C(OCCOC)C1 47619,C(CC1=CCN(C(c2ccc(CO)s2)=O)CC1)NC(c1n(C)nc(O)c1)=O 47620,C1(C(C)(C)C)CCCCN1C(=O)Cn1nccn1.n12cc(nn1)C2 47621,c1(C(=O)NC(CCCCNC(c2ccn(CC#C)n2)=O)=O)ccc(S(C)=O)cc1 47622,c1(CC(N2C(CN(C)C(C3CC3(Cl)Cl)=O)CC(F)C2)=O)ccc2c(c1)COCC2 47623,C1(C(N(C)C2CC2)=O)CC2(CCN(C(=O)Cc3cccc(Cl)c3)C2)C1 47624,c1(C(=O)NC2CC(NC(C)=O)C23CCC3)cccc2ncc(C)n12 47625,CCCCC(CC)C(=O)N1CCCN(C(c2ccc(Cl)nc2O)=O)CCC1 47626,N1(C(c2c(C)coc2)=O)CCC(N(C)C(c2nn(C)c(Cl)c2Cl)=O)C(C)C1 47627,O=C1CC(C2CC2)(C(=O)NC2CC(CC(=O)NC3CCCC(F)(F)C3)C2)C1 47628,C1(C(N2CC(=O)NCC2)=O)(C(F)F)CCCO1.n1(CCCNC)cccc1 47629,c1(NCCC(O)C(C)C)cc(Nc2nc(CCC)on2)ncn1 47630,C(=O)(C(F)(F)C(C)(C)O)NCC(=O)N(C(C)C(=O)NCC1CC1)CC 47631,C1(NC(CCC=C)=O)CCCC1(C)CNC(=O)C(c1cccc(COC)c1)(C)C 47632,n1(CC(C)NC(=O)C=Cc2ccco2)cc(CNC(=O)CC2CC(F)(CO)C2)nn1 47633,c1(C(C)C)cccc(F)c1C(=O)NC(C)CNC(=O)C(C)Cc1cccc(Cl)c1 47634,N1(c2cc(OCC)ncn2)CC(F)(F)CC1(C)CNC(=O)C=Cc1ccnn1C 47635,c1(CNC(CC(C)O)C)ccc2c(c1)CC(C)(C)O2 47636,N1(C(CC(=C=C)C)=O)CC2CCN(C(c3ccn(C(CC)CC)n3)=O)CC2C1 47637,C1(NC(C2(COC)C=CCN2C(c2ccco2)=O)=O)CCCC(C)(C)C1 47638,C1(CC(=O)OC)C(C)OCCN1C(CCC1CCC1)C(=O)NCc1ccccc1 47639,Cc1nc(N(C)CCOCCNC(=O)Cc2cnc(C)[nH]2)c2scc(C)c2n1 47640,N#Cc1cc(C(=O)N(C(C2CCCC2)=O)C2CC2)c[nH]1.N12CCC1C2 47641,n1(CC#C)cccc(C(N2CC(n3ccnc3SC)C2)C)c1=O.N12CCNC(C1)C2 47642,Cc1nn(C)cc1-c1cn(CCCCC(=O)O)nn1.C1(=O)C(CO)N1C(N)=O 47643,C1(NC(CSCC(C)C)=O)CC(C(=O)NC)C12CCC2.N12CC3C(C3C1)CC2=O 47644,C(=O)(CCC1=CCCCC1)NCC1(C)C(C)CN(C(COCC(=O)NC)=O)C1 47645,c1(C(C)(F)F)cccc(C(=O)NCC(CO)NC(c2cccn2C2CC2)=O)c1 47646,N1(C(c2ccc(C)[nH]2)=O)CCCCC(CCC(N2C3CCC2COC3)=O)C1 47647,C1(C(=O)NCCNS(CC)(=O)=O)CCCN(C(C2CC(C)N(C)C2)=O)C1 47648,Cc1cc(C(C)Nc2cc(CCN3CC=CC3)ncn2)cc(C)c1 47649,c1(NC(CC2CCCN(C(C3CC(=O)NCC3)=O)C2)=O)ccc(F)c(CO)c1 47650,C1(CCOC)CN(C(c2ccc(-c3nn[nH]n3)cc2Cl)=O)CC(C)O1 47651,C1(CC=C)(NC(c2ncccc2OCC)=O)CCN(C(=O)C(F)n2ccnc2)C1 47652,Cc1ccc(C(=O)NC2CC(N(C(=O)CCc3cncs3)C)C2)c(F)c1C 47653,C(CCN(C)C(C12CC(F)(C1)C2)=O)(C(C)C)NC(C(F)OC)=O 47654,N1(C(c2cn(C)nn2)=O)CCC2(CC1)CN(C(C1CC3CC3C1)=O)C1COCC21 47655,N1(C(C(C)n2cnnn2)=O)CCC(C2CCN(C(C3(C)CC(F)(F)C3)=O)C2)CC1 47656,C1(C(N2CCN(CC)CC2C)=O)CCc2nc(C)nn2C1.C(C)(C)N 47657,CC(CN=c1[nH]c(=NCC2CC(F)(F)C2)[nH]c2c1CCC2)n1ccnc1C1CC1 47658,C1(NC(C(C)NS(CC)(=O)=O)=O)CN(C(=O)Cn2nc(C)cc2C)CC1SC 47659,C(=O)(CCC(=O)C(C)(C)C)NCC=CC(=O)NC1CCC(CN(C)C)C1 47660,Cc1ccccc1OCC(=O)NC1COCC1C(=O)NC(C)CCO 47661,C(=O)(C(CC(C)C)C(C)C)N1C(CNC(N2CCC(C)(CC(=O)NC)C2)=O)CCC1 47662,c1(C(N2CCC(O)(C(C)NC(CNC(=O)NC)=O)C2)=O)cc2c(nc1O)CCC2 47663,C(C(CC(C)C)C(=O)NC1(CN(C(=O)CC(c2ccccc2C)C)C)CC1)OC 47664,CCCC(CCCO)C(=O)N1CCN(C(C2CCN(C(C)C)CC2)=O)C(C)C1 47665,CN(S(N)(=O)=O)CC(=O)NC1CC(CNC(c2ccn(C3CCC3)n2)=O)C1 47666,CCCCCCC(C(=O)NC1(C)CCN(C(=O)C(C)(C)C2CC2)C1)NC(C)=O 47667,c1(C(N2CC3C(CNC(C=C(C)C(=O)O)=O)(C3)C2)=O)ccnc(Cl)c1C 47668,Cc1nc(F)ccc1-c1cccc(OCC(C)O)c1 47669,C1(CNC(C2(NC(CCSCC(N)=O)=O)CCCC2)=O)CCCC(NC(N)=O)C1 47670,N1(C(C(C)(C)C2CCOCC2)=O)CC2CCCC(NC(c3cnsc3)=O)C2C1 47671,c1(C(=O)NCC23C(CN(C(C4(CC(C)C)CC4)=O)C2)CC3)cccn2cnnc12 47672,CCC(C)C(C)C(=O)N1CC(CNC(c2csc3nnsc23)=O)CC1C 47673,C(CC(C(=O)NOC(CO)C(C)C)NC(=O)C(C1CC1)SC)=CC 47674,CCC(C(=O)NCC(CNC(=O)CC1(C)CC1)OC)Sc1nc(=N)[nH][nH]1 47675,N1(Cc2ccc(CN3CCCC3)o2)CC(=O)N(C(C)(C)CC2CCCCC2)C1=O 47676,c1(CC)cc(N2CC(C3CC3)CCC2)n2ncc(Br)c2n1 47677,C1(NC(c2nc(OCC)sn2)=O)CCN(C(C2CC(=O)CO2)=O)CC1C 47678,C1(C(=O)NCc2c(C)noc2)C2CCN(C(=O)CCC(C)CN(C)C)CC12 47679,C(C)(C(C)(C)C(=O)N1CCC=C(Cl)C1)NC(c1cc(C)[nH]c1C)=O 47680,CC1CCN(CC(=O)NCC2C(C)CCN2C(c2cc(C#N)on2)=O)CC1 47681,c1(C(=O)NCC(CC)NC(c2ccc(O)c(N)n2)=O)cc(C(N)=O)ccc1F 47682,CC(C)C(C)CC(=O)NCC1(C(N)=O)CN(C(C2OCCCO2)=O)C1 47683,C(c1ccc([N+](=O)[O-])s1)=CC(=O)N(C)CC1CCCCN1C(=O)C1=COCCC1 47684,Cc1oc(C(C)(C)C)cc1C(=O)NCC1CC1NC(c1cnoc1C(C)C)=O 47685,c1(C(=O)NCCCCCNC(Cc2cc(C)sc2)=O)coc2ccccc12 47686,N1(C(C)(C)C)CCN(C(c2nccn2CC(F)F)C(=O)NC2CCC2)C1 47687,CCC(CCCO)N=c1[nH]c(N(C)Cc2ccc(Br)o2)nc2c1COCC2 47688,N1(C(c2ccc(F)s2)C(=O)NC2CC2)CCCCC2(CCC2)C1 47689,C1(C(C)(C)C)CN(C(=O)C=CC2CCCO2)CCN1C(=O)C(Cl)=CCl 47690,CC(CN(C(=O)C(CCN(C)C)NC(C1CC(O)C(F)C1)=O)C)C(C)(C)C 47691,c1(C(=O)NC(C)C(C)NC(=O)CSCc2ccccc2)cc(CCN(C)C)on1 47692,N1(C(C(C)(C)N(F)F)=O)CCC(C2CCCN(C(C3CC3C(C)(F)F)=O)C2)CC1 47693,c1(OC)cc(-c2cnc3cc(C(N4CCSCC4)=O)[nH]c3c2)cc([N+](=O)[O-])c1 47694,C1(CNCc2cccc(OCCCC)c2)CCCC1C1CC1 47695,C1(N(C(C2C(CC)C2)=O)C)CCCCC1N(C(=O)Cc1ccc(F)nc1)C 47696,N1(C(C(CC(C)C)F)=O)CCC2CCC(C1)N2C(c1cccc(SCC#N)c1)=O 47697,N1(C(c2cc(C)c(F)cc2N)=O)CCc2ccc(F)cc2C1C 47698,C(CC1c2ccccc2CCN1C(=O)Cc1ccon1)NC(=O)C(C1CC1)C1CC1 47699,CC1CN(C(C2(F)C(C)(C)C2(C)C)=O)CC(CCNC(=O)CC(F)(F)Cl)O1 47700,c1(NCCC(C)SC)cc(NCC2CCC(C(F)(F)F)CC2)ncn1 47701,C1(CC)CN(C(=O)C(=O)NC(C)CSc2ccc(Cl)cc2)CCC1C(F)(F)F 47702,CCCC(CC1CCCC1)C(=O)NCC(C)(C)CNC(c1c(C)cccc1F)=O 47703,c1(C(N)=O)ccccc1C(=O)NC1CCC1CNC(=O)C(C1C=CCC1)=O 47704,C1(C(=O)NCC=CBr)CCCN(C(=O)CCC2CCCO2)CC1 47705,Cc1ncc(C=CC(=O)NC(C2CCCN2C(=O)COc2cnn(C)c2)(C)C)s1 47706,c1(CCC)ccc(C(=O)N(CCC(C)NC(=O)CC2CCCO2)C)s1 47707,C1(CCNC(C=CC(C)(C)SC)=O)CCCN(C(C2(C)C=CCCC2)=O)C1 47708,CC(C)C(O)C(C)(C)C(=O)NCC1CCC(NC(=O)CSc2nnnn2C)CC1 47709,Cc1cc(C(=O)N(CCC(C)NC(c2c(C)n[nH]c2C)=O)C)ccn1 47710,c1(NC(c2cnc(C)[nH]2)C)ncnc(NCCc2nc(CO)cs2)c1C 47711,C1(NC(c2ncc(CC)s2)=O)CC2CCC(C1)N2C(c1cnc(OC)nc1C)=O 47712,N1(C(C(C(C)C)NS(C)(=O)=O)=O)CCC(NC(c2cncn2C)=O)C12CC2 47713,C1(CNC(C2C3CNCC23)=O)CCN(C(=O)CCC2CCCC2)CC1 47714,c1(C(N2CCN(C(C(C(C)(C)C)SC)=O)CC2C)=O)cc(Cl)cc(Cl)c1Cl 47715,O=C1CNC(=O)c2cc(C(=O)NCCOOC3CC3)ccc2N1 47716,c1(NC(C2N(C(CC(C)O)=O)CCOC2)=O)ccc(Cl)cc1O 47717,C1(CCC)(C(=O)NCc2ccoc2C(=O)O)CCN(C(c2ccsc2)=O)C1 47718,c1(CCC(=O)NCC(C)N(C(c2nc(OCC)oc2)=O)C)c(C)noc1Cl 47719,c1(C(N2CC(CNC(C=C(C)C(F)(F)F)=O)C(C)C2)=O)cnc2nncn2c1 47720,N1(C(c2c(N(C(C)=O)CC3CC3)cccc2)=O)CCCC(C)C1C1CCCCC1 47721,CN1CCN(C(=O)C(C)(C)Oc2ccccc2)CC1CNC(=O)C(C)(C)CO 47722,Cc1nccn1CCCC(=O)NC(C1CCN(C(c2cnn(C)c2)C)C1)=O 47723,c1(C(=O)Nc2ccc(I)cc2F)cnc(COC)nc1N1CC2CN(CC)C2C1 47724,Cc1nccn1CCCNC(=O)C(C1CC1)NC(=O)CC1CCO1 47725,Cc1nc(N2CC(NC(c3c[nH]c4ncccc34)=O)C(F)C2)c2sccc2n1 47726,c1(N(C(=O)COC2CCN(C(C)=O)C2)CC=C)cnc(C)c(OCC)c1 47727,C1(CNC(CCOC)=O)CCN(C(=O)C(C)(C)C2CC2)C1 47728,N1(C(CCCC)=O)CC(NC(C2(F)CCC2)=O)CC2(CC2)C1 47729,N1(C(COCCCC#C)=O)CC(NC(c2cc(C)ccc2C)=O)CC(F)C1 47730,c1(CCC(N2C(CCNC(C(C)n3ccnc3)=O)CCC2)=O)ccc(N)c(F)c1 47731,CC(C)CC(CNC(C1CCN(CC)CC1)=O)C(=O)NCC1(CO)CC(C)(C)C1 47732,c1(OC)ccc(S(=O)(=O)Nc2cncc3ncnn23)cc1Cl 47733,c1(C(N2CC(F)CC(C(=O)NCc3cccs3)C2)=O)cc(F)cc(F)c1I 47734,c1(CN(CC(C)Cc2cn[nH]c2)C(=O)CCn2cncn2)cnc(C#N)cn1 47735,N1(CC(=O)NCC(CCOC)NC(C2CC23CC(O)C3)=O)CCCCCC1 47736,C1(NC(c2nc(OCC)oc2)=O)CCN(C(C2CN(CC)CCO2)=O)C(C)C1 47737,C(=O)(C(CC1(C)CCC1)NC(=O)C(C1CCCCC1)C)NC1(C#C)CC1 47738,C(=O)(CCCC(=O)N1CC(C(=O)NCC(O)(COC)CO)(CO)C1)OC 47739,Cc1cc2ccc(C(N3CCN(C(c4cnn(C)c4F)=O)C(CO)C3)=O)cn2c1 47740,C=CC(C)CC(=O)NCc1cn(C2CN(C(=O)CCn3cnccc3=O)C2)nn1 47741,c1(CC)onc(C(N2CCC(NC(=O)CCc3cnn[nH]3)C2C(C)(C)C)=O)c1C 47742,c1(C(N(CCNC(C2C(C)C2C)=O)C2CC2)=O)cnc2ccc(F)cc2c1 47743,CC(C)CS(=O)(=O)CCC(=O)N1CC(CC(C)NC(=O)CCn2ccnn2)C1 47744,C(=O)(C#CC1(C)CCCO1)N1CC(N2CCN(C(C3(F)C(C)OCC3)=O)CC2)C1 47745,N1(C(c2nn(CC)c(C)c2)=O)CCN(C(c2ccnc(C3CC3)c2)=O)C(CO)C1 47746,C12(CNC(CC(C)(C)OC)=O)CCCC1CCN2C(=O)CC(F)(F)C(F)F 47747,C1(C(=O)NCC(CC=C)NC(=O)Cn2c(C)ccc2C)CCn2ncnc2C1 47748,c1(OCC)cccc(C)c1CNc1cc(Oc2ccccc2)cc(O)c1 47749,N1(C(c2cc(CC)sn2)=O)CC(C)(C)CC1C(=O)NCC1CCC(CC)CC1 47750,c1(C(=O)NC(C2CN(C(c3n[nH]c(CC)c3C)=O)C2)C)nnc(O)nc1O 47751,C(C(C)(C)CC(=O)N1CCCCC1C(=O)NC1CCN(C(C)C)CC1)OC(C)=O 47752,c1(C(=O)NC(CC)CN(C(=O)Cc2nc[nH]n2)CC)ccnc(N(C)C)c1 47753,CCC(C)C(O)C(C)C(=O)NCCCCC(=O)NC1CCC(C#N)CC1 47754,N1(C(CCc2ccc(C)nc2)=O)CCN(C(=O)CC2CCCC2)C2CC12 47755,c1(CN2CC(CNC(c3ccc(O)c(F)c3F)=O)OCC2)cc(F)cc(Cl)c1O 47756,CON(CCC(=O)NC(C)Cc1cnn(C)c1)C(=O)CCS(N)(=O)=O 47757,C1(CNC(=O)CN2CCN(C(=O)Cc3ccsc3)CC2)COCCOC1 47758,c1(CC)c(C(=O)NCC(C(C)C)NC(=O)CCC(C)(C)C#N)cnc2ncnn12 47759,c1(C(=O)NC2CCC(C)(CNC(C3(CCOC)CC3)=O)C2)nn(C)c(C)c1Cl 47760,C1(CNC(c2c(CC)ocn2)=O)C(C2CC2)CCN1C(c1scnc1C1CC1)=O 47761,C=CCCC(F)(F)C(=O)N1CC2CC2(CNC(=O)CC(C)(C)C(F)F)C1 47762,N1(C(C(CC)N2CCCC2=O)=O)CCC(N(C(=O)C(C)(C)F)CCO)CC1 47763,C1(CCC)CN(C(=O)Cc2occc2C)CC1NC(=O)C(C)CNC(C)=O 47764,C(C(=O)NC1CC(F)(F)C1)(C1=NOC2CC12)N1C(C(C)C)CC(F)(F)C1 47765,N1(C(C(C)SC(F)(F)F)=O)CCC(CNC(C23CC(CO2)C3)C)C1 47766,c1(N(C)CC2CCCN(C(C(C=C)O)=O)C2)ncc(C)c(C)n1 47767,C1(CNC(CCCCC)=O)CCC(C)CN1C(c1ccc(Cn2cccn2)o1)=O 47768,C1(NC(CCC#CC)=O)CCCCN(C(=O)CCCNC(C)=O)C1 47769,C1(CNC(c2n[nH]cc2Cl)=O)CN(C(c2coc(C(F)F)n2)=O)CC1O 47770,C(=O)(CC(C)(C)SC)NCC(CC=C)NC(=O)Cn1cc(Br)c(C)n1 47771,Cc1cc(C(C)C)ccc1C(=O)NC(C1CCN(C(=O)CC2CCOC2)CC1)C 47772,C1(CC)C(NC(C2(CN(C)C)CC2)=O)CCCN1C(c1ccc(SC)o1)=O 47773,c1(C(=O)NCC(C)NC(c2coc(N(C)C)n2)=O)cnn2cccnc12 47774,N1(CC)CCOC(C(N2CCCC(CNC(c3ncoc3C(C)(C)C)=O)C2)=O)C1 47775,Cc1cc2ncc(C(=O)NCC(C)(O)CNC(C3(C)CC4CC4C3)=O)c(C)n2n1 47776,CC1(C(N)=O)CCN(C(=O)N(c2nccnc2Br)c2cccc(F)c2)CC1 47777,C(=O)(C1=CCC(C)(C)CC1)NC(CCC)C(=O)Nc1ccsc1C 47778,C=C(Cl)CC(C(=O)NC(c1nc[nH]n1)CC)NC(=O)CN(C)C(C)C 47779,N1(C(COC2(c3n(C)ccn3)CC2)=O)CC2CCCC(C1)N2C(=O)CC=C(Cl)Cl 47780,CCC(C)C(C(=O)NC(c1cncn1C)CO)N(C(=O)C#CC(C)(C)C)C 47781,Cc1ccc2c(CN3CC4(CC4C(=O)Nc4c(C)cccc4Br)C3)c[nH]c2c1 47782,C1(NC(C2N(CC)C(=O)CC2)=O)CCC12CN(C(c1cnc(S)[nH]1)=O)C2 47783,N1(CN=c2sc(C#N)c(Cl)[nH]2)CCc2sc(NC(=O)CC3CC4CCC3O4)cc2C1 47784,CCCCC(CCC)NC(C1(N(C)C(C2CCOCC2)=O)CC1)=O 47785,N1(C(c2c(C)cccc2F)=O)CC(NC(=O)C=CC2CCCO2)CC2(CCC2)C1 47786,c1(C(=O)NCC(CN(C(C2COCCC2(F)F)=O)CC)(C)C)cc2occc2[nH]1 47787,C1(C(=O)NC(C=C)C2CC2)CCC(C)(C)N(C(=O)CCC(C)CN(C)C)C1 47788,CCC1C(=O)NC2CC(C2)OCC(=O)N1.c1(CC(C)N(C)C)nc[nH]n1 47789,N12CCC3(CC3C1)NC(=O)c1[nH]cc(c1)C2=O.c1(NC(=O)N)cccc(Cl)c1.CO 47790,C1(N(C(=O)CN(C)S(N)(=O)=O)CC)=NN=CC12CC(C)C2 47791,C=C1CCN(C(=O)C(CC2CCCC2)NC(C2(C)CC=CCC2)=O)CC1 47792,c1(CCC)ccc(NC(C2CN(C(=O)CCCOC(C)(C)C)CC2SC)=O)cc1 47793,N1(C(c2ccc(C)cn2)=O)CC(C)CCC1CNC(=O)C(C1CCC1)C1CCC1 47794,C1(C(=O)NC(CNC(C2(c3cccc(C)c3)CC2)=O)C2CC2)CCc2ccnn2C1 47795,C(C(N=c1ccnc(NCCCn2cccnc2=O)[nH]1)c1ccccc1)N(C)C 47796,C1(NC(C(C2CC2)SC)=O)CC(C)(NC(=O)CCC=CC(C)C)C1 47797,CCC(CN=C(NCC1CCCN1CC)N(C)Cc1cccc2[nH]ccc12)OC 47798,C(=O)(C(O)C1=CCCCC1)N(CCN(C(c1c(C)nc(CCC)s1)=O)C)C 47799,c1(C(C)C)ncc(C(N2CCN(C(=O)C=CC(C)(C)C)CC2)=O)cn1 47800,CCCC(CCCNC(=O)COc1ccsn1)NC(=O)C=Cc1c(C)coc1C 47801,N1(C(CC2C=C(C)CS2)=O)CCC(NC(C2CC(C)(C)C2)=O)C1c1ccccc1 47802,CC=C=CCCN=C(NCCC#N)NCc1cc(C)ccc1OC 47803,CC1CCC(c2nnnn2-c2ccccc2)(NCc2cccc(F)n2)C1 47804,C1(C(N2CC(=C(CNC(=O)CCc3nccs3)F)C2)=O)=NC2C(=C1)C=CC=C(O)C2 47805,c1(CC(N2C3(CNC(=O)CCC4OCCO4)CCC3CC2)=O)cc(F)c(F)cc1F 47806,n1(CC(=O)NC2C(C)N(C(=O)C=CC3CC3)CC2)sc(=O)c2ccccc12 47807,c1(CC)cc(C(=O)NCCCN(C)C(C2CCCCN2N=O)=O)ccc1Cl 47808,N1(C(CC2(OC)CN(C(=O)C=C(C)C3CC3)C2)=O)CC(C(N)=O)OC(C)C1 47809,C1(CCC)CCN(C(C2CCN(C(=O)CCc3cn(C)cn3)C2)=O)C1 47810,C1(C(=O)NC2CCCCN(C(c3ccc[n+]([O-])c3)=O)C2)CCn2c(O)nnc2C1 47811,c1(CC(=O)N(C2CCN(C(c3c(COC)cc[nH]3)=O)C2)C)cncnc1O 47812,C1(NC(C(=O)NCC)=O)COC2(C1)CN(C(c1cnc(OCC(F)F)cn1)=O)C2 47813,c1(C(=O)NC2CC3CN(C(C(C)(C)OC)=O)C(C2)C3)c(C)nc2sc(C)nn12 47814,N1(NC(c2c(F)cnc(Cl)c2)c2cccc(Cl)c2)CCCC2CCCC12 47815,c1(C(N2C(C(=O)NC(C)CO)C(O)CC2)=O)cc2c(s1)CCOC2 47816,C1(c2onc(C)n2)(NCCN2CCC2(C)C)CCNCC1 47817,C(=O)(C(F)C(C)CNC(=O)Nc1ccc(O)cn1)N(C)Cc1c(C)cco1 47818,C12(CNC(=O)C=CC(F)(F)F)CCC1CCN2C(=O)CCN1CCCC1 47819,C(=O)(CC(O)C(C)(C)C)N1CCC(NC(Cn2c(C)ccn2)=O)C1C 47820,N1(C(C(COC)C)=O)CCC(C)(CNC(=O)CN2CCC(C(N)=O)CC2)C1 47821,C12(CCN(CCCCc3cccs3)CC1)C(=O)N2.C(=O)(CCc1nn[nH]n1)OC 47822,c1(OC)ccc(NCCN2CCC(CO)C2)cc1.N12CCOC(C1)CC2=O 47823,c1(C(N2C(CN(C(CC(C)C3CC3)=O)C3CC3)CCC2)=O)c(C2CC2)cnn1C 47824,C1(C(N(C)CC2(NC(=O)COc3cccc(Cl)n3)CC2)=O)CCN(CCO)C(=O)C1 47825,C(CC(O)CC(=O)N(C)CCN(C(=O)C(C)(F)CC)C)SC 47826,[N-]=[N+]=Nc1ccnc(CNC(=O)NC2COC3(CCCC3)C2)c1 47827,c1(C(=O)NCCCC(CCC)NC(c2nc(Cl)oc2C)=O)cnc2ncccn12 47828,Cc1nc2ccc(C(=O)NC3CC(CCNC(=O)CSC(F)F)C3)cn2n1 47829,C(C)(CNC(c1ccncn1)=O)(CC(C)C)NC(Cc1nc(C(C)OC)sc1)=O 47830,N1(C(C(C(C)(C)C)NC(C(C2CCC2)SC)=O)=O)CCC(O)C(F)(F)C1 47831,c1(CC)nc(C)oc1C(N1CC2C(N(C(=O)C(CC)SC)C)C2C1)=O 47832,Cc1cc2c(C(N3CCC(CNC(=O)CSC(F)F)CC3)=O)cccc2[nH]1 47833,C1(C)(CN(C(CC)CO)C(c2ccco2)=O)CCCN(c2cc[nH]c(=N)n2)C1 47834,c1(N2CC(CNC(C(c3cccnc3)OC)=O)OCC2)cc(C)c([N+](=O)[O-])cn1 47835,n1(CCN(S(C)(=O)=O)C(C)C)c(Cc2cc[nH]n2)nnc1-c1cnn(C)c1 47836,Cc1nc(C(=O)NCC(C)(C)CN(C)C(C2CCSC(C)C2)=O)cn1C 47837,CC1(F)CN(C(=O)Cc2cccc([N+](=O)[O-])c2)CCN(C(c2cccc(=O)o2)=O)C1 47838,C1(CC=O)C(=O)N(C)C(C)(C(=O)NCCOC(F)F)C1CC 47839,Cc1ncc(N)cc1C(=O)NCC(C)NC(=O)C(c1cscn1)N(C)C 47840,Cc1cccc(Br)c1S(=O)(=O)NCCCc1ccc([N+](=O)[O-])cc1 47841,CN1C(C(=O)NC2CC(O)(CNC(=O)CC(F)(F)Cl)C2)CCS1(=O)=O 47842,c1(NC(c2n(CCC)ncc2)=O)ccc(NC(=O)C(C2(O)CCCC2)F)cc1C 47843,Cc1nsc(C)c1C(=O)NCC1CC(NC(C2CC2c2ccn(C)n2)=O)CCO1 47844,C(CC(=O)NCCS(C)(=N)=O)(C(F)F)NC(Cc1cc(C)n(C)n1)=O 47845,C1(O)(CCNC(C2(CCC)CCC2)=O)CCN(C(=O)Cn2ncc(Cl)c2C)C1 47846,c1(C2C(C=C)CC2)nc(-c2cnn(CCO)c2)nn1C1CCC(CC)CC1 47847,C(=O)(C(F)(F)CC(C)C)NC1(CCOC)CCN(C(=O)Cn2cc(Cl)cn2)C1 47848,C1(CCC(=O)N(C2CCN(c3ncccn3)C2)CC)CCCOC1 47849,C(CS(=O)(=O)CC(=O)N(C)CC1CCCCN1C(c1coc(C(F)F)c1)=O)OC 47850,N1(C(C2C(CCC)C2)=O)CC(CNC(c2cccc(CC)c2N)=O)CC12CCC2 47851,c1(NC(C)=O)cnc(O)c(C(=O)N(C)CC2CCCN2C(=O)C=C(Cl)Cl)c1 47852,C(C(C)(C(=O)N1CC(CC(F)C(=O)NC2CC(O)C2O)C1)OC)OC 47853,N1(C(C2(C)C(C)OCC2)=O)CC(C2(NC(c3cnnn3C)=O)CC2)C1 47854,C1(C(C(=O)CC(=O)NCC)N(C)C(C2SCCS2)=O)CC=CCC1.C1(C)CC1 47855,CCC1=NOC(C(=O)NCC(CO)NC(c2cccc(C(=O)OC)n2)=O)C1 47856,N12CCC(CC1C1CC1)C2=O.c1(NC(C2(F)CC2)=O)ccccc1-c1ccsc1 47857,Cc1nc(CC(N2CCC(CF)(NC(C3CCC(=O)O3)=O)C2)=O)c(C)s1 47858,C1(NC(=O)C(C)OC2CCCC2)CN(C(=O)CCc2cnc(C)s2)CC1CCC 47859,c1(CC(C)C)c[nH]c(C(=O)N(C)CCNC(=O)CC2C=CCC2)c1 47860,c1(C(=O)NCCCN(C(C2(F)CC=CC2)=O)CC)cc(C(C)C)nc(O)c1 47861,O=C(C(O)CC(F)(F)F)NCCC1CCCN1C(=O)Cc1cccc(C(F)F)c1 47862,CCCC(O)CC(=O)NCC(C1CCCC1)NC(=O)C(c1cccc(F)c1)C 47863,Cc1ncnc(C)c1CC(N1CC(NC(=O)C(=O)NC2CC2)CC(C)C1)=O 47864,C(N=c1[nH]c(C#N)c(Cl)s1)C1(F)CCN(C(C(C)Oc2cnccn2)=O)CC1 47865,c1(C(=O)NC(CC#C)CNC(=O)CCC=C=C)c(C)[nH]c2ccc(OC)cc12 47866,c1(SC)c(C(N2CCCC2C2CCN(C(c3[nH]cc(C)c3C)=O)C2)=O)cnn1C 47867,c1(C(C)=O)ccc(Cl)c(NC(c2ccc(-c3c(C)noc3C)c(C)n2)=O)c1 47868,CC1CCCN(C(=O)C=CC(C)(C)NC(C23CC2CNC3=O)=O)C1CO 47869,N1(c2cc(Nc3cc(SCC)cc(F)c3)ncn2)CCCC(C)(C#N)C1 47870,C(CCCCC(=O)NC(CC)C(C)(C)O)NC(C1C(=C)C1C(=O)OC)=O 47871,N1(C(c2nc(CC)oc2)=O)CC(C)C(NC(=O)CNc2cccnc2Cl)C(C)C1 47872,N1(C(C(CCSC)OC)=O)CCN(C(=O)Cc2cnns2)CC1c1ccccc1 47873,N12CCc3c(n[nH]c3C1)C2=O.c1(NCc2nc(C)[nH]n2)cc(Br)cc(Cl)c1F 47874,Cc1cc(F)ccc1C(=O)NCC(C)NC(c1cccc(OCC(F)(F)F)c1)=O 47875,C1(C(C(N2CC(CNC(=O)CCn3cccn3)OCC2)=O)O)CCCCCCC1 47876,N#Cc1cn(CC(=O)NC2CN(C(C3NC(=O)C4CC34)=O)C2)c(=O)nc1O 47877,c1(-n2cc(C(=O)NC3CCN(C(C(C=CC)O)=O)C3)nn2)ccccc1F 47878,C1(NC(c2c(C)nns2)=O)(CO)CCN(C(=O)C(C)CSC(F)(F)F)C1 47879,C1(NC(CC(c2ccc(F)cc2)C)=O)CCCN(C(=O)CC2COC(=O)C2)CC1 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47898,N(C(=NCCSc1ccsc1)NC(N1CCCC1)C)Cc1n(CCC)ncn1 47899,c1(CC(CO)CNC2(C(F)(F)F)CC3CC3C2)ccc(F)cc1 47900,Cc1nnc2n1CC(C(=O)N(CCCN(C(=O)CCCC1OCCO1)C)C)CC2 47901,C1(C2CC2)(CNC(COCC(C)C)=O)CCN(C(c2ccc(C#N)s2)=O)C1 47902,C1(CCNC(C2C(=C)CC2)=O)CN(C(=O)C=Cc2cnc(C)s2)CCCO1 47903,c1(C(C(=O)NCC(CC)(C)NC(=O)CCC=CC(C)C)C)ccc(OC)cc1C 47904,N1(C(C2CCC(=O)NC2)=O)CCOC2CN(C(c3cnc4ccccn34)=O)CC12 47905,c1(NC(C(=O)N(C2CC2)Cc2ccc(C)c(C)c2)=O)cc2cccc(Br)c2cn1 47906,N1(C(Cc2cc(C)ncc2)=O)CC2C3CCC(C2C1)N(c1nc(Cl)ncc1Br)C3 47907,c1(NC(=O)CCc2cncnc2)ccc2c(c1)CN(C(c1n[nH]cc1Cl)=O)C2 47908,C1(C)(C(=O)NC2CC(CCNC(C3(OC)CCC(C)C3)=O)C2)C(C)(C)C1(C)C 47909,Cc1cccc(CC(=O)N(C2CCN(C(c3ncc(C(F)F)s3)=O)C2)C)c1F 47910,C(=O)(C(F)(F)CC(C)C)NC1C(NC(C(CC)c2cccnc2)=O)CCCC1 47911,C(=O)(C(CC(C)C)C(C)C)NC1CC2(C(C(N(CCOCC)C)=O)C2)C1 47912,C1(CNC(C=CC(C)NC(C(c2cnn(C)c2)C)=O)=O)CNC(=O)C1 47913,c1(C(=O)NCC2CCN(C(=O)CC34CCCC3C4)C2)c(F)ccc(C2CC2)c1Cl 47914,CC(N=[N+]=[N-])C(=O)NCC1CC(F)CN1C(=O)CC1NC(=O)NC1=O 47915,c12cccc(n1)OC2=O.N1(C2CC2)CCC(CNC(C2(C(=O)NC)CC2)=O)C1 47916,C1(CSC)CCCN1C(=O)C(Cc1cc[nH]n1)NC(c1ccsn1)=O 47917,Cc1nc(S)sc1CC(N1CCC(N(C(=O)CCOC2CCCOC2)CC)C1)=O 47918,C1(C(N)=O)CCN(C(C2CCC2CNC(c2ccoc2)=O)=O)CC1 47919,c1(Nc2ncc(SC)s2)ccc2c(c1)CN(C(c1cnc(C)c(C)c1)=O)C2 47920,N1(C(CN2CC(C)C2)=O)CC2CC(NC(c3ccn(C4CCCCC4)n3)=O)C(C2)C1 47921,N1(CC)CS(=O)(=O)CC1C(=O)N(C)CCSc1cn(Cc2nccs2)nn1 47922,Cc1ccncc1C(=O)NCC#CC(=O)NCc1ccco1 47923,N1(C(C(F)OC)=O)CCC2CCN(C(C3CN4CCN3CC4)=O)CC12 47924,c1(CC)nn(C)c(C(=O)NCC2CN(C(c3ccc(SC)o3)=O)CCC2C)c1Cl 47925,C1(C(N(C(CCc2cnn(C)n2)=O)CC2CCCO2)=O)CC(C2CC2)C1 47926,c1(C(=O)OC)cc(=NCC2CCC(NC(c3cc(C(C)(C)C)on3)=O)C2)[nH]cn1 47927,C1(NC(C2C(C(N(C)C)=O)C2)=O)CC2CC(NC(C3(C4(O)CCC4)CC3)=O)C1C2 47928,c1(CC(=O)N(CCOCCNC(c2c(CC)scc2)=O)C)ccc(F)c(OC)c1 47929,C(CCCCCC(=O)Nc1cncc(C#N)c1)NC(CC1(OCC)CCC1)=O 47930,CCC(CC)C(C)C(=O)NCC1(C)CCCN(C(C2(C3CCC3)CCC2)=O)C1 47931,C#CC1(C(N2CC(O)(C(C)C)C2)=O)CCN(C(=O)C(c2ccn(C)c2)C)C1 47932,N1(C(C2(CC#C)CCCCO2)=O)CC(NC(=O)CCCC2CCCC2)CC(F)C1 47933,N1(C(=O)Cc2ccoc2)CC=C(CC(=O)N2CCC3CC23)CC1.C1CC1 47934,c1(C(C)(C)C)nnc(N2CCN(C(c3ccncc3)=O)CC2)n1Nc1ccccc1 47935,c1(C(=O)NCC2N(CC(=O)NC(N)=O)CCC2)ccn2ccnc2c1 47936,C1(C(C(=O)N(CCCC)CC)C)CCCN(C(=O)C(OC)OC)C1 47937,c1(N(C2CCCC(C#N)C2)C)ccc2c(c1)OCCO2 47938,c1(C(N2CC(NC(C(C3CCOCC3)OC)=O)C(F)C2)=O)cc(N)ccc1SC 47939,C1(CCF)(NC(c2ccsc2C(F)F)=O)CCN(CC2(O)CCOCC2)CC1 47940,c1(C(N2CC(NC(C3C(C)C3C)=O)C3(C2)CC3)=O)cc2cc(F)ccc2[nH]c1=O 47941,c1(CC)cc(F)c(N(c2ccnc(C3CC3)n2)CC2CC3CC3C2)c(F)c1 47942,CCCCC(O)C(C)C(=O)NCCC1CCCCN1C(c1cccn1CC)=O 47943,Cc1cc(CC(=O)NC(C)C(C)(C)NC(=O)Cc2csc(Cl)c2)n[nH]1 47944,N1(C(c2cccc(CC)n2)=O)CCC2C(CCCN2C(=O)Cc2cn[nH]c2)C1 47945,N1(C(c2ccn(CCNC(CCN(CCC)C)=O)c2)=O)CCC12CCC(O)CC2 47946,C1(F)(CNC(c2n(CC)ncc2Cl)=O)CCN(C(C2CC3CC3CC2C)=O)CC1 47947,c1(CC)nc(=N)[nH]c(=NCCCCN(C2CCn3nccc3C2)CC)[nH]1 47948,N1(C(C(C)NS(CC)(=O)=O)=O)CC2(CCC(NC(=O)C(C)CS(C)=O)CC2)C1 47949,C(=O)(C1CCCc2nncn21)N(CCCNC(C(C)SC)=O)CC1CCCC1 47950,C1(CNC(c2on(C)c(=O)c2)=O)(CO)CCN(C(=O)Cc2cnns2)CC1 47951,C(=O)(C1=NOC(C)C1C)NC1C(OC)CN(C(=O)CCC2CC2)C1 47952,c1(C(N2CC(CNC(=O)C=CC3CCCCCC3)C2)=O)ccc2nnn(O)c2c1 47953,C1(C(=O)NCC2(F)COCCN(C(=O)C3=NOCC3)C2)CC2(C1)CC21CCC1 47954,CC(CN(C(=O)C(Cn1cccn1)NC(=O)COc1ccccc1)C)C(F)(F)F 47955,C1(C(=O)NC(C)C(CO)NC(c2cnncc2O)=O)CN(C)CCN(C)C1 47956,CC1=C(C(=O)NC2(C)CC(NC(C3OC(=O)NC3(C)C)=O)C2)CCCO1 47957,Cc1nc(Cl)ccc1CNC1CCN(C(=O)CSc2nccn2C)CC1C 47958,CCS(=O)(=O)CC(CO)NC(=O)C(=O)NCCc1scnc1C 47959,C1(CC(=O)NCC2CCN(C(C3CC3C(F)(F)F)=O)C2)CCC2(CC1)OCCO2 47960,Cn1cc(SCC(=O)NCC2CC(O)(CNC(c3cc(C(N)=O)c[nH]3)=O)C2)cn1 47961,C(=O)(C1CC(=O)Nc2cc(F)ccc21)N(C(CNC(Cc1ncc(C)o1)=O)C)C 47962,Cc1nccc(CONC(C2CC(F)CN2C(=O)CC2CC=CCN2C)=O)n1 47963,N1(C(C2(CC#C)CCCC2)=O)Cc2[nH]nc(C(=O)NOCCCO)c2C1 47964,c1(C(=O)NC2C(NC(C(C)(C)n3ccnn3)=O)C2)cc(F)c(Cl)cc1Cl 47965,N1(C(c2nc(C(C)C)oc2)=O)CCCC(C)C1CCNC(c1cn(C)c(O)n1)=O 47966,CCCCC(CC)CC(=O)NCC1CCC2CN(C(c3ncc[nH]3)=O)CCC2C1 47967,C1(O)(C(C)N(C(=O)COC2CCCC2)C2CC2)CN(C(=O)CCC2CC2(F)F)C1 47968,CC(C)C(O)C(=O)NC(C)CCCNC(=O)CC(C)C1CCCCC1 47969,C(C)(CCC(=O)N(CCCNC(=O)Cn1nc(C)cc1C)C1CC1)SC 47970,C(=O)(C(CCC)OC)NC(CCC)CNC(=O)C(=O)NC1CC1 47971,C1(O)(CNC(c2nc(CNC(CS(=O)(=O)NC)=O)oc2)=O)CC2CCC1O2 47972,C12(NC(C(=O)NCC3CC3)=O)CCCN(c3ccn4nccc4n3)CC1C2 47973,Cc1cccc(CNC(=O)CC2CCN(c3cc(C(=O)O)ccc3F)C2)c1C 47974,n1(CC(=O)NC2C(SC)CN(C(C3(C(F)(F)F)CCCC3)=O)C2)nc(C)c(Cl)c1C 47975,CC1CC(C(=O)NC2C=CC(C)(C)CC2)CN(C(C2CCCN2C)=O)C1 47976,Cc1nc(O)sc1C(N1CC(CC(=O)NCc2ncccc2Cl)CC1C)=O 47977,N1(C(C(=O)N(C)C)=O)CC(CNC(=O)Cc2cccc(F)c2Cl)C2(CC2)C1 47978,c1(C(N(C2CCN(C(c3cscc3SC(F)F)=O)C2)C)=O)ccc(CO)nc1 47979,c1(C(N2C(CN(C(=O)C=CCO)CC#C)CCC2)=O)cc(Br)c(CC)o1 47980,C1(NC(=NCCC=C)NCC2(C3CCC3)CC2)CCOC2(CCOCC2)C1 47981,N1(C(CC(C)C2CC2)=O)CC(C(=O)Nc2cccc(O)c2)CC12CCC2 47982,Oc1cnc(Br)cc1CN1CCC(NS(C)(=O)=O)C1 47983,N1(C(C(N2CC(C)CC(C)C2)=O)=O)CCn2c(cnc2C(N2CCOCC2)=O)C1 47984,N1(CCC)C(=O)CCC1C(=O)NC(CNC(=O)C=C1CCSCC1)C1CCC1 47985,CCC1(C(=O)NCC(O)CN(C(=O)Cc2cscn2)C)CCCc2ccccc21 47986,Cc1nn(CC(=O)NCC2CCCN(C(=O)CC3(C)CCC3)C2)c2ncccc12 47987,C1(C(=O)NC2C(CNC(c3cnoc3-c3ccoc3)=O)CC2)CC2(C1)CC2(F)F 47988,c1(C(=O)NCC(CNC(C(C(C)(C)C)SC)=O)F)cc(Cl)c2n[nH]cc2c1 47989,Cc1cc(Cl)cc(C(N2CCOC(CN(C)C(c3ccc(F)s3)=O)C2)=O)c1N 47990,C(=O)(C1=CCOCC1)NCC(CCNC(C1(CCOC)CCC1)=O)O 47991,c1(C(=O)NC(CC=C)CNC(=O)CC(=O)OC)ccc(Br)c(OC)c1 47992,CCCCCC(O)CC(=O)NC(CC(C)(C)C)C(=O)NCc1conc1C1CC1 47993,c1(SC(c2ccc(F)c(F)c2)C)cc(Br)cc(COC(F)F)c1O.c1(=O)c(=O)[nH]1 47994,c1(OC(=O)NC(c2cn(CCO)nc2Br)CC(=O)OC)ccc(F)cc1Br 47995,Cc1ccc(CC(=O)NC(C2CN(C(C3CC3(C)C)=O)C2)C)cc1Cl 47996,C1(C(=O)OCC)CCCC1NC(=O)OCCCc1scnc1C 47997,Cc1cccnc1C(=O)N(CC(O)CN(C)C(c1cc(CC(C)C)nn1C)=O)C 47998,CC1(C(=O)Nc2cc(=O)n(Cc3ccccc3)[nH]2)CCN(C(C2CC2(C)C)=O)CC1 47999,c1(NC(c2cccc(C)c2)C)ccc(S(=O)(=O)NC(C)(CC#N)C2CC2)cc1Br 48000,c1(C(=O)NC(C)CN(C)C(c2ccns2)=O)cc(S(=O)(=O)N(C)C)oc1C 48001,C1(NC(C(C)SCCOC(C)C)=O)CC(C)(NC(=O)C(=O)NC2CCCCC2)C1 48002,N1(C(C2CC(=C)C2)=O)CCCC(NC(c2cccc(=O)o2)=O)C(F)C1 48003,c1(CCC(=O)NCCCCNC(C2CCC2C2CC2)=O)c(Cl)cccc1Cl 48004,c1(C(=O)NC(C2CCCN(C(C3=C(C)OCC3)=O)C2)C)cc2c([nH]1)CCOC2 48005,N1(Cc2cn(CCCC)nc2)CCC2C(CCN2S(=O)(=O)CCBr)C1 48006,C(=O)(CS(=O)(=O)CC1CCCO1)NC(CCCNC(CC1CC(OC)C1)=O)(C)C 48007,C1(C=C)(C(NCCSC)=O)CCN(C(c2ccsc2)=O)CC1.N1(CC)CCCC1 48008,c1(CN(C(C2CC(=O)C2)=O)C2CC2)c(F)cccc1F 48009,N1(C(=O)CN2CC3CC3C2)CC2CCCN(C(C3CCC(F)C3)=O)C2C1 48010,CN1CC(NC(c2cc(CNC(=O)C(C)(O)C3CC3)cs2)=O)CC12CCC2 48011,C(C(=O)NNC(=O)C(=O)OC(C)(C)C)(C(C)(C)C)SC.C(CS)O 48012,C12(NC(CCC3CCN(C(C(CC)OC)=O)C3)=O)CCCN(CCC1)C2 48013,N1(C(CC2C(C)CCC2)=O)CC2CCC1CC2NC(c1cnn(C)n1)=O 48014,c1(C(=O)NC2CN(C(c3cccs3)=O)C3CCCC23)cc2ccnc(Cl)c2s1 48015,Cc1nc2cc(C(=O)NCC3(NC(C4CCN(CC(F)(F)F)C4)=O)CC3)[nH]c2s1 48016,c1(C(N(CCCCNC(c2cc(C(C)=O)on2)=O)C)=O)cc(C)c(Cl)cn1 48017,c1(N(CCNC(C2(F)CCCC2)=O)CC)ncc(C#N)cc1F 48018,N1(C(C(c2ccnn2C)C)=O)CCCCC1C(C)(C)CNC(=O)C1=CCCC1 48019,n1(C(=O)OC)nccc1S(=O)(=O)N1CCSCC1CC.CC 48020,CCC(CNC(=NCc1cc(-c2ccccc2)no1)NCC(F)F)(CC)SC 48021,N1(C(C2N(CC#C)CCC2)=O)CCC(NC(C2C(C)OC(C)C2C)=O)C(F)C1 48022,CP(C)(=O)c1ccc(C(N2CCC(CNC(=O)C3=CCCCC3)C2)=O)cc1 48023,c1(C(=O)NCC2(NC(C3CC3Br)=O)CC2)cnc(C2CCC2)s1 48024,c1(NC(C)=O)ccc(F)c(C(=O)NCC(NC(C2CCCN2C)=O)CC2CC2)c1 48025,C1(CC(=O)NCCCOCCNC(N)=O)CCCCCN1C.C1CO1.C1CO1 48026,c1(OC)ccccc1C(=O)NCCC1CC(NC(c2ccc(CO)cn2)=O)C1 48027,N1(C(C2(COC)CCC2)=O)CCCC2(NC(=O)CCc3cccc(F)c3)CC2C1 48028,c1(C(=O)NC2CN(C(c3coc(Cl)n3)=O)CC23CC3)ccc2cccnn12 48029,c1(C(=O)NC2CCCN(C(CC(CCC)O)=O)C2)cnc2c(C)c(Cl)ccc2c1 48030,CC(CCNC(=O)CNS(N)(=O)=O)CCNC(=O)C(C)(C)C1CCOCC1 48031,C1(C(N(C2CC2C)C)=O)CC12CCN(C(=O)Cc1cccc(Br)c1)CC2 48032,CC(=O)CCCC(C)C(=O)N1CC(CC(N2CCC(F)(CF)CC2)=O)CC1(C)C 48033,C1(NC(CC2CC(CC)C2)=O)C2CC(NC(c3cc(C(N)=O)cs3)=O)CC12 48034,C1(C(N2CCOCC2CNCc2ccc(Br)[nH]2)=O)CCCCC1(F)F 48035,c1(C(N(CC(C)O)CCNC(c2c(C)n(C)nc2)=O)=O)cccn2c(C)cnc12 48036,CC1(NC(c2csc(Cc3ccccc3)n2)=O)CN(C(=O)CC2CC3(CC3)C2)C1 48037,N1(C(C=CC(C)C)=O)CC2CN(C(=O)Cn3ccccc3=O)CCC12 48038,C1(CCOC(C)=O)CCN(C(C2(NC(C(CC)(CC)CO)=O)CC2)=O)CCC1(F)F 48039,CCCCCCC(C)C(=O)N1CCN(c2nnc(-c3cc(Cl)cc(SC)n3)o2)CC1 48040,Cc1nc[nH]c(=NCC(C2CC2)N(C(=O)C(c2c(C)nn(C)c2C)=O)C)c1C#N 48041,c1(CC(N2CC(NC(CC(C)(C)O)=O)C(C)(C)CC2)=O)ccc2cccnc2c1 48042,C12(CNC(C3C(OC)CCC3)=O)CCCC1N(C(C1CCN(C)CC1)=O)CCC2 48043,N1(C(C(CC)C#N)=O)CCN(C)CC1C(=O)NCC1CC(OC)C1 48044,CCCC(CCCNC(=O)CNC(c1ccco1)=O)NC(=O)C=Cc1nc(C)cs1 48045,N1(C(C(CCCC)C)=O)CC(NC(c2cc(CC)on2)=O)C(C2CC2)C1 48046,CCCC(C)CCNC(C1(CNC(=O)C(C)OCOC)CC(C)(C)C1)=O 48047,C1(NC(CN(C)C2CC2)=O)CCCC(N(C(=O)CCN2CCC(C(N)=O)CC2)C)C1 48048,N1(C(C2N(C)CC(O)C2)=O)CCN(C)C(CNC(=O)COC2CCC2)C1 48049,c1(C(=O)NCC2(C)CCN(C(c3[nH]cnc3C#N)=O)C2)cnc2ccc(C#N)cn12 48050,Cc1cc(NC(C2CCCCCC2)=O)ncc1C(F)(F)F 48051,C(=O)(CC(O)C1CCC1)N(CCCOCC=CC(=O)NC1CCCC1)C 48052,C1(C(=O)NC(C=C)(C)C)CCC(C2CC2)N1C(c1cc(Cl)cs1)=O 48053,N1(C(c2cn(CC)nn2)C(=O)NCC2CCCO2)CC2(CO)CC2(C(F)(F)F)C1 48054,C1(C(N2CC(CCNC(C3(C)CCNC3=O)=O)C2)=O)CC12CCSCC2 48055,N1(C(C=C(CCC)C)=O)CCC(C2CC2)C1CNC(=O)Cc1c(C)cccc1C 48056,N1(C(c2c(CC)nc(C)[nH]2)=O)CC(C2CN(C(C34CC5CC3C4C5)=O)C2)C1 48057,c1(-c2nc(C(N3CCOC4CC34)=O)sc2)cccnc1C(F)(F)F 48058,C(=O)(C(C)CC(C)(C)C)N1C(CNC(c2ccc(OC)nc2C)=O)CN(C)CC1 48059,C#CCC(CC(=O)NCC1=CCCOC1)NC(C1CC1C1CC1)=O 48060,c1(N2CCC(C(C)NC(=O)CCNCC(F)(F)F)CC2)nc2ccc(F)cc2o1 48061,C1(CC2CCCC2)C(=O)N1.C(CC(C)O)N(C1C(C)C1)C 48062,N1(c2c(C=O)cncn2)CC2CCN(C(c3cn(C(F)(F)CO)nn3)=O)CCC2C1 48063,C12(C(=O)NCC(CNC(c3ccn4ncnc4c3)=O)O)CCC(O)(CC1)CC2 48064,C1(NC(CN(C)CCO)=O)CCCN(C(=O)CC(O)C2CCCC2)C1 48065,C1(CCNC(C(C)(C)OC)=O)C(C)CCCN1C(=O)C(=Cc1ccc(C)cc1)C 48066,C1(NC(c2c(C)nc(C3CC3)[nH]2)=O)CC2CC(NC(=O)C(O)CC(C)C)CC2C1 48067,C1(NC(c2nn(C)c(C(F)F)c2)=O)CC2CCC(C1)N2C(=O)C(C)(C)C1CCC1 48068,C1(C(=O)NCCCCC(C)NC(=O)CC(C)(C)c2cccs2)CC(=O)OC1(C)C 48069,N1(C(c2cc(C)c(O)nn2)=O)CCC(C2CCN(C(=O)Cc3scnc3C)C2)C1 48070,C(=O)(CCCC(C)(C)C#N)NCC(C1CCC1)NC(c1snc(C)c1N)=O 48071,C1(C(=O)N=c2cco[nH]2)N(C(=O)NC(=O)NC2CCS(=O)(=O)C2)CC12CCCC2 48072,Cc1n[nH]c(C)c1OCC(N1CCC(C)(NC(=O)C(C)OCCN(C)C)C1)=O 48073,C1(CNC(Cn2nc(C)oc2=O)=O)CC(C(=O)NCC(C)(C)C#N)=NO1 48074,CCC(O)C(C)C(=O)NC12CC(C1)N(C(=O)CCc1cncnc1)C2 48075,c1(CCCC(=O)NC2CCC(NC(c3c(Cl)cn(C)n3)=O)C2)cc(F)ccc1Cl 48076,S(=O)(=O)(c1cc(Br)cc2c1OCC2)NC(C1C(NC(Cc2ccc(C)cc2)=O)C1)=O 48077,Cc1cccc(CCNC(C2CCCN2C(=O)Cc2ccnc(C)c2)=O)c1 48078,CC1C(=O)N2CCCN2CC(C)(C)CCOC1CCCCNC(=O)CCS(C)(=O)=O 48079,C(=O)(C1CCCc2c[nH]nc21)N1CC(CNC(CC(C=C)C)=O)C1 48080,C12(CNC(c3c(CC)occ3)=O)CCC1CN(C(=O)Cc1cccc(F)c1F)C2 48081,c1(N(CC(=O)NC)C)nc(=NC)nc(N(C)Cc2cnc(CC(C)C)s2)[nH]1 48082,C12(C(=O)NCCCOC(=N)O)CC(CN1C(=O)CC1CCOC1)C2 48083,O=C(C#CC1CCOCC1)NCC1CN(C(c2ccc(C(F)F)o2)=O)CC1(F)F 48084,c1(C(=O)NCC(C2CC2)NC(C(C(=O)OCC)OC)=O)cc(S(C)(=O)=O)oc1C 48085,C1(CC)CN(C(C2(NC(=O)C(C)(C)OC)CC2C)=O)CCC1CO 48086,c1(OC)ccc(Cl)cc1C=CC(=O)NCC1CCC(NC(C2CC2(Cl)Cl)=O)C1 48087,CC(CS(C)(=O)=O)C(=O)NCCN(C(=O)C=Cc1cnccn1)C 48088,S1(=O)(=O)c2ccc(Br)cc2N2CCC(C2)N1CC.CCNC 48089,C#Cc1ccccc1CC(N1CC(F)CC1CNC(c1cc(OC)n(C)n1)=O)=O 48090,c1(C(=O)NCC(C)N(C(c2c(C)nns2)=O)C)cc(C2(Cl)CC2)n(C)n1 48091,C(=O)(C(C)(C)C(C)NC(c1ncccc1C)=O)NC(CCC)c1ccco1 48092,S(=O)(=O)(c1ccccc1C1CCN(C(=O)OC)C1)NC1CCN(CCC)CC1 48093,CC(C)CC(O)C(=O)N1CCN(C(=O)Cc2ccsn2)CC1c1cccc(F)c1 48094,CC(C)CC(C)(O)CNC(C1CC(CCNC(c2cccc(=O)n2C)=O)C1)=O 48095,c1(C(=O)NC2(CCCC(=O)N(CC(C)O)C)CCC2)ncn2c1CCC2 48096,CCCC(CNC(c1coc(C(C)C)n1)=O)C(=O)Nc1cn(C)nc1O 48097,C1(CNC(CCN(CCC)C)=O)C(C2CC2)CCN1C(c1cnc(CO)s1)=O 48098,C1(OC)CC(C(=O)NCCCN(C(=O)CS(=O)(=O)NC)C(C)C)CC1OC 48099,Cc1cc(Br)ccc1-n1nnnc1C1(NCCCc2ccsc2)CCC(C#N)C1 48100,C(=O)(C1=NN2CCCN=C2N1)NC1CCN(C(c2c(C)cc(F)s2)=O)CC1C 48101,c1(CC)nc(CC(=O)NCC2(F)CC(NC(C3CCOC3C)=O)C2)cs1 48102,c1(C(=O)NCCC2CN(C(c3cc(CC)cc(Cl)c3)=O)C2)c(F)ccc(C)c1F 48103,N1(C(C2(CCCC)CCC2)=O)CC(NC(=O)Cc2coc(C(F)F)n2)C(C)C1 48104,C1(C)(C(N(CCCCNC(c2ncoc2C2CCCO2)=O)C)=O)CC=CCC1 48105,N1(C(C(CCC)N(C)C)=O)CC2CC(NC(=O)C(C3(O)CCCC3)F)CC1C2 48106,c1(C(N(C2CCN(C(c3ccc(CC)s3)=O)C2)CC)=O)c(OC)nsc1OC 48107,C1(NC(=O)CC2CSC2)CCN(C(c2cscc2Br)=O)CC1 48108,C(C(=O)N1CC(NC(=O)Cn2nnc(C3CC3)n2)CC(F)C1)(C(C)(C)C)OC 48109,N1(C(C(C)(CO)OC)=O)CC(C(N2CCC23CCC3)=O)C2(CCC2)C1 48110,C(CO)(C(C)NC(=O)Cn1nnnc1C1CC1)NC(CN(S(C)(=O)=O)C)=O 48111,C(C(C)C(C)C(=O)NCCOCCN(C)C(c1cc(C)nn1C)=O)OC 48112,C1(CC#C)CN(C(C2CCN2C(=O)COCC2CCCO2)=O)CCO1 48113,C1(Cl)(C(=O)NC(CNC(C2CC(SC)C2)=O)C)CC12CCOCC2 48114,N1(C(CC(C)c2ccco2)=O)CC2(CCCC(CNC(c3cc(Cl)on3)=O)O2)C1 48115,c1(C(=O)NC2C(NC(C(CC=C)C)=O)CCC2)c(N)cc(OC)cc1F 48116,C=CCC(CC)C(=O)NCC=CCNC(C1CCCN1C(c1ccc(C)cc1)=O)=O 48117,c1(C(=O)OCCC(CCC)C)ccc(C(F)(F)F)c(F)c1 48118,C(=O)(C(COC)CC)NCC(=O)N(CC(CCC)O)CC.C(C)C 48119,c1(NC(CC)CC(F)(F)F)ncccc1S(=O)(=O)NC(c1ncccn1)(C)C 48120,Cc1nccc2c(=O)c(C(=O)NC3CCC4(C=C4)N=N3)c[nH]c12 48121,c1(NC(=O)CCN(C(=O)CCCN2CCCC2)CC2CC2)cccc2cncn12 48122,c12nc(C)c(o1)C(=O)NC2.C(CCCCC1CC1)NC(CN(C(C)=O)C)=O 48123,C(N=c1[nH]c(=NC(C)c2ccoc2)c2ccccc2[nH]1)c1snc(CC)n1 48124,C1(CCOC)CN(C(c2cnn(C(C)C)c2C2CC2)=O)CCN1C(=O)C(C)C1CC1 48125,Cc1cn2c(n1)CCC(C(=O)NC1CCC1NC(c1ccccc1[N+](=O)[O-])=O)C2 48126,C(=O)(C(C)(C)CC(=O)OCC)N1CCC(CCNC(C(CC(=C)C)C)=O)C1 48127,C(=O)(CCS(N)(=O)=O)N1CC2C(CNC(C(C(C)C)OCC(C)C)=O)(C2)C1 48128,c1(C(N(CCCNC(=O)CCCC2CC2)C(C)C)=O)c(F)ccc2cnn(C)c12 48129,C(C(=O)NC1CC(NC(c2nc(C)[nH]c2C(F)(F)F)=O)C1)(C(C)(C)C)NC(C)=O 48130,Cc1csc2c(C(N3CC4CC(NC(C5(Cl)CC5)=O)CC3C4)=O)ncnc12 48131,C(=O)(C(C)CCC(C)(C)C)NC1CC(NC(Cc2ccc(C)c(Br)c2)=O)C1 48132,C1(C(=O)NCCOC2CN(C(c3cc(C)nn3C)=O)C2)CCc2nncn2C1 48133,c1(C(N2CCC(N(C(=O)CC(C)F)CC)CC2)=O)ccc(-n2cnnn2)c(C)c1 48134,C1(NC(=O)CONC(=O)C2(C3(C)CCC3)CCC2)CC12CCCCC2 48135,c1(OCCC(N2C(CNC(C3CC(CC)(CC)C3)=O)CC2)=O)cccc(Cl)c1Cl 48136,C1(N(C(C(C2CN(C=O)C2)OC)=O)C)CCCC(=O)C1.C(CCN=[N+]=[N-])N 48137,N1(CC(COCC)O)CCC(C(N2CC(C(=O)O)C2)=O)CC1 48138,C(=O)(C1=CC2C=CC(C1)C2)N1CC(N(C(=O)CSC(F)F)C)OCC1 48139,C(C1CCCCCC1)=CC(=O)NC1CCN(C(CC2CCCN(C)C2)=O)C1 48140,N1(C(C(C)NC(CC)(C)C)=O)CC(C)C(NC(C2C3CC4C(C3)C24)=O)C(C)C1 48141,Cc1ccc(C)c(C(=O)NCC23CCCC2CN(C(=O)C2=CCCC2)C3)c1O 48142,c1(CC(=O)NC(c2nccn2C)C=C)c(C)cc(C)cc1C 48143,c1(C(=O)NCC(C2CC2)NC(CC(C)(C)OC)=O)nccc(Br)c1C 48144,CC1(CNC(C2CCCC3(CC3)C2)=O)CN(C(c2cn3ccnc3s2)=O)CCO1 48145,C1(C(=O)NC2(C)CC(NC(c3cccs3)=O)C2)C2CCC3C(C2)CC13 48146,c1(NC(CC2(OC)CN(C(=O)CNC=O)C2)=O)cccc2c1CCCC2 48147,C12(C(=O)O)COC(CCN1C(=O)CCc1n[nH]c3cccnc13)C2 48148,c1(C(=O)NC2CC(C)(NC(C3C=C(C)CS3)=O)C2)cnn(C(C)C)c1C 48149,C(CCC(C)C)(C(=O)N(CC(C)O)CCN(C)C)NC(C(CCC)NC(C)=O)=O 48150,c1(NC(c2c(C)nns2)=O)cnc(F)cc1C(=O)Nc1cccc(CCO)c1 48151,C1(NC(C=CC=CCC)=O)CN(C(=O)C=CC2CCOCC2)CCC1C(F)(F)F 48152,Cc1ccc(F)cc1NC(=O)C(C1CCCN(C(c2cc(O)nn2C)=O)C1)C 48153,N1(C(c2cc(OCC)no2)=O)CCCC(NC(c2cc(OC)ncn2)=O)C1C 48154,C(=O)(CS(=O)(=O)CCC(F)(F)F)N1C(CNC(=O)CCc2ncc[nH]2)COCC1 48155,C1(NC(C(C)OCCCCCC)=O)CN(C(=O)C(F)OC)CCC1(C)C 48156,CCC(C)(COC)C(=O)NC1CC(O)CN(C(=O)CCCc2ccsc2)C1 48157,S(=O)(=O)(c1cccs1)NCC(=O)NC(C1CN(C(=O)Cn2cccnc2=O)C1)C 48158,C1(C(N2C(C=C)CCC2)=O)CCN(C(C2CC(=O)OC2(C)C)=O)C12CCC2 48159,c1(C(=O)NCCC2N(C(C3(OC(C)=O)CC3)=O)CCC2)cnc2onc(C)c2c1 48160,c1(OC)nccc(CN2CCN(C(=O)Nc3c(C)nn(C)c3C(N)=O)CC2)c1F 48161,C(=O)(C(C)CS(C)(=O)=O)N1CCC(O)(C(C)NC(C(=O)NCC)=O)C1 48162,c1(CCN(C(=O)Nc2c(CC)ccs2)C)ccc(F)c(C)c1 48163,N(C1CCCc2c[nH]nc21)C(C(CN(C)C)NC(c1cc(OC)cc(F)c1)=O)=O 48164,C1(CNC(C2CCCC(C)C2)=O)CC2(CC2)CN1C(C1CCCSS1)=O 48165,c1(C(N2C(CC)CN(C(C3CC(C)(C)O3)=O)CC2)=O)ccc(C)c(S(N)(=O)=O)c1 48166,N1(C(C)=O)CCCC(C(=O)NC(CNC2(c3ccon3)CC2)C2CCC2)C1 48167,CS(=O)(=O)c1nc(NNC(=O)C2CCOCC2)nc2ccccc12 48168,CC(C)(C)C(CO)C(=O)NCC(F)CNC(=O)CCc1cccc(C(F)(F)F)c1 48169,C(=O)(C(F)C(F)(F)F)NCC(C)=CC(=O)NCCCOc1cccc(F)c1 48170,c1(CN(C(=O)C(=O)NCCc2ccc(C(C)(C)C)cc2)C)sccc1S(C)(=O)=O 48171,C1(NC(c2nncs2)=O)CC(O)(C2CCN(C(c3ccccc3)=O)CC2)C1 48172,CCCC(CC)C(=O)N1CCN(c2cc(CNC(C3CC3OC)=O)ccn2)CC1 48173,c1(C(N2C(CNC(CC(C)n3cccn3)=O)COCC2)=O)ccn2c1CCCC2 48174,N1(Cc2scc(C)n2)CCC2(CC1)CN(C(C1(C)CCOC(C)C1)=O)CC(C)O2 48175,C1(C(N2CCCC(C)C2)=O)CCN(C(=O)CCCC2CCCC2)C12CCC2 48176,N1(C(CC(CC)O)=O)CCCC(C2CC2NC(c2cn(C)nc2C)=O)C1 48177,N1(C(C2CCCCC(=O)N2)=O)CCCC12CCN(C(C1CC1F)=O)CC2 48178,C1(C(N2C(CNC(C3CC4(CC4)C3)=O)CCC(C)C2)=O)CCc2nnc(O)n2C1 48179,C(CC(O)C(=O)NCCC1CCN(C(=O)CCOC2CCN(C)CC2)C1)SC 48180,C(=O)(C(O)C(C)(C)C)N1CCN(CCNC(C(C2CC2)OCC)=O)CC1 48181,c1(OC)cccc(C(N2CCCC2CCCNC(=O)COc2ccc(F)cc2)=O)n1 48182,C1(C(=O)NCC(C)(F)CNC(=O)CC2CC(F)C2)CCOC1(C)C 48183,CC(C)(C)CC(O)CC(=O)Nc1ccc(-c2noc3c2COCC3)cc1 48184,C1(C(N2CC(CC(=O)OCC)C2)=O)CN(C)CCN1C(=O)CCc1ccco1 48185,c1(C(N2CC(CN(C(C(CC)(F)F)=O)C)OCC2)=O)cc(C(N)=O)cc(C)c1 48186,C(=O)(CCC(C)(C)C#N)NC1CCN(C(CCOCCOCC)=O)CC1O 48187,C(=O)(C(CC1COCCO1)C(F)(F)F)N(C1CN(C(c2ccn(C)n2)=O)C1)C 48188,c1(OC)cc([N+](=O)[O-])ccc1NC(=O)NC1(C(C)Nc2ccc(OC)cc2)CC1 48189,N1(CC(=O)NC)CCOC(CNCc2cnoc2-c2ccoc2)C1 48190,C1(NC(CN(CCC)C)=O)CCN(C(c2cccc(N)c2C)=O)CC1O 48191,CN1CC=C(CC(=O)N2CCC3CCN(C(=O)CN4CCCNC4=O)C3C2)CC1 48192,c1(OC)nc(N2CCN(C(c3ncn(C)n3)=O)CC2)ncc1Br 48193,C1(CNC(c2ncc(C)cc2C)=O)CC2CCCC2N1C(c1cc(Cl)ns1)=O 48194,N1(C(C(C(C)C)SC)=O)CCC(C2CCN(C(=O)Cc3nccn3C)CC2)C1 48195,N1(C(CCN(C(=O)CC2CCCC23CC3)CC#C)=O)CCCCC(NC(=O)C2CC2)C1 48196,C(=O)(CC(O)CNC(c1conc1C)=O)N(C)Cc1cnc(C)s1 48197,C(CC(N)=O)(c1cn(CCCC(=O)O)nn1)NC1CC(CCSC)C1 48198,CC(CCCc1ccc(Cl)cc1)C(=O)c1ccccc1.C1(NC(=O)N)CCCC(C#N)C1 48199,C1(NC(=O)COCC2CC2)CCC2(CC1)CCN(C(=O)C(F)C(F)(F)F)C2 48200,NC1COCC1CNC(=O)CNC(c1ccc(Cl)s1)=O 48201,C(=O)(CC(C)(CC)C(=O)OC)NC1(CO)CCN(c2n(CC=C)nnn2)C1 48202,C1(NC(C=C(C)Cl)=O)CCCCC1Nc1nnc(C2CC2)o1 48203,c1(C(=O)NCCn2c(C)ccn2)ccnc(CNC(=O)CC2(C)CCOC2)c1 48204,C1(C(=O)NCC2(O)CN(C(c3cc(C)on3)=O)C2)Cc2cc(F)cc(F)c2O1 48205,C(CC(C)C)(CS(C)(=O)=O)NC(c1cn(CCC)nc1C)c1nnnn1C1CC1 48206,C1(N(C)CC2CCC23CCC3)CCCCN(C(=O)C(C)(C)C#N)C1 48207,Cc1ccc2c(N3CCCC(COC(C)C)C3)nc(=NC3COCC3C)[nH]c2c1 48208,C12(C(=O)NC(CC)CNC(=O)COc3cccc(Cl)c3)CCC(COC)(CC1)C2 48209,c1(C(=O)NC2(CC(=O)N(C)Cc3sccc3CO)CCC2)cc(=O)n(C)cn1 48210,c1(C(=O)OC)c(C(=O)NC2(CC(=O)N(CCCO)C(C)C)CCCC2)n[nH]c1C 48211,C1(OC)CCCCC1n1cccn1.C1(=O)C(N)CN1C 48212,N1(C(c2ccn(COC)n2)=O)CCCC12CCCN(C(=O)C(C)CC(C)(F)F)C2 48213,C12(C(N3CCC(CC(C)C)C3)=O)C(C(=O)OC(C)(C)C)C3CC1C2C3 48214,c1(C(=O)NCC2(O)CCCN(C(COC(CC)(C)C)=O)C2)ccc(C#N)c(O)c1 48215,C=CC(C)(C)C(=O)N(CC(C)NC(=O)C(=O)NCC(=O)N)C.N1(CC)CCCC(C)C1 48216,Cc1nc2ccccc2cc1C(N1CCC1C(=O)Nc1ccc(N)c(C)c1C)=O 48217,CN1CCCC(CCC(=O)NC(C)(C)CN(C)C(c2csnc2Cl)=O)C1 48218,c1(C(C)C)ccc(NC(C2(N(C)C(C3(CO)COC3)=O)CC2)=O)cc1O 48219,C1(F)(C(=O)NCC(CC)NC(c2ccc(-c3ccco3)s2)=O)CCC(C)CC1 48220,Cc1cc(C(=O)NCCCCCn2cc(C(C)(C)CCNC(N)=O)nn2)nn1C 48221,n1(CCOC)nc(C)c(Cl)c1C(C(=O)NCC(F)F)CCSC1CC1.N(C)C 48222,C1(C(=O)NC(COC)CCO)CCCCC1(C)NC(c1cnc[nH]c1=N)=O 48223,N1(C(=O)COc2ccc(C(F)(F)F)cc2)CC2(C1)CN(C(C1CCC3CC13)=O)C2 48224,C12(COC)CC(CN1CC1C(O)CCN1C(=O)OC(C)(C)C)C2 48225,C=C(C)C1OCCCC1C(=O)NC1CN(C(c2ccccc2CC#N)=O)CC1O 48226,N1(C(C2C(C)(C)NC(=O)C2)=O)CCC=C(C(=O)NC2CCCC2(F)F)C1 48227,Cc1ccc(F)c(O)c1C(N1CC(CNC(=O)CCc2ccon2)C(C)C1)=O 48228,C1(n2cc(CC(C)(C)O)nn2)CCCCCN1C(=O)CCC12CCC(CC1)C2 48229,c1(C(C(=O)NCCCOC)N(C2CN3CCC2CC3)C)ccc(F)c(Br)n1 48230,C1(CC(=O)N(CC(C(=O)NCC(C(=O)NC)O)C)C)NC(=O)NC1=O 48231,CC1=C(C(=O)NC2CCCCC2N(C)C(C2CCOC2(C)C)=O)CCS1(=O)=O 48232,C12(C(N3CC=C(CNC(C4CCOCC4)=O)CC3)=O)CCCN1CC(O)C2 48233,CCC(C)C(=O)C(=O)N1CCC(C)(C(=O)NCC2CCCC2)C1 48234,c1(C(=O)NC2C(C)(C)CN(C(C3(F)CCOCC3)=O)C2)c(F)ccc2occc12 48235,C(C(C)(CC(C)C)NC(=O)C(C)N(C)C)NC(C1(CC)CC1)=O 48236,Cc1c(C(=O)NC2CC2NC(c2ccc(CCC#N)o2)=O)cnn1CCC#N 48237,N1CCC(O)C(c2n(C)cc(-c3ccccc3)n2)(C(F)(F)F)C1 48238,c1(C(=O)NCCCCC(=O)N2CCC(NC(C)(C)C)C2)ccc(C#N)cc1 48239,C=C(C)C1CN(C(=O)C(F)C2CC(NC(=O)C=Cc3ccncn3)C2)CCO1 48240,C12(NC(=O)COC3CC3)CCC(C(=O)NCC(F)Cl)(CC1)C2 48241,N1(C(C2CSC2)=O)CCC12CN(C(C13CC(O)C1C3)=O)C2 48242,N1(C(c2ccc(-n3cccn3)cn2)=O)CCCCC(NC(C2C=CCS2)=O)C1 48243,N1(C(CC2N(C(CC3C(C)CCC3)=O)CC2)=O)CCCCC12CC2 48244,C1(C(=O)NC2CCC(N(C)C)C2)CCC2(CC2)N1C(=O)CCc1nc(CO)n[nH]1 48245,N1(C(c2cc(C)cc(C)c2)=O)CCC2(CC1)CC2NC(C12CCN(CC1)C2)=O 48246,c1(N2CCC(C(=O)NCC)CC2)nccc(NCC(N2CCCC2)C)n1 48247,c1(OCC)cccc(NC(=O)C(N2CCCCC2CNC(C2(C)CCO2)=O)=O)c1 48248,c1(C(=O)NCCN(C(=O)C(C)(C)CF)CC(C)O)c[nH]c2cc(F)ccc12 48249,CN(CCCC(=O)N1CC=CC(NC(=O)C=CCOCc2ccccc2)C1)N=O 48250,N1(C(C2(C)CC(=C)C2)=O)CCC2OCCN(C(c3ccc(C(C)F)cc3)=O)C2C1 48251,N1(C(C(C)n2ccnn2)=O)CCCC2(CCC2NC(c2ccn(C)n2)=O)C1 48252,n1(CC(=O)NCC2(CNC(C3C(C(C)C)(CC)C3)=O)CCC2)c(C)csc1=O 48253,c1(C(N2CCC(CNC(CC3C(C)(C)CCCC3)=O)C2)=O)cncc([N+](=O)[O-])c1 48254,C1(NC(c2cc(SC)oc2)=O)CC(NC(=O)C2=CCCOC2)C12CCOCC2 48255,N1(C(c2c(C)occ2)=O)CC2C(NC(C3(c4ccc(F)cn4)CC3)=O)C2C1 48256,C1(NC(CC(C)OC)=O)CCN(C(=O)C(C)Sc2ccccc2)C12CC2 48257,C1(C(C)(C)C)(NC(c2n(CC)nnn2)c2cncn2C)CCOCC1 48258,C(=O)(C(Cc1ccoc1)NC(=O)C(F)=CCCF)NCC(C)OC 48259,c1(CC)nnc(N2CC(O)(C(C)NC(C3(C)CC3)=O)C2)c(C#N)c1CC 48260,C1(CNC(C(C2CCC(=O)N2)C)=O)CC2CCC(C1)N2C(=O)CS(=O)(=O)N(C)C 48261,CC1(CNC(=O)Cn2ccc(=N)[nH]2)CN(C(C2CCCCO2)=O)CCO1 48262,C1(CNC(CCc2cccc(OC)c2)=O)CN(C(=O)C(O)C2CCC2)CCCO1 48263,c1(C(N2C(C)CC(CNC(CCCCC)=O)C2)=O)ccc2oncc2c1 48264,c1(C(=O)NCC(C2CCC2)NC(C2(COC)CCCCO2)=O)cc(C)ccc1C 48265,N1(C(c2nnn(CC)c2C)=O)CCC(NC(C2CC2F)=O)CC(O)C1 48266,C1(NC(c2ccn(CC(C)C)n2)=O)CN(C(c2[nH]cnc2C)=O)CC1C 48267,N1(C(CCC2(NC(C3(C)CCC(=O)N3)=O)CCC2)=O)CC2CCC2(C)C1 48268,C1(C(=O)NC2C(C)N(C(C3COC(C)(C)CO3)=O)CCC2)CCC(C2CC2)CC1 48269,S(=O)(=O)(c1ccc(N2CCC(CO)CC2)c(C#N)c1)N1CCC(C)C(CO)C1 48270,CC1CSCCN(C(=O)CC2CCN(C(c3ccn(C)c3CC(=O)O)=O)CC2)C1 48271,C1(NC(Cn2cc(CNC(C3CC(C)OC3)=O)nn2)=O)CC(C)(C)C12CCC2 48272,C1(C(N2CC(CNC(Cc3cn(C)nc3)=O)OCC2)=O)CC2C=CC1C21CC1 48273,c1(OC)cc(C(=O)NC2CN(C(c3ccoc3Cl)=O)CC2F)cc2nc(O)[nH]c12 48274,c1(CC(=O)NCC2(NC(C(=Cc3cn[nH]c3)C)=O)CCCC2)ccncc1C 48275,c1(NC(C2NCCN(C(c3nc(CC)oc3)=O)C2)=O)cc(C)cc(Br)c1F 48276,Nc1ccc(C(=O)NC2CCN(C(c3ncc(F)cc3F)=O)CC2CO)nc1Cl 48277,C=Cc1ccc(C(=O)NC(Cn2cncn2)C(=O)N(CC(C)(CC)OC)C)cc1 48278,N1(C(Cc2cccc(COC)c2)=O)CCN(C(=O)CCCCSC)C2COCC12 48279,N1(C(=O)OC(C)(C)C)CCC(C(=O)O)C(O)C1.C1(C(C)C)CC(CCN)CNC1 48280,CC1CN(C(=O)Cc2cccc(CO)c2)CCCN1C(c1ncn2c1CCC2)=O 48281,N1(C(C2OCCN(CC)C2)=O)CCN(C(c2scc(C)c2C)=O)CCC1C 48282,C(=O)(C1=C(Cl)CCCC1)NCC1N(C(C2(N(C)C)CCCCC2)=O)CCC1 48283,CC1(C)COCCC1CC(=O)NC1(CNC(c2csc(Cl)n2)=O)CCCCC1 48284,N1(C(=O)OC)CCC=C(CNC2NC(=O)NC2=O)C1.c12ccc(cc1)C(=O)NC2 48285,c1(OC)cccc(C(N2CCC2CNC(C2(F)CCC2)=O)=O)n1 48286,c1(C(=O)NCc2nc(CNC(CCc3nc(=N)[nH][nH]3)=O)sc2)cccnc1S 48287,N1(C(C2C(C)(C)CCN(C(C(CCC)(C)C)=O)C2)=O)CCC2(CCCCO2)C1 48288,Cn1nnc2c(CN3CC(n4cc(C(=O)NC5CCC(F)CC5)nn4)C3)ccnc12 48289,c1(C(C(N2CC(COC)C(O)C2)=O)NC(CCSCC)=O)c(C)cccc1Br 48290,N1(C(C(OC)OC)=O)CCC(F)(CNC(=O)C(=O)NCC(C)(C)CN(C)C)CC1 48291,Cn1nc(Br)cc1CC(=O)NCCCC1CCCN1C(c1ccon1)=O 48292,C(N=c1[nH]c2ncc(Cl)cc2o1)C1N(C(C2(c3ccc(Cl)cc3)CC2)=O)CCCC1 48293,c1(C(=O)NCCC(C)NC(C2C3CCCCCC23)=O)c(F)ccc(F)c1Cl 48294,C1(OC(c2ccsc2C(=O)Nc2ccco2)=O)CCS(=O)(=O)C1 48295,C1(C)(NC(CCC2(NC(CC(C)(C)OC)=O)CCC2)=O)CCC(F)(F)CC1 48296,c1(C(=O)NC2CC(CNC(CCSCCC)=O)C2)cc(C)nc2c1nc(C)n2C 48297,c1(C(=O)NC2CC(NC(C(Cn3ccc(C)n3)C)=O)C2)nccc(F)c1Cl 48298,C1(C(=O)NCC(C)N(C(CSCCC)=O)C)(C(C(=O)C(C)SC)C)CCOCC1.O 48299,C1(NC(CCC=C)=O)CCN(C(c2cccc(CC(F)(F)F)c2)=O)C1C1CC1 48300,Cc1cc(C(N2CC(CNC(c3cc4occc4s3)=O)C2)=O)cc(N)c1O 48301,C1(COC)(NC(=O)C(C2(O)CCCC2)F)CCN(C(c2cc[nH]c(=N)c2)=O)CC1 48302,C1(NC(CCSCC(C)C)=O)CCC2CCN(C(c3c[nH]ccc3=O)=O)C12 48303,c1(C(c2nnnn2C2COC2)NCC(C2CCSCC2)(C)C)cccc(CF)c1 48304,N12CC3CCC1CN3CC1(CC(=C)C1)C2=O.C1(C(=O)OC)CCCO1 48305,CC1(C#CC(=O)N2CCCC2(C)CNC(=O)C(C)(C)C2CC2)COC1 48306,C12(C(N3CC4C(CNC(C5N(CCC)C(=O)CC5)=O)C4C3)=O)CCCC1OCC2 48307,C1(CC(N)=O)CCCN(C(=O)CNC(C2CCNCC2)=O)C1 48308,N1(C(C2C(CCC)C2)=O)CC(CNC(c2cccs2)=O)CC12CCOCC2 48309,c1(C(=O)NCCN(C(c2c(CC)cno2)=O)CC)sc2cc(F)ccc2c1Cl 48310,c1(CC(=O)NC(C)C(CO)NC(=O)Cn2nnc(=O)[nH]2)coc2ccc(F)cc12 48311,c1(C(=O)NCCC2(O)CCCN(C(c3ccns3)=O)C2)ccc2c(c1)CCCO2 48312,N1(C(C2CC2c2cccnc2-n2cccn2)C)CC(N(C(C)(C)C)C)C(F)C1 48313,CCCCCC(C)(C)C(=O)NC1CN(C(c2c[nH]c3cccnc23)=O)CC1SC 48314,CC1CN(CC(=O)N(C)CC2CNC2)CCS1(=O)=O 48315,c1(N(C(C2CCCO2)=O)CC)ccccc1Cc1ccncc1.C12(C)CN(C1)C2 48316,C(=O)CCCCCCS(N)(=O)=O.C(=O)(C1=COCCC1)N(C1CC1C(=O)NCC=CC)C 48317,N1(C(C2C(C)(C)CCC2)=O)CCc2nc(CNC(c3ccccc3F)=O)sc2C1 48318,C(c1ccc(C)c(C)c1)=CC(=O)NC1C2(CC(NC(C(CC3CC3)OC)=O)C2)C1 48319,Cc1cc(CC(=O)NC2CC2CNC(c2cn[nH]c2)=O)sn1 48320,Cc1ccc(C(N2CCN(C(=O)C(C#N)CC3CC3)C(C(C)C)C2)=O)nc1O 48321,Cn1ncc2c1CCC(C(=O)NC(CNC(c1ncc(C(F)F)s1)=O)CO)C2 48322,C1(NC(C2(CNC(=O)OC(C)(C)C)CCCCC2)=O)CCN(C(N)=O)CC1(C)C 48323,c1(N2CCN(CC)CC2)nc2cccnc2c(=NCC2CCCC(F)(F)CC2)[nH]1 48324,c1(C(=O)Nc2cccc(NC(CC3C(CC)C3)=O)c2)c(Br)c(C)nn1C 48325,C1(CC#C)(C(=O)NC(C)CCNC(c2cnc(COC)nc2)=O)CCCCC1 48326,C1(F)(C(N2CCC(NC(Cc3c(C)con3)=O)CC2)=O)CS(=O)(=O)CC12CCC2 48327,c1(C(N2CCC3C(NC(C4CCOC4)=O)C3C2)=O)cnc2nccn2c1 48328,Cc1cc(F)c(N)cc1C(=O)NC1CN(C(c2ccccc2S(C)=O)=O)C1 48329,C1(NC(C(C)(C)OC)=O)CN(C(c2ncnc(C)c2C)=O)CCC1F 48330,c1(OC)ccc2c(c1)N(c1ncc(C3CCCCC3)n1C)C(C)(C)C(=O)N2 48331,c1(C(N(C2CCCC2)CCNC(c2nnc(C)s2)=O)=O)cnc2c(c1)CCC2 48332,c1(COCC)ccc(CCNC(=O)C(=O)N(C(C)C(C)(C)C)C)cc1 48333,N1(CC(=O)N(C(C)CNC(=O)C(C)OCC(C)C)C)CCCC1CO 48334,CCCCCCC(=O)N(CCNC(c1sccc1C1CC1)=O)CC 48335,Cc1cc(C(N2CCCC(NC(C3C=CCC3)=O)C2C)=O)c(O)c(C)n1 48336,c1(OC)cccc(C)c1C(N1CC2C(NC(=O)C(N3CCN(C)CC3)C)C2C1)=O 48337,N1(C(C(c2cnn(C)c2)OC)=O)CCCC2(CCC(NC(=O)C(F)(F)C(F)F)C2)C1 48338,C1(NC(C(CC)SC)=O)CCN(C(=O)C(c2cncn2C)=O)C12CCC2 48339,n1(CC(=O)N(CCC)C)ccccc1=O.C12CC(C1)NC(=O)CC2 48340,C(=O)(C1=C(F)CN(C(C2CC(C#N)C2)=O)CC1)NCC1(N2CCCC2)CC1 48341,C1(NC(c2cc(C(C)C)on2)=O)(CO)CCCCC1.c12cc(no1)C(=O)NC2C 48342,c1(C(N(CCN(C(c2cc(C)[nH]n2)=O)C)C(C)C)=O)ccnc(C(C)C)n1 48343,c1(CC(c2cn(C)nn2)NC(C(CCC)C)=O)ccc(Cl)cc1Br 48344,c1(C(=O)NC2CC(CNC(CCn3ncc(C)c3)=O)C2)ccc2cccnc2c1 48345,CC1CN(C(c2nnn(C)c2C(F)F)=O)CCC1N(C)C(c1cc(Cl)n(C)n1)=O 48346,C#CC1(O)CCN(C(C2CCCC(NC(=O)CNC(=O)NC)C2)=O)C1 48347,C1(CCC=C)CCCN(C(C23CC2CCN3C(=O)C(=O)NOC)=O)C1 48348,CC1CN(C(c2cncn(C)c2=O)=O)CCC1N(C)C(c1ccc(CO)cn1)=O 48349,CC(C(C)NC(=O)CSCCC#N)NC(=O)CCOCC1CCCO1 48350,C=CCC(CC)C(=O)N1CC2(CC(CC(N3CCC(c4ccon4)C3)=O)C2)C1 48351,c1(C(=O)NC2C(C)CN(C(C3CC(C)(F)C3)=O)C2)ncnc2c1c(Br)cn2C 48352,C12(C(=O)OC)CCCC1(NCCCC(C)CO)CN(C(=O)OC(C)(C)C)C2 48353,c1(C(C(=O)N(CCNC(C(CC#C)O)=O)CCOCCO)C)cccc([N+](=O)[O-])c1 48354,CC1CCCC(CC(=O)NCC2CN(C(=O)C(C)CN(C)C)C2)C1 48355,c1(C(=O)NCCNC(CCCN(S(C)(=O)=O)C)=O)ccc(NC23CCC2C3)cc1 48356,c1(C(=O)OC(C)=O)cn(C)[nH]c1=NC(=O)COC(C1CCOCC1)c1ccco1 48357,c1(C(N2CC(N(C(COCCC=C)=O)CC)C(C)C2)=O)c(C(F)F)nn(C)c1C 48358,N1(C(CC(COC)C)=O)CC(CNC(c2c(F)ccc(C)c2F)=O)C2(CCC2)C1 48359,c1(CC)cnc(-c2cn(CC3CCCN3C(=O)CC3CSCCS3)nn2)nc1 48360,C(=O)(C1=CCN(C(C2CCNC(=O)C2)=O)CC1)NC(CSC)C 48361,C(CCCCC(=O)NCC1C(C)CCN1C(=O)CC1(C)CC1(Cl)Cl)OCC 48362,C(=O)(C(CC(F)F)N(C(=O)CN(C)C(=O)OCC)C)NC(CCC)(C)CC 48363,C1(C(=O)C2CC2)(CC)CC(F)(F)C1.c12nc(C)c(s1)CNC(=O)NC2C 48364,CCC(CCOC)C(=O)N1CC(C(=O)NCC(C)(C)SC)C2(CC2)C1 48365,N1(c2cc(CC)ncn2)CC2(C1)SCCC2NC(=O)CSc1cnn(C)c1 48366,c1(C)ccc(CCOC)c(CC2CC2)c1.C12(CCC1)NC(=O)N2 48367,C1(C)(CC)C=C(C(=O)N(CC(N2CC(CC)C2)=O)C2CCC2)C1 48368,N1(C(C(COC)OC)=O)CC2CCC(N(C(=O)CCS(C)(=O)=O)C)C2C1 48369,c1(-c2ccc(C)cc2OC(F)F)cccc2c1CCN(c1cccc(Cl)c1C#N)C2 48370,Cc1cc(=NC2CCN3CCCC23)[nH]c(=NCC23CC(CCO2)C3)[nH]1 48371,C1(C(=O)NCC(C(C)C)CO)C2CC3C(C2NC(c2ccccn2)=O)C13 48372,c1(C(=O)NC2CN(C(c3cc(C)ns3)=O)CC(F)(F)C2)cnc2ncnn2c1C 48373,c1(CC(=O)NC2C(C)CN(C(=O)CCCCN(C)C)C2)ncn2c1CCC2 48374,CCC(CC(=O)NCC1(N(C)C)CCCC1)N(C)C(C1CC(OC)C1)=O 48375,C1(NC(c2c(CC)cccn2)=O)CC(OC)CN(C(=O)CCS(C)=O)C1 48376,O=C(CCCC(F)F)NCC1CCN1C(c1ccc(CO)nc1)=O 48377,C1(=CCC)CCN(C(=O)CN(C2CCCO2)C2CCCC2)C1 48378,C1(C(=O)NCCCCC2CN(C(=O)C(F)CC3CCC3)C2)CC(F)(F)C1 48379,N1(C(c2nnnn2Cc2cn[nH]c2)C2CC2)CCN(Cc2ccccc2)CC1 48380,C1(NC(c2cnc(C)[nH]2)=O)CCCCC12CCN(C(c1cccc(=O)n1C)=O)C2 48381,c1(SCC)ccnc2nc(=NCCNC(CNC(=O)OC(C)(C)C)C3CC3)[nH]n12 48382,N12CCC3(CC1)CC(C)N2C3.c1(OC)ccccc1C(=O)C=O 48383,C(=O)(C(C)CC(C)CC(C)C)NC1CN(C(C(C(CC)(C)C)O)=O)CC(C)C1 48384,CCC(CC(=O)NC1CC(C(=O)NCc2cc[nH]n2)C(O)C1)C(C)C 48385,CC(C(=O)OC(C)(C)C)C(=O)N1CC=CC1CNC(=O)C=Cc1nccs1 48386,C1(C(=O)NC2(CC)CN(C(=O)C(C)C)C2)C2CC2C2CC12 48387,Cc1noc(C)c1CC(C)C(=O)NCC1CCN(C(=O)CCc2cccnc2)C1 48388,C(C1=CCN(C(=O)COc2cccc(OC)c2)CC1)NC(C(C(C)C)OCC)=O 48389,c1(-c2cn(C3CCN(C(c4nnn(CC)c4C)=O)C3)nn2)cc(F)cc(C#N)c1 48390,C(C)(C(=O)N(CCC(=O)NCC(C)Cc1cn[nH]c1)C)OCCOC 48391,C=CCC(CNC(c1cc(Cl)no1)=O)C(=O)NCc1cc(C)cc(O)c1 48392,c1(CN2CCCC(NC(CCC(C)C)=O)CC2)cc(Cl)c(O)cc1F 48393,Cc1cc(F)ccc1CC(=O)NCC(C)CN(C(=O)Cc1cccc(F)c1)C 48394,c1(C(=O)NCCC(C)NC(C2(NC(C)=O)CCOCC2)=O)cc(F)c(Cl)cc1F 48395,Cc1cc(=NC2C(C)CN(C(=O)CC3CC=CCN3C)CC2C)[nH]c(C(C)C)n1 48396,Cc1ccnc2c(C(N3CCC(CNC(=O)C(C)N4CCC4)C(C)C3)=O)cnn12 48397,C1(CC(=O)NC2CCC(N(C)C(c3nc[nH]c3C(C)(C)C)=O)C2)CC2CCC1CC2 48398,Cc1ccc(-c2ccc(NC(C3CC(=O)CCO3)=O)c(C)c2)cc1Br 48399,C1(NC(c2ccc(C#C)nc2)=O)CN(C(C2(C)CCC2)=O)CC12CCC2 48400,N1(C(=O)NCc2ccc(OCC)nc2)CCC(O)C2(CCC2)C1 48401,Cc1ccc(C)n1CC(N1CCC=CC1C(N1CCC(F)(CF)C1)=O)=O 48402,c1(C(=O)NC)cn(CCSC)nn1.c12ccc([nH]1)CNC(=O)C(C)NC2=O 48403,N1(C(c2sncc2Br)C(=O)NCC(=O)NCCCCCC)CCCC(C(N)=O)C1 48404,CC1CCC=C1C(=O)N1CCC(CF)(NC(c2cn(C)nc2C(F)F)=O)C1 48405,N1(C(CC=CC)=O)CCC(C2CCCN(C(=O)CS(=O)(=O)CC)C2)C1 48406,CC(C)CCCCCC(=O)NC1CCN(C(c2cnn(C3CC3)c2)=O)C1 48407,c1(CC)csc(CNC(C2(NC(=O)Cc3csc(C)c3)CSC2)=O)n1 48408,CCC(CC)(C(=O)NCC1(C)CCN(C(c2ccc(CO)c(Cl)c2)=O)C1)OC 48409,N1(C(c2cn(CC)nc2C)=O)CCN(C(c2ccc(N)c(C)c2F)=O)C(C)C1C 48410,CC#CCC(C(=O)N(CC(O)COC)C)NC(=O)Cc1cccs1 48411,C(C(O)C(=O)NC(C)(C)C=CC(=O)NC(c1ncc(C)o1)C)OC 48412,c1(OC)cnc(Cl)cc1C(N1CCC(N(C(=O)C(C)(Cl)Cl)C)C(C)C1)=O 48413,C1(C(C)(C)C)(CNC(C(C)OCC)=O)CCN(C(C2CCC(N(C)C)CC2)=O)C1 48414,C(=O)(C1=NOC2(CCC2)C1)N1CC(C)N(C(=O)CCP(C)(C)=O)CCC1 48415,c1(C(=O)NC(C(C)NC(C2CC(O)CN2C)=O)(C)C)n[nH]c2c1COCC2 48416,C1(CCC)CN(C(c2cc(OC)nn2C)=O)CCN1C(c1ccccn1)=O 48417,C(=O)(C1=CCCC1C)NCC1C(CNC(c2c(C)cncn2)=O)C1(F)F 48418,C(=O)(CCC(=O)NN(C)C)NC(CC#CC)C(=O)NCc1oc(C)nc1C 48419,N1(C(CC(C(C)C)C)=O)CCCCCC(NC(C2(n3cccn3)CCOCC2)=O)C1 48420,CC1(C)CC(CN2CC3(CCC3)C2C2CC2)CCO1 48421,Cc1ccc(C(N2CCCC(NC=O)C2CO)=O)c(Cl)c1.C1(CO)CCN1C(C)(C)C 48422,C(CCCN=[N+]=[N-])NC(C(Cc1cc[nH]n1)NC(C(C)c1cccs1)=O)=O 48423,N1(C=O)CC(F)(c2c(-c3sc(C)c(Br)c3)nn[nH]2)C2(COC2)C1 48424,C1(NC(C2N(C(CC=C=C)=O)CC(O)C2)=O)CNC(=O)C12CC2 48425,CCC(CC(=O)NCCCCNC(c1cccc(O)n1)=O)C(F)F 48426,c1(C(N2CCCN(CC(N)=O)CC2)=O)cccc2c3c([nH]c12)CCCCC3 48427,N1(C(c2cnc(Cl)s2)C(=O)NCC)CC(=O)NCC1C 48428,S(=O)(=O)(c1ccc(Cl)nc1)N1C(C(N2CC(C(=O)OCC)C2)=O)COCC1 48429,Cc1n[nH]cc1CC(=O)NCCC(=O)N1CC(OCCN(C2(F)CCC2)C)C1 48430,n1(CC)ncc(C(N2CC(NC(=O)C(C)c3ccsc3)C2)=O)c1C(F)(F)F 48431,CC1=C(C)CC(C)(C(=O)NC2CCC2NC(c2ncsc2C(F)(F)F)=O)CC1 48432,C=CCCCCC(=O)NC1CCC(CNC(=O)Cn2cc(C#N)cn2)CC1 48433,CCCC1=CCCCC1.C(=O)(C(O)CCn1cncn1)NCCSC 48434,N1(C(c2cc(C)no2)=O)CCC(C)C(CNC(=O)CCCOC(C)(C)C)C1 48435,C1(C(N2CC(C3CN(C(CNC(C)=O)=O)C3)C2)=O)Cc2cccc(Cl)c2C(=O)O1 48436,C(=O)(CCCCC(N)=O)N1CCC(NC(C(C)(C2CC2)NC(C)=O)=O)C1 48437,Cc1ccc(NC(c2sccc2CNC(=O)CC2(C)OCCO2)=O)cn1 48438,Cc1cccc(C)c1OCC(=O)NC1CCN(C(=O)CC2CCC2)C1C(C)(C)C 48439,C1(CC(=O)NCCCCCN(C(c2c(CC)scc2)=O)C)SC2=NCCN2C1=O 48440,c1(C(N2C3(CN(C(c4c(C)nns4)=O)C3)CC2)=O)n[nH]c2ccccc12 48441,c1(Sc2nnc(N3CCC(OCC)C3)s2)ccc(Cl)cc1 48442,C(CCCC(=O)NCC1(C#N)CC1)NC(CCc1n(C)ccn1)=O 48443,c1(C(N2CC(CNC(C3CC3(F)F)=O)C(F)(F)C2)=O)ccc2cnoc2c1 48444,C1(NC(=O)C2=NOCC2)CC2(CCN(C(C3CCCCC34CC4(F)F)=O)CC2)C1 48445,CC1COCCC1N(C(=O)C(C1(O)CCC1)NC(=O)CC1CCC(=O)C1)C 48446,N1(C(COC(CNCC(C)OC)(C)C)=O)CCCCC(C2CN(C(=O)C3CC3)C2)C1 48447,N1(C(C2(CC)CC2)=O)CCC(C2CCN(C(=O)C(c3ccc(Cl)s3)C)CC2)C1 48448,c1(NC(C(COC(C)C)NC(C(CC)OC)=O)=O)ccc(OC(C)C)c(C)c1 48449,c1(OC)cnc(C(N2CC3C(NC(=O)Cc4c(C)noc4C)C3C2)=O)nc1 48450,N1(C(CC(C)(F)F)=O)CC2COCCC2(NC(c2ccnc3[nH]cnc23)=O)C1 48451,c1(N2C(=O)CCC3(C)CN(C3)C(=O)O2)ccc(Cl)cc1.CCC(CSC)OC 48452,C1(NC(CC(COC)(C)O)=O)C2CC(O)C1N(C(=O)CCCc1cccs1)C2 48453,N1(C(CC2N(C(COC)=O)CCNC2)=O)CCN(C)C(=O)CC1 48454,n1(CCC(=O)OC2C(SC)CCC2)ncn(C)c1=O 48455,N1(C(C=C(C)C(C)(C)C)=O)CCC(C2CC2)(CNC(=O)C#CC(C)(C)C)C1 48456,C(=O)(C(C)=C(C)C1CC1)NC(CNC(C=CCC)=O)C 48457,n1(C(CC)C)nnnc1C(c1coc(Br)n1)NCC1(COC)COC1 48458,C1(C2CCC2)(C(=O)NCCCC2(NC(=O)CC3CCCC(=O)N3)CC2)CC1(F)F 48459,n1(CCCC)nc(C)c(C=CC(=O)NCC(C)NC(=O)C(C)C(C)C)c1Cl 48460,C1(C)(NC(c2n(C(C)C)ccn2)c2nnnn2C2CCCC2)CCC(=O)N(C)C1 48461,Cc1cnoc1C(=O)NCC1(CNC(=O)CCc2nc[nH]n2)CCC1 48462,N1(C(C2CCN(CC(C)C)CC2)=O)CCC(NC(=O)CCC(C)(C)C)C(C)(C)C1 48463,C1(C(N2C(C)CCC2)=O)CC(O)CCN1C(=O)CCc1cc(O)cc(F)c1 48464,N1(c2ncc(CCC)cn2)C2CCC1C(C(=O)N(C)C)C2.C(=O)(NCC1CC1)N 48465,C(CC(C(=O)NOCCC(C)O)NC(=O)C1=C(Cl)CCC1)OCC 48466,N1(C(CCC=CC)=O)CCC(NC(=O)CSCC(F)F)CC(O)C1 48467,Cc1cc(C(=O)N(CC(O)CNC(c2cc(Cl)nn2C)=O)C)c2[nH]cnc2c1 48468,c1(OC)cccc2c(C(=O)NC(C)CCNC(=O)CCc3cncn3C)csc12 48469,S(=O)(=O)(c1ccc2c(c1)CCCC2)N1CC2(OCCN(C(C3CC3F)=O)C2)C1 48470,c1(NC(C2CCC3(CN(C(C(C)n4cccn4)=O)C3)O2)=O)cccc2cnccc12 48471,c1(C(=O)NCC(C)NC(=O)C(O)CC2CCOCC2)cc(Cl)ccc1C(F)(F)F 48472,C1(C(N2C(C=O)CCC(C)C2)=O)CC2CCC(C1)C2O.C(C)CCC 48473,CN1CC(NC(C2C3CC3CN2C(c2nn(C)cc2Cl)=O)=O)CC1=O 48474,C1(CNC(CCCCC=C)=O)CCN(C(C2(OC)CCOC2)=O)CCC1(F)F 48475,C(=O)(CCCC(=O)N1CC(C(=O)OC)CC1C(=O)Nc1cnc(F)cc1C)OCC 48476,C1(OC)CCCC(CC(=O)NC(C2CCCN2C(=O)CCc2cncn2C)C)C1 48477,N1(C(c2cc(C)oc2C)=O)CC2CCCC2(NC(=O)CSCC2CCCO2)C1 48478,c1(C(=O)NCc2scc(CNC(C(CC)F)=O)n2)c(C)[nH]c(C2CC2)nc1=O 48479,c1(OC)cc(CNC(C23CC(CCO2)C3)C)cc(OC)c1Br 48480,C(CC(C(=O)N1CCC(N(C(C2CCN(S(C)(=O)=O)C2)=O)C(C)=O)C1)NC=O)SC 48481,c1(C(=O)NC2CN(C(c3cccc(CC)n3)=O)CC2F)cc2nccc-2oc1Cl 48482,C1(NC(CCN(CCC)C)=O)CCCC(NC(c2cn(CC(N)=O)nn2)=O)C1 48483,C1(C)(CNC(C(CCC)=CCC)=O)CCN(C(C23CCCCC2CCC3)=O)CC1 48484,CC1CC(NC(=O)CC2CC(=O)NC(=O)C2)CN(C(C2C(C)C2C)=O)C1 48485,N1(C(COC(C)(C)C)=O)CCC(OCCNC(C2C=CCCC2)=O)C1 48486,c1(OCC)ncc(C(N2CC(NC(=O)CCCC3CC3)CC(C)C2)=O)cc1Cl 48487,N1(C(=O)CSC(F)F)CCCN(C(c2ncoc2-c2ccon2)=O)CC1CO 48488,C1(C#N)(CC(=O)N(C(C)CCCNC(=O)C(C)n2cccn2)C)CN(C(=O)OC)C1 48489,C1(CN(C2(COC)CC(c3ncc[nH]3)C2)C)CCOC(C)C1 48490,CCC(C(=O)N1CCCC1CN(C(=O)Cc1scnc1C)C)c1ccccc1 48491,Cn1ncc(C#N)c1C(=O)NC1CN(C(=O)CC2CCCC(F)(F)C2)CC1CO 48492,C(CCC)(C(=O)NC1COCC1CNC(C1CSCCS1)=O)=CCC 48493,N1(C(c2n(CC)ccc2)=O)CCCC12CCN(C(=O)CC1CC3CCC1O3)C2 48494,C1(C)(CNC(C(C2CC2)NC(CCc2cn(C)nc2)=O)=O)CCCCO1 48495,c1(C(c2cn(C(C)C(N3CC4(CCC(=O)N4)C3)=O)nn2)=O)cc2ncccn2n1 48496,CC(CN(C)C)CC(=O)N1CCC(F)(CNC(c2ccncc2C2CC2)=O)C1 48497,Cc1cc(Br)ccc1COC(c1cc(C2CCOCC2)on1)=O.C1CO1 48498,C1(C(=O)NC2(C(N(C)C)=O)CCCCC2)CC2CCC1N2C(=O)COC(C)(C)C 48499,CCC(CCCC(=O)N(C)CC1CCCC1)NC(=O)C(C)SC1CC1 48500,c1(CC(=O)NC)cc(C)c(C(=O)NCCCCCNC(=O)C2=CCCC2)o1 48501,N1(C(c2cc(C)ncc2)=O)CCC2(NC(c3cc(C4CC4)cc(F)c3)=O)CC2C1 48502,C(=O)(C(C)(C=C)CC)NC(CC=C)CNC(c1cccc(OCCF)c1)=O 48503,C1(O)(CNC(C2(CS(C)(=O)=O)CC2)=O)CCCN(C(c2nnc(O)nc2O)=O)C1 48504,C1(CC(=O)NC2(c3ccnc(Cl)c3)CC2)CCN(C(=O)CC2NC(=O)NC2=O)CC1 48505,c1(CN(c2cc(Cl)c(Br)cc2O)C)cc2ccccc2nc1O 48506,n1(C(C)C)cccc(C(=O)NCc2cn(CCNC(C3CC(F)C3)=O)nn2)c1=O 48507,c1(CC)ccc(Cl)c(NC(=O)CC(C)(C)F)c1.N12CCC(CC1)C2=O 48508,CCC(C)C(O)C(C)C(=O)N1CCCC(C(=O)NCC2CCC(C)(C)CC2)CC1 48509,N1(C(c2c(OC)n[nH]c2)=O)CCC(CO)(CNC(c2c(Cl)cnn2C(C)C)=O)C1 48510,C1(CC(=O)N(CCN(C(=O)CC(C)(C)F)C)C)CCCCC1(C)C 48511,C1(NC(CCCCC=C)=O)C2CC3CN(C(=O)Cc4ccoc4)C1C3C2 48512,N1(C(c2c(OC)nc(C)cc2)=O)CCCCCC(NC(c2onc(C)c2C)=O)C1 48513,N1(C(C(=C)F)=O)CC(C(=O)Nc2ccn(CC)n2)CC(F)(F)C1 48514,C(=O)(C1CC(=O)c2ccccc21)NCC(C)NC(c1c(C)cc(C)[nH]1)=O 48515,N1(C(CC=CC)=O)C2CCCC1CC(NC(=O)Cc1c(C)[nH]c3ccccc13)C2 48516,c1(C(N2CCC(NCCCC(=O)NC(=O)OCC)C2)=O)c(C)cccc1[N+](=O)[O-] 48517,CCCC(C(=O)OC)C(=O)N(C(C)CNC(c1cccn2cnnc12)=O)C 48518,N1(C(CC2CC(=C)C2)=O)CCC2(C1)CN(C(=O)C(C)C1CCOC1)CCO2 48519,c1(C(=O)NC2C(NC(Cc3cn(C)nc3)=O)CCC2)ccc2cnnc(O)c2c1 48520,C(=O)(CCC(C)(C)C(=O)NCC(CO)NC(C1CCCc2ccnn2C1)=O)OC 48521,N1(C(c2cc(C)oc2)=O)CC2(C1)CN(C(=O)C(C)OCCN(C)C)CCO2 48522,C1(C(=O)NC2CC(CCNC(C(CC)(C)C#N)=O)C2)COc2cc(F)ccc2O1 48523,c1(NC(C2C(n3cc(-c4ccc(C)o4)nn3)CCC2)=O)ccccc1OCCF 48524,c1(C(=O)NCC2C(CNC(CNS(CC)(=O)=O)=O)C2)csc(CC)n1 48525,N1(C(C(CC)C#N)=O)CC2CCC(NC(=O)CCC3CCC(C)O3)C2C1 48526,C1(NC(c2cnc(CC)nc2)=O)CC2CN(C(=O)C(C)(C)NS(C)(=O)=O)CC2C1 48527,CC(C)C(=O)C(=O)NC1COCC1CC(=O)NCc1nccc(Cl)n1 48528,N(C(=NCc1ccccc1)N1CCOC(c2cnn(C)c2)C1)CC(CC)(C)C 48529,C1(NC(Cc2cc(C)ns2)=O)CN(C(=O)C(O)CC(=O)OC(C)(C)C)CCC1F 48530,c1(CC(=O)N(c2cc(OCC)ncn2)C2(C)CCC(N)C2)cc(C)cc(C)c1 48531,Cc1ccnnc1C(CC(=O)NC(C)C)N(C1CCS1)C 48532,c1(C(=O)NCC2CCC(NC(c3cc(C)oc3C)=O)C2)nccc2ncccc12 48533,c1(C(N2CC(NC(c3cc(O)ccc3F)=O)C(O)C2)=O)ccc(I)cc1Br 48534,Cc1scc(NC(=O)CC2CCN(CC(=O)NC(c3ccccc3F)C)C2)c1C 48535,C1(C(N2CC(OC)C2)=O)CC(C)CN1C(c1cn[nH]c1)=O 48536,CCC(CC(=O)NCCC1(NC(C2(S(N)(=O)=O)CC2)=O)CC1)C(C)C 48537,CC(CCC(=O)NCCOC1CC(C(=O)NC2CSC2)C1)n1cccn1 48538,CC1CCN(C(=O)C(C)OCC(=O)NC2CC2C)CC1.c12cn(nn1)CC(=O)N2 48539,C1(C(=O)NC(CC)CNC(C2(CC)CC2)=O)CCc2cc(OC)ccc2C1 48540,C1(CC(=O)N(CC(C)(C)NC(Cc2cnc(C)o2)=O)C)CCC(C)CO1 48541,N1(C(CNC(CC)=O)=O)CCCC1C1CCC(C(=O)OC)O1 48542,CC(C)C(C)CC(=O)NCC(C)(O)CNC(=O)CCc1cncc(O)c1 48543,N1(C(C(CC(=C)C)C)=O)Cc2ccnn2CC(NC(c2cc(CC)oc2C)=O)C1 48544,O=C1CCC(=O)N1CCC1CC(F)(F)C1 48545,c1(C2(CNC(=O)Nc3cccs3)CC2)ccc(Cl)nc1 48546,C1(C2CC2)(CNC(C(C)CF)=O)CCN(C(=O)CCC(C)(C)F)C1 48547,c1(C(=O)NCCN(C(C(CC)n2cccn2)=O)C(C)C)c[nH]cc(F)c1=O 48548,c1(Nc2c(OC)nsc2)cc(Cl)cc2cn[nH]c12 48549,N1(CC)CC(C(=O)N2CCC(N(C(=O)C(F)(F)C(C)(C)O)C)C2)c2ccccc21 48550,Cc1nc2c([nH]1)CC(C(=O)NCC1N(C(C3CC4(CC4)CO3)=O)CC1)CC2 48551,C=CC1CCCN(C(c2sc(Br)nc2C)C(=O)NCc2ccc(OC)cc2)C1 48552,C1(=CC(=O)N(CCC(C)(C)NC(CC2(C=C)CCC2)=O)C)CN2CCC1CC2 48553,CC1CN(C(=O)C(C2CCCCCC2)O)CC(C)N(C(c2cc(C#N)c[nH]2)=O)C1 48554,Cc1nc(NCc2cc(CO)on2)cc(=NC(C)c2cccc3c2CCCC3)[nH]1 48555,c1(Cc2n(-c3nc(C)nn3C)nc(C)n2)cc(F)cc(Cl)c1 48556,c1(C(=O)NC2CCN(C(CC(CCC)CC)=O)C2C)cccc2c1CC(C)(C)C2 48557,C1(OC)CC(CNC(C2CC3CC3C2)=O)N(C(=O)CN2CC(C)(C)C2)C1 48558,N1(C(c2ccc3oc(O)nc3c2)C(=O)NCCCC)CCCCC12CCN(C)C2 48559,C1(C(=O)NCCCN(C(COCCOCC)=O)CCO)OCCOC1(C)C 48560,c1(C(=O)NCCN(C(=O)CC2CCCO2)C(C)C)ccc(SC2CC2)o1 48561,Cc1oc2cc(C(=O)NCCN(C)C(C3(O)CC3(C)C)=O)[nH]c2c1C 48562,N1(C(CNC(C)=O)=O)CCc2[nH]nc(C(=O)Nc3cc(Cl)c(F)c(Cl)c3)c2C1 48563,C=CCC(C)(O)C(=O)NC(C)C(=O)NCC(C)(C)C1CCCO1 48564,C(=O)(C1CCCc2nc[nH]c21)NCC1(F)CN(C(c2c(OC)nsc2)=O)C1 48565,CC(C)CC(CCO)NC(=O)CC1CCC(NC(c2csnc2Cl)=O)C1 48566,c1(C(=O)NCCC(C)N(C(C(CC)n2cccn2)=O)C)cc(C)nc(N(C)C)n1 48567,N1(C(=O)Nc2nccn2-c2ccccc2)CCN(c2ccccc2)CC1CCO 48568,N1(C(CCC=C(C)C)=O)CCC(N(C2(C)CC(F)(F)C2)Cc2ccccc2)CC1 48569,c1(CNC2CC(C(=O)NCc3cnc(Cl)nc3Cl)C2)c(F)cc(Br)cc1F 48570,N1(C(C(C)O)=O)Cc2ccccc2C1C(=O)NCc1nc2ccccc2nc1O 48571,C1(C(=O)NCCCCC2CN(C(c3c(SC)n(C)nc3)=O)C2)CCC(O)CN1C 48572,C1(COC)CC(O)CN1C(c1c[nH]nc1CNC(c1ncncc1N)=O)=O 48573,CC(F)(F)CC(=O)N1CCC(CCNC(=O)CCN2CCCCCC2)C1 48574,C1(NC(C2C(CCOC)C2)=O)CCCCN(C(=O)Cn2nccc2C)C1 48575,CP(C)(=O)c1cc(Cl)ccc1C(=O)NCCCCCNC(=O)CCc1cnoc1 48576,C(CCC(C)(C)C(=O)NCc1cc(Cl)ccn1)NC(C(C(=O)OCC)CC)=O 48577,C(=O)(CCCC(=O)NCCNC(C1(NC(c2coc(SC)c2)=O)CC1)=O)OC 48578,N1(C(Cc2cn(CC)nn2)=O)CCCC2(CCC(NC(=O)C#CC(C)(C)C)C2)C1 48579,CC1CC2(CCN(C(=O)CSc3ccccc3Cl)CC2)CN1C(C1CC1C)=O 48580,CC(CC(=O)N1CC(CCNC(c2cncnc2)=O)C1)N(C)C(=O)OC(C)(C)C 48581,Cc1n[nH]c(C)c1CNC(C1(NC(=O)C(C)(C)SC2CCCC2)CCCCC1)=O 48582,CC1(NC(c2nnnn2CCC2CC2)CCC2CCC2)CC(F)(F)C1 48583,C#CCC(CC#C)C(=O)NCC1(C)CN(C(C2(C)CCC2)=O)CC1C 48584,N1(C(C=CCCC=C(C)C)=O)CC2CC1CN2C(c1ccc(CO)s1)=O 48585,N1(C(c2n(COC)ncc2)=O)CCC=CC1C(=O)Nc1ccsc1 48586,Cc1cc(C)cc(CN2CCCCC2C(=O)Nc2sccc2C(N)=O)c1O 48587,C1(C(N2C(C(=O)NC)CCC2)=O)(OC)CCN(C(c2sncc2C)=O)C1 48588,N1(C(C2(C)COC2)=O)CCCC(CNC(C23CCCC2(C(N)=O)C3)=O)C1 48589,N1(C(C(C)=CC)=O)CC2CCC(CNC(=O)C=Cc3cccc(C#N)c3)C2C1 48590,Nc1cc(C(=O)NC2CC(CNC(c3ccc(Cl)[nH]3)=O)C23CCC3)cnc1N 48591,C(=O)(CS(=O)(=O)C1CCCC1)NCC1(C)CCCN1C(C1CC12CC(O)C2)=O 48592,C=CCCCCC(=O)NCC1CC(O)CN(C(=O)CCCc2ccccc2N)C1 48593,Cc1ccc(F)c2[nH]c(C(N3CCN(C(c4cnn[nH]4)=O)CCC3C)=O)cc12 48594,C(c1ccc(Cl)cc1)=CC(=O)NCCO.N12CCC(CC1)C2=O.C1(C)(CC)CC1N 48595,c1(C(N2C(C(N3CCC(NC(=O)NC)C3)=O)CC3CC32)=O)c[nH]c2ncccc12 48596,c1(CN2CC3(CC(C(N4CC(C(N)=O)OCC4)=O)C3)C2)c(Br)cc(F)c(F)c1F 48597,N1(C(C(C)=C(C)C)=O)CCC2(CCN(C(=O)C(=O)Cc3ccccc3)C2)C1 48598,C#CCCCCC(=O)NCc1cc(C(N2CCC=CC2C(=O)OCC)=O)n(C)n1 48599,c1(C(=O)NCC2C(C)CN(C(c3ccncc3)=O)CC2)n[nH]c2cccnc12 48600,C1(NC(c2c[nH]nc2OC2CCCC2)=O)CCCCN(C(=O)C2=C(Cl)CC2)C1 48601,C=C(Cl)CC(C(=O)NCCCN=[N+]=[N-])NC(c1ccncc1OC)=O 48602,c1(NC2CCCN2C(N(CCOC(C)(C)C)CC)=O)cccc2c1CCOC2 48603,c1(C(N2CC(C(N3CC(n4c(C)ncc4)C3)=O)SCC2)=O)nccc2occc12 48604,C1(CCNC(CCC(=O)NC)=O)CCN(C(=O)CC2CN3CCC2CC3)C(C)C1 48605,CC(C)S(=O)(=O)C(C)C(=O)N1CCC(C=CC(=O)NCCC2CC3CC3C2)CC1 48606,CCC(C)C(O)C(C)C(=O)N1CCC(NC(c2cnnc(C)c2C)=O)C1 48607,C1(CC)CC(OC)CN1C(=O)NCC(=O)NC1CCCC1 48608,C1(C(=O)NC(C)CCNC(c2conc2C(C)(C)C)=O)CCN(S(N)(=O)=O)CC1 48609,C1(OCC)CCCCC1NC(c1c(Br)cnn1C)=O 48610,C12(Nc3nc(C)c(C)s3)CCCC1CN(C(C1CCCS1)=O)C2 48611,c1(C(N(CC(C)NC(COC(C)C)=O)C)=O)ncccc1N(C)C 48612,CCCCC(F)C(=O)N(C1CCCN(C(=O)C(C)(C)OCC)C1)C 48613,N1(C(CC(C)=CC)=O)CC2CCCC(CNC(=O)CCc3c(C)noc3C)C2C1 48614,c1(COC(Cc2ccc(CC)cc2)=O)nccc(C)c1F 48615,C1(C(=O)NC(CC#C)COC)(C(=O)NC)CCCN1C(c1cc(CO)[nH]n1)=O 48616,CC1CCC(CNC(c2csc(=N)[nH]2)=O)CN1C(=O)CC1(O)CCCCCC1 48617,C(CCCCC(=O)NCC1(NC(c2csc(C)c2N)=O)CCC1)OCC 48618,CCC(CNC(=O)C(C1CCOCC1)O)(CC)NC(c1cnn(C)c1C1CC1)=O 48619,C(=O)(CC(F)(F)CC)NC(CCC)CNC(C1CCCN(C(C)C)C1)=O 48620,c1(CC)cc(C(=O)N(C)CCOCCCN(C)C(C2SCCC2C)=O)no1 48621,C1(C(N(CCCNC(C2(C(F)(F)F)CC2)=O)CC)=O)CCCCN1c1ncccn1 48622,C(C)(CCC(=O)N1CC2C(N(C)C(C3CC(=O)N(C4CCCCC4)C3)=O)C2C1)OC 48623,CCC(CC(=O)NC(CN(C)C(c1cccc(C(C)C)n1)=O)CC)OC 48624,C(=O)(C1CCCn2c(Br)cnc21)NCC(CN(C(=O)C(O)C1CCC1)C)(C)C 48625,N(C1CCc2cccc3cccc1c23)CCn1ncn(C)c1=O 48626,c1(OC)c(C)cc(C(=O)NCCC(C)NC(C2(C(C)(C)C)CCC2)=O)cc1Cl 48627,C1(O)(C(C)NC(c2n(CC)ccc2)=O)CCN(c2ncnc(C)c2F)CC1 48628,C(CC(CNC(=O)CSS(C)(=O)=O)NC(c1ccnn1C(C)C)=O)OC 48629,CCCC(C#N)C(=O)N1CCN(C(c2ccncc2Cl)=O)C(C2CCC2)C1 48630,c1(C(=O)NCC2C(NC(=O)C(c3ccccc3)C3CC3)C2)cnn(C2CCC2)c1 48631,N1(C(c2ccc(CC)[nH]2)=O)CCOCC1CNC(=O)CCc1ccc(OC)cc1 48632,N1(C(CC(=O)NC)=O)CCC2(CCC(CN(C)C(c3ccccc3)=O)O2)CC1 48633,C1(NC(C(C)CO)=O)CN(C(=O)C=CC2CCCC2)CC2CCCC12 48634,c1(C(=O)NCC(C)NC(Cn2c(C)ncc2[N+](=O)[O-])=O)cncc2nc(O)[nH]c12 48635,c1(CC)cc(C(=O)N(C2CN(C(C3(N4CCCCC4)CCCC3)=O)C2)C)nn1C 48636,C1(CNC(=O)Nc2ccc(OCCC)cc2)CCN(C(=O)C(=O)NC)CC1C.C(N)=O 48637,CCCC(C)(O)C(=O)NCC1CCCN(C(c2cc(C(F)(F)F)nn2C)=O)CC1 48638,C1(NC(C(CC(C)C)OC)=O)CCCCC12CCCC2.C1CC(=O)O1 48639,C1(C(C)NC(=O)COC(F)F)CN(C(=O)CCCC2CCCO2)CCO1 48640,c1(CNC(=O)NC2CCN(CC(=O)OCC)C2=O)noc2c1CCCCC2 48641,c1(CC(CC(=O)NC(CNC(C=CCN(C)CC)=O)C)SC)ccc(F)cc1F 48642,C1(O)(CC)CCCN(C(C2CN(Cc3ccc(Cl)nc3)CCC2O)=O)C1 48643,C1(C(=O)NC(CCC)C2CC2)CCN(C(c2cc(O)ccc2C)=O)C(C)C1 48644,c1(COC)cccc(C(N2CC(N3CC(C)(O)C3)C(C)C2)=O)c1 48645,N1(C(c2c[nH]cc(C)c2=O)=O)CC(NC(=O)Cc2nc[nH]n2)C2(CCCC2)C1 48646,C(=O)(C(F)(F)C(F)(F)F)N1CC(NC(=O)COC(=O)CC2CCC(C(F)(F)F)O2)C1 48647,CC(C)C(C(=O)NOC(C(=O)OC(C)(C)C)C)C(C)OC(C)C 48648,C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NCC1C(NC(CC(CC)C(F)F)=O)COC1 48649,C=CC(C)(CC)C(=O)N1CCN(CC2CN(C(c3cc(Cl)no3)=O)CCO2)CC1 48650,C1(C(=O)NCCN(C2CCCCCC2)C(C2(O)CCC2)=O)CC2CCCCCC12 48651,N1(C(C(=O)NCC)=O)CC(NC(=O)C(C)Cc2c(C)n[nH]c2C)C(C)(C)C1 48652,c1(CCC)cc(C(N2CC(C(N)=O)(CNC(C3(F)CC3C)=O)C2)=O)no1 48653,C#CCCC(O)C(=O)N1CCCN(C(C2CCS(=O)(=O)CC2)=O)CC1 48654,Cc1cc(C(N2CCC(C(F)(F)F)(C(=O)O)C2)=O)nc(O)c1 48655,C1(CCNC(=O)CCN2CCCCC2)COCCN1C(=O)CC1CN(C(N)=O)C1 48656,C#CCCCCCCC(=O)NCC1(NC(=O)Cc2nccc(OC)n2)CCOC1 48657,C1(C(=O)NC(C(=O)N(CCCN(C)CCO)C)C2(NC(C)=O)CC2)(CC)CCOC1 48658,CC(C)CCC(=O)N1C(CNC(c2ccc(N3CCCC3=O)nc2)=O)CC2CC12 48659,N1(C(C)C)CCC(C(=O)NC2CCCC2Nc2ccc(F)cc2)CC1 48660,C1(C(=O)NCC(CC)NC(c2cc(N)ccn2)=O)(COC)CC(C)(C)C1 48661,c1(C(N2CC(CNC(CNC(=O)OC)=O)C(C)C2)=O)cc(C#N)[nH]c1C 48662,C#Cc1ccc(C(=O)NC2CC(C)(NC(c3cccc(C(C)C)n3)=O)C2)cc1F 48663,N(C(=NCCC(C)C)NC1CCCOC1)Cc1c(OC)ccc(Cl)c1OC 48664,C=C=CCCC(=O)NC(C1CCN(C(c2nccc(C(F)F)n2)=O)C1)C 48665,c1(C(=O)NCCC2CCCN(C(c3csc(C4CC4)n3)=O)C2)c(O)cccc1Cl 48666,N1(C(C2N(CC)CCCC2)=O)CCC(NC(c2cc(Cl)nnc2O)=O)C(CO)C1 48667,CCCCCC(O)CC(=O)NCCC1CC(NC(c2nc[nH]c3ncnc2-3)=O)C1 48668,C1(C(=O)NCC2(C(=O)NCC(=C)C)CC(=C)C2)CCC2(CCC2)C1 48669,Cc1cccc2c1C(NC(=O)CC1(CO)CCS(=O)(=O)CC1)CC2 48670,c1(-c2nc(C)[nH]n2)ccc(C(N2CC(NC(c3cc(Cl)ns3)=O)C(O)C2)=O)cc1 48671,n1(C(CC)C)ncc2cc(C(N3CC4CC3CN(C(C3CCSC3)=O)C4)=O)cnc12 48672,C1(CN(C(=O)CS(=O)(=O)N2CCOCC2)CC)CCCCN1C(=O)C(N)=O 48673,c1(OC)cc(C(=O)NCC(CC(C)C)NC(=O)C=CC2CCOC2)n(C)n1 48674,N1(C(CC(C)NC(C)=O)=O)CCCC(NC(C2CCC(C(F)(F)F)CC2)=O)CC1 48675,N1(C(C2C(C)CC2)=O)CCc2c(CNC(=O)CC3=CCCC3)cccc2C1 48676,c1(C(N2CCOCC2)C)cn2c(n1)CCCN2C(=O)Cc1nc(Cl)n[nH]1 48677,CC(C)CCCCC(=O)N1CCCC1CCNC(c1ccc(Br)s1)=O 48678,C1(CCOC)(NC(=O)CCC2CCCO2)CCN(C(=O)C(OC)OC)C1 48679,C#CCC(C)(CC)C(=O)NCCC1(O)CCN(C(=O)C(C)(C)OCCC)C1 48680,Cc1cc(NC(=O)CC2COCCO2)ccc1NC(=O)CNS(=O)(=O)C1CC1 48681,C(CC)(C(=O)NCC1CC(CC(C)Cc2ncn(C)n2)C1)OCC 48682,c1(OC(C)C(=O)NCCC(C)N(C(=O)CNc2cccnc2)C)ccccc1Cl 48683,C(=O)(C1CCc2nccn21)NCC1CC(OC)CN1C(c1cc2occc2[nH]1)=O 48684,N1(C(=O)CC(O)C2CC2)CCC(NC(C2CC(n3ccnn3)C2)=O)CC(O)C1 48685,C(CCCC(=O)NCCc1ccc(F)cc1)NC(C1C(C)(C)C1)=O 48686,C(C)(C)(CCCC(=O)NCC(O)C1CC1)NC(C(c1n(C)ccc1)=O)=O 48687,C1(NC(c2c(OC)cnc(Cl)c2)=O)CC2CCC(C1)N2C(C1(C#N)CC1(C)C)=O 48688,N1(C(c2cnc(SC)s2)=O)CC2(CCN(C(c3ccncc3N)=O)CC2)CC1C 48689,O=S(=O)(c1cccc(=NC2CCOC3(CCCC3)C2)[nH]1)NCCCF 48690,C1(CNC(=O)Cc2ccns2)CC(C(=O)N2CC3C(C2)C3(F)F)=NO1 48691,c1(N2CCC(C(C)C)CC2)ccc(S(=O)(=O)NCCCO)cc1Cl 48692,Cc1ccc2oc(C(N3CCC(c4cccc(O)c4)C3)=O)cc2n1 48693,N1(C(c2cc(C)c(F)c(C)c2)=O)CCN(C(=O)C(O)C(C)(C)C)C2CCCC12 48694,c1(OC)ccc2sc(C(=O)NC3CC(OC)CN(C(=O)C(C)CO)C3)c(C)c2c1 48695,C12CCC(C1)N2.c1(O)ccncc1.C1(C(=O)NCCNC(CNC=O)=O)CCOCC1 48696,C(C)(CC(=O)NCC1CCN(C(=O)Cc2csc(NC=O)n2)C1)OC 48697,Cc1snnc1C(=O)NC(CC1CCOCC1)C(=O)N(CC(C)O)CCF 48698,C(=O)(CN1C(=O)CCc2ccccc21)NC(C)CCN(C)C(c1ccnnc1)=O 48699,CC1CCCn2ncc(C(=O)NCC3(O)CC(NC(c4ncc[nH]c4=O)=O)C3)c21 48700,N1(C(CCCOCC=C)=O)CCC(C)(CCNC(=O)COc2ccon2)C1 48701,C#Cc1ccc(OC)c(C(N2CCC(CCNC(=O)C(C)CS(C)(=O)=O)C2)=O)c1 48702,CCCCCCCCCC(O)C(=O)NC1CN(C(C2(n3cccn3)CC2)=O)CC1C 48703,c1(C2N(CC(C3CCN(C4CCCCC4)C3=O)=O)CCCC2)ccc(Cl)cc1Cl 48704,CCCC(CCCNC(=O)CCNC(=O)C1CC1)NC(=O)CC1CCCO1 48705,C1(C(=O)NCC(C=C)O)CCC(C)N(C(c2cnc(CC)cn2)=O)C1 48706,c1(C(C)=O)cccc(NC(C2(C)CCCN2C(c2ccc(C)o2)=O)=O)c1F 48707,N1(CC(c2cn(CCC=C)nn2)C)CCCCC(C(=O)OC)C1 48708,C12(NC(C3C(CNC(C=CC(C)C)=O)OCC3)=O)CCC(C1)OC2C 48709,C1(C)(C(=O)NC(c2cccs2)CC)CC12CCN(c1cc([N+](=O)[O-])c(C)s1)CC2 48710,N1(C(c2scc(COC)c2)=O)CC2CCN(C(=O)CCCCCF)CC2C1 48711,N1(C(C2C(NC(C(COCC)N(C)C)=O)CC2)=O)CCCC(C)(CC)CC1 48712,Cc1ncccc1CCC(=O)N(CC(O)CN(C)C(C1C=CCS1)=O)C 48713,N1(C(COCc2n(C)c(O)nn2)=O)CCC2(CC1)CC2(C)C(=O)NCCO 48714,C12(NC(C(CCCC)NC(N)=O)=O)CCCC1CN(C(=O)CC1(O)CCCC1)C2 48715,C(=O)(CCCCCC(C)O)NCCC1(NC(c2c(CC=C)cccc2)=O)CCC1 48716,C(=O)(C(C)(C)CCCF)NCC(C)(CNC(=O)Cc1ncc(C)s1)OC 48717,c1(C(=O)NC2CC(F)(CNC(CC(COC)C)=O)C2)cccc(OC)c1C 48718,C(c1cc2ccccc2o1)=CC(N1C(C(=O)Nc2cc(C(C)(C)C)n[nH]2)CC1)=O 48719,O=C(C(=O)C(F)(F)F)NCC1CN(C(c2cn(Cc3ccc(CO)o3)nn2)=O)C1 48720,N1CC2(CC(NC(=O)CCC3CC3)c3nccn32)C1.c1(CC)conc1C1CCC1 48721,CC(C)(C)C(=O)NCCCC(=O)NC1CCC1NC(=O)Cn1ccc(C2CC2)n1 48722,C1(CC(=O)NC2CCC(CNC(C(CC)N3CCCC3=O)=O)C2)CCCOCC1 48723,N1(C(C2(C3(C)CC3)CC2)=O)CC(C(=O)NC2(C)CC2)C2(CCC2)C1 48724,N1(C(C(COC)(C)C)=O)CC2(C)CC1(C(=O)NC(C)CCc1cn[nH]c1)C2 48725,C(=O)(C1(C)CCOc2ccccc21)N(CCNC(C(CCCC)CC)=O)C 48726,C1(NC(C2N=C(C)SC2)=O)CCCC2CN(C(=O)CSc3ccccc3Cl)CC12 48727,C(=O)(C(CCCC)NC(=O)CNC=O)NC1CC(=C)C1 48728,Cc1nc(C(N2CCCC(NC(=O)C(C)Cc3cnn(C)c3)C2)=O)c(C)s1 48729,C#Cc1ccc(CC(N2CCC(C(C)C(=O)NC(C3CC=CCC3)(C)C)C2)=O)cc1 48730,C#CCCCCCC(=O)N(CCCN(C)C)CCNC(C1(F)CC=CC1)=O 48731,N1(C(CC2CCN(CC)C2)=O)CCC(CCCCNC(C2C3COCC23)=O)CC1 48732,C12(C(=O)NC3CC(NC(C4C(C(N)=O)CC4)=O)C3)CCC(OCCO)(CC1)C2 48733,NC(=O)N=Nc1ccc(C(=O)NCC2CC(NC(C3CCCN3C=O)=O)C2)cc1 48734,n1(C(C(=O)OC)C)nccc1C(=O)N(CC(C)CNC(=O)CN1CCSCC1)C 48735,Cn1nc(-c2nc(-c3ccc(C(F)F)cc3)nn2C2CCCSC2)c2c1CCCC2 48736,N1(C(CC(CNC(=O)CC=C(Cl)Cl)OC)=O)CC(C)(C2CCC2)C1 48737,N1(C(Cc2cccc(CC)c2)=O)CC(NC(c2cncn(C)c2=O)=O)CC1(C)C 48738,c1(OC)ccc(F)cc1CC(=O)N(C)C(c1cccc(Br)c1)C.C1(=O)CN1 48739,CC1CN(C(C2(C)CCCN2C)=O)CCC1C(N1CCCC(CO)(CO)C1)=O 48740,n1(CC=C)cccc1C(=O)NCC(C)NC(=O)Cc1ccoc1C 48741,Cc1noc2nc(C3CC3)cc(C(N3CCCC(F)(F)C3)=O)c12 48742,C1(NC(=O)C2CC2)CC2CCCC(C1)N2CC1CN(C)C(=O)C1 48743,C1(C(=O)NC2CN(C(C3C(=C)C3)=O)C2)CCCCCN1C 48744,c1(OC)cc(F)c(C(=O)NC2CC(C)(NC(c3ccnc(Cl)c3)=O)C2)cc1F 48745,c1(C(N(CC(O)CN(C(=O)C(F)CC2CC2)C)C)=O)cccn2ccnc12 48746,C(c1ccccc1F)=CCC(=O)N(CC(C)(C)NC(CCc1cc(C)no1)=O)C 48747,n1(CCOC)ncc(C(C(=O)NCSc2ccccc2)NCC(C)(O)C(F)F)c1C 48748,CC(C)(CCCF)NC(=O)CC=C(Cl)Cl.C123CC(C1)(C2)C(=O)N3 48749,C1(C(=O)NCC(=O)OCCCC)CCN(C(c2cc(C)c(C)cn2)=O)CCO1 48750,c1(C(N2CCC(O)(CCNC(C3C(C)(C)CO3)=O)C2)=O)cc2scnc2[nH]1 48751,Cc1ccc(C(C)NCc2scnc2-c2ccccn2)s1 48752,N1C(=NCCOCC2CN(C(=O)Nc3ccccc3)C2)NCC1C.C(C#N)OC 48753,C1(CNC(c2nccc(CCC)c2)c2nnnn2C)(CO)CC12CCC2 48754,N1(C(CC=CC)=O)CCCN(CCNC(c2ccc(OCCO)cc2)=O)CC1 48755,C(=O)(CCCCC(C(F)(F)F)NC(C(=O)NCCO)=O)NCC1CC1 48756,N1(C(c2cn(CC)nc2)=O)CCCN(C(=O)CSCCC(C)C)CC1C(C)(C)C 48757,C#Cc1ccccc1CC(N1CC(CNC(=O)CC(=C)Br)CC1C)=O 48758,c1(CC(=O)N(CCCOC)CCO)ccc2n[nH]cc2c1.c12ncccc1S2 48759,NC(CC(C(F)F)NC(c1cc(-c2ccc(Cl)cc2)[nH]n1)=O)C(=O)O 48760,Cn1nc(O)cc1C(=O)NCc1csc(CNC(=O)Cn2cc(C(F)F)cn2)n1 48761,C1(NC(C2N(C)C(=O)NC2)=O)CC2CN(C(C3CCOC(=O)CC3)=O)CC2C1 48762,C(C(C)(C)CC(=O)N(CCC(=O)NCC1CCCN1C1CC1)CCO)OC 48763,c1(OCC(=O)N(C2CN(c3nnnn3C)CCO2)CC)c(C)cccc1Br 48764,c1(C(=O)NCC2C(C(=O)NC(CC)C3CC3)CCO2)ccc(F)cc1C 48765,n1(CC)c(C(=O)NCC(C)N(C(=O)CC(=O)NC2CCCCC2)CC)cnc1O 48766,C1(COC(CC)(C)C)CCCC(CNC(=O)Cc2cnnn2CC(C)=O)C1 48767,C(=O)(C(C(C)C)C(C)C)NCC(C1CC1)NC(c1c(C)cc[nH]1)=O 48768,N1(C(CNC(C2ON=C(C)C2)=O)C)CCN(C(=O)C=CSC)CC1 48769,C(C#CCN=c1[nH]c(N2CCN(c3cccnn3)CC2)nc2c1CCC2)OC 48770,Cc1cc(Br)cc2c1CN(C(c1cnsc1)C(=O)NC1(C)CC1)CC2 48771,CC1ON=C(C(=O)NCC2CN(C(=O)CCC(F)F)CC(C)(C)O2)C1C 48772,CCC(C)C(C(=O)NC(C)CN1CCN(C(=O)CC2CC(C)C2)CC1)NC(N)=O 48773,N1(C(C(=C(C)C2CC2)F)=O)CC2CCC(C1)N(C(c1nc(C)c(C)s1)=O)C2 48774,C1(C(=O)NCC2=NOC(C)C2)CCCCCC1NC(C1C=CCS1)=O 48775,C12(NC(c3cnco3)=O)CCCC1N(C(c1cc(-c3ccccc3)co1)=O)CC2 48776,C12(NC(CCS(C)=O)=O)CCOCC1CN(C(C1(c3cc[nH]n3)CC1)=O)C2 48777,C=CCC(C(=O)N1CCCC(C(=O)NC2CC(CO)C2)(C(C)C)C1)C(C)C 48778,N1(CC(=O)NCC(C)(C2CCC2)NC(c2c(C)cc(C)s2)=O)CCC(=O)NC1=O 48779,c1(C(N2CC(NC(c3c(CC)onc3)=O)C3(C2)CC3)=O)ccc2n[nH]cc2c1F 48780,C1(CNC(C)(C)C)CCCC1SCCCC(=O)N(C1(C(=O)NCCC(N)=O)CC1)C 48781,C1(C(N(C2CCN(c3nnc(O)s3)C2)C)=O)CCc2ncncc2C1 48782,CC1CN(C(=O)CCC=CCN(C)C)CCC1N=c1[nH]c(Cl)ncc1[N+](=O)[O-] 48783,c1(C(=O)NC2(c3ccccc3)CCN(C(C(C=C)O)=O)C2)cc(C)nnc1O 48784,C1(C(=O)NCC(CC)NC(=O)CCc2cn(C)nn2)CCCC1c1ccccc1 48785,C1(N(C)Cc2ccccc2)CCCCN(C(c2cc(I)cnc2Cl)=O)C1 48786,C(=O)(C(C)(C)C#N)NCC1CC(CC(NOC(C(C)C)CO)=O)C1 48787,c1(C(N(C2CCN(C(C3(O)CCC3)=O)C2)C)=O)cc(C(F)F)cc(Cl)c1 48788,C(c1c(Cl)cccc1Cl)=CC(=O)NCC1CN(C(CC(=O)OCC)=O)C(C)C1 48789,Cc1nn(CC(F)F)cc1C(N1CC2C(N(C(=O)CC3C=CCC3)C)C2C1)=O 48790,C(CCCCC(=O)NCC1CC(NC(=O)CSC)C1)=CC 48791,C(C(C)(C(C)C)NC(=O)C)NC(C1(OC)CC1)=O.c1(OC2CCCC2)cccnc1 48792,CC(CCO)CCN=c1[nH]c(=NC(C)c2nc[nH]n2)c2ccccc2[nH]1 48793,CC1CCCC=C1C(=O)NC1CCN(C(=O)CC(F)(F)C(F)F)CC1(C)C 48794,c1(OC)cc(C(=O)NC23CC(CNC(=O)C(O)CSC)(C2)OC3C)cc(OC)n1 48795,c1(C(N2CCC(N(C(=O)CCC3CC(OC)C3)CC)C2)=O)ccnc(Cl)c1OC 48796,N1(C(C2N(C(c3c(C)c[nH]c3)=O)CC2)=O)CCC2(CCCO2)C1 48797,C=CC1CCN(C(=O)CC2CCN2C(=O)C(C)SCC)CC1 48798,C(CCC(C)C)(C(=O)N(C)CCc1ncccn1)NC(C1C(CCC)CCC1)=O 48799,CCS(=O)(=O)C=CC(=O)NCc1ncoc1CCNC(c1ccc(OC)c(Cl)n1)=O 48800,C1(OCC)CC(CN(C(=O)CNC(c2cc[nH]n2)=O)C)C1 48801,C(c1cn(C)cn1)=CC(=O)NCC(CN(C(CCc1onc(C)n1)=O)C)O 48802,C(=O)CC1=NNC(=O)C1.c1(-c2cn(C)c(-c3c[nH]nn3)c2)cc2sccc2s1 48803,N1(C(c2c(CC)cns2)=O)CC(O)CCC1C(=O)NCCn1ncnn1 48804,C(=O)(NNC(=O)C1CCC(C)O1)NC(c1cc(C)on1)C 48805,C1(S(N)(=O)=O)(CS(=O)(=O)NCCN(c2cncc(OC)n2)C)CCCC1 48806,N1(C(C(CC)(C)O)=O)CCCCC2(C1)CN(C(c1nn(C(F)F)cc1Cl)=O)C2 48807,c1(C(N2CC(O)(CNC(C(CCCC)O)=O)C2)=O)cc(=O)c2cc(F)ccc2o1 48808,C1(C2CCCN(C(c3ccccc3Cl)=O)C2)(NC(C#CC(=O)O)=O)CC1 48809,Cc1cc(=NC2CCOC(C3CC3)C2)[nH]c(=NCCCc2cn[nH]c2)[nH]1 48810,N1(C(CC2(C(N3CCC(C)(C)C3)=O)CC2)=O)CCOCC(CN(C)C)C1 48811,C1(C(=O)NCCNC(c2c[nH]cc2-c2ccccc2)=O)C2CCCC12 48812,CCCCCC(O)C(=O)N1C(C)C2CC1C2NC(=O)CC1(C#N)CCC1 48813,c1(C(N(C2CCCN(C(c3cc[nH]n3)=O)C2)C)=O)ccc(N)c(Br)n1 48814,CCC(C)(C)CC(=O)N1CCOC(C)(CNC(=O)CC(C)OC)C1 48815,C=CC(CCC)CC(=O)N1CCC(O)(CN(C)C(c2cc(C)n(CC)n2)=O)CC1 48816,N1(C(C2N(C)CCC2)=O)CCOCC(NC(c2cccc(O)c2O)=O)C1 48817,c1(OC)ncc(Br)cc1CNC1CCN(C(=O)CC2CCNCC2)C1 48818,C=CCC(CC(C)C)C(=O)N1CC(NC(c2cc([N+](=O)[O-])n[nH]2)=O)CC(C)(C)C1 48819,C1(C2CCOCC2)(C(=O)NCC2N(C(CCCN(C(C)C)C)=O)CC(O)C2)CC1 48820,N1(C(CCCC)=O)CC(=O)NCC1C(N1CCCC(C)(CO)C1)=O 48821,Cc1sc(O)nc1C(=O)NC(C1CCCN(C(=O)COCC2CCOC2)C1)C 48822,CC(C)(C(=O)NC1CCCC1n1cc(C(C)(C)C(=O)OCCBr)nn1)C1CCCC1 48823,c1(C(=O)NCC2(OC)CN(C(C3CCCS3)=O)C2)cnc2ncnn2c1C(C)C 48824,C1(CC)CNC(=O)CN1C(c1sccc1Br)C(=O)NCCOCC1CC1 48825,c1(C(=O)NCC2CC(C)N(C(c3ccc(C(N)=O)[nH]3)=O)C2)cccc2occc12 48826,C(C(C(C)(C)C)NC(=O)C(C)Cc1ccnn1C)NC(c1n(CC=C)ccn1)=O 48827,N1(C(c2ccc(SC)s2)=O)CCC2CN(C(C3OC(C)(C)OC3(C)C)=O)C2C1 48828,CC#CCCCC(=O)NC1CCC1CNC(c1ncn(CC)n1)=O 48829,CCC(CC(=O)NC(C)CC(C)NC(c1c(C)cncc1C)=O)C(C)(C)C 48830,C(=O)(CC(C)C)NC(C(=O)NCCCN(CC)CC)c1cccs1 48831,C1(C(=O)NC(C2CCCC2O)C)C=CCN(C(=O)CC2CC(=O)NC2=O)C1 48832,N1(C(N)=O)CCCC1C(=O)NC1CC(NC(c2cn(C3CCOC3)cn2)=O)C1 48833,c1(CC(=O)NCC(C2CCC2)NC(C2(CC)CCNC2=O)=O)c(F)cccc1Cl 48834,Cc1ccc(C)c(C(=O)NC2CC3CC2N(C(=O)CC2(O)CCCOC2)C3)n1 48835,C(=O)(C#CC1(C)COC1)N1C(C)CCC(C(=O)NC(CC)CO)C1 48836,C12CC3(CCC3)CN1C2=O.c1(CNC(=O)CCCc2cc[nH]n2)ccncc1Cl 48837,N1(C(CNC(CCC)=O)=O)CC(F)CC1CNC(c1c(C)ncn1C)=O 48838,c1(C(=O)NC2CN(C(c3c(OC)n[nH]c3)=O)C(C)CC2)cnc2ccncc2c1 48839,n1(CCC(=O)NC2CC(NC(CN3CCC(C)(C)C3)=O)C2)cc(S(N)(=O)=O)cn1 48840,C(=O)NNc1cc(F)cc(F)c1.c1(C(CN)C2CC2CC)ccccc1 48841,c1(CC)cccc(N(C)C(c2csc(CNC(=O)C(F)=CCC)c2)=O)c1 48842,N1(CC)CCOCC1C(=O)NCC(=O)NCC(N1COCCC1C(=O)OC)=O 48843,CS(=O)(=O)c1cscc1C(=O)NC1CN(C(C2(F)CC=CC2)=O)C1 48844,c1(C(N2CCCC(C(C)NC(=O)Cc3nc[nH]n3)C2)=O)cnn2c1OCC2 48845,c1(C(=O)O)cc(S(=O)(=O)NCCCc2cccc(C(F)(F)F)c2)cc2c1OCO2 48846,CC(C)CC(C)(O)C(=O)N1CCCC(CNC(=O)C#CC2CCC2)C1 48847,Cn1ncc(CC(=O)NC2CCC(NC(c3ccon3)=O)C2)n1 48848,c1(OC)ccc2c(c1)C=C(C(=O)NC(C)CCNC(=O)C(C)n1ccnc1)CO2 48849,CCC(C#N)C(=O)NCC(=O)NCCC1CCN(c2ncnc(C(C)(C)C)n2)C1 48850,C(=O)(C(CC1CN(C(=O)OC(C)(C)C)C1)NC(C1CC1F)=O)NCC(=C)C 48851,CC1(C(N2CCCC(CCO)C2)=O)CCCN(C(c2ccncc2Cl)=O)C1 48852,c1(C(=O)NC(CNC(c2c(CC)non2)=O)CCOC)coc2ccccc12 48853,c1(C(CN(C(=O)C(=O)N(C2CC2)Cc2ncc(Cl)s2)C)O)ccc(C#N)cc1 48854,c1(C(N2CCCC(N(C(C(C)=C3CC3)=O)C)C2)=O)ccc2cc(C)cn2c1 48855,n1(CCC(=O)NC2CCN(C(c3c(C)ncnc3)=O)C2)cc([N+](=O)[O-])nc1C 48856,c1(NC2CCCN(C3CCC(C(=O)OC)C3)C2=O)ncc2ccccn12 48857,C1(CNC(COCC(=C)C)=O)C2CN(C(=O)CSc3ccc(Cl)cc3)CC12 48858,C(=O)(C1CCCc2c1ncn2C)N(CCCCN(C(C(CC)C(=O)OC)=O)C)C 48859,C(C(=O)NC1(C)CN(C(c2noc(C3CC3)c2C)=O)C1)(C(C)C)SC 48860,c1(NCC2C(C)C2)ccc(S(=O)(=O)NCC2(Cc3nccs3)CCC2)cc1C#N 48861,C#CCC(C)(C(=O)Nc1nccnc1CC)NC(=O)CNC(N)=O 48862,C1(C(=O)NCCC(C)NC(c2c(OCC)nccc2)=O)CCc2c(cnn2C)C1 48863,C(=O)(C(F)(F)C(O)C1CC1)N(C)CC1N(C(C(C)OCC)=O)CCC1 48864,C(=O)(C(C)(C)C(C)O)NCCCN(C(C1C(C(=O)OC)CC1)=O)CC 48865,c1(OC)ccc2cc(C=CC(=O)NC3CCN(C(=O)C(C)C)C(C)C3)ccc2c1 48866,C#Cc1ccc(C(=O)N(C(C)CN(C(=O)COc2ccccc2OC)C)C)nc1 48867,C#Cc1ccc(NC(=O)C(C2CCN(C(c3cccc(C#C)c3)=O)C2)F)c(C)c1 48868,CCCCCS(=O)(=O)CC(=O)N1CCCC2(NC(c3ccc[nH]3)=O)CC2C1 48869,O=C(F)CN(Cc1nn[nH]c1Cl)N1CC(n2cc(-c3cccc(F)n3)nn2)CO1 48870,CCCCC(C(=O)NCC1CCCN(C(=O)CSc2cccc[n+]2[O-])C1)C(C)C 48871,C(=O)(CS(=O)(=O)C(C)C)N(C)CC1CCN(C(c2c(CCC)nco2)=O)CC1 48872,C(c1cc2ccccc2s1)=CC(=O)N(CC(c1ccccc1Cl)(C)C)CC(F)F 48873,C(N(C)N1CC2(CNC(=O)OC2)C1)C1(C(=O)NC)CCN(C(C)=O)CC1 48874,c1(OC)ncc(N(CCCN(C(=O)COc2ccc(Cl)cc2)C)C)nc1C 48875,c1(C(=O)NC23CCN(C(c4[nH]cc(C)c4)=O)CC2C3)cccc2c1OCCO2 48876,C1(C(N2CCCCC2CCO)=O)(CC)CCCN(C(c2cc(Cl)cs2)=O)C1 48877,c1(C(=O)NC(C(=O)NCC2CC(=C)C2)CC2CCCO2)c[nH]nc1[N+](=O)[O-] 48878,c1(OC)nc(N2CC3(CCN(C(c4cncc(C)n4)=O)C3)C2)ncc1C#N 48879,N(C(=NCCF)NC(C)CC(F)(F)F)C(C1CC(C(F)F)C1)C 48880,CC1C(NC(c2cnn(-c3cc(F)ccc3F)c2)=O)CCCN1C(=O)CO 48881,Cc1nc(CC(=O)NCC(CO)NC(=O)CCC2CCC(=O)N2)co1 48882,N1(C(=O)CC2(c3ccon3)CC2)CCC2(NC(C3CC3F)=O)CCCC12 48883,C1(CS(C)(=O)=O)CN(C(C2CCCC23CCC3)=O)CCN1C(C1CC2CC1C2)=O 48884,C(=O)(CC(O)C(C)C)N1C(C)(CNC(C2(OC)CCSC2)=O)CCC1 48885,C1(CC(=O)NCCN(C(C)C)C(c2cc(-c3ccns3)on2)=O)CC(C)(C)CO1 48886,c1(C(=O)NC(CC)CNC(=O)CC2COC(=O)C2)nnc2n1CCCCC2 48887,C(c1ccc(=N)[nH]c1)=CC(=O)NCC1C(NC(C2(C)CC=CC2)=O)CCC1 48888,C(C(=O)NNC(=O)c1ccc(=N)[nH]c1)Oc1cn(C)nc1 48889,CC1CCCCC1(CNC(c1ccc(=N)[nH]c1)=O)NC(=O)CSCC#N 48890,N1(C(C=CSC)=O)CC(N(C)C)C(CNC(c2cc(CF)on2)=O)C1 48891,c12ccccc1CN2.OC1COCC1COC1CCCCC1 48892,N1(C(c2c(C)ncn2C)=O)C2CCC1CN(C(c1ccncc1Cl)=O)C2 48893,CC1CCOCC1C(N1CCC(O)(CC(N2CCCC(C(N)=O)C2)=O)C1)=O 48894,C1(CNC(C=CCC)=O)CCCC2CN(C(c3ccc(CSC)cc3)=O)CC12 48895,N1(C(C2CCCCN2C(c2cccnc2O)=O)=O)CC2CC(O)CC2C1 48896,N1(C(C(CC)C)=O)CCN(C(C23COCC(C2)C3)=O)CC1CS(C)(=O)=O 48897,c1(C(=O)NC2CC(NC(C3C(C)(C)CCCC3)=O)CC2O)cc2ccccn2c1 48898,c1(NCC2CCCN(CCC(=O)OC)C2)cc(OC)ccc1[N+](=O)[O-] 48899,C1(NC(c2c(OC)cccc2)=O)CCCN(C(=O)C(=O)CC(C)C)C1C 48900,C1(CNC(CC2(C)CC2(Cl)Cl)=O)CCC(NC(c2cnccn2)=O)CC1 48901,c1(C(N2C(COC)(CNC(c3occc3C)=O)CCC2)=O)csc(=NC2CC2)[nH]1 48902,C(=O)(C1CCSc2ccccc21)NC(CC=C)CNC(=O)CCCC(=O)OC 48903,C(=O)(C1=NOC(NC(C=C(C)C)=O)C1)N(CCCCCCC(C)(C)C)C1CC1 48904,C(=O)(C#CC1CCOC1)NC1(C)CCCN1C(=O)Nc1ncsc1S(N)(=O)=O 48905,c1(C(=O)OC)ncc[nH]c1=NCC1(CNC(c2cnc(C(C)C)s2)=O)CC1 48906,C12(CCCCC1)CC=CC(=O)NC2.C1(C(=O)NCC2(CC)CC2)CCSC1 48907,N1(C(c2c(C)nc(CC)o2)=O)CC(CNC(=O)CCC2CCC(=O)C2)CC1(C)C 48908,c1(C(N(CCC)CCNC(C2CC(C)(C)CO2)=O)=O)cc(F)ncc1OCC 48909,c1(C(N(C2CCN(C(C3(C)CCNC3=O)=O)CC2)CCO)=O)occ2c1CCC2 48910,c1(C(=O)NCC(CC)(C)NC(C2CC(CC(C)C)C2)=O)ccc(F)c(CO)c1 48911,N1(C(C(C)C2CCC2)=O)CCCC(CNCc2cnc(N(C)C)nc2)C1 48912,C1(C)(C(=O)NC)CCCN1C(C1(n2cc(C(C)COC)nn2)CC1)=O 48913,Cc1[nH]c(C#N)cc1C(=O)NC1CC2CC(NC(c3cnsn3)=O)CC12 48914,c1(OC)cnc(C(=O)NC(CNC(=O)Cn2cc(Cl)cn2)C(C)C)cn1 48915,CC(C)(C)C(O)C(=O)N1CCCCCC1CNC(c1cn2c(n1)SCC2)=O 48916,CCCC(O)C(=O)N1CCC(C)(NC(=O)Cc2nc(C)sc2C)C1 48917,c1(C(=O)NCC2CC(CSC)C2)ccc2ccoc2c1.C1(NC(=O)C)CCOCC1 48918,Cn1nnc2c1CCN(N1CCC3C(CCN3C(=O)OC(C)(C)C)C1)C2 48919,CCC(CC)(CC)C(=O)N1Cc2occ(C(=O)NCCC3CCCCC3C)c2C1 48920,CC1(C)C(C(=O)OC)CC1c1cn(CC(=O)N(CC(F)(F)Cl)CCCO)nn1 48921,C12CC3CC(C1)N(C3)C2=O.Cc1nccn1CC(=O)Nc1cnc(N(C)C)s1 48922,N1(C(CCn2ccc(C)n2)=O)C(C(=O)NCC2(O)CC(CO)C2)CC2CC12 48923,C(=O)(C1=CCCN(C(c2cc(F)ncc2Br)=O)C1)NC(C)CN1CCCC1 48924,C1(CNC(C(C2CC2)OCC)=O)N(C(=O)C=C2CCCC2)CCCC1(C)C 48925,C12(CNC(c3ccc(OC)nc3)=O)CCCN(C(=O)CCc3nccs3)C1C2 48926,C1(=O)C(O)CCc2cn(nn2)CC2CC(C2)CN1.CCCCCOCC(=O)O 48927,C12(C(=O)NCc3c(C(=O)NC4CCC5(CC5)C4)occ3)CCCC1C2(F)F 48928,CCC(C)C(O)C(C)C(=O)NCC1CC(NC(c2ccc([N+](=O)[O-])cc2F)=O)C1 48929,C#Cc1cnn(CC(N2CCC(NC(=O)Cc3cc(C)on3)C2C(C)(C)C)=O)c1 48930,C=C(C)C(CC(=O)N1CCCCC1CNC(c1csnc1C(=O)OC)=O)OCC 48931,C(=O)(C(C(C)C)OCC)N(CC(CNC(C1C(=C)C1)=O)O)C 48932,Cc1cncc(C(=O)NC23CC(C(=O)NC4CCCC4C(F)(F)F)(C2)C3)c1 48933,O=C(CC1CCN(C(c2ccc([N+](=O)[O-])cc2)=O)CC1)N=c1cc(C2CC2)[nH][nH]1 48934,C(=O)(C(C)C(C)S(C)(=O)=O)N1CC(C2OCCN(C(c3c(SC)n(C)nc3)=O)C2)C1 48935,C(=O)(C1=NOC(C)(C)C1)NC(CC)(C)CCNC(C1CC12CCCC2)=O 48936,C1(N(C(=O)CC2(C)CCC2)CC)CCCN(C(C2(C)CCCOC2)=O)C1 48937,C1(CC(=O)NCCC2CSCCN2C(c2cc[nH]n2)=O)CCNC(=O)C1 48938,c1(CCC)cc(C)c(C(=O)Oc2cccc(C(C)SC)c2)cn1 48939,N1(C(=O)CCOC2CCC2)CC2(CC2)CC1CNC(C1(C(F)(F)F)CCC1)=O 48940,Cc1ccc(CC(=O)NCC(C)(C)Cn2cc(CC(C)C(=O)O)nn2)nc1 48941,CS(=O)c1ccc(C(N2CCCN(C(=O)CCC3(C)CC3)CC2)=O)cc1 48942,C1(O)(CNC(C2CC(OC)C2)=O)CCCN(C(=O)C(C)(C)F)C1 48943,C(=O)(C1COc2ccc(Cl)cc21)NCC1CN(C(c2cc(C)no2)=O)C(C)(C)C1 48944,CC(C)(O)CCCNC(=O)CCC1CCN(C(C2(CO)CCCCC2)=O)CC1 48945,c1(OC)ccc(C2(C(=O)NC3CC(NC(C4(C)CC(C#N)C4)=O)C3)CC2)cc1 48946,C(C1=NOC2(CCC2)C1)CNC(C(C(C)CNC(=O)C(=O)NC1CC1)F)=O 48947,c1(CCC(N2C(CN(C)C(c3cnc[nH]c3=N)=O)CCC2)=O)ccc(Cl)nc1 48948,C1(C(N2CC3(CN(C(=O)CCC4CC4(F)F)C3)C2)=O)CC(c2ccncc2)=NO1 48949,NS(=O)(=O)CCCC(=O)NCC1CCCCO1.C12CCCCN(C1)C2 48950,N1(C(C(CC)N(C)C)=O)CCOC(C2CN(C(=O)CCc3cc(C)no3)C2)C1 48951,C1(=O)CCCC(=O)NCC(O)C(=O)N2CCN1CC2.C(CCC1CC1)SCC=O 48952,C(=O)(C(C)(C)C(=O)N1CC2(NC(=O)CCc3ncccc3C)CC1C2)OC 48953,C(F)(F)(C(=O)NOCC1COCCC1(F)F)c1ccc(C(=O)OC(C)(C)C)cc1 48954,CN1CC(C)(C(=O)NCC(C2CC2)N(C)C(C2C=CCC2)=O)CCC1=O 48955,C(N=c1[nH]cnc2c(Br)nn(C)c12)C1(NC(C(C)CC2CCC2)=O)CC1 48956,C1(NC(c2cncs2)=O)CCCOC12CCN(C(c1cccc(Cl)c1Cl)=O)CC2 48957,n1(C2CCC(CNCC3(C(=O)OC(C)(C)C)CC3)C2)ccc(O)nc1=O 48958,C(C)(C)(CCC(=O)N(CC(N1CCCC(C(F)F)C1)=O)CC(C)C)OC 48959,N1(C(c2ccc(N(C)C)o2)=O)CCN(C(C2(C)CC2(C)C)=O)CC1CCO 48960,C1(NC(C(C)OCCC(C)C)=O)CN(C(c2coc(CO)c2)=O)CC(C)(C)C1 48961,c1(NC(=O)C(=O)NC2CCN(c3nncs3)C2)ccc2c(c1)C(=O)NCCO2 48962,Cc1c(C(=O)NCCC(C)NC(=O)CC2OCCCC2(C)C)cccc1CO 48963,C1(C(=O)NCCC(C(C)C)NC(=O)CC(C)C2CC2)CCCCN(C)C1=O 48964,O=S1(=O)CC2CCN(C(=O)C(c3ccc(Cl)c(C(F)(F)F)c3)(F)F)CC12 48965,c1(C(N2C(C)C(NC(=O)CC(C)(C)C)CC2)=O)cc(S(=O)(=O)NCC(N)=O)c[nH]1 48966,CC(C)C(C(=O)NCc1cnn(C(C)C)c1)c1ccnc(C(=O)O)c1 48967,Cc1nccnc1N1CCN(c2nnc(-c3ccns3)n2-c2ccon2)CC1 48968,C(C(=O)NC1CC1)(C(CC)CC)N(CC(CCCC)CC)C.CCCF 48969,C1(NC(CC(=C)C)=O)CC(O)CN(C(c2ccc(-c3cscn3)cc2)=O)C1 48970,CC(C)(C)C(CCNC(c1ccc(Br)c2[nH]ncc12)=O)C(F)F 48971,C(=O)(C(C)(C)CN1CCN(C)CC1)NCCCCCNC(Cc1cnc(C)s1)=O 48972,C1(NC(CC2C(C)C2(F)F)=O)CCCN(C(C2(C3CC3)CC2)=O)C1 48973,N1(C(C(CC#C)C)=O)CCC(NC(=O)C2=C(C)OCCS2)C(F)(F)CC1 48974,c1(COC(c2cccnc2NC2CCC2)=O)cncc(Cl)c1Cl 48975,c1(C(=O)NCC2N(C(CCN(CC)CC)=O)CCN(C)C2)cc2ncccc2o1 48976,c1(C(=O)NC(C2CN(C(c3cc(CC)c(CC)o3)=O)C2)C)c(N)ccc(F)c1F 48977,N1(C(C=CCC)=O)CC2CC(NC(c3cn(C)nc3-c3ccco3)=O)C1C2 48978,C(C)(c1cccnc1)=CC(=O)NCCN(C(C1(C)CC=CCC1)=O)CC 48979,C(c1ccccc1Cl)=C(C(N1CC(CNC(CN(C2CC2)CC)=O)OCC1)=O)C 48980,CCN=C(NCc1ccc(C)cc1)NC1CSCC1C 48981,C1(C(=O)NC(c2ncnn2C)C)CCN(C(=O)CN2CCSCC2)C(C)(C)C1 48982,Cn1ncc(Cl)c1C(=O)NC(C)(CNC(C1CCCCO1)=O)Cn1cccn1 48983,C1(CC(=O)N(CCCNC(C(C)=C2CCC2)=O)CCO)CCCC(C)O1 48984,c1(C(N(C(CCNC(C(CSC)OC)=O)C)C)=O)ccc2occ(C)c2c1 48985,N1(C(c2c(CC)ccs2)=O)CCC(NC(c2c(SC)cnn2C)=O)C(F)(F)CC1 48986,c1(C(=O)NCCC(C)(C)NC(c2cc(OC)no2)=O)ncccc1SC 48987,N1(C(CCSCC)=O)CCN(C(=O)CN2CC(C)C2)CC1c1nccn1C 48988,C1(OC)CC(CNC(=O)C(C)C)N(C(C2CCN(c3ccncc3)C2)=O)C1 48989,c1(C(=O)NC2CC(CNC(C(CC#C)O)=O)OCC2)cc(OC)cc(Cl)c1F 48990,C(CN=c1nc(N2CCN(C3CC3)C(C)C2)c2c(ncn2C)[nH]1)OCC 48991,N1(C(C2CC=C(C)CC2)=O)CC2=C(C1)CN(C(=O)CCN1CCCS1(=O)=O)C2 48992,N1(C(c2ncn(C)n2)=O)CC(F)CC1CNC(=O)CC1CCC2CC12 48993,c1(C(N2CCC(NC(NCCC=C)=NC)CC2)=O)ncc(C2CC2)cc1F 48994,c1(CC(=O)NCC2N(C(c3nc(CCC)oc3)=O)CC=C2)cc(F)cc(Cl)c1 48995,c1(C(N2CCN(C)C(CNC(=O)C3=CCC3)C2)=O)cc2ccccc2s1 48996,c1(OC)ccc(CN2CCCNC(=O)C2C(C)C)c(F)c1F 48997,c1(C(=O)NC(CN(C(C(CCOC)C)=O)C)C)cccc2nn(C)nc12 48998,N1(CC(c2ccc(C)cc2)C)CCC2(CC1)CCN2C(c1cc(Br)cs1)=O 48999,n1(CCC(=O)NC(CN(C(CC(C)c2ccco2)=O)C)(C)C)cnc([N+](=O)[O-])c1 49000,c1(C(=O)NCC2CN(C(c3cnc(NC(C)=O)o3)=O)C2)cc2ccsc2s1 49001,c1(C(C)=O)ccc(OCCCOC(=O)C(C(C)(C)C)c2cc[nH]n2)cc1Cl 49002,Cc1nc2cccc(C(=O)NCC34CCCC3CCN4C(c3cnsn3)=O)c2[nH]1 49003,N1(C(C(C)SCCCC)=O)CCCC(O)(CCNC(=O)CCCCC2CC2)C1 49004,C1(C(=O)NC(CC)CNC(c2cccc(C(N)=O)c2)=O)Cc2c(F)cccc2O1 49005,c1(OC(N(C)C(c2ccccc2OCC(F)F)=O)C2CC2)cc(F)cc(N)c1F 49006,[N-]=[N+]=NC1COCC1N(C(=O)CCC1NC(=O)N1)C1CCCC1.C1(=O)CNCCN1 49007,N1(c2[nH]c3ccc(C)cc3c2)C(=O)C2C(C)CCCN2C1=O 49008,C1(C(=O)NCc2cnc(C)s2)CN(C(c2c[nH]cc2C)=O)CC1(F)F 49009,c1(CNC(=O)Nc2ncoc2C2(C)CCN(c3cc(C)sn3)C2)c(C)ncnc1O 49010,c1(C(=O)NCC2CCCN(C(CSCC(C)C)=O)C2)ccc([N+](=O)[O-])c(F)c1 49011,c1(OC)c(Cl)ccnc1N(CC(N1CCN(c2cc(C)ccc2C)CC1)=O)C 49012,N1(C(=O)Cc2c(F)cccc2Cl)CC2CCC(C1)N(C(c1ccns1)=O)C2 49013,C1(NC(c2cccc(C)n2)=O)CC2CCC1CN2C(c1ccn(C(C)(C)C)n1)=O 49014,Cc1cc(Cl)c(C(=O)NCC2CCC2NC(c2ccc(CC3CCC3)cc2)=O)s1 49015,CCCC(C#N)C(=O)NCC1(C(=O)NCC(C)CCC)CC=CC1 49016,N1(C(=O)COCC(F)F)CC2(CCCCN2C(C2CCc3ccccc3C2)=O)C1 49017,C1(F)(CNC(c2cc(C)c(O)nc2)=O)COCCN(C(=O)C(C)(C)F)C1 49018,CC1CCC(C)(C(=O)NC2CC3(C2)CN(C(c2cnc(C(C)O)s2)=O)C3)C1(C)C 49019,Cc1cc(F)cnc1C(=O)NC1(CO)CCN(C(c2sccc2OC(F)F)=O)C1 49020,C(=O)(C(C(C(C)(C)C)OC)N1CCCCC1CC)NCC(=C)C 49021,C(=O)(CCCC(F)(F)F)N1C(COC)CN(C(C2CCCCN2C)=O)CC1 49022,CCCC(C)(C)NC(=O)CC1(C)CCN1C(=O)C(CC)SC 49023,N1(C(c2c(CNC(C(C)OC(C)(C)C)=O)nccc2)=O)CCC2(CNC(=O)O2)C1 49024,c1(C(=O)NC(CC(=O)N(CCCO)CC)C2CC2)ccnc(C)n1 49025,N1(C(C(C)(C)CF)=O)CC2(CCN(C(=O)CCCC3CCCCC3)C2)C1 49026,N1(C(C(C=CC)O)=O)CCOC(C)(CNC(=O)C(F)(F)CCC)C1 49027,C1(NC(C2CC3CCC2O3)=O)CN(C(=O)CCc2ncc[nH]2)C2(CCCC2)C1 49028,c1(C2C(NC(C=CCN(CCOC)C(C3CC3Cl)=O)=O)C2)cncn1C 49029,c1(C(N2CC(C(C)NC(c3occc3Br)=O)C2)=O)cc(N)c(F)cn1 49030,C12(C(=O)NC(c3cccs3)C)CCC(CN(C(=O)CCCCCC#N)C1)C2 49031,C1(C(=O)NCC(CC)N(C)CC)CCN(C(=O)CCC2(C)CC2)O1 49032,N1(C(=O)OC)C(CS(C)(=O)=O)C2CCCC12.c1(NC(C)=O)c(CN)nnn1C.C1C(=O)N1 49033,N1(C(CN(C(=O)C(C)=NOCC#N)CCC)=O)CCCCCC1 49034,CCC(C)(C)CCNC(=O)CCC(C)NC(=O)Cn1cc(CO)nn1 49035,C(=O)(C1CCc2nccn21)N1CCN(C(CC2C(C)(C)C2)=O)CC1CC(F)F 49036,c1(C(N2CC(C(=O)NCCCOCC)N(CC#N)CC2)=O)c(Cl)ccc(F)c1Cl 49037,CC(C)CCCC(=O)NCCC1CC(NC(=O)C(C)CC(N)=O)C1 49038,C(CC1C(=O)NCC(=O)NC(=O)CC(=O)N1)=CC.C(C)(C)(C)OC(=O)O.SC 49039,c1(C(N(CCOCCNC(c2ccn(CC)n2)=O)C)=O)ccc2ccsc2c1 49040,C1(CC(=O)NCC2N(C(c3c(C)nn(C)c3Cl)=O)CCC2)CCC2(CCC2)CO1 49041,C(C(COC)C(=O)N1CCC(CCC(=O)NC2CCCC2CCO)CC1)OC 49042,c1(C(CO)N(C2CCNCCC2C)C(C2CCC(O)CC2)=O)ccc(F)c(Cl)c1 49043,C(=O)(C1CCCc2nn(C)cc21)NCC=CCNC(CSCC(C)C)=O 49044,C(CC(C)(C)C(=O)N1C2CCC(C2)C1CNC(=O)C(C)SC(F)(F)F)SC 49045,c1(C(N2CC=C(CNC(CS(N)(=O)=O)=O)CC2)=O)[nH]nc2ncnc(O)c12 49046,C1(CC)CCC2CC1C2(C)C.c1(C(=O)NCCC(=C)C)ccc(C)n1C 49047,CN1C(=O)CCC1C(=O)NCC1CCCC(CNC(=O)Cc2csc(=N)[nH]2)C1 49048,C1(S(C)(=O)=O)(C(=O)NCC(CN(C(=O)Cn2cccnc2=O)CC)(C)C)CC1 49049,N1(CC)CCC(NC(C2(CCC(=O)NC(=O)CN(CC(C)(C)C)C)CCC2)=O)C1 49050,C(=O)(CCCCCN(C)C)NC(C(N1CC=C(C)CC1)=O)CN(C)C 49051,c1(C(=O)NC(C2(O)CN(C(=O)CCN3CCCCCC3)C2)C)nnc(O)cc1O 49052,C(C(=O)N1CC(C2CCCO2)(NC(=O)CCCCSC)C1)(C(C)C)SCC 49053,C1(NC(=O)C=CC=C(Cl)Cl)CCC(NC(=O)CC(=O)Nc2ccc(Cl)cc2)CC1 49054,N1(C(C2C(=C)CC2)=O)CCCC(C2CN(C(c3nc[nH]c3C(C)(C)C)=O)C2)C1 49055,C1(C(=O)NCC2(C(N)=O)CN(C(C=CCCC=C(C)C)=O)C2)CCC(=O)N(C)CC1 49056,c1(CCC)ccc(C(N2CCC(CCOC)(NC(=O)OC(C)(C)C)C2)=O)cc1 49057,C(=O)(C1=CC(O)CCC1)NC1CCN(C(C2CC(C)(C(=O)OC)C2)=O)CC1 49058,Cc1csc2c(NCC3CCN(C(c4cc(Cl)cc(Cl)c4O)=O)C3)ncnc12 49059,c1(CN2CCN(C(=O)CCc3cccc(F)c3)C3C2C3)cccc([N+](=O)[O-])c1Cl 49060,C1(NC(c2cn(CC)nc2C2CC2)=O)CCN(C(=O)Cc2ccns2)CC1C 49061,N1(CC(N2CCC(NC(c3ccoc3Cl)=O)C(O)C2)=O)Cc2ccccc2C1 49062,c1(CNC(c2cnc(Br)n2C)c2n(CCC)nnn2)cccc(-n2ccnc2)c1 49063,c1(C(N(C(C(=O)NCCCCC=C)CC)C)=O)cccc(CC)c1 49064,N1(C(c2c(N)ccc(CC)c2)=O)CCC2CN(C(=O)CC3(C)CC3(F)F)CCC12 49065,N1(C(Cn2c(C)ccn2)=O)CC(CCNC(c2occc2F)=O)OC(C)C1 49066,c1(NC(N2CC(CC3CCCC(Oc4c(C)scn4)C3)C2)=O)cc2c[nH]cnc-2n1 49067,Cc1c(C(N2CCC(C(C)(C)C)(CNC(c3nocc3Cl)=O)C2)=O)nnn1C 49068,c1(C(=O)OC)ccc(C(=O)NC(C)CCNC(c2cn(C)c(C)n2)=O)cc1 49069,C(=O)(C(C)(C)C(C)(C)O)NC1(CCCCNC(C2N(C(C)C)CCCC2)=O)CC1 49070,C(=O)(C(C)(C)S(=O)(=O)C1CC1)N1C2CC(NC(CC(CC)(F)F)=O)C(CC2)C1 49071,c1(OC(C)C)ccc(F)c(S(=O)(=O)N2CCC2NC(c2cccc(F)c2)=O)c1 49072,N1(C(C(C)C2CCC2)=O)CC2CC(NC(c3ccnnc3Cl)=O)CC2C1 49073,C1(C(=O)NC2(CC=C)CN(C(C3(CF)CC3)=O)C2)CCCCC1C1CC1 49074,Cc1nn(C)c(=O)c(C(=O)NCCCC(C)NC(c2csc(Cl)c2)=O)c1C 49075,CC1CC(CCNC(c2ncoc2-c2ccco2)=O)CCN1C(=O)COCCF 49076,C(=O)(C(F)CCC(C)C)NCCCCNC(CC(CC)OC)=O 49077,C1(CC)CN(C(=O)C(O)C(F)(F)F)CCC1NC(=O)Cc1cc[nH]n1 49078,N1(C(C(C)=C(C)C)=O)CCC2(CCN(C(=O)C(C)(C)C(F)F)C2)C1 49079,C1(NC(c2c(C)scn2)=O)CCCC(N(C)C(C2CCC(C)CC2)=O)C1 49080,C1(C(=O)NC2CC3C=CC2C3)CCCN(C(=O)CN2CC(=O)NC2=O)CC1 49081,c1(CC(N2CC(CCNC(c3cnc(C)s3)=O)C2)=O)ccc(C(C)C)c(F)c1 49082,c1(C(=O)NC2(C)CCN(C(C3CC(C4CC4)=NO3)=O)C2)csc(=NC2CC2)[nH]1 49083,Cc1cnc2cccc(C(N3CC(NC(=O)COCCCF)CC(F)C3)=O)n12 49084,CC(C)(C)CCC(N)CNCc1cnccc1Cl 49085,C(=O)(CCCS(C)(=O)=O)NCC1(F)CC(NC(C(c2c(C)cccc2)C)=O)C1 49086,c1(OC)cc(F)ccc1-c1cc(CCN)ccc1F 49087,N1(C(CCCO)Cc2ccccc2)CCc2cc(CC3CCCC3)ccc21 49088,CC1=C(C(=O)N2CCC(NC(=O)CC3CCCC3)C(CO)CC2)CCS1(=O)=O 49089,C1(C#N)(C(=O)OCc2cc(C)c(Cl)cc2)CCCCCCC1 49090,c1(CC(=O)NCCOC2CCN(C(C(C)=CC)=O)C2)nn(C)cc1Br 49091,Cc1cn(C)cc1C(=O)NCC(C(=O)NCCC(=O)NC1CC1)N(C)C 49092,N1(C(Cn2c(C)nc(C)n2)=O)CCC2CCN(C(C3CC3C#N)=O)CC2C1 49093,C1(NC(c2c(CC)cno2)=O)CCN(C(=O)Cc2ccncc2Cl)C12CCC2 49094,C(=O)(C1=NN(C(C)C)C(=O)CC1)N1CC2C(C#C)(CC2)C1 49095,CC(Cc1cccnc1)C(=O)NCCC(C)N(C)C(C1CCCCO1)=O 49096,N1(C(c2cnc(CC)nc2O)=O)CCC2CCN(C(=O)CCNC(C)=O)CC2C1 49097,c1(OC)ccc(C(=O)NCC2COCC2NC(C2CN(C)CCO2)=O)cc1Cl 49098,CCC(C(=O)NC(C1(C(N2CC(COC)C3(CC3)C2)=O)CC1)C)C(C)C 49099,C(C(=O)NOCCN(C)C)(C1(O)CCC1)NC(C(C)C1CCCC1)=O 49100,c1(CN(C(=O)NC(c2ccc(C(C)C)cc2)C)CC)onc(C)c1CO 49101,C(=O)(CC(C)(C)C(F)F)NC1C(NC(C(C)S(N)(=O)=O)=O)CCC1 49102,CN1CCN(C(c2cc3occc3s2)=O)C(CNC(c2ccc(O)c(N)n2)=O)C1 49103,Cc1nc(O)[nH]c1C(=O)NC1(CCNC(=O)Cc2csc(N)n2)CCC1 49104,N1(CC(=O)NC2CCC(NC(C3CCC(CC)O3)=O)C2)CCC(=O)NC1=O 49105,C#CCCCCCC(=O)N1CC(C)(C)CCC1CNC(c1cnn(C)c1Br)=O 49106,N1(C(C2CC=CC(NC(C=NOC)=O)C2)=O)CC2CCC(C1)N2C(C)=O 49107,c1(C(=O)NCC(C)N(C(C(C)NC(=O)OC)=O)C)c(C)nn(C)c1OC 49108,c1(CN2C(C(=O)Nc3cc(C(=O)OC)cc(Cl)c3)CC3CC32)c(F)cc(O)cc1F 49109,Cc1cnn(CC(=O)NC2CCC(N(C(=O)CCC3CCCCC3)C)C2)c(=O)c1 49110,c1(NC(C(C)(N(C)C(c2ccnnc2)=O)C2CC2)=O)ccc(O)c(=O)cc1 49111,c1(C(=O)NC2CN(C(C(C=CC)O)=O)CC2O)cnc2c(c1)COCC2 49112,C(CC(=O)N1CC2CC2(CO)C1)(C(F)F)NC(CC1C=NN(C)C1=O)=O 49113,C1(CNC(c2cc(C(=O)OC)no2)=O)CN(C(=O)Cc2cc(Cl)n(C)n2)CCCO1 49114,c1(CC)cc(C(=O)N(CC(C)(C)C(=O)NC(C)(C)CC2CCCC2)C)nn1C 49115,C(C)(CCC(=O)N1CC(O)(CNC(C2CC(=O)N(C(C)C)C2)=O)C1)SC 49116,C(=O)(CC(C)P(C)(C)=O)NC1C(CNC(C=C(C)c2cnn(C)c2)=O)COC1 49117,C1(CC(=O)NCCOCCNC(C(C)NC(CC)=O)=O)C(=O)NN=C1C 49118,C(=O)(C(C)C(F)(F)F)NCCC=CC=C.C1(=O)C(C)COCCN1 49119,c1(C(N2CC3C(CNC(CC=C(C)C)=O)C3C2)=O)ccc2nn[nH]c2c1O 49120,C1(CC)CN(C(c2cnc(O)c(F)c2)=O)CCN1C(=O)CCc1cncnc1 49121,N1(CC(=O)N(CC(O)CNC(=O)CCCC2CCCCC2)C)CCCOC1=O 49122,C(=O)(CC(CC(C)C)NC(=O)CC1CCC(C)(C)O1)NC(CCOC)CO 49123,C1(C(=O)NC23C(CN(C(c4cc(C)[nH]n4)=O)C2)C3)CCc2ccc(F)cc2C1 49124,c1(C(=O)NC(CC)CNC(c2cscn2)=O)cc(N)c(N)cc1F 49125,N1(C(CCN(CCCCC)CCC)=O)CCN(C(C2CC2F)=O)CC1C1CCC1 49126,c1(OC)ccc(CC(N2CCC(C(C)NC(C34CCC(C3)OC4)=O)C2)=O)nc1 49127,c1(C(N2CCN(C(C3CCCSC3)=O)CC3(CC3)C2)=O)cc([N+](=O)[O-])cnc1O 49128,CC(C)CC(O)C(=O)N(CCCNC(C1CC(=O)N(C2CCCC2)C1)=O)CCO 49129,C12(NC(c3ncn(CC)c3)=O)CCCC(NC(c3ccsc3C)=O)(C1)C2 49130,c1(C(=O)NCC2(NC(COCC)=O)CC3CCC2C3)ccc2snnc2c1 49131,C12(C(=O)NC(C3CCCO3)CC)CCC(CC1)N(C(=O)C(=CC1CCCC1)C)C2 49132,C(=O)(CCCS(=O)(=O)NC)NC1C2CCN(C(C(C)OCCCC)=O)CC21 49133,S(=O)(=O)(CC(=O)NCC1CC(C)CO1)N(CCC1CCN(C2CC2)CC1)CC 49134,C1(C(=O)OC)CC(n2cc(C3(O)CC3)nn2)CN1C(=O)CCC1CCCCC1O 49135,c1(OC)cccc(C=CC(=O)NC(C)CC(C)NC(c2ccc(C)nc2C)=O)c1 49136,c1(C(=O)NC2CC(CC(=O)NC(C=C)(C)C)C2)cn(C)nc1SC 49137,c1(C(=O)NCCCCN(C(C2C(C(=O)NCC#C)C2)=O)C)cccc(CC)c1F 49138,c1(C(C)C)nc(C(N2CC(CO)(NC(C3CCC3CF)=O)C2)=O)co1 49139,C(C)(C)(CCC(=O)N1CCN(C(c2sc(C)cc2Cl)=O)C2CC12)OC 49140,c1(C(=O)NCC=CCNC(CC2CCC(C#N)C2)=O)cccc([N+](=O)[O-])c1 49141,c1(C(=O)NC2(OC)CC2)nc2ccccc2cc1Cl.C1(=O)C(C)(C)N1C1CC1 49142,C1(C2(O)CN(C(=O)CC3(CN(C)C)CC3)C2)(CNC(CCCN(C)C)=O)CC1 49143,C1(C=O)CCCN1C(=O)CC1(C)CC1.c1(C(=O)NCC=C)ccn(C2CC2)n1 49144,CC1(C)C(CNC(c2ccnc(O)c2)=O)CCN1C(=O)CCNc1ncccn1 49145,C1(NC(c2cnc(OC)nc2)=O)CCN(C(=O)Nc2cnccc2C#N)CC1F 49146,C1(C(=O)NCC2(C(N)=O)CC2)C=CCCN1C(C1CC1c1ccccc1)=O 49147,N1(C(C2CCC(C)(C)C2)=O)C2CCC1CC(C(=O)NCCCS(C)(=O)=O)C2 49148,c1(C(N(C)CC2N(C(c3c(C)nsc3)=O)CCC2)=O)cc(C(F)(F)F)cc(Cl)c1 49149,C(N=c1[nH]ccn2cnnc12)c1c(OC(F)F)ccc(F)c1 49150,C1(CNC(c2cncnc2)=O)CCN(C(c2cnc3ccnn3c2)=O)CC1(F)F 49151,C=Cc1cnn(C)c1C(N1CC2CC1CC2NC(=O)C(=O)C(C)(C)C)=O 49152,CC1CC(C(=O)NCCNC(=O)CN(C)C)CN1C(=O)C1CC1.C1(=O)CN1 49153,Cc1ccc2c(c1C)OCCC2NCc1cc(F)ccc1C#N 49154,C(CCC(O)C(=O)Nc1ccc(C)nc1)NC(C(C)=C1CC1)=O 49155,n1(CCCC)ncnc1NC(c1cc(C)sn1)=O 49156,c1(C(C)C)ccc2cc(C(=O)N(CC(C)NC(C3CCO3)=O)C)[nH]c2c1 49157,C1(C(N2CCC(C(C)C)C2)=O)CC(F)CCN1C(=O)COCC(F)F 49158,C#CC1CN(C(=O)CCOCCCOCCCCC)CC1OC 49159,N1(C(c2cc(C)oc2)=O)CCC2(NC(c3n[nH]cc3Cl)=O)CCCC12 49160,c1(C(C)NC(CSCCC)=O)nocc1C(=O)NCC(F)CO 49161,c1(C(=O)OC)[nH]c2ccc(NC(=O)Nc3c(Cl)ccnc3[N+](=O)[O-])cc2c1C 49162,C1(C(NOCCN(C)C)=O)CC(NC(C2(c3ccoc3)CC2)=O)CCO1 49163,N1(C(C2C(C)(C)CO2)=O)CCC2(CCC2CNC(c2cncnc2)=O)CC1 49164,CC(C)CC(F)(F)C(=O)NCC(C)(C)CN(C)C(C1CC1C)=O 49165,CC(C)CCCOC(C(=O)N(CCCN1CCCC1)C)C1(O)CCC1.C(C)=O 49166,C1(OC)CCC12CC(C(N1CCCC(NC(C3CCC3)=O)C1)=O)C2 49167,c1(C(=O)NCC23C(NC(COCCOC)=O)CC(CC2)C3)cnc2n1CCCC2 49168,CC(C)(C(=O)NCC1(NC(=O)CC2(n3cccn3)CC2)CC1)c1ccns1 49169,C12(C(=O)NCC(N(C)C(c3c[nH]nc3C(F)F)=O)C3CC3)CCCC(C1)OC2 49170,Cn1nc(CC(=O)NC(C)(CNC(C2CC23CCC3)=O)CO)cc1C(F)(F)F 49171,c1(C(CNC(C)C(=O)OCCc2nc(-c3ccccn3)no2)=O)ccccc1Br 49172,N1(C(C(C)C2CCCC2)=O)CC2CCC2(CNC(c2cc(Cl)ns2)=O)C1 49173,c1(C(=O)NC(CNC(c2c(C)cno2)=O)C(C)(C)C)c(Cl)ccc2ccoc12 49174,C1(C)(C(N(CCOC)CCNC(n2ccnc2)=O)=O)CCOC1C 49175,c1(C(=O)NCCCCC2CN(C(C3CCCC(C)C3)=O)C2)ccc2n[nH]cc2n1 49176,c1(CSCC)cnc(Cl)n1C.C1(C)(C)C(c2nnnn2CC2CCOC2)N1 49177,n1(CC)nncc1C(=O)NCC(O)C(=O)NCC(CO)N(C)C 49178,N1(C(C(C)=C(C)C)=O)CC(C)(C)OCC1CNC(c1cccc(O)c1)=O 49179,C1(C(=O)NCC2(F)CC(NC(c3cnc(C)nc3)=O)C2)CCC(C)(C)CO1 49180,C=CCC(C(=O)NN1CCN(CC(O)Cc2ccccc2)CC1)=C(C)C 49181,N1(C(C(CC)C#N)=O)CC(C(=O)NC(CC(=O)OC)C2CC2)C(C)(C)C1 49182,C1(c2c(OC)cccc2)CCCN(C(C)C(=O)OC(C)(C)C)CC1 49183,n1(CC=C)nnnc1C(c1nccn1CC=C)NCc1ccc(C(F)F)o1 49184,C(=O)(C(C)(C)CCCF)NC(CCCCNC(C(C(C)C)OCC)=O)C 49185,CC12CCC(C(=O)NCC3CC3NC(=O)C(C)(C)c3cnc[nH]3)(CC1)CO2 49186,C1(N(C(CC(C)C)C)C(=O)OCC2CCC2)C2CN(CC(=O)O)CC12 49187,N1(C(C2(C)COC2)=O)CCC2CN(C(=O)CC3CC4(CC4)CO3)C2C1 49188,C1(C(N2C(C(C)O)CC2)=O)CCN(C(C2(C)CNC(=O)C2)=O)CC1(C)C 49189,c1(NC(N2CC(C#C)(N(C)C)C2)=O)ccc(Br)c2nccn12 49190,c1(CC=C)ccccc1C(N1CCCC(CN(C)C(C2CCCN2C=O)=O)C1)=O 49191,CCCCCOCC(=O)NC(C1CCOC1)CNC(=O)C1CC1 49192,C1(CC(=O)NC(CCNC(C(C)O)=O)C)CC(F)(F)C1 49193,C1(CNC(CC(C)(C)C)=O)CC2(CCN(C(c3ccc(N)c(Cl)c3)=O)C2)CO1 49194,N1(C(CC(=O)OC(C)(C)C)=O)CCC(NC(C2CC2(F)F)=O)C12CCCC2 49195,CCCC(C)CC(=O)NC1(C(=O)NC2CCCNC2=O)CCOCC1 49196,C(=O)(C(O)C(C)(C)C)NC1(C(=O)NC(C)CC2CCCC2)CC1C 49197,C12CC(C1)CNCCN2C.C1(C2CC2)CCNC(=O)N1.C(C)(C)(C)OC 49198,C(=O)(C1=CS(=O)CCC1)NCCCN(C(C)C)C(C1CCCN1N=O)=O 49199,CCC(C)CCC(=O)NCCCNC(=O)CC(C(F)F)c1ccc(F)cc1 49200,c1(C(=O)NCC2(NC(CC3C(C)CCC3)=O)CC2)ccc2c(c1)COB2O 49201,c1(NC(=O)C(c2ccc(F)cc2)N2CCC(C(=O)O)CC2)ccc2c(n1)CCC2 49202,N1(C(C(c2cnn(C)c2)C)=O)CCC12CN(C(c1cc(O)cc(Cl)c1)=O)C2 49203,c1(OCCC#C)ccccc1C(C)N(C)Cc1sc(Br)nc1C 49204,CP(C)(=O)c1ccc(C(=O)NC2CCN(C(=O)C3=COCCC3)C23CC3)cc1 49205,C1(NC(CNC(C=NOC)=O)=O)CCC=CCC1 49206,Cc1ccc(S(=O)(=O)NCC(C)C)cc1NC1CC1C1CCOCC1 49207,C1(CNC(C2(C(=O)OCC)CC=CC2)=O)CN(C(C2SCCS2)=O)CC12CCC2 49208,C=Cc1ccc(C(N2CC(N(C(=O)CSCC(=O)OCCC)CCO)C2)=O)cc1 49209,N1(C(c2c(CC)cns2)=O)CCOCC(C(N2CC(C)(N(C)CC)C2)=O)C1 49210,CN1CCCC(CCC(=O)NCC2CCN(C(C3CCC3)=O)CC2)C1 49211,c1(NC(=O)NC23C(CN(C(C4CN(CC)C(=O)C4)=O)C2)C3)cccc(C)c1C 49212,C#Cc1ccc(CNC(C2(CC)CCCN2NC(=O)C(C#N)CCC)=O)cc1C 49213,C(C(C)CC(=O)N(C1CC1)C1CC1)NC(CC=CCC)=O 49214,c1(C(=O)NC(CN(C)C)C(=O)NC2CCC(C)(C)C2)ccc([N+](=O)[O-])o1 49215,N1(C(c2cc(CC)nn2C)=O)CC(C(=O)NC(C)(CC)C2CC2)C(C2CC2)C1 49216,C1(C(=O)NC2C(CNC(C#CC(=O)N(C)C)=O)C2)OCCN(C)C1=O 49217,Cc1cc(C(N2CC3C(CNC(c4nccn4C4CC4)=O)C3C2)=O)n(C)n1 49218,CCC(C(F)(F)F)NC(C1CCCCN1C(=O)COCC(F)(F)F)=O 49219,CC(C)C(C(=O)N1CCC(NC(C2CC3(CC3)C2)=O)C1)c1noc(C2CC2)n1 49220,C1(NC(CC(C)NC(N)=O)=O)CC(NC(C2(C#N)CC2)=O)CC1O 49221,c1(C(=O)OCC(=O)NCC23CC2CN(C(c2ccco2)=O)C3)ccc2scnc2c1 49222,c1(OC)ccc(C(=O)NC(C2CCCN2C(c2coc(O)n2)=O)(C)C)c(O)c1 49223,CCC(C)(C)C(C)CC(=O)N1CCC(N(C(=O)CC(=O)NC(C)C)C)CC1 49224,C1(CCC)CN(C(C23CSCC2C3)=O)CC1NC(C1C=CC1C(=O)OC)=O 49225,C1(C(=O)NCc2nc(-c3ccc(C)cc3)oc2)CN(C)CC(C)O1 49226,N#Cc1ccc(C(N2CC(CCO)(NC(=O)C=Cc3cscn3)C2)=O)s1 49227,C1(NC(=O)CC2CCCC(=O)N2)CC(C(=O)NCC2CCCC3(CC3)C2)=CC1O 49228,c1(C2C(C(N3CCCN(C(=O)C=CC(F)(F)F)CC3)=O)C2)cccc2c1OCCO2 49229,C1(NC(=O)CCCC2CCCC2)CCCC(C(=O)NCCC(=O)N2CCCC2)C1 49230,c1(C(=O)NCC(C2CC2)OC)cc(O)nc2c1CN(C(=O)Cn1cccn1)CC2 49231,C1(NC(C=NOC)=O)CCC(O)CN(C(=O)CC(C(F)F)n2cccn2)C1 49232,C(=O)(CC(C)CCC)NC1(CNC(C2CCCN(C(CC=C)=O)C2)=O)CC1 49233,CCC(CC(=O)NC(CC1CC1)C(=O)OC)NC(=O)CCc1cn(C)nn1 49234,C1(C(N2CC(CNC(=O)Cn3cc(Cl)cn3)C(C)C2)=O)(OC)CCC(C)CC1 49235,CCCCC(C(=O)NC)NC(=O)C(CNC(c1nocc1C)=O)CC1CCCC1 49236,C1(NC(C2N(C(C(C)(C)C3CCOC3)=O)CC2)=O)CCC2CCCC12 49237,c1(OC)cccc(C(=O)NCCSc2ccc(F)cc2)c1OC(=O)CC(F)(F)Cl 49238,c1(COC)nc(NCc2ccc(Br)s2)cc(=NC(C)c2cscn2)[nH]1 49239,c1(C(=O)NCC2N(C(C3(OCC)CC3)=O)CC2)ccnc(CC(F)(F)F)c1 49240,S1(=O)(=O)c2ccc(c(C#N)c2)N1.N1(CC(C)SC)CCCC(C)C1.C1C(=O)N1C 49241,c1(OCC(Cc2ncn(C)n2)O)ccc(-n2cccn2)cc1 49242,c1(CC(=O)NC2CCN(C(=O)COc3ccsc3)C2)ccn(C2CCC2)n1 49243,N1(C(c2cc(-c3ccc(Cl)s3)on2)=O)CC2(CCN(C(C3(C(F)(F)F)CC3)=O)C2)C1 49244,C1(C(=O)NCC2CC(NC(c3ccn(C)n3)=O)C(O)C2)Cc2c(F)cccc2O1 49245,C1(C(c2nnnn2C2CC2)NC(=O)CCCNC(C)C)(OC)CCCC1 49246,N1(C(COCC#C)=O)CC2(CC1CNC(=O)Cc1cc(C)[nH]n1)CC2(F)F 49247,c1(C(N2CC(OCC(=O)OC)C2)=O)cc(C(C)C)[nH]n1 49248,C1(C2CCCN(C(c3csc(=N)[nH]3)=O)C2)(NC(CCC(=O)NCCC)=O)CC1 49249,C(=O)(CCCCCC)NCCC(CNC(C12OCC(COC)(C1)C2)=O)OC 49250,c1(C(=O)NC(CC)CNC(=O)C(C)c2cccs2)ccc(F)cc1OC 49251,C(=O)(CCC(C(C)C)NC(=O)CC(C)(C)CC)NC1CN(CC)CC1C 49252,CC(C)CC(F)(F)C(=O)NC1CC1CNC(c1ccc(Cl)c(F)c1N)=O 49253,O=C(CC(C(F)F)NC(C1(F)CC1)=O)NCC1(F)CCOCC1 49254,CN1CCC2C(CCN2C(c2[nH]ccc2CNC(=O)CC2CC3(CC3)C2)=O)C1 49255,C1(C(N(CCCNC(C(c2ccccc2)N(C)CC)=O)CCO)=O)CCCC1F 49256,C(=O)(N1OC2CCC1CC2)C1(F)CCN(C(c2cc(CO)ccn2)=O)CC1 49257,C1(NC(c2c(C)cno2)=O)CN(C(C2CC2c2ccccc2F)=O)CCC1C 49258,C1(C2CCC2)(C(=O)NCCOCCOCCNC(c2scc(C)c2)=O)CCC1 49259,C(=O)(N=c1[nH][nH]c2c1CN(C(c1cccs1)=O)C2)c1cccc(C(C)C)c1 49260,C(=O)(CCC(F)(F)F)NCc1ncc(C(N(CC)Cc2cccnc2)=O)cn1 49261,C(=O)(C1CCc2ccccc21)OC(=O)C(F)(F)F.C12(CCC13CCC3)N(C=O)C2 49262,N#Cc1c(C(=O)NCC2(O)CCCN(C(=O)C(=O)NCC(F)F)C2)cccc1F 49263,c1(NC(CC2N(C(CC(C)CN(C)C)=O)CC2)=O)cn(C)ccc1=O 49264,N1(C(c2c(CCC)[nH]cc2)=O)CCC(C)(CCNC(c2cn(CCO)nn2)=O)C1 49265,Cc1cc(F)c(C(c2nnnn2C2CCCCC2)NC2CCCC2)c(Br)c1 49266,c1(OC)ccc(CC(=O)N(CC2CCCN(C(=O)Cc3scnc3C)C2)CC)cn1 49267,C(=O)(CCS(N)(=O)=O)NCC(C)(C)OCC(=O)N(C)Cc1nccn1C 49268,C(=O)(CCCCC(C)(C)C)NCC(C)(C(C)C)NC(CCC(=C)Br)=O 49269,CCCCC(CN(C)C)C(=O)NC(CC(=O)NCC(C)C(C)(C)C)C(C)C 49270,C1(C(N(C2CCN(C(c3snc(O)c3Cl)=O)C2)C)=O)CCc2c[nH]nc2C1 49271,Cc1cc(O)cc(O)c1CC(=O)NC1C2CN(C(c3cc(C(C)C)no3)=O)CC12 49272,Cc1nc2sccn2c1C(=O)NC1CN(C(c2cc[nH]c2)=O)CC1C 49273,C1(C(=O)NC(C)C(=O)NO)CCC(C)(C)N(C(=O)C(C2CCCCCC2)O)C1 49274,C(=O)(CCC(=O)N(C)C)NC(C)C(c1cccc(O)c1)NC(c1nccs1)=O 49275,N1(C(CC(C)CF)=O)CCN(C(=O)CCC2OCCO2)C(CS(C)(=O)=O)C1 49276,c1(C(=O)NC2(C)CC(C(=O)Nc3cnc(OC)nc3)C2)nccc(C)c1F 49277,c1(N(C(c2ccco2)=O)CC2N(C(C=CC=CC)=O)CCC2C)cc(Cl)cc(Cl)c1 49278,Cn1cc(C(F)=CC(N2CC(NC(=O)CNC3CC3)C3(CC3)C2)=O)cn1 49279,C(=O)(C(CC(C)C)C(C)C)NCC1(C(=O)OCC)CCC1.N12CCOC(C1)C2=O 49280,c1(OC)ccc(NC(C2CC23CCN(C(c2cnnc(O)c2)=O)C3)=O)c(CO)c1 49281,c1(C(N2C(CNC(Cn3ncc(C)c3)=O)CC2)=O)cncc2cnccc12 49282,C12(C(N3CCC(=CCNC(CS(CC)(=O)=O)=O)C(OC)C3)=O)CCC(O)(CC1)CC2 49283,CCCCCC(F)C(=O)N1CCC(COC)(NC(C23CCC(C2)OC3)=O)C1 49284,C1(CC)CC(NC(=O)CC(C)(C)NC(C2CC(C(C)C)C2)=O)CCO1 49285,C1(NC(C2CC(N(C)C)C2)=O)CC2CC(NC(=O)COCc3nccn3C)C1C2 49286,C#CC1CCCN(C(=NCCOCC)NCC(CC)CC)C1.C1(C)CC1 49287,N1(C(C(C(=O)OCC)F)=O)CCN(C)C(C(=O)NCC2=CCCC2)C1 49288,c1(C(N2CC(c3cn(CCC(=C)C)nn3)OCC2)=O)ccc(C2CC2)c(F)c1 49289,c1(C(C)OC)nc(CO)cs1.C1CCCCCC2N(CCC2)C(=O)N1 49290,C(=O)(NNC(=O)NC(F)(F)CF)c1c(C)ncs1 49291,N1(C(c2cnc(C(F)F)s2)=O)CC2=C(C1)CN(C(C1OC3CCC1CC3)=O)C2 49292,C1(C)(C(N2CCC(N(CC#C)C(C3CCOC3CC)=O)CC2)=O)CCCNC1=O 49293,N1(C(C23CC(C)(C2)C3)=O)CCC2CCN(C(c3cc4c(cn3)CCCC4)=O)CC12 49294,c1(C(N2CC3CCN(C(c4c(OC)nsc4)=O)CC32)=O)nccc2ccccc12 49295,C(C)(CCCCNC(=O)C(C)c1cccs1)NC(C1N=C(C)SC1)=O 49296,C1(CNC(C(C)OCC)=O)CC2(CCN(C(=O)Cc3ccnc(Cl)c3)CC2)CO1 49297,c1(C(=O)NC(CCOC)CNC(C2(C)CC=CC2)=O)ccc2cnn(C)c2c1 49298,CC1(C(=O)NC2CC3(C2)CC3C(N2CC(CO)C3(CC3)C2)=O)CC2C=CC1C2 49299,CON(C(=O)C1CCCN1C(=O)C(C)CC1CCCC1)C1CCC1 49300,c1(C(=O)NCC23OCC(NC(CNC(=O)NC)=O)(C2)C3)cc(C(F)F)ccc1Cl 49301,Cn1ccc2c(C(N3CC4OCC(NC(C5CC=CC5)=O)C4C3)=O)ncnc12 49302,N1(C(c2cnc(CCC)s2)=O)CCN(C(C2CCCC2CC)=O)CC1 49303,C1(CNC(C2CC(C)SCC2)=O)CCCC2CN(C(c3ccncc3Cl)=O)CC12 49304,n1(-c2cn(SCC)nc2)nc(CC2CC2)nc1-c1coc(NC(C)=O)n1 49305,C(=O)(CCCCC(C)CC)N(CCCNC(C(CC)CC)=O)C(C)C 49306,C1(NC(C2(OCC)CCCC2)=O)CCN(c2cc(NC(C)=O)nc(Cl)n2)CC1O 49307,Cc1ccnc(C(=O)NCC(O)CCNC(C2CCCCCN2C)=O)c1F 49308,Nc1ncccc1C(N1CC2C(CNC(c3cc(=O)cc[nH]3)=O)C2C1)=O 49309,C(=O)(C(O)CC(C)(C)C)N1CCCC(CN(C(CCSc2nc(C)[nH]n2)=O)C)C1 49310,c1(NC(C=C(COC)C)=O)cccc(NC(=O)Cc2coc(Cl)c2)c1 49311,C1(NC(C2C(C(=O)OC)C2(C)C)=O)COC2(C1)CN(C(c1cc(C#N)c[nH]1)=O)C2 49312,N1(C(C(CC=C)C)=O)C2CCC1CC(NC(C1(SC)CC1)=O)C2 49313,c1(COC)cc[nH]c1C(=O)NCC1COCC1NC(=O)CCC1CCOC1 49314,C1(C(N2CCN(C)CC2)=O)CN(C(c2cc(C#N)c[nH]2)=O)CCC1(C)C 49315,C1(C#N)(C(=O)NCc2cn(C(C)C(N3CCC(N(C)C)C3)=O)nn2)CC(F)(F)C1 49316,CN=c1nc(C(N2CC(NC(C3CCCN3C3CC3)=O)CC2C)=O)cc(C)[nH]1 49317,N1(C(c2c(C)ocn2)=O)CCCC(CO)(NC(C2CCC2(C)C)=O)C1 49318,CCC(CC)CC(=O)N1CCCC1CCC(=O)NCc1ccc(C)cc1F 49319,C1(CNC(=O)CC(F)F)COCC2(CCN(C(C3CC4CCC(C3)C4)=O)CC2)O1 49320,c1(C(N2C(C3CCN(C(CC)=O)CC3)CCCC2)=O)cc([N+](=O)[O-])ccc1NC 49321,Cc1cnc(Cl)c(CC(=O)NCc2cccc(CN(C)C(C3CC3F)=O)c2)c1 49322,N1(C(CSCCC)=O)CC2CCN(C(=O)CN3CCC(C)(C)C3)C(C2)C1 49323,C(=O)(CS(=O)(=O)C1CC1)NC1CCCC(NC(=O)COc2cccnc2)CC1 49324,N1(C(C(C)OCC)=O)CCC2C(NC(c3sc(C)nc3-c3ccccc3)=O)CC12 49325,C1(C(N2C(CNC(CC3(C)CC(F)(F)C3)=O)CC3CC32)=O)CCc2nnnn2C1 49326,c1(SC)cn(C)nc1C(N1CCCC(CN(C)C(C2(C)CC2C)=O)C1)=O 49327,N1(C(c2ccc(C(=O)NC)cc2)=O)CC2CN(C(c3cc(C)ns3)=O)CCC12 49328,N1(C(Cc2cccc(COC)c2)=O)CCC(NC(C2CCCC23CC3)=O)CC1C 49329,c1(CNC(C23CC2CN(Cc2cccc(F)c2O)C3)=O)cc(F)ccc1[N+](=O)[O-] 49330,C(=O)(CCCCCN=[N+]=[N-])N(C1CN(C(C2CC(C(F)(F)F)C2)=O)C1)C 49331,Cc1ccc2cc(C(=O)NC3CC(CO)N(C(=O)CC(C)O)C3)cn2c1 49332,C1(NC(COCCCCC)=O)CC(C)(NC(C2CCCN2C2CCCC2)=O)C1 49333,CC(C)(C(=O)NCc1nnc(O)o1)NC(C12CCCC1C2)=O 49334,N1(C(COCCN(C)C)=O)CC=CC1CNC(=O)CCN1CCC(F)C1 49335,Cc1ccn2ncc(C(=O)NC3CN(C(=O)CC4CC=CCC4)CC3(C)C)c2n1 49336,c1(C(=O)NCC(CN(C(CN2C(C)CC2)=O)C)(C)C)n[nH]c2nccc(Cl)c12 49337,CC1CN(C(C2(F)CCOC2C)=O)CC1NC(C1CCCN1N=O)=O 49338,N1(C(C(COC)NC(=O)Cc2cccs2)=O)CCN(C)C(=O)C1C 49339,c1(C(=O)NCCC(CCC)N2CCOCC2)c(SC)ccc(Cl)c1Cl 49340,C(CS(=O)(CCO)=NC(=O)c1ccc(-n2ccnn2)cc1)N(C)C(=O)OC(C)(C)C 49341,C(=O)(C1=CC(C)(C)C1)N(CCCNC(=O)C(C)OCc1cccc(F)c1)C(C)C 49342,C12(C(=O)OC)CC(C(=O)NCC3CCC(NC(c4ccn(C)c4)=O)C3)(C1)C2 49343,c1(C(N(C)CCC2CCCCN2C(=O)CCc2ccc[nH]2)=O)cnc2n1CCS2 49344,C1(NC(=NCCCSC)NCc2ccc(C)c(F)c2)CCOC2(CCOCC2)C1 49345,c1(NC(C2N(C(c3c(CCC)[nH]cc3)=O)C(C)CC2)=O)cccc(OC)c1Br 49346,N1(C(C(c2c(C)n[nH]c2C)C)=O)CCN(C(c2cc[nH]n2)=O)C(C2CCCC2)C1 49347,c1(CC(N2CC(C)N(C)CC2)=O)c[nH]c2ccc(-c3cncc(N(C)C)c3)cc12 49348,c1(CN(C2(C)CN(CC3C4(CC(C5C(C)=C5)C4)C3)C2)C)ccc(N)c([N+](=O)[O-])c1 49349,c1(C(N2C(C(C)(C)NC(C=CS(C)=O)=O)CCC2)=O)cccc([N+](=O)[O-])c1O 49350,C#Cc1ccc(F)c(C(N2CC3CCC2C(NC(c2cnn(C)c2N)=O)C3)=O)c1 49351,C1(CC)CCCCN1C(N1CCC(CNc2cnn(CC(F)(F)F)c2)C1)=O 49352,O=C(C#CC1CCCO1)NCC(c1ccc(F)cc1)NC(c1cc(Cl)no1)=O 49353,C1(N(C(C(CC)C)=O)C)CCCCN(C(C2CC=CC2)=O)C1 49354,C12(OC)CC(C(=O)NCC(C)(C)NC(c3cccc(F)c3)=O)C(C1)C2 49355,c1(C(N2CCN(CC(N3CCOCC3)(C)C)CC2)=O)n[nH]c2c1CCC(F)(F)C2 49356,c1(C(N2CCC(C(C)NC(c3nc(C(=O)O)co3)=O)C2)=O)c(O)cccc1Cl 49357,c1(C(=O)NCC2CC(Nc3ncnc4[nH]cnc34)C2)cc(=O)c2ccccc2o1 49358,c1(OCCC)ccc2cc1C2.C12(C)CCCN(C1)NC2=O.c1(CO)nccn1C 49359,C1(NC(C(CCC)OCC)=O)CCN(C(c2cc(C)n(C(C)C)c2)=O)CC1F 49360,N(C1CCOc2ccccc21)(C(CNC1CCOC1=O)=O)CC#C 49361,CC1C(NC(c2n[nH]cc2C2CC2)=O)CCCN1C(=O)CN1CCCNS1(=O)=O 49362,c1(CC(C)C(=O)NCC#CCNC(C2CC3(CCCO3)C2)=O)ccc(C#N)cc1 49363,C1(C(N2CC(CNC(C=C(C)C)=O)OCC2)=O)CCN(C)S1(=O)=O 49364,c1(C(CCCOC)NC(=O)C(F)=C2CCCC2)cccc(F)c1 49365,Cc1cc(Cl)c(Br)c(C(=O)N(CCS(=O)(=O)N(C)C)CCO)c1F 49366,C=CC1(C(N2CCC(O)(C=C)C2)=O)CCN(C(C2CCC2(F)F)=O)C1 49367,N1(C(COCCCC)=O)CC2CCC1C(CNC(=O)CCCc1cnn[nH]1)C2 49368,N1(C(c2ncn(CC)n2)=O)CC(CNC(=O)C=Cc2ccsc2)C2(CCC2)C1 49369,c1(C(N2CCC(N3CCc4ccccc43)CC2)=O)cccc2nc(Br)sc12 49370,C1(C(=O)N(C2CC(SC)C2)C)(CC)CCCN1C(c1ccccc1O)=O 49371,n1(CC)ccnc1C=CC(=O)NCC12CC1CN(C(=O)CN1CCN(C)CC1)C2 49372,c1(OC)ccc(CCC(=O)NCC2CCC2NC(C2CC3C=CC2O3)=O)c(F)c1 49373,N1(C(c2c(OC)ccc(C)c2)=O)CCC2C(CCN2C(c2cccc(Cl)c2F)=O)C1 49374,c1(CCC)nc(C)c(C(=O)NCC2CCCN2C(=O)CCc2nc(C)no2)s1 49375,N1(C(C2(C)CCCCC2)=O)CC(CO)C2(CCN(C(C3COCCO3)=O)CC2)C1 49376,C1(CNC(C2(C)CCNC2=O)=O)CN(C(c2c[nH]nc2Cl)=O)C2(CCC2)C1 49377,c1(CC(=O)NCCN(C(=O)C(CCSC)N(C)C)CCC)cccc(O)c1 49378,C1(C(C)C)C(NC(=O)CCOc2cccc(F)c2)CCN1C(=O)CCCC1CC1 49379,N1(C(CC)=O)CCN(C(c2nncn2CC)=O)CC1c1cnn(C)c1 49380,C1(NC(c2c(CC)non2)=O)CCC(O)CC1.c12cc(n[nH]1)C(=O)N(C)C2 49381,Cn1cc(C=CC(=O)NC(Cc2cn[nH]c2)C(=O)NCc2ccc(Cl)o2)nn1 49382,N1(C(c2cc(C)c(O)nc2)=O)CCC=C(C(=O)N2CCCCC2C#N)C1 49383,C12(CN3C(C(=O)NC(c4ccc(N(CCCl)CC)cn4)=O)CC3)CC=CC(C1)OC2 49384,c1(NC)cccc(C(N2CCC(NC(c3cc(OC)n[nH]3)=O)C2)=O)n1 49385,CC12CCOC(C(N3CCC(C(F)(F)F)C(NC(C45CCC(C4)C5)=O)C3)=O)(C1)C2 49386,CCCC(CCO)NC(=O)CN(C(=O)C#CC(C)C)CC 49387,C(c1cccc(Cl)c1)=CC(=O)NC(C1CCN(C(c2cc(C)c(C)[nH]2)=O)C1)C 49388,N1(C(C=CCC)=O)C2CCC1CC(N(C)C(c1ccncc1Br)=O)C2 49389,S(=O)(=O)(c1ccc(C(N2CCC(C(C)NC(c3cc[nH]c3)=O)C2)=O)o1)NC 49390,c1(C(N2CCN(C(C=CCC)=O)CC2CS(C)(=O)=O)=O)ccc2ncccc2n1 49391,C1(C)(CNC(C2C(OC)CCC2)=O)CCN(C(=O)CC2CCC(=O)NC2=O)CC1 49392,C1(CC=C)(NC(=O)CC2CC2COC)CCN(C(=O)CSC(F)F)CC1 49393,N1(C(C(COC)OC)=O)CC(CC(N2CCC2(C)OC(C)C)=O)C2(CC2)C1 49394,c1(CNC(=O)CC2CCN(C(c3ccnn3CCO)=O)C2)cccc(CO)n1 49395,CC(C)C(O)CC(=O)NCC1CCN(C(=O)Cc2ccccc2OC(F)(F)F)C1 49396,C(C(CNC(=O)CN1CSCC1=O)C(F)(F)F)NC(c1c(C(C)C)nn(C)c1)=O 49397,Fc1cccc2c1CN(c1nccc(=NCCN3CCCS3(=O)=O)[nH]1)C2 49398,n1(CC(C)NC(C2CCC2)=O)cc(C(=O)NCCNC(C2CCC(=O)O2)=O)cn1 49399,c1(OCC(=O)NC2CCN(C(=O)CSc3cccnc3O)CC2)cc(F)cc(Cl)c1 49400,CCC(C)C(=O)NC(C1(O)CN(C(C2COCCO2)=O)C1)C 49401,c1(C(N2CC(NC(C(CCC)O)=O)C(OC)C2)=O)cnc2c(c1)CNC2=O 49402,c1(NCCC=CC=C)[nH]c(=NC2CC3C(C2)C3(F)F)nc2c1ncn2C 49403,CC(C)CCCC(C)NC(=O)CN1CCN(C(C2C=CC(=O)N=N2)=O)CC1 49404,N1(C(c2c(C)ocn2)=O)CCN(C(c2ccc(F)cc2O)=O)C2CCCC2(C)C1 49405,N1(C(C2(COC)C=CCC2)=O)CCCC(N(C)C(c2ncoc2C2CCC2)=O)C1 49406,CC1=C(C(=O)NC(CNC(c2ccc(C(F)(F)F)cc2)=O)CC(C)C)CCCO1 49407,N1(C(CCn2c(C)ncc2)=O)C2CCC(C2)C1CNC(C1COC2(CCC2)C1)=O 49408,N1(C(c2ncc(NC)nc2)=O)CC(C2CCCN(C(=O)C(C)(C)C(C)O)C2)C1 49409,N1(C(c2n(CC#C)cnn2)=O)CCC2C(C(=O)N(CCOC)CC)C2C1 49410,Cn1ccc(C(N2CC(C)(NC(=O)CC3(O)CCOC3)C2)=O)c1C1CCC1 49411,C1(NC(C2CC2F)=O)CCN(C(=O)C(C2CCCC2)C2CCCC2)CC1 49412,N1(C(C2CC(CC)C2)=O)CC2CC2(NC(=O)CNC(c2cccc(OC)c2)=O)C1 49413,C1(C(N2CC(C)C2C(=O)NCCCOCCCO)=O)CCC(C)(C)CO1 49414,c1(C(N2CC(NC(C3(OC)CCOC3)=O)C2)=O)cc2c(C)c(F)ccc2[nH]1 49415,N1(C(CCC2CC(OC)C2)=O)CCCN(C(c2cc(C#N)ccc2Cl)=O)CC1C 49416,Cc1cc(N(CC(C)Cc2ccccc2)C)cc(C(N)=O)c1 49417,C1(CNC(c2cn(C(C)C)nn2)=O)(CO)CCCN(C(C2CCCC(F)C2)=O)C1 49418,c1(NC(N2CC(C(C)NC(=O)CC3CCCO3)C2)=O)ccc(F)c(F)c1F 49419,c1(C(=O)NC2CC(CNC(Cc3c(C)nsc3)=O)C2)coc2c1CCCC2 49420,C1(C(N2CC(N(C(=O)C=Cc3cc[nH]n3)C)C(O)C2)=O)CCCCN1[N+](=O)[O-] 49421,CC1CCN(C(C2(COC)CCCC2)=O)CC1C.C12CCOC1CNC2=O 49422,CC1=NOC(C)(C(=O)NCCC(=O)NCCS(C)(=N)=O)C1 49423,C1(CC(=O)NCC2C(NC(C(N(C)C)C3CC3)=O)COC2)CN2CCN1CC2 49424,Cc1ccc(N2CC(C(=O)NCC3(C(=O)O)CCCC3O)CC2=O)cc1 49425,c1(N2CCN(CCCOC)CC2)nc(NCC(F)(F)Cl)nc2ncn(C)c12 49426,CC1CC(=O)NC1C(=O)NCC1CC(NC(c2cnn(C(C)(C)C)c2)=O)C1 49427,CC1CC(NC(c2cc(C(C)(C)C)on2)=O)CN(C(C2CC2C)=O)C1 49428,C12(NC(c3cnn(C)n3)=O)CCC1CN(C(=O)CSCc1ccccc1Cl)C2 49429,CCCC(C)(O)CC(=O)NC1CC(F)CN(C(=O)C=CC(=O)NC2CC2)C1 49430,Cc1oc(C(=O)NCCC2(O)CN(C(c3ccc(C(N)=O)cn3)=O)C2)cc1CO 49431,C#Cc1ccc(C(=O)NCC(C)CN(C(=O)COC2CCC(C)CC2)C)o1 49432,c1(-c2cn(C)c(=O)c(C(=O)NCC3CC=CCC3)c2)c(F)cc(Cl)cc1F 49433,c1(C(N2CCCC(O)(CNC(CCCOC)=O)C2)=O)cc(OC)cc([N+](=O)[O-])c1 49434,CC1CC(C)(C)CN1C(=O)C(O)C1CN(C(=O)CN(C)C)C1 49435,Cc1c(Br)sc(CNCC(C)(C)CN)c1Br 49436,c1(C(N2CCC(CNC(CSCCCC)=O)(OC)C2)=O)ccc(F)c(C(C)=O)c1 49437,N1(C(CN(C(C)=O)C)=O)CCC2(CCC2)C(NC(C2CC3CCC3C2)=O)C1 49438,N1(C(C2CC(c3ccc(F)cc3)C2)=O)CCC2C(C1)CN2C(=O)Cn1cncn1 49439,c1(N2CCCC(NC(C)=O)C2)ncnc(NCC2CCCC2(C)C)c1C 49440,C1(C(=O)OC(C)C)CCN(C(N2C(CCNC(C=C(CC)C)=O)CCC2)=O)CC1 49441,C1(N(C)C(C2(C)CC3(CCC3)C2)=O)CC2CC1N(C(c1ccc(N)cc1F)=O)C2 49442,C1(C(C)C)N(c2cc(O)ncn2)CC12CCN(C(=O)C(c1cnn(C)c1)C)CC2 49443,N1(C(c2c(SC)ccs2)=O)CCOC2(CCN(C(C3CCOCC3)=O)CC2)C1 49444,C1(NC(c2cnsn2)=O)CC12CCC(NC(c1cccc(F)c1Cl)=O)CC2 49445,Cc1cnc(C(N2C3CC2CN(C(C2CN(C(N)=O)C2)=O)C3)=O)c(F)c1 49446,Cc1oc([N+](=O)[O-])cc1C(=O)N(CCCNC(=O)C=CC1CCCN1C)C(C)C 49447,CN(CCCC(=O)NCC1(C)CCCN(C(C2COCCN2C)=O)C1)N=O 49448,c1(NC(C2CCC3(CN(Cc4c(C)nsc4)C3)O2)=O)cnc2ccc(Cl)nn12 49449,C1(COC)(CNC(C2CCCCC2O)=O)CCCN1C(=O)CC1(C)OCCO1 49450,c1(C(C)NC(C=CCN(C(C2(CF)CC(=C)C2)=O)C)=O)ncc(C)cn1 49451,C#Cc1ccc(C(=O)NC2CC3(C2)CC(NC(c2ccc(Cl)cc2)=O)C3)nc1 49452,N1(c2nc(OC)nc(C)c2)CC2CCCC1C2CNC(c1cnn(C)c1CO)=O 49453,c1(OC)ccc(CNC(c2cncc(Cl)c2)c2nnnn2C2(C)CC2)cc1OC 49454,O=C(CCCCc1cccs1)NC1CC(CCNC(C2(CF)COC2)=O)C1 49455,c1(C(=O)NC(C)CCNC(C2(F)CCCC2)=O)cc(Cl)cc(Br)c1N 49456,N1(C(C2(C3CC3)CN(C(C3CC4C=CC3C4)=O)C2)=O)CC2CCC(O)CC2C1 49457,C(=O)(CCN(OC)C(=O)CC1(OC)CC1(C)C)NC(CC)C 49458,n1(CC(=O)NCC(C)N(C(=O)CC(C)(F)F)C)ccc2ccccc12 49459,C(=O)(CC(C)(C)CNC(=O)CN1CC(=O)CCC1=O)NC(C(C)C)CO 49460,c1(CCC)onc(C)c1C(=O)NC1CC(NC(=O)Cc2cccnc2)C1 49461,C1(NC(=O)COCc2ccccn2)COCCN(C(C2CC3(CCC3)CO2)=O)C1 49462,C=C(C)C(CC(=O)NC1CN(c2cc(O)nc(SC)n2)CCC1C)OCC 49463,C12(C(=O)NCC(C)(C(C)C)NC(C3C(CC)CCCC3)=O)CC(C)(C1)OC2(C)C 49464,c1(C(C)C)cccc(C(=O)N(C(C)CNC(C2CC2Br)=O)C)n1 49465,C(CCCC(C)(C)C(=O)NNC(=O)C(F)(F)CC)NC(c1occ(C(N)=O)c1)=O 49466,N1(C(C2C=CCCC2CO)=O)CC2CCC(C(=O)NC3CCCC34CCC4)(C2)C1 49467,CC1CC(C)CN(CC(c2ccccc2)NC(=O)CN2CCCCC2C)C1 49468,C(=O)(C(O)CC[S+](C)C)NC1C(NC(c2cccc(CC(C)C)c2)=O)C1 49469,c1(C(=O)NCC(C(C)(C)C)NC(C=C=C(C)C)=O)cc2ccccc2cc1N 49470,c1(C(=O)NCCN(C)C(C2C3CC3C3CC23)=O)cccc(OCC(F)F)n1 49471,N1(C(C(c2c(OC)cccc2)=O)=O)CC2CC1CCN2C(=O)CN1CCCC1=O 49472,C=CCCCC(=O)N1CCC(n2cc(CNC(C34CC(F)(C3)C4)=O)nn2)C1 49473,C1(NC(C2CCC(C)O2)=O)CCCC(C(N2CCOC(C3CCC3)C2)=O)C1 49474,c1(OC)cnc(F)cc1C(=O)NC1(CNC(=O)CN2CCC(C)C2)CC(F)(F)C1 49475,Cc1ccc2c(C(=O)NC3(C)CCN(C(C4(S(N)(=O)=O)CCC4)=O)C3)coc2c1 49476,C1(C(=O)NCCC(=C)CNC(=O)CCOCC(F)(F)C(F)F)CCCC(C)C1 49477,c1(C(=O)OCC)ccc(NC(=O)C(C)=CCNC(=O)C=CC(C)CC)nc1 49478,CC(CCN(C)C)C(=O)NCCC1CSCCN1C(=O)CSCC(F)F 49479,c1(CC=CCNC(c2c(CC)ocn2)=O)ccc(F)c(OC)c1.C12N(C1)C2=O 49480,n1(CC(N2CC3C(NC(c4c(C)ncs4)=O)(C3)C2)=O)nc2n(c1=O)CCCCC2 49481,C(CC(C)C(=O)NC1CCC(C(=O)NCCC2(C)N=N2)CC1)=CC 49482,C1(C(=O)NCC23OCC(NC(c4ccnnc4)=O)C(C2)C3)CCc2nncn2CC1 49483,C1(C(N(C(CC)C(=O)N2CC(C(N)=O)(COC)C2)C)=O)CCCN(C(N)=O)C1 49484,CCC(C)(CNC(=O)C(F)OC(F)(F)F)C(=O)NCC1(CN=[N+]=[N-])CC1 49485,c1(C(=O)OC)cccc(C(C)OCc2cn(C)nn2)n1.C1(C=O)CCCN1C 49486,CC12CCC(C(=O)NCCCNC(=O)CC3CCCCCC3)(CC1)CO2 49487,c1(C(C)(C)C)ccc(F)cc1C(N1CC2C(C1)N2C(c1coc(Cl)n1)=O)=O 49488,c1(NC(C2(NS(CCC)(=O)=O)CC2)=O)cc(F)ccc1Br 49489,C1(CC(=O)NC(c2ccccn2)C)CCCN(C(C2CCCO2)=O)CC1 49490,N12CCC(C)C(C1)C2=O.C1(C(=O)OC(=O)C2CC2)(C(=O)NC)CCCC1.C(C)CC 49491,C1(NC(=O)CN2CCOCC2)CC2CCC1(C(=O)Nc1cnc(O)nc1O)C2 49492,c1(CC)c(C(=O)NC2CCCC2CNC(=O)Cc2csc(Cl)c2)csc1C 49493,N1(C(CCN(CCC)C)=O)C2CCC1C(C)C(NC(c1nc(C)oc1C)=O)C2 49494,c1(OC(C(=O)N(CC(C)NC(=O)C(C)n2cnnn2)CC)C)ccc(C)cc1 49495,c1(C(N2CC(F)(CNC(c3cc(C(F)F)no3)=O)C2)=O)nccc(F)c1Cl 49496,N1(C(=O)Nc2c(OCCOC)cccc2)CCCC(C(C)OC)CC1 49497,C(=O)(C(CNC(=O)Cn1ccnn1)N(C)C)N(C(C(C)SC)C)C 49498,N1(C(CN(C(=O)CCn2cccc2)CC)=O)CCSC(C)C1C 49499,c1(CC(=O)NC(C)CC2CN(C(C3CC(C)(O)C3)=O)C2)cc(F)ccc1Br 49500,Cn1cccc1C=CC(=O)NC1CCC1CNC(C1CCOC1=O)=O 49501,O=C(C(O)CC(F)F)Nc1ccc(N2CCNCC2=O)nc1 49502,C1(C(=O)NCCOCCNC(c2nn(CC)nc2C)=O)C2CS(=O)(=O)CC12 49503,N1(C(C(c2ccc(F)cc2)C)=O)CC(NC(C2CC3C=CC2CC3)=O)CC(O)C1 49504,C1(C(=O)NCCN(C(COc2cccc(C)c2)=O)C)CC2(CCCC2)C1 49505,C(CCCCCNC(=O)CCc1cccnc1Br)N(C(C1C(=C)CC1)=O)C 49506,C(=O)(CCCN(C)N=O)N1CC(CCCNC(CCC2CC(OC)C2)=O)OCC1 49507,c1(CC)cnccc1C(=O)NC1CC(C)(C(=O)NCC(c2ccsc2)O)C1 49508,N1(C(C2CCN(C(c3cc(C)c(=N)[nH]c3)=O)C2(C)C)=O)CCC2(CC(F)C2)C1 49509,C=CC(CCC)CC(=O)N(C(C(=O)NC1CCCCCCC1)C(C)CC)C 49510,N1(C(c2c[nH]nc2Nc2cn(CCNC(COC)=O)nc2)=O)CCCC(CC)C1 49511,c1(OC)cc(CN2CCNCC2)c(OC)cc1I.C12CCCN(C1)C(=O)COC2 49512,c1(C(=O)NCC(C2CC2)NC(C2N(C=O)CCC2)=O)cc(Cl)c(Cl)c(Cl)c1 49513,N1(C(c2cccc(SCn3c(C)cc(C)n3)c2)=O)CC2CNCC2(C)C1 49514,N1(C(c2nc(C(C)=O)sc2)=O)CC2(COC(CNC(c3coc(Cl)n3)=O)C2)C1 49515,NCCCC(C(=O)NC1(CO)CCSC1)c1ccccc1 49516,C(=O)(CC(F)(F)C(C)(F)F)N1CC(N(C(=O)C(F)n2cccn2)C)C2(C1)CC2 49517,N1(C(c2c(COC)noc2)=O)Cc2n[nH]cc2C1C(=O)N1CCCC1C1CC1 49518,c1(N(C2CCCC2O)C)nc2c(c(=NCC3CN(C4CC4)C3)[nH]1)CSC2 49519,C(=O)(C1=NOC2COCC12)N1C(C(=O)NC(CC#C)CO)(CC#C)CCC1 49520,Cc1nc(C2CCCOC2)sc1C(=O)NCCCOCCN(C)C(C1CC1C)=O 49521,N1(C(C(CC)CO)=O)CC2(CCCC2NC(=O)CC2(CS(C)(=O)=O)CC2)C1 49522,c1(COC)cc(CC(=O)NCC2CC(C(F)(F)F)CO2)co1 49523,CC(CCCNC(=O)C(O)Cc1ccccn1)NC(=O)C=CC=C(Cl)Cl 49524,C1(NC(C2C(C)(C)OCC2)=O)COCCN(C(c2ccnc(C3CC3)c2)=O)C1 49525,N1(C(c2occc2C(=O)O)=O)CC(F)(n2cc(CN3CCOCC3)nn2)C1 49526,n1(CCC)cc(C(=O)NCCC2CCCN2C(=O)C(C2CC(F)(F)C2)OC)nn1 49527,N1(C(=O)OC)CCC(C(N2CCC(C)C2C)=O)CC12CCC2 49528,C1(C(=O)NCC2CN(C(Cc3cc(C)on3)=O)C(C)C2)CCC2(CCOCC2)O1 49529,c1(CC)c(NC(=O)NC2CCN(S(C)(=O)=O)C2)nc(Cl)nc1NC 49530,c1(C(C)=O)ccc(C)o1.n1(C(c2nnnn2CC(F)F)C2CC2)cc(C(C)(C)F)nn1 49531,C=Cc1ccc(C(N2CCN(C(C3C(F)(F)C34CCC4)=O)C(CO)C2)=O)cc1 49532,CC1OCCCC1C(N1CCC(CCC(=O)NC(C)CN2CCOCC2)CC1)=O 49533,C1(C2CC2)(C(N(C)CC2CCCSC2)=O)CN(C(=O)CC2CC2(C)C)C1 49534,c1(C(=O)NN2CC(CC=C)(NC(C3CC=C(C)CC3)=O)C2)ccnc(OC)c1F 49535,n1(CC)ncc(C(=O)NCC(N2CCC(NC(=O)OC(C)(C)C)C2)=O)c1C1CC1 49536,C1(NC=O)(CSC)CCOCC1.c1(OCCNC(CC2C(C)(C)CC2)=O)cccc(O)c1 49537,c1(C(=O)O)cc(=NCCCNCc2ccc(OC)cn2)[nH]c(CC2CCCC2)n1 49538,Cc1nn2ccc(-n3cccn3)nc2c1N(C)CNC1(c2cccc(Br)c2)CC1 49539,N1(C(CC2CCC(=O)N2)=O)CCN(C2COCC2NC(=O)COC2CC2)CC1 49540,n1(CC=C)nnnc1CNCC1CC1c1cnn(Cc2cc(C(C)C)no2)c1 49541,c1(C(=O)NOCC)c(F)ccc(Cl)c1F.c1(COC(C)C=O)ccc(F)cc1 49542,CC1CN(C(=O)C=C2CCSCC2)CCCN1C(=O)CN1CC(=O)N(C)C1=O 49543,c1(OCC(=O)NC(C)C(CO)NC(c2ccc(C(N)=O)cc2)=O)ccc(Cl)cn1 49544,C12(NC(CC3(C=C)CCOCC3)=O)CCCC1CN(C(=O)CC1OCCC1C)C2 49545,Cc1cccc2c(C(=O)NCc3cccc(CNC(C4CC4(F)F)=O)c3)n[nH]c12 49546,N1(C(C2(F)C(C)OCC2)=O)CCC2(CCCN(C(=O)CO)C2)C1 49547,c1(C(N2CC(NC(=O)CCOc3ccc(Br)cc3)C(O)C2)=O)ccc2nncn2c1 49548,N#Cc1cc(C(N2CCC(NC(C3CCCSC3)=O)C2)=O)ccc1Cl 49549,C12(C(N3C4C(NC(c5cc6c(s5)CCC6)=O)C(C4)C3)=O)CCC(O)(CC1)CC2 49550,C1(C(N2CC3(C2)CCN(CC)C(CC=C)C(=O)N3)=O)CC2CCCC2C1.OC 49551,N1(C(c2c(C)nccn2)=O)CCC(NC(=O)COC2(C)CCC2)C12CC2 49552,CC1(C)COC1CC(N1CCC(c2ccccc2)C1)=O 49553,CN1CC2(CCN(C3CC4CC3N(C(C3CCS(=O)(=O)C3(C)C)=O)C4)CC2)C1 49554,C1(CCOC)CN(C(C2(Cl)CC2(C)C)=O)CCN1C(c1ccn(C)c1)=O 49555,N1(C(C2C(NC(CCC#CC)=O)C3CCC2C3)=O)CCc2nc[nH]c2C1 49556,Cc1cccc(CC(C)C(=O)NC2(CF)CCC2)c1.C12CC(C)(C1)CCNC2=O 49557,c1(NC(c2[nH]c(C)c(C(N3CC(F)C(F)C3)=O)c2C)=O)ccc2ncc(I)n2c1 49558,c1(CC)csc(C(=O)NC2(CC)CN(C(c3csc(Cl)c3)=O)C2)n1 49559,N(C(=NCC1CC1)NCc1ncc[nH]c1=O)C(c1ncnn1C)C 49560,c1(C(=O)NC2C(NC(CCOC)=O)CCC2)cc2c(cc1Br)OCO2 49561,c1(C(=O)NC2(C(=O)NC(CC=C)C)CC(O)C2)ccc(C)c(OC)c1 49562,N1(C(C(C(C)C)OC)=O)CC2CC1CN2C(c1cc(C2CC2)nc(O)c1)=O 49563,CC1CC=C(C(=O)NC23CCCN(C(C4CC(=O)NC(=O)C4)=O)CC2C3)CC1 49564,C(=O)(C1=C(c2ccccc2Cl)CCC1)N(C1CCCCO1)C.C12CCCN(C1)C2 49565,CC1CCC(CCNC(=O)C(Cc2cn[nH]c2)NC(=O)Cn2ncnn2)CC1 49566,C(C)(CCC(=O)N(CCCNC(c1cnc(C)o1)=O)C)SC 49567,c1(C(=O)NCC(C)(C)OCCNC(CCCCSC)=O)ccc(C(C)(C)C)cc1C 49568,C(C(C(C)C)NC(c1ccccn1)=O)(C1CCCCC1)NC(CCCC)=O 49569,Cn1cnc2c1CCCC2C(=O)N1CC(NC(C2OCCO2)=O)C(C)(C)C1 49570,Cc1cnc(CN=C(NCC2CCC2)NCC2CCCCC2F)c(C)c1 49571,N1(C(C(C2CCN(C(c3cc(C(C)=O)on3)=O)C2)C)=O)CCc2nnnn2CC1 49572,CCC(CNC(=O)C(C1CC1)SC)N=c1[nH]c(C(C)C)nc(C)c1Br 49573,N1(C(C2CCC(C)O2)=O)CCCC2C1CCN2C(c1cccc2c1CC(=O)N2)=O 49574,c1(CC)sc(C(=O)NCC2(C)CCN(C(=O)C(c3cccnc3)C)C2)cc1C 49575,CC1CC2(CC(C(=O)NC3CCN(C(C4CCS(=O)(=O)CC4)=O)CC3F)C2)C1 49576,c1(CN2CC(C(=O)Nc3ccc(CC(=O)OC)cc3)OCC2)cc(F)cc(Cl)c1 49577,C1(C(=O)NCC)C2CC3C(C2NC(=O)C(C)(C)CNC(=O)Cc2cn(C)cn2)C13 49578,C1(C)(CC)CC(NC(=O)CC(C)(C)CNC(=O)Cc2cccn2C)CCO1 49579,c1(NC(CCc2ncc(C)[nH]2)=O)ncccc1CNC(=O)C(O)C1CCCC1 49580,Cc1nnn(C)c1C(N1CCC(C)(CNC(=O)C(c2ccccn2)C)C1)=O 49581,c1(C(N2CC(C(C)NC(Cn3c(C)ncc3)=O)C2)=O)cnn2cccc(Cl)c12 49582,C1(C(N2CC3(CN(C(c4nn(C)c(O)c4)=O)C3)C2)=O)CCC2(CCOC2)O1 49583,C#CC1CN(C(=O)CC2(C3CC3)CC2)CCN1C(C1CCC1COC)=O 49584,N1(c2c(C#N)nccn2)CCCC(C2(NC(C3CC3Cl)=O)CC2)C1 49585,CC1(C(=O)N(CC(O)CO)CC2CCCO2)CCN(C(=O)CSCC(F)(F)F)CC1 49586,CC(O)C(C(=O)NCc1cn[nH]c1)NC(=O)CC1CC2C=CC1C2 49587,CC(C)(C)C(CNC(c1ccc2cc[nH]c2n1)=O)C(=O)N1CC2(CCC2)CC1CO 49588,C1(NC(c2cc(CC)[nH]n2)=O)CC2C1CCN2C(c1cnn(C(C)CC)c1C)=O 49589,c1(C(N2C(C)(CNC(CC(CC)OC)=O)C=CC2)=O)ccc2c(c1)CNC2=O 49590,Cc1cc(C)c(C(N2CC(O)(CCNC(=O)C(C)OCCN(C)C)C2)=O)c(O)c1 49591,N1(C(c2nccc(CO)n2)=O)CCN(C(c2cnsn2)=O)C(c2ccccn2)C1 49592,C1(CCOC)(NC(=O)CSc2nncs2)CCN(C(c2ccc(CO)cn2)=O)C1 49593,CC1CC(CO)(NC(=O)CCN(C(=O)C(c2cccn2C)=O)C2CC2)C1 49594,N1(C(C2(P(C)(C)=O)CC2)=O)CC(NC(C2CNC(=O)N2)=O)C2CCCC2C1 49595,Cc1ccc(C(=O)NCCC2(CNC(C3CCN(C)C3=O)=O)CC2)cn1 49596,C1(NC(=O)COC2CC2)CC2CN(C(c3cc(Br)c(F)cc3Cl)=O)CC2C1 49597,C1(n2cc(C(CC)O)nn2)CC2CCC(C1)N2C(=O)Cc1ccc2c[nH]nc2c1 49598,S(=O)(=O)(c1ccc(=NCCOCCOC)[nH]c1)NCC(COCC)(C)C 49599,C1(CNC(=O)CC2CCCCO2)CCCCN1C(C1(CO)CCCC1)=O 49600,N1(C(C2C(C(C)C)CCO2)=O)CCCC(C(=O)Nc2cnn(C(C)C)c2)CC1 49601,C1(n2cc(-c3nccc(C)n3)nn2)CC2CCC1(C(c1ccccc1)=O)C2 49602,N1(C(c2c(NC)ccc(Cl)c2)=O)CCC=C(C(=O)N(C)Cc2ccncc2)C1 49603,N1(C(C23CC(n4cc(CC)nn4)C2C3)=O)CCN(CC(=O)NCC(C)C)CC1 49604,C1(NC(C2(C)C(C(=O)OC)C2)=O)CN(C(C2C(F)(F)C23CCC3)=O)C2(CCC2)C1 49605,C#CCC(C(=O)NC)NC(=O)CC1(CNC(c2nccnc2C)=O)CC1 49606,C1(O)(CNC(CCOCCN(C)C(c2ncc[nH]2)=O)=O)CCOC1 49607,C1(C2CC2)(NC(CCC=CC)=O)CCN(C(=O)CC2OCCOC2(C)C)C1 49608,c1(OC)cccc(N2CCC(NC(=O)N(C3CC3)C(C)C3CC3)C2=O)c1 49609,CC1(C)CC(F)(F)CCC1C(N1CCOC(CCNC(=O)CCCCC2CC2)C1)=O 49610,n1(CC)cc(C(=O)NCCCC2CN(C(=O)C(C)c3cc[nH]n3)CCO2)c(C)n1 49611,c1(OC)ccc(F)c(C(=O)NC2CCCCC2NC(c2cccnc2)=O)c1F 49612,C1(C(=O)NC(C(=O)Nc2cn(CCOC)nc2)C2CCCO2)CCC(N(C)C)CC1 49613,Cc1cc(C(N2CCCC(CNC(=O)CC3OCCCC3(C)C)C2)=O)ccc1N 49614,C1(N(C2CCOC2)C(c2nccc(C(=O)NCCO)c2)=O)C2CCC(F)(F)C12 49615,C1(NC(C2(COC)C=CCN2C(=O)CCc2ccc[nH]2)=O)CCCCCC1(C)C 49616,c1(C(=O)NCCC2CCN(C(c3c(C)nc(C)o3)=O)C2)csc(N=S(C)(C)=O)n1 49617,CC1(C(=O)Nc2nc(Cl)ns2)CCc2ccccc21 49618,C1(C(N2CC(F)(CNC(C(C)(C3CC3)OC)=O)C2)=O)CCC(C)(C)OC1 49619,c1(CC(N2CCC(C3N(C(C=CSC)=O)CCC3)C2)=O)c(C)nn(C)c1Cl 49620,N1(C(C2C3CCCC23)C(=O)Nc2cccc(OC)c2)CCOC(C)(C2CC2)C1 49621,C1(n2cc(CNC(C)=O)nn2)CCN(C(c2occc2C)=O)CC1 49622,c1(C(=O)OC)nc(=NC2CCCN(Cc3nc(C)nc4[nH]ccc34)C2)c(F)c(Cl)[nH]1 49623,C1(NCC(C2CCC(C)CC2)(C)O)C(C)CCCN1C(=O)OC(C)(C)C 49624,c1(C(N(CC(=O)NC(CN2CCCC2)CO)CCOC)=O)cnn(CCO)c1 49625,N1(C(c2c(C)coc2C)=O)C2CCCC1C(CNC(C1CNC(=O)N1)=O)C2 49626,C=CC1(CC)COCCN1C(c1ncc(Br)s1)C(=O)NC(C)(C)C 49627,c1(CN2CC3CN(C(c4c(OC)nsc4)=O)CC3C2)cc2ccccc2nc1C 49628,Cc1ccc(CC(N2CC3(CNC(=O)C=C4CCC(C)C4)CC2CO3)=O)cc1F 49629,Cc1cc(C=CC(=O)NC2COCC2CNC(=O)CCc2cccs2)on1 49630,N1(C(C(COC(C)C)(C)C)=O)CCCC(NC(c2cnc(O)c(F)c2)=O)C(F)C1 49631,c1(C(=O)OCC)coc(OC)c1C(N1CCN(c2nnn(C)n2)CC1)=O 49632,N1(C(CCC=C)=O)CC2(CCC2)CCC1CNC(=O)CCCF 49633,N1(C(C(=O)NCCC2CCN(C)CC2)c2cccs2)CCC(C)(C)CC(C)(C)C1 49634,N1(Cc2cc(C)c(Br)cc2C)CCC2CN(c3ncc4[nH]cc(I)c4n3)CC2C1 49635,C1(NC(C2CCC(N(C)C)CC2)=O)CCN(C(=O)Cc2ccnn2C)CC1O 49636,N1(C(C2C(C=C)OCC2)=O)CCN(C(c2ncc([N+](=O)[O-])n2C)=O)C2(CCC2)C1 49637,c1(C(C)C)cccc(F)c1C(=O)NC1CCN(CCO)CCO1 49638,c1(C(=O)NC2C(NC(Cc3c(C)ccc(C)c3)=O)CC2)c(C)nc(C2CC2)nc1C 49639,C1(CC=C)(NC(=O)CC2CCCOC2)CCCN(C(c2ccc(C(=O)OC)[nH]2)=O)C1 49640,c1(C(N(C)CC2CCCN2C(C2CC(=O)N(C3CC3)C2)=O)=O)n[nH]c2c1COC2 49641,c1(OC)cc(C=CC(=O)NC23CCCC2CN(C(c2cscn2)=O)C3)ccc1F 49642,c1(C(=O)NC(C)CCCNC(c2ccc(F)s2)=O)nccc(Cl)c1Cl 49643,c1(NC(C2CSCCN2Cc2cc(F)c(O)c(Br)c2)=O)ncc(Br)cc1[N+](=O)[O-] 49644,C(=O)(C(C)CC(N)=O)NCc1cc(N2CCN(C(CN(C)CC)=O)CC2)ncc1 49645,C1(NC(CCCC#C)=O)CN(C(C2CCN(C(C)=O)CC2)=O)CCC12CCC2 49646,c1(C(=O)NCc2c(OC)nsc2)ccc(CNC(C2(C)CCNC2=O)=O)cn1 49647,c1(C(N(C(C)CNC(C2CC(F)CN2C(=O)NC)=O)CC)=O)cnc(O)c(C)c1 49648,C1(CNC(C(CC)(C)OC)=O)C2CCC(C2)N1C(=O)Cc1cc(C(F)F)nn1C 49649,c1(CC)ccc(C(=O)NCC(C2CC2)N(C(=O)C(N2CCOC2=O)C)C)[nH]1 49650,N1(C(C(CCCC)C)=O)CC2=C(C1)CN(C(C1CCCCC1CC)=O)C2 49651,Cc1cc(Cl)c(NC(C2(C)CN(Cc3cccc4occc34)C2)=O)cc1C 49652,n1(CC(N2CC(CN(C(CCC(C)OCC)=O)C)C2)=O)cccc(N)c1=O 49653,N1(C(C(C=C)c2ccccc2)=O)CCN(CCNC(=O)CC2(C)CC(F)(F)C2)CC1 49654,C1(NC(c2c(C)ncc(C)c2)=O)CCCC12CCN(C(c1[nH]c(O)nc1C)=O)C2 49655,c1(C(=O)NC2C(NC(C3CC(C)(C)OC3(C)C)=O)CCC2)cccc2c1CCN2 49656,c1(CC(=O)N(CC(CN(C(=O)CC(O)C2CCCC2)C)O)C)nncn1C 49657,C(=O)(C(F)(F)CC)N(C(CC)CNC(=O)CN1CCCC1=O)C(=O)CC1CSC1 49658,C1(C(=O)NCC(C(C)C)NC(=O)Cc2cccnc2)CCC2(CC2)C1 49659,c1(C(N(CC(C)(C)NC(c2ccc(C3(CO)CC3)s2)=O)C)=O)nc(O)nc(O)c1N 49660,c1(CNC(C2CC2NC(C#CC(=O)N(C)C)=O)=O)ccc(O)c(NC2CCC2)c1 49661,c1(C(=O)NC2(C(=O)NCc3cn[nH]c3)C(C)C2)ccc(=O)n(C)c1 49662,N1(C(C2(CCN(C)C)CC2)=O)CCCC1CNC(=O)CNc1ccccc1 49663,C(CC(F)F)(C(=O)NCCC1COCCO1)NC(CN1CC(=O)NCC1)=O 49664,C(C(=O)N(CCCN(C(=O)CN(S(C)(=O)=O)C)C)C)(C(C)C)CCO.CCC=O.N 49665,C1(C)(C(=O)NCCN(C(=O)Cc2cccnc2O)CC)SCCCS1 49666,C1(OC)CC(C(=O)NC(C2CCN(C(C3CCOCC3)=O)CC2)(C)C)C12CCC2 49667,Cc1nn(C)c(Cl)c1C(=O)NCC1CCCC1C(=O)NC1(C)CC(F)(F)C1 49668,c1(N2CCSCC(C)C2)nc(N2C3C=CC(C3)C2CO)nc2c1CSC2 49669,c1(NC2CC(NC(CC3(COC)CCOCC3)=O)C2)ncnc2cc(C)[nH]c12 49670,C1(CCC)CN(C(=O)Cc2nocc2Br)CCN1C(c1scnc1C)=O 49671,C#Cc1cnc(C(=O)NC(CC2CCOCC2)C(=O)N(CCC=C)C)c(C)c1 49672,C1(CCC)CN(C(c2cnc(Br)c(OC)c2)=O)CCN1C(=O)CCSC 49673,C(=O)(CC(CNC(C1(CC)CCOC1)=O)OC)NCCC 49674,N1(C(c2ccn(CC(C)C)n2)=O)CC2(C1)CN(C(c1ncc(Cl)n1C)=O)CCO2 49675,c1(NC(c2cc(CCNC(=O)C(C3CCCO3)C(N)=O)on2)=O)cc(C#N)cn1C 49676,C1(OC)CN(C(c2c(Cl)nsc2Cl)=O)CCC1NC(=O)C(F)C1CCOC1 49677,C1(C(N(CCCNC(CN(C(C)C)C)=O)C)=O)CCCN1S(C)(=O)=O 49678,N1(C(c2c(F)ccc(C)n2)=O)CC2CCN(C(=O)CCC3CCC(C)O3)CC12 49679,N1(CC(N2CC(O)(CNC(C3(c4cccnc4)CCCC3)=O)C2)=O)CSCC1=O 49680,N1(C(C(CC)N(C)C)=O)CC2(CC(CC(=O)NCCc3ccc(F)nc3)C2)C1 49681,N1(C(C2N(C(=O)OC)CCC2)=O)CCCC(NC(=O)Cc2cnc(C)[nH]2)CC1 49682,C(C(C(=O)NC(C)C(C)O)NC(c1ccc(CSC)s1)=O)OCC 49683,C1(C(=O)NCC2C3CN(C(=O)CCN4CCOC4=O)CC23)CCc2cnnn2C1 49684,c1(C(=O)NC2C(C)(C)CN(C(=O)CC3OCCO3)C2)cnc2nccn2c1 49685,CC1CC2CN(C(=O)CCc3cnn[nH]3)CC2N1C(=O)CCC12CCC(CC1)C2 49686,Cc1ccnc2ccc(C(=O)NC3CCC(C)N(C(c4cnn(C)c4)=O)C3)cc12 49687,c1(C(N(C(CNC(C(C)OC)=O)C)C)=O)ccc(F)c2c1OCC2 49688,CC(C)C(O)C(C)(C)C(=O)NC1CCN(C(=O)CC2CCCSC2)CCC1CO 49689,Cc1ccc(F)c(C(=O)NCC(c2nnnn2C(C)C)NN2CCOCC2)c1Br 49690,c1(OC)ccc(CC(=O)N(C(c2cn(-c3ccccc3)nn2)(C)C)C2CC2)c(C)c1 49691,C(N=c1ccnc(NC(CN(C)CCc2cccs2)=O)[nH]1)C1CCCC1 49692,C1(NC(c2c(C)csc2)=O)C2CC3CN(C(=O)CC(C)(C)C(F)(F)F)C1C3C2 49693,C(=O)(CCCCCC(C)(C)C)N(CCCNC(CCc1ccc(C)s1)=O)C1CC1 49694,c1(OC)ccc2c(c1)CCC(C(N1CC(NC(C3OCCO3)=O)C(C)C1)=O)C2 49695,N1(C(c2c(N)cc(F)cc2)=O)CCCC(C2(NC(C3CCCCO3)=O)CC2)C1 49696,CN1CCN(C(=O)CC2CCC(C)(C)O2)CC1CNC(C1CCC(C)(C)O1)=O 49697,c1(C(N(C(CC)C(=O)NC(C)COC(F)(F)F)C)=O)cccc2cc[nH]c12 49698,C(=O)(C1=CCCCCC1)NCC1(OC)CCN(C(CSCCCC)=O)C1 49699,C(=O)(CC(CC=C)NC(c1ccnc(O)c1F)=O)NC(C#C)CC1CCC1 49700,C(=O)(C(F)(F)C(O)c1ccccc1)NC1C(NC(COCC=C)=O)COCC1 49701,c1(NCc2scc(C(=O)OC)c2)cccc(C(=O)Nc2cc(C)ns2)c1C 49702,c1(C(N(CC(CC)NC(=O)CC2(O)CCC2)CC)=O)ccc2scc(C)c2c1 49703,c1(C(=O)NC23CC(C(N4C5(C)CC5CC4)=O)(C2)C3)cc2ccccn2n1 49704,C1(NC(C(C)(C)C(F)(F)F)=O)CC(C2CCN(C(=O)CNc3ccccc3)C2)C1 49705,c1(C(=O)OC)[nH]c(=NCC23CCC(C)(CC2)CO3)sc1Cl 49706,C(C(F)(F)C(F)(F)F)N(C(CC1(N(C(CCC#C)=O)C)CC1)=O)CC 49707,c1(C(=O)NCC(CCNC(=O)CC2CC(=O)NC2=O)O)cnc2[nH]cncc1-2 49708,c1(NCCCN(C(c2c(C(C)C)cccc2)=O)C)cnc(C#N)c(C#N)n1 49709,CCCC(CC)C(=O)NCCNC(c1cc(F)ccc1NS(C)(=O)=O)=O 49710,C1(CNC(CC(C=C)C)=O)CCN(C(=O)C(c2cc(C)ccn2)(C)C)CC1(F)F 49711,c1(OC)ccc(C(=O)NC(C)(CNC(=O)CC(C)(C)O)C(C)C)cc1C 49712,N1(CC)CCCC1CC(=O)NCC#CCNC(=O)CCOCC1CC1 49713,c1(OC)ccccc1C(=O)NC(C)C(CO)NC(=O)CC1CCCOCC1 49714,C1(OCC)(OC)C(C(=O)NCC2(C)CCC(=O)NC2)CC1(F)F 49715,c1(C(=O)NCCCN(C(c2cc(C)c(Br)o2)=O)C)n[nH]c2nccc(Cl)c12 49716,Cc1cncc(C(=O)NC2CCN(C(=O)C(c3c(C)n[nH]c3C)C)CC2C)c1Cl 49717,S(=O)(=O)(c1c(Cl)ccc2c1OCO2)Nc1ncnc2sc(C)c(C)c21 49718,c1(C(N2C(C)CC(NC(C34CCC3CC4)=O)C2)=O)ccc(N)cc1S(N)(=O)=O 49719,Cc1nc2c(CNC(c3c(C)cccc3C)C3CCCN3)ncnc2[nH]1 49720,C1(NC(C2CCN(CC)C2)=O)CCC12CN(C(=O)Cn1cc(C(F)(F)F)nn1)C2 49721,C1(CNC(=O)NCC2CN(c3nnc(C4CC4)o3)C2)CC(=O)N(C2CCCCC2)C1 49722,C(CC(C)C)(C(=O)NC1CC1CNC(=O)CNC(c1cscn1)=O)NC(C)=O 49723,CCCC(CCC)CC(=O)NC1(C)CN(C(c2cc[nH]c2C2CCCC2)=O)C1 49724,c1(C(=O)NC(CC=C)CNC(=O)Cc2ccsc2C)cc2c(O)ncnc2cn1 49725,c1(CC)nc(C2CCCN2Cc2ccccc2)n(-c2ccc(Br)cc2)n1 49726,C1(Nc2c(C(=O)OC)c(Cl)ncn2)CC1C1CCCN(C(=O)C2=NOCC2)C1 49727,c1(N(C)CCOC(F)F)nc(=NCC2COC(=O)O2)[nH]c2c1SCC2 49728,C1(C(N2CCN(C(C=C(CC)CC)=O)CC2C2CCC2)=O)CCn2ccnc2C1 49729,CCCCC(O)C(=O)NCCOCCOCCNCCCSc1ccc(Cl)cc1 49730,Cc1cc(C(=O)NC2CC2CNC(c2nnn(C)n2)=O)c2ncccc2c1 49731,C1(NC(C(C(C)O)N(C)C)=O)CCN(C(=O)CC2CC(C(C)(C)C)C2)CC1O 49732,c1(OC)cc(Cl)ccc1CC(=O)N(C(C)CN(C)C(C1CC2CCC1CC2)=O)C 49733,CC1(CNC(c2cn(C3CCC3)nn2)=O)CC(NC(c2cnc[nH]2)=O)C1 49734,c1(OC)ccc(-c2nc(Cc3cnn(C(C)C)c3)n(C3CCCCC3C)n2)cn1 49735,c1(C(c2nnnn2C)Sc2c(CC)cc(C#N)cc2)cc(Cl)cc(Br)c1F 49736,C(=O)(C1=CCc2ccccc21)N1C(CNC(c2ccn(C3CC3)n2)=O)CCC1 49737,CCC(C)(C)CNC(=O)C(C1CCCC1)NC(=O)C=CC(C)(C)SC 49738,c1(C(=O)NCCn2cc(C(=O)NCC(=O)NCC(C)C)nn2)ncccc1F 49739,C(=O)(C(O)CC(C)C)N1CC(C=C)(CC(=O)N(C)Cc2ccncn2)C1 49740,C1(CC(c2nccn2C)NC(=O)NCCc2nc(C)sc2)CC12CCOC2 49741,c1(OC)ccc2c(CCC(=O)N(CC(C)NC(c3ccc[nH]3)=O)C)c[nH]c2c1 49742,C(CC(=O)NOCC1(C)CC1)Cn1ncc(N(C(CNC(=O)NC)=O)C)c1 49743,N1(C(c2ccc(C)o2)=O)CC2(CCCC2)C1C(=O)NCC1=CCCN(C)C1 49744,C1(CNC(=O)CCC2CCC(O)CC2)CC(O)CN1C(=O)C=Cc1ncc[nH]1 49745,N1(C(c2n[nH]c(CC)c2Cl)=O)CCC2(CCC2CNC(=O)C(C)C(C)C)CC1 49746,c1(C(=O)NC(CNC(C2CC=CCO2)=O)C2CC2)sccc1S(=O)(=O)N1CCCC1 49747,c1(C2(C(N3C(CC(=O)OC)CCC3)=O)CCC2)ccc(C2=C(C)CCCC2)cc1 49748,c1(C(N(CCC(N2CCC(CSC)C2)=O)CC=C)=O)cccc(CO)c1 49749,c1(C(=O)NC(C2(O)CCN(C(C(=O)NCC)=O)C2)C)ccc2ncn(C)c2n1 49750,N(C(=NCC1CCCSCC1)NC1CCC1)C(C1CCC1)C 49751,CON(CCC(=O)NC12CC(C)(CO1)C2)C(=O)C(COC)N(C)C 49752,C(=O)(CCS(C)=O)NCCCN(c1ccccc1)C.C1(=O)CC(C2CC2)N1 49753,CCCC(CCCNC(=O)C(F)OC)NC(C1(C)CCN(C)C1=O)=O 49754,N1(C(CC2CC(SC)C2)=O)CC(NC(C2(C)CCCOC2)=O)CC(C)C1 49755,N1(C(C2(CCOC)CCCC2)=O)CC2CC(NC(=O)C=CC=C(Cl)Cl)CC2C1 49756,Cc1cccc(Br)c1C(C(N1CCC(CO)CC1)=O)NC(c1cnn(C)c(=O)c1)=O 49757,c1(C(=O)NC(C)CCCCNC(c2cnc(C(C)O)s2)=O)cccc2c1CCN2 49758,C(=O)(C(C)C(C)S(C)(=O)=O)NCC1CC(CC)(CC)C1 49759,CC(C)C(C)(CNC(c1cnc(C2CCC2)s1)=O)NC(=O)CCCn1cccn1 49760,c1(CNC(=O)CCc2cc[nH]n2)ccc(C(=O)NCC23CCC(CC2)O3)cn1 49761,c1(C(C)(C)C)c[nH]c2cc(NC(C3CC(F)CN3C(=O)CCS(C)(=O)=O)=O)ccc12 49762,C1(NC(C(CC)n2cncn2)=O)CCCN(C(=O)C=CCOCC(F)(F)F)C1 49763,CC1(C(=O)NC2CCC2CNC(=O)C=Cc2ccco2)CCCNS1(=O)=O 49764,C1(NC(C=CC=CC)=O)CCN(c2cnc(F)cn2)CC1O 49765,N1(C(c2cnc(C3(N)CCC3)s2)=O)CCC2CC2C1 49766,C1(C)(CNC(c2c(CC)c[nH]n2)=O)COCCN(C(C2CC2CC)=O)C1 49767,C1(OC)CC(C(N2CC=CC(O)C2)=O)N(C(=O)C(c2ccnn2C)C)C1 49768,Cc1cccnc1C(=O)NC1CC(C)N(C(C2CN(S(=O)(=O)C(F)F)C2)=O)C1 49769,N1(C(C2N(C(C(N)=O)=O)CC2)=O)CCOC2CC12 49770,C1(CC)C(NC(=O)CSc2cn[nH]c2)CCN1C(=O)COc1cccc(F)c1 49771,c1(C(=O)NCC2(NC(C3CN(C(C)C)C(=O)CC3)=O)CC2)nccn2ccnc12 49772,C(=O)(C1=NNC(=O)CC1)N1CCCC(C)(NC(C2CCC3CC3CC2)=O)C1 49773,c1(NC(c2cc(C)sc2N)=O)nncc2ccoc12 49774,c1(CCN(C)C(=O)NCC2CCCN2Cc2ccccc2)ccc(Cl)cc1 49775,Cc1cc(C(=O)NC2CC(F)(F)CC2NC(=O)C2=CCOCC2)cc(Cl)c1 49776,N1(C(CC2(C=C)CN(C(=O)CP(C)(C)=O)C2)=O)CCN(CC)C(=O)C1 49777,c1(C(N2CCN(C(=O)NCC)CC2)=O)cc(N(C)C)nc2cc(Br)ccc12 49778,N1(C(C(CC)=CCCC)=O)CCC2CN(C(c3sc(C)cc3Cl)=O)CCC12 49779,CCC(C)(C(=O)NCC1CCC1NC(c1nc(=O)n(C)[nH]1)=O)OC 49780,N1(CC2N(C)CC=CC2)CC(=O)N(Cc2ccc(C3CCC3)cc2)C1=O 49781,CCCC(C)(CC)C(=O)N1CCCCC(NC(c2nn(C)c3c2CCC3)=O)C1 49782,Fc1cccc(C(F)CNC(C2CCC2)C2CC2)c1F 49783,c1(C(N2CC(CC)N(C(C3CC(F)C3)=O)CC2)=O)c[nH]c2ccccc2c1=NC 49784,Cc1ccc(CC(=O)NC2CCCCN(C(c3cc(=N)[nH]c(Cl)n3)=O)C2)cc1C 49785,c1(NC(c2cccc(NC(CC(=O)OC)=O)c2)=O)cc(I)ccc1I 49786,C1(C(N2CC(C)(NC(c3cnn(-c4nccs4)c3)=O)C2)=O)CC2(CCCC2)CO1 49787,c1(OCC=C)ccc(Cl)nc1C(=O)NC1CCC1NC(=O)C(C)c1ccco1 49788,c1(Cn2c(-c3ccccc3F)nc(CCOC)n2)cc(F)cc(F)c1 49789,N1(C(C2C(NC(C3(C)CCC(C)C3)=O)CCO2)=O)CC(O)(C2CCC2)C1 49790,C1(NC(C2C=CCCN2C(c2ccc(F)cc2)=O)=O)CCOC12CCC2 49791,C(C1CN(C(=O)CC2CC3CCC2CC3)CC1C(=O)NCc1cccnc1)=CC 49792,N1(C(C2N(C(C(C)C)=O)CCCC2)=O)CCC(NC(c2cnc(S)[nH]2)=O)C(F)C1 49793,C(CCN(C)C(c1ccc(CC)s1)=O)(C(C)C)NC(c1cc(CCC)[nH]n1)=O 49794,C(CC(O)C(=O)N(C1CC1)Cc1ncnn1C1CCCC1)NC(N)=O 49795,CCCS(=O)(=O)C(C)C(=O)NC1CN(C(=O)CCn2cc(C)cn2)C(C)(C)C1 49796,c1(CN(C(=O)Cn2cnc(C(N)=O)n2)C)ccc(CNC(=O)CC(C)(F)F)cc1 49797,C1(NC(c2c(CNC(c3ncc(C(N)=O)nc3)=O)cc[nH]2)=O)C2CCCCCC12 49798,C12(NC(CC3C(CC)C3)=O)CC(CNC(c3ccn(C)c3C)=O)(C1)OC2C 49799,Cc1ccc(C(=O)NCC(C)(C2CC2)NC(=O)COCP(C)(C)=O)c(C)c1 49800,c1(C(C(=O)NCCCC(=O)OC)N(CC(C)C)C(C)C)cc(OC)cc(O)c1 49801,c1(NCCCC(=O)N(C)C)cc(Br)ccc1S(=O)(=O)NCC1CCOC(C(C)C)C1 49802,C1(N(C(COC(CC)CC)=O)C)CCN(C(C2C(C)CC2C)=O)C1 49803,C(CCCC(=O)N1CC2CC2(CNC(=O)CNC(c2ccc(Cl)cc2)=O)C1)OC 49804,c1(C(=O)NC(C2CCCN(C(c3n[nH]c(C)c3O)=O)C2)C)cc(Cl)cnc1O 49805,N1(C(CSCCCC)=O)CCC12CN(C(=O)CCC(C)(C)F)C2 49806,C1(CCNC(C2(C=C)CC2)=O)CN(C(c2cncc(N)c2C)=O)CC(C)O1 49807,C(CCCCC(=O)N(C1CCC1O)C)N(C(=O)Cc1cncnc1)C 49808,N1(C(CN(c2ccncc2)C)=O)CCCCCC1CNC(c1ccccc1F)=O 49809,CC1=C(C(=O)NC2COC3(C2)CN(C(=O)CCc2scnc2C)C3)CCS1(=O)=O 49810,c1(C(=O)NC(CC=C)CNC(C2(C)CCOCC2)=O)cc(C)cc2c1NCCC2 49811,CC1CC(NC(C2CCCCS2)=O)CCN1C(c1c[nH]c(=O)cn1)=O 49812,C(=O)(CCCCCc1cn(CC(F)(F)F)nn1)NC(CCC)C 49813,CC(C(=O)N=c1ccn(CCNC(c2cc[n+]([O-])cc2)=O)[nH]1)c1ccno1 49814,Cc1nccc(C(=O)NC23CC2CN(C(=O)C#CC2CC2)C3)c1C 49815,CCCCCC(O)C(=O)N1CCCC(CNC(=O)CC2(OCC)CCOCC2)C1 49816,C(C(CC(=O)NCCOc1ccon1)C1CCC1)NC(CCOC)=O 49817,N12CCCC1C2=O.N1(C(CNC(=O)CCC2CCCC2)=O)CCC(O)C1.C1(C)CCC1 49818,C#Cc1ccc(C(N2CCC(NC(C3CC3C3CCC3)=O)C(O)C2)=O)c(F)c1 49819,C#CC1CCC(NC(C2CCCN2C(=O)COC(=O)NC2CCCCC2)=O)C1 49820,CCCCC(C)CCC(=O)N1CCC(CNC(c2coc(Br)n2)=O)C12CC2 49821,c1(CNC(=O)NCc2cnc(C3CCC3)o2)cccc(C(F)(F)F)c1 49822,n1(CC)nnc(C(=O)NCC2(C)CCN(C(C3CCN3C)=O)C2)c1C 49823,C1(C(=O)NCc2n(C)ccn2)CC2CCC1N2C(=O)C(O)C1CCC1 49824,n1(CC(=O)NCC2CCCC(NC(c3ccc(SC)s3)=O)C2)nc(C)ccc1=O 49825,CON1CCC(CC(=O)NC2(C(=O)NCC(CO)C3CC3)CCCC2)CC1 49826,C(=O)(C1=CS(=O)CCC1)NC1(CCNC(C2(C)CCN(C(C)=O)C2)=O)CCCC1 49827,Cn1cnc2ncnc(Nc3cccc(-c4ccc([N+](=O)[O-])c(Cl)c4)n3)c12 49828,C(=O)(CCCS(C)(=O)=O)NCC1(N(C(=O)CC(C)(C)C(F)F)C)CC2CCC1C2 49829,c1(C(C2(CCCCNC(CN(CCOC)C)=O)CC2)=O)ccn2nnnc2c1 49830,c1(CC(=O)NCC(=O)NCCC(C)NC(C2(C3CC3)CC2)=O)ccccc1 49831,CC1CCC(NC(=O)CCCCCN(C)C)CN1C(=O)CC1CCC(=O)N1C 49832,C1(C(CNC(C(C2CCCO2)OC)=O)=O)CC=CCC1 49833,c1(C(=O)NC(CNC(CCC(=O)NC)=O)(C)C2CC2)ccc2c(c1)C=CS2(=O)=O 49834,Cc1ccc(C(N2CC(F)(F)CC2C(=O)Nc2cc(F)cc(Cl)c2)=O)c(O)c1 49835,C1(CC(c2n(C(C)(C)C)nnn2)NCCc2ccoc2)CC2CCC1O2 49836,N1(CC)CCC1C(=O)N(C(CNC(C1(CO)CC1)=O)C1CC1)C.C1(C)CC1 49837,N1(C(CSc2ccc(C)cc2)=O)CC(NC(=O)C#CC2CCC2)C(C)(C)C1 49838,CC1(C)CC(NC(c2ccc(Cl)cc2N)=O)CN1C(C1CS(=O)C1)=O 49839,Brc1cc(OC(F)F)c(NCc2cccc(Br)n2)cn1 49840,c1(OC)ccc(C(=O)C(N2CCC(C(F)F)(CNC(=O)C3CC3)C2)=O)cc1Cl 49841,N1(C(C2CC(=O)NC2)=O)CCCC(C2CCN(C(=O)CCc3ccc[nH]3)C2)C1 49842,C1(NC(CNC(CC)=O)=O)CN(C(c2cccc(N)c2)=O)CCC1CO 49843,C1(CNC(C2(C)CC2)=O)CCN(C(=O)CCc2ccncn2)CC1 49844,c1(C(N(C)CCOCCNC(c2cc3n(n2)CCO3)=O)=O)cn2c(n1)CCCC2 49845,N(C(=NCCC1CC1(F)F)NCC1CCCSCC1)C(C)C 49846,N1(C(c2c(CC)occ2)=O)CCCC(C2CN(C(=O)C(C)OCCC(C)C)C2)C1 49847,CCCC(O)CC(=O)N(CCC(C)NC(c1occc1-c1ccc(F)cc1)=O)C 49848,N1(C(c2ccc(OC)cn2)=O)CCN(C(C2CC(C)(C)CCO2)=O)CC(CO)C1 49849,N1(C(c2cncc(C)c2)=O)CCN(C(c2ccc(C)nc2)=O)CC(O)C1 49850,C1(CNC(C=Cc2ccc(C)o2)=O)CN(C(c2cnn(CCF)c2)=O)CCN1C 49851,N1(S(c2c(OCC)ccc(F)c2)(=O)=O)CC2CC3CCCN3C2C1 49852,C12(NC(=O)Cc3cc[nH]n3)CCCC1CN(C(c1c(F)cncc1Cl)=O)C2 49853,Cc1cn2ccnc(C(=O)NC(C3CCN(C(=O)Cc4cc[nH]n4)CC3)C)c2n1 49854,c1(CCNC(C2C(OCC)C2)=O)ccc(CNC(C2CC3(CCC3)C2)=O)cc1 49855,C1(C(C)C)CC(O)CN1C(=O)Cc1ccn(Cn2cc(CNCC3CC3)nn2)n1 49856,C1(C)(C(N)=O)CC(F)(F)CN1C(=O)CC1CNC12CCC2 49857,C1(C(N2C(C)(C(=O)NC(CC)C(C)CN(C)C)CCC2)=O)CCC(F)(F)CC1 49858,c1(NC(C2(F)CN(C(C3CNC(=O)O3)=O)C2)=O)c(Br)cccc1[N+](=O)[O-] 49859,c1(OCC=C)ccc(CC(N)=O)cc1.C1(C(C)C)CSCC(=O)N1.C1(=O)CN1 49860,Cc1nsc(C(=O)N(CCCN(C(=O)C(C)Cn2ccnc2)C)C)c1Br 49861,CC(C)(C#N)CCCC(=O)NOC(CC(C)C)C(=O)N1CCCCCC1 49862,c1(CC)cnccc1C(=O)NCC1CCN(C(C2CS(=O)(=O)C2)=O)C1 49863,CC(C(=O)NCCC1CCCN1C(=O)C(F)C1(O)CCC1)C(F)(F)C(F)F 49864,C(C(=O)NOC(CO)C(C)C)(C1CCCC1)NC(CCc1cc(C(=O)OC)no1)=O 49865,C1(CNC(C(CC)(C)C(N)=O)=O)CCN(C(=O)C2=NOC(C)(C)C2)CCC1(F)F 49866,c1(C(=O)NC(C(C)C)CNC(c2ncsc2C2CC2)=O)ccc(Br)cn1 49867,C(C(O)C(=O)NCC1(N(C(C2(C3CCCCO3)CC2)=O)C2CC2)CCOC1)N(C)C 49868,Cc1nn(CC(=O)N(CC(C)NC(c2n[nH]c(C)c2F)=O)C)cc1Cl 49869,C12(C(N(C3CCN(C(C(C(C)C)F)=O)C3)C)=O)C3CC(CC13)C2(F)F 49870,c1(C(=O)NCC2C(CNC(c3cc(SC)oc3)=O)C2)cnc2n1CC(C)CC2 49871,CC1(C)OCC(CCN=C(NCC2CCCO2)NC2CC2)CO1 49872,C(CS(=O)(=O)NC1CNC1)N(C(=O)CC1CCCC1)C 49873,C(=O)(CCCS(N)(=O)=O)N1CC(N(C(C(c2ccccc2)C)=O)C)C(O)C1 49874,C1(C(=O)NC2CCCC(NC(c3c(C)cc(F)s3)=O)C2)CC2C(C1)C2(F)F 49875,N1(C(CN(C(C(c2cnn(C)c2)OC)=O)C)=O)CCN(C(=O)COC(C)=O)CC1 49876,CCCC(C)(CCC)C(=O)NC(C)CN(C(=O)C(=Cc1ccncc1)C)C 49877,Cc1ccc(CNC(C2(CCNC(C3CN(C(C)C)C3)=O)CC2)=O)cc1C 49878,c1(CCC(=O)N(CCCOCCN(C(CSCC#C)=O)C)C)ccccc1Cl 49879,C1(C(=O)NC(CN(C(=O)CCNC(C)=O)CC)C)CC(F)CN1C 49880,c1(OC)noc(C)c1C(=O)NC1COCCC1NC(C1(C2CCCO2)CCC1)=O 49881,CCC(C(=O)NC1COCC1CNC(=O)CNC(c1ccoc1)=O)OC 49882,C1(C(=O)NCCCN(C)C(C2(C)CCN(C)C2=O)=O)COc2ccc(F)cc2C1 49883,C(C(=O)NNC(=O)c1cccc(Cl)c1F)C1CCN(C(=O)OC(C)(C)C)C1 49884,S(=O)(=O)(c1ccnc(C(F)F)c1)N1CCCC(C(C)=O)C1 49885,C1(CNC(CSCCCC)=O)N(C(=O)C(C)C(=O)OC)CCCC1(C)C 49886,CC(CC(=O)NCCC1(NC(=O)C(C)SCc2ccccc2)CC1)CC(C)(C)C 49887,CC(C)CCC(C(=O)NCC(CO)C(C)C)NC(=O)CCN(C)CCO 49888,c1(C(=O)NC(CNC(c2c(C)ccnn2)=O)C)cn2cccc(F)c2n1 49889,CCCC(CC)CCC(=O)NC1C2CC1N(C(=O)CCc1ccc(N)c(F)c1)C2 49890,C(=O)(C(C)(C)Cc1ccccc1)N(C(c1nnc(C)s1)(C)C)CCC#N 49891,c1(C2(NC(N(CC(C)(C)OC)C)=O)CCCC2)ccc(Br)cc1 49892,C(=O)(C(C)CC(F)F)N1C(C(C)NC(c2cc(OC(F)F)ccn2)=O)CCC1 49893,C(c1cnco1)=CC(=O)NC(c1cocn1)C 49894,C#CCCC(C(=O)NCC(F)(F)C(N)=O)NC(c1cnc(O)cc1C)=O 49895,c1(OC)cccnc1C(=O)NCCn1cc(CNC(C2CN(CC(C)C)C2)=O)nn1 49896,c1(CNC(c2n(CCC)nnn2)c2nnc(COC)s2)c(Cl)cnc(F)c1Cl 49897,C1(CNC(C=CCCC(C)C)=O)CC2(CC2)CN1C(=O)COCc1cccnc1 49898,N1(C(CN(C(=O)CC(O)C(C)C)CCC)=O)CCC(C)(C)C1C 49899,N1(C(C2C(C)C2)=O)CC2(C1)CN(C(C1CCC(=O)N(C)C1)=O)CC2CO 49900,Cc1cnncc1C(=O)NCC(C1CCC1)NC(=O)C(C)Cc1cccc(Cl)c1 49901,C1(OC)CN(C(=O)C=CSc2nc[nH]n2)CC1NC(c1cnn[nH]1)=O 49902,C(=O)(C(C)C(C)NC(=O)CCN1CCCC1=O)N(C)CC1C(C)OCC1 49903,n1(C(C)C)nnnc1C(c1ccn(C)n1)NCC1CCC(=O)O1 49904,c1(C(N(CCN(C(c2ccc(C=C)cc2)=O)CC)CC)=O)ccc2n[nH]cc2n1 49905,CCC(C)(Cl)CNC(c1cn(CCNC(c2ccsc2Cl)=O)nn1)=O 49906,C1(CCNC(C2CN(C(N)=O)C2)=O)CN(C(c2nnsc2C(N)=O)=O)CCO1 49907,N1(C(C(c2cccc(Cl)c2)C)=O)CCCC(NC(=O)CC2CCC(=O)N2)CC1 49908,c1(C(N(C(C)CNC(=O)CSc2nc[nH]n2)CC)=O)cnsc1 49909,CC1CC(NC(=O)C(C)(C)CC2CC2)CN(C(=O)Cc2cncn2C2CC2)C1 49910,C1(NC(C(c2cnn(C)c2)OC)=O)CC12CC(NC(=O)CCCC1CCCC1)C2 49911,CC1(CNC(=O)Cc2ccc(Cl)s2)COCCN(C(=O)CN(C)C2CC2)C1 49912,C=CCC(C)(C)C(=O)NCC1(C)CCN(C(C2CCCN2C(C2CCC2)=O)=O)C1 49913,Cc1cnn(C)c1C(=O)NC1CCCC1NC(=O)CSc1c(C)n[nH]c1C 49914,C12COC3(CCN(CC3)C1)C2.c1(C(=O)OCC)nc[nH]c1NCc1cc(Br)cs1 49915,C1(N(C(C(CCC)OC)=O)C)CC2CCC(C1)N2C(c1ocnc1C)=O 49916,c1(C(N2CCCC2C(C)(C)C)C(=O)NCCOCC)cnc(Br)n1C 49917,Cc1c(C(=O)N(CCCN(C)C(c2cccc(CO)n2)=O)C)c[nH]c2nccc1-2 49918,N1(C(C2CN(C)C2)=O)CC(C)(C)CC1C(=O)NCC(O)CO 49919,N1(C(c2cncc(CC)c2)C(=O)NC(C)(C)C)CCN(C)C2CC12 49920,[N-]=[N+]=NCC(C(=O)NCCN1CCC1)NC(c1nnsc1N)=O 49921,C1(NC(C2(CC)CC2)=O)CCC2CCN(C(=O)C(c3ccc(C)cc3)C)C12 49922,C1(NC(Cc2n(CC)cnc2)=O)CCCC(N)CC1 49923,N1(C(c2c(C)occ2)=O)CC(NC(=O)C(c2cccc(F)c2)F)C(C)C1 49924,c1(OC)cc(C)cc(CNC2CN(C(=O)C(=O)NC3CCCCCC3C)C2)c1O 49925,C(CCC(C(=O)N1CCC(N(C)C)CC1)NC(C1CC1(F)Cl)=O)OC 49926,N1(C(C(C2CCOC2)OC)=O)CC(NC(c2ccc[n+]([O-])c2)=O)C2CCCC12 49927,N1(C(CC(C)(C)O)=O)CCC2(CCN(c3ccnc(C4CC4)c3)C2)C1 49928,c1(OC)ccc2[nH]c(C(=O)NCCN(C(=O)C(C)CCCC(C)C)C(C)C)cc2n1 49929,c1(C(N2C(C)C(NC(=O)CCCC(F)F)CCC2)=O)cnc([N+](=O)[O-])n1C 49930,CC1CN(C(=O)C2=CCCC2)CC(C)N(C(c2cc(Cl)cc(Br)c2)=O)C1 49931,C=CCC(C)C(=O)N1CCC(C(C)C(N2CCC(CCO)CC2)=O)C1 49932,C1(CNC(=O)COC2CN(C(=O)CCC3CC3)C2)CC2(CCCO2)C1 49933,Cc1cc2ccccc2n1CC(=O)NC1(C)CCN(C(C2(C)CCN(C)C2)=O)C1 49934,Nc1cc(CN(CCCCCCO)c2ccccc2)cc(F)c1 49935,S(=O)(=O)(c1cccc(=NCc2ccc3sccc3c2)[nH]1)NC(c1ccc(Cl)s1)C 49936,N1(C(C=C(CCC)C)=O)CCc2nc(CNC(=O)CC3(C)CC3(F)Cl)sc2C1 49937,CC1CCN(C(C2CCCN(C(c3ccc(C#N)cc3)=O)C2)=O)CC(=O)N1 49938,c1(OCC)c(C(N2CC(C)(NC(c3c(C)cccc3Br)=O)C2)=O)cccc1F 49939,S(=O)(=O)(c1ccccc1Cl)NCC(=O)N(C1CC(NC(c2occ(C)c2)=O)C1)C 49940,c1(NCCCS(C(C)C)(=O)=O)[nH]c(=NC2CCSCCC2)nc2c1cnn2C 49941,N1(C(c2cncc(C(C)=O)c2)=O)CCC2C(NC(=O)C=C3CCC(C)CC3)CC12 49942,C1(C(=O)OC(C)C(=O)NCC(F)(F)F)C(C#N)C1(C)C 49943,c1(NC(CC2(C(F)(F)F)CC2)=O)cnnn1CC1CCN(C2CC2)C1 49944,C1(C(=O)NC2CC(C)(NC(C(CC)Sc3ccccc3)=O)C2)CC(F)CN1C 49945,C1(C(=O)NC(C2CCCC2O)C)CCCC1CNC(c1cc[nH]n1)=O 49946,c1(N2CC3(C(C(N4CCC(C)C4)=O)C3)C2)ncnc2[nH]cc(C#N)c12 49947,c1(CC)ccsc1C(=O)N(C)CC1CCN(C(C2CC3CC3C2)=O)C1 49948,Cc1nc2ccnn2cc1C(c1nc(CCC(C)F)n(-c2cnnn2C)n1)=O 49949,N1(C(C(C)C2CCC2)=O)CCC(CO)(CNC(c2ccnc(Cl)c2N)=O)CC1 49950,C1(C(=O)NCC(c2cccc(Cl)c2)NC(C2(OC)CCC2)=O)CC12CC2(F)F 49951,CCCC(C)C(=O)N1CCC(N(C(=O)C=C=C(C)C)C)CC1 49952,N1(C(c2c(CC)nn[nH]2)=O)CCC2(CC(C(N3CC(C(C)C)C4(CC4)C3)=O)C2)C1 49953,C1(C#N)(CNC(=O)NC(Cc2nc(C)[nH]n2)C)CCCC1 49954,CC1CCCCN1C(C1CC(NC(c2cc(Cl)cs2)=O)C(O)C1)=O 49955,CC1CC(=O)NCC1C(=O)NCC1CC(NC(c2cccc(Cl)n2)=O)C1 49956,c1(C(=O)NCC(C(C)(C)C)NC(CC(CC)C)=O)ccnc2c1CC(=O)N2 49957,C(CN=C(NCCN(C)C)N1CCC(C)C2(CCC2)C1)c1c(C)n[nH]c1 49958,N1(C(C(CC)CC)=O)CC2(C1)CN(C(C1CCC3(CC1)N=N3)=O)CC2CO 49959,Cc1cc(C(=O)NC(CC#C)C(=O)NCCCCF)cc(C)n1 49960,C12(C(=O)NC(CNC(C(C)OC3CCOC3)=O)C3CC3)CC(C)(CCO1)C2 49961,C1(NC(c2nccc(N)c2)=O)CC(C(=O)NCC(F)Br)C12CCC2 49962,CCCCC(C(=O)NCC(C)N(C)C(c1nc(C(F)(F)F)cs1)=O)C(C)C 49963,N1(C(CC(=C)C)=O)CCC2(CCCN(C(=O)C3=NOC(C(C)(C)C)C3)C2)C1 49964,C(=O)(CC1=NNC(=O)C1)NC1CCC(CCNC(Cc2n(C)ccc2)=O)C1 49965,CC#CCC(C(=O)NC1CCC12CCCC2)NC(C1CCC1COC)=O 49966,C(=O)(C(C)C(=O)NCc1ccoc1C(=O)NCC1CNC(=O)CO1)OCC 49967,C1(NC(C23CCC(OC)C2C3)=O)CN(C(=O)CC2CC3(CCO2)CC3)CCC1O 49968,S(=O)(=O)(c1ccc(C(=O)NCC2CC2NC(c2cnn(C3CC3)c2)=O)o1)NC 49969,N1(C(C23CC(COC)(OC2)C3)=O)CCCC(N(C)C(C2CCCO2)=O)CC1 49970,C1(CC=C)(NC(=O)C2=CCC2)CCN(C(c2ccc(CCC)cc2)=O)CC1 49971,c1(C(=O)NCC=C)nc(C(=O)NCCC(C)NC(C2COCC2COC)=O)cs1 49972,CC1(C)C(CC(=O)NC23CCCN(CC2)C3)CCN1C(=O)COc1ccsn1 49973,N1(C(C(COCC)C)=O)CC2CCC(C1)N2C(c1cccc(F)c1O)=O 49974,Cc1nc(C(C)C)sc1C(N1CC(NC(=O)C2=CCC2)CC1CO)=O 49975,c1(C(=O)NCC(C)N(C(COCCC)=O)C)sc(Cl)c(Cl)c1C.C(C)(=O)O 49976,c1(CC(=O)NCCC2(NC(c3cn(C(C)C)nn3)=O)CC2)ccc(F)cc1 49977,C1(C(C)NC(=O)CSCC(N)=O)CCCN1C(=O)CC1(C)CCCO1 49978,N1(C(c2c[nH]c(=NC)o2)=O)CC(C)(C)C(NC(=O)CC2(C)CCOC2)C(C)(C)C1 49979,C1(C(=O)N(C)SCC)(CO)CCN(C(=O)C(CSC)Sc2cncnc2)C1 49980,CC1=C(C(=O)NCC(C2CC2)N(C)C(c2c[nH]nc2C(C)(C)C)=O)CCCO1 49981,C(=O)(C(C)CCCOC)N1C(C(=O)NCCc2n(CC)cnn2)C=CC1 49982,Cc1c(Cl)c(NC(N2CC(c3cnn(C)c3)C(C)(C)C2)=O)nc2ccccc12 49983,CCCC(C)CCCC(=O)N1CCCC1C1CCN(C(c2ccc(C)nc2)=O)C1 49984,c1(OC)c(C(N2CCC(N(C)C(c3csc(SC)n3)=O)C2)=O)cccc1F 49985,c1(OC)cccc(CNC2CC2C(=O)Nc2cc(CO)on2)c1C 49986,c1(C(N2CCN(C(C3C(C)CC(=O)N3)=O)CC2)=O)ccnc(C#N)c1 49987,CCCC(C(=O)NC(CN(C(=O)C=Cc1cnc(C(C)(C)C)s1)CC)CC)C(C)C 49988,N1(C(CCC(CC)C)=O)CCC2CN(C(C3CCN(C(N)=O)CC3)=O)CC2CC1 49989,N1(C(C2=NC=C2C(=O)OC)=O)CCN(C(c2ccon2)=O)C(CC(F)(F)F)C1 49990,C(=O)(C1=NOC(C)C1)N1C(COC)CCCC1 49991,C(CCC(C)C(c1nnnn1C1COC1)NCCOCc1ncoc1C)=C(C)C 49992,CC(CNCc1cc(C2CC2)n[nH]1)CC(F)F 49993,c1(CC(=O)NC2(C3CCCCN3C(=O)Cc3nc[nH]n3)CC2)cccc(Cl)c1O 49994,c1(CCCC)ccc(C2(NCC3N(C(c4cc[nH]c(=N)c4)=O)CC3)CC2)cc1 49995,N(C(=NCCN1CC2CCC1C2)NCCN1CCCC1)Cc1[nH]cc(C#N)c1 49996,O=C(C1=CCC(NC(c2n[nH]c(O)n2)=O)C1)NCCCCO 49997,CCCC(F)(F)C(=O)NCCCCC(C)NC(=O)CCOc1ccc(C)c(C)c1 49998,C(=O)(C(C)(C)C(=O)NCC1CC(NC(=O)C(C(C)C)n2cc(Br)cn2)C1)OC 49999,N1(CC2N(C)CCNC2)CC(=O)N(Cc2c(I)ccnc2O)C1=O 50000,C12(NC(CCCOC(C)=O)=O)CCC(CC1)N(C(C)=O)C2 50001,c1(C(N(C2CCCN(C(=O)CCc3cocn3)C2)CC)=O)cc(F)cnc1O 50002,C1(CNC(CCC(C)OC)=O)(NC(C2CCC(F)(F)C2)=O)Cc2ccccc2C1 50003,c1(CSCCC(=O)NCC(CO)NC(C2N(CC)CC2)=O)n[nH]c(C)n1 50004,C12(NC(c3cc(C(C)C)no3)=O)CCC(CC1NC(c1csnn1)=O)C2 50005,c1(SCC(=O)NCC(CNC(CCOCCCC)=O)C)nnnn1C1CC1 50006,Cn1cc(C(=O)NCCOCCNC(=O)CCc2cccnc2F)c(C(F)F)n1 50007,C1(NC(=O)C=C2CCCC2)CCC2CCN(C(=O)Cc3coc(C4CC4)n3)C12 50008,CC(CN(C)C)CN=c1[nH]c(=NCC2CC23CCOCC3)[nH]c2c1CCCCC2 50009,c1(C(=O)NCC23CC(NC(CC(CC)C)=O)(C2)C3)c(F)ccc(C(F)F)c1Cl 50010,C(CC(C(=O)N1CC(CF)C1)NC(=O)C=CCn1cncn1)SC 50011,CC1CN(C(c2cnccc2Cl)=O)CC(CCNC(=O)CCn2cccn2)O1 50012,CCCCC(CN(CCNC(C1(C)CCC1)=O)C(c1ccc(Br)s1)=O)CC 50013,CC(C(=O)N1CCC(C(C)(C)C)(CNC(=O)C(CO)NC(N)=O)C1)S(N)(=O)=O 50014,CC#CCCCC(=O)NNC(=O)CC(c1ccc(N2CCOCC2)nc1)=O 50015,N1(C(C(=Cc2cn[nH]c2)C)=O)CCN(C(c2csc(CC(C)C)n2)=O)CCC1C 50016,N1(C(C(=CC2CCCC2)C)=O)CC2OCCN(C(=O)CCS(C)=O)C2C1 50017,CCCCC(F)C(=O)N(C1CCCN(C(c2cc(C3CC3)on2)=O)CC1)C 50018,C(=O)(CCC(C)S(C)(=O)=O)NC(CCCC)CNC(c1ncsc1CC)=O 50019,Cc1cc(CC(=O)NC2CC(C)(CNC(c3c(C)cccc3F)=O)C2)cc(F)c1 50020,Cc1ncc(C(N2CC(O)(C(F)C(=O)NCC3CCC3(F)F)C2)=O)c(=N)[nH]1 50021,c1(NC(C(C)NC2(C)CC2)=O)ccccc1C(c1nnnn1C)C1CCC1 50022,C(=O)(CCCCN1CCOCC1)N1CC(OCC)(CNC(C2(OC)CCOC2)=O)C1 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50040,C(=O)(CCC(C)(C)N(C)C)NC(C1C=CCCC1)C(N1CCC(C)(OCC)C1)=O 50041,c1(C(N(C(C)CCNC(c2nonc2N)=O)C)=O)ccc(Br)c(N)c1 50042,C1(C(=O)NCCCCC=C)CN(C(=O)C(CC(=C)C)OC)CC1(C)C 50043,S(=O)(=O)(c1cc(CCN=c2nc(SC)[nH]s2)c(C)o1)N(C(=O)OC(C)(C)C)CC 50044,C(=O)(CS(=O)(=O)N1CCN(CCCNC(C2(C)CC2F)=O)CC1)OCC 50045,N1(C(c2ccnc(C)n2)=O)CCC(C)CC1CNC(=O)COCCF 50046,C1(C)(CNC(C)=O)CCN(c2nnnn2CC2COC(C)(C)O2)CC1 50047,CN1CC(C(N2CC(CC(F)C(=O)NCC3CC(O)C(O)C3)C2)=O)CCC1=O 50048,c1(C(=O)NCC(CC)NC(C(CCC)O)=O)cccc(S(=O)(=O)NCCO)c1 50049,c1(CC(C(=O)N2C(c3onc(C)c3Cl)CCC2)C)c(C)nn(C)c1C 50050,C(=O)(CCS(=O)(=O)NCC1CCC(NC(CS(CC)=O)=O)CC1)NCCOC 50051,c1(C(C(N2C(C)CC(NC(C3CC(N(C)CCO)C3)=O)C2)=O)C)ccc(F)c(F)c1 50052,c1(C(=O)NCCCC(C)NC(C2(CC#C)CCOC2)=O)cc(C2CC2)cc(F)c1 50053,N1(C(c2cc(C(F)F)[nH]n2)=O)CCN(C(C2CC(n3ccnn3)C2)=O)CC1 50054,c1(OC)cccc(C(=O)NC(CNC(=O)CC23CC(C2)C3)CO)c1OC 50055,CS(=O)(=O)c1ccccc1CN1CC2C(C1C(N1CCOC(CO)C1)=O)C2(C)C 50056,C(=O)(C1CCc2cc(Cl)ccc21)N1CC=CC(NC(c2nc(C)n(C)c2)=O)C1 50057,c1(C(=O)NCC2CN(C(C(CC=C)NC(C)=O)=O)C2)cc2nc(OC)ccc2[nH]1 50058,C1(NC(c2ccc(C)s2)=O)CC(NC(C2CCC3(CCC3)C2)=O)C12CCC2 50059,C1(CNC(c2ccc(Cl)o2)c2nnnn2CC2CCCO2)CCCCCC1 50060,c1(-c2c(C(N3CCC(NC(CCC=C)=O)C3C)=O)nco2)ccc2c(n1)CCCC2 50061,C(CCCCNC(C1CC1(F)Cl)=O)N(C(C)C)C(c1ccc[nH]1)=O 50062,c1(CNC(c2c(C)snc2)=O)cccc(NC(C2CCCCC2C)=O)c1 50063,c1(C(=O)NC2CCN(C(COCC)=O)C2(C)C)cc2c(Br)c(C)ccc2[nH]1 50064,C1(C(N(CCCNC(c2ccc(C(=O)OC)cn2)=O)C(C)C)=O)CC1C1CCCC1 50065,N1(C(CCSC)=O)CCC(C)CC1CNC(c1ccc(C(F)(F)F)c(F)c1)=O 50066,C1(C(=O)NC(CCC(=O)OC)C)CN(C(=O)CCCCSC)CCC1(C)C 50067,C1(C=O)CC2CC1CC2O.N1(N2C(C=O)CSC2c2ccco2)CC2CC2(CO)C1 50068,c1(SC)ccc(Br)cc1C(=O)NC1CC(NC(=O)CC2CCOCC2)C1 50069,c1(N2C3CN(C(C(C(C)C)NC(C)C)=O)C(C3)C2)ccc(Cl)cc1Cl 50070,C1(NC(CCN(C)CC)=O)CCCN(C(c2cc(C)n(C(C)C3CC3)n2)=O)C1C 50071,CCCCC(C)(F)C(=O)NCC1CC(NC(=O)CC2(N(C)C)CCCC2)CCO1 50072,Cc1onc(Cl)c1C(N1CC2C(CNC(c3snc(Cl)c3Cl)=O)C2C1)=O 50073,N1(CC(C)C)CC(C(N2CCC2)=O)CC1=O.N1(CC(=O)NC(=O)C2CC2)CCNC(=O)C1 50074,C1(NC(C=C(C)C(C)C)=O)C2CC1N(C(=O)Cn1cc(C)cn1)C2 50075,C1(CNC(CCCN(C)C(C2(C3CC3)CC(=O)C2)=O)=O)CC2CCCC2C1 50076,c1(C(N2CCCC(CCNC(C(COCC)(C)C)=O)C2)=O)cnc2scc(C)n12 50077,N(S(=O)(=O)N1CCC2(CCCC2)C1)C(C1CC(CC)OCC1)=O 50078,C1(C2CC2)(C(=O)NCCCN(C)C)CN(C(c2ccc(Cl)cn2)=O)C1 50079,N12CCC(N=[N+]=[N-])(C1)C2=O.CCS(=O)CCNS(=O)(=O)Cc1ccccc1 50080,N1(C(C(C)OC)=O)CC2(CC(NC(c3cn4cc(C)ccc4n3)=O)CO2)C1 50081,C1(C(=O)NCC2N(C(c3n[nH]c(CC)c3Cl)=O)CC(O)C2)CCOC(C)(C)C1 50082,c1(CC)nc(C)c(C(=O)N(CCC(C)C)C2CC2)s1.C12CCCN1C2=O 50083,N1(C(CCCC#C)=O)CC2CCC(NC(c3nn(C)c4ccccc34)=O)CC2C1 50084,C12(CCOC1)C(=O)O2.c1(NC(C=CC)=O)ccccc1 50085,C1(CNC(CCC2C(C)(C)C2)=O)(NC(c2ccc(=N)[nH]n2)=O)CCCCC1 50086,C1(C(=O)NCC(C(C)(C)C)NC(c2c(CC)c[nH]c2)=O)CCCCC(=O)N1 50087,c1(OC)cc(OC)c(OC)cc1-c1ccc(C)c(OCc2ccncc2C)c1 50088,CC(CCNS(=O)(=O)Cc1ccc(C(=O)O)cc1)S(C)=O 50089,N1(C)CCC(C2(OC)CC2)CC1.c1(OC)nscc1CNC(=O)C(F)CC1CC1 50090,c1(OCC)ccc2c(c1)C(C(=O)NCCc1ccc(C(C)(F)F)cc1)CC2 50091,n1(CC)cc(C(=O)NC2CN(C(=O)CN3CCN(C)CC3)C2)c(C(C)C)n1 50092,C(=O)(C(CC(C)c1ccccc1)N(C)Cc1cccnc1)NCC(C)C 50093,C1(OC)CCCC(C(=O)NCCCN(C2CCCC2)C(c2cn(C)c(C)n2)=O)C1 50094,C(N=c1[nH]cnc(Cl)c1[N+](=O)[O-])C1C(NC(c2nccc(CO)n2)=O)CCCC1 50095,CCC(CC)CCC(=O)NCC1(C)CCN(C(=O)C(C)CNC(=O)OC(C)(C)C)C1 50096,C(=O)(C(F)C(=O)N(CCC(=O)N(C)CCN(C)C(C)=O)CC)OCC 50097,C(=O)(C(C)(CCC)CCC)NCCC(=C)CNC(=O)COC(=O)CO 50098,N1(C(c2n(CCC)nc(C)c2)=O)CCC2(CC2NC(=O)C(CC2CC2)OC)C1 50099,c1(C(=O)NC2CC(CCNC(CCSC)=O)C2)cc(SC2CCCC2)c[nH]1 50100,c1(OC)ncc(C(=O)N(C2CC3CC2N(C(=O)CSCC(C)C)C3)C)cc1Cl 50101,Cn1nc(Br)c2c(NCC(C3CC3)NC(c3ccc(Cl)cc3F)=O)ncnc12 50102,C(=O)(CCCC(C)(C)C#N)NC(C1(O)CCN(C(=O)CCS(C)(=O)=O)C1)C 50103,N1(C(CCCC#C)=O)CC2CCCC1C2CNC(=O)CC=C=C 50104,c1(COC)ncc(CNC(=O)C(=O)NC(C)(C)CC2CC2)c(=N)[nH]1 50105,c1(SC(c2nncn2C)C)ccncc1NCC(F)C1CCC1 50106,N1(C(c2cc(C#C)c(Cl)cc2)=O)CCC2(C1)CN(C(=O)CCOC(C)C)CCO2 50107,N1(C(C(C)C2CC2)=O)CC(C(N)=O)(CCO)C1.N12CCC(C1)C2 50108,Cc1cnc(NCc2csnn2)c(S(=O)(=O)NC2CC3CCCCC23)c1 50109,c1(C(N(CCN(C(=O)CC(C)(C)CC)CC)CC)=O)cc([N+](=O)[O-])c(C)cc1C 50110,c1(C(=O)NC2CC(CNC(C(C(C)c3ccccc3)O)=O)C2)ccnc(F)c1O 50111,C1(C)(NC(COCCC#C)=O)CCCN(C(=O)CC(CC)C2CC2)C1 50112,CC(C)C(O)C(C)(C)C(=O)NC1CN(C(=O)C=CS(C)=O)CC1C1CC1 50113,c1(NC(=O)OC(C)(C)C)cccc([N+](=O)[O-])c1.C1(NCCSC)CC2CN(C1)C2 50114,C1(NC(CCC(=O)NC)=O)CC(NC(=O)C(Cc2ccsc2)NC=O)C1(C)C 50115,N1(C(C(=O)N(C)C)=O)C2CCC1CC(CNC(C13CCCC(CO)(C1)C3)=O)C2 50116,N1(C(CSCCC)=O)CCC(C(F)(F)F)CC1CNC(C1COCCN1C)=O 50117,C1(C(=O)NC(C(C)C)CCN(C)C(C2CCC(=O)NC2)=O)CC1C1CCCCC1 50118,C(=O)(CCCCCCN=[N+]=[N-])NC1C(CNC(C2(C)CC(C)(C)C2)=O)COC1 50119,Cc1ccc(C(O)C(N2CCCC(NC(c3ccc(Cl)nc3)=O)C2)=O)cc1 50120,CC(CN(C)C)CC(=O)NCC1C2CC1N(C(C1COCCN1C)=O)C2 50121,N1(C(C(CC)(C)C(N)=O)=O)CCCCC(CNC(c2ccon2)=O)CC1 50122,c1(C(CNC2CC(CNC(CC#C)=O)C2)=O)cc(OC(C)C)c(OC)c(OC)c1 50123,C1(CC#C)(C(=O)NCC(O)C(F)F)CCN(C(=O)CCCC#N)C1 50124,c1(C(C(=O)NC(C(=O)OC)C)N(C2CCC2)Cc2cc[nH]n2)nc(C#N)cs1 50125,Cc1cc(C(=O)NC2(CNc3ncnc(Cl)c3C(C)=O)CCC2)nc(C)c1 50126,Cc1cnc2c(C(=O)NC3CC(C)(Oc4ccccc4)C3(C)C)nccc2c1 50127,C(C)(C)(CC(F)C(=O)NC1(c2ncc(C)o2)CC1)NC(c1c(CC)nn(C)c1)=O 50128,c1(C(N2C(CNC(c3nccc(C)c3)=O)C(C)CC2)=O)cc2c(ncn2C)[nH]1 50129,C1(NC(c2sc(C)c(O)n2)=O)CC2CC(C1)N(C(C1(C)CCCCC1)=O)C2 50130,c1(CC)nc(C(=O)NCC2C(NC(=O)Cc3cnnn3C)CC2O)co1 50131,c1(-n2cc(CN3CCCC(NC(c4ccns4)=O)C3)nn2)ccc2c(c1)CCO2 50132,C(=O)(C(C)(F)F)NCC(C)CN(C)C(c1ccc(CSC(F)F)o1)=O 50133,CC1CN(C(c2csc(C(F)F)c2)=O)CCCN1C(c1ncoc1C(F)(F)F)=O 50134,CC(CCCNC(c1nc(Cl)cs1)=O)NC(=O)C(C)(C)c1cncs1 50135,C1(COC)(NC(=O)CC2CCCC2C)CN(C(c2ccn(C)c2)=O)C1 50136,C(C)(CNC(c1ccn(C)n1)=O)(C(C)C)NC(C(=O)NCC)=O 50137,c1(OC)ccc(N)c(C(N2CCOCC2CNC(=O)Cc2cc(Cl)n(C)n2)=O)c1 50138,C1(C(=O)N(CCCCN2CCOCC2)CCl)CC12CCN(C(C1CCCO1)=O)CC2 50139,CC1N(C(C2N(C(c3ccc[n+]([O-])c3)=O)CCC2(C)C)=O)CCOC1(C)C 50140,c1(C(N2CCC(N(C(C(CC(C)C)C)=O)CCO)C2)=O)nn2cccnc2c1Cl 50141,Cc1cnc(CC(=O)N(C)CC2CCCN2C(=O)C(F)C2CCC2)o1 50142,c1(C(N2CCCCC3CCC23)C(=O)NC2(C)CC2)ccc(F)c2ncccc12 50143,C1(CC)CNC(=O)CN1C(=O)CC1CN(C(=O)Cc2cccc(C)c2)CC1C 50144,CC1(C)CN(C(c2ccc(C#N)[nH]2)=O)CC1C(=O)NCc1nc(O)n[nH]1 50145,Cc1ccc(Cl)cc1OCC(N1CC(NC(c2ccoc2)=O)CC(C)C1)=O 50146,C(=O)(C1=CNC2=NCCC2=C1)N(CCCOCCN(C)C(C1CCS1(=O)=O)=O)C 50147,CN1CCC(CC(=O)NCCCC2CCN(C(=O)C(O)c3ccco3)CC2)C1=O 50148,C1(C)(CNC(CN2CCC(C)CC2)=O)COCCN(C(c2cnsn2)=O)C1 50149,C(=O)(CCC(=O)NCC(CC)N(C)C(C1CCCN1c1ncccn1)=O)OCC 50150,C(=O)(C1=COc2ccccc2O1)N(C)CCN(C(=O)NC12CCCCC1C2)CCO 50151,c1(C2CC2)ncccn1.C(C(=O)N1CC(C(F)(F)F)C1)(C1CCCC1)NC(=O)C1CC1 50152,CC1CN(Cc2cccc(-c3ccccc3)n2)CCN1C(c1cccc(O)n1)=O 50153,N1(Cc2n(CC)cnc2)CC(C(N2CCC(NC)C2C(C)C)=O)C2(CC2)C1 50154,C#CC1(C(=O)NC2CC3CCCCN3C2)CCN(C(c2c[nH]c(C#N)c2)=O)CC1 50155,c1(CC(C(=O)NCCN(C(C(CC)(C)F)=O)C2CC2)=O)c(C)nn(C)c1C 50156,C1(CC(=O)NCCN(C(=O)Cn2cc(C3CC3)cn2)CC)CCC(=O)NC1=O 50157,Cc1cc(I)c(Cl)cc1NC(C1C(O)CCN1C(c1cc(C#N)ccc1Cl)=O)=O 50158,C(=O)(C(C)(C)C(=O)N1CCOCC(C(N2CCN(C)C(CO)C2)=O)C1)OC 50159,N1(C(c2c(CC)cns2)=O)CCN(C(=O)CC2CC(=O)C2)C(C2CC2)C1 50160,CCCC(C(=O)NCCC1CN(C(c2cc(C(F)(F)F)nn2CC)=O)C1)C(C)C 50161,C(CCCC(=O)NC1CCC(NC(C2(C)CSC2)=O)C1)SC 50162,C(=O)(CC(C(F)(F)F)N(C)CC1(COC)CN(C(C2CC2F)=O)C1)OC 50163,N1(C(C(CCC)NC(N)=O)=O)CCC(C(=O)NCc2nnn(C)n2)=C(F)C1 50164,C1(CNC(C(C)C(=O)N2CCOCC2)=O)CN(C(=O)CC2(CO)CC2)CC1(C)C 50165,CC1Cc2cc(N)ccc2CN1C(c1c(Br)ccc(F)c1N)=O 50166,CN1C(=O)CSC1=CC(=O)NC1CCC1NC(C1CC2(C1)CC21CC1)=O 50167,Cc1ncc(C=CC(N2CCC3CN(C(c4cc(C)c(C)o4)=O)CC23)=O)c(O)n1 50168,N1(C(c2cn(CC)nn2)=O)C2CCC1CC(CCNC(c1ccc[n+]([O-])c1)=O)C2 50169,Cc1ccc(C23CC(C(=O)NCCC(O)CNC(=O)C(C)O)(C2)C3)s1 50170,c1(CC(=O)NCC(C)N(C(=O)Cc2nccn2C)CC)ncc(F)cn1 50171,C1(OCC2(CC)CCC2)CCn2cncc2C1.c12cn(nn1)CC(=O)N2 50172,C1(COCC)CCN(C(c2cccc(Br)c2Cl)C(=O)NCCCSC)C1(C)C 50173,c1(C(=O)NC(CC)(C)CNC(C2C(C)(C)C2(F)F)=O)ccc2c(c1)OCC2 50174,N1(C(C(C=CCCC)O)=O)CCN(C(=O)Cn2ccc(=N)[nH]2)C2CC12 50175,CC1CC(C(=O)NC)CN1C(C1(C(=O)OC(C)(C)C)CC1)=O.C(=O)(C(F)F)NC1CCC1 50176,N1(C(c2c(OC)cccc2Cl)=O)CCC2(CC(C(=O)NCCCCO)CO2)C1 50177,c1(CCN=C(NC(C=C)C)NCC2(OCCO)CC2)nnc2n1CCCC2 50178,c1(OC)ccc2c(c1)OCC2C(=O)N1CCC(C)C(F)(F)CC1 50179,C(=O)(CCC[N+](=O)[O-])OCN1CCCC(C(C(C)Oc2cccc(F)c2)=O)C1 50180,c1(C(=O)NC(CNC(CNS(CC)(=O)=O)=O)(C)C2CCC2)cccc(F)c1Cl 50181,CC1(C)OCCC1C(=O)NC(C(=O)NC1(CF)CCCC1)c1ccco1 50182,CS(=O)(=O)C1CCC(CNC(=O)C(=O)NC2CCC(F)(F)CC2)CC1 50183,C1(CC(C)C)C(=O)NCc2ccoc2C(=O)NO1.N1(OC)CC(CO)OC(C)C1 50184,CC(C)CC(C)(O)C(=O)N1CCN(CCNC(=O)CC(=O)NC2CC2)CC1 50185,c1(C(=O)NCCNC(c2cc(C)n(C3CC3)n2)=O)c[nH]c2cccc([N+](=O)[O-])c12 50186,CCC(CC(=O)N1CCN(C(=O)C(=Cc2cccnc2)C)C2(CC2)C1)C(F)F 50187,c12c(cc(OC)cc1O)NC(=O)C1CCCN(C1)C2=O.c1(COC)ncnn1C 50188,c1(OC)cc(C(=O)NC2CCCC2NC(=O)CC2CC2(Cl)Cl)cc2c1OCC2 50189,C(=O)(CC1OCCc2ccsc21)NCC1C(C)CCCN1C(=O)CN1CCCC1 50190,CC1CCN(CC(=O)Nc2ccnc(CNC(=O)Cc3cccnc3O)c2)CC1 50191,N1(C(C=C(C)C(C)(C)C)=O)CCOC(CCNC(=O)CN2CC(C)C2)C1 50192,Cc1cc(CCC(=O)NCC2CC(NC(c3cnsn3)=O)C(O)C2)nn1C 50193,c1(C(=O)NCC(C2CC2)OC)cn(C2CN(C(=O)C=CC3CCCC3)C2)nn1 50194,C12(NC(C=C(C)C3CCCCC3)=O)CCCCCC1N(C(C1CC1CF)=O)CC2 50195,c1(CN(C)CC2CN(C(C3CC3F)=O)C2)cc2ccc(Br)cc2[nH]1 50196,Cc1cncc([N+](=O)[O-])c1N(CC(C)CNC(C1CCn2ncnc2C1)=O)C 50197,Cn1c(C(N2CCOC3C(O)CC23)=O)cc(=O)n(C)c1=O 50198,c1(C=O)ccc(OC)cc1Cl.N12CC(C(C)C1)N2C.C(CCC(=O)NC1CC1)OCC 50199,c1(CC)ncc(C(N2CCC(CF)(NC(=O)CC3COC(C)(C)C3)C2)=O)c(C)n1 50200,C1(CNC(C(CC#C)OCC2(C)N=NOC2)=O)CN(C(c2ccc(Cl)[nH]2)=O)CC12CCC2 50201,CCC(C(=O)NC(C)(C)C=CC(=O)NC(C)CC1CCC1)n1cncn1 50202,c1(-n2c(C3C(CC)C3)nc(C3CC3(C)C)n2)ccc(C)cc1OC 50203,CCC(C)CC(=O)C(=O)N(C(C)C(=O)NCCc1cc(C)on1)C1CC1 50204,C1(C(N2CC(COC)(NC(C3(F)CCOCC3)=O)C2)=O)(OC)CCOCC1 50205,C1(NC(C2CC(O)(CC#C)C2)=O)CC(Cc2ncc(OCOCC)cn2)C1(C)C 50206,c12cn3c(c1C)N(CCC3)C(=O)c1cccc(c1)C1(CC1)C(=O)C(=O)C2.CO 50207,S(=O)(=O)(c1nc(N2CCC(C(C)(C)C)CC2)ccc1Br)N(C(CC)CO)C 50208,c1(C(=O)NCC2(C)CCN(C(C3CCCCO3)=O)C2)ccc2cnsc2c1 50209,N1(C(C2C(=C)C2)=O)CCCCCC1CNC(c1cc(C(C)C)nn1C)=O 50210,C1(CC(=O)NCCCNC(c2cc(Cc3cccs3)on2)=O)CCCCO1 50211,c1(CC(=O)NC(CC)CNC(=O)CCN2C(=O)CCC2=O)ccccc1SCC 50212,c1(C(=O)Nc2c(C(N(C)Cc3ccc(CC)cc3)=O)c[nH]n2)cc2occc2[nH]1 50213,c1(N(C(=O)C(=O)NCC(=O)Cc2ccccc2)C)ccccc1CC(C)(C)O 50214,C(=O)(C(C)C(O)CCCC)N(C1CCCN(C(CN(CCC#C)C)=O)C1)C 50215,Cc1ccc2nnnn2c1C.C(C(C)C(F)(F)F)c1nc(S)nn1-c1ncnn1C 50216,CCCCCCC(CC)C(=O)N(CCc1nnn2c1CCC2)CCOCCO 50217,C1(C(=O)OC2CC(C(CC)CC)OCC2)CC2(CCOCC2)CCO1 50218,N1(C(c2ccccc2F)=O)CCC(N(CCO)C(C23CCC2C3)=O)CC1 50219,N1(C(CCC(C)C)=O)CCN(C(=O)C(C)c2cccs2)CC1c1ccc(F)cc1 50220,N1(C(C2N(C(C(CC#C)O)=O)CCOC2C)=O)CC(C)OC2(CCC2)C1 50221,C1(C(=O)NCCC2N(C)CCC2)CCCC(NC(C2(CO)CCCC2)=O)CC1 50222,N1(C(CCNC(CC(C)C)=O)=O)CC(NC(C2CCCCC2C)=O)CC(C)C1 50223,C1(C(N2C(C(=O)NCCn3c(C)ncc3)C(C)C2)=O)CCCC(C)(C)C1 50224,C12(C(=O)NCC#CCNC(c3cc(C)nc(O)n3)=O)OCCCC1C2(F)F 50225,C1(CC(N)=O)CCCCN1S(=O)(=O)NCC(=O)N(C1CCNCC1)CCO 50226,c1(C(N2CCC(NC(c3c(C(C)C)[nH]cc3)=O)C(C)C2)=O)cccc2cnnn12 50227,c1(C(N2CCC(NC(C3CC34CCC4)=O)(CF)C2)=O)cc2c(Br)cccn2n1 50228,N1(C(CC2C(C)C2)=O)CCOCC2(COCCN2C(c2cn(CC3CC3)nn2)=O)C1 50229,CCS(=O)(=O)CC(=O)N1CCCCC1C1CCN(C(C2CC2F)=O)C1 50230,c1(NC(=O)Cc2ccn(C(F)F)n2)cc2c(cc1Br)CCC(=O)N2 50231,N1(C(C2C(CC)C2)=O)CCC(O)(CCNC(c2ccc(CC3CCC3)cc2)=O)C1 50232,CC1CN(C(C2C(C)(C)C2(C)C)=O)CC1NC(c1ccc(C(F)(F)F)o1)=O 50233,c1(CC)cnccc1C(N1CCOC(C(=O)NCC2COC(=O)N2)C1)=O 50234,N1(CC(CC(C)C)OCC(=O)O)CCNCC(O)C1 50235,c1(C(N(CC(C)(C)CNC(C2CCC(C)C2)=O)CC)=O)cn2c(n1)SCC2 50236,CC1(C)CCCCC1(C)NC(c1ccc(CNC(C2(C#N)CCC2)=O)nc1)=O 50237,N1(C(C2OCCC(C)C2)=O)CC2CN(C)CC(C1)O2 50238,c1(C(N(CCCNC(CC2CC(OC)C2)=O)C2CC2)=O)cnn2ccc(C)nc12 50239,CCN(Cc1ccccc1C(F)(F)F)N1CC(C(F)(F)C(F)(F)F)C(N)C1 50240,c1(C(=O)NCC=C2CCN(C(CC(C)C3CC3)=O)CC2)cc(Cl)cc([N+](=O)[O-])c1 50241,C1(NC(=O)CCCC2CCCC2)CC2(C1)CC2C(=O)NOC1CCOC1 50242,c1(C(=O)NCCCCCCO)cc2cc(-c3cnc4occc4c3)ccn2n1 50243,N1(C(CCCCC#C)=O)CCC2(CC1)CC2CNC(c1c[nH]ccc1=O)=O 50244,C1(C(N2C(C(=O)Nc3cnccn3)CCC2)=O)CCCN(CC(F)(F)F)C1=O 50245,N1(Cc2cccc(OC)c2)C(=O)CN(CCc2ccnn2C)C1=O 50246,CC1CN(C(=O)CCP(C)(C)=O)CC1(C)C(N1CCCC(CN=[N+]=[N-])C1)=O 50247,c1(COC)ccoc1C(=O)NC1(CC(=O)NC(c2noc(CO)n2)C)CCC1 50248,C(C)(CN=c1[nH]c2ccccc2cc1C#N)NC(C1CCC(C)CC1)=O 50249,c1(NC(C2CCN(C(=O)CCC3CCC3)CC2O)=O)cncc(Cl)c1Br 50250,C(=O)(C1=NOC2(CCC2)C1)NCC(CN(C)C(c1ncc(C(F)F)s1)=O)(C)C 50251,c1(CNC(C2(n3nccn3)CC2)=O)cccc(Cl)c1F.C12(CC1)C(=O)N2 50252,C1(NC(C(Cc2ccsc2)NC=O)=O)CC2CCC1N2C(=O)Cc1ccn(C)n1 50253,N1(C(CCCCOC)=O)CCC(C2CCN(C(=O)Cc3c[nH]ccc3=O)C2)CC1 50254,c1(C(=O)NC(C)C(C)(C)NC(=O)CNS(C)(=O)=O)cc2nc(O)[nH]c2cc1N 50255,Cc1ccncc1C(=O)N(CCN(C)Cc1cscc1F)CCN(C)C 50256,CCC(CC)C(F)C(=O)NCC(O)CNC(=O)Cn1cnc(=N)[nH]1 50257,Cc1ccc(Cl)c(C(N2CCC(O)C(NC(=O)C(C(C)(C)C)C3CCC3)C2)=O)c1 50258,c1(C(=O)NCC(CNC(c2cccs2)=O)CO)cccc2c1OCCC2 50259,c1(N2CCC(C(C)NC(c3cc(C4CC4)nn3C)=O)CC2)nn(C)cc1S(C)(=N)=O 50260,N#CC1(CC(=O)NCC(C2CC2)NC(=O)CCOC2CCOCC2)CCCCC1 50261,c1(C(c2nnnn2C(C)(C)C)NCC(CC)OC)nc(O)c2cnn(C)c2n1 50262,c1(NC(C23N(C(C(CCSC)OC)=O)CC(C)(C2)C3)=O)ccc2cc[nH]c2n1 50263,C1(C(N2CCC(CNC(CCC#C)=O)C23CC3)=O)CC12CCC1(CC1)CC2 50264,c1(C(N2CC3C(NC(c4ccn(C(C)(C)C)n4)=O)C3C2)=O)ccc(O)nc1Cl 50265,c1ccc2c(c1)cc(C)n2C.C1(CNC(COC)C)COC(C)(C)O1 50266,C(C1CN(C(=O)CC2CCN(C)C2=O)CC1C(=O)NCC(F)C1CCC1)=CC 50267,c1(NC(C2N(C(C(CC)NC)=O)C3C(C2)C3)=O)nnc2ccc(Cl)nn12 50268,O=C(NN1CC(N2C(=O)CCC2=O)C1)C1CC(=O)N(Cc2ccccc2)C1 50269,CCC(C)C(CC(=O)N1CC(O)C(C#N)C1)NC(=O)CS(C)(=O)=O 50270,c1(-c2ccc(N3CCN(C(=O)CNC4CC4)CC3)cc2F)cc(F)cc(F)c1O 50271,C(=O)(CCCC(=O)N1CC2C(CNC(c3csc(Cl)c3)=O)C2C1)NC 50272,c1(Nc2ccc(CS(=O)(=O)NC(C)C#N)cc2)ncnc2sc(Br)cc12 50273,c1(C(N(CC(CNC(CSCC(C)C)=O)C)C)=O)cc([N+](=O)[O-])c[nH]1 50274,c1(C(N2CC(CNC(C3=C(CC)OCCC3)=O)C2)=O)cccc2nc(O)n(C)c12 50275,c1(CNC(C2CCCN(C(=O)Cc3ccccc3Cl)C2)C)ncc(C#N)cc1Cl 50276,N1(C(C(COC)(C)OC)=O)CC2CC2(CNC(c2cnc(C(N)=O)s2)=O)C1 50277,Cc1cnc(C(=O)NCCCOCCNC(c2snnc2C)=O)c(C)c1 50278,C1(NC(=O)CCC2CCC(NC(C3CC4CCC3C4)=O)C2)CCC(C2CC2)C1 50279,C1(O)(C(C(=O)N(C)CC2(NC(C3(C)CC3)=O)CC2)F)CCCC1 50280,C1(NC(CCC(C)C)=O)CCCC2CN(C(c3cnc(C(C)C)nc3O)=O)CC12 50281,C1(C(=O)NCCCCNC(C(C)(C)c2cc[nH]n2)=O)CCCCC1F 50282,N1(C(C(C)NS(C)(=O)=O)=O)CCC(C(CO)NC(c2ccon2)=O)CC1 50283,C1(C(=O)NC(C2CCN(C(=O)C(c3ccccc3)C)C2)C)(CC)CCCC1 50284,n1(CC(=O)NC2(CO)CN(C(C(C)Cc3cnc[nH]3)=O)C2)cc2ncccc2n1 50285,N1(C(c2cccc(C)c2O)=O)CCCC2(NC(c3nnc(O)nc3O)=O)CC2C1 50286,C#CC(CC(C)C)NC(=O)CCN(C(=O)C(C)(C)CC)C(C)C 50287,CN1CCCC12CN(C(C1(C)CCCN1C(c1ccnc(O)c1F)=O)=O)C2 50288,c1(OC(C)C)ccc(C(N2CCN(CC3CC(O)C3)C3CC23)=O)c(O)c1 50289,C(CC(C(C)C)NC(c1cccc(C2CCC2)n1)=O)NC(C=CC)=O 50290,C1CN=C2N=C(N=CN2)N(C)C2CCC1C2.C1(C(=O)OCC)(COCC)CCC1 50291,C(=O)(C1CCCc2nccn21)N1CCN(C(c2cc(C)oc2)=O)CC(O)C1 50292,c1(CC(C)C)cccc(C(N2CCC(C(N)=O)(N(C)C)C2)C(=O)NC2CC2)c1F 50293,c1(OC)c(F)ccc(F)c1C(N1CC2CC2(NC(=O)COCC(F)F)C1)=O 50294,N1(C(Cc2c(C)ccnc2)=O)CC2(CC2)CC1C(=O)NC1(C2CCCO2)CC1 50295,c1(CC(=O)NC2CCC(CCC(=O)NC(c3nn[nH]n3)CC)C2)cc(C)nn1C 50296,C12(NC(c3[nH]c(=NC)sc3)=O)CCOC(CNC(=O)Cn3nccn3)(C1)C2 50297,c1(C(=O)NCC2(O)CN(C(C(C)NC(=O)NC)=O)C2)ccc2cc[nH]c2c1 50298,C1(CCOC)CCN(C(C2CC(CNC(=O)C(C3CC3)N(C)C)C2)=O)C1 50299,C1(CNC(C(C)N2CCC2)=O)COCCN(c2nnc(C(F)F)s2)C1 50300,c1(C(=O)NCCC2(O)CN(C(CC3C(C)OCC3)=O)C2)ccc(S(N)(=O)=O)cc1 50301,c1(C(=O)NC2C(NC(C(C)(C)OC)=O)CC(F)(F)C2)ccnc2[nH]cnc12 50302,c1(C(=O)NC(C)CC2CN(C(C3(C)COC3)=O)C2)ccnn1C1CCC1 50303,C1(CC)CCCCC1C(N1CC2C(CNC(=O)CCc3ccncc3)C2C1)=O 50304,C(C)(CCC(=O)N1CCOCC1CNC(=O)Cc1cccc(OC(F)F)c1)SC 50305,N1(C(CS(=O)(=O)NC)=O)CC(NC(C2CC3CCC3C2)=O)CC(O)C1 50306,N1(C(C(C)O)=O)CCCCC(N(C)C(c2cnnc(-c3ccccc3)c2)=O)C1 50307,N1(C(c2c(C)cn(C)n2)=O)C2CCCC1CC(NC(c1cn(C)[nH]c1=N)=O)C2 50308,N1(C(CCc2cc(C)no2)=O)CC(=O)NCC1C(=O)NCCNS(N)(=O)=O 50309,C1(C(=O)NCCCCC2CN(C(C3CCC(C(=O)OC)C3)=O)C2)CC12CCOC2 50310,N(C(=NCCC1(F)CC1)N1CCCC(O)CC1)C(COC)C 50311,C(C(C)C(C)C(=O)N1CC(CNC(=O)Cc2cccc(C)c2Cl)C(C)C1)OC 50312,CCC(C)CCC(=O)NN1CC2C(NC(=O)C(=O)Nc3ncc[nH]3)(C2)C1 50313,N1(C(C2(CC=C)CCC2)=O)CC2(C1)CN(C(=O)C(C1CCCCC1)F)C2 50314,N1(C(C(c2cccc(C)c2)C)=O)CCN(C(=O)Cc2ccco2)CC1C(C)C 50315,C1(CC(=O)NCC2(CC)CCCCO2)CN(C(=O)C=C2CCC2)CC12CC2 50316,N1(C(CCC)=O)CCN(C(C2CC=CCO2)=O)CCC1C 50317,C1(C(=O)N(C(C(C)C)C)C2CC2)(CNC(C2CC(OC(F)(F)F)C2)=O)CC12CCC2 50318,c1(C(=O)NCCC(CNC(COCC#C)=O)OC)ccc2c(n1)CCC2 50319,C1(NC(C(C)Cn2cccn2)=O)CC(F)CN(C(c2cn(C3CC3)nn2)=O)C1 50320,Cc1c[nH]cc1C(N1CCC(N(C)C(c2ccsc2-n2cnnn2)=O)C1)=O 50321,Cc1cnn2ccc(C(=O)NC3CCCN(C(=O)C#CC4(C)CCCO4)C3)nc12 50322,N1(C(C2CN(CC(C)C)C2)=O)CCOC2CN(C(c3ccn(CCF)n3)=O)CC12 50323,C(N(O)C(=O)C(O)Cn1cc(C2CC(F)(F)C2(F)F)nn1)N1C(=O)CCC1 50324,C=C(C)CCC(C(=O)N(C(CC)C(=O)OC)C)NC(=O)COCCCC 50325,N1(C(C(CCOC)C)=O)CC2CCC1C(CNC(c1cc(Cl)ccc1O)=O)C2 50326,n1(CC(=O)NCCCCC2CCCN2C(=O)Cc2ccccc2)cc(F)ccc1=O 50327,c1(C(N2CC3CN(C(Cn4ncc(C#C)c4)=O)C3CC2)=O)c([N+](=O)[O-])c(C)nn1C 50328,C=C(Cl)C(C)(C)C(=O)N1CC(CNC(=O)CCn2cc[nH]c(=O)c2=O)C(C)C1 50329,c1(C(N2CCCCC(NC(C(COC)OC)=O)CC2)=O)nc2n(c1Cl)CCCC2 50330,O=C1CC2(C1)CC(C(=O)NCc1ccc(C(N3CC(F)C(O)C3)=O)cc1)C2 50331,N1(C(C(C=CC)O)=O)CC2CCCC1C2CNC(=O)CN(c1ccccc1)C(C)=O 50332,Cc1occc1C(=O)NC(CNC(=O)C(C)SCc1ccccc1)C(C)C 50333,C1(CC)CCCN(C(c2cc(CNC(=O)CCc3ccn(C)n3)nn2C)=O)CC1 50334,c1(C(N2CC(C(C)C(N3CC(O)C(F)C3)=O)C2)=O)ccn2nccc2c1 50335,C(=O)(C(C)(CO)NC(=O)CC1CCN(C(=O)CCC2CCC2)C1)OC 50336,N1(C(c2ccc(SCC)cc2)=O)CC2CC(C1)C2NC(=O)Cc1ccccc1F 50337,N1(C(C2CC(OC)C2)=O)CCC2(CCC(NC(C3(CO)CCCCO3)=O)C2)CC1 50338,N1(Cc2c(OC)nsc2)CCC(C(N2CCN(C)CC2)=O)C(C)(C)C1 50339,c1(C(=O)OC)ccc(S(=O)(=O)N(C(c2ccccc2)C2CC2Cl)C(C)C)o1 50340,n1(CC(=O)NC2(CCNC(C3C(CC(C)C)C3)=O)CC2)cc([N+](=O)[O-])nc1C 50341,N1(C(C(C)=CC)=O)CCOCC(C(=O)Nc2cccc(O)c2C(F)(F)F)C1 50342,c1(CNC(C2CCC(C)N2C)=O)cc2c(s1)CCN(C(=O)OC(C)(C)C)C2 50343,C1(C(=O)NC(COC)CO)N(C(=O)CCOC2COC2)CCCC1(C)C 50344,c1(CCC(=O)NC2CN(C(C3CCCCC3(F)F)=O)CC2F)cc(Cl)ccc1Cl 50345,Cc1ccc(C(=O)NC2(CNC(c3cscc3F)=O)CCCCC2)n1C 50346,N1(C(C(C(C)O)(F)F)=O)CCC2(CC1)CCN(C(C1(CCN(C)C)CC1)=O)CC2 50347,C1(CNC(C2(C)CC3CC3C2)=O)CCN(C(=O)CC2CC2)CC1(F)F 50348,c1(N(C)C)ccc([N+](=O)[O-])c(C(=O)NC2CN(C(C3CCC3(F)F)=O)CC2O)c1 50349,C1(C(=O)NC(C(C)NC(=O)OC)C)(NC(=O)OC(C)(C)C)CCCCC1 50350,CC1(C)CC(CCNc2cc(N3CCOC(c4ccc(F)cc4)C3)ncn2)CO1 50351,c1(C(N2CCCC(C(=O)NCc3ccc4c(c3)CC4)CC2)=O)ccc(Br)cc1Cl 50352,C1(CCNC(c2c(CC)noc2C)=O)CCN(C(c2cnsc2)=O)CCC1(F)F 50353,N1(C(C(c2cccnc2)NC(C2(F)CCCCC2)=O)=O)CCCC(CSC)CC1 50354,CC(CF)CC(=O)N(C(C)CNC(=O)C(=O)Cc1ccc(Cl)cc1)C 50355,c1(C(=O)NCC(C)NC(c2c(F)ncc(OC)c2)=O)ccc(F)c(C)c1N 50356,C1(NC(C2CCC(C)(C)C2)=O)CCCN(CCNCc2nnc(OC)s2)C1 50357,CCC(C)(CNC(=O)Cc1nn(CC)cc1Br)NC(C1CC2CCC2C1)=O 50358,c1(NC(N)=O)cccc(C(N2CC(NC(=O)C(O)C3CC3)C(F)C2)=O)c1 50359,c1(C(C)OC(c2c(C)ocn2)=O)ccnc(Cl)c1F 50360,C(=O)(C(CC(C)C)N(C)C(C1C2CN(C(C3(CC)CCCO3)=O)CC12)=O)OCC 50361,c1(NC(N2C(C(=O)Nc3ccc(CCC)cc3)CC2)=O)cc2cc(Cl)ccc2s1 50362,c1(C(=O)NC2(CN(C(C3CC(C)NC(=O)C3)=O)C)CC2)ccc(Cl)c(F)c1N 50363,c1(CC)ccc(C=CC(=O)NC2CN(C(=O)CCN3CCCC3)CC2SC)o1 50364,CC(CS(C)(=O)=O)C(=O)N1CCN(C(c2cc3c(ccn3C)s2)=O)C(COC)C1 50365,C1(OC)CC(NC(=O)NCC(C)Oc2ccc(C)cc2)C12CCOCC2 50366,c1(C(=O)NC2(CF)CCN(C(c3cccc(OC)c3)=O)C2)cc2ccccc2nn1 50367,C1(C(=O)NCC(CCC)C)(C(C)C)CCN(C(=O)C(CO)NC(N)=O)C1 50368,Cc1cc(C)n(CC(N2CC(N(C(=O)Cc3c(C)noc3Cl)C)C2)=O)c(=O)n1 50369,c1(C(=O)NCC2CC(F)(CNC(c3cncs3)=O)C2)cc2cccnn2n1 50370,C1(NC(=O)CCOC2CC2)CCCN(C(=O)C2=NOC(c3ccccc3)C2)CC1 50371,c1(OC)ccc2c(CNC(c3cnn(C(F)(F)F)c3C)=O)c[nH]c2c1 50372,c1(C(N2CCC(N3CCN(C(C4CCCC4F)=O)CC3)CC2)=O)cccc(F)c1Br 50373,C12CC(C)(C1)NC2=O.n1(CCC(C)=O)cc(CC2(O)CCC2)nn1 50374,c12ocnc1C(=O)NCC(CO)NC2=O.c1(CO)csc(CC2CC2)n1 50375,c1(CC(=O)NCCN(C(c2nc(CC)oc2)=O)C)ccc(C(F)(F)F)c(C)c1 50376,C1(NC(c2cnc(C3CCC3)s2)=O)CC2CC1N(C(c1csc(Cl)c1Cl)=O)C2 50377,c1(C(N2CC=CC(C(=O)NOCC3CCOC3)C2)=O)cnc2[nH]ccc2n1 50378,N1(C(c2c[nH]c(=NCC=C)s2)=O)CCC(C)N(C(c2cnc(C3CC3)[nH]2)=O)CC1 50379,N1(C(c2ccc(OC)nn2)=O)C2CCCC1CN(C(C1CC3CC3C1)=O)CC2 50380,Cc1cccc(C)c1C(=O)NCCOC1CN(C(c2ccnc(C)c2N)=O)C1 50381,C1(CC)(CC)CC(NC(c2cnn(C)c2SC)=O)CN1C(=O)CC1CCOC1 50382,C1(NC(Cc2c(C)ocn2)=O)CN(C(C2CN(C3CCCCC3)C2)=O)CC12CC2 50383,Cc1nc(-c2c[nH]c(C(=O)NCC3CCN(C(=O)C(C)n4cccc4)C3)c2)cs1 50384,N1(C(c2cc(C(C)C)on2)=O)CCC2(CCN(C(c3ccc(F)cc3Cl)=O)C2)C1 50385,C1(CC(=O)NCc2c(NC(C(CC)OC3CCCC3)=O)n[nH]c2)CC2C=CC1C2 50386,n1(CCO)ccc(=O)cc1.c1(C(N2C(=O)C2)C)nnnn1C1CC1.C(=O)(CCN)OC 50387,CC1CCC(C2CCCC2)CN1Cc1cn(CC2CCCOC2)nn1 50388,c1(OC)ccc(Cl)cc1C(N1CCC(CNC(=O)CC2CC2)C(O)C1)=O 50389,N1(C(CC2(C=C)CCC2)=O)CC2CC2(CNC(=O)CC2CCC(=O)N2C)C1 50390,c1(C(N2CCC(NC(C(C=C)c3ccccc3)=O)CC2)=O)cc(O)cc(C#N)c1 50391,COn1cnc(C)c1C(=O)NCc1ncncc1C(N1CC(C)(C(N)=O)C1)=O 50392,C(=O)(CC(C)CC(C)C)NCCCCN(C(c1cccc(NC(=O)NC)c1)=O)C 50393,C(=O)(C1CCCc2c[nH]nc21)NC1(CCCC)CCOCC1.c12ncc(cn1)[nH]2 50394,N1(C(CSC)=O)CC2CCC2(CC(=O)Nc2csnc2C)C1 50395,C(=O)(C1CCCc2scnc21)NC(C1CN(C(COCCSC)=O)C1)(C)C 50396,Cn1nc(COC)c2c1CCCC2.C1(NCCO)CCN(c2nnc(C(F)F)o2)CC1O 50397,C1(CNC(c2cc(C(C)C)n(C)n2)=O)C(C)CCCN1C(c1cnn(C)c1)=O 50398,C1(CNC(CCC2N(C)CCCC2)=O)CCN(C(c2ccc[nH]2)=O)CC1O 50399,CC1(NC(=O)C(O)C(C)(C)C)CCN(C(=O)Cn2cnnc2)CC1 50400,C(=O)(C(C(C)O)SC1CCCC1)NC(C1CCCN(C)C1)C1CCC(C)C1 50401,C1(C(C(=O)Nc2cnn(CCF)c2)NC(=O)COC2CCOC2)CC=CCC1 50402,Cc1noc2nc(C(=O)NC3CCCC(NC(=O)CC(C)O)C3)ccc12 50403,CC(c1ccccc1)=CC(=O)NC1CC1CNC(=O)C(C)n1ccnn1 50404,C1(C(=O)Nc2n(CC#C)ccc2)CC2CN(C(c3cccc(C4CC4)c3)=O)CC12 50405,C1(COC)CN(C(C2CCC(O)C2)=O)CCN1C(c1nc[nH]c1C(F)(F)F)=O 50406,N1(C(CC2OCC(C)(C)C2)=O)CC(C(N2CC(N3CCOCC3)C2)=O)C(F)(F)C1 50407,c1(C2C(C(=O)NC3(C)CN(C(C(C=C)O)=O)C3)C2)cc(Cl)cc(Cl)c1 50408,c1(-c2cnc(CC(N3CCC(C)(COCC)CC3)=O)nc2)ccc(C#N)c(F)c1 50409,c1(C(C)OC)nnc(CC2CCOC2)n1CC1CC1.C(COC)O 50410,c1(NCC2CN(C)C(=O)C2)ncnc2[nH]ccc12.C12CCC(CC1)N2 50411,c1(CCN(C)CCN(C(C(=O)NCCC(N)=O)C2COC2)C)ccccc1 50412,C1(C)(C(=O)OC)CNCCN1Cc1ccncc1 50413,c1(C(=O)NCC(c2ccccc2)OC)ccc(Oc2ccccc2)cc1 50414,CN(CCOCc1ccccc1)N1CC(CO)OC2(CCCNC2)C1 50415,n1(N(C)C)nc(-c2ccc(Cc3ccccc3)o2)nc1C1CCN(C(N)=O)C1 50416,C1(NC(C=C(C)C)=O)CCCCC12CCN(C(=O)C=Cc1ccoc1)CC2 50417,N1(C(C(Cc2cnc[nH]2)NC(C(CC#C)C2CC2)=O)=O)CC(O)C2(CCCC2)C1 50418,c1(OCC)cc(NC(c2cnc(OC)c(-c3cncc(C#N)c3)c2)=O)ccc1Cl 50419,Cc1nc2ccccn2c1C(N1CC(C(C)NC(=O)Cc2cncc(O)c2)C1)=O 50420,C12(CNC(c3ccn(CC(F)F)n3)=O)CC1CN(C(C1CC=CC1)=O)C2 50421,CCC(O)C(C)(C)C(=O)NCC1CCC1C(=O)NC1C2C=CC(C2)C1CO 50422,c1(OC(C(=O)NCCC(C)N(C(c2n(CC)ncc2)=O)C)C)cccc(C(C)C)c1 50423,c1(OC)ccc2c(n1)NC(C(N1CCN(C(C3(C4CC4)CC3)=O)CC(O)C1)=O)C2 50424,CCN(NC(=O)C(C)Oc1ccccc1F)CCCCO 50425,C1(C(N(CC(=O)NC(C)C)C)=O)(NC(c2ccc(F)cc2)=O)CCCC1C 50426,N1(C(C(=O)OC)=O)CC2C(Nc3c(Br)cnn3C3CCC3)CS(=O)(=O)C2C1 50427,CCCC(C)(C)C(=O)NCC1CN(C(c2nnc(CC)s2)=O)CCN1C 50428,C(=O)(CC(P(C)(C)=O)c1ccccc1)N(CC(O)CNC(C1(C)CCC1)=O)C 50429,C1(CCOC)CN(C(C2(CCN=[N+]=[N-])CC2)=O)CCN1C(=O)CCS(C)=O 50430,N1(Cc2scc(-c3c(C)cccn3)c2)CCN(S(=O)(=O)N2CCN(C)CC2)CC1 50431,CC(C)(C)S(=O)(=O)CC(=O)N1CCCCC1C(c1ccccc1)CC1CCCC1 50432,C(=O)(N=C1NC(=O)C2CCCN12)c1nc(C)c(C(C)(C)C)s1 50433,CCCCCCN(C(=O)C(C)NC(C)=O)CCNC(=O)C(F)CC1CC1 50434,C(C(C)NC(c1cccn1CC)=O)(C(C)C)NC(CCC)=O 50435,c1(C(=O)NCc2cc(C3N(C(CCC=CC)=O)CCC3)no2)c(SC)cnn1C 50436,C(c1ccccc1)=CCN1CC(CN(C(C2N(C(C)=O)CCC2)=O)C)C1 50437,C1(CNC(Cc2ccc(C)s2)=O)CCC2(CN(C(c3ccccc3O)=O)C2)O1 50438,CCC(CC(=O)N1CCC(N(C)C(c2ccc(F)c(C(=O)OC)n2)=O)C1)C(F)F 50439,N1(C(C2C(C=C)C2)=O)CC(O)(CN(C(=O)CC2COCC2O)C)C1 50440,Nc1cc([N+](=O)[O-])ccc1C(=O)NCCCCNC(c1nccc(Cl)c1Cl)=O 50441,C=CC(C)(O)C(=O)N(C1CC1)CC1CCCN1C(=O)CC(CC)OC 50442,CC#CCC(C(=O)NCCC(O)(CC)CC)NC(=O)C(OC)OC.OC 50443,c1(NC(CCC(C)NC(c2cnc(CC)nc2)=O)=O)ccc(C)cc1O 50444,N1(C(CCCOCC=C)=O)CCN(C(CNC(c2cc(C)cs2)=O)C(F)F)CC1 50445,C(=O)(CC(CC)CCCC)N1CCC(O)(CCNC(C=CCOC)=O)C1 50446,c1(C(N2CCC(NC(CC(CCC)C)=O)C2)=O)cc2c(nc1O)CCC(F)(F)C2 50447,n1(N(CC)CC)cc(-c2nc(-c3cccn3C)no2)c2ccccc12 50448,Cc1c(NC(=O)C(c2ccc(O)nc2)N2CC(CO)C2(C)C)cccc1Cl 50449,C(=O)(C(F)C(F)(F)F)NCC1(C(=O)NCCC(C)N2CCCC2)CC=CC1 50450,C=CCCCCCC(=O)N1CC2CC(NC(=O)Cc3cc(C)on3)CC2C1 50451,C=CCCCCC(=O)NC(C1CCN(C(=O)C=C(Cl)Cl)C1)C 50452,c1(CNC(CC2(C=C)CN(C(=O)CS(=O)CC)C2)=O)cnc(F)c(C)c1 50453,C1(C(CNC(C2(C)CCCC2)=O)O)CCN(C(c2ccc(O)nc2)=O)CC1 50454,C(CNC(c1cccc(CS(C)(=O)=O)c1)=O)(CC(F)(F)F)NC(C(=O)NC(C)C)=O 50455,S(=O)(=O)(c1ccc(-c2ccc(C(C)S)cc2)s1)N(CC=C)CC#N.C(C)C 50456,c1(C(N(C2CCCN(C(c3c(CC)c(C)sc3)=O)C2)C)=O)c(C)cc(O)cc1C 50457,C1(NC(COCCCC)=O)CC(CNC(=O)CCc2cccnc2)C1(C)C 50458,c1(C(N2CCC(C(C(=O)N(CC#C)CCF)C)C2)=O)ccnc(Cl)c1 50459,C=C(C)CCCC(=O)N1CCC(C)C(CC(N2CCCC2C(C)(C)C)=O)C1 50460,c1(OC)cc(C)cc(C(N2CC3(CC3)CC2CNC(=O)C(C)C(F)F)=O)c1O 50461,c1(N(CCC)C)nc2c(c(=NC3CCCn4nccc43)[nH]1)CC(C)CC2 50462,C(=O)(CCCCCN(C)C(C1CC2(CC2)CN1C)=O)OCc1c(OC)n(C)nc1 50463,C1(COC)CCN(C(=NCCc2ccnc(OC)n2)NCC2CCCO2)C1 50464,N1(C(C(C(=O)OCC)OC)=O)CC(=O)NCC1C(=O)NCC(F)(F)F 50465,c1(CC)cccc(C(=O)NCC(CC(=O)NC2CN(C)NC2=O)C2CCC2)c1 50466,C1(COC)(NC(c2nccn2C(C)C)=O)CN(C(C2CC2Cl)=O)C1 50467,c1(C(=O)NCCCN(C(C(C)C(C)(C)O)=O)C2CC2)csc2ccccc12 50468,C1(C)(C(N2C(C(C)=O)CCCC2)=O)CC12CCN(Cc1ncccc1Cl)CC2 50469,c1(C(=O)NCCC(CNC(C2(CSC)CCC2)=O)O)ccc(-n2cccc2)cc1 50470,N1(C(CCCCC)=O)CCN(C(c2ccc(OCCF)cc2)=O)C(CF)C1 50471,CCCCCC(F)C(=O)N1CCCC1(C(N1C2CSCC1C2)=O)COC 50472,Oc1nccc(=NC2CC(NC(=O)C(F)(F)C(F)(F)F)C23CCC3)[nH]1 50473,c1(CC)cc2c(cc1CNS(=O)(=O)Cc1c(C)nn(C)c1C)OC(C)C2 50474,c1(OC)c(Cl)cc(C(N2CCC(NC(=O)CCC3CCC(=O)N3)C2)=O)cc1Cl 50475,N1(C(C(n2c(C)ccn2)C)=O)CC2(CC(C(N3CC(C(C)(C)C)C3)=O)CO2)C1 50476,c1(N2CCC(F)(F)C3(C2)CCC3)nc(=NCc2cc[nH]n2)[nH]c2c1CCCCCC2 50477,c1(CN(CC(=O)NCC(F)CNC(=O)CCn2ccnc2)C)c(F)cccc1F 50478,CC(C)C(C)(C)C(=O)NC(CNC(=O)CC1(C(F)(F)F)CC1)Cc1ccccc1 50479,c1(C(N2CCC(NC(C34COCC3C4)=O)C2)=O)cnc2cc(O)ccc2c1 50480,C(=O)(C#CC1CCCCO1)N(C(CNC(C1C(C=C(C)C)C1(C)C)=O)C1CC1)C 50481,c1(CCC)cc(C(=O)N(CCC(C)NC(=O)C(=C2CCCCC2)F)C)ccn1 50482,Cc1cccc(CCNC(=O)CCC2(C)CN(C(C3CC(C(C)C)C3)=O)C2)n1 50483,C(C(CO)C(C)(C)C)c1onc(-c2ncc(C)o2)n1 50484,C1(C(N2CC3C(NC(c4cc(C)c(Cl)cc4)=O)(C3)C2)=O)CCCC(F)(F)CC1 50485,C1(C#N)(C(=O)NCC2OCCN(C(Cc3nc(NC=O)sc3)=O)C2)CCOCC1 50486,CN1CC=C(CC(=O)NOCC(=O)NCC(C)(F)C(C)(C)F)CC1 50487,C1(C(=O)NC2(CCNC(c3csc(CO)n3)=O)CCC2)CC2CC(=O)C1O2 50488,N1(C(C(CC)(F)F)=O)CCC(F)(C(=O)NC2(C3CCCCO3)CC2)CC1 50489,C12(C(N3CCC(c4cn(-c5cncc(C)c5)nn4)C3)=O)CCCC(CC1CO)C2 50490,C(=O)(C(F)CC(C)(C)NC(=O)Cc1cnccc1C)NC(CC#C)CCOC 50491,O=C1CCC(C(=O)NC(Cn2cccn2)C(=O)N(CC(F)F)CC(F)F)O1 50492,c1(OC)c(F)ccc(F)c1C(=O)NC1CCN(C(c2cc(C)ccn2)=O)CC1F 50493,C1(C(N2CCN(CC(C)NC(C3(C)CC3(C)C)=O)CC2)=O)Cc2cscc2C1 50494,N#CC1CN(Cc2ccc(O)nc2)CC1NC(c1sccc1I)=O 50495,N1(C(CC2CC(NC(c3ncn(C)n3)=O)C2)=O)CCC(O)C(F)C1 50496,Cc1ccccc1C(C)CC(=O)N(C1CCN(C(=O)C(C)(C)C)C1)C 50497,N1(C(C2C(CNC(C(OC)OC)=O)CCO2)=O)CC(COC(C)=O)C1(C)C 50498,C1(NC(C(c2scc(C)n2)C)=O)CC2CC(C1)N(C(=O)CC(C)C(F)(F)F)C2 50499,c1(CC)c(N2CC(CC(C)NC(=O)CC(C)C3CCCCC3)C2)ncnc1C 50500,CCC(C)(C(=O)N(CC(C)C(=O)N(C)Cc1n[nH]c(C)n1)C)OC 50501,CC#CCCC(=O)NCCCCN(C(=O)COc1ccc(O)cc1)C 50502,Cc1cn(C)cc1C(=O)NCCNC(c1ccnnc1S)=O 50503,c1(C(=O)NCC2(C(=O)NC(C#C)CC3CCCC3)CCC2)cn(CC=C)cn1 50504,CCC(O)(CCC(=Cc1ccccc1C(=O)O)C)CC.NC 50505,C1(NC(c2c(CC)scc2)=O)CC(NC(=O)C(C)C)C12CCOCC2 50506,N1(C(CCCOC)=O)CC(N=[N+]=[N-])CC1C(N1CCC(CO)C1)=O 50507,c1(OCC)nc(Cl)ccc1C(c1nnnn1C)NC1(c2ccc(Cl)cc2F)CC1 50508,c1(NC(c2cccc(N3CCCC3)c2)=O)cccc(F)c1.c12cn(nn1)CCS2 50509,N1(C(C=CC)=O)CC(CNC(c2cccn(C3CCSC3)c2=O)=O)CC(O)C1 50510,CC#CCCCCN=C(NCC1CCCCC1)NCC(O)C(F)(F)F 50511,N1(C(c2ccc(Nc3ncc(F)cn3)cc2)=O)CCCC2(CCO2)C1 50512,CC(CC(=O)N(CC(C)NC(c1cnc(C(F)(F)F)s1)=O)C)C1CC1 50513,CCC(C)(COC)C(=O)NCC(C)N(C(=O)CC1CCC=CCC1)C 50514,N1(C(c2ccc3n[nH]cc3n2)=O)CCc2cc(Cl)c(F)cc21 50515,c1(C(=O)NCCCN(C(C2CCS(=O)(=O)N2)=O)CC)c[nH]c2ccc(Cl)cc12 50516,CCCCC(CNC(c1cccc(OCCF)c1)=O)NC(=O)CC1(OC)CCC1 50517,CC1CCN(Cc2cnc(C(C)C)o2)C1C(=O)NCC1COCC1(C)C 50518,CC1CN(C(=O)CCN(CCCO)C(C23CC(C#N)(C2)C3)=O)CC(=O)N1 50519,N1(C(Cc2cc(C)ns2)=O)CC2CC(NC(C3CC4CCC3CC4)=O)CC1C2 50520,N1(C(C(COC)O)=O)CC2CCCC(CNC(=O)CC3CCCC3)C2C1 50521,N1(C(CC(C)C)=O)CCN(C(c2ccn(-c3cncc(F)c3)n2)=O)CC1CO 50522,N1(CC2(NC(C3C(C)C3)=O)CC2)CCN(C(c2cnoc2)=O)CC1 50523,C(C)(CNC(=O)CC12CC(C1)C2)(CC(C)C)NC(C1(c2c(C)cccc2)CC1)=O 50524,C1(NC(C=C(C)C(C)(C)C)=O)CCC(C)(C)CC1CNC(=O)C(C)(F)F 50525,C(C(=O)OCC1CC1)(C1=CCCCC1)OCCCN1C(C)COCC1 50526,C1(O)(c2cn(CC(=C)CC)nn2)CCN(C(=O)CC2CCC(=O)N2)CC1 50527,C1(C(=O)NC(C)Cc2cccnc2)CC2CCC1N2C(C1(C#N)CCCC1)=O 50528,N1(C(C(C)N(C(C)=O)C)=O)CCC(NC(C2CC(O)CN2C(C)=O)=O)C(C)C1 50529,S(=O)(=O)(c1ccc(N)cc1)NC(=O)CC(=O)NC(C(C)Nc1nc(C)sc1)C(C)C 50530,C1(CC(C)NC(C(COC)O)=O)CCN(C(c2cncc(F)c2)=O)CC1 50531,C=Cc1ccc(C(N2CCC(C)C(NC(=O)CCC(C)(C)F)C2)=O)cc1 50532,N1(C(C2C(=C)C2)=O)CC2(CCNC(c3cc(N(C)C)cnc3O)=O)CCC1CC2 50533,C1(CC)CN(C(=O)C(F)=C(C)C)CC1NC(c1cc(Cl)ccn1)=O 50534,C1(OC)CCn2cc(C(N3CC4(CCN(Cc5csc(C)n5)C4)C3)=O)nc2C1 50535,c1(C(N(C(CCNC(C2N(C(C)=O)CCOC2)=O)C)C)=O)nccc2n[nH]cc12 50536,c1(CC)cnc(O)c(C(=O)NCC(CO)NC(=O)C(c2ccnn2C)C)c1 50537,n1(C(c2cc(NC(=O)NCCNC3CCCC3)cs2)CC)nnnc1C(C)(C)C 50538,Cc1c(CNC2(C)CC2(C)C)cnn1-c1ccc(F)cc1 50539,c1(C(N(CC(C)O)CCNC(C(C)OCC#C)=O)=O)cc(C)c(O)c(N)c1 50540,C1(C(C)C)N(C(=O)C=C(Cl)Cl)CC12CCN(C(=O)Cc1ccc(F)cc1)CC2 50541,CC1(C)CN(C(=O)CCn2cnnn2)CC1C(N1CCOCC1CC1CC1)=O 50542,N1(C(c2cc(C)[nH]c2C)=O)CCC2C1CCN2C(c1c(C)cccc1C)=O 50543,C1(F)(C(=O)NCC2CC(C#N)C2)CCN(C(C2CCC2Cc2ccccc2)=O)C1 50544,CC1COC2(C1)CN(C(c1cnc(CNC(C3(C)CCC(O)CC3)=O)nc1)=O)C2 50545,C1(C)(NC(C(C)Cc2ccco2)=O)CCN(C(=O)CC2CCCN2C(C)C)CC1 50546,Cc1c[nH]nc1C(=O)NCC(C)N(C(c1cnc(C(C)C)s1)=O)Cc1ccccc1 50547,N1(C(CN(C(C)C)C)=O)CCC2(NC(c3cc(F)ccc3Cl)=O)CC2C1 50548,C1(NC(c2c(C)n(C3CC3)cc2)=O)CN(C(c2cc3c([nH]2)CCC3)=O)CCC1C 50549,C(C(C)C(F)C(=O)N(C)Cc1cccnc1O)NC(C1(SC)CC(=O)C1)=O 50550,c1(NC(=O)Cc2cccc(-c3cn[nH]c3)n2)cc(Br)cnc1O 50551,c1(C(N2C(C)CN(C(C3CC34CCC4)=O)CC2)=O)noc2c1COCC2 50552,CCCCC(F)C(=O)N1CCC(NC(=O)C(=Cc2cccnc2)F)C1 50553,N1(Cc2c(C)noc2)CCC2(NC(c3ccnn3CC3CCC3)=O)CCCC12 50554,C1(C)(NC(C=COCC)=O)CCN(C(=O)CN2CCP(C)(=O)CC2)CC1 50555,N1(C(CC(C)N(C)C)=O)CCCC12CCCN(C(=O)CC1(O)COC(C)(C)C1)C2 50556,c1(OC)ccc(C(=O)N(CCCCN(C(=O)C(C)OC)C)C)nc1N 50557,c1(C(=O)NC2CN(C(c3cn(CC=C)nc3)=O)CC(C)C2)cc(C)c(=O)n(C)c1 50558,C1(CNC(C(C)OC2CCCC2)=O)CN(C(=O)COc2ccc(F)nc2)CCN1C 50559,N1(C(Cc2cccc(C)c2C)=O)CC2CCN(C(c3cn[nH]c3)=O)C2C1 50560,c1(OCC#C)cc(C(N2CCOC(C3CCCC3)C2)C(=O)NC2CC2)ccn1 50561,c1(OC)cscc1C(=O)NCC1CCC1C(N1CCCC1C(C)(C)C)=O 50562,c1(OC)ccc(CC(=O)NC2(C)CCCN(C(c3ccc(F)c(O)c3)=O)C2)cc1C 50563,C(=O)(CCC(CC)CCC)N1CC(OCCNC(CC(=O)NC)=O)C1 50564,C1(NC(CSc2cc(C)no2)=O)COCCN(C(=O)COCC2CCOC2)C1 50565,c1(CC(=O)NC2CN(C(=O)Cc3cnc4ccccn34)C2)ccc2c(c1)OCO2 50566,C(=O)(C1CCCc2n[nH]cc21)N1CC(C(C)NC(CC=CC)=O)OCC1 50567,CC(C)(CCC(=O)NC1CCN(C(c2ccc(Cl)cc2)=O)C12CCC2)[N+](=O)[O-] 50568,C(=O)(C1=C(C)OCCC1)N1CCN(CC)C(=O)C(C)NC1.C(=O)(C(C)C)O.CCCCC 50569,c1(CCC)cc(C(N2CCC(N(C(=O)C=CSCc3ccco3)C)C2)=O)ccn1 50570,CC(C)(CC(=O)N1CCC(NC(c2conc2C2CCC2)=O)C1)c1cccs1 50571,C1(O)(CCN(C(=O)CC2CCC23CCC3)C)CCN(C(=O)NC)CC1.C1(O)CCC1 50572,c1(CC)cc(C(=O)NC2CN(C(C3(CC)CCCO3)=O)C2)ccc1C 50573,Cc1c([N+](=O)[O-])ccc(Cl)c1C(=O)Nc1cc(C2CCC2)nn1C 50574,Cc1cc(C(=O)NCc2cc(C(=O)NCCN3CCC(CO)C3)co2)ncn1 50575,CC(O)CCCC(=O)NC(C1CCN(Cc2nc(-c3ccsc3)no2)CC1)C 50576,N1(C(C(C2CC2)OC)=O)CCOCC(F)(CNC(C2C3CC4C(C3)C24)=O)C1 50577,CC(C)CCCCC(=O)NCC1CN(C(C2OCCC2C(F)(F)F)=O)CC1C 50578,N1(C(C(C=CC)O)=O)CCC(CC2COCCN2C(=O)Cc2cnsc2)CC1 50579,N1(C(C(C(CC)O)(C)C)=O)CCC12CCCN(C(c1cccs1)=O)C2 50580,C=C(C)c1cccc(NC(C2CCN(C(c3cscn3)=O)C23CCC3)=O)c1 50581,C(=O)(CCCCC(N)=O)NC1CN(C(C=CSC)=O)CC1O 50582,C1(CC)CCCCN1C(=O)C(CCN(C)C)NC(=O)C(CN(C)C)CC 50583,N1(C(C(CC#C)C2CC2)=O)CCN(C(=O)Cc2c(C)nn(C)c2Cl)C(CF)C1 50584,c1(C(=O)NC(CN(C(c2cnn(CC)c2)=O)CC)C)cc2cccc(C)c2nn1 50585,C(C(C)C(C)C(=O)NC(C1(O)CCN(C(c2cn(C)c(=O)n2C)=O)CC1)C)OC 50586,C(=O)(C1=CCC(F)(F)CC1)NC12CCN(C(c3ccc(C=C)cc3)=O)CC1C2 50587,C1(NC(C2(CC)CN(C(C=CCN(CC)CC)=O)C2)=O)CC2(CCC2)C1O 50588,C(=O)(CCCC(C)(C)C)N1CCC(C)CC1CNC(=O)CCc1cccnc1Cl 50589,C1(CC)CN(C(c2ccccc2SCC#N)=O)CCC1NC(C1CCCN1C)=O 50590,N1(C(c2c(Br)cn(CC)n2)C(=O)NCCCSC)CC(OC)C2(CCCC2)C1 50591,CC(C)C(O)C(C)C(=O)N1CC(C)(NC(=O)CCc2ccc(F)cc2)C1 50592,CC1CN(C(C2(CCF)CC2)=O)CCC1CNC(c1cc(N(C)C)ccn1)=O 50593,n1(CC(C)C)ncc2cc(C(N3CCC(c4cc5cccnc5s4)CC3)=O)cnc12 50594,C(=O)(CS(=O)(=O)C1CC1)NC1C2(CN(C(c3c(C)cc(O)nc3)=O)C2)CC1 50595,c1(C(C)NCc2occ(C(=O)OC)c2)c(C)ccc(F)c1N 50596,C1(CCOC)(NC(=O)CC(=C)Br)CCN(C(=O)C(C)(C)C2CCCCO2)C1 50597,C=C1CCN(C(C2CCN2C(C)(C)C)=O)C(C(=O)NC(CCO)C(F)(F)F)C1 50598,N1(C(=O)Cn2cc(C3CCCOC3)nn2)CCCC2(C1)C(O)CC2O 50599,N1(C(c2c(CC)ncc(Br)c2)=O)CC2CCC(C1)N(C(=O)C#CC(C)C)C2 50600,Cc1cc(F)c(N)cc1C(=O)NC(C)C.c12ccc(Cl)nc1S2 50601,N1(C(CNC(C)=O)=O)C(CC(N2CCC2C2CCCCC2)=O)C2CCCC12 50602,C1(C(N(C2CC(C)OCC2)C)=O)CCC(C)(C)N(C(=O)C(c2ccn(C)n2)C)C1 50603,N1(C(Cc2c(C)ccs2)=O)CC(CNC(C2CCC(C(C)C)CC2)=O)C(C)C1 50604,CC(C(=O)NC1C2CN(C(=O)CCc3cccc(C(F)(F)F)c3)CC12)C(C)(F)F 50605,c1(C(=O)NCC2CC(NC(=O)C(=Cc3cccnc3)F)C2)ccc2nsnc2c1 50606,CCC(C)C(O)CC(=O)NC1C2CC3C1C3C2C(N1CCC(C)(O)CC1)=O 50607,C1(CC)CN(C(=O)CCN2CCC(O)CC2)CCN1C(c1nc(Br)cs1)=O 50608,c1(C(=O)NC(CCNC(C(CC=C)C)=O)C)cnc2c(c1)N(C)CCO2 50609,c1(OC)ncccc1C(N1CCCC(CC(=O)NC(C)(C)CN2CCCC2)C1)=O 50610,CCC(CC)C(=O)NCC1CC1NC(C1CC(=O)N(Cc2ccc(F)cc2)C1)=O 50611,C(CC(=O)N1CC(CN(C)C)C2(CC2)C1)(C(F)(F)F)NC(C1C(CCC)C1)=O 50612,N1(C(c2cc(C)n(C)c2C)=O)CC2COCCC2(NC(=O)COCC(F)(F)F)C1 50613,c1(C(=O)NC2(C(N3CC(COC)OCC3)=O)CCCC2)cc2cccnn2n1 50614,CCCCC(O)CC(=O)N1CC(C(=O)NC23CCC(CO)(CC2)C3)C(C)C1 50615,CCCC(CCCNC(c1cnc(OC)cn1)=O)N(C)C(c1cnc(C)s1)=O 50616,Cc1ccc(C(N2CC(C(N3CCCC3C(O)CO)=O)C2)=O)c(O)c1 50617,C1(C(=O)NC(CC=C)CNC(=O)CSS(C)(=O)=O)CC(=O)N(CC)C1 50618,C1(NC(C(CC)N(CC)CC)=O)CCN(C(c2cc(C)cs2)=O)C(C)C1 50619,c1(C(=O)NC(C2CC(NC(=O)CN3CC4CC4C3)C2)C)cc(N)c(O)c(F)c1 50620,CC1CCC(CO)CN1C(c1cc(CNC(c2ccoc2)=O)cs1)=O 50621,C(=O)(C(O)CCCNC(c1cc(C#N)cn1C)=O)N(C(CCSC)C)C 50622,CC1(C)CCCC(C(=O)NC(CNC(=O)CCc2ncco2)C2CC2)C1 50623,c1(C(=O)NCCC(=C)CNC(C2(OC)CS(=O)(=O)C2)=O)ccc(-n2cccn2)nc1 50624,C=CCC(C(=O)NCCCN(C(=O)CC1CCC(C)(C)O1)CC)NC(C)=O 50625,C1(C(=O)NCC(c2ccccn2)C)CCC2(CC2)N1C(=O)C(C)CC(F)F 50626,CCCC(CCC)C(=O)NCC1CC2(CC2)CN1C(c1[nH]nc(OC)c1Cl)=O 50627,Cc1c(C(C(=O)NCCC#N)N(C2CCN(C)C2)C2CC2)cncc1Br 50628,Cc1cccc(C=CC(N2CC(F)CC2C(F)(F)F)=O)c1 50629,C1(C(=O)NCC(C(C)C)(C)F)CCCC(NC(C2CCCSC2C)=O)CC1 50630,N1(C(CCc2cc(C)on2)=O)CC(N(C(=O)Cc2nn(C)cc2Cl)C)C(F)C1 50631,C(=O)(C(CC(C)C)N(C(CCO)C(F)F)C)OC.C1(=O)C(C)N1 50632,N1(C(COCCCCC)=O)CC(CO)C2(C1)CN(c1cc(-c3cccs3)ncn1)C2 50633,N1(C(CCCSC)=O)CC(NC(=O)C(C)(C)c2cccnc2)CC1C 50634,C1(C(=O)NC2C(NC(c3c(C)coc3C3CC3)=O)CC2)CCCCCN1C 50635,C(=O)(C(O)C1=CCCCC1)NC(C(NOC(C(=O)OC)(C)C)=O)CC1CC1 50636,Cc1cc(Cl)nc(Cl)c1NC(=O)CC1CCC(C)N1Cc1cc(O)cc(Cl)c1 50637,C1(C(=O)NC2(C)CC(NC(c3ccc(C)cc3C)=O)C2)CC2CCC(C1)C2(F)F 50638,Cc1cc(C)c(C(N2CC=C(CNC(=O)C=Cc3cccnc3)CC2)=O)cc1N 50639,N1(C(c2ccc(SC)s2)=O)CCN(C(=O)Cc2cnc3n2CCOC3)CC(O)C1 50640,C(=O)(CC1CCCc2ccccc21)NC(CNC(C(CC#C)C)=O)(C)C1CC1 50641,c1(C(=O)OCC2CC(OC)C2)cc2ncccc2o1 50642,CC(C)CC(CN1CCOCC1)CC(=O)N1CC(C)C(P(C)(C)=O)C1 50643,c1(C(=O)NCC(C(=O)NC(CCC)C)N2CCCC2)ncccc1C 50644,c1(SC)nc(C(=O)NC2CC(F)(CNC(=O)CCOCC(C)(C)C)C2)cc(=N)[nH]1 50645,CS(=O)(=O)CCC(=O)NCC1CCCN1C(=O)CCc1cncc(F)c1 50646,N(C(=NCc1ccc(OC(F)(F)F)cc1)N1CCC(C2CCOC2)C1)C(CC)C 50647,c1(CC)ccc(C(=O)NC2CCC(NC(c3ccc(C(C)C)cc3)=O)CC2)cc1 50648,C1(NC(Cn2cc(NC(C=CC(CC)C)=O)nc2)=O)CCc2nncn2C1 50649,C1(NC(C2(OCC)CCC2)=O)CC2CN(C(C3CSC3)=O)CC2C1 50650,CC1(C)CN(C(=O)CCCCC2CCCCC2)CC1NC(C1(C(N)=O)CC1)=O 50651,C#CCCC(=O)N(C(C)C(=O)N(C1CCOC1=O)C)CC 50652,Cc1ccc(CCn2cc(C3(F)CN(C(=O)CC4CCCC4(F)F)C3)nn2)c(C)n1 50653,C1(C(=O)NC2CC(O)(CNC(=O)C(O)C3CC3)C2)(COC)CCCC1 50654,C12(CNC(CSCC=C)=O)CC1CN(C(C1C3CCCOC13)=O)C2 50655,C1CCC(C)C(=O)N2CCC(O)(C2)C(C)N1.c1(COC)cccc(Cl)c1C 50656,Cc1c(Cl)sc(Cl)c1C(=O)NCCCCNC(c1cc(C(F)(F)F)c[nH]1)=O 50657,Cc1cc(C(=O)N(CC(=O)NCC2CC(O)C23CCC3)C2CCC2)cnc1O 50658,N12CCOCC1CNC(=O)CC2.C1(COC)(COC)CC1C(=O)OC 50659,Cc1cc(C(F)(F)F)nn1CC(=O)NCCC1CCN(C(c2cncs2)=O)C1 50660,N1(C(C(C)NC(c2ccco2)=O)=O)CC(C)(C)CC1CNC(=O)CC1(C)CC1(F)Cl 50661,C1(CC)C(C(N2CCC2(C)CCO)=O)CCN1C(=O)Cc1cccnc1 50662,C1(CNC(c2ccc(CC)s2)=O)CN(C(=O)Cc2ccnc(O)c2)CCN1C 50663,C1(C2CCCO2)(C(=O)NCC2CCCCN(C(c3n(C)ccn3)=O)C2)CCCO1 50664,C1(NCc2c(C)ncs2)CCN(C(=O)C(C2(O)CCCC2)F)CC1C 50665,C(=O)(CC(=O)NC(C1(NC(=O)C(C)(C)C)CCCC1)=O)OC(C)(C)C 50666,C(=O)(CC(O)C(=O)N1CC2CC2(CNC(c2nsnc2O)=O)C1)OC(C)(C)C 50667,Cc1cnc(C(=O)NC2CC(F)CN(C(=O)C3=CCCCC3)C2)cc1C 50668,N1(C(CCC(C)(C)NC(=O)C=Cc2ccccn2)=O)Cc2ccccc2C1 50669,C1(CNC(CN(C)C(N)=O)=O)CC(F)(F)CN1C(c1cccnn1)=O 50670,c1(C(N(CCCNC(C2CCC(C)(C)CO2)=O)CC)=O)ccc2c(c1)NCCC2=O 50671,C1(NC(C(C)=C2CC2)=O)CN(C(c2nn(C)nc2C(F)(F)F)=O)CCC1C(F)(F)F 50672,C(=O)(CCCCCC(C)O)N1CCC(OCCNC(C(CC(C)C)O)=O)CC1 50673,C1(c2oncn2)CC(F)(F)CN1c1c(-c2cccs2)cn(C)n1.C(N)=O 50674,C1(C#N)(C(=O)NC2(C)CN(C(CN(CC(=O)NC(C)C)C)=O)C2)CCCOC1 50675,CN1CC(CC(=O)NOCC(N2CCC(F)(COCCF)C2)=O)CC1=O 50676,C1(NC(c2nc(C)n(C)c2)=O)CCCC(C(=O)N(CC(Cl)Cl)C)CC1 50677,CC1CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CCC1N(C)C(C12CCC(CC1)C2)=O 50678,c1(NC)ccc(F)cc1C(=O)NCC1CN(C(=O)CCOc2ccncc2)C1 50679,c1(CC)conc1C(=O)NC1(C)CC(C(=O)NC2C=CC(C(=O)NC)C2)C1 50680,CCC(CC)CC(F)C(=O)N(CCCNC(=O)C(F)=CCCF)C 50681,c1(C(=O)NC(c2ccc(Br)s2)C2CC2)cnc(O)c2ccsc12 50682,C1(C(N(C2CCOC2)CC)=O)CCC(NC(=O)C(C)=O)CC1 50683,N1(C(C=C(C)C(C)(C)C)=O)CCN(C(c2cc([N+](=O)[O-])c[nH]2)=O)C(C)C1C 50684,C1(NC(CC(c2cccs2)N(C)C)=O)CCCC(CNC(=O)C=Cc2nccs2)C1 50685,C(CC(C)C(=O)N(CCNC(c1cnc(O)o1)=O)C1CC1)=CCC 50686,C(=O)(C(C#N)CCC)N1CC2C(C(N(CCC#C)C)=O)(C2)C1 50687,CC(CCNC(=O)C(C)Cc1ccco1)CCNC(=O)CCc1cn[nH]c1 50688,N1(C(C2CCCC(C)C2)C(=O)NCC(C)C)CCC2(CC1)CCN(C)C2=O 50689,C1(C(=O)NC(CC(=O)NC)C)CCCCCN1C(=O)Cc1nocc1C 50690,C(C)(CN=c1ccn2ncc(S(=O)(=O)NC3(c4ccccc4Br)CC3)c2[nH]1)OC 50691,c1(OC)cnc(C(N2CCCC(NC(=O)CC3CN(C)C3)CC2)=O)c(OC)n1 50692,C1(NC(COCCC)=O)CC2(N(C)C(C3CCN3CC)=O)COC1C2 50693,C(C)(C(=O)N(CCCCC(=O)NC1(C)CC2(CC2)C1)C)(C(C)C)OC 50694,c1(C(=O)NC(CC=C)C(N2CCS(=O)C(C)C2)=O)ncc(F)cc1C 50695,CCC1=NOC(CC(=O)N(CC(C)(C)C(=O)NCCCc2nc[nH]n2)C)C1 50696,c1(C(=O)NC(C2(O)CCN(C(=O)CN3CCC(C)CC3)C2)C)cc2sccc2s1 50697,C1(OC)CC(NC(c2cc(C)nn2C)=O)C12CCN(C(c1scnc1C)=O)CC2 50698,c1(OC)cc(C(N2CCCC2CC(=O)Nc2ncc(C)cc2C)=O)cc(Cl)n1 50699,CC1(NC(c2ncoc2C(F)F)=O)CCC(NC(=O)Cc2ccccc2)CC1 50700,CC1CC(CNC(=O)CCCc2cnn[nH]2)CCN1C(=O)CC1CCCO1 50701,c1(C(=O)NC(C2CCN(C(=O)C=Cc3cnc[nH]3)C2)C)coc2c1CSC2 50702,c1(C(=O)NCC2CC2NC(C2CCC2)=O)ccc2nc(O)nc(O)c2c1 50703,N1(C(C(COC)OC)=O)CCC(CC(=O)N(CCC(C)C)C2CC2)CC1 50704,C1(NC(c2cccc(OCC)c2)C(=O)NC)CCS(=O)(=O)C(C)(C)C1 50705,N1(C(CCOC)=O)CCCCC(N(C(=O)CC(C(C)C)c2ccccc2)C)C1 50706,Cc1cc(C(=O)NCC2(F)CCC(CNC(=O)CCF)C2)c2cc(Cl)ccc2n1 50707,Cc1c(O)ccc(CNC2CC2C(=O)Nc2coc3ccccc23)c1O 50708,O=C(CC(C(F)F)NC(C1CC1(Cl)Cl)=O)NCC1(C2CCC2)CC1 50709,N1(C(C(=Cc2ccncc2)C)=O)CCN(C(=O)C(N)=O)C(C)C1C 50710,C(=O)(C(C(C)CC)N(C)C(c1ccc(CCOC)cc1)C1CC1)NCC 50711,c1(CC)c(C(=O)NC(CNC(=O)COCC2CCCO2)C2CCC2)cccc1F 50712,CN1CCC(C(=O)NCc2ccc(CNC(=O)C3=CCCC3)cc2)S1(=O)=O 50713,Cc1cnc(NCC2CCCCC2NC(C2CCCN2N=O)=O)nc1O 50714,C1(NC(CCCn2c(C)ncc2)=O)CC2(C(=O)O)COC1C2 50715,N1(C(COCc2cccc(C)c2)=O)CCC(NC(=O)CCOC2COC2)C(O)C1 50716,N1(C(c2n[nH]c(C)c2Cl)=O)CCC(O)(CN(C)C(C2CCC(C(N)=O)C2)=O)CC1 50717,CC(C)C(C)C(CNC(c1ncoc1C(F)(F)F)=O)NC(=O)CC(C)(C)C 50718,CCC(F)(F)C(F)(F)Br.C(=O)(C1=COCCC1)OC(C)(C)C 50719,CC(C)C(C(=O)NC12CC1CN(C(=O)CN(C)C(=O)C1CC1)C2)NC=O 50720,C1(NC(c2ccc(N(C)C)nn2)=O)CC2CN(C(=O)C3=CCCOC3)CC12 50721,C1(C(=O)NC(C(C)NC(=O)C(Cl)=CCl)C)CCCCC(=O)N1 50722,C12(C(=O)OC)CC3(CC1C2)c1nnc(o1)C(=O)N3.C1(C)C(OC)N1 50723,C1(C2CCOCC2)(C(=O)NC2CC(NC(C(C(C)C)OCC(C)C)=O)CC2O)CC1 50724,C(=O)(C(F)(F)C1=CCOCC1)N1CCC(NC(=O)C2=CCCSC2)C(CO)C1 50725,C=C1CCN(C(c2nonc2N)=O)C(C(=O)Nc2cnc(F)nc2)C1 50726,C(=O)(CC1=CCCC1)OC(C(C(=O)OCC)=O)C 50727,c1(CC)oc(C)cc1C(N1CCC(CCNC(c2cnco2)=O)C1)=O 50728,C(c1cc[nH]c1)=CC(=O)N(CC(C)NC(c1cn(CC2CCCOC2)nn1)=O)C 50729,c1(C(=O)NCC(CNC(c2ncn(CC)n2)=O)F)cccc(-n2ccnn2)c1 50730,N1(C(C(C)=C2CCC2)=O)CCC(NC(c2cc(C(F)F)ccn2)=O)CC1C 50731,C(C(=O)N1CCCN1)N(C(CC=CC=C)=O)CCC 50732,CC1CCN(C(=O)COc2cccc(C#N)c2)CCN1C(=O)CCc1cnoc1 50733,N1(C(C2(CC)CCC2)=O)CCC(O)(C2CCN(C(=O)CN3CCCCC3)CC2)C1 50734,N1(C(c2cncc(CNC(COC(C)=O)=O)c2)=O)CC2CCC(O)C(O)C12 50735,C(C(C)(CC(C)C)NC(c1ccc(C)c(O)n1)=O)NC(c1c(CC)cncc1)=O 50736,C1(C(=O)OCC)CCN(C(=O)C#CC2CN(C(c3c[nH]c(=O)cn3)=O)C2)O1 50737,C1(CNC(c2ccc(CC)c(Cl)c2)=O)CCC2(CCC2)C1NC(C1CCCC1)=O 50738,CC(C)CC(CNC=O)CC(=O)NC1CCCN(C(=O)C(N2CCOCC2)C)C1 50739,N1(C(c2c(C)ccnc2Cl)=O)CC(C)CN(C(=O)CC(=O)N(C)C)C(C)C1 50740,c1(CC)ccc(NC(=O)COCC(C)(C)C)cc1F.N12CCCC1C1(CC1)C2=O 50741,C(=O)(C1COc2ccc(Cl)cc21)N1CCC(CN(C)C(C2CCCOC2)=O)C1 50742,c1(C(N2C(C)(CNC(c3cnc(SC)[nH]3)=O)CCC2)=O)cccc(N)c1O 50743,C(=O)(C(F)(F)CCOC(c1cc(O)ccc1F)C)OC 50744,CC(C)C(F)C(=O)NCC1CCC(NC(=O)CC2CC(C)C2)C1 50745,N1(C(c2cn(C)c(=O)cn2)=O)CCC(NC(=O)CSS(C)(=O)=O)CC(O)C1 50746,C1(N(C(=O)CSc2cccs2)C)CCCC(NC(c2c[nH]cc2Br)=O)C1 50747,C1(NC(C=C(COC)C)=O)CN(C(c2cc(CC(C)C)c[nH]2)=O)CC1N=[N+]=[N-] 50748,c1(C(=O)NCC(C(C)C)NC(C2COCCO2)=O)sc(N2CCOCC2)nc1Cl 50749,c1(OCC(N2CCC(N(C(=O)CC34CC(C3)C4)CC)C2)=O)cc(Cl)ccc1Cl 50750,C=Cc1ccc(C(=O)NCC2(O)CCN(C(=O)CSc3nncs3)C2)cc1 50751,c1(C(=O)NC23CCN(C(=O)C(N4CCOCC4)O)CC2C3)ccc(Cl)cc1Cl 50752,N1(Cc2cc(OC)c(C#N)cc2)CC2(CCN(S(=O)(=O)c3ccc(OC)o3)C2)C1 50753,c1(OC)cc(C(=O)N(CC(C)CNC(=O)CC(C(N)=O)N(C)C)C)c(O)c(Cl)c1 50754,c1(C(=O)NC2(C)CN(C(C3(CC(C)C)CCC3)=O)C2)nn(C)c2ccccc12 50755,CCC(C)C(C)C(=O)NC12CC(C(=O)Nc3cnc4n3CCC4)(C1)C2 50756,c1(C(N2CC(OCCNC(CSCC)=O)C2)=O)cnc2c(c1)c(C)nn2C 50757,Cc1ccc(C(C)C(=O)N(C2CN(C(=O)C(C)Cc3ccccc3C)C2)C)cc1 50758,NS(=O)(=O)c1cccnc1N1CCC(OCC(F)F)CC1 50759,c1(OC)ccc(O)c(C(C)Nc2ccc(C(=O)O)c(F)c2)c1 50760,c1(C(N2CCN(C(=O)Cc3nc[nH]n3)C(CO)C2)=O)nc(Br)c2n1CCCC2 50761,C1(C(=O)NCCC(=O)NCC)CC2(CCN1C(c1cn(C)nn1)=O)CC2 50762,C1(CC(=O)NCCCCNC(=O)C=CC(C)SC)CCCCCC1.C(CO)OC 50763,c1(C(=O)NCCC(C)NC(C2(C(C)C)CC2)=O)cc([N+](=O)[O-])ccc1NCC1CC1 50764,c1(C(N2CCC(CC(C)NC(C3CC(C)C3)=O)CC2)=O)cc(C#N)c(F)cc1F 50765,N1(C(c2cccc(C(F)F)c2)=O)CNS(=O)(=O)c2cc(Br)ccc21 50766,CCCC(C(=O)OC)C(=O)NC1COCCC1NC(c1ccc2n[nH]cc2n1)=O 50767,c1(C(N2CCCC(NC(CCOCCOC)=O)C2C)=O)cc2c(s1)CCC(C)C2 50768,CCCCC(O)CC(=O)N1CC(CNC(=O)CCC2CCCC2)C(O)C1 50769,N1(C(C=CCNC(CCCCSC)=O)=O)C(CO)CCC12CCC2 50770,C12CN(CC1(F)Cl)C2=O.C(C(COC)C(=O)Oc1ccc(Cl)cc1)OC 50771,c1(OCCCC)ccc(Cl)cc1NC(N1CCC(C)C1(C)C)=O 50772,CC1CN(C(C2CCC3(C2)N=N3)=O)CCN1C(=O)CC(C)(C)C1CC1 50773,c1(OC)ccccc1NCCOC(=O)C(N)Cc1n[nH]nc1Br 50774,C1(NC(c2cc(C)nnc2)=O)(CO)CCCN(C(C2CC23CC(C)(C)C3)=O)C1 50775,N#CC1(C(=O)NCCc2ccc(Br)cn2)CC12CCC2 50776,N1(C(=O)OC(C)(C)C)CCN(C(C)C(=O)NC2CC(n3cccn3)C2)CC1 50777,c1(C(=O)NCC(CNC(c2cc(C)c(C)[nH]2)=O)C)ncc(Cl)cc1Cl 50778,N1(C(c2ncn(CC)c2)=O)CCN(C(=O)C(F)(F)C(F)F)CC1CO 50779,N1(C(c2n(C)cnc2)=O)CCCC2(CCC(NC(c3coc(Cl)n3)=O)C2)C1 50780,C=C(C)CC(C(=O)NCCC(=O)NC(C)CN1CCOCC1=O)NC(C)=O 50781,N1(C(=O)Nc2c(C)sc(-c3ccco3)n2)CCN2C3CCC(C3)C2C1 50782,C1(CC)CN(C(C2(NC(=O)C(CC3CCC3)OC)CCOCC2)=O)CCO1 50783,C(CC(=O)N1CC(F)(F)C1C1CC1)(C(F)F)NC(c1n(C)c(S)nn1)=O 50784,CCCS(=O)(=O)CCNc1cc(NCC2(C)CCCS2)nc(C)n1 50785,C1(C)(C(N2C(Cn3ccc(C(C)C(=O)N(C)C4CC4)n3)CCC2)=O)CCC(C)C1 50786,c1(C(=O)NCC(F)CNC(C2CC(F)C(=O)N2)=O)cc2cccc(O)c2[nH]1 50787,c1(N2CC3C(NC(c4ccc(S)cc4)=O)C3C2)ncnn2cccc12 50788,N1(C(c2c(CC)con2)=O)CCOCC1CC(=O)NC1CCOC(C)C1 50789,C=C1CC(CC(=O)NC(COC)COC)C1.C1(c2cccs2)C(=O)N1 50790,CCCS(=N)(=O)c1cccc(CNc2cccc(C#N)c2F)c1 50791,C=CC(CC)CC(=O)N(C1CCCC1)CCCNC(C12CCN(CC1)CC2)=O 50792,C=C(C)CCCC(=O)N1CC=CC(NC(C2(c3cccc(C(N)=O)c3)CC2)=O)C1 50793,C1(C(N(CCOC)CCNC(C2CN(C)CCO2)=O)=O)CC2(C1)CC1(CCC1)C2 50794,CC1(C)CN(C(c2ncccc2C(F)F)=O)CCC1NC(=O)CC1CCC(=O)N1 50795,c1(C(N(CC(C)NC(CSCC)=O)C)=O)[nH]c(C)cc1C 50796,N1(C(C(C#C)(C)C)=O)CCN(C(=O)CC2CCNC2=O)C(CC(F)(F)F)C1 50797,C(C(COC)C(=O)NC1CC(C(N2CCC=C(Cl)C2)=O)C1(C)C)OC 50798,C(C(=O)NCCCCCNC(c1c[nH]nc1-c1ccsc1)=O)(C(C)C)NC(C)=O 50799,Cc1cc(C(N2CC(CNC(c3ccn(CCF)n3)=O)C3CC23)=O)c(N)cc1F 50800,CC1CC(NC(=O)CCc2cnn[nH]2)CN1c1nncs1 50801,c1(C(=O)NC2(CNC(c3nc(CCC)sc3)=O)CC2)cccc2c1C(C#N)C2 50802,C1(O)(C(=O)NCC2C(C(=O)NCC(C(=O)NC)O)CCC2)CCCCC1 50803,CC1(C)C(NC(C2CCC(O)C2)=O)C(C)(C)C1N 50804,C=CC(CC(=O)N(c1ccccn1)CCNC(=O)COCCC)c1ccccc1 50805,Cc1ccnn1C(C)C(=O)NCCN(C1CCCCC1)C1CCSC1 50806,c1cn2c(n1)C(CN1CCNCC1c1ccncc1)CCC2 50807,N1(C(c2cnoc2)=O)CCN(C(=O)CN2CCC(O)CC2)C2CCC12 50808,C(CC)(C(=O)NCCC1CN(C(=O)CC2CC2C(F)(F)F)C1)=CC 50809,N1(C(C=CC(C)=O)=O)CCN(C(C2(CO)CCOCC2)=O)C(C)C1 50810,c1(OC)cccc2c1CCCC2N(C)C(=O)C(=O)Nc1ccn2ccnc2n1 50811,c1(OC)ncc(C(=O)N(CC(C)NC(=O)COC2CCCCO2)CC)cc1Cl 50812,c1(C(=O)NCC2=CCN(C(=O)NCCCl)CC2)c(F)cncc1Br 50813,c1(C(=O)NCC2CCN(C(CCC3C(C)C3)=O)C(C)C2)cn2ccccc2n1 50814,c1(CCCNC(CC)C2CC2c2ccccc2)ccccc1Br 50815,C1(C(=O)NCC2(CNC(C3(C(=O)NC)CCC3)=O)CCCC2)CCCCN1C 50816,C1(NC(CN2CC(C)(C)C2)=O)CC(NC(C2C(C)(C)C2(F)F)=O)CC1O 50817,N1(C(c2c(CC)nco2)=O)CCN(C(c2c(C)cc(C)nc2S)=O)CCC1C 50818,CCCCCCC(C(=O)NC(CCC)CCC)N1CCCC1 50819,N1(C(C(C)(C)c2cncnc2)=O)CCC(CNC(=O)C(=O)Nc2ncc[nH]2)CC1 50820,C(Nn1cccn1)C1(NC(c2ccccc2)=O)CCC1 50821,c1(C(N2C(C(=O)Nc3ncncc3Cl)CC(F)C2)=O)c(F)cccc1F 50822,C1(COC)(CNC(=O)CC2(C(F)(F)F)CC2)CCCN1C(c1nc(C)oc1C)=O 50823,c1(C(=O)NC2CC(CNC(c3c(C)nc(N)cn3)=O)C2)cnn2ccn(C)c12 50824,Cc1cccc(C(C)(C)C(=O)N(C(C)CNC(=O)C(F)CNC(=O)C(C)C)C)c1 50825,C#CC(N(N(C)CC1CN(S(C)(=O)=O)C1)CC(C)C)c1ccccn1 50826,Cn1cc(S(N)(=O)=O)c(C(=O)NCC(C)(CO)NC(C2CCS(=O)(=O)N2)=O)n1 50827,CC(C)(C)C(C(=O)NCc1cccc(F)c1)NC(c1cccc(F)c1F)=O 50828,CCCC(C)(CC)C(=O)NCC(C1CCC1)NC(c1cnc(OCC)c(Cl)c1)=O 50829,N1(c2ncnc(C)c2C#N)C2CCC1CN(C(C1CCOC1)=O)CC2 50830,Cc1csc(C(=O)NCCC(C)NC(C2(O)CC(F)(F)C2)=O)c1C 50831,N1(C(C(C2CCCC2)OC)=O)CC(=O)NCC1C(=O)NCCC(F)=C(F)F 50832,N1(C(CC(=C)C)=O)CCN(C(=O)COc2ccccc2C#N)CC1C1CCCC1 50833,C1(C(N2CCN(CCNC(C(CC)=CCCC)=O)CC2)=O)CCC(C)(C)CC1 50834,c1(OC)ccc2c(c1)CCN(c1nc(NC3CCOCC3C)c3ccsc3n1)C2 50835,C=CCC(C)(O)C(=O)N1CCCC(CCNC(c2csnn2)=O)C1 50836,CCCC(CCC)C(=O)NC1CCCC(NC(c2ccnn2CC#N)=O)CC1 50837,c1(CN(CC2(C(N)=O)CCCCC2)Cc2csc(C(N)=O)n2)c(OC)cccc1Cl 50838,c1(CC)oc(C(=O)NC2CC(CNC(C3CC34CCC4)=O)C2)cc1C 50839,C(C)(C)(CCC(=O)NC1CC(C(F)C(=O)NC2CC(n3cccn3)C2)C1)OC 50840,C1(CC)CC(C(=O)NCC2CC(F)C2)CCN1C(c1sccc1C)=O 50841,N1(C(C2(C(F)F)CC(=C)C2)=O)CCC(C)(NC(C2CN(C3COC3)C2)=O)C1 50842,C1(OC)CN(C)CC1NC(=O)C(C1(C)CC1)NC(C1CC1(C)C(F)F)=O 50843,c1(C(C(=O)NCC(=C)C)N(CCOCC)CC2CCCO2)ccc(F)c(Br)n1 50844,C(=O)(CCCC(C)=O)NCC(CC=C)NC(=O)C=Cc1ccco1 50845,CC1(C)CCCC(C(=O)NCCC(C)(C)NC(C2C3CCCCC23)=O)C1 50846,C1(C(F)(F)F)(C(N2CC(OCC3N(CC(=O)NCF)CCC3)C2)=O)CCCCC1 50847,C(=O)(C(CC)C(C)C)NC(CC(=O)N1CC(COCC)(CO)C1)C 50848,N1(C(C(COC(C)=O)C)=O)CCC(C(=O)NCCNC(=O)C(C)C)CC1(C)C 50849,c1(NC(=O)Cc2ccc(Br)cc2)c2c(cc3c1CCC3)CCC2.C12CCCN1C2=O 50850,N1(C(C=CC(C)(C)SC)=O)CCN(C(=O)CN(C2CCC2)C)C(CO)C1 50851,CCCC(C(=O)N(CCCN(C(=O)CCc1cc(C)sc1C)C)C)NC(N)=O 50852,Cc1nn(C)c(=O)c(C(N2CCN(C(=O)CC(C)F)CC3CCC23)=O)c1C 50853,CC1COCCC1NC(=O)C(=O)N(CCCC1CC2CCC1C2)C 50854,CN1CCC(CC(=O)NC2C=CC(CNC(=O)CCc3ccccn3)C2)C1 50855,Cc1cc(C(N2CC(NC(C3COC(=O)N3)=O)C(C(F)F)C2)=O)ccn1 50856,C12(C(N3CC(C)(CNC(=O)CCc4nccs4)OCC3)=O)CCC(N=[N+]=[N-])C1C2 50857,Cn1nccc(C(N2CCC(NC(=O)CCC3CCCO3)C(F)C2)=O)c1=O 50858,C1(NC(c2c(COC)noc2)=O)C2CCN(C(C3CC4(CC4)C3)=O)CC12 50859,c1(CC)ccc(C(=O)NC2(CNC(=O)CCOC(C)C)CCCCC2)cn1 50860,C1(C(N2CCC(CNC(c3ccc(C)s3)=O)C2)=O)C(Cl)(Cl)C12CC2 50861,N1(C(CN(C)C(C2(Cl)CC2(F)F)=O)=O)CC(N)CC(C)(C)C1.c1(SC)ccncc1 50862,C(=O)(CCCCCCC(=O)OC)NC1CN(C(C(C=C)O)=O)CC(F)C1 50863,Cc1ncc(C(=O)NC2CC2CNC(=O)CC(C)C)c(Br)c1Cl 50864,Cc1cccc2c1OC(C(N1CCC(CO)(NC(c3ccon3)=O)C1)=O)C2 50865,C1(C(=O)NC2CC(NC(c3ccc(NC4CC4)nc3)=O)C2)CCC(F)(F)C1O 50866,C(CN=C(NCc1csc(CC2CCC2)n1)NC1CC(OC)C1)SC 50867,C1(NC(C(c2ccc(C)cc2)C)=O)CCCC12CN(C(=O)Cc1cncn1C)C2 50868,CC(CC(=O)N1CCC(C2CCCN2C(=O)COCCCF)CC1)C(C)(C)C 50869,c1(C(=O)NC2CCC(N(C)C(C3(CF)CC3)=O)C2)n[nH]c(C(F)(F)F)c1Br 50870,NS(=O)(=O)c1n[nH]cc1C(N1CC2CCC1C2NC(=O)Cn1cnccc1=O)=O 50871,CCCC(CCC)C(=O)NC(C)CN(C)C(c1onc(OC)c1Br)=O 50872,c1(C(=O)NC2CN(C(c3ccc(C(C)C)o3)=O)C3C2C3)cc(F)cc(F)c1 50873,c1(OC)ccncc1C(=O)NC1(CCOC)CCN(C(c2ccccc2C)=O)C1 50874,c1(C(=O)NC(CNC(C2C(C)CC2)=O)(C)C)ccc(C(F)F)cc1Cl 50875,C(CN=c1ccc(C#N)c[nH]1)NC1(CCC)N(C(=O)OC(C)(C)C)CCC1 50876,Cc1ccc(C(=O)NC2CC(O)(CNC(=O)C(C)SCCOCCO)C2)c(Cl)c1 50877,CC1CN(C(C2C(F)(F)C23CCC3)=O)CCC1CNC(=O)CC1OCCC1(C)C 50878,C1(OC)CCC(C(=O)NC(C)CNC(c2sccc2C(C)(C)C)=O)CC1 50879,C(C)(C)(C(=O)NCCCN(C(=O)CC1CC(F)C1)C(C)C)COC(C)=O 50880,C1(C(=O)NC2CCCN(C(Cc3n(C)nc(C4CC4)c3)=O)C2)C2CC3C(C2=O)C13 50881,CC1Oc2ccc(C(=O)NCC(C)NC(c3cc(C(C)(F)F)on3)=O)cc2C1C 50882,N1(C(c2c(Cl)cnc(CC)n2)=O)CC2CCC1CN2C(C1(c2cc[nH]n2)CC1)=O 50883,CC1CN(C(c2nc(C(F)(F)F)cn2C)=O)C(C(=O)O)CC1C 50884,c1(C(C(=O)N)N(C2CCN(CC)C2)CCCC=C)cnn(C)c1Br 50885,C(=O)(C1CCc2c[nH]nc21)N1CCC(CCCNC(c2cnsc2)=O)CC1 50886,C1(C(=O)OC)N(C(C2CCc3nccn3C2)=O)CCCC1(C)C 50887,C#CCC(CC#C)C(=O)OCC1CCCC1c1ccccc1 50888,CC(C(=O)N1CC(NC(C2(C)COC2)=O)C1)C(C)C1CCC1 50889,c1(CNC(CCCOC)=O)nnc2n1CCN(C(=O)C(C)CS(C)=O)C2 50890,C(C(=O)NCC1(NC(c2c(Cl)cnn2C)=O)CCC1)(C(C)C)SC 50891,C1(C(=O)O)CCC(O)CN1C(=O)CCCc1cn(CC2C(F)(F)C23CCC3)nn1 50892,N1(C(CC2(NC(c3cnc(CC)o3)=O)CC2)=O)CCN(C2CC2)C(=O)CC1 50893,c1(C(N2CC(CNC(c3ccc(SC)cc3)=O)C3C2C3)=O)cncc(Cl)c1C 50894,Cc1ccc2c(c1)C(C(=O)NC(C)CC(C)NC(c1nc(C)cs1)=O)CC2.CC1CC1 50895,CC1CN(C(c2cccc(N(C)C)c2)=O)CCCN1C(c1ccc(C2CC2)s1)=O 50896,N1(C(CC(C)C(F)F)=O)CCC2CCCC12C(=O)NCCC1CCC1 50897,CCC(F)(F)C(C)(C)C(=O)N1CC(Oc2ccc([N+](=O)[O-])cc2)CC(C)C1 50898,c1(C(N2CCC(C(C)C(N3CC4(CCC4)C3)=O)C2)=O)ccc(O)cc1Cl 50899,C12(C(N3CC(OCCNC(=O)CCOC4CCCC4)C3)=O)CCCCC1OCC2 50900,C#CC1CC2CCC1N(C(C1CCN(C(=O)CC3CCCN3C)C13CC3)=O)C2 50901,c1(C2C(C(N(CCNC=O)CC)=O)C2)ccc(C(F)F)c(Cl)c1.C12CCC(C1)C2 50902,c1(C(N2CC(OC)(CNC(c3cnnn3C)=O)C2)=O)cc2ccccc2[nH]1 50903,c1(C(N2CCC(CCNC(C(C)SC)=O)C2)=O)cccc(=S)n1O 50904,CC(C)(C(=O)N(C1CCCC1)CCNC(C1OCCOC1C(F)(F)F)=O)C(N)=O 50905,N1(C(C)=O)CCN(C(=O)Cc2csc(C)n2)CC1CCO 50906,CCC(C)(COC)C(=O)N1CC(C2CC2C(N2CCOC(C(C)C)C2)=O)C1 50907,N1(C(CCP(C)(C)=O)=O)CC(C(=O)NCc2cc(=O)cc[nH]2)CC12CCC2 50908,c1(OC)ccc(Cl)cc1CC(=O)N(C1CC(NC(=O)CC2(O)CCCC2)C1)C 50909,c1(NC(=O)NC(c2cc(C)sc2C)C2CCCO2)cccc2c1CCO2 50910,C1(c2nc(CC)on2)CN(C(=O)CCc2ccncc2F)CCO1.n12cc(nn1)C2 50911,N1(C(CCC)=O)CCN(C(c2cc(C)nn2C)=O)C(C2CCC2)C1 50912,C1(C(=O)NCCN2CCN(C(=O)C(F)C(F)(F)F)CC2)CC2C=CC1C21CC1 50913,C(c1ccc(F)c(C)c1)=CC(N1CCC(=CCNC(C2C(=C)CC2)=O)CC1)=O 50914,CC1CCN(C(C2CNC(=O)O2)=O)CCN1C(c1cc(-c2ccccc2)on1)=O 50915,N1(C(c2ccc(C(CC)=O)cc2)=O)CCN(C(c2coc(C)n2)=O)CC1C1CC1 50916,Cc1ccc(C(=O)NCCSCC(=O)NCC(C)(C)O)c(F)c1 50917,c1(OC)cc(C)sc1C(N1CC(NC(C2(OC)CCOC2)=O)C(SC)C1)=O 50918,N1(C(CC=CC)=O)CCCC(N(C(=O)CCOc2cccc(C)c2)C)C1 50919,C1(C#N)(C(=O)NC(CCOC)C(=O)NCc2[nH]cnc2C)CCCOC1 50920,N1(C(CNC(C(C)(C)C)=O)=O)CCC2CCCC12CNC(c1ccc(CO)s1)=O 50921,CCC(C)(C)CC(=O)N1CC(N(C(=O)C(C)SC)C)C(O)C1 50922,C1(CNC(C=C(C)Cl)=O)CN(C(=O)C(=O)NCCOC)CCC1C 50923,N1(C(CN(C2CC2)CC)=O)CCCN(C(c2sc(=N)[nH]c2C)=O)CC1C 50924,N1(C(c2c(COC)noc2)=O)CC(C)N(C)C(C)C1.C12CC=CCC1C(=O)N2 50925,N1(C(CNS(CCCC)(=O)=O)=O)CCc2nc[nH]c2C12CCN(C(=O)C(N)=O)C2 50926,c1(C(=O)NCCC(C)NC(CC=CCC)=O)cnc2ccccn2c1=O 50927,Cc1ccc(C)c(C(=O)NCc2nocc2C(=O)NCCCO)n1 50928,c1(CN(C(C)CCC(C)C)C(C(=O)OC)COC(C)(C)C)ccc(F)cc1 50929,C1(CC(=O)NC(C)CCCCNC(c2ccsn2)=O)CCC(=O)NC1=O 50930,c1(NC2CC(C)N(C(=O)CCc3ccncc3)CC2)ncc2c(c1C#N)CCC2 50931,C1(OCC#C)(CNC(=O)C(c2ccccc2)NC)CCCS(=O)(=O)C1 50932,c1(C(N2CC(CN(C(C(C)C3CCCC3)=O)C)C2)=O)ccc(C2CC2)o1 50933,N1(C(CCCC(C)C)=O)CCC(N=[N+]=[N-])(C(N2CCCC(OC3CC3)C2)=O)C1 50934,Cc1cc(O)ncc1C(=O)N(CCCN(C(=O)CC1CCC(=O)N1)C)C 50935,N1(C(C(C)C(C)(F)F)=O)CC2(COC(CNC(=O)C(C(C)(C)C)N(C)C)C2)C1 50936,Cc1ccc(C(N2CCC(C(N3CCC(C)(CO)CC3)=O)(C(C)C)C2)=O)nc1C 50937,N1(C(CCCC(=O)NCCC)C(=O)OC)Cc2ccccc2OC(C)C1 50938,C1(C(=O)OCC)CCCN(C(C2(C)CCN(C(C3CC3(C)C(F)F)=O)C2)=O)C1 50939,Cc1ccc(C(=O)NCCCN(C(=O)C(C)(O)C(C)C)CCO)cc1I 50940,c1(C(C)C)cc(C(=O)NC2CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C2)cc(Br)c1 50941,C1(NC(=O)CS(=O)(=O)NC2CCOCC2)CN(Cc2ccccc2)CC(F)(F)C1 50942,CC(C)(CCNC(=O)CNC(N)=O)NC(C1OCCO1)=O 50943,C1(C2(O)CCC2)(C(N(CC(C)NC(=O)CC2CC3CC2C3)C)=O)CC1 50944,c1(CC)cnc(C(=O)NCC2(NC(C3CCC34CCC4)=O)CCCC2)cn1 50945,N1(C(Cc2nnc(C)s2)=O)CC2CC(NC(c3conc3C(C)(C)C)=O)CC2C1 50946,c1(C(N2C3C(NC(C(C(CC)CC)C)=O)C(C3)C2)=O)nc(N)cc2ccccc12 50947,N1(C(c2c(OC)csc2)=O)CCC(C)C(N(C(=O)C(=CC2CCCCC2)F)C)C1 50948,C1(NC(C2CCCN(C(Cc3c(C)cccc3)C)C2)C)CCC2CC2CC1 50949,C1(CO)(NC(c2cc(Br)ccn2)c2nnnn2Cc2cccs2)CCOCC1 50950,C1(C(N2CC(C#C)(F)C2)=O)C2CCN(C(=O)CC3CCCCC3O)CC12 50951,c1(OC)ccc(-n2cc(-c3ccc(=O)n(C)n3)nn2)cc1N(C)C 50952,CC1(C)CN(C(=O)Cn2cc(C3CCOC3)cn2)CC1NC(C12CC(C1)C2)=O 50953,c1(C(=O)NCC(CC=C)NC(c2cnc(C)nc2CC)=O)cnc(SC)nc1C 50954,CCC(C)C(C(=O)NCCn1ncnn1)NC(c1ncnc(O)c1F)=O 50955,CCCC(O)CC(=O)NCCO.N1(C(C(N2C(CN)CCC2)=O)C)CCCC(O)C1 50956,c1(-c2ccc(C(=O)NC(CNC(C3CCC3F)=O)CO)s2)cccc(F)c1 50957,C1(C(=O)NCC(CN(C(COCC(C)C)=O)C)C)CCC(N(C)C)CC1 50958,C1(C(=O)NCC(CN(C(=O)Cc2ccn(C)n2)C)O)CCCC1C(F)F 50959,C1(CNC(c2n(C)ncc2CNC(=O)CSCC(N)=O)=O)CC2C=CC1CC2 50960,C1(CC(=O)NCC2CC(NC(C=CC(C)C)=O)C2)CN(C)CC1O 50961,O=C1NC(=O)C2CN(c3ccncc3S(=O)(=O)NCCSC3CC3C3CC3)CC12 50962,C1(C(N2C(CCC(=O)NCCn3ccc(C4CC4)n3)CC2)=O)CC2CCC1C2 50963,CC(=O)N=c1nc(Cl)[nH]n2c(Br)cnc12 50964,N1(C(C=Cc2c(OC)cccc2)=O)CCCC(C)(NC(c2scnc2C)=O)C1 50965,C(C)(CCC(=O)N1CCCC1CCCC#N)NC(C1C(C)=CCS1)=O 50966,CCC(C)CC(=O)N1CCC(n2cc(CNC(C3CC=CC3)=O)nn2)CC1 50967,c1(C(=O)NC(C2CCN(C(=O)CC(C)(C)O)CC2)C)ccc(C#N)c(Cl)c1 50968,Cc1cccn2cc(C(=O)NC3CCOC3C3CCN(C(=O)C4CC4)CC3)nc12 50969,C1(C(N(CC(C)NC(=O)C(C)(C)N(C)C)CC)=O)CCC(O)CN1C 50970,Cc1ccc(C(C)C(=O)NC2(CN(C)C(c3nc[nH]c3C(F)(F)F)=O)CC2)cc1 50971,C1(CNC(CN(C)C2CC2)=O)CCC1NC(c1cc[nH]n1)=O 50972,c1(OC(C)C)cc(NC2CCCC(CNC(C3(C)C=CCCC3)=O)C2)ncn1 50973,C1(NC(C=Cc2cccc(OC)c2)=O)CN(C(=O)CNC=O)CCC1C 50974,C1(NC(CC(C)C2CCCO2)=O)CCC(C)N(C(=O)Cc2cnn(C)n2)C1 50975,N1(C(C=C(CC)C)=O)CCC(NC(C23CSCC2C3)=O)C1C1CC1 50976,C1(N(C)C(c2cnn(-c3cccnc3)n2)=O)CCc2nnc(Br)n2C1 50977,Cc1nccn2c(C(N3CCNC(=O)C3c3ccccc3Cl)=O)cnc12 50978,c1(C(=O)NC(CNC(C(CC=C)C)=O)CO)cccc2[nH]c(C)cc12 50979,c1(NC2(CCO)CCCC2)ccc(Br)c(S(=O)(=O)N2CC(CN(C)C)OCC2)n1 50980,c1(C2(NC(=O)NCc3cc(Cl)cs3)CC2)ccc(F)c(F)c1 50981,N1(CC2CCN(Cc3ccccc3)CC2)CCCC(O)(Cn2cccn2)C1 50982,N1(C(COCCCOC)=O)CCOC(C(C)NC(=O)C=Cc2ccc[nH]2)C1 50983,C1(C(=O)NCC(C2(O)CN(C(=O)CCC(F)(F)F)CC2)(C)C)COC(C)(C)CO1 50984,C(=O)(C1=NOC2(CCC2)C1)N1CC(C)C(C(=O)NC2(c3nn[nH]n3)CC2)CC1 50985,N1(C(CC2OCC(C)(C)C2)=O)CC(C2CCCCN(C(C3CCC(F)C3)=O)C2)C1 50986,c1(C(C)C)cc(C(N2CC(CNC(=O)Cc3ccoc3)C2)=O)nn1C.C1(C)CC1 50987,C1(C(N2CCC(CC#C)CC2)=O)CCN(Cc2csc(C3CC3)n2)C1(C)C 50988,C(=O)(C1=CCOC1)NCCCNC(C(C)CNC(=O)OC(C)(C)C)=O 50989,c1(C(C(=O)NCC2NCCC2CC(F)(F)F)F)ccc(Cl)cc1 50990,c1(C(N2CC(CC(=O)NC(C(=O)NCC)(C)C)C2)=O)cnc(N(C)C)nc1 50991,C1(C(=O)NCC(C2(O)CCN(C(c3cncc(Cl)c3)=O)C2)C)CCS(=O)(=O)CC1 50992,c1(C(=O)NC2(COC)CCCN(C(=O)CC(C)F)C2)ccc(C)c([N+](=O)[O-])c1 50993,C(=O)(C1=NNC(=O)CC1)NCC1(CNC(C(C)(C)CC2CCCC2)=O)CCCC1 50994,c1(C(=O)NC2(CO)CN(Cc3ncsc3Br)C2)cccc(C(F)(F)F)n1 50995,C1(NC(c2c(C)ccc(Cl)c2)=O)COC2(C1)CN(C(C1(C)CCS(=O)(=O)N1)=O)C2 50996,Cc1cccc(CN(CC(=O)OC(C)(C)C)C)c1-n1cc(C(O)C(C)(C)C)nn1 50997,C1(C(=O)OC)CCN(C(c2n[nH]c(CO)n2)C(=O)NCCSC(C)C)C1 50998,c1(C(N2CC(C)C(CNC(c3cnn(C)c3N)=O)CC2)=O)ccn2nccc2n1 50999,C(C)(C)(CC(F)C(=O)NC1CCOC1)NC(CN(C(COC)=O)C)=O 51000,CN1CCN(C(=O)Cn2cnnn2)CC1NC(C1CCSC1)=O 51001,C1(C(N2CC(O)(CN(C)C(c3n[nH]cc3F)=O)C2)=O)CC2(C1)CC2(F)F 51002,CCCC(C)(O)C(=O)NCC1CCC1NC(c1ccc(N)c(CC(C)C)c1)=O 51003,CC1CC(NC(=O)CC2CCN(C(C3CC(F)CN3)=O)C2)C(=O)O1 51004,N1(C(C2CC(SC)C2)=O)CCC(CCNC(=O)C(C)N2CCC2)C(F)(F)C1 51005,CN1CCC(C)(C(=O)NCCOC2CCN(C(=O)CNCC(C)(C)C)CC2)CC1 51006,C=CC(CC)CC(=O)NCC1(C)CCCN1C(c1cc(C2CC2)ccc1Cl)=O 51007,c1(OC)c(C(=O)N(CCC(=O)NCCCn2cnnc2C)C(C)C)cnn1C 51008,Cc1ccnc(O)c1C(=O)NC1CCC2(C(N3CC(SCC)(OC)C3)=O)C1C2 51009,Cc1c(C(N2CC(C(=O)NC3(C)CCCC3(F)F)CC2CO)=O)cccc1O 51010,C=CCCCC(C(=O)N(CCCCCO)C)NC(C1CC(CC2CC2)C1)=O 51011,[N-]=[N+]=NCCCCC(=O)NC1(CCNC(C2CCCCC2C2CC2)=O)CC1 51012,C(C(CNC(=O)CCc1nncs1)C(F)(F)F)NC(C1CC12CCCC2)=O 51013,C1(C(N2CC(C(C)NC(c3ncoc3-c3ccon3)=O)C2)=O)C(C)(C)C1(C)C 51014,c1(OC)ccccc1SCC(=O)NC(C)CC1CN(C(=O)CC2CCC3CC23)C1 51015,C=CC1(CC(N2CCCC(C(C)(C)C)C2)=O)CN(C(=O)CCOC(C)C)C1 51016,C(=O)(CC(C)CNC(=O)COC(=O)CO)NC1(CC)CCC1 51017,C1(NC(=O)NCC2(C(=O)O)CC3CCC2C3)CCCC2(C1)OCCO2 51018,N1(C(c2c(C)nc(N)cn2)=O)CCC2(CCC(NC(=O)C#CC3CCOC3)C2)C1 51019,c1(CC)ccc(CC(=O)NC(CNC(c2cc(=O)n(C)cn2)=O)C2CC2)cc1F 51020,C1(C(N2CC(CNC(c3ccc[nH]3)=O)C(F)(F)CC2)=O)CC2CCCCCCC12 51021,c1(C(N2CC(CNC(C(C=C)O)=O)OCC2)=O)ccc(C)c(S(=O)(=O)CCO)c1 51022,Cc1ccc2c(C(=O)NC(C)CNC(=O)CC3CC(=O)C3)coc2c1 51023,N1(C(C(CC=C)CC)=O)CC2COCCC2(NC(c2cnc(Cl)c(N)c2)=O)C1 51024,c1(C(N(CCCNC(C2N(CC)CC2)=O)CCO)=O)c(SC)cccc1F 51025,N1(C(C2C(C(=O)OC)C2)=O)CCC(C2(NC(c3cc(C)ccn3)=O)CC2)CC1 51026,C(C(CC)CO)NC(C=CCN(CC)CC)=O.C1=CCNC1=O 51027,c1(C(N(CC(C(=O)O)C)C)=O)sc(C)nc1C.C1(OC)CCN(CC)C1 51028,CCCCC(O)CC(=O)NCC#CCNC(=O)CC(n1nc(C)cc1C)C 51029,c1(CCC(=O)NCC(O)CNC(C2(F)CCCC2)=O)ccc2c(c1)OCO2 51030,C1(C)(CC)C(C(=O)N(C2CC(F)(F)C2)C)CCN1C(c1ccn(C)c1)=O 51031,C1(NC(=NC)NCC(c2ccc(Cl)cc2)O)CCCC2(CCCC2)O1 51032,CC1CN(C(C2CC(=O)NC2(C)C)=O)CCN1C(c1nn(C(C)(C)C)cc1Cl)=O 51033,c1(OC)c(F)cc(Br)c(C(=O)NNC(=O)C(F)F)c1F 51034,c1(C(=O)NCC(C2CCOC2)NC(c2cnns2)=O)cc([N+](=O)[O-])c2nsnc2c1 51035,c1(OC)nccc(C(N2CC(OCCS(=O)(=O)N)CC2)=O)n1.C(C)(C)O 51036,Cc1nn(C)cc1C(=O)NCC(C1CCCN(C(c2nnccc2C)=O)C1)(C)O 51037,c1(N(C)C)cncc(C(N2CC3C(CNC(C4(CO)CCCC4)=O)C3C2)=O)c1 51038,c1(N2CCCC(CCC=C)C2)cc(Br)ccc1S(=O)(=O)NC1CC1 51039,Cc1cccc(CN2CCC(C)(CN)C2)c1Br 51040,N1(C(C=NOC)=O)CCCCC1CC(=O)NC1C(C)C1C 51041,C(C(CC(=O)NC(CC1CCC1)CO)NC(=O)C(C)C1CCCC1)OC 51042,C1(CNC(=O)CCn2cncn2)COC(CNC(c2cc(-c3ccco3)[nH]n2)=O)C1 51043,c1(C(=O)NC(CCCNC(C(C(CC)C)O)=O)(C)C)cc2ncn(C)c2cn1 51044,CCC(COC)C(=O)NC1CN(C(=O)CC2(c3cccnc3)CC2)CC1C(F)F 51045,C(=O)(C(F)C(C)(C)O)NCC1C(C)CN(C(c2ccnc(OC(F)(F)F)c2)=O)C1 51046,C1(C(NOCCC#C)=O)N(C(=O)Cc2csnn2)CCC1(C)C 51047,C12(C(=O)NC(C3(C)OCCO3)C)CCC(n3cc(-c4nccs4)nn3)(CC1)C2 51048,Cc1sc(-c2ccccc2C2CC2)nc1CN1CC(C(=O)CS(N)(=O)=O)C2CC12 51049,c1(C(=O)NC2CC(CNC(C3N(C)CC(O)CC3)=O)C2)ccc2nc(=N)[nH]n2c1 51050,C1(NC(c2nccnc2Cl)=O)CC2CN(C(c3c(Cl)nsc3Cl)=O)CC12 51051,C#CC1CN(C(=O)Cn2ncccc2=O)CCN1C(c1cc(F)ccc1CC)=O 51052,C1(C(N(CCCC(=O)NCC(C)CNS(C)(=O)=O)C)=O)CCc2cnnn2C1 51053,CCCCCCCCC(C)C(=O)N1CCCC(CNC(c2coc(CO)c2)=O)C1 51054,N1(C(c2ncn(CC)c2)=O)CCC(NC(=O)C(C)Cc2ccc(F)cc2)C(F)C1 51055,Cn1cc(C(=O)NC(CCCNC(=O)Cc2ccc(Cl)s2)c2ccccc2)nn1 51056,N1(C(CCOCCC)=O)CC(CNC(c2c(NC(C)=O)c[nH]c2C)=O)CC1C 51057,c1(C(=O)NC2(CC)CN(C(=O)CC(COC)OC)C2)coc2c1COC2 51058,c12ccc(F)cc1CN(C(C)C)C(=O)N(CC)C2.C12(NC)CCCC1CNC2 51059,N1(C(=O)CCOCC2CC2)CCC(O)C(C(N2CCCC23CC3)=O)C1 51060,C1(O)(CNC(c2c(C)coc2)=O)CCN(C(c2cc(Br)ns2)=O)C1 51061,N1(C(c2ccc(OC)cc2)=O)CCCCC(CNC(=O)CCCCSC)C1 51062,CCCC(O)C(=O)NCC1(CNC(=O)C(C)SC)CCOCC1 51063,CCC(C)(CCC(C)C)C(=O)N1CCOC(C(N2CCC(F)(F)C2)=O)C1 51064,c1(C(N2CC(N3CC(C#N)C(c4ccccc4)C3)C2)=O)ccc2ccccc2n1 51065,CCC(CC(=O)NCCC(C(=O)Nc1cnc(C)nc1)OC)C(F)F 51066,C1(CNC(COc2ccn(C)n2)=O)CN(C(=O)CC2C(C)(C)C2(C)C)CC1(C)C 51067,N1(C(C(C)c2ccsn2)=O)CCCC(C2CN(C(c3cccc(C4CC4)n3)=O)C2)C1 51068,N1(C(C2COCCN(C(c3c(CC)ncs3)=O)C2)=O)CCCc2ccccc21 51069,c1(C(N2CCC(NC(c3n(C)ccn3)=O)C(F)C2)=O)cncc2[nH]ccc12 51070,C1(CC(=O)OC)CCN(C(=O)C(C2CCCCC2)C)CC1.C12CCN(CC1)CC2 51071,C1(C(C)(C)C)CC(C(=O)N2CC(CNC(=O)CCC3CC3)C(C)C2)=NO1 51072,c1(C(=O)NCC2(C(C)(C)C)CCN(C(c3c(C)snn3)=O)C2)ccc(N)cc1Cl 51073,c1(C(N2CC=CC(NC(=O)C3=CCC3)C2)=O)ccc2c(=O)ccoc2c1 51074,C(=O)(C#CC1(C)CCCO1)N1C2CC(CN(C(C3CCCN(CCC)C3)=O)C2)C1 51075,c1(C(N2CC3(CC(CC(=O)NC(C)C(C)(C)O)C3)C2)=O)ccc2ncccc2n1 51076,c1(OC)ccc(C(C)NCC2CN(c3cc(O)nc(C)n3)CCO2)cc1C 51077,N1(C(C2(NC(C3CCN(CC)C3)=O)CCN(C)C2)=O)CCCN(C=O)CC1 51078,c1(CC)noc2ncc(C(N3CCN(C(C4CCCSC4)=O)C(C)C3)=O)cc12 51079,c1(C(=O)NC(C(C)NC(=O)COc2ccc(F)cc2)C)ccc2c(n1)OCCO2 51080,S(=O)(=O)(c1cccnc1Cl)N1CCCC(N(C(c2cc(OC)no2)=O)C)C1 51081,C(=O)(C(C#N)C(C)C)N1CCC(C(C(=O)NC(c2nccn2C)C)F)C1 51082,C(=O)(CCCCCNC)NCC1C(SCC)C1.C(=O)(C(C)OCCOC)C1CCC1 51083,c1(C(=O)NCCC=CCC)cc(C(N)=O)ccc1C 51084,N1(C(c2c(CC)nco2)=O)CCOC(CCNC(=O)C(C)CF)C1 51085,c1(OC)cccc(CNC(=O)CC2CCN(Cc3nc(Cl)cs3)CC2)c1O 51086,C1(C(=O)NC2CN(C(C(CC=C)(F)F)=O)CC2O)CN2CCN1CC2C 51087,Cc1nc(Oc2ccc(F)cc2)ncc1C(=O)N(C1CC1)C1CC1 51088,C=CC(CCC)CC(=O)NC1CC2CCC(C1)N2C(C1CC(F)(F)C1)=O 51089,C(=O)(C(C)CC(N)=O)N1CCN(C2CCN(C(CCC=CC(C)C)=O)C2)CC1 51090,N1(C(CC(CC2CC2)NC(COCCC#C)=O)=O)CCC(C)=C(C)C1 51091,N1(C(c2cc(CC)[nH]n2)=O)CC(CNC(=O)C(N2CCOCC2)C)CC(C)C1 51092,c1(OC)cc(N)c(F)cc1C(=O)NCC1CCCN1C(=O)CCSC1CCCC1 51093,Cc1ccc(Cl)cc1C(N1CCC(CN(c2ncncc2I)C(C)C)CC1)=O 51094,C1(CC(=O)NC2CC2O)CCCCN1C(c1ccc(Cl)o1)=O 51095,C1(NC(CCc2c(C)cccn2)=O)CCN(C(C2(C)CCCC2)=O)CC1(C)C 51096,C(N=c1[nH]c(=N)[nH]c(=NC2CCN(CCN(C)C)C2)[nH]1)c1ccc(C)c([N+](=O)[O-])c1 51097,CC1C(NC(c2ccc(CC#N)cc2)=O)C(C)CCN1C(c1cnc2n1CCC2)=O 51098,C1(N(C)C)CC(C(C)(C)C)CN(C(=O)C(F)(F)C(F)F)C1.C1(=O)CCC(C)(C)N1 51099,N(C(=NCC1CC1)N1CCS(=O)(=O)C(c2c3c(ccc2)C(=O)NC3=O)C1)C 51100,C1(F)(C(NC(C(C)=C2CC2)=O)CC)CCN(C(C2CCN(c3ccccc3)C2)=O)C1 51101,N1(c2n(CC)c(C(c3cccnc3)(C)O)nn2)CCN(CC(F)(F)F)C(C)C1 51102,C1(O)(CN(C(=O)C(c2ccccc2)N(C)C)C)CCN(C(=O)C(C)(C)F)C1 51103,c1(C(=O)OC)cncc(C(=O)N(C)CCOCCNC(=O)Cc2cn(C)nn2)c1 51104,C(CN=c1ccc(Br)c(S(=O)(=O)NCCc2ccc(SC)cc2)[nH]1)SCCCC 51105,c1(NC(CSCC)C)nc(N2CCCC(COC)C2)nc2scnc12 51106,N1(C(C(C)(C)CCl)=O)CC2(C(N3CCN(S(C)(=O)=O)CC3=O)=O)CC1CO2 51107,c1(NC2CCCCCC2)sccc1C#N.CC12CCN1CCNC(=O)C2 51108,C1(F)(CNC(c2c(CC)noc2)=O)CCN(C(=O)C2CC2)CC1.S1(=O)(=O)C(F)CN1 51109,C=Cn1nccc1C(=O)NC1CCC1NC(C1CCN1C(=O)OCC(C)(C)C)=O 51110,c1(OC)cc(C)c(C(=O)NC2CN(C(=O)CCc3cnc(O)[nH]3)CC2O)c(C)c1 51111,n1(CC(=O)NCC2C3N(C(C(C)C(F)(F)F)=O)C(CC3)C2)ccc2ccc(F)cc12 51112,C1(CN(C(=O)CCc2nccs2)C)CCCN(C(c2cnsn2)=O)C1 51113,N1(C(C(C(C)NC(c2cc(=N)[nH][nH]2)=O)(C)C)=O)CC(O)C2(CCCC2)C1 51114,c1(C(N2C(C3CCN(C(C=CC(C)(C)SC)=O)C3)CCC2)=O)cc(C)c(C)o1 51115,CCC(C)(C)C(C(=O)NCC(C1CC1)N(C)C(C1(c2ncco2)CCC1)=O)OC 51116,N1(C(CS(CC)=O)=O)C(C)CC2CN(C(C3(C(=O)OC)CC3)=O)CC12 51117,Cc1sc(C(=O)NCC(C2CCN(C(=O)C(F)CC3CC3)CC2)C)cc1[N+](=O)[O-] 51118,C1(OC)CN(C)C(C)(C(=O)NCC(CO)NC(c2ccsc2SC)=O)C1 51119,N1(C(C(C)(F)F)=O)CCN(C(=O)CN2CC=CC2)CC(O)C1 51120,N1(C(c2cc(CC)no2)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)C(CC2CC2)C1 51121,C1(C(=O)OC)CC2CC2N1C(=O)C(N1CC2CC2C1)C 51122,CCC(C)(C)C(=O)C(=O)N(C)CCC1CC1.C1C(=O)NOCCCO1 51123,c1(-c2ccc(C(=O)NCCN(C(=O)CCCc3ncco3)C)[nH]2)ccccc1F 51124,c1(C(=O)NCC=C)ccc(C)nc1OC.C(=O)(C(C)(O)C1CCC1)NCC(CC)(C)OC 51125,Cc1ccc(C)n1CC(N1CCCC1CCNC(=O)CCc1cnco1)=O 51126,c1(C(=O)OC)cc(C#N)cnc1NC1CC2CN(C(C3CNC(=O)N3C)=O)CC12 51127,c1(C(=O)NC2(C)CN(C(C3CC(C#N)C3)=O)C2)nnn2c1CSCC2 51128,c1(CC)ccc(NC(C2(CO)CCC2)=O)c(C)n1.c12cccc(c1)CNC2=O 51129,Cn1ncc2c(N3CCC4CCN(C(c5ccccn5)=O)CC4C3)ncnc12 51130,C1(NC(C=C(CC)CC)=O)C2CC3C1C3C2C(=O)NCC(C)(C)CSC 51131,c1(C(=O)NC2CN(C(CC(CCC)O)=O)CC(C)C2)cc2ccc(F)cc2[nH]1 51132,C1(COC)(CNC(=O)C2=CCSC2)CCCN1C(c1ccc(C#N)s1)=O 51133,C[Si](C)(C)CC(C(=O)O)Nc1ccc(NC(=O)C(Cl)(Cl)Cl)cc1 51134,CCCC(CCC)CC(=O)NCC1CCC(C)(C)CN1C(c1sncc1CC)=O 51135,CN1CCC(C(N2CC(N(C(=O)C=CC(=Cc3ccccc3)CO)C)C2)=O)CC1=O 51136,c1(CN(C(COC(C(=O)N(CCC(C)SC)C)OCC)=O)C)cnccn1 51137,c1(C(N2CCCC(CCNC(CCCCCC)=O)CC2)=O)cc2cccnc2o1 51138,CCCCCC(O)CC(=O)N1CCCC(C2CCCCN2C(c2cnsc2)=O)C1 51139,CC(C)C(O)Cc1cn(C(C)CNC(=O)CSCC(=O)N(C)C)nn1 51140,C1(NC(CCC(=O)NC)=O)CCCC12CCN(c1ccc(C(=O)OC)cn1)CC2 51141,c1(CNC(C2(C)CN(C)C(=O)C2)=O)ccc2c(c1)CN(C(=O)CS(C)(=O)=O)C2 51142,c1(C(C(=O)N(CC(C)NC(C(CC)C)=O)C)=O)c(OC)cc(OC)cc1OC 51143,C1(C(N2C(C)(C)C(CO)C2)=O)N(C(c2cnccc2C#N)=O)CCCC1(C)C 51144,c1(C(N2CCC(OCC(N3C(CC)CC(O)C3)=O)C2)=O)cc2occc2s1 51145,N1(CCCc2cc[nH]n2)CCCN2CCCC12 51146,CC(C)CC(C)NC(=O)CCN(C(=O)CC1OCCO1)CCCO 51147,CCC(CC)(CCNC(=O)C(C(C)(C)C)SC)NC(=O)Cc1cc(C)nn1C 51148,C1(N(C(C2CCC(=O)C2)=O)CC)CCN(C(C2CCNC2=O)=O)CC1 51149,C1(C(N2CC(OC)C(NC(C3CC3C3(C)COC3)=O)C2)=O)CCC(O)CN1C 51150,c1(C(=O)NCC2C(CNC(C3(CC=C)CC3)=O)C2)cnc2[nH]ncc2c1 51151,N1(C(Cc2cc(=N)[nH]cc2)=O)CCCC(NC(c2cccc(CO)c2)=O)CC1 51152,c1(OC)ccc2[nH]c(C)c(C(=O)NC(CNC(=O)CCC(C)SC)C(C)C)c2c1 51153,CC(C1OCCc2ccccc21)NC(=O)NCCc1cn(CCS(=O)(=O)F)nn1 51154,c1(N2CC(C(C)NC(=O)CSC3CC3)OCC2)cc2nncn2cn1 51155,C#CCC(O)C(=O)N1CCOC(Cn2cc(-c3ccnn3C(C)C)nn2)C1 51156,N1(C(c2ncn(CC=CC)c2)=O)CCC2(CC1)CN(C(C1COCCN1CC)=O)C2 51157,c1(CN(C(C(=O)NC(CSC)(C)CO)=O)C)cc(C)ccc1Cl 51158,CCC(C)C(C(=O)NCC1(NC(c2ccc(C)cc2Cl)=O)CC1)NC(C)=O 51159,c1(OC)ncccc1C(F)F.c1(C2(C3CC3)CC2)nnc(C2CN(C(=O)OC(C)(C)C)C2)s1 51160,C1(C(=O)NC(CNC(C2C(=C)C2)=O)CC=C)CCC2(CC2)C1 51161,Cc1ccccc1C=CC(N1CCC1(C)CC(=O)NC1C2CCCC1CC2)=O 51162,C12(C(N3CCC(C#C)(O)C3)=O)CCCC1CCN2C(=O)C(F)=CCC 51163,C1(C(=O)NCCN2CCCCC2=O)CC12CCN(C(=O)CCCC1CCCO1)CC2 51164,CN1C(=O)CCC1CNC(=O)CC=CCNC(c1ocnc1C(F)F)=O 51165,C(C)(C(=O)N(C)CC1(NC(c2nc(OC)c(C)s2)=O)CC1)(C(C)C)OC 51166,c1(C(N2CCCC(N(C(=O)C3=CCCO3)C)CC2)=O)ccc2cncn2c1 51167,C=CCC(F)(F)CNC(=O)CN(C)C(C1CCN1C(C)(C)C)=O 51168,C1(C(N(C(C)CC(=O)N(C)CCC2CCCO2)C)=O)C2CN(C)CC12 51169,c1(C(=O)NCC2N(C(C3CC(C#N)C3)=O)CCOC2)ccc(Cl)c(C(=O)OC)c1 51170,c1(-c2ccc(CN3CC(C(=O)OC)C(C)CC3)s2)cccc(F)c1C#N 51171,C(CC(C)(C)CC(=O)NCC(C)(O)CNC(=O)C(C)=C1CCC1)OC 51172,C(=O)(CC(C)CC(=O)N1CCC(C)(C)C1C(=O)NCCc1cc(C)no1)OC 51173,c1(CC=C)ccccc1C(=O)NC(C)C=CC(=O)N(C)Cc1c(C)noc1C 51174,C1(NC(C=Cc2c(C)ccs2)=O)CN(C(=O)CC2CSCCS2)CC12CCC2 51175,c1(C(=O)NCCC2CCN(C(CCN(C)CC)=O)C2)cc2c(Cl)nccc2s1 51176,c1(C(=O)NCCN(C(C2CC(F)(F)C2(F)F)=O)CC)nccc(Br)c1O 51177,CC(F)(C(=O)N1CCC(CCCCNC(=O)Cc2ccccc2F)CC1)C(F)(F)F 51178,CCCC(C(=O)NCCCN(CCC)C(C1CCN(C)C1C)=O)NC(N)=O 51179,C1(NC(CCOCC)=O)COC2C(NC(C3CC3n3ccnc3C)=O)COC12 51180,c1(C(N(C2CCCN(C(C(C)NC(C)=O)=O)C2)CCO)=O)ccc(F)c(C)c1N 51181,c1(C(c2cn(C)nc2-c2ccnn2C)c2onc(C3CNC3)n2)ccc(F)c(F)c1 51182,CC1CN(C(C2CCN2S(C)(=O)=O)=O)CC1(C)CNC(=O)CNS(C)(=O)=O 51183,Cc1cnc2c(C(=O)NC3CN(C(=O)C=C4CCC4)C(C)(C)C3)cccn12 51184,C1(C(N(C(C)COC)CC)=O)(CNC(=O)C(N)=O)CCCCC1 51185,c1(C(=O)OC)n[nH]c(=NCC(O)CNC(=O)CC2CC(O)C2(C)C)s1 51186,N1(C(c2ncn(C)n2)=O)CCCC(C(N2CCC(F)(CF)CC2)=O)CC1 51187,N1(OC(c2c(CCCC)[nH]cn2)=O)CCN(C(=O)C(C)(C)Br)CC1C=C 51188,c1(CCC)cccc(C(N2CCC(C)(CNC(=O)CCS(C)=O)C2)=O)c1 51189,N1(C(C2CN(C(C)=O)C2)=O)CC(C(=O)NCC(C)(F)C(C)C)C(F)(F)C1 51190,c1(C2C(C(=O)NCC3CC(NC(=O)C(O)C4CCCC4)C3)C2)ccc(F)cc1F 51191,C(c1ccccn1)=C(C)C(=O)NC(C)C(C)NC(=O)CN(C1CCC1)C 51192,CC(c1cccs1)=CC=CC(=O)NCC1(C)CCCN1C(=O)CO 51193,N1(C(CC(=O)NCC#C)=O)CCC2CC12C(=O)NC(CO)C(N)=O 51194,C#CCC(CC(=O)NCC#CC1CC1)NC(=O)CN1CCC(C)C1 51195,C(C)(c1cnccn1)=CC(=O)N(CCC(=O)N(C)CC1CC1(F)F)CC=C 51196,C1(C(=O)OC)CC2(C1)NC(=O)N(Cc1cccc(I)c1)C2=O 51197,c1(C(N(CCOC)CCNC(=O)CC2CCCCC2O)=O)c(C)cc(C)cc1O 51198,C1(F)(C(N2CCC(OCC=C)C2)=O)CCCN(C(=O)CN2CCOC2=O)C1 51199,c1(C(CO)NC(=O)NC2N(C(CCC)=O)CCCC2)cc(F)cc(Cl)c1 51200,c1(C(=O)NC2CN(C(c3cc(CC)[nH]n3)=O)C(C)C2)ccc(=O)n2c1COCC2 51201,C1(C(=O)NCCC2(C(=O)NC(C34CCC(CO3)C4)C)CCC2)CCOC(=O)CC1 51202,c1(OC)ccc(CCC(N2CC(CNC(=O)Cc3ccsn3)C(O)C2)=O)cc1N 51203,c1(NC(=O)C(N2CC=CC2CNC(=O)C(F)(F)C(O)C2CC2)=O)cc(O)cc(Cl)c1 51204,C1(NC(C2C(C)(CC)C2)=O)CC2CCC(C1)N2C(C1(SC)CC1)=O 51205,c1(C(=O)NC(CC=C)CNC(C2CCCC(O)C2)=O)cccc2c1CCCN2 51206,C1(C(=O)NC2CC(N(C(C(C)OCC=C)=O)C)C2)CCC2(CC1)CC2(F)F 51207,Cc1cc(C(=O)NCCC(O)CNC(=O)CCC2CC2)n(CCO)n1 51208,CCCC(C)(O)C(=O)NCCOCCNC(=O)Cc1ccc(Cl)cc1Br 51209,C1(NC(=O)NC(c2ccc(OC)nc2)C)(CO)CCCCC1C 51210,N1(C(C2CCC(CCCCC)O2)=O)CC=CC(NC(=O)C(C)(Cl)Cl)C1 51211,CC1CN(C)CCN1C(c1ncccc1N(CCO)CCO)=O 51212,C(CCCCC(=O)N(C1CCN(C(=O)C(C)OCCOC)C1)CCO)=CC 51213,C(CC(C)C)(C(=O)N(c1ccn(C)n1)C)ONC(C(C)OC(C)=O)=O 51214,c1(C(=O)Nc2c(C(C)=O)cccc2C)nn(C)c(Cl)c1I 51215,C(=O)(C#CC(C)(C)O)N1CC(c2cn(C(C(C)Oc3ccccn3)=O)nn2)C(O)C1 51216,n1(CC(=O)N(CCCCCCCN)C)nc2ccccn2c1=O 51217,Cc1nncc(C(=O)NC2CCC(CCC(=O)NCCN3CCCC3C)C2)c1C 51218,c1(OC)cccc(C=CC(=O)NC2CC2NC(=O)CCc2nnc(S)nc2O)c1 51219,Cc1cc2c(CC(=O)NCCN(C(c3ccc(=O)n(C)n3)=O)C3CC3)csc2s1 51220,C1(NC(C2C(C)(Br)C2)=O)CC(F)CN(C(C)(C)C)C1.c12cc(ncn1)N2 51221,C1(NC(C2CCC(=C)CC2)=O)CCN(C(=O)Cn2cc(C(F)(F)F)nn2)C(C)C1 51222,C1(C(=O)NCC(C)C(=O)N(C)Cc2ccncn2)C(C)(C)C1(F)F 51223,C1(F)(C(=O)NC2C(C(C)C)CCCC2)CCN(C(c2ccccc2)=O)CC1 51224,C1(NC(=O)CS(=O)(=O)NC2CC2)CN(C(C23CC4CC2C3C4O)=O)CCC1(F)F 51225,N1(C(c2cnc(CC)nc2C)=O)CC2CC(C1)CN(C(C1CCCC1C(N)=O)=O)C2 51226,c1(NC(CC(c2ccccc2)CNC(C(C)=CC2CC2)=O)=O)ccc(F)cc1O 51227,N1(C(C(C)Sc2ccoc2)=O)CC2(C1)CN(C(=O)CC1(C#N)CCOCC1)C2 51228,CC1(CNC(=O)COc2ccsn2)CCCN1C(=O)CSCc1ncc[nH]1 51229,N1(C(c2[nH]cc(C(=O)OC)c2)=O)CC2C(CNC(=O)C=CCCC=C(C)C)C2C1 51230,C1(OC)CCCC(C(N2CCC(NC(C3(C(C)(C)C)CCC3)=O)C2)=O)C1 51231,c1(C2C(C(C(=O)NCCC#N)N(C(C3COC3)C)C)C2)ccc(F)c(F)c1 51232,C(CCCC(=O)N(C)CC1CCCN1C(=O)CCNC(c1ccccc1)=O)OC 51233,c1(C(N(C2CCN(C(CN(CCOC)C)=O)CC2C)C)=O)cc2cccnc2o1 51234,CC1C(NC(=O)CC2(O)CCCCC2)C(C)CCN1C(=O)CC1CC(C)(C)CO1 51235,Cc1nnc2n1CC(C(N1CCN(C(C3CC(C(C)C)=NO3)=O)CC1CO)=O)C2 51236,N1(C(C(NOC)=O)=O)CCC(C=CC(=O)N(CCN=[N+]=[N-])C)CC1 51237,C1(C(=O)NCC(F)F)CCCN(C2CC3C=CCC23)C1 51238,C1(NC(C(=O)NCCOC)=O)CCCCN(C(=O)Cn2ccnn2)C1 51239,CC(C)(CC(F)(F)F)C(=O)NCC1(F)CCN(C(C2CCC3(CCC3)C2)=O)CC1 51240,C1(O)(CN(C)C(c2ccnn2CCF)=O)CCN(C(=O)COC2CCOC2)C1 51241,C1(C)(C)CSCCO1.c12cn(nn1)C1CN(C1)C2=O.n1(CC)cc(C2CC2)nn1 51242,CC1CN(C(c2cccc(N(C)C)n2)=O)CC1NC(c1ncsc1Br)=O 51243,c1(OC(C)C)c(F)cc(-c2ccccc2C(N2CC3CCC2C(O)C3)=O)cc1F 51244,C1(NC(CSCC(C)C)=O)CCN(C(=O)Cc2cncn2C)CC1 51245,N1(CCNC(c2c[nH]nc2-n2cc(-c3cc(CC)on3)nn2)=O)CCCNC1=O 51246,C(=O)(C(C)CC(C)C)N1CCN(C2CN(C(C3(C=C)CCC3)=O)C2)CC1 51247,c1(CC)cncc(CNC(c2coc(CNC(=O)CCc3ccn(C)n3)c2)=O)c1 51248,C1(CNC(c2c(C)coc2)=O)CN(C(=O)C(O)C2CCC2)CC1(F)F 51249,C(CO)(CCCCNC(c1ccnn1C(F)F)=O)NC(c1c(C(C)C)ncs1)=O 51250,N1(C(CCc2scc(COC)n2)=O)CCCC(C)(NC(=O)C(O)C(F)F)C1 51251,c1(C(N(CCCNC(=O)C(C)CC2CCCCC2)CC)=O)nccc(C)c1F 51252,C1(NC(C2CCN(C(c3c(C)nsc3N)=O)C2)=O)CC=C(C(C)C)CC1 51253,N1(C(CCC#CC)=O)CCC2(CC(NC(=O)Cc3nc([N+](=O)[O-])n[nH]3)CO2)C1 51254,c1(CC)n[nH]cc1-c1cn(CC2(OC)CC(CO)C2)nn1.OC 51255,Cc1cc(Cl)cc(C(N2CC(NC(=O)CSc3ccncc3)CC(C)C2)=O)c1N 51256,C(=O)(CP(C)(C)=O)NC1CCN(C(c2n(C)nnc2)=O)C1 51257,c1(C(N(c2ncc(F)s2)C)=O)cccn2ccnc12 51258,c1(C(=O)OC)cc(C(=O)NC2(C)CN(C(=O)CC3(C)CCCO3)C2)cc(C)c1 51259,C(=O)(C(C)(C)CC(F)(F)F)N1C(C)CC(NC(C2NC(=O)OC2C)=O)C1 51260,N1(C(C2(C)CCCN(S(=O)(=O)CCBr)C2)=O)C2CCCC1COC2 51261,CCCCCC(CC)C(=O)NC1COCCN(C(c2cc(N)cnc2Cl)=O)C1 51262,C1(CC=C)(NC(COCCCC#C)=O)CCCN(C(=O)C(C)NS(=O)(=O)CCC)C1 51263,C1(C(=O)NC2(CNC(C(CC)C(F)(F)F)=O)CC2)Cc2ccccc2CO1 51264,c1(C(N(CC(=O)NC2CCC2NC(C2CC23CC3)=O)C)=O)ccccc1Cl 51265,c1(-n2cc(C(C)NC(c3ccoc3)=O)nn2)cccc(Br)c1Cl 51266,CN1CCC(C(=O)N(C(=O)C(N2CCC(O)CC2)C)CC2CCC2)CC1 51267,CC(C)(CC(F)(F)F)C(=O)N1CCN(C(=O)CCCCC(N)=O)C(C(F)F)C1 51268,C(=O)(C(C)(C)S(C)(=O)=O)NCC(CCNC(C(CC(C)(C)C)NC(C)=O)=O)C 51269,N1(C(CN(CC)CC)=O)CCCC1C1CCCN1C(c1cn(C)ccc1=O)=O 51270,c12cc([nH]n1)N2.C1(C2(C)N=N2)CC(CN2CCCC2)C1 51271,c1(C(N2CCC(CNC(c3cc(C(C)(C)C)n[nH]3)=O)CC2)=O)cnc2n1CCS2 51272,C1(C(=O)NCC(F)F)CC12CCN(C(=O)C=Cc1cscn1)C2 51273,Cc1cc(=NCCCN2CCC(N3C(=O)CCC3=O)CC2)[nH]c(NS(C)(=O)=O)n1 51274,N1(C(C(CC(=C)Cl)NC(=O)Cc2ccn(C)n2)=O)CC(=O)NC(C)(C)C1 51275,c1(C2C(C(=O)NCC(CNC(c3cc(OC)ns3)=O)(C)C)C2)cccc(C#N)c1 51276,C1(C(N2CC(OC)C(C(=O)NC3C(C)(C)C3(C)C)C2)=O)CCCCNC1=O 51277,c1(COC)nccc(=NC2CC3CN(C(=O)C(C)(C)c4ccccn4)CC23)[nH]1 51278,C1(C(C)NC(=O)CCNC(C2CCO2)=O)CCOCC1 51279,N1(C(CCCOC)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)CCc1nccs1 51280,N1(C(C(C)=C(C)C)=O)C(C(N2CSCC2C(=O)N(C)C)=O)CCC12CC2 51281,C1(C(N(C(C#C)C)C)=O)C2CCC(C2)C1NC(C1CCC1C#N)=O 51282,C=CCCCCC(=O)NCC(c1ccc(CNC(=O)CC(F)(F)F)cc1)(C)C 51283,Cc1occc(=O)c1OCC(=O)Nc1cncc(C(=O)Oc2ccccc2F)c1 51284,N1(C(C(C)n2cccc2)=O)CCC2(CC(C(=O)Nc3cncc(Br)n3)=NO2)C1 51285,c1(CC(C(=O)N(C2CCN(C(c3cnc(CC)[nH]3)=O)C2)C)C)c(C)n[nH]c1C 51286,N1(C(C=NOC)=O)C(C)CC2CN(C(=O)CC3C=CCC3)CC12 51287,C1(CC(=O)N(C(C)C(=O)NCCC2CCC2)C2CC2)CCN(C)CC1 51288,C12(C(=O)NC(CCCC)CNC(=O)C(F)n3ccnc3)C3CC(CC13)C2(F)F 51289,N1(C(c2c(OC)cncn2)C(=O)NCCCSC)CC(CO)C(C2CC2)C1 51290,c1(COC(CC)(C)C)cn(C(C)C)nn1.c12ccc(o1)NC(=O)C(C)OCCS2 51291,C1(C(=O)NC(CC=C)CNC(c2cnc(C)[nH]2)=O)CCC(n2cccc2)CC1 51292,c1(C(=O)NC2C(NC(CC(CC)C3CCC3)=O)CCCC2)ncnc(C)c1C 51293,C(CC(C)(C)NC(=O)Cc1ccccc1)NC(CN(C)C1CC1)=O 51294,C1(NC(CC2(C=C)CC2)=O)CCCCN(C(c2cc(C)n(CC)n2)=O)C1 51295,N1(C(CC(C)O)=O)CCc2c(C(N3CC(C(F)(F)F)C4(CC4)C3)=O)csc2C1 51296,CCCCCC(O)CC(=O)N1CC2CCCC2(C(=O)NCC(C)C(C)(F)F)C1 51297,C(=O)(C(CNC(=O)COCCOCC)C(C)C)NC(CCC(=C)C)C 51298,c1(OC)cncc(C(N2CCOC(CNC(c3sccc3C3CC3)=O)C2)=O)n1 51299,Cc1ccc([N+](=O)[O-])cc1C(=O)NC1CN(C(=O)C(C)CF)CCC1C 51300,C(CNC(=O)C(C1CCCCCC1)C)(CC(C)C)NC(CC1(C=C)CC1)=O 51301,C1(NC(CC2(COC)CC2)=O)CCCN(C(c2ccc(C3CC3)cc2)=O)C1 51302,C12(CNC(C3CCC(C)C3)=O)CC(CN1C(=O)C(C1CCCCC1)N(C)C)C2 51303,c1(N(C(c2cnc(NCCO)nc2)C(=O)NCCCF)C(C)(C)C)ncc(Cl)n1C 51304,c1(CC)nc(C(N2CCC2C(=O)NCc2nc(=N)[nH][nH]2)=O)cs1 51305,c1(CC(=O)NC(CCNC(CC(CC)SC)=O)C)ncn2c1CCCC2 51306,CC1CCC(NC(C2C(CNC(=O)CCOCC(F)(F)C(F)F)COC2)=O)CC1 51307,c1(C(=O)NCCN(C(Cc2c(C)ccs2)=O)C)ccc2[nH]ccc(=O)c2c1 51308,C1(C(=O)NC(CN(C(C2(COC)CCCO2)=O)C)(C)C)CC2CCC(C1)C2 51309,C12(C)NC(=O)N(C1=O)C2.C1(C)(c2nc(C)on2)CN(C(=O)OC)C1.C(C)(C)(C)O 51310,c1(C(N2CCC(CSCCCC)CC2)C(=O)NCCOCC)c(C)cccc1C 51311,Nc1cccc(C(N2CCC(CNC(=O)CCc3ccc(O)nc3)C2)=O)c1 51312,c1(OC)noc(C)c1C(=O)NC1CCC(C(=O)NC(c2cncs2)C)CC1 51313,c1(CCC)ccccc1.CCC(CNC(=O)CO)NC(=O)CC1CCC1.C1CN1S 51314,Nc1ccc(F)c(C(N2CCC(NC(=O)Cn3ccnc3)C(F)C2)=O)c1 51315,C(CCNC(C1CC(N)CCN1C)=O)(C(F)(F)F)OC 51316,c1(CN(C)C(C2COCCN2C(=O)CC2CC2)=O)ccc([N+](=O)[O-])cc1 51317,c1(OC)cc(C)c(C(N2CC(COC)(NC(c3ccc(C)c(C)n3)=O)C2)=O)cn1 51318,n1(CC(=O)OCC)nc(C)c(S(=O)(=O)N2CC(O)CC2C(=O)OC)c1C 51319,c1(C(=O)NCC(F)CO)cccc2ccnn12.C12(CC1)C(=O)N2 51320,c1(C(=O)NCC2C(C)CN(C(C3CC(O)C3)=O)CC2)nc(Cl)c(=O)[nH]c1N 51321,C1(C(=O)NC2CC(CNC(C(Cn3ccc(C)n3)C)=O)C2)CC(=O)N(C(C)C)C1 51322,c1(C(=O)NC(CNC(c2cnc(OCC)nc2)=O)CC(C)C)ccc(F)cc1C 51323,c1(C(=O)NCC(C)N(C)C(c2cnc3[nH]ccc3c2)=O)nc2cc(O)ccc2[nH]1 51324,N1(C(C(C=C)(F)F)=O)CCS(=O)(=O)C(CCNC(=O)C(C)N(C)C(C)=O)C1 51325,N1(C(CC(CC)OCCN(C)C)=O)CCC(C(=O)NC2CCCCC2O)C(C)C1 51326,C1(O)(C(=O)NCC(N2CCOCC2)C)CCCC(C)(C)C1.C12(CCC1)C(=O)NC2 51327,c1(OC)ccnc(NC(=O)C(N2CCNCC2C#N)=O)c1F 51328,S(=O)(=O)(c1cc(Br)c(Br)s1)N1CC2(CCN(Cc3cncc([N+](=O)[O-])c3)C2)C1 51329,C(=O)(C(Cn1cncn1)NC(=O)C(C)SC(C)C)N(CCC=C)CC 51330,C1(NC(c2cc(N)c(Cl)nc2)=O)CCCC12CN(C(=O)Cc1cncnc1)C2 51331,c1(C(=O)NCC(CN(C)C(C2(n3nccn3)CC2)=O)O)csc(Cl)c1 51332,C1C(=O)N=C2C=C(N(C)N2)O1.N12C(CC)C1CCCC2C(CCCCSCC)=O 51333,C(C(CNC(c1ccc(SC)cc1)=O)C(F)(F)F)NC(CCCC#C)=O 51334,c1(C(COC(C(C=C)OC)=O)=O)cc(C)cc2cccnc12 51335,C1(NC(c2nsnc2O)=O)C=CCCC1C(=O)NCC(CO)C1CC1 51336,c12ccccc1C(C)NC2=O.N1(CCC(C)C)CCCC1Cn1cc(CO)nn1 51337,c1(NC(C2(NC(C(CC)n3ccnc3)=O)CCSC2)=O)ccc2c(c1)COC2 51338,C1(Cc2cccc(Br)c2)CC(=O)N1.CCCS(=O)(=O)NCC1CC(F)(F)C1 51339,c1(CC)ncc(C(=O)NCC(O)CNC(C2CCCN2C(=O)NC(C)C)=O)s1 51340,c1(C(=O)NC(C2CCOC2)CNC(c2ccc(Cl)[nH]2)=O)ccc(F)c(C2CC2)c1 51341,N1(C(CC(=C)C)=O)CC2(CCC(CNC(=O)C(C)Cc3ccc(C)cc3)O2)C1 51342,N1(C(C2(C(=O)NC)CCC2)=O)CCN2CCN(C(=O)C(O)CC(C)C)CC2C1 51343,N1(C(C(CC=C)OC)=O)CCC(NC(=O)C(F)CCCCC)C(C)(C)C1 51344,c1(NC2CC(OC)C23CCC3)nc2c(cc1C#N)CCOC2 51345,CCS(=O)(=O)CCN(C)Cc1csc(-c2cccc(Oc3cccc(Cl)c3)c2)n1 51346,C1(CNC(C2CC(CCC)C2)=O)CN(C(=O)CC(F)F)CC1C(F)(F)F 51347,C(=O)(CCCCCN(C)C(C1COC(C)C1)=O)NC(CC)CO 51348,C(C(O)CNC(=O)CN(C(=O)COC)C)NC(C=CCC)=O 51349,N1(C(C(CC#CC)NC(=O)CCCC2CC2C=CC)=O)CC(C)OC2(CCC2)C1 51350,C#Cc1ccc(C(N2CCC(CNC(c3cnc(N)cn3)=O)CC2C)=O)c(F)c1 51351,CCC1C(=O)N2CC=CC2C(=O)NCC1.c1(C(=O)OC)ncccn1 51352,c1(C(=O)NCCN(C(C(CC)n2ccnc2)=O)C)cc(OC)c(Cl)cc1OC 51353,c1(C(N2CC(CNC(CCc3n(C)ccc3)=O)OCC2)=O)cnc2[nH]ccc2n1 51354,Cc1oc(C(=O)NC2CC3CCC2N3C(=O)C(O)C(C)C)cc1S(N)(=O)=O 51355,C1(NC(C2(CC)CC2)=O)CCCC(NC(=O)C(c2ccc(O)cc2)=O)C1 51356,N1(C(CSCC=C)=O)CCC(F)(CNC(c2ccc(N)cc2Br)=O)CC1 51357,c1(CNC(C=C(C)CNC(=O)COCC(C)C)=O)nc[nH]n1 51358,Cc1c(C(N2CCCN(C(=O)CC3CC(O)C3(C)C)CC2)=O)cc(F)cc1Br 51359,c1(NC(Cc2ccc(OC)nc2)=O)nc(F)ccc1OC(C)C 51360,C1(C(NOCC)=O)CN(C(=O)CN2CCC(=O)CC2)CC1(F)F.c1cc(CC)[nH]n1 51361,N1(C(C=COCC)=O)CCCC2(CC(NC(=O)Cc3sc(C)nc3C)C2)C1 51362,N1(C(C(CO)NC(c2ccc(F)cn2)=O)=O)CC2CC1CO2 51363,C(CN=c1[nH]c(=NC2COCC2SC)[nH]c2c1COC2)N(CCOC)CC 51364,c1(CCC)c(C(=O)NCC(CC)NC(=O)CC2CC=CCN2C)cnn1C 51365,C1(NC(C(C)=CC)=O)CC2CC1N(C(=O)CC(C(F)F)c1ccccc1F)C2 51366,c1(C(N2CCCC(NC(c3c(C)snn3)=O)CC2)=O)ccc2c(c1)COCCN2 51367,C1(C2(O)CN(C(c3n[nH]cc3[N+](=O)[O-])=O)C2)(CNC(=O)Cc2ncc(Cl)s2)CC1 51368,C(=O)(CCCC(F)F)N1CCC(N(C(C(C(C)C)C)=O)CC2CC2)CC1 51369,C1(NC(=O)C(CO)NC(c2ccon2)=O)CCCC(CO)C1 51370,N1(C(CN(CCOC)C)=O)CC(CNC(C2CCC(C)(C)OC2)=O)CC12CCC2 51371,C=CC(C)CC(=O)NCC(CC)NC(c1coc(SCC)c1)=O 51372,c1(SC)ccccc1CCNC(=O)NC1CCOC(C(F)(F)F)C1 51373,c1(COC(C2CC(=O)N(C3CCOCC3)C2)=O)ccnc(-c2ccccc2)c1O 51374,C(N=c1[nH]c(=N)[nH]c(=NCc2ccccn2)[nH]1)C1(N(C)C)CCCC1 51375,C1(C(C)=O)CC1(Cl)C(=O)NC1CC1NC(=O)COc1cn[nH]c1 51376,CCC(C)CC(C)C(=O)NCC1(C(N2CC(O)C(O)C2)=O)CCCC1 51377,c1(OC)ccc(C(C)C(=O)NC2CC3CC(NC(=O)CP(C)(C)=O)CC23)c(C)c1 51378,N1(C(CCC2CC(OC)C2)=O)CCN(C(=O)C(CN(C)C)N(C)C)CC1CO 51379,N1(C(CCc2ncc(C)[nH]2)=O)CCCCC(CNC(C2CCCN2C(C)C)=O)C1 51380,C1(NC(C(CC#C)NC(=O)C(C)CC2CC2)=O)CCCOC12CCC2 51381,C1(C(=O)NCC2(F)CC(CNC(=O)CC3CCCCC3O)C2)CCCCC12CCC2 51382,C(C)(CC(C)C(F)F)NC(CN(C(c1cc(CC)[nH]n1)=O)C)=O 51383,C1(O)(C(C)C)CCN(C(C2(NC(=O)C(C)C3CC3)CCOCC2)=O)C1 51384,CC1=C(C(=O)N2CC(C(O)C(=O)NC3COCC3CN(C)C)C2)CCC1 51385,Cc1ccc2cc(C(=O)NC(C)(C)CNC(C3CCC4(CCOC4)O3)=O)[nH]c2c1 51386,C1(CCC)CCCC1C(=O)NCC12CC(NC(=O)COC3CCC3)(C1)C2 51387,N1(c2nnc(C)n2C)C(=O)C23CCCC2CCN3C1=O 51388,C(C(C)(C)C#CC(=O)N(CCSC)CC)NC(C(CC)COC)=O 51389,C1(C)(CNC(CC=CC=C)=O)CCN(C(C2(C=C)CCOCC2)=O)CC1 51390,C1(C(=O)NCC2(C)CC3CC3C2)CN(C(=O)Cc2cscn2)CC1(F)F 51391,N1(C(CCc2n(C)ccn2)=O)CC2(CC(CNC(=O)CCc3ncc[nH]3)C2)C1 51392,c1(OC(C)C)ccc(F)c(C(=O)N(CCNC(c2cc(F)c[nH]2)=O)C2CC2)c1 51393,c1(C(N2C(CCNC(CCOC)=O)CC(OC)C2)=O)ccc(=NC)[nH]c1 51394,C1(NC(=O)COCCOC(C)=O)CC(C(CC)=O)CCO1 51395,N1(C(C2C(=C)C2)=O)CCC2(CC(NC(c3c(-c4ccccc4)coc3C)=O)C2)C1 51396,N1(CC(=O)NC2C=CCN(C(c3c(CCC)[nH]cc3)=O)C2)CCCCS1(=O)=O 51397,N1(C(C(C)SC)=O)CCC(C2CCCN(C(c3c(Cl)nn(C)c3Cl)=O)C2)C1 51398,C1(C)(NCCOCCCCC)CCC(C)CC1.N12CCN(CC1)C(=O)C2 51399,C12(C(=O)NC(CC(=O)O)C(=O)O)CC3CC(C(=O)N1)C2C3 51400,C1(NC(CCCCOC)=O)CC2CCCC(C1)C2NC(c1ccco1)=O 51401,CC(C)CC(=O)NCCO.c1(CC(c2ccco2)NC=O)ccccn1 51402,N1(C(C(C)OC)=O)CCN(CCC2CCCCN2C(c2ccnnc2)=O)CC1 51403,c1(C(N2C(C)CC(NC(CC(C)(C)OC)=O)C2)=O)cccc2[nH]cc(Cl)c12 51404,C(=O)(CC(O)CNC(c1cc(C2CC2)sn1)=O)NCc1ncn(CC)n1 51405,CON1CC(C(=O)NCC2CCCC2C(=O)NCC2(CO)CC=CC2)CC1=O 51406,C1(C)(c2nnnn2C2CC2)CCCN1.C1(C)(COCC(C=C)(F)F)C=CCCC1 51407,c1(N(CCNC(c2n[nH]c3c2CCSC3)=O)CC)nc(O)c2ccc(Cl)cc2n1 51408,N1(C(c2c(CC)cnnc2)=O)CC2CC(C)N(C(c3cccc(F)c3C)=O)C2C1 51409,c1(OC)ccc(NC(C2CC(NC(=O)C3=CCCOC3)C2(C)C)=O)cc1C 51410,N1(C(CC(CC)OC)=O)CC(N(C(=O)CCOC)CC)C2(CC2)C1 51411,c1(C(N2C(C(=O)NCCc3c(C)cccc3)CCCC2)=O)cc(C)c(C)cc1I 51412,O=C(CCCc1ccc2c(c1)OCO2)NNC(=S)NC1CCOC1 51413,C1(C(=O)NC2CC(N(C(=O)COc3cccnc3)C)C2)CCCC(=O)O1 51414,Cc1cc(N2CC3CC3C2)nc(=NCCc2ccc(C(F)(F)F)o2)[nH]1 51415,C1(CC#C)(NC(=O)C=CCNC(=O)CC2CCCO2)CCC1 51416,c1(OC)cc(OC)c(CC(=O)NCCCOCCC2CCC2)cn1.C1(=O)CN1 51417,C(CC(C(C)(C)C)NC(C1CCC(=O)C1)=O)N(C(c1cn(CCOC)nn1)=O)C 51418,N#CC1(C(N2CCOC(CNC(=O)CCC(N)=O)C2)=O)CC(F)(F)C1 51419,c1(C(=O)NC(C)CC(C)NC(C2CCCC2c2cnn(C)c2)=O)ccc(O)nc1 51420,C1(C(=O)NC(CN(C(c2c(C)nc(C)[nH]2)=O)C)(C)C)CC2COCC2C1 51421,C(CC(C)CC)(C(=O)N(CC(C)(C)CO)C)NC(CC1CC(=C)C1)=O 51422,Cc1ccc(C(=O)NC2CC3C(NC(c4ccc(C(C)C)cc4)=O)C3C2)cn1 51423,C1(C(=O)NCCC(=O)NC)CCc2cnnn2C1 51424,C1(CCCNC(C(C2CC(F)(F)C2)OC)=O)CCCN1C(=O)C=CCO 51425,c1(CC)c(Cl)nc[nH]c1=NCC1CN(C(C2CC(=O)N2)=O)CC1C 51426,N1(C(CCCOCC)=O)CCN(C(c2cc(OC)ns2)=O)CC1C1CC1 51427,N1(C(C(CCCC)O)=O)CCC2(CC1)CCN(C(C1(C(C)C)CC(F)(F)C1)=O)C2 51428,C1(C(N2C(CCNC(c3coc(CO)c3)=O)CCC2)=O)CCn2ccnc2C1 51429,c1(CN2CCN(C(c3ccc(C)[nH]3)=O)C3C2C3)cc([N+](=O)[O-])ccc1O 51430,Cc1cccc(CONC(C2(NC(c3cnc(O)o3)=O)CCCC2C)=O)n1 51431,N1(CC(C)(C)OC)CCC(S(=O)(=O)Nc2ccccc2)C1 51432,N1(C(CCCC(=O)NC)=O)CC(CO)C2(C1)CN(C(=O)C(C)C1CCCO1)C2 51433,c1(C(=O)NCC(=O)O)cc2n(n1)CCCN(Cc1ccc3nc(O)oc3c1)C2 51434,c1(CC(N2C(CC)C(NC(=O)CCF)CCC2)=O)c[nH]c2cc(C)ccc12 51435,C12(CNC(C3CC(C)(CC)C3)=O)CCCC1N(C(=O)C(C)CN(C)C)CCC2 51436,N1(C(=O)Cc2cccc(Cl)c2F)CCOC2(C1)CN(C(C13COCC1C3)=O)C2 51437,N1(C(c2cnc(SC)s2)=O)CCC(NC(c2sc(C(F)F)cc2C)=O)C(F)C1 51438,C12(C(N3CC4CC(NC(C5CC(C)(O)C5)=O)C4C3)=O)CC3CC(C1)CC(O)(C3)C2 51439,N1(C(C(C=C)(C)O)=O)CCCC(C)(C(=O)NC2CCCCC2)C1 51440,CCC(C(=O)NCC(C)N(C)C(C1(C#N)CC1(C)C)=O)C(C)C 51441,c1(C(=O)NC2C(Nc3ccnc(SC)n3)CCCC2)cc(O)cc(O)c1 51442,c1(CN2C(CNC(c3c(C)ncn3C)=O)CCCC2)cc(Br)cc2c1OCC2 51443,N1(C(CCCCOCC)=O)CCC2CN(C(=O)CCC(CF)CF)CCC12 51444,Cc1ccc(NC(C2CCCCN2C(=O)CC2CCCC(=O)C2)=O)c(C)c1 51445,c1(C(N(C(CCNC(c2c(C)snc2)=O)C)C)=O)nn(C2CCC2)cc1Br 51446,c1(C(=O)NCC(COC)(C)O)ccc(NC(=O)C(F)CC2CCCC2)cc1 51447,C1(CNC(C(CC(C)C)O)=O)CN(C(c2ccccc2N)=O)CCC12CCC2 51448,c1(SC)ccc(C=CC(=O)NC2CCCCC2CNC(=O)C(C(C)O)N(C)C)s1 51449,C1(CC(=O)NC2(C=C)CCC2)CCN(C(C2CN(C(C)C)C2)=O)C1(C)C 51450,c1(CC)ccc(C(N2CCC2CNC(=O)C(CC)n2cncn2)=O)c(F)c1 51451,Cc1ccc(Cl)c(C(=O)NCC2(CCN(C(=O)Cn3ccnc3)C3CC3)CC2)c1O 51452,CC(O)C(C)(C)C(=O)N(CCC(C(C)(C)C)NC(=O)CN(C)C1CC1)C 51453,C1(OCC(C)NC(=O)NC(C)CC2(O)CCC2)CCCCC1 51454,c1(C(=O)NCCC(=O)NCCC2CC(OC)CN2C(C)=O)c(F)ccc(F)c1Cl 51455,C12(CCNC(Cc3ncc(C)s3)=O)CCC(C1)N(C(=O)CNS(=O)(=O)NC)C2 51456,C1(CC)(CC)CC(C(N2CC(CC(=O)C(C3(CN)CCCO3)=O)C2)=O)C1.CS(C)=O 51457,c1(NC(CN(CCC)C(c2cn(C)nc2OC)=O)=O)cncc(C)n1 51458,Cc1cc(C(=O)NCC(CNC(=O)C(C)C(F)F)CO)c(Br)s1 51459,S1(=O)(=O)c2cccnc2N2C(C)CN1C(C)C2.C(C(C)(C)SC)OC 51460,C(=O)(C1CCOc2ccccc21)N1CC(NC(c2nocc2C)=O)CC(OC)C1 51461,C=C1CC2CCCC(C1)N2C(C1CCCN(C(c2csc(=N)[nH]2)=O)C1)=O 51462,C(=O)(C#CC1(C)CCCO1)NCC(CNC(c1cc(Cl)ns1)=O)OC 51463,c1(N2CC3CC(NC(=O)CC4(O)CCC4)CC3C2)c([N+](=O)[O-])cccc1[N+](=O)[O-] 51464,CCCCC(O)C(=O)N1CC(CN(C)Cc2ccc(C(=O)O)s2)C2(CC2)C1 51465,C1(C(=O)NC2(CF)CCN(C(C3CCC(C)(C)C3)=O)C2)CC2(CC(=O)N2)C1 51466,N1(C(c2ncc(CC)cn2)=O)CCC2CCCC12C(N1CC2C(C1)C2(F)F)=O 51467,C1(C(N2C(c3nc(C)[nH]n3)CCC2)=O)(CN)CCS(=O)(=O)CC1 51468,C1(NC(C(=O)NCCC(CC)O)=O)CCC(C(C)(C)C)CC1 51469,C(=O)(C1CC(=O)Nc2ncn(C)c21)N1C(C)C(NC(=O)CSS(C)(=O)=O)CCC1 51470,Cc1nn(C)c(F)c1C(N1CCC(C(C)(C)NC(c2ccnc(OCN)c2)=O)C1)=O 51471,CCC(CC(=O)NC(CC1CC1)C(N1CCC(CCF)CC1)=O)CC(C)C 51472,CC(CC(=O)N(C)CCc1ccccc1)NC(=O)CC1(C#N)CC1 51473,C(CC(C)C)(C(=O)NCC1C=CC(C(=O)Nc2cccc(C(C)C)c2)C1)OC 51474,CCCCS(=O)(=O)N1CCCC1C(=O)N(CC(C)NC(=O)Cc1ccsc1C)C 51475,C(=O)(C#CC1(CC)CC1)N(CCNC(c1ccncc1NC)=O)CC 51476,C12(C(=O)NC3CN(C(=O)COC4CCCOC4)C3)CCN(C1)S(=O)(=O)C2.C(C=O)O 51477,N12CCC(C1(C)C)CC2=O.C1(CC)CC(C(=O)N2CCCC(OCCF)C2)=NO1 51478,c1(C(=O)NCCC2(C)CCN(C(CC(C)NC(N)=O)=O)C2)ccc2snnc2c1 51479,N1(C(C(CCC)OC)=O)CC(N(C(=O)C=Cc2cccnc2)C)C2(CC2)C1 51480,CC1(C)CC(C(N2CCC(=CCO)CC2)=O)CN(C(c2cnn(C3CC3)c2)=O)C1 51481,C12(C(=O)NCC=CCNC(c3c(C)occ3)=O)COCC(C1)C2 51482,C(C(CC(C)C)C(=O)N1CCC(C)(C)C(C(N2CCC(C(=O)NC)CC2)=O)C1)OC 51483,CCC(CCC(=O)NCC1(C)CCCCC1)NC(C1CC1(C)CC)=O 51484,C(=O)(C(CC)OC)N(C1(CC(=O)N(CC(C)(C)C)CCC#C)CC1)C1CC1 51485,C12(NC(C3CC(C#N)C3)=O)CCC(CC1)N(C(=O)CCC1CCCCO1)C2 51486,NS(=O)(=O)c1cc(NC(=O)Nc2ccc3c(c2)CC(=O)NC3)c(F)c(Br)c1 51487,c1(C(=O)NC2CCC(NC(CC(=O)OCC)=O)CC2)cnc(OCC(F)F)cn1 51488,c1(CCC)cnnc(NC(CC(=O)NCc2noc(CC)n2)c2ccccc2)c1 51489,N1(C(CCSCC)=O)CCN(C2CCCN(C(=O)C(C)NC(C)=O)C2)C(=O)C1 51490,c1(CC)cc(NCC(C)CNC(=O)C(=O)NCC2CC2)ncn1 51491,c1(CNCCNC(=O)NC23CCC(F)(CC2)CC3)c[nH]c2ncc(Br)cc12 51492,C(c1ncc(C)[nH]1)=CC(N1C(CN(C(C2CC2(OC)CC2CC2)=O)CC)CCC1)=O 51493,Cc1cc(=O)c(C(=O)OCc2ncsn2)nn1-c1cccc(Br)c1 51494,C1(C(=O)NC(C2CCCC2(C)C)C)CN(C(=O)Cn2cnnc2)CC1C 51495,C(CCO)(C(F)(F)F)NC(C(CC1CCC1)NC(=O)COCC1CC1)=O 51496,CCCCC(C(=O)N1CCN(C(c2cnsc2C)=O)CC1CF)NC(N)=O 51497,c1(CNC2CC(CC(=O)Nc3occ(C)n3)C2)cnn2cccc(C)c12 51498,N1(C(C=Cc2ccc(C)o2)=O)C(C(N2CC3CCCC3C2)=O)C2CCCC12 51499,c1(CSC)nc(C)ncc1-c1nc(CC(c2ccc(F)cc2)(C)C)no1 51500,c1(CC(=O)NCCC2CC(NC(CCc3ccc(C)s3)=O)C2)cn(C)nc1C 51501,c1(CC)csc(COC(n2cc(CC(=O)OCCN3CCOC3=O)nn2)=O)n1 51502,N1(c2n(CCOC)c(C(c3ccsc3)(F)F)nn2)CCN(C)C2(CCOC2)C1 51503,C=CCC(Cc1ccccc1)C(=O)NC1CCCC1NC(=O)CC(F)F 51504,c1(C(N(C)CC2CN(C(C(C)=CC)=O)CC23CC3)=O)ccc(S(C)(=O)=O)o1 51505,N1(C(C(C(C)C)SCC)=O)CCN(C(c2ccncc2N(C)C)=O)C(C2CC2)C1 51506,c1(C(N2CC3C(CNC(C4(C)CCN(C)C4)=O)(C3)C2)=O)cc(F)ccc1C1CC1 51507,S(=O)(=O)(c1ccc(F)cc1O)N(c1scc(-c2n(C)ncc2)n1)Cc1ccco1 51508,C1(NC2CC(c3cc(F)cc(F)c3)C2)CC(C(N)=O)C12CCC2 51509,C(C(=O)N(CCCCNC(=O)C(C)N(c1ccccc1)C)C)(C(C)C)NC(C)=O 51510,CC1C(=O)N(CC(=O)NC2(CNC(=O)Cc3nncs3)CCC2)C(=O)C1C 51511,C#CCCCCC(=O)NC1CCC(N(C)C(c2ccnnc2NC)=O)CC1 51512,N1(CC)CC(C(=O)NC2CCCN(C(C3CN4CCCN3CC4)=O)CC2)CCC1=O 51513,n1(CCCN(C2CCCC(C)C2)C2CC2)c(C(F)(F)F)nc2ccccc12 51514,Cn1nnc2c1CC(C(=O)NCC1(C)CC(NC(=O)Cc3ccon3)C1)CC2 51515,c1(C(=O)NCC(CN(C(Cn2c(C)ncc2)=O)C)O)cc(C(F)(F)F)cc(N)c1 51516,c1(C(N2C(C(=O)NCC(C)(C)CCO)C(C)(C)CC2)=O)cccc2[nH]ncc12 51517,N1(C(C(C)OC(C)(C)C)=O)CCC(NC(=O)C(C)CC(N)=O)C12CCC2 51518,c1(OC)ncccc1C(=O)NC(C)(C)CN(C(=O)Cn1ccc(C)n1)C 51519,c1(C(=O)NCC(C2CCCCC2)NC(CC(C)SC)=O)cc2n(n1)CCCN2 51520,C(=O)(CCC(C)(C)C)NC1C2(CC(NC(C(CC)(C)OC)=O)C2)C1 51521,c1(C(=O)NC2CN(C(C(CSC)C)=O)CC(F)C2)cc2c(nc3ccccn23)s1 51522,Cc1cc(C(C)C(=O)N(C)CCN(c2nc(C(=O)C3CC3)cs2)C)c(C)o1 51523,C1(NC(=O)C=Cc2cnc[nH]2)COC2(C1)CN(C(C1CC(C(F)F)C1)=O)C2 51524,c1(CC)nc(C)[nH]c1C(=O)NC(CNC(=O)C(C(C)C)NC=O)CC(C)C 51525,CC(C)(C(=O)NCCC1CCCN(C(=O)COCC(F)(F)F)C1)C(F)(F)F 51526,C(N=c1ncc(C(C)(C)O)c[nH]1)C1CCC(NC(c2c(C)ocn2)=O)CC1 51527,N1(C(C(C(CC)O)C)=O)CC2CCCC(CNC(=O)C(C(C)(C)C)N(C)C)C2C1 51528,c1(C(=O)NCCCN(C(CC(CC)O)=O)C)coc2cc(F)cc(F)c12 51529,c1(OC)ncnc(N(C2CCNCC23CC3)Cc2ccc(Cl)cc2)c1CO 51530,CN1CCN(CCCNC(=O)C(c2ccc(F)cc2F)F)CC1CO 51531,CCCCCC(=O)N(CC(C)CNC(=O)C(C)CCOc1ccccc1)C.OC 51532,C1(C(=O)NC2(CC)CCCC2)CCCN(C(c2ccc(C)cn2)=O)C1C 51533,CC(CC(=O)N1C(C(=O)N=c2ccn(CC#N)[nH]2)CC1CO)CC(C)(C)C 51534,C1(NC(c2c(C)nn[nH]2)=O)CCC2CC1CN2C(=O)CCCCCC#N 51535,c1(C(=O)OC(C)C(=O)N(C)C)cccc2c3c([nH]c12)CCCCC3 51536,C1(C(N(CCCNC(c2ccc(C3CC3)s2)=O)CC)=O)CCCCCN1C 51537,C1(NC(c2c(C)ccs2)=O)CCCCN(C(c2cnc(C(C)(F)F)s2)=O)C1 51538,C1(NC(c2c(CC)n[nH]c2)=O)CC2(CNC(=O)CCC3CCOCC3)CC1CO2 51539,C(=O)C(C)C(F)(F)F.CCCC(CCC)=CC(=O)N(CC(CC)C1CC1)C 51540,N#Cc1cc(C(=O)NC2CC(CNC(c3scnc3Br)=O)C2)co1 51541,c1(C(C)NC(=O)NC2CCC3CC23)cccc(Br)c1F 51542,C(=O)(C1=CCC(F)(F)CC1)N1CCC(C2(NC(c3cc(C)no3)=O)CC2)C1 51543,C#CCCC(=O)NCCn1cc(CNC(c2ccn(C(C)C)n2)=O)nn1 51544,C1(C(=O)NCC(C)N(C(C=CCC(=O)O)=O)CC)CC(N)C1(C)C.C(C)(C)(C)OC 51545,c1(NC(c2c(NC(C3C(C=C)OCC3)=O)cccn2)=O)c(OCC)cccc1C 51546,c1(C(=O)NC(C)CNC(=O)CC(F)(F)F)c(O)nc(=O)n2c1CCC2 51547,C(=O)(CS(=O)(=O)C(C)C)NC(CC1CN(C(CCn2ccc(C)n2)=O)C1)C 51548,C1(C(N(C(C)CCNC(C2CC3(CC3)CO2)=O)C)=O)CCS(=O)(=O)C1(C)C 51549,N1(C(C(=O)NCC=C)C(C)C)CCOC(C)(C(F)(F)F)C1 51550,C(C(F)(C(=O)NCC(O)C(C)O)C(C)C)NC(c1c(C)cc[nH]1)=O 51551,CCC(CCC(=O)NC1CC2(C1)CC2C(=O)NCC(C)(C)OC)OC 51552,N1(C(c2c(NC)scn2)=O)CCC2CCC(C1)N2C(=O)CC1CCCSC1 51553,C1(CNC(CC)=O)CCC2(CCN(C(c3ccccc3COC)=O)CC2)O1 51554,CON1CC(C(=O)NCC2(O)CCN(C(=O)Cc3ccn(C)n3)C2)CC1=O 51555,C12(CNC(COCCN(C)C)=O)CCCN(C(=O)COc3ccsc3Cl)C1C2 51556,c1(C(=O)NC2C(CNC(COc3ccc(OC)cc3)=O)CC2)cnc(Cl)c(N)c1 51557,C1(NC(C)=O)CN(C(=O)CCc2cc(Cl)cc(Cl)c2)CC12CC2 51558,c1(-n2cc(C3N(C(Cc4cc(C)ns4)=O)CCC3C)nn2)nn(C)cc1Cl 51559,c1(NC(CC2OCCN(C(c3n[nH]c(CC)c3F)=O)C2)=O)ncc(C)cc1Br 51560,CCCCCC(O)C(C)C(=O)N1CCCC(CCNC(c2ccoc2Cl)=O)C1 51561,c1(C(N2CC(NC(C=CC(C)C)=O)C(O)CC2)=O)cc2c(Cl)c(Cl)ccc2[nH]1 51562,C(=O)(C1CCc2c[nH]nc21)NCCC(CC)CC(=O)N1CC(=O)NCC1(C)C 51563,n1(CC(C)CO)nc(-c2ccccc2)nc1CC1CC1(C)C 51564,c1(C(N2C(C(=O)NCC(Cl)=CCl)CC=CC2)=O)cc(F)cc(O)c1 51565,Cc1cnn(CCC(=O)NCC(O)CNC(c2csc(Cl)c2)=O)c1 51566,C12(C(=O)NC(C(C)NC(c3cncn3C)=O)C)CC(CCO1)C2 51567,C1(CNC(C(c2cnn(C)c2)C)=O)COC(C)(C)CN1C(c1ccoc1C)=O 51568,c1(OC)cccc(CCC(=O)NCC(C)NC(=O)C(C)C(F)(F)F)c1F 51569,C12(C(N3CC(C)C(NC(C4(F)CCCC4)=O)C3)=O)CC3CC(CC(C3)C1)C2 51570,c1(C(=O)NCC(CNC(CC(CC)OC)=O)CO)ccc2c(c1)nc(O)n2C 51571,c1(CCNC(=O)C(N2CC3CC(C(=O)NCC4CC4)C2C3)=O)c(Cl)cccc1Cl 51572,Cc1cc(CNC(=O)CC(C)NC(c2cc(C)ns2)=O)cc(C#N)c1 51573,c1(C(CNC(=O)C=CCOCCO)NC(C(C)=C(CC)C)=O)ccccc1 51574,N1(C(C2(C)CCCCO2)=O)CCC2(CC1)CC2C(=O)NC1(CF)CC1 51575,C=C=CC(C)C(=O)NCC(C)(C)C(=O)N(CCC(C)(C)C)C 51576,c1(-n2c(-c3ncn(C(C)C)n3)nc(CCC(C)C)n2)cccc([N+](=O)[O-])c1 51577,CC(CCCNC(=O)CCc1cnoc1)NC(=O)CSc1nncs1 51578,C1(NC(C2C(CC)C2)=O)CC2CC(NC(c3cc(Cn4cccn4)on3)=O)CC12.C 51579,c1(CC(=O)NC23CC2CN(C(c2ccoc2)=O)C3)nnc(O)nc1O 51580,Cc1ccc(O)cc1C(N1CCC(NC(=O)C=C2CCC(C)C2)C(F)C1)=O 51581,C#CC1(C(=O)OC)CCN(C(=O)C(C(=O)NC2CN(C(C)C)C2)OCC)C1 51582,c1(C(=O)NCC(C2CCCN(C(C(C)C)=O)C2)(C)O)cc2cccn2c(O)n1 51583,N1(C(c2ccc(C)cc2CO)=O)CCC2C(CCCN2C(=O)Cc2cccs2)C1 51584,CC(C)(C)C(O)C(=O)NC1CCN(C(c2cc(F)cs2)=O)C1c1ccccc1 51585,c1(C(=O)OC)c(C)[nH]c2ccc(NC(=O)NCC3CS(=O)(=O)C3O)cc12 51586,CCC(CC(=O)N(CC(C)NC(C1CC2(CCC2OC)C1)=O)CC)CC(C)C 51587,N1(C(C2(C(N(C)C)=O)CC2)=O)CC(NC(c2ccn(C(F)(F)F)n2)=O)CC(F)C1 51588,Cc1cnccc1-c1cn(CCO)nn1.C1(CC(N2CCCC2)=O)CC2CCC1O2 51589,C#Cc1cccc(NC(C2C(NC(=O)CCSCCCC)CCOC2)=O)c1 51590,c1(C(=O)NC2C(CC)CN(C(=O)C(C)(C)CNC(C)=O)C2)csc2nccn12 51591,C(C1=CCN(C(c2cc(CCCO)on2)=O)CC1)NC(=O)C(F)=CC1CC1 51592,C1(CC=C)(C(=O)OC)CCCN1C(c1cccnc1)=O.C1(CCO)CN1C1CC1 51593,C1(NC(c2cc(C)nc(C)c2)=O)CN(C(c2cnn(C)c2)=O)CC(C)(C)C1 51594,C(C(C)(C(=O)N1CCC(CC2CC2)CC1)NC(=O)CCC1CCC(=O)C1)SC 51595,c1(C(=O)NCCCCCO)nc2ccc(Br)cn2c1F 51596,C(CC(C)C)(C(=O)NCCC(=O)NCC1CCC(C)(C)C1)NC(C)=O 51597,C1(CCOC)CN(C(C2(C)C=CCC2)=O)CCN1C(c1cc(C)[nH]n1)=O 51598,C12(C(N(CCC)CC3CC3)=O)CC(CN(C(=O)CCc3nc(C)no3)C1)C2 51599,N1(C(C2C(CNC(C3CC4(CCC4)C3)=O)CCO2)=O)CCC(=C(F)F)CC1 51600,C=CCCC(C(=O)NCc1cn(C)nc1OC)NC(=O)Cc1ccccc1F 51601,Nc1cc(C(N2CC3CC2C3NC(=O)CCc2cscn2)=O)c(Cl)c(F)c1F 51602,Cc1ncnc(N2CC(c3ccccc3)(NC(=O)CC3CCC(=O)N3)C2)c1Br 51603,c1(CC(=O)NC(CC)(C)CNC(=O)COCP(C)(C)=O)ccc(Br)cc1 51604,N(C(=NCC(C)C)N1CCC(Nc2ccccn2)C1)C(CC)C 51605,c1(C(=O)NCC(CC)NC(C2(C)CCNC2=O)=O)c(C)nc2ccccc2c1C 51606,c1(OC)cncc(C(=O)NCCCCCCNC(=O)C(C2CCCCCC2)C)n1 51607,C1(=O)CC(C)CO1.C1(c2c(OC)c[nH]n2)CCCN(C(=O)NCCC(C)C)C1 51608,N1(CC(=O)NC2C(CC)CN(C(=O)C(C)(C3CC3)OC)C2)CCC(=O)NC1=O 51609,N1(C(c2cc(C)ncn2)=O)CCCC(N(C(=O)Cc2c(F)cccc2Cl)C)CC1 51610,C(C(C(C)(C)C)NC(=O)Cc1ccccc1O)NC(C(C)n1cncn1)=O 51611,C1(C(=O)NCC)(CC2C(NC(COCCCCOCC)=O)C2)CCOCC1 51612,n1(CC(N2CCC(CC=C)(NC(=O)C(CC)OCC)C2)=O)c(C)c(C)sc1=O 51613,C1(CNC(CNC(=O)OC)=O)CCCN(C(C2CCC(C)(C)C2)=O)C1 51614,C12(CNC(c3cc(C)sn3)=O)CC3CC(CC(C3)C1NC(C1CC13CC3)=O)C2 51615,CC(CN=c1[nH]c(N2CCOCC2)nc2cccnc12)(C1CCCC1)OC(F)F 51616,CCC(CC)C(=O)NCC(C)NC(c1nnn(C)c1C(F)(F)F)=O 51617,C1(CNCCCC(=O)OC(C)(C)C)C2(CC2)C12CC2 51618,C(=O)(C(C)N(CC(C)N(C(=O)C(C)C1CC1)CC)C)NCC#C 51619,n1(CC)nc(C)cc1C(=O)NC(C)C(C)(C)NC(C1CNC(=O)N1)=O 51620,C1(NC(c2c(C)ncn2C)=O)CCN(c2ncccn2)CC1C 51621,N(C1CCCn2nc(C)nc21)C(N(C(C)(C)C1CCC1)CC=C)=O 51622,c1(C(=O)NC(CN(C(C(C)OCC)=O)CC)C)cc(Cl)c(Br)cc1C 51623,C(=O)(CC1=CCOCC1)NC1C(CN(C(=O)CCCF)C)CC(C)(C)CC1 51624,N1(C(C(CC(C)=O)(C)C)=O)CCC2(CCCN2C2CCNC2=O)C1 51625,N1(C(c2[nH]cc(C)c2)=O)CCCC2CCN(C(c3n[nH]c4c3CCCC4)=O)CC12 51626,N1(C(=O)Cc2ccccc2)CC2CC(C1)N2C(=O)C(F)C1CCOC1 51627,C(C(C)(C)CC(=O)NC1CCOCC1NC(=O)CSCC(F)(F)F)OC 51628,C(C(C(=O)Nc1cnn(CCF)c1)C(C)(C)C)NC(c1c(C)n[nH]c1C)=O 51629,c1(CC)ncc(Br)cc1C(=O)NCCCCN(C(=O)CCC(C)CN(C)C)C 51630,N1(C(C(N2CCNC2=O)C)=O)CC2CN(C(C3C(C)(C)C3(C)C)=O)CC2C1 51631,c1(C(N2C(C(=O)NC(CC)C)CCCC2)=O)cc(C)cc(F)c1 51632,Cc1nc(CNC(=O)C=CC(C)NC(C2C=CCC2)=O)[nH]c1C 51633,CC1(C)CCC(CNC(=O)CC2CC(N(C)C)C2)(NC(c2ccccn2)=O)C1 51634,N1(C(C(C)(C)C2CCCCO2)=O)CCC12CN(C(=O)CCSc1ccccn1)C2 51635,C1(c2nc(CC(=O)N(CC(=O)NCC)CC)on2)CCC(C2CC2)C1 51636,C1(C(=O)NCC2(F)CN(C(C3(CC=C)CCCC3)=O)C2)COC2CCCCC12 51637,N1(c2nncc(C)c2)CCCC(O)(C2CC2)C1 51638,c1(C(=O)NC(C)C(F)NC(=O)CN2CCSCC2)ccc(CSC2CCC2)cc1 51639,N1(C(C2N(C(=O)CCCC3CCCO3)CC=CC2)=O)CCCC(O)(CO)C1 51640,c1(OC)c(C)csc1C(=O)NC1CN(C(=O)Cc2cn[nH]c2)CC1C 51641,CC1CCCc2ncc(C(=O)NC3CC34CCN(C(=O)Cc3cnoc3)CC4)n21 51642,C1(CC)(NC(c2ccnn2C)=O)CCCN(C(C2CCCN(CC(C)C)C2)=O)C1 51643,C12(CNC(C3(C#C)CCC3)=O)CCC(CC1)N(C(c1coc(C)c1)=O)C2 51644,c1(C(c2n(CCC)nnn2)NCc2conc2COC)ccccc1OC1CC1 51645,C1(C(N(CCOCC)CC)=O)CC(NC(c2cnn(C(C)C)c2)=O)CCO1 51646,S(=O)(=O)(c1ccc2c(=O)n(C)c(=O)n(C)c2c1)NCC(CCSC)N 51647,c1(C(=O)NC2CN(C(C(c3ccccc3)OC)=O)CC2C)nccc2cc[nH]c12 51648,C1(CC(=O)NCCc2ccccc2O)CN(C(c2cccnc2)=O)CC12CC2 51649,c1(CN(C(=O)C(N2CCCC2c2ccsc2)=O)C)cccc(Br)c1 51650,N1(C(CC2(COC)CCCC2)=O)CC2CCN(C(=O)Cc3csc(C)n3)CC12 51651,Cc1ccc(C(F)(F)C(=O)NC(C2CCCN2C(c2cc(C)c(C)o2)=O)C)cc1 51652,N1(C(C(CCCC)(C)F)=O)CCN(C(C2CCc3nccn3C2)=O)CC2(CC2)C1 51653,CCC(CCC(=O)NCC(O)CNC(=O)C#CC(C)(C)C)S(N)(=O)=O 51654,C1(NC(c2ncn(CC)c2)=O)CCC(N(C(=O)COc2cn[nH]c2)C)CC1 51655,C1(C(=O)NCCN(C(=O)C(F)C2CCOC2)CCOC)CCC=CCCC1 51656,Cc1cccc(C(=O)NC(CNC(=O)CN2CCOCC2=O)C(C)C)c1F 51657,c1(NC(CC2OCCN(C(C3C(C(=O)OCC)CC3)=O)C2)=O)ccc(C)nc1C 51658,c1(-c2ccc(C)o2)cc(C(=O)N=c2[nH]c(Cl)ncc2C)c2[nH]ccc2c1 51659,Cc1csc(C=CC(=O)NCCC(C)NC(C2(C)CC3CC3C2)=O)n1 51660,CC(CCCCNC(C1(C)CCC(=O)C1)=O)NC(=O)C=CC1CCOCC1 51661,N1(C(CC(C=C)C)=O)CC2CC(C1)CN(C(=O)CNC(=O)CC1CCCC1)C2 51662,N1(C(C(C=C=C)C)=O)CCC(CC(=O)NC(C2CCCC2)CC)C1(C)C 51663,CCC(C)C(O)C(C)C(=O)NCC1CC(C(=O)NCC2CCCC(C)(C)C2)C1 51664,CN1CCC(NC(=O)CC2COCCN2C(c2ccoc2)=O)C(C#N)C1 51665,N1(C(CCNC(CC(C)C)=O)=O)CC(NC(=O)CCc2cnc(O)[nH]2)C(O)C1 51666,C1(NC(C(NOC)=O)=O)CN(C(c2ccc(=N)[nH]n2)=O)C2(CCOCC2)C1 51667,c1(OCc2cnc(SC)n2-c2ccc(Cl)cc2)ccsc1[N+](=O)[O-] 51668,c1(C(N2CC(CNC(C3CCC34CCC4)=O)C2)=O)cccc(C#CCO)c1 51669,c1(C(=O)NCC2C(C)CCN(C(=O)COc3ccsc3)C2)cc2ccccn2n1 51670,C1(NC(c2[nH]ccc(=N)n2)=O)CCN(C(C2OC3CCC2CC3)=O)CC(O)C1 51671,C1(CNC(C=CSC)=O)CCN(C(=O)C(c2ccccn2)C)CC1(F)F 51672,c1(C(=O)NCCNC(C=CC(C)(C)SC)=O)nccnc1O 51673,CC1CC(C(N2CCN(CCCNc3ncccn3)CC2)=O)CC(=O)N1 51674,N1(C(CC(C)(C)N(C)C)=O)CCC2CCCC12C(N1CC2C=CC1CC2)=O 51675,C1(NC(=O)CC2CC=CCC2)CCC2(CC1)CCN(c1nc3ccccc3o1)C2 51676,c1(C(N2CCOCC(CNC(COCC=C)=O)C2)=O)ncc2ccccn12 51677,CC1(C(=O)OCCOc2ccns2)CCC(F)(F)CC1 51678,CC(C)C(N=c1[nH]nc(CC(F)(F)F)o1)C(C)NC(C1CC(C)(C)CO1)=O 51679,C1(C(=O)NC2OCCN(C)C(=O)C2)CC2(CO1)CN(C(=O)C(F)(F)C(F)(F)F)C2 51680,N1(C(C=Cc2ccc(C)s2)=O)CCCCCC1C(=O)NC1(C(O)C(F)(F)F)CC1 51681,CCCC(O)CC(=O)N(CCNC(=O)C(F)C(C)(F)F)CCOC 51682,C=CCN=c1ccc(=NCc2cnc(C)cn2)[nH][nH]1 51683,N1(C(CC2N(C(C)C)CCC2)=O)CC(C(=O)Nc2cc(C(F)F)ncn2)CC1(C)C 51684,C1(CC(=O)NCC2(C)CCCC2O)(NC(=O)OC(C)(C)C)CCCCC1 51685,CCC(CNC(c1cc(C#N)oc1C)=O)(CC)C(=O)NC(C12CCC(CO1)C2)C 51686,CCCCS(=O)(=O)CC(=O)N1CC(NC(=O)C(C)SC(C)C)C2(CCC2)C1 51687,Cc1ccc(C)c(C(=O)NC2CCCC2(C)CNC(=O)CC2CCCO2)n1 51688,C(=O)(C1=CS(=O)(=O)CCC1)NC1C(NC(CNC(CNC(CCC)=O)=O)=O)CC1 51689,N1(C(c2ccc(C)cc2C)=O)CC(NC(=O)CCOC(C)C)C2(CCC2)C1 51690,C12CCN(C(=O)CN(C3CCC3)C1=O)O2.c1(CC)cccc(C#N)c1 51691,C(C(=O)NC1CCC1CNC(=O)CC1(C#N)CCCCC1)(C(C)(C)C)N(C)C 51692,N1(C(C(C)=C(C)C)=O)CCC(C(=O)NCc2ncsn2)=C(F)C1 51693,c1(C(N(C2CCN(C(=O)CC3(OC)CC3)CC2)CCOC)=O)cnc(C)nc1 51694,C(C(C)(C1CCC1)NC(=O)CN(S(C)(=O)=O)C)NC(COC(CC)C)=O 51695,c1(SC)csc(C(C(=O)NC2(c3ccsc3)CC2)NC(C2CCC2)=O)c1 51696,Cc1cc(C)n(CCC(N2CC3CC2C3NC(c2ccc(C(F)F)cn2)=O)=O)n1 51697,C12(CC(N3CC(C(C)OC)C3)=O)CCC1CN(C(C1(C(C)(C)O)CCC1)=O)C2 51698,C1(NC(c2c(C)ccs2)=O)CC(F)(F)CC1NC(=O)COc1ccccc1 51699,Cc1cc(NC(=O)C(=O)NCc2ccccc2Cl)ccc1-c1ccncc1.C(C)(C)N 51700,C#CC1CC2CCC1N(C(=O)C(Cc1ccoc1)NC(c1cnn(CC)c1)=O)C2 51701,Cc1nsc(CNC(c2nnnn2CC(=O)NC)(C)CC2C=CCC2)n1 51702,C1(CC)(CO)CCCN(C(=O)C(=O)NCCOc2ccccc2)C1.C(CF)O 51703,c1(CN(C)CC)nc(C)c(C(=O)NC(C)CCNC(C2CC(O)C2)=O)s1 51704,C(C1COc2ccccc21)NC(NC(c1cccs1)C)=NCCF 51705,C(=O)(CC(=O)N=c1ccn(-c2nccc(S(C)(=O)=O)n2)[nH]1)NC1(C#C)CCCCC1 51706,c1(OC)ccc2c(c1)CC(C(=O)NC1CCCC13CCC3)O2 51707,CCCC(C)(O)C(=O)N1CCCC(NC(c2ccc(C(F)(F)F)c(F)c2)=O)C1 51708,C1(C(=O)NC2CC(CNC(c3cc(C4CCC4)no3)=O)C2)CC2(C1)OCCO2 51709,C12(C(N(CCNC(c3nn(CC)nc3C)=O)C)=O)CCC(C(F)F)(CC1)C2 51710,c1(C(=O)NCCC2(OC)CN(C(C3CC3F)=O)C2)c(O)cc(=O)n2c1CCCC2 51711,N1(C(C(C)NC(C)=O)=O)CCC(CC(=O)NCCF)C(C)C1 51712,c1(OC)cnc(Cl)[nH]c1=NC1CC2CCC1N(C(=O)C1CC1)C2.c1cc[n+]([O-])cc1 51713,c1(C(N2CC(C=C)(CC(=O)NC3(C)CCCC3O)C2)=O)nccc(C)c1F 51714,CC1COc2c(C(=O)NCCn3cc(CO)nn3)cnn2C1 51715,C1(CNC(c2cnc(CC(C)(C)C)s2)=O)CN(C(C2CSCCS2)=O)CC1O 51716,c1(C(=O)NCC2(CCNC(=O)CC3CC3)CC2)cccc(C(F)(F)F)n1 51717,C(=O)(CCCCCC(C)C)NC1CN(C(c2c(C)ccc(Cl)c2)=O)CC1C 51718,c1(CNC(=O)NC2(C(F)F)CCC2)ccc2c(c1)OCCO2 51719,C1(CC(=O)NC2(CC(=O)NCCc3n(CC)cnn3)CCC2)CCC(C)CO1 51720,N1(C(c2cccc(O)c2CO)=O)CCC(F)(F)C(NCc2ccccc2F)C1 51721,N1(C(C=NOC)=O)CCC(N(C(C2CC2OC(C)(C)C)=O)CC2CC2)CC1 51722,CCC(C(=O)N1CCCC(O)(CNC(c2cnccn2)=O)C1)C(C)(C)CC 51723,CC1(C=CC(=O)NCC2(C(=O)NCCC3CCCC3)CCC2)COC1 51724,S(=O)(=O)(c1cc(Br)cs1)N1C(CCC#N)CC(F)C1 51725,C(=O)(CCC1=NNC(=O)CC1)NCC1CC(NC(c2c[nH]cc(C)c2=O)=O)C(O)C1 51726,C(=O)(C(F)(CNC(c1ccccc1C1CC1)=O)C(C)C)N(CC=C)CC 51727,C1(CNC(C(CC)c2ccccc2)=O)CCC2(CN(C(=O)CC3CS(=O)(=O)C3)C2)O1 51728,c1(-n2c(SCCN(C)C)nc(-c3cncc(Br)c3)n2)ccc(Cl)c(Cl)c1 51729,CCC(CC)C(C(=O)NC1(C(=O)NCCn2ccnc2)CSC1)OC 51730,C(N=c1[nH]cnc(Cl)c1F)C1CN(C(c2ccn(CCC)n2)=O)CC1C 51731,c1(CC)nc2c(C(=O)NCC(C)(CO)NC(=O)C(C)C3CC3)ccnc2[nH]1 51732,CC1(C)CC(Cc2ccccc2)CN(CC2CC(F)CN2)C1 51733,Cc1nnc2c(C(N3CCCOC(CNC(=O)C(C)(C)C#N)C3)=O)cccn12 51734,C1(C(C(=O)NC(c2cccnc2)C(=O)N(C2(CC)CC2)C)C)CCOCC1 51735,c1(OCC)cncc(C(=O)NCCCC(C)(C)NC(c2cccn2C)=O)c1 51736,c1(OC)cc(Cl)c(Br)cc1C(=O)NOC1CCOC1 51737,CN1CCN(C(=O)CCCc2cccnc2)C(CNC(c2nccnc2Cl)=O)C1 51738,N1(C(=O)Cc2cnoc2)CCC2(C(=O)NCC3(C(=O)O)CC3)CCCC12 51739,C(c1ccnn1C)=CC(=O)NC(C(=O)NC(c1n(CC)ncc1)C)c1ccoc1 51740,c1(CC)ccc(CNC(C2(C3CCCN3C(=O)Cc3ncc(C)o3)CC2)=O)o1 51741,CCCC(C(=O)NCC(CNC(=O)Cn1cnccc1=O)OC)c1ccccc1 51742,C1(C(=O)NCC(CSC)OC)CCC(O)CN1C(=O)Cc1nocc1C 51743,N1(C(C2N(CC)CC2)=O)CC2CC(C(=O)NCc3cc(C)sc3C)(C2)C1 51744,C1(NC(c2cc(OC)n(C)n2)=O)CN(C(=O)CC2CCC=CCC2)CCC1CO 51745,CC1CCN(C(c2ccccc2C2CC2)=O)CC1NC(c1ccc(Br)o1)=O 51746,c1(CN(C(C)C)C(=O)Nc2cncc(Cl)c2)nc2c(s1)CCCC2 51747,c1(COC)ccc(C(N2CC(NC(=O)CC3COC(=O)C3)CC2C)=O)cc1 51748,c1(NC(N2CCSC2c2cccnc2)=O)cccnc1NC1CCCC1 51749,CC(CCCCNC(=O)COC1CCOC1)NC(=O)CCNC(c1cccs1)=O 51750,C12(C(=O)NCC(C)OC(F)F)CCCC1N(C(=O)Cn1cncn1)CC2 51751,n1(CC2CCCN(C(C)(C)C)CC2)cc(C#N)c(O)nc1=O 51752,C(=O)(C(C)(C)C(c1cccnn1)NC(C1(OC)CCCCC1)C1CCC1)OC 51753,Cc1c(C(=O)NC2CC(N(C(=O)Cn3cnnc3)C)C2)sc2ccc(F)cc12 51754,C(=O)(C(C)(C)C(=O)NCC(O)CNC(=O)CCn1cc[nH]c(=O)c1=O)NC 51755,C1(CC=C)(NC(=O)Cc2c[nH]ccc2=O)CCN(C(C2CC2(C)C)=O)C1 51756,C1(F)(C(=O)NCCC2CN(C(C3N(CC)C(=O)CC3)=O)CC2C)CC2(CCC2)C1 51757,c1(C(=O)NC2CCN(C(CN3CCP(C)(=O)CC3)=O)C2)ccc2nsnc2c1 51758,c1(C(N2CC3C(NC(C(C)S(N)(=O)=O)=O)(C3)C2)=O)cccc2cc(O)ccc12 51759,N1(C(CCCCCCC)=O)CCN(C(=O)C(F)CC2CCCCC2)CC1C1CC1 51760,CC1(C)CCC=C1C(=O)NCCn1ccc(=O)n(CC(=O)NC2CNC2)c1=O 51761,C(=O)(CCCCCCCCCO)NCC1C(C)(C)CN(C(C2C=CCCC2)=O)C1 51762,Cc1nc(NCc2ccc3c(c2)CCOC3)cc(=NCC2(C)CCOC2)[nH]1 51763,c1(C)ccc2c(c1)OCCO2.C1(CC=CC)C2CN(C(=O)C3ONS3)CC12 51764,C1(O)(CNC(C(CCOC)OC)=O)CCCN(C(c2cn(C)nc2C)=O)CC1 51765,c1(CC(=O)NC2C(CNC(=O)CCCCC3CC3)CCC2)c[nH]c2ncccc12 51766,c1(C(=O)NCC2(CNC(CC(COC)(C)C)=O)CC2)cc(OC)c(OC)cc1N 51767,N1(C(c2cc(C)cc(OCC)c2N)=O)CC2CC(C1)CN(C(C1CC13CCC3)=O)C2 51768,CCCCCC(O)C(=O)N1CCCC1Cn1cc(CNC(C2(F)CC2)=O)nn1 51769,N1(C(C(C=C)O)=O)CCOC2(CCN(c3ccc(F)cc3[N+](=O)[O-])CC2)C1 51770,c1(C(=O)NCCN(C(C2CC2CF)=O)OCCCCCC)cn(C(C)C)nc1C 51771,N1(C(CC(C)F)=O)CCN(C2CCC(NC(C3(C)CC(=C(F)F)C3)=O)CC2)CC1 51772,CCC(O)CC(=O)NCC1CCC(NC(=O)CC2CSC2)CC1 51773,CCCC(CCCNC(c1ccc(=O)n(C)c1)=O)NC(c1sc(C)cc1C)=O 51774,c1(C(N(CC(C)NC(c2cc(CC)[nH]n2)=O)C)=O)ccc2cnsc2c1 51775,N1(CCOC)CCN(C(c2cccc(CNC(=O)C(C)N=[N+]=[N-])c2)=O)CC1 51776,c1(C(N2CC3C(CNC(C4CC=C(C)CC4)=O)(C3)C2)=O)cc2cn[nH]c2cn1 51777,C(=O)(C1=NN(C)C(=O)CC1)N(CC)CC1CC(NCCCC(=O)OC2CCOCC2)C1 51778,CC(C)(CO)C(=O)NC(C1CCN(C(C2CCCCS2)=O)CC1)CO 51779,N1(C(C(C=C)O)=O)CC(N(C)C(c2oncc2CC)=O)C(CC)C1 51780,C1(CN2CC(n3cc(C(=O)CCn4c(C)cc(C)n4)nn3)C2)CCn2ncnc2C1 51781,C1(COC)(CNC(=O)C(C)n2cccn2)CCCN1C(C1CC=CC1)=O 51782,N1(C(CC(=O)OC)=O)CC(C2(NC(=O)Cn3ccc(O)nc3=O)CC2)C1 51783,CC1CCOCC1C(=O)NCc1cccc(C(=O)NC2(CO)CCC2C)n1 51784,C=CC1(C(=O)NC2CCN(C(C3CCCN3C)=O)C2C(C)C)CCOCC1 51785,C1(C(N2CC(CNC(C)=O)CCC(C)(F)C2)=O)(COC)CCCNS1(=O)=O 51786,C1(C2(O)CCC2)(C(=O)NC2C(CNC(c3cnc(C(C)(C)C)[nH]3)=O)C2)CC1 51787,n1(CCCN(C)Cc2ncc(C(F)F)s2)cc(CN2CCCC2)nn1 51788,C1(CC)CC(O)CN1C(C1C=CCN(C(=O)C(COC(C)(C)C)N(C)C)C1)=O 51789,C1(C(N2CC(NC(C=C(C)C(F)F)=O)C3(C2)CC3)=O)CCOCC12CCCCC2 51790,N1(C(Cc2cc(C(C)C)no2)=O)CCC(CO)C(NC(=O)COCCF)C1 51791,C(=O)(C1CCCc2ncnn21)N1CCN(C(c2[nH]nnc2C2CC2)=O)CC(C)C1 51792,N1(C(CN(CCCCCC)C)=O)CCC(CNC(=O)CCC2CC2(Cl)Cl)C12CC2 51793,c1(OC)ncc(CNC(=O)C(C2CCC(=O)N2)C)s1 51794,Cc1cc(C2(C(=O)NC34CCCN(C(=O)CC#N)C3C4)CC2)ccc1Br 51795,c1(CC(=O)NCC=CCNC(c2c(C)nc(CC)s2)=O)ccc2c(c1)OCO2 51796,N1(C(C(C2CCC2)OCC)C(=O)NCc2n[nH]c(C)n2)CCC(O)(CC)CC1 51797,c1(C(N2CC3(C(C(N4C(C(C)=O)CCCC4)=O)C3)C2)=O)ccc2ccn(C)c2c1 51798,N1(C(C(C=C)(C)O)=O)CC(C(=O)NOCCN(C)C)C2(CC2)C1 51799,c1(C(=O)NC2CCC(NC(=O)C(F)=CC3CC3)CC2)cc2c(cn1)OCCC2 51800,N1(C(c2cnc(N)[nH]c2=N)=O)CCCC2(CCCCC2NC(=O)C(O)C2CC2)C1 51801,C1(NC(=O)CN2C(=O)CCC2=O)CC2CC(C1)N(C(=O)Cn1cncn1)C2 51802,C(C(O)CCNC(=O)Cn1nccn1)NC(=O)C=CCOC1CC1.C1CC1 51803,c1(C(=O)NC(CNC(C(c2ccc(CC)cc2)C)=O)C2CC2)cc(C)cc(N)c1 51804,N1(C(C(C(CC)CC)C)=O)CCC(NC(C2CC3CC3C2)=O)C2(CCC2)C1 51805,CC1CN(C(C2(C)CCCOC2)=O)CCC1CNC(c1ccc(F)cc1F)=O 51806,C12CN(CCC1(C)C)C2=O.C1(CNC(C(C)NC(N)=O)=O)CC(F)(F)C1 51807,N1(C(C2CC(C#N)(OC)C2)=O)CC(NC(c2ccc(OC)s2)=O)C2(CCC2)C1 51808,C=C(C)C(O)CC(=O)N1CC(OC)CC1CNC(=O)C#CC(C)C 51809,CN1CCCC1(C)C(=O)NCC(C(C)(C)C)NC(=O)Cc1ccncc1Cl 51810,Cc1ncc(C(N2CCC(C(F)F)(CNC(=O)C(C)OCCC(C)C)C2)=O)n1C 51811,Cc1cc(Cl)ncc1CNC1CCC(NC(=O)NC23CCCNC2C3)CC1 51812,CC1CCCC1.C1(CNC(=O)C(=O)N)CCSCC1.C12(CC1)CC(=O)C2=O 51813,C(C(CC(C)C)NC(=O)C(C)(C)NC(C)(C)C)OCCCOC(C)=O 51814,c1(-n2c(C(CC=C)CC)nc(-c3occc3C)n2)ccc(C)c(F)c1 51815,C=C=CCCC(=O)N1CC(CNC(C2CN(C)C(=O)N2)=O)C1 51816,c1(C(=O)NCC(C)CNC(c2nnn3c2CCC3)=O)nccc2ccncc12 51817,c1(C(N2C(CCNC(C(CC#C)O)=O)COCC2)=O)cccc(F)c1C 51818,Cc1nc(C2CC2)[nH]c(=NC2CCCN(C(c3cnn(C4CC4)c3)=O)C2)c1Br 51819,CCC(F)(F)C(=O)NCC1CC(F)(CNC(c2cnc(C)nc2)=O)C1 51820,C1(C)(CNC(C(C)NC(=O)OCC)=O)CCN(C(C2C=CCCC2)=O)C1 51821,CC(C)(C)C(C#N)C(=O)N1CC=CC(C(=O)Nc2cccc(F)c2)C1 51822,C1(CNC(c2c(COC)cco2)=O)CCn2cnnc2C1.N12CCC(C1)C2=O 51823,C(=O)(C1=NOC2COCC12)NC(C(C)C)CCN(C(=O)CCC1CC(F)(F)C1)C 51824,C1(NC(C2CCCCO2)=O)(CO)CN(C(C2(CO)CCC2)=O)C1 51825,N1(C(CCCC)=O)CCCCC(NC(c2cc(C(F)(F)F)ccn2)=O)C1 51826,c1(SC(C(N2CC(O)(CNC(C=CSC)=O)C2)=O)C)ccc(O)cc1 51827,C1(CC(=O)NC(c2c(C)nns2)C)CC2(CC2)CN1C(c1nnn(C)c1N)=O 51828,C(=O)(C(C)(O)C(C)(C)C)N1C(C)(CNC(=O)C(c2ccc(F)c(F)c2)=O)CCC1 51829,c1(N2CCC(C(C)CC(=O)N(C)Cc3ccncc3)CC2)cc(=O)n(C)cn1 51830,C1(C(=O)NC)CCN(C(=O)CN(C)C(=O)NCCOC)CC1(C)C 51831,C1(C(=O)NCC2OCCN(C(C(C=C)O)=O)C2)CC2CCC1CC2 51832,Cc1nc(NC(N2CC3CCC3(c3nnc(C)o3)C2)=O)cc(N(C)C)n1 51833,CC(C)(COc1ccccc1)C(=O)NC1CN(C(c2cccc(OCCF)n2)=O)C1 51834,c1(CC(=O)NC(C)C(C)(C)NC(=O)CCCN2CCCC2)ccc2c[nH]nc2c1 51835,c1(C(=O)NC(C#C)(C)C2CCOC2)coc(CNC(=O)CCn2cc(C)cn2)c1 51836,C1(C(=O)OC)CCOC(C)(CC)C1.N1(C(CCC)C)CC(NC(=O)NCC)CC1=O 51837,N1(C(C2(c3ccccc3C)CCC2)=O)CCC(C)(NCc2cncc(C)c2)CC1 51838,CC1CN(C(=O)CC2CC2CNC(=O)C=Cc2cccnc2)CCS1=O 51839,c1(OCCC)ccc(C(=O)NC2(CO)CCOC2)cc1OC 51840,C1(C(N(CCC(C)NC(c2cc(OC)n[nH]2)=O)C)=O)Cc2cc(OC)ccc2O1 51841,C1(C(=O)NCC(CCOC)NC(=O)Cc2ccc(N)cn2)CCc2nn[nH]c2C1 51842,c1(C(N2CC(NC(C(C)SCCCC)=O)C(C)C2)=O)sc2nccnc2c1NC 51843,C(=O)(CCC1CCOc2ccccc21)N(CC(c1cccc(O)c1)O)C 51844,C1(NC(C2CN(CC)C(=O)C2)=O)CN(C(C2CC2c2ccccc2)=O)CCC1F 51845,C(=O)(C1=C(Cl)CCCC1)NC1CN(C(Cc2cc(C)on2)=O)CC(O)C1 51846,C(CN=c1[nH]c(=NCc2ccccc2C#N)[nH]c2c1CCC2)C1CC(C)OCC1 51847,C1(C(N(C(C)C2CC2)C)=O)CCN(C(=O)C(CO)NC(N)=O)C(C)(C)C1 51848,CC1OCCCC1C(=O)NC1CCC(C(=O)NCC(O)CN(C)C)CC1 51849,C(c1ccccc1)=CC(C(=O)NCCC(=C)CNC(c1ccn(COC)n1)=O)C 51850,C(=O)(C(O)C(C)(C)C)NC1(COC)CN(C(=O)C(=O)NCc2csc(C)n2)C1 51851,Cn1cc2c(n1)CCCC2C(=O)NC1CC(F)CN(C(=O)CC(F)F)C1 51852,N(S(=O)(=O)N(C)C)CC(=O)NC(C1CCCN1C(=O)CCc1ccco1)C 51853,CC1(C)CCC=C1C(=O)N1CCCCC1CNC(c1cn2cnnc2cn1)=O 51854,C(CC(F)(F)F)NC(C1CC(N)C1)=O.C1(CC(=O)CC#C)CCOCC1 51855,Cc1cccc(CC(N2CCC(NC(C3CC4(CC4)C3)=O)C2C2CC2)=O)c1 51856,c1(N(CC(C)NC(c2csc(C(C)(C)C)n2)=O)C)c(F)cc([N+](=O)[O-])cc1F 51857,c1(N2CCN(CCCC)CC2)ncnc(NC(C2CCC(C)CC2)C)c1C 51858,c1(C2(CNC(c3n(CCCC)nnn3)(C)CCOCC)CC2)cc(C)cc(F)c1 51859,C1(NC(C=COCC)=O)CN(C(=O)CC2(C#N)CC2)C2CCCCC12 51860,c1(C(=O)NC2(CNC(C(CSC)C)=O)CCCCC2)[nH]cc2c1CCS2(=O)=O 51861,c1(CC(=O)NC2CN(C(C(C)=C3CCC3)=O)CC(C)C2)ccc(S(N)(=O)=O)cc1 51862,CC1CN(C(=O)C(C)C2(O)CCC2)CC1(C)C(=O)NC1CC2(CCCO2)C1 51863,C1(CNC(C2(CCC)CC2)=O)CN(C(c2csnc2Cl)=O)CC1C 51864,CC(CCc1ccccc1F)C(F)(F)C(=O)N1CCC2(c3nn[nH]n3)CCCC12 51865,c1(C(=O)OC)cscc1C(=O)NCC1CCN1C(=O)C(C)O 51866,c1(C(=O)NC2(CNC(CC(CC)C)=O)CCCC2)cc2c(Cl)cccc2nc1C 51867,CC1CN(C(=O)C(c2cncn2C)O)CC(C)N1C(c1ncncc1Cl)=O 51868,c1(C(N2CC3CN(Cc4ccn(CC)n4)C3C2)=O)cncc(S(C)(=O)=O)c1 51869,C1(C(=O)NCC(CNC(C2CCC(C(=O)OC)CC2)=O)(C)C)Cc2nncn2C1 51870,C1(NC(c2cccc(-n3cccn3)c2)=O)CC(F)CN(C(c2n[nH]cc2Cl)=O)C1 51871,c1(CC(N2CC(NC(c3nc(C)oc3)=O)C(C)C2)=O)c(C)[nH]c2ccnn2c1=O 51872,CCC(C)(CNC(C1(NC(=O)CC2CCCCO2)CC1)=O)OC 51873,C=CCN=C(NCc1cccc(C(N)=O)c1)NC1CCN(C(=O)OC)C1 51874,c1(C(N2CCN(C(COCCC#C)=O)C(C3CC3)C2)=O)cc(Cl)cc2c1CCC2 51875,c1(C(N2C(C)CCC(NC(CS(CC)=O)=O)C2)=O)cccc2ccc(C)nc12 51876,C(C1CN(C(=O)CC2CSC2)CC1C(=O)NC(C)(C)C)=CC 51877,C1(c2cncn2C)(C(=O)OC)CCN(C(c2cc(C(F)(F)F)cs2)=O)C1 51878,c1(C(N2CC(C3(NC(c4c(OC)scc4)=O)CC3)OCC2)=O)cc(C)ncc1C 51879,C1(CCNC(C#CC2(C)CC2)=O)CCN(C(C2(C)CCCCO2)=O)CCC1(F)F 51880,CCC(C(=O)OC)C(=O)N(CCC(=O)OC)OC.c12nc(co1)C(=O)NC2C 51881,C(C1CCN(C(c2nccn2C2CC2)=O)CC1)=CC(=O)NCc1c(C)cnn1C 51882,c1(C(c2n(C(CC)(C)C)nnn2)NCc2cnc(C)cn2)nc(C)c(C)[nH]1 51883,CN1CCN(C(C2CC(F)(CO)C2)=O)CC1CNC(C1CSCCS1)=O 51884,N#CC1CCC(CNC(=O)C(CCOCCO)NC(=O)CCF)CC1 51885,C1(CC)(NC(=O)CCc2cc[nH]n2)CCCN(C(c2cnc(Cl)cc2Cl)=O)C1 51886,c1(OC(C)C(=O)NC2CCCC2NC(=O)COC(F)(F)F)ccc(Cl)cc1 51887,N1(Cc2ccc(Br)cc2)CC2CCC1CO2.N12CCCC1CC1CCC(C1)C2=O 51888,c1(CN(C(=O)CCN2CCCC2)C2CC2)cnn2c1CN(C(C13CC(C1)C3)=O)CC2 51889,C(=O)(C(C)(C)CS(C)(=O)=O)N1CC(NC(=O)CSC2CC2)CC(C)C1 51890,N1(C(c2cc(OC)ncc2)=O)CCCC(N(C)C(c2ccc(F)c(C)c2)=O)CC1 51891,CN1CCN2C(C1)C(=O)N(C)CC1CC(C1)C2=O.c1(CC2CC2)ncnn1C 51892,N1(C(Cn2ccc(C)n2)=O)CC2(CC(NC(=O)CCCC(N)=O)CO2)C1 51893,Cc1cc(C(=O)NCC(O)CN(C(=O)Cc2c(C)noc2C)C)sc1Br 51894,C(C)(C(C)C(=O)N(C1CN(C(C)C)C1)C(C)C)NC(C1(CC#C)CCC1)=O 51895,C(CC(C(C)(C)C)NC(c1ccc(F)o1)=O)N(C)C(c1cc(F)ccc1F)=O 51896,C1(C(=O)NC2CCCOC2)(NC(C(C)c2cccs2)=O)CCCCC1 51897,C=CC1(CC(=O)NC(c2cnn(C)c2)CC)CN(C(c2cc(C)[nH]c2C)=O)C1 51898,C1(C(=O)Nc2n(COC)ncc2)(OC)CCN(C(=O)CN(C2CCCC2)C)C1 51899,N1(C(C2N(C(c3ccc(SC)o3)=O)CC(=O)NC2)=O)CCOC2CN(C)CC12 51900,O1NC(=O)CN=C2N=C(c3ncccc3N2)C(=O)N(CC)C1.C1(C)CC1 51901,CC(C)(C)C(CO)C(=O)NCC(C1CC1)NC(=O)CCCCCO 51902,c1(C(=O)NCCC2CCN(C(C3CC3F)=O)C2)csc2cccc(F)c12 51903,C1(C(=O)NCCCC(C)(C)NC(=O)CN2CC3CC3C2)CCc2nnc(O)n2C1 51904,CC(O)C(C(=O)NCC1(NC(c2csc(-c3cn[nH]c3)n2)=O)CCCCC1)N(C)C 51905,c1(C(N2CC3CN(C(C)=O)CC3C2)=O)cc2cc[nH]c(=O)c2s1 51906,C1(CNC(=O)Nc2cnc(C)o2)CCCN(Cc2ccccc2Cl)C1 51907,c1(OC)c(Cl)cc(C(=O)NCC2CCCN2C(=O)CC2CCC23CCC3)cc1Cl 51908,CC1CN(C(=O)C=CC2COC(C)(C)O2)CCN1C(c1cncs1)=O 51909,C1(CNC(C2CCC(CC)CC2)=O)CC(C)(C)CN1C(c1nc(C)oc1C)=O 51910,C1(C(N2CC(CCC)C(NC(c3cnc(S)nc3)=O)C2)=O)CN2CCCN1CC2 51911,C(N=c1cc[nH]cc1S(=O)(=O)NC1(C(N)=O)CC1)C1CCC(C)O1 51912,c1(C(N2CC(C3CN(C(c4cnn(C5CC5)c4)=O)C3)C2)=O)ccc2c[nH]nc2c1 51913,CCS(=O)(=O)CC(C)NC(c1cc(N(C)C)ccc1C)c1nnnn1CC(F)F 51914,C(=O)(C1CCc2cccnc21)N1CC2C(NC(COC)=O)C(CC2)C1 51915,c1(C(=O)NC(CC(C)NC(Cc2cc(C)ns2)=O)C)cc(C(F)(F)F)ccc1F 51916,Cc1cc(C#N)ccc1C(=O)NC1CCN(c2ccnc(C3CC3)n2)CC1(C)C 51917,c1(CC)ccc(C(=O)N(CCC(C)NC(=O)CCC2CCC(=O)NC2)C)cc1 51918,C1(NC(c2c(CC)nc(C)[nH]2)=O)CCN(C(C2CCCN2S(C)(=O)=O)=O)CC1C 51919,c1(CC)cccc(C(N2CCOCC2CCNC(c2ncccc2F)=O)=O)c1N 51920,c1(CC)ccc(OC)cc1C(=O)NCC1CN(C(c2ccnc(Cl)c2OC)=O)C1 51921,C12(NC(C3(CNC(C4CC(C)(C(C)=O)C4)=O)CCCC3)=O)CCCCC1OCC2 51922,C12(NC(c3cnn[nH]3)=O)CC(CNC(C3CC3c3cccs3)=O)(C1)C2 51923,O=S(=O)(c1ccc(Br)cc1NC1CC(CCO)C1)N1CC2CC2C2CC12 51924,C(=O)(C1=C(C)CCCC1(C)C)NCCC(CNC(c1cc(C)oc1)=O)O 51925,c1(C(=O)NCCN(C(COCC)=O)CC(C)O)sc2c(Br)csc2c1C 51926,c1(C(C)NC(COC2CCN(C(c3c(C)noc3)=O)C2)=O)ccc(C)nc1 51927,CC1CCC(C)(NC(c2cccc(CNC(C3CCC(O)CC3)=O)n2)=O)C1 51928,c1(CC(=O)NCC(C2CCC2)NC(c2cnc(OC)nc2)=O)ccc(Cl)c(F)c1 51929,C1(C(=O)NC(c2cccc(Cl)c2)CNC(C(CC)O)=O)CCC(C(=O)OC)CC1 51930,c1(C(=O)NCC(C)(C)OCC(=O)NCC2C(C)CCOC2)cnn2c1CCC2 51931,Cc1cc(C(=O)Nc2ncc(CCNC(c3cc(Cl)ncc3Cl)=O)s2)cc(C)c1Br 51932,C1(C(=O)NCc2cc(CC)no2)CCN(C(=O)C2(C)CC(N=[N+]=[N-])C2)O1 51933,N1(c2c(C(C(=O)OC)=O)cccn2)CCCC2(C1)CN(C(=O)C(C)OC)CCO2 51934,C1(c2n(C)cnn2)CCCN(C(=O)CN2CSCC2=O)C1 51935,CC1(C)CCC2CN1C2=O.c1(C(N)=O)ccncc1.N12CCC1C2=O 51936,Cc1cccc(OC(C)C(N2CCC(CNC(=O)CC34CC(C3)C4)CC2)=O)c1 51937,c1(C(C)C)cccc(C(N2CC(NC(C3CC4CCC4C3)=O)C(C)C2)=O)n1 51938,n1(C(C)C)cnc2ccc(-c3ccnc(C(N4CCOCC4)=O)c3)cc12 51939,c1(NC(=O)C(=O)NCCc2cccc(C(F)F)n2)ccc(I)c(Br)c1 51940,C1(N(C(=O)C=Cc2cnccn2)C)CCCN(C(C2CCCN2C(N)=O)=O)CC1 51941,Cc1sc(O)nc1C(=O)N(C1CCCCC1NC(c1cc(C(F)F)ncn1)=O)C 51942,C(=O)(C1=CCC(C)(C)CC1)NCCC(C)NC(=O)CCCOc1cccc(F)c1 51943,N1(C(CC2(OC)CCC2)=O)CCC2(CCC2)C(NC(C2(S(N)(=O)=O)CC2)=O)C1 51944,c1(CNC(C2C(CNC(C3CC34CCOC4)=O)CCC2)=O)cnccc1Cl 51945,Cc1ccnnc1C(N1CCCC1C(C)(C)C(=O)N(C)Cc1ncco1)=O 51946,c1(OC)nc(N2CCC2(C)C(=O)NCCN2CCCCCC2)ncc1Br 51947,N1(C(C2=CCCC2C)=O)CC(CO)C2(C1)CN(C(c1sccc1Cl)=O)C2 51948,C1(C(=O)NCC(C)NC(=O)Cc2cccc(N)c2N)CC2CCC(C1)C2 51949,c1(C(=O)NC2C(C)N(C(c3csc(C(N)=O)n3)=O)CC2)cccc(S(C)(=O)=O)c1 51950,CCC(CN=c1cccc(S(=O)(=O)NCCN(C)CC2CC2)[nH]1)OC 51951,N1(C(c2cc(C)ns2)=O)CCC(C)(CC(N2CCC(F)CC2)=O)C1 51952,n1(CC)nc(C(=O)NC2CN(C(C3(Br)CC34CCC4)=O)C2)cc1C 51953,c1(OC)nc(C(=O)NC(C2CCCCC2)CNC(=O)C(C)(C)CF)sc1C 51954,c1(CNC(CC(=O)NCC#C)=O)nnn(C)c1C(=O)NC(CO)C(C)(C)C 51955,c1(C(N2CCN(Cc3scc4c3OCCO4)C3CC23)=O)ccc(O)c([N+](=O)[O-])c1 51956,C1(CC(N2CCC(NC(CCOC)=O)C2)=O)CCCC(C)C1 51957,N1(C(=O)Cc2cnoc2)CCC2CN(C(=O)Cc3cccc(F)c3F)CCC2C1 51958,c1(SC)ccc(C(=O)N(CC(Cc2ccccc2)NC(=O)COC(C)C)C)o1 51959,N1(C(c2ccc(CSCC)cc2)=O)CCC(O)C(NC(=O)CC(C)C(F)F)C1 51960,N1(C(C2C(CC)C2)=O)CCC2(CC1)CC(NC(c1cnc(C(C)(C)C)s1)=O)CO2 51961,C12(C(N3CC(C)(NC(C4CCC4c4ccccc4)=O)C3)=O)CCCC(CCC1)C2 51962,C1(C(=O)NCC(=O)NCC=C)(CC)CCCN(C(C2CC3CCCC3C2)=O)C1 51963,C(=O)(CCCCC(N)=O)NCC(CCC)NC(C1CCC2CC2CC1)=O 51964,n1(CC)ccc(=NC(c2nc(N(C)C)no2)C2CC2C2CC2)[nH]1 51965,C1(C(=O)NCC(C)NC(=O)CC2CN3CCC2CC3)CCC2CC1C2(C)C 51966,CC1(C)COC(CC(=O)N(CCNC(=O)CC(O)CC2CC2)CC2CC2)C1 51967,c1(C(=O)OC)cccc(OCC(=O)NC2CCCC2NC(C2(C)CC2C)=O)c1 51968,CC1(C)COc2cc(NC(C3CC4(C3)CC(CO)C4)=O)ccc21 51969,N12CCOCC1C2=O.C1(COC(C)C)CCN(C(=O)C(C)SC2(CO)CC2)CC1 51970,N1(CC(=O)NC(C#C)C(=O)OC)C(=O)NC(C)(CCOC)C1=O 51971,c1(OC)ncccc1C(=O)NC1CCCCC1NC(C12CC(C(=O)OC)(C1)C2)=O 51972,N12CC(O)CC1C2=O.N12CCSCC1C2=O.C(=O)(CC(=O)N)NC1CC1.CO 51973,C1(C(=O)NC2C(C(=O)OC)C2)CCOCCN1C(=O)CN1CCOCC1 51974,Cc1cc(CCC(=O)NCC(C)NC(C2CCCC2C2CC2)=O)cc(C)n1 51975,N1(C2CCCN(CCS(CC)(=O)=O)C2)CC(=O)N(CC(C)(C)C)C1=O 51976,CCCC(O)CC(=O)NC(CO)C(C)NC(c1cc(CC)ccn1)=O 51977,N1(C(CCN(C(Cc2c(C)ccnc2)=O)C(C)C)=O)CCC2CCN(C)C2C1 51978,N1(C(C(CCCC)O)=O)CCC(CNC(c2cccc(=S)n2O)=O)C(F)(F)C1 51979,Cc1coc(C=CC(=O)NC2CN(C(=O)Cc3nn(C)cc3Br)CC2O)n1 51980,C(=O)(C(C)(C)C(=O)OCc1c(Br)nnn1C)N(C)C 51981,CCCCC(CN=c1[nH]cnc(Cl)c1[N+](=O)[O-])NC(=O)C1CCc2cccnc21 51982,C(=O)(C(C)(O)CC(C)C)N(CCCNC(c1cc(OCC)cc(=O)o1)=O)C(C)C 51983,CCCCCCC(=O)NC1CC2(CNC(C3CC4C(C3)C4(C)C)=O)CC1CO2 51984,C1(C(NOC(C=C)C)=O)CN(C(C2CC(C)(C)CN2C)=O)CCN1C 51985,C(=O)(CC(C)CC(=O)NCCN(C)CCF)N1CC(C(=O)OC)C(C)(C)CC1 51986,c1(C(N2CC(NC(C(C)Cc3ccccn3)=O)C2)=O)cnnc2ccccc12 51987,N1(C(C2CC(C#C)(O)C2)=O)CC2CC(NC(=O)C(C)OCC(C)C)CC1C2 51988,Cc1ccc(N)c(C(N2CC(N(C(=O)C(c3cnn(C)c3)C)C)C3(CC3)C2)=O)c1 51989,N1(C(C(C)OCC(C)C)=O)CCN(C(c2cccc(N)c2C(F)F)=O)CCC1C 51990,CCC(C)CC(=O)C(=O)NC(c1ccc(F)cc1)C(=O)N(CC(C)(C)CSC)C 51991,C(CC(C(=O)OC(C)(C)C)N1CCCC1(C)CC(C)(C)C)SC.C(=O)C1CC1 51992,Cc1cccc2oc(C(=O)NC3CC(O)CN(C(c4ncc[nH]c4=O)=O)C3)cc12 51993,CC1(C(=O)NC2CCCN(Cc3ccccn3)C2)CCCN(CCCl)C1 51994,c1(C(=O)NCc2occ(C(N(C)CC3C(C)OCC3)=O)n2)cc2ccccn2c1 51995,c1(C2C(=O)NCC(=O)N2)cnn(C)c1.c1(CCSCC)nncs1 51996,CN1CC2CC1CN2C1(c2csc(-c3cn(-c4ncncc4Br)nn3)c2)CC1 51997,c1(CCCC(=O)NCc2cccc(OC)c2C)ccc2c[nH]nc2c1 51998,C(=O)(C(O)CC(=O)SCCC(=O)NCC(C)(C)NC(C)(C)C)Nc1cnc[nH]1 51999,C(c1cnccn1)=CC(=O)N(C1CCCN(C(=O)C(C(C)C)CCCC)C1)CC 52000,N1(C(C2CCC(C)(CC)O2)=O)CCN(C(=O)CCCn2cncn2)C2COCC12 52001,N1(C(=O)NC(C(C)C)(C)Cc2ccccc2)CCNCCC1C 52002,N1(C(CC=CC=C)=O)CCCCC(C(=O)NC(C2(OC)CCC2)C)C1 52003,C1(NC(c2c(OC)cccn2)=O)CCN(C(C2CC(CCO)C2)=O)CC1F 52004,Cc1cc2nc(N3CCC(C)C(NC(c4ccccc4F)=O)C3)cc(=O)n2o1 52005,c1(C(C(=O)NCC(CC=C)NC(=O)CCCOC)C)ccc(CC(C)C)cc1 52006,C1(C(CC)=O)CCCC1C(=O)NCCCC(C)NC(=O)CCc1cnn[nH]1 52007,N1(C(CC2(CC)CCCC2)=O)CCC(NC(c2ccsc2CC)=O)C(F)(F)CC1 52008,Cn1c(I)cc2c(N3CC(Nc4c(F)cc(I)cc4F)C3)ncnc12 52009,N1(C(CC#N)=O)CCC2C(C1)OCCN2C(=O)Cc1nc(=O)o[nH]1 52010,C=CC1CN(C(=O)CCN(C)CC)CC1NC(C1CCN(C2CCCCC2)C1)=O 52011,c1(C(=O)NC(C(C)NC(c2cn(CC)nc2C(C)C)=O)C)coc2ccccc12 52012,c1(C(=O)NCC2C(CNC(C(CC)CC)=O)C2)cc(OC)cc2c1OCC2 52013,CC(C)(CC(F)C(=O)N1CCC(C(F)(F)F)C1)NC(c1cc(COC)[nH]n1)=O 52014,C1(C(=O)NCC2N(C(CCC)=O)CC(O)C2)COc2cc(Br)ccc2C1 52015,N1(C(c2c(OC)scc2)=O)CCC(NC(=O)CNc2ncccn2)C(CO)C1 52016,C(=O)(C(F)CCC(C)(C)C)NC(CNC(C(C)=C1CCC1)=O)C(C)C 52017,CC(C)(CNC(=O)C1CC1)CC(=O)N1CCC(C#N)C1 52018,N1(C(C2C(C)C2)=O)CCCCC(CNC(=O)CCC2CNC(=O)N2)C1 52019,C=C1CC2(C1)CC(C(=O)N(C(CNC(c1ncccc1F)=O)C1CC1)C)C2 52020,C=C=CC(C)C(=O)N(C)CC1CCN(C(c2c(C(F)(F)F)ncn2O)=O)C1 52021,C1(NC(C(CC=C)CNC(C2CCCC(O)C2)=O)=O)C2CCN(CC2)C1C 52022,C1(CNC(Cn2cc(CCCSCC)nn2)=O)CN(CC)C(=O)O1.C(N)=O 52023,N1(C(C(c2n(C)cnc2)O)=O)CC=C(C(=O)NCc2ccc(F)c(F)c2)CC1 52024,CN1CCC(C(=O)NC2CS(=O)(=O)C23CCN(C(=O)C(F)F)CC3)c2ccccc21 52025,C1(CCCNC(COCC)=O)CN(C(=O)CNC(=O)CC2CCCO2)CCO1 52026,C(=O)(CC1=NNC(=O)C1)NCCOCCCNC(C1C(C(C)C)CCC1)=O 52027,C1(ONC(c2c(C(C)C)scc2)=O)CCCN(c2ccc(C(N)=O)cc2)C1 52028,C1(c2onc(C)n2)CCCCN1C(c1cnc(C)o1)C(=O)NC1CCOC1 52029,c1(C(N2CC3C(NC(C4N(CC)CCC4)=O)C3C2)=O)cc(OC)cc2c1CCC2 52030,c1(C(=O)NC(C(C)C)CNC(c2coc(CO)c2)=O)cc(Cl)cn1C 52031,Cc1cccc(C(N2CCCC(CNc3nccnc3C#N)C2)=O)c1Cl 52032,C1(CCCNC(CCCOC(C)C)=O)CCN(C(=O)CC2CCOC2)CC1 52033,CCC(C)CC(C)NC(=O)CN(C(=O)CN(C)C)C(C)C.C12(CC1)C(=O)N2 52034,c1(OC)ccc(C)c(CN2CCC3(CC3C(=O)N(CC#N)CC#N)C2)c1 52035,N1(C(CC=C)=O)CC2CC(C)N(C(=O)CCOc3ccc(Cl)cc3)C2C1 52036,c1(OC(C)C(=O)N(CC(C)NC(C2(CN(C)C(C)C)CC2)=O)C)cccnc1 52037,c1(C(=O)NC(CCCC)CNC(=O)CSCCN2CCC(C)C2)cnc(Cl)cc1C 52038,C12(CC)CC1CN(C(c1ccc(OC(C)C)nc1)C(=O)NC(C)C(=O)OC)C2 52039,CCCCC(C)CCC(=O)NCC(C)(C)C(=O)NC(c1cnn(C)c1O)C 52040,c1(CC2CC=CC2)nc(-c2cc(Cl)c(Cl)s2)n(CC2CC2)n1 52041,c1(SC)c(C(=O)NC2CC2NC(c2cnc(OC(C)C)nc2)=O)cnn1C 52042,C1(C)(NC(C(CNC(CC(=O)NCC#C)=O)(F)C(C)C)=O)CN2CCC1CC2 52043,N1(C(C(=Cc2cn[nH]c2)C)=O)CC2CCN(C(C3CCCCO3)=O)C2C1 52044,C(=O)(CC(F)(F)C(F)F)NCC(CC(C)C)NC(C1CC(c2ccccc2)C1)=O 52045,N(C1COc2c[nH]nc21)C(CCC(CC)NC(c1cccc(F)c1N)=O)=O 52046,CCC(C)C(O)CC(=O)N(CC(C)(C)CNC(c1ccnc2cc[nH]c12)=O)C 52047,O=C(CCCCCCBr)N1CCN(CCNc2c(Br)cc(F)cc2Br)C2CC12 52048,C(CCO)(C(=O)N1CC(NC(C2CCN(C)C2=O)=O)C1)N(C)C 52049,C(CCC(C)C)(C(=O)N(CC(C)C)CCC)N1CC(C(=O)OCC)C(O)CC1 52050,N1(C(C2(CC#C)CC=CCC2)=O)CCC2(CC1)CN(C(c1nccnc1C)=O)C2 52051,CC(CCC(=O)NCC1COC(C)(C)C1)NC(=O)C(F)C1CCC1 52052,c1(CNC2C(C(=O)NC)CCCC2)cccc(C(C)(C)O)c1 52053,Cc1ncc(C#N)c(N2CC3C(C(=O)Nc4c(C)cc(O)cc4C)C3C2)n1 52054,C(CC(F)F)(C(=O)NC1CN(C)NC1=O)NC(C1CCC(=C)CC1)=O 52055,C1(C(N2CC(C(C)OC)C2)=O)CSCN1C(=O)C(C)COC(C)=O 52056,C(c1cncn1C)=CC(=O)NC1CC(CNC(CN(CC(C)(C)C)C)=O)C1 52057,Cc1ccc(C(F)(F)C(=O)NCCN(C(C2CN(C3CCOC3)C2)=O)C2CC2)nc1 52058,n1(CC(=O)NCC(CCNC(CCCCSC)=O)O)cccc(C(F)(F)F)c1=O 52059,CCC(CN(C)C)CC(=O)NC(C)(CSC(C)CC)C(=O)NCCCC 52060,C1(CC)CCN(C(=O)COC2CN(C(=O)CC3(C)CCC3)C2)CCO1 52061,C1(C(N(CCCNC(C(C2COC2)SC)=O)C2CC2)=O)CC(O)C(F)C1 52062,N1(C(CSc2ccc(OC)cc2)=O)CCN(C(c2ccccc2Br)=O)CC1C 52063,N1(C(C(=O)NC)C2CCCC2)CCCC(C)(OC(c2ccc(NC)cc2)=O)C1 52064,C1(C(N(C2CCCC(N(C(=O)C=CCF)C)C2)C)=O)CC2(CCC2=O)C1 52065,C(=O)(C#CC1CCCCO1)NC1CCCN(C(C(C)=C2CCCC2)=O)C1C 52066,Cc1[nH]c(C#N)cc1C(=O)NC(C)(CNC(=O)CC(=O)NC1CC1)Cn1cccn1 52067,c12cnn(c1)C(=O)C(=O)C2.C1(CC(=O)NCCCSCC)(N)CCC1 52068,C1(OC)CC(C(=O)N(C(CNC(C)=O)C2CC2)C)CC1OC 52069,CCC(CC)C(C)C(=O)NC(CO)C(C)NC(c1cccc(COC)c1)=O 52070,CC(C)(CCC(=O)N1CCC(=CCNC(=O)CC2CCC(=O)N2)CC1)[N+](=O)[O-] 52071,C1(C(=O)OCc2cc(C)no2)CCC2(CCC3(CC2)OCCO3)O1 52072,C=CC1(C(=O)N(C)Cc2cnc[nH]2)CCN(C(c2cc(CCO)on2)=O)C1 52073,N=c1cc(C(=O)NCC2(CNC(=O)C=Cc3cccnc3)CC23CCC3)cc[nH]1 52074,C1(CNC(c2c(CC)c[nH]c2)=O)CCCC(CNC(=O)CCC2CCCCO2)C1 52075,CC(CC(=O)c1cccc(F)c1)C(=O)Nc1ccnc(N2CCCC2)c1 52076,c1(CC)nc(C(N2CCC(C(C)NC(C3(CO)CCOC3)=O)CC2)=O)c(N)s1 52077,c1(C(=O)NC(COC)C(=O)NC2COCC2OC)cc(C)ccc1O 52078,N1(C(C=CCC)=O)CCOCC(CNC(C2CCC(=O)N(C(C)C)C2)=O)C1 52079,c1(NC)ccc(C(=O)NC2CC2CNC(c2sc(F)cc2C)=O)c(Cl)c1 52080,C1(NC(C2(NC(CNC(CCC)=O)=O)CC2(C)C)=O)CCn2ccnc2C1 52081,C1(F)(C(N2CCN(C(c3cc(Br)cnc3Br)=O)C3C2C3)=O)CCCCC1(F)F 52082,N1(C(CCC=CCC=C)=O)CC(C)CCC1CNC(=O)Cc1cnsc1 52083,C1(NC(c2ccncc2F)=O)CCCC12CN(C(c1sccc1F)=O)C2 52084,CC1CCN(C(C2(O)CC2)=O)C1CNC(c1cnn(C2CC2)c1)=O 52085,N1(C(Cc2nnc(C)o2)=O)CC2CC(C)N(C(=O)Nc3c(C)cccc3C)C2C1 52086,CC1(C(N2CCOC(CNC(=O)CSCc3ccncc3)C2)=O)CC(C#N)C1 52087,C(=O)(C(C)(C)S(C)(=O)=O)NCC1CC(NC(C(c2c(OC)ccc(F)c2)=O)=O)C1 52088,C1(C)(CCN2CC(CNC(C3C(OCC)C3C)=O)C2)NC(=O)NC1=O 52089,C(=O)(C(C)S(=O)(=O)C(C)C)NCCC1CC(NC(c2cc(F)cc(C)c2N)=O)C1 52090,c1(N2CCC(C(N(C(C)CCO)C)=O)CC2)ncccc1C#N 52091,CC(C)CC(CNC(C1OCCC1n1cccn1)=O)NC(c1cnoc1)=O 52092,N1(C(c2cc(C)sn2)=O)CC2CC(C1)CN(C(c1ccc(C(=O)CF)cc1)=O)C2 52093,c1(SC)cccnc1C(=O)NCC1C=CC(NC(=O)CCC2CC(C)C2)C1 52094,O=C(C(=O)N=c1nc[nH]n1-c1cccc(F)c1)c1cccc(Cl)c1 52095,n1(CC)nc(C)c(C(c2nnnn2C2CCCC2)Nc2cccc(CO)c2)c1Cl 52096,c1(C2C(NCC(C)CC3CCCNC3)C2)ccccc1F 52097,C1(C(=O)NC(c2nn[nH]n2)C)C(CNC(=O)C(=O)NC(C)C)C1(C)C 52098,c1(C(=O)NC(CNC(C(C=C)O)=O)(C)CO)cc(C)c2nc(C)cn2n1 52099,CC1CC(C)N(C(c2cnn(CCF)c2)=O)CCN1C(c1nccc(N)c1Cl)=O 52100,n1(CC(N2CC(CNC(C3(CC)CC3(F)F)=O)(OC)C2)=O)nnc2c1CCCC2 52101,N1(C(C2(CN(C)C)CC2)=O)CC(NC(c2csc(CO)n2)=O)C2CCCC2C1 52102,C12(C(N3CCC(CNC(CCCC=C)=O)CC3)=O)CC3CC(CC(C3)O1)C2 52103,O=C(C#CC1CCC1)NC1CC(NC(=O)C=CCN2CCCCC2)C12CCC2 52104,C1(CNC(Cc2c(C)nc[nH]2)=O)CCCCCN1C(c1cnn(CC2CC2)c1)=O 52105,c1(C(=O)NCC(C2CCOC2)NC(C(N2C(=O)CCC2=O)C)=O)ccncc1F 52106,N1(C(c2cc(OC)ncn2)=O)CC2(CCN(C(c3ccc(Cl)nc3Cl)=O)C2)C1 52107,C1(C(=O)OC)CCCC1(C)NC1CCCC1CNC(c1cnnc(Cl)c1)=O 52108,C1(C(=O)NC2CC2)CC(F)(F)C1.C1C(O)CNC(=O)N1C 52109,c1(C2N(C(=O)Nc3cc(Br)cc(Br)c3)CCOC2)cc(F)c(Cl)cc1Cl 52110,CC(C)C(C(=O)NCCCS(N)(=O)=O)NC(=O)Cn1cnnn1 52111,c1(C(N2C(CNC(c3coc(Cl)c3)=O)CC(F)(F)C2)=O)cn2c(n1)CCCC2 52112,C1(NC(=NC)NCC(CO)C2CCC2)CCS(=O)(=O)CC1 52113,c1(OC)cc(SC)ccc1C(=O)N(C1CN(C(C23CC(F)(C2)C3)=O)CC12CC2)C 52114,N1(C(CC2(C)CCC2)=O)CC2(CCC2CNC(=O)C(C)(C)C2CC2)C1 52115,CC(C(F)(C(=O)O)C(=O)O)NC(C1CC1c1ccc(C(=O)N(C)C)cc1)=O 52116,C1(C(F)(F)F)CCOCCN1CCCc1cccnc1Br 52117,c1(C(=O)OC)ncnc(Cl)c1-n1nccc1NC(=O)NCCC=CBr 52118,C(CCC(C)C(C)C)=CC(=O)N(CCNC(C(c1ccc(C)cc1)C)=O)CC1CC1 52119,c1(OC)ncc(-c2cnccc2CN(C)C)cc1C=O.N1CCC(O)C(F)C1 52120,CC(=O)C(C)CC(C)C(=O)NC(CCN(C)C)C(N1CCC2(CCC2)C1)=O 52121,N1(C(=O)CCn2ccnn2)CCCC(C2CCN(C(c3cn(CCO)nn3)=O)C2)C1 52122,C(=O)(C1=CCC(C)CC1)NCC1(F)CCC(CNC(c2cncc(C)n2)=O)CC1 52123,n1(CC)cnc2nc(=NCc3cc(Br)cs3)[nH]c(NCCC(C)OC)c12 52124,c1(OCC(N2CCN(C(C3CCN3C3CC3)=O)C(CO)C2)=O)cccc(F)c1F 52125,c1(C(N2C(CNC(CC(C)SC)=O)CCC(C)(C)C2)=O)cnc2sc(C)c(C)n12 52126,C(=O)(C(C)(C)CCC#N)NC(C1CCN(C(c2c(C)nc(O)cc2)=O)C1)(C)C 52127,c1(C(=O)NC2CC(C)CN(C(C3CC4(C3)CC4(F)F)=O)C2)cccc2nonc12 52128,c1(C(=O)NC2C(NC(c3c(CC)n[nH]c3)=O)COCC2)n[nH]c2c1CCC2 52129,S(=O)(=O)(c1ccc(N2CCN(C(C3CC3(C)C)=O)CC2)nc1)NCCCCC 52130,c1(C(N2CCC(CNCc3c(C)c(Cl)ccc3)C2)=O)cc2[nH]ccc2cc1Cl 52131,C=CC1CN(C(=O)Nc2c(C(=O)OC)nnn2C)CC1O 52132,C#CCCC(O)C(=O)NC1(CO)CCCN(C(c2c[nH]nc2CC)=O)C1 52133,C1(CC)CN(C(C2CC(C)(C)O2)=O)CCN1C(C1CN(C(N)=O)C1)=O 52134,c1(C(N2CC(NC(Cc3c(C)noc3)=O)C(C)C2)=O)cnc2sccc2c1 52135,N1(C(c2c(C)nn(C)c2C)=O)CCN(C(c2cccc3c2CCC3)=O)CC(O)C1 52136,C1(NC(Cn2c(C)cnc2)=O)CN(C(C2CC(F)C(=O)N2)=O)CC2(CCC2)C1 52137,C(=O)(CCCC(=O)N1CC(NC(=O)C(CC)NC(N)=O)C(O)C1)OCC 52138,c1(OC)ccnc(N(C(C)(C)C)CC2CCN(C(=O)Cc3cc(Cl)n(C)n3)C2)n1 52139,N1(CC(C)NC(C=COCC)=O)CCN(C(c2ccnc(C(C)(C)C)c2)=O)CC1 52140,C1(C)(C(=O)NCC(C2(O)CCN(C(CCCOC(C)=O)=O)C2)C)CCCN(C)C1 52141,N1(C(C(C)SCCCC)=O)CC=C(CCNC(=O)CCc2cncc(O)c2)CC1 52142,N1(C(C(C)OC(C)=O)=O)CC2CCCC2C1C(=O)NC1CC(C)(C)OC1=O 52143,c1(C(=O)OC)ccc(C(C)NCCc2ccnn2C(F)(F)F)o1 52144,c1(CCC(=O)NC(C)CCCNC(=O)C(C)(C)Oc2ccccc2)cnn(C)c1 52145,C1(C(=O)NCc2c(C(N(CCn3ncc(C)c3)C)=O)scc2)CC2CCCC2C1 52146,CCC(C)C(O)C(C)C(=O)N1CCOC(CN(C(=O)CCC(C)C)C)C1 52147,C(=O)(C1Cc2ccc(Cl)cc21)N1CC(CNC(c2cc(F)ccc2O)=O)OCC1 52148,c1(OC)ccc(C(C(F)(F)F)NC(=O)CNC(=O)NC2CCCC2)cc1OC 52149,N1(C(C2(C)CCN(C(C(C)C#N)=O)CC2)=O)CCCC2(CC(O)C2)C1 52150,c1(C(=O)NCC(CNC(CC=C)=O)CO)c(Cl)ccc(OC)c1F 52151,c1(C(=O)NCCC2N(C(C#CC(C)C)=O)CCCC2C)ccn2ccnc2n1 52152,Cc1ccc(C(N2CC(F)CC2CNC(=O)C(C)NC(=O)C(C)(C)C)=O)nn1 52153,C(=O)(CCCCCC(C)(C)C)NCC1(F)CC(NC(C(C(C)O)C)=O)C1 52154,C1(CNC(c2nc(C(C)=O)sc2)=O)CC(F)CN1C(C1CC(N2CCOCC2)C1)=O 52155,C1(NC(CC2(CC=C)CCCC2)=O)COCCN(C(C2CC(N=[N+]=[N-])C2)=O)C1 52156,CC1(C)CN(C(C2COCC(C)(C)O2)=O)CC(CNC(=O)C(C)(F)F)O1 52157,C#CC1CCCC(NC(C2CCOC2CNC(=O)Cc2c(C)cnn2C)=O)C1 52158,C(=O)(CC1=CCCCC1)NCC(C1CCN(C(C2(C)CC2)=O)CC1)(C)C 52159,N1(C(C2(CC)CC2)=O)CCC(O)(CN(C)C(C2CCCC(O)C2)=O)CC1 52160,N1(C(C2C(=C)CC2)=O)CCC(NC(c2cccc(-n3ccc(C)n3)c2)=O)C(F)C1 52161,C=CCC(C)(C)CC(=O)NC1CC2CC1N(C(c1coc(OCCOC)n1)=O)C2 52162,C(c1ccccn1)=C(C)C(=O)NCC1(C(C)NC(c2ccnc(C)n2)=O)CC1 52163,C1(C)(NC(C(n2c(C)ncc2)C)=O)CCN(C(C2(C(C)C)CCCO2)=O)C1 52164,C(=O)(C(C)=Cn1ccnn1)NCC1C2CN(C(c3cc(CCC)oc3C)=O)CC12 52165,C(=O)(C1CCCc2ncc(C)n21)N1CCN(C(C(CCCC=C)(C)C)=O)CC1C 52166,C1(CNC(CNC(C)=O)=O)CCN(C(c2c[nH]c(=N)nc2C)=O)C12CCC2 52167,C(=O)(CC(O)CCCCC)NC(CC#C)(C)C(=O)NCCCN1CCC(O)C1 52168,N1(C(C=CC(CC)C)=O)CCC2(CCCC2NC(=O)C(=O)NCCOC)CC1 52169,C1(C(=O)NCC(O)Cc2ccccc2)C2CCC(C2)N1C(c1cccc(F)n1)=O 52170,C(=O)(CCC(O)C(C)(C)C)N1CC(CNC(c2nc(CC)oc2)=O)C(O)C1 52171,C(=O)(C(C(C)C)OCC)NCCn1cc(C(=O)NC(CCC)CO)nn1 52172,n1(C)cc(C2(O)CN(C(=O)C)C2)nn1.n1(CC(C)C2CCC2)cc(C2CC2)cn1 52173,CC1(C)CC(NC(=O)CCc2ccc(F)cc2Cl)CN(C(=O)Cc2nc[nH]n2)C1 52174,c1(C(N(C2CCCN(C(CC(C)OC)=O)C2)C)=O)ccc(C)c2c1NCCC2 52175,Cc1nc(NCC(C2CC2)NC(=O)CC(O)C(C)C)c(C)c(O)n1 52176,C1(CNC(C2CC23CCC3)=O)CN(C(C23CC(C(F)(F)F)(CO2)C3)=O)CCCO1 52177,n1(CC)ncc(C(=O)NC2CCOC2C(=O)NC2(C)CCOC2C)c1C 52178,N1(C(CC(C)F)=O)CCN(CC(C)(C)NC(c2cc(CCO)on2)=O)CC1 52179,CCC(C)(C)C(O)C(=O)N1CC(N(C)C(c2ccc(OC)cc2C)=O)C(C)(C)C1 52180,c1(C(=O)NCC(C)NC(c2n[nH]c3c2CC3)=O)ccc(CC2CCC2)cc1 52181,C1(NC(C=CSC)=O)C(C)CCN(C(=O)CCc2cnc(C3CC3)o2)C1C 52182,CC1CCCCC1(C)C(=O)NC1CCCN(C(c2csc(O)n2)=O)C1C 52183,N1(C(CS(CC)=O)=O)CCCCC2(CCN(c3cc(C(=O)OC)ncn3)C2)C1 52184,N1(C(C(CC(=O)OC)N(C)C)=O)CC2CCC1CN2C(c1coc(N(C)C)n1)=O 52185,N1(C(c2c(CC)nco2)=O)CCCN(C(c2ccc(O)c(O)c2)=O)CC1C 52186,C1(CCCC(N2CC(O)(CCNC(CCC3(C)CC3)=O)C2)=O)CCCC(=O)N1 52187,N1(C(C=CC=CC)=O)CCCCC2(C1)CN(C(c1ccc(OCOC)cc1)=O)C2 52188,c1(C(=O)NCC(CNC(C2CC2F)=O)OC)cc2c(C#N)c(F)ccc2[nH]1 52189,C1(C)(CNC(CCC2COC(C)(C)O2)=O)CCCN(C(C2OCC3CCCC23)=O)C1 52190,C1(C(=O)NC(CC2CCN(C(c3c(C)[nH][nH]c3=N)=O)CC2)C)CCC2(CCC2)O1 52191,C(=O)(C(O)C(C)(C)C)NCCC1(O)CCN(C(c2cc(C)c(Cl)s2)=O)C1 52192,c1(NC(=O)Nc2scc(C(C)N)n2)ccc2cc(I)ccc2n1 52193,Cc1cc(C(N2CCC=CC2C(=O)NCC2(Cl)CC2(F)F)=O)ncc1N 52194,N1(C(c2c(-c3ccc(SC)cc3)cccc2)=O)CCn2[nH]c(=N)nc2C1 52195,CCCCC(CC)NC(=O)C(=O)NCCNc1nccc(C(F)(F)F)n1 52196,CN1CCCC(F)(C(N2CCC(CO)(NC(c3coc(C(F)F)c3)=O)CC2)=O)C1 52197,CCCC(C(=O)NCC(F)CNC(c1ccccc1Cl)=O)NC(N)=O 52198,Cc1ncnc(C)c1CC(=O)NC1CC2CN(C(=O)C(C)n3ccnc3)CC12 52199,C=CC(CC)CC(=O)N1CCN(C(=O)C2=CCSC2)C(CCO)C1 52200,CC1(C)NC(=O)CCC1NC(=O)COc1cccc(Cl)c1 52201,CCCC(CC)CCC(=O)NCc1cc(C(=O)NC(C)(C(=O)OC)C2CC2)n(C)n1 52202,CC1CN(C)CC(C(N2CC(NC(c3cccc(=S)n3O)=O)C(C)C2)=O)O1 52203,n1(CC(=O)NC(C)(C)CNC(=O)C(c2cccc(F)c2)O)nnc2c1CCCC2 52204,O=C(C1=NOCC1)Nc1ccccc1.C12CN(C(=O)Cc3cncnc3)CC1C2 52205,C12(C(N(CC(C)O)CCNC(=O)CC3CCCC(=O)N3)=O)CCC(C)(CO1)C2 52206,C(C1CCc2c[nH]nc21)NC(C1=NOC(CNC(C(CC)OC)=O)C1)=O 52207,c1(SC)ccccc1C(=O)NC1CN(C(=O)COc2ccsc2Cl)CC1F 52208,C1(CNC(CC(C)c2ccncc2)=O)CCC(NC(C2(C)C=CCC2)=O)CC1 52209,C1(NC(CC2C(C)OCC2)=O)CC(C(=O)NCC2CC2CCN=[N+]=[N-])C1(C)C 52210,Cn1ncc2cccc(-c3ccccc3CN3CC(S(C)(=O)=O)CC34CC4)c12 52211,N1(C(CC(C)(C)C#N)=O)C(CNC(C2(C)CCCS2)=O)CC2CCCCC12 52212,N1(CC(=O)NCCC(C)N(C(=O)C(=O)N(C)C)C)CC(=O)N(C)C1=O 52213,c1(CNC2CC(CC(=O)Nc3cnc4cnccn34)C2)c[nH]c2nccc(Cl)c12 52214,C1(CCNC(c2cn(C(C)C)nc2)=O)CCCN(C(=O)Cc2ccsc2)CC1 52215,c1(C(C(N2CCCC(NC(C(CC)(C)C)=O)C2)=O)=O)ccc2c(c1)CCCC2 52216,CCCCC(O)C(=O)NC(C1CCCC1)CNC(c1ncc(F)cn1)=O 52217,Cc1cnc2cc(C(=O)NCC3CN(C(=O)CCC4CC4(F)F)CCO3)ccn12 52218,CCC(CC1CCCC1)C(=O)NC1CCOC(CNC(=O)C=C2CCCCC2)C1 52219,N1(C(=O)NC2CCC(C)C2)CCC2(CCN2)CC1 52220,C(CCCC(=O)NCC(C)N(C(=O)Cn1nnc(-c2cccs2)n1)C)OCC 52221,N1(C(=O)NCC(C2CCCC2)(C)C)CCC(CCNC(N)=O)C1 52222,c1(C(C(=O)NCCOCC)N(CCNn2cccn2)C)ccc(S(C)(=O)=O)cc1 52223,N1(C(c2cc(CC)n(C)n2)=O)C2CCC1(CNC(C1CC=CC1)=O)CC2 52224,c1(OC)ccc(C(=O)NCC2CN(C(C3CCC3C3CC3)=O)C2)c(F)c1 52225,C1(NC(Cc2ccc(C(=O)NC)cc2)=O)CCN(C(=O)CCNC(C)=O)C(C)C1 52226,c1(NCCCOC(C)C)nccc(=NC2CC=CCC2)[nH]1 52227,C1(C(C)NC(=O)Cc2ccon2)CN(C(=O)CC2NC(=O)NC2=O)CCO1 52228,N1(C(C(N2CCC(C3(c4ccccn4)CC3)C2)=O)=O)CCCCCC1c1ncc[nH]1 52229,c1(C(CC)C)ccc(C#N)c(NCC(C)CNC(C2C=CC=CC=C2)=O)n1 52230,c1(C(N2CC(CCNC(C3C(OCC)C3)=O)OCC2)=O)cnc2c(n1)CCCC2 52231,c1(C(=O)NCC2(CNC(Cn3ccc(C)n3)=O)CC2)c(C)cc(Cl)cc1C 52232,Cc1ccccc1C(=O)NCCCCCNC(C1CCC(C(F)(F)F)C1)=O 52233,c1(C(=O)NC(CC2CC2)C(=O)NCCc2cncs2)cccc[n+]1[O-] 52234,N1(C(C)=O)CC(N(C(=O)C(C)CC(N)=O)C)C(C)(C)C1.C1CC(=O)N1 52235,c1(SC)ccc(C(=O)NC2CCC2NC(=O)CCc2cnc(C)o2)cc1[N+](=O)[O-] 52236,c1(C(N2CCC(O)(CN(C(C3(OC)CCOC3)=O)C)C2)=O)c(C)nc2sccn12 52237,c1(C(=O)NCC2OCCC2C(=O)NCCSCCO)cnc(Cl)s1 52238,c1(C(N2CC(NC(C(N)=O)=O)C(O)C2)=O)ccc(Cl)c2ccccc12 52239,C1(=O)CCCC(C)NC(=O)C2CN1CCN2C.CC(C)CC(CO)N 52240,C(=O)(C(O)CCCNC(=O)CCCC1CC1C)N(CCC(=O)NC)CC 52241,C(=O)(C(C)CCCC(C)C)NCCCCNC(C(C(C)C)SC)=O 52242,CC1(C)CCCN(C(=O)C=Cc2cnc[nH]2)C1CNC(C1CC1[N+](=O)[O-])=O 52243,c1(CNCC(CCC)(C)C)cc(OC)c2cc(F)ccc2n1 52244,n1(CC)nc(C)cc1C(=O)NC(C(=O)N(C(C)CC1CC1)C)C1CCCO1 52245,c1(C(=O)NC2CC(CNC(C3(C)CN(C)C(=O)C3)=O)C2)cc2c([nH]1)CCCC2 52246,C12(C(=O)NCC3(NC(CNC(N)=O)=O)CCCCCC3)CCCCC1C2(F)F 52247,c1(CCN2CCC(CCOCC#C)CC2)c(Cl)cccc1Cl.C(C)=O 52248,CN1CC(C)(C(N2CC(N(C(=O)CSc3nncn3C)C)C2)=O)CCC1=O 52249,C1(C(=O)OC(C)(C)C)CC2CCC1(CC(=O)O)C2.C12CC(C1)CCC(=O)N2 52250,C1(CC(N2CC(CCCNC(COC)=O)OCC2)=O)NC(=O)CN(C)C1=O 52251,N1(C(C(=O)NCC)C(C)C)CCC(=O)N2CCCCCC12.C(=O)OC 52252,C1(CC)CN(C(=O)CC(F)(F)CC)CCN1C(=O)COc1cc(F)ccc1F 52253,C1(NC(c2n(CC)ncc2)=O)CC(NCCCOC(C)C)C12CCC2 52254,CCC(CC)C(=O)NC(Cc1cnn(C)c1O)C(=O)NCCc1noc(=O)n1C 52255,c1(SCC(=O)NCC(F)CNC(=O)CCN2CCOC2=O)ccccn1 52256,C1(NC(C=C(C)C)=O)CCC(C)N(C(C2C3COCC23)=O)C1 52257,C=C(C)C1OCCC1C(=O)NCCC1CC(NC(=O)CCOC)C1 52258,C1(C(COC)(C)O)CCN(C(C2(N(C)C)CC2)=O)CC1.C12CC1NC2=O 52259,Cc1ccn2c(C(N3CCOC(CCNC(c4ccccn4)=O)C3)=O)cnc2c1 52260,C1(C(=O)NCC2(F)CCCN(C(CCCNC(C)=O)=O)C2)CC2CCC1C21CC1 52261,C1(CNC(C2CCS2(=O)=O)=O)CCN(C(c2csc(C(F)(F)F)c2)=O)C1 52262,c1(C(N2CC(c3ccccc3)(NC(C)=O)C2)=O)cc(N)c(N)cc1F 52263,C(=O)(C1=NOC(C)(C)C1)NC1CCCC(NC(c2c(CC)[nH]cc2)=O)C1 52264,c1(CNC(c2c(C)c[nH]n2)=O)cccc(C(=O)NC(C)CN2CCCC2=O)n1 52265,C#Cc1cccc(CC(=O)NCC2(NC(c3[nH]cc(C)c3C)=O)CCOCC2)c1 52266,c1(C(=O)NCC(CC)NC(=O)C(F)(F)c2csc(Cl)c2)n[nH]c2c1CC(C)CC2 52267,S(=O)(=O)(c1cccc(NC(=O)C(=O)NC(C)CCN(C)C)c1)NCC 52268,C#CCCCC(C)C(=O)NC1CC(C(=O)NCCCN2CCCC2)C1 52269,Cc1cc(C(=O)NC23CC(CNC(c4csc(C(F)F)c4)=O)(C2)C3)cc2nc[nH]c12 52270,C1(NC(=O)CC2COC3CC2C3)CCC2(CCN(C(=O)C(O)CF)CC2)C1 52271,c1(COC)nc(C(=O)NCCC2CCC(NC(=O)C(F)C(C)C)C2)cc(O)n1 52272,C(=O)(C(C1CCCC1)NC(=O)CN(C)C(C)=O)NCC(C)OCC#C 52273,N1(CC(=O)NC(C(C)C)CNC(=O)C(C)n2cccn2)CCC(=O)NC1=O 52274,C1(N(C(c2ccn(CC(F)(F)F)n2)=O)CC)CCCN(C(C2(CF)CCC2)=O)C1 52275,n1(CC)ncc(C(=O)N(C2CN(C(=O)COc3ccc(CO)cc3)C2)C)c1Cl 52276,O=S(=O)(c1ccc(Cl)cn1)NC1CCC(NCc2ccc(Cl)cc2F)C1 52277,C(=O)(CC(CN(CC(=O)NC)CC1CC1)C1CCC1)N(C1CCCCC1)CCC 52278,CC1CC(NC(=O)C(C)(O)Cc2ccccc2)CCN1C(=O)C1=NOCC1 52279,c1(C(=O)NC(C)CNC(C2CCCCO2)=O)ccc2nc(O)sc2c1 52280,c1(CN2CC(CC(=O)NCCCC#C)OCC2)nc2ccccc2[nH]1 52281,N1(C(C#CC(C)C)=O)CCCC(C2CC2NC(=O)CC2CCCCCC2)C1 52282,c1(C(N2C(CN(C(=O)C=CC3CC3)C)CCC2)=O)c(O)nc(=O)n2c1CCC2 52283,n1(CCC(=O)N(C(C)CNC(c2cccnc2C)=O)CC)cnc(C)c1C(=O)OC 52284,c1(C(=O)NC(C2CN(C(c3conc3C3CC3)=O)CCO2)C)c(Cl)nsc1Cl 52285,O=S(=O)(c1[nH]cc2c1CCCC2)N1CCCCC1C(F)F 52286,Cc1ccnc(NC2CCCN(C(=O)CCOCC3CCC3)CC2)c1[N+](=O)[O-] 52287,C12(NC(C3CCC(C(F)(F)F)CC3)=O)CCC(CC1)N(C(C1CC1F)=O)C2 52288,c1(OCC)ncc(NC(=O)CCCN(C)C(c2sccc2CC)=O)cn1 52289,C1(F)(NC(CSCCOC)=O)CC2CCC(C1)N2C(c1cc(OC)nc(C)n1)=O 52290,C(=O)(C(CCOC)NC(=O)CCc1nc(C)no1)NC(C=C)C1CCC1 52291,N1(C(C2C(O)CCN2Cc2cncc(O)c2)=O)CCN2CC(O)CC2C1 52292,CC1CC(C(=O)NCCC2CN(C3CCC3)C2)N(C(=O)CC23CCCC2C3)C1 52293,N1(C(C2=CCN(C(c3cnc(C)[nH]c3=N)=O)CC2)=O)CCC2CCC(O)C1C2 52294,c1(C(N(CCCOCCNC(C(C)OCCC=C)=O)C)=O)cc(Cl)c(Cl)[nH]1 52295,C(=O)(C(F)(F)C(F)(F)F)NCC1(F)CCCN(C(C(c2cn(C)nc2)(C)C)=O)C1 52296,C(=O)(CCCCCCS(N)(=O)=O)NCC1N(C(CC2COC(C)(C)O2)=O)CCC1 52297,c1(N2CC3(C(NC(C4CC5C=CC4C5)=O)CCC3)C2)c(Cl)cc([N+](=O)[O-])cc1Cl 52298,Cc1cc(C(=O)NC(CNC(=O)C(C)(C)OCC(F)(F)F)CO)nc(O)c1 52299,C#CC1(O)CN(C(=O)C=CCC2(NC(=O)C(n3cc(C)cn3)C)CCC2)C1 52300,C1(C(N2CC(CO)C(O)C2)=O)(COC)C=CCN1C(=O)CN1CCCCCC1 52301,C=CCCC(C(=O)N1CCC(CCO)C1)NC(c1ccc(C)cc1)=O 52302,CN1CC=C(c2ccc(C3CCC(CNc4ncc5cn[nH]c5n4)C3)cn2)CC1 52303,C1(CCNC(C2(CC=C)CC=CC2)=O)CC(OC)CN1C(C1CCC1COC)=O 52304,c1(C(N(CC(C)(C)C(=O)NC(C2CCCO2)CO)C)=O)cccc2[nH]ccc12 52305,c1(CNC(=O)CC2C=CC(NC(C3CNC(=O)N3)=O)C2)cccc(CO)n1 52306,C1(C(=O)NCC(C)NC(=O)C(C2CC(F)(F)C2)O)CCCN(C)C1 52307,CN1CCC(C2CCN(C(c3c(Br)cnn3C)=O)C2)CC1 52308,N1(C(=O)C=Cc2ccncc2)CCC(C2CCN(C(c3ncccc3F)=O)C2)C1 52309,C(=O)(C(F)(F)CN1CCCC1)NCC(C)(CO)NC(C1(F)CCCCC1)=O 52310,c1(C(=O)NC2CCC(C)N(C(C3CCC(C(N)=O)C3)=O)C2)ccc2cnoc2c1 52311,N1(C(C=CSC)=O)CCC2CCC(C1)N2C(c1cccc(N2CCOCC2)c1)=O 52312,Cc1c(C(N)C(=O)N)cnn1C.c1(C2CCC2)ccc(F)cc1 52313,C1(CCCCCNC(C2CC2C2CC2)=O)CCN(C(c2nc(Cl)c(Cl)s2)=O)CC1 52314,C1(OC)(OC)CC(CNC(C2CCN(C(=O)CCC3CCCOC3)C2)=O)C1 52315,c1(C(=O)NC2CN(CC3CC34CCCCC4)CC2F)ccc2c(c1)OCCO2 52316,C(=O)(C(CCF)NC(=O)CN(C)C(=O)C1CC1)NC(C)CCCO 52317,C(=O)(C(O)P(C)(C)=O)NCCC(C)CCNC(c1c[nH]nc1C1CCOCC1)=O 52318,N1(C(CC2CC(SC)C2)=O)CC2(C(=O)N(C)CC3CCSC3)CC1CCO2 52319,C(=O)(C1=CCCCCC1)NCC(CC=C)NC(C1CC(Cl)(Cl)C1)=O 52320,C1(O)(CNC(c2cc(C)c(F)cc2)=O)CCCN(C(C2C=CCS2)=O)CC1 52321,C1(NC(c2nc(C)sc2C)=O)CC2(CNC(=O)CC(O)C(C)C)CC1CO2 52322,n1(CC)cnc(C(=O)NC(C)C(C2CCCCC2)NC(C2CC(C)(F)C2)=O)n1 52323,N1(C(CNC(C2(C3CCC3)CC2)=O)=O)CCN(C(=O)CC(F)(F)F)C2COCC12 52324,c1(C(N(CCC(=O)NC(c2ccco2)CO)C)=O)c[nH]c(=O)cn1 52325,N1(C(C2CCN(C(CC)=O)CC2)=O)CCC2(CCCN2C(=O)Cn2ncnn2)C1 52326,Cc1cccc2[nH]cc(CC(N3CCC(CN(C(=O)CSC(C)C)C)C3)=O)c12 52327,c1(C(N(C(CN2C(NC3CCN(C)CC3)CC2)=O)CC)=O)cnc2c(n1)CCCC2 52328,N1(C(C=CCCC)=O)CC(NC(=O)C(C)(C)C#N)C(c2ccnn2C)C1 52329,CCCCC(O)CNC(=O)COC1CCN(C(c2cn(C(C)C)nn2)=O)C1 52330,C1(C(N2CCC(C)(CNC(C3CCCN3C)=O)C2)C)CCCN(CC(F)(F)F)C1 52331,N1(C(c2cc(OCC)no2)=O)C2CCCC1CC(NC(c1c(Cl)cnn1C)=O)C2 52332,C1(CNC(C(C)O)=O)CC(F)CN1C(=O)C(F)=CCCF 52333,CCC1(CNC(C)CCC(C)C)OCCc2ccccc21 52334,N1(C(C(C)NC(CC)(C)C)=O)CC(C)(C)CC1CC(=O)N(C)CC1CC(F)(F)C1 52335,c1(C=O)n[nH]c2c1CC(C)CC2.CC(=O)CCCc1cn(C2CC3CCC2C3)nn1 52336,CCC(O)C(C)C(=O)N1CCCC(CNC(c2cc(C3CC3)ns2)=O)C1 52337,c1(C(N2CCCCC(CNC(Cc3cc(C)[nH]n3)=O)C2)=O)cnn2c(=N)[nH]cnc12 52338,N1(C(C(CC)CO)=O)CC2(C1)SCCC2NC(c1cccn2cncc12)=O 52339,C1(C(=O)NCCC#C)CC(O)CN1C(C1CC(=O)NC(=O)N1)=O 52340,C#Cc1cc(C(=O)NCCC(O)C(=O)N(CC)Cc2ccoc2)ccc1C 52341,C1(C2CCCCO2)(C(=O)NCC(C)CN(C)C(c2ccc(CO)o2)=O)CCCO1 52342,n1(CC(=O)NCC2(CNC(CCSC)=O)CCC2)cc2ccccc2n1 52343,C(C)(CN=C(NC(C)CCc1ccco1)NC1CCCC1)n1c(C)cc(C)n1 52344,C1(C(N2CCCC(N(C(CCN3CCN(C)CC3)=O)C)C2)=O)CC(C2CC2)=NO1 52345,CC1CN(C(c2nccc3nn[nH]c23)=O)C(C)CN1C(c1n[nH]c(O)n1)=O 52346,C1(NC(C2CC(C)(O)C2)=O)CN(C(=O)CC2CCCS2(=O)=O)CCC12CCC2 52347,c1(CNC(CCCOCCOCC)=O)ccc(NC(C)=O)nc1.n12cc(nn1)C2 52348,c1(CNC(CC2CCN(C(C(C)OCCOC)=O)C2)=O)nc(C)c(C)nc1C 52349,N1(C(=O)C=CC2CCCC2)CCC2OCCN(C(C3CCCCS3(=O)=O)=O)C2C1 52350,c1(C(N2CC(O)CC(NC(C(CC)N(C)C)=O)C2)=O)n[nH]c2c(C)cccc12 52351,C1(C(C)NC(=O)C(C)SC(F)(F)F)CCN(C(c2cnn[nH]2)=O)CC1 52352,c1(C(=O)NCC(CC)NC(c2coc(C(C)=O)c2)=O)nc(C)ccc1Br 52353,CCC(C)C(=O)C.N1(CC2CC2)CC(=O)NC(C(C)C)C1 52354,C1(CN(C(COCC=C)=O)C)C2CN(C(=O)CCCc3nc(C)no3)CC12 52355,c1(C(=O)NC(c2cc(=O)n(-c3ccccn3)[nH]2)C)ccc(F)cc1C(N)=O 52356,N1(CC)CCC(C(=O)NC23CC(C(=O)NCC(O)C(F)F)(C2)C3)C1 52357,CCC(C#N)(CC)C(=O)N1CC2CCCN(C(C3C4CC5C(C4)C35)=O)C2C1 52358,C(=O)(C(c1cnsc1)C(=O)OC)NCC(=O)OCC(=C)C 52359,N1(C(CCc2ccc(C)cc2C)=O)CC(CNC(C2(C)CC2F)=O)CC(C)(C)C1 52360,N1(C(C2C(C)CCOC2)=O)CCOCCC1C(=O)NCC1(F)CC1 52361,N1(C(C(C)N(C(c2cnnn2C)=O)CC)=O)CCN2C(=O)NCC2C1 52362,C1(OCC(=O)NCCC(C)(C)NC(c2cc(C)c(C)s2)=O)C#CCCCCC1 52363,CC(=O)C(C)(C)CC(=O)N1CC2(CC(C(=O)NCC3(C)CC3)CO2)C1 52364,N1(C(C(=O)NCC(N2CCc3sccc3C2C)CC)=O)CCC2(CCCCC2)CC1 52365,N1(C(c2c(C)cno2)=O)CC2CC(NC(=O)Cn3ccc(C(F)F)n3)C2C1 52366,CC1(CC(=O)NC(CC2CC2)CC2CC2)CCN(C(c2nccs2)=O)C1 52367,CCC(C)CC(C(=O)NCC(O)C(F)(F)F)NC(=O)CN(C)CC 52368,C1(C(N(C(C)C)CCN(C)C(c2ccnnc2O)=O)=O)CCC(C)NC1=O 52369,C1(=CCNC(C(C)(O)C2CCOCC2)=O)CCN(C(=O)C(F)OC(F)(F)F)CC1 52370,C1(NC(c2cnc(C(F)F)nc2)=O)CC2CC(C1)N(C(c1cnco1)=O)C2 52371,CCC(F)(F)CC(=O)NC(CC1CC1)CC(=O)Nc1cnn(C(C)(C)C)c1 52372,C1(C(=O)OC)CN(C(CC2C=CCC2)C(=O)NCCC2CC2)CC1C1CCCC1 52373,c1(CC(=O)NCCC(=C)CCNC(c2cc[nH]n2)=O)nc(C(F)(F)F)nn1C 52374,c1(C(C(=O)NCCCC2CC2)N(C2CCCS2(=O)=O)C)cccc(Cl)c1Br 52375,c1(C(=O)NC(C(C(C)C)NC(=O)COC2(C)CCCC2)C)cc2cc(Cl)ccn2n1 52376,C(=O)(C1=NOC2(CCC2)C1)N1CCC(COC)(CNC(=O)Cn2cnnc2O)C1 52377,C(=O)(CCS(=O)(=O)CC(C)C)N(CC(CN(C(c1ncc(C)cc1C)=O)C)O)C 52378,C1(C(C)NC(c2ccc(C)o2)=O)CCCN(C(c2ccc(NC(C)C)nc2)=O)C1 52379,C1(OCCOC)CCCC(C(=O)NC(C)CN(c2cc(Br)cnn2)C)C1 52380,c1(C(=O)NCC2(O)CCCN(C(C(C)=C(CC)C)=O)C2)cc2c(=O)[nH]ccn2n1 52381,C(=O)(C(F)C(C)(C)O)NCC1(C(=O)NCC=Cc2ccco2)CC(=C)C1 52382,c1(CCCC(=O)NCC23C(CN(C(C(C)OC)=O)C2)C3)ccc(C(F)(F)F)cc1 52383,Cc1cc(F)ccc1NC(c1ccc(CC2CC2)cc1)=O 52384,N1(C(c2n[nH]c(C)c2Cl)=O)CCC(CNC(=O)C(F)(F)C2(CO)CCC2)C1(C)C 52385,C(=O)(C=CS(C)=O)NCC(C(C)C)NC(c1cnn(C)c1)=O 52386,Nc1ccc(C(N2CCCCC(CNC(=O)COCC(F)(F)F)C2)=O)nc1F 52387,N1(C(C2C(CC)CCN2C(c2cc(C)oc2C)=O)=O)CCSC2(CCC2)C1 52388,N1(C(=O)COC2CCCC2)CCC2(CCN(C(C3CCCCS3(=O)=O)=O)CC2)C1 52389,N1(C(c2c(OC)nccn2)=O)CC(C2CCCCN(C(=O)C(=O)NC3CC3)C2)C1 52390,C1(CCC)C(=O)NCCN1C(=O)CC1C(NC(=O)Cn2cc(C#N)cn2)CC1O 52391,N1(C(CS(=O)(=O)NC)=O)CCCC(C)(C)C1C(=O)NC1CN(C)C(C)(C)C1 52392,C1(NC(c2cn(CC(C)C)nc2)=O)COCCN(C(c2ccc(=O)n(C)n2)=O)C1 52393,c1(C(=O)NC2CCC(CNC(c3nocc3Cl)=O)C2)ccc(F)c2occc12 52394,c1(CC(=O)NC2CC2NC(C2C3CCC(=O)C23)=O)ccc(F)cc1Br 52395,N1(C(C(COCC)NC(=O)CN(C)C(=O)OC)=O)CCCC1COC 52396,C1(NC(c2cnc(C)[nH]2)=O)C2CCC(C2)C1C(N1CCC(C)(F)C1)=O 52397,C(CNC(c1ccc(-n2cnnn2)cn1)=O)(C(C)(C)C)NC(C(C)(C)OC)=O 52398,C(=O)(C(C)Cn1ccnc1)N.C1(C(=O)OC)CC(CC(=O)N(C2CCCC2)CCO)C1 52399,C(c1cncn1C)=CC(=O)N(CC(C)O)CCNC(C(C1CCC1)OCC)=O 52400,c1(C(N2CC(OCCNC(c3cccc(O)n3)=O)C2)=O)cc(C(F)(F)F)ccn1 52401,Cn1nc(Cl)c(C(N2CCCC2CNC(c2cnc3n2CCC3)=O)=O)c1Cl 52402,C1(S(N)(=O)=O)(C(=O)NC2C(CNC(c3cc(C)oc3)=O)C2)CCC1 52403,C1(C(=O)NCCCC(C)NC(C(CCOC)OC)=O)CCCC(=O)CC1 52404,C1(C(=O)OCC)(C(C)NC(=O)C(c2ccc(Cl)cc2)(C)C)CC12CCC2 52405,C(=O)(C(C)(C)NC(=O)OC(C)(C)C)N1CC(C(C(=O)NCC2C(C)C2)O)C1 52406,C1(C)(CC(N2C(CN(C)C(C3(C)COC3)=O)CCC2)=O)CCCCC1 52407,CC(C(=O)N1CCC(C)(CNC(C2CCCC(C(N)=O)C2)=O)CC1)S(C)(=O)=O 52408,S(=O)(=O)(c1cc(Cl)ccc1F)NC1C(C(=O)Nc2ncc(OC)cc2O)CCC1 52409,CS(=O)(=O)c1ccc(C(=O)NCC(C2CC2)NC(C2(CO)CC2)=O)o1 52410,C#CCC(C)(C(=O)NC1CC1CCC)NC(c1cnc(NC)cn1)=O 52411,C1(NC(C(c2c(C)cccc2)C)=O)CN(C(C2(CO)CC2(F)F)=O)CC(C)(C)C1 52412,C1(NC(CC=CC(C)(C)C)=O)CCN(C(C2(CF)CC2)=O)CCC1CO 52413,N1(C(COC)=O)CCN(C(C2CC3CC2C3)=O)C(CS(C)(=O)=O)C1 52414,CC(C)(CCS(C)(=O)=O)C(=O)NC1C2CN(C(=O)C=Cc3cc[nH]n3)CC12 52415,C=CCCC(F)(F)C(=O)N(C1CCC(NC(=O)Cc2ccccc2F)C1)C 52416,C(=O)(C(O)CCSC)NCc1c(C2CN(C(C3(COC)CCOC3)=O)C2)ocn1 52417,c1(CNC(C(C)(C)C(F)(F)F)=O)cnn2c1CN(C(c1csc(CO)n1)=O)CC2 52418,N1(C(C2CCC(C)CC2)=O)CC2(CO)CC1(C(=O)NC1CCN(CCF)C1)C2 52419,N1(C(Cc2c(C)nsc2)=O)CC(C(N2CCCC2C(=O)N(C)C)=O)C2(CC2)C1 52420,Cc1ccc2c(C(=O)NC(C3CCCN3C(c3cc(Cl)c[nH]3)=O)(C)C)c[nH]c2c1 52421,C(CC(CNC(=O)CN1CCC(C)C1)NC(=O)C=Cc1ccoc1)OC 52422,C(=O)(C(C(C)C)C(C)C)N1C(CNC(C2CCCC(=O)N2)=O)CC(OC)C1 52423,CCCC(CCO)NCCCNC(C1(C#N)CCCC1)=O 52424,N1(C(c2c(SC)scc2)=O)CCOC(CCNC(=O)CCCn2cccc2)C1 52425,C12(NC(C(CC)=CC)=O)CCC(C(N3CCN4CCC3CC4)=O)(CC1)CC2 52426,C(C)(C)(CCC(=O)NC1CCN(C(=O)CC(O)C2CCCC2)CC1C)OC 52427,Cc1cc(NCc2ccc(S(C)(=O)=O)cc2)ncc1S(=O)(=O)NC(C)CS(C)=O 52428,c1(C(=O)NCC(CCCC)NC(=O)C2=C(C)OCC2)cnc2ncnn2c1O 52429,CS(=O)(=O)C=CC(=O)NC1CC(CNC(C2CC23CCOCC3)=O)C1 52430,c1(C(=O)NCC2CCCCN2C(c2cn3c(n2)SCC3)=O)cc(F)c(Cl)cc1Cl 52431,CC(C(C)C(=O)NC(C)C(C)C(=O)OC)NC(c1nc(=N)cc[nH]1)=O 52432,c1(C2N(C(=O)C3CC3)CCC2)ccc(F)c(F)c1.c12cncc(c1)NC(=O)CO2 52433,C1(CC)CC(C(=O)NC2C=CCC2)C1.C12(CC1)C(=O)N2C 52434,Cc1ncc(C=CC(=O)NCCOc2ccc(F)c(F)c2)c(O)n1 52435,C(CCCC(CO)NC(c1cc(C)ccc1F)=O)NC(CSCCC(=O)OC)=O 52436,Cn1ncc2c(NCCC34CC3COC43CCC3)[nH]c(=NCC3(CO)CC3)nc12 52437,C(CC1=CCCCC1)NC(C(Cc1ccco1)NC(C1CCN(C)C(=O)C1)=O)=O 52438,c1(C(=O)NCCN(C(C2CCC3(C2)N=N3)=O)CC)cccc(OC)c1OC 52439,Cc1ncc([N+](=O)[O-])cc1C(=O)NC(CNC(=O)CN1CCCC1)C(C)C(C)C 52440,C1(OCCNC(C2C=CCCN2)=O)CC(F)(CF)C1 52441,CC1C(C(=O)NC(CCO)c2ccco2)CCN1C(c1ccco1)=O 52442,N1(C(COCc2cc(C)on2)=O)CCCC(NC(c2cncc(Cl)c2C)=O)CC1 52443,C1(NC(c2cc(C)[nH]n2)=O)COC2(CCN(C(C3(CO)CCOCC3)=O)C2)C1 52444,CCCS(=O)(=O)CC(=O)NCC1CC2(CO1)CN(C(c1c(C)ncn1C)=O)C2 52445,c1(-c2n(-c3cccc(C)c3)nc(-c3ccn(C)n3)n2)cn(C)cc(Br)c1=O 52446,c1(NC)ccc(C(=O)NC(C)(CNC(=O)CC2CC2c2ccccc2)CO)nc1 52447,C(=O)(C1=CCCN(C(=O)OC(C)(C)C)C1)N(c1nc(F)ccc1Cl)C 52448,N1(C(C(CCSC)O)=O)CC(O)(C2CCN(C(c3ccc(CO)nc3)=O)CC2)C1 52449,c1(NC)ccc(C(=O)NC(C2CC2(C)Br)=O)cn1.C12(O)CN(C1)CC2 52450,c1(SC)ccc(NC(C2CS(=O)(=O)CC2N2CCCC2)=O)c(C#N)c1 52451,c1(NC(CNC(c2ccn(C(CC)CC)n2)=O)C2CC2)cc(O)nc(O)n1 52452,C1(C(=O)NC(c2cccc(O)c2)CO)CC12CCN(C(C1CC=CCC1)=O)CC2 52453,N1(C(C(C2(O)CN(C(c3ccc(C(C)=O)o3)=O)C2)F)=O)CC(=O)NCC1C 52454,N1(C(c2cc(C)oc2)=O)CC(NC(=O)C(C)Cc2cnc[nH]2)C(N=[N+]=[N-])C1 52455,C(C(F)(C(=O)NC(CC)C(N)=O)C(C)C)NC(c1ccn(CCC)n1)=O 52456,c1(N2C(CCCNC(CCCOC)=O)CCC2)cc2nncn2cn1 52457,n1(CCC(=O)N(C(=O)C(C)(C)O)C)cc(CNS(C)(=O)=O)nn1 52458,c1(-c2nn(-c3c(OC(F)F)cccc3)c(C3CC(F)C3)n2)ccc(F)c(Cl)c1F 52459,c1(CNC(=O)C=CC2CCCNC2)cn2c(n1)CCCC2 52460,N1(C(C=NOC)=O)Cc2nccn2CC(NC(c2cccc(C(F)(F)F)n2)=O)C1 52461,c1(C(N2C(C)CC(NC(=O)C(F)F)C2)=O)ccc2ncn(C)c(=O)c2c1 52462,C1(C)(CC(=O)NC(C)CN2CCOC2=O)CCN(C(c2cnccn2)=O)C1 52463,Cc1cc(CN2CC(NS(=O)(=O)c3cnoc3C)C(C(F)(F)F)C2)c(O)c(C)c1 52464,N1(CCNC(C2(F)CCC2)=O)CCNC(=O)C1.c12cccc(n1)CN(C)C2=O 52465,c1(NC2CC(CC)C3N2CCC3)cc(Br)c(CC)cc1C 52466,c1(C(=O)NCC(CC=C)NC(c2ccns2)=O)ccc2cc(C(C)C)ccc2c1 52467,N1(C(c2c(C)nc(C3CC3)nc2)=O)CCN(C(c2ccccc2O)=O)CC12CCC2 52468,C1(CCC(=O)NCC2(Cl)CCC2)CCCCN(C(c2ccc[n+]([O-])c2)=O)C1 52469,C(=O)(CCCCC(F)F)NC(CNC(C(C(C)C)n1cccc1)=O)CO 52470,N1(C(C(c2ccccc2F)(C)C)=O)CCCC(C)(CN=c2[nH]nc(CO)s2)C1 52471,CC1CC(NC(c2ccnn2C2CCOCC2)=O)CN(C(C2CCOCC2)=O)C1 52472,N1(c2nc(COC)nc(Cl)c2)CC2(CCC2)CC1CNC(C1(CCF)CCC1)=O 52473,C(F)(F)(C(F)(F)F)C1(SC)CCC1.c12ccc(cc1)C(C)NC2 52474,c1(C(=O)NCC2(F)CC(NC(C(CN(CC)CC)F)=O)C2)ccc(N)c(C)c1F 52475,n1(CC)nc(C(=O)NCC2CCCCN2C(=O)Cc2cccc(OC)c2)cc1C 52476,Cc1[nH]nc(C(C)C)c1C(=O)NC1CC(C)N(C(=O)CC(=O)NC2CC2)C1 52477,C1(C(=O)NCC23CC(CNC(C4CCC(F)CC4)=O)(OC2)C3)Cc2cscc2C1 52478,C1(NC(c2cn(C)nc2)=O)CN(C(c2cc(Br)no2)=O)CC1N=[N+]=[N-] 52479,c1(CC(=O)OC(c2ccnc(C)n2)C)ccc([N+](=O)[O-])c(C)c1 52480,CC(Cn1cccn1)C(=O)N(C(C)CNC(=O)Cc1ccn(C)c1)C 52481,C1(NC(C2CC(OC)C2)=O)CCN(C(c2n[nH]c(=N)s2)=O)C1 52482,N=c1cc(CO)cc[nH]1.N12CCN(CC1)C1CC(C1)C2=O 52483,C1(C)(C(=O)NC(C(C)NC(=O)CC2(CO)CCCC2)C)SCCCS1 52484,C#CC1C(C(N2CCC2CNC(=O)CN2CCC(O)CC2)=O)C1(C)C 52485,C(=O)(CC(O)CC(C)C)N(CCN(C(=O)Cn1nc(C)nc1C)CC)CC 52486,Cc1c(C(=O)NC23CCC2CN(C(c2cc(Br)n(C)n2)=O)C3)nn(C)c1N 52487,Cc1c(Br)csc1C(=O)OCCCc1ccc(C(F)F)o1 52488,n1(CC(=O)NC(C)CNC(C2(S(C)(=O)=O)CCCC2)=O)ncn2nccc2c1=O 52489,c1(CCC(=O)N(CCN(C(CN2C(C)CCC2)=O)CC)C)ccccc1C(F)(F)F 52490,N(C(=NCCC1CCC2(CCC2)O1)NCC1CCCC1)Cc1ccccn1 52491,C1(NC(=O)Cc2cncnc2)CC12CCC(NC(c1cc(Cl)cs1)=O)CC2 52492,c1(OC)ccn2ncc(-c3ccnc(NC(=O)C(F)(F)C(O)C4CC4)c3)c2c1 52493,CC1(OC(C(F)(F)F)C2CCOC2)CCOC1.C1C(=O)O1 52494,N1(C(c2sccc2I)=O)CC2CC2(C(=O)NCCC(F)(F)F)C1 52495,c1(C(C(=O)NCCCCCN(C(=O)COC(F)(F)F)C)O)ccc(Cl)cc1 52496,c1(SC)cc(NC(c2cn(C3CC(C(=O)N(C)C)C3)nn2)=O)ccn1 52497,C12(C(=O)NCCNC(C3CN(C(C(c4cnn(C)c4)C)=O)C3)=O)C=CC(CC1)C2 52498,Cc1ccc(C(N2C3CN(C(=O)Cc4scnc4-c4cccs4)CC23)=O)c(F)c1 52499,CCCC(C(=O)NC1CCCCN(C(=O)Cc2cccnc2)C1)S(N)(=O)=O 52500,C1(NC(c2c[nH]ccc2=O)=O)CN(C(C2CC3(C2)CC2(CC2)C3)=O)CC12CCC2 52501,C(=O)(CC(C)(C(F)F)N(C)C)NCCN(C(C1(C)CCC(=O)N1)=O)CC 52502,CC12CCC(C(=O)NC3CC3NC(C3(O)CCC3)=O)(CC1)CO2 52503,CC1CC(C)C(CNC(C2CCN(C3CC3)C2=O)=O)CN1C(=O)C1=CCCCC1 52504,c1(CNCCCc2ccc(F)cc2)ccc(F)c(F)c1Br 52505,c1(C(=O)NCC2N(C(CCCCCC)=O)CCCC2)cn(CCO)c(=O)nc1O 52506,C(CC(=O)N(C)CC1CCCCC1O)(C(C)(C)C)NC(c1cc(C)c(=N)[nH]c1)=O 52507,c1(C(=O)NCC(C)N(C(C(CC)CCOC)=O)C)cc2c(OC)ccc(C)c2[nH]1 52508,C(=O)(CCN(CCCO)C(C1CC1C(C)(C)C)=O)N(C(C#C)C)C 52509,C(c1ccncc1)=C(C)C(=O)NC(CN(C)C)C(=O)NC(c1ncc[nH]1)CO 52510,C1(N(C(c2ccco2)=O)CC)CCCN(C(=O)C=Cc2ccn(C)c2)C1 52511,O=[N+]([O-])c1cc(S(=O)(=O)N2CCC(F)(F)C(c3ccccc3)C2)ccc1Cl 52512,c1(CC(N2CCC(CC=C)(NC(=O)C(C(C)C)SC)C2)=O)ccc(C)c(OC)c1 52513,c1(NC(C2(C(=O)OC)CCC2)c2nn[nH]n2)cnc(C(F)(F)F)c(C)c1 52514,c1(CCN(C)C)cn(C)nc1C(=O)NCC1CC1NC(c1ccc(SC)cc1)=O.CS 52515,c1(C=O)nnc(O)cc1O.C1(CO)CCCN(N(C)NC(CCOCCC)=O)C1 52516,c1(C(=O)NC2CCC2)ccccc1C(=O)N(C(C)CNC(COC)=O)C(C)C 52517,C1(CNC(c2c(N(C)C)noc2)c2nnnn2CCC2CC2)CCCCCC1(F)F 52518,N1(C(CSc2cn(C)nc2)=O)CC(C2CC2NC(c2cc(C3CC3)on2)=O)C1 52519,c1(CNC(C(CCC)NC(=O)CC2CCOCC2)=O)ccc2ocnc2c1 52520,c1(C(=O)NCC2(NC(C(C)NC(C)=O)=O)CCCCC2)cc2c([nH]1)CCOC2 52521,C(=O)(C1=CCCCC1C)NCC1CN(C(C2(C(=O)OCC)CC=CC2)=O)CC1O 52522,n1(CC(C)C)c(CCCN(C2CCCCC2)C)nnc1-c1noc(C2CCC2)n1 52523,C1(CNC(C2(CC)CCC2)=O)(NC(=O)CC(C)(C)C(C)(F)F)CCC(C)(C)CC1 52524,CC1(C)CCN(C(=O)C=CC=C(Cl)Cl)CC1NC(=O)CCCOc1ccccc1 52525,O=C(C1CCc2ccccc21)NCC12CC1CN(C(C1(C(N)=O)CC1)=O)C2 52526,N1(C(C=Cc2n(C)ncc2)=O)CC2CC(NC(=O)Cc3ccc(Cl)c(F)c3)C2C1 52527,C1(C(N2C(CNC(CSc3nc(C)[nH]n3)=O)CC2)=O)CC(=O)N(C2CCC2)C1 52528,CN1CC(CC2C(C)(COC(=O)C)C(=O)NCCOCCNC2=O)C1 52529,CC(C)C(C(=O)N(C)C)NC(C1(F)CCN(C(=O)CCc2ccccn2)C1)=O 52530,Cc1ccc(C(CNC(c2cnc(S)n2C2CC2)=O)NC(=O)CC(C)F)cc1 52531,C1(C(N(C(CC(=O)OC)C)C)=O)(NC(=O)CCn2ccnc2C)CC(F)(F)C1 52532,C12(NC(C(c3cnn(C)c3)C)=O)CC(CNC(=O)CC3(C(F)F)CC3)(C1)C2 52533,CCCCCCCCC(=O)NCC1(C(N)=O)CN(C(c2cn(C)c(=O)n2C)=O)C1 52534,c1(C(=O)NC2CCCC2NC(c2nnc(O)cc2O)=O)ccc2cccnc2c1 52535,C(=O)NC(N(C1CCCc2ccccc21)c1c(C2(CC)CCC2)cccc1)=O 52536,N1(C(CCC(C)CN(C)C)=O)CCC2CN(C(c3ccc4snnc4c3)=O)CC12 52537,c1(NC(=O)NC(C(=O)NCc2cnc(CC)nc2)F)ccc(S(N)(=O)=O)cc1 52538,Cc1ccc(Cc2nc(C3CCC4(CC4)C3)n(-c3ccn(C)n3)n2)cc1C 52539,N1(C(C2(OC)CC2)=O)CC(CNC(C2(C)CC(F)(F)C2)=O)OC(C)(C)C1 52540,c1(C(N(CCNC(CS(CC)=O)=O)Cc2ccccc2)=O)cc(C#N)cc(C)n1 52541,C(c1ccc(Br)s1)=CC1CCN(C(CC)C(C)(C)c2ccccc2)C1 52542,C1(C(F)(F)F)(NC(C(=O)NCC2N(C(CCC)=O)CCCC2)=O)CC2CCC1C2 52543,CN1CCn2nc(C(=O)NCC3CCN3C(c3cccc([N+](=O)[O-])c3)=O)cc2C1 52544,Cn1cc(CCC(N2CCCC2CNC(C2CC(C)(O)C2)=O)=O)nn1 52545,CCC(C)(C(=O)NC1CCC(NC(c2ccnc(C)n2)=O)CC1)C(N)=O 52546,c1(C(N(CC(=O)NCc2c(CC)nns2)CC)=O)ccc(C)n1C 52547,N1(C(CCC2C(C)=NNC2=O)=O)CCN(C(=O)Cc2ccc(C)c(O)c2)CC1C 52548,N(C1CCC=C(c2nc(C(=O)OC(C)(C)C)c(C)s2)CC1)C(C1C2CCCC12)=O 52549,C1(NC(C=CC=CC)=O)CCCN(C(C2CN(C3CCOC3)C2)=O)C1 52550,CC1(C)CC(CNC(N2CCCC2CCOc2cccnc2)=O)C1 52551,Cc1c(CNC(C2(F)CN(C(C)(C)C)C2)=O)oc2ccc(Cl)cc12 52552,C(C)(C(CCc1ccccc1)NC(c1cnn(C)c1)=O)NC(Cc1cc(C)[nH]n1)=O 52553,c1(C(N2CCC(C(NOCC)=O)C2C(C)C)=O)cnn2cccc2c1 52554,Cc1c(CNC(=O)C(n2cc(CCC3(CO)CCC3)nn2)C)oc2ccccc12 52555,C(=O)(C1=CCCCC1C)NC(C)CC1CN(C(=O)C(C)CN(C)C)C1 52556,N1(C(CCN(CCC)C)=O)CC2CCCC2(C(=O)NCC(C)C(C)(C)C)C1 52557,C1(NC(C(C(C)C)OC)=O)C2CC3C1C3C2C(N1CCC(c2ncco2)C1)=O 52558,c1(OC)ccc(C(=O)NCC2(NC(=O)C=C(C)C)CC2)c(O)c1F 52559,C1(COC)(NC(=O)CC2(OC)CCC2)CCCN(C(=O)C(C)(C)CCOC)C1 52560,N1(C(C2CC23CCOC3)C(=O)NCCSC)CCOc2cc(C)ccc2C1 52561,c1(N(CCNC(C(=O)NC(c2ccccc2)C#C)=O)C)c(C)noc1C 52562,C=CCCCC(C)(C)C(=O)N1CC(CNC(C2(OC)CCOC2)=O)C(CCC)C1 52563,c1(OC(C)C(=O)NC2CCCN(C(=O)CCCF)C2)ccccc1Br 52564,C1(NC(C#C)=O)CC2(CCN(C(c3cccc(F)c3Br)=O)CC2)C1 52565,N1(c2nc(C)c(Br)cn2)CC(C)CN(C(C2CN3CCC2CC3)=O)CC1C 52566,N12CCOCC1C2c1cn(C2(C(C3(C)CC3Br)=O)CC2)nn1.C(=O)O.CO 52567,N1(C(C(C)N(C(CN(C(C)=O)C)=O)C(C)C)=O)CCCN(C=O)CC1 52568,c1(C(=O)NC(CC=C)CNC(=O)C(C)OCCN(C)C)ccc(O)nc1Cl 52569,CN1CCCC(C(N2CCC(C)(c3ccccc3)C2)C(=O)NC2CCC2)C1 52570,N1(Cc2c(C)nn(C3CCOCC3)c2Cl)CC=C(c2ccnn2C)CC1 52571,c1(C(=O)NC(CC(C)(C)O)C(=O)O)ccc([N+](=O)[O-])c(O)n1 52572,c1(OC)sccc1C(=O)NCC1(NC(=O)Cc2cc[nH]n2)CCOC1 52573,N1(C(CC=CCC)=O)CC(OC)CC1(C)CNC(c1ccc(C)cc1N)=O 52574,N1(C(c2c(OCCC)cccc2)=O)CCC(NC(c2cncnc2C)=O)C(C)C1 52575,N1(C(c2c(Cl)ccc(C)c2)=O)CCC2CN(C(C3(C(C)C)COC3)=O)CCC2C1 52576,c1(CN2CCCC(C(=O)NC(COC)C)CC2)cc2ccccc2o1 52577,Cc1cc(C)c(C(=O)OC2N(C(=O)C3CC3)CC(O)C2O)c(Cl)n1 52578,C(=O)(C1=CC2(CCOC2)C1)N(CC(CNC(c1cc(N)c(C)c(N)c1)=O)C)C 52579,CC(C)C(F)(F)CC(=O)N1CC(CNC(c2c[nH]c(C(N)=O)c2)=O)CC1C 52580,c1(SCC(=O)NC2(C)CN(C(c3c[nH]ccc3=N)=O)C2)ccsc1[N+](=O)[O-] 52581,N1(CC(=O)N(CCC(=O)NC(C2CCCC2)C)CC#C)CCCC1C 52582,CC(C)CCCCC(=O)N1CCC2CN(C(=O)COCc3cccc(Cl)c3)C2C1 52583,CCCCC(O)CCC(=O)NCC1CCN(C(=O)OC(C)(C)C)CC1(C)O 52584,CCCC(O)CC(=O)NCCN(C(=O)C(c1ccc(CC(C)C)cc1)C)C 52585,N1(C(CCSCCCC)=O)CCC(NC(C2CC(N3CCCC3)C2)=O)CC1 52586,CC1(NC(c2ncc(Cl)nc2Cl)=O)CCCN(C(=O)Cc2csc(C(F)(F)F)n2)C1 52587,N1(C(c2c(C)cn(C)c2)=O)CCC(O)C(N(C(=O)CCN2CCC(F)C2)C)C1 52588,C1(NC(c2c(OC)cc(O)nc2)=O)CCC2(CC1)CN(C(c1ncsc1C)=O)C2 52589,C(=O)(C(C)(C)CC(F)F)NC(CC(C)NC(c1cn(C)nc1C1CCCC1)=O)C 52590,N1(C(C(C)SC(F)(F)F)=O)CCOCC(NC(C2(c3ccno3)CCC2)=O)C1 52591,c1(C(=O)NCc2ccc(C(C)NC(=O)C(O)C(C)C)cc2)cnc(O)n(C)c1=O 52592,N1(C(C(C)CC2CCCC2)=O)CCC(C2CC2)(CNC(=O)COCCF)C1 52593,Cc1c(C(=O)NCCN(C(=O)CCN2CCCC2=O)C(C)C)cc(F)cc1Br 52594,c1(NCc2c(C3CN(C(c4cc(C)on4)=O)C3)ocn2)ncnc2sccc12 52595,C1(C(C)(C)O)(C(=O)NCCN(C(C2CC2F)=O)CC)CCCC1 52596,Cc1nnc2cc(NCCCCNC(=O)C(c3cccc(Cl)c3F)(C)C)ncn12 52597,C1(NC(CC2=NNC(=O)CC2)=O)CN(C(C23CC(F)(C2)C3)=O)C2(CCOC2)C1 52598,C1(N(C(C(C=C=C)C)=O)C)CN(C(=O)C=Cc2cccc(F)c2)CCC1O 52599,C1(NC(C2C(C(=O)OC)CC2)=O)C2CC3CN(C(=O)CC4=NNC(=O)C4)C1C3C2 52600,CC(CC(=O)NCCCN(C(=O)CC1CC(F)(F)C1)C1CC1)c1ccco1 52601,c1(CC(=O)NCC(CO)NC(=O)CCc2nncs2)c[nH]c2cnc(Cl)cc12 52602,Cc1ccc([N+](=O)[O-])c(NCC(=O)NCC2CC2NC(C2CC(CF)C2)=O)c1 52603,C(=O)(C1=CCCCC1P(C)(C)=O)N1CCN(C(c2c(C)nc(C)o2)=O)CC1C 52604,c1(CCS)cn2ccccc2n1.c1(-c2n(C3C(C)C3)nc(-c3nc[nH]n3)n2)cnn2cc[nH]c12 52605,c1(OCc2cn(-c3ccc(C(C)(C)C)c(Br)c3)nn2)ccc(C#N)c(F)c1 52606,C1(CC(=O)N(C)CC2(C3CCCO3)CC2)(NC(=O)CSC(F)F)CCCCC1 52607,C(CNC(=O)C(N1CCCC(C)C1)=O)(C(F)(F)F)OCC(=O)OC 52608,c1(C(N(C(C(=O)NCc2nnc(CC)s2)C2CC2)C)=O)cc(C#N)ccc1N 52609,C1(C(N2C3CCC2CN(C(C2(C4CCCO4)CC2)=O)C3)=O)COC2CCCCC12 52610,N1(C(c2c(C)nc(COC)s2)=O)CCC(NC(=O)C(C(C)C)NS(C)(=O)=O)C(O)C1 52611,C12(NC(CC3C(CC)C3)=O)CCC1CN(C(C1CCC(=O)N1C)=O)C2 52612,C1(F)(C(=O)NC2CN(C(C(C)N3CCC3)=O)CC2C)CCCCCC1 52613,Cc1ccc(F)cc1CC(=O)NC1(C)CCN(C(C2CCC3CC23)=O)CC1 52614,n1(CC(=O)NC2CC(NC(C(C)NC(N)=O)=O)C2)cc(CC2CC2)nn1 52615,C12(CNC(CCCN(C)C)=O)CCC(CC1)CN2C(=O)C(c1ccc(F)cc1)O 52616,c1(CN2CC(F)CC(C(=O)Nc3ccc(OC)nc3Cl)C2)nc2ccccc2[nH]1 52617,N1(Cc2cn(-c3c(Cl)ccc(C)n3)nn2)CCCC1C1CCCO1 52618,C(C(F)C(=O)NOCC(O)CO)C1CN(C(Cc2n(C)c(Cl)nc2)=O)C1 52619,C1(N(C(c2ccc(COC)cc2)=O)C)CC2CCC(C1)N2C(=O)C(C)(Cl)Cl 52620,Cc1ccc2[nH]c(C(=O)NCC(O)CCNC(=O)CCC(C)(C)C)cc2c1 52621,C1(C(=O)NCc2nnc(C)n2C)CCN(C(=O)C(C)C)C(C)C1 52622,c1(C(N2C(CNC(C3CC4(CC(=C)C4)C3)=O)CC2)=O)ccc2nc(C)cn2c1 52623,C1(N2CC(C)C(NC(C3(C)CS(=O)(=O)C3)=O)C2)CCc2ccccc2NC1=O 52624,c1(C(N2CCCC(C)(NC(C3C(C)C3)=O)C2)=O)cncc2ccsc12 52625,c1(OC)ccc(CC(N2CC(NCc3ccc(CO)nc3)CC(F)C2)=O)cc1Cl 52626,N1(C(c2c(CNC(=O)CCCCC3CC3)nccc2)=O)CCSC2CCC12 52627,c1(NC(c2[nH]cc(C(=O)OC)c2)=O)cccc(NC(C2(C)CCCO2)=O)c1 52628,N1(CCCOc2ccc(CCC(C)C)cc2)CCOC(C(F)(F)F)C1(C)C 52629,c1(N2CCSCC(C)C2)nccc(=NC2CCCn3nccc32)[nH]1.C(C(F)(F)F)N 52630,N1(C(c2csc(F)c2)=O)CC2OCCN(C(C3CCCN4CCCCC34)=O)C2C1 52631,C1(NC(C2(CNC(C(C)=C3CC3)=O)CCCCC2)=O)CC(O)C12CCC2 52632,C1(C(=O)NC(CC(C)NC(=O)CCOCCN(C)C)C)CC12CCC1(CC1)CC2 52633,c1(NC(CN(C(c2ccc(Cl)cc2)C(=O)NC)C2CC2)=O)cccc(NC(N)=O)c1 52634,C1(NC(CCSc2nc(C)[nH]n2)=O)CC2CN(C(=O)CN3CCCC(C)C3)CC12 52635,c1(OCC)ccc(NC(=O)CN2CCC(c3ccccc3F)C2)cc1 52636,C1(C(N2CC(C)(NC(CCc3cc(C)no3)=O)C2)=O)CCCCC1n1cccn1 52637,N1(C(c2ccc(F)c(C3CC3)c2)=O)CC(CO)c2ccccc21 52638,c1(C(N2CC(NC(C(C)(C)CCl)=O)(CO)C2)=O)cc2[nH]ccc2cc1Cl 52639,C1(C(=O)NC2(C#C)CC(F)(F)C2)C(C2CC2)CCN1C(=O)C=Cc1ccoc1 52640,N1(C(c2n(CC#C)cnn2)=O)CCC2(CCCC2NC(c2ccc(CO)s2)=O)C1 52641,C(C(CC(C)C)NC(c1ccc(-c2cc[nH]n2)s1)=O)NC(CC=CC=C)=O 52642,c1(N(C)Cc2nc(CC(=O)O)cs2)nnc(CCCN(C(c2cnn[nH]2)=O)C)o1 52643,C1(OC)CN(C(=O)C(c2cccc(Cl)c2)O)CC1NC(c1cc(C(N)=O)[nH]n1)=O 52644,C1(COC(N(C)Cc2ccccc2Cl)=O)COc2ccccc2O1.C1CS1 52645,N1(C(C(c2n(C)cnc2)O)=O)CC2(CCC(NC(c3ccccc3)=O)CC2)C1 52646,C(=O)(CC(C)CC(F)(F)F)NC1CCC(NC(c2nn(CC)c(C3CC3)c2)=O)C1 52647,c1(NC(C2C3(CN(C(Cc4nnc(C)o4)=O)C3)C2)=O)cc(Br)cnc1I 52648,c1(C(N2CCOC(c3ccccc3F)C2)C(=O)NC)ccc(COC)c(F)c1 52649,C(=O)(CC1CCc2ccccc21)N1CCN(C(=O)Nc2c(C)nsc2N)CC1 52650,C(=O)(CS(=O)(=O)C1CCCC1)NC1CCN(C(CCC2CC(OC)C2)=O)C12CC2 52651,CCCC(C(=O)NCCCCCNC(=O)C=Cc1cn[nH]c1)S(N)(=O)=O 52652,C(=O)(C(C)(C)CCCC(=O)NCC1(O)CN(C(c2c(C)nn(C)c2F)=O)C1)OC 52653,C1(CNCC(c2ccc(Br)cc2)C)CCC2(C1)CC2(F)F 52654,C1(NC(c2[nH]cc(CC)c2)=O)CC(F)CN(C(c2cccc(F)c2)=O)C1 52655,C1(CNC(CCc2c(C)n[nH]c2C)=O)CN(C(C2CCCOC2)=O)C(C)(C)C1 52656,Cc1nc(C(N2CC23CCN(C(c2c[nH]cc(F)c2=O)=O)C3)=O)cc(O)n1 52657,c1(SCC(=O)OCC(c2n(C)ccc2)=O)c(F)ccc(Cl)c1Br 52658,CC(N=c1ccc(C#N)n[nH]1)C1CCCCN1C(=O)CCN1CCCC1 52659,N1(C(C(Cc2c(C)n[nH]c2C)C)=O)CCCC2(NC(c3n[nH]cc3Cl)=O)CC2C1 52660,N1(CC(CC)C)CCC2(CC1)OCCc1sc(C(N3CC=CC3)=O)cc12 52661,C1(CNC(C(CCC)F)=O)CN(C(C2CCCCC23CC3)=O)CC12CCC2 52662,N(C(=NCc1cc2c(cc1Cl)CCCC2)N1CCCC(OC(C)C)C1)C(C=C)C 52663,C#Cc1cccc(C(N2CCC(C3CCN(C(=O)CN(C)C)CC3)C2)=O)c1C 52664,c1(C(=O)OC)cc2n(n1)CCCC2NC(C1CCN(C2CCCCC2)C1)=O 52665,C(=O)(C1=CC(C)(C)C1)NC1C=CCN(C(C(c2ccc(N)cn2)C)=O)C1 52666,C(C(C)(C)CC(=O)N(C)CC1CCCN(C(c2ccc(CSC)cc2)=O)C1)OC 52667,Cc1cc(C(=O)NCC(CC(=O)NCC2(C)CCCC2O)C2CCC2)nnc1C 52668,C(CC(F)(F)F)(c1ccc(C(F)(F)F)cc1)N(C(C1(c2ccccc2)CCC1)C)CC 52669,C1(CC=C)COCC1NC(=O)C(C1(O)CCC1)NC(=O)C(C)=C1CC1 52670,c1(C(=O)NC(CCCNC(C2C=CCC2)=O)c2ccccc2)ccc([N+](=O)[O-])[nH]1 52671,N1(C(C(C)Cc2ccnn2C)=O)CCC(C)(CNC(=O)Cc2cncs2)C1 52672,C1(NC(C2C(OCC)CC2)=O)CC1C1CCCN(C(c2cccnc2Cl)=O)C1 52673,c1(C(N2C(C)CC(NC(=O)C=Cc3cccc(Cl)c3)C2)=O)cccc2[nH]ncc12 52674,C(=O)(CC(C)C(C)C(C)C)N1CC(C(C)(C)O)(CNC(C(CC(C)C)C)=O)C1 52675,C1(NC(c2ccc(OC)cc2)=O)CC2(C1)CC(N=[N+]=[N-])C2.c12nc(cs1)C(=O)N2C 52676,C12(CNC(c3ccc(-c4ncc[nH]4)nc3)=O)CC1CN(C(c1coc(Cl)n1)=O)C2 52677,c1(C(N(C2CCN(C(c3nc(CC)oc3)=O)C2)C)=O)cc(Br)ccc1C#N 52678,C1(C(N2CC3CCCC3C2)=O)CN(Cc2cc(Br)ccc2Br)CCC1(F)F 52679,C1(C(=O)NC2CC(CO)N(C(C3CCC(O)CC3)=O)C2)CC2C=CC1CC2 52680,c1(OC)ccc(Br)c(C)c1C(N1CC(CNC(c2cc(C)c(C)s2)=O)C1)=O 52681,C(=O)(C1=CC(C)CC1)N1CCC(N(CCOC)C(c2cc(C)ccn2)=O)CC1 52682,C1(C(N2CCCC(N(C)C(c3scnc3Cl)=O)C2)=O)CCc2cncn2C1 52683,c1(COC)cc(CC(=O)NCC(C)N(C)C(c2c[nH]nc2C(C)C)=O)no1 52684,C(=O)(C(C)(C)C(F)F)NC1C(C(=O)NCc2cc(C)c(C)s2)COC1 52685,c1(NCC=C=C)cc(N2CCCC(OC(C)(C)C)C2)nc(SC)n1 52686,N1(C(c2n(C)nnc2)=O)CC2(CC2)CC1CC(=O)NCCC1(C)CCCC1 52687,CC1CN(C(=O)C(=O)C(F)(F)F)CC2(CCN(CCOCCO)C2)O1 52688,N1(C(N2C(CC(=O)OCC)COCC2)=O)C2CCC1CC1(C2)CC1(F)F 52689,C(=O)(CCCn1ccnn1)NC(C)C(=O)NCC1(CCO)CCCC1 52690,CC(C)C(O)CC(=O)NC12CC(NC(C3(C)CC3(F)F)=O)(C1)C2 52691,c1(SC)nc(=NC(CNC(C2CC3(CCCCO3)C2)=O)C(C)C)s[nH]1 52692,CC1(C2CC2)CCCN1C(=O)NC(c1cccc(F)c1)c1cccs1 52693,c1(C(=O)NC(CCC(=O)N(C2CC3OCCCC23)C)(C)C)cn2ccccc2n1 52694,c1(-c2nccc(NC(c3c(C(C)=O)c(C)ccc3)=O)c2)c(F)cc(CO)cc1F 52695,c1(C(C(=O)N(C2CN(C(=O)OC(C)(C)C)C2)C)O)cc(F)c(F)c(Cl)c1 52696,C1(N(C(c2c(COC)ncs2)=O)C)CC2CCC(C1)N2C(c1ccc(F)s1)=O 52697,C1(CNC(C2(COC)CC2)=O)CN(c2ncns2)CCC12CCOC2 52698,C(=O)(NNc1cc(C(F)(F)F)cc(Br)c1)c1c(C)nn(C)c1C 52699,N1(C(CC=CC=C)=O)CCCC2(C1)CN(C(=O)CC1CCCOC1)CCO2 52700,CC(C(=O)NC(CNC(=O)CCCn1c(O)nnc1O)C(C)(C)C)C(C)(F)F 52701,C1(NC(C2CC(O)(CC#C)C2)=O)CN(C(C2(NC(C)=O)CCOCC2)=O)CC1F 52702,c1(C(N2CCCC(CN(C(=O)Cc3nc[nH]n3)C3CC3)C2)=O)ccnc2[nH]nnc12 52703,c1(C(C)C)nn(C)c(C(=O)NC2CC2C(=O)O)c1Cl 52704,Cc1cc(C(=O)N(C2CCN(C(C3CCC4(CCC4)C3)=O)C2)C)nc(O)c1 52705,C1(C(N2CC(C)=C(C)CC2)=O)N(C(c2cn(C3CC3)cn2)=O)CC12CCCC2 52706,O=C1C2CC(O)CCN2C(=O)N1c1nnnn1CC1CCCCC1 52707,C1(CNC(CC2CC(C)OC2C)=O)CC2(CO1)CN(C(C1CCC1(C)C)=O)C2 52708,N1(CCn2c(Cc3ccc(Cl)c(Cl)c3)nnn2)CCc2c(Nc3ccccc3)cccc21 52709,CC1=C(C(=O)NCC2CCN(C(C3C(c4nc(C)no4)C3(C)C)=O)C2)CCO1 52710,C1(C(N(CCOC(C)=O)C)=O)(CCNC(C2SCC=C2C)=O)CCCC1 52711,C(=O)(CC(C)CN(C(c1cc(C)nn1C)=O)C(C)C)OCC 52712,C1(CC(=O)NC2CCC(CNC(COCCC)=O)C2)COCCN1CC 52713,C(CCCCCNC(C1OC2CCC1C2)=O)c1cn(CCCOCC(C)C)nn1 52714,c1(C(C2CCCO2)NC(CNC(=O)CCC2CC2(F)F)=O)ccc(Cl)nc1 52715,N#CC1CCCC1CN1CC(O)CC1c1ccc(Br)cc1 52716,CCCCC(C)C(=O)N1CC2(CCC2NC(c2ccc(F)c(CN(C)C)c2)=O)C1 52717,C1(CC)CCCCC1C(=O)N(C)CCN(C(c1cc(Br)co1)=O)C(C)C 52718,C1(NC(c2cc(CCCCC)[nH]n2)=O)CC2CC1N(C(=O)Cc1cnno1)C2 52719,c1(NC(CCCCn2cc(NC(C(COC)C)=O)nn2)=O)ccc(F)c(Cl)c1 52720,C1(CNC(c2c(CC)nccc2)=O)CN(C(C2CCC(C)CO2)=O)CCN1C 52721,Cc1cc(C(=O)N(C2CCN(C(=O)CCCN3CCCC3)CC2C)C)nnc1C 52722,C(=O)(C1CCCc2nncn21)NCCN(C(=O)C(C)n1ccnc1)CC 52723,C1(NC(C2(CN(C)C)CCCC2)=O)CCCN(C(=O)CCC2CNC(=O)N2)CC1 52724,C1(NC(C2(C(C)C)CCC2)=O)CN(C(c2ccc(N)c(Cl)c2)=O)CCC1CO 52725,C(=O)(C(O)CC(C)C)NC(C(=O)NCc1c(C)cccc1)c1ccco1 52726,C1(CCCC)CN(C(c2cn(CC)nc2C)=O)CCN1C(n1cnccc1=O)=O 52727,C1(N(C(CC2(OCC)CCC2)=O)C)CCC(NC(=O)C=Cc2nc(C)cs2)CC1 52728,C(=O)(C1CNc2ccccc21)NCCN(CCNC(C(CC)OC)=O)C 52729,C1(NC(CN(C2CCCCC2)C)=O)CCCN(C(=O)CCC2CCCO2)C1 52730,N1(c2nccc(C)n2)CC2CC(NC(c3c[nH]nc3C)=O)C2C1 52731,C(=O)(CCCC(F)F)N1C(CNC(=O)CCc2nc(C3CC3)no2)CC(OC)C1 52732,c1(C(N2CCC(C(=O)NCC3(C)CCCO3)C2)=O)ccc2ccc(Cl)cc2n1 52733,C(C)(C(O)C(=O)Nc1cccc(NC(c2ccc(NC(C)=O)cn2)=O)c1)OC 52734,C1(C(CNC(C2(CC)CCOC2)=O)C)CCN(C(c2cccn2COC)=O)CC1 52735,c1(CNC(c2cc(O)cs2)=O)csc(CNC(=O)CCOC2COC2)n1 52736,C1(CCCC)CCCN(C(=NCC2CCSC2)NCc2ccnn2C)C1 52737,c1(CNc2c(SCC)noc2)cc(F)cc(Cl)c1 52738,c1(C(=O)NCCOC2CCN(C(CCNC(C)=O)=O)C2)c(Cl)ccc2c[nH]nc12 52739,Cc1c(C(=O)N(C)CCOCCNC(=O)CN2CCC(C)CC2)cccc1Cl 52740,N1(C(C(C)CSc2ccccc2)=O)CCC2CN(C(=O)CC3CCC3)CC12 52741,c1(CC(=O)OC)ccc(C(=O)NC(C)(C)C(C)NC(C2CC23CCC3)=O)cc1 52742,CCS(=O)(=O)CC(=O)NC(CCNC(c1cnc(CC(C)C)[nH]1)=O)C(C)C 52743,c1(CSCCC(=O)N(c2ccccc2)C(C)C)ccccc1-c1cnc(F)cc1 52744,CC1CC(N(C)C(=O)N(N2CCN(c3ccccc3)CC2)C)C1(C)C 52745,c1(C(N(CCNC(C(C)OCCOC)=O)C(C)C)=O)cnc2ncnn2c1C 52746,C1(C(CC)C(=O)N2CC(N(C)C(C3CCCO3)=O)C2)CCC(C)CC1 52747,C1(NC(N2CC(C(C(=O)O)OC)C2)=O)C2Cc3ccc(Br)cc3C12 52748,C1(C(=O)NC(CC=C)CNC(=O)CCn2ccnn2)CCCOCC1 52749,N1(C(CC2CCCC(NC(CCCC(=C)C)=O)C2)=O)CCn2ccnc2C1C 52750,c1(C(c2n(CCCC)nnn2)NC2CC(C)(CCOC)C2)cccc(C)c1C 52751,c1(C(=O)NCC23CC(NC(=O)COc4ccon4)(C2)C3)ccc(F)cc1F 52752,c1(C(N(C)CC2(NC(=O)CCc3csc(=N)[nH]3)CC2)=O)cnc(-c2ccccc2)o1 52753,N1(C(CCCNC(c2ccc(Cl)cc2)=O)=O)CC2CCC(C1)N2C(C1(F)CC1)=O 52754,C12(C(=O)O)CC3(CC(C3)N1C)C2.C(C(=O)NC)(C(C)CC1CCC1)NC 52755,Cc1cc(F)c(N)cc1C(=O)NC1CCCCC1CNC(c1nncs1)=O 52756,CC(C)CC(C)C(=O)NCC(F)CNC(c1nccc(Br)c1O)=O 52757,CC(C)C(C(=O)NCCC(C)N(C)C(c1ccn(CC(F)F)n1)=O)c1cccs1 52758,N1(C(C(C)OCC2CC2)=O)CCC(N(C(=O)C(O)CC2CC(F)(F)C2)CCO)C1 52759,C(CN(C)C)(CC(C)C)NC(=O)CCO.C1=CCNC1=O.C1CO1.CC=CC 52760,N(C(=NCCCCl)N1CCCC2(CC2)C1)CC1CC(C(C)(C)C)OCC1 52761,C1(NC(Cc2n[nH]c(=N)s2)=O)(CNC(=O)C#CC2CCOC2)CC2CCC1CC2 52762,CN1CCC(C(=O)N(C2CCCN(C(=O)CCc3nncs3)C2)C)C1=O 52763,S(=O)(=O)(c1ccc(C(F)(F)F)c(F)c1C)C(=O)NC1(C(=O)NCC#C)CCCCC1 52764,C(=O)(CC(C)CC(F)(F)F)NCC1CN(C(C=CC)=O)CC12CC2 52765,c1(CNC(C(C)(F)F)=O)ccc(C(N2CCNC(C(F)(F)F)C2)=O)nc1 52766,C1(NC(CC(C)(C)C)=O)C2CC1CN(C(=O)CC(c1ccc(Cl)c(Cl)c1)O)C2 52767,c1(NC(C2C(CNC(C(COC)COC)=O)CCC2)=O)cnc2ccccc2c1 52768,C1(NC(CC(C(C)C)C)=O)CC2CC(C1)N(C(C1CC(=O)NC(=O)N1)=O)C2 52769,N1(C(C(C)N(C(=O)CC(C)(C)C)C)=O)CCC(O)(C(=O)N(C)C)CC1 52770,c1(C(=O)NCCC2CCCN(C(c3cc(OC)ncc3)=O)C2)cc(C#N)[nH]c1C 52771,c1(C(c2n(CCCOC)nnn2)NC(C)CCCCO)cc(C)ccc1C 52772,CN1CCN(C(C2C3CCC(=O)C23)=O)C(CNC(c2ccno2)=O)C1 52773,C1(NS(CC(C)C)(=O)=O)CC2CCC(C1)N2C(=O)C(C)(C)C 52774,c1(COC)ccc(C(=O)NC2(CCn3cc(C4(O)CCC4)nn3)CCC2)o1 52775,c1(C(N2CC(O)(CN(C(C(CC)CC)=O)C)C2)=O)cnc(C(F)F)cc1C 52776,c1(SC)cc(C(=O)N(CC(O)CN(C)C(c2ccc(C)cc2)=O)C)c(Cl)cc1Cl 52777,CCC(C)CC(C)N(C(=O)C(CCOCCO)NC(=O)C=CC(F)(F)F)C 52778,c1(CC(N2CC(NC(C(C=C)c3ccccc3)=O)(COC)C2)=O)cccc(O)c1 52779,c1(C(=O)NCCN(C(=O)C(C)(C)N(C)C)C)cccnc1N1CCCC1 52780,C(CC(C)C(=O)NC(CNC(c1coc(CS(C)(=O)=O)n1)=O)CO)=CC 52781,C12CCCN(C1)C2.c1(NC(CSC)=O)cnc(CO)s1 52782,N1(C(CC(COC)C)=O)CCCC2(C1)CN(C(=O)CC(C)CN(C)C)C2 52783,C1(N(C(C)=O)CC)CCC(CN2CCCC2NC(=O)COC2CCOCC2)CC1 52784,c1(C(=O)OC(C)=O)cc(O)nc2c(OC3CCCN(C(C=CC)=O)C3)cccc12 52785,C1(CCN(C(=O)COC2CC2)C2CC2)CCCN(c2nc(C(F)(F)F)ns2)C1 52786,C(=O)(N=c1ccn(C2CCC2)[nH]1)C1(CNC(=O)CC23CCCC2C3)CCCC1 52787,C(=O)(C(C)CC1CCC1)NCC(CC)N(C(=O)CSCc1cccs1)C 52788,CCC(CNC(C1CN(C(C2CC2Br)=O)C1)=O)(CC)NC(C)=O 52789,n1(C(CC)C)ccc(=NC(=O)C2C3CC2N(C(=O)Cc2ccns2)C3)[nH]1 52790,n1(CC(=O)NCC#CCNC(C(C)CC2CC2)=O)cnc2ccccc2c1=O 52791,O=C(CNC(C(=O)NCC1CC1C(F)(F)F)=O)N=c1ccc(Br)n[nH]1 52792,C1(C(=O)NCCN(C(=O)C=NOC)CCC)CCN(c2cnccn2)CC1 52793,N1(C(CNC(CC)=O)=O)CCC(CN2CCN(C(=O)CC(C)C3CC3)CC2)CC1 52794,c1(O)ccc(F)c(Br)c1F.C1(C(N(C)C)=O)CCCN(C2CC2)C1 52795,c1(C(=O)NC2C(CNC(c3c(C)noc3C)=O)CCCC2)cc(Cl)ncc1O 52796,C=CCC(CC=C)C(=O)N1CCCC(C)C1CNC(c1cnc(S)nc1)=O 52797,C(CC1CCOCC1)(C(=O)NCCCc1cc[nH]n1)NC(C1(n2nccn2)CC1)=O 52798,c1(OCC(N2CC(CNC(C(n3c(C)cc(C)n3)C)=O)C2)=O)ccc(Cl)c(F)c1 52799,Cc1c(Cl)ccc(C(=O)NCCCCCN(C)C(c2ccc(C3CC3)s2)=O)c1Cl 52800,c1(CN2CCCC(C(C)NC(c3cnc(Cl)cc3I)=O)C2)cc(Br)cc(O)c1O 52801,Cc1nc2ccc(C(=O)NC(CNC(C3CC(=O)N(C)C3)=O)C(C)C)cc2s1 52802,c1(C(=O)NCCNC(CC2CC(C)(C)OCC2)=O)cc(Br)cn2ccnc12 52803,C12(NC(C(C3CCCOC3)OCC)=O)CCCC1N(c1nc(CC)ns1)CC2 52804,c1(C(N2CC3(CN(C(C(CC)CCOC)=O)C3)C2)=O)[nH]c2cc(C)ccc2c1C 52805,C(CCS(=O)(=O)NCC(=O)NC1(CNC(=O)C=C(C)C(C)C)CCOC1)OC 52806,C#Cc1ccc(OCC(=O)NCCNC(=O)CC2CC(CC)=NO2)cc1 52807,N1(C(C2OCCN(C)C2)=O)CC2CC(C1)C2NC(=O)CSCCC(F)(F)F 52808,CC(CCCO)N=c1[nH]c(N2CC(C)OC(C)C2)nc2c1SCC2 52809,c1(C(=O)NCc2ccc(-c3nccc(N(C)CC)n3)cc2)cc(F)cnc1O 52810,c1(C(=O)NC(C(CO)NC(C2CCN(CCC)CC2)=O)C)cc(OC)cc(C)n1 52811,CC1(C)CC(NC(=O)CC2COCC2(C)C)CN(C(c2ccoc2Cl)=O)C1 52812,Cc1cc(C(=O)N(c2nc(Cl)ncc2-c2nn[nH]n2)C)cc2nc[nH]c12 52813,c1(CSCCCC=C(C)C)ccccc1.C(C)(C1CC1)=CC(=O)NCCOCCOCCO 52814,c1(C(=O)OC)cc(C(=O)NCC=CCNC(=O)C(C)(C)C2CCCCC2)n(C)n1 52815,c1(-n2cc(CCC3CCN(C(c4cscn4)=O)C3)nn2)ccc(C(=O)O)c(F)c1 52816,n1(CC(=O)NCCC(CC)(CC)NC(C(CC)O)=O)ccc(=O)c2ccccc12 52817,Cc1c(C(=O)NCC(C)CNC(C2(C(C)C)CCCO2)=O)cnc2ncnn12 52818,CC(C)(O)C#CC(=O)NC1CN(C(=O)COC(C)(C)C(F)(F)F)CCO1 52819,N1(C(C=C(C)C(C)(C)C)=O)CCCCC(Cc2c(C(=O)NC3CC3)c(C)ns2)C1 52820,Nc1cc(F)c(C(N2CC=CC(NC(=O)C3=CCCC3)C2)=O)c(F)c1 52821,CC1(C)CN(C(c2ccn(C3CCC3)n2)=O)C(CNC(=O)CNS(N)(=O)=O)CO1 52822,c1(C(=O)NCC(=O)NCC=C)coc(CNC(=O)Cc2cscn2)n1 52823,CCCCC(CC(=O)NC(COC)CCO)NC(C1(C2(C)CC2)CC1)=O 52824,C12(CC(N3CC(NC(CC4(C)CCO4)=O)C3)=O)CC3CC1(CO)CC3C2 52825,c1(C(=O)NCC2C3CN(C(CCC(N)=O)=O)C2CCC3)cc2cccc(F)c2o1 52826,c1(C(=O)NCCCC2N(C(c3cc(C(=O)OC)[nH]n3)=O)CCC2)n[nH]c(C)c1C 52827,c1(C(N2C(CNC(CC(=O)OC)=O)CC2)=O)cc(C(F)(F)F)ccc1Cl 52828,N1(C(c2ccc(CCCCC)cc2)=O)CCN(Cc2ncccc2F)CC1C#N 52829,c1(CC(=O)NCC(CC)NC(c2cc(O)cc(N)c2C)=O)ccc([N+](=O)[O-])cc1 52830,N1(C(C(C(C)C)NC(CC(C)C)=O)=O)CCCN(C(c2snc(Cl)c2Cl)=O)CC1 52831,c1(CCC)cccc(C(N2CC(NC(=O)C3=C(Cl)CC3)C(O)C2)=O)c1 52832,C1(O)(C(C(=O)N(CC(C)O)CCNC(C2CC2(F)F)=O)(F)F)CCOCC1 52833,Cc1cccc(Br)c1C(C(=O)NCc1c(C)n[nH]c1C)NC(=O)Cc1csnn1 52834,c1(OC(c2cccc([N+](=O)[O-])c2)C(=O)OC)cc2c(cc1Cl)OCCO2 52835,Nc1cc(Cl)cc(F)c1C(N1CC(CNC(C2CC=CC2)=O)C2(CCC2)C1)=O 52836,c1(OC)ccc(NC(=O)NCCCOc2c(C)cccc2Cl)c(F)c1 52837,CC(CCO)C(=O)N1CCCC1C1(NC(c2ccc(Cl)cc2)=O)CC1 52838,C=CCC(CNC(c1ccc(C#N)cc1)=O)C(=O)N1CC(C)(COC)C1 52839,N1(C(C(=O)OCC)=O)CCC(NC(c2cn(CC(N)=O)nn2)=O)C(F)C1 52840,C12(NC(C(C3CCC(=O)N3)C)=O)CC1CN(C(C1(O)CCCCC1)=O)C2 52841,CCCC(CCC)CC(=O)N1CCC(O)C1C(=O)NCC(O)C1(Cl)CC1 52842,C1(CC)CCCN(C(=O)C(COC)CNC(C2CCC=CCCC2)=O)CC1 52843,c1(NC(C(CC)CCOC)=O)cc(C#N)cnc1C 52844,c1(C(=O)NC(CNC(c2nnc(C)s2)=O)C(C)C)cccc(S(=O)(=O)CF)c1 52845,C1(c2ccccc2)(NC(C2C(C)C2C)=O)CC(NC(=O)C(C)CO)C1 52846,C1(C(=O)NCc2cnc(C)s2)CC(O)CN1C(C1CC1[N+](=O)[O-])=O 52847,C1(NC(C(C=CC)O)=O)C(C)(C)C(NC(=O)CCc2scnc2C)C1(C)C 52848,C=C(C)CCCC(=O)N1CCCC1c1cn(-c2cc(C(=O)O)ccc2C)nn1 52849,c1(C(=O)NC(CC)CNC(=O)CCNc2ccc(OC)cc2)cc(N)ccc1O 52850,S(=O)(=O)(c1ccc(C(=O)O)cc1)NC(c1cccc(OCC(C)O)c1)CF 52851,c1(C(=O)NC(C)CNC(C2(C)CCCCC2)=O)cncc(F)c1Cl 52852,N1(C(Cn2ncc(CC)c2)=O)CC2(C1)CN(C(c1ccc(Cl)cc1C)=O)CC2CO 52853,N1(C(C(=O)NC(c2cc(-c3ccccc3)no2)C)=O)CC(C)OC2(CCOCC2)C1 52854,C1(C)(C(N2CC(CN(C)C(C3OCC3(C)C)=O)OCC2)=O)CCCCNC1=O 52855,c1(C2CN(CCN(C)C(c3csc(C(C)(C)C)n3)=O)C2)ccc(Cl)cc1 52856,c1(C(N(C)CCN(C)C(c2cc(C(N)=O)c[nH]2)=O)=O)cc(C(F)(F)F)n(C)n1 52857,CC1=C(C)CC(C)(C(N2CCCN(C(c3cnc[nH]c3=N)=O)CC2)=O)CC1 52858,N1(C(CCCC=C)=O)CC2(CCN(C(C3CC3c3cscn3)=O)CC2)C1C(C)C 52859,Cc1c(C(=O)NCc2cn(-c3cccc(F)c3)nn2)oc2ccc(F)cc12 52860,C1(C(N(CC)CC2CCCN2C(=O)CP(C)(C)=O)=O)OCC2CCCC12 52861,c1(NC(C)=O)nc(C(C)(C)C)co1.C(=O)(C(C)N1CC(C)C1)N(C1CC(O)C1)C 52862,C(=O)(C(O)CC(C)C)N1C(CN2CCN(C(c3c(C)nns3)=O)CC2)CCC1 52863,C=CC(C)(C)C(=O)NC(C1CC(F)(F)C1)CNC(C1(C(=O)NC)CC1)=O 52864,c1(C(=O)OC)cc(C(=O)NCC(O)CN(C)C(c2ccn(C)n2)=O)c(C)s1 52865,C=Cc1cncc(C(=O)NCC2C=CC(NC(=O)C(C)O)C2)c1 52866,c1(C(=O)NC2CN(C(CCN(C)CC)=O)CC23CC3)cc(S(N)(=O)=O)ccc1Cl 52867,N1(C(c2scc(C)c2C)C(=O)NCCSC)CCCC2C1CCN2C 52868,C1(C(=O)NC(C)CN(C)C(c2cc3cscc3s2)=O)CCCC(F)(F)CC1 52869,C1(C)(C(=O)Nc2c(C(=O)OCC)scc2)CCN(C(c2cc[nH]c2)=O)C1 52870,C1(C(=O)NCC(COC)C)CCN(C(=O)CC2C(C)(C)C2(C)C)CC1O 52871,C1(CNC(c2nc(C)sc2)=O)CC2CCC1N2C(=O)CNC(C1CCOCC1)=O 52872,c1(SC)nn(C)cc1C(=O)NCC1(O)CN(C(=O)C=C(C2CC2)C2CC2)C1 52873,C=CC(C)(O)CC(=O)NCCOC1CCN(C(C2CCC(=O)NC2)=O)CC1 52874,CC1(C)C(CC(=O)NCC(O)(CO)c2ncco2)C1(C)C 52875,C1(NC(=O)CCn2cccn2)CCCCCN(C(c2cc(C(N)=O)co2)=O)C1 52876,Cc1ccc(F)c(C(=O)N(C)CCOCCN(C)C(C2CC(C)N(C)C2)=O)n1 52877,c1(CC)nc(C(N2CCC(O)(Cn3cc(-c4csnn4)nn3)C2)=O)c(C)o1 52878,c1(C(=O)NC2(CF)CCN(C(c3[nH]c(=NCC)sc3)=O)C2)cnc2ncccn12 52879,C(CN=c1nc(N2C3CCC2CC(F)C3)c2cc(Cl)ccc2[nH]1)(OC)OCC1CC1 52880,c1(CCNC2CCC(SC)C2)nc2c(s1)CC(C)CC2 52881,N1(CNC(C(C2CC=CCC2)NC(C(c2cncnc2)C)=O)=O)CCCNC1=O 52882,N1(C(C(C)OC)=O)CCCCC2(C1)CN(C(=O)Cc1csc(S)n1)C2 52883,CCC(CC)C(C)C(=O)N1CCC(CC(N2CCCNC(=O)C2)=O)C1(C)C 52884,c1(OC)cc(C#N)ccc1C(N1CCC(C(C)C)CC1)C(=O)NC1COC1 52885,C1(C(C)NC(C2N(CC)CC2)=O)CCN(C(=O)CC2CCC(=O)C2)CC1 52886,C1(C(N2CCCC(N(C(c3ccsc3)C)C)C2)=O)CC(c2ccccc2)=NO1 52887,C(C(=O)NNC(=O)C1CC1c1ccc(C)cc1)SCC=C(C)C 52888,N1(C(c2c(C)cno2)=O)CC(NC(c2c(Cl)cncc2Cl)=O)CC(O)C1 52889,C(CNc1nn(C)c(C)c1Cl)(N=c1cc(C)nc(CO)[nH]1)c1ccc(CC)cc1 52890,N(C1CCc2c(Cl)ccc(F)c21)CC(=O)N(c1ccc(C)cc1)C1CC1 52891,C1(Oc2c(C(N3CC(OCC(=O)OC)C3)=O)nco2)CCCC(C)C1 52892,C1(CC)C(NC(c2cc(C3CCCC3)n(C)n2)=O)CCN1C(=O)CCSC 52893,N1(C(C=CC(=O)OCC)=O)CCC2(C1)CN(C(C1(C)CCOC1)=O)CCO2 52894,c1(C(C(=O)NCCCF)N(C(C)C2CC2)CC)nc(C)ccc1F 52895,C1(CCCO)CCC(N=c2ccnc(NCc3cc(Cl)cc(Cl)n3)[nH]2)CC1 52896,C1(CCC(=O)NCC(CC)N(C)C(C2CC(=O)N(C)C2)=O)CCCCN1C 52897,NS(=O)(=O)c1ccc(-c2nnc(N3CCCC4(CCO4)C3)n2CCC2CC2)cc1 52898,C1(C)(C(=O)NC(C)(C)CNC(C2COCCN2CC2CCC2)=O)CCCNS1(=O)=O 52899,C(=O)(C1CCCc2scnc21)NCC(CNC(C1CCC(C(=O)OC)C1)=O)(C)C 52900,N1(C(C(CSC)OC)=O)CCCC(C(=O)N(C)Cc2cc(C)cs2)C1 52901,Cc1oc(Cl)nc1C(=O)NCC(C)(O)CNC(c1coc(C2CC2)n1)=O 52902,C1(C#N)(C(=O)NCC2CN(C(c3c(C)n(C)nn3)=O)C2)CCOCC1 52903,c1(NC(c2coc(CN3CCCCC3)c2)=O)c(F)cc(F)cc1F 52904,C1(CC)CN(C(=O)COCC2(F)CC2)CCC1NC(=O)CCc1ncc[nH]1 52905,CC(C)C(F)(F)CC(=O)NC(C)(CNC(c1cc(Cl)ccc1F)=O)C(C)C 52906,c12cnc(OC)c(c1)C(=O)N1CC(CC1C)CNC(=O)C2.C1CC12CC2.COC 52907,c1(C(=O)NC(C2CC(NC(=O)CCS(C)=O)C2)C)c(C(F)(F)F)cnn1C 52908,Cc1nc(CCC(=O)NCCC2CCN(C(c3c[nH]nc3C(F)F)=O)C2)cs1 52909,c1(CC(=O)N(C)C(C2CCCO2)C)ccc(COC)c(OC)c1.CO 52910,C1(NC(c2n(C)nnc2)=O)C2CCN(C(=O)CCCC(=O)OC(C)(C)C)CCC12 52911,C1(CCC=O)CCCCN1.C1(CCC=C)CCCN1C(c1cnnn1CC)=O 52912,CC1CN(C(=O)C(C)(C)CN(C)C)CC(C)N1CC#N 52913,N1(C(C(C)NC=O)=O)CCC(CCNC(c2cc(CCO)on2)=O)C1 52914,c1(C(N2C(C)CC(CNC(CC3CC(=C)C3)=O)C2)=O)ccc2nccn2n1 52915,n1(CC(=O)OC)nnc2c(NCC3(NC(=O)CC(C)(C)O)CCC3)ncnc12 52916,C1(C(=O)NCCN(C(C(C)OCCCCCC)=O)CC)CCCN(CCF)C1 52917,N1(C(C2CC(C#N)C2)=O)CCC2CCN(C(c3ncccc3Br)=O)C2C1 52918,C1(O)(C(N(CC(C)CNC(=O)C(C)(C)c2ccno2)C)=O)CC2CCC1C2 52919,C1(C(=O)NCC(CN(C(C2(CC=C)CC=CC2)=O)C)O)CC(F)(F)C1(C)C 52920,c1(-c2n(C(C=C)COC)ccn2)ccc(-c2ccc(C)s2)c(F)c1 52921,c1(C(N(CC(CN(C(=O)CSc2nncs2)C)O)C)=O)cc([N+](=O)[O-])cnc1O 52922,c1(OCC)cnc(C(N2CC=CC(NC(c3ccc(CC)[nH]3)=O)C2)=O)cn1 52923,CC1(C)C(C(N2CC(O)(CNC(=O)C(F)=C3CCCC3)C2)=O)C1(F)F 52924,C1(NC(Cc2cccc(OC)c2)=O)COCCN(C(=O)CC2(C)CC2(Cl)Cl)C1 52925,C(=O)(C(O)C(F)F)NCC(CC(C)C)NC(=O)C(C)N(C)C(C)=O 52926,N1(C(c2ccc(CC)nc2)=O)CCCC(NC(c2cn[nH]c2)=O)C1C 52927,c1(C(N2CC(C)C(C)(CO)C2)C(=O)NCCC)cc(Cl)c(Br)cc1F 52928,N1(C(C2=CCCC2C)=O)CCC(C(=O)NCC2CC3CCCC3C2)C12CCC2 52929,c1(C(=O)NC(C)C(C)NC(C2(CCO)CC2)=O)cnc(-c2ccccn2)nc1 52930,N1(C(Cc2n(C)ccn2)=O)CCCC1(C)CNC(c1cnc(-c2cccs2)s1)=O 52931,C#Cc1ccc(C(=O)NCCC(C)CCNC(C2(O)CCSC2)=O)c(C)c1 52932,N1(C(c2n[nH]c(C)c2Cl)=O)CCCCC(NC(C2(c3cccnc3)CCC2)=O)C1 52933,c1(OC)c(C(=O)N(CC(C)C(=O)N2CC(N(C)CCO)C2)C)cnn1C 52934,C1(CCNC(c2c(C)n[nH]c2)n2c(S)nnn2)CC(F)(F)C1(C)C.C1CC1.C1CC1 52935,N1(C(CC=C(C)C)=O)CCCC2(CNC(C34CCC(C)(C3)OC4)=O)CCCC12 52936,C(CCC(=O)NCCCC1(C)CC1)(C(C)C)NC(c1ccc(C)c(F)c1)=O 52937,Cc1ccc2c(N3CCC3(C)NCc3ccc(Cl)cc3C(F)(F)F)ncnc2c1 52938,c1(NC)cccc2nc(CNC(c3c(OC)cccc3F)=O)c(C)nc12 52939,n1(CC)cc(C(=O)NC2CCN(C(=O)CCC#N)C(C3CC3)C2)c2ccccc12 52940,c1(CC(=O)Nc2ncc(SC)s2)cn2c(n1)CN(C(c1cc(Br)cnc1C)=O)CC2 52941,N1(C(CSCC)=O)CCc2ccccc2C(NC(=O)CC2(COC)CC2)C1 52942,c1(CN(C(=O)CC2(O)CNC2)NC)ccc(COC)cc1F.c1ccccc1 52943,CCC(CC(=O)NCC=CCNC(=O)C(C1(CN(C)C)CCOCC1)C)C1CC1 52944,c1(C(N2CC3CN(c4ccncn4)CC23)=O)cc2ccccc2o1 52945,C1(CC(=O)NC2C=CCN(C(c3ccc(CC)o3)=O)C2)NC(=O)CN(C)C1=O 52946,C1(F)(CNC(c2c(C)[nH]nc2C2CC2)=O)CCCN(C(c2ns[nH]c2=O)=O)CC1 52947,c1(CN2CCc3n(C)c(C4CC4)nc3C2)nc2ccccc2c(=NCC(F)(F)Br)[nH]1 52948,C1(C(=O)NCCOC2CCN(C(C3CCCCO3)=O)C2)CCc2nc[nH]c2C1 52949,N1(C(c2c(Cl)c(C)n(C)n2)=O)CCC2CCCN(C1)N2C 52950,C#CCC1C(=O)N2CC(C2)CONC(=O)C1.c1(SC)c[nH]ccc1=O 52951,Cn1cc(CNC(=O)C(N2CCC(N3CCOCC3)C2)=O)c(C(F)(F)F)n1 52952,N1(C(CNS(NC)(=O)=O)=O)CCCOC(CNC(=O)C(C2CCCCCC2)O)C1 52953,N1(C(C(C(C)C)(C)C)=O)CC2OCC(NC(C3CCCN(S(C)(=O)=O)C3)=O)C2C1 52954,c1(C(=O)NCC2(O)CC(NC(C3CC(F)(CO)C3)=O)C2)cc2ccccc2o1 52955,Cn1nc(C(N2CC3CC3C2C(N2CCC3CC23C)=O)=O)cc1C#N 52956,N1(C(=O)Nc2cnc(OC)nc2)CCn2c(NC(C)(CO)C(=O)O)nnc2C1 52957,C(=O)(C(CCC)=CCC)NCCC1(NC(C2(C=C)CC2)=O)CCC1 52958,c1(COC)ccc(C(=O)NCC2CCC2NC(=O)C(C)(C2CC2)NC(C)=O)o1 52959,c1(-c2c(C(c3nnnn3C3CC3)NCC(C)F)occ2)ccc(Cl)cc1 52960,c1(C(=O)NC(C2(CNC(CCN(C(CCC)C)C)=O)CC2)C)csc(Cl)c1Cl 52961,Cc1nn2c(C(=O)NCCCCNC(=O)C(C)C(C)C)c(C)nc2s1 52962,Cc1cc(=NC(=O)C(=O)C(C)(C)C)[nH]n1-c1ccc(C)c(Cl)c1 52963,N1(C(C(C)(N(C(C2CCC(C)(CC)O2)=O)C)C2CC2)=O)CCCC(C)(COC)CC1 52964,c1(C(N2CC(CNC(C(CC)F)=O)C(C)C2)=O)cc2cc(Cl)cnc2[nH]1 52965,c1(NC(C2C(NC(C3CC(=O)NC(=O)N3)=O)CCOC2)=O)cccc2c1CCO2 52966,C1(CCNC(CCCCN(C)C(c2ccn(C)c2)=O)=O)CCCC(C)(C)C1 52967,C1(C(=O)OC(C)(C)C)(NC(C2CCC(C3CC3)C2)=O)CC2(CCCCC2)C1 52968,CC(CCNC(C1CCC(=O)O1)=O)CCNC(c1ccn(CCC(F)(F)F)n1)=O 52969,C(C)(C)(CCCCNCC1(SC)CCOC1)NC(C1(C(=O)NCC=C)CCC1)=O 52970,c1(C(=O)NCc2nc(CNC(C3C(C)(C)C3)=O)sc2)cc(S(N)(=O)=O)ccn1 52971,C1(NC(C2(C#C)CN(C(=O)C(C)C#N)C2)=O)CCOCC12CCC2 52972,C1(NC(c2cnc(CNC(C(c3cccs3)OC)=O)s2)=O)CCC(=O)N(C)C1 52973,N1(C(c2cn(CCC)nc2)=O)CCC(C(=O)NCC2CC(C)=NO2)C12CCC2 52974,N1(C(c2c(CC)c[nH]c2)=O)CC(C)N(C(=O)C=CC(=O)NC2CC2)CC1C 52975,c1(C(=O)NC2CN(C(CNC(CC)=O)=O)C(CC)(CC)C2)ccc(CC)cc1C 52976,N1(c2snc(C)n2)CCC2CC(CNC(C3C4CC5CC(C4)CC3C5)=O)CCC2C1 52977,O=C1CC2CC(C(=O)NCc3cc(C(N4CCCC4C4CCCC4)=O)no3)C1O2 52978,CC1CN(C(=O)CN(C2CCC2)C)CCCN1C(C1CC(n2cccn2)C1)=O 52979,CCCC(C)CC(=O)N1CCCC(CN(C)C(c2ccc(C3CC3)s2)=O)CC1 52980,Cn1cc(C#N)cc1C(N1CCCCC1CN1CC2(CC(N)C2)C1)=O 52981,c1(C(N2CC(COC)(CNC(=O)C(F)(F)C3(O)CCC3)C2)=O)ccnc(C)c1O 52982,C1(C(=O)NC(CC)C)CCCN(C(=O)Cc2csc(C(F)(F)F)n2)C1 52983,C1(CC)CCN(C(=O)CC2(C)CCC2)C(C(=O)NC2CC(C)C2)C1 52984,N1(C(c2c(C)ocn2)=O)CCN(CCN(C)Cc2ccnn2C2CC2)CC1 52985,c1(C(C)(C)C)cc(NC2CC(NC(=O)CCC(N)=O)C2(C)C)ncn1 52986,C(=O)(C(CCC1CCCC1)N(C)Cc1cn(C)nn1)NCC=CC 52987,c1(C(N2C(CNC(=O)C(O)c3ccsc3)CC(O)C2)=O)cnn2c1OCCC2 52988,C1(N(C(=O)CC2N(CCC(C)C)CCC2)CC2CCCO2)CCN(C(C)=O)CC1 52989,C12(C(=O)NCC=CCNC(COc3c(Cl)ccc(C)c3)=O)C3C4C1C1C2C3C41CO 52990,N1(C(C(C)C2CCCC2)=O)CC2CCC1C2NC(c1ccc(Cl)c(O)c1)=O 52991,Cc1ccc(C=CC(=O)NC2CCN(C(C3CS(=O)(=O)C3)=O)CC2CO)nc1 52992,N1(C(CC2C(NC(=O)OC)CC2)=O)CCC(OC(C)C)C1 52993,C=CCCCC(C(=O)N1CCn2ncnc2C1)OC.c12cc(no1)N(C1CC1)C2=O 52994,Cc1c(CC(=O)NCCCNC(=O)CC2C=CCC2)cccc1[N+](=O)[O-] 52995,c1(CC)cc(C(=O)NCC(C(C)C)NC(=O)C(C2CCC2)OC)ncn1 52996,CC1(C(=O)NC2CC(=O)N2)CCN(C(=O)NCC(F)F)C1 52997,C1(NC(=O)CCc2ccc[nH]2)CC2CN(C(c3cccc(Cl)c3Cl)=O)CC12 52998,C1(NC(C2CCN(C(c3cn(CCC)nc3)=O)C2)=O)CCN(C)CC1C#N 52999,C1(C(=O)NC(C2CCOC2)C#C)CCC(C)N1C(C1CCOCC1)=O 53000,C(CCN=c1[nH]c(N2CCOC(CF)C2)nc2c1SCC2)OCC(C)C 53001,c1(NC(C(=O)Nc2oc3ccc(OC)cc3c2)=O)ccc2c(Cl)cccc2c1F 53002,Cc1cccc(C(F)(F)C(=O)NCCN(C(=O)CSC(F)(F)F)C(C)C)c1 53003,N12CC(C3(CCN(C(=O)CCC)CC3)C1)C2C(=O)NCCCC.C(C)(=O)OC 53004,C1(NC(C2C(C)CCC2)=O)(CNC(C2CC(F)(F)C2)=O)CCOCC1 53005,C1(CC(N2CCN(C(C(C)Cn3ccnc3)=O)CC2)=O)COc2ccccc2O1 53006,C(c1cncnc1O)=CC(=O)NCCC(C)N(C)C(C1CCS1(=O)=O)=O 53007,C1(CN(C(=O)CCN2CCC2)C)CCN(C(c2cn(C3CCCC3)nn2)=O)CC1 53008,C1(C(=O)NCC(C)CC2CCC2)CCC2CCC1N2C(=O)Cn1cnnc1O 53009,c1ccc2c(c1)nc(N1CCc3c1cccc3I)c1cc[nH]c21 53010,CC(CC(=O)NOC(c1ccccn1)C)C1CC1.C1(=O)C(F)(F)CO1 53011,C(=O)(CC(C(F)(F)F)OC)N1CC(F)(CNC(CC2(CC=C)CCCC2)=O)C1 53012,N1(C(C2(CC#C)CCCCO2)=O)CCC(NC(=O)Cc2ccco2)C(F)(F)CC1 53013,C(=O)(C1=CC2CCCC12)NCC(C)CNC(c1c(O)cccc1Br)=O 53014,N1(C(C(CCF)NC(C(CC=CC)C)=O)=O)CCCNC(=O)C1 53015,C1(NC(C2CC3CC2C2CC32)=O)CCC2CN(C(=O)C=Cc3cscn3)CC2C1 53016,N1(C(C(CC2CCC2)NC(Cc2cccc(C#C)c2)=O)=O)CC(F)(F)CCC1C 53017,c1(OCCC)ccc(NCC=CCNC(=O)NCC)cc1OC1CC1(F)F 53018,Cc1sc2ncnc(N3CCC4CCC(C3)N4C(C3CC34CC(O)C4)=O)c2c1C 53019,c1(C(N2CCC(CNC(CC(C)OC)=O)CC2)=O)ccc2c(c1)CC(C)(C)C2 53020,c1(CN(C)CCN2CCOC2=O)ccc(-c2cnn(C)c2)cn1 53021,Cn1cc2c(n1)CCCC2C(=O)NCC(C)(O)CNC(=O)CC1(O)CCC1 53022,N1(C(C=CSC)=O)CCCC(NC(C2(c3ccnc(Cl)c3)CC2)=O)C1C 53023,C#CC1(CCOC)COCCN1C(C(=O)NC1CC(F)(F)C1)C1CC1 53024,C1(C(N2CCSCC2C2CCC2)C(=O)NC2(C)CC2)CCOC2(CCOCC2)C1 53025,N1(C(CC(CC)O)=O)CC(C)CN(C(c2cc(F)n(C)n2)=O)CC1C 53026,Cc1c[nH]c(=NCCCC2NC(=O)N(C)C2=O)c2ccccc12 53027,C1(NC(CCC(C)CN(C)C)=O)CCCCC12CCN(C(=O)CNS(N)(=O)=O)C2 53028,c1(CCNC(C2C(=C)CC2)=O)ccc(CNC(C2C3CCC2CC3)=O)cc1 53029,CC1CN(C(c2cnc(C3CC3)s2)=O)CCCN1C(=O)CC1CCCCC1O 53030,Cc1sc(O)nc1C(N1CCCC(NC(c2cnc(Br)s2)=O)C1)=O 53031,C(=O)(CCCCC(N)=O)N(C1CCN(C(c2cnc(C)s2)=O)CC1)CCOC 53032,N1(C(CC2CC(C)(C)C2)=O)CC2CCCC(NC(c3nc(Cl)c(Cl)s3)=O)C2C1 53033,C1(C(N(C)CCNC(c2cccc(=O)o2)=O)=O)CC(C)(C)OC1(C)C 53034,C(=O)(C(C)(C)S(C)(=O)=O)NC1CN(C(c2c(OC)c(F)ccc2)=O)CC(C)C1 53035,CC(C)CCC(=O)NCC(=O)OCCOCCO.C12CC1CC(=O)N2C1CC1 53036,C1(C#N)(C(=O)NCC(C)(C)NC(C2CCCN(CC(F)(F)F)C2)=O)CC12CCC2 53037,N1(C(=O)CNc2cccc(CO)c2)CCN(C(=O)CN2CCCCC2=O)C2CC12 53038,C1(C(=O)NC(C(=O)N(CCC(C)C)CCCO)C2CCCC2)CC(C)(F)C1 53039,N#Cc1ccc(CC(=O)NC2(C(N3CCCOCC3)=O)CC(F)C2)cc1 53040,C(CN=C(NCc1cc(Cl)ccc1Br)N1CCC(C2CCOC2)C1)N(CC)CC 53041,N1(C(c2c(C)cc(OC)o2)=O)CCC2(C1)CN(C(c1ccn(CCO)c1C)=O)C2 53042,c1(CC(=O)NC(CC(=O)NC)C(C)C)noc2ccc(O)cc12 53043,Nc1c(C(N2CCSCC2CCNC(C2(O)CC(F)(F)C2)=O)=O)cccc1F 53044,C1(C(=O)NCC2C(CNC(CN(C(=O)OC)C)=O)C2)(OC)CS(=O)(=O)C1 53045,c1(CC)cc(N)c(C(N2CCCCC2C2CC2)=O)cc1F 53046,c1(C(N2C3(CN(C(c4cnccn4)=O)C3)CC2)=O)cnc2c(F)cccc2c1 53047,CC1(C)CCCCC1C.C1(c2nc3n(n2)-c2ccccc2-3)CCCCCCC1 53048,c1(OC)ccc(CC(=O)NC2(C)CCN(C(C34CCC(OC)C3C4)=O)C2)cc1Cl 53049,C1(C(=O)NC2(C(=O)NCC(C=C)O)CC(F)C2)CN(C)CCO1 53050,c1(NC(=O)COC(C23OC(C)C(CC2)C3)=O)cc2cccnc2s1 53051,c1(C(C)C)ncc(C(=O)NC(C)CCNC(c2nncs2)=O)s1 53052,Cc1nc(NC2CCN(C(=O)Cc3ccc(C(N)=O)cc3)C2)c2c[nH]nc2n1 53053,C1(NC(C=CC=CC)=O)CS(=O)(=O)CC1NC(C1(S(C)(=O)=O)CC1)=O 53054,C1(C(N(c2cccc(O)c2)CC)=O)CCC2CCC1N2C(=O)C(O)CC(C)C 53055,C1(CC)CCN(C(=O)C(CC)N(C)C(C2CSC2)=O)O1 53056,C(=O)(C(CC(C)C)NC(C1CC(n2cncn2)C1)=O)NCCNC(C)=O 53057,CCCCC(=O)C(=O)N1CC(C)CC1C(N1CCCC(CN(C)C)C1)=O 53058,C1(C(N(C)CC2CCCN2C(c2ccc(Cl)o2)=O)=O)CC2CC1C1CC21 53059,C1(CNC(C(C)C)=O)COCC2(CCN(C(C3(F)CCC3)=O)C2)O1 53060,CCCCCC(=O)N1CCC(C)(NC(=O)C(c2ccc(Cl)cc2)OC)C1 53061,C(=O)(C1CCCc2cn(C)nc21)NCCC(C)NC(c1cccc(O)n1)=O 53062,C1(NC(Cc2cnc(C)o2)=O)CCC(C)N(C(c2c(Br)nnn2C)=O)C1 53063,C(=O)(CCC(C)(C)F)NC1C(C)CN(C(=O)CCCOc2ccc(N)cc2)C1 53064,C1(CNC(c2n(C)cnc2)=O)CCC(F)(CNC(C2(C)CCCNC2=O)=O)CC1 53065,N1(C(C(CCC)C(C)C)=O)CCC2(CC1)COC(CNC(c1cscn1)=O)C2 53066,c1(OC)cc(C(=O)OC(C2CCOCC2)C)cc(F)c1F.N12CCSC(C1)C2=O 53067,CC(C)CCC(O)C(=O)NC1CCN(C(=O)C2=C(Cl)CC2)CC(O)C1 53068,N1(C(c2c(C)scc2)=O)CCCC2(NC(c3ccccc3[N+](=O)[O-])=O)CC2C1 53069,Cc1oc(Br)cc1C(N1CC(C)(NC(C2CC23CC(O)C3)=O)C1)=O 53070,N1(C(C=COCC)=O)CCOCC1CNC(c1ccnn1CC(F)F)=O 53071,Cc1c(F)ccc(-c2ccc(C(=O)NCc3ccncc3F)nc2)c1Cl 53072,c1(N(CC(C(F)(F)F)OCC)CC)cc(C)nc2c(F)cccc12 53073,C1(C(=O)N(C2CCCCC2)CCNC(C2(C3CC3)CCC2)=O)Cc2ccccc2S1 53074,N1(C(c2cn(C)nc2C(F)F)=O)CC2CCC(C1)N2C(=O)CC1CC1C(F)(F)F 53075,C1(C(N2CC(C(N)=O)(CNC(C3CC34CC4)=O)C2)=O)CC2CCC1C2 53076,CC1(C)CN(C(C2CCN(C(c3ccncn3)=O)C2)=O)CCO1 53077,Cc1coc(C)c1C(=O)NCc1csc(CNC(=O)CCN2CCCCC2)n1 53078,n1(CC)nc(C)cc1C(=O)NCC1CCC1NC(=O)CN1CCCCC1C 53079,CCC(O)C(C)C(=O)NCC(C)(C(C)C)NC(=O)Cc1ccc(Cl)cc1 53080,c1(CC)nccnc1CNC(=O)C(C(C)C)NC(C1CCCN1C(N)=O)=O 53081,Cc1cn2c(n1)C(C)CC(C(=O)NCC(CO)NC(c1ccc(CO)cn1)=O)C2 53082,N1(C(Cc2c(F)ccc(C)c2)=O)CC2CCC(C1)N2C(c1cc(C(N)=O)co1)=O 53083,c1(C(N2CCC(C)(NC(c3n(C)c(S)nc3)=O)C2)=O)nc2c(s1)COCC2 53084,C(=O)(CCC(F)(F)CN=[N+]=[N-])NC1CC(C)(CNC(C=CCOCCOC)=O)C1 53085,CC1(O)CCCN(C(C2CN(Cc3cccc(F)c3I)CCO2)=O)C1 53086,C(=O)(CC1CCCc2ccccc21)NC1CC(CNC(C2(C)CC=CCC2)=O)C1 53087,C(=O)(C1=COCCC1)NCCC1CCN(C(C(C(C)C)OCC(C)C)=O)C1 53088,N1(C(C(CC)=CCCC)=O)CC(NC(=O)CC(C)C2CCCC2)C(C)C1 53089,n1(CC(N2CC(SC)C(NC(=O)C(F)CCC(C)C)C2)=O)nc2c(n1)CCCC2 53090,CN1CCCC1(C)CNC(=O)Nc1nc(-c2ccncc2)cs1 53091,C12CC(N(c3ncc(Br)cn3)C1)C(=O)N2.c1(C(N)=O)ccccc1OCC(F)(F)F 53092,C(=O)(C1=CCCN(C(=O)Cc2ncccc2F)C1)NC(c1ccc(O)nc1)C 53093,C1(C(=O)NCC)CN(C(=O)C(c2ccn(C)n2)C)CC12CCC2 53094,c1(OC)cc(NC(=O)C(C)N(C(=O)CC(C)n2cccc2)C)ccc1F 53095,c1(CC(N2CC(CCCCNC(CSC)=O)OCC2)=O)cccc(Cl)c1Cl 53096,N1(C(CS(=O)(=O)NCC)=O)CCN(C(C2CC3CCCC(C2)C3)=O)C2(CC2)C1 53097,c1(N(CCCNC(=O)CC2=NNC(=O)C2)C(C)C)cnc2cc(F)c(F)cc2n1 53098,n1(C(C(=O)N)C)cc(CO)nn1.C(CCN(C)C(C)=O)SC 53099,C1(OCC)CCN(c2nnc(Cc3ccccc3Cl)n2CC2CCCOC2)CC1 53100,C#CCC(C)(C)C(=O)NC1COCCC1C(=O)NCC(CC)C(C)(F)F 53101,CC1=NN(C)C(=O)C1CC(=O)N(CC(=O)N(CC(=O)OC(N)=O)C)C1CC1 53102,C1(C(=O)NCC(C)NC(=O)CC2COCCO2)CCCCN1C 53103,N1(C(C2C(OCC)C2C)=O)CCC(NC(=O)COCCN(C)C)CC1 53104,C1(NCc2ccc(C(=O)O)cc2)CC2(C1)CC(C(=O)NCCSc1cccs1)C2 53105,c1(OC)ccc(C(N2CCN(C(=O)N(C)C)CC2)C(=O)NCCC(C)O)nc1 53106,C1(C(N(CCc2cn(C(C)(C)OC)nn2)C)=O)CCCC(=O)C1 53107,c1(NC(N)=O)cc(C(=O)NC2CCC2NC(=O)CCOC2CC2)ccc1F 53108,N1(C(C(CC)C#N)=O)CCCC2(CCN(C(=O)C(C)CCC(C)(C)C)C2)C1 53109,c1(NC(CC2CCN(C(COC(CC)C)=O)C2)=O)cc(C)cnc1O 53110,C1(CCC)CC(C(=O)NC2CN(C(=O)Cc3cnc(C(C)C)[nH]3)CC2C)CCO1 53111,CC#CCCC(=O)NC(CC1CCC1)C(=O)NCC(N1CCCCC1)C 53112,c1(C(=O)NCCOC2CN(c3ncnn4cccc34)C2)nnc2ccccc2n1 53113,N1(C(Cc2cc(C)[nH]n2)=O)CCCCC1CCNC(C1(CC(C)C)CCC1)=O 53114,Cc1cc2c(C(=O)NC3(CNC(=O)CC4CC4C)CCCC3)cccc2o1 53115,N1(C(c2ccc(-c3c(C)nc(C)s3)nn2)=O)CC=C(c2ccccc2)CC1 53116,C(=O)(C1=C(C)OCCC1)NC1C(NC(c2nc(OC)c(F)cn2)=O)CC(F)(F)C1 53117,c1(CNC(=O)CC2CCOCC2)cncc(NC(C2CCC(=O)N2C2CC2)=O)c1 53118,Cc1ccnc2sc(-c3nc(CC(C)(C)C)nn3CC3CCCO3)c(C)c12 53119,c1(CC)ccc(C(C)=O)cc1C(=O)NCC1(CO)CN(C(=O)CC2CC2)C1 53120,Cc1nnc(O)c(C(=O)NCC2C3CCCC2N(C(=O)Cc2ccco2)C3)c1C 53121,N1(C(Cc2c(C)nc(C)s2)=O)C2CCC1CC(NC(c1ccc([N+](=O)[O-])s1)=O)C2 53122,c1(NC)ccc(C(=O)NCC(C)(C(C)C)NC(=O)C(c2cccnc2)C)cc1 53123,C1(C(=O)NCC(C)(CO)CO)CCC(C)(C)N(C(C2CC3(CSC3)C2)=O)C1 53124,N1(C(C(C)OC(CC)=O)=O)CCCCC1C(c1cccc(C)n1)OCC 53125,Cc1cc(NC(C2CC(CCNC(c3[nH]ccc(=O)c3C)=O)C2)=O)ccc1F 53126,C1(NC(c2occ3c2CCCC3)=O)CCC12CCN(C(=O)CSC1CC1)CC2 53127,N1(C(c2c(C)cn(C)n2)=O)CCCC2(NC(c3cccc4c3CCC4)=O)CC2C1 53128,N1(C(C(=O)NC(C)(C)C)CC2CCC2)CCOCC1(C)C1CC1 53129,C1(C(C)C)CN(C(=O)CN2CC=CC2)CC1C(=O)N(C1CC12CC2)C(C)C 53130,c1(CC(=O)N(C2CCN(Cc3nc(C)no3)CC2)CC)nn(C)c2ccccc12 53131,C1(CC)(NC(c2nc(C)n(C)n2)=O)CCN(C(=O)CC(C)c2cccnc2)CC1 53132,C1(NC(C(C)CO)=O)CN(C(C2CC2c2ccc(O)cc2)=O)CC1F 53133,C1(CNC(C(C)N(C)CC2CCCO2)=O)CCN(C(=O)CCc2ccc[nH]2)C1 53134,C1(CCOC)(C(=O)N)CCN(C(c2ccc(CO)o2)=O)C1.c1(OC)csnc1OC 53135,c1(C(N(CCNC(c2c(C)nc(CCC)o2)=O)CCC)=O)cncc(Cl)c1C 53136,C(C(CC(=O)NCCSC)NC(=O)CC1CCC(C)(C)O1)OC 53137,N1(CC(=O)N(C2CCOC2=O)C2CC2)CCCC(C(F)(F)F)C1=O 53138,C(=O)(CCC(C)N(C)C)NCC=CC(=O)NCC1(COC)CCCO1 53139,c1(CN=C(NC2C(C)C2)NCC2(C)CCOCC2)ccc2c(c1)CC(C)O2 53140,C(=O)(CCP(C)(C)=O)N1CCC(N(CC#C)C(c2nc(C)oc2C)=O)C1 53141,CC1CCC2(CC2)N(C(c2cc(OC(F)(F)F)ccc2Cl)=O)C1 53142,C(C(=O)OC(C)(C)C)(C(=O)N1CC2CC2(CNC(=O)C2=CCCS2)C1)OC 53143,Cn1ccc(C(=O)NCCC2CCCN(C(C3(C)CCCC3O)=O)C2)cc1=O 53144,c1(C(C)(C(=O)NCC(CNC(=O)CCCC2CC2)CO)N(C)C)ccc(F)cc1 53145,N1(C(c2cc(N)c(Cl)cn2)=O)CCOC2CN(C(=O)CC3C=CCC3)CC12 53146,C(C(CC(F)(F)CNC(C1CCOCC1C)=O)OC)OC 53147,n1(CC)cc(C(=O)NC2CC(NC(c3cc(C4CC4C)on3)=O)C2)cn1 53148,N1(c2c(C)c(Nc3nn(C)cc3Cl)ncn2)CCC(S(=O)(=O)C(F)F)C1 53149,C1(C(=O)NCC2CCC(NC(c3cnc(Cl)s3)=O)CC2)CC2C=CC1C2 53150,N1(C(c2cc(-c3cccc(OC)c3)no2)=O)CC2ON=C(C(F)F)C2C1 53151,c1(C(=O)NC(C)(C)CCNC(c2cnc3[nH]cncc2-3)=O)ccc(Cl)c(F)c1F 53152,N1(C(C=CCCC)=O)CC2CC(C(N3CCC(CO)C(C)C3)=O)C(C2)C1 53153,Cc1ccccc1C=CC(=O)NC1CC2(C1)CC2NC(C1CCC(=O)N1C)=O 53154,N1(C(CC(CC)(C)C)=O)CC2CC(CNC(=O)C(C)(C)SC)CC1C2 53155,CCC(CC(=O)NC(C)(CNC(c1nc(C(F)(F)F)cn1C)=O)CO)C1CC1 53156,c1(C(CC)CC)ccccc1NC(=O)C(=O)NCc1ccn(C(F)(F)F)n1 53157,C(=O)(C(C(C)(C)C)OC)N1C(C(=O)NCCC(C=C)(C)C)CCC1 53158,Cc1cc2c(o1)S2.C1(CO)CC(C(F)(F)F)C1 53159,CCC(CC)NC(=O)CC1(NC(C2CC2C2CCCO2)=O)CC1 53160,C1(C(N(CC(C)NC(=O)CCCF)C)=O)CCC(CC2CCCC2)O1.C(CCOC)S 53161,C1(CN(C)CC2(C#N)CC2)CCCN(C)C1c1cccc(Cl)c1 53162,N1(C(C2CNC(=O)N2)=O)CC(NC(c2ccoc2Br)=O)C2(CCC2)C1 53163,c1(CN2C(C(=O)NC3CC(O)C3)C(O)CC2)c(Br)ccc2c1OCO2 53164,C1(CCOC)(C(=O)NC2CCC2(OC)OC)CCN(C(C2CCN(C)C2)=O)C1 53165,N1(C(C2C(NC(C3CCC(=O)N3)=O)CC=CC2)=O)CC2CC2C2CC12 53166,c1(C(=O)NCCCN(C)C(c2cnc3ccoc3c2)=O)cncc(P(C)(C)=O)c1 53167,C(C1=NOC2CCCC12)NC(C1(N(C(C(=O)NCCC(N)=O)=O)C)CC1)=O 53168,C1(O)(CNC(=O)C(O)c2ccco2)CCCOC1.C12CN(C1)C2=O 53169,c1(N2CCN(C)C(CNCC3CN(C4CCOCC4)C3)C2)cncc(C#N)n1 53170,c1(CNC(N2CC(C)(C#N)C2)=O)ccc(N=[N+]=[N-])cc1 53171,C(=O)(C1COc2ccccc21)NC(CNC(c1ncnc(OC)c1F)=O)C(C)C 53172,c1(C(=O)NCC2(NC(C(CC)F)=O)CCC2)ncn2ccc(C)cc12 53173,CCC(C)CCC(O)CC(=O)N1CCCCC1CNC(=O)Cc1cccnc1N 53174,C1(CNC(C2C(C(N)=O)C2)=O)C2CC1N(C(C1CCCC1F)=O)C2 53175,c1(C(=O)NC(C(C)NC(C(C)Sc2nncn2C)=O)C)nc2c(s1)COCC2 53176,C1(CNC(=O)CNC(=O)C2CC2)C2CN(C(=O)CC3(n4cncn4)CC3)CC12 53177,c1(C(N2C(CC)COCC2)=O)cc2sc(C(=O)OC)cc2[nH]1 53178,CCC(F)(F)CC(=O)NC(C)(CNC(c1ccc(C)cc1F)=O)C1CC1 53179,c1(C(=O)NCC(CNC(c2c(C)onc2O)=O)F)ccc(S(=O)(=O)C(F)F)cc1 53180,c1(C(C)(C)C)cc(Br)ccc1NC(C1CC1NC(=O)Nc1cccnc1O)=O 53181,C(=O)(CC(N)C(C)(O)C(F)(F)F)NC(c1c(OCC)cccc1Cl)C 53182,N#Cc1ccc(N2CCC(C(=O)Nc3cccc(NC(=O)CC4CC4)c3)C2)cn1 53183,c1(C(C)C)ocnc1C(N1CC(O)(CCNC(=O)CCOCC2CC2)C1)=O 53184,CC1(C#CC(=O)OC(C)(C)C)CN(OC(=O)NCC(c2ccccc2F)CO)C1 53185,c1(C(C(=O)NC2CCCCC2)N(CC(=O)OC)CC(C)C)cc(F)c(F)c(Cl)c1F 53186,N1(C(C2(C)CC(=C)C2)=O)CCCN(C(c2cnc(C(F)(F)F)nc2)=O)CC1C 53187,n1(CC)ccnc1C=CC(N1CCOC(CCNC(C2CCS2(=O)=O)=O)C1)=O 53188,C(=O)(C1=CC2C=CC(C1)C2)N(C)NC(CC(CCCC)CC1(O)CCCC1)=O 53189,c1(CCC)cc(C(=O)NC(C)CC(C)NC(=O)CC2COCC2O)no1 53190,N1(C(C(C)OCCOC)=O)CCCC(C)(NC(=O)CCc2cc(C)nc(C)c2)C1 53191,C1(CCNC(C)=O)CC(NC(C2CCN(c3ccc(C)cc3)CC2)=O)C1(C)C 53192,C1(NC(C(C=C)C)=O)CCCCC1NC(=O)CCc1cc(C)no1 53193,c1(NC(C2(C)CCCN(C(C34CC(C3)C4)=O)C2)=O)nc2c(s1)COCC2 53194,CC(C)CCC(F)C(=O)NC(CC1CCCC1)C(=O)NCC1CC(C)(O)C1 53195,c1(C(=O)NC(CNC(C2(C)CC2Br)=O)CO)cncc2sccc12 53196,O=C(N=c1cc[nH]c2cc[nH]c12)C1C=CC(NC(c2cnc3ccoc3c2)=O)C1 53197,N1(C(C2N(C(c3ccc(NC)cn3)=O)CCCC2)=O)CCC(C)C(C)C1 53198,c1(NC(C2C(NCc3nc(C)[nH]n3)C2)=O)c[nH]c2ccc(Cl)cc12 53199,c1(C(N(CC(C)NC(CC2(OC)CCC2)=O)C)=O)csc(Br)c1 53200,C1(CNC(C(c2cncnc2)C)=O)CC2CCC1N2C(c1ncccc1Cl)=O 53201,C(C(C)(C)CC(=O)NC(C)C(=O)NC1CCC1)NC(c1c(C)oc(Cl)n1)=O 53202,CCCC(C)(C)CC(=O)N1CCC(NC(=O)C(C)(C)CC(C)C)C(C)C1 53203,c1(C(=O)NCC2N(C(=O)C(C)(C)CC3CC3)CCN(C)C2)cc2c(o1)CCCC2 53204,C1(NC(c2cc(N)ncn2)=O)CC2(NC(C3CCCCN3C(N)=O)=O)COC1C2 53205,CON=C(C(=O)NC(CNC(=O)C(C)(C)SC)C1CC1)c1ccco1 53206,N1(C(C2CCCCN(C(CC3CC(OCC)C3)=O)C2)=O)CCC2(CC1)CC(O)C2 53207,c1(C(=O)NC2C(C)N(c3cncc(Cl)n3)CCC2)ccc2c(c1)ncn2C 53208,N1(C)CC(C)N(C(=O)CN(c2c(OC)cccc2)CC(C)C)C(C)C1 53209,c1(NC)cccc(C(N2CC(F)CC2CNC(c2cnn(C(C)C)c2)=O)=O)n1 53210,N1(C(c2c(CC)nc(C)o2)=O)CC(NC(=O)C(C(C)C)C2CCC2)CC(F)C1 53211,c1(-c2nnc3n2CCC2CN3CCO2)cc2cc(Cl)ccc2s1.C1(CSC)CC1 53212,c1(C(=O)NC(CN(C(CCCOCCC)=O)CC)C)cc(Cl)ccn1 53213,c1(C(CNC(C2(O)CCC2)=O)NC(C23CCC(CC2)C3)=O)cc(F)cc(Cl)c1 53214,N1(C(c2ccn(C(CC)CC)n2)=O)CCC(C(=O)OC)C12CC2 53215,C1(NC(C(CNC(C)=O)O)=O)CCCC(C(=O)NC2CS(=O)(=O)C2)CC1 53216,N1(C(C(C)CO)=O)CCC(CCC(=O)NC2(CCF)CC2)CC1 53217,c1(OC)ccc(CC(=O)NC(C)(C)CNC(c2cc(CN(C)C)on2)=O)c(C)c1 53218,c1(C(=O)NCC(CC)(C)NC(C2CC2F)=O)ccc(F)cc1OC 53219,C1(NC(c2cc(COC)oc2C)=O)CC(NC(C2C(C)(C)C2(C)C)=O)C12CCC2 53220,C=CC(C)C(=O)N(CCC(=O)NC(C1CCC1)C)C 53221,C1(C(=O)NCc2cn(C3CCN(C(CC)=O)CC3)nn2)CCS(=O)(=O)C1(C)C 53222,N1(C(C(C)(C)CC2CC2)=O)CCC2(CCN(C(c3csc(CO)n3)=O)C2)C1 53223,Cn1cc(S(C)(=O)=O)c(C(=O)NC2CCCC2NC(C2CC(F)C2)=O)n1 53224,Fc1cncc(NC(c2nc(Br)cs2)c2nnnn2C2CCCCC2)c1 53225,C(N=c1[nH]c(=NC2CCOCC2)[nH]c2c1CCC2)C1(S(C)(=O)=O)CC1CC1CC1 53226,C1(COC)CN(C(c2ncn(C)n2)C(=O)NCC(C)C)CC(C)O1 53227,C1(CNC(C2(N(C)C)CCC2)=O)CC2(CCC2)CN1C(=O)CCC1CC(F)(F)C1 53228,C12(NS(C)(=O)=O)CCCN(C1)C2.n12cc(cn1)C(c1nnnn1C)CC2.CO.CO 53229,C(=O)(C(C)P(C)(C)=O)N(CCNC(c1occc1Cn1cc(Br)nn1)=O)CC 53230,C1(C)(CNC(c2c(C)nsc2)=O)CCN(C(c2cc(C3CC3)ns2)=O)C1 53231,N1(C(C(C)c2ccsc2)=O)CCOCC1CCNC(c1cc(C2CC2)no1)=O 53232,C=CCC(C)(C)CC(=O)NC1CCCCN(C(c2cc(CCO)on2)=O)C1 53233,c12cc(cc(F)c1F)ONc1ccc-2s1.CCOC 53234,n1(CCOC)cc(Cl)c(C(N2CC(C(=O)Nc3cccc(F)c3)(OC)C2)=O)n1 53235,CC(C)CC(O)C(=O)NCCCOC1CCN(C(=O)CSC(F)F)C1 53236,c1(OC)ncnc(N2CCOC(C(C)NC(c3cnccn3)=O)C2)c1OC 53237,N1(C(C(C)(F)F)=O)CC2CCN(C(c3ccnc(C(C)(F)F)c3)=O)C(C2)C1 53238,C(=O)(C(C)(C)S(C)(=O)=O)NC1C(C)CCN(C(c2ccc(F)c(C(F)F)c2)=O)C1 53239,N1(C(=O)NC(C(C)C)C)c2ccc(Cl)cc2OCC1C 53240,N1(C(CC2(C=C)CN(C(=O)Cc3cccc(C)c3O)C2)=O)CC2CCCC2C1 53241,C12(C(=O)NCCC3(NC(c4cocn4)=O)CCCC3)COCC1CS(=O)(=O)C2 53242,C=CC(CCC)CC(=O)N(C)CC1CN(C(c2ccccc2)=O)CCO1 53243,CC1(NC(=O)C(c2cccc(F)c2)O)CCN(C(=O)CNc2ncccn2)C1 53244,C=CCC(C)(CC)C(=O)N1CCC(NC(c2ccnc(C(F)(F)F)n2)=O)CC1 53245,C1(C#N)(C(N2CC(NC(c3ccc(COC)[nH]3)=O)C(C)C2)=O)CCSCC1 53246,c1(C(N2CCC(CNC(=O)COCC3CCCO3)C2)=O)cccc2[nH]cc(Cl)c12 53247,C=CCC(C)(C)CC(=O)NC(CCF)C(=O)NC(CN(C)C)CC(C)C 53248,C1(C(N2CC(N(C)C)C2)=O)CC1C1CN(C(=O)CCC2CCCCO2)C1 53249,c1(C(=O)NCC(C)CNC(c2c(Cl)nsc2Cl)=O)cc2sccc2[nH]1 53250,N1(C(C(C)(C)CF)=O)CC(NC(=O)Cc2nc3ccccc3s2)C(C2CC2)C1 53251,C12(C(N3CCC(OCCN(C)C)CC3)=O)COCCC1C2(F)F 53252,C(=O)(C1OCCc2ccccc21)NC(CCN(C(c1c(COC)nn[nH]1)=O)C)C 53253,CC1(C#CC(=O)N2CC(OC3CCN(C(C4CN(CC(F)(F)F)C4)=O)CC3)C2)CC1 53254,C#CC1(C(=O)NCC(c2nncn2C)C)CCN(C(c2ccc(CC)cc2)=O)C1 53255,N1(C(CN(C2CC2)CC)=O)CC=CC(NC(c2cccc(C(F)(F)F)n2)=O)C1 53256,CCCCCCC(CNC(c1nc(C)cs1)c1nnnn1C(C)(C)CC)CC 53257,CN1CCN(C(=O)Cc2cncs2)C(C(=O)NCC2CN3CCC2CC3)C1 53258,c1(OCC)cc(C(N2CCC(O)C2C)C(=O)NCc2ccccc2)ncn1 53259,c1(C(N(C2CN(C(=O)CCc3ccc(O)c(Cl)c3)C2)C)=O)n[nH]c2c1CC1CC21 53260,C1(NC(=O)CNC(=O)OC(C)(C)C)CN(C(C2CC(=C)C2)=O)CC2CCCC12 53261,c1(C(=O)NCCN(C(C2CC(O)CN2C(N)=O)=O)CC)cc2cc(Cl)ccn2n1 53262,N1(C(C(c2ccc(F)cc2)C)=O)CC2(CC(NC(c3cccc(O)n3)=O)CO2)C1 53263,c1(CNC(c2nnc(C)n2C)c2n(CCOC)nnn2)cccc(Br)c1 53264,C(=O)(C(CCC(C)C)NC(=O)C(=O)NCC)NC1C(CC=C)COC1 53265,C1(NC(C2OCCN(C)C2)=O)CCCC12CN(C(=O)C=Cc1ccccc1F)C2 53266,Cc1cncc(C(=O)NC2C=CCN(C(C3(CS(N)(=O)=O)COC3)=O)C2)c1 53267,C(C(C(F)(F)F)N1CCCCC1)NC(=O)N(C1CCCCC1)CCO 53268,N1(C(C2C(C(C)C)C2)=O)CCC(C(N2CCC(F)(C#N)C2)=O)C(C)(C)C1 53269,c1(C(=O)NCCCCn2cc(CCOCC(N)=O)nn2)cc(Br)sc1Cl 53270,Cc1cccc(C)c1C(N1CC(CCn2cc(C3CC3COC)nn2)C1)=O 53271,NC1CN(c2nc(CSc3ccc(Br)cc3)co2)CC1C(F)F 53272,C1(C(=O)NC2CCN(C(CCCC)=O)C23CC3)CCn2nccc2C1 53273,C1(C(=O)NCC2CN(C(C3CCC(C)S3)=O)C2)(OC)CCC(F)(F)CC1 53274,c1(C(N2C(C(=O)NCc3cnc(C)nc3)CC3CC32)=O)ccc(Cl)c(Br)c1 53275,c1(NC(C2C(NCCNC(C)=O)CCO2)=O)ccccc1OC(F)F 53276,CC(C)C#CC(=O)N1CCC(O)(N(C(=O)C(C(=O)OC(C)(C)C)OC)C)C1 53277,C1(C(N2CCC(NC(CCCCCC)=O)C(O)C2)=O)CCc2cnn(C)c2C1 53278,Cc1[nH]c2ccccc2c1C(N1CC(C)CN(C(=O)CCOC(C)C)C(C)C1)=O 53279,c1(C(N(CCCNC(C2(n3nccn3)CC2)=O)CCC)=O)ccc[nH]1 53280,C(C(F)(F)C(=O)NC(C)CC1CN(C(=O)Cc2cccc(Cl)c2)C1)OC 53281,CN=c1[nH]nc(CC(=O)NC(C2(O)CCN(C(c3cocc3Br)=O)C2)C)s1 53282,C1(C(=O)NCC(C2CC2)OC(C)=O)CC(C)CCN1C(=O)C(C)SCC1CCC1 53283,N1(C(c2c(C)n(C)cc2)=O)CCN(C(=O)CNC(=O)CN(C)C)CCC1C 53284,c1(CN2C(C(=O)NCC3N(CC)CCC3)CSCC2)c(Cl)ccc(F)c1F 53285,C(=O)(C(C)(C)S(=O)(=O)C1CC1)NCCN(C(c1cccc(C(C)C)c1)=O)C1CC1 53286,N1(C(C(C)SCCCC)=O)CC2(CCCC2)C1C(=O)NC1CCCC1 53287,N1(C(C(C)O)=O)CCC2CCC(NC(c3ccn(C(F)F)n3)=O)C12 53288,C1=CC(=O)Nc2c(N)ccc1c2.C1(CC=C)C(OC(C)C)CC1OC 53289,n1(CCC(=O)NC(CN(C(C(C)OCCCCCC)=O)CC)CC)cccnc1=O 53290,c1(C(=O)NCC(C)(C2CCC2)NC(c2ccc(OC)s2)=O)nn(C)c(C)c1Cl 53291,N1(C(=O)C(O)C(F)F)CCC2(CCCN2C(C2(Cc3cnn[nH]3)CCCC2)=O)C1 53292,c1(C(=O)NC(CC)(C)CNC(=O)C=CCF)cc2c(cn1)NC(=O)CO2 53293,N1(C(CN(S(C)(=O)=O)C)=O)CC(C(C)(C)O)(CNC(=O)Cc2cc[nH]c2)C1 53294,c1(CCC(=O)NC(CC)(C)CNC(=O)Cc2c(C)noc2C)n[nH]c2ccccc12 53295,C1(O)(C(=O)NCC(CNC(CC(=O)NCC)=O)S(C)(=O)=O)CCCC(C)CC1 53296,C1(O)(C(C)NC(=O)CC2CCOCC2)CCN(C(=O)CCc2cc[nH]n2)C1 53297,CN1CCOC(NC(=NCC2CC2)NCCN2CCOC(c3cccs3)C2)C1 53298,CC#CCC(C(=O)NCC1CC1(F)F)NC(c1c[nH]c(C)c1)=O 53299,C1(C(N(C2CCN(C(=O)C(C)N3CC(C)C3)CC2)CC)=O)CCC(F)CC1 53300,c1(C(=O)NC2CCN(C(=O)C3=CCCC3)C(C3CC3)C2)ccn2cccc2c1 53301,N1(C(C(CN(C)C)N(C)C)=O)CC2CCC(C(=O)Nc3cncnc3O)(C2)C1 53302,c1(CC)c(C(=O)NCC(C)NC(=O)COCCSC)cnn1-c1ccc(F)cc1 53303,N1(C(C(CC(C)C)F)=O)CCc2sccc2C1CNC(=O)CC(C)(C)CC(F)F 53304,N1(C(c2c(C)ocn2)=O)CC2CCOCC2(NC(=O)C(=Cc2cccnc2)F)C1 53305,CC(C(=O)NOCC(N1CC(C(N)=O)(N(C)C)C1)=O)NC=O 53306,C(=O)(C(C)(O)C(F)(F)F)N(C)CCOC(C)(C)C.C12(CC1)C(=O)NCCCS2 53307,Cc1ncc2c(n1)CCC(C(=O)NC1C=CCN(C(=O)C#CC3(C)COC3)C1)C2 53308,N1(C(c2cc(C3CCOCC3)[nH]n2)=O)CC2OCCN(C(C3CCOC3)=O)C2C1 53309,C1(=O)CCN1CCO.C12CN(C1)C(=O)C(C)N2.C1(OCC)CCCC1 53310,c1(CC)nocc1C(=O)NCCN(C(=O)C(C)COC)C 53311,C(=O)(CC(C)(O)CCC)N(C1C(C)CCN(C(C(C=C)c2ccccc2)=O)C1)C 53312,c1(C(=O)NCC(CC)(C)NC(C2(COC)CCOC2)=O)cccnc1C 53313,N1(C(c2cn(CCF)nn2)=O)CCCCC(C2CN(C(C3CCCOC3)=O)C2)C1 53314,N1(C(CCCC=C)=O)CCC(CO)C(NC(c2ccc(Br)c(C)c2)=O)C1 53315,c1(C(=O)NC2CC(F)(CNC(C(CC=C)CC)=O)C2)cc2nn[nH]c2cc1F 53316,Cc1ccc2c(c1)CCN(Cc1cc3cc(Cl)ncc3o1)C2 53317,c1(C(N2C(CNC(CC3(OCC)CC3)=O)CCC2)=O)nc(C(F)(F)F)sc1C 53318,N1(CCNc2scc(-c3ccc(Br)cc3)n2)CCC2CCCC(C1)N2 53319,N1(C(c2ccc(SC)s2)=O)CC(NS(=O)(=O)CCSC)C(C)C1 53320,c1(CC)[nH]nc(Cl)c1C(=O)NC1CC2C(NC(c3ncsc3C)=O)C2C1 53321,N1(C(CN(C(C)C)C)=O)CC(CNC(c2ncc[nH]c2=O)=O)C2(CC2)C1 53322,Cc1cc(CC(c2ccccc2C#N)=O)cc(C)c1Br.C1(=O)C(C)O1 53323,C(=O)(CCCC(=O)NCC1CCC(C(=O)NCCC(F)F)O1)OCC 53324,c1(C(=O)NC(CNC(C=C(CCC)C)=O)CO)ccc(C(F)(F)F)c(Cl)c1 53325,c1(C(=O)NCC2N(C(C(CSC)C)=O)CCCC2)c(OC)ccc([N+](=O)[O-])c1N 53326,c1(NC(CCNC(CC(C)CN(C)C)=O)(C)C)ncnc2ccc(Cl)cc12 53327,C#Cc1cc(F)c(C(=O)NC2CC2CNC(C2CCC(C)(C)CC2)=O)c(F)c1 53328,c1(C(=O)NC2C(NC(C=CC(C)(C)SC)=O)CCCC2)ncc(Br)cc1N 53329,Cc1ccc(-c2ccc(CNC(=O)CCCNn3nnc(-c4ccsc4)n3)s2)s1 53330,CCCC(C#N)C(=O)N1CC(C)(C)CC1C(=O)NC(c1n[nH]c(CC)n1)C 53331,c1(OCOC)cc2ccc1-2.c1(CC(N2CC(NC(=O)OC)C2)=O)cc(Cl)ccc1I 53332,c1(C(N2CCCC(C)C2CNC(=O)C(C)C2CCCO2)=O)cncc2[nH]ccc12 53333,c1(C(=O)NCC2CCCN2C(=O)CSc2nc[nH]n2)cccc(-c2nccs2)c1 53334,c1(C(C(=O)NC(CC)CN(C(=O)CC(C)(C)O)C)O)cc(Cl)cc(Cl)c1 53335,N1(C(CCCC2C(C)C2)=O)CCC(C)(C)C(CNc2cc(O)ccc2C(=O)O)C1 53336,C1(CC(=O)NCCCC2CCC2)CCN(C(=O)CC2CCOCC2)CC1 53337,C(CC(CC)C(=O)NCC1(CCNC(=O)C(C)N2CCCC2)CC1)=CC 53338,c1(CNCC2N(C(c3nc(Br)cs3)=O)CCOC2)ccc(F)c(O)c1 53339,C(=O)(CCCCCCC(=O)N1CCN(Cc2c(O)cccc2Br)C2CC12)OC 53340,Cc1cc(C(F)(F)F)cc(S(=O)(=O)NC(=O)CNCc2cc3ccccc3nn2)n1 53341,C1(=O)C(C(C)C)N1.C1(CCOC)CCN1C(=O)Cc1cnoc1 53342,N1(C(C(=O)N(C(CNC(C(OC)OC)=O)C)C)C2CCC2)CC(=O)N1 53343,Cc1nc([N+](=O)[O-])cn1CC(N1CC(OCCNC(c2cnn(C)c2F)=O)C1)=O 53344,C1(CCOC)(C(=O)Nc2cncnc2C)CCN(C(=O)C(C(C)C)SC)C1 53345,C(=O)(CS(=O)c1ccc(Cl)cc1)NCC(C1CC1)NC(=O)Cc1cnsc1 53346,c1(-n2c(C)cnn2)ccc(C(=O)NCC2CN(C(=O)C(O)c3ccsc3)C2)cc1 53347,C(=O)(N=c1[nH]onc1C1CC1)NCc1cn(C(=O)OC(C)(C)C)cc(Cl)c1=O 53348,C(N=c1[nH]c(=NCCCN(C)C2CC2)[nH]c2c1COCC2)C1CC(C)OC(C)C1 53349,CC12CN(C(N3CCC(O)C(F)C3)=O)C(C(=O)N(C)C)(C1)C2c1ccccc1OC 53350,c1(OC)cncc(C(N2CCCC2CCNC(C2(C)CC3CC3C2)=O)=O)c1 53351,CC1(CNC(C2(F)CCCC2)=O)CCCN1C(C1CCCCO1)=O 53352,CS(=O)(=O)c1cc(OC(F)F)ccc1NS(=O)(=O)C1CC1F 53353,N1(C(C(CC)C2CCOCC2)=O)CCN(c2ncc(F)cn2)CC1C 53354,C1(C(=O)OC)(NCc2nnc(C(=O)OC)s2)CC1(C)C 53355,C(=O)(C1=Cc2ccccc2OC1)N1CC(NC(CC(C)(F)F)=O)C2(CC1)CCC2 53356,C(=O)(CC(C)C(C)C)NC1CC(CCNC(c2c(C)noc2C(F)(F)F)=O)C1 53357,C1(=O)CC(O)CNCCO1.c1(OC(C)(C)C)cc(Br)no1 53358,C1(NC(C=C(CSC)C)=O)CCC(CC(=O)NC(CO)CCO)C1 53359,N1(C(C(CCC)O)=O)CC(NC(c2cc3sccc3s2)=O)C(C#N)C1 53360,c1(NC2C(C)NC(=O)C2)ncc(F)cc1F.N1(CC)CC(=O)NC(C(C)C)C1 53361,C1(NC(Cc2c(C)con2)=O)CCCCC1NC(=O)C(C)(C)c1cc[nH]n1 53362,N1(C(C2C(CC)C2)=O)CCCCC1CCCNC(=O)Cc1cncn1C1CC1 53363,N1(C(c2c(C)nc(O)nc2C)=O)CCC2(CC1)CN(C(=O)CC13CCCC1C3)C2 53364,c1(C(=O)NC2C(NC(C3C(C(C)C)CCO3)=O)C2)ccccc1[N+](=O)[O-] 53365,c1(C(N(C2CCCC(NC(c3ccc(C)s3)=O)C2)C)=O)cc(C)c(C#N)cn1 53366,c1(C(C(=O)N(C2CC(=C3CCC3)C2)CCC(C)Cc2cn[nH]c2)O)cccnc1 53367,C(=O)(C#CC1CCCCC1)NCCC1N(C(c2c(CC)cco2)=O)CCCC1C 53368,N1(C(C(C)Cc2ccco2)=O)CC(C(N2CCS(=O)CC2)=O)CC(F)(F)C1 53369,N1(C(c2n[nH]c(CC)c2Cl)=O)CC2(CCCC(CNC(c3oncc3C)=O)O2)C1 53370,C1(CNC(C=Cc2cc(OC)ns2)=O)CC2CC(C1)N(C(=O)CC(C)C)C2 53371,C1(CC)CN(C(=O)C(C)(C)COCC(F)F)CCN1C(C1CCCSC1)=O 53372,N1(C(CC(C=C)C)=O)CC2(C1)CN(C(c1[nH]nnc1CC1CC1)=O)CC2CO 53373,CC(C)CC(C)(CNC(=O)CN(C)C(=O)C1CC1)NC(c1cnc(O)nc1O)=O 53374,c1(C(=O)NC(C(=O)OC)Cc2cn(C)cn2)cnn2c(Br)cccc12 53375,C(=O)(C(C)C(O)CCCC)NCCCCCC(=O)N1C(CCCCC#C)CCC1 53376,N1(C(c2cc(Cl)cc(Br)c2F)=O)CCCC2(CCCO2)C1 53377,Cc1cc(C(=O)N(C)CC=CC(N2CCCCC2CCO)=O)cc(O)c1 53378,C1(NC(c2c(C)sc(-c3ccco3)n2)=O)CCN(C(C2CCC2)=O)C(C2CC2)C1 53379,c1(CC(=O)NC(C)CC2CCN(c3ccnc(C#N)n3)CC2)cc(Cl)ccc1Cl 53380,Cn1cncc(C(=O)NCC2(O)CCC2C(=O)NC2COC3(CCC3)C2)c1=O 53381,N1(C(C2(SCC)CC2)=O)CC2CN(C(=O)CC(CC)C(F)(F)C(F)(F)F)CCC12 53382,C(=O)(CC1=CCCCC1)N1C2C(N(C(C(C)c3ccsc3)=O)C)CC(C2)C1 53383,CCCS(=O)(=O)C(C)C(=O)N(C1CN(C(c2cnc3cccnn23)=O)CC1O)C 53384,c1(OC)ccc2c(c1C(=O)NCCN(C(=O)C1=CCCSC1)C1CC1)CCC2 53385,c1(C(=O)NCC2(OC)CN(C(c3ccc([N+](=O)[O-])s3)=O)C2)cc(F)cc(Cl)c1N 53386,N1(c2c3cccc(OC)c3ncn2)CCCC2(CCCCC2O)C1 53387,c1(C(=O)NCCN(C(=O)CCn2ccnn2)C)ccc2cc(F)c(F)cc2n1 53388,C1(CNC(=O)Cc2cc(Cl)cs2)CCCC2(CN(C(C3CC4CC4C3)=O)C2)O1 53389,C1(c2cn(-c3cccc(OC)c3)nn2)CN(C(=O)CCOC2COC2)CC12CC2 53390,c1(C(=O)NC(CCC2CC2)C(=O)NC2CC(Cl)(Cl)C2)ccc2nccn2c1 53391,c1(C(=O)NC2C(CC)N(C(=O)Cc3nc[nH]n3)CC2)cnn2c(C)cccc12 53392,c1(C(=O)N(C2CC2)Cc2nncs2)oc(C(F)F)nc1-c1ccccc1 53393,c1(C(=O)NC2CCC(C(C)NC(c3cnc(Cl)nc3)=O)CC2)ccc(I)cc1Cl 53394,C(=O)(CCCC(F)F)NCCCN1CCC(CNC(c2ccc(C(N)=O)[nH]2)=O)C1 53395,C(CCCCC(=O)O)NCc1c(C)non1.N12CCC(C1)C2 53396,c1(C(=O)NC2CC3(C(NC(c4c(C)onc4)=O)C3)C2)ccn2ncc(C)c2n1 53397,C1(C2CN(C(COC3(C)CC(=C)C3)=O)C2)CN(C(=O)CC(C)(F)F)CCO1 53398,C1(C(=O)NC(C)CCN(C(=O)CSc2nc[nH]n2)C)CC1[N+](=O)[O-] 53399,C1(C(=O)NCCc2ccccn2)C2Cc3ccc(Cl)cc3C12 53400,C(=O)(C(F)(F)CC=C)N1CCC(CN(C(CC2C(C(=O)OCC)CC2)=O)C)CC1 53401,N1(C(C2C(CC)C2)=O)CCCN(C(c2c(OC)cccc2F)=O)C(C)C1 53402,O1C2CCc3ccc(cc32)C1=O.c1(C(C)(C)C)cccc(OC(F)(F)F)c1Br 53403,N1(C(C2(C)CC2(Cl)Cl)=O)CC2C3CCC(C2C1)N(C(=O)CCN1CCOCC1)C3 53404,N1(C(C=CC=CCC)=O)CC(N=[N+]=[N-])CC1C(=O)NC1CCC(CCO)CC1 53405,Cn1[nH]c(C2CCNCC2)nc1=NC(=O)NCc1nnc(CCO)s1 53406,C1(CN2CCC3CC23)CC2CCC1N(C(c1cnc3ncccn13)C)C2.O=C1CN1 53407,C1(OC)CC(NC(=O)Cn2ccc([N+](=O)[O-])n2)C12CCN(C(=O)C=C(C)Cl)CC2 53408,c1(OCC(N2CC(NC(C(COC)(C)C)=O)C(F)C2)=O)cc(Cl)ccc1Cl 53409,C1(NC(c2ccc(F)nc2)=O)CCOC(CNC(c2c[nH]nc2Br)=O)C1 53410,C(CCCC(C)(C)C)NC(c1n(CC)nnn1)CC1CCOC1 53411,Cc1cc(C#N)ccc1C(N1CCC(C(=O)NCCS(C)(=O)=O)C(O)C1)=O 53412,N1(C(c2cncc(C)n2)=O)CCCC(CO)(NC(=O)CC2CCCN2C2CC2)C1 53413,Nc1c(C(N2CC(CNC(c3cc[nH]n3)=O)C3CC23)=O)cnn1-c1ccccc1 53414,C(C(O)C(=O)N(C)CC1CCCN1C(c1cc(C(C)(C)C)on1)=O)SC 53415,N1(C(C2C(OC)C2)=O)CCC(C2CC2C(=O)NC2(CC(C)(C)C)CC2)CC1 53416,N1(C(C=CC=C)=O)CC(N(C)C)C(NC(=O)CS(=O)(=O)N(C)CC)C1 53417,C1(c2cn(CCOC)nc2)CN(C(c2ccc(-c3ccncc3)o2)=O)CC1C 53418,c1(C(N2C(C(C)(C)NC(C(CCC)C)=O)CCC2)=O)cc(S(N)(=O)=O)ccc1F 53419,c1(N)cc(C(N2CC(CNC(C3(C4CC4)CCC3)=O)C2)=O)ccn1.CC(C1CC1)=CC 53420,C1(NC(CC=C=C)=O)CCC(C)N(C(=O)CCC=CC)C1 53421,N1(C(c2n(CCC)ccc2)=O)CC(C(=O)NC2(C(=O)NC)CC2)CC(C)C1 53422,C1(NCCNC(CCCOCC#N)=O)CCCN(NS(C)(=O)=O)C1 53423,C(=O)(C1=CCCOCC1)N1CC(O)(CCCOC(=O)C=CC(=O)NCCCC)C1 53424,C1(C)(COC)CC(NC(=O)CCc2ccco2)CN1C(=O)CC(C)(F)F 53425,C(C(CCCC)NC(=O)CC=CC)NC(C(C=C)O)=O 53426,S(=O)(=O)(CC(=O)NC1(C(=O)NCCC2CCCO2)CCSC1)NC 53427,c1(C)cnn2c1CN(C(=O)CC(F)(F)F)CC2.CNC(CN1CCC(C)(O)C1)=O 53428,N1(C(C2C(OCC)C2C)=O)CC2(CCN(C(C3CC4(C)CC3CO4)=O)C2)C1 53429,CCCCC(C(=O)NCCC1(C(C)(C)O)CC1)N(C)C.C12(CC1)C(=O)NC2 53430,Cc1cc(C(=O)NC2CC(NC(=O)C(C)Sc3ccc(Cl)cc3)C2)c(C)s1 53431,C(=O)(C(F)C(=O)NCC)OCC.C(C)(CCCC)NC(=O)C(C)(C)n1cnc(C)c1 53432,c1(C(=O)NC(C)CNC(c2ncccn2)=O)sc2cccc(F)c2c1Cl 53433,c1(N2CCN(C(C3(C4CC4)CC3)=O)CC2)nc2ccccc2[nH]1 53434,N1(C(Cc2nc(C)[nH]n2)=O)CCC2(CNC(c3ccccc3F)=O)CCCCC12 53435,Cc1ccc2ccnc(NC(c3ncoc3C3CCC3)c3nnnn3C(C)C)c2c1 53436,CON=Cc1ccc(C(=O)N(C(C)CCNC(c2cncc(Cl)c2)=O)C)cc1 53437,c1(CN2CCCC(NC(C(C)CC3CCCCC3)=O)CC2)ccc2c[nH]nc2c1 53438,N1(C(C(CC)NC(C2C(C)C2C)=O)=O)CCC(CC)C1CC 53439,C(=O)(C(O)C1=CCCCC1)NC1CN(C(CC(CCCCC)O)=O)C(C)C1 53440,C1(C(N2CC(C)(NC(CCC(=O)NC)=O)C2)=O)CCC(=O)C(C)C1(C)C 53441,c1(C(N(CCCN(C(C(C)n2ccnn2)=O)C)C)=O)cc(S(N)(=O)=O)sc1Cl 53442,C12(CNC(CC)=O)CCCC(CN1C(=O)C(O)CN1CCCC1)C2 53443,C1(C(N2C(CC(=O)NCCC(C)(C)N(C)C)CCCC2)=O)CCCCCN1C 53444,N1(C(C(C=C)O)=O)CC(C(=O)NCC(C)N(C)C2CC2)C(C)(C)C1.C(=O)NC 53445,C1(NC(c2ccc(F)cc2)=O)C2COCC1CC(NC(c1cnsn1)=O)C2 53446,c1(CCNC(CN(CCCCCC)CC(=O)NCc2ccccc2)=O)cccc(C)n1 53447,C1(CC)(NC(C2COCCO2)=O)CCN(C(C2CN(CC3CC3)CCO2)=O)CC1 53448,CC(C)CC(CNC(C1CCN(C2CCCCC2)C1)=O)NC(N1CCCC1)=O 53449,C1(CNC(C2(C)CC(=C)C2)=O)CCCN(C(c2ccnn2CCC)=O)C1 53450,N(C(=NCCSc1ncccc1N(C)C)NCC1CCCO1)Cc1ccc(Br)o1 53451,N1(C(c2cc(C)n(C)n2)=O)CCCN(CCNC(C2CC2CF)=O)CC1 53452,CC1(CCCCNC(=O)NC2CCCC2C2CC2)NC(=O)NC1=O 53453,c1(C(C(=O)NC(CNC(c2c[nH]c(=NC)s2)=O)C)C)cccc([N+](=O)[O-])c1 53454,C12(C(N3CC(NC(CCc4ccc(CC)cc4)=O)C3)=O)CC(C)(C1)OC2(C)C 53455,C1(OCC)CC2(C1)CC2C(=O)NCC1(O)CN(C(C2CC23CCCC3)=O)C1 53456,C1(NC(Cc2nnc(C)s2)=O)CCC12CN(C(C1CCCN1CCC(C)C)=O)C2 53457,C(=O)(C(F)CC(C)(C)C)N1CCCC(N(C(C=CCCC)=O)C)CC1 53458,N1(C(C(c2ccc(OC)cc2)C)=O)CC2CC(C)N(C(=O)CSC(C)(C)C)C2C1 53459,N1(CCNC(C(=O)N(CCNC)C)=O)CCN(c2ccccc2)CC1 53460,c1(CCC)cc(C(=O)N(CCNC(=O)C(C)SC)CC2CC2)no1 53461,C1(CCC)CCCCN1C(=O)CC=CC(=O)OCC.C1(=O)CC2(CC2)CN1 53462,c1(SC)ccc(NC(C23CC2CN(C(C2(C4CC4)CC2)=O)C3)=O)c(F)c1 53463,CC1c2ccccc2CC1NC(=O)NCc1cn(-c2cccc(Cl)c2N)nn1 53464,Cc1cc(C)c(OCC(N2CCCC2CCNC(=O)C(F)(F)C(C)O)=O)c(C)c1 53465,Cc1nncc(C(N2CC(CC(=O)NCCC3=CCCCC3)C2)=O)c1C 53466,N1(C(CC(C)n2ccnc2)=O)CC(C(=O)N(C2CC3CCC2CC3)C)C2(CC2)C1 53467,c1(C(=O)NCCC2OCCN(C(C3(C=C)CCC3)=O)C2)cc2nccnc2[nH]1 53468,CCC(CC(=O)NCC12CC1CN(C(=O)CCCC1CCCO1)C2)c1ccco1 53469,C(=O)(C(C)CC(C)(C)C)NC(C(=O)NCC1=CCCC(C)C1)CN(C)C 53470,N1(C(c2cc3n(c2)CCSC3)=O)CCC2CN(C(=O)C3=CCOC3)CC2C1 53471,c1(CC(N2CCC(c3cn(C4(C)CC4)nn3)C2)=O)cn2cc(F)ccc2n1 53472,C(CCCC(=O)OC)(c1nnnn1C)NC(C(c1nnc(CC)s1)(F)F)=O 53473,C(CC(C(C)(C)C)NC(=O)Cc1nc([N+](=O)[O-])n[nH]1)N(C)C(C1CCSC1)=O 53474,CC1(C)CC=CCN(C(C2(NC(=O)CC3(C#N)CC3)CCCC2)=O)C1 53475,C12(NC(c3cc(C)sc3C)=O)CCCC1CN(C(=O)CC1CC3CC3C1)C2 53476,C(c1cncn1C)=CC(N1CC(CCO)(NC(c2c(C)n[nH]c2)=O)C1)=O 53477,C1(CONC(=O)Nc2cnsc2)CCCCO1 53478,c1(C(C(=O)NCCCCCNC(=O)CSC(C)(C)C)N(C)C)ccccc1Cl 53479,Cc1ccc2c(c1)C(NC(=O)C(=O)NCCSCC(F)(F)F)CO2 53480,c1(OC)cccc2cc(C(C)NC(c3ccc(F)c(C)c3)CO)oc12 53481,C1(C2CC2)(CNC(CC2CCC(C)(C)O2)=O)CCN(C(=O)C(Cl)=CCl)C1 53482,C(C1=NOC2CN(C(c3cnn[nH]3)=O)CC12)NC(c1ccc(C(C)(C)C)cn1)=O 53483,C(=O)(CC(C)C(C)C)NCCC1(C(=O)NCCCC(=O)OC)CCCC1 53484,CCC(C(=O)OC)C(=O)N1CC(C)(NC(C2CC(F)CN2C)=O)C1 53485,c1(CNCC(C)CC2CCCCC2)cnn(CCF)c1 53486,CC1(CNC(C2CC2C(C)NC(=O)CNC(C2CCC2)=O)=O)CC2(CC2)C1 53487,C1(NC(=O)Cc2csc3nccn23)CC(C2CCN(C(c3cn[nH]c3)=O)C2)C1 53488,c1(NC(c2ccccc2)(C)Br)nccc(N2CCOC(c3cccc(F)c3)C2)n1 53489,N1(C(CS(N2CCN(C)CC2)(=O)=O)=O)CCCC2C1CCN2C(C1CCOC1)=O 53490,n1(CC)cccc1C(=O)N(CC(=O)NC1(CC)CC1)C(C)C 53491,C1(C(N(C(CC(C)C)C(=O)NCCN2CC(C)(O)C2)C)=O)CC(=O)CC12CCC2 53492,c1(N)ccc(OC(F)F)cc1.C12CCC1CC(=O)NC(CO)CNC2=O.CCS 53493,C12COC3(C1)CN(C3)C2=O.c1(NC(C(N2CCC(C)C2)=O)=O)ccc(C#N)[nH]1 53494,C(=O)(C1=CC2C=CC1C2)NCC#CCNC(c1c(O)ccc(C)c1)=O 53495,C1(NC(C(C)n2ccnc2)=O)CCCC12CN(C(=O)C1CC1)C2 53496,N1(C(CSCCC)=O)CCOCC(CNC(C2(C#N)CC2(C)C)=O)C1 53497,C(CCF)(C(=O)NCC1(F)CC1)NC(CC1CC(OCC)C1)=O 53498,C1(C(N2CC(O)(c3nn[nH]n3)C2)=O)CN(C(C2(F)CCCCC2)=O)C2(CC2)C1 53499,c1(CC)cc2c(CC(=O)NC3CC(CCNC(C4CCOCC4)=O)C3)csc2s1 53500,N1(C(C2(C#N)CC(=O)C2)=O)CCC(C2(NC(C3CC3C3CCCC3)=O)CC2)CC1 53501,C1(C(=O)NC(CCOCC)C)CCCN(CC(=O)NC(c2cccc(C)c2)C)C1 53502,c1(CC)cc(Br)c(C(c2nnnn2C2CCCCC2)NCC2CC(O)C2)s1 53503,c1(CC)ccc(C(=O)NCCN(C)C(C2(COC)CCOCC2)=O)cc1N 53504,CCCC(C)CC(=O)N(CCNC(C1CCCCC1(F)F)=O)CCOCCO 53505,N1(C(C2C3CC2N(S(=O)(=O)Cc2c(F)cccc2Cl)C3)=O)CCC2(CCCO2)C1 53506,N1(C(c2cncc(F)c2)C)CC2CC1CN2C(C1CCC1)=O 53507,C(CC(N)CC(=O)O)NC(=O)Nc1cccc(CSc2onc(CC)n2)c1 53508,C1(NC(c2ncn(C(C)(C)C)n2)=O)CCCN(C(c2cnc(C(F)F)cn2)=O)C1 53509,C(CCC(=O)NC1CCC(CCNC(=O)C(C)(C)c2cccnc2)C1)OCCC 53510,c1(CC)ccc(C(=O)N(CCNC(c2ccc(C)o2)=O)CC2CC2)c(F)c1 53511,C1(CN(C(=O)Cc2csc(SC)n2)CC)CCCN(C(=O)CN2CC(C)(C)C2)C1 53512,CCC1=NOC(C(=O)NCCCCC(C)NC(c2cc(C(C)C)no2)=O)C1 53513,CCCN=C(NCC(CC)C(C)C)NCc1ccc(F)cc1.O1NC(=O)C1 53514,CC1CCN(C(=O)CN)CCN1C1C2CCC1(c1cncs1)C2 53515,C(C(=O)NNC(=O)CCCN)N(c1cc(C)cc(C)c1)C(=O)Cc1ccccn1 53516,C1(C(=O)NCCC(CNC(c2cnc(CC)[nH]2)=O)O)CCC(F)(F)CO1 53517,N1(C(c2nccc(C)n2)=O)CCN(C(C2CCC(C)(F)CC2)=O)CC(C)(F)C1 53518,c1(C(=O)NC(CCOC)CNC(=O)C(C)SC(C)C)ccc(OC)c(Br)n1 53519,CCC(CC)C(C)N=c1nc(N2CC3C(=O)NC(=O)C3C2)c2ncccc2[nH]1 53520,c1(C(=O)NCCC2CCN(C(c3ccc(CC)o3)=O)C2)cncc2ncn(C)c12 53521,C1(NC(CSC(C)C)=O)CC(NC(C2CC(S(C)(=O)=O)C2)=O)C12CCOCC2 53522,C1(CC)(NC(=O)CC2(CC(C)C)NC(=O)N(CC)C2=O)CCCN(C(C)=O)C1 53523,C1(C(N2CCC(C)C2)=O)C2C=CC3(CN(C(N4CCc5ccccc54)=O)C(=O)C13)O2 53524,c1(CC(N2CC(C)(C(=O)NC3(C(N)=O)CCCCC3)C2)=O)ccc(O)nc1Cl 53525,C(c1cnn(C)c1)=CC(=O)NC1(CO)CN(C(c2c(OC)csc2)=O)C1 53526,c1(NC=O)ccc(C(N2CCCC2C2(NC(=O)C(F)C3CCC3)CC2)=O)cc1 53527,C1(NC(Cc2ccc(C)s2)=O)CN(C(C2CCCCC2(F)F)=O)CC12CCC2 53528,O=C1COC(CNC(C2CCN(C(=O)C(F)C3CCC3)CC2)=O)CN1 53529,c1(C(=O)NCC2(NC(C(CC#C)C)=O)CCOC2)cc(C(=O)C(C)C)ccc1F 53530,c1(OCCC)ccc(CC(=O)OCC)cc1.c12cnn(C)c1COC2=O 53531,N1(C(c2ccn(COC)n2)=O)CC(CNC(=O)CCc2cc(OC)no2)C2CC12 53532,c1(NC2CCN(Cc3c(OC)cc(OC)c(Cl)c3)C2)n[nH]c2ccc(C)cc12 53533,C(=O)(CCCCC1CCCCC1)NCCCCNC(CCCOC(C)C)=O 53534,C(c1ncco1)=CC(=O)NCC1CCN(C(c2ccoc2C2CC2)=O)C1 53535,CC(C)(C)C1=NOC(C(=O)NCCOCCNC(=O)C(F)CC2CCOC2)C1 53536,C1(CCC)CN(C(=O)CC2CC2c2ccccc2)CCN1C(=O)Cc1nc[nH]n1 53537,Cn1cc(C(N2CCC(CO)C(NC(=O)CC3CC4CC4C3)C2)=O)c2sccc12 53538,C1(OC)(CNC(C2CC3(C2)CC3F)=O)CCN(C(=O)C(C)C(C)C)CC1 53539,C1(NC(CC(=O)OC)=O)C2CCN(C(c3nn[nH]c3Cl)=O)CCC12 53540,C1(CCC)(NC(c2nn[nH]c2Cl)=O)CCCN(C(c2c(C)nn(CC)c2C)=O)C1 53541,c1(CC)ccc(C(c2nnnn2C)NC(Cc2ccccc2)CC(=O)O)cc1F 53542,C1(C(=O)NCC(C2CCCC2)NC(C(CN(CC)CC)F)=O)CCC(C)CC1 53543,N1(C(c2cnn(CC)c2Br)=O)CCC(C)C(NC(c2ccc(CO)o2)=O)C1 53544,NS(=O)(=O)CCC(=O)NCCNC(C1CCCN(C(c2cnns2)=O)C1)=O 53545,c1(N(C(=O)NC(C)COc2ccc(F)cc2)C)cc(Cl)nc(=N)[nH]1 53546,C=C=C(C)CC(=O)NC1C2CCN(C(=O)CC3CC3CC(=O)OCC)C12 53547,C#Cc1ccccc1CNC(C1CCN(C(=O)C(C)C=CC)CC1O)=O 53548,c1(C(=O)NC(CC)C(=O)NCC(C)NC(C)=O)cncnc1C 53549,N1(C(Cc2c(C)ccnc2)=O)CCCC(C(=O)N(C)Cc2nc(=O)o[nH]2)CC1 53550,C12CCCC(C1)NC2=O.O=C1C(=O)NCCCCN1.C1(C(=O)NC2CC2)CC1 53551,N1(C(COCCC(C)C)=O)CCN(C(c2nnn(C)c2C(F)(F)F)=O)CC(O)C1 53552,Cc1nccc(C(=O)NCC2(F)CC(CNC(=O)C=CC3CCCO3)C2)n1 53553,N1(C(c2c(OCC(C)C)nccc2)=O)CCCC(C)(NC(=O)CCC(C)(C)F)C1 53554,C1(C(=O)Nc2nnc(-c3ccc(Cl)cc3Cl)s2)C=CC2(CCCC2)CC1 53555,C(CC(C(N)=O)NC(C1(NC(C2CC2(F)Cl)=O)CCOCC1)=O)OC 53556,N1(C(CC2CCC(C)CO2)=O)C2CCC1CN(C(C1CCn3nncc3C1)=O)C2 53557,c1(CNC(C2CCCNC2=O)C)ncccc1Cl 53558,c1(CC(C(=O)NCCC(C)OC)NC(=O)C(C)Cn2cccn2)cnn(C)c1O 53559,CCCCCC(F)C(=O)NC(C)C(=O)NOCC(O)CO 53560,Cc1nsc2ncc(C(N3CC4(C3)CN(C(=O)Cn3nnc(=N)[nH]3)C4)=O)cc12 53561,c1(C(N(C)CCOCCN(C)C(C2C3COCC23)=O)=O)nn(C)cc1S(C)(=O)=O 53562,C12(C(N3C(CNC(C4CSCCS4)=O)C4CC4C3)=O)CCC(F)(CC1)CC2 53563,Cc1ccc(F)c(C(=O)N(CCCN(C)C(c2cnc(-c3ccsc3)s2)=O)C)c1 53564,c1(C(=O)NC2(COC)CN(C(C3OCC4CCCC34)=O)C2)cc(Cl)c(Cl)cc1N 53565,C(=O)(C(C)(C)C(F)(F)F)NC(C1CCCN(C(CCOC(C)=O)=O)C1)C 53566,C1(C2CC2)(NC(CCN(C(C)=O)C)=O)CCN(C(c2coc(Cl)n2)=O)C1 53567,CN1CCN(C(=O)Cc2cnns2)C(CNC(=O)CC2CCCCC2(C)C)C1 53568,c1(C(=O)NCC(=O)N(C(C(=O)OC)C)C2CC2)nc2cc(Cl)ccc2s1 53569,C12(CNC(CCCOCC=C)=O)CC1CN(C(=O)C(C)Cc1cnc[nH]1)C2 53570,C(C(=O)NCCCOC)(C1=CCC2CC1C2(C)C)N1C(C)(CC)CC1 53571,CC1(C)CCC(CNC(C2CCC(=O)NC2)=O)N(c2nnco2)C1 53572,c1(C(=O)NCCC2CCC(NC(=O)CCCC3CC3)C2)occ2c1CCOC2 53573,CS(=O)(=O)CCCC(=O)NC1(CNC(=O)COC2CC2)CCOC1 53574,N1(C(=O)Nc2n(C)ncc2C2CCC2)CC2C3CCC(C(O)C3)C2C1 53575,C(CCC(C)C(=O)N(CCC(C)NC(=O)Cn1cnc([N+](=O)[O-])c1)C)OC 53576,c1(C(=O)NC)ccccc1NCc1cscc1Br 53577,C1(C(=O)NCC2CCC(CO)CC2)CN(C(=O)C(O)Cn2cncn2)CCC1O 53578,C1(C(=O)OC)CC(C(=O)NCCCCNC(=O)C(C)(C)C2CC2)C1(C)C 53579,c1(OC)cc(F)cc(C(N2CCOCC(CNC(=O)C3=NOCC3)C2)=O)c1N 53580,c1(C(=O)NC23CCN(C(c4cccc(F)c4O)=O)CC2C3)c[nH]c2nccc-2c1 53581,c1(CC(=O)NC2(CCCC(=O)NCCC=C=C)CCC2)ccc(C)c(F)c1 53582,C(=O)(C(C)(C)C(C)O)N1CC(CNC(C2(CC=C)CCC2)=O)C(C)C1 53583,c1(COC)nc(C)c(C(N2CC(CNC(=O)C(C)(C)CF)C(C)C2)=O)s1 53584,CC(C(=O)NC1CN(C(=O)CC(F)F)CCC1CO)S(N)(=O)=O 53585,C1(C(=O)NCC(C)NC(c2cnc(C(C)(C)C)s2)=O)CC(c2ccccn2)=NO1 53586,C(=O)(C#CC1CCCO1)N1CC(NC(C2CC(C)C2(C)C)=O)C1 53587,Cc1ccc(-c2csc(C(=O)NC(CNC(=O)CN(C)C3CC3)CO)n2)cc1 53588,C(=O)(C(C)CC(C)(C)C)N1CC(CNC(CSSC)=O)C(C(F)(F)F)C1 53589,C=CCCCCCC(=O)N(C1CCCCN(C(=O)C(C)(C)OCCC)C1)C 53590,N1(C(C2(C)CCCC2O)=O)CC2(CC(CNC(c3nc(Cl)sc3Cl)=O)C2)C1 53591,C1(C(=O)NC(CC(=O)OC)(C)C)CCN(C(=O)CCC(C)=O)CCO1 53592,C1(NC(C(C)=CC2CC2)=O)C(C)CN(C(=O)CC2(C)CCCCC2)CC1C 53593,c1(C(=O)OCC)c[nH]c(=NC2CCC3CCC23)cn1 53594,C1(C(N(CC(=O)NOCC2CCCCC2)CC#C)=O)CCCCC1F 53595,Cc1cc(N)cc(C(=O)NCC2CC2NC(=O)Cc2n[nH]cc2Br)c1F 53596,N1(C(N2CCCCC2)=O)CCCC(Cc2ccccc2)C1.O=C1CCN1 53597,C(=O)(CC1=NN(C)C(=O)C1)NCCCCCN(C)C(C1CCCSC1)=O 53598,C=CCCCC(C)NC(C1C=CCCN1C(c1cc(C)oc1C)=O)=O 53599,c1(NC(c2ccc(-c3ccc(C)nc3)cn2)=O)cccc([N+](=O)[O-])c1F 53600,NC(=O)CCN=c1ccn2ncc(S(=O)(=O)N3CCN(CC(F)(F)F)CC3)c2[nH]1 53601,CC(Cn1cccn1)C(=O)NCC(C)N(C(=O)Cc1nnc(-c2ccco2)o1)C 53602,C1(C(N2C(CCCNC(c3ccsc3)=O)CCC2)=O)CCC(C(N)=O)O1 53603,C1(NC(CN(C)C2CC2)=O)CCN(CC(c2ccc(NS(C)(=O)=O)cc2)=O)C1C 53604,c1(C(=O)NC(CN(C(C2(CCCC)CC2)=O)CC)C)ccc2c(c1)N(C)C(=O)C2 53605,N1(CC(=O)N(CCCC)CC=C)CCc2c(Cl)cc(Cl)cc2C1 53606,Cn1cc(C(=O)NCC(C2CCOC2)NC(c2ncccc2N)=O)c(C(F)F)n1 53607,C1(C(=O)NC2CCCCC2O)(NC(C2CN(c3nccs3)C2)=O)CCCCC1 53608,c1(C(N2CCC(CC(C)NC(C3CC(F)C3)=O)CC2)=O)ccc(Cl)c(C#N)c1 53609,Cc1cccc(O)c1C(N1CC2(CCC2NC(=O)C=Cc2ccccc2)C1)=O 53610,Cc1nc(CC2CC2)sc1C(=O)NCC1CCCC(NC(c2c[nH]nc2F)=O)C1 53611,C1(NC(c2ccccc2F)=O)CN(C(c2ccc(C3CCOC3)s2)=O)CC1F 53612,C1(C(=O)NC(CN(C)C(C2(C(C)(F)F)CC2)=O)(C)C)CC12CCOCC2 53613,C(=O)(C1=CSCCO1)NC1C(NC(C(Cn2cncn2)OC)=O)C1 53614,c1(C(N(C2CC(NC(C3CC3c3ccn(C)n3)=O)C2)C)=O)nccnc1N 53615,CC1CC(N(C(=O)C(F)C2CC(NC(c3c[nH][nH]c3=N)=O)C2)C)CCO1 53616,c1(C(=O)NC2CC(CNC(C(C)N3CCC3)=O)C(O)C2)ncc(Cl)cc1F 53617,C12(C(=O)OC)CCCC1CCN2C=O.c1(C(=O)NCCSC)cnc2ccccc2n1 53618,C(=O)(C1=NOC2(CCC2)C1)NC(CCC)CCCNC(=O)C(C)(F)F 53619,CC1CCC1C(=O)NCCCC1(NC(C2CC(OC(C)(C)C)C2)=O)CC1 53620,C(=O)(CC(C(F)F)NC(c1cnco1)=O)NC(C)(C)C(F)F 53621,c1(C(N2C3CC(NC(=O)COCCF)CC2CC3)=O)ccc(F)c2[nH]ccc12 53622,C1(C(=O)NCC=CCNC(=O)CCSCCCNC(C)=O)(OC)CCC(C)C1 53623,N1(C(=O)CCCc2cc(Cl)sc2Cl)CC2(CCN2C(=O)CCOC2CC2)C1 53624,c1(CC(C)C(=O)N(CCNC(C23COCC2C3)=O)CC2CC2)ccccc1F 53625,c1(CC)onc(C)c1C(=O)NCC1(C)CCC(NC(=O)CSc2cccs2)C1 53626,N1(C(c2c(OCC#C)nccc2)=O)CCCC(NC(=O)CCN2CCCC2)CC1 53627,N1(C(CCCN(C)C(C2CC3OC2C2CC32)=O)=O)CC(C2=NOCC2)C1 53628,C1(C(=O)NC2CCOC2)CN(C(c2ccn(CCF)n2)=O)CC1(F)F 53629,C1(O)(CN(C)C(c2ccc(C(N)=O)s2)=O)CCN(C(C2(CO)CCCCC2)=O)C1 53630,C1(n2cc(COC)nn2)CCN(C(C23CCCC2CC3)=O)CC1 53631,C(=O)(C1=N[N+]([O-])(CCO)CC1)NCCN1CCCN(C(CCC(C)SC)=O)CC1 53632,CC(CC(C)(C)C)C(=O)N1CCC1CNC(c1ccncc1Br)=O 53633,Cc1ccc(Cl)cc1OCC(=O)OC(C1CCCCC12CC2)CO 53634,N1(C(CC2C(C)OCC2)=O)CCC2(CC1)CCN(C(C1CC13CC(C)(C)C3)=O)CC2 53635,c1(C(=O)NCCC2(C(=O)OC)CCC2)cc(F)ccc1OC.C1C(C)=CC(=O)N1 53636,c1(C(N2C3C(NC(c4cnc(CC)nc4)=O)CC(C3)C2)=O)ccn2nccc2n1 53637,C(CCOC)(C(=O)NCCC(C)N(C)C)NC(C(C)OC)=O.C(=O)NC 53638,C1(=O)C(CCC(N)=O)N1.C(=O)(C(C)(C)CC#N)NCCC(C)C(=O)Cn1cnnn1 53639,CC(C)C(CCN(C)C(c1ccc(Cn2cccn2)o1)=O)NC(c1cc[nH]c1)=O 53640,Cc1cc(C(C(=O)Nc2ccoc2)N(C(C)C(=O)Nc2ccc(F)cc2)C)c(C)o1 53641,c1(CC(C(=O)N(CCCNC(C2(CC#C)CCCO2)=O)CC)C)ccc(F)cc1 53642,Cc1ccc(S(=O)(=O)NC2CCC(C(=O)Nc3ccccc3CO)CC2)cc1Cl 53643,C1(CNC(C(C)Cc2ccon2)=O)CC2(CC2)CN1C(c1ccc(F)nc1F)=O 53644,CCC(CC)CC(=O)NC1CCN(C(c2cccc(N)c2O)=O)CC1F 53645,c1(C(N2CCC(N(C(COCC=C)=O)CC)C2)=O)cccc2nc(O)[nH]c12 53646,C(N=c1[nH]c2ccc(F)cc2o1)C1C(C)CN(C(c2sccc2C(F)F)=O)CC1 53647,C1(NC(C=CC(C)(C)SC)=O)CN(C(=O)CCc2ncc[nH]2)CC1SC 53648,C1(CN(C)CC)CCN(C(c2cnoc2CC2CC2)=O)C1 53649,Cc1ccc(C(=O)Nc2cn(C)c(C(=O)Nc3nc(Cl)nc(Cl)n3)n2)c(C)c1Br 53650,Cc1ccc(CCNC(=O)C(C)CN(C(=O)CSc2cccnc2)C)cc1 53651,c1(C(=O)NCC2(OC)CN(C(c3ncc(C(F)F)s3)=O)C2)ncc(C)cn1 53652,c1(CN(C(=O)CN2CCSCC2)CCNC(C2CC(C#N)C2)=O)cccc(Cl)c1 53653,N1(C(COC)=O)CCC(NC(c2ccc(C(O)CF)cc2)=O)C(F)C1 53654,c1(C(N(CC(C)N(C(=O)Cc2cccc(F)c2F)C)C)=O)cc(F)ccc1F 53655,c1(C(=O)NC2CC(F)(CNC(C3N(N=O)CCC3)=O)C2)cc2cn[nH]c2cn1 53656,c1(C(N2CCC(N(C(c3c(SC)cccc3)=O)C)C2)=O)ccc([N+](=O)[O-])o1 53657,CC1(C)OC2(Cc3ccccc3)CCC1(NC(c1ccc(F)c(O)c1)=O)CC2 53658,CC(O)C(C(=O)N1CCC(C)(NC(c2cnn(C3CCC3)n2)=O)C1)N(C)C 53659,c1(NC(C2(F)CCN(Cc3ccc(C)nc3Br)CC2)=O)cnc(C)c(Cl)c1Cl 53660,c1(C(N(CC(O)CNC(=O)CN2CCC(C)(C)C2)C)=O)cc(Cl)cc2c1OCC2 53661,C(CN=c1[nH]c2cccc(F)c2o1)(C1CC1)NC(=O)C#CC1CCCCC1 53662,CS(=O)(=O)c1ccccc1C(N1CCCCC(NC(=O)C2=C(Cl)CCC2)C1)=O 53663,C1(NC(CC(C(C)OC)NC(=O)Cn2ccccc2=O)=O)CC2(CNC(=O)O2)C1 53664,C1(CC(=O)NCC2(CNC(C3N(C)C(=O)CC3)=O)CCC2)CCCCC12CC2 53665,C1(OC)CN(C(c2cnc(Cl)s2)=O)C(C)(CNC(=O)C(F)(F)CN(C)C)C1 53666,CN1C(=O)c2ccc(C(=O)NCCCNC(C3CCC3(F)F)=O)cc2C1=O 53667,CC(C)C(C)(O)C(=O)N1CC(CNC(C2CCC3CCC2O3)=O)C1 53668,N1(C(CCC(C)SC)=O)CC2CCCC2(NC(=O)Cc2ccn(C)n2)C1 53669,N1(C(C(C)Cn2ccnc2)=O)CCCC(N2CCCC2)C1.CC(C)(C)OC(=O)O 53670,c1(C(N2CC3(C(F)(F)F)CC3(CO)C2)=O)cc(=O)c2ccccc2[nH]1 53671,N1(C(C(C)NC(COC)=O)=O)CCC2CCN(C(=O)Cc3cncnc3)CC12 53672,c1(C(=O)NC(c2ccc(OC)cc2)c2nccn2C)coc2c1COC2 53673,C(=O)(CCCC(=O)N(C)C)NCCCN(C(=O)CN1CC(C)C1)CC 53674,CC(C)CCC(=O)NCC(=O)NC1CC(CNC(c2ncn(C)n2)=O)C1 53675,C(=O)(C(O)CCNC(=O)C=CC1CCOC1)N(CCOCCOC)C 53676,N1(C(CC(CCC)NC(=O)C(C)(CO)OC)=O)CCC(C2CCCC2)C1 53677,C(=O)(C(C)CCN(C)C)N(CCCNC(CC(=O)NCC)=O)CC1CCCC1 53678,C(=O)(CCC(F)(F)C(F)F)N1CCCC(NC(CCc2cc(C)no2)=O)C1C 53679,N1(C(c2cncc(CC)c2)=O)CC(C)CCC1CNC(=O)Cc1nc[nH]n1 53680,C#CC1(C(N2CC(C(N)=O)C2)=O)CCN(C(=O)C(C)c2cc[nH]n2)CC1 53681,c1(COC)nc(C(=O)NC(C)C(C)(C)NC(C2CC2(C)C)=O)n[nH]1 53682,C1(C(=O)NCC(F)(F)C(C)(C)O)(CC)CCCN(C(=O)C=Cc2cc(C)no2)C1 53683,N1(C(C)=O)CCC(C)(NC(C2CCCCC2NC(=O)C(C)C#N)=O)C1 53684,CCN(Cc1cccs1)N(CCOC)CC(=O)N(c1ccc(F)cc1)c1nccs1 53685,Cc1c(C(=O)N(CCC(C(C)C)Nc2ncccn2)CC(C)C)cccc1F 53686,c1(C(=O)NCC2(CCNC(CC3C(C)CCC3)=O)CC2)c(F)cc(F)cc1Cl 53687,C1(CC)(CC)CC(O)CN1C(=O)C(C1CCN(C(c2cc(F)n(C)n2)=O)C1)F 53688,n1(CCCC)nnnc1C(c1ccccc1)NC1CCC(C(=O)NC)C1 53689,C1(CNC(C2(CC)CC2(F)F)=O)CN(C(=O)CCc2cccn2C)CCC1(C)C 53690,C1(CC)CN(c2cc(F)n[nH]2)CC12CCN(Cc1conc1C)CC2 53691,C1(NC(C(C)=CC)=O)CCN(C(=O)Cc2nonc2C)CC1O 53692,C1(CNC(c2nccnc2N)=O)CC(C(=O)NCc2nc(CSC)sc2)C(O)C1 53693,C1(C)(NC(C(N2CCCC(C)C2)=O)=O)CCCN(C(c2cc(Cl)ccc2O)=O)C1 53694,Cc1nc2cccc(C(=O)NCC3CC3NC(C3(CC(C)C)CCCC3)=O)c2[nH]1 53695,CC1CCOC1C(=O)N(C(C)(C)C)Cc1cn(C2CC(N(C)C)C2)nn1 53696,N1(C(CC=CC=C)=O)CCCCCC1CNC(=O)CCS(C)(=O)=O 53697,N1(C(c2ccc(C(=O)NC)cc2)=O)CCCCC(CNC(=O)C(C)CSC)C1 53698,c1(C(N2CC(NC(C(COC)(F)F)=O)C(OC)C2)=O)ncc(F)cc1F 53699,C(=O)(C1=CC2CCCCCC12)N1CCC(C(C)NC(c2ccc(C(C)=O)s2)=O)C1 53700,C(c1ccc(S(=O)(=O)NC)cc1)=CC(=O)NCC(CC=C)NC(=O)CC1CC1 53701,C=CCCC(C(=O)OC)NC(=O)CSC.C12(CCSC1)C(=O)N2 53702,Cc1nsc(C(N2CC(C(=O)N(C)CCOC(F)F)CC2C)=O)c1N 53703,O(C1CCc2c(Br)cccc21)C(=O)C(c1ccc(F)c(F)c1)=O 53704,N1(C(C2(F)CCN(C(CC=C)=O)C2)=O)CC(C)OC(C)(C)C1C 53705,C(=O)(CS(=O)(=O)CC(=O)N1CCCC1CCCNC(=O)C=Cc1nccs1)OC 53706,c1(C(N2CCC(CC3N(C(CC(C)C)=O)CCCC3)CC2)=O)cc(N)cc(O)c1 53707,c1(C(=O)NCC2(CCNC(C3CC3C(=O)O)=O)CC2)cc2c(cn1)CCCC2 53708,Cc1nsc(N)c1C(=O)NCC1CCN1C(c1cc(Br)c[nH]1)=O 53709,N12CCN(CC1)C1(CC1)CCNC2=O.C(C)(C(=O)OC(C)(C)C)OCC=C 53710,Cc1c(NC(C)(C(C)C)c2nnnn2C2CCCCCC2)ccc(Br)c1Cl 53711,C1(CNC(CCCCC#C)=O)CCCC2CN(C(=O)Cc3ccc(F)nc3)CC12 53712,n1(CC(=O)N(C2CN(C(=O)COCCN(C)C)CC2F)C)cnc2ccccc12 53713,Cc1cnn(CCC(=O)N(C)CC2(CNC(=O)COc3cccnc3)CC2)c1 53714,CCC(CC(=O)NCCCOCCCNC(C1OCCC1C)=O)C(F)F 53715,N1(C(C(CC=C)(C)C)=O)C2CCC1CC(NC(C1(C(C)C)CNC(=O)C1)=O)C2 53716,N1(C(C2C(C)=C2)=O)CC2CCCC(C1)N2C(=O)CC(C)c1ccco1 53717,C1(CC(=O)NC2CN(C(Cc3cn(C)nc3)=O)C2)CCNC(=O)C1 53718,C(=O)(C1=Cc2ccccc2C1)N(CCC(=O)NC1COCCC1O)CC=C 53719,C(=O)(C1=C(Cl)CCOC1)NCc1ccc(C(N2CC(C#C)OCC2)=O)cc1 53720,N1(C(C(C(C)C)OC)=O)CCC2(CNC(=O)CCCn3cccn3)CCCC12 53721,C=C(C)C1CC=C(C(c2nnnn2CCCF)NCCC(C)C(C)(C)C)CC1 53722,N1(CC(=O)CCNC(=O)C(c2ccc(Br)cc2)(F)F)CCC(CO)CC1 53723,c1(C(=O)NCCCN(C(=O)CCC2CCCCN2C)CC)cc[nH]c(=N)c1 53724,Cc1ccc(CN(C(=O)CC2CCN(CC3CCCO3)C2)CC2CC2)c(C)c1 53725,N1(C(c2c(CC)nccc2)=O)CC2CCC(C1)C2CNC(=O)C(C)NC(=O)NC 53726,C12(C(=O)NCC(C(C)C)O)CCC(NC(=O)CC(C)O)(CC1)C2 53727,CC(C)(CNC(=O)CCCC1CCCC1)C(=O)NC1(c2ncc[nH]2)CC1 53728,C(=O)(CC(O)CNC(=O)CC1CCCC1O)N(CCOC(C)=O)C(C)C 53729,Cn1nc(CNC(=O)CC2CCOC2=O)c2c1CCN(C(c1cc[nH]n1)=O)C2 53730,c1(CC)ccc(C(C)C(=O)N(CCNC(=O)CC(C)n2cccn2)C(C)C)cc1 53731,C(=O)(C(CC(C)C)OC(c1sccc1C)=O)N(C)CC1(OC)CCN(C(C)=O)C1 53732,C(=O)(C1=CCCCC1C)N1CC(NC2C(NC(Cc3ncc(C)[nH]3)=O)CCCC2)C1 53733,c1(C(C(=O)NCC(C)C)N(C(CCC)C)CC)cnc(Cl)c(F)c1 53734,c1(COCC)nnc(N2CCCC2CC(C)(C)NC(c2ccon2)=O)s1 53735,CC1CC(NC(c2cc(C#N)n(C)n2)=O)CCN1C(c1cnc(C2CC2)s1)=O 53736,C=CCN(OC)C(=O)CCC1CN(C(=O)CC2CSC2)C1 53737,C(C1=NOC2(CCC2)C1)NC(C1CCN(C(C(CC)N(C)C)=O)C1)=O 53738,Cn1nc(-c2ccncc2)cc1C(=O)NCC(CO)NC(=O)OC(C)(C)C 53739,c1(NC(c2cn(-c3c(C)cc(F)nc3)nn2)C2(O)CCC2)cccc2c1CCO2 53740,C1(C(=O)NC(c2nccn2C)CC)CCCN(C(c2nn(C)cc2C)=O)C1 53741,C1(C(F)F)(OC)CC(C(=O)N(C2CCN(C(c3cccnc3)=O)C2)C)C1 53742,c1(C(=O)NCCN(CCC)C(C2(C)CC(C)=NO2)=O)nc(C)n(C)n1 53743,Cc1nc(CC(=O)NC(Cc2cn[nH]c2)C(=O)NCC2CC2(C)C)n[nH]1 53744,C1(NC(=O)C(F)F)CN(C(C23CCCN2CCC3)=O)CCC1O 53745,c1(-c2cc(NC(C3CCCCCC3)C)sc2)ccc(F)cc1 53746,c1(C(=O)NC(C)CNC(C2CCN2S(C)(=O)=O)=O)cnc2n1CCS2 53747,C1(NC(C(OC)OC)=O)C2CCC(C2)C1C(=O)NCC1CC(O)C(O)C1 53748,CCCCC(CC)CC(=O)NC1CCC(C)N(C(=O)C=CS(C)(=O)=O)C1 53749,c1(CC(C(=O)NC2(CNC(CCOCCOC)=O)CCOC2)C)ccccc1Cl 53750,C1(C(=O)NCc2cc(C)n(C)n2)CC(F)CN(C(c2cnc(Cl)c(I)c2)=O)C1 53751,C1(C(N(C)Cc2cncc(O)c2)=O)C2CCC(C2)C1N 53752,C1(NC(c2c(COC)cc[nH]2)=O)CC(C)CN(C(=O)CCOC(C)C)C1 53753,Cc1cc(Br)ncc1C(c1nnnn1C(C)(C)C)NCC1CCCN1S(C)(=O)=O 53754,N1(C(COc2cc(C)on2)=O)CCC(O)C(c2cn(C3CCCNC3=O)nn2)C1 53755,c1(OCC)ncccc1C(=O)NC1CCCC1NC(=O)CC(C1CCCC1)SC 53756,c1(C(=O)NCCN(CCOC)C(C2OCCC2C)=O)cc(C)ncc1Br 53757,Cc1cc(F)ccc1C(=O)N(c1ccc(Br)c(N(C)C)c1)C1CCNCCC1C 53758,C(C)(C)(CC(F)C(=O)N(C1CCOC(C)(C)C1)C)NC(C1C(C)OC(=O)N1)=O 53759,C1(CNC(c2c(C(C)C)nns2)=O)CCN(C(C2CN(C)CCO2)=O)C12CC2 53760,C1(NC(CCN(C(=O)C(C)CC2CC2)CC)=O)CC1C1CC1 53761,N1(C(c2ccon2)=O)CCCC2(CCN(C(c3nccc4ncccc34)=O)C2)C1 53762,C1(C(=O)Nn2cc(OC)nn2)CCCCN1CCNC(=O)NC(CSC1CC1)=O 53763,C1(CNC(C(N2CC(CC)OC(C)C2)=O)=O)CC2(CO1)CC1(C2)OCCO1 53764,C1(CC(=O)NC)CN(C(=O)CC2(CSC)CC2)CCN1C(=O)C(C)C(C)(F)F 53765,C(=O)(CC(C)(O)C(F)(F)F)N1C2CN(C(c3n(C=C)ncc3)=O)CC1CC2 53766,C1(NC(CN(C(CCOC)=O)C)=O)CC2CC1N(C(C1C3CCCOC13)=O)C2 53767,CN1CC(C(=O)NCC(C)(C)NC(=O)CNC(N)=O)c2ccccc2C1=O 53768,C1(NC(C2(C)N(C)CCC2)=O)CC12CCN(C(C1CCc3nn[nH]c3C1)=O)CC2 53769,N1(C(C(CC=C)C)=O)CCC2(CC1)CC2CNC(c1ccc(OCCF)cn1)=O 53770,C1(NC(c2cnoc2)=O)CC1C1CCCN(C(c2c(F)ccnc2F)=O)C1 53771,N1(c2nc(OC)c(OC)cn2)CC2CCCC(C1)C2C(N1CCCC(F)C1)=O 53772,C(=O)(C1=C(C)CCCC1(C)C)N(C1CC(C(c2cccc(N)c2)=O)C1)CC=C(C)C 53773,c1(NC(=O)NC2C3CCC(C3)C2C(=O)NOc2ccccc2)cccc2c1CCC2 53774,Cc1nc2oc1C(=O)NC(=O)CCC(=O)NC2.c1(C)ccccc1.C1(CN)CC1Cl 53775,C1(CC(=O)NCC(C)NC(=O)C(C)(C)NC(c2cccs2)=O)CCC2(CCC2)O1 53776,Cc1cc(C(N2CC(C)(C)OCC2CNC(=O)CC(C)C(F)F)=O)cc(N)c1O 53777,C1(NC(C(C)OCC=C)=O)C2CCC1N(C(c1nc(C)n(C)n1)=O)C2 53778,c1(NCC(C)NC(c2ccc(OC)c(C)c2)=O)ncnc2[nH]ccc12 53779,N1(C(C2N(C(C3CCN(C)C3)=O)CC3CC32)=O)CCOCCc2ccccc2C1 53780,C(C(=O)NNC(=O)c1ccccc1-n1cccc1)C1CCN(C)C1 53781,c1(C(=O)NC(C2CCN(C(C3C(C)(Br)C3)=O)C2)(C)C)coc2ccc(F)cc12 53782,Cc1ccccc1C(C)(C)C(=O)N(C1CCC(NC(=O)C(C2CC2)N(C)C)C1)C 53783,C(C(C)CN=c1cc(C)nc(C2CC2)[nH]1)NC(C=Cc1cccc(OCC)c1)=O 53784,c1(OC)cccc(OC)c1S(=O)(=O)NC1COC2(CCCC2)C1O 53785,C1(C(N(C)CC2(NC(c3ccn(CC(F)F)n3)=O)CC2)=O)CC2(CCC2)CCO1 53786,CC12COCC1CN(C(C1CCCC1NC(C1(C)C=CCC1)=O)=O)C2 53787,c1(C(=O)NCC(CCC)NC)ccc([N+](=O)[O-])cc1.C(C(F)F)=C 53788,c1(C(=O)NCCn2cccc2NC(C2CC2)C2CC2)cc(Br)ccc1I 53789,c1(OC)c[nH]ccc1=NCC1CN(C(=O)OC(C)(C)C)CCC1CC(=O)O 53790,Cc1nn(C)c(Cl)c1C(=O)NC12CC(CNC(c3ncccc3O)=O)(C1)OC2C 53791,N1(C(CCN(C(CCC)C)C)=O)CC2(CNC(c3[nH]c(O)nc3C)=O)CCC1CC2 53792,c1(OCC(=O)NC(CC)CN(C(=O)CCCN(CC)CC)C)ccc(C)c(C)c1 53793,c1(OC)cc(O)c(C(=O)NCC(C)NC(C2CC=CC2)=O)cc1S(N)(=O)=O 53794,C1(CNC(c2cc(C)on2)=O)CC2COCC2N1C(C1CC(C)(C)CN1C)=O 53795,Cc1c(C(N2CCN(CCNC(=O)C=CC(F)(F)F)CC2)=O)cnn1C1CCC1 53796,C(=O)(Nn1ccccc1=O)C1CC(NC(C(C2CC2)OC)=O)C1 53797,N1(C(C2C(C)CC2)=O)CC(C(N2CC(n3ccnc3)C2)=O)CC1(C)C 53798,C(C(=C)CC)NC(CN(C(C1(CC=C)CC1)=O)C)=O 53799,c1(C(=O)OCC)cccc(NC(=O)NC(C)C(C2CCCCC2)O)n1 53800,C1(NC(C(C)NC(C)=O)=O)CN(C(c2[nH]c(=N)sc2C(F)(F)F)=O)CC1C 53801,N1(S(CCOC)(=O)=O)CCOC(C(=O)N(C2CC(O)C2)C)C1 53802,C(CCCCCF)N(C(=O)COC(=O)C=CC(F)(F)F)C 53803,Cc1cn2c(CC(N3CCC(C4CC4NC(C4(CN(C)C)CC4)=O)C3)=O)csc2n1 53804,Cc1nn(CCO)cc1C(N1CCC(N(C(=O)C(O)Cc2ccccc2)C)C1)=O 53805,c1(CC)cc(C(=O)N(C(C)C#N)C(c2ccccc2Br)C)cc(Cl)c1 53806,N1(C(C2(COC)CC2)=O)CCOC2(CCN(C(=O)Cn3c(C)c(C)sc3=O)C2)C1 53807,c1(C(=O)NC2CC(C)N(C(c3cc(Cl)n(C)n3)=O)C2)ccc2ncsc2c1 53808,c1(C(=O)NC2CN(C3CCC(C)CC3)C(=O)C2)cc2cc(Cl)ccc2n1C 53809,c1(C(N2CC(C(C(N3C(C(=O)NC)C=CC3)=O)OC)C2)=O)ccnnc1C 53810,S(=O)(=O)(c1c[nH]c(C(=O)NCC(C)(C(C)C)NC(C2CCCC2O)=O)c1)NCC 53811,N1(C(C(CCC)C)=O)CCN(C(c2ccc[nH]2)=O)CC1c1cn[nH]c1 53812,N1(C(C)=O)CCC(C)(C(N2CC(CNC(c3cn(CC(F)(F)F)cn3)=O)C2)=O)C1 53813,C1(C(N(CCCNC(=O)C(F)=C(C)C)CC)=O)CN2CCN1CC2 53814,C12(NC(Cc3ccc(C#C)cc3)=O)CCN(C(=O)CC(C)CCC)CCC1C2 53815,N1(C(C2C(C(C)C)C2)=O)CC(C)(CNC(c2onc3c2CCCC3)=O)CC1(C)C 53816,CC1C(=O)C2CCCCC(C(F)(F)F)N(C1=O)CCN2CC.N(C)C 53817,c1(OC)cncc(C(=O)NC2CCCC(C(N3CCC(F)CC3)=O)C2)c1 53818,C1(NC(COCCN(C)C)=O)C2CC(O)C1N(C(=O)Cc1cscn1)C2 53819,c1(C(N2C(CCCC)CN(C(=O)C(O)CF)CC2)=O)ccc2c(=O)[nH]ccc2c1 53820,c1(C(N2C(C(N3CCC(C#C)CC3)=O)C(O)CC2)=O)cc(Br)c(O)c(Br)c1 53821,C1(NC(C(CC(C)C)(F)F)=O)CN(C(C2CC23CCCC3)=O)C2(CCCC2)C1 53822,C1(S(N)(=O)=O)(C(=O)NC(C)CCNC(=O)C(O)CCc2ccccc2)CCCC1 53823,CCCC(CNC(=O)C(C1(O)CCCC1)F)NC(=O)CC1CCOC1C 53824,C(=O)(C(CN(C)C)NC(=O)CCNC(C1CCC1)=O)N1CC(CC)C1 53825,N1(C(NC2CCc3cccnc32)=O)CC2(CCOCC2)c2ccccc21 53826,c1(C(C#C)NC(=O)C(=O)NC(c2n[nH]c(C)n2)CC2CC2)ccccc1 53827,C(=O)(C1=CCCCO1)NC1(CCCNC(CN(c2ccccc2)C)=O)CC1 53828,CCCCC(CNC(=O)CN1CCCCC1=O)NC(=O)CCNC(=O)CO 53829,c1(C(=O)NC2C3CN(C(C4C(C)OCC4)=O)CC2C3)cc(Br)cc([N+](=O)[O-])c1 53830,N1(C(C(c2ccc(Br)cc2)=O)=O)CCC(F)C(NC(C2CS(=O)(=O)C2)=O)C1 53831,c1(C(=O)NC2CC(CNC(CC(CCC)O)=O)C2)cc(F)cc2nccnc12 53832,c1(C(=O)NCC2C(NC(CCC(C)SC)=O)CCCC2)ncc(F)cc1N 53833,N1(C(c2c(C(C)C)noc2)=O)CCN(C)C(C(=O)NCC2CCCCS2)C1 53834,O=C(C1Cc2c(Cl)cccc21)NCC1(F)CC(NC(c2c(F)cccc2F)=O)C1 53835,C(=O)(C(CCNC(=O)C(C1CC1)SC)OCC)N(C1CCCC1)CCC 53836,c1(C(=O)NCC(CO)NC(=O)CC2(O)CCC2)cccc(-n2ccnc2)c1 53837,c1(C(=O)NC2CCC(N(C)C(c3ccccc3Cl)=O)CC2)cc(F)ccc1F 53838,c1(COCCNC(=O)NCCCC2CC(CC(C)C)OCC2)ccc(Cl)cc1Cl 53839,CC(C)CC(C(=O)NC1CCN(C(=O)C(C)OCC(C)C)CC1)N1CCCC1=O 53840,N1(C(CC(CN(C)C)(C)C)=O)CCC2(C=C(C(=O)N3CCCCC3C(F)F)C2)C1 53841,C1(N(C(CCc2c(C)ncs2)=O)C)CCC(NC(=O)C(C)OCCN(C)C)CC1 53842,N1(C(C(CCCC)O)=O)CCCC(C2CCCN(C(=O)CC3CC(OC)C3)C2)C1 53843,c1(C(=O)NCC2C(CNC(CCC(=C)Br)=O)C2)cc2ccccc2n1C 53844,N1(C(C2CC3C=CC2CC3)=O)CC2CCN(C(c3cnc4cccnn34)=O)C2C1 53845,C(=O)(CCCC(=O)O)N(C(C)(C)C)C1CC1.Cn1cncc1C(N1CCC(C(=O)N)C1)=O 53846,c1(CCC)onc(C)c1C(=O)NC(CNC(c1cc(C(F)F)ccn1)=O)C1CC1 53847,N1(C(CC2CCC(=O)N2)=O)CCC2(CC1)CC(NC(=O)Cc1cccnc1Cl)C2 53848,c1(C(=O)NCC2(O)CCC(C)C2)ccc(F)c2[nH]ccc12 53849,C12(C(=O)NC(N3C(C(=O)Nc4ccccc4)CCC3)=O)CCC(CF)(C1)OC2 53850,c1(CCCCNC(=O)Nc2ccc(C)s2)cn2ccccc2n1 53851,C1(NC(COCCCCC)=O)CCN(C(=O)CC(O)C(C)C)CC1O 53852,C(c1cn(C)cn1)=CC(=O)NC(CC=C)CNC(C1OCCCO1)=O 53853,C1(CNC(C2CN(C)C(=O)C2)=O)CC(C(=O)NCc2cn[nH]c2)=NO1 53854,CCCCCCC(C(=O)NCC)N1CCC(C2CC3(CCC3)C(=O)N2)CC1 53855,C1(CC(=O)N(CCNC(CC2N(CC)C(=O)CC2)=O)C(C)C)CC2C=CC1CC2 53856,c1(-c2scc(C(=O)NCC3N(C(C(C)NC(C)=O)=O)CC3)n2)cccc(C)c1 53857,c1(C(N2CC(CNC(C(C=C)O)=O)C(C(F)(F)F)C2)=O)c(NC)cccc1F 53858,C1(CC(N2CC(NCC(=O)NCCSC)C2)=O)CCC2CC12 53859,N1(C(Cc2c(C)occ2)=O)CC(NC(c2cocc2C(N)=O)=O)CC(F)C1 53860,c1(C(=O)NCC(=C)CCNC(=O)C(Cc2cnc[nH]2)NC(C)=O)ccc(F)cc1 53861,c1(C(=O)NCC2(O)CN(C(C(C(C)O)C)=O)C2)ccn(CC(F)(F)F)c(=O)c1 53862,N1(C(c2cc(C)ns2)=O)CCCN(C(C2CCn3nccc3C2)=O)C(C)C1 53863,c1(C(=O)NCCC2(CNC(C(C)(C)C3CCCO3)=O)CC2)ccc([N+](=O)[O-])cn1 53864,N1(CC(=O)NCC(C)N(C(c2c[nH]c(=N)s2)=O)CC)CCCCCC1 53865,N1(C(C(C(C)O)NC(=O)CN2CC=CC2)=O)CC(C)c2ncccc21 53866,N1(C(CC2CCC(C)(O)CC2)=O)CC2(CCCC(CNC(C3CCC3)=O)O2)C1 53867,N1(C(CC2ON=C(C)C2)=O)CCC(O)(CCNC(c2cc(C(F)F)cs2)=O)CC1 53868,CC(C)CCCCC(=O)NCCCC(O)C(=O)NCc1cc(Cl)ccn1 53869,C1(NC(CCN(C(C)C)C(C2C=CCS2)=O)=O)C(O)CC1O 53870,c1(CCNC(=O)NCCCN(C)C(c2ccsn2)=O)ccccc1Br 53871,c1(N(C(=O)CC2CC(NCc3cn[nH]c3)C2)CC)cnncc1Cl 53872,C(=O)(CCCCCCCCN)N1C2CN(Cc3c(OC)cccc3)CC21 53873,c1(C(=O)NC2CC3C(NC(c4cc(C5(C)CC5)n[nH]4)=O)C3C2)ccc(O)cc1O 53874,CC1(NC(C2CCCC2O)=O)CCN(C(=O)Cn2cc(Br)cn2)C1 53875,C1(N(C(COCC(=C)C)=O)C)CN(C(=O)C(C2CCOC2)NC(C)=O)CCC1(C)C 53876,C1(C(N(CC(C)(C)NC(c2cccnn2)=O)C)=O)C2(CC2)C12CC2 53877,Cc1c(C(=O)NCC(C)CNC(=O)C(C(C)C)NS(C)(=O)=O)ccc2c1CCC2 53878,CC(C)CC(C(F)(F)F)NC(=O)C(=O)NC(Cc1cccnc1)C1CC1 53879,c1(OCC)ccc(NC(c2cc(OC)cc(C(=O)O)c2Cl)=O)cc1[N+](=O)[O-] 53880,C1(n2cc(C(CC)N(C)C)nn2)CCCN(C(=O)Cc2cnc(=N)[nH]c2)C1 53881,c1(C(=O)NC(CNC(C(CCC)(C)O)=O)CCOC)cn2cc[nH]c(=O)c2n1 53882,C1(OCC)CC(NC(=O)CN(C)C(=O)OC(C)(C)C)C1C.C1(=O)CCCN1 53883,N1(C(CN(CC)CC)=O)CCN(C(=O)CCC(=O)NC23CCCC2C3)CCC1C 53884,C#CCC1C(=O)N1.c1(NC(=O)OC(C)(C)C)cc(-c2ccccn2)on1 53885,c1(SC)cccc(F)c1C(=O)NCC1COCCN(C(c2cnccn2)=O)C1 53886,C1(CC(=O)NC2C(NC(c3cc(=N)[nH]cc3)=O)C2)CCC2(CC1)OCCO2 53887,c1(C(=O)NCCCCCNC(C2CC(C)C2)=O)ccc(F)c(Cl)c1F 53888,c1(N2CC(C(C=O)NC3CC4(CCC4)C3O)C2)ccccc1C#N.CC1(C)CC1 53889,C(=O)(N1OC2CCC1CC2)N1CC(C#C)(CO)C1.c1(C=O)cnn(C)n1 53890,Cc1cc(Nc2ccccc2C)ccc1NC(C1(NC(c2cc[nH]n2)=O)CC1)=O 53891,CCCCC(CC)C(=O)NC1CCCC1NC(=O)C(C)(C)c1cnco1 53892,c1(C(CC)CC)cc(C(N2CCC(CN(C(=O)CCn3cnnn3)C)C2)=O)on1 53893,C=CCC(C)(O)C(=O)NC1CC(F)(F)CC1NC(=O)C=Cc1cscn1 53894,c1(CCCC(=O)NCC2CC(NC(=O)C(F)C3CCC3)C2)nc2ccccc2s1 53895,c1(N2CCOCC(CNC(Cc3cccc(OC)n3)=O)C2)cc2nncn2cn1 53896,C1(NC(c2csc(O)n2)=O)CN(C(=O)C(F)n2cccn2)CCC12CCC2 53897,CC1(C)CCC(C)(NC(C2(NC(c3sccc3Cl)=O)CC(CO)C2)=O)C1 53898,Cn1nc(CCNC(=O)C(C2CCOC2)NC(=O)OC(C)(C)C)cc1C(F)(F)F 53899,N1(C(C)=O)CCS(=O)(=O)CC1.c1(CC23CN(C2)C3=O)cccnc1O 53900,C(=O)(C1=CC(O)CCC1)NCCC1CCCN(C(c2ccc(C3(C)CC3)o2)=O)C1 53901,C(C(C)C)(C(O)C(=O)NC(CNC(c1cc(C)ns1)=O)CO)OC 53902,c1(C(c2nnnn2C2CC(F)(F)C2)NC(CC=C)CC)cn(C(C)C)nc1Br 53903,CCCCC(C(=O)NC1CCN(C(=O)CC2CC2(Cl)Cl)CC1F)NC(N)=O 53904,C1(CC(=O)N(C)CC2N(C(C(F)OC)=O)CCC2)CCCN(CCF)C1 53905,Cc1cccc(C(N2CC=CC(NC(C3CC(N=[N+]=[N-])C3)=O)C2)=O)c1F 53906,C(=O)(CCCC(C)(F)F)N(C1CCCN(C(C(C=CCCC)O)=O)C1)CC 53907,N1(C(C(C)OCC=C)=O)C2CCC1CC(C(=O)NC1(N3CCOC3=O)CC1)C2 53908,C(=O)(CC(C)(C)CC(F)(F)F)N1CCC(COC)(NC(=O)C(F)=CCCF)C1 53909,C1(NC(c2cc(CC)n(CCO)n2)=O)CN(C(C2CC(=O)N(C)C2)=O)C(C)(C)C1 53910,N#CCCCC(=O)N1CC(F)CC1CNC(c1cccnc1-n1nccn1)=O 53911,c1(OC)c(Cl)ccc2[nH]c(C(N3CCCC(NC(=O)CCC4CC4)C3)=O)cc12 53912,C=CC1(CC(=O)NC2(C)CCN(C(c3c[nH]c(=N)nc3C)=O)C2)CCCCC1 53913,CCC(CO)CN=c1cc(C)[nH]c(=NCc2ncc(Cl)cn2)[nH]1 53914,c1(C(N2CC(NC(C(C=C)(C)C)=O)C(C)C2)=O)c(C)ccn1C 53915,C1(CCNC(CC2(C=C)CC2)=O)CCN(C(=O)CCCCN(C)C(C)=O)CC1(F)F 53916,N1(C(C2CC(CC)C2)=O)CCC2(NC(=O)C=Cc3cnc[nH]3)CCCCCC12 53917,N1(C(C2OCCN(CC)C2)=O)CC2(CCN(C(=O)CCC(C)C)CC2)CC1C 53918,N1(C(CC(CN(C(=O)COC2CCCC2)C)O)=O)CCCC(C)(C)C1CO 53919,N1(C(=O)C=CC2CCC2)CCN(C(=O)C(CC(F)F)c2ccc(F)cc2)C(CO)C1 53920,c1(NC(Cn2cc(-c3ccc(C)s3)nn2)=O)cc(OC(F)F)nc(C(=O)O)n1 53921,C(C(C)C(C)C(=O)N1CC(O)CC1CNC(=O)C(C)=CC1CC1)OC 53922,C(=O)(CC(C)CC(C)C)NCCC(C(=O)N(CCCOC)C)(C)C 53923,c1(CC)cc(C(=O)NCC(N2CC(NC(c3cccc(C)c3)=O)C2)=O)ccc1Cl 53924,N1(C(C2(OC(C)=O)CC2)=O)CCC(C)(C)C(CNC(=O)C(C2CCCCO2)O)C1 53925,N1(C(C2(C)CCCO2)=O)CC2(NC(=O)CC3(C#N)CCC3)CC1C2 53926,C=CCC(C(=O)N1CCC(OCCNC(c2cc(N)cc(O)c2C)=O)C1)C(C)C 53927,C1(CN(C(C2CCC(N(C)C)CC2)=O)CC)CCN(C(C2CC(C)C2)=O)CC1 53928,c1(C(N(c2cc(C)nc(C)n2)CC2(F)CCCNC2)=O)n[nH]c2cccnc12 53929,c1(C(=O)OCC)nc(=NC(C)CN(C)C(c2ccnnc2C)=O)cc[nH]1 53930,C12(CNC(C(CC#C)(C)C)=O)CCCC(CN1C(=O)CNC(=O)OCC)C2 53931,C1(CCC)CN(C(=O)Cn2cnc(C#N)n2)CC1C(=O)N(C12CC(C1)C2)C 53932,C1(C(=O)NC(C(C)NC(=O)Cc2cnn(C(C)(C)C)c2)(C)C)CC2(CCC2)CO1 53933,C1(C(=O)NCC2N(C(c3c(OC)c(C)ncn3)=O)CCC2)CCCC1S(C)(=O)=O 53934,CC1COCCN1C(=O)C(C)N1CCC1c1cccc(Br)c1 53935,C1(NC(C2CC=CCO2)=O)CCOC12CCN(C(=O)Cc1ccccc1F)CC2 53936,C12(CC(=O)N(C3CC4CCC3CC4)C)CCC1CN(C(c1cc(Cl)c[nH]1)=O)C2 53937,C#CC1(C(N2CC(CNC(c3cnc(C)[nH]3)=O)C(C(F)(F)F)C2)=O)CCOCC1 53938,c1(NC(CCC)=O)nc2ccc(CC(=O)NC)cc2[nH]1 53939,c1(OC(C)(C)C)ccc(NC(C2CCC(=O)NC2)=O)c(Br)n1 53940,c1(C(=O)NCC(CN(C(=O)C(C)=CC(C)(C)C)CC)(C)C)cccc2c[nH]nc12 53941,N1(C(c2cc(C)no2)=O)CCN(CC2CN(C)CCN2C)CC1C(C)C 53942,N1(C(c2c(CC)c[nH]n2)=O)CC(O)CC1(C)C(=O)NCC(C)C(C)(F)F 53943,N1(C(C2N(CC)CC2)=O)CC2CCN(C(=O)CC3(C(F)F)CC3)CC2C1 53944,C(=O)(C(O)CC[S+](C)C)NCC1(OC)CCN(C(c2ccc(F)cc2Cl)=O)C1 53945,c1(OC)ccc(C(=O)NCCOCCCN(C(=O)CC=C(C)C)C)c(F)c1 53946,CC1(C)CCCC(CC(N2CCC(c3ccc(I)cc3)(CO)C2)=O)O1 53947,C1(NC(=O)C(O)CN2CCCC2)CN(C(=O)COCCCF)CC1F 53948,c1(NC2C(OC(C)C)CCC2)ccc(S(=O)(=O)N2CCC(C)OC(C)C2)c(Cl)c1 53949,c1(C(=O)NC2C(CNC(C3N(C)CCC3)=O)COC2)cnc2c(c1)CNC(=O)N2 53950,c1(C(N(CCC(=C)CNC(C2CC23CCC3)=O)CC=C)=O)scnc1CC 53951,c1(SC)ccc(CN(C(C(CNC(=O)CC2CC2(Cl)Cl)C2CC2)=O)C)o1 53952,C(=O)(CCC(C)(C)C#N)N1CC(C(=O)NCC(C(=O)NC)O)N(C)CC1 53953,N1(C(C2CCCOCC2)=O)CCOC2(CCN(C(C3CCS(=O)(=O)CC3)=O)C2)C1 53954,c1(C(N(C)C(C2CCCO2)=O)NC2CC2)cccc(F)c1.C12(S(=O)(=O)N1)CC2 53955,O=C(C1=COCCO1)NCC1CC(F)CN1C(=O)CCCC1CCCC1 53956,Cc1nocc1C(N1CC(O)(CC(=O)NC(C2CCCC2O)C)C1)=O 53957,N1(C(C(C2CCN(C(C(CCC)OC)=O)CC2)C)=O)CCC(C)C(F)(F)C1 53958,C1(CCNC(C=CCNC(COC(CC)C)=O)=O)COCC1O 53959,C(=O)(C1=C(Cl)CCC1)NCC(CC(=O)NCCC(C)CO)C1CCC1 53960,c1(CC(N2CC(NC(C(COCC)C)=O)C(C#N)C2)=O)nc2cc(Cl)ccc2s1 53961,C1(CNC(CC2(CSC)CC2)=O)CCCN(C(c2[nH]c(C3CC3)nc2C)=O)C1 53962,c1(NC(C2CCN(Cc3ccc(I)cc3O)CC2O)=O)ccc(F)c(CO)c1 53963,C1(Oc2cn(NC(C(=O)OCCC(N)=O)=O)nc2)CCCOC1C(C)(C)C 53964,C1(C(N(C(CNC(c2ccc(C(C)=O)cc2)=O)C)C)=O)CC12CCS(=O)(=O)CC2 53965,c1(CCC)cc(C(=O)NCCC(C)(C)NC(C2CCC2(OC)OC)=O)n[nH]1 53966,C1(CNC(CCN(CCC)C)=O)CCCCC1NC(c1cccc(C(F)F)n1)=O 53967,C#CC1CC2CC1CN(C(=O)NC1CC3OC(=O)OC3C1C(=O)OCC(C)(C)C)C2 53968,C1(C(N(CCCNC(=O)CCc2nccs2)CC)=O)CNC(=O)CC12CCOC2 53969,c1(C(C)NC(c2cccc(Br)c2)c2nccn2C)ccc(F)c(F)c1F 53970,Cc1cn2cc(C(N3CCC(F)C(NC(c4ccc(O)cc4F)=O)C3)=O)sc2n1 53971,CCC(C)(C(=O)NCCCN(C(=O)C(F)(F)C1(OC)CCC1)C)C(F)F 53972,N1(C(C)=O)CSCCC1C(N1CCN(Cc2nc(C3CCC3)no2)CC1)=O 53973,CCC(C)C(O)C(C)C(=O)NCCCNC(=O)CN(C)C1CC1 53974,C1(N(C(c2nc(C(C)(F)F)sc2)=O)C)C2CN(C(c3nc(C(N)=O)cs3)=O)CC12 53975,CC1CN(C(c2ccncc2Sc2ccccc2)=O)CC1NC(=O)C(C)(F)F 53976,C#CC(C)(CC)NC(=O)C(CC)NC(=O)Cc1sccc1C 53977,n1(CC(CC)O)cc(C(=O)NC2CCC(CCNC(c3cnc(C)s3)=O)C2)nn1 53978,C#Cc1ccnc(C(N2CCCC2CCC(N2CC3CCC3(C)C2)=O)=O)c1 53979,S(=O)(=O)(c1ccc(C#N)cc1)NCC=O.CC1CN2CCN12.c1(SCC)ncccc1F 53980,N1(C(c2c(N)cccc2Cl)=O)CCN(c2nccc(-n3ccnc3)n2)CC(O)C1 53981,c1(C(=O)NC2CN(C(C(C3CCCOC3)OC)=O)C2)nonc1N 53982,C1(NC(C2CCC(F)(F)C2)=O)CN(c2ccncc2[N+](=O)[O-])CCC12CCC2 53983,C1(CC)(CC)C(Cc2cccs2)CC1NC(=O)Cc1csc(C(F)F)c1 53984,C1(F)(C(=O)NCC2(O)CN(Cc3c(OCC(=C)C)cccc3)C2)CCC(F)(F)CC1 53985,C(=O)(N=c1ccn(CCCO)[nH]1)C1N(C(c2ccc(COC)cc2)=O)CC(C)C1 53986,C1(C(=O)NC2CCC(Cn3cc(Cn4cccc4)nn3)CC2)(CC)CCCCO1 53987,N1(C(c2cc(C)c(O)cc2)=O)C(C(N2CCC([N+](=O)[O-])CC2)=O)C2CC(O)C1C2 53988,C(=O)(CC(CNC(c1c[nH][nH]c1=N)=O)C1CCC1)N(CCCO)CC#C 53989,c1(OCCCC(=O)N(CC(C)NC(=O)OC)CC)ccc(SC)cc1Br.OC 53990,C(=O)(C1=CCC(C)(C)CC1)NC(CNC(c1c(C)c(F)cnc1)=O)C1CC1 53991,C1(C)(C(=O)NC2C(NC(C3OCCC(C)C3)=O)COCC2)CC(=O)N(C)C1 53992,C(=O)(C1CCCc2ncnn21)NCc1ccc(C(C)NC(=O)CC2=CCCC2)cc1 53993,c1(NC(CC2C(NC(C3N(CC)CCC3)=O)CCCC2)=O)ccc(F)nc1 53994,c1(C(=O)NCC(c2ccc(C)cc2)O)coc(S(C)(=O)=O)c1 53995,C1(NC(CNC(C(CC)C)=O)=O)CCCCN(C(C2(C)CC2C)=O)C1 53996,Cc1cc(C(N2CC3C(CNC(=O)CSC4CC4)C3C2)=O)c2sc(=N)[nH]c2n1 53997,CCC(C)CN(C)N(CCCOC)CC(=O)OC.C12CCCCN1C(=O)N2 53998,N1(C(CCC=C)=O)CCC(NC(C2CC(=C(F)F)C2)=O)C(F)C1 53999,c1(N2CCC(C)COCCC2=O)ccccc1.C1(CC(=O)NCC)C=CCCC1 54000,Cc1cc(Cl)c(C(N2C3CCC2C(NC(=O)CCn2ccnc2C)C3)=O)cc1N 54001,C1(CCC)CC(O)C(O)CC1C(=O)NC1(C)CCC1 54002,CCC(CC(C)C)C(=O)N1CCCC(C)(CNC(c2ccc(CF)cc2)=O)C1 54003,C(C)(CN=c1[nH]c2c(c(=NCCCN=c3cc[nH]c4ccccc34)[nH]1)CSC2)SC 54004,C(=O)(CCCCCO)NCC1(OC)CCOCC1.c12cc(no1)C(=O)NC2 54005,CCC(C)(C(=O)N1CCCC(COC)(NC(c2ccc(Cl)c(C)c2)=O)C1)C(F)F 54006,C1(C(N2CCC(NC(c3ccnn3C3CCC3)=O)(CF)C2)=O)CN2CCC1CC2 54007,c1(OC)cc(N)ccc1-c1cn(CCC(=O)NCC(C)(C)OC(F)F)nn1 54008,N1(C(C(C=CC)O)=O)CCCC2(CCCCC2NC(c2cc(C)c(C)cn2)=O)C1 54009,c12cc(Br)ccc1CC1CCN(C1)C2=O.c1(CNC(C)=O)ccc(F)cc1F 54010,c1(C(=O)NC2C(NC(Cc3c(C)ncs3)=O)C2)cc([N+](=O)[O-])cn1C 54011,N1(C(CCCC(C)=O)=O)CC2(CC(NC(=O)CN3CCS(=O)(=O)CC3)CO2)C1 54012,C1(NC(CN(C(CCOCC)=O)CC2CC2)=O)CCOC(C(C)C)C1 54013,C1(C(=O)NC(CNC(C(CC(=O)OC)C)=O)C)Cc2ccccc2C1 54014,c1(CC)nc(C)[nH]c1C(=O)NCC1COCCN1C(=O)C(C)Sc1ccccn1 54015,N12CCC(C(O)C1)C2=O.N1(CC(=O)NCCn2cncn2)CC2CC2C1 54016,c1(C(=O)NC(C(C)NC(C2(O)CCCCC2)=O)CO)ccc(Cl)c(C#N)c1 54017,CC(C(=O)N1CCCC(CNC(=O)COCCF)CC1)C(C)(F)F 54018,Cc1cc(C(=O)NCCCCNC(c2cncc(C(N)=O)c2)=O)sc1Br 54019,C1(C2CCC2)(C(=O)NC2C(NC(C3(C(F)F)CCCO3)=O)CCC2)CC1 54020,N1(C(C(C)OC)=O)CCCN(C(c2cc(C)n(C(C)(C)C)n2)=O)C(C)C1 54021,CC(C)C(CC(=O)NC12CC(CNC(c3ccnc(S)c3)=O)(C1)C2)C(C)C 54022,C1(N(C(=O)CCC2NC(=O)NC2=O)C)CCCN(C(=O)CCc2cnoc2)CC1 54023,O=C(CC(C(F)(F)F)c1ccon1)N1CC2(C1)CN(C(=O)CCn1cncn1)C2 54024,c1(-c2cn(C3(CC(CCC)NC(=O)C4=C(C)OCC4)CC3)nn2)cnc(N)c(N)c1 54025,c1(C(N2C(CN(C(C(C=C)(C)O)=O)CC)CC(F)C2)=O)nccc(C)c1F 54026,C1(C(N(CCc2cc(C(=O)NCCC3CC3)cs2)CCSC)=O)CC(=O)N(OC)C1.CO 54027,N1(C(N(CC#CC)CC#C)=O)CCc2cccc(Br)c2C1C 54028,c1(C(N2C(C(C)(C)C)C(NC(C3CC(CF)C3)=O)CC2)=O)csc2ccncc12 54029,c1(CC)ccc(C(N2CCN(C(=O)CCCCCOC)C3CC23)=O)cc1[N+](=O)[O-] 54030,c1(C(=O)NCC(CCNC(Cc2cn(C)nc2)=O)(C)C)c[nH]c2ncccc12 54031,C1(NC(CCC2C(C)C2)=O)CCN(C(c2ccc(OC(F)F)cn2)=O)C1(C)C 54032,N1(C(c2ccn(CC(F)F)n2)=O)CCN(C(c2cnc(C(F)F)s2)=O)C(CF)C1 54033,c1(NC(=O)NCC(=O)NC(CC)CNC(=O)C2CC2)cccc(C2CCOC2)c1 54034,c1(CNC(=O)CC2CC2)cc(NC(C2(C3CCCO3)CCC2)=O)n[nH]1 54035,CCCC(CC)CC(=O)NC1CCN(C(c2ccc(C)cc2)C)C1 54036,C=C1CC(C(=O)N(CCCCO)C(C)(C)C)(CNC(=O)OC)C1 54037,N1(C(C2C(NC(CCCCC#C)=O)CCOC2)=O)CC(O)CCC(C)(C)C1 54038,c1(NCCC(C)(C)SC)cc(C)c(S(=O)(=O)NC(c2ccn(C)n2)C)cn1 54039,C1(CC(=O)N(CCO)CCO)OCC2CCN(C(=O)CCc3ccccc3)CC12 54040,CC(F)(F)C(F)C(=O)NCC1CN(C(=O)CN(C2CCC2)C)CC1O 54041,c1(C(=O)NCC2(O)CCN(C(Cc3cnc(C)[nH]3)=O)C2)cc2cc(Cl)ccn2n1 54042,C#CCCC(O)C(=O)NC1COCCN(C(c2ncc(C)cc2C)=O)C1 54043,C(CCCCNC(c1c[nH]nc1F)=O)N(C)C(c1cnn(CC2CCCO2)c1)=O 54044,N1(C(C(C)(C)C2CC2)=O)CC(NC(c2cccc3c2NCC3)=O)C(S(C)(=O)=O)C1 54045,C(C1CCCN1C(=O)CCN1CCCCC1)=CC(N1CC(N(C)CC)C1)=O 54046,C(N=c1ccc(Br)c(C(C)C)[nH]1)c1cccc(OC)c1F 54047,C(c1ccc(F)cc1Cl)=CC(N1CC(C(C)C)N(C(c2ccn(C)n2)=O)CC1)=O 54048,C1(NC(=O)NCCCN2CCCC2=O)CC1C1CC1 54049,c1(C(N(C2CCOCC2)C)=O)cccc(CCO)c1.C1(=O)C(CC2(C#N)CC2)N1 54050,N1(CCCN(CCOCCN(C(C)=O)C)C)CC(C)(C)OC2(CCCOC2)C1 54051,c1(C(N2CC3(CN(C(CC(=O)NCC#C)=O)C3)C2)=O)cc(S(N)(=O)=O)cs1 54052,N1(C(CCC(CC)C)=O)CCCN(C(c2cnc(CC3CC3)s2)=O)CCC1 54053,N1(C(c2cc(CCC)n(C)n2)=O)CCC(C)C(NC(c2ocnc2CCC)=O)C1 54054,c1(-c2cc(C)c(OCC(C)C)nc2)ccc2[nH]c(NCc3cc[nH]n3)nc2c1 54055,C1(C(=O)NCc2cnsc2)(CNC(CC(C)n2ccnc2)=O)CCCCC1 54056,C(=O)(C(F)CC(C)(C)NC(c1ccns1)=O)NC1CCN(C)C1=O 54057,c1(CC(=O)N(C2CCN(C(c3cccn3C)=O)C2)CC)ccc(Cl)c(F)c1 54058,c1(OCC)ccc(F)c(C(=O)NC2CCCC2CNC(=O)COCCN(C)C)c1 54059,Cn1cc(Br)c(C(C(=O)NC(C)(C)C)N(CCC=Cc2ccccc2)C)n1 54060,Cc1ccnc(-c2cccc(C(C)CS(=O)(=O)Oc3ccccc3)c2)n1.C(C)(C)O 54061,CC1CCC(NC(=O)CN2CCN(C)CC2)CN1C(=O)CCc1cc(Cl)no1 54062,[N-]=[N+]=NCCCOCC(N1CCCC1CCCNC(C1CC1NC(=O)OC)=O)=O 54063,C(=O)(CCCCC(=O)N1CCN(C(c2cccc(OC)c2)=O)CC1C1CC1)NC 54064,CCCC(C)(O)CC(=O)N1CCCCC(NC(c2nc(C(F)(F)F)cs2)=O)C1 54065,N1(C(CNC(CC)=O)=O)CCCC(C2CCCN(C(C3COC(=O)O3)=O)C2)C1 54066,CCCCCC=CC(=O)NCC1CC1.N12CCC(C1)C2.C1(C(=O)N)(C(=O)OC)CC=CC1 54067,n1(CC(N2CC(N(C)C)C2)=O)cc(CNC(=O)C(O)C2CCCC2)nn1 54068,N1(c2nn3cc(C)nc3s2)CCC2C(CCCN2n2ncc3ccccc23)C1 54069,n1(CC(=O)N(CCC2CN(C(C)=O)C2)C(C)C)cc(C)cn1 54070,c1(CC(N2C(CC(=O)NCC3CC(N(C)C)C3)CC2)=O)ccc(O)c(F)c1 54071,C1(NC(COC(c2nccn2C)C)=O)CCN(C(c2occc2F)=O)CC1F 54072,C1(N(C(=O)COCC2CCC2)CC#C)CCN(C(c2csnn2)=O)CC1 54073,C1(NC(CCCC=C)=O)CCN(C(C2CC3(CSC3)C2)=O)C(c2ccccc2)C1 54074,c1(Cc2nc(-c3cccc(C(C)(C)C)c3)nn2CC(F)(F)F)c(F)cccc1Cl 54075,C(CCCCCCCC(=O)NCCO)n1cc(C(C)OC(C)(C)C)nn1 54076,CC1CC2CC2CC1C(=O)NC1CN(C(=O)C=Cc2cncs2)CC1(C)C 54077,C1(N(C(CC(=O)NCC)=O)C)CS(=O)(=O)C12CCN(C(C1CCCCC1)=O)CC2 54078,N1(C(C2(CC)CC2)=O)CCN(C(c2ccc(C(F)F)o2)=O)C(c2cccnc2)C1 54079,C(=O)(C1=NOC2(CCC2)C1)N(CC(CC)NC(=O)Cc1ccc(Cl)nc1F)C 54080,C(CCCCCCNC(c1ccco1)=O)n1cc(COCC)nn1 54081,C1(C(N2CCC(CC(C)NC(C(C=C)O)=O)CC2)=O)Cc2ccccc2C1 54082,c1(CC)cc(N)ccc1C(=O)NCC1CCC(NC(c2cnoc2C2CC2)=O)C1 54083,C(=O)(C(F)CC(C)(C)NC(=O)CC(C)(C)CN(C)C)Nc1c(CC)noc1 54084,C1(CCC)CC1N=c1[nH]c(=NCc2ccc3scc(C)c3c2)[nH]c2cc[nH]c12 54085,c1(C(=O)NCC2N(C(CCC(C)OCC)=O)CCC2)ccc(S(N)(=O)=O)cn1 54086,C1(NC(C2CC(F)CN2C(=O)C2CC2)=O)CCN(CCOC2CCCCC2)CC1 54087,N1(C(CSCCOC)=O)CCCCC(C2CN(C(c3cc(C(C)=O)cs3)=O)C2)C1 54088,Cc1n[nH]cc1C(=O)NC1CC(O)C1CC(=O)NCCC(C)(C)C1CC1 54089,c1(N2CCC(NC(c3ccc(CC)nc3)=O)C2)c(Cl)cncc1[N+](=O)[O-] 54090,CC1CCN(CC(=O)NC2(CF)CCN(C(=O)CC3CCCCN3C)C2)CC1 54091,C12=NC3=C(C(=NCC4CN1C4)N2)CCC3.Cc1cc(N(N2CCOCC2)C)no1 54092,Cc1cc(C(N2CCN(C(C3CCCCC3O)=O)CC2C)=O)ncc1C#N 54093,C1(CCNC(CC(C)C)c2ccccc2)(CO)CCN(C(=O)OC(C)(C)C)CC1 54094,C1(OC)CN(C(=O)C(O)CNC(C2CC2C(N)=O)=O)CC12CC2 54095,C(=O)(C1CNc2ccccc21)NCC1C(CNC(CC(C)(C)SC)=O)C1 54096,N1(C(C2(COC)CN(C(=O)CC(C)(C)CC(=O)OC)C2)=O)CCc2c(F)cccc21 54097,N1(Cc2cccc(C)c2)CCC2(CC1)CC2C(=O)Nc1c(Br)ccc(F)c1F 54098,N1(C(C2C(C)CCC2)=O)CCCC(CCNC(=O)COCC2CCOCC2)C1 54099,c1(CC(=O)NCC2(F)CN(C(=O)C(C3CCCCC3)O)C2)cc(F)ccc1Cl 54100,c1(NC)ncccc1C(N1CC(NC(=O)Cc2cscc2F)C(C)C1)=O 54101,C#CC1(C(=O)Nc2ccc(OC)cn2)CCN(C(C2CC(=C)C2)=O)C1 54102,C1(NC(CC2(C)CC2)=O)CC(NC(C2(C3CCCCO3)CCC2)=O)C12CCC2 54103,c1(-c2cn(CCCN(C(=O)C(N3CCCC3)C3CC3)C)nn2)c(F)cccc1Cl 54104,n1(NC(=O)NCCOCCN(C)CC)nccc1C 54105,c1(C(N2C3CC(C(=O)NCCOCCCC)C(C3)C2)=O)cn2cc(C)ccc2n1 54106,c1(C(N2CCCC2)=O)cc2c(s1)CCC21CCCO1.c1(N)cc2n(n1)CCCO2 54107,CC1CN(C(=O)CCOC2CCC2)CC1CCNC(=O)CC#N 54108,C(C(C(=O)NCC12CCC(CC1)CC2)C(C)C)NC(C(C(C)C)OC)=O 54109,N1(C(C2C(=O)NCCC2)=O)CC2(CNC(c3ccn(CCF)n3)=O)CC1CO2 54110,c1(C(=O)NCC(CNC(c2cccs2)=O)OC)cc2ccc(F)cc2o1 54111,c1(OC)ccc2[nH]c(C(=O)NCC3CCN(C(=O)CC(C)O)CC3O)c(C)c2c1 54112,N1(C(C(C)=C2CCC2)=O)CC(NC(c2cc3sccc3s2)=O)CC(F)C1 54113,C1(C(N(CCOC)CCNC(c2ccnc(C3CC3)c2)=O)=O)CCCN(C)C1C 54114,CC(C)CC(C(=O)NC(CC(C)(C)C)C(=O)NCc1ccccc1CO)C(C)C 54115,C1(CN(C(C)(C)CNC(=O)OC(C)(C)C)CCC)CC(=O)N(CC)C(C)(C)C1 54116,c1(C(C)OC)nc(CN(C)CCN(C)C(c2sccc2C2CC2)=O)cs1 54117,C1(N(C(c2ccc(-c3ccc(F)cc3)s2)C(=O)NCCI=O)C)CCc2ncnn2C1 54118,CN1C(=O)CCC1C(N1CCCCC1CCNC(=O)C=CCN1CCCC1)=O 54119,C1(NC(C=NOC)=O)CC2(CCN(C(C34CCCC3(C(N)=O)C4)=O)CC2)C1 54120,C1(C(=O)NC(CC(C)NC(N)=O)C)CCN(C(=O)CCOc2ccccc2)CC1 54121,c1(C(=O)NCC2(NC(=O)C=Cc3ccoc3)CC2)ccc2cncn2c1 54122,C1(O)(CNC(C(CC)(C)C)=O)CCCN(C(=O)CC2CCCC(C)(C)O2)CC1 54123,O=C(N1CC(O)C(O)CO1)C1CNCCC1(F)F 54124,C(C1=CCCN(C(=O)C(C)NC(C)=O)C1)NC(C(CC)(C)C)=O 54125,C1(N(C(c2c(CC)n(C)nn2)=O)C)CCN(C(=O)CC2CC2)CC12CC2 54126,N1(C(COC(CC)CC)=O)CCN(C(C2CCCN2C2CC2)=O)C(CC2CC2)C1 54127,CC1CC(C)N(C(c2nn3c(c2C)CCCC3)=O)CCN1C(=O)Cc1cccs1 54128,c1(NC2C(OC)CCCC2)ncnc2c([N+](=O)[O-])cccc12 54129,C1(c2nnnn2CCCF)(NCC(CC)C)CCC(NC(=O)OC(C)(C)C)C1 54130,c1(CCN(C(CC2(NC(COCC(=O)NC)=O)CC2)=O)C)cccnc1 54131,C(c1cn(C)nn1)=CC(=O)NC1(CNC(C2C(C)C2)=O)CC1 54132,C=C(C)C1CCC(C)=CC1CC(=O)NC1CCN(C(c2ccc(Cl)cc2F)=O)C1 54133,C(=O)(C1=C(c2ccccc2)CCC1)NCC1C(NC(=O)C=CC2CCC2)C1 54134,C1(O)(C(=O)NCCC(=O)OC(C)(C)C)CCN(Cc2cccc(O)n2)CC1 54135,C=C=CCCC(=O)NC1CCN(C(=O)CSCc2ccncc2)C1 54136,N1(C(CN(C)C2CC2)=O)CCCC(C2N(C(c3cnc(O)o3)=O)CC2(C)C)C1 54137,n1(CC)cc(C(=O)N(C)CC2CCN(C(=O)C(C)OC3COC3)C2)nn1 54138,Cc1ccc2c(C(=O)NCC(O)CN(C(=O)C(C)C3CCC3)C)coc2c1 54139,c1(C(N2C(CNC(=O)C3=CCSC3)CCC(C)C2)=O)ccc2c(c1)CCC2 54140,Cc1cc(-c2cccc(C3CC3C(=O)Nc3ccc(Cl)nc3Br)c2)cnc1C#N 54141,C(=O)(C(C)(F)C(C)(C)F)N1CC(CN(C)C(c2cn3cnnc3cn2)=O)OCC1 54142,n1(CC)cc(Cl)c(C(=O)NCC2CCCN2C(c2sc(C)cc2C)=O)n1 54143,c1(C(=O)OCc2ccco2)cc2ccccc2cc1O.c1(S)cc(Cl)ccc1F 54144,C(=O)(C(CC1CCCC1)NC(=O)C=CCN1CCC1)NCCCCSC 54145,C(=O)(CCCCC(=O)N(C)C)NC12CCN(C(C(=O)NCCOC)=O)CC1C2 54146,CC(C)CC(C(=O)N(C1CCC1O)C)ONC(C1CCC1(C)C)=O 54147,C1(NC(c2nnnn2C)C2CC(CC)C2)Cc2ccc(Br)cc2C1 54148,N1(C(C2(NC(C(COC(C)=O)C)=O)CCN(C)C2)=O)CCC2OCCC2C1 54149,Cc1nc(C)c(C(N2CCCC(CNC(c3cccc(O)n3)=O)CC2)=O)nc1C 54150,c1(C(=O)NCC(C2CCN(C(C3C(CC)OCC3)=O)CC2)F)c(C)cc(C)nc1Cl 54151,C1(CNC(CC2C(C)(C)C2)=O)CN(C(=O)Cc2ccc(Cl)s2)CCC12CCC2 54152,C(c1cncc(F)c1)=CC(N1CC(C)C(NC(=O)CC2CCCCC2(F)F)C1)=O 54153,CC(C)C(C)(CNC(c1cnc(N)cn1)=O)NC(=O)CC1(C(F)(F)F)CNC(=O)C1 54154,c1(CCC(=O)NCC(C)(C2CC2)NC(C(C)OCCCC)=O)c(C)n[nH]c1C 54155,c1(NC(C(CC(CC(=O)OC)O)CNC(=O)OC(C)(C)C)CC)cnn(C)c1C#N 54156,C(CC(C)C)(C(=O)NCC(C(C)(C)C)NC(=O)CC(O)C1CC1)NC(C)=O 54157,C1(C(N2CC(CNC(c3ncccc3F)=O)C3(C2)CC3)=O)CC2(C1)CC(F)(F)C2 54158,N1(C(C(C)N(CC)CC)=O)CCC(NC(=O)C(CO)OC)C1C 54159,N1(c2nc(C)nc3c2cc[nH]3)CCCC2(CCCO2)CC1 54160,C(CN=C(NCC(C)N(C)C)NCC1CC1C1CC1)SC 54161,C(C1=CCN(C(c2cnn3c2CCC3)=O)CC1)NC(=O)CCN1CCC1 54162,C(=O)(C1CCCn2cnnc21)N(CCNC(c1ccc(CC)nc1)=O)C1CC1 54163,C1(CNC(=O)OC(C)(C)C)CC2CC2N1C(=O)C(O)Cc1ccccc1Cl 54164,Cc1nn(C)cc1C1CC1C(=O)NCCCNC(C1CC2CCC1O2)=O 54165,c1(C(=O)NCC2N(C(Cc3c(C)n(C)nc3)=O)CCCC2)nn(C)c2c1CCC2 54166,C(C(C)C)(C(O)C(=O)NCC1CCOC1C(=O)N(C)Cc1ncco1)OC 54167,C1(C)(C(=O)NC(c2cccnc2)C(=O)NCC(CC)(C)Cl)CC(F)(F)C1 54168,C(=O)(C1=CC2CCC(C1)C2)N1CCCC(C(=O)OC)(Cn2cc(COC)nn2)C1 54169,C1(C)(C(N(C(C)CNC(C2CC2C(C)(F)F)=O)C)=O)CCCC1 54170,Cc1nccc(C(=O)NCC(CO)NC(=O)CSCC(c2ccccc2)=O)c1O 54171,N1(C(C(COC)O)=O)CC(NC(c2ccc(F)s2)=O)C2CCCCC12 54172,CC1=C(CNC(=O)C(c2ccco2)NC(=O)OC(C)(C)C)S(=O)(=O)CCO1 54173,C1(CC)CN(C(c2c(Cl)csc2Cl)=O)CCC1NC(c1cn(C)nc1Cl)=O 54174,C12CC(C)(C1)NC(=O)C2.C(=O)(C(N)=O)N(CCCN(C)C)C 54175,N1(C(C2C(CCOC)C2)=O)CC23CCCC2(C1)CN(C(C1CCC(OC)C1)=O)C3 54176,C1(Cc2ccc(C(C)(C)C)cc2)CCN(S(=O)(=O)N2CC=CC(N)C2)C1 54177,c1(C(=O)NCC2N(C(C(C(=O)OC)C)=O)CC(C)(C)C2)cccc2c1cnn2C 54178,C1(C)(C(N(CCCCN(C(=O)C(c2ccccc2)O)C)C)=O)CC(C#N)C1 54179,c1(NC(C(=O)NC(CC=C)CO)=O)ccc(OC(F)(F)F)c(Cl)c1 54180,C(=O)(CC(F)(F)CCN(C)C(=O)OC(C)(C)C)OC(c1ncccc1O)=O 54181,C(=O)(C(C)(C)C(N)=O)NCC1CNC(=O)c2c(cncc2)O1.CCS 54182,C1(C(=O)NC2CCN(CCNC(c3ccc(F)nc3)=O)CC2)Cc2nncn2C1 54183,N1(C(CSCC)=O)CCC2CN(C(c3ccc(OC)nc3C)=O)CCC2C1 54184,c1(C(=O)OC)cccc(C(=O)NCC(C)(C)CNC(=O)CCF)c1C 54185,c1(C(N(CCCNC(C2CN(C(=O)NC)C2)=O)C2CC2)=O)ccc(C)c(F)n1 54186,CCC(C)(C)CCCC(=O)N1CC(NC(c2cnc(S)[nH]2)=O)C2(CC2)C1 54187,C1(CCC#C)CCCN(C(=O)CCCC2(NC(c3cnc(=N)[nH]c3)=O)CCC2)C1 54188,c1(C(=O)NC2N(C(CCC(=O)OC)=O)CC3(CC3)C2)c(C)cc(Br)c(C)c1OC 54189,CCC(CNC(=O)CN1CCC(C)CC1)(CC)NC(=O)Cc1c[nH]nc1C 54190,CC(CNC(=O)C(c1ccccc1)=O)C(F)C(=O)NCc1c(F)cncc1F 54191,N1(C(C(C)=C2CCC2)=O)CC2CCC(CNC(c3n[nH]c4c3NCCC4)=O)(C2)C1 54192,CS(=O)(=O)CCC(=O)NC1CCN(C(c2csc(-c3cccnc3)n2)=O)C12CC2 54193,n1(CCCC)nnnc1C(C1(C)COC1)NCc1ccn(CC(F)F)n1 54194,CCCCCC(F)C(=O)NCC(c1ccccc1)NC(C12CC(C)(C1)OC2C)=O 54195,CC1(C)CC(CC(=O)NC2COCCC2NC(=O)CCC2CC3CCC2C3)CO1 54196,C1(CC)CCC(C)CN1C(c1cn(CCNC(=O)CCSC)nn1)=O 54197,Cc1coc2ccc(C(=O)N(CC(C)NC(c3cc(Cl)cc(F)c3F)=O)C)cc12 54198,c1(C(N2CCCC2=O)CC)nnc(N2CCCC2)n1CCCC1COCCO1 54199,N1(C(c2cc(C)nc3n2ncc3)=O)CCCC2CN(C(C3(C4CC4)CC3)=O)CCC12 54200,Cc1[nH]c2ncccc2c1C(N1CCOC(CNC(=O)C(O)CC(F)(F)F)C1)=O 54201,C1(CCOC)(NC(=O)C(C)Cc2cnco2)CCN(C(=O)CSS(C)(=O)=O)CC1 54202,C1(NC(CCC)=O)CS(=O)(=O)C12CCN(C(c1c[nH]c(C)cc1=O)=O)CC2 54203,c1(C(N2CC(CNC(C=NOC)=O)C(O)C2)=O)c(N)c(F)cc(F)c1F 54204,C(C(C)C)(C(O)C(=O)NC1CC(N(C(=O)CCc2cc(C)no2)C)C1)OC 54205,N1(C(c2ccn(CC)c2C)=O)CC(CC(=O)NOCC=CCl)C2(CC2)C1 54206,C1(C)(C(N(CC=C)CCC)=O)CN(C(C2CCC(COC)C2)=O)CC1C 54207,n1(CCC)nnnc1C(c1cc(C)[nH]n1)NCCc1cnoc1 54208,CC(CN(C(=O)CC1CCCO1)C)C(=O)NC(C=C=C)C(=O)OC(C)(C)C 54209,C1(C(=O)NC)C2CCC(C2)C1NC(COC(C)=O)C(C)(C)C 54210,CCC(CC(=O)N1CC(=C(F)CNC(=O)CSC(F)(F)F)C1)C(F)F 54211,CCCC(CC)CCCC(=O)N1CC(C)CN(C(=O)CC2CCOCC2)C(C)C1 54212,C(=O)(C(CCCC(C)(F)F)N1CCC2(C)C(F)(F)C2(C)C1)NCCCOC 54213,C(=O)(CN=c1cc[nH]cc1)N1C(C(=O)NCC2N(C(C)=O)CCC2)CCCC1 54214,C(=O)(C(C)C(=O)NC(C)(C)CC=CC(=O)Nc1cncnc1O)OC 54215,C(=O)(C1CNC(=O)c2ccccc21)N1C(CNC(C2(C(C)C)COC2)=O)CCC1 54216,C(=O)(CCCCCS(N)(=O)=O)NCC1(O)CCN(C(c2cc(C)nc(C)n2)=O)C1 54217,C1(CNC(C2(Cl)C(C(=O)OC)C2)=O)CCCC1NC(C1CCC(C(N)=O)C1)=O 54218,c1(C(=O)N)cc(C)cc(O)c1.c1(OC)cnc(C(=O)N(CC(C)O)CCOC)cn1 54219,CC(CC(N)=O)C(=O)NCC1(C)CCCN1C(c1cc[nH]c(=N)c1)=O.C(C#N)O 54220,c1(C(=O)NCC2CCN(C(C(CC)F)=O)C2)cc2cscc2s1 54221,Cc1c(N)ccc(C(=O)NCC(C)CNC(=O)COc2ccc(F)c(F)c2)c1Cl 54222,C(CCCCCF)NC(C1CCOC1CNC(c1cncc(F)c1)=O)=O 54223,c1(CC)ncc(Cl)c(C(N2CC(N(C)C(c3ncc(F)cn3)=O)C(F)C2)=O)n1 54224,N1(CC)CCC(C(=O)NCC(=O)NC(C(=O)N(CC(=O)NC)C)C2(C)CC2)C1 54225,C1(NC(=O)CC2CCCCN2C(C2CCC3CC2CO3)=O)CCCCCC1F 54226,C1(NC(CCC=C)=O)CC2CN(C(=O)COc3ccc(F)c(C)c3)CCN2C1=O 54227,C1(C(=O)NCC(C(=O)NCc2cccc(C)c2O)OC)CC(=O)CC(=O)N1 54228,C1(F)(COCc2ccc(C(=O)NOC3CS(=O)(=O)C3)cc2)CCCCCC1 54229,CC1CCN(CC(=O)NC2CCCN(C(=O)C(N3CCN(C)CC3)=O)C2)CC1 54230,C(=O)(C(C)(C)C(=O)N1CCC(F)(C(=O)NC(C)CN(C)C2CC2)CC1)OC 54231,Cc1cc(C(=O)N(C2C3CN(C(C4CN(C)CCO4)=O)CC23)C)c(Cl)cc1F 54232,CC1Cc2ccc(C(N3CC4CCC3CN(C(=O)COC3CCC3)C4)=O)cc2C1 54233,c1(C(=O)NCC2CCC(C(=O)Nc3ccc(C)cc3)C2)cc(C#N)cn1C 54234,C1(C(N2CCN(C)C(=O)C2)=O)CC(C)(C)CCN1C(C1CN2CCC1CC2)=O 54235,N1(C(CCCN(C(C)=O)C)=O)CCC=CC1C(=O)NCC1CCCCCC1 54236,N1(C(C2CCC(N(C)C)C2)=O)CC2(CCN(C(c3cn(C)c(=O)cn3)=O)C2)C1 54237,C1(COC)(CNC(c2c(C)noc2C)=O)CCN(C(=O)C(C(C)C)SC(C)C)C1 54238,c1(C(C)=O)cnc[nH]c1=NCC1CC2(CC(NC(=O)CSCC3CCCO3)C2)C1 54239,N1(C(c2c(SCC)cc(Cl)cc2)=O)CCC12CCCN(C(=O)Cc1cccs1)C2 54240,c1(C(N2C(CNC(C(COC)(C)Oc3ccccc3)=O)CC2)=O)cc(Cl)ccc1Cl 54241,CCC(C)C(O)CNC(c1csc(CNC(C2(NC(C)C)CC2)=O)c1)=O 54242,N1(C(C2(N(C)C)CC2)=O)CCOC(CCCN)C1.C1(NC(C)C)CN(C(=O)CO)C1 54243,CC(C)CC(CC(C)C)C(=O)N1CCC(O)C(N(C)C(C2CC(F)C2)=O)C1 54244,c1(C(=O)NCCNC(c2c(C)cc(C)nc2O)=O)sc2[nH]c(C)nc(=O)c2c1C 54245,CC1(C(=O)NCCCC2CCCN2C(c2cnc[nH]2)=O)CCCC1(F)F 54246,C1(C(=O)NCCCCNC(c2coc(C(F)(F)F)n2)=O)(COC)CCCO1 54247,c1(CCC)onc(C)c1C(=O)NCC(CC(C)C)NC(C1CCCN(CC)C1)=O 54248,C1(CC(=O)NC(C)C(C)NC(c2ccccn2)=O)CCCCC12CC2 54249,C1(N2CC(C)(C)OC(C)(C)C2)CCN(N2CCC(=O)CC(=O)N2)CC1 54250,Cc1[nH]nc2c1CC(C(=O)NCC1CCCCN1C(=O)C1=C(Cl)CCCC1)CC2 54251,N1(C(C2(CC#C)CCOC2)=O)CC=C(C(=O)NCC2=CCC2)CC1 54252,c1(C(=O)NC2(C(=O)NCCC(COC)O)CC2(C)C)cccc2[nH]ccc12 54253,c1(C(=O)NCC2C3CN(C(CCC#C)=O)CC32)cccc(P(C)(C)=O)n1 54254,N1(C(c2cncs2)=O)CC(C2CCN(C(=O)CC3CCCN(C(F)F)C3)CC2)C1 54255,c1(OC)csc(C(N2CC(O)(CCNC(C3CSC(C)=N3)=O)C2)=O)c1 54256,CC#CCCCC(=O)NC(CNC(c1nnsc1C(F)F)=O)CC(C)C 54257,c1(C(N2C(C(=O)NCc3cscn3)CCOCC2)=O)cccn2ccnc12 54258,N1(C(C2CCC(C)(C)C2)=O)CCc2[nH]nc(CNC(C3CCOC3)=O)c2C1 54259,CC1CCc2onc(C(=O)NC3CCN(C(=O)C=C(C4CC4)C4CC4)C3C)c2C1 54260,c1(N(CC)CC2CCN(C)C2)cc(N)nc(CC(C)C)n1.C12CC(C1)C2 54261,c1(CC(=O)NCCC2CCN(C(CCCc3onc(C)n3)=O)C2)cccc(F)c1 54262,N1(C(C)=O)CCOC(C(=O)NC2CCC(N(C(=O)C=CBr)C)CC2)C1 54263,Cc1nn(C)c2c(NC3C=CCC3)nc(=NC3CCCOC4(CCCO4)C3)[nH]c12 54264,c12cncc(n1)C(=O)N1CC(C(C)C1)CC(=O)N2CCCO.C(C)(=O)N.CO 54265,C(=O)(CC(C=C)CCC)NCC1CCCC(NC(CSCC#C)=O)C1 54266,C1(C(=O)Nc2c(C)ccnc2)CN(C(c2cccc(Cl)c2I)=O)CC(F)(F)C1 54267,C1(CC)CCCN(C(=NCCC2(F)CCCCC2)NCC(CO)CC(C)(C)C)C1 54268,c1(C(N2CCCCC2CCO)C(=O)NCC=C)ccccc1Br 54269,N1(C(C(c2ccccn2)C)=O)CCCC(CO)(NC(C2CC3C=CC2O3)=O)C1 54270,c1(C(=O)NCC(CC(C)C)NC(=O)CO)ccnc(C(F)(F)F)c1N 54271,Cc1[nH]c(C)c(C(=O)NCC(C)(C2CC2)NC(=O)CCC(=O)NC2CCCC2)c1C 54272,N1(C(C(CCCC)F)=O)CCC2(CC(C(=O)N(C3CC(C(N)=O)C3)C)C2)C1 54273,N1(C(C(C=C)O)=O)CCCN(CCNC(=O)C(C)c2cncs2)CC1 54274,C1(NC(C2CCCC(OC)C2)=O)CCCN(C(c2ccc(N(C)C)cn2)=O)C1C 54275,CCCC(CCC)CC(=O)N(C1CC2CC1N(C(c1ccc(F)c(C)c1)=O)C2)C 54276,C1(C(=O)NCC)Cc2nccnc2C1.CCCCC(O)C(=O)N(CCC)CC 54277,c1(C(=O)NC2CCC(N(C(=O)CN3CCCC3=O)C)C2)n[nH]c2c1CCSC2 54278,c1(NCC=CC)cc(C)c(S(=O)(=O)N2CCOC(c3ccccc3Cl)C2)cn1 54279,C1(CNC(CCN(CCC)C)=O)(CNC(=O)C(C)CO)Cc2ccccc2C1 54280,CC(C)CC(CNC(=O)CC1CC2(CCC2)C1)NC(=O)CCc1cccc(Cl)c1 54281,N1(C(c2cc(COCCC)on2)=O)CCN(c2ccc(F)cc2)CC1 54282,N1(CCN(CCC(CC)O)C(=O)Nc2ccccc2)CCSC(C)(C)C1 54283,Cc1cccc(CCC(=O)NC(C2CN(C(C3CCCN(C)C3)=O)C2)C)c1 54284,N1(C(c2cn(CC(C)C)nc2)=O)CCC(N(C(=O)CN2CC=CC2)C)C(C)C1 54285,N1(N(C(c2ccc(CC)o2)=O)CCC2CC2)CC(C(=O)OC)C2(CC2)C1 54286,CC(C)C(CNC(C1CNC(=O)N1)=O)C(=O)N(C1CCOCC1)C 54287,c1(CC)cccc(NC(C2CCC(CN(C)C)CC2)=O)c1.C12CCCN1C2=O 54288,c1(C(N2CCCC(CCCO)C2)C(=O)NCCOCC)nc(C)[nH]c1Br 54289,Cc1cc(C(=O)NCCOC2CCN(C(=O)CC(C)C)C2)c(C)n1C1CCOC1 54290,n1(CC)ncc2c1CC(C(N1CCC3(C1)CN(C(=O)C=CC(C)C)C3)=O)CC2 54291,c1(N(C)NCc2ccc(C)cc2)cc(NC2CCC3CC23)nc(C(C)C)n1 54292,C1(NC(C(C2(O)CCC2)NC(C=C(C)C)=O)=O)COC(C(F)F)C1 54293,N1(C(c2n[nH]c(CC)c2Cl)=O)CC(C)C(NC(=O)CN(S(=O)(=O)CC)C)C(C)C1 54294,C1(C(=O)NC2CCC(N(C)C(C34C(=O)C5CC3C4C5)=O)C2)CC1C1CCOCC1 54295,c12cccc(F)c1C(=O)NC1CN(CC1F)C2=O.CC1(C(F)(F)F)CC1C(=O)O 54296,CCC(C)C(O)C(C)C(=O)N1CC(OC)CC1C(=O)NCc1ccc(F)c(Cl)c1 54297,S(=O)(=O)(c1ccsc1)Nc1ccc(CC2(C)CCN2Cc2cccnc2)cc1 54298,C(CCC)(C(=O)NC1CCOC(c2ccc(Cl)cc2)C1)=CCC 54299,c1(CNC(Cn2c(C)csc2=O)=O)nc(CNC(c2csc(Cl)n2)=O)cc(O)n1 54300,C1(N(C(C(C2CN(C(C(N)=O)=O)C2)O)=O)C2CC2)CCC(=O)NC1 54301,c1(N(C)Cc2nc(-c3ccc(C)cn3)sc2)cc(N(C)C)nc(C)n1 54302,c1(-c2ccnc(C(N)=O)c2)ccc(O)c(C)c1C.n1(CC)ccnc1CN 54303,c1(N(C2(CC=C)CC2)C)ncnc2c1ncn2CC(CC)(CC)CS(C)(=O)=O 54304,C#CCC(C(=O)NCc1nn(C)cc1Cl)NC(=O)CCCCN(C)C 54305,Cc1nc2cccc(C(=O)N(CC(C)NC(c3cc4c(s3)CCCC4)=O)C)c2[nH]1 54306,c1(C(=O)Nc2ccc(NC(C(COCC)C)=O)c(C)c2)c(C)[nH]c2ccccc12 54307,c1(C(=O)NC2CC3(C(NC(C(C)Cc4ccnn4C)=O)C3)C2)ccc(Cl)c(O)c1 54308,N1(C(c2cnc(CC)s2)=O)CC(NC(=O)CC2CC(C)(C)CO2)C2(CCCC2)C1 54309,c1(C(=O)NCC(CNC(c2cnccn2)=O)O)ccn2ccccc12 54310,C1(C(N2CCN(C(C3(CC)CCC(O)CC3)=O)C(C)C2)=O)CCC2C(C1)C2(F)F 54311,C1(CC)CCCN(Cc2cccc(-c3ncc(C(=O)OC)nc3)c2)C1 54312,c1(C(=O)NCC(CCCC)NC(C2CC3(CC3)CO2)=O)ccc(O)c([N+](=O)[O-])c1 54313,C(C(C)(O)CC(=O)NC(c1cncn1C)C(=O)N(C)Cc1cccc(F)c1)OC 54314,C1(C(=O)NCC2(COC)CN(C(C3CC=CC3)=O)C2)CNC(=O)CC1C 54315,N1(C(c2ccc(C)c(C#N)c2)=O)CCC2CN(C(=O)CC(C)C(C)(C)C)CC2C1 54316,N1(C(C(CC)(C)C#N)=O)C2CCC1CC(O)(CNC(=O)CC1=CCCCC1)C2 54317,c1(C(=O)NCCCN(C(C2(C)CC2Br)=O)CC)c[nH]cc1COC 54318,C1(C(N(C2CN(C(=O)NC(C)(C)C)C2)C)=O)(CCF)CCOCC1 54319,c1(CC(=O)NCC(C)(C)NC(C2CCC(C(=O)OC)C2)=O)cc(F)ccc1OC 54320,CC1(C)CN(C(=O)C(c2cscn2)NC(=O)OC(C)(C)C)Cc2ccccc21 54321,c1(OC)ccc(CCC(=O)NC2CCN(c3ccccn3)CC2)cc1 54322,C1(C(=O)NC(CNC(CCC(=O)NCCC)=O)CC(C)C)CC(C)CC(=O)N1 54323,Cc1ccc(S(=O)(=O)NC(C)C(N2CC3(C2)CN(C(C2CNC(=O)N2)=O)C3)=O)cc1 54324,C1(COC)CN(C(C2CCN(C)S2(=O)=O)=O)CCN1C(c1ccc(O)cc1C)=O 54325,C1(c2nnnn2C2CC(COC)C2)(NC(c2ccc(C)cc2)(C)C)CCC1C1CC1 54326,C12(C(N3CC=C(C)C3)=O)COC(C1)C(NC(C1CCC1)=O)C2 54327,c1(OC)cc(C(N2CCC(C(N3CCC(CO)(OC)C3)=O)C2C(C)C)=O)ccn1 54328,C1(C(=O)NCCC(C)N(C)C(C23CC(C)C2C3)=O)CCCCC1 54329,C1(NC(=O)COCCOCCO)COCCN(C(=O)Cn2cccn2)C1 54330,C12(C(N(CC(=O)NCCCN(c3cnccn3)C)C3CC3)=O)CCCN(CC1)C2 54331,C(=O)(C1=NN(C)C(=O)CC1)N1C2C(C2)C1.c1(-c2cn(C)nc2)sc(CO)cc1C 54332,N1(C(c2c(CC)cc[nH]2)=O)C(C(=O)NC(c2snnc2C)C)CCC1C1CC1 54333,CON=CC(=O)NCC(O)CCNC(c1cncnc1)=O 54334,C1(C(=O)NCCOC2CN(C(=O)CO)C2)CC1C1CC(F)(F)C1 54335,c1(NC(C2(O)CN(C(CNC(C=C)=O)=O)C2)=O)cc(C)ccc1C(C)=O 54336,c1(C(N2CC3CCC(C2)C3NS(=O)(=O)c2ccccn2)=O)cn2cccnc2n1 54337,C12(CCCCC1)C(=O)N2.c1(CNC(N)=O)ccc(CC(=O)CCCCC2CC2)cc1 54338,N1(C(c2cccc(NC(C3C(C(=O)OC)C3)=O)c2)=O)CCC(OC)C(F)C1 54339,CC1(C)CC(=O)NC1CNC(=O)C(c1cccs1)NC(=O)CN1CC2CC2C1 54340,c1(C(=O)NC2(CC=C)CN(C(=O)C(C3CCC(=O)N3)C)C2)cc2cccn2cn1 54341,C(C(CO)CC(C)(C)C)NC(c1ccc(OCC=C)cc1O)=O 54342,Cc1nc(NCC2(CNC(=O)N)C=CCC2)cc2nncn12.c1(C)ccccc1 54343,C1(CNC(=O)CCc2cccs2)CCCN(C(C2CCC(F)(F)C2)=O)CC1 54344,c1(OCCC(N2C(CNC(COC(C)C)=O)CC2)=O)ccc(Br)cn1 54345,c1(C(=O)NCC(CN(C(=O)CC2COC(=O)N2)C)(C)C)cn2ccccc2n1 54346,N1(C(c2nn(CC)c(O)c2)=O)CC(NC(=O)CNc2nccs2)CCC1C 54347,Cc1cc[nH]c(=N)c1C(=O)NC(C1CN(C(=O)CC2CCC(F)(F)C2)C1)C 54348,c1(CC)ccc(C(N2CCC(CNC(=O)CN3CCCC3=O)C(C)C2)=O)cc1N 54349,Cc1nc(CCC(=O)N2CC(C(C)NC(c3sccc3C(C)C)=O)C2)[nH]c1C 54350,S(=O)(=O)(c1cccc(=NCC2CCC3(C2)CC3(F)F)[nH]1)N(C(CC)C1CC1)C 54351,C1(C)(CC)CC(NC(c2c(OC)cccc2C)=O)CN1C(c1cnc(S)nc1)=O 54352,N1(C(CC(CNC(C2CCCOC2)=O)OC)=O)CCCC(C2CCC2)C1 54353,C12(NC(c3cc4occc4s3)=O)CCCN(C(c3ccccn3)=O)CC1C2 54354,c1(NC(C2CCCC(NCc3cccc(OC)c3Cl)C2)=O)cnc2sccc2c1 54355,CC1COC2(CCC2)CN1C(=O)CSCCNC(=O)C(O)Cn1cncn1 54356,c1(CC)cc(C(=O)NC)ccc1C(=O)N(C)CCCOc1ccc(Cl)cc1Cl 54357,C(=O)(C1=CCCCC1)N(C)CC1CCCC(NC(C2C(CC)N(C)CC2)=O)C1 54358,C1(C2CC2)(C(N2C(CNC(C3(C#C)CC3)=O)CC(OC)C2)=O)CC=CC1 54359,c1(OC)ccc(I)c(NC(=O)CC2CCCN2c2cc(C#N)ncn2)c1 54360,CS(=O)(=O)CCC(=O)NCC1(O)CCCN(C(=O)CC2CCCS2(=O)=O)C1 54361,N#CC1(NC(c2ccc(I)cc2I)=O)CCN(C(c2ccc(Cl)nc2Cl)=O)C1 54362,c1(C(=O)NC2C(NC(CCCOCCOC)=O)C2)occ2c1CCC2 54363,Cn1ncc2nc[nH]c(=NC3CC(NC(c4ncc(OC(F)(F)F)cn4)=O)C3)c12 54364,CC(C)(CCC(=O)N1CC(C)(C(=O)NC2CCCCC2(F)F)CC1(C)C)[N+](=O)[O-] 54365,CC1CC(NC(C2(C)CCCC2(F)F)=O)CN(C(c2ccc(NC=O)cc2)=O)C1 54366,c1(C(N2CCC(N(C)C(c3cnc[nH]3)=O)C2)=O)cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 54367,c1(N(CC(=O)N(C(CNC(=O)C(CO)c2ccccc2)C2CC2)C)C)ccncc1 54368,C(C(C(=O)NCc1cnc(F)c(C)c1)C(C)(C)C)NC(C1C(C)=CCS1)=O 54369,C(Cn1cncn1)(C(=O)N(C1CC1)C(C)C1CC1)NC(C1CC(C)C1)=O 54370,C(=O)(C(F)C(C)CC(C)(C)C)N1C(C)CN(C(C2C(OC)CCCC2)=O)C(C)C1 54371,C(=O)(C1CCc2ccccc21)NCC(C)CNC(=O)CCc1cccc(F)c1F 54372,N1(C(C)C(=O)N2CCCC2)CC2C(C(=O)NCc3ccc(Cl)cn3)C2C1 54373,N1(C(C23OCC(C(C)C)(C2)C3)=O)CCN(c2ccc(C(=O)O)cn2)C(C)C1 54374,c1(C(N2CCC=C(Br)C2)C(=O)NCCCOC)cccc(C(=O)OC)n1 54375,C1(C(N2CC(CC(C)C)OCC2)=O)CC2CCCC2N1C(=O)CCC(N)=O 54376,c1(C(=O)NC(CNC(Cc2nnc(C)s2)=O)C(C)C)c(Cl)cnn1C 54377,c1(CCC)cc(C(=O)NCC(C)CN(C(=O)CCCC2CCOCC2)C)ccn1 54378,c1(C(=O)NC(CC=C)CNC(=O)CCn2ccccc2=O)cc[nH]c(=NCC)c1 54379,C1(C(F)(F)F)CC(=O)N1.c1(CC)ccc(C)c(C(=O)NC2CC(C(=O)OC)C2)c1 54380,c1(C(=O)NC(CN(C(c2cnn(C(C)C)c2F)=O)C)C)cccc([N+](=O)[O-])c1C 54381,C1(C(=O)NCC=CCNC(C2(c3cccs3)C(C)C2)=O)CCC(F)(F)CC1 54382,C=Cc1cncc(C(N2CCC(NC(C3SCCCS3)=O)C2)=O)c1 54383,C=Cc1ccc(C(N2CC(CNC(=O)Cn3nnc(-c4ccsc4)n3)C2)=O)cc1 54384,c1(N2CC(OC)(CNC(=O)Cn3nnc(C)n3)C2)cc(=O)n(C(C)C)c(O)n1 54385,C(CNC(COCC#C)=O)(C(=O)NCC(=O)NCC=C)NC(N)=O 54386,C(=O)(C1=CC2(CCOC2)C1)NCc1c(CCNC(c2ccc(SC)o2)=O)ocn1 54387,c1(C(N2C(CNC(C3CC(C)N(C)C3)=O)CCCCC2)=O)nc(Cl)cc(N)c1Cl 54388,C12(N(C(=O)C3CC3)CC3(O)CN(C(C(C)OCC=C)=O)C3)CCOC(C)(C1)C2 54389,C(=O)(CCCCC(=O)N1CCC(NC(=O)CCCn2nc(C)c(C)c2C)C1)NC 54390,c1(CC(=O)NCC(CNC(c2n(C=C)nnc2)=O)C)cc(Br)ccc1O 54391,N1(C(CSC(C)C)=O)Cc2ccccc2C(CNC(c2ncc[nH]c2=O)=O)C1 54392,n1(CC)cnc(C(N2CC(CCCCNC(C3CCC(COC)C3)=O)C2)=O)c1 54393,C=CCC(C(=O)N(CCCNC(c1cc(F)ccc1C(F)(F)F)=O)CC)C(C)C 54394,Cc1ccc(CO)cc1NC(=O)C(C)(C1CC1)N(C)C(C1CC(=O)CS1)=O 54395,Cc1cccc(C(=O)NCC2CC(NC(C3(C#N)CC3)=O)CC2O)c1Br 54396,N1(C(C(C)NC(N)=O)=O)CCC2(CC1)CCN(C(c1cc[nH]c1C1CC1)=O)C2 54397,c1(OC)ccc(Cl)c(Cl)c1C(=O)NCC1CCN1C(=O)C(F)OC(F)(F)F 54398,O=C(C#CC1CC1)NCC1CC(F)CN1C(=O)Cc1ccc(Cl)nc1.C12CC1C2 54399,C1(C)(C(N(CCOC)CCNC(C2CSCC(=O)N2)=O)=O)CCC(C)=C(C)C1 54400,N1(C(CC2CCN(C)C2)=O)CCN(C(c2cnoc2-c2ccc(Cl)s2)=O)CC(O)C1 54401,N1(CCC#C)CCC(C(=O)NC(C)(CNC(=O)C2=CCCS2)C2CC2)CC1 54402,C1(NC(Cc2cnc(C)o2)=O)CCCC1(C)CN(C(=O)CC1(O)CCC1)C 54403,N1(C(C(c2ccc(OC)cc2)O)=O)CCC(F)C(NC(=O)CN2CCC(C)CC2)C1 54404,C(CC1=CCN(C(C2CCCCN2CC(F)F)=O)CC1)NC(C=C(C)C(F)F)=O 54405,C=C1CON(C(=O)C2CC=CC(NC(=O)CCC3CCCOC3)C2)C1 54406,O=C(C1=CC2C=CC(C1)C2)NCC1CC(F)CN1C(=O)CSc1cccs1 54407,c1(C(N2CCC2C(=O)Nc2ccncc2)=O)cnn(C2CC2)c1Cl.C12(CC1)C(=O)N2 54408,C1(NC(=O)CCc2ccco2)CC2(C1)CC2NC(=O)CCCc1ncco1 54409,C(=O)(C1CCCc2sccc21)N1CCN(CC2(NC(=O)C=CCO)CC2)CC1 54410,c1(C(=O)NCCC(=C)CNC(=O)CCC(F)F)cc2c(C(=O)OC)nn(C)c2s1 54411,c1(CCN(CCN(C(C)C)C(C2CCNC2=O)=O)C)ccc([N+](=O)[O-])cc1 54412,C1(C)(NC(c2n(C(CC)(C)C)nnn2)c2ccc(Br)o2)CCC2(CC1)CC2 54413,N1(C(C(CC(F)F)N(C(=O)CN2CC=CC2)C)=O)CCC(F)(F)C(F)C1 54414,C1(C(=O)NCCOCCO)CC(=C(F)F)C1.C1(C(C(C2CCC2)=O)=O)(N)CCOC1 54415,N1(C(CN(CCC)C)=O)CCOCC1CN(C(=O)C(F)C(C)C)C 54416,S(=O)(=O)(c1cccnc1NCc1csc(C2CC2)n1)NC1C(C)COCC1 54417,c1(OC)cnc(OC)c(C(=O)NNC(=O)C2CC2(Br)Br)c1 54418,Cn1nnnc1CC(N1CCC(C(F)(F)F)C1)=O.C1C(=O)N1 54419,c1(C(=O)NCC(C(C)C)NC(C(C)(CO)NC(C)=O)=O)cnc2cc[nH]c2c1 54420,C1(NC(c2onc(C)n2)C2CCOCC2)CCn2nnnc2C1 54421,C1(C(=O)NCCC2(NC(c3c(Cl)cn(C)n3)=O)CCCC2)CC12CC(F)(F)C2 54422,c1(C(=O)NC(C)(C)CCNC(=O)CC2(O)CCOC2)cc2ccncc2cc1F 54423,CC1(C)CCC(C(=O)NCC2(CF)CC2)CN1C(C1CN(C2CCC2)C1)=O 54424,c1(OC)ccc(I)c(C(N2CCOC(CCNC(=O)Cc3cccnc3)C2)=O)c1 54425,C1(C(=O)NCCC2CCCN2C(c2nocc2Cl)=O)CN2CCC1CC2 54426,C1(NC(C2CN(C(N)=O)C2)=O)CN(C(c2ccc3n[nH]cc3n2)=O)CC2(CC2)C1 54427,N1(C(C2(C)N(C(c3n(CC)cc(Cl)c3)=O)CC=C2)=O)CCC2(CO)CCCC12 54428,C12CCCCC1NC2.c1(N(C)C(c2cncnc2C2CC2)=O)nnc(C#N)s1 54429,O=C(NNCC(F)(F)C(F)(F)F)c1cnc2cccc(O)c2n1 54430,C12(CNC(CSCCOC)=O)CCCCC1N(C(=O)C=C(C)C1CC1)CC2 54431,C1(C(=O)NCCSCC)CC2(CCC2)CN1C(c1[nH]ccc(=O)c1C)=O 54432,C(=O)(CS(=O)(=O)O)N(CCCNC(C1CCC(C)O1)=O)C.C1(OCC2CC2)CCC1 54433,C(=O)(C(C#N)C(C)(C)C)NC(C(NOCC(C)C)=O)Cn1cncn1 54434,c1(C(=O)NCC2(CN(C)C(C3(S(N)(=O)=O)CC3)=O)CC2)ccc2c(c1)NCCC2=O 54435,C1(C)(C(=O)NCC2(OC)CN(C(c3c(C)oc(C(C)C)c3)=O)C2)CCCS1(=O)=O 54436,N1(C(CC(C)(C)C)=O)CC2CCC(NC(c3n[nH]c4c3CCC4)=O)CC2C1 54437,N1(C(=O)Nc2ccc(C(F)(F)F)o2)CCOCC1c1ccc(C(F)(F)F)o1 54438,C1(COC)CC(CNC(C2CCC(C)O2)=O)N(C(c2[nH]c(O)nc2C)=O)C1 54439,C1(F)(CNC(=O)C(F)CC2CCC2)CCN(C(=O)CCc2cncnc2)C1 54440,CC1C(O)CC2CCC1N2C(=O)Nc1ccc(-c2ccccc2)cc1 54441,c1(C(=O)OC)cc(C)nn1CC(=O)NC(C)CC(C)NC(=O)C(C)CC1CC1 54442,c1(OCCNC(C2N(C(c3c(C)n[nH]c3)=O)CCOC2)=O)ccc(Cl)cc1Br 54443,c1(C(=O)NCC2N(C(C3N(C(C)=O)CC(O)C3)=O)CCC2)ccc(N)cc1Cl 54444,CON(C(=O)CCc1ccc(CNC(=O)C(C)(O)C(C)C)cc1)C1CCC1 54445,CCC(CC)(CO)C(=O)NC1CCN(C(c2cccn2Cc2cccs2)=O)C1 54446,C(C(C)C)(C(O)C(=O)N1CC(C(C(=O)NCC2CCOC2=O)OC)C1)OC 54447,C1(OCC#C)CCN(C(=O)C(Cc2cn[nH]c2)NC(=O)CCSC)CC1 54448,C(C(C)(C)C(=O)NC1CCCC1NC(=O)C(c1ccn(C)n1)C)OC 54449,c1(C(N2CC(F)(CNC(C(CCC#C)O)=O)C2)=O)cc(F)c(F)c(Cl)c1F 54450,Cn1ncc(NC(c2cccn2Cc2ccncc2)=O)c(Cl)c1=O 54451,c1(C(=O)NC2CCC(C)(CNC(c3n(C=C)ncc3)=O)C2)ccc(Cl)c(O)c1 54452,c1(C(=O)NC(CNC(CCC(C)OCC)=O)CO)cc(=O)n(C)cc1Br 54453,C1(C(=O)NC2CC(OC)C23CCCC3)CC2(CCCCC2)N1C(=O)OC(C)(C)C 54454,C1(COCC)CCN(C(c2nonc2C)C(=O)NCc2ccccc2)C1 54455,N1(C(c2cn(CC)nc2)C(=O)NCC2CC2(Cl)Cl)CCN(C2CCOCC2)CC1 54456,N1(C(Cc2ccc(C)s2)=O)CC=CCC1C(N1CCC(C(N)=O)C1)=O 54457,N1(C(C2CC(CC)C2)=O)CCCC2CN(Cc3c(C)cccc3[N+](=O)[O-])CC12 54458,c1(C(N2CCC(N3CCN(c4nnc(C(F)F)o4)CC3)C2)=O)ccccc1Cl 54459,c1(C(C(=O)N(CCCNC(Cc2c(C)scc2)=O)C)C)ccc(F)cc1 54460,c1(CC(N2CC3(C(NC(C(C)O)=O)CCC3)C2)=O)c[nH]c2cccc(Cl)c12 54461,C1(c2ccccc2)(C(N(CCCNC(C2(COC)CC2)=O)C2CC2)=O)CC(OC)C1 54462,C1(C(C)(C)C)CCCCC1NC(=O)C(C)(C)C1CCN(C(c2ccco2)=O)C1 54463,c12cc(cc(F)c1)CN1CCN(C(CO)C1)C2=O.c1(C=O)cc(Cl)c(Br)s1.CO 54464,C(C(C)C(F)C(=O)NCCCC1CC(C)C1)NC(c1c(C)cc[nH]1)=O 54465,C(=O)(C(CC)(CC)CC)NC(C(=O)OC)Cc1cn(C2CCCC(CN)C2)nn1 54466,N1(C(c2ccc(C(F)(F)F)cn2)C(=O)NC)CCCC(C)(C(F)(F)F)C1 54467,c1(-n2ccc(C(=O)NCC3C(NC(C4(SC)CCC4)=O)C3)n2)cnccc1C 54468,c1(C(N2CC(C)C(CNC(=O)Cc3csc(Cl)c3)C2)=O)cc(Cl)cc(F)c1N 54469,CC1(C(N2CC(O)(CNC(=O)C#CC3CCOC3)C2)=O)CCCCC1(F)F 54470,N1(C(C(CCSC)O)=O)CCOCC(C(=O)NCCC(=O)N(C)C)C1 54471,C(c1cccc(Cl)c1)=CC(=O)NCC1CCC(NC(c2cn(C)[nH]c2=N)=O)C1 54472,C1(NC(C2CC(=C)C2)=O)COCCC1C(=O)NCc1ncc(CC)o1 54473,n1(CC(=O)NC2CC(CCNC(C=CC(CC)C)=O)C2)cc(C#N)c(O)nc1=O 54474,c1(C(=O)NC2C(NC(c3nccc(C)n3)=O)COC2)ccc2cccnc2c1N 54475,N1(C(C2(C(=O)O)CCC(F)(F)CC2)=O)CCN(C2=NCCCN2)CC1 54476,C(C)(CCC(=O)N1CCC(C)(CCNC(c2cc(F)n(C)n2)=O)C1)SC 54477,C#CCCCC(C)C(=O)NCC(C(C)C)NC(=O)Cc1cccc(SC)c1 54478,C1(NC(CC2CN(C(C)=O)C2)=O)CC12CC(NC(c1cccc[n+]1[O-])=O)C2 54479,N1(CC(C(C)(C)C)CC(=O)O)C(=O)NC2(CCCCC2)C1=O 54480,C(=O)(NNC(=O)C(C)OC)c1ccc(OCC)cc1.c12cn3c(cccc3n1)[nH]2 54481,C1(CC)CN(C(C2CCC(C(N)=O)CC2)=O)CC1NC(C1CC(C)(O)C1)=O 54482,C1(NC(CCc2ccc(OC)c(OC)c2)=O)CCNC12CCOCC2 54483,N1(C(C(CSC)C)=O)CCC(C)(CNC(c2c(C)coc2-c2ccccc2)=O)C1 54484,C(=O)(CN=c1cc[nH]cc1)N1C(CCNC(C2(O)C(C)(C)OCC2)=O)CCCC1 54485,CC(C)C(O)C(C)C(=O)N1CC(n2cc(CNCc3ccc(F)cc3O)nn2)C1 54486,CC1(O)COCCN(C(c2cc(CNC(=O)CCc3ccncn3)no2)=O)C1 54487,N1(C(CCC#CC)=O)CC(NC(C2(OC)CCOCC2)=O)C(C2CC2)C1 54488,Nc1ccc(C(=O)NC2CC2NC(c2cnc(C(F)(F)F)cn2)=O)nc1Br 54489,Cc1[nH]nc(Cl)c1C(N1CCOC(C(C)NC(C23COC(CF)(C2)C3)=O)C1)=O 54490,Cc1c([N+](=O)[O-])c(C(N2CC(NC(=O)CSc3nc[nH]n3)CCC2C)=O)nn1C 54491,C1(CNC(=O)CCc2ccccn2)C(C2CC2)CCN1C(=O)Cn1cccn1 54492,c1(C(=O)NC(CC)CNC(=O)C(C)SCCNC(N)=O)ccc(N(C)C)c(C)c1 54493,C(=O)(C(=O)NNc1cc(C)cc(C)c1)N1CCC(C)(C(=O)NC)C1 54494,C1(CN(C(=O)CNC=O)C)CCN(C(C2(C#N)CC2C(F)(F)F)=O)C1 54495,C1(C2CC2)(CNC(c2c[nH]nc2[N+](=O)[O-])=O)CCN(C(=O)Cn2cnnc2O)C1 54496,N1(C(Cc2cc(=N)[nH]cc2)=O)CCC2CN(C(=O)CSc3ccc(Cl)cc3)CC12 54497,C(C(CC(=O)N1CCCC1CN(C)C)NC(=O)C(C)CCN(C)C)OC 54498,N1(C(c2cc(CCC)c(C)s2)=O)CC(NC(=O)CCNC(C)=O)C(C)(C)C1 54499,C1(c2cn(CC3CCCN3C(C3C=CC3C(=O)OC)=O)nn2)(OC)CCCC1 54500,N1(C(C(CCC)CC)=O)CCCC2(C1)CN(C(c1cnn(CC)c1C)=O)C2 54501,C1(NC(C(CSC)O)=O)CC2CCC1CN(C(C1(F)CCCCC1)=O)C2 54502,c1(C(=O)NC(CC)CNC(=O)CCOC(C)=O)cnoc1CC(C)C 54503,N1(C(CC2N(C(C3ON=C(C(C)C)C3)=O)CC(O)C2)=O)CCCN(C=O)CC1 54504,O=C1NC2(CCO1)CN(C(=O)CCC1CCCN1C(c1nsnc1O)=O)C2 54505,C1(C)(C(N(C)CC2CC(=C)C2)=O)CC(O)CN1C(=O)C(CC1CCCC1)OC 54506,CN1CCCC(CNC(C2CC(NC(c3cc(F)n(C)n3)=O)C23CCC3)=O)C1=O 54507,C(=O)(C(C)(F)C(=O)OC)N1C(CNC(C(CC=CCC)C)=O)CC(F)C1 54508,C1(NC(c2ccccc2)C2(OC)CC2)CN(C(c2n[nH]c(C)c2Br)=O)CC1C 54509,C(=O)(C(CO)C(C)(C)C)NCCC(C)(C)NC(CN(C)C(c1ccoc1)=O)=O 54510,c1(N2CC(O)(C(C)NC(CC(=C)C)=O)C2)ncc(C)c(-n2nc(C)cc2C)n1 54511,Cc1sc(CN2CCC(CC3(O)CC3)CC2)c(Br)c1C 54512,c1(SC(C(=O)N(CCNC(COCCOC)=O)C2CC2)C)cc(OC)cc(F)c1 54513,c1(C(C)C)nccc(C(=O)NC(c2cccc(Cl)c2)CNC(C2CC2F)=O)n1 54514,NS(=O)(=O)c1ccc(C(=O)Nc2ccc(Br)c(C(F)F)c2)cc1 54515,c1(CN2CC(CC(=O)Nc3cccc([N+](=O)[O-])c3)C2)c(O)ccc2ccccc12 54516,c1(SC)nc(C(=O)N(CCCN(C)C(C2CC(F)CN2C)=O)C)c2ccccn12 54517,c1(C(N2C(C(C)NC(C3(C)CCC(=O)N3)=O)CCC2)=O)cc2nc[nH]c2cn1 54518,N1(C(c2c(CSCC)cccc2)=O)CCC(N2CCCC2)C(C)C1 54519,C(C(C(=O)NC1CC(N(C)C(c2cnn(C)c2CC)=O)C1)C(C)(C)C)OCC=C 54520,N(C1CCCc2nc(O)ccc21)C(N1CC2(C1)CC2(F)Br)=O 54521,CC1(C)CCCC(NC(C2CCN(C(c3ncc(F)cc3F)=O)C2(C)C)=O)C1 54522,c1(OC)cc(-c2cnc(CN)cc2C)ccc1OC 54523,N1(C(CCc2cc(C)on2)=O)CCN(C(c2cnn(C3CCC3)n2)=O)CC1CO 54524,C123CCC(CC1)(C2)NC(=O)CCC1CCN(CC1)CC=CCN3.CCC.N(C)C 54525,C(=O)(CCC(=O)C1CCSC1)NC(C(C)NC(c1n[nH]cc1CN(C)C)=O)CO 54526,c1(C(=O)NCCN2CCN(C(C(C)C(C)O)=O)CC2)cc(F)c(Cl)cc1Cl 54527,C1(NC(C2(SC)CCC2)=O)CCCC(CC(=O)NC23CC(C)(C2)C3)C1 54528,c1(C(=O)NCC(CO)NC(C2CCC(F)(F)CO2)=O)cnc2[nH]nc(O)c2c1 54529,c1(CC(COC)N(C(=O)CN2CCCCC2)C)ccc(O)cc1.C1C(O)C(=O)N1 54530,c1(C(CNC(C2N(C(=O)NC)CSC2)=O)=O)ccc2ccccc2c1 54531,N1(C(=O)OC(C)(C)C)CCC2(CCN(C(c3ccc4ccc(O)cc4n3)=O)C2)C1 54532,c1(C(=O)NC(CCCNC(c2c(CC)cno2)=O)C)ncc(C)cc1OC 54533,c1(NC(=O)NC(CC(=O)OC)c2ccccc2)ncnc(Cl)c1Br 54534,N1(C(c2c(C)cccn2)=O)CCCC(N(C)C(C2CSCCS2)=O)CC1 54535,N1(c2nnc(CCC)s2)CCC(NC(=O)CCC(=O)N2CCCC2)CC(C)(C)C1 54536,C12(NC(c3nc(C)oc3)=O)CCC(C(=O)NC3CCNC3=O)(CC1)C2 54537,C1(NC(C(C(C)C)SC)=O)C2CC3C1C3C2C(=O)NCCCC(=O)N(C)C 54538,c1(C(=O)NC2C3CN(C(CCc4nc(C)c(C)o4)=O)CC2C3)c[nH]c2nccc-2c1 54539,C1(NC(C(CCNC(C2COCCC2C)=O)OC)=O)COC2(CCC2)C1 54540,C1(CN(CC2CCCCC2CCC)CC=C)CC12CCOCC2 54541,n1(CC)nnnc1C(c1cscc1Br)NCc1nnc(SC)s1 54542,c1(C(=O)NCC2N(C(c3cc(C)c(N)cn3)=O)CC2)ccc(S(N)(=O)=O)cc1 54543,O=C(C(F)(F)CO)NCC(C1CCN(C(=O)Cn2cc(C3CCOC3)cn2)CC1)F 54544,C1(F)(Cn2cc(CCOCC(=O)OC)nn2)CC(NC(=O)CN2CCCC2=O)C1 54545,Cc1nc(NCCCC2CCSC2)cc(=NCC(C(C)(C)C)N(C)C)[nH]1 54546,C#CCCCCC(C)C(=O)N1CCC(C(=O)NCCN(C)C2CC2)(CC)C1 54547,S(=O)(=O)(c1ccc(NCCc2ccsc2Br)cc1Br)N(CCCC(=O)NC)C 54548,C(=O)(CC(O)(c1ccccc1)c1ccccc1)N(C(=O)CC(C)(C)O)C 54549,N1(C(C=CC2CCN(C(C(CC)C(F)(F)F)=O)CC2)=O)Cc2ccnn2CC1C 54550,CC1(C#CC(=O)NC2C=CC(CNC(=O)CCc3nc(=N)[nH][nH]3)C2)COC1 54551,C1(C(=O)NC(C)(C)CS(C)(=O)=O)CN(C(=O)CC2CCC2)CC12CC2 54552,CC1(C(=O)NC(c2ccccc2Br)CNC(C2(C)CC2(F)F)=O)CC(F)(F)C1 54553,Cc1c(N2CCCC(Cc3ncn(C)n3)C2)ncnc1N1CCC(C(C)C)CC1 54554,C1(NC(C2(CCOCC)CCC2)=O)CCCN(C(=O)CC(F)(F)CC)C1C 54555,C1(COC)(CNC(=O)C(C)NC(=O)CC)CCCN1C(C1CCCN1S(C)(=O)=O)=O 54556,c1(C(=O)NC(C(C(C)C)NC(C(=C(C)C2CC2)F)=O)C)cnc2n1CCCC2 54557,c1(C(N2CC(C(C)NC(c3cc(C)ns3)=O)C2)=O)c(C)ccnc1O 54558,c1(C(N2CCC(CC#N)C2)C(=O)NC)cccc(Cl)c1F 54559,S(=O)(=O)(CCC(=O)NCC1C=CC(NC(=O)C(c2ccccc2)F)C1)NC 54560,c1(CNC(c2c(CC)cc[nH]2)=O)ccc2c(c1)CCN(C(c1c[nH]nc1C)=O)C2 54561,c1(NC(c2ccsc2C(N2C3COCC2C3)=O)=O)cnc(I)cn1 54562,N1(CCC)CCCC(C(=O)NC(C)CCNC(c2cc(CC)no2)=O)C1 54563,C(N=c1[nH]c(=NC2CCCC(F)(F)C2)c2ccccc2[nH]1)c1nc(C)c(C)[nH]1 54564,c1(C(N2C(C(C)(C)NC(CCC#CC)=O)CCC2)=O)ccc2c(c1)OCCO2 54565,Cc1nc([N+](=O)[O-])cn1CC(N1CC(NC(C2(C)CC=CC2)=O)CC1C)=O 54566,c1(C(=O)NCC(C(C)(C)C)NC(c2ccc(F)c(N)c2)=O)cc2c(s1)CCCC2 54567,Cc1cn2c(CC(N3CCC(CNC(C4(C)C(C)(C)C4(C)C)=O)C3)=O)csc2n1 54568,c1(C(=O)NCCCC2(N(C(C3C(C)(CC)C3)=O)C)CC2)cnc(N(C)C)cn1 54569,c1(C(N2C(CCC)CN(C(=O)C(C)SC(C)C)CC2)=O)cnc2sccc2c1 54570,C1(CNC(CCC(=O)OC)=O)CC2CCCC2N1C(=O)COCc1cc(C)on1 54571,Cc1cc(C)c([N+](=O)[O-])c(C)c1C(N1CC(CC(C)NC(c2cc[nH]n2)=O)C1)=O 54572,c1(C(=O)NCCN(C(C2(O)CCC(CC)C2)=O)C2CC2)cccc2c1CC(=O)N2 54573,c1(C(=O)NCc2c(C(N3CCC(CC=C)C3)=O)con2)ccc(O)nn1 54574,C1(=CC(N2CC(C)(NC(C(C)Oc3ccccc3)=O)C2)=O)CC2CCC(C1)N2C 54575,c1(C(=O)NC2CCN(c3nc(SC)c(Br)cn3)C2)c[nH]c2cc(C(C)C)cnc12 54576,C1(CC(=O)N(CC(O)CNC(=O)C2=CCCC2)C)CC(C)(C)OC1=O 54577,Cc1ncc(Cl)c(C(N2CCC(NC(c3cc(O)ncn3)=O)CC2C)=O)n1 54578,c1(C(N(C(C)COC(F)(F)F)Cc2cncn2C2CC2)=O)c([N+](=O)[O-])cnn1C 54579,C1(C(=O)NC(CC)(C)CNC(C2(N(C)C)CCCC2)=O)CC(C#N)(OC)C1 54580,Cn1cc(C2=CCCC2)cc(C(N2CCNCC2C(C)(C)C)=O)c1=O 54581,C1(C(N2CCC(C)C2CNC(c2cn(C)nc2Cl)=O)=O)CC2(C1)CC2(F)F 54582,C1(C(N2CC(CNC(c3c(OC)ccs3)=O)OCC2)=O)OCCN(C)C1=O 54583,n1(CC(=O)NCCC2(O)CN(C(COCCCC)=O)C2)ncc2ncccc12 54584,c1(OC)c(F)cc(C(=O)NC(C)(C)C(C)NC(=O)CC2CC=CCC2)c(N)c1F 54585,c1(C(N2CCC3CN(C(CSCCC#N)=O)CC32)=O)coc2c1C(=O)CCC2 54586,c1(C(=O)NC(C2CCN(C(c3cc(C(F)(F)F)n[nH]3)=O)C2)C)ccc(O)cc1Cl 54587,C1(C(N2CCCC(OC)CC2)=O)CN(C(=O)CS(C)(=O)=O)CC(C)(C)C1 54588,C(C(C)(F)C(C)(C)F)NC(C(C(C)C)NC(C1C(OC)(OC)CC1)=O)=O 54589,CCC(C(=O)N1CCC(C(=O)NCC2CCC(=O)O2)C1(C)C)C(C)(C)CC 54590,C(N=c1[nH]c(N2CCc3sc(Cl)cc3C2)nc2cc[nH]c12)C1(C)CC1Br 54591,C(C1CCCN1C(=O)CC1CCSC1)=CC(=O)NC(C)C(C)(C)C 54592,c1(OC)ccc(CCC(=O)NCC2(CO)CCNC2)cc1C 54593,C1(C(=O)NCC2(NC(=O)C(c3ccc(F)cc3)F)CC2)CC2CCCC(C1)C2 54594,N1(C(CC)=O)CCC(F)(C(=O)NC2(C)CCCC2N(C)C)C1 54595,Cn1cc(C(F)=CC(=O)NCCCCNC(=O)Cc2cccnc2O)cn1 54596,C1(CNC(c2ccc(F)cn2)=O)C(C2CC2)CCN1C(=O)COCC1CCC1 54597,c1(C(C)OC(C2(CC=C)CCOC(C)(C)C2)=O)cc(OC)c(OC)c(OC)c1 54598,C(C1=CCCN(C(=O)Cc2ccc(F)cn2)C1)C(N(CCCCC)CCC=C)=O 54599,C1(n2cccn2)(C(=O)NCCCN(C(=O)COC2CCOC2)C2CC2)CCCC1 54600,C1(C(N2CC(CC(C(=O)NCC(C)C)F)C2)=O)CCCN(C(N)=O)C1 54601,Cc1c(C(=O)N(CCCNC(C2CCCCS2)=O)C2CC2)[nH]c2ccccc12 54602,C(=O)(C1=NOC(C)C1C)NCC1CC(NC(Cc2c(C)nc(S)s2)=O)C1 54603,C1(C(=O)OC)CCN(C(C2CC(O)(CNC(C3C4CCCOC34)=O)C2)=O)C1C 54604,C1(C(N2CC(O)(C(C)NC(C3CCCC(F)(F)C3)=O)C2)=O)CCC(C)(C)CC1 54605,c1(C(N2CCC(N(C(=O)C(C)SC)CCC)CC2)=O)cc2sc(C)cc2[nH]1 54606,c1(CNC(C(CNC(=O)CCc2nc[nH]n2)OC)=O)ccc(CO)cn1 54607,C(CC(=O)NCCCCC1CCCC1)(C(F)F)NC(c1cc(C#N)[nH]c1)=O 54608,Cc1csc(C2(C(=O)NNCC3(c4ccnn4C)CC3)CCC2)c1 54609,N1(C(CC2CC(=C)C2)=O)CCC(CCOC)(NCC2CC2C(C)C)C1 54610,C(=O)(CCCCC(C)CC)N(C1CN(C(Cc2cc(CC)c(OC)cc2)=O)C1)C 54611,c1(C(N(CC(CN(C(=O)C=CCN2CCCC2)C)O)C)=O)cc2sc(Cl)cc2s1 54612,c1(OCC)ccc(C)nc1C(=O)NC1(CO)CCN(C(C2CC3(C2)CC3(F)F)=O)C1 54613,c1(C(N2CC(O)(CNC(c3cc(Cl)cc(Cl)n3)=O)C2)=O)cc(Cl)cc(Cl)c1O 54614,c1(C(N(C(CNC(C=C(CCC)C)=O)C2CC2)C)=O)ccnn1CC 54615,c1(CC(=O)NCc2ccc(C(C(C)CN)=O)cc2)cc(F)ccc1Cl 54616,CC1(C(=O)NCC23COC(C2)C(O)C3)CCCCC1O.C12(CC1)C(=O)NC2 54617,c1(C(N2CCN(CC(F)F)C3CC23)=O)nnc(O)cc1O.C12CCC(CC1)C2=O 54618,Cc1c(C(N2CC3(CCC3NC(C34CCC3C4)=O)C2)=O)cccc1C1CC1 54619,Cc1c(C(=O)NCC2CCN(C(=O)CCC(C)N(C)C)CC2)cnn1C(C)(C)C 54620,CCC(CC(=O)NC(CCOCCO)C(=O)NCc1cncs1)C1CC1 54621,CC(C)(C)CC(O)CC(=O)NCCC1(O)CN(C(c2cc(CCO)on2)=O)C1 54622,CCC(CC)(C(=O)NC1CCC(CNC(c2ccc(=O)n(CC)n2)=O)CC1)OC 54623,C1(CNC(CC=CCC)=O)(CO)CCCN(C(=O)C(F)C2CCC2)C1 54624,C1(OC(C)C(=O)Nc2ncoc2C2CN(C(=O)C(C(C)C)OC)C2)CCCCCC1 54625,C1(CCC(N2C(CNC(c3c(C)coc3)=O)CCC2)=O)CCCCN1C 54626,CCC(C#N)C(=O)N1CC(F)CC1CCNC(=O)COCCF 54627,N1(C(=O)CCOCc2ccccc2)CCC2(C1)CN(C(=O)C=CCF)CCO2 54628,n1(C(C)(C)C)cc(C(=O)NCC2CC2NC(C2CCC(C(F)(F)F)O2)=O)nn1 54629,N1(C(c2n(C)ccn2)=O)CCC2CN(C(C3OCC4CCCCC34)=O)C2C1 54630,Cc1nc2ccc(C(N3CC4(CC(CC(=O)NCC(O)CO)C4)C3)=O)cc2o1 54631,N1(C(CNc2nccc(OC)n2)=O)CCOCC(NC(=O)CCC2CC2(F)F)C1 54632,CCC(C)(CC)C(=O)NCCC1CCN(C(=O)COCc2cccnc2)C1 54633,C12CCc3cc(ccc3C1)OC2=O.C(=O)(C(F)CC1CC1)N(CC)CC 54634,CCC(CCC(=O)NCC1CCN(CC)C1)NC(=O)CC(O)C1CCCC1 54635,c1(CC)cc(C(=O)N(CCCNC(=O)Cc2cccnc2Br)C)sc1C 54636,C1(CNC(C2(CS(N)(=O)=O)COC2)=O)CCCCN(C(=O)C2=CCCCO2)C1 54637,N1(C(C2CCCN(CC)C2)=O)CCC2CN(C(c3cncn3C)=O)CC12 54638,c1(CC)nn(C)c(CN(C=O)Cc2ncsc2Br)c1Cl 54639,N1(CCN(C(C=C(CC)C)=O)C)CCN(C(c2ncoc2C2CCCO2)=O)CC1 54640,C1(NC(c2cnc(C(C)O)s2)=O)CC(F)(F)CC1NC(=O)C1=CCSC1 54641,Cc1ccc(NCC(N2CC(NC(=O)CC34COC(C)(C3)C4)C(C)C2)=O)cc1 54642,O=C(C1=C(F)CN(C(C2CC23CCCCC3)=O)CC1)NC1(c2ccco2)CC1 54643,c1(CC(=O)NC(CC)CNC(=O)CNS(=O)(=O)CC)c(C)cccc1Cl 54644,N1(C(c2nc(C)oc2)=O)CCC(CNC(=O)CCC(C)(C)[N+](=O)[O-])C(F)(F)CC1 54645,N1(C(C(C(=O)NC)(C)C)=O)CCN(C(=O)CCNC(C2CCCO2)=O)CC(O)C1 54646,CCCC(CC)CC(=O)N1CCN(C(c2c[nH]nc2-c2cccnc2)=O)CC1C 54647,C1(O)(CNC(c2ccccc2F)=O)CCCN(C(c2nc3c(s2)COCC3)=O)C1 54648,C(N=c1nc2c(cnn2C)c(Nc2cnc[nH]2)[nH]1)C1CCCC(CC)CC1 54649,N1(C(C2C(CC)CCO2)=O)CC(S(=O)(=O)N2CCN(C(C3CC3(F)F)=O)CC2)C1 54650,c1(C(=O)OC(C(=O)NCC(CC)NC(C)=O)F)ccc2c(c1)CCCN2C(C)=O 54651,N1(CC(=O)Nc2n(C)ncc2)CCCC(NC(N2CC3CC3C2C#N)=O)CC1 54652,N1(C(COCC)=O)CCC(C2CCCCN2C(c2ccn(C3CCC3)n2)=O)CC1 54653,c1(C(=O)NC2CC(F)(CNC(C3CC(C)N(C)C3)=O)C2)cccc(S(N)(=O)=O)c1 54654,Cc1c(C(=O)Nc2ccc(NC(C3(C(N)=O)CCC3)=O)cc2C)cc(O)cc1N 54655,C1(NC(C2N(C(CN(C)C3CC3)=O)CC2)=O)CCCC(=O)N1 54656,C1(C(=O)NC2CC2CNC(=O)C=CC2CCCC2)(COC)CC=CC1 54657,C1(N(C(Cn2cc(-c3cccc(C)n3)nn2)=O)C)CCCCC1(C)C 54658,C1(CC(=O)NCCCN2CCN(C(C(CC)O)=O)CC2)OCCOC1(C)C 54659,n1(CC(=O)NC2CCN(C(C(C)CF)=O)CC2O)nc2n(c(=O)c1=O)CCOC2 54660,c1(C(=O)NCC23OCC(CNC(C(CC)(F)F)=O)(C2)C3)cc2ccccn2c1 54661,C(CNC(=O)Cc1csc(Cl)c1)(C(C)C(C)C)NC(Cc1cnc(C)[nH]1)=O 54662,C(=O)(CCCC(C)NC(N1CCOC(C(F)(F)F)C1)=O)OC(C)(C)C 54663,c1(OCC)cccc2c(NC(=O)NC3CCC(SC)CC3)c([N+](=O)[O-])cnc12 54664,N1(CC(N2CCCC(N(C)C(C3CNC(=O)O3)=O)CC2)=O)C(=O)C(=O)N(C)C1=O 54665,C1(C(=O)NCCC(C)(C)NC(CC(C)c2cccnc2)=O)C(C)(C)C1(C)C 54666,C(C)(CC(C)NC(c1cncs1)=O)NC(CN(C(COC)=O)C)=O 54667,C1(NC(C(COC)(C)C)=O)CCN(C(c2cccc(CCN(C)C)c2)=O)C(C)C1 54668,C=Cc1cncc(C(=O)NCc2ncoc2C2CN(C(=O)CC(O)C(C)C)C2)c1 54669,Cc1nsc(N)c1CNC(C1CC=CCC1C(F)(F)F)=O 54670,C1(NC(C(=Cc2cn[nH]c2)C)=O)CC(C)N(C(c2nnsc2N)=O)C1 54671,Fc1ccsc1S(=O)(=O)NOCCCOc1ccc(-c2cccs2)cc1 54672,N1(C(CC=C)=O)CCCC(C(C)C(=O)NCCCCCC2CC2)C1 54673,c1(OC)nc(=Nc2sc(C(=O)NC(C)Cn3ccnc3)nc2)[nH]cc1Cl 54674,c1(C(N2CCN(C(C(C)SCC)=O)C(CCOC)C2)=O)cc2ccsc2c(O)n1 54675,CC(C(=O)NCCC1CC(NC(c2ccn(C3CC3(F)F)n2)=O)C1)C(F)F 54676,N1(C(C(C)N(CC)CC)=O)Cc2nccnc2CC1N(C)CC1CCCC1 54677,c1(N(C)C)cc(Cl)ccc1C(=O)NCC(F)CNC(=O)CO 54678,C1(CC(N2C(CC)CN(C(c3nc(C)sc3C)=O)CC2)=O)NC(=O)CN(C)C1=O 54679,N1(C(c2c(CC)nccn2)=O)CCCN(C(=O)C(O)Cn2cncn2)C(C)C1 54680,CCCC(C)(CCC)C(=O)NC1CC(F)(F)CC1NC(c1scnc1Cl)=O 54681,C(N=c1[nH]c(C)nc2[nH]ccc12)C1CC2(CC(NC(C3CC(=C)C3)=O)C2)C1 54682,CCC(F)(C(=O)OC)C(=O)NCC=CCNC(C1(OC)CC(C(F)F)C1)=O 54683,C(=O)(CCCC(F)(F)F)N1CC(CCCNC(c2cn(C(C)C)nc2)=O)C1 54684,C1(C)(OC(=O)OCC(=O)OC(C)(C)C)COCCN1OC(c1c(C)[nH]c(=N)s1)=O 54685,CC1(C)CC(CNC(c2cnc(=N)[nH]c2)=O)N(C(=O)C(N)=O)C1 54686,C1(C(=O)NCc2n(C)cnn2)CC2(CCC2)CN1C(=O)CCC1OCCO1 54687,C(=O)(C#CC1CCC1)NCC(CC=C)NC(=O)Cc1cccc(C(N)=O)c1 54688,C1(NC(Cc2c(CC)con2)=O)CN(C(=O)CCC2CCOCC2)CC12CC2 54689,N1(C(C(C)OC)=O)CCCC1(C)CNC(c1ccsn1)=O 54690,N1(C(C23CC(NC(CC4CC(=C)C4)=O)(C2)C3)=O)CC(C)CC(C)(C)C1 54691,CCC(C)(C(=O)NCCC1(OC)CN(C(=O)C=C(CC)CC)C1)OC 54692,Cc1onc(-c2ccccc2F)c1C(=O)OCC(n1cnc(C#N)n1)=O 54693,C1(NC(CC(C(F)F)NC(C=CC(C)C)=O)=O)CCn2ncnc2C1 54694,c1(NC(C2C(CC)CN(C(C3(F)CCC(COC)C3)=O)C2)=O)ccc(O)c(O)c1 54695,c1(C(=O)NC(CCC)CNC(=O)C(F)(F)C2(O)CCC2)oc(C)nc1CC 54696,c1(C(=O)NCC2CC(NC(C3CN4CCN3CC4)=O)C2)cccc([N+](=O)[O-])c1O 54697,C1(C(N(C2CCN(C(c3cnn(CC4CC4)c3)=O)CC2)C)=O)CCCCNC1=O 54698,N1(C(CCC(=O)OC(C)(C)C)=O)CC(O)CC1(C)NC(=O)CNS(=O)(=O)C1CC1 54699,C1(CC=C)(NC(=O)CC2CCCC3CC23)CCCN(C(C2CC3CC(=O)C2O3)=O)C1 54700,c1(NCCN(C(=O)C(CSC)NC(=O)CCN2CCOCC2)CC)cn(C)nn1 54701,C1(CNC(CCCOCCOCC)=O)(COC)CCN(C(C2CC(C)=NO2)=O)C1 54702,N1(C(C(C)NC(COC)=O)=O)CC2CCCCC2(NC(c2ccncc2)=O)C1 54703,c1(C2(C(N(C3CCN(C(C(CC)CC)=O)C3)C)=O)CC2)cccc(F)c1Br 54704,C12(NC(Cc3c(C)scc3)=O)CC1CN(C(c1cc(C3CCCCC3)on1)=O)C2 54705,C1(C(N(CCNC(=O)CN(C)C)CC)=O)CC(=O)C1C 54706,Cn1cc(C(N2CCC(N(CCO)C(C3(C(F)F)CCCC3)=O)C2)=O)cn1 54707,C1(NC(C2C(=C)C2)=O)CC2CCC1CN2C(=O)CC1CCC(C)CC1 54708,c1(C(N(CCNC(CCCOCCC)=O)CC)=O)ccc(C)nc1 54709,c1(N)cc(Br)c2ccccc2n1.N1(C(c2cc(C)sc2C)=O)CC2(C1)CN(C(C)C)C2 54710,C(=O)(C1CN(C)C(=O)c2ccccc21)NC(C)CNC(=O)C=CCF 54711,c1(C(=O)NCC(CC=C)NC(c2ccsc2COC)=O)cncc(C2CC2)c1 54712,C1(C2CCN(C(c3ccc(S(C)(=O)=O)o3)=O)C2)(NC(C=C(C)C(C)C)=O)CC1 54713,C1(NC(c2c(C)nn(CCO)c2)=O)CC2CN(C(=O)C(C)CC(C)(C)C)CC2C1 54714,C(C1=NOC2COCC12)NC(C1(CC)CCCN(C(=O)Cc2cscn2)C1)=O 54715,CN1CCCN(C(c2nc(C(=O)NC3CC4CCC3N4)cs2)=O)CC1 54716,C(CNC(c1c(C)n[nH]c1C)=O)(C(C)(C)C)NC(CCOCCC)=O 54717,C12(C(=O)NCC(C)(C3CCC3)NC(C3(COC)CC3(F)F)=O)CCC(CO)C1C2 54718,c1(NC(CNC(C=CC(C)OCCOC)=O)=O)cnc(C2CCOCC2)nc1 54719,Cc1cccc(C(=O)NCC2(C)CCCN2C(=O)COc2ccccc2)c1F 54720,Cc1cc(C(N2CCN(C(C34CC(C)(C3)C4)=O)CC2c2ncc[nH]2)=O)nnc1C 54721,C12CC(C(C)(C)C)CN(C1)C(=O)N(C1(F)CCC1)C2.Cc1nnc(C(C)(C)C)o1 54722,c1(CC(N2CC(N(C(C(C)N(C)CCO)=O)C)C3(C2)CC3)=O)c(F)cccc1C#N 54723,C1(CC)CN(C(=O)CC(C)(C)C)CC1C(N1CCC(F)(C(C)C)C1)=O 54724,c1(OC)cc(C(=O)N(C2CCC(NC(c3[nH]ccc3C)=O)CC2)C)cc(F)n1 54725,CS(=O)(=O)c1cc(C(N2CCN(C(=O)C3=C(Cl)CC3)C(CCO)C2)=O)ccc1F 54726,c1(OC)c(Cl)cc(CN2CCC(O)C(C)(C(N3CC(NC)C(F)C3)=O)C2)cc1Cl 54727,CCCC(CNC(c1cnn(C2CC2)c1)=O)C(=O)NCc1ncccc1F 54728,c1(CCNC(CN(C(=O)C(COC)N(C)C)CCOC)=O)ccc(C)c(C)n1 54729,C(=O)(CCC(N)C(=O)O)N1CCN(Cc2c(OC)cccc2)CC1C 54730,Cc1ccc2c(c1)N(C(c1cccc(C)c1N)=O)CCC2 54731,c1(C(=O)NCC(N(C(CCOC(C)C)=O)C)C2CC2)cc(Br)c2cccnn12 54732,N1(C(c2ccn(CCCC)n2)=O)CCN(C(c2cnn3ccsc23)=O)C2CC12 54733,CC1(CNC(=O)CN2CC=CC2)CN(C(c2csc(Cl)c2)=O)CCO1 54734,N1(C(c2cc[nH]c(=N)c2Cl)=O)C(CNC(=O)CCc2cscn2)CC2COCC12 54735,C1(C2CN(C(=O)CCc3nc(O)n[nH]3)C2)(NC(CC2N(C)CCCC2)=O)CC1 54736,C(N=C(NCc1cc(C)on1)N1CCC2(C1)CC2(F)F)c1cc(C)oc1C 54737,c1(OCC(=O)Oc2cccc3[nH]ccc23)cc(F)c(N2CC(O)C2)c(F)c1 54738,C1(C(N(CCCC)C(C)(C)C)=O)CC2CCC1N2C(=O)C(C(C)C)SCCCC 54739,C1(C(N2CCC(F)(CF)C2)=O)(OC)CCN(C(=O)C(C)SCC2CC2)C1 54740,N1C2CCc3c(cccc32)C1=O.n1(CC(=O)N(C)C)nc2n(c1=O)CCCC2 54741,CC(O)C(F)(F)C(=O)N1CCC(CC(=O)NC(C(N)=O)C2CCCC2)CC1 54742,C1(CCC(=O)NC2C(C(=O)OC)CC2)CCCN1C(=O)CCCNC(C)=O 54743,CCS(=O)c1ccc(-c2ccc3nnc(C(=O)NCC(C)O)n3c2)cc1 54744,C1(NC(Cn2ncc(C)c2)=O)CCCC2CN(C(c3cccc(C#N)c3)=O)CC12 54745,Cn1nccc1C1OCCC1C(N1CCC(CCNC(c2cnns2)=O)C1)=O 54746,C(=O)(C(C)CNc1ccccc1)NCCN(C(=O)CC=C(C)C)CCOC 54747,C1(C(=O)NCC(C)NC(C(=O)NCC)=O)CCC(C)(C)CC1 54748,N(C(=NCCC1(C)OCCO1)NCc1cnccc1Cl)CC1C(OCC)C1 54749,CCC1=C(C(=O)NC2(CNC(=O)C#CC3(C)CC3)CC2)SCCO1 54750,c1(NCC2CN(C(c3cccc(NC(CC)=O)c3)=O)C2)nc(O)c2ncnc-2[nH]1 54751,C1(NC(c2cn(CC(C)C)nc2)=O)CCCCCN(C(=O)CC(C)F)C1 54752,CC1(C(N2CCC(C(F)C(=O)NCCc3nnc(O)o3)C2)=O)CCCC1 54753,CC1(C)C2COC1(CNC(=O)NCc1n[nH]c(C(F)F)n1)C2 54754,CCC(F)(F)CC(=O)NCC1CC1NC(C1C(c2ccccc2)C1(F)F)=O 54755,c1(C(=O)NC2CN(C(=O)COCCCF)CC2CO)c(O)cccc1F 54756,C1(NC(C)(C)CCC2CCCCN2C(=O)OC(C)(C)C)CCCCC1C 54757,c1(C(=O)NCC(C)(C(C)C)NC(C(CCOC)C)=O)nc[nH]c2nccc1-2 54758,C1(C(=O)NCC2C3CN(C(C(C(C)C)F)=O)C2C3)C2(CCC2)C12CCC2 54759,CCCCCCCCC(=O)NC1(CNC(C2CCC23CCC3)=O)CCCCC1 54760,C1(C(n2cc(C(CC)NC(=O)CS(=O)(=O)N(C)C)nn2)C)CC(OC)C(OC)C1 54761,C1(C(=O)NCC(C)C(=O)NC2CC(O)(CO)C2)CCCCC1(F)F 54762,c1(NC(C(C(C)CNC(=O)C=C2CCOCC2)F)=O)cccc(N=[N+]=[N-])c1 54763,c1(NCc2nnc(N(CCC=C)C)n2Cc2cccs2)cc2c(cn1)CCCC2 54764,C(=O)(CCC1CCc2ccccc21)NCC(n1cc(C(C(C)C)O)nn1)C 54765,N1(C(CCC(C)C)=O)CCCC(C)C1CNC(=O)CC1CCCCCCC1 54766,C(=O)(CCC(C)(C)NC(c1nccn1CCF)=O)NCCc1cn(C)nc1 54767,C(=O)(C(CO)C(C)(C)C)N1CCCC(C(N2C(C)CC(CO)C2)=O)CC1 54768,c1(C(=O)NCC2C(NC(CCCN(C)C)=O)CCC2)cc(O)cc(F)c1 54769,C1(C(=O)NCc2conc2C)(OC)CCN(C(=O)C(F)C2CCCC2)C1 54770,Cc1ncc(CNC(C2(NC(=O)CCCn3cncn3)CC2C)=O)o1 54771,N1(C(C2CCC3(CC3)C2)=O)CCCC2(CCCN2C(=O)Cc2cccc(O)c2)C1 54772,C1(N(C(=O)CN(C)C2CC2)CC)CCCN(C(=O)Cc2c[nH]nc2C)C1 54773,Cc1cc(NC(=O)CC2CCCN2C(c2cncs2)=O)cc(O)c1 54774,C1(C(=O)NC(C)CCNC(=O)C(O)C2CCC2)CCc2cnnn2C1 54775,n1(CC(N2CC(C(C)NC(Cc3c(C)occ3)=O)C2)=O)ccc2c(C)cccc12 54776,C(=O)(C1(C)OC(=O)c2ccccc21)NC1Cn2c(C)ncc2CC1 54777,C#CCCCCC(=O)N(C(CC)CC(N1CCCC(CO)C1C)=O)C 54778,C(=O)(C(C(C)(C)C)NC(=O)CCOCCC)NCC(CCC=C)O 54779,c1(C(=O)NC2CCN(C(CCCOC(C)=O)=O)CC2)cccc(Cl)c1O 54780,c1(-c2cc(C(=O)NC(CC=C)CNC(=O)CCSC)sn2)cccc(Cl)c1 54781,Cc1c2cccc(NC(C3CC3C(=O)NCC3CCCOC3)=O)c2nn1C 54782,c1(Oc2ccc(Br)cc2)cc(O)ccc1F.CC1CN(c2nnnn2CCF)CCO1 54783,CC(C)(O)C(C)(C)C(=O)N1CC(=O)CC1C(=O)NC1CC2(C1)CC2(F)F 54784,c1(NC(C)CC(=O)NCCCN(CC)CC)ncc(Br)c(C(F)(F)F)n1 54785,C1(CNC(C(CN(C)C)N(C)C)=O)CC(NC(=O)C(C)(C)CF)CC1O 54786,O=C(N=c1cc(C(F)(F)F)[nH][nH]1)NCC1CCCOCC1 54787,N1(C(CCCCN(C(c2nn(CC)nc2C)=O)C)=O)CCC2CCN(C)C2C1 54788,N(C(=NCC1CCCC12CC2)Nc1ccccc1Cl)Cc1scc(C)n1 54789,N1(C(CCNC(CCNC(=O)OC)=O)=O)CC(O)(C#C)C1 54790,c1(C(=O)NCC(CCCC)NC(C2CCC(C)O2)=O)c(COCC)nn(C)c1Cl 54791,c1(C(C)C(=O)NC(C)(CNC(=O)Cn2cncn2)CO)cccc(Cl)c1 54792,N1(C(CCC#C)=O)CCC2(CC2NC(=O)Cc2cc(Br)ccc2C)C1 54793,N1(C(c2nc(OC)oc2)=O)CC2(CC(NC(=O)C(C)C3CCCC3)CO2)C1 54794,C1(NC(C2(CC#C)CCN(C(=O)CC3(CSC)CC3)C2)=O)CCCCCC1C 54795,N1(C(CCNC(COC)=O)=O)CCC(NC(C23COCC2C3)=O)C2CCC12 54796,Cc1nc2ncc(C(=O)NCCNC(=O)C(C)N3CCCC3)c(=O)n2[nH]1 54797,c1(N2CCC(CNC(CCNC(=O)C=CCl)=O)CC2)ccn2ccnc2n1 54798,C1(C)(CNC(C2C(C(C)O)C2)=O)CCN(C(=O)CN2CCC(F)(F)C2)C1 54799,c1(C(N2CCC(O)(C(C)NC(COCCCC)=O)C2)=O)nc(Cl)c(=O)[nH]c1N 54800,CC(C)(F)C(=O)NCC1CCN1C(c1cc(-c2ccccc2)on1)=O 54801,c1(OC)cccc2c1C(CNCc1cccc(SC)n1)CC2 54802,c1(C(=O)NCCCCNC(c2c(C#C)c[nH]n2)=O)cccc2c1ccn2COC 54803,c1(C(C)C)cc(C(=O)NCC2CC(CNC(C3CCN(C)C3)=O)C2)on1 54804,n1(CCCC)cc(C(N2CC(Cc3cn(-c4ccc(Cl)cc4)nn3)C2)=O)c(C)n1 54805,c1(NC(C2CCOC2)=O)cccc(CNC(=O)C(F)CC2CCC2)c1 54806,Cc1nn(C)c(C)c1CC(=O)NCC1C(C)CCCN1C(c1cnco1)=O 54807,c1(C(=O)NCCN(C(=O)C(C)c2cc[nH]n2)CCOC)nc(O)sc1C 54808,C1(C(N(CCCN(C)C(c2nnn(C)n2)=O)C)=O)CC2CCC1CC2 54809,c1(S)cccc(Cl)c1.C1(C(=O)NC(C)CNC(=O)CCOCC2CC2)CC2CCC1O2 54810,CC1C(C(=O)N(C)C)CCCN1N(CCO)CCO 54811,Cc1cn(C(C)C)cc1C(N1CC(NC(C2(CF)CC2)=O)C(F)C1)=O 54812,Cc1ccc(Br)nc1NC(C12CCC(NC(c3cncs3)=O)(CC1)CC2)=O 54813,n1(CCNC(=O)NCCC(C)OC)c(-c2ccnnc2)nc2c(C)cccc2c1=O 54814,c1(SCCC(=O)N(c2ccccc2)CC)ccc(N(CC(F)F)C)cc1 54815,N1(C(=O)C=Cc2ccco2)CCCC(C2CN(C(=O)C3=CC4CCCC34)C2)C1 54816,N1(C(C(CC)COC)=O)C(C)CN(C(C2CC3(C2)CC3(F)F)=O)CC1C 54817,N1(CC(=O)NC2C3CN(C(CC(C)SC)=O)CC32)CCCCS1(=O)=O 54818,N1(C(c2ccc(SCC)nc2)=O)CCC(NC(C2(C(F)F)CC2)=O)C(C)C1 54819,N1(C(CN2CCC(=O)CC2)=O)CC(NC(=O)CCc2cnn[nH]2)C(C2CC2)C1 54820,C(=O)(C(C1CC1)NC(=O)CC1CN(C2CCC2)C1)N(CC)CC 54821,N1(c2c(S(=O)(=O)N(C)CCOC(F)F)cncc2)CCC(F)(F)C2(CCOC2)C1 54822,c1ccccc1.C(=O)(C(C)C#N)NCC1(CCNC(CCSCCC)=O)CC1 54823,c1(OC(CC(=O)NCCCNC(C2C(=C)CC2)=O)C)cc(Cl)cc(Cl)c1 54824,N1(C(C(=O)NC(C)C)C2CC=CC2)CCOC2(CCCS(=O)(=O)C2)C1 54825,c1(C(N2CCN(CC)C(C)C2)C(=O)NCC2CCCO2)ccc2c(n1)OCCO2 54826,c1(O)ccccc1O.CCS(=O)(=O)N1CC(C(=O)N(CCCN(C(=O)CSC)C)C)C1 54827,CC(C)C(C(C)NC(=O)Cc1csc(-c2nc[nH]n2)n1)NC(=O)Cc1ccsc1 54828,N1(C(C(C)Cn2cccn2)=O)CC(C(=O)Nc2cc(F)ccc2I)CC(F)C1 54829,C1(C)(CNC(CC(C)c2cnn(C)c2)=O)CCN(C(C2C(C)(C)C2(C)C)=O)CC1 54830,N1(C(Cc2cc(C)sc2)=O)CC(NC(c2ocnc2C(F)F)=O)CC1CO 54831,N1(C(c2c(C(=O)OC)nns2)=O)CCC(OCCCNC(=O)C(F)C(C)C)CC1.CC 54832,Cc1nc2nccc(C(=O)NCC(C)(O)CNC(=O)C3=CCCC3C)n2n1 54833,N1(C(c2cc(OC)c(OC)cc2)=O)CC(C)(C)NC(=O)c2ccccc21 54834,c1(N(C)C)nc2c(C(N3CC4(CCCN(C(=O)C(F)(F)F)C4)C3)=O)cccc2o1 54835,c1(C(N2CC3C(NC(c4ccc(C(=O)OC)cn4)=O)(C3)C2)=O)cc(C)c(C)cn1 54836,C1(NC(COC(C)(C)C)=O)CC2COCC(C1)N2C(=O)C(O)C1CC1 54837,C(C(=O)NC1CC(F)(CNC(c2cccn(O)c2=O)=O)C1)(C(C)(C)C)N(C)C 54838,C(=O)(C(CO)C(F)(F)F)N1CCC2(C(C(=O)NCCCc3n(C)nnn3)C2)C1 54839,c1(C(C)=O)c[nH]c(C(=O)NC(c2cn(C)nn2)C(=O)N(CCCF)C)c1 54840,N1(C(c2c(C)nco2)=O)CCC2(CCC2NC(C2CC23CCCCCC3)=O)CC1 54841,C(=O)(C(CC(F)F)c1ccccc1)NCC(C(C)C)NC(c1nc(OC)c(C)s1)=O 54842,C1(NC(C(C(C)C)O)=O)CCN(C(=O)Cc2csc(C(F)(F)F)n2)C12CC2 54843,c1(COC)nc(C(=O)NC2(CO)CN(C(=O)C(C)C3CCOC3)C2)co1 54844,C(=O)(C(O)CC(F)(F)F)N(CC)CC1CCCN(C(=O)CCn2cnnn2)C1 54845,C1(C(=O)NCC2C(C(=O)NC(C3CC(O)C3)C)CC2)CCCC1F 54846,N1(C(COC2CC(NC(C(CCCC#C)C)=O)C2)=O)CCN2C(=O)OCC2C1 54847,C1(NC(c2cc(C)c(C)o2)=O)CC2(C1)CC(CNC(=O)CC1CC(C)(C)C1)C2 54848,Cc1c(C(N2CCN(C(=O)C(C)(O)c3cccs3)CC2C)=O)ccc2c1CCC2 54849,c1(C(CC)O)cn(Cc2ncoc2CNC(c2ccc(F)s2)=O)nn1 54850,C1(CNC(c2c(C)onc2Cl)=O)CN2CCCCC2CN1C(=O)C1=CCOCC1 54851,C1(NC(c2cc(C)oc2C)=O)CC(C)CN(C(C2(O)COC2)=O)C1 54852,c1(CNC(c2ccc(F)c(O)c2)=O)cnn2c1CN(Cc1cnco1)CC2 54853,Cc1c(CC(N2CC3CC3(CNC(C3CCCC3(F)F)=O)C2)=O)ncn1C 54854,c1(C(=O)NC2C(C(N(CC#CC)C)=O)CC2)cnc(CC)nc1 54855,c1(C(N2C(CC(N3CC(OCC#C)C3)=O)CC2)=O)ccc(CSC)o1 54856,C(=O)(C(C)(C)n1cc(Nc2ncn(C(C)C)n2)cn1)OC 54857,C1(CCC#C)(C(C)NC(=O)C(=O)NCC(C)CC2CCCNC2)OCCO1 54858,N1(S(c2ncn(CCCOC)c2)(=O)=O)CCc2cc(C)ccc2C1 54859,Cc1cccc(O)c1NC(=O)OCCCCOCC(=O)NCC1(F)CC(CO)C1 54860,Cc1cc(C)c([N+](=O)[O-])cc1C(=O)NCC1CCN(C(=O)CC(C)CF)C12CC2 54861,C=CCC(C)(C)CNC(=O)C(C(C)C)NC(=O)CC1COCC1O 54862,Cc1cccc(CC(=O)N(CCCNC(=O)C(C)Cn2cccn2)C(C)C)c1Cl 54863,C12(CC(N3C(C)CC(CNC(=O)CC4(F)CCC4)C3)=O)CC3CC(CC(C3)C1)C2 54864,Cc1cc(N2CCC3CN(C(=O)C(C)CCN(C)C)CC3C2)ncc1[N+](=O)[O-] 54865,Cc1cc(Cl)cc(Cl)c1OCC(=O)NC(CNC(c1ncn(C)n1)=O)C1CC1 54866,C1(C(N2CCCC(NC(c3cn(CC)nn3)=O)(CO)C2)=O)CCCCCS1(=O)=O 54867,c1(NC(=O)CN2CCN(Cc3cc(O)cc(F)c3)CC2)ncc([N+](=O)[O-])cc1O 54868,N1(c2snc(OC)n2)CCC(NC(=O)CC2OCCC2(C)C)C12CC2 54869,c1(C(N(C(C)C)CC)=O)cc(Br)cnc1C.c12ccccc1N(C(C)C)C2=O 54870,Cc1cnc2n1C(C(=O)NCC(=O)OC(c1cc(S(N)(=O)=O)cn1C)=O)CCC2 54871,Cc1cc(C(=O)N(C2CN(C(c3nnc(S)n3C)=O)C2)C)c2c(c1)CCO2 54872,C1(C(=O)NCCCCC=C)CCC2(CC2)N1C(=O)Cc1n[nH]c(C)n1 54873,CCC(CC)C(F)C(=O)N1CCCC1CNC(C1CNC(=O)C1)=O 54874,CCCC1C(=O)N2CC(C)(C2)O1.c1(CNC(=O)CSC)n[nH]c(O)n1 54875,C(=O)(CCC(=O)N1CC1)NC.c1(CNC(=O)OC(C)(C)C)ncc[nH]c1=O 54876,c1(C(=O)NCC(C(C)(C)C)NC(=O)C2=NNC(=O)C2)ccc2c(c1)CCCC2 54877,N1(C(CC(C)CF)=O)CCCC(O)(CCNC(c2coc(CC3CC3)n2)=O)C1 54878,c1(C(=O)NC2CCN(C(C(CCSC)O)=O)CC2O)ccc2c(c1)NC(=O)C2 54879,C1(O)(CCNC(c2ccn(C(C)C)n2)=O)CCN(C(C2CCCCC2F)=O)CC1 54880,C=CC(C)CC(=O)NCC1CC(CNC(C2CN(C)C2)=O)C1 54881,CC1(OC(F)(F)F)CC(C(=O)O)C1.c12csc(n1)-n1cc(nn1)N(CCO)C(=O)C2 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54899,C1(C(=O)NCC(C)CNC(=O)C(C)(C(F)F)c2ccccc2)CN2CCN1CC2 54900,CN1CCCC1CCC(=O)NCC1(CF)CCNC1 54901,N1(C(C2C(C)(C(C)C)C2)=O)CCC2(CCN(C(C3COC(C)C3)=O)C2)C1 54902,N1(C(C(C)OCC2CC2)=O)CCC(F)(CNC(=O)C(=Cc2cccnc2)F)C1 54903,N1(C(c2c(SCC)cccn2)=O)CC(c2ccccc2)C(C#N)C1 54904,CCCCC(C)(CO)NC(C1CC=CC(NC(=O)CCc2cscn2)C1)=O 54905,c1(-c2cnc(NC(C3C(NC(c4ccc(Cl)cc4)=O)C3)=O)[nH]2)cccc(Br)c1 54906,C1(C(=O)NCCC#C)CN(C(C2(CN(C)C)CC2)=O)CCO1 54907,C1(NC(C(CC=C)(C)C)=O)CC1C1CCCN(C(C2CCCC(O)C2)=O)C1 54908,c1(OC)c(C(=O)NC2CC2C(=O)Nc2ccc(Cl)c(C)n2)cc(Cl)cc1Cl 54909,Cc1nncn1NC(=O)c1c(CNC(=O)CC2C=CCC2)nnn1C 54910,c1(OC)ccc(CN(C(=O)C(=O)Nc2csnc2C2CC2)C)c(C(F)(F)F)c1 54911,C(=O)(CC(=O)NC1(CNC(=O)CCc2nc[nH]n2)COC1)NCC#C 54912,C1(C(N2CC(CCCCC)C2)=O)N(C(=O)CCCCC(N)=O)CCCC1(C)C 54913,CCC(C)(CO)C(=O)NCC(C1CCN(C(=O)CN(CC(C)(C)C)C)CC1)(C)O 54914,C1(F)(C(=O)NC2(C(=O)NCC3(CC=C)CCCC3)CSC2)CCOC1C 54915,N1(C(c2nncc(OC)c2)=O)CC(NC(c2cc(C(F)F)[nH]n2)=O)CC12CCC2 54916,C12(CNC(C(CC)OC)=O)CCC(CC1)N2C(=O)C(c1cccs1)SC 54917,C1(NC(=O)C2=COCC2)CC(F)CN(C(c2ccc(=O)n(-c3ccccc3)c2)=O)C1 54918,c1(C(=O)NCC(CC)NC(c2ccoc2)=O)c(-c2ccccc2)noc1CC 54919,Nc1c(F)cc(C(N2CC3(CC(NC(=O)C(O)C(F)(F)F)CO3)C2)=O)c(F)c1F 54920,C#CCCCC(=O)NCCC1CSCCN1C(=O)COC(C)(C)CC 54921,CC1C(O)CCCN1C(c1sccc1NC(c1ccc(=O)nc(O)c1)=O)=O 54922,c1(NCCNC(N2C3CNC(=O)C3CCC2)=O)cc2cccc(Br)c2s1 54923,c1(N(C2CNC2)C(C2CN(C(CCC)C)C(=O)C2)=O)ccn2ncc(Br)c2n1 54924,C12(NC(Cc3c(C)scc3)=O)CCC(CNC(=O)C(n3cc(Cl)cn3)C)(C1)OC2 54925,S(=O)(=O)(c1cc(Br)c(F)cc1F)N1CCC(C)C2(C1)CCCC2 54926,c1(CN(C(CCN(C(C(CC)OC)=O)C)(C)C)C)cccc(OC)c1.C1CO1 54927,N1(C(C(c2cccs2)SC)=O)CCCN(C(=O)CN2CCCC2)CCC1 54928,c1(C(C)=O)cccc(C(N2CCC(N(CCO)Cc3cccnc3C)CC2)=O)c1 54929,C1(C(=O)NCC(C)N(C(c2cccc(Br)c2)=O)CC)CCc2cnnn2C1 54930,CCC(C)(F)C(=O)N1CCCC(C(=O)NCC2CCCC2)C1 54931,C(=O)(C(O)CCCNC(=O)CCN(CC)CC)NC(CC)CC(F)(F)F 54932,C(=O)(CC(CC)C1CCC1)N(CC(CN(C)Cc1onc(CCC)n1)O)C 54933,O=S(=O)(c1ccc(-n2cc(-c3cccc(F)c3Cl)nn2)cc1)C(F)(F)F 54934,CCCCC(C(=O)N1CC2CC1CN2C(c1nn(C)cc1C)=O)N(C)C 54935,CCCCCCCCC(=O)NCC1CCC(CCNC(=O)CCOCC(C)C)C1 54936,C(=O)(C1=NOC2COCC12)NC(CNC(c1nn(CCCC)c(=O)cc1)=O)CC 54937,c1(CNC(C2(C)CCN(C(C(CCC)OC)=O)C2)=O)cccc(F)c1F 54938,n1(-c2cccc(C)c2)nc(C(N2CCCc3[nH]ccc3C2)=O)c2c1CCCC2 54939,C1(CC(=O)NCCCCSC)(NCC2CC3CCC3C2)CCCCC1 54940,CCCC(CNC(=O)CN1CCCC1=O)C(=O)N1CCC1C(=O)OCC 54941,C1(C(N(CCCNC(c2cnsn2)=O)C(C)C)=O)CC2(CCCCC2)S1(=O)=O 54942,c1(C(N(CCNC(CC(C)OC)=O)CCOCCO)=O)ccc(N)c(Cl)c1O 54943,C12CCN(CC1O)C(=O)N2.c1(C(=O)OC)cscc1NC(c1ccccc1)=O 54944,C#CC1(C(=O)NCC2CCC(F)C2)CN(C(=O)CC2CC(N(C)C)C2)C1 54945,c1(N(C)C)ccc(C(=O)NCC2CCC(NC(=O)C(=O)NCCC3CC3)C2)nn1 54946,c1(C(N2CCCC(N(C(C3CC=C(C)CC3)=O)C)C2)=O)cc2c(nc1N)CCC2 54947,N1(C(C(COC)C)=O)CC2CCCC(C1)N2C(c1ccnnc1O)=O 54948,c1(C(=O)NCC2(N3CCN(C(C)CO)CC3)CC2)c[nH]c2cccc(F)c12 54949,N1(C(C(C2CCN(C(CN(C)CC)=O)C2)F)=O)CCC12CC(CC(N)=O)C2 54950,c1(CCC(=O)NCc2cn(CC(C)(C)C)nn2)ccc([N+](=O)[O-])cc1 54951,CCC(F)(F)C(C)(C)C(=O)N1CCC2=C(C1)CN(C(=O)CC1CCOC1)C2 54952,C(=O)(CCS(C)(=O)=O)NC1C(CNC(c2ccc(CC)[nH]2)=O)CCCC1 54953,c12ccn3c(nnc3c1)C(=O)NC1CC(C1)CNC2=O.C(C1CC1)CO 54954,CC1CCN(C(C23CCC(O)(CC2)CC3)=O)C(C)C1NC(=O)Cn1cnnc1O 54955,N1(C(c2c(CC)non2)=O)CCC(NC(=O)C=C2CCCC2)C(F)C1 54956,CC(C)CCN=C(NCC(C)(C)C1(O)CC1)NC(C1CC1)C1CC1 54957,C(=O)(C1=CC2CCC(C1)C2)N(C1CCC(NC(C(C(C)C)C)=O)CC1)C 54958,N1(C(Cc2cc(OC)no2)=O)CC(C)N(C(=O)Cc2cc(Cl)ccc2Cl)CC1C 54959,O=C(C1=CCCCC1)NC1C=CCC(C(=O)NCCCCc2cnc[nH]2)C1 54960,C1(C(=O)NC(CC#C)CCOC)CNC(=O)CN1C(=O)C(C)NC=O 54961,CC(C(=O)NCCCC(=O)N1CC(C(N)=O)(N(C)C)C1)C(F)F 54962,C1(NC(C(CN(C)C)OC(=O)OCc2ccccc2)=O)CCCC1(C)C 54963,N1(C(C2CC(SC)C2)=O)CCC2(CC1)CC2NC(c1ccc(N)c(F)n1)=O 54964,c1(C(N2CC(CNC(C3(C)CCOCC3)=O)C3C2C3)=O)ccc(Cl)nc1N 54965,C1(C(=O)OC)CCCN(c2nnc(CC(F)(F)F)s2)CC1.CCCC1C(=O)N1C 54966,N1(C(c2nc(C)[nH]n2)C)CC=C(CNC(C2CCCCN2N=O)=O)CC1 54967,CC1(NC(c2conc2CCNC(=O)CNc2ncccn2)=O)CCCCC1 54968,c1(C(=O)NCC2CCN(C(C(CSC)C)=O)CC2)c(S(N)(=O)=O)ncn1C 54969,c1(NC(C2C3CN(C(C4CN(C)CC4C(F)(F)F)=O)CC32)=O)nc2ccccc2o1 54970,C(=O)(C(O)CNC(=O)C(C)CSC)NCC1CC(C(=O)OCC)C1 54971,c1(C(=O)NCCCN(C(C(C(=O)OC)C)=O)CCO)ccc(C#N)cc1F 54972,c1(CNCC(O)COc2ccc(Cl)cc2)nccc2c(I)cnn12 54973,C(=O)(C(CO)C(C)(C)C)N1C(C(N2CC(OCCC)C2)=O)CC1 54974,Nc1cc(F)cnc1C(=O)NCC(CC(=O)N1CCC(N2CCC2)C1)OC 54975,c12cccc(c1)COCCC(=O)N2.C(CCC(c1ccccc1)c1nn[nH]n1)OC 54976,c1(OC)cc(C(N2CCC(C(C)NC(=O)CC(C)C)C2)=O)cc(Cl)n1 54977,c1(CC)onc(C)c1C(=O)NCCC(C)N(C(=O)C(N1C(=O)CCC1=O)C)C 54978,c1(C(=O)NCC(C)(C2CCC2)NC(C(C)NC(CC)=O)=O)cc([N+](=O)[O-])c(C)s1 54979,Cc1cc(C)c(C(c2ccccc2)NC2CCC(C(N)=O)C2)cn1 54980,CCCC(C(=O)N1CCC(N(C)C(c2cnoc2C2CC2)=O)C1)OC 54981,Cc1nc(C)n(CC(=O)NC2CC(C)(NC(=O)Cc3cc(C)n(C)n3)C2)n1 54982,c1(C(N(CC(C)NC(C2CC3(CCO2)CC3)=O)CC)=O)cnc2ccncc2c1 54983,N1(C(CCC2C(C)C2)C)CCC(C#N)(c2ccc(C)o2)CC1 54984,c1(C(N(C)CC2CN(C(=O)C3=C(Cl)CC3)CCO2)=O)cc2cnccc2o1 54985,CC1(C)CN(Cc2c(F)cc(I)cc2F)c2cc(C(F)(F)F)cnc21 54986,CC(C)CC(C(=O)NCC1CCN(C(c2cncc(Cl)n2)=O)CC1C)C(C)C 54987,N1(C(CCOCC#C)=O)CC=CC(NC(=O)CC2OCCC2C)C1 54988,c1(CN(CCN(C(C2C(OC)CN(C)C2)=O)C)C)ccnc2ccsc12 54989,C1(CC)C(NC(c2ccc(=O)n(C)n2)=O)CCCN1C(c1ccn(C)n1)=O 54990,C1(C(=O)NC2(CC(=O)NC(c3ccco3)CO)CCC2)CNC(=O)N1 54991,c1(CN2CCC(F)(C(=O)NC(C)CCO)CC2)cnc2ncccn12 54992,C1(C(=O)NCc2cc(C)nn2C)C2CC(CNC2)N1Cc1ccc(C)c(C)c1 54993,C1(F)(CNC(C2(C)CC=CCO2)=O)CC2CCC(C1)N2C(c1cnc(C#N)s1)=O 54994,CCC(C)CC(=O)C(=O)N1CCCC(C(=O)NC2(COC)CCC2)C1 54995,C(C1CN(C(c2ccn(CCC)n2)=O)CC1C(=O)N(CC(O)COCC)C)=CC 54996,c1(CC(N2CCCC(NC(C(CCCOC)C)=O)CC2)=O)ccc2occc2c1 54997,C(c1csc(Br)c1)=CC(=O)NC(C1CN(C(CC(=O)OCC)=O)C1)C 54998,C(=O)(C1=C(C)OCCS1)N1CCC(CCOC)(NC(C2CCC2(F)F)=O)C1 54999,c1(OC)ccc2ccnc(-n3cc(CNc4cc(F)cnc4Br)nn3)c2c1 55000,C1(C(=O)NCC(C)N(C)C2CC2)CCN(c2ncncc2I)CC1 55001,N1(C(c2cc(OC)no2)=O)CCCCC1CCCNC(C1(CN(C)C)CC1)=O 55002,CC1=C(C(=O)NC23CC(C(=O)NC(Cc4cnc[nH]4)CO)(C2)C3)CCCO1 55003,Cc1ccc(CC(=O)NCC2(C)CCCN2C(=O)C=Cc2ccncn2)cc1C 55004,c1(C(=O)Nc2c(CC)nccc2)c(Cl)ccc(NC(=O)Cc2csc(C)n2)c1F 55005,C1(C)(CNC(CC2CC(OC)C2(C)C)=O)CCN(C(=O)CN2CCC(C)CC2)CC1 55006,N1(C(c2nnc(C)s2)=O)CC2CCCC2(NC(c2cc(Cl)cc(F)c2F)=O)C1 55007,CC(O)(C(=O)NCCCOCCNC(=O)CC1(CO)CC1)C1CC1 55008,C1(NC(CC2C(C)=NOC2=O)=O)CCOC12CCN(C(c1ncoc1C)=O)CC2 55009,C1(C(=O)NC(C)CCCO)CCN(C(C2CCCC(C#N)C2)=O)C12CC2 55010,N1(C(C(CC)C)=O)CC(O)(C2(CNC(=O)CC3CCCN3C(C)C)CC2)C1 55011,C(=O)(CCCCCF)NC1(CNC(c2c(C)cc(CC)o2)=O)CCC1 55012,N1(C(C(CCCC)N(C)C)=O)CCCCCC(NC(=O)CC2CCC2)C1 55013,C1(COC)(NC(=O)C(C)CN(C(=O)Cc2coc(C)n2)C)CCOC1 55014,N1(C(C(C)OCC#C)=O)CCCCC(NC(CC(F)(F)F)c2ccc(Br)cc2)C1 55015,C1(N(C(c2cn(C(C)C)nn2)=O)C)CN(C(c2coc(C(N)=O)c2)=O)CC1O 55016,C12(C(=O)OC)CCC(Nc3cnc(NC(=O)CC4CCCCN4C)nc3)(CC1)C2 55017,c1(CCC(=O)NCC2(F)CC(NC(C(C)(O)C3CC3)=O)C2)ccc(Cl)c(F)c1 55018,c1(C(=O)NCCCOCCCNC(C2(SC)CC(O)C2)=O)cc(Cl)c(C)cn1 55019,Cc1nccn1C(C)C(=O)NCCC(O)CNC(c1cc(C(N)=O)cs1)=O 55020,C(=O)(CC(CN(C)C)C(F)F)N1CCN(C(c2nn(CC)c(C3CC3)c2)=O)C(C)C1 55021,C(=O)(C#CC1CCCCC1)N1CCC2(CN(C(C(C(C)C)F)=O)C2)C1 55022,c1(N2CCN(C(C)(C)CF)CC2)nc(=NCc2cncnc2)[nH]c2c1COC2 55023,C(C1=CCCN(C(=O)C=Cc2cc[nH]n2)C1)NC(C(C1CCC1)OC)=O 55024,Cc1nn(C)c(Cl)c1C=CC(N1CC2CC1C2NC(=O)CC1C=CS(=O)(=O)C1)=O 55025,c1(N2CCC=C(C(=O)N(C)[Si](C)(C)C)C2)cc(Br)cc(F)c1C#N 55026,Cc1nc(Cl)ccc1CC(=O)NC(C)C(C)(C)NC(=O)Cc1ncoc1C 55027,C(=O)(C1=CNS(=O)(=O)N=C1C)NC1CCC(CNC(CC(C(F)(F)F)OC)=O)C1 55028,c1(C(=O)NCCC2OCCN(C(C(C)SCC)=O)C2)ccc(Br)cc1C#N 55029,S(=O)(=O)(c1cc(Cl)ccc1Cl)N1CC2C(NC(c3cncnc3)=O)C(C2)C1 55030,N#Cc1cnn(CC(=O)NCCCCCNC(c2cc(C3CC3)on2)=O)c1 55031,C(=O)(CCC(C(C)C)NC(=O)C(F)C(C)(F)F)NCC(CC)C(C)C 55032,N1(C(CC2N(Cc3ccc(OC)cc3F)CCOC2)=O)C2COCC1CC(F)C2 55033,c1(C(=O)NCC2(O)CC(CNC(C(C)NC(N)=O)=O)C2)cn(C)c(=O)nc1O 55034,C1(C(=O)NCc2cc(C(C)C)no2)CN(C(c2ccnc(F)c2)=O)CC(F)(F)C1 55035,c1(CNC2C(CCCC(=O)NCC3(SC)CCOCC3)CCC2)cccc(F)n1 55036,CCCCC(=O)C(=O)NC(CCCNC(=O)C=CS(C)=O)c1ccccc1 55037,CCC(F)(F)CC(=O)NC(C)C(C)C(=O)NCc1nc(C)cs1 55038,c1(C(N2CC(O)(CN(C(Cc3c(C)scc3)=O)C)C2)=O)ccc(S(C)(=O)=O)cc1 55039,N1(C(C(C2CCCCC2)OC)=O)CCC(C2(O)CN(C(=O)C3=CSCS3)C2)CC1 55040,c1(OCC(=O)NCCCNC(=O)CC(O)c2ccccc2)ccc(Cl)cc1Cl 55041,c1(CN(c2n(CC=C)c(C3COCCC3(F)F)nn2)C)ccc2ccccc2c1 55042,CC(C)CC(C)CC(=O)N1CCC(C(=O)NCCc2c[nH]nc2O)CC1C 55043,S(=O)(=O)(c1c(C)cnn1C1CCOCC1)NCc1c(SC)cnc(C)n1 55044,C1(COC)CN(C(c2cn(CC(N)=O)nn2)=O)CCN1C(=O)CN1CCOCC1 55045,c1(CC(=O)NC2C(CNC(C3(CC#C)CC3)=O)C2)cnccc1C 55046,N12CC3(CC3)CC1C2.CCC(C(=O)N1CC(OCC(=O)NC)C1)C1CCC1 55047,C1(C(=O)NC2(C[Si](C)(C)C)CC2)C2CN(C(C3CCC4(CC4)C3)=O)CC12 55048,N1(C(CCC#CC)=O)CCCC(CO)(CNC(=O)C=NOC)C1 55049,C1(C(N(C2CCC2(C)C)C)=O)CCN(C(C2CC2(F)Cl)=O)CC1(C)C 55050,C(=O)(C1=CC2CCCCC12)N1CC(NC(c2sc(CCC)c(CC)c2)=O)C(O)C1 55051,N1(C(c2c(CCC)[nH]cc2)=O)CCC(C)N(C(c2c[nH]nc2CCC)=O)CC1 55052,c1(C(=O)OCC)c[nH]ccc1=NCC12CCC(NC(=O)COC)(CC1)CO2 55053,N1(C(c2c(C)nc(C)c(C)n2)=O)CCC2(C)CN(C(c3cc(C)c(C)o3)=O)CC12 55054,CCCCC(O)CC(=O)N(C(C)CO)CC=C.C(CCC)=CC=CC 55055,CC1CN(C(C2C=CC=CC=C2)=O)CCCN1C(=O)CCCC1CCC1 55056,N1(N2C(C3(C=O)CC3)CCC2)CCc2nncn2CC1.C12CC3CCC1N3C2=O.CC 55057,C1(C2CN(C(=O)COCCF)C2)(NC(c2c(OC)cccn2)=O)CC1 55058,c1(C(=O)NC(CCNC(C(CC2CC2)OC)=O)(C)C)ccc(CO)cn1 55059,CC1C=C(C(=O)NCCCCCN(C)C(C2(C)CNC(=O)C2)=O)C1 55060,C1(NC(Cc2cn(C)nc2)=O)C2C=CC(C2)C1C(=O)NC1CC(C(N)=O)C1 55061,c1(COC)ccoc1CNC(=O)CC1COCC1NC(=O)C(C)n1ccnn1 55062,C1(F)(CNC(CC=C)=O)CCC(CNC(=O)C(CCC)c2ccccc2)CC1 55063,Nc1nc2ncccc2cc1C(=O)NCC1CC1NC(C1CCC1(F)F)=O 55064,C1(CNC(c2c(C)onc2C(F)(F)F)=O)CC2CCC(C1)N2C(=O)CC1(C)CC1 55065,Cc1ccc(C)c(CC(=O)NC2CCC2CNC(=O)CN2CC(=O)N(C)C2=O)c1 55066,c1(C(=O)NCC2CN(C(COc3c(C)cccc3)=O)C2)cccc2cccnc12 55067,c1(CNC2CCC(C(=O)Nc3c(C#N)cc(F)cc3)C2)ccc(Cl)c([N+](=O)[O-])c1 55068,S(=O)(=O)(c1ccc(NCc2cc(C)no2)c(Cl)c1)NC(c1cc(C)cc(C)c1)C 55069,Cc1cc(C(N2CCOC(C(C)Nc3ncccn3)C2)=O)c(C(F)(F)F)o1 55070,c1(OC)ccc(CC2CCC(C(=O)NCC3CC(=C4CC4)C3)C2)cc1Cl.NC 55071,C1(NC(c2ccc(SC)o2)=O)C=CCN(C(=O)CNC(=O)CCCCO)C1 55072,N1(CCC(=O)N(C2CC(NC(c3ccn(C)n3)=O)C2)C)C(=O)NC(C)(CO)C1=O 55073,Cc1cnc(C(N2CC(C)(NC(=O)Cc3ccnn3C3CCC3)C2)=O)cc1Cl 55074,c1(NC(C)=O)ccc(-c2nc(C(N3CC(NC(=O)C(C)O)C3)=O)cs2)cc1 55075,CC(Cc1nccn1C)N=c1cc[nH]c(=NCCCC2(C)CC2)[nH]1 55076,c1(OC)nc(NNC(=O)C2CC(O)CN2)ccc1Cl 55077,C(=O)(C1CCc2nccn21)NC1CN(C(CSc2nc(C)[nH]n2)=O)CC1C 55078,C1(C(=O)NCC(C)N(C)Cc2cccnc2Br)CC2CCC1CC2 55079,c1(C(N(C2CN(Cc3nc(CCC)sc3)CCC2C)C)=O)cnc2ccccn12 55080,C=C1CCCN(C(=O)CSCCNC(c2ncn(CC)n2)=O)C1 55081,C(=O)(CCCCC(C)C)N1C(C(=O)NCc2ccc(C)s2)CC(C)(C)C1 55082,C12(C(N3CC=C(CCNC(C4C(C)C4)=O)CC3)=O)CC(C)(C1)OC21COC1 55083,N1(C2CCC(NC(C(C)=C3CC3)=O)C2)CCN(C(=O)C2=CCSC2)CC1 55084,Cc1ccc(CC(=O)NCC2CC(C)CN(C(c3cnsn3)=O)C2)cc1Cl 55085,c1(CCC(=O)NCC2CN(CC(O)COc3cccs3)C2)ncc(F)cn1 55086,c1(-c2ccc(F)c(C)c2C)cnc2cc(C(N3CCCCC3C(N)=O)=O)ccn12 55087,Cc1ccn2cnc(C(=O)NC3C=CCN(C(C4(CCS(N)(=O)=O)CC4)=O)C3)c2c1 55088,C1(CC(=O)NCCOCCN(C(C(C)n2cncn2)=O)C)CCOCC1(C)C 55089,C(=O)(C1CCc2cc(OC)ccc21)NC1CCC(NC(CN(C(=O)OC)C)=O)C1 55090,C1(N(C(C2CCCN(C(c3c(CC)cno3)=O)C2)=O)C)CCCC(C)C1C 55091,C12(CNC(C3N(C(=O)NC)CCC3)=O)CCC(NC(c3cccs3)=O)(CC1)CO2 55092,C=C=C(C)CC(=O)NCCN(C(=O)C(CC)NC(=O)OC)CC(C)O 55093,C1(C(=O)NCCOC2CN(C(CC3C(C)CCC3)=O)C2)(CO)CCCCC1 55094,c1(C(C)=O)cc(C(=O)NC(C(=O)NCCS(C)(=N)=O)C2(O)CCC2)no1 55095,c1(CNc2c(C(=O)Nc3ncc(C)c(F)c3)n[nH]c2)ccc(F)c(C)c1Cl 55096,c1(CC(=O)NCC(C)(CC)NC(C(CCC)O)=O)ccc(S(N)(=O)=O)cc1 55097,c1(CC(=O)NC)c[nH]c2cc(OC(CC)CN(CC(C)(C)CNC(N)=O)C)ccc12 55098,c1(C(N2CC(C)C(NC(c3cnn4c3N(C)CC4)=O)C2)=O)snc2ccccc12 55099,c1(C(=O)NCC2C(NC(C3C(CCC)C3)=O)CC2)ccc(CC)cn1 55100,C1(C(=O)NC(CCC=C)C2CC2)C2CC1N(C(=O)C=Cc1ccncc1)C2 55101,CCC1=C(C(=O)N2CCC(C)(CNC(C3CCN3CC(C)C)=O)CC2)CCCO1 55102,c1(OC)cccc2ccc(C(=O)N(C)CCN(C(=O)CCCC(C)(F)F)C)nc12 55103,S(=O)(=O)(c1ccc(C(=O)Nc2cccc(Cl)c2)cc1)N1C2(CN)CCC2CC1 55104,C(=O)(C(F)C(C)CC(C)(C)C)NC(CC)(C)CNC(=O)C(=O)N=S(C)(C)=O.OC 55105,S(=O)(=O)(c1ccc(NCC=CBr)c(Br)c1)NCc1ccc(OC)nc1C 55106,c1(CC(C(=O)NC(C2CCCC2)COC)NC(c2cc(C)no2)=O)cnn(C)c1O 55107,C=CC1CN(C(=O)CCCC2CCC2)CC1NC(=O)C=C1CCC(C)C1 55108,c1(N2CC(N(C)C(c3cc4cccnc4s3)=O)C2)ncnc2cc(Br)ccc12 55109,Cc1nc(C)c(C(N2CCC(O)(C(C)NC(=O)Cc3nn(C)cc3Cl)C2)=O)s1 55110,Cc1cc(C)c(CN2CCN(C(=O)C=Cc3ccoc3)C3CC23)cc1C 55111,C=CC1(CC(=O)NCC2CN(C(c3cc(C4CCCC4)no3)=O)C2)CCC1 55112,c1(C(=O)Nc2ccc(C(=O)Nc3cc(F)ccc3I)cn2)cc2sccc2[nH]1 55113,c1(C(=O)NCC(CN(C)C(c2cc(C(F)F)cs2)=O)(C)C)cccc(F)c1Cl 55114,C(=O)(C(CC)C(F)(F)F)N1C(CC)C(C(=O)NC(C)C(C)(C)OC)CCC1 55115,C(=O)(C(C)(C)Cc1cn(CC(C)NCc2cnc(C3CCC3)o2)nn1)OCC 55116,N1(C(C(c2cnccn2)C)=O)CCC2CCC12CNC(c1cn(CCO)nc1C)=O 55117,N1(C(CC)C(=O)O)CCC2(CC1)CC2(C)C(=O)NC1CCOC(C(F)(F)F)C1 55118,c1(CCC)c(C(=O)N(CC(C)NC(=O)C(c2ccccc2)C)C)cnn1C 55119,c1(CS(=O)(=O)NC(c2cc(C3CCC3)no2)=O)coc2ccccc12 55120,c1(C(=O)NCC(CC(C)C)NC(C2(C)CCCN2C)=O)cc2c[nH]cnc-2n1 55121,c1(N2CCC(c3nccs3)C2)nc(N2CC3CC3C2)nc2c1COCC2 55122,CN1CCC(C)(C(=O)NCC2(C)CCN(C(c3cccnc3OC(F)F)=O)C2)C1 55123,C1(C(=O)NC2(CNC(=O)Cc3nc[nH]n3)CCCCC2)CC2CCC(C1)O2 55124,c1(C(=O)NC2CC(CCC(=O)NCCOCC(C)(C)O)C2)cc(O)ncc1F 55125,C(=O)(CS(=O)(=O)C(C)C)N1C(CNC(CC2(C=C)CCCCC2)=O)CC1 55126,CN1CCN(C(=O)Cc2csnn2)CC1CNC(=O)COc1ccon1 55127,N1(C(CC2(OC)CCCCC2)=O)CCC2C(O)C(C)(C)C12.C1(C)CCC(=O)N1 55128,C(=O)(C#CC1CCCC1)NCCCCC(C)NC(C1(c2cccc(O)c2)CC1)=O 55129,C1(=O)C(C(C)CCC(C)C)N(C2CC2)CCN1.c1(OC)ccccc1 55130,Cc1ccc(N(C(=O)CC(C)(C)CNC(c2nnsc2C)=O)C)cc1F 55131,c1(C(=O)NC(C(C)C)C(C)NC(=O)C#CC2CCCO2)cccc2sccc12 55132,C1(NC(c2n(CCC)ccc2)=O)CCN(C(c2cn[nH]c2)=O)C1(C)C 55133,C#Cc1nc(C(=O)N(CC(N2CCN(C(=O)CCCC)CC2)=O)C(C)C)cs1 55134,N1(C(c2c(N)ncc(C)c2)=O)CCC2(C1)CN(C(=O)C(F)Cc1ccccc1)C2 55135,CC(=O)CCCC(C)C(=O)NC(CC(=O)N1CCCC(C)(CN(C)C)C1)CC(C)C 55136,CC1(C)COc2cc(C(=O)Nc3ncc(-c4cncc(F)c4)s3)nn2C1 55137,CCC(CC)C(C(=O)N1CC(C)(C(N2CC([N+](=O)[O-])C2)=O)C1)OC 55138,N1(C(c2ccc(C(C)C)o2)=O)CCCC(C)(CNC(c2cnc(O)c(Cl)c2)=O)C1 55139,Cc1cc(CNC2CCN2c2nnnn2Cc2ccccc2)cc(C)c1Br 55140,C#CCCC(C)NC(c1ncc(Br)s1)c1nnnn1CCC 55141,C1(C(=O)NCC(CC(=O)N(CCCO)CC)O)CC2C(C1)C2(C)C 55142,N1(C(CCC2CC(C)C2)=O)CCCC(CO)(CNC(=O)CS(C)(=O)=O)C1 55143,C(=O)(C(C)(C)CCCNC(C1CCCN1C=O)=O)N(C(C)CC1CC1)C 55144,C1(CC(=O)NC)CN(C(C2CCC2(C)C)=O)CCN1C(C1CCC=CCC1)=O 55145,C#CC(CNC(=O)C(Cn1cncn1)NC(=O)CN1CC(C)(C)C1)CC(C)(C)C 55146,n1(CC)nc(C(F)(F)F)cc1C(N1CC(CNC(=O)CCCn2ccnn2)C1)=O 55147,C(=O)(C(O)P(C)(C)=O)[N+](CC(CN(CCC(=O)N)CCOC)C)([O-])C(C)CCC.C1(N)CC1.O 55148,c1(C(C)(C)C(=O)OCC(c2ncccc2Br)=O)ccc(C(F)F)cc1 55149,N1(C(C(N(C(=O)CN2CCCCCC2)C)C2CC2)=O)C2CCCC1CN(C)C2 55150,CC(C)CC(CCO)CN=c1[nH]c2c(c(=NCC3C(F)(F)C34CCC4)[nH]1)CCCC2 55151,C1(C(N2CC(C(C)(C)O)(CNC(C3C(C)(C(=O)OC)C3)=O)C2)=O)CC2(C1)CC(F)C2 55152,Cc1ccc2nc(C(=O)NCCC3CN(C(=O)C(C)C#N)CCCO3)cn2c1 55153,c1(NC(CN2CCC(c3cccc(C)c3C)CC2)=O)ccc2c(c1)OC(C)C2 55154,Cc1nccc(NCC2CCC(NC(=O)C=CC(C)(C)C)C2)n1 55155,C12(C(N(CCCCN(C(=O)C(c3ccc(O)cc3)(C)C)C)C)=O)CC3CC1C2C3 55156,CC1(CNC(c2cnc(CCC(F)(F)F)s2)=O)CCCN1C(C1CC2CC2C1)=O 55157,C#CCC(CC#C)C(=O)NC(CNC(c1csc2ccncc12)=O)(CC)CC 55158,C1(NC(CN(C(=O)OC)C)=O)CC=C(C(=O)N(C)Cc2occc2C)C1 55159,CC#CCCC(=O)N(CCNC(c1cncnc1-c1ccccc1)=O)C1CC1 55160,c1(C(=O)NCCCN(CCCNC(c2[nH]cc(C)c2)=O)C)cnc(C)c(C)c1 55161,N1(C(C2(C)CNC(=O)C2)=O)CCC(C2CCN(C(=O)CC(F)F)C2)C1 55162,C1(C(N(C(CC)C(=O)NC(C)(C)CCCF)C)=O)CN2CCC1CC2 55163,N1(C(C2(C=C)CC2)=O)CCC(C)(NC(=O)C(C)C)C1 55164,n1(C(C)C)ccnc(C(=O)NC2(C)CCN(C(C3CS(=O)(=O)C3)=O)C2)c1=O 55165,C(C)(C)(CC(=O)NC1(CC(=O)NC2CCC3CCC23)CC1)OC 55166,C1(C(=O)NC(CCC2N(C(COC)=O)CCCC2)(C)C)(CF)CC2(CCC2)C1 55167,c1(NC(C(c2cccs2)NC(C(CCC)NC(N)=O)=O)=O)cc(C#N)ccc1O 55168,N1(C(C2N(C)CC(C)(C)C2)=O)CCN(C(C2(N(C)C)CCOC2)=O)CCCC1 55169,S(=O)(=O)(c1cccc(=NC2CCC=CCCC2)[nH]1)NC1CN(C)C2(C1)CCOC2 55170,c1(N2CCC(N(C(=O)C(O)CCSC)CCC)C2)cc(C)c(C#N)cn1 55171,CC1CC(C(=O)NCC2CC3(CC3)CN2C(c2cc(O)cs2)=O)CCC1C 55172,c1(OCC(=O)NCC2CCCC(CNC(C3C=CCC3)=O)C2)ccc(F)nc1 55173,C(CCN(C)C)(C(=O)NCCC(C)(O)C1CC1)NC(Cc1c(C)nsc1)=O 55174,CC(CC(=O)c1cccc(Br)c1)C(=O)NC(Cc1ccccc1Br)CO 55175,C1(NC(c2scc(OC)c2)=O)CS(=O)(=O)CC1NC(=O)C=CSC 55176,C(C)(C)(CC(=O)N1CCC(C(=O)NCc2cc(C)co2)(C(C)C)C1)OC 55177,N1(C(CSC(C)(C)C)=O)CC2(CCC(NC(=O)CC3C=CCC3)CC2)C1 55178,S(=O)(=O)(C=Cc1ccccc1)N1CCN(S(=O)(=O)CCCCl)C2C1C2 55179,n1(CC(=O)OC)ncc2c(O)nc(=NNC(=O)CC3(CO)CC3)[nH]c12 55180,C(=O)(NN1CCCC1C(=O)N(C1CCCC1O)C)c1cc(COC)on1 55181,N1(C(C(C)NC(=O)NC)=O)CCCC(CO)(NC(=O)CC2C=CS(=O)(=O)C2)C1 55182,C1(CNC(C2(COC)CC2)=O)C=CC(NC(C2CCC(C)C2)=O)C1 55183,C1(NC(C2C(CNC(CCCC3C(C)C3)=O)OCC2)=O)CCOC1(C)C 55184,C1(C(=O)NCCC2(CNC(=O)COC3CC(F)(F)C3)CC2)CCCCCS1(=O)=O 55185,c1(C(N(CC(CC)OC)C)=O)coc(CNC(C2(C3CC3)CC2)=O)n1 55186,C1(C(=O)NCC(C)O)CC=CC(n2cc(-c3ccc(F)cc3)nn2)C1 55187,c1(C(=O)NCCCCNC(C#CC(C)(C)C)=O)cc2n(n1)CCCC2=O 55188,C1(NC(=O)NCC(C(=O)NC)NC(=O)OC(C)(C)C)CCN(c2cn[nH]c2)C1 55189,C12(NC(COCCC)=O)CCCC1CN(C(c1cc(CC)nnc1C)=O)C2 55190,CCC(c1ccnc(NCC2CC23CCOC3)c1)=CCO 55191,N1(C(COC(C)C)=O)CCOCC(CNC(c2ccccn2)=O)C1 55192,C=CC1CCCN(C(c2nnn(CC)c2C)=O)C1.c12sccc1CNC2=O 55193,N#CC1CN(C(C(c2ccc(OC(F)F)cc2)=O)=O)CCN1C(C1CCOC1)=O.O 55194,N1(C(C(=Cc2cccc(Cl)c2)C)=O)CCCC2(CCC(NC(=O)C3=CCC3)C2)C1 55195,c1(CC(=O)NC(C(=O)OCC)Cc2ccccc2)cccnc1F 55196,c1(NC2CCCCN(C(CC(CC)O)=O)C2)c(Cl)cc([N+](=O)[O-])cc1Cl 55197,C(=O)(CC(C(F)F)NC(c1scnc1C)=O)Nc1cccc(CC)c1 55198,c1(C(N2CCC(CC=C)C2)=O)cncc(N(C)CC)n1 55199,C1(CC)C(NC(C2CCC(CC)CC2)=O)CCCN1C(=O)CCn1ccnn1 55200,n1(CC(=O)N(C2CCN(C(C3(CC=C)CCCC3)=O)C2)CCO)ncn(C)c1=O 55201,N1(C(=O)COC2CCC2)CC(C2CCN(C(=O)CCSC3CCOC3=O)CC2)C1 55202,N1(C(CCC=C)=O)CCC(OCC2CN(C(=O)CCc3ccnc(Cl)c3)C2)CC1 55203,Cc1ccc2c(c1)C(n1cc(CNCc3cc(F)ccc3F)nn1)CCC2 55204,C(=O)(C#CC1CCOCC1)NC(CCC)CCCNC(C1CC(OC)C1(C)C)=O 55205,N1(C(C2C(C)CC=CC2)=O)CCC(F)CC1C(=O)NCC1(C#N)CC(C)(C)C1 55206,C1(=O)C(C(C)C)N1.C(C1=C(C)CCC1)NC(C(C)N(C(CC)=O)C1CC1)=O 55207,CCC(CN(C)C)CC(=O)N1CC(NC(=O)CC(C)(C)COC(C)=O)CC1C 55208,c1(C(=O)OCC)cccc(CNC2CC2NC(=O)CCOc2cccc(C)c2)c1 55209,C1(CC)CN(C(c2cc(=O)n(C)o2)=O)CCN1C(C1CCCOCC1)=O 55210,c1(OC)ccc(CNC(=O)NNC(C)CN2CCCCCC2=O)c(F)c1Br 55211,C1(C(=O)NCC(C2CCN(C(C3(C)CCC(=O)N3)=O)CC2)C)CCS(=O)(=O)C1 55212,Cc1cc(C(N2CCC3(NC(=O)CCCc4ccccn4)CC3C2)=O)nnc1O 55213,C1(C(=O)OC)COC(C)CN1C(C1CCCC1)=O.C12CN(C1)C(=O)CCO2 55214,OC1CN(Cc2cccc(Cl)c2)CCc2ccccc21 55215,c1(C(=O)Nc2cc(C)c(NC(c3ccnnc3C)=O)cc2)ccn2cncc2c1 55216,C(CCC(=O)NC1CC(C)(NC(c2ncsc2Br)=O)C1)OCC=C 55217,O=C(C1=CCOC1)NCC1CC1NC(C1CCCC1(F)F)=O 55218,CCCCCCC(C)(CCC)C(=O)N(C)CC1CCCN1C(C1CSCCS1)=O 55219,c1(NC(C2C3CN(C(C4(F)CC4)=O)CC23)=O)cnccc1[N+](=O)[O-] 55220,C1(CCN(C)CCN2CCN(CCO)CC2)CC1C1CC1.C(C)(C)(C)O.C1CC1 55221,c1(CN2C(C(=O)Nc3c(C#N)cccc3O)CC(O)C2)nccc2ccccc12 55222,Nc1ccc(NCCNC(=O)OC2(c3nnnn3C3CC3)CCC2(C)C)c(O)c1 55223,c1(C(=O)NCC(CNC(C(COC)(F)F)=O)F)cccc2c1ncn2C 55224,Cn1cc([N+](=O)[O-])cc1C(=O)NCC1(F)CN(C(c2cnn(C)n2)=O)C1 55225,c1(OC)cc(C)c(C(=O)NC2CCCC2CNC(c2c(C)coc2C)=O)cn1 55226,c1(CC(=O)NC2(CNC(C(CC)COC)=O)CCOC2)ccc(CC(C)=O)c(F)c1 55227,C1(C)(CCC)CCCN(C(c2ccc(CN3CCCCC3CO)nc2)=O)C1 55228,C1(CC#C)(C(=O)NC(C2CCOC2)CNC(c2cnc(S)[nH]2)=O)CCOCC1 55229,N1(C(c2c(OC(C)C)n[nH]c2)=O)CC(NC(C23CCCC2C3)=O)C2(CCC2)C1 55230,c1(C(N(CC(CC)NC(C2C(CCC)CCC2)=O)C)=O)ccc(C)cc1O 55231,Cc1nccc(CNC(=O)NC2CC=CC(NC(=O)C(C)(C)C)C2)c1C 55232,c1(N)cnc(F)c(F)c1.N12CCCOC(C1)N1C(=O)C(CC1)C2=O.CO 55233,CC1(C(=O)NCCCc2[nH]c(=N)sc2C2CCN(C(N)=O)CC2)CC(C2CC2)=NO1 55234,C(=O)(C1CCCc2n[nH]cc21)NC(C)(CNC(=O)CCc1cscn1)CO 55235,c1(C(N2CCC3CC23C)C(=O)NCC(=O)NCC)cc2c(OC)cc(OC)cc2o1 55236,CC1(C(=O)NC2CCCC(CNC(=O)CN3CCCCC3=O)C2)CCCS1(=O)=O 55237,Cc1cc(C)c(C(=O)NCC2(NC(c3cc(F)c[nH]3)=O)CCOC2)cc1C 55238,N1(C(c2[nH]c(CC)c(Cl)n2)=O)CCC12CN(C(=O)CC(C)(C)C)C2 55239,CC(C)C(C(=O)NC1CCN(C(c2conc2-c2ccccc2Cl)=O)C1)N(C)C 55240,c1(C(=O)NCC2N(C(C(C=C)O)=O)CCN(C)C2)ccc2[nH]ccc2c1F 55241,c1(NC(C)=O)ccc(C(=O)NCC2(O)CC(NC(C3CCC3(F)F)=O)C2)s1 55242,c1(C(=O)NC2C(NC(c3cnc(CC(F)(F)F)s3)=O)CCC2)ccnnc1S 55243,Cc1cc(C(N2CCCC(N(C(=O)C(C)C3=CCCC3)C)C2)=O)cc2nc[nH]c12 55244,c1(C(=O)NC2C(CC)N(C(C)=O)CCC2)c(Cl)ccc(Br)c1F 55245,Cc1[nH]c2ncccc2c1C(N1CC(CC)C1)=O.C1(C)CCC(=O)N1 55246,C(=O)(C1=CCCC1C)NC(CCC)C(=O)NC1Cc2cscc2C1 55247,C(=O)(C1=CC=CN2CCS(=O)(=O)N=C12)NCCC(C)OC 55248,N1(C(C#C)C)CCN(C(C2C=CCN2C(=O)CC2(COC)CC2)=O)CC1 55249,C1(NC(CCc2ccc(CC)cc2)=O)CCC(C)N(C(C2C=CCCC2)=O)C1 55250,C(=O)(CC(C)n1cccc1)NCCCN(C(C1CC(O)C1)=O)CC 55251,CCCCCC(CCCCC)C(=O)NCC1(CNC(c2cc(C#N)oc2C)=O)CC1 55252,Cc1cc(Br)c(N)cc1C(=O)NCC1(CNC(=O)CCCC(F)(F)F)CC1 55253,c1(C(=O)NC(CCNC(c2cn(C)[nH]c2=N)=O)(C)C)cccc2nsnc12 55254,N1(C(c2ccc(C(N)=O)s2)=O)CCC2(CC1)CC(NC(C1C3CC4C(C3)C14)=O)C2 55255,c1(C(=O)NC2(C)CC(NC(=O)CC3(C(F)F)CC3)C2)ccc2c(c1)C(=O)C(=O)N2 55256,C1(C(=O)NCC(CNC(c2c(F)cc(C)cc2F)=O)F)CC(F)(F)CCC1(C)C 55257,c1(C(N2CCCC(OC3CCCC3)C2)=O)cnn2c(=O)cc[nH]c12 55258,N1(C(c2cc(C)[nH]c2)=O)CCN(C(=O)CC(C)C(F)(F)F)CCC1C 55259,c1(C(=O)NCC(C)NC(c2c(C)cc(C)s2)=O)c(N)sc2ccccc12 55260,c1(C(=O)NC2CCC(CNC(C3CC4CCCC34)=O)C2)ccc2n[nH]cc2c1Cl 55261,c1(NC(CC)C(=O)N(C)CC2(NC(=O)C(N)=O)CC2)cccnc1Cl 55262,C(=O)(C1=CCCN(C(=O)Cc2ccccc2C)C1)N(CCCCO)CCCC 55263,N#Cc1cccc(C2(C(N3CC(NC(C4CCC4CF)=O)C3)=O)CCCCC2)c1 55264,Cn1cc(C(=O)NC2CCCCC2CNC(=O)C(C)(C)c2cscn2)n(C)c1=O 55265,c1(CC(=O)NC2(COC)CCN(C(C3(C)CC(C)(C)C3)=O)C2)ccc(C#N)cc1 55266,C1(C(N(CC(C(=O)OC)C)C)=O)CC(C)(C)CN1C(c1cc(C)c(F)cn1)=O 55267,N1(C(c2c(C)cccc2)=O)CCC(C)C(CC(=O)NCc2cnccn2)C1 55268,CC(C)CC(C)NC(=O)C(C)(CC1CCC1)NC(N1CCCC1)=O 55269,C(=O)(C1=CC2CCCCCC12)N.N1(C(C)=O)CC(CC(O)C(=O)OC)(CC2CC2)C1 55270,N(C(=NCCCSC)NCC1(OC)CCCC1O)Cc1ccc(OC)cc1Br 55271,C(=O)(C(CC(C)C)n1ccnc1)NC(CC=C)CNC(C1(COC)CC1)=O 55272,c1(C(=O)NCC2CC(NC(C3(C)CC4CCC3O4)=O)C2)ccc(Cl)c([N+](=O)[O-])c1 55273,c1(C(N2CC3=C(CN(C(C(C)CC(C)(C)O)=O)C3)C2)=O)cc2c(cn1)COCC2 55274,CCCCC(C(=O)N=c1ccn(C(C)CC)[nH]1)NC(=O)Cn1ccnc1C 55275,C1(NC(C(C)OCC#C)=O)CC1C1CCN(C(C2(C#N)CCN(C)CC2)=O)CC1 55276,Cc1nc(C(N2CCOC(C(C)NC(=O)C(C)C3CCCO3)C2)=O)[nH]c1C 55277,C1(C(=O)OC)(CC)CCN(C(=O)C=CC(C)NC(=O)C(C)C2CCC2)C1 55278,c1(NCC2OCC(CNC(c3c(C)coc3)=O)C2)ccc([N+](=O)[O-])cc1Br 55279,c1(CNC(C(C)n2ccnn2)=O)ccc(C(=O)NC(c2cscn2)CO)s1 55280,Cc1ccc(C)n1CCC(=O)NCC1CCCN1C(=O)Cc1cccnc1Br 55281,Cc1onc(Br)c1C(N1CC(CNC(c2ccc(O)nn2)=O)C(C)C1)=O 55282,c1(C(=O)NCC(CNC(=O)Cn2cccn2)F)cccc(C(=O)NCCO)c1 55283,c1(C(N2CC(CC(=O)N(C(C)C3CC3)CC)OCC2)=O)ccn2ccnc2c1 55284,Cc1cc(C(=O)NCC2CC(NC(c3cc(Cl)sc3Cl)=O)C(O)C2)cn(C)c1=O 55285,C(=O)(CCC(C)S(C)(=O)=O)NCC1(CNC(C(=Cc2cccnc2)C)=O)CCC1 55286,C1(NC(CN(C)CC)=O)CC2(CCCN(C(C3CCCC(=O)N3)=O)C2)C1 55287,N1(C(Cn2c(CCC)ncc2)=O)CCOCC1(C)c1ccccc1 55288,C(=O)(C(CO)C(C)(C)C)NCC(CCCC)NC(c1cc(C)ccc1OC)=O 55289,S(=O)(=O)(C(F)(F)F)CCNC(C)=O.C12(C(F)(F)F)CN(C1)C(=O)CCN2 55290,c1(N2CC(CCC)OCC2)nc2c(c(=NCCS(C)=O)[nH]1)CSC2 55291,c1(SC)ccc(CCC(=O)NC2CC(CNC(c3oc(C)nc3C)=O)C2)cc1 55292,N1(CC(F)=CC=CC=CCOC(C)C)C2CCC(C(=O)OC(C)(C)C)CC1CC2 55293,C12(NC(c3ncc(OC)cn3)=O)CCC(CC1)N(C(c1nocc1C)=O)C2 55294,C1(C(=O)NCCC2(OC)CN(C(C3CC3CF)=O)C2)OCC2CCCC1C2 55295,C1(N(CC(=O)NC2C3CC(OCC)CC32)C(C)(C)C)CC(C)NC(C)C1 55296,c1(OC)cc(C)cc(C(=O)NCC(C(C)C)NC(=O)CC(O)C(C)C)c1N 55297,c1(CCC(=O)NCC(CC)NC(C2CCC(C(F)(F)F)O2)=O)c(F)cccc1F 55298,CC1(C)CC(C(N2CCN(C(=O)CCCF)CC(O)C2)=O)CC(C)(C)C1 55299,Cc1cc(C(=O)NC(C(=O)N2CC(C(F)(F)F)C2)C2CCOC2)nn1C 55300,Cc1ncc2n1CCN(C(C1CCN(C(c3cncn(C)c3=O)=O)CC1O)=O)C2 55301,N1(C(c2c(CSC)cccn2)=O)CCC(CNC(=O)CCCOC(C)C)C(O)C1 55302,C12(NC(C(CC)C)=O)CCCC(NC(c3ccc(C)cc3F)=O)(C1)C2 55303,CC1CC(NC(C2(C)CC2(F)F)=O)CCN1C(c1coc(O)n1)=O 55304,C1(C(=O)NCc2ccc(C#N)cc2)CN(C(=O)CCC(N)=O)CC12CCC2 55305,N1(Cc2cccc(CC(F)(F)F)c2)CC2(C(F)F)CC2(C(F)(F)F)C1 55306,C(=O)(C1CC=Cc2ccccc21)NC1CC(F)(CNC(C(C)(C)N2CCC2)=O)C1 55307,C(=O)(CCCC(C)(C)C#N)N(CC(CNC(C(C(=O)OCC)C1CC1)=O)O)C 55308,c1(C(=O)NC(C2CCCN(C(=O)CCc3cnn[nH]3)C2)C)cc2ncccn2n1 55309,CCCC(C(F)(F)F)NC(=O)CSCCNC(=O)Cc1ccoc1C 55310,CN1CCN(C(C2CCC(C(N3CCC(CO)C3)=O)C2)=O)CC1C1CC1 55311,n1(CC(=O)NCC2C3CN(C(C4CC=C(C)CC4)=O)CC32)c(C)cc(C)nc1=O 55312,N1(C(c2ccc(NC)cc2)=O)CCC(NC(C2CCC(C(N)=O)C2)=O)C12CC2 55313,C(CCC(=O)N1CCCC1CC(N1CC(N(C)C)C1)=O)N(C(C)=O)C 55314,C1(CC)CC(C(=O)N(CCC(=O)NCCCCN(CC)CC)C(C)C)C1 55315,N1(C(C(C)OCCC=C)=O)CC(NC(=O)C(c2ccc(Cl)nc2)(F)F)CC1C 55316,C(c1ccc(=N)[nH]c1)=CC(N1CCC(C)(NC(C(CCSC)OC)=O)C1)=O 55317,C(=O)(CCCC1CC1)NCCCN(C(C(C1CCC1)N(C)C)=O)CCOC 55318,CC(CNC(c1cc(CO)ccn1)=O)CC(=O)NC(C)C(C)CC1CC1 55319,CCCC(CNC(C1CCN(OC)CC1)=O)C(=O)NCCN1CC(C)(O)C1 55320,C1(C)(C(N(CCC)CCO)=O)CCN1C(=O)C(C1(O)CCCC1)F 55321,c1(CCCC)nc(-c2ccc(NC(C)(C)C)cn2)nn1CCC(=O)OC(C)(C)C 55322,C1(C)(NCc2nc(CC)oc2)CCN(c2ccnc(-c3cc(OC)ccn3)n2)C1 55323,C12(C(=O)NCC3CC4CN(C(C5(C)CC5(F)F)=O)CC43)CC(C)(C1)OC21COC1 55324,c1(C(=O)NC(C)CNC(=O)C(C)OC2CCCCCC2)nnc(O)nc1O 55325,C(C)(C(=O)N1CCC(CCNC(c2ccc(C)cc2F)=O)C1)(C(F)(F)F)OC 55326,N1(C(C(C2CCN(C(c3cc[n+]([O-])cc3)=O)C2)C)=O)CCC(C)(O)C(O)C1 55327,C1(C(N(C2CCC2O)C)=O)CC12CCN(C(=O)Cc1cn[nH]c1)CC2 55328,CCC(C)(CC)C(=O)N(CCCCNC(C1CC1c1ccccn1)=O)CCO 55329,c1(C(N(CC(CN(C(c2c(C)cncc2)=O)C)O)C)=O)c(Cl)cccc1[N+](=O)[O-] 55330,c1(C(=O)NCCCCCCNC(c2c(C)nc(C)[nH]2)=O)cccc2oc(C)cc12 55331,c1(C(=O)NCC2(F)CC(NC(c3n(CC)ccn3)=O)C2)ccc(F)cc1C 55332,c1(C(=O)NCC2CCN2C(=O)C(O)Cc2cnc[nH]2)cc2c(F)c(F)ccc2[nH]1 55333,c1(C(=O)NCCC(=O)N2CC(C3CCCO3)C2)cc2ccccc2[nH]1 55334,C1(NC(c2c(CC)csc2)=O)CC2CN(C(=O)CC(F)(F)CC)CCN2C1=O 55335,C1(NC(C(C)OC)=O)CCCCCC1CNC(=O)CC1(O)CCC1 55336,C(N=c1[nH]cnc(NCc2ccc[nH]2)c1C)c1ccc(CC)cc1F 55337,C(=O)(C1=NNC(=O)CC1)N1CCC(F)(CNC(c2c(CCC)occ2)=O)C1 55338,c1(C(C(=O)NC2C(CNC(=O)C=CBr)C2)=O)ccc(Cl)s1 55339,N1(C(C(C)OC)=O)CCCN(C(=O)C(C)CC(=O)c2ccccc2F)CC1 55340,CCC(O)C(C)C(=O)NC(C)(C)CCCNC(c1cnc(C2CCC2)s1)=O 55341,c1(C(N2CCC(N(C)C(c3n[nH]cc3F)=O)CC2)=O)cccc(C2CC2)c1Cl 55342,C(=O)(C1=CC2(CN(C(C3(C)CC(=O)N(C)C3)=O)C2)OC1)NCCCOC(C)C 55343,N1(C(CCCCC2CCN(C(C(CC(C)C)F)=O)C2)=O)CCNC(=O)CC1C 55344,CC1(C)CN(C(c2coc(C#N)c2)=O)CCC1NC(=O)CN1CCCCC1=O 55345,CC1(C)CCOC1C(=O)NC1C=CCN(C(c2cnc(-c3ccccc3)s2)=O)C1 55346,CC(C)C(=O)C(=O)N(C1CCCN(Cc2ccc(-c3ccc(CO)o3)cc2)C1)C 55347,N1(C(c2cccc(CSC)c2)=O)CC2CC(NC(=O)C3=CCCC3C)C1C2 55348,C1(NC(c2ccccc2)CC)CCCCCC1c1ccccc1 55349,N1(C(C2CC(CNC(=O)C3=C(Cl)CC3)C2)=O)CC(O)C(N=[N+]=[N-])C1 55350,C(CS(=O)(=O)CC(=O)NCC1(C(=O)NCC2CSCCO2)CC12CCC2)OC 55351,C(=O)(C(C)(C)C(F)(F)F)N(CCCCCNC(c1c(C)cn(C)c1)=O)C 55352,C1(C(=O)NCC2OCCC2C(N2CC3(CCOC3)C2)=O)CC2(CCC2=O)C1 55353,O=C(O)CC(Cc1ccccc1)NC(c1ncncc1Br)=O 55354,C1(C)(CNC(c2ccc(OC)nn2)=O)CN(C(=O)CC2(C)CC2)C(C)(C)C1 55355,C(CCF)(C(=O)NCC1CC1(Cl)Cl)NC(Cc1cn(CC)nn1)=O 55356,C(=O)(C#CC(C)(C)CNC(c1nccnc1N)=O)N1CCC(OC)C1C 55357,CC(C)C(F)C(=O)NC1CC(CNC(C2CC2c2cccnc2)=O)C1 55358,Nc1ccnc(C(N2CC3(CCC3NC(c3csc(C(F)(F)F)n3)=O)C2)=O)c1Cl 55359,c1(C(=O)NC2C(NC(COC(CC)C)=O)CCC2)cc(F)cc(S(N)(=O)=O)c1 55360,c1(C(N2CCC(NC(COCCCOC)=O)C(O)C2)=O)cc2n(n1)CC(F)C2 55361,c1(SC)ncc(C(=O)NCC(C)CNC(c2ccnnc2)=O)s1 55362,CC(C)CC(C)(C(N)=O)NC(=O)CCCN(C)C(C1CCC2(CCC2)C1)=O 55363,C#CCCCC(=O)NCC(N1CCCC1CNc1ccccn1)=O 55364,C1(CNC(C2N(C(C)=O)CCC2)=O)CC2(CO1)CN(C(c1sccc1C)=O)C2 55365,C12(C(=O)NCC(CC=C)NC(C3CC4C=CCC(C3)C4)=O)CCC(O)(CC1)CC2 55366,CC(C)CC(C(=O)N1CC(NC(C2CCC(C)(F)CC2)=O)CC(F)C1)C(N)=O 55367,Cn1c(CNC2(CC3COc4ccccc4C3)CC2)cc2ccsc12 55368,N1(C(c2c(C)ocn2)=O)CCC(NC(=O)CCCc2cccnc2)C12CC2 55369,c1(N(C)C)cccc(C(N2CCC2CNC(C2CCN(C)C2=O)=O)=O)n1 55370,N1(C(C)=O)C2CCC1C(F)C(NC(c1nc(Cl)ccc1C#N)=O)C2 55371,C=CCC(C(=O)N(C1CC1)CC1CCCN1C(C1CC2(CC2)CO1)=O)C(C)C 55372,c1(C(C(N2CCC(NC(C(CSC)(C)O)=O)C2)=O)(F)F)cccc(F)c1F 55373,O=S1(=O)CCC2(CCN2C(=O)CCCCc2ccc(C(F)(F)F)cc2)C1 55374,C(N=c1cc(C)[nH]c(=NCCc2ccnn2C)[nH]1)C1N(C(C)=O)CCC1 55375,CC1(CC(=O)NCCCNCCCNC(=O)CCc2cscn2)CCCC1 55376,C1(O)(CC(N2C(CC(=O)OC)CCC2)=O)CCN(C(C2CCCC2O)=O)CC1 55377,CC(C)(C)C(CNC(c1ccc(=N)[nH]c1)=O)C(=O)NC1CCC2(CC2)C1 55378,CCCC(O)C(CO)NC(=O)C(C)(COC)NC(=O)C(C)(C)C(C)O 55379,C(=O)(C(F)(F)CCn1cc(CO)nn1)NCCC(C)N(C)C.C(=O)N(C)C 55380,c1(C(=O)NC2CCC(NC(CN(S(C)(=O)=O)C)=O)C2)cnn2cccc(Br)c12 55381,Cc1cc(CCC(=O)N(C)CCN(C(C)Cc2ccccn2)C)ccn1 55382,C1(NC(C2CCC(C)O2)=O)CC1C1CCCN(C(C2(CO)CC2)=O)C1 55383,c1(CCC(N2CC(O)(CNC(CC(C)O)=O)C2)=O)ccc(CN(C)C)cc1 55384,N1(C(C2(N(C)C)CC2(C)C)=O)CCCN(C(C2CS(=O)C2)=O)CC1 55385,N1(C(C2(C)CCOC2)=O)CCN(C(c2cc(CO)on2)=O)C(CCO)C1 55386,CC(c1cccnc1)=CC(=O)NC1CCN(C(c2c[nH]nc2C2CC2)=O)C1 55387,Cc1ccc(OCC(=O)NCCCC(C)NC(C2(S(C)(=O)=O)CC2)=O)cc1 55388,C1(C(=O)NC(C2CCCC2)CNC(C2CCSC2)=O)Cc2ccccc2N1 55389,c1(C(=O)NCC2C(NC(C(CC=CCC)C)=O)COC2)coc2cc(F)ccc12 55390,C(=O)(CC1CCOc2ccccc21)N1CCC(C(C)Nc2ncccc2C#N)C1 55391,C(N=c1nc(N2CCC(C(N)=O)C2)c2ccccc2[nH]1)c1ncn(C)c1Br 55392,c1(C(CCN(C(C(CC(=C)C)NC(C)=O)=O)C)=O)cnn2ncccc12.C(CN)O 55393,C1(C(=O)NCC23CC(NC(C(C)SC)=O)(C2)C3)COC(=O)N1C 55394,N1(C(CC)C(=O)N(c2ccccc2C)C(C)C)CCC(C#N)(C(N)=O)C1 55395,c1(OCC)ccc(C(N2CSCC2NC(C23C=CC(CC2)C3)=O)=O)cn1 55396,Cc1cc(Cl)c(Cl)cc1C(N1CC2CC2(C(=O)Nc2ccnc(C(C)(C)C)c2)C1)=O 55397,C1(C(=O)NCC2(C)CC2)CC2(CCN(C(c3cccs3)=O)CC2)C1 55398,CC(C)(C)C(=O)CCC(=O)N1CC(C(=O)NC2CC(=O)N(O)C2)C(C)(C)C1 55399,CC1ON=C(C(=O)NCCN(CC(C)O)C(c2cc(-c3ccncc3)no2)=O)C1C 55400,c1(C(N(C)CC2CCCN2C(=O)C=CC2CCCC2)=O)cnc(N)cn1 55401,C=CC1(C(=O)N(C(C)CN(C)C(C)=O)C)CCN(C(=O)CC2CC=CCC2)C1 55402,C(c1ccccc1)=C(C(=O)NC(COC)CNC(C1(CO)CCCC1)=O)C 55403,C(=O)(CS(=O)(=O)C1CCCC1)NCCCC(C)NC(c1c(OC)csc1)=O 55404,Cc1nc(=N)[nH]c(=NCC(C)N(C)C(C2CC=CCC2)=O)[nH]1 55405,C(=O)(CC(C)(C)CC(F)F)N1CC(CN(C2CCCC2)C)C1 55406,c1(OC)ncc(CNC2CCC(C(=O)Nc3cnc(C)nc3)C2)cn1 55407,c1(CC)cccc(C(=O)NC2CC23CC(NC(=O)CCNC(=O)CC(C)C)C3)c1 55408,C1(OCC)CCCN(C(=O)C(C2(C)CC2)NC(C2CCC=CCC2)=O)C1 55409,c1(CC(=O)N(C2CCN(C(=O)C(F)CC3CC3)C2)C)ccn(C(F)(F)F)n1 55410,CC(C)CC(C(=O)NCC(=O)OCC1CC1)NC(c1cnn(C)c1C#N)=O 55411,CC1(C)CN(C(c2ncoc2C(F)F)=O)CC(CNC(=O)CCC2(C)CC2)O1 55412,Cc1nc2cc(C(=O)NCC(C)N(C(=O)CC3CC(O)C34CCC4)C)ccc2o1 55413,c1(C(=O)OCC)ccc(C2CCCCN2C(C2COC(C)C2)=O)n1C 55414,C(=O)(C1(C)CCc2ccccc21)N1CC(F)CC(NC(COCC(=O)OC)=O)C1 55415,CC(O)C(C)(C)C(=O)NCC(O)CC(N1CC2CSCC2C1)=O 55416,C(=O)(C1CCc2ccccc21)NCC1CN(Cc2sc3c(c2)CC(CC)CC3)C1 55417,C(C(=O)NN1CCCC1C(=O)NOC(CO)C(N1CC(C)N(OC)C(C)C1)=O)C 55418,S(=O)(=O)(c1ccc(Cl)cc1-c1ccc(O)c(SC)c1)N(CC(F)(F)F)CC 55419,c1(CC(=O)NC(C2OCCN(C(CC=CCC)=O)C2)C)c[nH]c2cc(F)ccc12 55420,C(CCc1ccccc1)(C(F)(F)F)NC(N(C1CCC1(C)C)C)=O 55421,Nc1cc(F)cnc1C(=O)NC1CC(CCNC(c2sccc2C2CC2)=O)C1 55422,N#Cc1ccsc1C(=O)NCc1ncccc1C(=O)NOCC1CCCCC1 55423,N1(C(c2c(N)ccc(CC)c2)=O)CC(NC(c2cnn3c2OCC3)=O)CC1(C)C 55424,C12(NC(CC=CC)=O)CCCC1N(C(=O)C(O)CC(C)(C)C)CCC2 55425,C1(SC)CN(C(c2[nH]c(O)nc2C)=O)CC1NC(=O)CC1CCC(=O)N1C 55426,C(=O)(C1(C)CCn2ccnc21)NC1CC(N(C(c2cc(OCC)ncc2)=O)C)C1 55427,c1(C(N(CCNC(CC=CCC)=O)CCC)=O)cc(Cl)cn1CC 55428,N1(C(C(=O)Nc2c(NCC)ccc(Cl)c2)=O)CCC2(CC1)CC2c1cccnc1 55429,C1(NC(CCCCCC)=O)CN(C(c2cnn(C(C)C)n2)=O)C2(CCOC2)C1 55430,C1(C(N2C(C(=O)NC3C(C(C)(C)C)C3)C(O)CC2)=O)CC2CC(=O)C1O2 55431,CC1(C)CC(NC(C2CCCCS2)=O)CN1C(C1CCCCC1n1ccnc1)=O 55432,C1(=O)C2c3c[nH]nc3CN2C(=O)C2CC(C2)N1C.C1(C(=O)OC)CC12CCCCC2 55433,c1(CC(N2CCN(C(C(CCCC)C)=O)CC2COC)=O)cc(F)c(Cl)cc1F 55434,C=CCCCCC(=O)N(CC(C)NC(C1CCN(C(C)C)CC1)=O)C 55435,C1(C(=O)NCC(C(C)C)NC(C2CCN(C3CCCCC3)C2)=O)CCCC2CC12 55436,c1(C(=O)NCC2C(NC(C(CCSC)O)=O)C2)occ2c1CCOC2 55437,c1(C(=O)NC2C(NC(C=NOC)=O)COC2)cnc2c(c1)NC(=O)CS2 55438,N1(C(c2cncc(N)c2)=O)CCC2CCC(C1)N2C(C1CCCS(=O)(=O)N1)=O 55439,C(=O)(CC(C)C(F)(F)F)NCC(C(=O)NCCc1nnc(C)o1)N(C)C 55440,c1(C(N2C(CNC(C(CCSC)OC)=O)CCC2)=O)cc(F)cc2nc(S)[nH]c12 55441,N1(C(C(N2CCSCC2)C)=O)CCCOC(CNC(=O)CC(C)CN(C)C)C1 55442,C12(C(N(CC#C)CCOC)=O)COC(C1)C(NC(=O)C(C#N)C(C)C)C2 55443,C1(C)(NC(C(N2CCCCC2=O)C)=O)CCN(C(=O)Cc2c[nH]c(=N)nc2O)CC1 55444,C(=O)(C(O)C(C)(C)C)N1CC(CNC(c2cc(C)sc2C)=O)C(C(F)(F)F)C1 55445,c1(C(N2CC3(CCCN(C(CCC(=O)OC)=O)C3)C2)=O)cn(C)c(=O)c2cncn12 55446,c1(C(N2CCC(NC(C3C(CC(C)C)C3)=O)CC(O)C2)=O)ccc(F)c2occc12 55447,c1(C(=O)NCC2CCN(C(C=CC(C)C)=O)C2)cc([N+](=O)[O-])cc2c1OCCO2 55448,CC1c2cc(Br)ccc2OC1C(=O)Nc1coc(C(C)(C)C)n1 55449,N1(C(C(C(=O)NCC)F)=O)CCN(C(c2cc(OC)nn2C)=O)C(CC(F)F)C1 55450,C(=O)(C1=C(C#N)CCC1)NCCCC(C(=O)NC(C)Cc1ccccn1)O 55451,C12(N)CCCC1OCC2.NC(=O)CCN(C(C(=O)NCCO)=O)CC(F)(F)F 55452,C12(NC(C(C)OCCCC)=O)CCC(CNc3cc(CC)nc(C)n3)(CC1)OC2 55453,C(=O)(C(=O)C(C)CC)N(C(COC)C)C(=O)CNC(=O)OC 55454,C(C)(C)(CCC(=O)NC1CC2(C1)CC(C)C2)NC(C(c1ccccc1)C)=O 55455,N1(C(CC2C(C)(C)C2(C)C)=O)CCOCC(NC(c2cccc(Cl)c2Cl)=O)C1 55456,c1(C(=O)NC2CC(F)(CNC(CC(CC)OC)=O)C2)ccc(OC)cc1F 55457,C(C1=CCCSC1)(c1nnnn1C1CCCCC1)Nc1cccc(NC(CC)=O)c1 55458,S1(=O)(=O)c2ccc(cc2Cl)NCC2CN1C2.N1(C(C(C)CO)C)CCOCC1C 55459,CC1c2c[nH]nc2CCC1C(=O)NC1CCN(C(=O)CC(C)(F)F)CC1F 55460,c1(C(=O)NCC2C(C(=O)NCCCc3nc(=N)[nH][nH]3)COC2)ccc(Cl)cc1 55461,C(CCC(C)C(=O)NC1C=CCN(C(c2cc(-c3ccccn3)[nH]n2)=O)C1)OC 55462,C(=O)(C1SCc2cccnc21)N1CC(CNC(CN(C)CC)=O)C(F)(F)CC1 55463,c1(C(=O)NC(C2CN(S(=O)(=O)CBr)C2)C)ccc2c(c1)CCCC2 55464,C(CC(C(=O)N(C)Cc1ccoc1)NC(c1c[nH]nc1C)=O)OCC 55465,N1(C(C(c2c(C)cccc2)(F)F)=O)CC(CNC(c2cncn2C)=O)CC(C)C1 55466,c1(OC)ccc(C(=O)NC2CCN(C(c3nc(C)ccc3C)=O)CC2C)c(F)n1 55467,C1(CC)CN(C(c2ccccc2NC(=O)NC)=O)CC1Cc1nc(=O)n(C)[nH]1 55468,c1(OC)cc(CC(C(C)C)NC(C2CC2C(N)=O)=O)ccc1O 55469,CCCCC(C(=O)N1CCN(C(C2CCCN2CC)=O)C(C(C)C)C1)C(C)C 55470,C(=O)(CCC(N)=O)NC1(C(N(C)OCC#N)=O)CC1c1ccccc1 55471,CC1OCCC1CNC(C1CC(NC(c2ccc(C3CC3)s2)=O)C1)=O 55472,Cn1ncc2cc(C(N3C4CCC3COC4)C(=O)NCc3ccccc3)ccc12 55473,N1(C(C2(C(C3CCOCC3)=O)CCC2)=O)CC2CC(C1)C2N=c1[nH]nc(CO)s1 55474,N1(C(c2cnn(CC)c2Cl)=O)C2CCCC1CN(C(C13CCCN1CCC3)=O)C2 55475,N1(C(C(Cc2ccc(OC)cc2)C)=O)CCN(C(=O)C=CCBr)C(C(C)(C)C)C1 55476,c1(CC)c(C(=O)N(C)CC2CCN(C(=O)CSC)C2)nnn1C 55477,N1(C(c2cc(CC)c(F)cc2)=O)C(CNC(=O)C(C)OC)CC2CCCC12 55478,C(C(N=[N+]=[N-])C(=O)N1CC(NC(C2CC2C2CCCC2)=O)CCC1C)OCC 55479,CN1CCN(C(c2cc(Cl)cs2)=O)C(C(N2CCCC2(C)C2CCC2)=O)C1 55480,C(CC(=O)NNC(=O)C(C)(C)CCCCOC)(CC)(O)OC(C=CC(=O)OCC)=O 55481,c1(OCc2cc[nH]n2)ccc(NC(c2ccccc2)C2CCOC2C2CC2)cc1 55482,N(C(=NCCCC1CC1)NC1CCS(=O)(=O)C1)CCC(=O)NC.C(Cl)S 55483,c1(C=O)cc(F)cc(Br)c1C.C1(OC)C=CCN(C(C2CCCC2C(N)=O)=O)C1 55484,CCCC(CCC)=CC(=O)NCC(C)N(C(=O)CNC(c1ccc(Cl)nc1)=O)CC 55485,CC(C)C1=NOC(C(=O)N(CC)CC2(O)CCCN(C(=O)CCC=CC(C)C)C2)C1 55486,Cc1ccnc(O)c1C(=O)NCC(C)NC(=O)Cc1nnc(-c2ccccc2)o1 55487,C(=O)(C1=CC2C=CC(C1)C2)NC1C(CNC(CN(C(C(C)C)=O)C)=O)CCCC1 55488,N1C(=NCCC(F)F)NCCc2cccc(c2)C1.C1(=CC)CCNC1 55489,C1(NC(CCCc2onc(C)n2)=O)CN(C(=O)CC23CCCC2C3)CC1C(F)(F)F 55490,c1(C(=O)NCCC(CNC(CCc2cc(C)on2)=O)O)cccc(CC#N)c1 55491,C(CCN=c1[nH]c2ccc(Br)cc2s1)OCCNC(=O)CC1CC2C=CC1C2 55492,c1(C(=O)NC(CNC(c2c(CC)ncs2)=O)C(C)C)ccc2nnn(O)c2c1 55493,CC1(CNC(c2nc(Cl)c(Cl)s2)=O)CCCN1C(c1cc(=O)cc[nH]1)=O 55494,C#Cc1cnc(C(=O)N(CCC(C)NC(c2cccc(CC)c2F)=O)C)c(C)c1 55495,n1(CCC(=O)NC)c(=O)c2ccccc2n1C(=O)C(CCCC(C)C)C(C)C 55496,c1(NCC2CCN(C(C)=O)C2)cccc(F)c1[N+](=O)[O-].c12ccc(cc1)CN2CC 55497,C1(CNC(CNC(CC)=O)=O)(NC(=O)C2=CCOCC2)CCCCC1C 55498,c1(CNC(C2(CC)CCN(C(c3c(CC)n(C)nn3)=O)C2)=O)nn(C)c(=O)n1C 55499,c1(C(=O)NC(C(=O)N(CCO)CC)c2ccco2)cccc(O)c1F 55500,C1(C(N2CC3(CC3)CC2CO)=O)N(C(c2cc(C3CC3)[nH]n2)=O)CC12CCCC2 55501,C1(C(N2C(CCNC(=O)C(C)NC(C)=O)CC(OC)C2)=O)Cc2nccnc2C1 55502,C(=O)(C(C)CCCOC)N1C(CC(NOCC(CC)C)=O)CCC1 55503,C1(CNC(C2N(CC#C)CCC2)=O)CC2(CO1)CN(C(=O)C(C)(C)CC=C)C2 55504,C1(C(N2CCC(C)(NC(C3CN(C(=O)OC(C)(C)C)C3)=O)C2)=O)CCC2CC1CO2 55505,C1(C(=O)NC(CNC(C=CC=CC)=O)C)CCC(C)C1 55506,C12(CNC(CCOC)=O)CCCC1N(C(c1cc(C3CC3)ncn1)=O)CCC2 55507,c1(OC)ccc(NC(=O)C(c2ccc(N(C)C)cc2)N2CCC3CC23)cc1 55508,n1(CCS(C)(=O)=O)nc(CC2CC2)nc1-c1ccc(Cc2cccc(F)c2)nc1 55509,C(CCCC(C)NC(=O)CC1CC1(Cl)Cl)NC(C1(OCC)CCCC1)=O 55510,C=C1CON(C(=O)CC2CCC(NC(c3ccc(C)cc3)=O)C2)C1 55511,N1(C(C(COC)(C)O)=O)CC(NC(c2ccc(OC(C)C)cc2F)=O)CC(O)C1 55512,N1(C(C(=O)NC(CC(C)C)c2ncccn2)=O)CCc2cc(Cl)ccc2C1 55513,C=CCC(C)C(=O)NC1(C(=O)NCc2cnn(C)c2C(C)C)CC1(C)C 55514,C1(NC(c2cn(C(C)C)nc2)=O)CCCCC1CNC(c1coc(Cl)n1)=O 55515,N1(C(c2ccsc2)=O)CCN(C(N2CCC(c3cc(O)ns3)C2)=O)CC1 55516,C1(C(=O)NCCn2ccc(C(N(c3ccccc3)C)=O)n2)CC12CC(F)(F)C2 55517,C1(O)(C(C)NC(=O)Cn2cccn2)CCN(C(=O)C=CCn2cncn2)C1 55518,CC(CC(=O)N(C)CCC1CCCCN1C(C1CCCO1)=O)P(C)(C)=O 55519,CC(C)C(CNC(=O)CC(=O)N(C)C)C(=O)N(C1CCCC(O)C1)C 55520,CCCC(CCC)=CC(N1CCC(CNC(=O)CSc2nnnn2C2CC2)C1)=O 55521,CC(C)CC(O)CC(=O)NCC1CCCN1C(=O)CCc1ccccn1 55522,C1(NC(C2CC2(F)C(=O)OC(C)(C)C)=O)CCN(C2CC2)CC1.C(=O)(CO)N 55523,C(=O)(CCCCCO)N1C(C)CC(NC(c2ccc(C(=O)CF)cc2)=O)C1 55524,N#Cc1c[nH]cnc1=NCC1(CNC(c2ccnc(Cl)c2Cl)=O)CC1 55525,C1(C(C)NC(CSCCOC)=O)CC2CCC(C1)N2C(=O)C=CC(C)CC 55526,C1(C(=O)NCC)CS(=O)(=O)CCO1.[NH+](C)(C)C 55527,c1(CC(=O)NCC(CC=C)NC(C2(Br)CC2)=O)cc(OC)ccc1F 55528,N1(C(C(=CC2CCCC2)C)=O)CCCC(CCNC(c2cc(C)ccn2)=O)CC1 55529,c1(C(N2C(C)(CNC(c3c(C)cn(C)c3)=O)CCC2)=O)cc2c(C)n[nH]c2cn1 55530,C12(C(=O)N)CC(C)(C1)OC2(C)C.c1(N2CCC(CNC(C)=O)C2)cccc(CO)c1 55531,c1(CN2C(C(=O)Nc3ccc(CCO)cc3)CC(F)(F)C2)cc(Br)c(O)cc1O 55532,C#CCC(C)(C)C(=O)N1CCC(COC)(NC(C2CC2CCC)=O)C1 55533,c1(CC(N2C(C)(CNC(C(C)OCCC#C)=O)CCC2)=O)cc(F)cc(Cl)c1 55534,c1(C(=O)NCC(CN(C(C2CC(C)SCC2)=O)C)C)ccc(F)c(CO)c1 55535,c1(NCC(C(C)C)O)ccc(S(=O)(=O)NC2CC3OCCCC23)c(Br)c1 55536,N1(C(C(C)N(C)C)=O)CCN(C(c2cncs2)=O)CC1c1cc(F)ccc1F 55537,C(=O)(CC1CCCc2c1[nH]c1ccccc21)NC1C(NC(CC=C)=O)COCC1 55538,C1(CNC(=O)C2=CCCCCC2)CN2CCCCC2CN1C(=O)Cc1ccon1 55539,C1(CC(=O)NC2(CC=C)CN(C(c3ccn(C4CC4)n3)=O)C2)C=CS(=O)(=O)C1 55540,N1(C(C(C)OCC=C)=O)CCCC(O)(c2cn(-c3ccc(=O)n(C)c3)nn2)CC1 55541,C1(OCC)CC2CC(NC(CC)C(=O)NCC(F)(F)F)CC12 55542,N1(C(C2CN(C(C)=O)C2)=O)CCC2CN(CC(=O)C(F)(F)F)CC12 55543,C1(C(=O)NC2C(SC)CN(C(C3CCOC3(C)C)=O)C2)COCC(C)(C)O1 55544,N1(C(C)=O)CCCCC1C(=O)NCC=CCNC(c1sc(F)cc1Br)=O 55545,c1(C(=O)NCCCNC(=O)CCNC(=O)NC2CC2)cccc2oncc12 55546,c1(OC)cc(C(=O)NC(C2CN(C(=O)C(C)(C)CN(C)C)CCO2)C)cc(Cl)c1 55547,C1(NC(CSCC#C)=O)CCN(C(c2cnn(C3CC3)c2C)=O)CC1(C)C 55548,C1(NC(C2(C)CC2(Cl)Cl)=O)CC2CC(C1)N(c1ncc(Br)c(O)n1)C2 55549,Cn1cncc1C(=O)NCc1ocnc1C(=O)NCCC1CC1C1CC1 55550,Cc1ccc(CNC(=O)Nc2nc(C3CCCN(C(=O)C(F)Br)C3)n[nH]2)c(C)c1 55551,C1(O)(CCNC(=O)C(O)C2CCC2)CN(C(=O)CC2CCOC2=O)C1 55552,C(C(CC(C)C)C(=O)N1CCOCC1CNC(c1cn2cnnc2cn1)=O)OC 55553,c1(C(=O)NCC(C)N(C(c2cccc(CC)c2)=O)CC)cnc2n1CCC(C)C2 55554,Cc1cnc(CN2CCCC(N(CC(N3CCCC3)=O)C)C2)cn1 55555,C(=O)(C1(C)OCCc2ccccc21)NCC(C(C)C)(C)NC(=O)CC12CC(C1)C2 55556,c1(C(N2CCC(O)(CNC(C3C(OC)C3)=O)CC2)=O)cc([N+](=O)[O-])ccc1C 55557,c1(OC(C2CCC(C)(C)CC2)C(=O)OC)cc(=O)c2cc(Br)ccc2[nH]1 55558,c1(Cn2ccnn2)ccc(OC)c(OC)c1.C1(C(=O)OCC)C2CN(C(C)C)CC12 55559,c1(NC(C(=O)NCC2CC(=C3CC3)C2)=O)cncc(C2CCOCC2)c1 55560,CCCCC(O)C(=O)NC(C1CCN(C(c2cccc(CN(C)C)c2)=O)C1)C 55561,N(C1CCc2cc(Cl)ccc21)C(C1(C(F)(F)F)CC(O)C1)=O 55562,N1(C(C2(CC)CCCN(C(=O)CC3CC4CCC3O4)C2)=O)CC(C)CCCC1C 55563,c1(C(C(=O)OCCC)NCCSCCC=C)nccc(Cl)c1F 55564,c1(C(C(=O)NC(C)C)N(CC=C)Cc2cccnc2)c(Cl)c(C)nn1C 55565,c1(CC(=O)N(c2cccnc2)CC=C)ccoc1C 55566,c1(C(=O)NCCC2CN(C(=O)Cc3ccsc3)CCO2)cccc2c1OCC2 55567,N1(C(C(c2ccccc2)C)=O)CCC(CCCNC(C2CCC2)=O)CC1 55568,C(=O)(C(C)C1=CCCC1)N1CCCCC(NC(c2cccc(C#C)c2)=O)C1 55569,CCC(C)C(C)NC(C1(C=CCN(C(=O)C(C)c2cccs2)C)CC1)=O 55570,CCC1=NOC(C(=O)NCC2CC(C)N(C(=O)CCc3cnccn3)C2)C1 55571,c12ccc(nc1)[nH]c2=O.CCC(C(=O)NCC(C)(O)C1(C)CC1)NC(C)=O 55572,c1(C=O)cc[nH]n1.C1(=O)CCN1.C1(=O)CN(C)N(CC)CCN1.C(=O)OC 55573,C(CC(C)C(=O)N1CC(OCCNC(c2cnc(N(C)C)s2)=O)C1)OC 55574,c1(C(=O)NC2CC(=O)N(C3CN(C(=O)Cc4ccoc4)C3)C2)ccc(Cl)c(F)c1 55575,c1(C(C(N2CCC(NC(=O)OCC)CC2)=O)=O)ccc(F)c(C)c1.C1CS1 55576,CCCCCCC(C)C(=O)NC(CC1CC1)C(N1CC2CCC(C1)N2CC)=O 55577,CC(Cc1ccnn1C)C(=O)N1CCC1CNC(=O)CCc1ccccc1 55578,c1(N2CCn3c(C)ncc3C2)nc2c(c(=NCCSC(F)F)[nH]1)CCCCC2 55579,c1(CC(=O)N(CCNC(C2CCC(C)O2)=O)CC)cc(OC)cc(OC)c1 55580,Cc1ccc2c(c1)C=C(C(=O)NC1CCOC(CNC(C3CC3F)=O)C1)CO2 55581,N1(C(C=CC=CCC)=O)CC2CCCC2(NC(c2cc(C)cnc2OC)=O)C1 55582,C(=O)(C(CC1CCCC1)C(C)C)N1CCC(NC(Cc2c(C)onc2)=O)CC1 55583,C(CC(F)CN=[N+]=[N-])NC(C1(CCN(C(C(CC=CCC)C)=O)C(C)C)CC1)=O 55584,c1(OC)[nH]c(=N)ccc1C(N1CCN(C(C)CNC(C2(CF)CCC2)=O)CC1)=O 55585,N1(CCNC(C2C(C)C2(F)F)=O)CCC(C(c2cncn2C)c2nnnn2C)C1(C)C 55586,CC1CN(N2CCNC(=O)C2)CC(C=O)O1.C(=O)(C(C)(F)c1ccon1)CCO 55587,CCC(CC)(C(N)=O)NC(c1cn(CCNC(=O)CC2CC(F)(F)C2)nn1)=O 55588,CC(C)C(CCC(=O)NC1CC=CCC1C)NC(c1cn(C)c(=O)cn1)=O 55589,C#CCCC(C(=O)NCc1cc(C(N)=O)n[nH]1)NC(=O)COCC#CC 55590,c1(CC)ccc(C)nc1NCC(C)NC(C1CCOC(=O)N1)=O 55591,C1(C(=O)NCCNC(=O)C=C(Cl)Cl)CCC2CCC(=O)N12 55592,C1(F)(CNC(C(C)C)=O)CC2CCC(C1)N2C(=O)C=Cc1nccs1 55593,C(=O)(C(F)C(F)(F)F)N(C(CNC(c1cccc(CC)n1)=O)C)CC 55594,C(=O)(C1=NNC(=O)CC1)N(CC(CC)NC(c1ccc(Br)c(N)c1)=O)CC 55595,C=CCC(C(=O)NCCCN(C(=O)C(C=C)CC)C1CC1)C(C)(C)C 55596,CC1=C(C(=O)N2CC(NC(C3(C)CCCS3(=O)=O)=O)C2)SCCO1 55597,N1(C(C(CC)CO)=O)CCC(NC(C2(O)CCSC2)=O)C(C)C1 55598,[N-]=[N+]=NCC(C(=O)NCCOC1CC1(F)F)NC(C1CCN(CCF)C1)=O 55599,c12cnc(cn1)[nH]2.c1(C(=O)NC2CC(C(=O)NCCF)C2)cccc(Cl)c1 55600,N1(C(C(CCC)C)=O)CCC2(CC1)CN(C(C1C=C1C)=O)C2C(C)C 55601,c1(OC)ccc(CCC(C)N)cc1.C(C(C)(C)CF)Cc1nnnn1CCCF 55602,c1(CC)cc(C(N2CCC(NC(=O)C=CCN(C)CC)C2(C)C)=O)c(C)nn1 55603,CCC(CC)C(C)C(=O)NC1CCN(C(c2ccnc3ccsc23)=O)C12CC2 55604,C1(NC(CCC=C)=O)COC2(CCN(C(c3cncc(O)c3)=O)CC2)C1 55605,C1(OC)(CNC(c2cccc(C3(C)COC3)c2)=O)CCN(C(=O)C(N)=O)C1 55606,N1(C(c2cn(CC)nn2)=O)CCC2CN(C(=O)Cn3c(C)cc(O)cc3=O)CC12 55607,c1(C(N(C2CN(C(C=CCC)=O)CC2F)C)=O)ccc(=O)n(-c2ccccc2)n1 55608,CC1(C)CC23N=C1S(=O)CCN1C2=NN=NN2C(C)(CCC3CCC2CC)CC1 55609,C(CCCCC(=O)N1CC2CC(C1)C2NC(c1ncc(N)cc1Cl)=O)OC 55610,N1(C(=O)CCc2ccccn2)CC2CCC2(CNC(C23CC4CC2C3C4O)=O)C1 55611,CC1(C)CCN(C(C2CCN(C(=O)c3cccc(CN(C)C)n3)O2)=O)CC1 55612,c1(CC(=O)NCCCOCCNC(c2cc[nH]c2)=O)ccc([N+](=O)[O-])cc1Cl 55613,C(C(=O)N1OC2CCC1CC2)C1OCCN(C(=O)CC2CCOCC2)C1 55614,Cn1nc(C(N2CC=C(CNC(=O)Cc3cccnc3)CC2)=O)c2c1CCSC2 55615,C(=O)(CC(CC)C(C)(C)C)N(CC(C)(C)CNC(=O)CNC(=O)CCCF)CC 55616,CC1(C)C2CCC1(CC(N1CCN(C(=O)C(O)CC3CC3)CC1C(F)F)=O)CC2 55617,N1(C(C(CC)N(C)C)=O)CCCCC(NC(c2cc(COC)on2)=O)C1 55618,c1(NC(C2CC23CN(C(C2CC2c2ccccc2F)=O)C3)=O)cc(I)ccc1CO 55619,N1(C(c2cc(COC)oc2C)=O)CCC(C)C(N(C)C(C2CC3(CC3)C2)=O)C1 55620,c1(C(=O)NCC2(C)C(C)CN(C(=O)Cc3ccnn3C)C2)nnn2ccccc12 55621,N1(C(c2ccnc(C)c2O)=O)CCOC2(CCN(C(C3CCCC3(F)F)=O)C2)C1 55622,N1(C(C(C)N(C)C(C2CCC(CO)CC2)=O)=O)CCCC(C(C)O)CC1 55623,C=CCC(CNC(=O)CCn1cncn1)C(=O)Nc1ccc(O)nc1 55624,c1(C(C)C(=O)N2CC(CCNC(C34COCC3C4)=O)C2)c(Cl)cccc1Cl 55625,C1(C(N2CCC(SCC)CC2)=O)CC2(CC2)CN1C(C1CCCC1OC)=O 55626,c1(C(N2CC(CNC(C=CCOC)=O)C3C2C3)=O)ccc(=O)n(C)n1 55627,CC(C)CCCC(=O)N1CC(O)CCC1C(=O)NCc1cccnn1 55628,Cc1cc(CCCOc2ccc(Br)c(F)c2)c(C)n1C.C12CC(C1)C(=O)N2 55629,c1(C(=O)NC(C(C)C)(C)CNC(C2(O)CC2)=O)ccn2cnnc2c1 55630,c1(NC(=O)N(C(c2c[nH]c3c2CC(C)CC3)=O)C2CC2)cc2c(cc1O)OCO2 55631,c1(NCC(C(F)(F)F)OCC)nc(N2CCCC(C)(F)C2)nc2sccc12 55632,C(=O)(CCCCC(N)=O)NC(c1cccc(C)n1)C.C12CCC(C1)NC2=O 55633,C(C(CC(F)(F)F)NC(C1(C2CC2)CCCO1)=O)NC(c1cnc(OC)nc1)=O 55634,C(C)(CNC(=O)Cc1cnc(C(F)(F)F)s1)(CO)NC(C(C)OCCC(C)C)=O 55635,C1(CNC(C2CCCC2c2nc[nH]n2)=O)CCCCN1C(c1ccsc1Cl)=O 55636,Cc1coc(C)c1C=CC(N1CCC(NC(=O)C(c2cncn2C)O)C1C)=O 55637,C(=O)(C1=Cc2ccc(Cl)cc2OC1)N1C2CC(NC(C(C)CF)=O)CC1CC2 55638,c1(OCC)nc(C(=O)NC(CNC(c2ccn(C3CCOCC3)n2)=O)CC)ns1 55639,c1(CC(=O)N(CC(=O)NCC(=O)NCCC(O)C2CC2)C2CC2)cccc(F)c1 55640,c1(C(=O)OC)cc(Cl)ccc1NC(C)C.c1(C2C(=O)N2C)cccc(Cl)c1 55641,N1(C(C(CC)(O)c2ccccc2)=O)CCC(C2CCN(c3ncncc3Br)C2)CC1 55642,C(CCNC(=O)CCc1ncc(C)[nH]1)(C(C)(C)C)NC(c1cnn(CC)c1C)=O 55643,C12(CNC(CC3(C=C)CCC3)=O)CC(CO1)N(C(=O)CCC1CCCN(C)C1)C2 55644,C(=O)(CCC(C)CN(C)C)N1C(C(=O)N(C)Cc2cncnc2)(CC)C=CC1 55645,CC1(C)CN(C(=O)C#CC2CCOC2)CCC1NC(c1ccccc1)=O 55646,C#Cc1cc(C(=O)NCCn2cc(CNC(=O)CC(C)SC)nn2)cc(F)c1 55647,c1(OCCCC)ccc(Cl)cc1NC(=O)NCC1CC2(CCC2)C1 55648,C1(C2CC2)(C(N2CCC(NC(c3sccc3F)=O)CC2)=O)CC=CC1 55649,Cn1nnc2cc(C(=O)NC3CC4CCC(C3C)N4c3ncccn3)cnc12 55650,C(=O)(C(CNC(=O)CCC1CC1C)CC(C)C)NCc1ccc(C)s1 55651,C(=O)(C(CO)C(C)(C)C)NC(CC=CC(=O)NCC(CCC)O)(C)C 55652,N1(C(c2cccc(C)c2)=O)CCN(C(=O)Cc2csc(C3CC3)n2)C(C)C1C 55653,Cc1cc(F)ccc1NC(=O)C(Cc1cc[nH]n1)NC(c1ccncc1O)=O 55654,C(=O)(CCCS(N)(=O)=O)N1CCC(NC(C(C(C)C)n2ncc(C)c2)=O)C1 55655,C12(NC(C=CC(C)N(C(=O)Cc3cnns3)CC)=O)CCCC1CCC2 55656,c1(-n2cc(CN(C=O)C(C3CCS(=O)CC3)=O)nn2)ccnc(C(=O)O)c1 55657,C(CN=c1[nH]c(NCCC=CCn2cnnc2)nc2ccccc12)=CC 55658,N1(C(C2CC2CN)=O)CCOCC1c1nc(C(F)(F)F)cs1.c12ncc-1s2 55659,c1(C(=O)NC2C(NC(C3(CC(=O)OC)CC3)=O)C2)ccc(-c2ccncc2)o1 55660,O=C1CN(CC2CCCCC2O)C(=O)N1CC1COC1 55661,CC(C)C(C(=O)NCCCCCNC(c1ccccn1)=O)SCc1ccccc1 55662,C1(CCNC(C(C=C)(C)O)=O)CN(C(=O)C(C)OC2CCOC2)CCCO1 55663,N1(C(CC(=C=C)C)=O)CC2(CCN2C2CC2c2ccc(-c3cccnc3)cc2)C1 55664,C1(C(C)NC(C(Cn2ccc(C)n2)C)=O)CCN(C(=O)CSCC(N)=O)CC1 55665,CCC(C)CC(C)C(=O)NCC(=O)NC1CC1CCN1CCCCC1 55666,N1(C(C2CCCC(C)C2)=O)CCCN(C(=O)C=Cc2ccc(=O)n(C)c2)CCC1 55667,N1(C(c2c(C)cn(C)c2)=O)CCCC(O)(CCNC(=O)C=C2CCC(C)CC2)C1 55668,C12(N(C(CSCc3nc(C)sc3)=O)CC)CCCC1CN(C(=O)C(F)(F)CC(C)C)C2 55669,C(N=c1ccnc(NC2CC2C2CC2C)[nH]1)c1cncc(C)c1 55670,C1(C#N)(CC(=O)NCCCN(CC)CC2CCCS2)CC1 55671,c1(NC(c2nnn(C)n2)c2n(CC3CC3)nnn2)ccc2c(c1)CC(O)C2 55672,C(N=c1[nH]cnc(C(C)C)c1Br)C1N(C(C(COCC)OC)=O)CCCC1C 55673,C(c1ccnc2ccccc12)=CC(N1CCC(F)(CNC(C(C)CO)=O)C1)=O 55674,Cc1nn(CC(=O)NC2CC(NC(=O)C(C)N(C)C)C2)c(C)c1[N+](=O)[O-] 55675,c1(N2C(S(C)=O)CCCC2)[nH]c(=NCc2cnsc2)nc2c1CCC2 55676,c1(C(N2CCCC(CCNC(CC(C)F)=O)C2)=O)ccn2ncccc12 55677,CC(C)(CNC(c1cc(Cl)cs1)C1CC1)CC1CN(C(=O)Cn2ccnn2)C1 55678,CCCCCC(=O)NC1COCCC1NC(c1cnc(C2CC2)[nH]1)=O 55679,C1(CC(N2CCC(O)(CN(C(C3CC(OC)C3)=O)C)C2)=O)CC2(CCC2)CO1 55680,c1(CNC(C(=O)Nc2cn(CCOC)nn2)=O)cccnc1O 55681,CC1C(C(=O)NC2CC3CC(C2)NC3)CCCN1C(=O)OCC(F)(F)F 55682,C(=O)(C1=NOC(C)C1C)NC(C1N(C(c2ccc(OC)cc2OC)=O)CCC1)C 55683,C(CC(C)(C)C)(C(=O)NCc1ccccc1Cl)N(C1CCN(C(=O)C2CC2)C1)C 55684,c1(C(=O)NC(C)Cc2nncn2C)n[nH]c2c1CN(C(=O)C(=O)C1CCCC1)C2 55685,C1(NC(c2cn(C)cc2C(F)(F)F)=O)CN(C(=O)CC2C=CCC2)CCC1F 55686,Cc1ccc(C(N2CCC(NC(=O)C=CC3CCCO3)C(F)C2)=O)c(N)c1 55687,C(CN=c1[nH]c(=NC2CCC(C3CC3)CC2)[nH]c2c1COCC2)C1(SC)CC1 55688,C1(C(N(CCC(C)NC(c2ccnc(OC)n2)=O)C)=O)COc2ccccc2O1 55689,CN1C(=O)CCC1CC(=O)NC1CC(CC(=O)NCC=CCl)C1 55690,CC(C(=O)N1CCCC(NC(c2cnc(N)c(CO)c2)=O)C1)C(C)(F)F 55691,C(C(=O)N(CCCN(C)C)C(C)C)(SC)SC.C(=O)(CO)N 55692,C1(C)(C(N(C(C)CNC(c2ccc(F)c(C(F)F)c2)=O)C)=O)CC(C2CC2)=NO1 55693,N1(C(C(CC=C)C)=O)CCC2(CC2C(=O)NCC2CCNC(=O)C2)C1 55694,c1(NC(=O)NCc2onc(CC)n2)cccc2ccncc12 55695,Cc1c(C(N2CCCC2CCCNC(=O)CC(C)CF)=O)ccn1C(C)C 55696,c1(C(=O)NC(C)CCN(C(=O)CC2CC3(CCC3)C2)C)cccc2nccn12 55697,C1(OC)CN(C(c2ccncc2)=O)CC1NC(c1ccc(-n2cccn2)nc1)=O 55698,N1(C(C(C2(C)CC2)NC(CC(=O)OC(C)(C)C)=O)=O)CCOC(C)(C2CC2)C1 55699,N1(CC(=O)NC(C(=O)N(c2cccc(O)c2)CC)C(C)C)CCN(C)C(=O)C1 55700,N1(C(C(COC)C)=O)CC2(CCN(C(=O)C(C)Cc3ccncc3)CC2)C1 55701,N1(Cc2nc(C(C)NC(c3ccc(F)o3)=O)on2)CCC(C)(C(C)(C)N(C)C)CC1 55702,c1(C2C(OC(C)(C)C)C2)nc(-c2cc[nH]n2)nn1CC(C)(C)O 55703,C(C)(C(CC(=O)NCCC(C(C)C)OC)NC(C1CN2CCC1CC2)=O)OC 55704,Cc1cnc(CC(=O)N(C2CCN(C(C3CCSC3)=O)C2)CC2CC2)s1 55705,N1(C(C2CC=C(C)CC2)=O)CCCC(CNC(=O)C(F)=CCCF)CC1 55706,C1(CCNC(C2(NC(C)C)CC2)=O)CN(C(=O)CN2C(=O)CCC2=O)CC(C)O1 55707,C1(C(C)NC(=O)C(F)Cc2cccnc2)CN(C(C2(C#N)CC2)=O)CCO1 55708,C(CC(C(=O)NCCC(F)C(C)C)NC(=O)CC1CC=CCC1)OC 55709,Cc1c(C(=O)NCC(C2CCC2)NC(C2CSCCS2)=O)cnn1CCC(C)C 55710,Cc1c(C(=O)NCC2CCN(C(c3ccn4c3CCC4)=O)CC2C)sc2cncn12 55711,C1(CNC(C=CCCC)=O)CN(C(=O)Cc2c(C)n[nH]c2C)CC(C)(C)C1 55712,C1(O)(C(CNC(c2c(CC)noc2)=O)C)CCN(C(=O)Cn2cnnc2)C1 55713,c1(CC)nn[nH]c1C(=O)NC(C(=O)NC1CC2CC2C1)c1ccco1 55714,C1(NC(c2cc(C)[nH]c2)=O)CCCCC12CCN(C(c1cnc(F)c(C)c1)=O)C2 55715,C(=O)(C1=NOC(C)C1C)NC1(CC(=O)NCC(C2CC2)OC)CCC1 55716,N1(C(c2c(C)nc(O)cc2)=O)CC(CNC(=O)C(C)n2cnnn2)CC(C)(C)C1 55717,C1(NC(CCN(C)CC)=O)CCC(NC(=O)CCn2cnc(=N)[nH]2)CC1 55718,N#Cc1ccc(CN2CCCC(C(N3CCCC3CO)=O)C2)c(Br)c1 55719,c1(N2CCC(C(C)NC(c3cc(O)n(C)n3)=O)CC2)nc2ccccc2o1 55720,N1(C(c2ccc(C)c(C)c2)=O)CCC(NC(c2cnc[nH]2)=O)C(CO)CC1 55721,C1(NC(c2nn(C(CC)CC)c(C)c2)=O)C2CCC1N(C(=O)CC(C)COC)C2 55722,CN1CC(C(=O)NCC2(CNC(C3CCCCC3O)=O)CCCCC2)CCC1=O 55723,N1(C(C(C)(C)OC)=O)CCCC(CCNC(c2ccc(C)nn2)=O)CC1 55724,c1(C(=O)NCC(C)N(C)C(C2CCC(C)(C)O2)=O)cccc(O)c1F 55725,C1(CNC(C(CC)NC(C)=O)=O)C2CN(Cc3ncsc3Br)CC12 55726,N1(C(c2cc(OC)ncc2Br)=O)CCC(C)N(C(c2cnnn2C)=O)CC1 55727,c1(CNCc2cn(CCC)nn2)ccccc1C(=O)NCc1nncn1C 55728,C1(CC(=O)NC(CCC)CO)CN(C(=O)Cc2cncnc2)CCC1C 55729,C(=O)(CC(N=c1[nH]nc(C2CCC2)s1)c1cccnc1)Nc1ccccc1 55730,C1(C(=O)NCCc2cc[nH]n2)(CC)CCN(C(C2CCNC(=O)C2)=O)C1 55731,C1(C(F)(F)F)(C(N2CC(CC(C)NC(=O)CCc3cncs3)C2)=O)CCCC1 55732,C1(CO)CN(N2CC3CCCC(O)C23)CC12CCOCC2 55733,C(=O)(C1OCCc2ccccc21)NCC(C(C)C)NC(C(F)=C(C)C)=O 55734,c1(OCC(=O)N(C(CNC(C2(C=C)CC2)=O)C)CC)ccccc1C 55735,N1(C(=O)NCC2CC(C(=O)OCC)C2)CCC(C)=C(C)C1 55736,n1(C(C)C)ccc(=NC(=O)C(C)(C)CN(C(=O)C2=NOCC2)C)[nH]1 55737,C1(NC(CC2CC(C)NC2)=O)CCC2(CCC2)C1 55738,n1(CCOC)cnc(C(N2CC(NC(C3CC3(C)C(F)F)=O)C2)=O)c1 55739,N(C(=NCc1cnc(C)cn1)NCC(=O)NC(C)C)CCC 55740,C12(CNC(c3c(C)ccc(N)c3)=O)CCC(NC(=O)CSS(C)(=O)=O)(CC1)CO2 55741,c1(CC)cnc2ccccc2c1N1CCC(C)(C(=O)N(CC(C)(C)CO)CC)CC1 55742,C1(NC(C2CCC3(CC2)CC3)=O)CS(=O)(=O)C12CCN(C(CCO)C(F)(F)F)CC2 55743,CC1(C)C(C(F)F)CCN1C(c1cc(C(F)F)ncn1)=O 55744,N1(C(C(C=CC)O)=O)CCC(CNC(=O)C(O)C(C)(C)C)C(CC)C1 55745,N1(C(C(=O)NC)CCC2CC2)CCS(=O)(=O)CC1CCO.C=C1CC(C(=O)OC)C1 55746,CCCCC(C)(F)C(=O)N1CC2CCCC2(NC(c2cccc(C)n2)=O)C1 55747,c1(-c2cc(NC(=O)NC)ccc2)c[nH]c2cc(C(=O)NC3(C)CC3)ccc12 55748,C(=O)(C(C)S(N)(=O)=O)NCCC1N(C(c2cc(SCC)ncc2)=O)CCSC1 55749,c1(CC)ccnc(C(N2CCC(C(=O)N(C)CC3(O)CCC3)C2C(C)C)=O)c1 55750,C1(CN(C(=O)CC2CCCC2)CC)CCCCN1C(C1CSCN1C(C)=O)=O 55751,CCC(CC(=O)NCC(CO)NC(c1cnc(C2CC2)s1)=O)C1CC1 55752,N1(C2CCN(C(=O)C=CI)C2)CCN(C(=O)C(C2CCCCC2)O)CC1 55753,c1(NC(=O)NCCC2COCC2O)ccc(I)c(Br)c1 55754,C=C1CC2CCC(C1)N2C(=O)C(F)C(C)CNC(C1(C(N)=O)CCC1)=O 55755,c1(-c2cc(C)nn2C)ccc2[nH]c(C(=O)NC(c3cc[nH]n3)C)cc2c1 55756,C1(CNC(C2(OC)CCC2)=O)CCN(C(c2cccc(=O)n2C)=O)C12CC2 55757,C1(O)(C(=O)NC2C(NC(C3CC3c3ccc(O)nc3)=O)CCC2)CCCCCC1 55758,c1(C(N2C(CC)CN(C(=O)CCC3OCCO3)CC2)=O)cncc2cnccc12 55759,CCC(C)C(C(=O)NC1CC(C)(NC(=O)CCNS(=O)(=O)c2cccs2)C1)OC 55760,C1(C(=O)NC2(CC=C)CCN(C(c3nsnc3O)=O)C2)C2CCCCCC12 55761,C1(NC(C(C)CCO)=O)CC2CCC(C1)N2c1ncc(C#N)cc1F 55762,c1(C(=O)NCCCN2CCCC2)ccc(CNC(CNC(=O)OCC)=O)nc1 55763,c1(CN2C(C(=O)Nc3nnc(C)o3)CC(C)C2)c(C)nn(C)c1Cl 55764,C=C(C)CN=C(NCC1NC(=O)CC1(C)C)N1CCC(F)(F)C(C)C1 55765,C1(CC(=O)N(C(CNC(C=C(C)C)=O)C2CC2)C)CC(=O)c2ccccc2C1 55766,c1(C(=O)NCC23N(C(C4CCC(=O)C4)=O)CC(C2)C3)cc2c(s1)CCC2 55767,c1(C(=O)NCC(C2CCC2)NC(c2ccc(SC)o2)=O)nccc2n[nH]cc12 55768,C(c1ccc(O)cc1)=CC(=O)NC1(CCOC)CCN(C(C=CC=CC)=O)C1 55769,C1(NC(C(COC(C)C)NC(c2ccc(SC)o2)=O)=O)COCC1C1CC1 55770,c1(C(N2CCC(CN(C(=O)C=CC3CCC3)CC)CC2)=O)c(C)nn(CC)c1C 55771,C1(CN(C(=O)Cc2cccs2)C)CN(C(=O)CCNC(C2CCC2)=O)CCO1 55772,C(=O)(CC(O)C(C)C)NCC1(OC)CN(C(c2ccnc(-n3cccn3)c2)=O)C1 55773,Cc1nsc(C(N2CCC3C(NC(=O)CC4COCCN4C)C23)=O)c1N 55774,c1(C2(C(N(CCN(C(=O)CP(C)(C)=O)CC)CC)=O)CC2)ccnc(F)c1 55775,C(=O)(C(O)(C(F)(F)F)C1CC1)NCCC1(C)CC=CC1 55776,C1(CC(C(=O)NCC(C(C)C)(C)NC(=O)CC(F)F)C)CCC(F)(F)CC1 55777,C1(CNC(c2c(C)nc(C)s2)=O)CC(C(C)(C)C)CN(C(=O)Cc2cnoc2)C1 55778,C1(CC=C)(C(=O)NC2CCN(C(=O)Cn3cc(C#N)cn3)C2CC)CCCCC1 55779,CCC(C(=O)NCC1CC1NC(=O)C=CCN(C)C)NC(N)=O 55780,C1(C(=O)NCC2(NC(C(C(C)C)OC)=O)CCCC2)CCC(F)(F)CO1 55781,C(=O)(C1=Cc2ccccc2C1)NCC12C(CN(C(CCC)=O)C1)CCCC2 55782,CCS(=O)(=O)CCCN=C(NCC1CCCO1)N(C)CC1OCCO1 55783,C(C(=O)NCC(CCOC)NC(c1cnn(C)c1C)=O)(C(C)C)OCC 55784,CCCCCC(O)C(=O)N(C1C(N)C2CCCCCC12)c1ccccc1OC 55785,N1(C(CCC(C)OCC)=O)CCC(C)(C)C(NC(c2cc(C(N)=O)no2)=O)C1 55786,Cc1nc2cccc(C(N3CCN(C(C4COC(=O)O4)=O)C(C4CC4)C3)=O)c2[nH]1 55787,N12CCC(CC1)CC2=O.C1(C)(CSC)C(=O)N1.C1(C(C)C2CC2)CCC(C)C1.C(C)C 55788,C1(CN(C(C23COC(C2)C3)=O)CC)CCCN(C(c2nc(O)sc2C)=O)C1 55789,c1(CNC(C2CCC(C)(CC)O2)=O)nc2c(s1)CN(C(=O)COC(C)(C)C)CC2 55790,N1(C(C(C=C)O)=O)CC2CN(C(=O)Cn3c(C)cc(O)cc3=O)CCC12 55791,C1(O)(C(=O)NC2CN(C(CC(=O)OC)=O)c3c(cccc3)C2)CCCC(C)(C)CC1 55792,N1(C(c2cc(C)nn2C)=O)CC(C)CN(C(c2ccc(=O)oc2)=O)CC1C 55793,C1(CC(=O)NCC(C2CC2)N(C)C(c2cc(C)c(C)s2)=O)(OC)CCCCC1 55794,C(=O)(N=S(C)(=O)CCO)N(C(CC)Cc1ccc(Cl)cc1)C 55795,c1(CC(C)C(=O)NC(C2CN(C(C3COCCC3C)=O)C2)C)cccc(Cl)c1 55796,c1(CC)occc1C(=O)NCC(=O)NCC(N1CCCC1C1CCCO1)=O 55797,C(=O)(CC1=CCOCC1)N1CCN(C(c2c(Cl)c(C)n(C)n2)=O)C(C)C1 55798,C(=O)(CCCC(CC)NC(=O)CCCCCC)NC(C1CCOC1)C#C 55799,N1(C(C(CC)F)=O)CC2C(CNC(=O)CCc3nnc(C(F)F)o3)C2C1 55800,N1(C(CC=CC=C)=O)CCC2CCN(C(c3cc(C(N)=O)co3)=O)C2C1 55801,C(=O)(C1CCCn2nccc21)N1C(C2CN(C(CC3C=NN(C)C3=O)=O)C2)CC(F)C1 55802,Cc1cc(N)ccc1C(=O)NC(CNC(c1nc(O)c(C)s1)=O)C1CCC1 55803,c1(-c2ccc(OCCC)cc2F)nc2ccc(C(N3CCC(CO)C3)=O)cc2s1 55804,NS(=O)(=O)c1cncc(C(=O)NC23CC2CN(C(C2CCCCC2)=O)C3)c1 55805,N1(C(CC)CC)CC(C(=O)NC2CN(C(=O)CC(=O)NC3CC3)CC2C)CC1=O 55806,N1(C(CCC#C)=O)CCC(C)C1CNC(c1cnc(C(F)(F)F)s1)=O 55807,CON(C)C(=O)C1(c2nccs2)CC1.C(=O)(CC1CCC1)N 55808,C(C(O)C(=O)NCCCCC1CCC1)NC(C(C)C1CCC1)=O 55809,C12CCCN(C1)C2=O.N1(C(=O)CCc2csnn2)CCC(O)(C(F)F)C1 55810,c1(CSCC)cccc(C(=O)NC2CC2NC(C2(O)CCOC2)=O)c1 55811,C1(C(N(C)CC2(O)CN(C(=O)CN3CCSCC3)C2)=O)SC2C=CC1CC2 55812,C1(C(=O)NC(CCCNC(=O)CSc2nc[nH]n2)C)OCCOC12CCC2 55813,Cc1coc(C2CC2)c1C(=O)NCCCCNC(C12CCCCC1C2)=O 55814,Cc1cc(C(c2nnnn2C(C)C)NC(C)Cn2cnnc2)c(Br)cc1F 55815,c1(C(N2CC(SC)C(NC(=O)CCC3CC(F)(F)C3)C2)=O)n[nH]c2c1CSCC2 55816,N1(C(=O)NC(c2ccncc2)C)CCC(NS(=O)(=O)NCCC2CC2)CC1 55817,C1(CNC(COCC(C)C)=O)CC2(CCN(C(=O)C(O)CC[S+](C)C)C2)CO1 55818,C#CC1CCN1C(=O)C(Cn1ccnn1)NC(=O)C=C(C)C(C)C 55819,CCC(CCC(=O)Nc1ccccc1CCO)NC(=O)CC1CCCCC1O 55820,C1(NC(CC2(C)C(C(=O)OC)C2)=O)CC2C1CCN2C(c1ccnc(S)c1)=O 55821,N1(C(=O)COCC(F)F)CCC(O)(CCNC(C2(c3ccc(F)cn3)CC2)=O)C1 55822,N1(C(C2N(C(C)=O)CCCC2)=O)CCN(C)CC1CNC(=O)Cc1coc(C)n1 55823,N1(C(CC(=O)OCC)=O)CCC2(CC1)CC(NC(=O)CSc1cccc(O)c1)C2 55824,C1(C)(NC(C(C)OCCC(C)C)=O)CCCN(C(c2[nH]nnc2C2CC2)=O)C1 55825,C(CCSC)(C(=O)NC1CC2C(NC(c3cc(O)n(C)n3)=O)C2C1)OC 55826,CC(C)C(C)(O)CNC(=O)C(C1(O)CN(C(c2cc(C3CC3)ccn2)=O)C1)F 55827,CC1CN(C(c2ccnc(C(C)(C)C)c2)=O)CCC1NC(c1cc(=O)cc[nH]1)=O 55828,C1(N(C)C)CCC(C(N2CCC(CCNC(=O)CCc3nccs3)C2)=O)CC1 55829,N1(C(CS(=O)(=O)NC(C)(C)C)=O)CC2CN(C(=O)C(C)(C)CC#N)CC2C1 55830,N1(C(CC(CC)C2CC2)=O)CC(NC(=O)CCC(=O)NC)CC12CCCCC2 55831,c1(C(N2C(C3(NC(C(C)OCC#C)=O)CC3)COCC2)=O)ccccc1NC(C)=O 55832,C1(F)(CNC(Cc2ccn(C)n2)=O)CCN(C(C2CC(N3CCCC3)C2)=O)CC1 55833,C1(CCOC)CN(C(=O)CSc2n[nH]c(O)n2)CCN1C(=O)C(C)SC 55834,C(N1CCC(F)(F)CC1C)c1nnc(C(CC)C(=O)N2CCOCC2)o1 55835,c1(-c2nnc(N3C(C)(C)CC=CC3)n2CC2CCOC2)ccc2nc[nH]c2c1 55836,CCC(O)C(C)C(=O)NC1(c2ncc(C)o2)CC1.C123CC(C1)(C2)C(=O)N3 55837,C1(O)(CNC(=O)Cc2ccccc2O)CCN(Cc2cc(O)cc(Br)c2)CC1 55838,N1(C(CC(C)(C)O)=O)CCC2(CC(C(=O)Nc3cc(Br)ccc3I)=NO2)C1 55839,Cc1ncc2n1CC(C(=O)NC1CN(C(C3CCOC(C)(C)C3)=O)CC1C)CC2 55840,N1(C(C(c2ccnn2C)C)=O)CC(NC(=O)Cc2cnoc2)CC12CCCOC2 55841,C12(OC)CCC(CO)(C1)N(C(=O)C(c1cccc(Cl)c1)N)C2 55842,N(C(=NCC(C)(CC)C(C)O)NCC1(NC(=O)OC(C)(C)C)CCC1)OC 55843,c1(NC(C(=O)NCC(CNC(C2CC(C)(C(=O)OC)C2)=O)C)=O)cccc(F)c1 55844,S(=O)(=O)(c1ccc(F)cc1Cl)NC(c1ccc(S(C)(=O)=O)cc1)C 55845,N1(C(CN(C(=O)C=C(C)C(C)C)CC#C)=O)CCC(C(C)(C)C)(CC)C1 55846,C1(CC(=O)N(CCOCCCN(C(CCOCCOC)=O)C)C)CCCC12CC2 55847,c1(C(C)=O)c(Cl)nc[nH]c1=NCCCNC(=O)C=C(C)C1CCCCC1 55848,C1(CC)C(C(=O)NC(CCN(C)C(c2cc[nH]n2)=O)C(C)C)CCN1C 55849,Cc1ccn(C(C)CC(=O)NCC2(C)CC(NC(c3cc(F)cs3)=O)C2)n1 55850,N1(C(C(C2CCN(C(=O)CC3CCCC3)C2)C)=O)CC(C)NC(=O)C12CC2 55851,C#CCC(O)C(=O)N1CC(C(=O)NCCc2ncn(C)n2)(CC)C1 55852,C1(CNC(C2C(C(C)NC(Cc3c(C)n[nH]c3)=O)C2)=O)CC2(CCC2O)C1 55853,c1(C(=O)NC2CC2C(N2CCn3ccnc3C2)=O)ccc([N+](=O)[O-])cc1I 55854,CCCC(C(=O)NCC(C)(C)CNC(c1cc(Br)cc(N)c1C)=O)C(C)C 55855,CC1=C(CNC(=O)C(C)(C2CCC2)NC(c2cnc(C)cc2C)=O)COCC1 55856,c1(C(=O)NC(C2CCOC2)CNC(C(C)=C2CCC2)=O)cc(F)cc(Cl)c1O 55857,C(c1cc(C)cc(C)c1)=CC(N1CC(C)(NC(c2cccc(OC)c2F)=O)C1)=O 55858,N1(C(C2N(C(C(CC)OC)=O)CC=C2)=O)CCCCC1COC.C1CCC1 55859,CCCCC(CN(C)C(C1CC12CC(NC(=O)C(C)CCOC)C2)=O)CC 55860,c1(-c2n(C)c(N3CC(O)CC34CCC4)nn2)ccc2ccccc2c1Br 55861,C1(NC(C2CC3CCC2O3)=O)C=CCN(C(=O)CCc2ccco2)C1 55862,CC1(C)CC(CNC(C2CC3CC2C3)=O)CN1C(C1CC1F)=O 55863,c1(CCC(=O)NC(CNC(CCOCC(C)C)=O)(C)C)cc(Cl)no1 55864,N1(C(C(C2CCN(C(CC=C(C)C)=O)C2)(C)C)=O)CCCC(C)(CO)C1 55865,c1(NC(=O)NCc2cc(Cl)c(Cl)s2)ccc(-c2cnn(CC(O)CO)c2)cn1 55866,CC(CC(C)(C)C)C(=O)N1CCOC(C)C1C(=O)NCc1noc(C(C)C)n1 55867,c1(CN2CC(NC(C(CCC)(C)C)=O)C2)cnc2ncccn12 55868,c1(CNC2C=CC(C(N=c3nc(C)[nH]s3)=O)C2)ccc2c(c1)CCCCN2 55869,N1(C(C(=O)NCC)=O)CC2CC1CCC2NC(c1ccc(OC(C)C)nn1)=O 55870,Cc1cc(NC(c2nnnn2C2CCCC2)CC2CCCC2)c(F)cc1Cl 55871,C(=O)(CCCCC(=O)N(CCC(=O)NC(C)CC1CC(C)C1)C(C)C)OC 55872,N1(CC(=O)N(C(CC)CNC(=O)CC2(CS(C)(=O)=O)CC2)C)CCCCCC1 55873,c1(OC(C)(C)C)ccc2c(c1)C(NC(c1oc3ccccc3c1Br)=O)CC2 55874,c1(CC(=O)N(CC(C)NC(=O)CC2CCN(C)C2=O)C)cccc2nsnc12 55875,C(=O)(CCc1ccsc1)NC(N)=O.C(=O)(CCN)NCCCOCCCN(C)C 55876,Cc1nc(C)c(C(N2CC(NC(c3ccnn3C(F)F)=O)C(C)(C)C2)=O)nc1C 55877,CC(C)C(CNC(=O)CCCC1CCCO1)NC(=O)CCC1(CO)CCCC1 55878,Cn1cc([N+](=O)[O-])c(OCC(N2CCCC2C(C)(C)C(=O)O)=O)n1 55879,c1(OC)ccccc1C=CC(N1CC2(CNC(c3cc(Cl)ns3)=O)CC1CO2)=O 55880,CCCCC(O)C(C)C(=O)NC(C)(C)CNC(C1CC1c1cnn(C)c1)=O 55881,c1(C(N(C2CN(C(Cn3ccc(C)c3)=O)CC23CC3)C)=O)ccn2cccc2c1 55882,C12(CNC(c3cc4n(n3)CCC4)=O)CCC(CC1)N(C(C1CCCC(CF)C1)=O)C2 55883,Cc1cccc(CC(=O)NC2CC2NC(=O)C(C)C2CCCC2)c1 55884,N1(C(Cc2n(C)nnc2)=O)CCC2(CCOC2)C(CNC(C2(CCO)CC2)=O)C1 55885,C(N=C(NCc1cnccn1)NC1CCN(C2CC2)CC1)C1(C)COC1 55886,C1(NC(CCC2(C)CN(C(c3ccc(NC)cc3)=O)C2)=O)CC2CCCC2C1 55887,N1(C(C=C(COC)C)=O)CC(OC)C(C(=O)NCCN2CCC(CO)C2)C1 55888,C1(NC(C(C)(C)c2cncnc2)=O)CC2CN(C(=O)CC3OCCO3)CC2C1 55889,C1(NC(c2ccc(O)cc2)=O)CN(C(C2CCC3(CCC3)OC2)=O)CC2(CC2)C1 55890,Cc1c(C(=O)NC2CCCC(NC(=O)C(F)=C3CCCC3)C2)sc2ccccc12 55891,c1(C(N(C(CC)CNC(=O)CCOCC2CC2)C)=O)cc(C2CCC2)[nH]n1 55892,N1(C(CC#C)=O)CC2CCCC2(NC(=O)Cc2cc(OC)cc(Cl)c2)C1 55893,O=C(C#CC1CC1)N1CCCC1c1cn(C2CCOC2)nn1 55894,C1(C(C(=O)NCC2CCCO2)N(c2ccc(Br)cc2)C)CCC2(CC1)CC2 55895,C1(NC(CNC(=O)OCC)=O)CN(C(=O)C(C2CCCCC2)F)C2(CCCC2)C1 55896,C(=O)(CCCCC#N)N1C(C(=O)NCC2(C)COCCO2)CC(F)C1 55897,N1(C(C(c2ccccc2)SC)=O)CC(NC(c2cc(C#N)oc2C)=O)CC(O)C1 55898,C1(C#N)(C(N(CC)CC2CCN(C(=O)CCS(N)(=O)=O)CC2)=O)CC2C=CC1C2 55899,C(CN=c1[nH]c(=NCc2ccc3c(c2)OCO3)[nH]c2c1COC2)n1c(=O)scc1 55900,c1(C(N(C2C3CN(C(C4ON=C(C)C4)=O)CC32)C)=O)ncc2c(F)cccn12 55901,C=CCCC(C(=O)OC)NC(c1csc(O)n1)CCN(CC(=O)OCC)C1CC1 55902,C1(NC(C2C(C)(C)C2)=O)CCCCCC1CC(N1CC(OC(=N)O)C1)=O 55903,C1(CNC(c2c(C)nsc2)=O)CCCC(NC(C2OCC2(C)C)=O)C1 55904,C1(NC(c2ccc(COC)o2)=O)CC2CCC1N(C(=O)C(C)n1cnnn1)C2 55905,C1(C(=O)NC2(C#C)CCOC2)CCC2(CC2)N1C(C1CN2CCN1CC2)=O 55906,c1(OC)ccc(CCC(N2CC=CC2CNC(C2CCCO2)=O)=O)cn1 55907,N1(C(C2CC3CCN(CN)CC23)CC)CC(CC2CCCCO2)CC(C)(C)C1 55908,Cc1cccc(Br)c1C(=O)NC1CCC1C(=O)NC1(C)CC(C)OC1=O 55909,C=CC(C)(O)C(=O)NC(C1(CNC(c2csc(-c3cocn3)n2)=O)CC1)C 55910,CN1CCOc2c(C(N3CC(NC(=O)C(O)C(F)(F)F)C3)=O)cccc21 55911,c1(C(=O)NCC(C2CCC2)NC(C2C(CC(C)C)C2)=O)nsnc1O 55912,C1(C(=O)OC)CN(C(=O)C2CC2)C1.C12(CCC1)C(=O)N2.C1(=O)CO1 55913,C(C)(C)(CCCCC(=O)NC1CCN(C(c2ccc(Cl)c(Cl)c2)=O)CC1)OC 55914,Cc1cnnc(O)c1C(N1CCC(O)(C(C)NC(=O)CC2CC3CC3C2)CC1)=O 55915,CC(CN=c1nc(N2CC3C(C)C3C2)c2c([nH]1)CCCCC2)Sc1nccs1 55916,C1(C(=O)NC(CNC(CC2(C(=C)F)CCC2)=O)CC(C)C)CC(C)(C)CN1C 55917,c1(C(N2CC3C(CN(C(C(C=C)O)=O)C)C3C2)=O)cc(C)cc(C)c1 55918,CCCCC(C)(C)OC(=O)C(Cc1ccc(C)cc1)C1CC1 55919,CC1CC=C(C(=O)NCC2CCC2NC(=O)CSc2nnnn2C2CC2)CC1 55920,Cc1ccc2c(CC(N3CCN(C(C45CC(C)(C4)C5)=O)CC3)=O)c[nH]c2c1 55921,c1(CNC(C)Cc2ccnn2C)ccoc1C(=O)NCC1CCCO1 55922,C(C1=C(C(=O)O)CC(O)C(O)C1)N1CCC(NC(=O)C(F)(F)F)CC(C)(C)C1 55923,N1(C(C(C(=O)OCC)(C)C)=O)Cc2occ(C(=O)N(CCCN(C)CC)C)c2C1 55924,N1(C(CC2C(C)CCC2)=O)CCC2(CC(NC(=O)C=Cc3cncs3)C2)C1 55925,CC1CN(C(=O)COC2CC(NC(C3CCCC(=O)N3C)=O)C2)CC(=O)N1 55926,C(=O)(C(C)(C)CCCCC)NC1CN(C(CC2(C(=C)F)CCC2)=O)CC(C)C1 55927,C1(NC(c2cc(CSC)on2)=O)CC2CC1N(C(=O)C(C)(C)COCC(F)F)C2 55928,N1(C(C2(CO)CCN(C(c3cc(C)ncc3C)=O)C2)=O)CCCC12CCCOC2 55929,N1(C(c2nccn2-c2ccccc2F)=O)CCC(O)(C(F)(F)F)C(O)C1 55930,CC1(C)CN(C(=O)CC2(C(F)(F)F)CC2)CCC1NC(c1cc2ccsc2s1)=O 55931,C(=O)(CCCCCC#N)NC(C(=O)NC(C#C)CC(C)(C)C)(C)C1CCC1 55932,Cc1cc2nc(C(=O)N(C3CC3)C(c3cccc(Cl)c3)C)ccc2c(=O)n1C 55933,C=CCCCCC(=O)N1CCN(C)CC1C(=O)NCc1c(F)cccc1F 55934,Cc1cc2c(cc1C)OC(C(N1CCN(C(=O)CC3(CO)CC3)C(CF)C1)=O)C2 55935,C(=O)(C(C)C(=O)NCc1cc(C(=O)NC(c2cnn(C(C)C)c2)C)n(C)n1)OC 55936,c1(C(N(CCCOCCNC(C(CSC)C)=O)C)=O)ccc2c(c1)COCCN2 55937,CC1CCC(C(N2CCC(CN(C(=O)C(C)(F)F)C3CC3)CC2)=O)CC1C 55938,N1(C(C2(NC(C3C(C)C3)=O)CCCCC2)=O)C2CCC1CN(C)C2 55939,N1(C(CC2(OC)CN(C(c3cnc(Cl)n3C)=O)C2)=O)CCC(C)(C2CC2)C1 55940,Cc1nc2ccccn2c1C(=O)O.c1(C(N2CC(N(C)CCO)C2)=O)ccccc1C#N 55941,c1(OC)cc(CC(N2CC3C(C2)N3CC)=O)ccc1Br.c12ccc(cn1)c(=O)[nH]2 55942,c1(CC)[nH]nc(C(N2CCCC2C2CCN(C(c3cn(C)cn3)=O)C2)=O)c1Br 55943,CN1N=CC(CC(=O)NC2CC(NC(=O)C(C3CCCCCC3)O)C(O)C2)C1=O 55944,S(=O)(=O)(CC(=O)N(CCCNC(=O)Cc1cnn(CCO)c1)CC)NCC 55945,Cc1ccc(C(F)F)cc1C(N1CCC1CNC(c1cccc(C#N)c1)=O)=O 55946,C12(C(=O)NCC(=C)CCNC(c3[nH]nnc3C(F)F)=O)CCC(C(C)=O)(CC1)C2 55947,c1(OC)cccc2c(N3CCCC(CC(C)C)C3)ncnc12 55948,c1(C(=O)NC(c2cnc(C(C)C)[nH]2)C)ccc(C(F)F)cc1 55949,C=C1CCC(C(c2nnnn2C2(C)CC2)NCC2CC(Br)=NO2)CC1 55950,C(C(O)CC(=O)NC1CN(C(=O)C(C)(C)N2CCCCC2)CC1F)N(C)C 55951,C(=O)(CCS(N)(=O)=O)N1CCC(NC(c2occ(C(C)=O)c2)=O)C1C(C)(C)C 55952,C(=O)(CCCC(C)(C)NC(=O)C(C#N)C(C)(C)C)NCC1CN(CC)C(=O)O1 55953,Cc1ccc(C)c(C(N2CC(CCNC(C3CC(C(C)C)=NO3)=O)C2)=O)c1 55954,c1(Nc2ccc(-c3n(C)ncc3)cc2F)ncnc2c1ccn2C 55955,CC1(C)COC1C(N1CCCC1C(=O)NCc1cc[nH]c1-c1ccccc1)=O 55956,Cc1scc(C(=O)NCCCOCCC(=O)NCC2CC3CC3C2)c1C 55957,N1(C(c2cccc(CC)c2)=O)CCC2CCN(C(C3CC3CC(C)(C)C)=O)C2C1 55958,C1(CNC(CC(CC)(C)C)=O)CC2CCC(C1)N2C(C1(COC)CCCCC1)=O 55959,c1(CCC(=O)NC(C)CNC(=O)CC2CCC(=O)O2)ccc(C(N)=O)cc1 55960,N(C1CCCc2sccc21)C(C(c1ccc(C(=O)OC)cc1)N)=O 55961,CC1CCN(C(C2C3COCC23)=O)CCN1C(c1ccc(C(F)(F)F)cn1)=O 55962,C(=O)(C1=NOC(C)(C)C1)N(CC)CC1CCCN(C(C2CSC2)=O)C1 55963,c1(NCCC(C)(C)CC(F)(F)F)nnc(S(=O)(=O)N2CCCCCC2)c(Br)c1 55964,C1(C=O)CN(N2CC(C)(CC#N)C2)CC1S(=O)(=O)c1cccc(Br)c1.CCOC 55965,c1(CC)cc(C(=O)NC2(C)CN(C(=O)CCNC(N)=O)C2)cc(C)c1 55966,C1(C(=O)NC(C=CC(=O)NC(CCOC)(C)C)(C)C)CCCC(C)(C)C1 55967,c1(NC(CCC=C(C)C)c2nnnn2C2(C)CC2)cc(C(F)F)cc(C(C)C)c1 55968,C1(CC=C)(NC(=O)Cc2cccc(C)c2C)CCN(C(=O)CSS(C)(=O)=O)CC1 55969,c1(C(N(C)CC2CCN(C(=O)C(O)C3CC3)CC2)=O)[nH]cc2c(=O)n(C)ccc12 55970,N1(C(C(CC(C)C)(C)O)=O)CC2(C=C(C(=O)NCC3CCSC3)CO2)C1 55971,CC(C)(CCC#N)C(=O)N1CCN(C(c2sc(C(F)(F)F)cc2Br)=O)CC1 55972,C#CC(C)(C)C(=O)NCC1CC(COC)CN1C(c1ccc(C2CC2)cc1)=O 55973,C1(NC(C(C)CC2CCCC2)=O)CC12CCN(C(=O)CC1CCCN1C)C2 55974,C1(NC(C(c2cc(C)oc2C)C)=O)CCCCN(C(=O)C(F)(F)c2nccs2)C1 55975,C1(NC(c2c(CC(C)C)onc2)=O)(CO)CCN(C(C2(C)C=CCC2)=O)CC1 55976,C1(NC(C2CC(C)(CC)C2)=O)(CO)CCCN(C(=O)C(C)(C)c2ccccn2)C1 55977,c1(C(CNC(C2N(C)CC(O)C2)=O)NC(C2CC23CCC3)=O)ccc(F)cc1F 55978,C(=O)(C(F)(F)CC(C)C)N(C(C)CNC(=O)COc1c(F)cccc1Cl)CC 55979,c1(C(=O)N(C2CCC(=O)N2)C(CC)CNC(c2cc(C)cs2)=O)cc(N)c(Cl)c(O)c1 55980,C1(C(=O)OC)CCCCC1C(N1CCCC1CNC(C)=O)=O.C1(=O)C(C(C)C)N1 55981,C1(NC(=O)Cn2nc(O)ccc2=O)CC1C1CCCN(C(=O)CCOC2CC2)C1 55982,C1(CC(=O)N(CC(CC)NC(c2cnc(C(C)C)o2)=O)C)CC(C)(C)OC(C)(C)C1 55983,N1(C(C(C)=C(CC)C)=O)CCCCC1CN(C(=O)CCc1cnn(C)n1)C 55984,N1(C(CCCSC)=O)CC(CNC(C23CSCC2C3)=O)C2(CCC2)C1 55985,C(=O)(C1=NNC(=O)CC1)NCC(CNC(c1n[nH]cc1Br)=O)O 55986,C(=O)(C1CC(=O)c2ccccc21)NC1CN(C(COCc2cc(C)no2)=O)C1 55987,c1(CNC(=O)OC(C)(C)C)ccc(CNCC2CC(C(F)(F)F)CO2)cc1 55988,C1(C(N(CCN(C(C)C)C)C(C)C)=O)CC1C(F)(F)F 55989,O=C(C(O)CC(F)(F)F)NC1CCN(C(=O)C=Cc2cccc(O)c2)C1 55990,Cc1nnc2n1CC(C(=O)OC1CCC1)CC2 55991,O=C(N=S1(=O)CCN2CCCCC2C1)c1cc([N+](=O)[O-])nn1-c1ccc(Cl)nn1 55992,c1(C(N2CC3C(CNC(COCCCC)=O)(C3)C2)=O)nccc(Cl)c1C 55993,C(=O)(CCCC1CC1C)N(CCOCCCNC(CC1(CC)CC1)=O)C 55994,N1(C(C2CNC2=O)=O)CCC(CO)C12CC2.c1(COCC)ccn(C(C)(C)C)c1 55995,N1(C(CC2CC(OC)C2)=O)CCOCC1CNC(c1ccsc1Cl)=O 55996,C(CC)(C(=O)N1CCC(c2ncco2)C1)N(C(CSCCC)=O)C 55997,c1(OC)noc(C(N2CC=CC2CNC(C2CC(C(F)F)C2)=O)=O)c1Br 55998,c1(C(N(CC(C)NC(=O)Cc2cnc[nH]2)C)=O)cc([N+](=O)[O-])n[nH]1 55999,C1(C(=O)NC2(CC=C)CCC2)CCN(C(=O)c2cccc(C3CC3)c2)O1 56000,C(CC(=O)NCc1ncnn1C1CC1)(C(C)OC)NC(C1(CSC)CC1)=O 56001,C1(CNC(C2CC23CCOCC3)=O)CC(C(C)C)CCN1C(C1(SCC)CC1)=O 56002,c1(CNC(C(N2C(C)CSCCC2)=O)=O)c(Br)ccc(Cl)c1F 56003,CC(CC(C)(C)C)C(=O)N1CC2CC(C1)N(C(=O)CNc1ncccn1)C2 56004,C(=O)(C(C)CN1CCOCC1)NC(C1CCN1C(c1noc(C(C)(C)C)n1)=O)C 56005,Cc1c(C(=O)N(c2nccc(Cl)n2)C)cccc1C(F)(F)F 56006,C1(NC(C2CC3(CCC3OCC3CC3)C2)=O)CCN(C(C2CCC(=O)O2)=O)C12CC2 56007,C1(NC(C(CCC)OC)=O)CN(C(C2(C)CCC(=O)N2)=O)CC2(CC2)C1 56008,CC1C(C(=O)NCC(CO)C(=O)NC2CCCC2C#N)CCN1C 56009,c1(C(C)C)cc(COC(C)(C)C)cc(Br)c1.N12CCC(C1)NC2=O 56010,C(=O)(CC=C(Cl)Cl)N(CCN(C(C1C(C(=O)OCC)(C(C)C)C1)=O)C)C1CC1 56011,N1(C(CCOCC#C)=O)CC(CNC(c2cnn(C3CC3)c2Cl)=O)CC1C 56012,n1(CC)cc(CN(C(=O)CNC(=O)CN(C(=O)C(C)CO)C)C)nn1 56013,CC1CC(CCNC(c2cc(Cl)no2)=O)CCN1C(=O)Cc1ccc(F)nc1 56014,N1(C(c2ccc(CC)[nH]2)=O)CC(NC(C2CC(OC(F)F)C2)=O)CC1C 56015,N1(C(CC(C)CF)=O)C2CCC1CC(NC(=O)CN1CSCCSC1)C2 56016,CCS(=O)CC(=O)NC1CC(CNC(C2(CC)CCC(=O)N2)=O)C1 56017,C(=O)(C(C)(C)CNC(C1CCC(O)C1)=O)NCCC1C(C(=O)OC)C1 56018,C1(C(=O)NC2CCN(C(C(CC)c3ccccc3CC)=O)CC2)CCCC(C)(C)O1 56019,c1(C(=O)NC(CC2CCCC2)CO)cnc(-c2ccccc2Cl)nc1 56020,CC1CCCc2cc(C(=O)NCCN3CCS(=N)(=O)CC3)nn21 56021,CC1CC(C(=O)N(C(=O)CCCC(F)c2ccccc2)C2CC2)CCN1C 56022,C=C(C)CC(C)C(=O)NCC(CC)NC(=O)C(C)(C)C(F)F 56023,N(C(=NCCc1ccccc1F)NC(C)(C)C)OC.C1(C)CCCC1 56024,C(c1cncnc1O)=CC(=O)NCC1CN(C(CCNC(C)=O)=O)C1 56025,CC1CN(C(C2CCC3(CC2)CC3)=O)CCC1NC(c1cnc(C2(C)CC2)s1)=O 56026,Cc1cc(N)c(C(N2CCC(O)(C(C)CNC(c3ccco3)=O)C2)=O)c(F)c1 56027,C1(C(N2CCC(C)(NC(=O)CC3COC(=O)C3)C2)=O)C2Cc3ccccc3C12 56028,C(=O)(CC(C)CC(=O)NC1CN(C(c2cc(C3CC3)no2)=O)C2(CCC2)C1)OC 56029,c1(C(=O)NC2CCC(NC(c3c(CC)ncs3)=O)C2)ccc(OC)nc1Cl 56030,Cc1cncc(C(N2CCCC(O)(CCNC(=O)C(C)CC(N)=O)C2)=O)c1C 56031,c1(OC)c(C(N2CC(NC(c3onc(C)c3C)=O)CC(O)C2)=O)cccc1Br 56032,c1(C(N(C(CNC(C2(c3cc[nH]n3)CC2)=O)C2CC2)C)=O)cscc1C1CC1 56033,C=CCCCCCCCC(C(=O)NCC=C)N1CC2CCCN2C(=O)C1C 56034,CC(CCC(=O)NCC(F)Br)N(C)C.C1(C)C(=O)N1 56035,CC(C)CCCCC(=O)NC1C=CCN(C(c2ccn(C(C)(C)C)c2)=O)C1 56036,NS(=O)(=O)c1cccc(C(=O)NC2C3CC2CN(C(c2ccc(CO)o2)=O)C3)c1 56037,N1(C(c2cnc(OC)nc2)=O)C(C(=O)Nc2cnc(Cl)nc2C)CCC1C 56038,CCC(CO)(C(=O)N(C)CCN(C)C(c1c(C)ccnc1O)=O)OC 56039,C1(C(N2CC(C)(OC)C(F)(F)C2)=O)CNCCC12CCOCC2 56040,C1(O)(CNC(C=CC)=O)CCN(C(c2cn(C)nc2-c2ccccc2F)=O)C1 56041,N1(C(C)=O)CC(NC(c2ccc(C(C)(C)C)s2)C2CCC2)C2CC2C1 56042,Cn1ccc2cc(C(N3CCCC(NC(=O)CSC(F)(F)F)C(F)C3)=O)cnc12 56043,N1(C(CC#C)=O)CC2COCC2(C(N2CCCC2C(C)(C)O)=O)C1 56044,c1(COC)ncc(C(=O)NCC2CC(CNC(c3cnn(C(F)F)c3)=O)CO2)s1 56045,N1(C(C2ON=C(C)C2)=O)CC(O)(C2CCN(C(c3cc4c(s3)CCC4)=O)CC2)C1 56046,Cc1cccc(-c2nc(C3OCCC3C)n(CC3CCSC3)n2)c1 56047,c1(N(C)CC)nnc(C(C)OC)n1CCO.c1(OCC)ccccc1 56048,CCCCN=C(NCc1ccc2c(c1)OCO2)NCC1CCCCC1 56049,N1(C(C(c2cccnc2)C(N2CC(C(F)(F)F)C2)=O)=O)Cc2cccc(O)c2C1 56050,N1(C(c2cc(=N)[nH]cc2)=O)CCC2CCN(C(=O)CSCCC(F)(F)F)CC12 56051,CC(C)CC(C(=O)N1CCC(O)(CO)CC1)NC(=O)C(c1ccccc1)F 56052,C1(CNC(C(C)CN(C)C)=O)CC2(CCN(C(c3ncccc3N)=O)CC2)CO1 56053,C1(n2cc(CNC)nn2)CCCN(C(C2(C3CCS(=O)(=O)C3)CCC2)=O)C1 56054,C(C(=O)NC(CNOC)CO)(C(C)C)(C(C)C)NC(C1CC(C)C1)=O 56055,Cc1ccccc1COCC(N1CC(NC(C2CC3(CC3)CO2)=O)C(O)C1)=O 56056,CCC(C)(CO)CN=c1cc[nH]cc1S(=O)(=O)N(C)C(C1(NC(N)=O)CCCC1)=O 56057,C1(NC(C(c2c(C)cc(C)cc2C)N(C)C)=O)CCC2C3CCC(C3)C12 56058,CC(C)CCC(F)C(=O)N1CCC(O)(CCNC(C2CCCCCC2)=O)CC1 56059,c1(OC)cc(NC(c2nnnn2C(C)C)C2(OCC3CC3)CC2)cc(O)c1 56060,c1(C(=O)NC2CCCC(NC(C3(CC)CC3)=O)C2)ccc(Cl)c(N2CCCC2)n1 56061,c1(OC)ccc(F)cc1CCC(N1CC2CN(C(c3cc(O)ncn3)=O)C2C1)=O 56062,C1(C(=O)NC(CNC(C(=O)N(CC)CC)=O)CC)C(C2CC2)C1(F)F.c1nccs1 56063,C1(C(=O)Nc2ccc(COC)cc2)CCOCCN1C(c1cnn[nH]1)=O 56064,CC1CCCCN1C(c1ccnc(N2CCCC2c2ccccc2)n1)=O 56065,c1(C2C(C(=O)NC3CC(CNC(C=C(CCC)C)=O)OCC3)C2)cccc(C#N)c1 56066,N1(C(C(C=C)(C)C)=O)CCC(CO)C(NC(c2nnc(C)cc2O)=O)C1 56067,CC(C)CCC(O)C(=O)N1CCN(C)CC1C(=O)NCC12CC(CN1C)C2 56068,c1(C(N(CCOCCN(C(C2C(C=C)C2)=O)C)C)=O)cc(Cl)c(Cl)cc1O 56069,c1(OC)ccc(C2(NC(=O)NCc3ccnc(CC)n3)CC2)cc1OC.CSC 56070,c1(-c2nc(C)sc2)ccc(CN2CCCC2CC(N2CCC(CO)CC2)=O)cc1 56071,N1(C(Cc2c(C)scc2)=O)CCN(C(=O)CS(=O)(=O)C2CC2)C2COCC12 56072,c1(C(=O)OC2C(C(=O)OC)(CC)C2(C)C)cc(C(C)C)n2nccc2n1 56073,C1(C(N(CCCNC(C2(OC)CCC2)=O)C(C)C)=O)OCC2COCCC12 56074,C1(NC(C(C(C)C)OCC(C)C)=O)CN(C(C2(C)CCN(C)CC2)=O)C(C)(C)C1 56075,c1(OC)cc(CC(=O)NC2CCC(CNC(=O)CC3(CO)CC3)C2)ccc1C 56076,c1(CC)nc(C)c(C(=O)NC(C(=O)NOCC2CC3C=CC2C3)C2CC2)o1 56077,N1(C(CCCC#C)=O)CCC(NC(C2CCCN(C(C)=O)C2)=O)C1(C)C 56078,CCC(C)(C)C(C(=O)NC1(CNC(c2csc(C#N)c2)=O)CCOCC1)OC 56079,C1(CNC(CC(C)N2CCCC2=O)=O)CCN(C(C2CCC(=O)N2)=O)C(C)C1 56080,c1(C(N2CCC(C(=O)O)C2)=O)ccc(F)c(S(=O)(=O)N2CCN(C3CC3)CC2)c1 56081,C1(C(=O)NCC(c2ccccc2)C)CCc2ccncc2C1 56082,N1(C(C2CC=C(C)CC2)=O)CC2(CCC(NC(c3ocnc3C)=O)C2)C1 56083,C12(NC(c3ccoc3)=O)CC1CN(C(c1ccccc1-n1cnnn1)=O)C2 56084,N1(C(C(N2CCCC(CC(F)(F)F)C2)=O)=O)CC2(C1)OCC1CC21 56085,Cc1cc(C)cc(C=CC(N2CCCC2CN(C(=O)CCSCC(N)=O)C)=O)c1 56086,N(C1CCNC(=O)c2[nH]ccc21)C(C1CCC(C(=O)OC)CC1)=O 56087,c1(OC)ccc(OCC(=O)NC(C)C(C)(C)NC(C23CCCC2(CO)C3)=O)cc1 56088,C1(C(N2CCN(Cc3cc(C4CCCCC4)no3)CC2)=O)CC2(CSC2)C1 56089,c1(C(N(C2CCN(C(C(COC)C)=O)C2)C)=O)c[nH]c(=N)c(C)c1 56090,C1(C(=O)NC2(CC)CC2)C2CC1N(C(c1ccc(CO)s1)=O)C2 56091,C12(NC(c3cc(C)sc3)=O)CCCC1CN(C(c1n[nH]c(C)n1)=O)C2 56092,C1(C(N2C(CCN(C(=O)Cn3cc[n+](C)c3)C)CCCC2)=O)C(F)(F)C12CCC2 56093,C1(CC=C)(C(=O)NCc2ncccn2)CCN(C(c2cccc(C)n2)=O)C1 56094,CCC(CC(=O)NCC1C2CN(C(=O)CC3CC4(CCO3)CC4)CC12)C(C)C 56095,c1(C(=O)NCC23CC(CO2)N(C(=O)CC=C(Cl)Cl)C3)c(F)ccc(Cl)c1F 56096,C1(NC(c2cc3c(s2)CCCC3)=O)CC(C2CCN(C(C3CCCC3F)=O)C2)C1 56097,C1(N(C(C(=O)NCC2CCC2)c2cnc[nH]2)C2CCC2)CCC(F)(F)CC1 56098,C(C)(C)(CN=c1[nH]nc(C#N)s1)NC(C(C)Oc1cccc(C)c1)=O 56099,C12(NC(=O)CSCC3CC3)CCCC1(C(F)(F)F)C2 56100,Cn1cc(C(=O)C(=O)NCC(=O)NCC(N2CCC(CO)C2)=O)cn1 56101,c1(C(CNC(=O)C(CSCCN(C)CC)NC(=O)COC)OCC)ccccc1F 56102,CC1CC(N(C(=O)C(C)(C)CN(C)C(C2CCCC(C)C2)=O)C)CC(C)O1 56103,N1(C(C2(c3cccc(OCF)c3)CCC2)=O)CC(NCC2CCOC2)CC(O)C1 56104,N1(C(CCC=C)=O)CC2NCC2(C)C1 56105,C(=O)(C(C)CC(C)C(C)=O)NC1C(C(=O)NCC2(CC(=O)OC)CC2)CC=CC1 56106,CCCC(CC)C(=O)NCCCNC(=O)C(O)Cc1c(F)cccc1Cl 56107,C(CN=c1[nH]c(=NCC2CCC3(CC3)C2)[nH]c2c1CCCC2)c1occc1 56108,c1(OC(C)C)cc(NC(C2CCC(C)(C)CO2)=O)cc(C#N)c1 56109,c1(C(N2CC(c3cccc(Cl)c3Cl)(O)C2)=O)cc(Cl)c([N+](=O)[O-])s1 56110,n1(CC2C(CC)CCO2)c(NN2CCCC2)nnc1-c1nnc(C(=O)N(C)C)s1 56111,N1(C(c2cc(C)n(C)c2)=O)CC(NC(C2CC3(CCCO3)C2)=O)CCC(O)C1 56112,c1(OC)ccc(CNC2C(Cc3ccc(Cl)c(Cl)c3)N2)c(OC)c1.C1CC1.OC 56113,c1(C(N2CC(C(=O)Nc3nccs3)C2)=O)cc(Cl)cc(Cl)c1O 56114,C=CCC(C)(C)CC(=O)N1CCC(NC(c2cc(C(C)C)no2)=O)C1 56115,CC(C)CCCCCC(=O)NCC1=CCN(C(C2(c3cccs3)CC2)=O)CC1 56116,C1(C#CC(=O)NCC(F)CNC(=O)C(C)Cc2ccc(O)cc2)(CC)CC1 56117,N1(C(c2c(C)nc(O)s2)=O)CCN(C(=O)CCc2cn(C)nn2)CC(C)C1 56118,N1(C(COCC=C)=O)CC(NC(c2cnc(OC(F)(F)F)cn2)=O)CC2(CC2)C1 56119,c1(C(=O)Nc2ccc(F)c(F)c2F)n[nH]c2c1CN(Cc1cnc(C3CC3)s1)CC2 56120,C1(C(NOC(C)C)=O)CCC(NC(=O)COCCF)CC1 56121,Cc1cncc(C(=O)NCCC(C)CCNC(=O)C(F)CC2CCCCC2)c1 56122,CC1=C(Br)CN(C(=O)C(=O)N(C)Cc2cccnc2)CC1 56123,c1(CC(=O)NC2CCC(n3cc(C(C)NC)nn3)CC2)cccc(C)c1Cl 56124,c1(OC)cc(Cl)c(C(N2CCCC(C(=O)NC(C)CC#N)CC2)=O)cc1OC 56125,c1(C(N2CC(C(C)NC(c3c(Cl)cc(C)s3)=O)OCC2)=O)ccc(F)c(CO)c1 56126,c1(SC)cc(C(=O)NCC2(C(N)=O)CN(C(=O)CC3CCCC34CC4)C2)c(C)o1 56127,c1(C(N2C(C(N3CCC(C)(C#N)C3)=O)CC3CC32)=O)ccc2cc(O)ccc2n1 56128,C1(C(=O)NC2CCN(C(C)C)C2=O)CCC(C)(C)N(C(=O)CP(C)(C)=O)C1 56129,Cc1cc(C(=O)NC2(CNC(C3CC4(C3)CC4F)=O)CCOC2)c(F)cc1F 56130,CON1CCC(C(=O)NC(C2CCN(C(c3cc[nH]c3C)=O)C2)(C)C)CC1 56131,C(=O)(CS(=O)(=O)CC(=O)OC)NC1C(NC(CSC)=O)C1 56132,CC1CC(C(=O)NCC2(F)CN(C(c3cc(O)cc(O)n3)=O)C2)Cc2nn[nH]c21 56133,C1(CC)(NC(=O)C(CC)C2CC2)CCCN(C(=O)CCOc2cccc(C)c2)C1 56134,N1(C(c2cc(C)nc(O)n2)=O)CC2(CCCN(C(c3ccc(CF)cc3)=O)C2)C1 56135,C1(C)(NC(c2n[nH]c(C)c2F)=O)CCN(C(c2cccc(O)c2Cl)=O)CC1 56136,CC1CC(=O)NC1C(=O)NCCOC1CCN(C(c2nc[nH]c2C(F)(F)F)=O)C1 56137,C(C(C)(C)C#CC(=O)NCCC1(C)CCOCC1)NC(C(C=C)(F)F)=O 56138,Cc1cnc(C(N2CC(N(C(=O)C3=CCCCO3)C)C2)=O)cc1C 56139,C1(NC(C(C)OCCOC)=O)CCN(C(=O)CCF)CCC1CO 56140,c1(C(=O)NC(C2CCCCC2)C(C)NC(C2(O)CCSC2)=O)cc(Cl)ccn1 56141,N1(C(c2cc(C)nn2C)C(=O)N(CCCSCC)C2CC2)CCC2(C1)CC2(F)F 56142,N1(C(c2c(CC)[nH]cc2)=O)CCN(C(=O)C(C)(C)OC(C)C)CC1CO 56143,Cc1cncc(C)c1C(=O)NCC(C)NC(C1CCC(=O)N1CCC(F)(F)F)=O 56144,CC1CCC(C(N2CC(O)(CCNC(=O)C(F)=CCCF)C2)=O)CC1C 56145,C1(NC(CC(C)(C)c2cccs2)=O)CCN(c2ccc(C#N)nc2)CCC1CO 56146,C1(O)(C(=O)OC)CN(C(C2CC(F)(NC(=O)C(=O)Nc3ccccc3)C2)=O)C1 56147,C1(OC)CCC(C(N2CC(N(C)C(c3cnn(C(C)C)c3F)=O)C(O)C2)=O)CC1 56148,c1(OC)cc(CN(CCCNC(c2csc([N+](=O)[O-])c2)=O)C2CC2)c(OC)cc1C 56149,CCC(C)(CO)C(=O)N1CC2(CCN2C)C1 56150,CCCCCC(F)C(=O)NC1CC=C(C(=O)N2CCC(O)CC2C2CC2)C1 56151,C1(NC(CCCC=C)=O)C(C)CCN(C(=O)CCS(C)=O)C1C 56152,C1(CNC(CC(C)c2ccsc2)=O)CCCCN(CC2CC2)C1.C(C1CCOCC1)=C 56153,CC1CN(C(=O)CC2(O)CCCCC2)CC1(C)CNC(=O)C(CCO)N(C)C 56154,C(CC(C)C(=O)N(C(C)C(=O)NC1CC(C)(C)C1)C1CC1)=CC 56155,CC(O)CC(C)(C)CNC(C1CN(C(c2ccc(N)c(F)n2)=O)CC1(F)F)=O 56156,c1(C(N(CC(CC)NC(c2coc(Cl)c2)=O)C)=O)ncc2[nH]ncc2n1 56157,Cc1ncccc1CCCNC(=O)N(C(=O)Oc1ccccc1)CC1CC1(Cl)Cl 56158,C(C(=O)NC1CCCCN(C(c2ccc(O)c(Cl)n2)=O)C1)(C(C)(C)C)N(C)C 56159,N1(C(C(C)N(C(C)=O)C)=O)CCC(C(=O)NC2CCC(O)C2)C(C)C1 56160,C=CC1(C(N2CCCC(CO)(NC(=O)CCN3CCC(F)C3)C2)=O)CCCCC1 56161,c1(C(=O)NCC2N(C(C(CC#C)C)=O)CCC(C)C2)ccc2nc[nH]c2c1F 56162,C(=O)(C(CC)CC(F)(F)F)N1CCC(CNC(c2cc(CCC)on2)=O)C12CC2 56163,c1(C(N(C2CCN(C(c3c(CCC)nns3)=O)CC2)CC)=O)cc(C)ccc1F 56164,c1(N2CCC(NC(C3N(CC)C(=O)CC3)=O)C(F)C2)ncc(C#N)cc1Br 56165,C(=O)(C1=C(C#N)CCC1)NC1CC(CCN(C)C(c2ccc(C(=O)OC)o2)=O)C1 56166,c1(CC(=O)NCCC(=C)CNC(=O)C(F)(F)CC2CC2)cccc(C(F)(F)F)c1 56167,N1(C(c2cc(C)oc2)=O)CCN(C(c2ncc3[nH]ncc3n2)=O)CC2(CC2)C1 56168,CC1CC(C(N2CCC(N3CC=CC3)C2)=O)CCN1C(=O)CC1CCCC1 56169,c1(CCC(=O)NC(C)CNC(C2CC3(F)CC2C3)=O)ccc2c(c1)CCO2 56170,C1(C)(C(=O)NCC(CC)N(C(c2ccc(SCC)nc2)=O)CC)CC2C=CC1C2 56171,Cc1ccnc(CNC(=O)CC2CN(C(C3(CF)CC3)=O)CC2C)n1 56172,C=CC(C)(C)C(=O)N1CCC(CCCCCNC(=O)Cc2cc(C)n(C)n2)CC1 56173,c1(C(CO)NC(C(=O)OCc2ccccc2)C2CC2)cccnc1Br 56174,C1(NC(CCCNC(=O)OC)=O)CCCCN(C(=O)C(C)OCCN(C)C)C1 56175,C1(F)(C(N(C(CO)C2CC2)C)=O)CN(C(c2ccsc2)=O)C1 56176,N1(C(CN(C(=O)COCC(C)(C)C)CCOC)=O)CCC(CO)(CO)C1 56177,c1(C(N2CCC(F)(CF)C2)C(=O)NCCCSC)cccc2c1OC(C)(C)O2 56178,Cc1csc2ncnc(NCC3CCCCN(C(C4CCC45CCC5)=O)C3)c12 56179,C(=O)(C(C)CC(C)(C)C)NCC(CC)NC(=O)CSC(F)F 56180,c1(C(N2CCCC(N(CC#C)C(c3nc(C)c(C)[nH]3)=O)C2)=O)nc(C)ccc1F 56181,C(=O)(C(F)CC(C)C)NCc1cccc(NC(C=CC(CC)=CC)=O)c1 56182,C1(C)(N(C)CC)CCN(C(C2(C(C)NC(=O)CC3CC(C)(C)C3)CC2)=O)C1 56183,c1(C(=O)NC(CNC(c2cc(C(=O)OCC)ncc2)=O)CO)ccc(=O)n(C)n1 56184,N1(C(CSCC=C)=O)CC2(CCCC(CNC(c3nn(C)cc3SC)=O)O2)C1 56185,C(N=c1[nH]c(=NCC(=O)N2CCCO2)c2c(F)cccc2[nH]1)c1scc(CC)n1 56186,Cc1ccc(Cl)cc1NC(C1(NC(C2CCCN2c2ccc(F)cc2)=O)CC1)=O 56187,N(C(=NCc1ncc[nH]1)NC1CC(OCC2CCOCC2)C1)C(CC)C 56188,C=C(CNC(=O)CCC1CC1(C)C)CCNC(C1CCN1C(c1ccsc1)=O)=O 56189,C=C(C)C(C)(C)C(=O)NC1CCC(C)(CNC(=O)CNC(C)=O)CC1 56190,C(c1ccccc1F)=CC(=O)N(C(C)CCNC(C1(CF)CCOCC1)=O)C 56191,c1(OC)cc(C(=O)NC2CCCC2NC(=O)CCN(C)CCO)cc2c1OCCO2 56192,c1(C(N(CCNC(=O)CC(O)CC(C)(C)C)CC)=O)cc2cc(Cl)c(Cl)cc2[nH]1 56193,C1(NC(CC2(OC)CCCC2)=O)CCN(C(=O)CC(C)N(C)C)CC(O)C1 56194,C1(NC(C=C(C)c2ccsc2)=O)CN(C(=O)CCC2CC(F)(F)C2)CCC1O 56195,N1(CC(N2CCC(OCC=C)C2)=O)CCCC(NC(=O)Cc2ccon2)C1 56196,c1(C(=O)NCCN(C)C(c2ccc(OCC(F)F)nc2)=O)cc2sccc2s1 56197,c1(N(C(c2ccco2)=O)CC)ccccc1C 56198,C(=O)(CCCCCC(C)(C)C)N1C(CNC(=O)C=C(C)C2CC2)CC(COC)C1 56199,Cc1cnsc1C(=O)NC1(CNC(C2CCC(OC(F)(F)F)C2)=O)CCCC1 56200,N1(C(C)=O)CC(S(C)(=O)=O)C1.C1(CCC)C(=O)N1SCCCCC(=O)OCCCO 56201,C1(CC(=O)NC(C)CC(C)NC(=O)C2=CCC2)(Cc2ccccc2)CCCCC1 56202,N1(CCCNC(C2CCN(C(=O)NC)C2)=O)CCN(C(C2CCC(=O)C2)=O)CC1 56203,N1(C(c2cncc(C3CC3)c2)C(=O)NC(C(=O)OC)C)CCC(O)C2CCCCC12 56204,C1(CC)CN(C(C2CC(O)(C#N)C2)=O)CCC1NC(=O)C(C(C)C)NC(N)=O 56205,CCCC(C(=O)N(CCNC(=O)C(c1ccccc1)F)CCOCC)NC(N)=O 56206,c1(NC(=O)NC2CC2C(N2CC(F)C(F)C2)=O)cnnc(Cl)c1 56207,C1(N(C(Cc2nnc(C)n2C)=O)C)CC2CC1N(C(=O)C(C)NC(C1CCC1)=O)C2 56208,N1(C(C(C)Oc2ccc(C)cc2)=O)CC2CC1CC2CNC(=O)C#CC(C)C 56209,Cc1ccccc1N=c1[nH]c(N(C)C(C)C)nc(=NCCOCCOC)[nH]1 56210,c1(N(CC(N2CC(NC(CCCC(=C)C)=O)C2)=O)C)nc(C)c(C)c(C)c1C#N 56211,Cc1nc2sccn2c1C(=O)NCC(C)CN(C(=O)CC1CCC(F)(F)CC1)C 56212,CC1(C(=O)OCC(c2ccc(O)c(O)c2)O)CCCN(CCN2CCCCC2=O)C1 56213,c1(C(N(C2CCN(C(C3CCS(=O)(=O)N3)=O)C2)CC)=O)ccc(P(C)(C)=O)nc1 56214,c1(-c2cc(Cl)c(Br)cc2)nc(C2SCCc3ccccc32)no1 56215,c1(C(N(C2CCCN(C(=O)C(F)=CCCF)C2)CC)=O)cnc(CC2CC2)nc1O 56216,CCN=c1ccc(C(=O)NCCCNC(=O)CSc2nncs2)c[nH]1 56217,c1(CC)nccn1CC(=O)NCCN(C(C1CC(n2cncn2)C1)=O)C(C)C 56218,C1(C(=O)N(C2CCCC(O)C2)C)(CNC(c2c(C)nco2)=O)CC12CCC2 56219,N1(C(c2c(CC)scc2)=O)CCN(C(c2cc(C#N)no2)=O)C(CS(C)(=O)=O)C1 56220,C1(C(C)C)CCCCN1C(=O)C(CCN(C)C)NC(=O)Cc1cscn1 56221,C1(NC(Cc2cc(CC)nn2C)=O)CC(O)CN(C(=O)CCC2(CO)CC2)C1 56222,c1(C(=O)NC(CNC(CN(CCC)C)=O)C(C)C)cc(C)c(C)c(S(N)(=O)=O)c1 56223,CCC(C)C(O)C(C)C(=O)N1CCC(CCNC(=O)C#CC(C)C)C1 56224,CC1C(NC(C2CC2CF)=O)CCCN1C(=O)C=Cc1nccs1 56225,Cn1ncc(C(N2CCCC2CNC(c2cnn(C3CCC3)c2)=O)=O)n1 56226,c1(OC)c(Cl)ccc(C(=O)NC2(C)CN(C(c3cc(N(C)C)ccn3)=O)C2)c1N 56227,C1(C(N2CCCCC2C2CCC2O)=O)CC(F)(F)CCO1 56228,N1(C(C(CO)N(C)C)=O)CCC(NC(c2ccc(-n3cncn3)nc2)=O)C12CC2 56229,C(CCN=c1[nH]c(=NC(C)c2nccs2)[nH]c2c1CSC2)OCC 56230,C(=O)(C1=CCCN(CC)C1)NC12CC3CCC(C1C2)N3CC12CC(C)(C1)NC2=O 56231,C1(NC(C(C)NC(CC)=O)=O)CCCC1NC(c1cn(CCO)nn1)=O 56232,c1(NC(C)=O)ccc(-c2nc(C(C)O)n(CC3CCCO3)n2)cc1 56233,C1(NC(c2c(C)scn2)=O)CCC(O)CN(C(=O)COC2CCC2)C1 56234,N1(C(c2cc(C3(C)CC3)on2)c2scc(Cn3cc(Br)cn3)n2)CCC(C)(O)C1 56235,N1(C(c2csc(C)c2C)=O)C(C)CC2CN(C(c3coc(CO)c3)=O)CC12 56236,Cc1ccc2oc(C(=O)NC3(C)CC(NC(=O)C(=O)NC4CCCCC4)C3)cc2n1 56237,CCC(CC)(CC)C(=O)N1CCN(C(c2nc(C(C)(C)C)no2)=O)C(C)C1 56238,N1(C(CC2CC(OCC)C2)=O)CCN(C)C(CNC(c2cc3ccsc3s2)=O)C1 56239,C(=O)(CCCN=[N+]=[N-])NC(C1CC=CCC1)C(=O)NCc1[nH]nc(C(C)C)n1 56240,C(N=c1[nH]c2cc(Cl)c(S(=O)(=O)NCC(Cl)=CCl)cc2s1)C1C(C)OCC1 56241,C1(NC(c2c(CC)ncs2)=O)COC2(C1)CN(C(C1(C)CCC(C)CC1)=O)C2 56242,C1(F)(CNC(C2(C)CC(=C)C2)=O)CCCN(C(c2ccnn2C2CCC2)=O)CC1 56243,N1(C(c2cccc(C)c2Br)=O)CC(NC(C2CC(O)C2)=O)CC12CCCC2 56244,c1(NC(N2CCCC2CC2(O)COC2)=O)ccc(F)cc1.c12ccc(o1)C2 56245,C1(CN(C(C(CC)F)=O)C)CCCCN1C(=O)C(C)N(C)C 56246,C1(CNC(C2CC3CCC2O3)=O)CN(C(=O)CSc2ccccc2O)CC1(F)F 56247,c1(C(N2C(C)CC(NC(Cc3c(C)cccn3)=O)C2)=O)cnc2c(Cl)cccn12 56248,N1(C(C(C)SC(C)C)=O)CCCCC(C(=O)NCC2CCCOC2(C)C)C1 56249,c1(C(=O)NC2CCC(CNC(c3nn(C)c(CO)c3)=O)C2)c[nH]cc(Cl)c1=O 56250,N1(C(c2ccccc2OC(F)(F)F)C)CCC2CCN(Cc3ccccc3)C2C1 56251,CCS(=O)(=O)CC(=O)NC(c1cc(-c2ccc(Cl)cc2)on1)C 56252,c1(C(N(CCCNC(C2CC23CCOC3)=O)C)=O)ccc(Br)c(F)c1F 56253,C1(CC=C)(N(CCC(=O)OC)C2CC2)CCCCC1.c12c[nH]cc1NC2=O 56254,c1(C(=O)NC2C(NC(C=CCC)=O)CC2)cc2ccc(Cl)cc2c(=O)o1 56255,Cc1c(C=CC(=O)NC2CCN(C(C3(CO)COC3)=O)CC2O)cnn1C 56256,C(=O)(CC(C)(C)Cc1ccc(Cl)cc1)NC(CC)(C)CNC(c1cccnn1)=O 56257,n12nnnc1C(c1cnsc1)NCC2.C(CC(C)CC)SC 56258,c1(C(N2CCCC(CCC(=O)NCCCNC(=O)OC)C2)=O)ccc(C)c(O)n1 56259,C12(OC)CC1CN(C(=O)C(C1CN(C(=O)C(C(C)C)N(C3CC3)CC)C1)OC)C2 56260,CCCC(C(=O)NC(C(=O)Nc1cnn(C)n1)C1CCCC1)NC(N)=O 56261,c1(C(C(=O)NC)N(C2CCOC2=O)C)ccc(C)c(C)n1 56262,C#CC1CN(C(C2CCC=CO2)=O)CCN1C(c1ncc(F)cc1F)=O 56263,c1(-c2cn(CC(C)NC(c3cnns3)=O)nn2)c(F)cccc1F 56264,C1(NC(Cc2nc(C)sc2C)=O)CC2(NC(=O)C(C)(C)C3CCCO3)COC1C2 56265,Cc1cc(=NCCCC(C)(C)NC(c2ncc(F)cn2)=O)[nH]c(C(F)(F)F)n1 56266,C1(N(C(=O)CC(CC(C)(C)C)C2CC2)C)CCN(C(=O)C(C#N)C2CC2)CC1 56267,C1(C(N2CCC(CC)(CO)C2)=O)CC2C=CC1N(C(=O)Cc1ccns1)C2 56268,C1(CNC(c2c(OCC)cccc2)=O)CCN(C(c2cnsc2C)=O)CC1(F)F 56269,c1(C(=O)NC2C(NC(C(Br)=C(C)C)=O)CC2)cc2ncccc2o1 56270,N1(C(c2ccnc(C)n2)=O)CC2CCCCN2CC1CNC(=O)Cc1cnc[nH]1 56271,N1(C(C(C=C)O)=O)CC2CCC1C1CN(C(c3c(F)cc(F)c(F)c3F)=O)CC21 56272,C1(COC)COCCC1NCCc1csc(CNC(=O)OC(C)(C)C)n1 56273,c1(NC(CC(C)NC(=O)CNC2CCCS2(=O)=O)C)ncccc1C#N 56274,O=C(C(F)CC1CC1)NC1CCCC1NC(c1ccn(Cc2ccccc2)n1)=O 56275,C1(=O)C(C)C(=O)N1CCCC(C)O.C(C(=O)OC)CCC 56276,c1(C(=O)OC)ccc(NC(N2CCCC(N(C)C(=O)OC(C)(C)C)CC2)=O)cc1Cl 56277,N1(C(c2ccc(OCC)cc2)=O)CCN(C(C2CCCN2N=O)=O)CC1C1CCC1 56278,CCC(c1ccc(C)cc1)=CC(=O)NC(C)CN(C)C(c1n[nH]cc1OC)=O 56279,c1(C(N2CCC(C)(NC(CCN(CC)CC)=O)C2)=O)ccc2c(c1)OCC2 56280,N1(CC(=O)NC2CC(CCNC(C3(SC)CCC3)=O)C2)CCCCCC1=O 56281,C(=O)(CCC(=O)NC(C)(C)CC(=O)NC1CCN(C(N)=O)C1)NCC 56282,CC1(CNC(C2(c3cccc(O)c3)CCC2)=O)CCCN1C(C1CC(=O)N1)=O 56283,C1(CC)CN(C(c2c(C)nsc2C)=O)CC1N(C(=O)CC(C)(C)C1CC1)C 56284,c1(SCC)ccccc1-n1nc(C(C)OC)nc1-c1cccc(C2CCOC2)c1 56285,c1(CCS(C)=O)sncc1Br.C1CCOCCN1 56286,N1(C(CC(CC)(C)C)=O)CCC2(CCCN2C(c2sccc2C)=O)C1 56287,C1(C(=O)NC2C(NC(CC)=O)CCC2)CC12CC(F)(F)C2 56288,CCCCC(C(=O)NCC1(F)CCN(C(=O)C(O)(C2CC2)C2CC2)C1)C(C)C 56289,N1(C(C(F)=CC)=O)CCC(C2CCCN(C(c3n[nH]c(CC)c3Cl)=O)C2)C1 56290,C12(NC(=O)Cc3ccno3)CC1CN(C(C1CCCOC1c1cc[nH]n1)=O)C2 56291,C1(CCNC(CCN(C)C(N)=O)=O)COCCN1C(=O)COC(C)(C)C(F)(F)F 56292,c1(C(=O)OC)cc(Cl)c(OC)cc1CN1CCCC(CS(C)(=O)=O)C1 56293,C1(C(=O)NC(CCC)c2nn[nH]n2)N(C(c2c[nH]c(=NC)o2)=O)CCCC1(C)C 56294,N1(C(C2N(C)CCOC2)=O)CC2(CNC(C3(CC4CC4)CC3)=O)CC1CCO2 56295,Cc1nc(Cc2ccccc2)oc1C(=O)NCC1CCN1C(C1CC1F)=O 56296,C1(NC(CC(CC)O)=O)CC2CCC(C1)N2C(=O)C(c1ccc(F)cc1F)C 56297,C(c1cccc(Br)c1)=CC(=O)NCC1C(NC(C(CC#C)C)=O)CC1 56298,C(=O)(C(=O)N=c1ccn(C2CC2(F)F)[nH]1)N1C(c2n(C)cnc2)CCC1 56299,C(CNC(=O)C=CC(F)F)(CC(=O)NCC1COC(C)(C)C1)OC 56300,C1(NC(C(C)NC(=O)NC)=O)CCN(C(c2c(C)ccoc2=N)=O)CCC1(F)F 56301,c1(C(=O)NCC2(O)CN(C(C3CC(OC)C3)=O)C2)nn(-c2cnn(C)c2)nc1C 56302,c1(OC)cc(C(=O)NC2CCC(CNC(C3(C)CCCCC3C)=O)CC2)cnc1C 56303,N1(C(c2c(C)nco2)=O)CC2(C(=O)Nc3cn(C)c(=O)nc3O)CCC1CC2 56304,c1(C(=O)NCCCC2N(C(Cc3ccc(C)o3)=O)CCC2)ccc(C)nc1O 56305,N1(C(CCC2C(C)C2)=O)CC2CC(N=c3cc(Cl)nc(OC(C)(C)C)[nH]3)CC1C2 56306,N1(C(c2cn(C)c(=O)cn2)=O)CC2CCN(C(=O)CCNS(C)(=O)=O)CCC2C1 56307,c1(CC(=O)NCc2c(C3CN(C(c4cc(C)sn4)=O)C3)ocn2)ncccc1C 56308,c1(CN2CC=C(CNC(C3OCC(C)C3)=O)CC2)cccc2cc[nH]c12 56309,C1(COC)CCN(C(=NCC2SCCS2)NCCSC)CC1 56310,N1(C(CCc2cc(OC)no2)=O)CC(NC(C2CC2CC(C)(C)C)=O)C2(CC2)C1 56311,c1(C(N2CC(NC(C3CC4CSCC(C3)C4)=O)C(O)C2)=O)ncc2[nH]ncc2n1 56312,N1(C(CC=C)=O)CCC(NC(C2(C)CC2(F)F)=O)C(C)C1 56313,C1(OC)CN(C(C2CC3(CCC3)C2)=O)C(C)(CNC(c2ccc(F)cc2Cl)=O)C1 56314,N1(C(c2c(C)cno2)=O)CC(NC(=O)Cn2cc(C#N)cn2)C(CC2CC2)C1 56315,CC1CCC(CO)N1C(C12CC1CN(C(c1cnsn1)=O)C2)=O 56316,C(=O)(C1CCCc2nncn21)NC1C(C)CCN(C(C2C(C(=C)C)OCC2)=O)C1 56317,N1(C(C(C(C)C)OC)=O)CCC(CNC(=O)C(C)(C)O)C(F)(F)CC1 56318,c1(-n2cc(CCN(C(CN3CCN(CC)CC3)=O)C)nn2)ccc(F)c(C)n1 56319,N1(C(C=CC(=O)N(C)C)=O)CCC2(CC2)CC1C(=O)NCC1(C#N)CCC1 56320,CC(C)C(O)CC(=O)N1CC(F)CC1CC(=O)Nc1ccc(Cl)nc1 56321,Cc1ccc(CC(=O)N(C(C)CNC(c2c[nH]nc2-c2ccncc2)=O)C)cn1 56322,C1(CC(N2C(COC)CCC2)=O)(NC(=O)Cn2nccn2)CCCCC1 56323,c1(NCCC(=O)NC2CC(C)CN(C(=O)C(F)(F)F)C2)ccccc1[N+](=O)[O-] 56324,C(c1cnc[nH]1)=C(C)C(=O)Nc1ncoc1CCNC(=O)CCC1CCOCC1 56325,c1(C(N(C)CC2CCN(C(CCCCCC)=O)C2)=O)ccc2cccnc2c1 56326,c1(OC)ccc(C(=O)NCC(=O)NCC(C)CNC(C2(C)CC(C)(C)C2)=O)cc1 56327,CN1CCC(C(N2CCCC2CCC(=O)NC2COC(C)(C)C2)=O)C1=O 56328,CC(C)(F)CCC(=O)NC1CC1CNC(C1COC(Cn2cccn2)C1)=O 56329,O=CN1CCCC1C(=O)N(CCC(=O)NCCN1CCOC1=O)CCO 56330,C1(NC(C2OCCN(CC)C2)=O)(CO)CCN(C(C2(C(N)=O)CCCC2)=O)CC1 56331,C1(CCC)COCCN1C(c1cccnc1)C(=O)NC1CCOCC1 56332,C1(N(CCC)C(N2CCC(CC(=O)O)C2)=O)CCC(CCn2cccn2)CC1 56333,N1(C(C(C)OCOC)=O)CC2CCC(C1)C(NC(c1cccc(NC(C)C)c1)=O)C2 56334,N1(C(c2nccc(CNC(CC3(OC)CCC3)=O)c2)=O)CC(C)CC1(C)C 56335,C1(C2CCN(C(c3c(Cl)n[nH]c3C)=O)C2)(NC(c2cncc(C=C)c2)=O)CC1 56336,CC1(C)CN(C(C2CCCCC2O)=O)CCC1NC(C1CC12CCSCC2)=O 56337,C(=O)(C(F)CC(C)C)N(CC(CC)NC(c1ccc(OC)cc1)=O)CC 56338,N1(c2c(Cl)cnc(OC)n2)CCC(C)C(NC(c2cnc3n2CCC3)=O)C1C 56339,Cc1ccc(C2=CCC(C#N)CC2)c2[nH]c(C(=O)NCc3ccncc3Br)cc12 56340,c1(NC(c2n(C)nnc2)c2nnnn2CC2CCCO2)ccc(O)c(F)c1 56341,C=CC1(C(N2CCOC(C#N)C2)=O)CCN(C(c2cc(CC)no2)=O)CC1 56342,C(=O)(CCCOC(C)(C)C)N1CC(NC(C=C(C)C(F)F)=O)C1 56343,C(=O)(C(C)(COC)OC)NCC(CNC(C(C=C)C)=O)OC 56344,N1(C(C2CC(=C3CC3)C2)=O)CCCC2C1CCN2C(=O)CN1CSCCSC1 56345,C(CCCCC(=O)N1CCN(C)C(C2CC2)C1)SCC.C(C(C)O)O 56346,c1(CC)ccc(C)cc1C(N1CCC(C2CCCN(C(C3C(C)C3C)=O)C2)C1)=O 56347,N1(C(c2n[nH]c3c2CCC3)=O)CCC2CN(C(C3(CC(F)F)CC3)=O)CCC2C1 56348,C#Cc1cc(C(=O)NCC(C)(C2CCC2)NC(=O)C=CC2CCCC2)ccc1C 56349,C(CCO)(C(C)(C)C)NC(CCC(C)NC(=O)CCc1ncccn1)=O 56350,c1(NC(=O)CNC(=O)NCC2CCCN2CC(c2cccnc2)=O)ccc(F)cc1 56351,c1(C(N2CCC(CC(C)O)CC2)C(=O)NCCCC2CC2)cc2occc2s1 56352,c1(SCC(=O)NCC2C(CNC(C(N)=O)=O)C2)ccc(F)c(F)c1 56353,c1(CC)nnsc1C(=O)NCC(C)(O)CNC(=O)CCC1CCCOC1 56354,C(=O)(C(C)(O)CC(F)F)NCC(CNC(CCn1c(C)nc(C)n1)=O)(C)C 56355,c1(C(N2CC(CC(F)C(N3CC(F)(C4CC4)C3)=O)C2)=O)ccc(F)cc1F.C 56356,ON(CC)C(=O)CNC(=NCCc1ccc(SC)cc1)NCC.C1(C)CCCCC1 56357,CC(C)(CC(=O)NCC(C)(C)NC(=O)Cn1nnc(=N)[nH]1)CC(F)F 56358,c1(CC(C)C)ccc(C=CC(=O)NCC2CC(CNC(=O)CO)CO2)cc1 56359,Cc1ccc(-n2cc(CN(C3CCNCC3)C(C)C(=O)O)nn2)c(Br)c1 56360,C(=O)(C(C)(CC)C(=O)N1CC(CNC(=O)COC(C)C)C(F)(F)C1)OCC 56361,C1(NC(CC(C)C)=O)C2CC1CN(C(=O)CC1CCS(=O)(=O)C1)C2 56362,c1(C(=O)NC(C(N2CC(C#CC)C2)=O)CCC2CC2)cnc(C)c(C)c1 56363,C=CCCCCC(=O)OCc1csc(CC(=O)O)n1 56364,C1(NC(C2C3CN(C(C(=O)NCC)=O)CC32)=O)(CO)CCC(F)(F)CC1 56365,C(=O)(N=c1[nH]c(S(C)(=O)=O)ncc1Br)c1c(CCCCCC)c(CC)n(C)n1 56366,N1(C(C(C2CCCN(C(c3cnnn3C3CC3)=O)C2)C)=O)CCc2sccc2C1 56367,N1(c2cc(OCC)ncn2)CC2(C)CN(C(=O)C(C)Cc3ccco3)CC2(C)C1 56368,CC1CC(CNC(=O)CC(C)(C)NC(C2(C)CC(O)CN2C)=O)CC(=O)N1 56369,C1(N=[N+]=[N-])(C(=O)NC(CC)C(F)(F)F)CCN(C(C2CNC(=O)C2)=O)C1 56370,C1(CC=C)(C(=O)NCCOCC=C)CCCN1CCN1CCOC1=O 56371,C1(NC(CCc2ncc(C)[nH]2)=O)(CO)CCN(C(c2occc2F)=O)CC1 56372,S(=O)(=O)(c1cccc(N2CCN(C3CCC3)CC2)c1)N.N1(C(=O)C=C)CCCC1 56373,N(C1CCc2ccccc21)C(C(CCSC)NC(C1CCCCO1)=O)=O 56374,C1(COC)(NC(=O)C(C)CC(N)=O)CCCN(C(=O)CCc2cccc(C)c2N)C1 56375,c1(CC)ccc(C(c2nnnn2C2COC2)Nc2ccc(C)nc2)c(C)c1 56376,N1(C(c2ccnc(OC(C)C)n2)=O)CCC(NC(=O)C(=CC(C)(C)C)N)C(C)C1 56377,Cc1nc(N(CC(C)CNC(c2cn(-c3ccn(C)n3)cn2)=O)C)c(C)c(C)n1 56378,C(=O)(NN1CCCC1C(=O)NC1(CN(C)C)CC1)c1c(C)ncs1 56379,CC(C)CC(C(=O)NC(C1CCOC1)CO)ONC(c1ccc(N)cn1)=O 56380,C(=O)(C(O)CC(C)C)N1C(CCNC(c2c(OC)noc2C)=O)CSCC1 56381,c1(C(=O)OCC)cnc(N(C)CC2CCCN2C(C2CC23CC3)=O)s1 56382,N1(C(CCOCC)=O)CC2(CCC(NC(=O)C(=O)NCC(F)F)CC2)C1 56383,c1(C(=O)OC)ccc(C2COC2)cc1.N12CCCC1C(=O)C1CC1CNC2=O 56384,c1(NC)c(C(N2CCCC(CCF)C2)=O)sc2nccnc12 56385,C1(NC(Cc2nc(C(C)C)sc2)=O)CCN(C(=O)Cc2cnsc2)CC1C 56386,C1(C2(O)CCOCC2)(C(=O)NC2CC3CC(NC(C(CC=C)C)=O)C2C3)CC1 56387,C=CCC(CC(=O)OCC)OCC.c12ccc(cc1)ONCCCNC2=O 56388,N1(C(c2cnc(OC)nc2)=O)CCC2C(NC(=O)C=CC3CCCC3)CC12 56389,C1(C(=O)NCC(O)C(=O)NC2CC(CO)C2)CCC(O)CC1 56390,C(C)(CCC(=O)N(Cc1ccccc1)Cc1cccc(C)c1)OC(C)=O 56391,Cc1nc(C2CC2)ncc1C(N1CCOC(C2(O)CC2)C1)=O 56392,C(=O)(C(CC(N)=O)NC(c1ccccc1)=O)N(CC(O)C1CCC1)C 56393,C1(CNC(CCC=C)=O)(OC)CCN(C(=O)C=Cc2nccs2)C1 56394,C(=O)(C1=CCCN(C(C2CCN(C(c3ccc[n+]([O-])c3)=O)CC2)=O)C1)OC 56395,c1(CC(=O)Nc2ccc(CNC(CC(C)(C)O)=O)o2)ccc2c(c1)CC2 56396,c1(C(N2CC=C(CNC(C(C)OC(C)(C)C)=O)CC2)=O)cnc2[nH]nnc2c1 56397,CC1(CC(N2CCC(OCC3CCC3)C2)=O)CN(C(=O)CCn2cccn2)C1 56398,c1(C(N2CCN(C(C(CC)C)=O)C(c3ccccn3)C2)=O)ccn2cncc2c1 56399,c1(C(=O)NCC(N(C(=O)CCn2cncn2)C)C2CC2)cccc(CO)c1 56400,N1(CC(C)C)CCN(C(C23CC(CN2C(=O)C(F)(F)CO)C3)=O)CC1 56401,c1(Nc2[nH]nc(SC)c2C#N)ccc2ncc(-c3cccc(F)c3F)n2c1 56402,C1(NC(C(C)Cc2cccnc2)=O)COCCN(C(c2cc(F)ccc2N)=O)C1 56403,c1(CC(=O)NCC(CN(C(=O)C=CC(F)(F)F)C)O)ccc2ccoc2c1 56404,C(=O)(C1=NOC(C)(C)C1)N1CCC(C(C)NC(=O)C=CC(N)=O)C1 56405,c1(CN2C(Cn3cc(-c4n(CC)ncc4)nn3)CCC2)ncccc1OC(F)F 56406,C(=O)(C(O)C(C)C)NC(C(N1CC(O)(CC=C)C1)=O)CO 56407,c1(CN(C(=O)CC2(c3ccccc3)COC2)CC=C)cccc(F)c1F 56408,c12ccc(c(F)c1)NC(=O)CC2.N1(CC)CCC1C(=O)OC.N12CC(C1)NC2=O 56409,N1(C(c2c(C(C)C)sc(Cl)n2)=O)CCC(C)C(NC(=O)C=CC=C(Cl)Cl)C1 56410,CN1CCC(Nc2cc(NCc3nc(Cl)cs3)ncn2)CC1=O 56411,c1(NC(N2CC(n3cnnn3)C2)=O)ccc(Cc2ccc(Cl)c(F)c2)c(F)c1 56412,c1(C(N2C3CC(NC(c4ccc(SC)o4)=O)C2CC3)=O)c(C)ccc2n[nH]cc12 56413,C(CC(=O)NC(CO)C(N)=O)(C(C)(C)C)NC(C(C)=C1CCC1)=O 56414,N1(C(CC2CC(=C)C2)=O)CC2CC1C1CC21.C1CCC(=O)N1C 56415,C1(C(=O)NCC(CN(C(=O)CC23COC(CF)(C2)C3)C)O)CC2OC1C1CC21 56416,S(=O)(=O)(c1cccnc1NC1CCCC2(CCC2)C1)NCC(CC)C(C)C 56417,N1(C(c2cc(C)c(F)cc2Cl)=O)CC(C)CN(C(c2ccc(N)cc2)=O)C(C)C1 56418,N1(Cc2cc(OC)c(Cl)cc2)CCC(F)(F)C(C(=O)Nc2ncc(Cl)cc2Br)C1 56419,c1(COC)nc(N2CC(O)(C(C)NC(C3CC(OC)C3)=O)C2)cc(O)n1 56420,c1(C(=O)NC2C3CCN(C(CCSCCC)=O)C32)cc2ccc(OCC)cc2[nH]1 56421,C1(C(=O)NC2CCC(NC(=O)Cc3ccsn3)CC2)CN2CCN1CC2 56422,c12ccccc1C2OC.C1(=O)C(CC2CCCC2)N1.N(C(=N)N)CC 56423,CC1CN(C(=O)CC(=O)NCC(F)(F)F)CC1CCNC(=O)CC1(C)CCCO1 56424,C1(C(N2CCCC2c2ccccc2)=O)(NC2CCC(O)C2O)CCOCC1 56425,N1(C(C2COCCN2C2CCCC2)=O)CCC(CO)C1(C)C.N1(CC)CC1 56426,C(=O)(C1=CCCCCC1)N1C(CNC(C2CC(OCC)C2)=O)C(C)CC1 56427,N1(C(C(C=C=C)C)=O)CCC(C2CCN(C(c3ccc(=O)n(C)c3)=O)CC2)CC1 56428,C1(C(CC)(C)C)CC(C(N2CCN(C(=O)CCF)CC2)=O)CCO1 56429,c1(NC(C(Cc2cc[nH]n2)NC(CCC(CC)=O)=O)=O)cn(C)c(=O)cc1C 56430,C1(NC(c2ccc(C(C)C)s2)=O)CC2CC(NC(C3(c4cc[nH]n4)CC3)=O)C2C1 56431,C1(C(=O)NCC(CC)(C)C(N)=O)CC(C)(C)CCN1C(c1ccc(C(F)F)o1)=O 56432,C1(N(C)C2CC2)CCCN(C(C(=O)CCC(=O)OC(C)(C)C)=O)CC1 56433,N1(C(c2c(COC)cc[nH]2)=O)CCN(C(=O)Cc2ccc3c(c2)CC3)C2(CC2)C1 56434,CCC(CC(F)(F)F)C(=O)NCCCNC(C12CC(F)C1C2)=O 56435,Cc1cc(C)c(CC(=O)NC2CCC2NC(=O)CC2CCC3(CCC3)O2)c(C)c1 56436,C=CC(C)CC(=O)NC1CC(O)C1CC(=O)NCc1cnc(CC)cn1 56437,CCCC(O)CC(=O)N1CC(NC(=O)CC2=CCCC2)C(C)(C)C1 56438,c1(NCCSC)ccc(S(=O)(=O)NC2CCC3CC23)cc1Cl 56439,c1(C(N(C(CS)C)C)=O)cccc2nc(N(C)C)oc12.N1(CC=O)CCCC1C(=O)OCC 56440,C(C)(C)(C(=O)N1CC(C2C(=O)N2)C1)OC.C1(C(N)=O)(CSC2CC2)CCC1 56441,c1(OC)ccc(OCC(N2CC(NC(=O)CSCC(N)=O)CC2C)=O)cc1 56442,N1(C(C=COCC)=O)CCN(C(c2cc(-c3ccco3)c[nH]2)=O)C2(CC2)C1.C1CC1 56443,C1(=O)CC(C(F)(F)F)ONC(=O)C2CCCN12.C(=O)(C(F)(F)C(F)F)OCC 56444,C(=O)(C1(C)CCc2ccccc21)NCCC1CC(NC(c2n(C)c(S)nn2)=O)C1 56445,CC1(C(=O)NC)CCN(Cc2cccnc2Cl)CC1.c1(CC(=O)N)cccc(CO)c1 56446,C(C(C)C(F)C(=O)NCCC(F)(F)C(C)C)NC(c1cc(C)ns1)=O 56447,C1(N(C(CCC(=C)Cl)=O)C)CCCN(C(c2nocc2Br)=O)CC1 56448,CC(=O)C(C)(C)CC(=O)N1CCC(N(C(=O)C(C)OCC(C)C)C)C1 56449,C(=O)(C1=CCS(=O)(=O)C1)N(CCNC(c1cccc(-n2ccnc2O)c1)=O)CC 56450,c1(C(=O)NCCNC(c2cn3c(n2)SCC3)=O)cc2ccc(Cl)nc2s1 56451,C(=O)(C(CC(F)F)NC(C1CCOCC1(C)C)=O)NCCc1n(C)ncn1 56452,C1(NC(C(c2ccccc2)NC(=O)CCn2cncn2)=O)CCSCC1 56453,C(=O)(C(C)(C)CC(C)C)N1CC(OCCNC(C(F)=CCC)=O)C1 56454,Cc1ncc(C(=O)NCCC2(C(=O)NC(C)C(C)(C)CO)CCC2)c(=N)[nH]1 56455,C(=O)(CCC(F)(F)C(F)(F)F)NC(CC)CN(C(=O)CC1(C)CCOC1)CC 56456,C1(C(N2CCC(NC(c3cc[n+]([O-])cc3)=O)C2)=O)CC2CC1N(CCO)C2 56457,c1(C(=O)NCC2C(C)CN(C(C3C=CCC3)=O)CC2)cc2cc(F)ccc2s1 56458,c1(NC(CC)=O)ccc(C(=O)NCCCN(C(=O)C(C)CN(C)C)CCO)cn1 56459,N1(C(c2c(C#C)cnn2C)=O)CCC2(NC(=O)CCC(=O)NC)CCCC12 56460,C1(NC(CCN(CC(=O)OCC(=O)NC2CC2)C)=O)CCOC(C)C1 56461,N1(C(C(COC(C)C)NC(C)=O)=O)Cc2[nH]nc(C(=O)NC3(Cl)CCC3)c2C1 56462,c1(N(C2CC(F)C2)C(C)C)ccc2c(c1)OCO2 56463,C1(C(=O)NCC2(C#N)CCCC2)(OC)CCN(C(=O)C(C(C)C)SC)C1 56464,CC1CCCC(C(=O)NCCOC2CCN(C(=O)CCC3CCCC3)C2)C1 56465,CCC(CC)CC(=O)NCc1ncoc1C1CN(C(=O)C(C)(C)C(C)C)C1 56466,Cc1cccc(C(=O)NCCOC2CN(C(C3(C(C)(C)O)CC3)=O)C2)c1F 56467,c1(C(=O)NC2CCN(C(CCc3cncc(C)c3)=O)C2)ccc2c(c1)CCC2=O 56468,C1(C(=O)NCCC(C)N(CCC)C)C=CCCN1C(=O)Cc1ccsc1 56469,C(c1ccc(Cl)cc1Cl)=CC(N1CC(C(=O)Nc2ccc(Cl)cc2O)OCC1)=O 56470,N1(C(COCC(=C)C)=O)CCCC(N(C)C(c2ccc(Cl)s2)=O)CC1 56471,c1(NC(=O)CCc2ccc(-c3nn[nH]n3)cc2)ccc(F)cc1O 56472,c1(COC)cccc(C(=O)NC2CCCC(NC(=O)CSC(C)(C)C)C2)c1 56473,C1(C)(NC(C(C)Cc2cccnc2)=O)CCN(C(=O)C(C)(C)C)C1 56474,CC1(C)CC(C(N2CCCC(NC(=O)Cc3ccsc3)CC2)=O)CC(C)(C)S1 56475,C1(C(=O)OC)CC12CCC(NC(c1sc(SC)cc1C)=O)CC2 56476,c1(CC(=O)NC2(CCNC(Cc3cc(C)n(C)n3)=O)CC2)ccc(Cl)c(Cl)c1 56477,C12(CNC(=O)COC3CC3)CCC(CC1NC(=O)C(C1CCOCC1)O)C2 56478,c1(OC)cc(F)cc(F)c1S(=O)(=O)N1CCN(C(C)(C)C)CC(C)C1 56479,c1(-c2ccc(CC)cc2)cccc2c(C(N3CCC(N(C)C)C3)=O)csc12 56480,N1(C(c2[nH]cc(COC)c2)=O)CCC12CCN(C(c1cc(C)cc(F)c1)=O)CC2 56481,C1(C(N2CC(C(=O)OC)C2)=O)CC12CN(c1nncs1)C2 56482,c1(C(=O)OC)cc(C(=O)NC2(CC(c3coc(C4CC4)c3)=O)CCOC2)cn1C 56483,c1(CC(N2C(CN(C(CC(CC)(F)F)=O)C)CCC2)=O)nnc2n1CCOC2 56484,c1(C(=O)NC(CN(C(C2(F)CC(C(=O)OCC)C2)=O)C)C)csc2nccn12 56485,c1(C(=O)NCC2(COC)CN(C(C3CC4CC4C3)=O)C2)cnc2n1CCCC2 56486,C(CC(C(=O)NC(c1cn[nH]c1)C)NC(c1[nH]ccc1C)=O)OCC 56487,C(=O)(C(C)(F)C(=O)NCC(C)(F)CNC(=O)CC1CC1(Cl)Cl)OC 56488,S(=O)(=O)(c1ccc(I)s1)N.C(C(F)(F)CCO)c1ccc(OC)cc1 56489,N1(S(CCC)(=O)=O)CCCC(OC(C2(F)CCCCC2)=O)C1=O 56490,C1(NC(c2c(C)nccn2)=O)(CNC(C2CCCC2C)=O)CC2CCC1CC2 56491,N1(C(Cc2cn(CC)nc2)=O)CC(C)(C)OCC1CNC(=O)C(CN(C)C)N(C)C 56492,C=C(C)CC(C)C(=O)NC1CCCCC1NC(=O)C(C)(C)Cc1cccc(Cl)c1 56493,Cc1ccc(C(C)C(N2CCCC2(C)C(=O)Nc2cncnc2Cl)=O)cc1 56494,c1(C(=O)NCC(C2CC2)NC(C(C=CCCC)O)=O)cccc(C(C)(F)F)n1 56495,C(=O)(C1c2c[nH]nc2CN1C(c1ccc(CC)nc1)=O)N1C(C=C)CC1 56496,S(=O)(=O)(c1ccccc1N)N(CCC)Cc1ccc(SC(F)(F)F)cc1 56497,CC(O)(CNC(C1CC12CC(NC(c1coc(C3CC3)n1)=O)C2)=O)CCO 56498,c1(C(=O)NCCC2N(C(c3ccc(C(C)=O)o3)=O)CCC2)ccc2c(n1)CCC2 56499,C1(NC(c2cccc3ncsc23)=O)CN(C(c2cnco2)=O)CC12COC2 56500,c1(C(N(C)CC2(CNC(C3CCC4CCC34)=O)CC2)=O)ccc(S(N)(=O)=O)s1 56501,N1(C(c2cn(C)nc2)=O)CCC(CO)(NC(=O)CC2(N(C)C)COC2)C1 56502,O=C(CCC(=O)c1ccncc1)NC1CCCCC1NC(C1CC2CC2C1)=O 56503,c1(C(=O)NCCCCNC(C2C(C)CCOC2)=O)c(F)ccc(Cl)c1[N+](=O)[O-] 56504,C1(O)(CC(=O)N(CC(C)(O)C2CC2)C)CCCCC1.C12CCC(C1)NC2=O 56505,C(C(=O)N1CC2CC2(CNC(c2c(CO)noc2C)=O)C1)(C(C)C)OC 56506,C1(NC(c2c(C)coc2C(C)C)=O)C2CCC1N(C(=O)CC1COCCO1)C2 56507,n1(CC)nnnc1C(c1nc(C(=O)OC)co1)NC1CC1c1ccccc1 56508,C(C(=O)OCC1(CO)CC1)(C(C)C)NC(CC1CCN(C(C(CC)C2CC2)=O)C1)=O 56509,Cn1nccc1C=CC(=O)NC1CC(NC(c2ccsc2C#N)=O)C1 56510,N1(C(c2c(CC)nccc2)=O)CC(O)CC1(C)C(=O)NC1CN(c2ncco2)C1 56511,N1(C(C2CC(=C)C2)=O)CC2(CC(NC(C3(OC)CCCCC3)=O)c3nccn32)C1 56512,CC1(C)CC(C(=O)NCC(O)(CO)CO)CN(C(=O)Cn2cnnc2O)C1 56513,c1(-c2cccc(OCC)c2F)c(C(=O)NCCC2CC2)[nH]c2ccccc12 56514,C(=O)(C(F)C(C)CNC(=O)CC1CC(=O)C1)N1CC(CSCC)C1 56515,CC1CC(NC(C2COCCOC2)=O)CN(C(c2ccsc2C(F)F)=O)C1 56516,N1(C(=O)CC2CCCCC2O)CC2(C=C(C(=O)N3CCOC4C(O)CC34)CO2)C1 56517,Cn1ccc(CC(=O)NCCc2n[nH]cc2C(=O)NOC2CCC2)n1 56518,CCCC(C)(C)CC(=O)N1CC(C(=O)NCC2CN(C(C)C)C2)C(F)(F)C1 56519,N1(C(C(C)=C(CC)C)=O)C2CCC(C2)C1CC(N1CCOC2CC12)=O 56520,N1(C(C(CC)C)=O)CC(F)CC1C(=O)NCc1ccnc(Cc2ccccc2)c1 56521,C1(N(C)C(C2CC(C(F)(F)F)C2)=O)CC(C)(N(C)CCO)C1.C(=O)CCN(S(C)(=O)=O)C 56522,C(=O)(C(C)(C)C(C)(C)O)N1CC(C)C(CCNC(C2CCCN2C)=O)C1 56523,c1(C(N2CC3C(CNC(c4cnc(C(C)C)s4)=O)C3C2)=O)ccc(Cl)c(F)c1N 56524,c1(C(CN2C(C(C)O)C2)Sc2ccccc2)cccc(Cl)c1O 56525,C(=O)(CCCCCCCC)NC1(C)CC(C(N2CCC(OCC#C)CC2)=O)C1 56526,Cc1snnc1C(=O)NCCC1CCC(NC(c2cnc(S)[nH]2)=O)C1 56527,N1(C(c2n(CC)ncc2)=O)CC2(C(=O)NC(COC)CCO)CCC1CC2 56528,C(=O)(C1=CC2CCC(C1)C2)N1CC(CC(=O)NC2CCCC2CF)(OC)C1 56529,C(C(C)(F)C(C)C)NC(C1C(NC(c2cc(CC)[nH]n2)=O)COC1)=O 56530,n1(CC(C)(C)CO)nc(-c2ccc(Cl)s2)nc1-c1cc[nH]n1 56531,C1(CNC(C2CCC(O)(c3ccccc3)C2)C)CC(C)CC(C)(C)C1 56532,N1(C(c2sc(C)cc2C)C(=O)NCCC(=O)OCC)CCC(C#N)CC12CC2 56533,C1(CC(N2C(CN(C(=O)Cn3cc(Br)cn3)C)CCC2)=O)COCC(C)(C)O1 56534,c1(CNC(C2CC(=C)CN2C(C2(O)CCC2)=O)=O)cc(C(F)(F)F)cc(Cl)c1 56535,C1(CCNC(CCCOCCOCC)=O)CN(C(=O)CCn2ccnc2)CC1C 56536,c1(C(=O)NCCOCCNC(c2sccc2CC#N)=O)nn[nH]c1Cl 56537,C=C(C)CCC(=O)N1CCC(NC(C2CC(C)=NO2)=O)C1CC 56538,C1(CNC(=O)CC2CCCOCC2)COCCN(C(C2C=CCS2)=O)C1 56539,Nc1cc(C(=O)NC2CC3(C2)CC(NC(c2ncncc2F)=O)C3)cc(F)c1O 56540,N1(C(c2nc(CCCC)sc2)=O)CCC(NC(=O)C2=CSCS2)CC1C1CC1 56541,C(=O)(C(F)CC(C)(C)NC(c1cccnc1)=O)N(C(C)CCO)C 56542,C(CNC(=O)CCn1c(C)csc1=O)(C(C)(C)C)NC(CSCCCC)=O 56543,C(c1cccc(F)c1F)=CC(=O)NCC1C(NC(c2cc(=N)[nH]cc2)=O)CC1 56544,N1(C(c2c(CC)scc2)=O)CCCN(C(c2cnc(O)c(OC)c2)=O)C(C)C1 56545,c1(CCC(N2CC(NC(C(CC)N(C)C)=O)C(F)C2)=O)cnc2ccccn12 56546,Cc1cc(Br)cn2c(CNCc3c(I)cc(Cl)nc3Cl)cnc12 56547,C1(NC(CN2CCN(C)CC2)=O)CCSC12CN(C(c1n[nH]cc1Cl)=O)C2 56548,CC1Oc2ccc(C(=O)OCC(=O)N(C)Cc3ccccc3F)cc2NC1=O 56549,c1(C(=O)NCC(C2CC2)NC(C2(C)CC=CCO2)=O)nnn2c1CCC2 56550,c1(C(=O)NCC2C(NC(COC)=O)COC2)cc2ccccc2cc1NC(C)=O 56551,C1(C(N2CC(C(C(=O)N(C)Cc3noc(C)n3)OC)C2)=O)CCC(N=[N+]=[N-])C1 56552,N1(C(C2C(C)=C2)=O)CC(CNC(=O)Cc2nc[nH]n2)C2(CCC2)C1 56553,c1(C(N2CCC(CC(=O)Nc3c(OC)cc(Cl)cn3)C2)=O)cc(Br)c(O)cc1O 56554,C(=O)(C1CCc2nccn21)NCCC1(C)CCN(C(COCC(=O)OC)=O)CC1 56555,C(=O)(C1=NOC(C(C)(C)C)C1)NC(CNC(C(C=C)(C)C)=O)(C)C1CC1 56556,c1(C(=O)NCC2CN(C(c3c(N(C)C)cncc3)=O)C2)ccc2nc(O)cn2c1 56557,Nc1nonc1C(=O)NCC1(CC(N2CCC(F)C2)=O)CC1 56558,C1(CC(=O)N(C)C)CCCN(c2ccnc(N3CCC(C)(F)C3)n2)C1 56559,CCN(Cc1ccc(F)cc1)N1CCCCC12CCS(=O)(=O)CC2.CO 56560,N1(C(=O)NC)CC2C=CC1C(C(N1CC(C(=O)NCC3CCCCC3O)C1)=O)C2 56561,C12CCCC1NC2=O.c1(C(=O)NCC2(O)CCC2)cc(C2CC2)no1 56562,Cc1cn(C)cc1C(N1CC2CC2(CNC(c2cccc(=O)o2)=O)C1)=O 56563,C(CCCCNC(=O)CC12CCCC1C2)N(C(C1(C(C)(C)OC)CC1)=O)CCO 56564,c1(C(N2CC(C=C)(CC(N3CC(C)C3)=O)C2)=O)cccc2ccnn12.C(C(C)CC)=N 56565,c1(C(N2C(C(N(c3cccc(C)n3)CCCC)=O)CC(C)C2)=O)ccc(Cl)cc1Cl 56566,N12CCCN(CC1C)C(=O)c1nc(C)c(s1)C2=O.C1(COCC)(OCC)CCC1 56567,c1(C(=O)NCC2N(C(c3cn(C4CCOC4)nn3)=O)CC2)c(F)cccc1F 56568,c1(C(=O)NCC2CC(NC(C#CC)=O)C2)ccc(I)c(C)c1 56569,C1(C(=O)NCC2CCN(C(c3ncoc3C3CC3)=O)C2)CC(=O)NC(=O)C1 56570,Cc1cc(C(=O)N(C(C)CNC(=O)C(C)SC2CCCC2)C)nc2ccccc12 56571,N1(C(c2nc(C)oc2C)=O)CCC(CO)(CNC(C2CN(C3CCC3)C2)=O)CC1 56572,CS(=O)(=O)c1cc(C(=O)NCC(F)CNC(C2(F)CC=CCC2)=O)ccc1F 56573,c1(C(N(C2CCN(C(=O)C(C)N3CCCC3)C2)CC)=O)ccc(=O)oc1 56574,C#CC1CC2CCC1N(C(C1CC3(CCN(C(c4cnc(Cl)s4)=O)C3)C1)=O)C2 56575,CC(C)CC(C)(CNC(C1(Cl)CC1(C)C)=O)NC(c1cccc(-c2cc[nH]n2)c1)=O 56576,Cc1cc(C(=O)NCCOC2CCN(C(=O)Cn3cccc3)C2)cc2ccsc12 56577,CCC(C(=O)N1CCC(CC(=O)NCC(C)(O)Cn2cccn2)C1)C(C)(C)CC 56578,c1(OCC)cccc(C(N2CC(NC(C3(CC)CCCO3)=O)CC2CO)=O)c1N 56579,C1(C(=O)NCCN(CCC#C)C)CC2(CCC2)CN1C(=O)C(F)C1CCC1 56580,c1(C(N2CCCC(N(C(C(CC)N(C)C)=O)C)CC2)=O)cc2n(n1)CCNC2=O 56581,N1(C(Cc2ccn(CC)n2)=O)CC(NC(c2ccoc2COC)=O)CCC1C 56582,N(C=CC(=O)C(F)(F)F)C(C1CCCCN1C(c1cc2ncsc2[nH]1)=O)=O 56583,CC(C)CC(C)CC(=O)N1CCN(C(c2cccc(SCC#N)c2)=O)C2CC12 56584,C1(C(=O)NCC(CN(C(c2n(CC#C)cnn2)=O)C)O)CCC2(CCC2)C1 56585,C#Cc1cccc(C(=O)NC2CC(CNC(c3cc(OC)n[nH]3)=O)C2(C)C)c1F 56586,c1(SC(C(N2C(CNC(c3c(C(C)C)onc3)=O)CCC2)=O)C)cccc(F)c1 56587,N1(C(C2CCC(C)C2)=O)CCOC2(CCN(C(c3cc(Cl)ccc3N)=O)C2)C1 56588,C1(CC(=O)NC2(C(N(CCOC)C)=O)CC2)CCC(C#N)C1 56589,c1(C(=O)NCC2(F)CC(CNC(COCCC(C)C)=O)C2)ccc(F)c(N)c1F 56590,CCCC(C(=O)N1CCC(NC(c2cncs2)=O)C(O)C1)C(C)C 56591,N1(C(c2c(C)ncs2)=O)CCC2(CCCC2NC(c2cc(O)nc(O)c2)=O)CC1 56592,N1(C(C(CC)O)=O)C2CCC1CN(C(c1c(C(F)(F)F)cccc1C(F)F)=O)C2 56593,c1(SCC(=O)NC2CCC2NC(C2CNC(=O)N2)=O)c(F)cccc1F 56594,c1(OCC(N2CCC(C)(NC(=O)CC(C3CC3)C3CC3)C2)=O)ccc(F)cc1Cl 56595,c1(C(N2CCC(NC(C(C)OCC#C)=O)C(F)C2)=O)csc2cccnc12 56596,CCC(CC)CC(C(=O)NCSc1ccccc1)N1CCCC(C)C1C 56597,C12(F)CCN(CC1)C2.O=C(C(Cl)=CCl)NCCNC(C1(CCc2ccccc2)CC1)=O 56598,C1(NC(c2n(C)nc(C3CC3)c2)=O)CC2CN(c3cnc(C#N)cn3)CC12 56599,N1(c2cc(NCCC3CCCOC3)nc(COC)n2)CCn2nccc2C1 56600,c1(CCC(=O)NC(CN(C(=O)C(C)(C)NS(C)(=O)=O)C)(C)C)cccc(O)c1 56601,Cc1cc(=NCC2CCCN(C(c3ncc([N+](=O)[O-])n3C)=O)C2)[nH]c(C2CC2)n1 56602,C1(CC)CCC(C(=O)NC2CCC2C(=O)NCCC2=CCCC2)CC1 56603,C1(NC(C2CC(F)CN2C(=O)Cn2cnnc2O)=O)CCn2ncnc2C1 56604,C#CCC(CC(F)F)C(=O)NC(CNC(c1nccnc1C(N)=O)=O)CC(C)C 56605,Cc1cccc(C(=O)NC(C(=O)NC2COCC2F)C(C)O)n1 56606,N1(C(c2ccno2)=O)CCC2(CC1)CCN(c1ncc3ccccc3n1)CC2 56607,C(=O)(CC(C)(C)NC(C1COCCC1C)=O)NCC(=O)NCCOC 56608,c1(C(=O)NCC2(CNC(C3(C)CCC(=O)N3)=O)CC2)cnn2c1OCC1(CC1)C2 56609,Cc1nn(C(C)(C)C)cc1C(=O)NCC(CO)NC(=O)C(C(C)C)N(C)C 56610,Cc1ccnc(C(=O)NCCC(C)N(C)C(C2CCC2(F)F)=O)c1N 56611,c1(C(=O)NCC2C(C)CCN2C(=O)CC2CCC(F)(F)C2)ccn2c1CSCC2 56612,Cc1cncc(C(=O)NCCN(C(=O)Cc2cnc(C3CC3)[nH]2)C2CC2)c1 56613,S(=O)(=O)(c1cccc2nsnc12)N1C2CCN(C(CN(c3cccs3)C)=O)CC2C1 56614,N1(C(CC2N(C(CCC)=O)CCCC2)=O)CCN(C(=O)COCC(F)F)C(C)C1 56615,CCCC(C(=O)NC1CC2C(NC(c3[nH]nnc3C(F)F)=O)C2C1)OC 56616,C=C1COCCN(C(C2C(CC)CCCN2C(c2oc(C)nc2C)=O)=O)C1 56617,S(=O)(=O)(c1cc(C(F)(F)F)ccc1Cl)NC1CCN(C(c2cscn2)=O)CC1F 56618,N1(C(C(C=C)c2ccccc2)=O)CCN(C)CC1CNC(c1ccn(CC)n1)=O 56619,c1(OC)ccc(F)c(N)c1C(N1CC(CCCCNC(C2C=CCCC2)=O)C1)=O 56620,N1(C(CCN(C(C2(C)CCCO2)=O)CC)=O)CCC(O)C(C)(C)C1 56621,C(=O)(C(C)(C)CC(C)(C)C)NC(C)C(C)C(=O)N1CCCC1C1CCOC1 56622,C(CCNC(C1CC1C(C)(F)F)=O)(C(=O)NCC(c1ccncc1)C)OC 56623,CCCCCCC(F)C(=O)N1CCOC(C2CN(C(c3ccc(=O)n(C)n3)=O)C2)C1 56624,C(=O)(C(O)CC(F)F)N(C1CCCN(C(CC2(OC)CCC2)=O)C1)CCF 56625,CCCCCC(O)CNC(=O)CC(CNC(c1cn(CCO)nn1)=O)C1CCC1 56626,C1(NC(CCCN(C)C(C2CC23CCC3)=O)=O)CN2CCC1(F)CC2 56627,N1(OC)CCC(O)C(CC(=O)NOCCO)C1.c1(C)csc(C(=O)OC)c1 56628,N1(C(CCC)=O)CCC2CCCC12C(=O)NCc1c(C)cccc1F 56629,C1(CC)CN(C(C2CCOCC2NC(C2CCCC2OC)=O)=O)CCCO1 56630,c1(C(N2C(COC)CN(C(=O)C(C)(O)C3CCC3)CC2)=O)cc2ccccn2c1 56631,C1(C(=O)NCCN(CCCCCC)C(C)=O)(Cc2ccccc2)CCNC1=O 56632,C1(CC#C)(C(=O)N(CC(=O)N(CC(F)Cl)C)CC2CC2)CCOC1 56633,C1(c2c(C)n(C)nc2)C(C(=O)N(C)Cc2cnco2)CC(=O)N1C 56634,C(C)(C(C)(C)NC(C1CC(F)(CO)C1)=O)NC(C(=C(C)C1CC1)F)=O 56635,c1(C2CN(CC(=O)Nc3c(NC(=O)OCC)scc3)C2)cccc(Br)c1 56636,C1(CNC(CN(CC(C)C)C(C2CCCC2)=O)=O)CCCN(c2ccncc2)C1 56637,c1(C(=O)NCC2CCC(NC(CCCOCC)=O)C2)cccc(C(N)=O)c1 56638,C(=O)(C(CC)C(C)C)NC(C(=O)NCCOCC#C)CCC1CC1 56639,C(=O)(C1=NOC(C)C1C)NCC(CCOC)NC(c1ccc(C(F)F)c(Cl)c1)=O 56640,C1(CNC(CCCC(C)(C)C)=O)CN(C(=O)CCc2cnco2)CCC12CCC2 56641,N1(C(C2(C)CC2)=O)C2CCC1C(F)C(NC(c1ccc(Cl)c(C(F)F)c1)=O)C2 56642,N1(C(CSCCCC)=O)CCC(CNC(C2(SC)CC2)=O)CC1C 56643,C(C(CC(=O)NC(C)(C)CCO)NC(=O)CCc1ccncn1)OC 56644,C1(CNC(C2(OC)CCOC2)=O)CN(C(c2coc(C)n2)=O)C2(CCC2)C1 56645,c1(C(N(CC(CN(C(C(C(CC)C)O)=O)C)O)C)=O)ccc(Cl)c(C)c1F 56646,N1(C(Cc2c(C)cccn2)=O)CCC(N(C)C(c2cnco2)=O)C(C)C1 56647,C12(CNC(c3cc(COC)no3)=O)CCCC1N(C(C1CCOC1C)=O)CCC2 56648,C(CC1=CCN(c2ncc(I)cn2)CC1)NC(CCC(C)OC)=O 56649,c1(OC)cc(CN2CC(O)CC2(C)C)ncc1-c1ccc(-n2ccnc2)cc1 56650,C(=O)(CCCCCF)NC1C(NC(C(N2CCCCC2=O)C)=O)CCCC1 56651,c1(NC2C(C)(O)CCC(C(=C)C)C2)cncc(S(C)(=O)=O)c1 56652,C(=O)(C1CCCc2c1ncn2C)N1CCC(N(C)C(C2CC2C(F)F)=O)C1 56653,c1(C(=O)NCC2C(C(=O)NC(CN(C)C)CCO)CCO2)cnc[nH]c1=N 56654,N1(C(CCSCCC)=O)CCC2(CC1)CC(CNC(=O)C(C)OCCCC)C2 56655,CCCCC(O)C(C)C(=O)NCCC1CN(C(C2(O)CC(C)(C)C2)=O)CC(C)O1 56656,N1(C(C(C)(C(C)C)OC)=O)CCC2(CC1)CC(CNC(c1cc(CO)[nH]n1)=O)C2 56657,c1(C(N2CCN(C(c3cncc(C)n3)=O)CC2)=O)cc(C(C)C)cnc1O 56658,N1(C(c2cc(CC)[nH]n2)=O)CCC(C)(C)C(C(=O)NC(C)Cc2cc(C)[nH]n2)C1 56659,C(=O)(C1=CC(O)CCC1)NC(C)C(C)(C)NC(C1SCCCS1)=O 56660,C1(NC(CNC(CC)=O)=O)CC2C=CC1N(C(c1cscc1C)=O)C2 56661,C1(NC(CCC(=O)N(C)C)=O)CCCN(S(=O)(=O)Cc2ccc(O)cc2)CC1 56662,c1(C(=O)NCC2C(NC(C(C)n3cnnn3)=O)C2)coc2cccc(O)c12 56663,Cc1c(NC(C)(CCCl)c2nnnn2C2CC2)cccc1F 56664,N#CC1=C(C(=O)NCC(C2CC2)NC(c2cn3c(n2)SCC3)=O)CCC1 56665,N1(C(Cn2c(=N)scc2)=O)CCC(C(N2CC(n3cccn3)C2)=O)(CO)C1.C1(CF)CCC1 56666,CCCC(C)(CCC)C(=O)N(C)CC1CN(C(=O)C(C)OCCC(C)C)CCO1 56667,N1(Cc2cc(C(C)C)no2)CC(CO)CC(F)(F)C1.N12CCCC(CC1)C2=O 56668,c1(C(N2CCCC(n3cc(CC(CC)(C)C)nn3)C2)=O)ccc([N+](=O)[O-])o1 56669,c1(OC)ccc(COCC(=O)NCCCn2cc(CC3CC3(Cl)Cl)nn2)cc1 56670,CC1CC(F)(F)CCN1C(C1CCN(C(=O)CCn2cccc2)CC1)=O 56671,Cc1c(CC(=O)NCCC2(CNC(C3(C(F)(F)F)CC3)=O)CC2)cnn1C 56672,c1(C(=O)NCC(=C)CCNC(C2CC2OC)=O)[nH]c2cc(Cl)cc(Cl)c2c1C 56673,CCCCCCCN=c1[nH]c(=N)[nH]c(=NCc2cn(C(C)C)nn2)[nH]1 56674,C(=O)(C(C(C)CC1CC(F)(F)C1)N1CCC(CC(=O)OCC)C1)NCCC 56675,c1(C(N2CC(C(C(N3CCC(CC#C)C3)=O)OC)C2)=O)cc(F)cnc1O 56676,S(=O)(=O)(C(F)(F)F)N1CC(NC(=O)CCc2cnco2)C1 56677,N1(C(CC(C)(C)O)=O)CC(NC(c2csc(Cl)c2)=O)CC(O)C1 56678,C(C1=CCN(C(C2CCCS2)=O)CC1)NC(C1CCCN(Cc2ccc(Br)o2)C1)=O 56679,N(C(=NCCC1COC(C)(C)C1)NCCN1CCCC1)Cc1ccc(OC)cc1 56680,CC1CCCN(C(c2cncc(NS(C)(=O)=O)c2)=O)C1CCNC(=O)C(C)(F)F 56681,N1(C(C2(S(N)(=O)=O)CC2)=O)CC(NC(=O)Cn2cc([N+](=O)[O-])cn2)C(C2CC2)C1 56682,N#Cc1ccc(S(=O)(=O)N2C3COCC2CN(C(C2CCC(=O)N2)=O)C3)cc1 56683,C(=O)(CC(C)(F)F)N(CC(CC)NC(c1ccnc(NC(C)=O)c1)=O)C 56684,C(=O)(C(F)(F)C=Cc1ccccc1)N1CC(=C(CNC(C(=O)NC(C)C)=O)F)C1 56685,C(=O)(CCC(C)(C)C#N)NCc1ccc(OC)cc1.C12CC(C13CCC3)C(=O)N2 56686,C(C(C)C)(C(O)C(=O)N1CC2(CC2)CC1CC(=O)NC1CN2CCCC1C2)OC 56687,Fc1ccc(Cl)c(F)c1CNc1ccnc(-c2ccccc2)n1 56688,c1(OC)ccsc1C(N1CCC(C(=O)N(CC(F)F)C(C)C)C1)=O 56689,C(=O)(CC(C)(C)C)NC1CC(C(C(=O)N(C)Cc2cnccn2)F)C1 56690,c1(NC(C2CCCC(O)C2)=O)cccc2c1CN(CC1CCCN1)C2 56691,C1(OC)CN(C(=O)C(O)CN(C)C)CC1C(=O)NC1CC(O)(CSC)C1 56692,c1(OC)ccc(C(=O)NCC(CNC(C2(C)SCCCS2)=O)CO)cc1N 56693,Cc1c(C(N2CCOCC2CCNC(=O)CC(C)N(C)C)=O)cccc1Cl 56694,c12nsc(n1)N1CCC(C1)N(C)C2=O.c1(CC)ccc(CC)s1 56695,C1(C(=O)NCC)CCCN(S(=O)(=O)CC)C1.C1(=O)C(=O)NCCCN1C(C)C 56696,N1(C(C(C)OCCN(C)C)=O)CC2=C(C1)CN(C(c1cc3ccccn3c1)=O)C2 56697,C(=O)(C1CCc2nccn21)NC(c1c(C(=O)NC2CC(OCC)C2)con1)C 56698,C1(C(=O)O)(C(N2CSCC2CO)=O)CC=CC1 56699,C1(NC(C2(NC(CC(C)O)=O)CC(O)C2)=O)CCN(C)C1=O 56700,Cc1c(NC(=O)NCC(C)C(F)CNC(=O)OC(C)(C)C)ccc(F)c1F 56701,CC(C)C(F)(CNC(C1=CC=C(C)CC1)=O)C(=O)NOC1CC1 56702,C=CC1(C=CC(N2CC(CC(C)NC(C3C=C(C)CS3)=O)C2)=O)CCOCC1 56703,c1(N(CC(F)(F)F)C(=O)NC2CC(SC)C2)ccc2c(c1)OCCO2 56704,N1(C(c2cc(COC)on2)=O)CC(CNC(=O)CC(C)(C)OC)OC(C)(C)C1 56705,C1(CC)C(C(=O)NC2(CCO)CN(C(c3cnc(C)nc3)=O)C2)CCN1C 56706,N1(C(C2CN(C(CCCN(C)C)=O)CC2(F)F)=O)CC2(N(C)C)CCC1CC2 56707,c1(C(=O)NCCCC(C)NC(=O)CC2CNC(=O)C2)cc2c[nH]cnc-2n1 56708,CCC(C)(C)C(=O)N1CCC(C(C)CNC(=O)Cc2csnc2C)CC1 56709,N#Cc1cc(Cl)cnc1N1CCCC(NC(C2CC(O)C2)=O)CC1 56710,C1(NC(Cc2c(C)nc[nH]2)=O)CN(C(C2(CCO)CC2)=O)CCC1F 56711,Cc1cc(CNC(c2cnn(CCNC(=O)C(O)C(C)(C)C)c2)=O)cnc1F 56712,N1(C(c2c(Cl)cc(C)s2)=O)CC(C)CCC1CNC(c1ccc(F)s1)=O 56713,CCC(C)(C)C(=O)N(CC(O)CN(C)C(=O)C1CC1)C.C123CC(C1)(C2)CC(=O)N3 56714,C(Cc1cc[nH]n1)(C(=O)NCC1CC1c1ccsc1C)NC(C(=O)NCC)=O 56715,C=CCC(C)C(=O)NC1CCN(C(c2cn(-c3ccc(N)cc3)nn2)=O)CC1 56716,C(=O)(C(C)(O)C(C)C)NCC1CC(F)(CNC(c2cc(C)no2)=O)C1 56717,c1(NC(CC2CC(NC(Cc3ccc(C)cc3Br)=O)C2)=O)ccc(C#N)c(Cl)c1 56718,N1(C(c2nc(C(C)C)sc2)=O)CC(NC(=O)C2=CCSC2)C2(CCC2)C1 56719,C1(NC(c2cc(CNC(CC(C)C)=O)[nH]n2)=O)CCCC1(C)C 56720,N1(C(C2(C(F)F)CCNC2)=O)CCC(F)(CC(F)(F)F)C1 56721,C(CC)(CC)(CCNC(c1cccc(Cl)c1F)=O)NC(C(CC)n1ccnc1)=O 56722,N1(C(c2oc(CCC)c(Br)c2)=O)CCC(C)(C)C(CNC(C)=O)C1 56723,c1(NC(CC(CC2CC2)NC(C(CC)n2ccnc2)=O)=O)cnc(Cl)nc1C 56724,C1(OC)CN(C(=O)CC2CCOCC2)C(C)(CNC(=O)Cn2cnnc2O)C1 56725,C(C(C1CCCCC1)NC(=O)CCF)(C(C)C)NC(c1ccc(SC)s1)=O 56726,C=CCC(C)(CC)C(=O)NC1CN(C(=O)CC2(O)CCOCC2)CC2(CC2)C1 56727,N#Cc1ccc(C(CF)NCCCc2nnco2)cc1 56728,c1(NC(c2nc(C3CCC3)cs2)C)[nH]c(=NCC2CC(CO)C2)nc2c1ncn2C 56729,n1(CC)cc(C(=O)NC2CCCC2NC(C2(C(C)C)COC2)=O)c(C2CC2)n1 56730,c1(C(C(=O)OC)C)cn(CCCOCCNC(c2cnn(CCN(C)C)c2)=O)nn1 56731,c1(CC)[nH]ccc1C(=O)NCC(=O)NCC(F)Cl 56732,c1(N2CC3CC(NC(c4ccc(OC)nn4)=O)C3C2)ncnc2[nH]ccc12 56733,c1(C(=O)NC2C(OC)CN(C(=O)C(CO)N(C)C)C2)cc2cc(Cl)ccc2n1C 56734,n1(CC)ccnc1CN1CCCCC1.C12CCCC1C(C)(C)NC(=O)N2 56735,c1(COC)ccc(NC(C2CN(C(=O)CCc3ccc(F)nc3)CCS2)=O)cc1 56736,c1(NC(CCC2N(CC(=O)OC)CCC2)=O)cnc(Oc2ncncc2Cl)c(Cl)c1 56737,N1(C(CCCOCC)=O)CCCC(CN(C(=O)C(n2cc(Cl)cn2)C)C)C1 56738,N1(C(C(C)O)=O)CCCC(C2CN(C(C3CCc4n[nH]cc4C3)=O)C2)C1 56739,c1(N2CCCCC(NC(=O)CCCCc3cnn[nH]3)C2)nc(Cl)nc2[nH]ccc12 56740,C1(CCC)C(=O)NCCN1CCNC(c1ccncn1)=O 56741,C1(CCOC)(NC(=O)CC(C)(C)C2CC2)CCN(C(C2(CSC)CCOC2)=O)C1 56742,N(C(=NCc1ccc(O)c(O)c1)N1CCC(CC(N)=O)C1)CC(=C)OC 56743,Cc1cc(NC(C2CC2c2cccc(F)c2)=O)nc(C(C)S(C)(=O)=O)n1 56744,C12(CNC(C(C(C)O)C)=O)CC(NC(c3ccc(CN(C)C)cc3)=O)(C1)C(C)O2 56745,C1(C(=O)NC2C(CC(=O)NC(CCCCC)C3CC3)C(O)C2)CC2(CCC2O)C1 56746,N1(C(COCC(N)=O)=O)CCC(CCCNC(c2cccc(CCO)c2)=O)CC1 56747,c1(C(=O)NC(CN(C(COCCC=C)=O)C)(C)C)cc2ccccc2nc1O 56748,Cc1cc(C(=O)NCC2CC(F)(CNC(C3CC3C)=O)C2)ccn1 56749,c1(OC)ccc(C(N2CC3CC3C2C(N2CCCC2CC(C)C)=O)=O)cc1Cl 56750,N1(C(C2(C)CCCCC2(F)F)=O)CCn2nnc(-c3ccccc3)c2C1 56751,CC1COCCN1CCNC(=O)C(=O)NCC1CC12CC(O)C2 56752,CP(C)(=O)C(O)C(=O)N1CCC(CCCCCNC(C2CCCC(=O)O2)=O)CC1 56753,NS(=O)(=O)CCCC(=O)N1CCN(C(=O)CCCN2CCCCC2)C2CC12 56754,c1(OC)cc(C(C)NC(c2ccc(N)cc2Cl)=O)ccc1OCC(n1cncn1)C 56755,c1(OC)c(F)cc(C(=O)NC2CCC2NC(=O)CC2CC(C)(C)CO2)c(N)c1F 56756,N1(C(C2(C3CC3)CN(C(C(C3CC3)SC)=O)C2)=O)CC(C2=NOCC2)C1 56757,CC12CN(C(=O)Cn3cncn3)CC1CN(C(c1c(F)ccc(Cl)c1F)=O)C2 56758,c1(OC)c(NC2CN(C(C3C4Cc5ccccc5C34)=O)C2)nc(O)nc1O 56759,C1(=CC(=O)NC2CC(NC(Cc3ccn(C(C)C)n3)=O)C2)CN2CCC1CC2 56760,C1(C(N2C(C3CCN(C(c4ccc[n+]([O-])c4)=O)C3)CCC2)=O)OC2CCC1CC2 56761,C(=O)(C(F)(F)C(F)F)N1CCC(CNC(c2ccsc2)=O)CC1 56762,c1(C(=O)NC(CC)CNC(=O)CN(CC)CC)cc(F)ccc1C(F)(F)F 56763,C#CCC(CCCO)NC(C1CCCCC1CNC(C1CC2(C1)CC21CC1)=O)=O 56764,c1(CC(=O)NCCCN(C(C2C(SC)CCC2)=O)C)ncn2c1COCC2 56765,c1(C(N(CC(C)NC(CCNC(CC)=O)=O)C)=O)n[nH]c(O)n1 56766,C(=O)(CCC(=O)NC1C2CC1N(C(=O)C(C1CCCCCC1)C)C2)NCCC 56767,C1(C(=O)NCC(CNC(=O)CC2(NC(C)=O)CCC2)OC)CC(C)CC(C)(C)C1 56768,c1(OC)ccc(C(=O)C(=O)ON2CCC(N3CCCC3)C2)cc1 56769,CCCC(C)(C)CC(=O)NCC(C1CC1)N(C)C(c1cnoc1CC)=O 56770,c1(NC(C2(NC(CC3CC(=C)C3)=O)CC(F)C2)=O)ccc(F)cc1C 56771,CN1CCN(C(=O)CCCC2CCCC2)C(CNC(c2nscc2N)=O)C1 56772,C=CCC(CNC(=O)CCC(=O)NC(C)CC)C(=O)N(C(C)CC)C 56773,c1(NC(N(CCC)Cc2cccnc2)=O)nn(C)c(Cl)c1I 56774,N1(C(C2CCN(C)S2(=O)=O)=O)C2CCC1CN(C(C1CC(CCO)C1)=O)C2 56775,Cn1cc(Cl)c(CC(=O)NC2CC(C(=O)Nc3cnccc3C(N)=O)C2)n1 56776,C1(NC(C2CC(SC)C2)=O)CCCC(NC(=O)CC2CCCCO2)C1 56777,CC(C)C1=NOC(C(=O)N(C)CCOCCNC(=O)Cn2cc(Br)cn2)C1 56778,Cc1cc(NCCC(=O)NC(Cn2cc(C(C)(O)CCO)nn2)CC(C)C)c(C)s1 56779,CC1CCC=C1C(=O)NCCn1ccc(C(=O)N(C)CC2CC(F)(F)C2)c1 56780,c1(CNC(C2C(CC)CCO2)=O)cnn(C)c1C(=O)NCCC(O)C1CCCC1 56781,C1(C(=O)OC(C)=O)CC12CCOC2.CON(C)C(=O)C1C2(CC2)CN1 56782,N1(C(c2ncnc(C)c2C)=O)CC2CCCC1C2CNC(c1ccc(F)nc1)=O 56783,c1(C(N2CC3N(C(C(C)OC)=O)C3C2)=O)noc2ccccc12 56784,CC1(C)CCC(C(N2CCCC(CNc3ccccn3)C2)=O)C1 56785,C(=O)(CCCCCCCBr)NC1C(C(=O)Nc2c(C(=O)OC)cccn2)CCC1 56786,C(C)(C)(C(C)CC(=O)OCC1CNC2CCC1C2)c1cc(OC)c(F)cc1 56787,C1(CNC(c2ccnn2CC2CC2)=O)CN(C(=O)CCCc2cc[nH]n2)CCO1 56788,CC(O)CCCNC(=O)CC1CCCC1NC(=O)Cc1ccsn1 56789,c1(C(N2CCC(CO)C2)=O)cnc2ccc(-c3ccc(Cl)cc3)cn12 56790,N1(C(C(CC)(C)C)=O)CCCC2(CCN(C(C)C(=O)NC(C)(C)C)C2)C1 56791,c1(CNC(C(N)=O)CO)cccc(OCC(F)F)n1 56792,c1(C(=O)NC(CNC(CSCC(=O)OC)=O)CO)ccc2c(c1)CCCS2 56793,C(=O)(C(O)CC(C)C)N1CCCC(CN(C(C2CN(C(C)C)C2)=O)CC)C1 56794,c1(Nc2cccc(N3CCN(CC(=O)OC)CC3)c2)ccc(F)c(OC)c1F 56795,C1(C(=O)Nc2c(C(=O)OCC)ccs2)C(C)CCN1C(=O)Cn1cc(CO)nn1 56796,c1(CCC)cc(C#N)c(N(C)CC2CCC(C)O2)s1.C12CCN(C1)C2=O 56797,N(C1CN(C(C2CC(C)OC2C)=O)Cc2ccccc21)C(CCS(=O)(=O)NC)=O 56798,c1(C(N2CCCC(CCNC(CC(C)CF)=O)C2)=O)ccc2occc2n1 56799,C1(C2(NC(N(CC(C)Cn3ccnc3)CC)=O)CC2)CCCCO1 56800,Cc1cc(C(N)=O)ccc1NC(C)(C)C.c12cn(C)nc1NC2 56801,C1(NC(c2c(OC(C)C)n[nH]c2)=O)CCN(C(c2n[nH]cc2Cl)=O)C12CC2 56802,C(=O)(C(C)C(C)COC)N1CC(N(CC(COC)(F)F)Cc2ccc(OC)nc2)C1 56803,C(=O)(C(O)C(C)(C)CC)NCC(=O)NC(C1CC(Sc2cc(O)ncn2)C1)CC 56804,C1(CC=C)N(c2ncnc(NCCC(O)C(C)C)c2C)CCCC1(C)C 56805,Cn1ncc2nc(Cl)nc(N3CCCC3(C)CNC(C3CCCS3(=O)=O)=O)c12 56806,C1(NC(c2cc(CNC(C3C(CCC)CCC3)=O)[nH]n2)=O)CCC(O)C(O)C1 56807,C(=O)(C(C)C(C)(C)C)NCC1N(C(CCCc2c(C)ccs2)=O)CCCC1 56808,c1(OCC)cccc2c1OCC(C(=O)NCC1C3CN(C(=O)CCOC)CC13)C2 56809,CC1CCN(C(=O)C(F)CC2CCC2)CCN1C(c1cnc(N)c(Cl)c1)=O 56810,c1(C(=O)NC(C)CCN(C)C(C2(CO)CCOC2)=O)cc(Cl)ccc1N 56811,C(=O)(C#CC1CCCCC1)N1CCC(N(C)C(c2ccc3sncc3c2)=O)C1 56812,C1(Cc2nnc(N3C(C)C(C)CCC3)n2Cc2cccs2)CCC2CCCCC2C1 56813,N1(C(C2(NC(C3CC(CC)(CC)C3)=O)CC(CO)C2)=O)CC2CCCCC12C 56814,c1(C(CNC(CCCC)=O)NC(c2[nH]cnc2C)=O)ccc(Cl)cc1 56815,N1(C(C2C(CNC(C(CC)C(F)(F)F)=O)C2)=O)CCC2(CCOC2)CC1 56816,C(=O)(CCCCCN(C)C(C)C)NC1(CCNC(C(CC)C)=O)CCC1 56817,CCC(CC(=O)N1CCCC1CCNC(=O)C=C1CCC1)SC 56818,C#CCC(CO)NC(c1n[nH]cc1CNC(c1c[nH]cc1C(C)C)=O)=O 56819,C1(C(C)(C)NC(C=CCOC)=O)CCCN1C(=O)C(n1nccc1C)C 56820,N1(C(CCOCC(C)C)=O)CCC(NC(C2(C)CC(O)CN2C)=O)C(F)C1 56821,C1(C(=O)NCC2(SCC)CC2)CNC(=O)CN1C(=O)C=CC1CCCN1C 56822,C(=O)(CS(=O)(=O)CC(=O)N1CCN(C(C)=O)C(C)C1)OC 56823,C(=O)(C#CC(C)(C)C)N1CCC(NC(c2n(C)nc(C3CC3)c2)=O)(CO)C1 56824,C1(CNC(=O)COC2CCC2)CC2(CO1)CN(C(C1CCC(=O)O1)=O)C2 56825,C(=O)(C(C)S(N)(=O)=O)NCC1(C(C)NC(C2CC3CC2CC3O)=O)CC1 56826,CN=c1[nH]cc(C(N2CC(O)CC2C(=O)NCC2C=CCOC2)=O)o1 56827,C1(NC(=O)C2CC2)CN(C(C2CC2C(F)F)=O)CCC1(F)F 56828,C1(C(=O)NC2CN(C(CCC(=O)OC)=O)CC23CC3)CCC2(CC1)CNC(=O)C2 56829,C(=O)(CCCCC(=O)N1CCC(C)C(NC(c2ccc(Cl)o2)=O)C1)NCC 56830,C1(CCNC(C(C2CCCO2)C2(CC(=O)OCC)CC2)=O)OCCCC1(C)C 56831,N1(C(C)=O)CCCC1C(N1CSCC1C(N1CC(N(C)CCOC)C1)=O)=O 56832,Cc1ccc(S(=O)(=O)N2CCCC(NC(c3c(C(C)C)cccc3F)=O)C2)cc1C 56833,CCC(O)C(C)(C)C(=O)NCCOC1CN(C(=O)COc2ccc(Cl)nc2)C1 56834,C(=O)(C1CCCC2(C#N)CC(C2)N1C)NCC.OCC 56835,Cc1nc(C2CCCO2)sc1C(=O)NC1COCC1NC(c1ccccc1O)=O 56836,N1(C(=O)OC)CCCC(C(=O)NCC2CC(NC(=O)Cn3ncnn3)C2)C1 56837,c1(CC)cc(Cl)ccc1NC(=O)CCC1CNC(=O)N1 56838,C1(NC(C2CCN(C(C(C)OCCC=C)=O)C2)=O)CCC(SC)CC1 56839,C1(O)(CNC(C(C)C2CC2)=O)CC2CCC(C1)N2C(c1cnc(S)nc1)=O 56840,N1(CC(=O)NCc2oc3ccc(C)nc3c2)CCCC2(CC1)CNC(=O)C2 56841,N#Cc1cc(S(=O)(=O)N2Cc3c[nH]c(=N)nc3C2)ccc1NCC1C2CCCC12 56842,C1(C)(NC(C2C(=C)C2)=O)CCN(C(c2ncccc2C(F)(F)F)=O)CC1 56843,C1(NC(=O)Cn2cc(Br)cn2)C2CC3CN(C(=O)C=Cc4ccsc4)C1C3C2 56844,CC1Oc2ccc(CN=c3ccn4nccc4[nH]3)cc2NC1=O 56845,N1(C(C(C)NS(C)(=O)=O)=O)CC2CC1CN2C(C1CC(C)(C)CN1C)=O 56846,C1(C(=O)NC2C(C=C)CN(C(C3(CO)CCCC3)=O)C2)CCCC(C)(C)CC1 56847,C1(NC(C(C)C2CC2)=O)CCC2(CC1)CN(C(=O)Cc1csc(S)n1)CCO2 56848,Cc1cccc(C)c1CC(N1CCC(CO)C(NC(c2cccc[n+]2[O-])=O)C1)=O 56849,N1(C(C(C(CC)C)O)=O)CCN(C(=O)CCCNC(N)=O)C2(CCC2)C1 56850,N1(C(CCCOCC)=O)CCCCC1.c1(CCC(=O)NC(C)C)ccc(Cl)cc1 56851,N1(C(C(C)C2CCC2)=O)CCOCC1C(=O)NCC(N)=O 56852,C1(NC(CCCC)=O)CCCN(C(=O)C=CCOCC(F)(F)F)C1 56853,C1(C)(CC(=O)NC(CC=C)CNC(=O)Cc2cccnc2Br)NC(=O)NC1=O 56854,C12(CNC(C(C)(C)F)=O)CN(C(c3ccc(OC(F)F)cc3F)=O)CC1CCO2 56855,c1(C(C(=O)NC2CC(CCNC(C3(C(C)C)CCC3)=O)C2)C)ccccc1 56856,n1(CC(=O)NC2CCCN(C(C3N(CC)CCC3)=O)C2C)ncc2cccnc12 56857,C(c1ccc(C2OCCO2)cc1)=CC(N1CCNCC1C1CCCCC1)=O 56858,N1(CC)CCN(c2cc(Cl)ncn2)CC1.C1(NC(=O)OC)CCN(C(C)=O)C1 56859,N1(C(CP(C)(C)=O)=O)CCC2(CCCC2NC(c2[nH]nc3ncccc23)=O)C1 56860,CCCC(C(=O)N1CCC(C)C1)NCc1ccc(Br)cc1 56861,c12ncc(cn1)[nH]c2=O.C1(CC)(NC(=O)COC(C)C)CC(F)(F)C1 56862,CC(C)C(CNC(=O)CCC1CCCCO1)NC(=O)CCCN(C)C 56863,C1(C(NOCC(CC)C)=O)CCCN1C(=O)C(C)OCCCN(C)C 56864,c1(OC)cccnc1-c1cn(C2(C(=O)OC)CN(CCCc3csnc3C)C2)nn1 56865,N1(CCSS(C)(=O)=O)CCCN(C(C2(C(=O)CC3CCC3)CC2)=O)CCC1 56866,O=C1CCOC(C(N2CCCC2C2(O)CN(C(=O)C=CC=CCO)C2)=O)C1 56867,C1(NC(CCN(C(=O)COc2ccc(CC)cc2)CC=C)=O)CCCN(CC)C1 56868,C1(C(=O)NC2CC(CCC)C2)CNCCC(O)C1 56869,N1(C(C2(CCC=C)CN(C(=O)C(O)C(C)C)C2)=O)CC(C)(C)C1COC 56870,N1(C(C=C(C)C)=O)CCN2CCN(C(=O)CCc3ccccn3)CC2C1 56871,CC1(CNC(=O)CCC2CNC(=O)N2)CCCN1C(=O)C=CC(F)(F)F 56872,c1(C(=O)NCC2N(C(C(COC)C)=O)CC2)nc(-c2nc[nH]n2)sc1C(C)C 56873,CC(C)C#CC(=O)N(CCCCNC(=O)CC(C)C1CCCO1)CCO 56874,c1(CC)nncn1NC(=O)C1CC(NC(c2cc(CC)on2)=O)C12CCCC2 56875,C1(C(N2CC(NC(c3cccc(C)n3)=O)C3C(C2)C3)=O)CN2CCCN1CC2 56876,c1(N2CCCC(CN(C(C3(OC)CCCC3)=O)C)C2)ccc(C#N)cc1[N+](=O)[O-] 56877,Cc1ncc(Br)c(N2CCC3(CC3C(=O)Nc3cccc(C)c3I)C2)n1 56878,C1(=O)CCCCC(=O)NC2CN1CC2C.c1(CC)cccc(NC(C2CC2)=O)c1 56879,Cc1nscc1C(N1CC=CC1CNC(c1cc(C(C)(C)C)n[nH]1)=O)=O 56880,C1(OC)CN(C(=O)CC2(C)CCOCC2)CC1C(=O)NCC1(SC)CCOCC1 56881,c1(C(N(CCCN(C(CSC2C(C)CCC2)=O)C)C)=O)cccc(C(F)(F)F)c1 56882,C1(C(=O)NC2C(C(=O)OC)CCC2)CCCCN1C(=O)Cc1ccoc1 56883,C(CCC1CCC1)(C(=O)NC(C)(C)C(C)(C)C)NC(C(=CC1CCCC1)C)=O 56884,C1(C(=O)NCCC(COC)(C)C)CCC(C)(C)N(C(c2csnc2C)=O)C1 56885,c1(NC(N(c2cc(C)cc(F)c2)C2CCNCCC2C)=O)cnc2ccccc2c1 56886,C1(COC)(NC(=O)CCC2CCCO2)CCCN(C(c2ncc(N)nc2C)=O)C1 56887,CC1=C(C(=O)NC(CNC(C2(C)CCC(C)=C(C)C2)=O)CC(F)(F)F)CCO1 56888,Cc1nnc(O)c(C(=O)NCC(O)CN(C(=O)Cc2cn3ccsc3n2)C)c1C 56889,CC1(C)CC(CNC(=O)CNC(=O)C(C)(C)C)N(C(C2SCCCS2)=O)C1 56890,c1(CCC(N2C(C)(C(=O)NC(CCC)C)CC2)=O)c[nH]c2c(C)cccc12 56891,CC1CCN(C(c2cccc(SC(F)(F)F)c2)=O)CCN1CC1CCCC(=O)N1 56892,c1(CCC(=O)N(CCNC(=O)Cc2cc[nH]c2)CC)c(F)cccc1F 56893,C(=O)(CC(C)(C)C#N)NC1CCN(C(C)CNC(=O)CN2CCCCC2)CC1 56894,N1(C(C2CC(C#C)(O)C2)=O)CCC(C)C(NC(C2CC(O)C(F)C2)=O)C1 56895,CC(c1ccccc1)=CC(N1CC(C)(OCC(=O)NCC2CC(C)CO2)C1)=O 56896,N1(C(C(C)(C)C2CCCO2)=O)CCC2C(C1)CN2C(c1cnn(C(F)F)c1)=O 56897,c1(N(CC(N2C(CNC(C(C)SC)=O)CC2)=O)C)ccccc1[N+](=O)[O-] 56898,CC(C)C(C(C)NC(=O)Cn1cnccc1=O)NC(=O)CCn1cnccc1=O 56899,CN1CCN(C(=O)CC2(C#N)CCCCC2)CC1CNC(c1cnc[nH]1)=O 56900,CC1CCC(O)(CNC(c2ccc(CNC(=O)CC3CC3(C)C)nc2)=O)C1 56901,C(=O)(C(C)(C)C(=O)N1CCC(C(C)C(=O)NCC(C)(O)CC(=O)OC)CC1)OC 56902,c1(N(C2CC3(C2)CC(N)C3)C(c2ccc(C)c(Cl)c2)=O)ncc2ccsc2n1 56903,N1(C(C2CN(C(=O)NC)C2)=O)CC2C(CNC(c3ccncc3O)=O)C2C1 56904,c1(C(=O)OC)[nH]c2cc(NC(c3ccc(I)c(Cl)c3)=O)ccc2c1-c1nn[nH]n1 56905,c1(C(C)C)nnnn1CCCC(=O)N1CC(O)(CNC(C2C(C)(C)C2(F)F)=O)C1 56906,Cc1[nH]c2ccccc2c1C(=O)NC(C)CN(C(=O)CC1CC(F)C1)C 56907,C1(C)(C(=O)NCC(CNC(c2ccc(CC)nc2)=O)O)CC(C(C)C)=NO1 56908,C(=O)(C1CCCn2cncc21)Nc1c(OC)cccc1 56909,Cc1ccc(C(=O)NC2CCN(C(=O)Cc3nc(=N)[nH][nH]3)C(C)C2)cc1CO 56910,CC(C(C)(C)C(=O)NC1CCN(C2CC2)C1=O)NC(=O)C1=COCC1 56911,Cc1cc2[nH]c(C(N3CCCC(CCNC(c4ccccn4)=O)C3)=O)cc2o1 56912,C(CCCCNC(=O)Cc1cncnc1)NC(c1cnn(C(F)F)c1)=O 56913,C1(NC(C(C2(O)CCCCC2)CC)=O)CCN(c2cc(C(F)F)ncn2)CC1O 56914,c1(C(N2CCC(OCc3cc(C)ns3)C2)=O)ccc(CN2CCCCC2)cc1 56915,CCCC(CC)CC(=O)N(C1CCN(C(C23CCC(N=[N+]=[N-])C2C3)=O)CC1)CC 56916,c1(CNC(C(CCC)(C)CC)=O)cccc2c1CN(C(C1CC1(C)CC)=O)C2 56917,c1(CCCC(=O)NCCN(C(C2C(C=C)C2)=O)C)ccccc1Br 56918,Cc1nn(C)c(Br)c1C(N1CCCC(N(C(=O)CCOC2CC2)CCO)C1)=O 56919,C(=O)(CCCC(C)(F)F)CNC(C1(C(=O)NCc2cccc(COC)c2)CC1)=O 56920,C1(NC(C2CC(=O)NC2)=O)C2CC1CN(C(C1CCN(C(N)=O)CC1)=O)C2 56921,C(C)(CCN(C(=O)C(F)n1cccn1)CC)NC(COC(CC)C)=O 56922,c1(CC)cc(C(=O)NC(CNC(=O)CN2CCCC2=O)CC)ccc1C 56923,C(=O)(CS(=O)(=O)CC(=O)OC(C)(C)C)N(CC(C)C(=O)Cc1ccnc2c1CCO2)C 56924,N1(C(COCC(N2CCCC2)C)=O)CCC(O)(NC(=O)CSc2ccccc2)C1 56925,O=C(C1=NOC2(CCC2)C1)NC1CC1CNC(=O)COc1c(Cl)cccc1Cl 56926,C1(NC(CSc2ccc(C)cc2)=O)CN(C(=O)CNc2cnn(C)c2)CCC1F 56927,C1(C)(C(N(CC(C)SC)C)=O)CCCN1C(c1sccc1CO)=O 56928,n1(CC)cnc2c(NC(C)CC(C)C)[nH]c(=NCc3cc(Br)cs3)nc12 56929,CC(C)CCCC(C)NC(C1CC2(C1)CN(C(c1cccc(F)c1O)=O)C2)=O 56930,C1(C(=O)NCCCCNC(c2ccnn2-c2ccncc2)=O)(CC)CC1(F)F 56931,CCCCCCCC(=O)N1C2CCC(C2)C1CNC(C1CCCS(=O)(=O)C1)=O 56932,CCCCCCCCC(C(=O)NC1CCCCC1)N1CC2CSCC(C2)C1 56933,C=C(C)CC(C(=O)N1CCC2(CC2C(=O)NCCCc2ccccn2)C1)OC 56934,C(C(N=c1c(C#N)c[nH]c2ccccc12)C1CCC1)NC(c1cc(OC)no1)=O 56935,c1(C(C(=O)N(CCNC(CCN(C(C)=O)C)=O)C)NC=O)ccccc1F 56936,c1(C(=O)NC(CNC(c2c(COC)cno2)=O)C2CCC2)ccc(Br)c(N)c1 56937,C1(CC(=O)NCC(CNC(c2c(C(=O)OC)csc2)=O)CO)CC=CCN1C 56938,CCC(C(=O)N1CCC(CF)(NC(=O)CCc2ccccc2Cl)C1)C(C)C 56939,c1(NC(=O)NCC(CC)C)ccnc(F)c1 56940,N1(C(C(C)OCc2ccccc2)=O)CCN(C(=O)C(F)C(C)(C)O)CC12CCC2 56941,CCC(CC(=O)NCC(c1nccs1)C)N(C)C(c1cc(C(C)C)on1)=O 56942,CCC(CC)(CO)C(=O)NCC1CCC2CN(C(C3CCCC(F)(F)C3)=O)CC12 56943,N1(C(C2C(=C)C2C(=O)OC)=O)CCCN(C(C2CC2(Cl)Cl)=O)CCC1 56944,Cc1cc(C(=O)NCC(=O)NC2CCC2CNC(=O)C(C)(C)CF)c(C)o1 56945,c1(C(=O)NC2C(CNC(C3CCC(C)O3)=O)CCC2)cnc2ccccn12 56946,c1(C(=O)NC(C(C)(C)NC(C(C)NC(C)=O)=O)C)c[nH]c2ccc(F)cc2c1=O 56947,C1(CNC)CCCN(C(C2C(C(=O)O)C2(C)C)=O)C1 56948,C(=O)(CC1=NNC(=O)C1)NCC1CN(C(c2cc(C)nc(Cl)c2)=O)C(C)C1 56949,C1(C(N(CC(C)O)C2CC2)=O)CCN(C(C2CC2C2(C)COC2)=O)C(C)C1 56950,C(C(C)S(C)(=O)=O)(c1n(CC=C)nnn1)NC1C(OCC)CC1C(=O)OCC 56951,C(=O)(C(C)S(C)(=O)=O)NC(CCNC(c1cccc(-c2nc(C)on2)c1)=O)C(C)C 56952,C1(NC(C2C(CC)CCCC2)=O)CCN(C(=O)C(=O)NCC(F)(F)F)CC(O)C1 56953,N1(C(C(CCC)F)=O)CCC(C)CC1CNC(c1ccc(OC)nn1)=O 56954,N1(C(C(C)SC(C)C)=O)CCCC2(CNC(c3ccc([N+](=O)[O-])o3)=O)CC12 56955,N1(C(CCCC)=O)CCC12CN(C(C1(C)CCOCC1)=O)C2 56956,c1(OC)c(Cl)cc(NC(=O)NC(C)CNC23CC(CCO2)C3)cc1Cl 56957,CS(=O)(=O)C(C(=O)NCCCOCCNC(=O)C(c1cccnc1)O)C1CC1 56958,C(N=c1cc(NCC2CC3CCC3C2)nc[nH]1)C1(COC)CCC1 56959,n1(CCC(=O)NCC2N(C(C(C)C(C)(C)C)=O)CCCC2)cnc2ccccc12 56960,CCC(C)CCC(=O)NC(Cn1cncn1)C(=O)NC1CC(C#N)C1 56961,N(C(=NCCC(=O)N1CCCCC1)NCc1cnco1)CC(CC)(CC)OC 56962,c1(CC)cccc(C(N2C(C(=O)NCC3(F)CCCCC3)CC3CC23)=O)n1 56963,C12(C(=O)NCC(CN(C(C(CC)n3cncn3)=O)C)O)CC(CN1C1CC1)C2 56964,C(=O)(CC(C)(C)CNC(C)=O)N1CC(OCC)CC1C 56965,C1(NC(C(C(CC)C)CC(=O)O)=O)CCc2nc(-c3ccccc3)ncc2C1 56966,n1(CC(=O)NC(C)CCNC(=O)CC2CCC23CCC3)nc2ccccn2c1=O 56967,Cc1cc(C(=O)NCC(CC(C)C)NC(c2cc3sccc3[nH]2)=O)nc(C)n1 56968,Cc1n[nH]c(C)c1OCC(=O)NCC1(F)CCC(NC(c2ccnc(O)c2)=O)C1 56969,CCCCC(O)C(C)C(=O)NC(C)CN(C)C(c1ncc[nH]c1=O)=O 56970,C1(CC)CN(C(c2ccccc2C(=O)N(C)C)=O)CCC1Nc1cc(O)ncn1 56971,n1(C(C(=O)NC(CNC(c2c(CC)n[nH]c2)=O)CC)CC)cnc(C#N)n1 56972,C(=O)(C(C#N)CC)N(CC(=O)NC(C=C)(C)CC)CCC 56973,CC1CC=C(C(=O)N2CC(CC=O)CC2(C)C)CC1.N1CCN(CCO)CC1 56974,C1(C(=O)OC(C)(C)C)CCC2(CO1)CC(NC(C1CC1(Cl)Cl)=O)C2 56975,Cc1[nH]nc2c1CC(C(N1CC(C(N)=O)(CNC(C3COC(=O)N3)=O)C1)=O)CC2 56976,N1(C(C(C)NC(c2cnccn2)=O)=O)CC2(CC(NC(c3cc[nH]n3)=O)CO2)C1 56977,Cn1nc(C(=O)NCCCCCC(=O)NCCCc2cscn2)cc1C#N 56978,c1(CC(=O)N(CCCNC(C2ON=C(CC)C2)=O)CC)c[nH]c2cccc(C)c12 56979,C12(CCCCC1)C(c1nnnn1CCSC)N2.N1(CC)CCCOC1 56980,c1(C(=O)NCC2(CN(C)C(C3(C)CC3)=O)CC2)cc(C#N)ccc1Cl 56981,Cc1cnccc1C(=O)NC1CCCCC1NC(=O)CN1CCCCC1=O 56982,N1(C(C2(OC)CCCOC2)=O)CCC(NC(=O)CCn2nc(C)nc2C)C(O)C1 56983,Cc1cc(C(=O)NC2CC(CNC(=O)COC3CCC3)C23CCC3)c(N)c(F)c1 56984,c1(C(=O)OC)cnn(C2CN(C(CC(c3ccccc3)C)=O)C2)c1C(F)(F)F 56985,N1(C(CC2CCCC(OC)C2)=O)C2CCC1CC(CNC(c1ccc(Cl)s1)=O)C2 56986,O=C(N=c1[nH]nc(C2CC2)s1)C1CCCN(C(c2nc(Cl)sc2Br)=O)C1 56987,CN1CCC(CNC(=O)C(O)O)(CNC(=O)CC23CCC(CC2)C3)C1 56988,C1(C)(COC)CCCN(C(C2CCN(C(c3cc(C)c(C)[nH]3)=O)CC2)=O)C1 56989,N1(C(CNC(C2C(C(C)C)OCCC2)=O)=O)CC2(C1)CN(Cc1ccccc1)C2 56990,Cc1cccc2c1OCC2C(=O)NCCOC(C)(C)CNC(C1CC1C(C)(C)C)=O 56991,C1(C(=O)NC(CC)CNC(c2coc(OCC(F)(F)F)n2)=O)(CC)CCOC1 56992,C12(C(=O)NC(CNC(c3nc(COC)sc3)=O)CC)C3C4C1C1C2C3C41C 56993,Cc1cc(OCC(=O)NC2COC3(C2)CN(C(c2nc[nH]n2)=O)C3)cc(C)c1F 56994,CCC(CC)C(C)C(=O)N1CCCCC1CCCNC(=O)C=CCN1CCC1 56995,C(CN(C)C)(C(=O)NC(CC(=O)N1CCOCC1)C1CCCC1)NC(CCC)=O 56996,N1(C(c2c(CC)nc(N)s2)=O)CC(C)N(C(=O)Cc2cc(C3CC3)n[nH]2)CC1C 56997,C1(CNC(c2cccc(C3CC3)c2)=O)C2CCC(C2)N1C(=O)CC1(O)CCC1 56998,Cc1cc2cc(C(N3CCC(CN(C)C)C3C)C(=O)NCC3CC3)oc2cc1C 56999,CCC(C)C(=O)C(=O)NCCc1cc(C(N2CCCCC2C(N)=O)=O)no1 57000,C(=O)(CCCCN1CCCCC1)N(CCNC(=O)CCOCC1CC1)C1CC1 57001,c1(C(N(C(C)CC(=O)NCCCCC2CC2C)C)=O)cc(F)ccc1F 57002,C(CCC(C(=O)N1CCC(CC(=O)OC)C1)NC(C1CCOCC1C)=O)OC 57003,c1(C(N(CC(C)NC(c2nc(OC)sn2)=O)C(C)C)=O)c(Cl)oc2ccccc12 57004,N(C(=S)N1CCCC1c1ccc(Cl)nc1)C(C)COC(F)(F)F 57005,c1(C(N(CCCN(C(C(C)C(C)C(C)(C)C)=O)C)C)=O)cc([N+](=O)[O-])ccc1Cl 57006,C1(OC)CN(C(=O)CC2C=CCN2C(=O)C=Cc2cnn(C)c2)CC12CC2 57007,CC(C)C(F)C(=O)NCC(C1CCN(c2nccnc2F)CC1)(C)C 57008,c1(C(=O)NC2C(NC(CCC)=O)C2)cccc(N)n1 57009,c1(C(=O)NCCN(C(COCCCC#C)=O)C(C)C)csc(-c2cccnc2)n1 57010,c1(C(=O)OCC)cccc(C(N2CC(OCCOCCOC)C(C)C2)=O)c1 57011,C1(C(N2CCC(CC=C)(NC(=O)CCCOC)C2)=O)OC(C)(C)OC1(C)C 57012,CCC(C)CC(C)C(=O)N1CC2CC(C1)N2C(C1OCCC1(C)C)=O 57013,CC(C)C(C(=O)N1CCC(F)(F)CC1)C(C)NC(c1nc(=N)cc[nH]1)=O 57014,N1(C(CNC(c2cn(CC)nn2)=O)=O)CCCN(C(C2CCS(=O)(=O)C2)=O)CC1 57015,c1(CC(=O)NC2(CNC(=O)CC3COCCO3)CCOC2)ccccc1O 57016,Cc1n[nH]c(C)c1CCC(=O)NC1CC1CNC(c1c(C2CCC2)cnn1C)=O 57017,C1(NC(CCOCC#C)=O)CCCN(C(c2cc(N)nc(Cl)c2)=O)C1C 57018,c1(OC)ccc(C2(C(=O)N(C(C)CCNC(=O)COC3CCC3)C)CC2)cc1F 57019,c1(C(=O)NC2CN(C(C(C(C)(C)C)(C)O)=O)C2)ccc2nc(S)[nH]c2c1 57020,CC1=C(C(=O)NCC2CC(NC(c3ccc(Cl)c(Cl)c3)=O)C2)CCCC1 57021,c1(CC=CCNC(=O)Cn2ccnc2)ccccc1Br.N12CCC(C1)C2 57022,C1(NC(c2c(SC)cccc2)=O)CC2(CCCCN2C(=O)Cc2cccn2C)C1 57023,N1(C(C2CN(C(C)C)C2)=O)CCCC(O)(CNC(c2cnc(C(F)F)s2)=O)C1 57024,c1(CC(=O)NC(C(C)C)C(=O)NCc2ccn(C(C)C)n2)cnc2[nH]ccc2c1 57025,CCCCC(C(=O)NCC1CN(C(=O)C(=CC2CCCC2)C)C(C)(C)C1)N(C)C 57026,c1(CNC(COC)=O)oc2ccccc2c1CNC(=O)CCC(C)(C)F 57027,C12(C(=O)NCC3CC(C)N(C(c4ccnc(O)c4)=O)C3)CCCC1CCC2 57028,c1(C(c2n(CCC)nnn2)NCCOc2cccc(C)c2)cc(Cl)c(Br)cn1 57029,N(C1COc2cc(Cl)ccc21)C(=O)Nc1cc(C2CC2)ccc1Cl 57030,C1(CNC(CCC=CC(C)C)=O)CC2CCC1N2C(c1ccnn1CCF)=O 57031,C(=O)(C(C)C(=O)NC1CCCCCC1C(N1CCCC(CO)C1C)=O)OC 57032,c1(CNC(c2n(CC)nnn2)CCCC2CC2)ccc(F)cc1Br 57033,c1(-c2c(CC)cccn2)c(C(N2CCNC(=O)CC2)=O)nn2c1CCCC2 57034,c1(C(=O)OCC)cn2cc(NC(c3ccc4sc(C)nc4c3)=O)cccc1-2 57035,C1(CC)CCCCCCN1C(c1nnn(C)n1)C(=O)Nc1cc(Br)ccc1OC 57036,C1(C(=O)NCC(C)N(C)C(c2csnc2Cl)=O)CCCCC12CCC2 57037,C1(C(=O)NC2CC2C(F)(F)F)C2CN(CCNC(C3CCCCC3)=O)CC12 57038,C1(C(=O)N(CCCNC(C2CCCN2CCC(C)C)=O)C2CC2)(OC)CCSC1 57039,CC1(C(=O)NCCC2(NC(=O)Cc3cccc(C(F)F)c3)CCC2)CCCCCC1 57040,N1(C(C2(CO)CC(C)(C)C2)=O)CCC2(CC1)CC2CNC(C1COC1)=O 57041,C12(C(=O)NC(CC)CNC(=O)CC(C3CC3)C3CC3)COC(C(F)(F)F)(C1)C2 57042,C(C(CC(=O)NCC(C1CCCCC1)O)NC(=O)C(C(C)C)SC)OC 57043,C1(NC(=O)Cc2c[nH]nc2O)C2CCN(C(c3n[nH]c(C4CC4)c3Br)=O)C12 57044,c1(NC(CCN(C(=O)CCOC2COC2)C)=O)cncc(C(F)F)c1 57045,C(=O)(C(F)CC(C)(C)NC(c1ccc(O)c(F)c1)=O)NCC1CC(=C)C1 57046,C1(F)(CNC(C(=O)NCC)=O)CCC(NC(=O)C=C(C)Cl)C1 57047,N1(C(c2cc(CC)c(F)cc2)=O)CC(C)N(C(=O)CC(F)(F)CC)CC1C 57048,N1(C(CC=CC=C)=O)CCN(C(C2CCC(C(C)C)N2C)=O)C(CO)C1 57049,C(=O)(C(CCc1ccccc1F)N1CC(O)(C(Cl)(Cl)Cl)C1)NC(CC)C 57050,C=C(C)C(C)(O)C(=O)NC1CCC(NC(c2ccc(COC(C)C)cc2)=O)CC1 57051,C1(NC(=O)COC2CCOC2)CC2CC(C1)N(C(C1C=CC=CC=C1)=O)C2 57052,C1(C(N2CCCC(CNC(C(C)C3CCCO3)=O)C2)=O)CCCCC12OCCO2 57053,C1(OC)(CNC(=O)COCCC(=O)NC)CCN(C(=O)CS(=O)(=O)C2CC2)CC1 57054,C1(CCC(=O)Nc2cn(CC(=O)NC)nc2)CCN(C(C2CCC(=O)CC2)=O)CC1 57055,c1(C(=O)NCC(N(C)C(C2(C)C=CCC2)=O)C2CC2)cc2n(n1)CC1(CC1)C2 57056,C(=O)(C(C)(C)S(C)(=O)=O)N1CC(O)(CN(C)C(C2CCC3(CCOC3)O2)=O)C1 57057,N1(C(C(CCCCC)O)=O)CC2(CCCCN2C(C23CC(C)(C2)OC3(C)C)=O)C1 57058,c1(CC)nnc(N2CCC(CN3CCCCC3)CC2)n1Cc1ccccc1 57059,C1(F)(CNC(=O)C(=O)NC2CC2)CCCN(C(=O)C=Cc2ccccc2)CC1 57060,N1(C(c2ccc(CNC(CC(C)C3CCCO3)=O)s2)=O)CCC(C2(C)CC2)CC1 57061,c1(C(=O)NCC2N(C(COCC)=O)CC(C(F)(F)F)OC2)ccc2occ(C)c2c1 57062,C=CC1COCCN1C(C1CC(C)N1C(c1nocc1C(C)C)=O)=O 57063,Cc1cc(Br)c(C(=O)Nc2ccc(C)c(C(F)(F)F)c2)cc1Cl 57064,C1(C(=O)NCCCNC(C2SC3C=CC2C3)=O)C2CC3C(C2=O)C13.C1CN1 57065,c1(NC(C23CC2CN(Cc2cnn(C4CC4)c2)C3)=O)cc(F)ccn1 57066,Cc1ccc(O)cc1NC(C1CN(C)CC1C)=O.C1(CC2CC2)CC(=O)N1 57067,c1(C(N2CCC(N(C(=O)CCC3(C)N=N3)C)CC2)C)cccc(C#N)c1 57068,C(=O)(C1CCc2ccccc21)NC1CCC(NC(=O)Cc2cc(C3CC3)on2)C1 57069,CCC(C)(CNC(=O)COc1cnn(CC)c1)NC(=O)CC1C=CCC1.OCC 57070,c1(C(N(CCC(C)NC(=O)Cc2c(F)cccc2Cl)C)=O)cccc2ncnn12 57071,CC1(C)CN(C(=O)CNC(N)=O)C(CNC(C2SCCS2)=O)CO1 57072,C1(O)(C(C)NC(=O)Cc2cnns2)CCN(C(c2cc(-c3ccoc3)[nH]n2)=O)C1 57073,C1(S(C)(=O)=O)(C(=O)NCC(CC)(C)NC(C2CCN(C)C2C)=O)CCC1 57074,C1(C(=O)NC(C(C)C)c2cn[nH]c2)CCC2CCC1N2C(=O)C(c1cnn(C)c1)=O 57075,Cc1ccc(C(N)=O)cc1NC(c1cocc1Br)c1nnnn1C.CC(F)(F)F 57076,C(=O)(CCC(C)(C)C)N1CC(O)(C(C)NC(COCCC#C)=O)C1 57077,c1(OCCC)ccccc1CNC(=O)C(=O)NCC1CCCN1CC 57078,N1(C(c2ccc(Cl)c(Cl)c2)=O)CCC2(CC1)CN(C(c1ccc[nH]1)=O)C2 57079,c1(C(=O)NCC(C)CNC(=O)CC2CC23CC3)c[nH]c(C(N)=O)c1 57080,C1(N(C(=O)CC2CCC2(C)C)CC)CCCN(C(c2cccnc2S)=O)C1 57081,C1(N(C(C(C)OCC)=O)C)CCC(NC(c2ccc(=O)oc2)=O)CC1 57082,C(CS(=O)(=O)CCO)NC(c1cc(C(F)(F)F)n(C)n1)C 57083,C1(CN(C(=O)COC2CCN(C)CC2)C)CCCN(C(C2CCC(CO)CC2)=O)C1 57084,c1(N(C(CC)CC)C(c2nnnn2CC2CCOC2)C2CCC2)cccc(Br)c1 57085,C(=O)(CCCCCCNC(=O)C(=O)C(F)(F)F)NC(C)=O 57086,CCC(F)(C(=O)OC)C(=O)N1CC2CC(NC(c3cccc(F)c3SC)=O)C1C2 57087,N1(C(Cc2c(C)n[nH]c2)=O)CCC2(CCN(C(=O)CNC(C3CC3C)=O)CC2)C1 57088,N1(C(C(C)NC(CC)=O)=O)Cc2[nH]nc(C(N3Cc4c[nH]c(=N)nc4C3)=O)c2C1 57089,C1(C(N(CCOc2ccccc2C)CC)=O)CCCN(Cc2cnoc2C)C1 57090,C1(C(=O)NC2(CCNC(CCC3C(C)(C)C3)=O)CCC2)CC(=O)N(O)C1 57091,N1(Cc2ccc(C(=O)OC)s2)CCCN(C(=O)Cn2c(Cl)cccc2=O)CC1C 57092,C(c1c(Cl)cccc1Cl)=CC(=O)NC(CC=C)CNC(C1(n2ccnn2)CC1)=O 57093,C(CCC(=O)NCCC1(SCC)CC1)NC(C1CC1(F)Cl)=O 57094,c1(NC(C2(CNC(COC(CC)(C)C)=O)CCC2)=O)cc[nH]c(=N)c1 57095,C1(CN(C)C(C2C3CCCCC23)=O)CCCCN1C(=O)CCC1CCOCC1 57096,N1(C(C(CNC(C2C(OCC)CC2)=O)C(C)C)=O)CCCN(C)CC1CC 57097,Cc1c(F)ccc(N)c1C(=O)NCC1(NC(=O)C(c2cccnc2)C)CC1 57098,CC1CN(C(C23COCC2C3)=O)CC2(CCN(C(c3cnc(O)c(F)c3)=O)C2)O1 57099,C1(CC(=O)NC2C(CC)N(C(C3CNC(=O)C3)=O)CC2)CCC2(CC1)OCCO2 57100,CC(C)CCC(O)C(=O)N1CCC2(CC2)CC1C=O.CCN(C)C1CC1 57101,c1(C)cc(C(=O)N(C)CCOCC)n[nH]1.N12CC(OC)(C1)C1C(=C)C1C2=O.OC 57102,c1(C(CNC(=O)Cn2cncn2)NC(c2cc(F)ccn2)=O)ccc(F)cc1 57103,N1(Cc2ccc(OCC)c(OC)c2)CCN(C(=O)Nc2ccnn2C)CC1(C)C 57104,CC1CC2CN(C(=O)CCc3cccc(C(N)=O)c3)CC2N1C(=O)COC(F)F 57105,C=C(F)C1(CC(=O)NC(C)CCNC(c2cc(C)cs2)=O)CCC1 57106,CC(C)C(C(=O)N1CC(O)(CNC(=O)CN2CCNC(=O)C2)C1)NC(=O)C1CC1 57107,Cc1cnc(Cl)c(C(=O)N(C)CC2CCCN2C(=O)C(=O)C2CCCC2)c1 57108,c1(Nc2n(C)cc(NC(c3ccc(C)c(C)c3)=O)n2)ccc2oncc2c1 57109,C(=O)(CC1=CCCCC1)N(C1CN(C(c2cc(S(N)(=O)=O)cs2)=O)CC1O)C 57110,C1(NC(C(C)(C)OCC)=O)CN(C(=O)CCCCCNC(=O)COC)C2CC12 57111,C(=O)(CCN(OC)C(=O)C1CCC(=O)O1)Nc1c(OC)cccc1 57112,c1(NCc2ccc(C)o2)cccc(C(=O)Nc2sccc2Cl)c1 57113,C(C(C)C(F)C(=O)N(C)CC1CC(F)(F)C1)NC(Cn1nnc(C)n1)=O 57114,CCCCC(CNC(C1CCN(C(=O)CCCOC(C)=O)C1C(C)C)=O)CC 57115,Cc1cccc(C(N2CC(O)(C(F)C(=O)N(CC(O)C3CCC3)C)C2)=O)c1F 57116,N12CCC3(CC1)CC3C2=O.C1(=CC(=O)NCC(C)(C)C2CCCO2)CCSCC1 57117,N1(C(c2c(C)cc(Cl)cc2)=O)CCC2C(CCCN2c2ncnc3c(C)csc23)C1 57118,C1(C(N2CCN(C(C3C=CC=CC=C3)=O)CC2)=O)(CC)CCC(F)(F)CC1 57119,CCCCC(C(=O)NCC1(C)CCCOC1)NC(=O)C(C)(C)C(=O)NC 57120,c1(CC(=O)NCC2N(C(CSCC#C)=O)CCN(C)C2)cccc2c1OCCO2 57121,c1(OCC)cncnc1N(C(C)CNC(=O)CCC1CC(OC)C1)C 57122,C=CCC(CC)C(=O)NCCC1(NC(=O)Cc2csc(-c3ccoc3)n2)CC1 57123,C1(NC(C=Cc2scc(C)n2)=O)CC(C)CN(C(C2CC2C(=O)OC)=O)C1 57124,C(CC(O)CNC(c1cn(C2CCOC2)nn1)=O)NC(c1csc(Cl)c1)=O 57125,Cc1scc(C(=O)NC2CC3C(NC(=O)Cc4nccn4C)C3C2)c1C 57126,N#CC1CCC(CC(=O)NCc2nocc2C(=O)NCC2CCOCC2)C1 57127,n1(CC(=O)NCCN(C(C23CCC(CC2)CO3)=O)CC)nc2n(c1=O)CCOC2 57128,C(c1cn(C)c(=O)n(C)c1=O)=CC(N1CC(NC(c2c(C)ccs2)=O)C(C)C1)=O 57129,c1(CC(C)NC(=O)NCCCC(C)c2ccccc2)cccc(F)c1 57130,C(N=c1[nH]c(=NCC23CCCCC2C3)c2ccccc2[nH]1)C1(c2cnccc2)CC1 57131,c1(C(=O)OC(c2ccccc2F)C)cc2n(c1)CCS(=O)(=O)C2 57132,CC(C)(CNC(C1CCC2(CCC2)C1)=O)CC(=O)NC(C(C)(C)CO)C1CC1 57133,N1(C(C2C(=C)CC2)=O)CC2CCN(C(c3cccc(Cl)c3Br)=O)CC12 57134,CC(C(=O)N1CC(N(C)C(c2coc(C3CCC3)n2)=O)C(C)(C)C1)S(C)(=O)=O 57135,Cc1nc2scc(-c3ccccc3)c2c(=O)n1CCC1(C(F)F)CCNC1 57136,c1(C(=O)NCC2CCCN(C(CS(CC)=O)=O)C2)cc2c(C)cccc2o1 57137,C(=O)(C(C)S(N)(=O)=O)NC(CC(C)C)CNC(C1(COCC(F)(F)F)CC1)=O 57138,O=C(CN=c1cc[nH]cc1)NC1(C(=O)NCCCC2CCOC2)CC(CO)C1 57139,C1(NC(=O)C(CO)c2ccccc2)CCCCCN(C(c2cc(Cl)ccn2)=O)C1 57140,C1(C(=O)NCC2(CNC(c3ccnnc3Cl)=O)CCCC2)CCC=CCCC1 57141,CC(C)(C)C(O)CC(=O)N1CC(NC(=O)COC2CCCC2)C(O)C1 57142,c1(C(N2CCC(CC)C2)=O)cccc(CN(c2cn(C)cn2)C)c1 57143,C(=O)(C1CCc2nccn21)N(C)C.C12(O)CCN(C1)C(=O)c1ccc(cc1)CS2 57144,c1(C(N2CC(CNC(=O)Cc3cnccc3Cl)C3C2C3)=O)cc2n(n1)CCC2 57145,c1(C(C)C)occc1C(=O)NC(c1ccccc1)C(N1CC(N(C)C(C)C)C1)=O 57146,N1(C(CCC(C)C)=O)CC2(CC(NC(=O)CC3CCOCC3(C)C)CO2)C1 57147,N1(C(C(F)=CC)=O)CCC2(CC1)CC(C)N(C(C1CC13CC3)=O)C2 57148,c1(C(=O)NC2CCC(NC(CN3CC(CC)C3)=O)C2)ccc2[nH]c(=N)sc2c1 57149,C1(C)(CNC(c2cc(COC)[nH]n2)=O)CCN(C(c2snnc2C)=O)C1 57150,Cc1cc(C(=O)NCC(C)(F)CNC(=O)Cn2nnnc2C(C)C)ns1 57151,C1(OC)CCC12CC(C(=O)N(CCCCNC(C1(C(C)C)CC1)=O)C)C2 57152,N1(C(C(c2ccccc2)OCC)=O)CCCCC12CC(NC(C1C=CCC1)=O)C2 57153,c1(CNC(C(Cn2cncn2)NC(c2cnc(Cl)s2)=O)=O)cncnc1O 57154,N1(C(C(C)NC(=O)NC)=O)CC(CNC(=O)C=C2CCN(C)C2)C(C)C1 57155,c1(CNC(CC2(CSC)CC2)=O)cn(C)nc1C.c12ccoc1CNC2=O 57156,Cc1cc(NC(C2CSCCN2Cc2ccc(Br)cc2O)=O)c(C)cc1Br 57157,N1(CC2CC2)CCCN(C)CCC1.N1(C(c2ccc(SC)cc2)C)CCOCCC1 57158,C1(CCC)CN(C(c2ccc[n+]([O-])c2)=O)CC1C(N1CCC(COC)C1)=O 57159,C=CC1(C(=O)NCCOCCCN(C(=O)CCS(C)=O)C)CCOCC1 57160,Cc1c(C(=O)NCC(O)CN(C)C(C2CCCN2C=O)=O)cnn1CCN(C)C 57161,CC#CCC(C(=O)N(CCC(=O)OCC)C)NC(=O)CCc1cn[nH]c1 57162,c1(CC(N2CCC(C)C(NC(c3ccncc3)=O)C2)=O)ccc2cccnc2c1 57163,N1(C(CCCN(C(C)=O)C)=O)CCCC2(CNC(=O)Cc3cccc(Cl)c3)CC12 57164,C12(CCCC1)C(=O)NC1C(C1)C(=O)NCC2.C(C)(C(=O)NC)OCC#C 57165,c1(C(=O)OCc2ccc(SC)c(Br)c2)c(F)cc(OC(F)F)cc1F 57166,c1(C(N(C)CC2CCCCO2)=O)coc2c1CN(C(=O)C(F)=CC1CC1)C2 57167,N1(C(C2CCC(C(N)=O)O2)=O)CCCC2(CCN(C(c3cccnc3F)=O)C2)C1 57168,C(=O)(CCCC(C)(C)C)NC1CC2(CC(NC(C(C)c3ccon3)=O)C2)C1 57169,C1(C)(C(=O)NC(C(C)O)CO)CCCN(C(=O)CCC2CC2)C1 57170,c1(C(N)=O)ccnc(C(=O)NC2CCCC2CNC(=O)CS(=O)(=O)N(C)C)c1 57171,C1(C(N2CC(CCOC)C2)=O)C2CCC(C2)N1C(C1CC2C(C1)C2(F)F)=O 57172,c1(N(C)C)cncc(C(N2CC3CC2(CNC(=O)C=CC=CCO)C3)=O)c1 57173,c1(CC)sc(=N)[nH]c1C(=O)NCCN(C)C(c1cncc(C(F)F)c1)=O 57174,CC12CN(C(=O)COC(F)F)CC1CN(C(=O)Cn1cnc3c(N)ncnc13)C2 57175,c1(C(N2CC(C(C)NC(C3(CO)CCOCC3)=O)C2)=O)cccc2c1NCCC2 57176,C1(CNC(COCCCC(C)C)=O)CCN(C(=O)C(c2cncn2C)=O)C12CCC2 57177,CC(C(=O)NCCC1CN(C(c2cnc[nH]c2=N)=O)CCO1)C(C)(F)F 57178,C=C1CC2(C1)CC(C(=O)N(C1CCN(C(=O)CC3(C)OCCO3)CC1C)C)C2 57179,C1(CC)CNC(=O)CN1C(=O)C(O)CNC(C1COCOC1)=O 57180,c1(NC(=O)CC2CN(Cc3cc(O)ncc3Br)CCO2)ncnc2occc12 57181,CCC(CC(=O)NC(C)CCCNCC=Cc1ccc[nH]1)C1CCC1 57182,c1(C(=O)NC(CCN(C(C(CCC)CC)=O)C)C)ccc([N+](=O)[O-])cc1CC 57183,N1(C(c2c(C)noc2Cl)=O)CCCC(C2(NC(=O)C(F)(F)C(O)C3CC3)CC2)C1 57184,CCCCCCC(=O)NC(C1CCN(C(C2CC2(Cl)C(=O)OC)=O)CC1)C 57185,C1(NC(=O)CCc2cscn2)COC2(CCN(C(c3ccns3)=O)CC2)C1 57186,C(C1CCC(C)CC1)=C(C(N1CCC(N(C(C2CCN(C)C2=O)=O)CC)C1)=O)C 57187,C1(C(N2CC(N3C(=O)CC(OC)C3)C2)=O)COc2cc(OC)ccc2C1 57188,C(=O)(CS(=O)(=O)C1CC1)N(CC(c1ccc(C)cc1)F)CCNC(=O)CC(C)C 57189,C(=O)(C(C)(CC)C(N)=O)NC1(COC)CN(C(c2ccc(Cl)cc2OC)=O)C1 57190,c1(C(N(CCCCCNC(c2n(CC)ncn2)=O)C(C)C)=O)occ2c1CCC2 57191,N1(C(CSC)=O)C2CCC1CN(C(C1CCOC(C(C)C)C1)=O)C2 57192,C1(C(=O)OC)N(C(=O)C=CCNC(=O)CC2CCOC2(C)C)CC1(C)C 57193,N1(C(CC(C(C)C)NC(=O)Cn2cncn2)=O)CCN(C)CC(C)C1 57194,CN(C)NC(=O)CCC(=O)NC(C(=O)Nc1ccccc1C1CC1)C1CCCO1 57195,C1(=O)C(C(C)(C)C)N1.C(=O)(C(=O)NC(C1CCC1N)C)NC 57196,C1(CNC(C(c2cnn(C3CC3)n2)N(CCCCC)C)=O)CCOC(C)C1 57197,C1(NC(C2(n3cnnn3)CC2)=O)CCN(C(c2cc(Cl)cs2)=O)C12CC2 57198,c1(CCCNc2c(C)nsc2CC2CC(F)(F)C2)cccc(F)c1Br 57199,N1(C(c2c(-c3cn(C)nc3)cco2)=O)CC(NC(=O)COC2CCOC2)CC1CO 57200,N1(C(CCc2cnc(C)s2)=O)CCCC(CNC(C2CC2(F)F)=O)CC1 57201,c1(CC(=O)NCC2CC(C(=O)NC(c3ccns3)C)C2)ccc(Cl)cc1 57202,C(=O)(C1=Cc2cc(Cl)ccc2OC1)N1CC(NC(c2ccc(C)[nH]2)=O)C(C)(C)C1 57203,C1(c2nnnn2C)(NC(CCC(=O)OCC)c2ccccc2)CCCC(C=C)C1 57204,CC1CCC(NC(C2CNC(=O)C2)=O)C1 57205,N1(C(C2COCCN(C(CCC(CC)=O)=O)C2)=O)CCCC(C2CCC2)C1 57206,c1(C(=O)NCC2CCCN2C(=O)CCC2CCCCO2)ccc(SC2CCC2)o1 57207,C1(n2cnnn2)(C(=O)NCCN(C(=O)CCn2cnnn2)CCC)CCOCC1 57208,C(CCCC(=O)NCC1CC(CCO)C1)N(C(CSCC#C)=O)C 57209,Cn1[nH]c(=NC(=O)CC2(C)NC(=O)NC2=O)c2c1OCCC2 57210,Nc1ncccc1C(N1CCC(N(C(=O)CC2CS(=O)(=O)C2)CCO)CC1)=O 57211,c1(-n2cc(CN3CCNCC3)nn2)cc(F)cc(Cl)c1.O=C1CCC2(CC2)CC1 57212,C(=O)(CC(C)(C)C1CC1CN)NCCCN(C(c1cn(C2CCOC2)nn1)=O)CC 57213,C1(F)(C(=O)NCC(CC)(CC)OC)CCCN(C(c2ccc(C)o2)=O)C1 57214,C1(CC(=O)NCCCC(N2CC(O)(CN(C)C)C2)=O)CC2CCC(C1)C2 57215,c1(-c2nc(CCOCC)nn2C)cccc2nc(C(=O)NCCOC3CC3)cn12 57216,Cc1cnn(C)c1CC(=O)NCC(C)(C)CC(=O)N1CC(OCCC2CC2)C1 57217,C1(C(=O)N(CCO)CCN(C)C)CC(=O)N(C(c2n[nH]cc2[N+](=O)[O-])=O)C(=O)C1 57218,C(c1cc(Br)ccc1OC)=NCC1=CCN(Cc2ccc(CCCC)cc2)CC1 57219,n1(C2CC(CC(C(=O)Nc3nn(CCOC)c(=O)cc3)F)C2)cc([N+](=O)[O-])cn1 57220,C1(S(=O)(=O)NC(N2CCC(N(CC(C3CCCCC3)(C)O)C)CC2)=O)(CC)CC1 57221,n1(CC(=O)NCC(C)NC(c2sccc2-n2cnnn2)=O)cc(C(F)(F)F)nn1 57222,c1(N2C(CNC(c3ccc([N+](=O)[O-])s3)=O)CCCC2)ccc2nnnn2n1 57223,C1(OC(F)F)(CNc2cc(C)c(Nc3cccc(Br)c3)cc2)CCCN(C)CC1 57224,c1(NC(C2CN(C(C(OC)OC)=O)CC2O)=O)cn(C2CCCC2)c(=O)nc1O 57225,N1(C(C(N2CCC3(OCC(CC)C3N)CC2)=O)=O)CCc2ccc(Cl)cc2C1C 57226,C(=O)(CC1=NN(CC(C)(C)C)S(=O)C1)OCC.CCCC(C)CCN 57227,C1(C(=O)NCCCCNC(Cn2cc(C(C)=O)nn2)=O)CC12CCSCC2 57228,N1(C(C(C(C)C)C2CCC2)=O)CCCCC(C(=O)NOCCC(F)F)C1 57229,C(CCCC(=O)NC1CCC1(C)C)NC(C1(OC)CC1)=O 57230,O(NC(=O)C(CNC(=O)CNC=O)CC(C)C)CCC 57231,N1(C(C2CNC(=O)N2)=O)CCN(C(=O)CC2COCCOC2)CC1 57232,c1(NC(C(N)=O)=O)cncc(C(=O)NCCN2CC3CCC2C3)c1 57233,C=CCC(CNC(c1ccc(CC(C)C)s1)=O)NC(c1csc(C(F)F)n1)=O 57234,c1(C(N2CC(C(=O)NC(c3ccccc3)CO)(SC)C2)=O)cn2ccccc2n1 57235,N1(C(C)C)CCN(C)C(c2ncc[nH]2)C1.N12CCCC1CCCC2=O 57236,c1(C(=O)NC2C(NC(CC(=C)C)=O)CCC2)cn2cc(Br)cc(C)c2n1 57237,C(c1ccc(F)cc1)=C(C)C(=O)N(CCCNC(c1ccc(CN=[N+]=[N-])o1)=O)C 57238,C1(C(=O)NC(C(C)C)CN)CCCN(Cc2ccc(C(C)C)cc2)C1 57239,CS(=O)(=NCC(=O)NCCn1cc(CCS(C)(=O)=O)nn1)c1ccc(Cl)cc1 57240,N1(C(CCN(C(C2CCC(=O)CC2)=O)C2CC2)=O)CC2(CCC2)CC1CO 57241,c1(OCCNC(c2cnsn2)C)ccccc1F 57242,c1(C(=O)NC(CC)CNC(c2ccc(-c3ncc[nH]3)cc2)=O)cc(=N)[nH]c(Cl)n1 57243,CC1CC2(CO1)CN(C(=O)CCC1CCN(C(C3(F)CCCCC3)=O)C1)C2 57244,Cc1ccc(NNC(=O)c2ccc(OC(c3cnc(Br)s3)=O)cc2)nn1 57245,N1(CC)CCCN(c2cc(NCc3cccc(COC(C)C)c3)nc(C)n2)CC1 57246,N1(C(CC2(C)CCN(C(COC)=O)C2)=O)CC2CCC(C1)N2CC1CCOC1 57247,c1(C(=O)NCC(C)(C)NC(CC(C)C2CC2)=O)n[nH]c(C(C)C)c1[N+](=O)[O-] 57248,c1(OC(CC)C)ccc(C(=O)OC2(c3ccccc3)CC2)cc1 57249,c1(CNC(CCNC(C2C(OC)CCC2)=O)=O)csc(C)c1C 57250,c1(CC)cc(C(=O)NC2(CN(C(=O)Cn3cncn3)C3CC3)CCC2)cc(N)c1 57251,C(=O)(CC1=CCOCC1)N1C(C(=O)NCc2c(CC)nn(C)c2)CC(F)CC1 57252,CC1(C)CCCN(C(=O)Cc2nnc(O)s2)C1CNC(c1cnc(Cl)s1)=O 57253,c1(OC)ccc(C(C)C(=O)N(C(C)CCNC(=O)C(C)(F)F)C)c(C)c1 57254,C1(C(N2CCC(N(CCCOC)CC3CC3)CC2)=O)CCn2cncc2C1 57255,N1(C(c2ccc(C)c(C)n2)=O)Cc2n[nH]cc2C1C(=O)N1CCC(C)(C2CC2)C1 57256,CN1CCC(CC(C(=O)O)NC(C2CCCC2CN)=O)CC1 57257,C1(C(=O)NC2CC(CCOC)C2)CC2CCC1N2C(=O)Cc1cncnc1 57258,C1(C(=O)O)(NC(CC2(COC)CCOC2)=O)CCCC2CC12 57259,N1(C(C2CC(C(=O)OC)C2)=O)CC2CCC2(CCNC(c2n[nH]c(C)c2F)=O)C1 57260,C(=O)(CS(=O)(=O)C1CC1)N(CCCCCNC(c1ncn2c1CCC2)=O)C 57261,c1(NC(C2CCCN2C(c2cc(Br)cc(I)c2)=O)=O)cc(F)c(Cl)cc1I 57262,CC1=C(C(=O)NC2CCCC2NC(=O)CC2CC=CCN2C)CCC1 57263,Nc1ccc(C(=O)NCC2(O)CN(C(C3C4C5CCC(C5)C34)=O)C2)c(O)c1Cl 57264,C1(N(C(c2c(C)c(O)ccc2)=O)CC2CCCS2)C(C)OCC12CCNCC2 57265,S(=O)(=O)(c1ccc2c(c1)N(C(=O)Nc1ccc(S(C)=O)cc1)CCC2)N(C)C 57266,c1(C(=O)NC(C)CNC(C2CCCCCCC2)=O)cccc(S(=O)(=O)CCO)c1 57267,N1(c2nnc(CC)s2)C2CCC1C(CNC(=O)CCCOc1ccc(OC)cc1)C2 57268,c1(CNC(C(C)NC(c2cc(F)ccc2F)=O)=O)nccc2ccccc12 57269,CC(C)C(C(=O)NCC1(CNC(c2cc(C#N)cs2)=O)CC12CCC2)N(C)C 57270,C(=O)(C1OCCc2c(O)cccc21)NCCNC(C12CC3CC1C2C3)=O 57271,C1(C#CC(=O)NCc2ccc(C(=O)NC(C)CCOC)nc2)(CC)COC1 57272,c1(CC(=O)NCC(O)CNC(c2nocc2Br)=O)cccnc1F 57273,c1(OCC(=O)NCC2CCN(C(CC(CC)(C)C)=O)C2)cc2cccnc2nc1O 57274,C1(C(N(CCN(C(c2cc(OC)ncc2)=O)C(C)C)C)=O)CCCCC12CCC2 57275,Cc1cc(CC(=O)NC2CC(CCNC(=O)C=CCO)C2)cc(C)c1 57276,c1(CCC(=O)NCC(CN(C(C(CSC)OC)=O)C)(C)C)cccc(Cl)c1Cl 57277,CC1OC(C)C(C(N2CCN(C(=O)CC3(C)CC3(Cl)Cl)C(CCO)C2)=O)C1C 57278,COn1cnc(C)c1C(=O)NC1COCCN(C(=O)CCCC(C)C)C1 57279,c1(C(=O)NC(C)CNC(c2ccc(C(F)F)cn2)=O)cc2cccnc2nc1N 57280,N1(CCC)CCCCC1C(N1CCC(CF)(NC(c2nc(O)sc2C)=O)C1)=O 57281,C(=O)(CC(C)CC(=O)OC)NCC(CC)(C)NC(=O)CN(C)C(C)C 57282,N1(C(c2cc(CCCCC)[nH]n2)=O)CCCC(NC(C2(C)CCOCC2)=O)C1 57283,N1(C(C2C(COC)C2)=O)CCC(C(C)(C)NC(=O)C(=CC2CCCC2)C)C1 57284,CC(F)(F)C(C)(C)CC(=O)NCC12CC(CN1C(=O)Cc1ccccc1O)C2 57285,NS(=O)(=O)c1ccc(C(N2CCC(F)C(NC(=O)CCc3cscn3)C2)=O)nc1 57286,C(=O)(C(F)(F)C(F)(F)F)N(C(C)C(N1CCCC1C1(OC(N)=O)CC1)=O)C1CCCC1 57287,C(CS(=O)(=O)CC(=O)NCC(C1CCCCN1C(=O)C(F)C1CCC1)(C)C)OC 57288,CC(CCCCl)NCC1(C(F)(F)F)CCCO1 57289,C1(CNC(c2ccc(COC)[nH]2)=O)CCN(C(=O)COCC2CCCO2)C12CC2 57290,C1(C(=O)NCC(C(N2CCC(NC(CC)=O)C2)=O)N(C)C)CCC2(CCC2)O1 57291,c1(C(=O)NC2C3CN(C(C(C)(C)CO)=O)CC2C3)csc2c(F)cccc12 57292,N1(C(C2(CCC=C)CN(C(=O)CC3CC(=O)C3)C2)=O)CCC(C)(O)CC1 57293,O=C1CCC(CCC(N2CCCC2C2(NC(c3ccncn3)=O)CC2)=O)CN1 57294,N12CC3CC3(C1)C2=O.Cc1nscc1CNC(=O)C(C)N1CC(C)C1 57295,c1(C(=O)NCC2CC(NC(C3C(=C)C3)=O)C(O)C2)ccn2c(C)cc(C)nc12 57296,C1(CCNC(c2c(C)con2)=O)CN(C(C2CC2(Cl)Cl)=O)CCO1 57297,N1(C(C(C=C)(C)C)=O)CCC(NC(c2oc(C)nc2C)=O)C(F)(F)CC1 57298,N1(C(CS(C(C)(C)C)(=O)=O)=O)CCC2CCN(C(C3CC4(CC4)C3)=O)CC2C1 57299,N1(C(C(C)(C)OC)=O)CCOCC(NC(C2CN(CC)C(=O)N2)=O)C1 57300,CC1(C)CCCN(C(c2ccccc2N)=O)C1CNC(c1cc(C(N)=O)[nH]n1)=O 57301,N1(C(CCN(C(Cc2cccc(C#C)c2)=O)C2CC2)=O)CCOCC2(CC2)C1 57302,C1(C(=O)NC2(COC)CCN(C(c3c(CC)[nH]nc3Cl)=O)C2)CCCCCN1C 57303,Cc1cc2[nH]nc(C(=O)NCC(C)CNC(c3ccc(C#N)s3)=O)c2cc1C 57304,C(C(C)(O)CC(=O)NCCCCN(C)C(c1c[nH]nc1C(=O)O)=O)OC 57305,Cc1cc(=O)c(C(N2CCC(C(=O)NCC3CC4OC3C3CC43)C23CC3)=O)c[nH]1 57306,c1(-c2ccc(OCC#C)cc2)cccc2sc(CC(=O)N=c3nc(C)[nH]s3)cc12 57307,C(=O)(C(CNC(c1n[nH]c(C)c1O)=O)C(C)(C)C)NC(c1cnccn1)CC 57308,C1(OC)(CNC(C2C3CC3CN2C(C2CC(F)(CF)C2)=O)=O)CCOCC1 57309,n1(CC(=O)NC2CC3CN(C(Cc4nnc(C)o4)=O)C2C3)c(C)cc2ccccc12 57310,CC1CCN(CC(=O)NC2CCCC2NC(=O)COC2CCCOC2)C1 57311,Cc1c(Br)ccc(N2CCN(CC3(NC(=O)CSC(F)F)CC3)CC2)c1[N+](=O)[O-] 57312,Cn1nc(C(N2CC(NC(c3cscc3F)=O)CC(O)C2)=O)c(Cl)c1Cl 57313,C12(C(=O)NCCCNC(=O)CCN3CCOCC3)CC(c3ccccc3)(CO1)C2 57314,CCC(C)CCCC(=O)NCC(CC)(CC)NC(=O)Cc1cc(C2CC2OC)on1 57315,Cc1csc(C(=O)NCCCN(CCCN(C)C)C)c1Cl.c12nc(n[nH]1)NC2 57316,CCC(CNC(=O)C(CC1CCCC1)NC(=O)CN1CCNC(=O)C1)C(C)C 57317,c1(C(N2C(C3(NC(=O)C(F)C4CCC4)CC3)CCCC2)=O)ccc(Br)c(F)c1F 57318,C(CC(=O)N(CC(=O)N(CCCC1CC1)C)C(C)C)SC 57319,N1(C(CN(C(=O)OCC)C)=O)CCC2CC12C(=O)NC(C)Cn1cccn1 57320,C1(NC(CC)=O)CN(C(=O)Cc2csc(Cl)n2)CC1c1cnn(C)c1 57321,c1(CC)nn(C)c(Cl)c1C(=O)NC(CCNC(=O)C(C)(C)NC(C)=O)CC(C)C 57322,N1(CC(N2CC3C(CNC(C45CC(C(=O)OC)(C4)C5)=O)(C3)C2)=O)CCS(=O)(=O)CC1 57323,C1(C(=O)NCCCC)(CN(C)C)CCCN1C(=O)CN1CCN(C)CC1 57324,C1(NC(C2ON=C(C)C2)=O)C2CN(C(C3(NC(C)=O)CCSCC3)=O)CC12 57325,C(C)(CO)(C(=O)NCCN1CC(CF)C1)NC(c1ccc(C(C)C)o1)=O 57326,CC1=CCC=CC1C(N1CC(C)(CNC(C2(C(F)(F)F)COC2)=O)C1)=O 57327,C1(C(N(C)Cc2ccc(Br)cc2)=O)CCCCN(C(C2OCC2(C)C)=O)C1 57328,C1(CC)CN(C(c2cnc(OC)c(F)c2)=O)CCC1NC(=O)CC(=O)OC 57329,N1(C(C(C)OCC#C)=O)CC2CCCN(C(c3cc4c(cn3)OCCC4)=O)C2C1 57330,C(=O)(C(C(C)C)C(C)C)N(C1CCN(C(=O)C(c2cncn2C)O)C1)CCC 57331,c1(CCC(=O)NC(C)Cc2ccccc2)ccc(OC(F)(F)F)cc1 57332,c1(C(=O)NC2CC(NC(C(CC)OCC)=O)C2)ccnc(F)c1N 57333,C1(C(N2CCC(CNC(c3n(C)ccc3)=O)C2)=O)C2CCCOC12 57334,C1(N(C(c2cnc(SC)s2)=O)CC)CCCN(C(c2cc(C#N)on2)=O)C1 57335,C(=O)(C(F)(F)CCn1ccnn1)NCC(C)CN(C)C(c1cc(Cl)no1)=O 57336,Cc1cnsc1C(=O)NC(C1(C(C)C)CC1)C.c12cnn(c1)C(=O)NC2 57337,Cc1nc(C)c(C(=O)NC2(CNC(=O)Cc3cnn(C(C)(C)C)c3)CC2)o1 57338,c1(CN2CC(C(=O)Nc3n(CC)ccc3)OCC2)ccn2ccnc2c1 57339,CC1(C)CN(C(C2CCC(NCc3c[nH]c(Br)c3)C2)=O)CCO1 57340,c1(C(N2CCC(C)(NC(C3C(C)CCCC3)=O)C2)=O)cnc2n1CCS2 57341,c1(C(=O)NCCOCCNC(C2CC(C)(C)O2)=O)ccc(C(F)(F)F)nc1 57342,c1(CC(N2CC(c3cn(CC(CC)O)nn3)(N(C)C)C2)=O)ccc(F)cc1C 57343,C#CCC(C)(CC)C(=O)NCC1(O)CN(C(c2cnn(C)c2F)=O)C1 57344,C(=O)(C(C(CC)=Cc1ccsc1)N1CCC(CC)C1)NCCCCCC 57345,C(C1=C(C)OCCS1)NC(c1n(CCSC)nnn1)(C1CCCOC1)C(=O)OC 57346,N1(C(c2c(C)con2)=O)CCCC(N(C)C(c2ccn(CCC(F)(F)F)n2)=O)C1 57347,N1(C(CN(CCOC)C)=O)CCCC(O)(CNC(=O)CC(C)c2cccnc2)C1 57348,C(=O)(C(CCC1CCC1)NC(=O)CC(C)(C)SC)N(C(COC)COC)C 57349,N12CC3(CC(CO3)C1=O)C2.CC1(C)CCC1NC(=O)CSCC(N)=O 57350,c1(N2CCC(C(=O)OC)(C(=O)OC)C2)ncc(S(C)(=O)=O)cc1Cl 57351,c1(C(N(C)CC2CCN(C(C(CC)SC)=O)C2)=O)cc(O)cc(F)c1 57352,CC1=C(C(=O)N2CCC(C)N(c3ncnc4ccccc34)CC2)CCS1(=O)=O 57353,C1(NC(Cc2c(C)ocn2)=O)CCN(C(C2(C#N)CCCCC2)=O)CC1CO 57354,c1(CC)ccc(Cl)c(-c2cnc(CC(CC)CC)cc2)c1 57355,c1(C(=O)NC2(C)CCN(C(C(COC)(F)F)=O)C2)ccc2nnn(C)c2c1 57356,C(=O)(C(C)CC(=O)NC(CO)C(C)N(CC(C)CCCO)C1CCC(=O)N1C)OC 57357,C1(C(=O)NCC(CCC)OC)CN(C)CCN1C(c1coc(C(F)F)c1)=O 57358,O=C1CCCC(C(=O)NC(C(=O)NCC=Cc2ccccc2)C2CCCO2)C1 57359,N1(C(C=C(C)C)=O)CCC(C(F)(F)F)C(NC(=O)C(C)S(N)(=O)=O)C1 57360,CC1(CNC(C2C3COCC23)=O)COCCN(C(=O)C2=NOC(C(C)(C)C)C2)C1 57361,Cc1cnsc1C(=O)NCCC(O)CNC(C1C=CCC1)=O 57362,C1(N(C(=O)CN(CC(C)(C)C)C)C)CCN(C(C2COC(=O)O2)=O)C1 57363,C(CC(C)CC)(C(=O)NCc1c(C)cccc1F)NC(c1c(CC)cco1)=O 57364,C1(C(=O)NCc2cncnc2)CCC2CCC1N2C(=O)CCNC(C1CCC1)=O 57365,C1(NC(c2nc(C(C)(C)C)oc2)=O)CC2CCCC(C1)N2C(=O)C(F)CC1CC1 57366,C1(C(=O)NCCc2ccc(CC(C)C)cc2)CC2(C1)CC(C#N)C2 57367,C(CCCCCN=[N+]=[N-])NC(C1N(C(=O)Cn2ncccc2=O)CCC(=C)C1)=O 57368,C12(F)CCCN(C1)C2=O.c1(CC(=O)NCC2(C(F)(F)F)CCC2)cnsc1 57369,N1(C(CC(C=C)CC)=O)CCC(C)(C)C(C(=O)NCCc2cnnn2C)C1 57370,N1(C(C(C)OC(C)(C)C)=O)CCC(N(C)C(C2CC=CC2)=O)CC1 57371,c1(C(=O)NCC(=C)CCNC(=O)C=Cc2cnccn2)nncc2c1CCCC2 57372,C1(CC)OCCCC1C(=O)NC1CN(C(c2c(C3CCCC3)noc2C)=O)C1 57373,C1(NCCOc2c(C)cccc2)CCCN(C(C)C(N)=O)CC1 57374,C1(C(=O)NCC2CCN(C(=O)CCN3CCCS3(=O)=O)C2)CNc2ccnn2C1 57375,Cc1cc(C(C)(C)C(N2CC3CC3C2CNC(=O)CC2(C)CC2)=O)ccc1Br 57376,C(=O)(CC(C)CC(=O)N1CC2CC1C2NC(c1cc(C)cs1)=O)OC 57377,C(C)(CNC(=O)COCCC(C)C)(CNC(=O)CCc1nncs1)OC 57378,N1(C(C2C(OC)CCC2)=O)CCC(CC(=O)NCC(C)(C)C(C)O)CC1 57379,c1(C(C(=O)NCCC2CC2)N(C2CCCS(=O)(=O)C2)C)ccn2ncnc2c1 57380,n1(CCC(=O)NCCCNC(C2(C)CC2)=O)ncc(=O)c2ccccc12 57381,N1(C(C(CNC(C2(OC)CC(C)C2)=O)N(C)C)=O)CCc2ccc(C#N)cc21 57382,C1(C(=O)Nc2c(OC)nsc2)CCN(C(=O)COCCN(C)C)C1C 57383,C1(NC(=O)Cc2cscn2)CCC2(CCN(C(=O)C3=CC4(CCOC4)C3)C2)C1 57384,CCC(C)(C)CC(=O)N1CCC(CNC(c2cc(C)c(C(=O)O)s2)=O)C(C)C1 57385,C1(NC(C(Cc2cn(C)nc2)F)=O)COCCN(C(=O)CN2CSCC2=O)C1 57386,c1(C(=O)NCC(CC)(C)C(=O)NCC(n2cccc2)C)cccc2ccnn12 57387,C(=O)(C(C)(C)NC(C)C)N1CC(CN(C(CCOC(C)=O)=O)C)C1 57388,Cc1cc(CC(=O)NC23CC(C2)N(C(=O)CN2CC4CC4C2)C3)cc(F)c1 57389,C(CCNC(=O)CC1CCCN(C(=O)Cc2cc[nH]n2)C1)(C(C)C)OC 57390,C1(COC)(NC(=O)C(n2nccc2C)C)CCN(C(=O)CSS(C)(=O)=O)CC1 57391,C1(CCNC(C2CCCCC2)=O)(OC)CN(C(=O)CNC(c2ccco2)=O)C1 57392,c1(C(=O)NCc2cn(C3CCOC3)cn2)cc(Br)c(Br)cn1 57393,N1(C(C(C(C)C)(C)O)=O)CC(CO)C2(C1)CN(C(=O)Cn1cnc(=N)[nH]1)C2 57394,N1(C(c2sc(C)c(C)c2C)=O)C2CCC1CC(O)(CNC(=O)Cc1ccco1)C2 57395,N1(Cc2ccc(C)c(C)c2)C2CCC1CC(NC(c1ccc(I)cc1)=O)C2 57396,C12(C(=O)NC3(C)CN(C(Cc4ccc(OC)cc4)=O)C3)CCCCC1C2(F)F 57397,CCCCC(C)CCC(=O)NC1CC1NC(c1ccncc1C(=O)OC)=O 57398,c1(CC)sc(C(=O)NC(C)(C)CN(C)C(c2ccccn2)=O)cc1C 57399,C=CC(C)(C)CCNC(C1(OC)CCN(C(=O)COCC(C)(C)C)C1)=O 57400,c1(OCC(=O)N(C(CCNC(C=CCC)=O)C)C)cc(F)cc(F)c1 57401,c1(C(N2C(CNC(Cc3cn(C)nc3)=O)CC2)=O)ccc(OCC(N)=O)cc1 57402,N1(C(c2nc(NC(C)=O)sn2)=O)CC2(CC(NC(C3CCCN3C=O)=O)CO2)C1 57403,C12(NC(c3ccoc3)=O)CN(C(c3cnsn3)=O)CC1CS(=O)(=O)C2 57404,N1(C(C(c2cn(C)nc2)=O)=O)CCN(C(C2CCCOCC2)=O)C(C2CCC2)C1 57405,c1(C(=O)OC)sc(C(=O)N(C2CCN(C(C3(CCF)CC3)=O)C2)C)cc1N 57406,C1(CC(=O)N(C2(CCNC(CC3CC(OC)C3)=O)CCC2)C2CC2)CCN(C)CC1 57407,C1(NC(c2n(CC)nnn2)c2ccn(CC(F)F)n2)Cc2ccc(C#N)cc2C1 57408,N1(C(C(=O)NCC(C(=O)N(C2CC2)CC)C)=O)CCCC(C2CCNCC2)C1 57409,CC(C(=O)N1CCCCC1CCN(C)C(C1(F)CCC1)=O)C(F)F 57410,C=CCC(C)(C)CC(=O)NC(CCN(C)C(C1CCCOC1)=O)C(C)(C)C 57411,c1(C(=O)NC(CC)CNC(=O)C(CC2CC2)OC)cnncc1OCC 57412,N1(C(COCCCCC)=O)CC(CNC(c2c[nH]nc2OC)=O)CC1(C)COC 57413,N1(C(C(C)Sc2nncn2C)=O)CCC2(CC1)CCN(C(c1cocc1Cl)=O)C2 57414,c1(C(N2C(CNC(C3N(CC)CCOC3)=O)CCC2)=O)c(C)nn(C)c1C 57415,c1(OC(F)(F)F)cccc(CN2CCN(Cc3cc(C4CC4)no3)CC2)c1 57416,C(=O)(C(F)(F)C(F)F)NC(CN1CCN(C(C(C)SC(C)C)=O)CC1)(C)C 57417,c1(OC)cc(C)c(CNC2CC(NC(C3(c4cccnc4)CCC3)=O)C2)cn1 57418,c1(Sc2c(C)cncn2)cnc(Br)c2ccccc12 57419,C(C1c2ccsc2CCN1C(C1CC(O)C1)=O)NC(C(P(C)(C)=O)O)=O 57420,Cc1cnc(F)c(C(=O)NCC(C)N(C)C(c2ncsc2C)=O)c1 57421,C(=O)(CCCC(C)(F)F)N1C(CNC(C2CCC(SCC)CC2)=O)C(C)CC1 57422,C12CCN(C1)C(=O)NCC(C)N(C)C2.C1(C(=O)OC)(CC)CCC1 57423,CC(C)C(C)C(C)CC(=O)N1CCOC(CNC(=O)C(C(C)C)NC=O)C1 57424,N1(CCC)CCCCC1C(=O)NCCN(C(=O)CCCCC1CC1)C 57425,c1(CC(COC)C(=O)NCCNC(c2ccc(C)nn2)=O)ccc(F)cc1F 57426,C#CCCC(O)C(=O)N1CCN(C(c2ccc(C(F)(F)F)[nH]2)=O)C(CCO)C1 57427,C1(CC(=O)OCC)CN(C(=O)Cn2nccc2N)CC12CCN(C(=O)C=CCF)CC2 57428,c1(N2CCCC(CNC(C=C(C)C3CC3)=O)C2)nc(C)nc2sc3c(c12)CCC3 57429,C1(SCC(N2CCN(C(CCC)c3ccco3)CC2)=O)C=CS(=O)(=O)C1 57430,C1(C(N2CC(NC(C3(CC=C)CCC3)=O)C2)=O)CC(=O)N(CCC)C1 57431,n1(C(C)C(=O)NC(C)CC(C)NC(C2CC(O)C2)=O)cnc2ccccc12 57432,C(N=c1[nH]c2c(c(=NCc3c(OC)ccc(Cl)c3Cl)[nH]1)CCCC2)C1C(C=C)CC1 57433,C1(NC(C=C2CCC(C)C2)=O)C2CC3CN(C(c4ccc(N)cc4)=O)C1C3C2 57434,N1(C(=O)CSC(F)(F)F)CCCCC1C1CCCN1C(=O)CN1CCCNC1=O 57435,C1(CCNC(C2(CO)CC2)=O)CCN(C(C2CCCC2c2nc(S)n[nH]2)=O)CC1 57436,C(=O)(C(CCSC)NC(=O)C(C)C#N)N1CC(CC(CC)C)C1 57437,N1(C(C(CC)CC)=O)CC2OCC(NC(=O)C(c3c(C)noc3C)C)C2C1 57438,c1(NC(C23CC(C(=O)OC)(C2)C3)=O)c(OC)cccc1C.CCC(C)(C)C(=O)NC 57439,C(COC)(CC(=O)Nc1cccc(C#N)c1)NC(COCCOCC#C)=O 57440,CSC1=C(C(=O)NC2CCCCN(C(C3(CO)CC3(F)F)=O)C2)CCCC1 57441,Cc1ccc(SC(C)C(=O)NCCCCCN(C(c2c[nH]nc2C)=O)C(C)C)cc1 57442,N1(C(c2ncc(CC)s2)C(=O)NCCC2CC2)CCCOCC1C 57443,Cc1cc([SH](c2csnn2)(=O)C(C)C)nc(=NCCSC(F)F)[nH]1 57444,n1(CCC)cccc1C(N1C(C(=O)N(C)CCc2ncccn2)CC1C)=O 57445,CC(C)(CNC(C1(C)CC1F)=O)CNC(c1occc1C1CC1)=O 57446,N1(C(C2CC(CNC(c3c(CCC)nco3)=O)C2)=O)CC2CC(C)C2C1 57447,Cn1nccc1CC(=O)NC1CC(CC(=O)NCCF)C1 57448,N1(C(C=NOC)=O)CC2=C(C1)CN(C(=O)Cc1ccsc1C)C2 57449,C1(CNC(c2ncc(C)nc2)=O)CC2CCC1N(C(=O)CC1CC(C)(C)CO1)C2 57450,C1(c2nnnn2C)(CCSC)CCOC2(CCCC2)C1 57451,S(=O)(=O)(c1ccc(C2CC2)s1)N1C(C)CC(C2CCCN2)C1.c1ccccc1Cl 57452,N1(C(c2ccc(COC)[nH]2)=O)CCCC(CCNC(c2cc(Cl)n(C)n2)=O)CC1 57453,N1(C(c2c(C)[nH]cc2)=O)CCC(O)C(N(C(=O)CSc2nnnn2C2CC2)C)C1 57454,CC1CN(C(=O)Cc2csc(=N)[nH]2)CCN1C(c1nccn1C)=O 57455,CC(C)(C)CC(O)CC(=O)N1CCOCC1CC(N1CCNC(=O)CC1)=O 57456,c1(N2CCCC(C)(C)CC2)nc(N2CCSC(C)(C)C2)c2ncsc2n1 57457,C1(CNC(C(C(=C)Cl)(C)C)=O)C(C2CC2)CCN1C(=O)CCc1cnc(C)s1 57458,C1(C2(O)CN(C(c3cc(O)ccc3O)=O)C2)(CNC(c2c(C)snc2)=O)CC1 57459,N1(C(C2ON=C(C(C)C)C2)=O)CC2CCC(NC(=O)C(C)C)CC2C1 57460,C12(C(=O)NC3CCC(Cc4n(C)ccn4)CC3)CCC(=O)N1CC1(CC1)C2 57461,c1(N(C2CCCC2C)C(=O)CCn2cc(Br)ccc2=O)ccc(Br)cc1COC 57462,C1(CN(C(c2ccon2)=O)CC)CCCN(C(=O)CN2CCC(C)(O)C2)C1 57463,C1(C(=O)NCC2C(NC(CC(C)C)=O)CCCC2)CS(=O)(=O)CC(=O)N1 57464,N1(c2nc(=O)cc(C)[nH]2)CCC2(CC1)OCCc1cc(C(=O)NC3CC3)sc12 57465,c1(CC)cc(C(N2CCC(C(C)(C)C(=O)NCC(C)N(C)C)C2)=O)c(C)o1 57466,Cc1c(Cl)c(C(N2CC3CC3(NC(=O)CC3CC(F)C3)C2)=O)nn1C 57467,C12(C(N3C(C)(C)C(CNC(=O)CCC[N+](=O)[O-])CC3)=O)CCOC1CCOC2 57468,C12(CNC(CCOC)=O)CC(CNC(c3cnccc3N(C)C)=O)(CCO1)C2 57469,Cc1cc(Br)cnc1C(N1CC(N(C)C(c2cc(O)n(C)n2)=O)C(F)C1)=O 57470,S(=O)(=O)(c1ccc(-c2cccc(C(F)F)c2)cc1)NC1CCC(=O)NC1 57471,O=C(CC1NC(=O)c2ccccc21)NCC1CCN(C(c2coc(O)n2)=O)C1 57472,N1(C(CCOCC(C)C)=O)CCc2ccccc2C(NC(C2CCC(F)C2)=O)C1 57473,CCCC(C)CC(=O)NCCC1(CO)CC1.C123C(C4CC1C2C4)NC3=O 57474,C1(C(=O)NC2C=CCN(C(C(n3cc(C)nc3)(C)C)=O)C2)CC2CCCC2C1 57475,N1(C(CS(CC)(=O)=O)=O)CCC2CN(C(=O)COCCC(C)C)C(C)C12 57476,c1(C(=O)NCC2CN(C(Cn3c(C)cc(C)n3)=O)CC2C)nc2ccccc2[nH]1 57477,C1(C(N(C(C)C)Cc2cscc2Br)=O)CCc2ccccc2C1 57478,c12nc(n(C3CC4CCCC34)n1)CCNCCC2.c1(COC)ccccc1 57479,CCCC(CCC)=CC(=O)N(C1CC(C#N)C1)CC(=O)N(C(C)CC)C.C1CO1 57480,C1(CNC(CNC(C(C)OCCN(C)C)=O)=O)CCCCC1NC(=O)C(F)(F)F 57481,C1(C(=O)NC2CC3(C(NC(c4c(C)cccc4C)=O)C3)C2)CCC12CCOCC2 57482,N1(Cc2cn(C3CCC3)nn2)CCc2ccncc2C1.c1(N2C(=O)C2)cccnc1 57483,N1(C(C2CC2c2ccccc2)=O)CCC2(CCCN2C(c2csc(Cl)n2)=O)C1 57484,Cc1nnc2n1CCC2(C)C(=O)NC(c1ccc2c(n1)NCC(=O)N2)=O 57485,c1(C(c2n(CCC)nnn2)NCCSc2ccsc2)ccccc1Br 57486,c1(N(C(CN2CC(n3cc(COC)nn3)C2)=O)CC2CCCO2)ccnc(C)c1 57487,Cc1ccc(Br)c(C(=O)NC2CCCCC2NC(C2CN(C)C2)=O)n1 57488,CN1CC2CC2(CNC(c2ccccc2Nc2ccc(F)cc2F)=O)S1(=O)=O 57489,C(=O)(C1=NOC(C(C)(C)C)C1)N1CC(C)(NC(=O)CCOCC2(O)COC2)C1 57490,C(CCCCCCC(=O)NCC(C)(C(=O)O)n1nnc(-c2ccccc2)n1)SC 57491,Cc1ccnc(C(F)(F)C(=O)NCC2CCCN(C(C3CCCN(C)C3)=O)C2)c1 57492,N1(C(C=CCOC)=O)CCC(NC(=O)CCCc2ccccn2)C1 57493,N1(C(CN(C(=O)OC(C)(C)C)CC)=O)CC2(CCC2)CC1C(=O)Nc1ccno1 57494,CCCC(C)(O)C(=O)N(CC(C)N(C(=O)Cc1ccco1)C)C 57495,CC#CCC(C(=O)NC1CC2CC(O)C1C2)NC(c1ccnc(C)c1)=O 57496,N1(CCC)CCCC1C(=O)NC(c1cncn1C)C(=O)NCC=CC(C)C 57497,C(=O)(C(C(=O)OCC)C(C)(C)C)NC1(C)CCN(C(c2ccn(CC)n2)=O)CC1 57498,CC1CN(C(C2CN(CCCSc3ccccc3)CC2C)=O)CC(C)O1 57499,c1(C(=O)NC2C(C)CN(C(=O)C3=CCC3)CC2)cnn2c1CC(C)CC2 57500,C12(C(=O)NC3CCCN(C(=O)Cc4ccccn4)C3)C(=O)C3CC1C2C3 57501,c1(C(=O)NCCC(C)N(C(C(C(C)(C)C)SC)=O)C)cc([N+](=O)[O-])ccc1SC 57502,c1(C(N(C2CN(C(=O)Cc3ccoc3)CC2O)C)=O)cnc2ccccc2c1 57503,Cc1c(C(=O)NCC(F)CNC(=O)C(c2ccn(C)c2)C)cnn1CC(F)F 57504,N#Cc1cc(C(=O)NC2CCN(C(c3ccc(C(F)(F)F)s3)=O)C2)c[nH]1 57505,C1(C(=O)NCC2(NC(C3C(C)C3)=O)CC2)COC2CC1C2 57506,Cc1ccc2c(=NCC(=O)N=S(C)(C)=O)[nH]c(N3CCOC(C)(C)CC3)nc2c1 57507,n1(CC)cc(C(=O)NC(C2CCN(C(c3cc(C)cn3C)=O)C2)(C)C)c(C)n1 57508,N1(C(Cc2c(C)ccc(C)c2)=O)CC(C)(C)OCC1CNC(C1CCCC1)=O 57509,C(=O)(CCCCCC#N)NCc1cc(C(=O)NC(CC(=O)OCC)C)ncc1 57510,N1(C(c2cccc(COC)c2)=O)CCC(C2CCN(C(=O)C=C3CCC3)C2)CC1 57511,C1(NC(c2ncc(F)cc2F)=O)CC2CN(c3ncc(F)cn3)CC12 57512,C1(NC(C(N2CCC(O)CC2)C)=O)CCN(C(C2CC(C)(C(C)(C)C)C2)=O)CC1 57513,C(=O)(C(F)CC(C)(C)NC(=O)CCn1ccc(C)n1)N1CC(C#C)C(OC)C1 57514,Cc1cccc2cc(C(=O)NCC3CN(C(=O)COCC(F)F)CCC3C)oc12 57515,C(CCCCCC(=O)N1CCC(NC(C2CC(OC(F)(F)F)C2)=O)C(O)C1)SC 57516,c1(NC(=O)NC2CC(C)(NC(C3(C)CC3C(F)(F)F)=O)C2)ccccc1 57517,n1(C(C(N2CCCC(NC(CSCC(=O)OC)=O)C2)=O)C)cnc2c(N)ncnc12 57518,CC1(C(=O)NCCC(O)C(=O)NCC(O)C2CC2)C=CCCC1 57519,c1(CCOC(C(=O)OCC)C2CN(C(=O)Cc3cc(C)no3)C2)cncc(C)n1 57520,CCC(C)C(C(=O)N1CCC=CC1C(=O)N(C(C)C(C)SCC)C)OC 57521,N1(C(c2n[nH]c(C)c2Cl)=O)CC2CCCC(NC(C3CN4CCN3CC4)=O)C2C1 57522,CC(CS(C)=O)C(=O)N1CCN(C(=O)CN(C(=O)Cc2cnns2)C)CC1 57523,C1(CC(=O)NCC(C)CN(C)C)CCCN(C(c2nc[nH]n2)=O)C1 57524,CC1(C)CCc2cc(C#N)c(NC3CN(C(=O)CC4CCC5(CCC5)O4)C3)nc21 57525,CC(C)(CNC(c1ccc(-c2cnccc2F)cn1)=O)CC(F)F 57526,C(=O)(C1=CCOC1)NC(C(=O)NC(c1ccc(Cl)cc1)c1cn(C)nc1)=O 57527,C1(NC(C2(CCN(C)C)CC2)=O)CCC(NC(=O)CN2CCOCC2)C1 57528,C1(C(=O)NCC(C(C)O)C)CCOCCN1C(C1CCC(O)CC1)=O 57529,N1(C(C2CN(CC)C(=O)C2)=O)CC(NC(c2cnc(C)n2C)=O)C(C2CC2)C1 57530,CCCCCCC(C)CC(=O)NC1(COC)CN(C(c2c[nH]nc2[N+](=O)[O-])=O)C1 57531,c1(C(N(CCCC)C2CCC2)=O)cc(CNC(c2coc(C3CC3)n2)=O)[nH]n1 57532,C(=O)(CCCC(=O)NCc1csc(C(N2CCC(COC)C2)=O)c1)OC 57533,CC(C)CC(C(=O)N(C)C)N(C)C(c1nccnc1C(N)=O)=O.C1(=O)CN1C 57534,C(C(C)(C)C(C)C)N(CCOCC(=O)N(CC(=O)N)CC)C.C1(SCC)CCC1 57535,C1(NC(C(N2C(=O)CCC2=O)C)=O)CCN(CCc2ccc(F)c(F)c2)CC1F 57536,c1(C2(C(N3CC(C)(NC(c4c(Cl)cn(C)n4)=O)C3)=O)CC2)ccccc1C#N 57537,C1(OC)CCCC1C(=O)NC(C)CCNC(c1cn(C)cn1)=O 57538,C(C(CO)CC(C)(C)C)NC(=O)NC(CC(C)C)CCc1ccc(F)cc1 57539,N1(C(c2c(CNC(c3nc(CCC)oc3)=O)c[nH]n2)=O)CC(O)CC1CC 57540,c1(OC)ncnc(C(N2CCCC2CCNC(C2(CC(C)C)CC2)=O)=O)c1F 57541,C1(NC(CCn2c(C)ncc2)=O)CCCC(CN(C)C(c2nn(C)cc2Cl)=O)C1 57542,C(=O)(C1CCCc2cc(C#N)ccc21)NCCN(C(C(CN(CC)CC)F)=O)C 57543,C=CC(C)CN=C(NCC1CCCO1)NCC1(C(C)(F)F)CCOCC1 57544,Cc1c(C(=O)NCC#CCNC(c2[nH]c3ccccc3c2Cl)=O)nc2sccn12 57545,N1(C(=O)Cc2cccc(O)c2)CC2CN(C(=O)C=Cc3cnccn3)C2C1 57546,C(CCC(O)CO)NC(C=C(C)CNC(C1CCNC(=O)C1)=O)=O 57547,C1(NC(CCNC(COC)=O)=O)CN(C(c2cncc(F)c2)=O)CC1C 57548,c1(SCC(=O)NC2CN(C(C34CC(C)C3C4)=O)CC23CC3)ccccc1[N+](=O)[O-] 57549,c1(C(N(C2CCN(C(=O)Cc3ccon3)CC2)CC)=O)cc(C)nc2ncnn12 57550,c1(OC)cc(F)c(F)cc1C(=O)N(C)CC1CCN(Cc2cnn(CC)c2Br)C1 57551,C1(CC)CN(C)C(=O)CN1C(c1cc(C#N)n(C)c1)C(=O)NC1CCC1 57552,C#Cc1ccc(Cl)c(C(N2CCC(C)C(NC(c3cc(C)c[nH]3)=O)C2)=O)c1 57553,CC1Oc2c(C(=O)NCCN(C(=O)CCC(=O)NS(C)(=O)=O)C)cccc2C1C 57554,C1(C(=O)NCCN(CCCCCC)C(c2conc2C2CC2)=O)CCS(=O)(=O)C1 57555,C1(C(c2ccco2)C)CN(C(c2cscn2)=O)CCN1C(=O)C(c1cc(C)sc1C)=O 57556,c1(CNC(C2CCN(C(=O)OC(C)(C)C)C2)C)ccc(Cl)cc1C(F)(F)F 57557,N(C1CCCOc2c(F)cccc21)C(c1ccc(SC(F)(F)F)c(F)c1)=O 57558,C(=O)(C(O)CCCNC(c1c[nH]c(=NC)s1)=O)N(CC=C)CCOC 57559,c1(OC)ccc2ccccc2c1CC(N1CC(CNC(c2csc(Br)c2)=O)C1)=O 57560,C1(C2CCCC2)(C(N2CC3(CC(NC(C4CCOC4C4CC4)=O)C3)C2)=O)CCC1 57561,CC1(C)CC1(C(=O)NCCOc1ccccc1)NC(=O)C=CC(F)F 57562,c1(NC2C3N(C(c4cc(CCC)on4)=O)CC(CC3)C2)ncc(Cl)cc1[N+](=O)[O-] 57563,C1(CC#C)CCCCCN1CC(=O)Nc1cc(O)cc(O)c1.c12ccc(cc1)s2 57564,N1(C(c2c(CC)occ2)=O)CCC(C)C(NC(c2cc3c([nH]2)CCCC3)=O)C1C 57565,c1(CN2CC(NC(c3nc(Cl)ccc3F)=O)C(F)C2)ccn2ccnc2c1 57566,N#Cc1cncc(NC(c2nc(C3(O)CCOCC3)cs2)=O)c1 57567,Cc1cc(C)c(C(=O)N(C)CC2CCCCN2C(=O)C2=CC(C)C2)cn1 57568,C1(NC(=O)C(O)C2CCCC2)CCN(C(=O)CCc2cnc(-c3ccsc3)o2)C1 57569,C12(C(N(CCCn3cc(C(CSC)C)nn3)C)=O)CC3CC(C1)CC(C)(C3)C2 57570,c1(CC)ccc(N)c(C(=O)NC2CC3CC(NC(C4CCN(C)C4=O)=O)CC23)c1 57571,N1(C(C)COC2CCCCC2)CCCC(NC2CC2)C1 57572,N1(C(c2c(C)nc[nH]2)=O)CC(C)CCC1CNC(c1cc(C(N)=O)c[nH]1)=O 57573,N1(C(CSC)=O)CCC(CNC(=O)C=Cc2ccccc2C(F)(F)F)C12CCC2 57574,C#CCC(O)C(=O)N1CCC(NC(c2cnn(COC)c2CC)=O)C1 57575,S(=O)(=O)(c1ccc2c(c1)NCC2)NCC(=O)Nc1ccccc1C(F)(F)F 57576,N1(C(Cc2c(C)non2)=O)CC2C(CN(C(=O)C=CC(=O)NC3CC3)C)C2C1 57577,C1(=O)C(C(C)(C)C)N1.N1(CCC)CCCCC1C(=O)N(CCN(C)C)C(C)C 57578,c1(C(N2CCC(S(N)(=O)=O)C2)C(=O)NCC(C)C)noc2c(Cl)cccc12 57579,N1(C(c2csnn2)=O)CC2CC1(C(=O)NCC1CC(C(F)(F)F)C1)C2 57580,c1(C(=O)NCC(=C)CCNC(C2(C)CCCCO2)=O)ccc(S(N)(=O)=O)c(C)c1 57581,CC1ON=C(C(=O)N2CC(CNC(=O)CN3CCCCCC3=O)C3CC23)C1C 57582,c1(C(N2C(CCOC)CN(C(c3coc(C)c3)=O)CC2)=O)cccc2c1NCC2 57583,CCCCC(C)C(=O)NC(CNC(C1(CSC)CC(F)(F)C1)=O)CC 57584,CCC(C)C(O)C(=O)NCC1CC2CN(C(c3cc(C)cs3)=O)CC12 57585,C(=O)(C(C)C(C)C)NCC(c1ccccc1F)NC(C1(C(C)(C)OC)CC1)=O 57586,C(=O)(C1CCc2ccccc21)N1C(COC)CN(C(=O)CC(C)(F)F)CC1 57587,C(CCC(C)C)(C(=O)N(C)Cc1cc(C)cs1)NC(C(C=C)C)=O 57588,N1(C(c2c(CC)onc2C)=O)CCC(NC(=O)C=NOC)C(F)C1 57589,C(=O)(C(CC(C)C)NC(=O)CC(COC)NC(C1CC2CCC(C1)O2)=O)NC 57590,c1(C(N2C(CCNC(C=C(C)Cl)=O)CCC2)=O)cnc(C)cn1 57591,c1(CN2C(NC(CC)C(=O)OC)C(O)CC2)ccc(OC(F)F)cc1Cl 57592,c1(C(N(C(CNC(CC(C)OC)=O)C2CC2)C)=O)cc2cc(Cl)sc2[nH]1 57593,C(CCC(C)(C)C(=O)NC1CCn2nnnc2C1)NC(C(COC)C)=O 57594,c1(C(=O)NCC2(OC)CN(C(=O)C3=C(C)CC3)C2)ccc(C(F)(F)F)c(N)c1 57595,C1(C(=O)NC2C(NC(C(c3cn(CC)nc3)(F)F)=O)CC2)CCCC1(C)CO 57596,C(=O)(C(COC)COC)N(C(CC)C(=O)NC(CC)C1CCC1)C 57597,CC1CC(NC(c2cc3n(n2)CCC3)=O)CCN1C(C1CN(C)CC(C)O1)=O 57598,c1(OC)ccccc1OCC(O)CN(C1COCC1(C)C)C.C(C(C)(C)NC)O 57599,N1(C(CCN(C(CCC)C)C)=O)CCCC1C(C)NC(=O)Cn1cn[nH]c1=N 57600,C1(C(=O)NCC2(SC)CCOCC2)CN(C(C2CCCO2)=O)CC1C1CC1 57601,C12(NC(c3ccc(=O)n(CCF)n3)=O)CCCC1N(c1ncc(Br)cn1)CC2 57602,c1(C(=O)Nc2c(NC(c3cc(C)cc(F)c3)=O)cccc2O)cc(Br)cc(C)c1C 57603,CC(C)CCCOCC(=O)NC1CC1CNC(C12CSCC1C2)=O 57604,c1(NCC(N(C)C)C2CC2)[nH]c(=NC2CC(N3CCC3)C2)nc2scnc12 57605,c1(C(=O)NCC(CC)NC(=O)CSC2CC2)ccc(-c2cnn(C)c2)o1 57606,N1(C(C2(CC)CCCCC2)=O)CCCCC(CNC(c2nccc(Cl)c2C)=O)C1 57607,C1(CNC(=O)CCOCC2CCCO2)CCN(C(C2CC(=C(F)F)C2)=O)CC1 57608,C(CN=C(NCC(C)C#N)NC(C1CCC(F)(F)CC1)C)c1ccc(OC)cc1 57609,CC1(C)CC(C(=O)NC(C)(C)CCCNC(=O)CCc2nc[nH]n2)=NO1 57610,C1(CNC(c2c(COC)noc2)=O)CCCC(NC(C2CCC2)=O)C1 57611,C12(NC(C=NOC)=O)CCCCCC1N(C(c1cncc(C(=O)OC)n1)=O)CC2 57612,C1(COC)CN(C(C2CCS(=O)(=O)N2)=O)CCN1C(=O)CCSc1ccccc1 57613,c1(CNC(N2CC(CN(C(C)=O)C)C2)=O)csc(C)n1 57614,N#CC1(C(=O)NCC2CCCC2NC(=O)CN2CCOCC2)CCC1 57615,c1(OCC(=O)NCC(C)NC(c2ccc(CC)cn2)=O)ccc2c(c1)CCC2=O 57616,C1(NC(C(CO)OC)=O)CN(C(c2ocnc2C2CC2)=O)C2CCCC12 57617,c1(C(N2CCCN(C(c3c(C=C)cnn3C)=O)CC2)=O)ccc2c(c1)NCCC2 57618,CCCCC(CC)CC(c1nnnn1C1CC1)OC.c12nccn1CCS2 57619,N1(C(CN(C2OCCC23CCC3)CCC)=O)CC2CC3CC2C1C3 57620,C(=O)(CC(C)C(=O)NCC(C)CC(=O)NC(c1cncn1C)CO)OC 57621,C1(NC(c2c(C)noc2)=O)CN(C(=O)C=C2CCCCC2)C2CCCC12 57622,c1(OC)c[nH]c(C(=O)NC2CCC(NC(=O)CCN(S(C)(=O)=O)C)C2)cc1=O 57623,Cc1[nH]c(=NC(CCO)c2ccsc2)ccc1F 57624,c1(CC)oc(C)cc1C(=O)NC(C1CC=CCC1)C(=O)Nc1ccsc1 57625,CC(CO)(C(F)F)NC(=O)CC1(NC(=O)C(N)=O)CC1 57626,C1(C(=O)NC2(CC)CN(C(c3occc3C3CC3)=O)C2)OCCOC1C 57627,c1(C(=O)NCC(C2(O)CCN(C(C3(F)CC3)=O)C2)C)ccnc2c1ncn2C 57628,C1(NC(CC(=C)Br)=O)CC(NC(=O)CCCC2(OC)CCC2)C(O)C1 57629,N1(C(CCCCC#C)=O)CC2CC(NC(c3ccc(C(N)=O)c(Cl)c3)=O)C(C2)C1 57630,Cc1ccc2[nH]c(C(=O)NC3C4CCC3N(C(C3CCC(C)(C)C3)=O)C4)cc2c1 57631,C(CC(O)CO)NC(C1N(C(COCCOC)=O)CC1)=O 57632,CCC(N=c1cccc(S(=O)(=O)NC(C)(C)C2CC2)[nH]1)c1cc(C)ccc1F 57633,C(=O)(C(CC(C)C)ONC(=O)C1CC(F)C1)N1C(C=C)CCC1 57634,CC12CC1CCN2c1nnc(-c2nc[nH]n2)o1 57635,N1(C(C=NOC)=O)CCC2(CNC(c3c(F)cc(F)c(F)c3F)=O)CCCCC12 57636,n1(CCNC(C2(C3N(C(CC4CC(O)(CC)C4)=O)CCC3)CC2)=O)nc(C)cc1C 57637,CCC(C)(COC)C(=O)NCC1(NC(=O)C(C)OCCCOC)CC(F)(F)C1.CSC 57638,C(c1ccc(OC(F)F)cc1)=CC(=O)NCC(C)NC(C1CCC(C)(C)CO1)=O 57639,c1(C(=O)NCCCCN(C(C=Cc2ncc(C)[nH]2)=O)C)cnc2ccccc2c1 57640,c1(NC2(C(=O)NC(CCCNC(C3C(OC)CC3)=O)C)CC2)ccc(C)c(C)c1 57641,C#CC1(C(=O)NCC(CO)N(C)C)CCN(C(=O)Cn2cc(C)cn2)C1 57642,N1(C(CC(C)n2cccn2)=O)CCCC(C)(NC(c2ccc(CO)cn2)=O)C1 57643,c1(CC(=O)NC23CCCC(NC(=O)Cn4nccn4)(C2)C3)csc2ccccc12 57644,C1(COC(CSCCCC)=O)CN(C(=O)OC(C)(C)C)CCO1 57645,N1(C(C(c2scc(C)n2)C)=O)CCCCC(NC(c2ccc(N)c(F)c2)=O)C1 57646,N1(C(c2c(C)c(F)ccc2)=O)CCC(C2CCCN(C(c3ocnc3Cl)=O)C2)C1 57647,CC(C(C)(C)O)N(C(=O)C(C)CNC(C1CCC(C(N)=O)C1)=O)C 57648,c1(C(=O)NC2C(CNC(C3N(C)C(=O)CCC3)=O)C2)cc(F)c2ccccc2c1 57649,c1(CO)ccnc(-n2cc(CNC(C3CC3C(F)F)=O)nn2)c1 57650,N1(CC)CCCCC1C(=O)NCC1CC(C(=O)NCCC2CCC(=O)NC2)C1 57651,c1(C(N(C)CC2CCCN(C(C(C)SC(C)C)=O)C2)=O)cc(F)c(F)cc1O 57652,CC(F)(F)CCCC(=O)NCC1CC1NC(C1(Sc2ccccc2)CC1)=O 57653,N1(C(c2ccc(=N)[nH]c2)=O)CCC(F)(CNC(=O)CC2CNC(=O)C2)CC1 57654,c1(C(=O)NCC(CNC(c2cc(C)c(C)nc2)=O)CO)ccc2cn(C)nc2c1 57655,CC1CN(CCNC(C2CC=CCC2n2cc(-c3cccs3)nn2)=O)CCO1 57656,C(=O)(CN=c1cc[nH]cc1)N1C(CNC(c2ccc(F)c(C)c2C)=O)C(C)CC1 57657,C1(n2cc(CNC(CCC=C)=O)nn2)CCCN(C(=O)CC2(CO)CCC2)C1 57658,c1(NC(C2C3CN(C(c4cc(C)cc(F)c4)=O)CC32)=O)cc2nc[nH]c2nc1C 57659,c1(C(C)C(N2CCC(c3cn(CCCCC(=O)O)nn3)CC2)=O)cccc(C#N)c1 57660,c1(NC(C2CC(C)(O)C(Cc3nn(C)c(Cl)c3)C2)=O)cc(Cl)nc(C2CC2)n1 57661,CC1(C(=O)NC2CCCC(NC(c3cccc(CC(F)(F)F)c3)=O)C2)CCCCO1 57662,Cc1nc(N2CCC3CCN(C(c4cn(C)nc4C)=O)CC3C2)ncc1[N+](=O)[O-] 57663,Cc1nc(=O)n(C2CCN(C(C3CCN(C4CCSCC4)CC3)=O)CC2)[nH]1 57664,C1(C(N2CCC(N(C(=O)Cc3cnns3)CC3CC3)CC2)=O)C2CC3C(C2=O)C13 57665,C1(CCC(c2cncnc2)O)(CC)CCN(CN(C)C)C1.N12CCC(C)(C1)C2=O 57666,C1(C(N(C2CN(C(=O)Cn3ccnn3)CC2O)C)=O)C(C#N)C1(C)C 57667,C=C=CCCC(=O)NC(C)(C)C=CC(N1CCCCC1COC)=O 57668,c1(SC)ccc(C(=O)NCCCC(C)NC(=O)CCOC(C)=O)s1.C1(O)CC1 57669,n1(CCOC)ccc(CC(=O)NC2CC(OCC(=O)N(C3(C(C)C)CC3)C)C2)n1 57670,c1(NCC)cc(C(=O)NC(CNC(=O)C(CC(C)C)OC)CC(C)C)c(C)nn1 57671,C(=O)(CCCCC(F)F)NC(C)CN(C)C(c1ccc(Cl)cc1Cl)=O 57672,c1(NCCc2cnc(C)s2)ncc(C)cc1S(=O)(=O)N1CCCC(N(C)C)CC1 57673,c1(C(=O)NC(C)CS(C)(=O)=O)coc2c1CN(C(c1cc3n(n1)CCO3)=O)C2 57674,c1(C(=O)NC2CCC(CCNC(c3c(C)ncs3)=O)C2)cc(F)cnc1O 57675,N1(C(C2CCC(NC(c3cccc(C#C)c3)=O)CC2)=O)CC2CC3CC2C1C3O 57676,Cc1cc(C(=O)NCC2CC2CNC(c2ccsc2)=O)c(C)s1 57677,C1(CNC(C2CCC(=O)NC2)=O)CC(C(=O)N2CC(F)(CO)C2)=NO1 57678,c1(CN(C(C2C(NC(C(C)=C(CC)C)=O)COC2)=O)C)cccnc1O 57679,n1(CCOC)nnnc1C(C(C)C1CCC1)NC1CCC(C(=O)NCCO)C1 57680,c1(CC)onc(C(=O)NC2CCOCC2C(N2CCCC2C2(CC)CC2)=O)c1C 57681,CCC(C)(C(=O)Nc1ccccc1CN(C(=O)C(C(=O)OC)OC)C)C(N)=O 57682,c1(C(N(C(C)CNC(C23CCCC2(C(N)=O)C3)=O)C)=O)cccc(Br)c1F 57683,Cc1nc(-c2nccs2)sc1CNC(=O)CSCc1ccccc1Br 57684,C(=O)(CC1=CCCC1)NC(CC#CC)C(N1CCC(O)(C2CC2)C1)=O 57685,N1(C(C2(CC)CCN(C(=O)C(C)C3CCCC3)CC2)=O)C(CC)C2CC(O)C1C2 57686,N1(C(C2CCC(C(=O)OCC)CC2)=O)CCCC(N(C)C(C2CC(F)C2)=O)CC1 57687,Cc1cnsc1C(=O)NCCN(CC(C)O)C(c1cn(-c2ncccn2)cn1)=O 57688,N1(c2nnc(CCC)s2)CC2CCC1C1CN(C(=O)CCC(C)N(C)C)CC21 57689,N1(C(C=CC(C)(C)C)=O)CCN(C(=O)COc2ccc(F)c(Cl)c2)C2CCC12 57690,CP(C)(=O)c1cccc(C(=O)NCC(C2CC2)NC(c2ccc[nH]2)=O)c1 57691,C1(CC(N2CCC(C)(CCC)C2)=O)CC(C)(C)CN1C(=O)CC(C)(C)C 57692,C(=O)(C1=CS(=O)(=O)CCC1)NC1CN(C(CN(C(=O)OCC)C)=O)C(C)CC1 57693,c1(C(=O)NC(C)CN(C)C(C2C(C)C2C)=O)cc(S(=O)(=O)Nc2cccs2)c[nH]1 57694,Cc1[nH]nc2c1CN(c1nnc(-c3cc4ccccc4o3)n1CCCCF)CC2 57695,c1(NC(C2N(c3nc(C)cc(C)n3)CC(O)C2)=O)c(C)ccc2n[nH]cc12 57696,N1(C(C(C=CC)O)=O)CC(C)CN(C(=O)CC(O)C2CCCC2)C(C)C1 57697,c1(C(=O)NC(C)CCCCNC(c2cccc(CO)n2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 57698,C1(CNC(CCSCCCC)=O)CCC(CCC(=O)N(C)C(C)C)C1 57699,c1(C(=O)NC2CC(CCNC(C3C(C)(CC)C3)=O)C2)ccc(Cl)c2occc12 57700,CC1C(N(C(=O)CCC2CCC(NC(c3cc(C#N)cs3)=O)C2)C)CCCC1C 57701,c1(C(C(=O)C(Cc2ccccc2Br)N)=O)cccc2c1CCC2.C1(CN)CCOC1 57702,Cc1ccc(C(=O)NCC2CCN2C(=O)CCCc2ccccn2)c(C)n1 57703,c1(C(=O)NC2CCC(N(C(Cc3c(C)con3)=O)C)CC2)cnc(CO)nc1C 57704,N1(C(C(C)(C2CC2)NC(C2CCO2)=O)=O)CCC2(CC1)N=N2 57705,c1(C(=O)NCCCNC(c2ccc(N)c(F)c2)=O)ccc2c(c1)S(=O)(=O)NC2 57706,c1(NC(N2C(CCc3c(C)[nH]nc3O)CCC2)=O)cnc(N2CCCC2)nc1C 57707,N(C1c2ccccc2CC1NC(=O)C(C)N(C)C)C(c1n(C(CC)C)ncc1)=O 57708,N1(C(CC(CC)CC)=O)CC2CCC1CN2C(=O)C(C)N1CCC1 57709,C=CC1(CC(N2CCC(C#N)C2)=O)CN(C(=O)CCSCCC)C1 57710,C(CS(C)(=O)=O)(C(=O)O)NCn1nc(C(CCCC)n2cc(CO)nn2)c(C)n1 57711,C1(C2CCN(C(=O)C=CCN(c3ccncc3)C)C2)(NC(CSCCC)=O)CC1 57712,C1(C(N2CC3C(NC(c4ccc(C(N)=O)s4)=O)C3C2)=O)CCCC2(CC2)C1 57713,c1(C(N2CCOCC(CNC(C3CC3F)=O)C2)=O)cc2c(nc1O)CCCC2 57714,C(=O)(C(CC)N(C)N1CCCc2nc(C)ccc21)NCCCC(=O)OC 57715,C1(CC(=O)N(CC=CC(=O)NCC2(N(C)C)CCCC2)C)CCCCC1O 57716,C1(C#CC(=O)NCCC(C)(C)CNC(c2cccc(COC)c2)=O)(CC)COC1 57717,Clc1cccc2c1CCC(N=c1[nH]c(=NCc3nncs3)[nH]c3c1SCC3)C2 57718,N1(C(C(n2ccc(C)n2)C)=O)CCC2OCCN(C(=O)CCc3cnc[nH]3)C2C1 57719,c1(C(=O)NCC2(F)CC(NC(=O)CC3CC34CC4)C2)nn2cccnc2c1Cl 57720,c1(C(N2CC(O)(CN(C(Cc3c(C)scc3)=O)C)C2)=O)ccc(Cl)c(O)c1 57721,N1(C(c2ccc(C)nn2)=O)CCN(C(=O)C(C(C)(C)C)n2ccnn2)CC1C 57722,c1(C(=O)NCCC(Cn2cc(CCC(C)O)nn2)F)cc(F)c(F)c(F)c1 57723,c1(C(N2C(C(=O)Nc3cncnc3O)CSCC2)=O)cnn2ncccc12 57724,C12(NC(CCCC(C)C)=O)CCCC1N(C(c1ncccc1S(C)(=O)=O)=O)CC2 57725,c1(C(=O)NCC(C)NC(=O)CCc2cnn(C)n2)cccc2c1OC(C)C(=O)N2 57726,C1C(C(F)(F)F)CNC(=O)CCC(=O)c2ccc(C(C(C=C)(C)O)=O)c(c2)CCN1 57727,c1(OC(=O)NC2(NC(N3CC(N(CCN)CCO)C3)=O)CC2)ccccc1F 57728,N1(C(c2cnc(=N)[nH]c2)=O)CCCC(C2(NC(=O)CCc3cnn[nH]3)CC2)C1 57729,c1(C(N2CC(NC(c3ccc(C)c(F)c3)=O)C(C)C2)=O)cccc2c1OCCC2 57730,N1(C(CN(C)C)=O)CC23CCCC2(C1)CN(C(=O)C1CCc2ccc(Br)cc21)C3 57731,C#CCC(O)C(=O)N1C(C(N2CCC2C)=O)CCC1C1CC1 57732,N1(C(CNC2(CC(=O)OC(C)(C)C)CC2)=O)C2CSCC1C2 57733,n12c(nc3ccccc13)C(C)NC(=O)C2.C(C(F)CO)NC(=O)OC 57734,C1(NC(CC2C(C)CC2)=O)CC2CC(NC(c3cnn(C)c3C(F)F)=O)CC12 57735,N1(C(C2(C(=O)NC)CC2)=O)CC=C(CNC(C2SCC=C2C)=O)CC1 57736,c1(C(C(=O)NCC(c2c(C)cccc2)C)(F)F)ccc([N+](=O)[O-])cc1F 57737,C(=O)(C(C)CC(N)=O)NC1C(NC(c2ccc(CSC)o2)=O)CC1 57738,c1(C(N2C(C(N3CCOC(CCO)C3)=O)CCC2)=O)cncc(C(F)F)c1 57739,C1(C(=O)NCC(C)NC(C2CC(O)C2)=O)CCCC1O 57740,C1(C(=O)NCc2c(C(=O)NC(CCCOC)(C)C)cccn2)CC(C)CC(=O)N1 57741,N1(C(C2(COC)CC2)=O)CC2(C1)CN(C(c1cnc3c(c1)CCCO3)=O)CCO2 57742,n1(CC)nc(C)c(COC(c2ccc(N3CCCC3)nc2Cl)=O)c1C 57743,c1(OCC)ccc(NC(N2CCCC(NC(=O)CC3CCCC3)CC2)=O)cc1O 57744,CC1(CC(=O)NCC2CCC=CO2)CCN(C(=O)C=C2CCC2)CC1 57745,c1(C(N(CCN(C(c2n(CC)ncc2)=O)C(C)C)C)=O)cnnc(Cl)c1 57746,Cc1ccc2c(CC(N3CCC(C(C)NC(=O)CC(C)(F)F)C3)=O)coc2c1 57747,CC1(C)C(C(=O)NCCc2ncon2)CC1CC(N1CCOC(CC(N)=O)C1)=O 57748,Cc1cnccc1C(C)(C)NC(=O)CSCCC#N.C1CN1 57749,N1(C(CSCCCC)=O)CC2CCC1CN2C(=O)C(C(C)C)N(C(C)=O)CCC 57750,N1(C(C2CN(C(C(C)(F)c3ccon3)=O)CC23CC3)=O)CC2(CCC(=O)NC2)C1 57751,c1(CC)nn[nH]c1C(=O)NCC(C)(C)CNC(c1ccn(CC)n1)=O 57752,c1(OC)cc2cc(Cl)nc(NC(c3cnc(C)n3C)=O)c2cc1Br 57753,CCCCCCCC(F)C(=O)NC1CCN(C(c2ccc(Cl)c(Cl)c2N)=O)C1 57754,N1(C2CC2)CC(C(c2n(CC)nnn2)N2CCC2)CC1=O.C1CC1.C(=O)(NCC)OC 57755,C1(OC)CN(C(=O)C(F)CC2CCC2)CC1NC(c1cnc(S)n1C)=O 57756,n1(CCCCN(C(CNC(=O)NC)=O)C(C)C)cnc2ccccc12 57757,N1(C(CCSC)=O)CC(C(=O)N(CC(CO)(CO)OC)C)C2(CCC2)C1 57758,c1(CC)cncc(C(N2CC=CC(C(=O)NC(C3CCC3)C3CC3)C2)=O)c1 57759,c1(NC)cccc(C(=O)NC(C(C)NC(=O)CCCc2cccs2)C(C)C)n1 57760,C(=O)(C(O)C(F)(F)F)N(CC(=O)NC(C#C)CCC)CC(C)C 57761,CC1(C)COCCC1CC(=O)NCC12CC(NC(C3CCCCCO3)=O)(CO1)C2 57762,c1(C(=O)NCC2CCN(C(c3scnc3C3CC3)=O)C2)csc(CC2CC2)c1 57763,C1(NC(Cc2ccc(OC)cc2)=O)(CO)CCN(C(C2CCCC(C)C2)=O)CC1 57764,N1(C(C2C(CC)N(C)CC2)=O)C2CCC1C(CNC(=O)CCc1ccsc1)C2 57765,C#CCCCCC(=O)N1CC(N(C(=O)C(C)c2ncco2)C)C(O)C1 57766,N1(C(C(CCC)CC2CCCC2)=O)CCC(C2(NC(c3ccc(C)s3)=O)CC2)C1 57767,c1(C(C)CC(=O)NCCC2CCN(C(C3(F)CC=CC3)=O)C2)ccc(F)c(F)c1 57768,Cc1cc(C(=O)NC(C)CC(C)NC(C2(O)CC2)=O)cc(Cl)c1 57769,c1(C(=O)NC23C(NC(CC(C)O)=O)CC(CC2)C3)ccc2sccc2c1 57770,CC1c2c[nH]nc2CCC1C(=O)NC1CC1CNC(=O)CCSC(F)(F)F 57771,n1(CC(=O)NCCCCNC(C(CC)(C)C(F)F)=O)ncc2ccccc2c1=O 57772,CC1CC(C(=O)NC2CCCC2C(=O)NCCNC(N)=O)CCS1 57773,C1(F)(NC(=O)CCOCCOCCCO)CN(C(=O)Cc2csc(C(F)(F)F)n2)C1 57774,C1(n2cc(C(N3CCCC3)(C)C)nn2)CCCN(C(C2CC23CCCC3)=O)C1 57775,c1(C(=O)NCCCNC(CCCC(CC)C)=O)ccc2c(c1)OCCN2 57776,c1(OCCOC)cccnc1C(=O)NC1CC(C)N(C(=O)C=C(C)C(C)C)C1 57777,N#Cc1cc(NC(C23CC2CN(Cc2ccccc2Cl)C3)=O)cc(Br)c1 57778,c1(OC)ccc(F)c(C(=O)NC(C2CCN(C(C3CCC3(C)C)=O)CC2)C)n1 57779,C(CN=c1[nH]cncc1I)(N(C(c1ccc(C#C)cn1)=O)C)C1CC1 57780,N1(C(c2scc(C(C)C)n2)=O)CCC(CO)(NC(=O)CCCn2ccnn2)CC1 57781,CCC(C)CCC(=O)N1CCC(C(=O)N(CC(N2CCCC2)C)C)C1(C)C 57782,O=C(C1COc2ccccc21)NCCOC1CN(C(=O)C(O)C2CC2)C1 57783,N1(C(CC(=C)Br)=O)CCCC(NC(=O)Cc2cc(Cl)sc2Cl)CC1 57784,C=C1CC(C(=O)NCC2CCC2C(=O)OCC)N(C(c2ccc(CC)[nH]2)=O)C1.NC 57785,COn1cnc(C)c1C(=O)NC(C1CCCN1C(c1ncc(C)nc1OC)=O)C 57786,C=CC1(CC(=O)NCc2[nH]nnc2C2CC2)CN(C(c2cc(C(C)=O)on2)=O)C1 57787,C1(C2CCN(C(c3ccc(C)s3)=O)C2)(NC(CNC(C)=O)=O)CC1 57788,C(=O)(C(C)(C)C(C)NC(=O)CC(C)N(C)C)NCc1c(C)nn(C)c1 57789,c1(C(N2CCC3CC3(C(=O)Nc3nccc(Br)n3)CC2)=O)cc2ccccc2[nH]1 57790,c1(NC(C2CC2CNc2cc(OCC)ncn2)=O)c(Cl)nc(C)nc1Cl 57791,c1(C(=O)NCC2(O)CCN(C(C3CCCCO3)=O)C2)cc(Br)cnc1S 57792,c1(SCC=C)ccccc1C(=O)NCCNC(c1cnn(C)c1CCC)=O 57793,C(=O)(C(C(C)(C)C)OC)NC(C=CC(=O)NCc1c(CC)nns1)(C)C 57794,C1(C#CC(=O)NC(c2ccccc2)C(N2CCCC(C(F)F)C2)=O)(CC)COC1 57795,C1(NC(C2CCC(C)(C)C2)=O)CC2(CCN(C(c3cc(Cl)c(N)cc3F)=O)C2)C1 57796,n1(CC(=O)NCCCCNC(=O)CSc2ccc(F)cc2)ccccc1=O 57797,C1(C(N2CC(C)(CCO)C2)=O)(NC(C2CCC3CC23)=O)CCOCC1 57798,C1(NC(c2nnnn2Cc2cccc(F)c2)C(C)C2CC2)CC(=O)N(C(F)F)C1 57799,c1(C(=O)NCC2OCCN(C(C3CCC(C)CC3)=O)C2)c(F)ccc2nc[nH]c12 57800,c1(OC)cccc(C(=O)NC2CN(C(C3(C(F)(F)F)CCC3)=O)CCC2O)c1F 57801,N1(C(c2c(C)nn(C)c2C(F)F)=O)CC(C2CN(C(=O)C(C)OCC(C)C)C2)C1 57802,c1(CCCCC)nc(C(=O)NCC(O)CCNC(=O)C(O)Cn2cncn2)cs1 57803,N1(C(CC2N(CC)CCC2)=O)CCC(CO)(CNC(c2cnnn2CC)=O)C1 57804,Cc1c(NC(c2cccc(C(C)C)n2)c2nnnn2C(C)(C)C)cccc1F 57805,C1(CNC(C2CC(C)OC2)=O)CCCCN(C(c2ccnc(Cl)c2F)=O)C1 57806,C12(NC(C(CN(CC)CC)F)=O)CC1CN(C(c1cc(C)[nH]n1)=O)C2 57807,N1(C(C(=O)NCc2c(C)nn(C(C)C)c2C)=O)CC2CCCOC2C1 57808,c1(C(N2CCCC(C)(NC(=O)C=CCF)C2)=O)cnc2c(c1)OCCN2 57809,Cc1ncc(CNC(=O)CC2CC(NC(=O)CC3CC4(CCC4)C3)C2(C)C)n1C 57810,N1(C(c2c(NC(N)=O)cncc2)=O)CCN(C(C2C=CCC2)=O)C(CO)C1 57811,c1(C(=O)NCC2(OC)CN(C(c3cc(Cl)ncc3N)=O)C2)cccc2nccn12 57812,C12(NC(c3cc(C)n(CCO)n3)=O)CCCN(C(=O)CS(N)(=O)=O)CC1C2 57813,c1(C(=O)NCCCN(C(=O)CCc2cncn2C)CC)cccc2c1OCC2C 57814,N1(C(C(OC)OC)=O)CCC2(CCC(CNC(C3CC4CC(=O)C3C4)=O)O2)CC1 57815,c1(N(CC(F)C2CCC2)C)ccc(S(=O)(=O)N2CCC(c3ccccc3)C2)cc1F 57816,C12(CCC)CCCN(C(=NCCCCC(C)(F)F)NC(C)C1)C2 57817,Cc1ccccc1C(C(=O)NCC1CCC12CCC2)NC(=O)OC(C)(C)C 57818,C1(N(C(C2C(=C)CC2)=O)CCOC)CCN(C(c2nccn2C)=O)CC1 57819,Cc1cc(C#N)nc(N2CCCC(NC(c3ccccc3C3(C)CC3)=O)C2C)n1 57820,Cn1ncc2ncc(C(N3CCC4(CCCN4C(C4CC4F)=O)C3)=O)cc12 57821,CCS(=O)(=O)CCn1nc(-c2ccc(F)cc2)nc1C12CCC(C1)OC2 57822,C(C(C)C(F)C(=O)N(C)C(c1cccs1)C)NC(C(C)=C(C)C)=O 57823,Cc1onc(CO)c1C(=O)NCC1C(CNC(C2CCOC(C)C2)=O)C1(F)F 57824,C1(CNC(C(C(C)C)C)=O)CCN(C(c2ccc(-c3cccs3)o2)=O)CC1(F)F 57825,C1(CC(=O)NC)CN(C(=O)C2=CCSC2)CCN1C(=O)C=C(C)C(C)(C)C 57826,C1(N(C(=O)CSCc2ccncc2)C)CC2CC1N(C(=O)C(F)=C1CCC1)C2 57827,c1(N2CCC(C(CN(C)C)Cc3ccccc3)C2)ccc(F)cc1I 57828,Cc1cc(C(N2CCSCC2CCNC(=O)C(C)OCC(C)C)=O)c(C)n1C 57829,CN1CCCCC1CCC(=O)NCC(C)(C)C(=O)NC1CCCC1 57830,N1(C(CC(CC)SC)=O)CCCC(C)(NC(c2oc(C)cc2C)=O)C1 57831,C#CCCC(O)C(=O)NCC1(CCNC(=O)C(C)Cc2ccccc2Cl)CC1 57832,S(=O)(=O)(c1ccc(NC2CCCC2CCO)cc1Cl)NCc1c(C)nns1 57833,C1(CNC(C2C(CCOC)C2)=O)CCN(C(c2ccnn(C)c2=O)=O)CC1(F)F 57834,N1(C(C)=O)CC2(C1)CN(C(=O)Cc1cnc(C)n1C)C2.C1(C)C(=O)N1C(C)=O 57835,C1(NC(CC=C(C)C)=O)CC2(CCN(C(C3CC3Br)=O)CC2)C1 57836,C1(CNC(c2cc(C)c(F)cn2)=O)CN(C(C2(COC(C)C)CC2)=O)CCC1C 57837,c1(CN2CCCC(C(N(CCCC)CCOC)=O)CC2)nc2ccccc2n1C 57838,c1(C(=O)NCC(CC)NC(=O)C(C)(C)C(C)C)nn(C)c(Cl)c1Cl 57839,c1(C(=O)NCC(N2CCN(Cc3ccccc3CO)CC2)=O)ccc([N+](=O)[O-])o1 57840,C1(C)(CNC(Cc2ccn(CC)n2)=O)CC(F)(F)CN1c1nc(C2CC2)ns1.NC 57841,Cc1c(NC(=O)C(O)CC(F)(F)F)cc(F)cc1-c1ccc(OC(F)(F)F)cc1F 57842,Cc1cc(C(=O)NC(CC(=O)NCC(F)(F)Cl)C2CC2)cnc1O 57843,CCCC(CNC(c1[nH]nnc1C)=O)C(=O)NC1CC12CC(OC)C2 57844,c1(CNC(CC(=O)O)Cc2cn(-c3ccncc3)nn2)ccc([N+](=O)[O-])cc1 57845,C1(CCC)CN(C(C2CC2C)=O)CCN1C(=O)CNC(=O)C(F)(F)F 57846,c1(C(=O)NCC(CC=C)NC(c2cc(CC)on2)=O)cc2ccsc2n1C 57847,C1(C(=O)NCC(CNC(Cc2cc(CC)no2)=O)(C)O)CCC([N+](=O)[O-])CC1 57848,N1(CCCCCNC(C(CC)C)=O)CCC(n2cc(-c3ncc(F)cn3)nn2)CC1 57849,C(c1ccc(Cl)c(C(F)(F)F)c1)=CC(=O)NC(CN(C(=O)C(C)OC)CC)C 57850,C1(NC(CC(C=C)(C)C)=O)CCC(O)CN(C(=O)CCOCC2CCC2)C1 57851,c1(NCC(N2CCC2c2ccccc2)C)ccc(F)cc1F 57852,CCC(C)CC(C(=O)N1CCC(N2CCC2)C1)NC(c1n[nH]cc1C)=O 57853,C1(NC(C2C(C)(COC)C2)=O)CN(C(=O)CCc2cccc(OC)c2)CC1O 57854,C12(C(=O)N)CCCN1CCC2.c1(CSCC(N)=O)ccc(C(N2CCC2CC)=O)cc1 57855,c1(NC)ccc(C(=O)NCCn2cc(C(=O)NCC3CCOC3)cn2)cc1 57856,C1(OCCC)CCN(C(c2c[nH]nc2CNC(=O)C(c2cnn(C)c2)O)=O)CC1 57857,C1(NC(CSc2nc(C)[nH]n2)=O)CCN(C(C2CC3C=CC2O3)=O)CC(C)(C)C1 57858,N1(C(CSc2cn(C)nc2)=O)CCC2CCN(C(=O)CC3CC3(C)C)CC12 57859,Cn1c(C(=O)NC2CCN(C(=O)CCC3CC3(Cl)Cl)CC2)nnc1S 57860,c1(C(C(=O)NCC(CC=C)NC(=O)Cc2ncc(C)s2)(C)C)cc(C)cc(C)c1 57861,N1(C(C(C(C)C)n2ncc(C)c2)=O)CC2(C1)CN(C(C1CCCCS1)=O)C2 57862,c1(C(N2CC(C(=O)OC)N(C(C3CC(F)C(=O)N3)=O)CC2)=O)ccc(F)c(F)c1 57863,C1(NC(CCC)=O)CCCC(NC(=O)CCOCC(F)(F)F)C1.C1CN(CC)CC1 57864,C(CNC(c1ccc(C(C)C)cc1)C)(CS(C)(=O)=O)OCC 57865,C1(C(=O)NCCCN(C(=O)CC2(C)CCC2)C)CC2(CSC2)C1 57866,C(=O)(C(CC)(CC)CCOC)N1CCC(C)(NC(c2cc(CC)cc(C)c2)=O)C1 57867,c1(C(=O)Nc2ccc(C#C)c(Cl)c2)ccc(S(=O)(=O)C2CC2)nc1 57868,C=C(Cl)C(C)(C)C(=O)NC1CCC(NC(=O)Cc2cc(Cl)n(C)n2)CC1 57869,Cc1cc(C(=O)NCCC2CC(NC(=O)C(F)CC3CCOC3)C2)nc(C)c1 57870,C1(NC(c2scc(C)c2Cl)=O)CCC2CCN(C(C3CC3(F)F)=O)C12 57871,c1(C(=O)NCC2CCN(C(=O)C(O)C(F)F)C23CC3)cc(O)cc(F)c1 57872,C12(C(N(C3CN(C(C(C4CCOCC4)OC)=O)C3)C)=O)CC3CC(CC(C3)C1)C2 57873,CC(CNC(=O)CC1CCC(O)C1)C(F)C(=O)N(C)Cc1ncn(C)n1 57874,Cc1cc(NC(C2CN(C(=O)CN(C)C(c3ccccc3)=O)C2)=O)n(C(C)(C)C)n1 57875,c1(C(=O)NCC(CCOC)NC(=O)CC(C)C)cccc(C(=O)N(C)C)n1 57876,N1(C(=O)CC2CC3(CCC3)CO2)CC2OCCN(C(c3ns[nH]c3=O)=O)C2C1 57877,c1(C(N2CC(NC(c3ccc(SC)cc3)=O)C(F)CC2)=O)c(F)ccc(F)c1O 57878,C=C1CCN(C(c2cn(C)cc2C)=O)C(C(=O)NC(CN2CCCC2)CC)C1 57879,C1(C(=O)NCc2c(C)cnn2C)CC(N=[N+]=[N-])CN1C(c1cc(F)n(C)n1)=O 57880,S(=O)(=O)(c1ccc(O)c([N+](=O)[O-])c1)N(C(=O)CCCS(=O)(=O)N1CCOCC1)C 57881,c1(C(N2CCCCc3ccc(I)cc32)=O)cc(F)c(Br)c([N+](=O)[O-])c1Cl 57882,c1(OC)ccc2c(NC(=O)C(=O)NCC(C)(C3CCC3)NC3CC3)c[nH]c2c1 57883,CC#CCCCC(=O)NC1COCC1C(N1CC(OC)CC(C)C1)=O 57884,Cc1cc(C)c(C(=O)NC2CCC(CNC(=O)C=Cc3cn(C)nn3)CC2)o1 57885,CN1CC(N(C)C(C2CSC(C(F)(F)F)C2)=O)CC1=O 57886,c1(N(C)C)cccnc1C(=O)NC(C)CC(C)NC(=O)COC(C)(C)C 57887,C1(O)(C(C2CC2)NC(=O)Cc2ccsc2)CCN(C(=O)C=Cc2ccccc2)C1 57888,N1(C(C)=O)CC2CC2(C(=O)NC2(c3cccnc3)CC2)C1.N12CC(C1)C2=O 57889,c1(C(=O)NC(CNC(c2cc(C(C)C)nn2C)=O)CO)ccc(N)cc1O 57890,c1(NC(C)CN(C(=O)C2=CCSC2)C)ncnc2c1nnn2C1CC1 57891,c1(C(=O)NCC2(C)C(C)CN(C(=O)CC3CC(F)C3)C2)cc2c(s1)CCOC2 57892,N1(C(c2cc(C)sc2)=O)CCCOC(CNC(C2CCCN(C)C2)=O)C1 57893,O=S(=O)(c1ccc(=NCC2(CO)CC2)[nH]c1)NCC12CC(CCO1)C2 57894,c1(CC)noc(C)c1C(N1CCCC1C(O)CO)=O.c12csc(c1)C(=O)NC2 57895,N1(C(C2C(CCC)C2)=O)CC2(C1)CN(C(c1cc(CC)ccn1)=O)CCO2 57896,C(CCCCC#N)(c1n(CC(=C)C)nnn1)(C1CC1)Nc1ccc(Br)c(Cl)c1 57897,c1(OC)sccc1C(=O)NCc1c[nH]nc1C(=O)NC1(C(C)(F)F)CC1 57898,c1(N2CC(C)(C)C2CNC(=O)CC2CC3(CCC3)C2)ccc(C#N)c(C(F)(F)F)n1 57899,CC12CCC(C(=O)NCC3CCN3C(=O)CCCOc3ccccc3)(CC1)CO2 57900,c1(OC)ccc(CNC2CCC(C(=O)NCc3ncn(C)n3)C2)c(Br)n1 57901,c1(C(c2nnnn2CC(F)F)OC(C)(C)C)ccnn1CCF.c1(C)csc(Br)c1.C 57902,c1(CC)[nH]c(C(=O)NC2CC(CO)N(C(=O)Cc3nonc3C)C2)nc1Cl 57903,c1(C(N2CC(NC(C(CSC)O)=O)C(C)C2)=O)coc2c(C)cccc12 57904,C1(NC(C2CC3C=CC2C3)=O)CC(=O)N(C2CCCC2)C1.C12CCC1C(=O)NC2 57905,C(c1ccc(F)c2ccccc12)=CC(N1CC(NC(CC2C(C)C2)=O)C1)=O 57906,c1(C(=O)OC)c(C)ccc(NC(=O)NCCC2CC2C(F)(F)F)c1C 57907,Cc1ccc(CC(=O)NC2CC2CNC(=O)C(C)CN(C)C)cc1F 57908,C(=O)(C1CCCc2nccn21)N1CC(F)(CNC(c2ncc(OC)cn2)=O)C1 57909,c1(C(N(CCCOCCNC(C(C)C(F)F)=O)C)=O)n[nH]c2cccnc12 57910,c1(CC)ccoc1C(=O)NC1CCC(CNC(C2(CCO)CC2)=O)C1 57911,CC1CC(C(N2CCC2CC(C)(C)CNC(C2CN(C)CO2)=O)=O)C(=O)O1 57912,CCCC(C(=O)N1CC(NC(C2CC(C)CO2)=O)C(C)C1)N(C)C 57913,C1(CNC(=O)Cc2cncnc2)CC2CCC(C1)N2C(C1CC12CCOSC2)=O 57914,C(=O)(CS(C)(=O)=O)NCC(C)N(C(=O)CCC(=O)C1CC1)C 57915,c1(NC(C2CCN(Cc3ccno3)C2)=O)cc(C(F)(F)F)cc(Br)c1 57916,C1(Cc2cn(C(c3ccncc3F)C)nn2)OCCOC1(C)C.C1(C)CC1 57917,N1(C(C(C)c2ccco2)=O)CCCC12CCN(C(=O)CCC(C)(C)N(C)C)CC2 57918,N#Cc1cc(Cl)c(C(=O)NCC2CC2NC(c2c[nH]nc2-c2ccncc2)=O)s1 57919,c1(C(=O)NC(CNC(c2cn(CCC=C)nn2)=O)CC)noc2ncccc12 57920,c1(N(CC(=O)Nc2c(C)nn(C(F)F)c2C)C)cccc2ccccc12 57921,C=CC1(NC(C2CC23CCN(C(=O)Cn2nccn2)C3)=O)CCOCC1 57922,N1(C(Cc2cc(CC)no2)=O)CCC(C(=O)NC)(C(=O)Nc2cncnc2O)C1 57923,N1(Cc2c(C)ncs2)CCCCC(NC(=O)C=Cc2ccnn2C)C1 57924,C(=O)(CCCCCCCCSC)NC1C(NC(CC(C=C)CC)=O)COCC1 57925,c1(CC(=O)NC(CNC(C(C)=CC2CC2)=O)C)cccc(F)c1 57926,c1(C(=O)NCCCNC(C2C(OC)CC2)=O)c(OC)ccc(Cl)c1F 57927,CC(C)(C)C(O)C(=O)NCC1CCCCN1C(=O)Cc1n[nH]c(=N)s1 57928,c1(C(=O)NCC2CCN(C(C=CCCC)=O)C2)ccc(F)c(C(C)(C)F)c1 57929,N1(c2cccc(C)c2)N=C(C(=O)N(C)CCNC(c2ccn(C)c2)=O)CCC1=O 57930,c1(N(CCC)CCNC(c2coc(C)c2)=O)ncccc1[N+](=O)[O-] 57931,C1CCCCN1CCc1csc(N(CC(CCC)OC)C)n1.C(=O)O 57932,C(=O)(C(C)(C)C(=O)OC)NCCCNC(c1nnn(COCC)c1N)=O 57933,c1(C(=O)NCC(CNC(C(C)=C2CCC2)=O)(C)C)n[nH]c2ccc([N+](=O)[O-])cc12 57934,C12(CNC(=O)CN3CCCCC3=O)CCC(CC1)N2C(=O)C(c1ccccc1)F 57935,CN1CCOCC1C(N1CC2CC2(C(N2CCC2c2ccccc2)=O)C1)=O 57936,C1(NC(c2cnc(C(C)O)s2)=O)CC2CCC(C1)N2C(C1COC2(CCC2)C1)=O 57937,N(C(=NCC1CC(F)(F)C1)NCC(=O)NC1CCC1)CC(c1ccccc1)(C)O 57938,c1(CC)ccc(C)c(C(=O)NC2CCN(C(c3c(F)cncc3Cl)=O)CC2C)c1 57939,C1(CC(N)=O)CCCN1C(C1COC(CNC2CC2)C1)=O.C12(CCC1)C(=O)NC2 57940,C1(CC)CN(C(c2cnccc2C)=O)CCC1NC(c1csc(=N)[nH]1)=O 57941,C1N=C2NC(=NC(C)Sc3ccccc31)c1sccc1N2.C(=O)(N(C)C)OC 57942,S(=O)(=O)(c1c(Br)cccc1[N+](=O)[O-])N1C(C)CCC(C)(C)C1 57943,C1(OC)CCN(C(C2CCOCCN2C(C2CCSCC2)=O)=O)C12CCC2 57944,C12(NC(C(COC)OC)=O)CCCC1N(C(c1cc(C)cc(Br)c1O)=O)CC2 57945,c1(C(=O)NC2CCN(C(C3(C)ON=C(C)C3)=O)C2)ccc2c(ccn2C)c1 57946,c1(N2CCC(N(C(C(C)Cc3cnc[nH]3)=O)C)C2)ncc2c(n1)CCOC2 57947,C1(C(N(C2C3CN(C(=O)Cc4cc(F)ccc4F)CC23)C)=O)CC2CCC(C1)S2 57948,c1(CC(=O)NC(CC)CNC(=O)C(C)OC)cccc(C(F)(F)F)n1 57949,c1(-c2nnc(Nc3ccc(CCCC)cc3)o2)ccc2c(c1)N(C)C(=O)C2 57950,C1(C2(O)CN(C(C3CN(C)C(=O)N3)=O)C2)(CNC(c2ccc(C)cn2)=O)CC1 57951,C=CC(C)C(C)C(=O)N1CCC(CNC(c2cccc(Br)c2N)=O)CC1 57952,N1(C(CCNS(C)(=O)=O)=O)CCN(C(c2ccsc2)=O)C(C2CCC2)C1 57953,c1(OC)ccncc1C(=O)NCCC1(C)CCN(C(=O)Cc2n[nH]c(C)n2)C1 57954,C1(C(=O)NCC2CN(C(C3(CN(C)C)CC3)=O)C2)C2CCC3(COC(=O)C13)O2 57955,Cc1nc(C)c(CN2CCCCC2CNC(C2CCS(=O)(=O)C2)=O)[nH]1 57956,c1(-c2n(C(C)C3CC3c3ccccc3)nc(CCC(F)(F)F)n2)cc2ccsc2s1 57957,CC1(C(=O)NCC2CC(C(=O)NCCn3ncccc3=O)C2)C=CCCC1 57958,C1(CN(CCC)CCN(C)C)CCCN(C(c2cccc(Br)c2)=O)C1 57959,C12CCN(CC1)C2.CC1CCC(C(=O)NCc2cnn(-c3nccnc3Br)c2)C1 57960,N1(C(Cn2cc(CC)nn2)=O)C2CCC1CC(CNC(C1(C)CCC(C)C1)=O)C2 57961,C12(C(=O)NC3CC(NC(C(C)n4cnnn4)=O)C3)CC3CC(C(=O)N1)C2C3 57962,CC1(C)C(NC(c2ccc(C(F)(F)F)nc2)=O)CCN1C(=O)C(F)C(F)(F)F 57963,C1(C(N(CC(O)C(F)(F)F)C)=O)CC2CCC(C1)N2C(=O)CC1CCC(=O)O1 57964,CCC(CNC(=O)CC1CCNC1=O)(CC)C(=O)N(C1CC(C)C1)C 57965,C(=O)(C(CO)C(C)(C)C)NCC(CNC(C=C(COC)C)=O)OC 57966,c1(C(=O)NCC2CCC(NC(=O)C3=C(Cl)CCC3)C2)ccc2c(c1)CC(=O)NC2 57967,C1(NC(C(C)SCCCC)=O)CCN(C(c2cnc(C3CC3)o2)=O)CC(O)C1 57968,C1(N(C)C)CC(CC(=O)NC(C(=O)NCCSC(F)F)C2CCOC2)C1 57969,c1(C(C(N2CCC(n3ccnc3)C2)C)=O)ccc(F)cc1 57970,n1(CC)cc(C(=O)NCC(CCNC(=O)CCC2(O)CCC2)OC)nn1 57971,C1(F)(C(N2C3CN(C(C)=O)CC32)=O)CCCC=C1F 57972,CC(C)CCC(F)C(=O)N1CCC(C(=O)NCCCc2cn[nH]c2)C1(C)C 57973,C(=O)(C(C)(C)S(C)(=O)=O)N(C(CNC(=O)C(=O)Nc1ccccc1)CO)C 57974,CS(=O)C1CN(C(c2sccc2CNC(=O)CN2C(=O)CNC2=O)=O)C1 57975,c1(CC(=O)NC2(CF)CCN(C(CCNS(C)(=O)=O)=O)C2)cccc(Cl)c1Cl 57976,N1(C(C2CC(C(=O)OC)C2)=O)CCCCC1CC(=O)NC(=O)C1CC1 57977,CC12CCOC(C(=O)NC3CCN(C(c4scnc4Cl)=O)CC3O)(C1)C2 57978,C1(=CC(=O)NC(C2CC(NC(C3CCCC3F)=O)C2)C)CCCCC1 57979,N1(C(C=C(CC)CC)=O)CCC(C(C)CNC(=O)COCCCOC)CC1 57980,c1(C(N(CCNC(C(C(C)O)C)=O)CC2CC2)=O)cccn2cncc12 57981,C1(OC)CN(C)C(C)(C(=O)NCC2CN(C(=O)CCc3cnn[nH]3)CCC2C)C1 57982,C(=O)(CCCCC(C)(C)C)NCC1(CNC(C2(NC(C)=O)CCCC2)=O)CCC1 57983,Cc1cccc(C(C)NC(c2cccc(Br)c2Cl)C)c1C 57984,N1(C(Cn2c(C)ncc2)=O)CCC(C)(C(N2CCC(O)C(C)C2)=O)CC1 57985,CC(CS(C)(=O)=O)C(=O)NC(=O)C1CC1.C12CN(C1)C2=O 57986,c1(NCCCNC(C2CN(C(C)=O)C2)=O)cnc2n1CCCC2C 57987,N1(C(CC(C(=C)C)OCC)=O)CCC(C(=O)OC)C(C2CC2)C1 57988,Cc1cccc2c(C(=O)NCC3CCCN(C(C4CC(C)CO4)=O)CC3)cnn12 57989,C=C(C)CC(C(=O)N1CC2C(NC(c3ccc(OCCC)nc3)=O)C2C1)OC 57990,C1(O)(CNC(CCCC#CC)=O)CCCN(C(=O)CCC(=O)N2CCOCC2)CC1 57991,N1(C(C(C)C)=O)CCC(C(=O)NCc2ccnc(Cl)c2)CC1 57992,N1(C(=O)NCC2CCC(C)O2)CCN(Cc2ccccc2)c2ccccc21 57993,N1(c2nc(NCc3scc(CC)n3)nc(C)c2)CCC(O)C(C)(C)C1 57994,C1(C(N2CCC(C(=O)OC)C2)=O)(NC(C2N(CC)CCC2)=O)CCN(C)C1 57995,c1(C(N(C(CC2CCC2)C(=O)NCCSC)CC)=O)ccncc1C(=O)OC 57996,CCC(C)(C(=O)N1CCC(CN(C(C2COCCC2(F)F)=O)C2CC2)CC1)C(N)=O 57997,c1(C(C)NCc2cn(CC(O)Cc3cscc3Br)nn2)c(F)cccc1F 57998,CC1(CNC(C2CC(CF)C2)=O)CCC(NC(=O)CNC(=O)C2CC2)CC1 57999,C12(CNC(=O)CCc3cccs3)CC(CO1)N(C(=O)Cn1nnc(C3CC3)n1)C2 58000,C1(C)(CC(=O)NC2CN(C(C(COC)NC(=O)OC(C)(C)C)=O)C2)CCCCC1 58001,c1(C(N2CC3C(C(=O)NC)C3C2)=O)c(Br)ccc2[nH]c(C(=O)OC)cc12 58002,N1(C(C2CCCCO2)=O)CCC2CN(C(=O)CCc3ccccc3F)CC2C1 58003,CS(=O)C=CC(=O)NCC1(CNC(=O)CSc2cn[nH]c2)CC12CCC2 58004,c1(C(N2CC3C(CNC(C4C(C(C)C)CCC4)=O)(C3)C2)=O)n[nH]c2c1COCC2 58005,C(=O)(CCC(C)(F)F)NCC(CNC(C1(CC)CC(F)(F)C1)=O)(C)C 58006,C1(CC(=O)N(C)CCN(C)C(C2(CCO)CC2)=O)CCC2(CCC2)O1 58007,c1(C(=O)NCC(CN(C(=O)CCNS(C)(=O)=O)C)O)cnn(C)c1 58008,Cn1ccn2ncc(C(=O)NC3CC(CNC(=O)CC4CCCO4)C3(C)C)c12 58009,N1(C(c2c(C)c[nH]n2)=O)CCC(CCNC(c2conc2C(C)(C)C)=O)CC1C 58010,c1(C(=O)NC(CNC(C2C(=C)C2)=O)C2CC2)cc(F)c(OC)c(Cl)c1 58011,CC1CN(C(c2cnc(F)c(Cl)c2)=O)CCC1CNC(C1(C(N)=O)CCC1)=O 58012,C1(CCC(=O)N(C2C3CN(C(C4(C)CCCOC4)=O)CC23)C)CCCCCC1 58013,C1(F)(C(=O)NC(COCCOCC(=O)C2CC2)C2CC2)CC2(CCCCC2)C1 58014,N1(C(C(C)c2cc[nH]n2)=O)CCCCCCC1C(=O)NCC(F)F 58015,c1(C(N2C(C)C(NC(c3ncncc3Cl)=O)CC2)=O)cc2n(n1)CCCC2O 58016,N1(C(C2CCC(C(=O)OC)C2)=O)CC(C2(NC(c3ccc(Cl)cc3OC)=O)CC2)C1 58017,CC1CCC(CNC(=O)Cc2ccc(F)nc2)CN1C(c1cncn1C)=O 58018,C1(C(=O)NCC(CNC(C2(C=C)CCC2)=O)(C)O)CCOC1(C)C 58019,CC1(C)CN(C(=O)C(N2CCC3(CO)CC3C2)=O)CCC1C(c1ccccc1)=O 58020,C1(NC(c2ccc(F)c(Cl)c2)=O)CC2CN(C(c3cnco3)=O)CC12 58021,c1(C(=O)NCC2(O)CC(C(NOCC(C)O)=O)C2)cc[n+]([O-])cc1 58022,C1(CC(C)NC(C(=O)NC(C)C)=O)CCCN1C(C1CC1C(F)(F)F)=O 58023,c1(C(=O)NCC2(C(C)(C)O)CN(C(CC)=O)C2)cnc2c(Cl)cccn12 58024,N1(C(C2C(C(C)C)C2)=O)CCN(C(=O)Cc2c(Br)cnn2C)C(CCO)C1 58025,c1(Sc2nc(-c3ccccc3)[nH]n2)nnc(C2CCCC2)n1CCCCCCCO 58026,C12(NC(=O)CCc3ccoc3)CCCC1(F)CN(C(C13CCC(F)(CC1)C3)=O)C2 58027,N1(N(C(CSCCOC)=O)C(C)C)CCOC(C)C1.C(C=O)NCC 58028,N1(C(COC2(C)CCOCC2)=O)CC=C(CCNC(C2CCC(=O)O2)=O)CC1 58029,Cc1nc(CN=c2cc(C(C)(C)C)nc[nH]2)cn(C)c1=O 58030,c1(CC(=O)NCCN(C2CCCCC2)C(c2cnc(C)[nH]2)=O)ccccc1Cl 58031,C12(C(=O)NC3CC4(CCC4)C3)CCC(CC1)CC2.C12CC1C(=O)NC2 58032,N1(C(C2OCC(=O)C2)=O)CCCOC(CNc2nccc(CO)n2)C1 58033,C1(NC(CC2(C)OCCO2)=O)C2CN(CC(F)F)CC12.C12CCCN(C1)CCC2 58034,CC(C)C(O)C(C)C(=O)OCCCC(C)CN(C)C 58035,C1(C(C)C)CN(C(=O)CCC(=O)C2CC2)CC1C(=O)NC(C)C1CC1 58036,c1(CCC(=O)NCC2C(NC(C(Cn3ccc(C)n3)C)=O)C2)ccc(C#N)cc1 58037,c1(C(=O)NCC(CC)(C)NC(c2c[nH]nc2OC)=O)cc(C)cc(Cl)c1 58038,C1(NC(c2cc(C)sn2)=O)CCC12CCN(C(c1cc(Cl)c(F)cc1Cl)=O)CC2 58039,CC1=NN(C)C(=O)C1CC(N1C2CCC1C(NC(c1cccc(F)c1Cl)=O)C2)=O 58040,C1(CN2CC(n3cc(CC=C)nn3)C2)CCCN(C(C2(C3(C)CC3)CC2)=O)C1 58041,c1(C(=O)NC(CNC(C(CC)O)=O)C2CCC2)cc(C)cc([N+](=O)[O-])c1 58042,c1(C2(C)CC2)cc[nH]c1C(=O)NCC1CC(CNC(=O)Cn2cccn2)C1 58043,Cc1cncc(C(N2CC(O)(C3CCCN3C(=O)CN3CCN(C)CC3)C2)=O)n1 58044,CC(CCCCO)NC(=O)C(CCF)NC(c1cncc(O)c1)=O 58045,c1(C(N2CCCC(Br)C2)=O)ccc(NCCc2ccncc2Cl)cc1 58046,C1(C(N2CC(CNC(C(COC)C)=O)CC2(C)C)=O)CN2CCCN1CC2 58047,N1(C(c2c(-n3c(C)ncc3)cccc2)=O)CC(CO)OC2(CCC2)C1 58048,c1(CC(=O)NC(C2CCCCN2C(c2ccc(CO)nc2)=O)C)cccnc1Cl 58049,C1(NC(c2nc(C(C)(C)C)oc2)=O)CCCCN(C(=O)C(F)(F)C2(O)CCC2)C1 58050,c1(C(=O)NC(C(C)NC(=O)CCNC(=O)NC2CCOCC2)CO)cccnc1O 58051,Cc1ccc(O)c(C(=O)NCC2(CNC(C3(C)CC4(CCC4)C3)=O)CCCC2)c1 58052,C12(C(=O)NCC(C3CC3)SC)CC(C)(CN1C(=O)CCn1ccnn1)C2 58053,N1(C(C=CCC)=O)CCC2(CCCC2NC(c2cnn3c2OCC3)=O)CC1 58054,C1(C(N2CCCCCC(NC(c3nnc(C)s3)=O)C2)=O)Cc2cccnc2C1 58055,C(=O)(CC(O)C(C)C)NC(CC)CC(=O)NCc1nc(C)c(C)s1 58056,N1(C(Cc2cc(C)sc2C)=O)CCC(C2CN(C(c3ccns3)=O)C2)CC1 58057,c1(CCC(=O)NCc2ccc(CCCCCCC)cc2)ccc(O)c(O)c1.C(C)(=O)O 58058,CC1CCC(NC(c2ccc(CO)c(Cl)c2)=O)CN1C(=O)CCC1CCC1 58059,C(=O)(C(F)C(C)(C)O)NCCC1(O)CN(C(CC2ON=C(CC)C2)=O)C1 58060,[N-]=[N+]=Nc1ccccc1C(=O)NC1CC2CC1N(C(=O)CCC(N)=O)C2 58061,c12ncoc1CCNC2=O.C1(C(=O)NCCC(=O)NC2CC2)CCCCC1 58062,Cc1cccc(Cl)c1CN(C(c1ncccc1-c1nn[nH]n1)=O)C1CC1 58063,Cn1nc(O)cc1C(=O)OCc1ccccn1.c12nccn1C2 58064,Cc1cnc(C(=O)NC2CCC(C(=O)NCc3ccnn3C)C2)cc1C 58065,c1(C(=O)NC23CCCC(NC(C(C)C)=O)(C2)C3)cc(=O)n2nccc2[nH]1 58066,N1(C(C(C)N(C)C)=O)CCN(CCCNC(=O)C(C)OCc2nccn2C)CC1 58067,c1(C(=O)NCCN(C)C(C2CCC2c2nncn2C)=O)ccc(F)c(Br)c1 58068,C1(NC(c2ccc(OC)s2)=O)CCCC(NC(c2ccnc(C(F)F)c2)=O)CC1 58069,Cc1cc(C(=O)NC(c2cnn(C)c2)C)cc(C)c1O 58070,C(=O)(C1=Cc2ccccc2C1C)NCCN1CCCN(C(CCCCOC)=O)CC1 58071,c1(C(N2CCCN(C(c3nc(CC)oc3)=O)CCC2)=O)cccc2cnccc12 58072,CC1CC(C)N(C(c2ccc3cc[nH]c3n2)=O)CCN1C(C12COCC(C1)C2)=O 58073,Cc1ncc(C=CC(=O)NCC2CN(C(c3cc(F)cc(F)c3O)=O)C2)c(O)n1 58074,N1(C(c2c(CC)cco2)=O)C2CCC1C(C(=O)NCCCc1nc(C)no1)C2 58075,CC1(C)CC(CNC(=O)C2=CSCS2)CN1C(=O)C=CC(c1ccccc1)=O 58076,Cc1cncc(C(=O)NC(C2CC2C(N2CCOC(CN=[N+]=[N-])C2)=O)C)n1 58077,S(=O)(=O)(c1cnc(Cl)nc1)NC1C(C(=O)Nc2c(OC)ccc(Cl)c2)CCC1 58078,C1(N(C(c2cnc(CC)s2)=O)C)CN(C(C2CC2C(C)(F)F)=O)CC1(C)C 58079,c1(NC(N(CC)CC2CC(OC(C)(C)C)C2)=O)cc(C)n(C)n1 58080,O=C1NC(=O)C2(CC(C(=O)NCC3CN(C(c4ccc(F)nc4F)=O)C3)C2)N1 58081,c1(OCC)cnc(NC(C2(CNC(=O)C(O)C3CCCC3)CC2)=O)c(Cl)c1 58082,CCCCC(C(=O)NCCC1CN(C(=O)C(C)(O)C2CCOC2)C1)NC(=O)OC 58083,c1(N(C(=O)CC(C2CC2)C2CC2)C)cc(NC(CCC)CC)nc(C)n1 58084,C1(O)(CNC(C(C)n2ccnc2)=O)CCN(C(=O)C(F)CC2CC(F)(F)C2)CC1 58085,C1(NC(C(C)OCCC=C)=O)CC2(CCCN(C(=O)C(C)(C)CNC(C)=O)C2)C1 58086,C(=O)(CCCCc1cnn[nH]1)NCC1(CCNC(CCc2nnc(C)o2)=O)CC1 58087,Cc1cc(=NC(=O)C(=O)NC2CC3CN(C(=O)CC=C(Cl)Cl)CC3C2)[nH]o1 58088,CCCC(C(=O)NC1(CO)CN(C(c2ccc(N)cc2[N+](=O)[O-])=O)C1)S(N)(=O)=O 58089,C1(C(=O)NC(c2ncn(C)n2)C)CC12CCN(C(=O)C(C)N1CCCC1)CC2 58090,c1(OC)c(F)cc(S(=O)(=O)N(C)CC2CCCC2(C)C)cc1Br 58091,CC1(C)CC(O)(CC(=O)NCCCCCCNC(c2cc(N)cnc2Cl)=O)CO1 58092,C(=O)(C(C)(C)CCNC(=O)CC1CCCNC1=O)N(CCC(N)=O)C 58093,C1(N(C)C(c2ccccc2O)=O)CCN(CCNC(=O)C=C2CCOCC2)CC1 58094,CC#CCCC(=O)NCCCN(C(c1oc(C)nc1-c1ccccc1)=O)CC 58095,c1(C(=O)NCC(C)(C)NC(C=CC)=O)nc(CC(F)(F)F)sc1C 58096,C12(C(N(c3cn(CC)nc3)C)=O)CCCC1CCN2C(c1cnn(C)c1C)=O 58097,CCC(CC(C)C)C(=O)NCC1CC2CCC1N2C(=O)CCn1cccn1 58098,c1(OC)ccc(C(=O)NC2CC2CNC(=O)CC(C)F)c(NC(C2CCCC2)=O)c1 58099,C1(C(=O)OC)CC12CN(C(C13CC1CCN3C(c1cc(C)sc1C)=O)=O)C2 58100,C12(C(=O)NCC3CN(C(c4scc(C)c4C)=O)CC3(F)F)CCCCN1CCC2 58101,C(CC(C)C)(C(=O)NCC(c1cnn(C)c1)C)OCc1ccc(C)cc1 58102,c1(C(=O)NC(CNC(CCOC(C)C)=O)C2CC2)occc1F 58103,Cn1ccc(=NC(=O)CCC2CCN(C(c3cc(CC4CC4)on3)=O)CC2)[nH]1 58104,C1(C(N2CC(CC)(CC)C2)=O)CN(C(=O)C=C(C)C(F)F)CC(C)(C)C1 58105,C1(CC(=O)OCC)CCCCC1C(=O)NC1CN(C(C2CC=CCC2)=O)C1 58106,n1(CC(C)(C)C)nc(-c2cncc(F)c2)nc1CCn1cnccc1=O 58107,C1(F)(CNC(CC2CCC(C)C2)=O)CCN(C(=O)Cc2csc(C(C)C)n2)CC1 58108,C1(CC(=O)NC2CCCC2CNC(=O)CNc2ccccc2)CCC(F)(F)C1 58109,c1(C(C)C)ccc(C(=O)NC2C3CN(C(C4CCC(=O)N4C)=O)CC23)cc1 58110,C1(C(=O)NC(CNC(C=C(C)CN2CCOCC2)=O)(C)CO)CCC(F)(F)C1 58111,c1(C(N2CC(F)CC(NC(C=C(CC)C)=O)C2)=O)cccc2nccnc12 58112,C1(NC(C2(N)CCCC2)=O)CCn2cnnc2C1.C=C1CC1C(=O)NC 58113,N1CCC2(CNC(=O)N2)C1.Cn1ccc(=O)c(-c2cn(CCCCCCF)nn2)c1 58114,N1(C(COCC(C)C)=O)CCC2(CCC(CNC(c3ccc(Cl)s3)=O)OC2)CC1 58115,C1(C)(CNC(C2(F)CN(C(c3c(C)scn3)=O)C2)=O)CCCC1O 58116,Cc1ccc(Cl)cc1NNC(=O)NCC1Cc2cc(Br)ccc2O1 58117,c1(C(N(CC(N2CC(COC)C3(C2)CC3)=O)C)=O)cnc2sc(C)cn2c1=O 58118,C(CC1=CCN(C(=O)C(C)(COC)SC)CC1)NC(c1ccc(CCC)s1)=O 58119,c1(NC(c2cccc(OCCCOC)c2)=O)cc(Br)c(N)cc1[N+](=O)[O-] 58120,c1(C(=O)NCC2CC(NC(c3cccc(C)c3C)=O)C2)ccc2nc[nH]c2n1 58121,N1(C(C(C)Cc2cccc(F)c2)=O)CCC2(CC(NC(=O)COC3CCOC3)C2)C1 58122,C(C1CN(C(=O)C=CC=CCC)CC1C(N1CCC(C)CC1C)=O)=CC 58123,C(CC(C(C)(C)C)NC(N1CC(O)CC1CC1CN(C)CCN1C)=O)N(C)C 58124,C1(CNC(c2cnc(CNC(C)=O)o2)=O)CCCC2(CC2)C1 58125,Cc1noc(C)c1S(=O)(=O)N(C1CC2CC1CN2)CCCC(=O)O 58126,C(=O)(CCC(CF)CF)N(C(C)CNC(C1CCOC1)=O)C 58127,CC(CC(F)(F)F)C(=O)N1CCCCC(N(C)C(c2snnc2C2CCC2)=O)C1 58128,c1(NC)c(C(=O)NCCc2cn(Cc3cccnc3F)nn2)cccc1F 58129,C(CCN=c1ccnc(NCC2(Br)CC2)[nH]1)NC(c1c(C)c(F)ccc1)=O 58130,c1(NC(C2N(Cc3cc(C)cc(C)c3)CCOC2)=O)csc2nccnc12 58131,N1(C(CC(CC)SC)=O)CCC2C(CCCN2C(C2(C)CCN(C)CC2)=O)C1 58132,C12(C(=O)NCc3c(C)noc3)CCC(CNC(=O)CC=CC(C)(C)C)(CC1)C2 58133,c1(C(=O)NCC(=C)C)cnc2ccc(-c3cc(OC)cc(C)c3)cc2c1Cl 58134,Cc1ccc([N+](=O)[O-])cc1C(=O)NCCOC1CN(C(=O)C(C)(C)S(C)(=O)=O)C1 58135,C1(NC(C=CCC)=O)CCN(C2CCN(C(=O)COC3CCC3)CC2)CC1 58136,CC1CN(C(c2ccn(CC(F)F)n2)=O)CC1NC(c1cc(N)ccn1)=O 58137,N1(C(C(CC)(C)C#N)=O)CC2(CC(NC(c3ncccc3C3CC3)=O)CO2)C1 58138,N1(C(C2C(NC(c3cnsn3)=O)CCC2)=O)CCC(F)(F)C(F)C1 58139,N1(C(C2CCCC(C)C2)=O)CCC(F)(C(N2CC(C)(C#N)C2)=O)CC1 58140,C(C(=O)N1CCCCO1)(c1ccco1)N(C(COCC(=O)OC)=O)CCO 58141,c1(C(N2CCC(N(C(=O)CCC3CCOCC3)C)C2)=O)ccc2c(ccn2C)c1 58142,N#Cc1ccc(OC(F)F)c(C(N2CCC(S(N)(=O)=O)C2)=O)c1 58143,Cc1c(C(=O)NC(CO)CCCCNC(c2cccc(C#N)c2)=O)cccc1Cl 58144,C(C(=O)NNC(=O)C(C)(C)CCCCNC(C1CCC(F)C1)=O)OCCOC 58145,CC(CNC(c1n[nH]c(=N)[nH]1)=O)CC(=O)N(C(C)C(C)(C)O)C 58146,N1(C(C(CSC)C)=O)CCC(C)C1CNC(c1ccc(C(N)=O)nc1)=O 58147,C1(C)(NC(C(C2CCCCC2)NC(c2cc(CC)no2)=O)=O)CCOC1=O 58148,c1(C(N2CCN(C)C(C)C2)C(=O)NC(C(=O)OC)C)cc(F)cc(F)c1Br 58149,C1(NC(c2c(CC)nns2)=O)CC(CNC(=O)CCc2c[nH]c(=N)[nH]2)C12CCC2 58150,C1(OCC)CCCCN(C)C1=O.C12(C)CN(CCO1)C(=O)C2.COC 58151,N1(C(C(C=CC)O)=O)CCCCC(C(=O)N(C(C)C(C)SC)C)C1 58152,N1(C(c2cc(C)n(C)n2)=O)CCC(C)C(NC(c2csc(C3CCCO3)n2)=O)C1 58153,Cc1cc(C(=O)NCC=CCNC(C2CC2C2(C)COC2)=O)cc2c1CCC2 58154,CCC(C(F)(F)F)NCC1CC(CC#N)(CC)C1 58155,C(c1cccc(Cl)c1Cl)=CC(=O)NCCC(C)N(C(=O)CC1NC(=O)NC1=O)C 58156,CC(C)C(C)(CNC(c1nsnc1O)=O)NC(C1C=CCC1)=O 58157,c1(C(N2CC(O)(CNC(C(CN(CC)CC)F)=O)C2)=O)cnc2n1CCC(C)C2 58158,CC(C)(C)C#CC(=O)N1CC(C(F)(F)F)OC(CNC(c2csc(CO)n2)=O)C1 58159,c1(OC)ccc2cccnc2c1COC(C1CCC2(CC2)C1)=O 58160,N1(C(COCCOCC)=O)CC(C(=O)NC(CO)C2(C)CC2)C(C)(C)C1 58161,c1(C(N2C3CC(N4CC(C)C=C(C)C4)C(C3)C2)=O)ccccc1[N+](=O)[O-] 58162,c1(OC)nc(=NCCNC(c2ccc(N(C)C)c(F)n2)=O)[nH]c(C)c1F 58163,Cn1cnnc1CCCC(=O)NCC1(F)CC(CNC(C2CCCO2)=O)C1 58164,CC1OC(C)CN(C(c2c(F)cccc2Br)=O)C1C 58165,C1(NC(C(c2n(C)cnc2)O)=O)CCN(C(=O)CCN2CCCC2=O)CC1 58166,N1(C(C(C=C)C)=O)CCOCC1c1ccc(C(=O)CCCC2CCCC2(F)F)[nH]1 58167,CC#CCCCCNC(=O)CC(O)CNC(=O)C(F)C1CCCC1 58168,CC(C)(O)C(F)C(=O)N1CC(C(N)=O)(CNC(C2CCCC(C(F)(F)F)C2)=O)C1 58169,C1(CN(C(C(C)CF)=O)C)CCCN(C(=O)CN2CSCC2=O)C1 58170,c1(OC)cc(C(=O)NC2CN(C(=O)COC(C)C)C2)cc(Cl)c1 58171,C1(NC(CC(C)(C)F)=O)CC2CN(C(=O)CCc3ccoc3)CCN2C1=O 58172,N1(C(C(=O)NCCCOc2cccc(C)c2)=O)CCC2(CCOC2)CC1 58173,CCC(F)(F)C(C)(C)C(=O)N1CCN(C(c2ccc(C(C)=O)o2)=O)CC1C1CC1 58174,C1(C(C)C)CCOCCN1C(=O)COC1(C)CN(C(=O)C(F)n2ccnc2)C1 58175,c1(OC)ccc(C(N2CC(CO)(NC(=O)CC(=O)N(C)C)C2)=O)cc1S(C)(=O)=O 58176,CN1CCN(C(C2C(C)(C)C2(C)C)=O)CC1CNC(=O)CCC1CCCOC1 58177,NS(=O)(=O)c1scnc1C(=O)NC1C=CCN(C(c2cn3ccccc3n2)=O)C1 58178,CN1C(=O)c2ccccc2C1C(=O)N1CCCCC1CNC(c1nsnc1O)=O 58179,CC#CCCCC(=O)NCC1(C)CCCN(C(=O)Cc2ccccc2Br)C1 58180,O=C1Cc2ccc(NC(c3c(F)cccc3Cl)CC(=O)O)cc2N1 58181,S(=O)(=O)(c1cccc(=NCC(C)c2ccncc2)[nH]1)NC(CC#CC)C 58182,N1(c2cc(CC)ncn2)CCCC(CO)(NC(c2nc(Cl)c(Cl)s2)=O)C1 58183,C1(NC(C(C)(N(C(=O)CSCC(F)F)C)C2CC2)=O)CCOC(C)(C)C1 58184,c1(C(N(C2CN(C(C(F)OC)=O)C2)C)=O)n[nH]c(C)c1C 58185,N1(C(CN(CCOC)C)=O)CCCC1CC(=O)N(CCC12CC(CO1)C2)C1CC1 58186,N1(C(COCCOC)=O)CC2C3CCC(C2C1)N(C(C1CCC(C)S1)=O)C3 58187,CN1CCCCC(C(=O)NC2CC(CNC(c3ccc(Cl)o3)=O)C2)C1=O 58188,C12(NC(C(CSC)OC)=O)CCC(CN(C(c3cc(CO)on3)=O)C1)C2 58189,N1(C(C)Cc2csnn2)CCCC(C(=O)NC(CC2CC2)CO)C1 58190,c1(OC)cc(CC(=O)NC2CCSC23CN(C(=O)C=C(C)C)C3)c2c(c1)CCO2 58191,c1(C(=O)NCC2(F)CCN(C(=O)Cc3cnsc3)CC2)coc2cccc(F)c12 58192,N1(C(C=CC(C)(C)SC)=O)CC=CC(C(=O)N(C)Cc2sccc2C)C1 58193,C(CNC(=O)C(F)(F)C1(O)CCC1)(CCNC(c1sccc1CO)=O)OC 58194,c1(OC(C)C)cncc(C(=O)NC2(CNC(c3cc(C#N)c[nH]3)=O)CC2)c1 58195,C(C)(CCC(=O)NC1CCC1C(=O)NCC(O)CF)OC 58196,C(=O)(CC(COC)COC)NCCC1CCN(C(CS(CC)=O)=O)C1 58197,n1(CC)ncc(C(N2CCCC2C2(NC(C3CS(=O)(=O)C3)=O)CC2)=O)c1C 58198,N1(C(CC=CCC)=O)CCC(C)C(CC(=O)Nc2cccc(F)c2O)C1 58199,CC(C)(CS(N)(=O)=O)C(=O)N1CCCC1CNC(=O)C1=CC2CCCC12 58200,CCC(CN(C)C)CC(=O)NC1CN(C(c2cc(C(C)=O)on2)=O)C(C)(C)C1 58201,c1(C(=O)NC(C)CNC(=O)COCCc2nncn2C)cccc2sncc12 58202,N1(C(C2CCC(N(C)C)C2)=O)CCC(NC(=O)C#CC2(C(F)(F)F)CC2)C1(C)C 58203,N1(C(C2(C)CSC2)=O)CC(C(=O)NCCCN2CCC2)C2(CC2)C1 58204,C1(C(=O)NCCCNc2cccc(F)c2)CC(O)CN1Cc1cc[nH]c1 58205,N1(C(Cc2ccn(C)n2)=O)CC2CCN(C(c3ccc(C4CC4)cc3F)=O)C(C2)C1 58206,c1(C(=O)Nc2c(C)cc(Br)cc2Br)cnc2[nH]cc(-c3cccc(CO)c3)c2c1 58207,N1(C(Cc2nc(C)sc2)=O)C2CCC1C1CC1(NC(c1cccnn1)=O)C2 58208,C1(C(C)C)CN(C(c2sccc2CO)=O)CCN1C(=O)CNS(C)(=O)=O 58209,C1(CC(=O)N(C2CCN(C(c3ccnc(F)c3N)=O)C2)C)CC(C2CC2)=NO1 58210,C=CC(CCC)CC(=O)N1CC(C(=O)N(CCC(=O)OC)CC(C)C)C1.C1CC1 58211,C1(C(=O)NCCCC(C)NC(=O)Cc2cccs2)(N(C)C)CC(F)(F)C1 58212,C(=O)(C#CC1(C)CC1)NCCC1(OC)CN(C(=O)C(C)OCC2CCCO2)C1 58213,Cc1cc(C(=O)NCCCC2(NC(C3CC4(CCCO4)C3)=O)CC2)c(N)c(F)c1 58214,Cc1cnc(C(N2CC(C(N)=O)(CNC(C3CSCCS3)=O)C2)=O)cn1 58215,c1(C(N2CCCC2c2nn[nH]n2)=O)cccn2ncnc12.C12CC1CNC2 58216,C1(C(C)C)CC(C(=O)NCCC2CCCN2C(=O)CC2C(C)(C)C2(C)C)CCO1 58217,C(=O)(C(C(C)C)C(C)C)N1CC(CCC=C)(C(=O)NCCC2=CCOCC2)C1 58218,c1(-n2cc(CONC(Cc3cc(C)no3)=O)nn2)ccc(C)c(Br)c1 58219,c1(-c2c(F)ccc(C(N=c3ccnc(C)[nH]3)=O)c2F)cc(OC)cc2[nH]ccc12 58220,N1(C(c2c(C3CC3)ccc(C)c2)=O)CCC2(CC1)CN(C(C1(O)CC1(C)C)=O)C2 58221,CN=c1nc(C(N2CCCC(O)(CNC(C3CC3Br)=O)C2)=O)cc(C)[nH]1 58222,c1(C(N(C)CC2CN(Cc3sccc3Br)C2)=O)c(F)cccc1[N+](=O)[O-] 58223,C1(C(=O)NCc2n(CC)nnc2C)CC2CCC1N2C(c1n[nH]cc1CC)=O 58224,c1(C(=O)NCC2CCCN(C(c3ncc(F)cc3F)=O)C2)cc(F)cc(Br)c1F 58225,c1(NC(c2cncc(-n3c(C)ncc3)c2)=O)cc(Br)c(F)cn1 58226,C(=O)(CS(=O)(=O)CC(=O)NCC1CC(O)CN1C(=O)C(c1ccc(C)s1)C)OC 58227,C1(CN(C(C(OC)OC)=O)C)CCN(C(C2(Br)CC2)=O)C1 58228,C1(NC(C(N2CCCCCC2)C)=O)CCN(c2ccncc2C#N)CC1O 58229,C1(C(=O)OC2CC(OCC)C2Cc2ccc(C)cn2)CC2CC(CO)CC12 58230,C1(NC(C(C)C)=O)CC(=O)N(C2CN(C(=O)CC(C)NC(N)=O)C2)C1 58231,Cc1cc(O)ccc1CC(=O)NCC1COC(CNC(C2CC(C)(C)CO2)=O)C1 58232,c1(CC)nn(C)c(Cl)c1C(N1CC(CNC(=O)CC2(C(F)F)CC2)C(C)(C)C1)=O 58233,CCCCCCC(CC)NC(C1CC(CCNC(=O)CC(C)n2cccc2)C1)=O 58234,Cc1cc(C(N2CCC(C3CC3)C2CNC(=O)CC(C)(C)O)=O)cc2nc[nH]c12 58235,C=CCCC(C(=O)N(C)Cc1ccc(C)cn1)NC(CC(C1CCC1)OC)=O 58236,N1(C(CCCNC(c2cc(C)sc2)c2nnnn2CCOC)C)CCN(C)CC1 58237,c1(C(=O)NCCCN(c2nc(CC)nc(C)c2)CC)cc(C)ccc1[N+](=O)[O-] 58238,C1(C(=O)NCCCCC2CN(C(c3cc(OC)ns3)=O)C2)CCCC1S(C)(=O)=O 58239,c1(C(=O)NCC=CCNC(c2c(C(N)=O)cccc2)=O)cnc2nccn2c1 58240,c1(C(=O)NC(C(=O)NCC(CC)C(C)C)CCSC)ccc2cncn2c1 58241,C1(N(C)C(c2cc(=O)n(C)cn2)=O)CCCN(CCN2C(=O)CNC2=O)CC1 58242,c1(C(N2CC(CNC(C3(CC=C)CC3)=O)C3C2C3)=O)cc(C)ccc1[N+](=O)[O-] 58243,c1(C(N2CCC(NC(C=CCN(C)CC)=O)C2)=O)cncc2c[nH]nc12 58244,N12CCCCC1C(=O)N1C(CCC1)C2=O.C1CC=CC(O)C1.c1(N)nccs1 58245,N1(c2cncc(C#N)n2)CCC2(CC1)OCCC2NC(C1(C2CCCO2)CC1)=O 58246,C1(C(N(C2CC(NC(CCSC)=O)C2)C)=O)CCOCC1C 58247,C1(CNC(c2cc[nH]c2)=O)CN(C(=O)CSCc2ccccc2)C2CC12 58248,N1(C(CC(C)(C)O)=O)CCN(C(=O)CCc2nccs2)C(CO)C1 58249,CC(C)(CC(=O)N1CCC2(CCC2)CC1C(=O)ON)CC(F)F 58250,n1(CC(N2CC(C)(CNC(c3c(OC)nn(C)c3)=O)C2)=O)cc(C)c(O)nc1=O 58251,c1(CC(=O)NC2C(NC(c3n(CC)c(O)nc3)=O)CCC2)n[nH]c2c1CCCC2 58252,c1(OC)ccc(CCC(N2CC(NC(c3cc(C#N)[nH]c3C)=O)CC2C)=O)cc1C 58253,C1(CCCNC(Cc2c(C)nc[nH]2)=O)CCN(C(c2ncc(Br)cn2)=O)CC1 58254,C1(C(=O)NC(C2CCCN(C(C3(C#N)CC=CC3)=O)C2)C)CCC(C(F)(F)F)CC1 58255,C1(C(=O)NCC(=O)NCC)CCC(O)CN1C(c1cn(CC)nc1C)=O 58256,N1(C(c2c(NC)nccc2)=O)CCCOC(CNC(C23CC(C)C2C3)=O)C1 58257,CC(C)CC(C(=O)N1CC2COCCC2(NC(c2ccc(O)nc2)=O)C1)C(N)=O 58258,C1(CC=C)(NC(C2C=CCC2)=O)CCN(C(c2ccc(C(N)=O)cn2)=O)C1 58259,c1(C(=O)NCC2(C(C)(C)C)CCN(C(CNC(CC)=O)=O)C2)sc(C)c(C)c1C 58260,N1(Cc2c(C)nn(C)c2)C2CCC1CN(C(c1ccc(C(N)=O)o1)=O)C2 58261,C1(NC(C(C)OC)=O)COC2(C1)CN(C(c1cc(C)c(C)nc1C)=O)C2 58262,N1(C(c2cc(SC)c(N)cc2)=O)C2CCC1CN(C(C1(OC)CCSCC1)=O)C2 58263,c1(C(C(=O)NCC2N(C(C3(C(=O)OCC)CCCC3)=O)CC=C2)C)cccc(O)c1 58264,n1(CC)ncc(Cl)c1C(=O)NCC(C)CNC(=O)CCc1cc(C)[nH]n1 58265,C1(N(C(CC(=C)C)=O)CC)CCN(C(C2CCCCN2C(=O)C2CC2)=O)CC1 58266,C1(C(=O)NCCC(CNC(c2cc(O)ccc2F)=O)O)CCC2(CCC2)O1 58267,C(C(F)(F)C(F)(F)F)N(CCCNC(CC(=O)N)(C)C)CC.CCOC 58268,N12CCC(C)(C1)C2.CCCC(C)NC(=O)CCN(C)C 58269,C1(OC(C(=O)OC)C)CCCN(C(c2c[nH]nc2OCC(C)C)=O)C1 58270,n1(-c2c(C(=O)NCCN(C)C(C3(C)C=CCC3)=O)cccc2)ccc([N+](=O)[O-])n1 58271,c1(CS(C)(=O)=O)ccc(C(ONC(=O)NC2CC2(c2ccccc2)F)=O)cc1 58272,Cc1ccnc(N2CC(NC(=O)N(C)CCN(C)C(c3ccccc3)=O)C2)n1 58273,c1(COC)nocc1C(=O)NCCCC1CCCN1C(=O)CCCn1cncn1 58274,C=CCN(CC=C)N1CCC(S(C)(=O)=O)(C(c2ccccc2)=O)C1 58275,CC(C)(C#Cc1cn(CCOCCSC2CCCO2)nn1)NC(C1CC1C(N)=O)=O 58276,C#CCCC(O)C(=O)NCCC1CCN(C(C2CCS(=O)(=O)N2)=O)CC1 58277,Cc1nc(N2C3CCCC2CC(NC(=O)C2=CCC(C)CC2)C3)c2ccsc2n1 58278,C#CC1(O)CCN(C(C2CC(C)CN(C(C3CCCSC3)=O)C2)=O)CC1 58279,C1(C(CNC(C(C)OCC=C)=O)(C)C)CCCCN1C(=O)CN(C1CC1)CC 58280,Cc1ncn2ccc(C(N3CC(CNC(=O)C=CC(C)C)C4(CC4)C3)=O)cc12 58281,c1(C(N2CC3(CC(COC)C3)C2)=O)cc(C)cc(Br)c1F.c12sccc1NC2=O 58282,CC(CC(=O)NCC1(CNC(C2CC23CCCCC3)=O)CC2(CC2)C1)C(C)(C)C 58283,CCCN=C(NCC1(C)CCCc2ccccc21)N1CCC(OC(C)(C)C)C1 58284,CC(C)C(CNC(C1CC(OCC2CC2)C1)=O)C(=O)NCC12CCCN1CCC2 58285,C1CN=C2N=C(C3=C(N2)COC3)N2CCC(C2)O1.C(CCCNCC)OCC 58286,c1(C(=O)NC(C(=O)NOCC2CCOC2)c2cn(C)nc2)ccc(=O)n(C)c1 58287,C(=O)(CCC(C)(C)NC=O)NCC(=O)NCCC(=O)NCC(N)=O 58288,C(=O)(C(C)CNC(=O)CC1CCOCC1)N(CC(COC)O)C 58289,C(=O)(C(C)CC(F)F)NCC(CC)(CC)NC(=O)C(C)Oc1ccc(SC)cc1 58290,c1(SC)cc(C(=O)NC(C)CCN(C(=O)C#CC(=O)N(C)C)C)oc1C 58291,c1(N2CCN(c3nnc(C(C)C)n3CCOCCOC)CC2)c(F)cccc1F 58292,C1(CNC(C(N2CCC(O)CC2)C)=O)CC(C)CN(C(C23CC(C2)C3)=O)C1 58293,N1(C(C(C)OCCCC)=O)CC2CCC2(CNC(=O)C=Cc2cnc(C)s2)C1 58294,c1(CC)cn(C)nc1C.C(CCC(=O)NCCCC1CCCN1C(C1CC1)=O)OCC 58295,C1(COC)(CO)CCN(C(=O)CC(C)(C)NC(=O)C=Cc2ccnn2C)CC1 58296,c1(CC(N2C(C(=O)OCC)CC(F)CC2)=O)cc2ccc(Br)cc2s1 58297,N1(C(CCN(C2CC2)C)=O)CCC2(NC(=O)Cc3cnn(C)c3)CCCC12 58298,C=CC1(C(=O)NCCCC)CN(C(=O)CNC(c2ccccn2)=O)C1 58299,C=CCC(CC(C)C)C(=O)N(C)CC1CCN(C(C2CC3(CC(OC)C3)C2)=O)C1 58300,C1(CNC(C2(C)CC2(F)Cl)=O)CCN(C(c2n[nH]cc2Br)=O)C1(C)C 58301,C(=O)(C(F)(F)CCc1ccccc1)NCC1CN(C(C2C(C(=O)OCC)C2)=O)C1 58302,C=CC1(C(=O)Nc2cnc3c(c2)CCC3)CCN(C(=O)C(N)CC2CC2)CC1 58303,Cc1cc(CN(C)CCN(C(=O)CCc2conc2C)C)cc(C)c1Cl 58304,C#Cc1ccc(OCC(=O)NCCN(C(c2conc2C2CC2)=O)CC)cc1 58305,Cc1cc(C(=O)NN2CCN(S(C)(=O)=O)CC2C)cnc1C.c12ccccc1NC2 58306,C(=O)(C(C)CN(C(=O)CNc1ncccn1)C)NC(C#C)C1CCC1 58307,n1(CC)ncc(Cl)c1C(=O)NC1CCC(C)(CNC(=O)CCCC2CCCC2)C1 58308,c1(OC)cc(C(=O)NC2CCCCC2NC(=O)CCC2CC2C)cc(C)n1 58309,C1(C=O)CC2CCC(C1)N2C(C1(F)CNC1)=O.C(C(CO)C(C)(C)C)OC 58310,N1(Cc2cc(F)cc3c2OCOC3)CCc2nc[nH]c2C1c1cccnc1 58311,c1(C(=O)NC(CC)CN(C(=O)C(C)C2=CCCC2)C)oc2ccc(C)cc2c1C 58312,c1(C(N2CCC3(NC(c4cscn4)=O)C(C2)C3)=O)n[nH]c2c1CCCC2 58313,CC1CCC=C1C(=O)N1CCCC1C(=O)NCC=Cc1ccco1 58314,CC1CN(C(C(=O)NCC2CCCO2)C(C)CC2CCC2)CC(=O)N1 58315,c1(N(C)C)ccc(CNC(C2(NC(=O)C(O)CN3CCCC3)CCC2)=O)cc1 58316,C12(C(=O)NC(C3(N)CCN(C)C3)C)COCC1CN(C(=O)CCn1ccnc1)C2 58317,c1(C(N(C2CN(C(=O)CCCN3C(=O)CNC3=O)C2)C)=O)n[nH]c2ccccc12 58318,N1(C(CCCCCSCC(=O)Nc2cccs2)=O)CCCC(O)(C2CC2)C1 58319,c1(C(N(CCNC(CS(CC)(=O)=O)=O)CCOC)=O)cc2sc(=O)n(C)c2s1 58320,C1(CC=C)(C(=O)NC2(CC=C)CC(F)(F)C2)CCCN1C(=O)C(C)C=C 58321,Cc1ccc(Cl)c(O)c1C(=O)NC1CCN(C(=O)CC(F)(F)F)C1C1CC1 58322,C(C)(CNC(C1CC(=O)N(c2ccccc2)C1)=O)(C(C)C)NC(C1C(=C)C1)=O 58323,C(=O)(C(C)(C)CS(C)(=O)=O)NCC1CCN(C(CCNC(=O)NC)=O)CC1C 58324,CC1(C)OCC2CC12NC(C1(NC(c2ccnn2CCF)=O)CC(F)(F)C1)=O 58325,C1(CCCC=C)(CO)CCN(C(=O)CCc2ccccc2I)CC1 58326,CC(C)(CCNC(C1CCC(F)C1)=O)NC(=O)COCCN(C)C 58327,c1(N(C(C)=O)C)ccc(NC(C(=O)N(C(C)CCNC2CCCC2)C)=O)c(Br)c1 58328,c1(SCCC)ccc(C(=O)N(CCNC(=O)C(C)OCC(C)C)CC2CC2)o1 58329,Cc1ccc(O)c(C)c1NC(C1(O)CCCN(C(=O)COCC2CCC2)C1)=O 58330,c1(C(=O)NCCN(C(=O)CC2CN(C)CC2O)CC)ccc2c(c1)OC(C)(C)C2 58331,N1(Cc2c(C(=O)OC)c(-c3nn[nH]n3)sc2)CC2CS(=O)(=O)CC2(C#N)C1 58332,CNS(=O)(=O)NCC(N1CC(C(C)NC(=O)Cn2nnc(CC3CC3)n2)C1)=O 58333,C12(C(N3CCN(C(c4c(C)coc4C)=O)CC3CO)=O)CCC(N(C)C)(CC1)CC2 58334,C1(NC(c2c(CC)cco2)=O)CCN(C(c2cccc(OCC)c2)=O)CC(O)C1 58335,N1(C(C(F)=CC)=O)CC(NC(=O)CCC(=O)c2ccncc2)C2CC12 58336,C(=O)(C(C)(CC1CCC1)OC)NC(CN(C(c1cc(CCC)[nH]n1)=O)C)C 58337,CC1(C)CN(C(=O)C=Cc2ccsc2)CC1CNC(c1sccc1C#N)=O 58338,CC(C(=O)NCC1CCN(C(C2CC=CC2)=O)C1)C(C)(F)F 58339,CCCC(C(=O)NCC)N1CCCCC1CN1CCC(C(N2CCCCC2)=O)C1 58340,C1(NC(C2N(C(C)=O)CCC2)=O)CC2CCC1(Cc1cnn(C3CC3)c1Cl)C2 58341,c1(C(=O)NCC2(C(=O)NC(C(=O)OC)CO)CC2)ncc(Br)cc1F 58342,c1(C(=O)Nc2cncc(Cl)n2)ccc(=O)n2c1CNCC2 58343,C1(C)(CNC(C(COC)O)=O)CN(C(=O)C(C)(C)OCC(F)(F)F)CCO1 58344,C=Cc1cncc(C(N2CC(OCCNC(C3CC(O)C(F)C3)=O)C2)=O)c1 58345,N1(C(CC(C)F)=O)CCN(C(c2cc(Br)cc3cn[nH]c23)=O)CC2(CC2)C1 58346,C(=O)(C1=CCN(C(=O)Nc2cn(C)c(=O)cn2)C1)N1CC(COC(C)=O)C1 58347,N1(C(CN(CCOC)C)=O)CCCC2CN(C(=O)C(CCSC)N(C)C)CCC12 58348,c1(C(C(=O)NCCN(C(=O)CCc2cnoc2)CC(C)O)O)ccc(Cl)cc1 58349,C1(COC)(CN2C(C(=O)OC)CC(C(C)CCO)C2)CCCN1C(=O)COC 58350,N1(C(C=Cc2cnc(C)s2)=O)CC2OCCN(C(=O)CSCCN3CCCC3)C2C1 58351,c1(CC)nn(C2CC2)cc1C(=O)NCCNC(c1cncnc1)=O 58352,c1(OC)ccc(C(=O)NC(C)CCNC(c2cscc2C(=O)OC)=O)cc1C 58353,Cc1nc2ccccc2cc1C(=O)N(C1CCCC(NC(C2COC2)=O)C1)C 58354,N1(C(c2cc(COC)no2)=O)CC2CCC2(CCNC(c2c[nH]nc2SC)=O)C1 58355,C=C(C)CCCC(=O)NCCCCNC(c1ccn(C(F)(F)F)n1)=O 58356,Cc1ccc(C(=O)NC2(C)CC(NC(=O)CCC3CC3(C)C)C2)c(N)n1 58357,N1(C(C(CCC)CCC)=O)CC(CO)C2(C1)CN(C(=O)C(CC)OC)C2 58358,C12CCC(O1)CCCC(=O)N(C)C2.C=C(CNC(=O)OC(C)(C)C)CO 58359,C(CCC(C)(C)C(=O)N1CCC(O)(C=C)C1)C1CCN(C(C(C=C)CC)=O)C1 58360,C1(c2n(CCC)nnn2)(Nc2ccn3nnnc3c2)CCCC(C2=NOCC2)C1 58361,c1(C(=O)NCC(C)NC(C(CC)N(CC)CC)=O)ccc2c(c1)C(=O)CCC2(C)C 58362,CCC(C)CCCC(=O)N1CCC(C(C)(C)NC(c2cnnc(O)c2)=O)C1 58363,N1(C(CCCC2C(C)C2)=O)C(C(=O)NC(C)(CO)C(C)(C)O)CCC12CC2 58364,C1(NC(C2(C(=O)NC)CC2)=O)CCCN(C(c2ccnc(C(C)C)n2)=O)C1C 58365,C=CC1CN(C(C2CCN2C(C)=O)=O)CC1NC(C1CCCCCCC1)=O 58366,CC1(C)C=C(C(=O)NC2(CNC(C3(F)CCCOC3)=O)CCC2)C1 58367,C1(C(=O)NC(CC)C(O)c2ccccc2)CCc2cnn(CCCC)c2C1 58368,C(C)(c1cnn(C)c1)=CC(=O)NCC(CNC(CN(C(=O)OC(C)(C)C)CC)=O)F 58369,C1(CNC(c2cn(CC=C)nn2)=O)CN(C(C2(C(=O)NC)CC2)=O)CCC1C 58370,C#CC1CCCC(NC(=O)C(CNC(=O)CC2C=NN(C)C2=O)C(C)C)C1 58371,N1(C(C2(C(CC)=O)CC2)=O)CCC2C(CCN2C(C2C=CCS2)=O)C1 58372,C1(C(N(CC(C)C(=O)NC(C)Cc2nc[nH]n2)C)=O)C2(CC2)C12CC2 58373,C=C=CC(C)C(=O)NC1CN(C(=O)CC23COCC(C2)C3)CC1c1ccccc1 58374,C12(NC(C(CSC)O)=O)CC(C1)N(C(=O)C(c1cccc(C(F)(F)F)c1)O)C2 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58427,N1(C(c2cc(C3CCC3)on2)=O)CC2CC1CCC2NC(c1ccccc1CO)=O 58428,C1(COC)(NC(C2(c3ccno3)CC2)=O)CCN(C(=O)C(C)Cc2cnco2)C1 58429,C(C1CCCCC1)=CC(=O)NC1C(NC(CCc2cc(C)[nH]n2)=O)CC1 58430,c1(SCC(=O)NCC(CN(C)C(c2noc(C(C)(C)C)n2)=O)O)ccc(Cl)cc1 58431,N(C(=NCCC(C)(C)C)NC1CCCCC1)C1C(C)CCCC1 58432,c1(N(C(=O)NC(c2cc(F)ccc2F)C)C)ccc(S(C)(=O)=O)o1 58433,C1(NC(C=CCN(CC#C)C)=O)CCN(C(c2c(C(F)(F)F)coc2C)=O)CC1 58434,CCCCC(F)C(=O)N1CC(OCCC(=O)Nc2cccc(COC)n2)C1 58435,S(=O)(=O)(c1ccc(NC2CCOC3(CCCC3)C2)c(F)c1)NC(CC(C)C)C 58436,CC1CC2(CC(NCC3(C)CC3C(=O)NOCCOCCF)C2)C1 58437,C1(NC(c2cc(C)sc2C)=O)CCC12CCN(C(c1ccc(O)cc1)=O)CC2 58438,C1(CNC(CCC#CC)=O)COC2(CCC2)CN1C(=O)CCc1cncc(Cl)c1 58439,CC1(C)CCCC(O)(C(N2CCC2CNC(=O)CC2OCCO2)=O)CC1 58440,CC1(C)C(CC(=O)N(CCNC(=O)CSc2ccco2)C2CC2)CC1O 58441,CC1(C)COC(C(=O)NC2CCCC(CNC(c3cc(Cl)ccc3Cl)=O)C2)CO1 58442,C1(C(N(CC(c2ccc(O)cc2)O)CCOC)=O)C2C=CC(C2)C1N 58443,C1(NC(c2nccnc2Br)=O)CCCC12CCN(Cc1cc(F)c(Br)cc1F)C2 58444,Cc1[nH]c(C#N)cc1C(=O)NC1CCCC1NC(c1ccc(F)c(C(F)F)c1)=O 58445,C(CCNC(=O)Cc1cn(C)cn1)(C(C)C)NC(COCC(=C)C)=O 58446,C(=O)(CC(CSCC(c1cc(C2CCOCC2)no1)NC(=O)C)OC)NCC 58447,C(=O)(C(C)CC(F)(F)F)N(CCN(C(=O)Cc1ccn(C)c1)CC)CC 58448,C(CCC(O)C(=O)N(c1ccsc1)C)NC(Cc1cc(C)sc1)=O 58449,C(=O)(CCCC(=O)N1CC(CNC(=O)CC2CCNC2=O)C(O)C1)OC(C)(C)C 58450,CN1CCCC(CNC(c2cc(CNC(C3CCC(O)C3)=O)nn2C)=O)C1=O 58451,C1(CNC(c2n[nH]c(C)c2Cl)=O)CCC2CN(C(C3COC(C)(C)O3)=O)CC12 58452,N1(C(C2CC(SC)C2)=O)CCC(NC(C2CN3CCC2CC3)=O)C(O)C1 58453,N1(C(Cn2ncc(C#C)c2)=O)CCC2(CCCN2C(c2ncoc2C2CC2)=O)C1 58454,C1(O)(C(=O)NCC2N(C(c3c[nH]c(=N)s3)=O)CC(C)(C)OC2)CN2CCC1CC2 58455,c1(C(=O)NC2C(NC(C(C(C)C)N(C)C)=O)C2)c(O)nn(C)c1C(F)(F)F 58456,c1(OC)cc(C2CC2C(C)(C)CCCO)cc(I)c1OC.N1(C=O)CC=CC1CO 58457,C1(CC(=O)NC2CCC(NC(CC3CN(C)C3)=O)C2)CCC(C(F)(F)F)CC1 58458,c1(OCC(N2CCC(Cn3cc(C4CCCCO4)nn3)C2)=O)cc(Cl)ccn1 58459,C1(CC)CC(=O)N(C2CN(CC3OCC(NC(c4nc(CC)sc4)=O)C3)C2)C1.CC 58460,CCCC(C#N)C(=O)NC(C(=O)NOCC(=O)OC)c1ccoc1 58461,c1(N2CCCC(OCCN(C)C)C2)nc(=N)[nH]c(=NCCc2ccc(CO)cc2)[nH]1 58462,CC1CC=C(C(=O)N2CCC(F)CC2C(=O)NOCCF)CC1 58463,C(=O)(C(CC=C)C(C)C)NCC(C1N(C(C2CCCC(C#C)C2)=O)CCC1)(C)C 58464,C1(OC)CN(C(N2CCC(OC3CC3)CC2)=O)C(C)(CO)C1 58465,C#Cc1ccc(C(=O)NC2CC3CCC(C2)N3c2ccnc(SC)n2)cc1F 58466,C1(F)(C(=O)NCCN(C)C(c2cncc(-n3cncn3)n2)=O)CCOCC1 58467,Cc1ccc(C(=O)NCCCCCCNC(C2CC2Cl)=O)c(O)c1 58468,N1(C(C2C(CCOC)C2)=O)CC2(COC)CC1(CNC(c1cnccn1)=O)C2 58469,C1(CNC(c2scc(OC)c2)=O)C(C)CCN1C(=O)Cn1cncn1 58470,C1(C(=O)OC)CN(C(=O)NCCCN2CC3CC3C2)C2(CCC2)C1 58471,Cc1cccc2c1CC(C(N1CCC(C)C1CNC(C1C(F)(F)C13CCC3)=O)=O)N2 58472,N1(CC)CCCC1CC(=O)NCC(C)(C)CNC(=O)C=C(C)C(C)CC 58473,C(=O)(CCC(=O)N1CC(c2ocnc2C(=O)NCC2COCCO2)C1)NC 58474,c1(OC)coc(C(=O)NCC2(C)CCCN2C(=O)COCCN(C)C)cc1=O 58475,C1(OCC)CCCCC1NC(=O)C#CCNC(=O)CCC1CCC1 58476,C1(NC(C23C(CN(C(=O)C=Cc4ccoc4)C2)C3)=O)CC2(CCCO2)C1 58477,C1(O)(CCNC(c2c(C)nsc2)=O)CCN(C(=O)C(n2nccc2C)C)CC1 58478,C(=O)(CCCCCC(C)O)N1CCN(C(C(OCC)OCC)=O)CC1CO 58479,c1(N(C)C)ccc(C(=O)NC2CCN(C(C3CC3(F)F)=O)C2C2CC2)c(O)c1 58480,C1(CC(=O)NCC2CC(NC(c3cc(C)[nH]n3)=O)C2)CCC2(CCOCC2)CO1 58481,C1(C(=O)NC(C)CCN(C)C(c2ccc(C(C)(C)C)[nH]2)=O)CC2(C1)CC21CC1 58482,N1(C(C(CSC)C)=O)CCN(C(C2CCC(=O)N2C(C)C)=O)CC1c1cn[nH]c1 58483,C12(CNC(C(C)(N(C(=O)CCC3CCCCO3)C)C3CC3)=O)CCC(CO1)C2 58484,N1(C(C(N2CCC(CC3CCC(C)(CC)O3)CC2)=O)=O)CCC2(CC1)OCCO2 58485,c1(C(=O)OCC)ccc(C(=O)NCC2(F)CC(NC(C3(C)CC3)=O)C2)cc1F 58486,C1(NC=O)CC(OC)C12CCOCC2.c1(OCCCC)ccc2cc1-2 58487,C1(c2ncccn2)(C(N)CNC2CCOC2)CCCC1 58488,N1(C(C(C)(C)CO)=O)CC2CCN(C(C3CN(S(C)(=O)=O)C3)=O)CCC2C1 58489,C1(C(=O)NC(CC)CNC(C2CCN(CC)C2)=O)CCOC(C)C1 58490,c1(C(=O)NC(C(=O)NCC(C)NC(C2CC(C)OC2C)=O)C)ccc(N)cc1 58491,c1(CC)nccnc1C(=O)NCC1(CNC(=O)CC2CC(SC)C2)CCCO1 58492,c1(OC)ccc(SCCC(N2CC3CC3(NC(C34CCC(C3)C4)=O)C2)=O)cc1 58493,CC1(C(=O)NCCc2ncccn2)CCN(C(C2CC23CC3)=O)CC1 58494,C#Cc1ccccc1C(=O)NC1C2CC1N(C(=O)C(c1ccccc1)F)C2OC 58495,c1(N(CCC)CCNC(c2ccccc2F)=O)nc(CCN(C)C)nc(=N)[nH]1 58496,c1(C(N2C3C(CNC(c4c(CCC)nco4)=O)C(C3)C2)=O)ccn2c1CSCC2 58497,N1(C(C(CCC)CN)=O)CCC2CCCCC2CC1 58498,C1(=CC(=O)NC2CCN(C(c3ccc(F)s3)=O)C2)CN2CCC1CC2 58499,C12(CNC(c3ccn(CCNC(C(CCC)F)=O)c3)=O)CCCN(CC1)C2 58500,Cc1nn(CC(=O)NC2CCN(C(=O)CSC(C)(C)C)C2C)c(C)c1Cl 58501,CC1CC(NC(=O)C(=O)NCC2CC2)CN1C(c1cnc(C(F)F)nc1)=O 58502,CC(C)C(CNC(c1ccncc1)=O)NC(=O)CN(CCCCO)C(C)C 58503,N1(C(CNC(=O)OC)=O)CCC(C(=O)NCC23CCCC2C3)C1(C)C 58504,C=CC(C)C(C)C(=O)NCC1(CNC(c2cn(C)c(-c3ccccn3)n2)=O)CC1 58505,N1(CCC(=O)NC23CC(NC(C(C)SCC)=O)(C2)C3)CCCC(C(N)=O)C1 58506,N1(C(C(c2ccoc2)NC(c2ncc(F)cc2F)=O)=O)CC2CC1CC2O 58507,C1(F)(C(N(CCOCC#C)C)=O)CCN(C(C23CCN(CC2)CC3)=O)CC1 58508,N(C1CCCc2occc21)C(C1(C=C)CCN(C(=O)CC2CCC(O)C2)C1)=O 58509,C1(N(C(Cc2c(C)non2)=O)CCO)CCCN(C(=O)C(F)CC2CC2)C1 58510,c1(C(=O)NCC2(F)CC(NC(C(C(CC)C)O)=O)C2)c(C)ccc2ncccc12 58511,Cc1nnc(CCC(=O)N(C)CCNC(c2ccc(C(C)(F)F)cn2)=O)n1C 58512,Cc1nc(CC(=O)NC(CO)C(C)NC(=O)CSc2nncn2C)n[nH]1 58513,C(=O)(CC(C)C(=O)N(CCCNC(=O)C(C)SCc1ccc(C)cc1)C1CC1)OC 58514,CN1CCC(n2cc(C(N3CC(C(=O)NC4CC(F)(CO)C4)C3)=O)cn2)CC1 58515,N1(C(C2=CCC(C)CC2)=O)CC(NC(C2C3CCCC23)=O)C2CCCCC12 58516,C(=O)(CC(C)(C)C(C)(F)F)NC(CN(C(C1N(CCC(C)C)CCC1)=O)C)C 58517,c1(C(N(CCOCCN(C(c2c(C)c[nH]n2)=O)C)C)=O)ccc2ncnn2c1 58518,c1(CN(C)N(C)Cc2cnc(N)s2)cnn(C)c1.C(C)(C)(C)OC=O 58519,N1(C(c2nc(CC)sc2)=O)CC(N(C(=O)CN=S(C)(C)=O)C)C2(CC2)C1 58520,C1(CCNC(C2CNC(=O)O2)=O)CCCCN1C(=O)C1CC1.C(COC)N.CC 58521,C(=O)(C#CC1CCC1)NCC1N(C(C(CC)Cc2ccccc2Br)=O)CC1 58522,C1(CNC(Cc2cc(C)[nH]n2)=O)CCN(c2nnc(CN)s2)CC1.C1(C)CC1 58523,c1(C(N(CC(O)CNC(C2(C3CCCO3)CC2)=O)C)=O)ccc2nn[nH]c2c1 58524,CC(CC(C)NC(=O)CC(C)C1CCCC1)NC(c1sccc1C(F)F)=O 58525,N1(C(c2ccc(C=C)cc2)C(=O)NC(C)(C)CC)c2ccccc2C(C)C1C 58526,C(CNC(=O)Cc1ccc(F)cc1)(CC(=O)NC1CCCOC1)OC 58527,C1(CNC(c2c(CC(C)C)onc2)=O)CCCCCN1C(=O)CCn1cnnn1 58528,N1(C(CCCCCN(C)C)=O)CC2CC(NC(=O)CCc3cnccn3)CC1C2 58529,c1(N(c2cnnn2C)CC)nc(C(F)(F)F)ccc1C(N1CCCC1)=O 58530,C1(C(=O)NCCCOCC#C)CCC2CCC1N2C(c1cccc(=O)n1C)=O 58531,C1(CCNC(CNS(NC)(=O)=O)=O)CN(C(c2cnccn2)=O)CCO1 58532,c1(C(=O)NC2(C(CC(=O)NCCOC)C3CCCCC3)CCC2)ccc(Cl)cc1 58533,c1(NC(=O)NCC2(Cc3ccc(C)cc3)CC2)ccc(C)c(Cl)c1 58534,C(=O)(C(CNC(C1CN(C(=O)C2CC2)C1)=O)Cc1ccc(O)cc1)OC 58535,N1(C(C2(CC#C)CCCC2)=O)CCC(CNC(=O)CC2COCCO2)(OCC)C1 58536,c1(C(C)(C)C)cc(CNC(=O)NCCCn2cnnc2)ccc1F 58537,N1(C(C2N(CC)CCCC2)=O)CCC(C(=O)NC2CCC(=O)N(C)C2)C1(C)C 58538,CN1CC(C(=O)NCCC2CN(C(c3cnn(C(F)F)c3)=O)C2)CC1=O 58539,CSC1=C(C(=O)NCC2CCC(NC(C3CCC(C(C)C)CC3)=O)C2)CCCC1 58540,Cc1occc1CC(=O)NCC(C)(F)CNC(C1(c2ccn(C)n2)CC1)=O 58541,C1(CNC(C(C)NC(C)=O)=O)(NC(c2n[nH]cc2C2CCC2)=O)CCOC1 58542,C(=O)(C(C(C)NC(c1ncncc1Cl)=O)C(C)C)NCc1nccc(C)c1F 58543,N1(C(C2CC=C(C)CC2)=O)CC2(CCC2NC(c2cc(Cl)no2)=O)C1 58544,Cc1cccc(O)c1C(N1CC(NC(=O)C(c2cncnc2)C)C(C)(C)C1)=O 58545,S(=O)(=O)(c1ccc(NCCC(C)(C)F)c(Br)c1)N1CCCC(CCC)C1 58546,C(CC(=O)NCCCNC(=O)C(c1cccs1)C1CC1)N(CC)CC 58547,C1(O)(CNC(c2n(C(C)C)ncc2)=O)CCN(C(=O)CN2C(=O)CCC2=O)C1 58548,N1(C(CCCC#C)=O)CCC(C2CCN(C(=O)C(C)SC(C)C)C2)CC1 58549,C1(NC(=O)C(F)CC2CCC2)C2CC1N(C(=O)CC1(N3CCCCC3)CC1)C2 58550,CC(CN(C)C)C(=O)NC1CCC(CNC(C2(C)CC2Br)=O)C1 58551,C1(C(=O)NCCC(CNC(c2cnc(C3CC3)[nH]2)=O)OC)C(C#N)C1(C)C 58552,Cc1c(NCC2(CN(C)C)CCCC2)ncnc1N1CCS(=O)C(C)C1 58553,c1(NC(N2CCCC(NCc3sccc3F)C2)=O)cccc(C(F)(F)F)c1F 58554,c1(OC)nscc1NC(C1(CCNC(C2CC3(CC3)C2)=O)CCCC1)=O 58555,C12(CCN(C(c3cncc(Oc4cncnc4)n3)=O)CC1)COCC(=O)N2.CO 58556,N1(C(C2CC(=C)C2)=O)CCCCC2(CCN(C(c3cnn(C(C)C)c3)=O)C2)C1 58557,c1(C(C(=O)N(CC(C)O)CCNC(C2(OC)CC2)=O)OC)ccccc1 58558,Cc1ncccc1CC(=O)NC(CNC(C1CC1C(=O)OC(C)(C)C)=O)CC(C)C 58559,C1(CCN(C)C(c2ccc(Cl)o2)=O)CCN(C(c2c[nH]cc2C(F)(F)F)=O)CC1 58560,C(=O)(C(F)C1CC(NC(=O)C(F)OC(F)(F)F)C1)N(CCC)CCO 58561,C#CCC(C)(CC)C(=O)NCCC1CCN(C(=O)Cn2[nH]cnc2=N)CC1 58562,CCC(CC(=O)NC1(C(=O)NC23CC2COC3(C)C)CC1)CC(C)C 58563,c1(C(=O)NCC(C)NC(=O)CC(C(F)F)n2cccn2)cc(O)ccc1OC(F)F 58564,Cc1cnc(N(C2CCN(C(=O)Cn3cccn3)C2)C)nc1C 58565,C1(C(=O)NCC(COC)(C)C)(CF)CCN(C(=O)COCCCN=[N+]=[N-])C1 58566,C#CCC(C)(C)C(=O)NCC1(O)CC(C(N2CCCCCCC2)=O)C1 58567,C1(OC2(c3cnc(N(C(C)C)C)o3)CC2)CC2(C1)CC2NC(COC)=O 58568,Cc1c(F)ccc(Cl)c1C(=O)NCCN(C(=O)CC1=CCOCC1)CC(C)O 58569,Cc1csc(CCCC(=O)OCCNC(C2CC(OC3(C)CCOC3)C2)=O)n1 58570,C1(C(N2CC(N(C)C)CC(C)C2)=O)(NC(Cn2nc(C)oc2=O)=O)CCC(C)(C)C1 58571,C1(C(=O)NC2(C)C(C)CCC2)CCOCCN1C(=O)C=CCC1(N(C)C)CCC1 58572,N1(C(C=CCOC)=O)CCC(CCNC(C2CCC2(C)C)=O)C1 58573,c1(C(N2C(CNC(C(C=C)(F)F)=O)CCCC2)=O)cccc(C)c1Br 58574,N1(Cc2cn(C)nc2)CCC(NC(=O)CCc2ccccc2)C(C)(C)C1 58575,C(=O)(C1=CCCOC1)N1CCC(CCOC)(NC(=O)CC2CCCN2C)C1 58576,c1(-c2ccc(C)cc2)cnc(Nc2ccnc(-c3cccc(CO)c3)c2)c(O)c1 58577,C(CNC(=O)CC)(CC(F)(F)F)NC(C1CCC(CCCC)CC1)=O 58578,CCC(C)C(O)C(=O)NC1(CNC(=O)CCCOCCC(C)C)CCOCC1 58579,c1(CC(N2CC(CNc3ccnc(C)n3)OCC2)=O)cc(F)c(F)cc1F 58580,C12(CCNC(c3c(C#N)scc3)=O)CCC1CN(C(=O)C(C1CCCCC1)F)C2 58581,C1(C)(C(=O)NC2C(NC(C3CCC(OC)CC3)=O)CCC2)CCC(C)(C)CC1 58582,c1(SCC)nc(N2CCCC2C2(NC(c3cnc(C)o3)=O)CCC2)cc(C)n1 58583,c1(CC(=O)NC2C(N(C(c3cc(C)sc3)=O)C)CCCC2)cc(F)cc(F)c1F 58584,c1(C(N2CCC(C)N(C(c3ccnc(F)c3)=O)CC2)=O)cccc(F)c1[N+](=O)[O-] 58585,CC(N=c1[nH]c(N2CCOC(C3CCCC3)C2)nc2c1SCC2)c1ccncc1 58586,C1(NC(c2c(SC)cccn2)=O)CN(C(=O)C(C)(O)CC(C)C)CC12CCOCC2 58587,C1(OCCC)CCCN(C(C2(C(C)NC(c3cnc(C)o3)=O)CC2)=O)C1 58588,c1(-c2nnc(SC3C(C)SCC3)n2C2CC2)ccc2ccccc2c1 58589,CC(CC1=CCCCC1)(c1nnnn1C1CC1)NCCc1ccccc1COC 58590,CC1(C)CN(CCO)Cc2cccc(NCC3CCCC4CC34)c2O1 58591,C1(NC(CNC(=O)NC)=O)CCC2CCC1N2C(c1cnc(NC(C)C)nc1)=O 58592,C1(CNC(C=CC=CC)=O)CN(C(=O)CCc2ncccn2)C(C)(C)C1 58593,C1(C(N(CC#C)C)=O)CC12CCN(C(c1cn(C)ccc1=O)=O)CC2 58594,C(C(C(=O)NCC(COC)OC)C(C)C)NC(C1(C#C)CC1)=O 58595,C1(CC)CN(C(C2(C3(O)CCC3)CC2)=O)CCC1NC(c1ncccc1OC)=O 58596,c1(N(CC(N2CCCC2c2cn(C(C)CO)nn2)=O)C(C)=O)c(F)cccc1Cl 58597,Cc1nc[nH]c1C(=O)N(C)CCOCCN(C)C(C1CS(=O)(=O)C1)=O 58598,c1(C(=O)NC(CC)CN(C(=O)C=CC(F)(F)F)C)c(C)cc(C)nc1C 58599,C1(C)(C(=O)NC(CNC(CC2N(C)CCCC2)=O)C2CC2)CCC2CC2C1 58600,N1(C(C)Cc2cc(F)ccc2F)CCC2CCN(c3cc(=O)n(C)cn3)CC2C1 58601,C1(NC(c2ccc(OC)s2)=O)CC(CNC(c2cc(C(C)=O)cs2)=O)C(O)C1 58602,c1(C(N2C(CNC(c3ccc(OC)nc3)=O)C=CC2)=O)cnn2c1OCCC2 58603,C(CNC(c1nc(C)oc1C)=O)(C(C)C(C)C)NC(CCCC)=O 58604,C1(C#N)(CC(=O)NC2C(NC(CCCc3c(C)ccs3)=O)CC2)CCCCC1 58605,C1(NC(C(C=CC)O)=O)CCC2(CC1)CN(C(=O)CC1CCCC(C)C1)C2 58606,C1(O)(CN(C(C(C)c2cc[nH]n2)=O)C)CCN(C(=O)CCn2ncn(C)c2=O)C1 58607,N1(C(CC=CC=C)=O)CCCC2CN(C(c3cc(Br)ccn3)=O)CCCC12 58608,Cc1ccnc(C)c1C(=O)NCC12CC1CN(C(C1CCOC1)=O)C2 58609,N1(C(=O)NC)CCC(C(N2CCC(ON(C(=O)Cc3cc(C)cs3)C)C2)=O)C1 58610,CC(C(=O)NC1CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC1C(F)F)C(F)(F)C(F)F 58611,Cc1cn2cccc(C(=O)N(C)CC3(NC(c4cnoc4C4CC4)=O)CC3)c2n1 58612,c1(C(N2CC(NC(C(CC)n3ccnc3)=O)C(C)CC2)=O)ccc2scnc2c1 58613,C1(CNC2(c3n(CC=C)nnn3)CCCCC2)CCC2(CC1)CC2 58614,CC(CC(C)(F)F)C(=O)NC1COCC1NC(c1cccc2c1COC2)=O 58615,C(=O)(CCC(C)(C)[N+](=O)[O-])N(C1CCCN(C(=O)C=Cc2csc(C)n2)C1)CC 58616,Cc1ccc(C(N2CC=CC2CNC(c2ccnnc2C(F)(F)F)=O)=O)cc1F 58617,N1(C(c2c(C)nc[nH]2)=O)CCC(C2CCN(C(C34CSCC3C4)=O)CC2)CC1 58618,c1(C(=O)NC2(CO)CCN(C(Cc3nc(C)sc3)=O)CC2)cc2ncccn2n1 58619,c1(SC)cscc1C(=O)N(CC(C)CNC(=O)CC(C)O)C 58620,C(=O)(C1CCc2cc(F)ccc21)NC1CN(C(c2cncc(OC)c2)=O)C(C)CC1 58621,N1(C(COc2cccc(C)c2C)=O)CCC(C2CC2NC(=O)CC(C)F)CC1 58622,C12(C(=O)OC(C)(C)C)CC(C(=O)NCCNC(c3csc(Cl)n3)=O)(C1)C2 58623,C1(C2CCN(C(C3(C)CC3(F)F)=O)CC2)(NC(CCc2ccn(C)n2)=O)CCC1 58624,C1(CNC(C2C(OCC)CC2)=O)CC(F)(F)CN1C(c1cccc(N)c1)=O 58625,N1(C(C(C)OCCC=C)=O)CCCC1C1(C(=O)NCc2scnc2Cl)CC1 58626,C1(C(=O)NC(CC(=O)NCCCS(C)=O)CC2CC2)CC(=O)C12CCC2 58627,C1(OC)CC(C(N2CC(=O)N(C)C2)=O)N(C(=O)Cn2cccc2)C1 58628,C1(C(=O)NCC=CCNC(c2ccccc2C(F)(F)F)=O)CCCCC1C1CC1 58629,N1(C(C(CC2CCC2)OC)=O)CC(NC(=O)C(N)=O)C(c2cscc2C)C1 58630,c1(CCC(=O)NC(CNC(CC=C(C)C)=O)C(C)C)cc(Br)c(C)o1 58631,CC1(F)CN(C(c2cnc(S(C)(=O)=O)s2)=O)CCN(C(C2OCCC2CN)=O)C1 58632,CCC(C)C(O)C(=O)N1CCCC(CC)(NC(=O)CC2CC3C=CC2CC3)C1 58633,C1(C(=O)NC(C)Cc2ccco2)CSCCN1C(=O)CC1CCC(=O)NC1 58634,N1(C(c2cc(C)oc2C)=O)CCC(NC(=O)COCc2nc(C)no2)CC1C 58635,N1(C(Cc2cccc(C#C)c2)=O)CCC2C(CCN2C(c2cnnc(O)c2)=O)C1 58636,c1(C(C(=O)NCC(C)(C)NC(c2ccn(CC)n2)=O)C)cccc(C(=O)OC)c1 58637,CC1(C(N)=O)CCCN(CCc2c(C(F)(F)F)cccc2Cl)C1 58638,CC1CC(c2cn(C3CCC3)nn2)CCN1C(c1cc[nH]c1C1CC1)=O 58639,C(=O)(CCC(C)CN(C)C)NC(CC(C)NC(c1sc(C(=O)OC)c(N)c1)=O)C 58640,CC1CN(C(C2CC(O)CCN2)=O)CCN1C.c1cc(Cl)cnc1F 58641,CC1(C)CC(C(N2CC3(CCC(=O)N3)C2)=O)CN(C(C2CCCC23CCC3)=O)C1 58642,c1(OC)cc(F)c(NC(C2(C)CCN2C(=O)Cc2ncccn2)=O)c(F)c1 58643,C1(NC(=O)CCOCC(F)F)CC2CCC(C1)N2C(c1cc2c([nH]1)CCCC2)=O 58644,c1(C(N2C(CN(C(CC3(C=C)CC3)=O)C)CCC2)=O)cncc(Br)c1C 58645,c1(C(=O)NCC23C(NC(C(C4CC4)SC)=O)CC(CC2)C3)ccc(C#N)c(C)c1 58646,N12CCCCC1CC2=O.C1(CNC(C)=O)CN(C(C2CC(C(C)C)C2)=O)CCO1 58647,N1(C(c2c(C)onc2)=O)CC(NC(c2cccc(N)c2F)=O)C(C2CC2)C1 58648,C1(NC(CC2C(NC(C(C(C)O)N(C)C)=O)CC2O)=O)CCCC(O)C1O 58649,C12(C(N3CCC(CNC(C(C)SCC)=O)C3)=O)COCC1CS(=O)(=O)C2 58650,N1(C(=O)NC2C(CC(C)C)C2)CCC(N2CC(F)C2)CC1 58651,C12(C(N3CC4CC(NC(c5cccc(C)c5F)=O)C4C3)=O)CCCCC1OCC2 58652,Cc1oc(C)c(C(=O)NCCN(CCOCCO)C(c2nc(Cl)oc2C)=O)c1C 58653,C(=O)(C#CC1CCCCO1)NC1CCC(NC(c2sc(C)c(C)c2C)=O)CC1 58654,c1(CC(=O)N(C(CCNC(c2c(C)n(C)nc2)=O)C)C)ccn2cncc2c1 58655,S(=O)(=O)(c1ccc(Br)cc1F)C(N1CCC2C1CC2(O)C(F)(F)F)=O 58656,CCC(F)(F)CC(=O)NCCCC1CN(C(c2coc(C3CCC3)n2)=O)CCO1 58657,c1(C(=O)NCC(CC)NC(c2ccc(F)cc2C#N)=O)c(F)cc(C)cc1Cl 58658,CC(CC(=O)NCC(CNC(=O)C=CC(F)(F)F)CO)c1cnn(C)c1 58659,c1(OC)nccc(C(N2CCN(C(=O)C(C)Cc3cnc[nH]3)C(CO)C2)=O)c1N 58660,N1(C(C(CC(=C)C)OC)=O)CCCC(O)(CNC(=O)C(C)OCC)CC1 58661,c1(C(N2CCN(C(C3(CC)CC3(F)F)=O)CC2C2CC2)=O)ccc2c(c1)CCC=C2 58662,C1(CNC(Cc2c(C)nc[nH]2)=O)CCCC(C(=O)NC2(C)CCCC2)C1 58663,c1(C2C(C(=O)NC(CC(C)NC(c3n(CC)nnc3)=O)C)C2)cccc(C#N)c1 58664,C(C(C)C)(C(O)C(=O)N1CCCCCC1C(N1CC([N+](=O)[O-])C1)=O)OC 58665,C1(CNC(c2ncn(C(C)C)n2)=O)CC(C)CCN1C(=O)CP(C)(C)=O 58666,C(=O)(CC(C(F)(F)F)NC(=O)CC(C)C1CC1)NCCN(CCC)CCC 58667,Cc1cc(C(=O)N(C2CN(C(=O)Cc3cnn(C)n3)C2)C)cn1C(C)C 58668,C1(CN(C2CCN(c3cccc(Br)c3)CC2)C)CC(F)(F)C12CCC2 58669,CCC(CN(C)C)CC(=O)N(CCCC(=O)NCC1(C)CC1(F)F)C 58670,c1(CNc2c(F)cc(C(F)(F)F)cn2)ccc2ncc(Br)cc2c1 58671,c1(C(CO)NC(C(C)C#N)=O)ccc(F)c(Cl)c1 58672,N1(C(CC(=O)NCC#C)=O)C2CCC1CC(N(C)C(C1Cc3nccn3C1)=O)C2 58673,C(=O)(C(C)(C)C(C)C)N(CCCc1onc(C)n1)C.C1(=O)C=CCN1 58674,C1(C(=O)NCCNC(CC=C)=O)CCCC1NC(=O)OC(C)(C)C 58675,C(=O)(C(O)CC(=O)OC)NCCCOCCN(C(COCC#C)=O)C 58676,N1(C(C2(CC3CCC3)CC2)=O)CCCC(O)(CNC(C2(F)CCS(=O)(=O)C2)=O)C1 58677,c1(CC(N2C(C(=O)NCc3n(CC)nc(C)c3)CC2)=O)cc(F)cc(Cl)c1 58678,c1(C(N(CCCNC(C=CCCC)=O)CC)=O)ccc(F)c(S(N)(=O)=O)c1 58679,C1(N(C)C(C2(C)C=CCN2C(=O)CSc2cccnc2)=O)CCCCCC1O 58680,N1(CC(C2CCCC2)=O)CCS(=O)(=O)C(CCNC(=O)CCc2cn[nH]c2)C1 58681,CCC(CC)(CCNC(c1ncccc1O)=O)NC(c1ccc(Cl)cc1F)SC 58682,n1(CC)ccc(C(=O)NCCC(C(C)C)NC(c2csc3nccn23)=O)cc1=O 58683,C1(C(N(CCC(=O)NCC(C#C)CC2CC2)CCO)=O)C2CCCCCC12 58684,N1(C(C(CNC(c2c(CC)con2)=O)C)=O)CC(C)OCC1C 58685,CCCC(C)(C)CC(=O)N1C2CCC1CN(C(C1(n3nccn3)CC1)=O)C2.C 58686,N1(C(CCNC(c2ccc3c(c2)CC3)=O)=O)CCSC2CCCC12 58687,C1(C(=O)NCC2CCCN2C)(NC(c2c(CC)nns2)=O)CCCCCC1 58688,c1(OCCC(=O)NC(C2(O)CCN(C(C3(CC)CC3)=O)C2)C)ccc(C)c(C)c1 58689,c1(C(N2CCC(NC(CC)=O)CC2)=O)cc(C2(C)CCO2)ccc1F 58690,C1(CNC(c2sccc2Cc2cnncc2Cl)=O)CCCCCCC1 58691,c1(C(=O)NCC(CN(C(CCC(=O)NC)=O)C)O)ccc(OC)c(S(N)(=O)=O)c1 58692,C1(NC(c2c(OC)cncc2)=O)CCN(Cc2ccc(Br)[nH]2)CC1O 58693,C1(C(=O)NC(CN(C(Cc2c(C)nn(C)c2Cl)=O)C)(C)C)CN(CP(C)(C)=O)C1 58694,C(=O)(CC1CC2(CCC2)CCO1)NCCCOCC(C)(C)NC(COCCC)=O 58695,C(CCC(c1nnnn1C(C)(C)C)(C1CCCC1)CCn1cncn1)OC 58696,c1(C(=O)NCCC2(CNC(CCC(C)OC)=O)CC2)cnn2ccncc12 58697,c1(C(=O)NC2(CCNC(C(CC#C)C3CC3)=O)CC2)ccc(C)cc1C 58698,C1(CNC(c2c[nH]c(=O)cn2)=O)CCCCN(C(C2CC3(C2)CC3F)=O)C1 58699,C1(C(C)(C)C)(CNC(C2(C)CCCS2)=O)CCN(C(c2ccc(F)s2)=O)C1 58700,C1(C(=O)NC2CCCN(C(C(C)(C)C)=O)C2)(C(N2CCCC2)=O)CC2(CCC2)C1 58701,CC(=O)CC(C)(C)CC(=O)NCC(C)N(C(=O)C#CC1(C)CCCO1)C 58702,CON(CC1CCCCC1)C(=O)C(F)C(C)COC.C12CCCCCCN1C2=O 58703,Cc1ccc(C(=O)NCCC2CCC(NC(c3cnnn3C)=O)C2)cc1C 58704,N1(C(C=C)=O)CC(C)(C)CC1CC(=O)NC1CCC(O)(C(=O)O)CC1 58705,C1(C2CC2)(C(N(C(CNC(C(C=C)O)=O)Cc2ccccc2)C)=O)CCC1 58706,c1(C(N2CCN(C(C)=O)CC2c2cccc(F)c2)=O)cccc2ccn(C)c12 58707,Oc1c(CNCc2ccccc2F)cc(Br)cc1Cl 58708,N1(C(CC2N(C(C3CC(OCC)C3)=O)CCC2)=O)CCC2(CC1)CSC2 58709,C1(C(=O)NC2C(C(N(CC)Cc3cncn3C)=O)OCC2)CC1C1CCC1 58710,C=CCN=C(NCCc1nc(C)cs1)NC(c1nccc(C(F)F)n1)C 58711,c1(C(=O)NCCOCCNC(COCCCC)=O)c(F)cc(F)c(F)c1F 58712,c1(C(=O)OC)c(C)[nH]c(C(=O)N(C2CC(NC(=O)C(F)C3CCOC3)C2)C)c1C 58713,N#CC1(CC(=O)N(C2(C(=O)NCC(C3CCCO3)O)CCC2)C2CC2)CCC1 58714,Cc1cc(NC(=O)C(Cn2cncn2)NC(=O)CC2CSCCO2)cs1 58715,C1(OCC(=O)Nc2ncc(C3CC3)s2)CCN(CCNC(=O)C2CC2)C1 58716,c1(CN2CC(=O)N(Cc3c(C(C)C)noc3)C2=O)nc(O)c2ccc(Cl)cc2n1 58717,Cc1noc(C)c1C(=O)NC1(CCNC(=O)CCN2CCOCC2)CC1 58718,C(=O)(C1(C)CCn2c(C)nnc21)N1CCCC2(CCN(C(COC)=O)C2)C1 58719,C(C(COC)CC(=O)N1CCOC(C)(C)C1)OC.N1CCC2CC12C=O 58720,N1(C(C=CC(CC)C)=O)CC(C2CC2)(C(=O)NCc2ccc(CO)o2)C1 58721,C(=O)(C(CCNC(=O)CCC(C)C)OC)N(CCC1CC1)CC 58722,N1(C(c2ccccc2O)=O)CC(F)CC1C(=O)NCC(O)C(F)(F)F 58723,CC(C(=O)NCC1CCC1NC(=O)Cc1c(F)cccc1F)C1=CCCC1 58724,Cn1cnc2nc(=NCCc3ncoc3C3CC3)[nH]c(NCC3CCCC3(F)F)c12 58725,c1(C(N2CCN(C(=O)N(c3ccns3)C)CC2)C)cccc(O)c1 58726,C1(CNC(c2c(C)csc2)c2nnnn2-c2ccc(I)cc2)CCC2(CCC2)O1 58727,C(C(F)(C(=O)N(C)CCCCCC)C(C)C)NC(C1CCC(=C)CC1)=O 58728,CC(C)C(C(=O)N1CCC(O)(C(=O)NC(C)C(F)(F)F)C1)c1ccccc1 58729,c1(C(=O)NCC2(C(N(C3COCC3O)C)=O)CCC2)cn(C)cn1 58730,Cc1cccc(C(=O)NC2CCCCC2N(C)C(C2OCCCO2)=O)c1 58731,N1(C(C(C2CCC2)OC)C(=O)NC2CCOC2)C2CCC1CC(=O)NC2 58732,C1(CNC(CNC=O)=O)CN(C(c2ccc(NCCO)cc2)=O)CC1C(F)(F)F 58733,N1(C(C(C(C)C)NC(COC)=O)=O)CC2(CCN(C(=O)C(=O)CC(C)C)C2)C1 58734,N1(C(C(c2nccc(C)c2)(C)C)=O)CCN(C(=O)Cc2ccc(O)c(C)c2)CC1C 58735,CN(NC(=O)C(F)c1cncs1)C(N)=O 58736,c1(C(C)NC(CNC(C(=O)OC)C(N2CC(C)C(F)(F)C2)C)=O)ccc(F)c(F)c1 58737,c1(C(=O)NCCCN(C(CCOCC#C)=O)C)c(C)nc2sc(C)nn12 58738,c1(NC(C)=O)ccc(NC(C2CCCN(CCF)C2)=O)cc1C 58739,C1(OC)CC2CCC(C1)N2C(=O)CC(CC(C)C)NC(=O)C(C)OCCC(C)C 58740,C1(OCC)CC2(C1)CC2C(=O)NCCC(C)NC(=O)C(F)(F)COC 58741,c1(C(N2C(CCCNC(C(COC)(C)OC)=O)CCCC2)=O)nc(O)[nH]c(=O)n1 58742,CCCCCC(O)C(=O)N1CCC2C(NC(=O)CN(c3ccccc3)C)C2C1 58743,c1(CCC(=O)NCCCOCCCNC(C(CC#C)C)=O)cccc(F)c1F 58744,n1(CC(=O)N(C2CCN(C(C3CCC(F)(F)C3)=O)C2)C)ccc(=O)c([N+](=O)[O-])c1 58745,C1(OC)CCC2C3CC1N2C(=O)c1cc3cc(Cl)c1.C(C)=O.C1CC1 58746,C1(CC(=O)NCCN(C(C=CC=C)=O)CCOC)CC(C(F)F)(OC)C1 58747,c1(SC)ccc(F)c(C(=O)N(C2CCN(C(c3cn[nH]c3)=O)C2)CCO)c1 58748,C1(OC)CC2CN(C(c3c[nH]c(=S)cn3)=O)CCN2C1 58749,CCCCCC(=O)NCC(CC)N(C(=O)C(C1CCCOC1)OC)C 58750,Cc1nc(C(=O)O)oc1C(=O)NCC(F)(F)CCn1cc(C(C)(C)C(=O)O)nn1 58751,C1(NC(C(CC)C2CCOCC2)=O)(NC(=O)CN2CCCNC2=O)CCCCC1 58752,C1(CNC(C(F)=CCC)=O)CCCC1NC(=O)COCC1(F)CC1 58753,CC1CN(C(=O)C(C)CNC(=O)C(C)(C)N=[N+]=[N-])C(C)CCO1 58754,C1(C(=O)NCCC2(C)CCOC2)(OC)CN(C(=O)Cc2cn(C)nn2)C1 58755,CC(C)C(CNC(=O)CC(C)(F)F)C(=O)NCC(O)CF 58756,CC1c2cccc(F)c2CCN1C(c1ccc(-n2cc(C3CCC3)nn2)cn1)=O 58757,C1(C(N2CCC(O)(CNC(c3nn(CC)nc3C)=O)C2)=O)CC(C(C)(C)C)=NO1 58758,CCC(CCOC)C(=O)NCC1(NC(=O)Cc2cnn(C(C)(C)C)c2)CCC1 58759,c1(CC(=O)NCC(=C2CN(C(=O)CCc3nncs3)C2)F)cc(Cl)ccc1Cl 58760,c1(CN2CC(NC(C(C)OCC=C)=O)C(C)C2)cccc([N+](=O)[O-])c1 58761,NC(=O)CC(C1CC1)NC(=O)CC1(NC(C2CCC(F)C2)=O)CC1 58762,N1(C(C=C=C(C)C)=O)CC(C(=O)NC2(CN(C)C)CCC2)C(F)(F)C1 58763,Cc1cccc(CNC(C23CCC(NC(C4CCC(CO)O4)=O)(CC2)C3)=O)c1F 58764,c1(C(N2CC2CNC(CC2C(C)C2)=O)=O)ccoc1-c1ccccc1 58765,N1(C(CCCCSC)=O)CCC2(CC1)CC2C(=O)NC1(C(C)C)CCC1 58766,C(c1cccnc1)=CC(=O)NCC1CC1NC(=O)CC1(c2ccon2)CCC1 58767,CC#CCC(C(=O)O)NC(=O)C(c1ccc(Cl)c(F)c1)F 58768,c1(C(C)NC(N2C(C=C)CCC2)=O)ccc(C#N)cc1F 58769,CC1CCC(C(=O)NCC2(NC(=O)CCCNC(=O)C(C)(C)C)CCC2)C1 58770,C1(C(N(C2CCN(Cc3ccnn3C)C2)C)=O)CC(=O)N(c2ccccc2)C1 58771,Cc1cnc2c(C(=O)N(C(C)CCNC(=O)C(O)CN(C)C)C)cnn2c1 58772,C(C(F)(C(=O)NCC(C)C=O)C(C)C)OC(C12CCC(OC)C1C2)=O.OC 58773,C1(CNC(C(=O)NCCC2CCN(CC)CC2)=O)CC(N(C)C)C12CCC2 58774,CCCC(C)(C)C(=O)NCCNC(c1nc(C)oc1Oc1ccc(Cl)c(C)c1)=O 58775,N1(C(c2nc(CC)sc2)=O)CCCC(O)(CNC(c2ccnc(Cl)c2OC)=O)C1 58776,n1(CCC(=O)N(CCCNC(C2(OC(C)C)CCC2)=O)C2CC2)ncn(C)c1=O 58777,c1(NCc2ccc(C(=O)NC(CN(C)C)(C)C)o2)scnc1C#N 58778,O=C(C1=COCCC1)NC1CCN(C(c2cnn(CCO)c2)=O)C(C2CC2)C1 58779,c1(C(N(C)Cc2cn(Cc3nnc(C)s3)nn2)=O)csc2c1CCOC2 58780,C12(CNC(c3ccc(CSC)o3)=O)CN(C(=O)C(C)N(C)C)CC1CCO2 58781,c1(C(=O)NCC2C(NC(CC3C(CC)C3)=O)CC2)cc2c(=O)cc[nH]c2s1 58782,Cn1nc(C(=O)NCC2CC2NC(c2cccnc2C(F)F)=O)cc1Cl 58783,c1(C(=O)NCCN(C(c2cc(C)on2)C)CC)ccc2nccnc2n1 58784,N1(C(c2nc(CC(C)C)sc2)=O)CCC(n2cc(CNC(=O)CO)nn2)CC1 58785,C1(C(=O)NC2CCCC2c2cc(F)cc(F)c2)CC2CN(C3CC3)CC12 58786,N1(C(C(C2CCC2)OC)=O)CC2CCCC2(NC(c2cccc(CCO)c2)=O)C1 58787,C1(OC)(CNC(=O)C=CC2CC2)CCN(C(=O)C(F)=C(C)C)CC1 58788,c1(C(=O)NC2CCC(N(C(C(C)NC(CC)=O)=O)C)CC2)cc([N+](=O)[O-])ccn1 58789,c1(C(=O)NC2(COC)CN(C(C(CC=CC)CC)=O)C2)cc(C)cc(C)c1O 58790,c1(C(=O)NCC(CC)NC(C2CCCC(F)C2)=O)c(OC)cccc1O 58791,c1(C(=O)NC(CNC(C(C2CCC2)OC)=O)C(C)(C)C)c(C)cc(C)nc1O 58792,C(=O)(C(O)CCCNC(=O)CC1(O)CCCOC1)N1CCC(C(C)OC)CC1 58793,c1(N(C)Cc2ccc(CO)cc2)ccc(S(=O)(=O)NC2CSC2)cc1Br 58794,C(c1cc(Cl)cc(Cl)c1)=CC(=O)NCC(CNC(C1CC(CC)C1)=O)(C)O 58795,C12(NC(C(C3CC3)SC)=O)CC(NC(=O)CN(C)S(N)(=O)=O)(C1)C2 58796,CCC(CC)C(C)C(=O)NC12CCC(NC(=O)C(=O)N(CC)CC)(CC1)OC2 58797,C(CC(C)C)(C(=O)NCC1CN(C(c2cccnc2O)=O)CCCO1)NC(C)=O 58798,C1(C(N(C)CCOC(F)F)=O)CC2CCC1N2C(=O)Cn1cnnn1 58799,C1(C(=O)OC)CC2(CCN(CC(Cl)C(F)(F)F)CC2)S1(=O)=O 58800,C(=O)(CCCC(=O)OC)NC(CCCCNC(c1nc(SCC)sc1)=O)C 58801,Cc1ncc(C(N2C(C(=O)Nc3cnc(N(C)C)nc3)CCC23CC3)=O)c(C)n1 58802,C1(C(=O)NC2CC(F)(CNC(c3ncc(C)cn3)=O)C2)CC2CCC1CC2 58803,C(=O)(C1=CCN(C(=O)CC)C1)N1CCC(C(=O)NCC2(C(=O)OC)CC(=C)C2)C1 58804,Cc1ncsc1C=CC(N1CCC(C(C)NC(C2C(C)(C)C2(F)F)=O)CC1)=O 58805,c1(C(=O)NCC(CN(C)C(C2CS(=O)(=O)CC(=O)N2)=O)O)cn2ccncc2n1 58806,C(C)(CCC(=O)N(C1CCN(C(=O)CC2OCCO2)C1)C)SC 58807,C(=O)(CCCCN(C)C(C)C)NC(c1ccc(F)cc1)CNC(C(CC)=CC)=O 58808,C1(C(=O)NC(C2CCCC2)C#C)CN(C(=O)C(O)c2ccco2)CCC1(C)C 58809,CCC(CN(C)C)(CC)C(=O)NCC1CN(C(=O)CCC2CC(OC)C2)CCO1 58810,C1(C2CCCCC2)(NC(c2ccc(C)cc2Cl)c2n(CC=C)nnn2)CC1 58811,C1(NC(C(C)Cc2ccccc2)=O)CC12CC(NC(=O)CCCC1CC1)C2 58812,CCC(C)C(C)C(=O)N1CCCCC(NC(c2c(N)cccc2F)=O)C1 58813,c1(C(=O)NCCCNC(c2ccc(COC)[nH]2)=O)cc(N)c(O)c(F)c1 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58831,C1(CNC(CC)=O)(CO)CC12CCN(C(=O)CC1CC(=O)C1)CC2.C#CCOC 58832,Cc1nc(C(N2CCSCC2C(=O)NCc2cc[nH]n2)=O)ccc1Br 58833,N12CCC3(CCC3C1=O)CC2.C(=O)(C(F)(F)C(C)O)Nc1c(SCC)cccc1 58834,C=CCC(C(=O)N(C1CCCCN(C(=O)Cc2cccnc2OC)C1)C)C(C)C 58835,c1(C(=O)NC23CCCN(C(C4=C(C)OCC4)=O)C2C3)ccc2ncn(C)c2n1 58836,CC1CCCc2cc(C(=O)NCCCN(C)C(C3CCC4(CCC4)OC3)=O)nn21 58837,N1(C(CC(C)N(C)C)=O)Cc2nccn2CC(NC(=O)Cc2cnccc2Cl)C1 58838,N1(C(c2ccc(C)c(F)c2F)C(=O)NCCOC)CC(C)OC2CCCCC12 58839,Cc1n[nH]c(C)c1CC(=O)NCCC(C)NC(c1coc(-c2cnn(C)c2)n1)=O 58840,C1(CC(C)NC(=O)C=Cc2cn[nH]c2)CCN(C(C2CC3CC3C2)=O)CC1 58841,c1(C(=O)NCC2CCN(C(c3cn(C)nc3Cl)=O)CC2)coc2ccc(F)cc12 58842,c1(C(N2CC(CC(C)NC(=O)CNC=O)C2)=O)cc([N+](=O)[O-])ncc1Br 58843,c1(OC)ccc(Cl)c(CN2CCCC(C(=O)Nc3ncc(F)cc3Br)C2)c1 58844,c1(C(=O)NCC=CCNC(C2(C#N)CC3CC3C2)=O)ccnc2ccccc12 58845,C1(C(N2C(C(C)(C)CNC(c3ccoc3)=O)CCC2)=O)CC12CCOC2 58846,C1(CC(=O)N(CCCOCc2ccccc2)C)CCc2ccccc2C1 58847,C(C(CO)(CO)N)NC.C(=O)(C(C)CN(C)C)C(C(n1ccc(C2CC2)n1)C)=O 58848,CCCCCC=CCNC(=O)C(C1CN(C(=O)CC2CCOCC2)C1)OC 58849,N1(C(C2CC(C)(O)C2)=O)CC2CCC(NC(=O)Cn3ccsc3=N)CC2C1 58850,N1(C(CCN(C(CCC(CC)C)=O)CC)=O)CC(C2CC2(F)F)C1 58851,N1(C(C(C)NC(C)=O)=O)CC=CC1C(=O)N(C)CCN1CCCCC1 58852,N1(C(c2ccccc2)N(CC(C)C#N)C)C(=O)C=CC1=O 58853,N1(C(C2N(C(c3ccc(C)cc3F)=O)CC=C2)=O)CCC2(CCCNC2=O)CC1 58854,C1(C)(C(N(CCCO)C)=O)CC12CCN(CCC1CC3CCC1O3)CC2 58855,CC1CN(C(c2cc(O)no2)=O)CC(C)CN1C(=O)CC1CCN(C)C1=O 58856,CCCC(CCC)CC(=O)NCC(O)CNC(c1sccc1CC)=O 58857,c1(C(=O)NC(CNC(C2CC(OCC)C2)=O)(C)C)cc(Cl)c(Cl)cc1OC 58858,CN1CCC(CC(=O)N(C)CC2(O)CCN(C(=O)CCC3CC3(C)C)C2)CC1 58859,c1(C(N2CCC(CC)C2c2cc(F)cc(F)c2)=O)cc(F)c(C(F)(F)F)c(F)c1 58860,CC1(CNC(=O)C=CC(=O)NC2CC2)CCCN(C(=O)CC(F)(F)Cl)C1 58861,C(N=c1[nH]c(=NC2CC3CC4C(C3)C24)c2ncccc2[nH]1)c1cc(C)c(F)cc1 58862,O=C(C1CCNc2ccccc21)NC1(CO)CN(C(C2CCC3CC3CC2)=O)C1 58863,S(=O)(=O)(c1ccc(=NCCn2cccn2)[nH]c1)NC(C)C1CC1 58864,C(=O)(C1=CC2CCC(C1)C2)N1CCC(CNC(c2c(C)cc(O)nn2)=O)CC1C 58865,c1(C(=O)NCC2N(C(C3CCN(C)C3)=O)CC(F)(F)C2)cn(C)c(=O)nc1O 58866,c1(CC)ccc(C(N2CC(C(C)NC(c3ccc(C(=O)OC)s3)=O)C2)=O)cc1 58867,C1(NC(c2cc3ccsc3[nH]2)=O)CC2CC(C1)N(C(C1Cc3nccn3C1)=O)C2 58868,C(c1ccc(S(C)(=O)=O)o1)=CC(=O)NCC(C)(C)NC(C1OCCO1)=O 58869,c1(C(=O)NC2C(CNC(c3c(C)cc(SC)o3)=O)CC2)cccn2cnnc12 58870,C(=O)(C(CC)C(C)(C)CC)NC1CCC(CCNC(c2ccc(C#C)o2)=O)C1 58871,C1(CNC(C#CC(C)(C)C)=O)C2CCC1CN(C(=O)CCN1CCCCC1=O)C2 58872,C1(C(=O)NC(CCCNC(Cc2cc(C)ns2)=O)C)CCN(C)C(=O)C1 58873,Cc1c(C(=O)NCC#CCNC(=O)CC2CCCC2(F)F)sc2ccccc12 58874,c1(CNC(c2ccc(OCF)nc2)(c2nnnn2C2COC2)C)ncc(Cl)cc1Cl 58875,C12(NC(c3cccc(Cl)c3)=O)CCCCC1N(C(c1ccncc1)=O)CC2 58876,O=[N+]([O-])c1cncc(-n2ccc(=NCc3ncnc4ccsc34)[nH]2)c1 58877,Cn1nc(Cl)c(C(=O)NC2CCN(C(=O)C(C3(O)CCCC3)F)C2)c1Cl 58878,C#Cc1cnc(NC23CCN(CC2)CC3)nc1.c1(C(=O)OC)nc(Cl)c(Cl)s1 58879,c1(C(=O)NCC(CC)NC(c2ccc(-c3ccccc3)o2)=O)csc(CSC)n1 58880,c1(NC(C(CNC(C)=O)C)=O)ccn2c(O)nnc2c1 58881,N1(C(COC)=O)CCC2(NC(c3cncc(C(=O)OC)c3)=O)CC2C1 58882,C1(CNC(C(n2ccc(C)n2)C)=O)C(C)CCCN1C(c1cc(C(N)=O)co1)=O 58883,c1(C(=O)NC2CCCC(NC(c3c(C(C)C)nn(C)c3)=O)C2)nccc(Cl)c1O 58884,C1(NC(CC(C=C)C)=O)Cc2ccccc2C1NC(C1(COC)CCCCC1)=O 58885,c1(C(=O)NC(CN(C(C2CCC3(CC3)C2)=O)CC)C)ccc(C(F)F)c(F)c1 58886,N#CC1CCN(C(C2(NC(c3ccoc3)=O)CCOCC2)=O)C1 58887,n1(CCC)nnnc1C(c1noc(C(C)(C)C)n1)NCC1(F)CC1 58888,C1(C#N)(C(=O)NCC2CN(C(C3CCN(C)C(=O)C3)=O)C2)CC2C=CC1C2 58889,C1(N(C(=O)C(N)=O)C)CN(C(=O)Cc2cnn(CC(F)F)c2)CC12CC2 58890,C1(N(C(c2cccc(OCC)c2)C(=O)NCC)C2CC2)CCS(=O)(=O)C1 58891,N1(C(C(C)N(C)C)=O)CCN(C(=O)CC(C)(C)c2ccccc2)C(CO)C1 58892,CC1(C)CCCC(CC(=O)NCCC2CCCN2C(=O)CN=S(C)(C)=O)O1 58893,N1(C(c2ccn(C(C)C)n2)=O)CC(C)CN(C(=O)CS(=O)(=O)C(C)(C)C)C(C)C1 58894,c1(C(N(C)CCN2CC3(CC3CO)C2)=O)nnc2c(Cl)cc(C(F)(F)F)cn12 58895,C1(NC(COC)=O)CC(NC(c2cnc(NC3CCCCC3)nc2)=O)C12CCC2 58896,N#CC1(C(=O)NCCC2CC(C(=O)NOCC(N)=O)C2)CCCO1 58897,C1(C(N(C2(C(F)(F)F)CCC2)C)=O)CS(=O)(=O)C12CCN(C(=O)OC(C)(C)C)CC2 58898,C#CC1(NC(=O)CC2CN(C)C2)COC1.C12(CC1)C(=O)N(C)CC2 58899,c1(CCNC(C(N2CC3C(C(=O)OC(C)(C)C)(C3)C2)=O)=O)cc(F)ccc1Cl 58900,C1(NC(c2c(C)ncs2)=O)CCCCC1NC(c1ccc(C(C)(C)C)s1)=O 58901,c1(C(=O)NC2C(C)(CNC(c3nc(C)oc3)=O)CCC2)ncc(C(N)=O)cc1Cl 58902,n1(CCC)cc(C(=O)NC2CN(c3ccnc(-c4nccs4)n3)CC2C)c(C)n1 58903,C12(CCNC(CC(C)(C)C3CC3)=O)CC(Cn3cc(C(C)(C)C)nn3)(CO1)C2 58904,S(=O)(=O)(c1ccc(NC2CCCC3(CCCCC3)C2)c(C#N)c1)N(CC(CC)C)C 58905,c1(Cc2cn(CCO)nn2)oc(C(N2CCSC(C3CCOCC3)C2)=O)cc1Br 58906,c1(C(C(=O)NCCCF)N(CCC2=NNC(=O)C2)C)cc2cc(Cl)ncc2o1 58907,N1(C(c2nnn(C)c2C2CCC2)C(=O)Nc2ccccc2)CC2CCCC2C1 58908,n1(CC(N2C3CC(CNC(C(CC=CCC)C)=O)C2CC3)=O)cnc2ccccc12 58909,c1(OCC)cc(Br)c(F)cc1C.c1(CC2CC2)nnnn1C1CCC1 58910,C(C(CC(C)C)C(=O)NCCN(C(C1CCn2nccc2C1)=O)C(C)C)OC 58911,C(=O)(C(O)CNC(=O)Cn1cc(C)cn1)N(CC)Cc1cccs1 58912,N1(C(Cc2ccc(OC)nc2)=O)CCC(C)C(NC(C2(OC)CCSCC2)=O)C1 58913,CCCCCCC(C)C(=O)N1C2CCC1(CNC(c1nc(C)oc1OC)=O)CC2 58914,c1(C(N(C2CC2CNc2nccc(C(C)(C)C)n2)C)=O)ccc(Cl)c(Br)c1 58915,N1(C(C(C)NC(C)=O)=O)CC(NC(c2cc(C(C)C)ccc2C)=O)C2CC2C1 58916,C(C(CC1CCCC1)C(=O)NC1CCC(CO)CC1)NC(=O)C=CC=CO.C(C(F)F)=C 58917,c1(C(N2CCC(CNC(C3C(C)OCC3)=O)C2)=O)cnn2ccn(C)c12 58918,C12(C(N(CCCC)C)=O)CCC(n3cc(C4CCCO4)nn3)(CC1)C2 58919,CCS(=O)CC(=O)N(CC(C)CNC(=O)CCCSC(C)(C)C)C 58920,CC1CN(C(C2CCO2)=O)CC1NC(=O)Cc1ccnn1C1CCOCC1 58921,c1(OCCC)cc(-c2ccc(NC(c3ccc(Cl)s3)=O)s2)cc(C#N)c1 58922,C(CC(C(=O)NC(CC1CC1)CC1CC1)NC(C1CC(COC)C1)=O)SC.C1(C)CC1 58923,S(=O)(=O)(c1cccc(C(N(CC)CC)=O)c1)NC1(C)CCC(NC(C)=O)C1 58924,c1(C(C)C)nnsc1C(=O)N.C(C)(CCN)C(C1(F)CC1C)=O 58925,C(N=c1[nH]c(=N)[nH]c(=NCCS(=O)(=O)CC(F)(F)F)[nH]1)C1(C=C)CCOC1 58926,S(=O)(=O)(c1ccc(NC2CC2)c(Cl)c1)NC1CC2(C=C2)C1 58927,N1(Cc2ccc(OC)nc2Br)Cc2ccccc2C1C(=O)Nc1ncccc1I 58928,c1(C(=O)NC2CCC(CCNC(C3C(C)=CCS3)=O)C2)cc(C)ccc1O 58929,c1(CCCC)cc(C(=O)NCC2(NC(=O)C=Cc3cocn3)CCOC2)c(C)o1 58930,c1(OC)ccc2occ(C(=O)NC3CCCCC3CNC(=O)C=CC(C)C)c2c1 58931,C1(CC#C)(C(=O)N(C2CCCC2)CCCNC(C23CCC2CC3)=O)CCCCC1 58932,C(=O)(CCCS(C)(=O)=O)NC1CCCC(NC(CCCCOC)=O)C1 58933,c1(C(=O)NCCOC2CN(C(=O)C(F)(F)CO)C2)ccc(=O)n2c1CCCC2 58934,c1(C(=O)NC(CC(C)NC(Cc2cc(C)no2)=O)C)c(C(F)F)cnn1C 58935,C(C(C(=O)NCC(C)CCO)NC(=O)CC1(C#N)CC1)OC(C)C 58936,N1(C(C=C(C)C2CC2)=O)CCCC12CCN(C(c1ccsc1C)=O)C2 58937,C(=O)(CC(F)(F)CC)N1CCC(CC)C1CC(=O)NC1(COC)CC1 58938,c1(C(N2CC(NC(C(C(C)C)(C)C)=O)C(C(F)(F)F)C2)=O)ccc2nccn2n1 58939,C1(C(N2CC(COC)(CNC(=O)Cc3cn[nH]c3)C2)=O)CC(C(F)(F)F)=NO1 58940,C12(C(=O)NCCNC(c3cccc(OC)n3)=O)CCCCC(OC)(C1)C2 58941,C1(C(=O)NCC(CC)N(C(=O)CCc2cncs2)C)CNC(=O)CC12CCC2 58942,N1(C(C(C)OCCC#C)=O)CCCC(NC(C2(C(C)(F)F)CC2)=O)CC1 58943,C(=O)(CCC(C)=O)NC(C(=O)Nc1c(OC)nsc1)CC1CC1 58944,C1(NC(C(N2CCOC2=O)C)=O)CCN(C(C2C3(CC3)C23CC3)=O)CC(O)C1 58945,N1(C(CN(CCOC)C)=O)C2CCC(C2)C1CNC(=O)Cn1nc(C)oc1=O 58946,C12(C(=O)NC3CN(C(c4c(N)nccc4)=O)C3)CC3CC(CC(C3)C1)C2 58947,C1(NC(c2nc(C(C)OC)oc2)=O)CN(C(=O)CC2(OC)CCC2)CC(C)(C)C1 58948,Cc1ccc(Br)c(NC(=O)Nc2ccccc2)n1.N12CC3(CC1C3)C2=O.CC 58949,C(=O)(C1=NOC2COCC12)N1C(C(=O)NCCC2=CCOCC2)C=CCC1 58950,Cn1nc(C(N2CCCC(CO)(NC(c3ccc(F)s3)=O)C2)=O)cc1C#N 58951,C(=O)(C(C)(C)CNC(C1CC(C)N1C(=O)CCc1cnco1)=O)OC 58952,N1(C(c2cc(CC)c(CC)o2)=O)CC(C2CN(C(=O)C(C)(O)CC)C2)C1 58953,c1(C(=O)NC2CCN(C(C(CC)SC)=O)C2)c(C)nn(CC)c1C(F)(F)F 58954,C(=O)(C1=NOCC1)NCCC(CNC(C(CSC)OC)=O)O 58955,C(c1ccc(Cl)c(F)c1)=CC(N1CCC(NC(C(C)(C)OC)=O)C(F)C1)=O 58956,C(CCCCC(=O)NC(CC1CC1)CO)NC(c1cc(OC)ns1)=O 58957,Cc1cc(C(N2CC(NC(c3cnc(C)n3C)=O)C(C)C2)=O)c2c(C)noc2n1 58958,C1(CC)CN(C(=O)C=CC2CCCO2)CC1NC(=O)C(Cl)=CCl 58959,Cn1c(O)nc2c(C(=O)Nc3ncc(C(F)(F)F)c(Br)n3)cccc12 58960,Cc1ccc(C)n1CCC(N1CCCC(F)C1)=O.c12cn(nn1)C1CCCC21 58961,C1(C)(CC)CCC(C(=O)NNC(=O)c2cnoc2)O1 58962,c1(N2CC(C)(C3CC3)OCC2)nc(=NCCC2CCCCO2)[nH]c2c1COCC2 58963,c1(C(=O)NC2C(NC(CN(C(=O)OC)C)=O)C2)cc2n(n1)CCO2 58964,C(=O)(C(c1ccccc1)=C(C)C)NCC1C2(N(C(C(COC)OC)=O)C2)C1 58965,c1(NCCS(=O)(=O)NC(c2ccc(C)o2)=O)ccc(F)cc1C#N 58966,C1(NC(=O)OC)CC(C)N1C(=O)C(O)C1CN(C(c2ncn(C)n2)=O)C1 58967,C(=O)(C(C)CC(C)C(C)=O)NC(C)(C)C1CC1.n1(CC)ccc(C(N2CCCC2C)=O)n1 58968,Cc1ccc(Cl)cc1-c1cn(CCCNC(=O)CCNC(N)=O)nn1 58969,c1(OCCCC(=O)NC(CNC(C2CC(CC)(CC)C2)=O)C)c(C)cccc1C 58970,N1(CCNC(CCN(CCCCOC)C)=O)CCN(C)CC1.C1(=O)C(C)(C)N1 58971,C(=O)(C(F)C(C)(F)F)NC(COC)CCO.c12conc1C(C)NC2=O 58972,C12(NC(c3nc(C(C)C)oc3)=O)CCCC1CN(C(=O)CN1CC3CC3C1)C2 58973,c1(CC)nccnc1C(N1CC(NC(c2c[nH]c(=O)cn2)=O)C1)=O 58974,S(=O)(=O)(c1cccc(F)c1Cl)Nc1ccc(C=C)cc1 58975,c1(C(N2C(CNC(c3cc(C)sc3)=O)C(C)CCC2)=O)ccc2c(n1)CCCC2 58976,c1(CN2C(C(=O)Nc3c(C(C)=O)cccn3)CC3CC32)c(C)cc(Br)cc1C 58977,c1(C(C(C)C)C(=O)NC2CC(CF)C2)ccc(Br)cc1F 58978,c1(C(N2CC(N(C)C(c3cccnc3)=O)C(F)C2)=O)ccc(Cl)c(F)c1F 58979,c1(C(=O)NC2CCCCN(C(=O)CS(=O)(=O)NC3CC3)C2)cnc2[nH]ccnc1-2 58980,C(=O)(CC1CCc2ccccc21)NCC1CN(C(C(C)=CC)=O)CC1C 58981,c1(C(N2CC(O)C(C3CC3)C2)C(=O)NCC(C)C)cc2cccc(Br)c2o1 58982,C(C#Cc1ncccn1)N1CCC(NC(CC=C)=O)CC1 58983,C(CCC1CC1)(C(=O)NCCc1ncn(C)n1)NC(C(n1c(C)ncc1)C)=O 58984,CCC(C)CC(C(=O)OC)NC(C12CC(C)(C1)OC2(C)C)=O 58985,C=C(C)CC(C(=O)N1CCC(C(F)(F)F)C1)NC(=O)C(C1CCOCC1)F 58986,c1(CC(=O)NCCN(C(=O)CN2CCCC2C(N)=O)CCOC)nonc1C 58987,CCCCC(O)C(=O)NC1CC(CNC(=O)CCC(=O)c2ccc(Cl)cn2)C1 58988,C1(N(C(C2(OC)CC2)=O)C)CCCCN(C(c2sccc2C(C)=O)=O)C1 58989,C1(C(N2C(CCNC(C(C=C)C)=O)CCCC2)=O)CCC(=O)N(C)C1 58990,C(=O)(C1=NN(C)C(=O)CC1)NC(C1(O)CN(C(c2c(C)nns2)=O)C1)C 58991,N1(C(CCC=CC)=O)CCC(NC(=O)C=Cc2cccc(OC)c2)C(CO)C1 58992,c1(C(=O)OCC)n[nH]c2c1CN(C1CCN(c3ccc(F)cc3)C1=O)C2 58993,N(C(=NCCCF)NCC1CC2(CCC2)C1)CC(N(OC)C)=O 58994,c1(C(=O)NC(CC)CN(C)C(C2CCOC(C)(C)C2)=O)ccc(=O)n2c1CCC2 58995,N1(C(C23N(C(=O)Cc4ccc(F)nc4)CC(C2)C3)=O)CCC2(CC1)CC2 58996,N1(C(c2cc(F)c(Br)cc2F)C(=O)NC)CC(C2CCCOC2)C1 58997,Cc1occc1C(=O)N(C)CCN(C(=O)C(CC1CC1)NC(N)=O)C 58998,C1(NC(c2c(C)sc(Br)c2)=O)CC2CCCC(C1)N2C(C12CC(C)C1C2)=O 58999,C12(CNC(C3CC(F)(F)C3)=O)CCC1CN(C(C1CCN(CC(F)(F)F)C1)=O)C2 59000,Cc1ccc(C(=O)NCc2nccs2)c(O)c1.N12CCN(CC1)CCCNC2=O 59001,Cc1nc(C(=O)NC2CC(O)(CNC(=O)C(O)CC(C)C)C2)cc(O)n1 59002,N1(C(c2n[nH]c(C)c2C)=O)CCC2(CC1)CC2C(N1CCC(CC2CC2)C1)=O 59003,N1(C(C=CC)=O)CC(C(=O)NC(C)CC(=O)NC)C(F)(F)C1 59004,c1(C(N(CC(C)O)CC)=O)cn(CCNC(C2OCCO2)=O)nn1 59005,C(C(C)(C)C(=O)N1CCC(CC2CC2)C1)NC(CC)=O 59006,C(C)(CCC(=O)NCC(Cn1cc(-c2nn(C)cc2C)nn1)SC)OC 59007,C1(C(=O)NC2C(CC=C)COC2)CCC2(CC2)N1C(=O)CC1CSCCO1 59008,N1(C(COCCCC)=O)CC(C)CN(C(c2cnoc2-c2cnccn2)=O)CC1C 59009,CC1=C(C)CC(C)(NC(C2(C)CN(C(=O)Cc3coc(C)n3)CC2C)=O)CC1 59010,C1(C(=O)OCC)CCCN(C(C23CC2CN(C(C2COCOC2)=O)C3)=O)C1 59011,c1(OC(C(CC)N2CSCC2=O)=O)cc(Br)c(C(=O)OC(C)(C)C)s1 59012,N1(C(C2C(CC)CCO2)=O)CCC(C(=O)NC(CN(C)C)C(C)(C)C)C12CCC2 59013,C(=O)(C1=CC2C=CC(C1)C2)NC(CCC=C)C(=O)N1CCCC(CC)C1 59014,Cc1nc(C(C)(C)C)c(C(=O)NCC2(NC(=O)CC3(O)CCCOC3)CCC2)s1 59015,N12CCc3cccc(c3C1)NC2=O.N1(C(CSC(C)(C)C)=O)CCNCC1 59016,c1(CC)ncc(C(=O)NC(C2CCCN2C(c2cnn(CCOC)c2)=O)C)s1 59017,N1(C(C)=O)CCC2CN(CCNc3ccc(C(=O)OCC)cc3)CC12 59018,c1(C(=O)OCC(=O)NCc2ccc(OC)c(OC)n2)ccc(C)c(S(C)(=O)=O)c1 59019,N1(C(CC(C)N(C)C)=O)CCCCC1C(=O)NCC1COCCO1 59020,c1(N2CCCC(O)CC2)ccc2nccc(CO)c2c1 59021,C1(NC(c2ncn(C(C)C)n2)=O)CN(C(C2CCCCS2)=O)CCC1(C)C 59022,C1(NC(C(C)OC)=O)C2CCN(C(=O)CC3CC(=O)NC(=O)C3)CCC12 59023,C1(C(=O)NC2C=CCCC2)CC(O)C(O)CC1CNC(C1(CO)CCCO1)=O 59024,c1(OC)ccc(Cl)c(C(=O)NCC2CC(NC(c3[nH]c(C)cc3C)=O)C2(C)C)n1 59025,N1(C(c2n(CC)nnc2)=O)CCC2(NC(=O)Cc3cc(Cl)sc3Cl)CC2C1 59026,N(C(=NCC1CC1)NC1CCN(C(C2(CCC)CCC2)C)CC1)C(N1CCCC1)=O 59027,C1(NC(CC2CCC(=O)N2)=O)CCN(C(=O)CC2C=CCCC2)C12CCC2 59028,C#CCCC(C(=O)NC(CCC)C(=O)NC)NC(=O)C(F)C(F)(F)F 59029,N1(C(CCC(=O)NC)=O)CCC2(CO)CN(C(c3coc(Cl)n3)=O)CC2C1 59030,C1(C(=O)NCCN(C(c2cc(C)c(C)s2)=O)CC)CCc2ncsc2C1 59031,c1(C(N2CCCCC(C)C2)=O)cnc2c(-c3ccc4[nH]ncc4c3)cccc2c1 59032,C1(=CC(=O)NCC2CCN(C(c3ccc(C(N)=O)[nH]3)=O)C2)CC2CCC(C1)N2C 59033,C1(NC(C2CCN(C)C2)=O)CC2(C1)CC1(CC(NC(C3(C)CC3(F)F)=O)C1)C2 59034,C(=O)(C1=C(NC(C2CN(C(c3ccccc3Br)=O)CCO2)=O)CCCC1)OC 59035,N1(C(C2CCCC3(CC3)C2)=O)CCC2(CC1)CN(C(=O)C(F)(Cl)c1ccon1)C2 59036,c1(OC)cc(-c2ccc(F)nc2)c(OC)cc1CN1CCCC(N(C)C)C1 59037,C1(NC(c2ccc(COC)o2)=O)(CF)CCN(C(C2CC(C)(OC)C2)=O)C1 59038,C#Cc1cn(C)nc1C(N1CCC(CNC(C2CCC2C(N)=O)=O)C1)=O 59039,C(=O)(C1=CCCOCC1)N1CC(C(C)Nc2nc(C(=O)OC)c(Cl)cn2)OCC1 59040,CC1CCN(C(c2nonc2N)=O)CC1NC(c1cn(C)c(=O)n1C)=O 59041,N1(C(C(C)NC=O)=O)CC2(CCN(C(=O)CCCCl)CC2)c2cc(F)ccc21 59042,N1(CC(=O)NCC(C)CN(C(=O)CC2(C)CC2(F)F)C)CCS(=O)(=O)CC1 59043,C1(OC)(CNC(=O)Cc2nccn2C)CCN(C(C2(C)CC=CCO2)=O)C1 59044,c1(C(=O)NCCC2(OC(C)C)CN(c3cc(C(C)=O)ncn3)C2)cc(F)ccc1F 59045,C1(C)(C(=O)NC(C#C)C)CCN(C(c2n[nH]cc2I)=O)C1 59046,C1(CC(=O)N(C2(C)CN(C3CCNC3=O)C2)C2CC2)CCCCN1C1CCCC1 59047,c1(OC)ccc(C(=O)NCCCNC(c2nocc2NC(=O)OC)=O)cc1OC 59048,C1(OC)C(NC(=O)C(C2(O)CCC2)NC(=O)C=CC2CCOC2)CC1O 59049,C1(NC(=O)Nc2cn(C(C)C)nc2)COC2(COC2)C1 59050,C1(NC(CCc2c(C)cccn2)=O)C(C)CCN(C(c2ccc(C#N)[nH]2)=O)C1C 59051,C12(C(N3CC(CCC)C(CO)C3)=O)CCC(CC1)N(C(=O)C(CO)OC)C2 59052,c1(C(=O)NCC=C(C)CNC(C2CC(=O)N(C)C2)=O)cnc(C)cn1 59053,C1(CCNC(c2ccc(C(CCC)=O)cc2)=O)NC(=O)CNC1=O 59054,CC(C)CC(C(=O)NC1CC1(C)C(F)F)NC(c1cnn[nH]1)=O 59055,O=C(C1=Cc2cc(F)ccc2OC1)NC1CCN(C(C2CC=CC(O)C2)=O)C1 59056,C1(C(C(=O)NCCCN(CC)CC)OC(=O)C(F)CC2CCOC2)CC(F)(F)C1 59057,N1(CCC(=O)CC(c2ccccc2F)C)CCN(C(=O)CNC(C2C(C)C2)=O)CC1 59058,c1(C(N2CC(CN(C(C3(C(=O)OC)CCCC3)=O)C)C2)=O)ccncc1Br 59059,Cc1nc(C(=O)NCCCN(C(C2CNC(=O)N2)=O)C2CC2)cc(O)n1 59060,c1(C(=O)NC(C(C)NC(=O)C=Cc2cc[nH]c2)(C)C)ccc2nn[nH]c2c1 59061,c1(C(=O)NCC2CC(F)(CNC(C3C(OCC)C3)=O)C2)cc2sc(F)cc2[nH]1 59062,Cc1cc(Cl)c(NC(=O)C(=O)NC2CCN(S(=O)(=O)C(F)F)C2)cc1O 59063,c1(CNC2C(F)(F)CCN(C(CC#C)=O)C2)ccc2cccnc2c1 59064,N1(C(CC(C)C2CC2)=O)CCCC(N(C)C(c2ccc(N)c(N)n2)=O)CC1 59065,c1(C(=O)NCC2(NC(c3cn(C)nc3)=O)CCOC2)cnc(C#N)s1 59066,C1(NC(c2n(CC)ncc2)=O)CCN(C(c2ccc(CO)cc2)=O)CCC1CO 59067,C(CC(=O)N1CC2(CC(CO)CO2)C1)(C(F)(F)F)NC(c1n(CC#C)ccc1)=O 59068,C1(N(C)C(c2cnsn2)=O)CCCN(C(c2cc(O)n(C)n2)=O)C1 59069,C12(CNC(=O)Nc3cn(C=C)nc3)CCC(CO)(CC1)CC2 59070,N1(CCC=C)CC(C)C(C)(CNC(=O)CC2CCC(C)(C)CC2)C1 59071,C12(CO)CC(C(N)=O)(C1)C1(CN(C(=O)C(C)CNC(C=CCOC)=O)C1)O2 59072,C(=O)(C=C1SCC(=O)N1C)N(C1CCCC(NC(COCC#C)=O)C1)C 59073,C1(C(=O)NCc2c(COC)nco2)(NC(=O)C(CSC)OC)CCCCC1 59074,C12(C(=O)OC)CC1CCC2NCC(C)(Cc1ccccc1)CO 59075,C12(NC(=O)CCCF)CCOCC1CN(C(=O)COc1cccc(Cl)c1Cl)C2 59076,C1(COC)CN(C(=O)CC(C)C(F)F)CCN1C(c1cncn(C)c1=O)=O 59077,c1(OC)cc(C(N2CC(NC(=O)CCc3n[nH]c(=N)s3)CC(O)C2)=O)cc(C)c1 59078,C=CCC(CC)NC(c1nnnn1C1CCCC1)CCC1(C#N)CCC1 59079,N1(C(c2n(CC)cc(Cl)c2)=O)CCCC(O)(CNC(C2CC2[N+](=O)[O-])=O)CC1 59080,c1(NC(c2ccc(C#N)cc2Br)=O)cccc2c1OCCC(=O)N2 59081,N1(c2cccc(COC)c2)N=C(C(=O)NN2CCC(OC3CNC3)CC2)CCC1=O 59082,C(CCCCC(=O)N1CCN(C(C2CCOC2C)=O)C(C)C1)=CC 59083,N1(C(C(C)P(C)(C)=O)=O)CCOC2(C1)CN(C(C1CC13CC(O)C3)=O)C2 59084,C1(C(=O)NCC(C)CC2CC2)CCN(C(=O)c2ccnc(O)c2)O1 59085,c1(CNC(c2n(CCCSCC)nnn2)c2ncc(C)s2)ccc(F)c(C)c1Cl 59086,C1(NC(CC=C=C)=O)CCN(C(c2ccc(CNC(C)=O)o2)=O)C1C(C)(C)C 59087,C(=O)(C1CCCc2sc(=N)[nH]c21)NCC(CCCC)NC(=O)CC(C)CF 59088,C(C(=O)NCC1(CNC(=O)CCNC(=O)C(C)(C)C)CC1(F)F)(C(C)C)SC 59089,Cc1cc(Cl)c(C(=O)NCCC2CCCN(C(=O)COCc3nc(C)no3)C2)s1 59090,c1(C(N2C3CCN(C(c4c(CC)nc[nH]4)=O)CC3C2)=O)cn2ccc(F)cc2n1 59091,c1(NC(C23CC(C(=O)Nc4cccc(F)c4Br)(C2)C3)=O)cc(F)cc(Cl)c1 59092,c1(C(=O)NC(C)CNC(C2CC(n3ccnn3)C2)=O)[nH]nnc1-c1ccccc1 59093,C(=O)(CCC(C)CC)N1CCC(CC=C)(C(N2CC(CS(C)=O)C2)=O)C1 59094,C1(CC(=O)NCCN2CCN(C(C3C(SC)CCC3)=O)CC2)CCCC(C#N)C1 59095,O(P(C)(=O)CNC(C1CC=CCN1C(=O)CC1CCCOCC1)=O)CC 59096,CCCCCCCCCC(=O)NCC(C)CNC(c1cc(N)nc(Cl)c1)=O 59097,N1(C(CC(C2CC2)SCC)=O)CCCN(CCCNC(c2cccc(C)c2)=O)CC1 59098,C12(CNC(c3c(C)nsc3)=O)CCCC1N(C(=O)C(C)C1CCOC1)CCC2 59099,C1(CN(C(C(C=CC)O)=O)C)CN(C(=O)CC(CC)c2ccccc2)CCO1 59100,N1(C(=O)CNC(N)=O)CC(NC(C2(COCC)CC2)=O)CC(C)C1 59101,c1(C(N(CCNC(C(CC)(CC)OC)=O)CC2CC2)=O)cnc2[nH]nnc2c1 59102,C1(CNC(c2nc(COC)oc2)=O)CCN(C(C2CC3(CC3)C2)=O)CC1O 59103,C1(CCNC(=O)CCc2nc[nH]n2)CSCCN1C(=O)Cn1cc(C(F)F)cn1 59104,C(=O)(C(C(C)(C)C)NC(C)(C)C)NCC1(CNC(c2c(C)cno2)=O)CCC1 59105,CCC(C(=O)OC)C(=O)NC1CC2(C1)CN(C(=O)CSc1nnnn1C1CC1)C2 59106,Cc1ccc(C(=O)NCC2CN(C(C3CCC3C(C)(C)C)=O)CCO2)c(F)c1Cl 59107,C(=O)(CCCCN(CC)CC)NC1CC(NC(=O)CC2CC(C)(C)CO2)C1 59108,c1(C(=O)OC)ccn2cc(C(N3CCC(Oc4ccccc4)CC3)=O)nc2c1 59109,C1(C(CNC(C2CC(C(F)(F)F)(OC)C2)=O)C)CCN(C(C2CC(O)C2)=O)CC1 59110,C(N=c1nc(N2CCC(Cn3cccn3)CC2)c2ccccc2[nH]1)C1(CO)CC1 59111,C1(C(N2CC(NC(=O)CC3CCC3)CC(OC)C2)=O)CS(=O)(=O)CC(=O)N1 59112,N1(C(COCCCOC)=O)CC(O)CC1(C)C(=O)O.C1CC(C)N1 59113,c1(C(N)=O)ccccc1C(=O)NC1CC(C2C(CNC(C3CCCCO3)=O)C2)C1 59114,N1(C(c2cnc(CC)o2)=O)CCC(CC)C1CNC(c1ccsn1)=O 59115,C1(Br)(C(=O)NCC(C)(C)OCCNC(C2CC2F)=O)CC1(F)F 59116,N1(C(c2cn(C)nc2Cl)=O)CC2CC(C1)C(CO)C2NC(c1cccc[n+]1[O-])=O 59117,N1(C(C2C(CC)N(C(=O)C(C)OC(C)(C)C)CCC2)=O)CCn2ncc(C)c2C1 59118,c1(C(CC)CN(C(C)C(=O)O)Cc2nc[nH]n2)ccccc1 59119,CCCC(C)CC(=O)NC1COCCN(c2ncnc(CC)c2F)C1 59120,CC1(NC(C2CCCN(C(N)=O)C2)=O)CCN(C(=O)C(F)C2CC2)C1 59121,N1(C(C(CC)F)=O)CCC(N(C)C(c2ccn(C3CCOCC3)n2)=O)C2(CC2)C1 59122,CC(C)CC(O)C(=O)NC1CN(C(C2C3COCC23)=O)C12CCC2 59123,CC1CC(N=c2c(Br)c[nH]cc2[N+](=O)[O-])CN1C(c1cc2cnccc2[nH]1)=O 59124,C(CC(C)CCNC(c1cc(C(C)(C)C)no1)=O)NC(CCCOCC)=O 59125,c1(C(N(C2CN(C(c3c(O)ccc(F)c3F)=O)C2)C)=O)cc(F)cc2nc[nH]c12 59126,C(=O)(C(CCOCC)NC(=O)C(C)C1CCCC1)N(CC=C)CCOC 59127,CC1(C)CCCC(NC(N2CCC(c3cccc(F)c3)(C(F)(F)F)C2)=O)O1 59128,c1(C(=O)NCC(C)(C2CCC2)NC(CC(C)OC)=O)c(Cl)c2ccccc2n1C 59129,C1(NC(c2cnn(CC(F)(F)F)c2C)=O)CCN(OC(C2C(SC)CCC2)=O)CC1 59130,C(=O)(C(C)CC(F)F)NCCCC1N(C(CCc2cccc(C)n2)=O)CCCC1 59131,c1(C(N2C3C(CNC(c4cocn4)=O)(CCC3)CC2)=O)cccc([N+](=O)[O-])c1Cl 59132,C(=O)(C#CC(C)(C)C)NCCC1(C(=O)NCC2(C)CCN(C)C2)CC1 59133,C(=O)(C(C)(C)CC#N)N1CCC(N(C(=O)CC2C=NN(C)C2=O)CCC)C1 59134,CN1CCN(C(=O)CSCC(=O)OC(C)(C)C)CC1CNC(C1CCOCC1)=O 59135,C1(C2(O)CCOC2)(C(N2CCCC(CNC(=O)COC(F)(F)F)C2)=O)CC1 59136,n1(CC(=O)NCC2CC(NC(=O)C(O)C3CC3)C2)cc(Br)cn1 59137,c1(OC)cc(OC)[nH]c(=NCC2CCCC2NC(=O)C(c2cccc(F)n2)(F)F)n1 59138,Cc1nc(C2CCC2)sc1CC(=O)NCCC1CCN(C(=O)CCC2CC2)C1 59139,C1(C(=O)Nc2cccc(OCF)c2)(OCC(N)=O)CCN(CCCF)CC1 59140,n1(CC2(C)CC2)nc(C2CC2)nc1CC1CSC1 59141,C1(NC(=O)NCc2nc(CC(C)C)on2)CCCC(O)CC1 59142,C1(C(=O)OC)C(C)OCCN1C(c1cnc(CC2CC2)s1)C(=O)NC(C)(C)C 59143,C1(N(C(CCC(=C)C)=O)C)CCCN(C(c2cnc(Cl)c(C3CC3)c2)=O)CC1 59144,CC1(C2CC2)CCCN1C(c1ccnc(CNC(=O)CC2CCC(=O)N2C)c1)=O 59145,C1(N(N2CCC(C=O)C2)CC#C)CCN(C(c2cnn(C)c2C)=O)CC1 59146,C1(CC(=O)NCCOCCCNC(c2c(OC)scc2)=O)CC(O)CC(C)(C)C1 59147,C(=O)(CC(C)(C)CNC(c1ccoc1Cl)=O)NC(c1nccs1)CC 59148,C1(c2ncc(C(=O)OC)s2)CCN(C(=O)N(C)C)CC1.C1CCS1 59149,C(=O)(C(C)C(C)COC)NCC#CC(=O)NCCC#C 59150,N1(C(=O)CCc2cscn2)CC(NC(C23CC(c4ccccc4)C2C3)=O)C(O)C1 59151,c1(C(N(CC(CNC(CSC)=O)O)C)=O)cc(C)cc(Cl)n1.C(C)(C)(C)O 59152,C(c1cc[nH]n1)=CC(=O)NC(C1CCCN1C(=O)C(O)CC1CCCCC1)(C)C 59153,C1(NC(C(CC)(C)OC)=O)CC=C(C(=O)NCC(C)(C)CO)C1 59154,N1(C(CCC=CCC=C)=O)CCN(C(C2(C)CN(C(=O)C(C)CC=CC)C2)=O)CC1 59155,C1(C(=O)NC2(C)CN(C(c3sc(C)c(Br)n3)=O)C2)CNC(=O)C(C)(C)C1 59156,c1(C(CC)O)cn(CCN(C2(c3ccnn3C)CC2)C)nn1 59157,N1(C(C(C)CC(C)(C)C)=O)CCC2CCN(C(=O)Cc3cc[nH]n3)C2C1 59158,C1(C(N2C(C)(C3CC3)CCC2)=O)N(C(c2cc[n+]([O-])cc2)=O)CC12CCCC2 59159,c1(-c2cn(C)nc2)cccc(C(=O)NCC2(O)CN(C(=O)CC3CC3)C2)c1 59160,C(C)(CNC(CC1C(CC)C1)=O)(C(C)C)NC(=O)C(C)CF 59161,c1(C(C(=O)OC(C)C(=O)N(C)Cc2ccc(Cl)cc2)C)ccc2ncccc2c1 59162,c1(CCNC(=NCC)NCC2CC3(C2)CC32CC2)cccc2oc(C)nc12 59163,CC1(C)CCN(C(C23CC2COC32CCC2)=O)CC1CNC(=O)CC1CCC1 59164,C1(C(=O)NC(C(C)C)CO)(CO)CCN(C(c2ccc(C(F)F)o2)=O)C1 59165,c1(C(C)OC)ncc(C(=O)N(CCCCN(C(=O)CCCC2CCCO2)C)C)s1 59166,C(=O)(C1=CCCN(C(=O)Cc2cc(C)cs2)C1)NCCCCC#CC 59167,Cc1[nH]c(C#N)cc1C(=O)NC1CCCCN(C(=O)CC2CC3CCC2CC3)C1 59168,CCCCC(C)C(=O)NCC1CN(C(C)C(=O)NCc2ccn(C)c(=N)c2)C1 59169,CCCCC(C(=O)NCCN1CC(CF)C1)NC(C1CCOC(C)(C)C1)=O 59170,C12(NC(c3cnc(C4CC4)o3)=O)CCCC1N(C(c1ncccn1)=O)CCC2 59171,C1(C(=O)NCC2C(CC)C2)CCCCC1(C)NC(=O)Cc1cncnc1 59172,N1(C(c2n[nH]c(C)c2C)=O)CC2CCC1CN2C(C1(C)CCCNC1=O)=O 59173,c1(C(=O)NCCC(C)(C)NC(=O)COC(F)F)ccnc(SC(F)(F)F)c1 59174,c1(C(=O)NC2CCN(C(C(C)(C)OC(C)=O)=O)CC2F)coc2c(F)cccc12 59175,Cc1ccc2c(c1)NC(=O)C2CC(=O)N1CCNC(=O)C1C 59176,CC(C)CCCC(=O)N1CCC(C=CC(=O)NC(CO)CC(C)C)CC1 59177,C1(COC)CN(Cc2ccc(OC(F)F)cc2)CCN1c1ccncc1 59178,c1(OC)cc(Cl)ncc1C(N1CCN(C(c2oncc2C)=O)CC1C(C)C)=O 59179,n1(CCC)nccc1C(=O)NCC(c1ccccc1)NC(C12CSCC1C2)=O 59180,C1(NC(c2cc(CO)[nH]n2)=O)CCN(C(c2ccccn2)=O)C12CCCC2 59181,C(C(C)CCCC(C)C)NC(C1CCCN(C(c2cccc(C#C)c2)=O)C1)=O 59182,c1(C(N2C(CC)CC(C)CC2)=O)cnc2c(Br)c[nH]c2c1 59183,N1(C(C=CC2N(C)CCC2)=O)CCC(NC(=O)Cn2cc[n+](C)c2)C2(CCC2)C1 59184,C1(C(=O)NC2(C)C(C)OCC2)C2CC3C(C2NC(=O)CN2CCC(F)CC2)C13 59185,c1(OC)cc(C(N2CCC(C3CCCN3C(=O)CCF)C2)=O)ccc1O 59186,C(=O)(C(CCC(C)C)NC(=O)CN1CCCCC1C)NC1CN(C(CC)=O)C1 59187,C(CN(C(C(=O)NC1COC1)c1cnsc1)C(C)=O)(CO)(CO)OC 59188,Cc1cc(-c2cn(CCNC(c3ncccc3CO)=O)nn2)cc(F)c1 59189,Cc1nc(Cl)[nH]c(=NC2CN(C(=O)CSc3ccco3)CC23CCCCC3)c1F 59190,C(=O)(C(=O)C(C)(C)C)NC1(CNC(c2n[nH]c(C)c2C)=O)CCCCC1 59191,N1(C(Cc2nc(C)[nH]n2)=O)CCCN(CCNC(C2CCCNC2=O)=O)CC1 59192,c1(C(=O)NC2CC(N(C(c3sc(C)c(Br)c3)=O)C)C2)cccc(F)c1N 59193,CN=c1[nH]nc(CC(=O)NCCN(C)C(C2(CC(C)C)CCCC2)=O)s1 59194,C1(N(C(=O)CC2(CO)CC2)CC)CCCN(C(=O)C=Cc2ccncc2)CC1 59195,N1(CCNC(C(=O)N(CC(=O)Nc2n(CCC)ncc2)C)=O)CCN(C)CC1 59196,c1(CC(CNC(C2CN(C(C)=O)C2)=O)C(N(C)Cc2cnc[nH]2)=O)ccccc1 59197,c1(NC(C)Cc2ccco2)[nH]c(=NCc2cccc(F)c2Cl)nc2c1cnn2C 59198,c1(CCC(=O)NC(C)CCNC(=O)CCC2(C)N=N2)ccc2c(c1)NC(=O)CO2 59199,Cc1cc(C(=O)NC(CNC(c2c(C3CCC3)cnn2C)=O)CO)cc(F)c1 59200,C1(C(=O)NCCOCCNC(Cc2c(C)ccnc2)=O)C2CCN(CC2)S1(=O)=O 59201,C1(S(=O)(=O)N2CCCC(N3CCCCCC3=O)C2)(CC(=O)O)CCC1 59202,CCC(C)(C)C(O)C(=O)NC1(CNC(=O)CC2(CO)CC2)CCCCC1 59203,C(CN=C(NCC(F)F)NCC1(C)CC1Br)c1nc(CC)c(C)s1 59204,CC1(F)CC(C(=O)NCC(CNC(=O)CSS(C)(=O)=O)CO)C1 59205,N1(C(C2CC(C)(CC)C2)=O)CC2(CCN2C(c2ccc(Cl)cc2OC(C)C)=O)C1 59206,C1(C(=O)NCC(O)CC)CC(C)(C)CCO1.C1(CCC)CN2CC1C2=O 59207,c1(C(N2CCC(N(C(CN(C)CC)=O)CCO)C2)=O)ccc(C(C)(C)C)cc1C 59208,N1(C(c2ccc(Cl)cc2)=O)CCC2C(C1)OCCN2C(c1ccoc1)=O 59209,C(=O)(CCC(=O)N1CC(CNC(=O)C=Cc2cccs2)C(O)C1)N(C(C)C)C 59210,C(=O)(C(C)C(F)(F)C(F)F)N1C(CNC(c2c(CC)n(C)nc2)=O)CC(F)C1 59211,C1(C(N2C(CCNC(C(C)(C)CO)=O)CCC2)=O)Cc2ccc(Cl)cc2C(=O)O1 59212,c1(NC(c2nnnn2C2CCC2)C2(C(=O)OCC)CC2)ccc(Br)c(Cl)c1 59213,CC1(C(=O)NCC2(CNC(C3SCCS3)=O)CCCC2)CCC(O)CC1 59214,Cn1cnc2c1CCN(C(=O)C(F)C(F)(F)F)C21CCN(C(=O)CC2(C)CC2)C1 59215,c1(C(=O)NC2(C3CCCN3C(=O)C(F)=C3CCCC3)CC2)cc(C(N)=O)c[nH]1 59216,C1(C(=O)NCCCC2CCC3(C(C=C)C3)C(=O)N2)CCOC2(CCCCC2)C1 59217,Cc1[nH]nc2cc(NC(c3cccc4c3OCCO4)=O)ccc12 59218,C12(CC(=O)NC(CC=C)CNC(=O)C=Cc3cncs3)CCC(C(F)(F)F)(CO1)C2 59219,C1(C(=O)NCC2(C(C)(C)C)CCN(C(Cc3c(C)ccs3)=O)C2)CCC2(CCC2)C1 59220,C1(CC(=O)N(CC(CC)O)C)CCN(C(=O)COCC2CC2)CC1 59221,c1(CC)cn2ccc(C(=O)OCCc3ccc(C(C)C)cc3)cc2n1 59222,c1(C(N2CCC(CN(C(CCC=CC)=O)C)C2)=O)csc(Br)c1C 59223,c1(C(=O)NC2CCCCN(C(C(CC)(C)CC)=O)C2)cccc(F)c1C#N 59224,C=CCCCC(C(=O)NCCCC(=C)Cl)NC(=O)C(C)OCC 59225,c1(COC)ccc(C(=O)NC2CCCC(C(N3CCSCC3)=O)C2)cc1 59226,C1(C)(C(N2CC(CN(C(C(CC)(C)C)=O)C)OCC2)=O)CC(=O)N(C)C1 59227,CN1CCC(CC(N2CC(C(=O)NC3CCN(c4ccccc4)C3=O)C2)=O)C1=O 59228,C1(OC)CN(C(=O)CC2CN(C(c3c(O)cccc3Cl)=O)CCO2)CC(=O)N1 59229,N1(C(Cc2ccc(C)o2)=O)CCC(CNC(=O)Cc2nc(Cl)cs2)C(O)C1 59230,CC1(C)CN(C(C2CC(O)C(F)C2)=O)CCC1C(=O)NCCC1CCCCCC1 59231,C(=O)(C(CO)C(F)(F)F)N1C(C(=O)NCc2n(CCC)cnc2)CCOCC1 59232,C=CC(C)(C)CC(=O)NC1CC(F)(F)CC1NC(=O)Cc1cccc(F)c1F 59233,C1(NC(c2onc(C)n2)C(C)C)CNCC(P(C)(C)=O)C1 59234,C1(NC2CCC(CNC(c3cccc(NC(C)=O)c3)=O)CC2)CC12CC(C)(C)C2 59235,C(C(CNC(c1cncc(N)n1)=O)C(F)(F)F)NC(c1c(C)ccs1)=O 59236,c1(CN2CCC(NC(c3ccc(C)cc3Cl)=O)C2)cc(Br)cc2c1OCC2 59237,c1(CC(=O)NC(C2CCN(C(C3CCC3(C)C)=O)C2)C)coc2ccccc12 59238,Cc1nn(CCO)cc1C(=O)N(C)CC1CCCN1C(c1ccccn1)=O 59239,CCC(C)C(C)C(=O)N1CC=CC(NC(=O)CN2C(=O)CNC2=O)C1 59240,CC1CN(C(C2CC2c2ccnn2C)=O)CC1NC(c1cnsn1)=O 59241,Cc1cc(CCC(=O)NCCC2CN(C(=O)CN3C(C)CCC3C)C2)cc(C)n1 59242,C12(C(N(C3CCCCC3)CCNC(c3c(C)noc3)=O)=O)CSCC1C2(F)F 59243,CC1CN2CCN1C(C(N1CC(F)(CNC(=O)Cc3ccc(N)cc3)C1)=O)C2 59244,O=C1NC(=O)c2c(C(=O)NC3CC(NC(=O)CC4CCC5CC45)C3)cccc21 59245,C1(CC=C)(C(=O)NC(COCC)CC)C=CCN1C(=O)CCn1ccnc1C 59246,CC1(C)CN(C(=O)CC(CNC(C2(C)CC3CC3C2)=O)C2CCC2)CCCO1 59247,C1(C(=O)NCC(C)N(C(c2c(OC)nn(C)c2)=O)C)CCc2ccc(F)cc2O1 59248,C1(C(N(CC(C)(C)NC(C(n2ncc(C)c2)C)=O)C)=O)C2(CC2)C12CC2 59249,Cc1cc(S(N)(=O)=O)cc(-c2noc(C3C(C)N(C)CCN3C)n2)c1C 59250,C(=O)(CCC(F)(F)F)N(C)CC1CCCN1C(C1CC(CC(F)F)C1)=O 59251,C12(C(=O)NCC3CCC(C)N(C(c4ccc(CO)o4)=O)C3)CC=CCN1CCC2 59252,N1(CC(=O)N(C)CC2(CNC(C(C)OCCC=C)=O)CC2)CCCNS1(=O)=O 59253,Cn1nc([N+](=O)[O-])cc1C(=O)NCC(O)CNC(c1ccc(F)c2ccsc12)=O 59254,c1(C(=O)NCCN(C(=O)CCc2ncc(C(C)(C)C)o2)CC)cc(SC)oc1C 59255,C(C)(CCC(=O)Nc1ccc(C(=O)NOCC(=O)N(C)C)o1)OC 59256,c1(OC)nccc(N(CC(C)NC(=O)Cc2ccns2)C)n1 59257,c1(C(=O)NC2CCCCCN(C(CC(C=C)C)=O)C2)cc(F)c(Cl)c(N)c1Cl 59258,CCC(C)CC(C)C(=O)N(C)CC1CCCN1C(c1ccccc1Cl)=O 59259,C1(NC(c2cc(C#N)[nH]c2)=O)CC2CCC1C(NC(=O)C=CC1CCC1)C2 59260,C12(C(=O)NC3C(NC(c4cc(C)n(C5CC5)n4)=O)C3)CCC(C)(C(=O)O1)C2(C)C 59261,C1(C(=O)NCC2(CCN=[N+]=[N-])CC2)CC2(CCC2)CN1Cc1cccc(C)c1 59262,c1(C(=O)NCCCN(C(=O)CCC2CCCO2)C)ccc2c(Cl)nccc2c1 59263,C=CC(C)(C)C(=O)NC(C1CCCN1C(=O)C=C(C)C(C)C)C 59264,N1(C(=O)CC2CC(F)CN2C(=O)Cc2nc(Cl)cs2)Cc2cccc(F)c2C1 59265,c1(SC)ccc(C(N2CCOCC2C2CC2)C(=O)NCC2CCCO2)cc1F 59266,C(=O)(CCCCCNC(C)=O)NCC(CC)N(C)C(C1CCC1OC)=O 59267,c1(C(N2CCC(NC(CC(CC)O)=O)CC2C)=O)c(C)nn2cccnc12 59268,N1(C(C2(c3ccccc3)CCC2)=O)CCC2CCC(C1)N2c1cnc(F)cn1 59269,c1(COC)nc(C)c(C(=O)NC(C)(CNC(C2SCCCS2)=O)C(C)C)s1 59270,C1(C)(c2cn(CC(=O)OCC)nn2)COCCN1C(C1CC(=O)CO1)=O 59271,N1(C(c2cnsn2)=O)CCC2(CCCN2C(c2ccn(CC(F)F)n2)=O)CC1 59272,N1(C(c2cc(OC)cc(F)c2)C(=O)NCC(F)F)CC2CCCCCC2(C#N)C1 59273,c1(C(N2CCCC(N(C(C3C(CCC)C3)=O)C)C2)=O)ccc(=O)n2c1CCCC2 59274,C(=O)(CS(C)(=O)=O)N(CCC(C)NC(=O)COc1ccsc1Cl)C 59275,Cc1cc2scc(C(=O)OCC(C3Cc4ccccc4N3)=O)c2s1 59276,Cc1cn2cc(CC(N3CCC(C)(CNC(=O)C(C)C)C3)=O)nc2s1 59277,C(N=c1[nH]nc(O)s1)C1CCN(C(CCCc2onc(C)n2)=O)C1 59278,N1(C(c2c(CCC)nns2)=O)CCCC(C)C1CCNC(c1ccnc(S)c1)=O 59279,N1(C(C(N)c2ccco2)=O)CC2COCC2(C(N2CC(O)C(F)C2)=O)C1 59280,C(CCN=C(NCC(c1ccc(Cl)cc1F)O)NC1CCC(=O)NC1)SC 59281,N1(C(C23CCC(OC)C2C3)=O)CCCN(CCNC(=O)CC(=O)N(C)C)CC1 59282,c1(CC)cc(C(=O)NC2(CO)CN(C(c3c(C#N)cnn3C)=O)C2)cc(C)c1 59283,c1(C(N2CCCC(O)(CNC(C3C=CC=CC=C3)=O)C2)=O)ccc2nncn2c1 59284,C1(N(C)C(c2cn(C)nc2O)=O)CC2CCC(C1)N2C(=O)CN1CCCNC1=O 59285,N12CC3CCC(C1)N3C(=O)c1cccc(c1)C2.c1(C(=O)OC)cccc(CO)c1 59286,C1(CNC(C2N(C(C(c3cnn(C)c3)C)=O)CC2)=O)CC2(CC2)CO1 59287,c1(OCCN(C(C2CC3CCC2C3)=O)Cc2ccccc2)cccc(Cl)n1 59288,c1(C(N2CC3C(CNC(c4[nH]cc(C)c4)=O)(C3)C2)=O)ccsc1S(N)(=O)=O 59289,c1(C(N(CCCNC(c2n[nH]c(C)c2CC)=O)CCC)=O)occ2c1CCCC2 59290,N1(C(C2CCCCC(=O)N2)=O)CC2(NC(=O)C3CC3)CCCC2(F)C1 59291,N1(C(COC(c2cccc(F)c2)C)=O)CCCN(C(C2CC2(C)C)=O)C(C)C1 59292,Cc1nc2ncccc2cc1CC(=O)Nc1cn(C)nc1C(N)=O 59293,c1(OCC)cc(OC)c(NC(c2cc(C(=O)O)c(C(C)(C)C)o2)=O)cc1Cl 59294,c1(CC(=O)NCC(CNC(c2cccc[n+]2[O-])=O)OC)nnc(S)n1C 59295,c1(C(N2CCCC(CNC(c3cccc(C)c3I)=O)C2)=O)cnc2snnc2c1 59296,c1(CNCC2N(C(C3CCCC(C)(C)O3)=O)CC=C2)ccc2nnnn2c1 59297,N1(C(C(C)(C)OC)=O)CCC(C)(CCNC(C2(CC(C)C)COC2)=O)C1 59298,C(=O)(CCCCCNC(=O)NCC1CC1)NC(C)CCNC(C1CCC(=O)N1)=O 59299,CC1CC(=O)NC1C(N1CC(OCCNC(c2conc2C2CC2)=O)C1)=O 59300,c1(C(CNC(N2CC(CS(N)(=O)=O)C2)=O)O)ccc(Br)cc1 59301,C(CC(=O)N1CCC(CC(C)C)C1)(C(F)(F)F)NC(c1ccnc(OC)n1)=O 59302,Cc1nc(C)n(CC(=O)NC(c2ccc(F)cc2)CNC(=O)C=CC=C(Cl)Cl)n1 59303,c1(OC)ccccc1OCC(=O)N(c1ccccn1)CC1(CN)CC1.c1(C)nncs1 59304,c1(C(=O)NC(C=CC(=O)NCC2N(CC)CCC2)C)cc2ccccn2n1 59305,c1(CC)cc(C(=O)N(CCCCC(=O)NC2CC(=O)NC2=O)C)ccn1 59306,N1(C(C(CNC(CC(CC)(C)C)=O)O)=O)CCN2CC(C)CC2C1 59307,N1(C(C2(C)C(C)OCC2)=O)CCC(NC(=O)Cc2nn(C)cc2Br)C(F)C1 59308,CCCCC(C(=O)N1CC(OCCNC(=O)CCNC(=O)C=CCl)C1)N(C)C 59309,c1(C(C)=O)cc(CCC(N2CCC(N(C)C(C3CC3C)=O)CC2)=O)oc1C 59310,CC1=NOC(C)(CNc2cc(N3CCC(C(F)(F)F)(CO)C3)ncn2)C1 59311,C(=O)(CCCN=[N+]=[N-])NC1CCC(C(=O)OCC)C1.C12CCC1C(=O)N2 59312,Cc1ccc(C)c(C(N2CC(OC)CC2CNC(C2CCC(=O)N2)=O)=O)n1 59313,c1(C(CC)=O)ccc(N2CCC(NC(c3nccc(Cl)c3O)=O)C2)c([N+](=O)[O-])c1 59314,C(=O)(CCCCC1CC1)N(C1CCN(C(=O)CCC2C(=O)NN=C2C)CC1)CC 59315,C1(CC(=O)NC(C)CN(C)C(C2CCCN2c2cnccn2)=O)CCCC12CC2 59316,c1(C(N2CCC(OC)(CNC(=O)C=C3CC3)C2)=O)ccc(F)c(F)c1N 59317,C(=O)(C#CC1CCCC1)N(CC(CC)NC(C1CN(C2CCOCC2)C1)=O)C 59318,c1(OC(C)(C)C)ccc(CNC(=O)NC2CC(F)(CC3CCC(F)C3)C2)cc1 59319,CC1(C)CCCC(C(=O)NC2CCN(CCCNC(=O)Cc3ccon3)C2)C1 59320,c1(NC(CC2(COC)CC2)=O)ccc(C)cc1F.c12coc(c1)C(=O)N2 59321,C(=O)(C1OCCn2ccnc21)NCC(CNC(c1c(NC)ccc(F)c1)=O)CO 59322,C=C(Cl)CN=C(NC1CCOCC1)NC1CCC1(C)C 59323,CC1ON=C(C(=O)N2CCN(C(=O)COC(F)F)CC2CC2CC2)C1C 59324,CCCCCC(C)CC(=O)NC(C)(C)C(C)NC(=O)CC(C)(C)CN(C)C 59325,CC1CN(C)CCC1NC(=O)CC1(C)CCN1C(=O)C(F)F 59326,C1(NC(c2n(CC)nnn2)c2csc(-c3ncccn3)n2)CCOCC1(C)C 59327,N1(CC)N=C(C(=O)NCC2CC(O)(CNC(c3cnc(SC)s3)=O)C2)CCC1=O 59328,Cc1ccc(C(=O)NCC2C(C)CCN2C(=O)CCc2ccnc(Cl)c2)n1C 59329,N1(C(c2cnc(CC)[nH]2)=O)CC(C2CCN(C(=O)CCCNC(C)=O)C2)C1 59330,c1(C(N(CCNC(=O)C(=O)NCCC(C)C)CC)=O)c(F)ccc(OCC)c1F 59331,Cc1ccc(O)cc1-c1nc(NC(c2ccc(O)c(Br)c2)=O)cs1 59332,Cc1nc2cccc(C(=O)NC(C)CCCNC(c3nccc(N)c3Cl)=O)c2s1 59333,C1(NC(c2ccc(Cl)nc2)=O)CC=CCC1C(N1CCC(O)(C(=O)O)C1)=O 59334,c1(COC)occc1C(=O)NCC(C1CC1)N(C)C(C1CC=CCC1)=O 59335,C(=O)(C1OCCc2c(O)cccc21)NC(C(C)(C)C)CNC(c1ccc(Cl)s1)=O 59336,C1(CNC(c2c(C(N)=O)coc2)=O)CN(C(c2ccc([N+](=O)[O-])o2)=O)CC1(C)C 59337,CCCC(C(=O)NCc1cccc(CNC(C2(C)C=CCC2)=O)c1)OCC 59338,c1(C(C)C)ccc(C(N2CCCC2CN(C)C(C2CNC(=O)N2)=O)=O)s1 59339,Cc1cc(Cl)c(C(N2CCC(c3cn(Cc4cccc(Cl)n4)nn3)C2)=O)s1 59340,C(C)(C(CC(=O)NCC1CC2C(C1)C2(F)F)NC(=O)CSC(C)(C)C)OC 59341,C1(C)(C(=O)OCC)C=CCN1C(=O)CC1CCCN(C(=O)CSC(C)C)C1 59342,N1(C(CN2CC(CC)C2)=O)CCCC2(CCN(C(c3cc(CO)cs3)=O)C2)C1 59343,c1(OC)ncc(NC(c2ccc(OC)c(C3CC3)c2)=O)c(C)n1 59344,c1(CCC(N2CC3C(CNC(=O)C=CI)C3C2)=O)cc2ccccc2o1 59345,C1(CNC(Cc2c(C(C)(C)C)con2)=O)(COC)CCN(C(C2CC=CC2)=O)C1 59346,CCCC(F)(F)C(=O)N(CC(O)CNC(=O)C(C(C)C)NC(C)=O)C 59347,c1(C(N2CC(CNC(CCc3cc(OC)no3)=O)C2)=O)cnccc1NC(C)C 59348,C(CCC(=O)N(CC(C)NC(c1cnc(CC2CC2)s1)=O)C)N(C(C)=O)C 59349,CC1CC(C(=O)NCC2(C)CCOCC2)CN(C(=O)COCCCN(C)C)C1 59350,C(=O)(C1=CC2C=CC(C1)C2)NC(CC(C)NC(c1c(OC)c(C)sc1)=O)C 59351,N1(C(c2n(C)c(C#N)cc2)=O)CCCC2(C1)CN(C(=O)CSc1n[nH]c(O)n1)C2 59352,CCCC(C)(O)C(=O)NC1CCC(CNC(C2CC(=O)N(C(C)C)C2)=O)CC1 59353,c1(N2C(COC(C)=O)CCC2)cc(C(C)C)nc2ncnn12 59354,C=CC1CN(C(C2CN(C(c3cnn(C)c3OC)=O)CC23CC3)=O)CCO1 59355,C(C)(C(C)C)(c1nnnn1C(c1ccccc1)C)NC(C)CCOC(C)C 59356,c1(C(N2CCOCC2CC2CCCC2)C(=O)NC(CC)C)ccc(N(C)C)nc1 59357,c1(C(=O)NC2C3CN(C(c4ccc(Cl)cc4Cl)=O)CC23)ccc(Cl)c2[nH]ccc12 59358,C=CC(C)CC(=O)N1CC(CO)(NC(=O)CSCc2c(C)noc2C)C1 59359,N1(CC(=O)NCC2CCN(C(c3cn(CCC)nn3)=O)C2)CCN(C)CC1 59360,c1(N(C)C)ccc(C(=O)NCC2CN(C(C3(CO)CCC3)=O)CCO2)cn1 59361,C(=O)(C1=CCCOC1)NC(CNC(C1(CC#C)CC=CCC1)=O)CO 59362,c1(C(C)=O)cc(C)c(C(=O)NCCCCCNC(=O)C(=O)Nc2ccccc2)o1 59363,c1(NS(CCOCC)(=O)=O)ccccc1NC(=O)NC(C)C(C)CC 59364,c1(C(N2CCCC(NC(C3(NC(C)=O)CCCC3)=O)C2)=O)cccc2c1COC2 59365,Nc1ccc(C(=O)NC2CCCC2NC(c2ncoc2C(F)(F)F)=O)cc1Cl 59366,N1(C(c2cccc(CCC)c2)=O)CC2(CC(NC(C3CCC(=O)N3)=O)CO2)C1 59367,c1(C(=O)NC2CC(CC)(CC)N(C(=O)C3=NOC(C)C3)C2)c(C)ccc(C)c1O 59368,N1(C(C2CSCCS2)=O)CCOC(C(N2CCC(c3nc[nH]n3)C2)=O)C1 59369,c1(C(=O)NCC(C2CC2)NC(CCc2c(C)noc2Cl)=O)cnc2c(c1)OCCN2 59370,Cc1cnc(CCNC(=O)C(COC)NC(=O)CC(=O)NC2CC2)o1.C(C)C 59371,C1(CNC(c2c(OCCOC)cc(C)cc2)=O)C2CCCC1N(c1nncs1)C2 59372,N1(C(C(CCC)N(C)C)=O)CCC2(C1)CN(C(C1CC1(C)C)=O)C2 59373,N1(C(CCC2(C)CN(C(CNC(C3C(C)C3)=O)=O)C2)=O)CC2CC(O)CC1C2 59374,C1(C(N2C(C(=O)NC)CC(O)C2)=O)CN(C(=O)CC2C=CCCC2)CCC1(C)C 59375,O=C1NCc2c1ccnc2C(N1CC(NC(c2cccc(F)c2)=O)CC1CO)=O 59376,C1(C(N2C(C)(C(=O)NCCC3CCN(C)C3)C=CC2)=O)CCCC(C#N)C1 59377,C(C(C)(C)CC(=O)NC1CN(C)CC1C)NC(C1(CC)CCC1)=O 59378,c1(CC(=O)N(C(C)=O)CCN(C2CCCC2C)C2CCC2)cccc(Br)c1 59379,Cc1cccc(NC(C2CCN(C(=O)CCc3cc(F)ccc3Br)C2)=O)c1O 59380,C1(C)(CNC(CSc2n(C)cnn2)=O)CCC(NC(c2cc(CCO)on2)=O)C1 59381,N1(C(C2(CNC(C3COCC3(C)C)=O)CC(=C)C2)=O)CCC(OCC)(CO)C1 59382,N1(C(CCc2cc(OC)no2)=O)CC2CCN(C(C3CS(=O)(=O)C3)=O)C2C1 59383,c1(C(=O)NC2C(NC(CCC=C)=O)CCC2)nc2ncccn2n1 59384,C1(C(=O)NCC2CCC3(CC3)C2)(COC)C=CCN1C(=O)CC1CCCCC1 59385,c1(C(N)=O)cccc(C(N2CCC(CO)(NC(C3CCNC3=O)=O)C2)=O)n1 59386,Cc1sc2ncc(C(=O)NC3CC3CNC(c3ncoc3C(C)(C)C)=O)n2c1C 59387,Cc1cc(C(=O)N(C)CC2C3CN(C(=O)CSCC(C)C)CC23)cc2nc[nH]c12 59388,c1(CN(C(C2CC(C(C)NC(C(C)NC(N)=O)=O)C2)=O)C)ncc(C)o1 59389,n1(C(C)C)cc(C(=O)NCCC2CCN(C(=O)CCN3CCC3)C2)c(Br)n1 59390,C=CCC(C)(C)CC(=O)NCc1cncc(C(=O)NCC(N2CCC(O)CC2)=O)c1 59391,C1(C(=O)NCC(C)(C)CNC(=O)C(c2ccc(Cl)s2)=O)CC2(CC2)CO1 59392,Cc1ccc(F)c(O)c1C(=O)NCC1(CNC(C2OC(C)(C)OC2(C)C)=O)CC1 59393,C1(C(N2CCOCC2CCO)=O)(CNC(C(C)OCC=C)=O)CC12CCC2 59394,c1(C(N2CCN(CC(=O)NCC3N(CC)CCC3)CC2)=O)cc(F)cnc1O 59395,c1(C(=O)NC2CC(CCNC(C(C)OCCCC)=O)C2)cn(C)nc1C(C)(F)F 59396,CC(C)C(C(=O)N(C)Cc1ccon1)NC(c1cccnc1)=O 59397,c1(C(C)NC(=O)CCc2cncs2)ccc(CNC(c2c(C)ccn2C)=O)cc1 59398,c1(OC)cccc2sc(C(=O)NCC(O)CNC(=O)CCc3cccs3)cc12 59399,c1(C(=O)NC2C(NC(C)=O)COC2)cnn(C)c1Cl.c12ccc(s1)C2=O 59400,C1(NC(C(c2cncnc2)C(=O)NCCC(=C)CSC)=O)CCC(C(N)=O)CC1 59401,C(=O)(N=c1nc2cccc(F)n2[nH]1)C1(Cc2cn(C)nc2C(F)(F)F)CCC1 59402,C1(COC)C=CCCN1C(=O)CC(O)CNC(c1ccncc1N)=O 59403,c1(OC(C2C=CC(C(N(C)C)=O)C2)=O)cc([N+](=O)[O-])c(C#N)cc1Br 59404,C1(NC(COCCC#C)=O)(CO)CCN(C(=O)CCC2CCCCN2C)C1 59405,c1(C(=O)OC)c[nH]c(=NCCCN(C)C(C2CCc3cncn3C2)=O)s1 59406,CC1(C#CC(=O)NCC2(C(=O)O)CC(C)(c3cn(C4COCC4F)nn3)C2)COC1 59407,C1(C)(C(=O)NCC(CC(C)C)NC(CCC(=C)Cl)=O)CCCC1(F)F 59408,c1(C(=O)NCC2(F)CCCN(C(CCC)=O)C2)cnc2scc(Br)c2c1 59409,c1(OC)cc(C(=O)Nc2cc(C)cc(C)c2Br)c(N)cc1Cl 59410,c1(C(=O)NC2C(NC(C(C)CN3CCCCC3=O)=O)CCC2)cccc(F)c1N 59411,C(CC(=O)N1CC(C2(NC(c3cc(SC)c(CC)o3)=O)CC2)C1)(C(F)(F)F)OC 59412,C1(NC(=O)COc2ccnn2Cc2ccc(Cl)cc2)COc2ccccc2C1 59413,N1(C(C(C2CCOC2)NC(C2C3CC(=O)CC32)=O)=O)CC2(CCNC2=O)C1 59414,c1(C(N(CCNC(C2C(C)C2C)=O)CC)=O)cnn(CC(C)C)c1O 59415,C=CC(C)CC(=O)N(C)CC1CN(C(=O)CCc2cncnc2)C1 59416,C1(C(=O)NCC2(C(C)(C)O)CN(C(COCC(=O)OC)=O)C2)CCc2ccnn2C1 59417,c1(C(=O)NCCOCCN(C(=O)Cc2csnn2)C)cccc2c1OCC2 59418,N1(Cc2c(F)cc(C#N)c(F)c2)CCC(N)c2cc(Cl)ccc21 59419,c1(C(N(C2C3CN(C(=O)CC4CCCS4(=O)=O)CC23)C)=O)cncn(C)c1=O 59420,c1(C(=O)NCCCN(C(CSCC=C)=O)C(C)C)ccc(Cl)c(OC)c1 59421,Cc1ccc(C(=O)NC2(CNC(C3(C)CC3)=O)CCC(C)(C)CC2)cc1[N+](=O)[O-] 59422,c1(C(N2CCC(NC(CCCN(C)C)=O)C2C(C)(C)C)=O)nccc2cc[nH]c12 59423,C(CC(=O)NC(C(C)C)C1CC1)(C(F)F)NC(c1cc(OC)ncc1)=O 59424,N1(C(C2(C)CCCN2C(c2ccn(C3CC3)n2)=O)=O)CCCCCCCC1 59425,Cc1nc2ccc(C(=O)Nc3cccc(Cl)c3C(N)=O)cc2o1 59426,Cc1n[nH]c(C)c1CC(C)C(=O)NC(C)CC(C)NC(=O)C(c1ccccc1)F 59427,C(=O)(C(CNC(=O)CC(C)(F)F)CC1CC1)NCc1ccc(CC)o1 59428,C1(CCNC(c2ccc(CC3CC3)s2)=O)CCCCN1C(C1(O)CCC1)=O 59429,c1(C(N(CCCCOCC2CC2)C)=O)c[nH]ccc1=O.Cc1cc(C(=O)N)co1 59430,CCCC(F)C(=O)NCCC1(NC(=O)CCCC2CC2C)CCC1 59431,CC(C)(C)C(=O)C(=O)N1CCN(C(c2sccc2C(F)F)=O)CC1CF 59432,CON1CCC(CC(=O)NC2CC(F)(CNC(C3CCN3S(C)(=O)=O)=O)C2)CC1 59433,C1(NC(c2nccc(OC)c2)=O)CCCC12CN(c1nccc(C(C)(C)C)n1)C2 59434,C1(NC(=O)Cc2cnccn2)(CO)CCN(C(=O)CSc2ccccc2Cl)C1 59435,C1(C(N2CC(NC(N)=O)C2)=O)CCCCCN1C(C1CC=CC1)=O 59436,C1(CCCC)CCC(N=c2[nH]c(N3CCOC(C4(C)CC4)C3)nc(=N)[nH]2)C1 59437,CC(C)(C)C#CC(=O)N1CCN(C(=O)CC2CCCCC2)C(CS(C)(=O)=O)C1 59438,C1(OC)CN(C(c2ccccc2OC)=O)CC1C(=O)NC1(c2cnccn2)CC1 59439,C(CCC(=O)NC(CN(C)C)C(=O)N(C1CCC1(C)C)C)OCCOC 59440,C1(C(=O)NCC2(CO)C(C=C)C2)CC(F)CCN1C(=O)CCCCCOC 59441,CCC(C)C(O)C(=O)NC1(CNC(c2cc(-n3ccnc3)ccn2)=O)CC1 59442,C(CC(C(C)(C)C)NC(=O)Cn1nnnc1C)N(C(c1c(C)nccc1)=O)C 59443,CCC(CC)(CCNC(=O)C(C)Cn1ccnc1)NC(c1cc(F)n(C)n1)=O 59444,Cc1c(Cl)c(C(N2CCC(C)(NC(C3(C4CCCCO4)CC3)=O)C2)=O)nn1C 59445,N1(C(C(COC)NC(=O)C(C(C)C)NC(C)=O)=O)CCCC2(C=CCO2)C1 59446,C12(NC(CSCC(=O)OC)=O)CC1CN(C(=O)C(c1cnn(C)c1)C)C2 59447,C1(C(N2CC(O)(CNC(C3(C(=O)N(C)C)CCCC3)=O)C2)=O)(CC)CC1(F)F 59448,CC(C)(C)CC(N)CCNC(c1nnnn1CCCF)C(N)=O 59449,N1(C(COCCCCC)=O)CCCC1CN(C(C1CCC1CF)=O)C1CC1 59450,N1(C(Cc2n(C)nnc2)=O)CC2(C(=O)NC3CC(CO)C34CCC4)CCC1CC2 59451,c1(C(=O)NCCN(CCC)C(C2CCCO2)=O)cnc(C(F)(F)F)s1 59452,c1(OC)nccc(C(N2CC=CCC2C(=O)NCC2C(C)C2(F)F)=O)n1 59453,CC1(F)CCN(C(C2CC(O)CN2C(=O)CN2CCCNC2=O)=O)C1 59454,CC(C)CC(C(=O)N1CC2CC(NC(C3CCCS3)=O)CC2C1)C(N)=O 59455,c1(SC)c(C(N2CCN(C(=O)C(C)(C)F)CC2C2CC2)=O)cccc1F 59456,N1(C(C2CN(C(C(C(C)(C)C)OC)=O)CC2C2CC2)=O)CCC2(CCCO2)C1 59457,C1(C(=O)NCCCNC(=O)CNC(C2CCOCC2)=O)CN=C2N=CNN2C1 59458,c1(C(=O)NCCCN(C)C(C2CCCCN(C)C2)=O)ccc2c(c1)C=CS2(=O)=O 59459,C1(CNC(c2n(C(CC)C)ncc2)=O)CCCN(C(=O)C(C)(C)CC)C1 59460,C1(C)(CNC(c2ccc(CC)s2)=O)CCC(NC(=O)CCn2ccnc2)CC1 59461,C(=O)(C(F)C(F)(F)C(F)(F)F)NCC1C(C(=O)NC2CC(C)(C)C(=O)NC2)C1 59462,C(CCCCC(=O)NC(C)C(C)(C)CC1CC1)N(C(C(C)(C)SC)=O)C 59463,n1(C(C)C)cnc2c(NCC(=O)NC3CC3)[nH]c(=NCC3CCOC3C)nc12 59464,C(C)(C(=O)NC1CN(C(C2CC(n3cnnc3)C2)=O)C1)(C(C)C)NC(C)=O 59465,C1(Cl)(C(=O)NC2(CNC(=O)COCc3nc[nH]n3)CCC2)CC12CCC2 59466,c1(C(=O)NCC(CC)NC(=O)COCC2CCCC2)cc(C(F)F)ncn1 59467,c1(C(=O)NC2(CNC(C=C(C)C(F)F)=O)CCC2)ccc2nc(S)oc2c1 59468,C(CNC(=O)CC1(N(C)C)CC1)(C(C)(C)C)NC(C(C=C)C)=O 59469,c1(C(C(=O)NC)N(CC(C)OC)CCOCCO)cc(C)c(C)c([N+](=O)[O-])c1C 59470,[N-]=[N+]=Nc1ccc(C(=O)NC2CCC3CN(C(=O)Cc4cccnc4)CC23)cc1 59471,C1(C(=O)N(C2C=CCN(C(=O)CC34CCC(CC3)C4)C2)CCO)CC1C1CCOCC1 59472,C1(CNC(c2n(C)ncc2)=O)CN(C(c2cc(F)n(C)n2)=O)CCN1C 59473,C1(CNC(CC=C)=O)CN(C(C2(O)CC(CF)C2)=O)CCO1 59474,c1(COCC)cn(CC2CCN2Cc2ccc(-c3cccs3)[nH]2)nn1 59475,N1(CCNC(c2n(CC)ncn2)=O)CCCN(C(C2CC(C#N)(OC)C2)=O)CC1 59476,C12(C(=O)NC(CNC(CCC=C(C)C)=O)CO)CCC(C)(C1)OC2 59477,n1(CC(N2CC(CCCOC)C2)=O)nc(C(F)(F)F)c2c1CCC2 59478,N1(C(CC(Cc2ccc(OC)cc2)N)=O)CCC(O)CC1(C)C 59479,O=C(CC(C(F)F)n1cccn1)Nc1ccnn1CC(=O)OCn1cccn1 59480,C1(NC(=O)Cn2cc(C3CCC3)nn2)(CNC(c2cnc[nH]2)=O)CCOC1 59481,c1(CC(=O)NC2(CC=C)CN(C(=O)C(C)CO)C2)ccc(NC2CCCC2)cc1 59482,N1(C(c2c(CC)cns2)=O)CCN(C(=O)CCc2cncc(F)c2)CC1CCO 59483,C1(C)(CC)CC(NC(c2cc(O)n(C)n2)=O)CN1C(=O)COCc1nccn1C 59484,C1(NC(C(C(C)C)C2CCC2)=O)CCCC12CN(C(=O)CC1CC(C)C1)C2 59485,N1(C(C2(C)CCCS2)=O)CCC2(CC1)CC(NC(c1ncc(Cl)cc1F)=O)CCO2 59486,C1(c2cnc(C)[nH]2)NC(=S)N(CC(C)C)C2=C1C(=O)NC(C)C2 59487,C1(C)(C(=O)NCCN(C(=O)COCC2CCCO2)CCC)CCC(C)=C(C)C1 59488,C1(NC(c2cc(C)sc2C)=O)CC(NC(=O)CCOC2CC2)C12CCOCC2 59489,c1(C(N)=O)ccnc(CNC(C2CC=CCC2NC(=O)CC2OCCCO2)=O)c1 59490,CCC(CC(=O)NCC1CCCC1C(N1CC(C)(C#N)C1)=O)C(F)F 59491,N1(C(C(C=C=C)C)=O)C2CCC(C2)C1C(N1CCC(NC(=O)NC)C1)=O 59492,C#CCC(C)(C)C(=O)N1CC2(NC(=O)CC3(O)CCCC3)CC1C2 59493,N1(C(Cc2c(OC)ccc(C)c2)=O)CC(C2CN(C(C3CC(C)CCO3)=O)C2)C1 59494,CC1(C)CCC(O)(c2cn(C3CC4(CC(CO)C4)C3)nn2)CC1 59495,C1(CNC(c2nccnc2Cl)=O)CC(N=c2[nH]ncs2)C1 59496,Cc1ccc(OCC(=O)NC2CC3CCC2(NC(c2cnsc2C)=O)C3)cc1C 59497,C=CC1CN(C(c2cccc(COC)n2)=O)CC1NC(C12CC(F)(C1)C2)=O 59498,N1(C(C(CCC)CNC(C2CC(=O)NC(=O)C2)=O)=O)CCC(O)C12CCC2 59499,C1(C(C)C)CCc2c(sc(NC(c3cc(C4CC4)ns3)=O)c2C#N)C1 59500,C(=O)(CCS(C)(=O)=O)NC(C)C(C)C(=O)NC1CCCSC1 59501,c1(SCC)nccnc1C(=O)NCC1(CN(C)C(C2CC=CC2)=O)CC1 59502,c1(-c2cc(C)cc(C)c2)cccc2c1CCN(C(c1ccc(CCO)cc1)=O)C2 59503,C(=O)(CS(C)(=O)=O)N(CC(=O)NCC(COC)(C)O)CC(C)C 59504,c1(C(=O)NCC(CN(C(c2c(C)noc2C(C)C)=O)C)O)cn2c(n1)CCC2 59505,N1(C(C(CC)(F)F)=O)CC2CC(C)N(C(c3cc(N)cc(Br)c3)=O)C2C1 59506,CC(C)(CC(=O)N1CCN(C(c2ccc(N)c(F)n2)=O)CC1)C(F)F 59507,C1(CCNC(c2c(C)cnn2C)=O)CCCN(C(=O)C(F)(F)C(F)F)CC1 59508,c1(CNC(CC2(C)CN(Cc3c(C)cco3)C2)=O)c(F)cccc1Br 59509,C#CCCN=C(NCC(c1ccccc1)CO)NCC1(C)CCCCO1 59510,c1(C(N(C2CCN(C(c3c(CC)csc3)=O)C2)C)=O)ncc(NC)cn1 59511,c1(C(=O)NC2(CC)CCCN(C(=O)C(C(C)C)NC=O)C2)cnc2n1CCCC2 59512,CC(C)CN=C(NCc1cnnn1C)NCC1(S(C)=O)CC1 59513,c1(C(N2CCC(NC(C3(NC(C)C)CC3)=O)C2)=O)ccc(Cl)c(C(F)F)c1 59514,C(CC(F)F)(C(=O)NCC1(C)CC(C)(C)C1)NC(c1cn(C)nn1)=O 59515,C12CC1C2(C)C.C1(c2cn(CC=C)nn2)COCC1C(C)=O 59516,c1(C(=O)NC23CC(NC(=O)CCc4ccccn4)(C2)C3)cc2cccc(Cl)c2nn1 59517,C1(CNC(c2ccc(CSC)o2)=O)CC(F)CN1C(C1OCCC1(C)C)=O 59518,N1(C(C(COC)C)=O)CC2(C)CN(C(c3ccn(CC4CC4)c3C)=O)CC2(C)C1 59519,CCCCCC(O)C(=O)NC1CN(C(=O)COc2ccc(CC)c(C)c2)CC1C 59520,c1(C(=O)NCCCCc2cn(-c3ccc(Br)cc3Cl)nn2)ccc2ncsc2c1 59521,C12(C(=O)OCc3ccc(Cl)s3)CCCCC1C2 59522,Cn1cc2cccc(-n3cc(CN4CCCC4)nn3)c2n1.N12CCCC(C1)C2=O 59523,N1(C(c2c(N)cc(Cl)c(Cl)c2)=O)CCCC2CN(C(C34CC(F)(C3)C4)=O)CCC12 59524,n1(C(c2nnnn2C2CC2)NC(CCC)Cc2ccccc2)nc2c(n1)CCCC2 59525,C=CCC(C)(C)CC(c1nnnn1-c1ccccc1Cl)NCC1(C(N)=O)CC1 59526,Cn1ncc2nc(O)c(C(N3CC(CCCCNC(c4ccc[nH]4)=O)C3)=O)cc12 59527,C1(CCC)CN(C(C2CC(C)(F)C2)=O)CCN1C(c1cnc(SC)s1)=O 59528,Cc1cc(C(=O)NC2(C(=O)NCC3CC(C)CO3)CC(O)C2)n(C)n1 59529,C(CN(C)C(c1cc(CNC(=O)CC2CCC(=O)C2)no1)=O)(C(C)C)OC 59530,c1(C(=O)NC2CCCN(C(C3CCCCC3)=O)C2)c(O)cc(Br)cc1F 59531,N1(C(C(C)=C2CCC2)=O)CCC(NC(=O)COC2CCOCC2)C2(CCC2)C1 59532,C(=O)(C(C)C(CC)CC)NCC(CC)NC(=O)CCCC1CCOCC1 59533,c1(CCC)cc(C(=O)NC(C)(CNC(C2CCS2(=O)=O)=O)CO)n(C)n1 59534,CC(O)C(C)C(=O)NCc1ncc(C(=O)NCC2CC(F)(F)C2)cn1 59535,CCC(C)C(C(=O)NC1(CO)CC2CCCC12)NC(=O)C=CC(F)(F)F 59536,c1(C(C)=O)ccc(=NCCNC(c2ccc(-c3cccs3)cc2)=O)[nH]c1 59537,Cc1cnc2c(cnn2CC(=O)N(CC(C)NC(=O)CC2CCOC2)C)c1 59538,C12(NC(CCCN(C)C)=O)CCC1CN(C(=O)CCN1CCCS1(=O)=O)C2 59539,N#CC1CN2CC1C2.c1(CC(=O)Nc2ncc(Br)cn2)ccc(Br)cc1F 59540,C(=O)C1=CSCS1.n1(CC(CC)O)cc(C(=O)NCCN(CCOC)C(C)=O)nn1 59541,C1(NC(CCCOCC=C)=O)C2CC3C1C3C2C(=O)NCCC1CCCC2CC12 59542,CN1CCC(O)C(N(C(=O)CN2CCN(CC3CC(C4CC4)C3)CC2)C)C1 59543,N1(C(c2c(C)nc(COC)s2)=O)CC2CCN(C(=O)CCC3CC3(Cl)Cl)C2C1 59544,CC1(C)CC(C)(CNC(c2cnsn2)=O)CN1C(c1ncoc1Br)=O 59545,c1(C(=O)NCC(C(C)C)NC(c2oc(CC)c(C)c2)=O)scc2c1CCCC2 59546,Cc1ccc(OCC(=O)NC2C3CN(C(C4(C#N)CC45CCC5)=O)CC23)c(F)c1 59547,C(=O)(C1=NNC(=O)C1)N1CC(SC2(C(N3CCCC(C)C3)=O)CC2(C)C)C1 59548,c1(C(N2C3C(NC(CCCC=C)=O)CC(C3)C2)=O)cc([N+](=O)[O-])cn1C 59549,c1ccc(Br)cc1.C(C(=O)NC)(C1CC1Cl)N(C1CC(C(F)F)C1)C 59550,C1(C(N(CCC(=O)NC(c2cccs2)C)C)=O)C(C)(C)C1(F)F 59551,CCCCCCCC(F)C(=O)NCC1CCN(C(C2(C)CCCC2)=O)C1 59552,N1(C(C2CCC(CCCCOC)C2)=O)CCN(C(C2CCCC23CC3)=O)CC1 59553,N1(C(C23CC(C)C2C3)=O)CCN(C(=O)C(C)(F)F)C2COCC12 59554,C1(Cc2cn(C(C)(C)C)nn2)CCN(C(=O)CCC#N)CC1(F)F 59555,N1(C(c2ccc(CSC)o2)=O)CCN(C)CC1CNC(=O)C1=CC(C)(C)C1 59556,N1(C(C2N(C)CCC2)=O)CC2CC1C2NC(=O)CCN(c1ccccc1)C 59557,c1(C(=O)NC2(CC=C)CN(C(C3(CSC)CC3)=O)C2)ccnc(F)c1 59558,C1(NC(CC2(C)CCN2C(=O)C(C2(O)CCCC2)F)=O)CCCC(O)C1 59559,C1(CC)CN(C(c2nn(CC(F)(F)F)cc2Cl)=O)CCC1NC(=O)CN1CCC1 59560,c1(C(N2CCC(CC=C)(NC(=O)CCCC(N)=O)C2)=O)cccc2ncc(C)n12 59561,C1(NC(c2c(NCC)scn2)=O)CCCC12CN(C(c1cc(C#N)[nH]c1C)=O)C2 59562,N1(C(=O)CSCCN(C)C)CCCC(C)(C(=O)NC(c2ccccc2)C)C1 59563,C1(CC(=O)NCCN(CCCN(C)C)C(=O)C=C(C2CC2)C2CC2)NC(=O)NC1=O 59564,N1(C(C23CC(C#N)(C2)C3)=O)CC(C(=O)NCCCOC(F)(F)F)C(F)(F)C1 59565,c1(CC(=O)NCC2N(C(C(CC)(C)OC)=O)CC2)ccc(Cl)c(Cl)c1 59566,C(=O)(C#CC(C)(C)C)NCCN(C(c1snnc1C(C)C)=O)CC 59567,Cc1ccc(Cl)cc1C(=O)NCCC1(O)CN(C(C2COCC(C)O2)=O)C1 59568,N1(C(C(C)OCCOCC)=O)CC(Nc2ccccc2F)C2(COC2)C1 59569,S(=O)(=O)(c1cnc(NCCc2cc(Br)no2)c(Cl)c1)N1CCn2c(C)ncc2C1 59570,CCC(C)C(O)C(=O)N1C2CCC1(CNC(C1(C)CCC1)=O)CC2 59571,c1(C(N2CCN(C(C(C)=CC)=O)C3C2C3)=O)cccc2c1CCOC2 59572,C1(CC)(NC(=O)C(C)Oc2ccc(C)cc2)CCN(C(=O)CC2(OC)CC2)CC1 59573,C(CNC(=O)Cc1cnnn1C)(CC(F)(F)F)NC(C(C)SC)=O 59574,C12CCCCN(C1)C(=O)CC2.C1(C(=O)NCc2ccn(C)n2)CCCC12CCC2 59575,c1(OCC(=O)NC(CNC(CCC(=C)Cl)=O)C2CCC2)ccc(F)cc1O 59576,c1(SC)nc(Cc2ccc(COC(C)=O)cc2)ncc1Br 59577,N1(C(C(C)SCCCC)=O)CCN(C(c2c(C)noc2C)=O)CC1c1ccccc1 59578,N1(C(C)C)CC(NC(=O)C(Cc2cn[nH]c2)NC(=O)CCc2cccs2)C(C)C1 59579,N1(C(C(=O)NCC)=O)CCCC(C)(NC(C2CC23CC(O)C3)=O)C1 59580,CCC(C)C(O)CC(=O)NC1(C)CC(NC(c2n[nH]c3c2CCSC3)=O)C1 59581,N1(C(COCC(=O)OC)=O)CC2C(NC(C3CN(C(C)C)CCO3)=O)C2C1 59582,N1(C(c2cc(CC)on2)=O)CC2(CC2)CC1C(=O)NCCN1CCCC(O)C1 59583,C(=O)(CS(=O)(=O)C1CCCC1)NC1CCCCN(C(Cc2ncc(C)s2)=O)C1 59584,C(=O)(C(CCC(N)=O)n1cc(-c2ccc(Cl)cn2)nn1)NCc1c(C)nc(C)o1 59585,C(c1ccccc1Cl)=CC(=O)N(CCC(C)NC(CCc1c(C)nn(C)c1)=O)C 59586,C(c1ccncc1)=CC(=O)NC(C(C)NC(c1cscc1F)=O)C 59587,C1(CC(=O)NC2C(OC)CN(C(c3cc4ccsc4s3)=O)C2)CC(C)(C)OC1=O 59588,C1(CC)CC1N=c1[nH]c(N(C)Cc2nn(C)c3ccccc23)nc2ccsc12 59589,c1(NCC2N(C3CCN(C(C)=O)CC3)CC(O)C2)ccc(C)c(Cl)c1 59590,c1(N2CCC(C)SCC2)ccncc1S(=O)(=O)N1CC(C)(C)OCC1CO 59591,c1(C(=O)NC2CC(NC(C(C=C=C)C)=O)CC2O)cc(O)nc(C)n1 59592,c1(C(=O)NCC2C(NC(C3(COC)C=CCC3)=O)COC2)[nH]c(O)nc1C 59593,CCCC(C(=O)NC(C)CNC(=O)CCc1cc(C)on1)C(C)C 59594,N1(C(CCNC(=O)OC)=O)CCC(NC(=O)CC2COCCN2C)C1C(C)(C)C 59595,C1(C(=O)NCCC(C)CCO)(OC)CCN(C(C2(OC)CC(=O)C2)=O)C1 59596,c1(CNC(CCN(C(=O)C(c2cncnc2)C)CC#C)=O)ccc(Cl)cn1 59597,N#Cc1cc(C(N2CCC(CC(=O)Nc3ccc(F)c(F)c3Cl)C2)=O)ccc1F 59598,C1(CNC(C(C)NC(=O)C(C2CCCCC2)O)=O)CCOC1(C)C 59599,N1(C(=O)NCc2ccnn2-c2ccccn2)CCC2CCC12C(F)(F)F 59600,N1(C(c2c(C)cc[nH]2)=O)CCCC(C(=O)N(c2ccc(F)cc2)CC2CC2)CC1 59601,C1(C)(C(=O)NCCCCC(=O)OC)CCCN(Cc2cccc(O)n2)C1 59602,CC(C)CC(C)ONC(c1coc(C(N2CC(O)C2)=O)c1)=O 59603,C(=O)(C(F)C(C)CNC(c1cccc2c1CC2)=O)NCc1ncc(C)s1 59604,C(=O)(CC1C(=O)Nc2ccccc21)N1CC(C)C(NC(C2CSCC(=O)N2)=O)C1 59605,C(CCN=C(NCC1(C)CCCS1)NC1CCNC(=O)C1)OC(C)C 59606,C(=O)(C1CNc2ccccc21)NCC1CN(C(CC2C(C)(C)CCCO2)=O)C1 59607,C12(C(N3CCN(C(Cc4c(C)n[nH]c4)=O)C(C)C3)=O)CC(C)(C1)OC2(C)C 59608,c1(C(N(C(CNC(C2(Cl)CC2(F)F)=O)C2CC2)C)=O)cc(-c2cnn(C)c2)[nH]n1 59609,CC1CN(C(=O)C(F)C2CC2)CC(C)CN1C(=O)Cc1cc(C(F)(F)F)co1 59610,c1(C(=O)Nc2ncc(F)cc2O)cc(Cl)cc(Cl)c1F 59611,Cn1cc(C(=O)NCC2CCCC2NC(c2ccccc2Cl)=O)nc1O 59612,c1(C(=O)NCC(CN(C(=O)C(CC)OC)CCC)O)ccnn1C1CCC1 59613,C1(C(N2CC3CC3(CO)C2)=O)C2CC(O)C(C2)N1C(C1(CC2CCC2)CC1)=O 59614,CC1=NN(C)C(=O)C1CC(N1CCC(CO)(NC(c2cc(CO)on2)=O)CC1)=O 59615,C1(O)(C(N(C(CCNC(c2ncn(CC)n2)=O)C)C)=O)CCC(C)CC1 59616,c1(C(=O)Nc2ccc(O)c(F)c2)ccc(F)cc1Cl 59617,c1(CC(=O)N(C(C)CNC(c2cscn2)=O)CC)conc1C 59618,N1(C(C=Cc2scc(C)n2)=O)C2CCC1C(F)C(NC(C1(Cl)CC1(C)C)=O)C2 59619,C(=O)(CC(C(F)(F)F)NC(=O)C(C)OCC(C)C)NC1(CCC)CCSC1 59620,N1(C(c2ccc(CC)o2)=O)CC=CC(C(=O)Nc2cc(OC)ccn2)C1 59621,C(=O)(C1CCCc2ncccc21)NC(C(C)C)CNC(c1ccnnc1O)=O 59622,C#Cc1cncc(NC(C2CCN(C(c3n[nH]c(C)c3Cl)=O)CC2O)=O)c1 59623,C(=O)(CCC(C)(F)F)NCCCCC(C)NC(C(C)C)=O 59624,c1(N2C(COC)(CNC(=O)Cc3ccccn3)CCC2)ccccc1[N+](=O)[O-] 59625,C(=O)(C(C(C)C)NC(C1(O)CC1)=O)NCC(C)NS(CC)(=O)=O 59626,c1(C(N)=O)ccccc1C(=O)NCC1C2CC1N(C(C1CC3CCC3C1)=O)C2 59627,c1ccc(I)cc1.C(=O)(C(C)N1C(=O)C2CC2C1=O)OC(CC)C.C(C)(C)(C)O 59628,C1(C(=O)NCCCNC(CC2(OCCNC(C)=O)CCC2)=O)CC12CCOC2 59629,c1(N2CCC(C(N3CCC(S)CC3)=O)C2)ccccc1F.c1(OCCN)ncccn1 59630,C12(NC(c3ccc(C)cc3)c3nn[nH]n3)CC=CCN1CCC2.C1C(=O)O1 59631,c1(NCCCOCC)ncc(S(=O)(=O)N2CCS(=O)(=O)CC2C)cc1Cl 59632,Cc1cccc(Cl)c1CC(N1CCC(C)(CNC(=O)CC2CCCC2)C1)=O 59633,C(=O)(CC(C)CC(=O)OC)N1CCCC(CC(=O)N(CC(C)OC)C)C1 59634,c1(N2CCC(NC(=O)C=Cc3cccs3)(CF)C2)cc(Cl)nc(C2CCC2)n1 59635,CC(C)CC(C)(CNC(=O)Cc1cnsc1)NC(=O)CN1CCC(O)CC1 59636,C1(CNS(=O)(=O)c2ccoc2)CCC2(CCOCC2)CO1 59637,c1(NCCN2CCC(NC(=O)OC(C)(C)C)CC2)cc(F)c(Cl)cc1I 59638,Cn1cnc2c(N3CCOCC(NC(c4ccc(F)c(O)c4Br)=O)C3)ncnc12 59639,C1(NC(C(=O)NC(C)C)=O)CCC(C(=O)NCC2C(C)(C)C2(C)C)CC1 59640,C1(C(C)NC(c2coc(CO)c2)=O)CCCN(C(=O)CC2(N(C)C)CCCC2)C1 59641,C1(CN(C(=O)C=Cc2ccoc2)C)CCCN(C(C2CCC(=O)N2C2CC2)=O)C1 59642,c1(C(=O)NCC(C)N(C(N)=O)C)ccn(CC(=O)NC(c2ccco2)=O)n1 59643,S(=O)(=O)(CC(=O)NCC1CN(C(C2(N(C)C)CC2)=O)CC1C(F)(F)F)NC 59644,C1(C)(CC)CN(C(C2CCCN(C(=O)C=CC(C)(C)SC)CC2)=O)CCO1 59645,C1(COC)(CNC(=O)CC(C)F)CCCN1C(c1cccc[n+]1[O-])=O 59646,CCCC(CCC)C(=O)N1CCCN(C(c2cnc(O)s2)=O)C(C)C1 59647,C1(C(N(C(C(=O)OC)C)C)=O)C(C)OCCN1C(C1CS(=O)C1)=O 59648,S(=O)(=O)(C1CCCN(C(c2ccccc2OC)=O)C1)N1CC(C(C#C)C)C1 59649,N1(C(C2C(C(=O)OCC)C2)=O)CCC(CC(=O)NC(c2noc(C)n2)C)C(O)C1 59650,N1(C(CC2CCC(C)C2)=O)CC2(C1)CN(C(c1cn(C)cc1C(F)(F)F)=O)C2 59651,C1(C(=O)NCCOC)CC12CCN(C(c1ccsn1)=O)C2 59652,C1(c2n(C(C)C)nnn2)(NCc2ccncn2)CC2CC1CC2(F)F 59653,c1(C(=O)NC(C(C)NC(c2c(C)n(C)cc2)=O)(C)C)cc(F)ccc1Cl 59654,C(CNC(c1cc2n(c1)CCC2)=O)(C(C)C(C)C)NC(C(C)=C1CCC1)=O 59655,N1(C(c2c(CC)n[nH]c2)=O)CCCC(N(CCO)C(c2ccoc2C)=O)C1 59656,Cc1nscc1CCNC(=O)NCCc1nocc1C(C)C 59657,c1(CC(=O)NC2CCCC2C(N2CCC(O)CC2)=O)ccc2occc2c1 59658,C12(CCCN(C3CN(C(C4CCOC4)=O)C3)C)CCC(CC1)C2 59659,c1(NC(C2CC(F)CN2C(c2cnc[nH]2)=O)=O)nc(Cl)cc(Cl)n1 59660,CCC1=C(C(=O)N2CCCCC2CCNC(=O)CC(O)CN(C)C)CCCO1 59661,N1(C(C(c2ccn(C)c2)C)=O)CCCC1CC(N1CC(F)C1)=O 59662,C(=O)(C(C(C)(C)C)NC(c1ccccn1)=O)N1CCN(C(CC)=O)CC1 59663,C1(C(=O)NCCC2(CNC(Cc3c(C)ocn3)=O)CC2)CCn2ccnc2C1 59664,c1(Nc2c(C(F)(F)F)ccc(OC(F)F)n2)ccc(N=c2ncnc3[nH][nH]c(Br)c2-3)s1 59665,C1(C(N(CCC=C)CC)=O)CC2(CC2)CN1C(c1cn(CCO)nn1)=O 59666,C1(NC(c2nc(C(C)C)sc2)=O)CC2(CCCCN2C(C2(O)CCC2)=O)C1 59667,C(=O)(C(F)(F)c1cncs1)NCC(C)NC(=O)C(c1ccc(Cl)s1)C 59668,N1(CCCC(=O)NC(Cc2c(C)cccc2)C)C(=O)CN(C)C1=O 59669,Cc1nc(N2CCC(c3cccc([N+](=O)[O-])c3)C2)nc2ccccc12 59670,C1(O)(C(=O)NCC2CC(NC(C(C)(C)OC(C)=O)=O)C2)CN2CCC1CC2 59671,C#CCCN=C(NCCc1ccccc1C#N)NCCc1ccn(C)c1 59672,CC1C(C)N(C(=O)Cc2nnn(C(C)(C)C)n2)CCN1C(=O)C(=O)C(F)(F)F 59673,N1(C(COC(C)=O)=O)CC(NC(C2(C)CCN(C)C2=O)=O)CC12CCC2 59674,C(CC(O)CN=c1ncnc2[nH][nH]c(C)c1-2)NC1C(CC)CCCC1.C1C(=O)N1 59675,c1(C(=O)NC2C(C)CN(C(C3CCC(C)CC3)=O)CC2)nc2ccccn2n1 59676,c1(C(C)C(=O)N(C)CC2CCCN(C(c3ccnnc3)=O)C2)ccc(F)c(F)c1 59677,N1(C(CC2CC(OC)C2)=O)CC(C(=O)Nc2cc(C)cnc2O)CC(C)C1 59678,C(=O)(C1=CCCCO1)NCCCCCCNC(CCC1CCCN(C)C1)=O 59679,c1(C(=O)NCCCNC(C23CC4CC2C3C4)=O)ccc2c(n1)CCCN2 59680,C(C1C(C(=O)NCC2CCC2NC(=O)CC(F)F)C1(C)C)=C(C)C 59681,CC1(C)CNC(=O)C1NC(=O)C(F)C1CC(NC(c2ccc(F)cn2)=O)C1 59682,c1(C2(C(=O)NCC=CCNC(CCC(C)OC)=O)CC2)ccccc1C#N 59683,C1(NC(C(C)NC)=O)C2CCCC1CC(C(=O)Nc1ccccc1)C2 59684,c1(C(=O)NC(C2CC(NC(C(c3ccccc3)SC)=O)C2)C)cc[n+]([O-])cc1 59685,C1(O)(CNC(c2c(C)cno2)=O)CCCN(C(C2(N3CCOCC3=O)CC2)=O)CC1 59686,C1(NC(C(CNC(c2c(NC)scn2)=O)(C)C)=O)CN(C)C(C)(C)C1 59687,Cc1ccc(C)c(C(C(=O)NC2CC(C)(NC(C3(N(C)C)CC3)=O)C2)C(C)C)c1 59688,C#CC1(C(N2CCC(OC)C2C)=O)CCN(C(=O)Cc2cccnc2)CC1 59689,c1(CC(=O)NCCC2CCCC2)ccc(Cl)cc1.C1(C(=O)OCC)(NC=O)CC1 59690,C(C(=O)NC(CCSC)C(=O)NCc1cnn(CCF)c1)(C(C)C)SC 59691,C(=O)(C(C)(C)C)NC(CNC(C1CC1C(C)C)=O)C.C(C)(C)(C)OCC 59692,c1(C(=O)NCC2(O)CCN(C(C(C)SC)=O)C2)coc2ccc(OC)cc12 59693,C(=O)(C1=C(Cl)CCOC1)N1CCC(CC)CC1C(N1CCC1(C)C)=O 59694,C12(C(N3CC(C(CCC)O)C3)=O)CCCC1CCN2C(c1cncc(C)c1)=O 59695,CC1(C)CCCN(C(=O)CSCCc2ccccc2)C1CNC(c1cscn1)=O 59696,C1(C(=O)NCC2(NC(=O)C(=O)N(C)C)CC(OC)C2)CCCC(F)C1 59697,C=C(C)CCC(=O)NC(CN(C(=O)C(C)(c1ccccc1)OC)C)(CO)CO 59698,CC1(C)Cc2cc(Br)ccc2C1NC(c1nnsc1C(F)F)=O 59699,N1(C(CCNC(C)C)=O)CCCN(C(=O)CC2COC(=O)C2)CC1 59700,C1(F)(C(=O)NCCCC(C)NC(C2(c3cccnc3)CCC2)=O)CCCN(C)C1 59701,Cn1ccc(CCNC(=O)C(c2ccccc2)NC(C2CC=CCO2)=O)n1 59702,c1(C(=O)NCC2N(C(c3cncc(C=C)c3)=O)CCC2C)ccc2c(c1)CCO2 59703,C1(OC)(CNC(=O)Cc2cnc(C)[nH]2)CCN(C(=O)CSCCC(C)C)C1 59704,N1(C(c2cc(C)[nH]n2)=O)CC2ON=C(CNC(c3ccc(N(C)C)cc3)=O)C2C1 59705,c1(NC(C(c2csc(Cl)n2)N(CC(=O)OCC)CCC)=O)ccc(CC#N)cc1 59706,c1(OC)ccc(C(CCO)NC(=O)NC(c2ccc(Cl)cc2)C#N)cc1 59707,C1(CN(C)CC2CCN(C(C3CCC(=O)N3)=O)C2)C(C)(C)C1(C)C 59708,Cc1nc(C)c(CC(=O)NCC(C)(C)CNC(c2cc(C3(C)COC3)no2)=O)s1 59709,C1(NC(Cc2c(C)ccs2)=O)CCN(C(c2ccnc(OC(C)C)c2)=O)C(C)C1 59710,N1(C(C(C)=C(C)C)=O)CC2CC(NC(=O)C(C(C)C)n3ccnc3)C1C2 59711,N1(C(c2scc(CC)c2)=O)CCCC(C)(NC(=O)COCC2CCOC2)C1 59712,Cc1c(F)ccc(N)c1C(=O)NC1CC(NC(C2(OC(C)C)CCC2)=O)C1 59713,c1(C(N(CCNC(=O)C(C)(O)COC)CC)=O)cc(F)c(F)c(Cl)c1F 59714,c1(C(N2CC(CN(C(CC(=O)N(C)C)=O)C)OCC2)=O)cc2cccc(O)c2[nH]1 59715,Cc1cc(F)c(CC(=O)N(CC(C)(C)NC(=O)CC2CC3(CC3)CO2)C)cc1F 59716,CC1=C(C(=O)N2CCC(CNC(C3OCCO3)=O)C(C)C2)C(=O)OC1(C)C 59717,C1(NC(C2CC2c2ccccc2F)=O)CC(F)CN(C(c2ccc[n+]([O-])c2)=O)C1 59718,CC1(C(=O)NCc2cc(F)cc(Cl)c2)CCN(c2nccc(SC)n2)CC1 59719,C1(CC(=O)N(C(C2(O)CN(C(c3cc(C(N)=O)co3)=O)C2)C)C2CC2)COCCOC1 59720,N1(C(Cc2ncc(CC)[nH]2)=O)CC2=C(C1)CN(C(=O)Cc1ccoc1C)C2 59721,C(=O)(C(F)(F)C(F)F)NCC(N1CC(CC(CC2C(CC(C)C)C2)(C)C)C1)=O 59722,C(CCC)(C(=O)N1CCC(CN(C(c2onc(C)c2C)=O)C2CC2)CC1)=CCC 59723,C1(NC(CCOC)=O)CCC12CCN(C(=O)CCc1cnn(C)n1)CC2 59724,c1(N2C(CN(C(CCCC(C)=O)=O)C)COCC2)nc2cccnc2s1 59725,CC1CN(C(C2(C#N)CC2)=O)CCN1C(=O)C(C)C(F)(F)F 59726,Cc1cccc2cc(C(=O)NCC(C3CCC3)NC(C3CCCN(C)C3)=O)nn12 59727,C1(C)(C(=O)NCCN(C(c2cn(CC)nn2)=O)C)CC(C(F)(F)F)=NO1 59728,N1(CCCC=O)C(CCNC(C=CC(C)(C)SCC)=O)CC(C)C1=O 59729,Cc1ccc(C=CCC(=O)NC2(CCNC(C3CC3F)=O)CC2)cc1 59730,Cc1c(C(=O)NC2(C)CC(NC(=O)C(O)C(F)(F)F)C2)sc2nnc(S)n12 59731,N1(C(CC(CC)C2CC2)=O)CCC(NC(C2COCCO2)=O)C(CO)CC1 59732,c1(CC(=O)NCC(CCOC)NC(C2(O)CC(CF)C2)=O)cccc(Cl)c1F 59733,c1(CC(=O)NC2C(CNC(CNC(C)=O)=O)CCC2)cc(O)ccc1Br 59734,C1(NC(C2C(OC)C2)=O)CN(C(=O)CC2CC2)CC1c1ccnn1C 59735,N1(C(C(CC)CC)=O)C(CNC(C2CCN(S(C)(=O)=O)C2)=O)CC2CCCC12 59736,CCC(C(=O)NCC1(C2(O)CN(C(=O)CC3(O)CCCC3)C2)CC1)C(C)(F)F 59737,n1(CC(=O)NCCn2nccc2C(=O)NOCCCF)cccnc1=O 59738,c1(NC(C2C3(CN(C(C(c4ccc(OC)cc4)C)=O)C3)C2)=O)ccc(O)c(C)n1 59739,O=[N+]([O-])C1C2CCCC(N(c3ncnc(C(F)(F)F)c3Br)C3CC3)C12 59740,C=C1CCCN(C(=O)CCN(CC(N)C(C)C)C(=O)CN(C)C)C1 59741,N1(C(c2c(C)occ2Br)=O)CC2(CC(NC(=O)C(C)(C)C(C)O)c3nccn32)C1 59742,CCC(C)(COC)C(=O)NC(C1(NC(=O)C(N)=O)CC1)C 59743,C1(F)(CNC(c2n(CC=C)ccn2)=O)CCCN(C(c2cc(N)ccc2O)=O)C1 59744,N12CC(F)(C1)C2=O.C(C)(C(=O)NC(C)C(C)O)OCCOCC 59745,Cc1cc(NC(N2CCCC2C2CC2(F)F)=O)c(C)s1 59746,N(C(=NCCc1ccc(F)cc1C)NN1CCN(C(=O)NC2CC2)CC1)C(C=C)C 59747,C(CCC(C)C(=O)N1CCN(C(c2sc(=N)[nH]c2C)=O)C(c2ncc[nH]2)C1)OC 59748,N1(C(C2CN(C)CC(C)O2)=O)C2CCCC1CN(C(=O)CCc1cnn[nH]1)C2 59749,c1(SCCC(=O)N(CC(CN(C(C(C)(C)OC)=O)C)O)C)cc(F)ccc1F 59750,O=C(CCN=c1nc(N2CCCC3(CCCC3)C2)c2sccc2[nH]1)NC1CC1 59751,N1(Cc2ccc(F)cc2)C2CCCC1CN(n1cc(-c3sccc3Cl)nn1)C2 59752,C1(CNC(c2csc3nnsc23)=O)CC2CCC(C1)N2C(c1cscn1)=O 59753,c1(NCC(F)=C(C)C)cc(Br)ccc1S(=O)(=O)N1CCCC1C 59754,c1(C(N2CC3C(C2)N3C(=O)Cn2nc(O)ccc2=O)=O)ncc(Br)cc1Cl 59755,O=CN1CCCC1C(N1CCC(CCNC(c2cnco2)=O)C1)=O 59756,c1(N)nc2c(F)cccc2n1C.c1(CC)ccc(CF)cc1 59757,Cc1ccc2ncnc(N(C3CNCC(C)C3)c3ncccn3)c2c1 59758,c1(C(N2CC(CC=C)(NC(=O)Cn3ccnn3)C2)=O)cnc2[nH]cncc1-2 59759,C1(CCC(=O)N(C2C(C)CC2)C)CCCC1.C(=O)(CCCOC(C)=O)NC(C)C 59760,N1(C(c2nc(COC)oc2)=O)C2CCC(C(=O)Nc3csnc3OC)C1CC2 59761,C(=O)(C(F)CC(C)(C)NC(C1CNC(=O)O1)=O)NCC1(O)CCCC(C)C1 59762,C12(NC(c3ccco3)=O)CC(C1)N(C(=O)CCc1sccc1Br)C2 59763,Cc1nc(-c2ccccn2)sc1C(=O)NCC1C=CCN1C(C1(O)CCC1)=O 59764,c1(C(N2CCC(Cn3cc(C(C)(C)C)nn3)C2)=O)ccc2c(c1)C(=O)C(=O)NC2 59765,CN1CCN(C(=O)NC(c2ncccc2F)C2CCC2)C(c2cccs2)C1 59766,C12(NC(C(C)Oc3cccnc3)=O)CCC(CC1NC(=O)COCCN(C)C)C2 59767,c1(CNC(C(F)OC)=O)ccccc1CNC(=O)Cn1ccnc1C 59768,c1(OCC)cc(C(=O)NCC(CNC(C2(CC)CC2(F)F)=O)CO)ccn1 59769,c1(C(N2CCC(N(C(=O)COCC(F)F)CC)C2)=O)c(C)ccc(C)c1O 59770,C(CNC(C1CC1c1ccn(C)n1)=O)(CC(C)C)NC(c1nc(OCC)sn1)=O 59771,c1(C(=O)NC2CC(CCNC(C3(COC)COC3)=O)C2)sc(C)c(C)c1C 59772,C(=O)(CCC(C)(C)NC(C12CC1CN(C(=O)CCC1CCCOC1)C2)=O)OC 59773,C1(NC(c2ccc(CNC(C(CN(C)C)(C)C)=O)nc2)=O)COC2(CCCC2)C1 59774,C1(NC(C2CCC3CCCCN23)=O)CC2CCC(C1)N2c1ncnc(Cl)c1Br 59775,CC1CN(C(c2ncc(F)cc2F)=O)CC(CCNC(=O)C(C)(C)CO)O1 59776,N1(C(=O)COCC2CC2)CC2CCC1(CO)C2 59777,N1(C(C=Cc2nc(C)sc2)=O)CCC2CC1CN(C(=O)C(C)(C)n1cnnn1)C2 59778,CC1(C)OC2CCN(C(c3ncc(Cl)cc3F)C(=O)NC3CCCC3)CC2O1 59779,Cc1cc(=NCc2nnc(C(C)C)s2)[nH]c(NC2CCCC2C)n1 59780,Cc1nc(C(=O)NCC(C)N(C(=O)C(C(F)(F)F)C(F)(F)F)C)ccc1[N+](=O)[O-] 59781,N1(C(c2ccc(CC)[nH]2)=O)CCOCCC1C(=O)NC(c1cc(C)on1)C 59782,c1(C(=O)NC2(C3N(C(c4nc(C)sc4)=O)CCC3)CC2)cc(F)cc(F)c1 59783,c1(C(=O)NCC(C)N(C)C(C23CCC2C3)=O)ccccc1C(N)=O 59784,C12(CNC(=O)C3=CCCCCC3)CCCC1N(C(c1cccc(O)n1)=O)CCC2 59785,c1(C(N2CCC(C(C)NC(C(C(CC)C)O)=O)C2)=O)cnc2c(c1)c(C)nn2C 59786,c1(C(=O)NCc2cc(F)cc3c2CCC3)cncc2nc(O)[nH]c12 59787,C1(CNC(CC2CCN(C(c3c(OCC)scc3)=O)C2)=O)C(C)(C)C1(F)F 59788,CN1CC2CC1CN2C(C1C=CCN1C(C1CNC(=O)O1)=O)=O 59789,C1(CC(=O)N(CC(C)C#N)CCOC)CC2(CCC2)CO1 59790,C12(CC)CN(C1)C(=O)CC1C(C1(F)F)CC1CN(C1)C2=O.C1(COC)CC1 59791,C12(CCNC(=O)Cc3sc(O)nc3O)CCC1CN(C(c1ccc(F)o1)=O)C2 59792,C(=O)(C1(C)CCn2ccnc21)NCCN(C(CCCCC=C)=O)CCC 59793,C(=O)(CC(C)C(F)(F)F)NCC1CN(C(C2N(C(CC)=O)CCCC2)=O)CC1C 59794,C(CC)(CC(=O)NCC(F)Cl)NC(COCCCC)=O 59795,C1(F)(CNC(=O)Cc2ccc(Cl)s2)COCCN(C(c2ccon2)=O)C1 59796,N1(C(C(C)CC(C)(C)C)=O)CC2(CCCCN(C(=O)Cn3cccnc3=O)C2)C1 59797,c1(C(C)C)scnc1C(=O)NCC(O)CNC(c1ncc(C(F)F)s1)=O 59798,C=C(C)CC(C(=O)NC1C2CCC1CC2)NC(C1CCCN1C(C)C)=O 59799,c1(C(=O)NCC2(CNC(CC(C)(C)OC)=O)CC2)ccc(OC(F)(F)F)cc1F 59800,n1(CC(=O)NCC(CNC(C(CC=C)C)=O)O)cc(P(C)(C)=O)cn1 59801,Cc1ccc(C(N2CC(F)CC2C(N2CC3C(C(=O)N(C)C)C3C2)=O)=O)nc1C 59802,c1(CC(=O)NCCC2(CNC(C(C)S(N)(=O)=O)=O)CC2)cccc2c1OCC2 59803,CC1CCCCC1(CNC(C1CC2CCC1O2)=O)NC(C1CCCC2(CC2)C1)=O 59804,c1(C(CCC)NC(=O)NCCc2nccn2C(C)(C)C)ccc(Br)cc1 59805,S(=O)(=O)(c1cnn(C2CCCC2)c1)NCCOCC=C 59806,N1(S(Cc2cccc(C)c2)(=O)=O)Cc2ccc(C(=O)Nc3cncc(Cl)n3)cc2C1 59807,C1(C(=O)NC2(CC=C)CN(C(C3CC4CCC3CC4)=O)C2)CC2CCC1CC2 59808,c1(CCC(=O)NC2C(NC(CC(C)F)=O)C2)ccc(Cl)cc1Br 59809,c1(SC)nccc(=NC(=O)Cc2ccc(C(=O)NC3(C)CCCOC3)nc2)[nH]1 59810,N1(C(CC)C(=O)NC2CC3CC2N(C(=O)C(C)N(C)C)C3)CCc2ccccc21 59811,C(=O)(C(CCF)NC(C1CC(C)CCO1)=O)NCCCNC(C)=O 59812,N1(C(C2C=CC(=O)N=N2)=O)CC(NC(c2cc(Br)ncc2F)=O)C(F)(F)C1 59813,CC1(C)CCCC1(C)NC(c1cnc(CNC(c2cn(CCO)nn2)=O)nc1)=O 59814,c1(C(N2CCC(C3C(=O)NC(=N)S3)CC2)=O)nc[nH]c1[N+](=O)[O-] 59815,c1(OCC(=O)NC2CCCC(C)C2)cc(Cl)c(Br)cc1F 59816,c1(N2CCCC(SC)C2)nc(N(C)Cc2ccc(F)cc2)nc2cc(C)ccc12 59817,C1(n2cnnn2)(C(=O)NCCCCNC(C2C(OC)C2)=O)CCCSC1 59818,c1(OC)cc(=NC(=O)C2CCCN2C(C2CC(=O)C2)=O)[nH]n1C 59819,N1(C(c2c(=N)[nH]cnc2)=O)CCC2CCN(C(C34CC(CC(F)F)(C3)C4)=O)C2C1 59820,C(=O)(C(F)C(F)(F)C(F)(F)F)NCC=CCNC(c1cc(N)c(Br)cn1)=O 59821,C(=O)(C(CCC(C)C)N=C1NS(=O)(=O)c2ccccc21)NCCNC(=O)NC 59822,c1(C(N2C(C3(NC(C(C)SC)=O)CC3)CCC2)=O)cc(S(C)(=O)=O)cnc1O 59823,c1(C(N2CC(SC)C(NC(=O)C(O)CN3CCCC3)C2)=O)cncc(Cl)c1C 59824,N1(C(CC(C)N(C)C)=O)CC2(C1)OC1(C)CC2(NC(=O)COc2ccccn2)C1 59825,C1(NC2(C(=O)NC(C)C)CCC2)CCC(C)N(c2nccc(CO)n2)C1 59826,N1(C(CC(COC)C)=O)CCC(C)(C)CC1C(N1CCC12CC(C)(OC)C2)=O 59827,CC1(C)OC(=O)c2cc(C(N3CC(O)(CNC(C4CC4F)=O)C3)=O)ccc21 59828,C(=O)(C(CC)CCCCC)N1CCCC(O)(CNC(CCCC=C)CO)CC1 59829,C1(C(=O)NCC2CC(NC(CN(C(COC)=O)C)=O)C2)CC(C(C)=O)C1(C)C 59830,c1(OC)ccc2c(=NCC3CCCCS3)[nH]c(=NC(C)CS(C)(=O)=O)[nH]c2c1 59831,Cc1cc(OCCC(=O)NCC2(F)CCCN(C(=O)CCC(F)F)C2)cc(C)c1 59832,C#CCC(C)(CNC(=O)CCCN(C)C(C1CC2CC2C1)=O)CO 59833,N1(C(CC(CC(=O)OC)C)=O)CCCCC2(C1)CN(C(=O)Cc1cscn1)C2 59834,C=CC(CCC)CC(=O)NC(C)C(=O)NCC=CCNC(N1CCOCC1)=O 59835,c1(OC)c(C)cc(C(N2CCC3C(C2)C3(F)F)C(=O)NCc2ccccc2)cc1C 59836,C(=O)(CC(=O)NC1C=CC(CNC(=O)C(F)CC2CCC2)C1)OC 59837,N1(C(c2cnc(CC)s2)=O)CCCN(C(c2cnc(O)c(C)c2)=O)CCC1 59838,c1(C(=O)NCCC=CC)cc(O)nc2c1CN(C(C1CC1(F)Cl)=O)CC2 59839,C1(Cn2c(=O)cccc2)CCCN(N2CCC(OCc3cccnc3)C2)C1 59840,C1(C(=O)NC(C(=O)N(CCCC)CCOC)c2ccco2)CCS(=O)CC1 59841,C=CCC(C(=O)N(C)CC1CCCN(C(=O)C2=NNC(=O)C2)C1)C(C)(C)C 59842,C=CC1(O)CN(C(=O)CC2CCN(C(=O)C(C)(C)NC(=O)OC)CC2)C1 59843,Cc1nc2ccc(C(=O)NCC3CC4(CC(NC(=O)C(C)N(C)C)C4)C3)cc2[nH]1 59844,C1(CNC(c2c(OC)nc(C)s2)=O)CCN(C(=O)Cc2cnsc2)C1(C)C 59845,C(C(=O)NC1(CNC(=O)C(C(C)C)n2cnnc2)CCOC1)(C(C)C)OCC 59846,C1(F)(CNC(C=CCCC)=O)CCCN(C(=O)CCn2c(C)c(C)sc2=O)C1 59847,Cc1cncc(F)c1C(=O)NC1CCC(CCNC(=O)CC#N)C1 59848,C1(C(=O)N(C)Cc2ccn(C)n2)(CC)CCCN(C(=O)CSC2CC2)C1 59849,C(=O)(CC(C)(C)C(F)(F)F)NCC1N(C(CCOC)=O)CCC1C1CC1 59850,c1(CC(=O)NC)ccc(C(=O)NCC2CCN2C(=O)CC2COC(=O)N2)cc1 59851,CC(C)(C(=O)NCCC1CCCN1C(c1cnns1)=O)C(F)(F)F 59852,Cc1cc(C(=O)N(C)CCN(C(=O)C#CC2CCCCO2)C)c2[nH]cnc2c1 59853,N1(C(C=CCCC)=O)CC23CC1(C2)C(=O)NC3.C1(OC)CC2(C1)CC(C)(C)C2 59854,CCC(CC)C(F)C(=O)NCC1(C(=O)NCC2(C)COCCO2)CC=CC1 59855,Cc1cc(C)c(C)c(C(N2CC(O)(C(C)NC(=O)CCc3cscn3)C2)=O)c1C 59856,C1(C(N2CCCCC(CNC(CC3(C)CCCC3)=O)C2)=O)CC2CC1C1C2C1(F)F 59857,C1(NC(Cc2cc(C)no2)=O)CC(O)CN(C(c2c(O)cccc2F)=O)C1 59858,c1(C(C(=O)NC2CCSC2)C2CCCC2)cccc(NCC2CCCO2)c1 59859,C1(C)(NC(c2c(OC)oc(C)n2)=O)CCCN(C(=O)CCn2ccnn2)C1 59860,c1(OC)nc(OC)nc(N2CCC(C(N3CC4CCCC4C3)=O)C2)n1 59861,c1(C(=O)NC(C(C)F)=O)ccc(Br)c2cccnc12.C12CCN(CC1F)C2 59862,C(CCN(C)C)(C(N)=O)NC(C(CC)NC(CC1(OC)CCC1)=O)=O 59863,C1(C(N2CCC(=C)CC2)=O)CN(C)CCN1C(C1CC(=O)N(CC)C1)=O 59864,c1(C(=O)NCC2N(C(CC(C)(C)C3CC3)=O)CCOC2)cccc(C(N)=O)c1N 59865,C1(C(=O)NC(c2c(C)nns2)C)CCCCC1NC(=O)CN1CCCCC1=O 59866,CCC(CC(=O)NCC1OCCC1C)NC(=O)CCCOCCOC 59867,c1(CN(S(=O)(=O)c2cccc(C(F)(F)F)c2)C)cc2c(O)cccc2s1 59868,C(CC(C)CCO)NC(c1cncc(C(C)(C)C)c1)c1n(CC(=C)C)nnn1 59869,N1(C(C(C)NC2(CO)CCCC2)=O)CCN(C(=O)CS(N)(=O)=O)CC12CC2 59870,c1(CC)nc(C)c(NC(=O)NC(c2ccccc2)(C)CNC(=O)OC(C)(C)C)s1 59871,C=C(C)CCC(=O)NC(C1CCN(C(=O)C(C)NCC(F)(F)F)CC1)(C)C 59872,N1(C(C(C)OC)=O)CCC2CN(C(C3(O)CCC3)=O)CC2C1 59873,c1(C2(C(N3CC(C(C)NC(CCOCC#C)=O)C3)=O)CCCC2)cccc(Cl)c1 59874,C=C(C)C(CC(=O)NCCC(C(N1CC2C(C1)C2(C)C)=O)N(C)C)OOCC 59875,C1(C(=O)NCCc2cn[nH]c2)CN(C(C2CSC2)=O)CC12CCC2 59876,C1(NC(C2C=CCC2)=O)CC2(C1)CC2C(=O)Nc1ccc(Cl)cc1 59877,c1(CC)cc(C(=O)NCC2C=CC(NC(c3ccn(COC)n3)=O)C2)c(C)o1 59878,CC12CSCC1CN(C(=O)NCc1ccc(F)c(-c3nn[nH]n3)c1)C2 59879,c1(C(=O)NCCC2CCCN(C(CC3(C)CCCC3)=O)C2)ccc2ccsc2c1 59880,c1(C(=O)OCC)nnc2n1CCN(C(C=C(C)C)C(=O)NC1CCC1)C2 59881,C1(C)(C(=O)NC(CC(C)NC(=O)Cc2ccc(Cl)c(Cl)c2)C)CCS(=O)(=O)CC1 59882,c1(C(=O)NCCC#N)ncccc1NC(=O)Cc1ccc(SCCO)cc1 59883,c1(OC)cccc(C2(O)CN(C(C3CC(c4cccc(OC)c4)CC3)=O)C2)c1 59884,C1(N(CCNC(C2N(CC)CCC2)=O)C(=O)N(C)C)CCCCCC1 59885,C12(CNC(C3CCCO3)=O)CCCC1N(C(c1cc3sccc3s1)=O)CCC2 59886,C1(NC(c2cn(C3CC3)nn2)=O)C2CN(C(=O)CC3(OCC)CCCCC3)CC12 59887,C(C)(C)(C(C)CC(=O)NCC1(O)CCOCC1)NC(Cc1cn(CC)nc1)=O 59888,C(C(C)(CO)NC(=O)CC=CC(C)(C)C)N(C)C(c1csc(CCP(C)(C)=O)n1)=O 59889,C(=O)(C(C)(C)CN1CCOCC1)NCCC1CCN(C(C2C(C)C2C)=O)C1 59890,C12(C(=O)NC(CC(=O)NC)C3CC3)CC1CN(C(=O)CCc1cn(C)nn1)C2 59891,N1(C(CC=C)=O)CCN(C(=O)C(C)C(=O)C2CCCC2)C(CS(C)(=O)=O)C1 59892,C(=O)(C(F)C(C)CNC(=O)Nc1cn(CC)nn1)OCC 59893,C1(C)(C(N2C(C(=O)NCC(C3CCOCC3)C)CC2)=O)CC1(F)F 59894,c1(NC(N(CC(c2ccccc2)(C)F)C)=O)ncnc(F)c1F 59895,c1(C(=O)NC(CC)CNC(c2cc(Cl)n(C)n2)=O)c(O)nnc2c1CCC2 59896,c1(C(=O)NC2C(NC(c3ccc(C(N)=O)cc3)=O)C2)cccn2ccnc12 59897,Cc1cc(O)ccc1C(N1CCC(N(C(=O)CSc2ccccc2O)C)CC1)=O 59898,C1(NC(C(C)OC)=O)CN(C(=O)CCS(=O)(=O)N(C)C)C(C)(C)C1 59899,C(=O)(CCCn1cc(CCC(N)=O)nn1)NCC(=O)NC(C)(C)C 59900,C(CC)(CCC(=O)NCC(C)(C)N1CCCC1)NC(CCC=CC)=O 59901,C1(NC(c2cc(Cl)sc2Cl)=O)CCC2CN(c3nc(Cl)ncc3F)CC2C1 59902,C(C(CC(C)C)C(=O)NC1CC(CNC(C23CCC(N=[N+]=[N-])C2C3)=O)C1)OC 59903,CC(CC(=O)N(C(C)C(=O)NCCN)C)C(=O)OC(C)(C)C 59904,N1(C(C2=CCC(C)CC2)=O)CCC(N=c2cc(Cl)nc(C(=O)OC(C)(C)C)[nH]2)C1 59905,c1(C(=O)NCCCCC2CN(C(Cc3cc(C)ns3)=O)C2)cc2n(n1)CCCC2O 59906,CCCCC(C(=O)NCCCNS(C)(=O)=O)NC(c1cnn(C)c1)=O 59907,CCC(C)CCCC(=O)NCC1(CN(C(=O)COc2ccccc2Cl)C)CC1 59908,N1(C(CCC#C)=O)CC=C(C(C)(C)C(=O)N(C(C)COC)C)C1 59909,C(CC(N)=O)(CC(=O)N=c1ccn(C2CC2)[nH]1)NC(CC1C(C)CCO1)=O 59910,C1(CNC(c2c(CN(C)C)ccs2)=O)COCCN1C(=O)CC1CCC(C)(C)C1 59911,c1(C(=O)NC2CC(NC(c3c(C)cccn3)=O)C2)cnc2c(c1)OCC(=O)N2 59912,C(Cn1cccn1)(C(=O)N=c1cc(C(N)=O)n(C)[nH]1)NC(C(C1CCCC1)C)=O 59913,C(C(=O)NCCN(C)C(C1(C(O)C(C)C)CC1)=O)(C1CCCC1)OCC 59914,CC(C)CC(C(=O)NCC1CCOC1(C)C)NC(=O)CCC(F)(F)F 59915,CC1(C)OC(=O)CC1C(N1CC(C(O)C(=O)NCCC2NC(=O)NC2=O)C1)=O 59916,C1(CCCC)CN(C(c2c[nH]cc(C)c2=O)=O)CCN1C(C1CC1C1CCC1)=O 59917,N1(C(c2cnc(C)s2)=O)CCC(C2CC2)C1CNC(C1CCC1(C)C)=O 59918,C(C(C)(C)C(=O)NC1CCC(C(=O)NCC2CC2(C)C)C1)N(C)C 59919,C1(C2CC2)(C(N(CCCNC(c2c(C)nc(CC)s2)=O)C(C)C)=O)CC=CC1 59920,c1(CC(N2CCC(NC(C(COC)C)=O)C23CC3)=O)cnc2n1CCOC2 59921,CC1C(C(N2CCC(c3ccco3)C2)=O)CCN1C(C1CC12CCC2)=O 59922,C(=O)(CCCC(C)(C)C#N)N1C(C(=O)NC(CC)C2CC2)C(CC)CC1 59923,c1(SCC(=O)NCCCC2(N(C(CSCC)=O)C)CC2)ccccc1Cl 59924,O=C(C1CCSc2ccccc21)NC1CCC(NC(C2CCS(=O)CC2)=O)CC1 59925,c1(C(N(C2CC(NC(c3cncc4sccc34)=O)C2)C)=O)n[nH]c2c1NCCC2 59926,N1(C(CCC(C)C#N)=O)CC2(C1)OC1(C)CC2(NC(c2c(Cl)cnn2C)=O)C1 59927,CC1(C(=O)NCCCN(C(=O)Cn2ccnn2)CCO)CCCS1(=O)=O 59928,Cc1cnc2nc(C(=O)N(CC(C)(C)CNC(=O)C=CC3CCCO3)C)nn2c1 59929,N1(C(c2cn(C3CC3)cn2)=O)CC2CC2(C(=O)NCCN(C)C)C1.C(=O)C1CC1 59930,C1(C)(CC)C=C(C(=O)NCC(C)CC(=O)N2CCC(CSC)CC2)C1 59931,N1(C(C(C)(C)CF)=O)CCC2(CCCCN(C(=O)C(F)(F)C(C)(C)O)C2)C1 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59949,CC1CN(C(C2(NS(=O)(=O)C3CC3)CC2)=O)CCC1NC(c1cc(Cl)no1)=O 59950,C1(C)(OC)CCC(NC(C2CN(C(C3CCC3C)=O)CC2(F)F)=O)CC1 59951,c1(C(N(C2CCC(NC(=O)CCSC3CCCCC3)C2)C)=O)ccn2nccc2n1 59952,c1(SC)c(NC(=O)C(C2(C)CC2)NC(=O)CN2CCNC2=O)cnn1C 59953,C1(F)(C(N(CCN(C(C(C)SCC)=O)C(C)C)C)=O)CCOC1 59954,N1(C(C(CCC)CNC(=O)C2=CCCC2C)=O)CC2(CCC(=O)N2)C1 59955,c1(CC(C)C(=O)NC2CC2NC(C2(CO)CC2)=O)cccc(Cl)c1 59956,C1(C(c2n(CCC)nnn2)NC(C(=O)NC)C2CC2)CCC(C)(C)CC1 59957,C1(CN(C)C(C23CC(F)C2C3)=O)CCCN(C(c2cnccc2Br)=O)C1 59958,C1(NC(C(C(CC)C)N(C(=O)Cn2nnc(C)n2)C)=O)CC2CCC(C1)C2O 59959,C(=O)(C1=CS(=O)CCC1)NC12CC(CNC(c3ccc4ccoc4c3)=O)(OC1)C2 59960,C1(CNC(c2cc(CF)on2)=O)CN(C(C2(O)CCSCC2)=O)CC12CCC2 59961,C1(CNC(=O)C2=CCCS2)CCCCN(C(c2cc(Cl)cc(C(F)(F)F)n2)=O)C1 59962,C1(CSC)CN(C(=O)OC(C)(C)C)CC(C(F)(F)F)O1.C1C(C)N1 59963,c1(C(=O)NC2CC(C(C(=O)NCCCCSC)F)C2)nocc1Cl 59964,c1(C(=O)NC(C)CCN(C)C)n[nH]cc1-c1ccccc1 59965,c1(CNC(c2cccnn2)(C)CO)csc(SC(F)(F)F)n1 59966,c1(C(=O)NCC2(F)CC(CNC(C(C)=C3CC3)=O)C2)ccc(C2CC2)nc1 59967,C1(NC(=O)COCCCF)CN(C(=O)CCCn2cncn2)C2(CCC2)C1 59968,N1(C(c2ccc(C)s2)=O)CC=C(C(=O)NC2CN(C(N)=O)C2)CC1 59969,C(=O)(C(C)CCCCCC)NC(C(N1C(C)(CCC)CC1)=O)COC 59970,C1(CNC(c2c(SC)cccc2)=O)CCCN(C(=O)Cn2nc(C)cc2C)CC1 59971,c1(C(N(CC(C)O)CCNC(C2C(OC)CC2)=O)=O)cocc1C 59972,C1(C(=O)NCC(CC(C)C)NC(C2CC=CCO2)=O)CCc2ccccc2NC1=O 59973,N#Cc1c[nH]c(=NC(=O)c2nccc3c(Br)cccc23)cc1F 59974,N1(CC(=O)NC(C(C)C)CNC(=O)CCc2cnoc2)CCCCC(O)C1=O 59975,C(=O)(CC(C)(C)CC(F)F)NC1(CO)CN(C(Cc2ccc(C)s2)=O)C1 59976,c1(OC)ccc(C(=O)NC2CC(NC(c3cnc(O)s3)=O)C(O)C2)c(N)c1 59977,C#CC1CCC(C(N2CCCC(N(C)C(c3cccc(F)c3OC)=O)C2)=O)CC1 59978,c1(CCn2ncc(C(c3c(C)cccc3)NC(N)=O)c2)c[nH]c2cc(F)ccc12 59979,n12cc(nn1)CNC(=O)C2.C1(C(NOCCC#C)=O)CCCN1C1CCC1 59980,S(=O)(=O)(c1cccc(Cl)c1)NC1(CCC=C)CC1.C12(C)CCN(C1)C(=O)CCN2 59981,CC(C)C(C(=O)N1CCCC(CC(=O)NCc2ncccn2)C1)N(C)C 59982,n1(C(C)C(N2CCC(n3cc(CC4CCC4)nn3)CC2)=O)ncc2ccccc12 59983,c12ccc(c(I)c1)[nH]c2=O.C1(C)(C(=O)OC)C=CCN1C(C)=O 59984,C(=O)(CC1=CCOCC1)NC1C(CNC(CCOc2cc(C)cc(C)c2)=O)CC1 59985,c1(OC)ccc2c(=NC3CC3)[nH]c(=NCC(C)N3CCN(C)CC3)[nH]c2c1 59986,C1(C(N2CCC(N(C(=O)CC3CC=CC3)C)C2)=O)CCC(=O)N(C2CC2)C1 59987,Cc1cccc(N(C(=O)C(N2CC(C(N3CCOCC3)=O)CC2C)=O)C(C)C)c1 59988,CC(C)(CC#N)C(=O)N1CC(=O)CC1C(=O)NC1COC2(CCC2)C1 59989,c1(C(=O)NC2(CC(N)=O)CN(C(C(=O)NC(C)C)=O)C2)ccc(C2CCC2)nc1 59990,C1(C(=O)NCC(C)N(C)C(C2(CC(F)F)CCC2)=O)CC2(CC(=O)C2)C1 59991,CCCCCCC(F)C(=O)N(C1CN(C(=O)CCC2CC2(F)F)C1)C 59992,CC(CO)C(C)N=c1nc(N2CCN(CCCC#N)CC2)c2c([nH]1)COC2 59993,CC1(F)CC2(CN(C(=O)C(CNC(=O)CSC(C)(C)C)CC3CCCC3)C2)C1 59994,C1(n2cnnn2)(C(=O)NC(C)CCCNC(=O)C(F)OC(F)(F)F)CCCCC1 59995,C1(NC(C(=O)NCCOCCOC)=O)CC2(CCNC2)CO1 59996,C1(F)(Cn2cc(C(C)(C)NC(c3cccc(C(=O)O)c3)=O)nn2)CC2C=CC1C2 59997,Cc1cc(N(C2CCN(C(c3ccsc3Cl)=O)CC2)C)nc(C)c1C#N 59998,C12(NC(CN3CC(C)(C)C3)=O)CCC(CC1NC(=O)C=C(Cl)Cl)C2 59999,C1(N(C(=O)CCF)CC)CCCN(C(=O)CSc2nnc(S)s2)C1 60000,c1(C(N2CC(C#N)C(NC(c3cc(Cl)cnc3F)=O)C2)=O)c(F)ccc(I)c1F 60001,C(CCCOC)(C(=O)NCC(C)(C)C(F)F)NC(C(C1CC1)OCC)=O 60002,CCCC(C)(C)CNC(=O)CC1CC1CNC(=O)CCc1ccc[nH]1 60003,C(CCCNC(C1(C2CCCO2)CCC1)=O)NC(=O)Cc1ccon1 60004,c1(CN2Cc3c(C(N4CCC(C)C4)=O)n[nH]c3CC2)ccc(S(C)(=O)=O)cc1Cl 60005,c1(C(=O)NC2CCCN(C(N(C)Cc3ccc(N(C)C)nc3)=O)C2)ccc(O)cc1 60006,c1(C(C(=O)NCC=C)N2CCC2c2ccc(Cl)cc2)n[nH]c2cc(Br)ccc12 60007,n1(C(=O)OC)cc(NCCCNC(c2cc(Cl)ccc2OC(F)F)=O)ccc1=O 60008,CC1(C)CC(C(=O)NCC(C)(O)CNC(C2CCS(=O)CC2)=O)CNC1=O 60009,S1(=O)(=O)c2cn(C(C)C)nc2C(=O)N1CCOC.CCCCNC(C)=O 60010,N#Cc1ccc2c(c1)CC(NC(=O)CC1CNCC1O)C2 60011,C#CCC(C)C(=O)NC1CCN(C(c2n[nH]c(C)c2C(F)(F)F)=O)C1 60012,c1(C(N2CC3C(CNC(c4c(C)n[nH]c4)=O)(C3)C2)=O)cnc2snc(C)c2c1 60013,N1(C(CSCC#C)=O)CC(CNC(C2CCCN2C(=O)NC)=O)CC1(C)C 60014,N1(C(CN(C)C(C2CCSC2)=O)=O)CCCC2CN(C(=O)CC3(N(C)C)CC3)CC12 60015,C1(OC)CCCCC(=O)O1.c1(CC(=O)N(C)CCO)cccnc1Br 60016,c1(OCC)cc(C(=O)NCCC(C)N(C)C(c2cc(C)[nH]n2)=O)cc(Cl)c1OC 60017,CCCC(F)C(=O)NCC1CCCC1C(=O)N(CC(O)COCC)C 60018,c1(CCC(=O)N(C(C)C(=O)NCCN(C(C)CC)C)CCC)nccn1C 60019,O=C1CC2OCCC2(C(N2CCC3(CC(NC(=O)C(O)C(F)(F)F)C3)C2)=O)CN1 60020,c1(CC(=O)NC(C(CO)NC(CC(=C=C)C)=O)C)ccc(Br)c(C)c1 60021,C1(CC(=O)NC23CCN(CC2)CC3)CCN(C(C2C(C)(C(F)F)C2)=O)C1(C)C 60022,c1(OC)noc(C)c1C(=O)NCC1CC(F)CN1C(=O)C(c1ccccc1)OC 60023,N1(C(C(SC)SC)=O)CC2CC(NC(c3cccc(=O)o3)=O)CC(C2)C1 60024,C(=O)(C1CCCn2cncc21)N(C)CC1(CNC(C(CCCC)O)=O)CC1 60025,C1(C)(C(=O)NC(C2CCCN2C(=O)C(C)(C)C(F)F)C)CC(C(C)C)=NO1 60026,C(C)(CCCC(=O)NCC1SCCS1)NC(C1C(OC)CCCC1)=O 60027,N1(C(COC(C(C)Nc2ccc(Cl)cc2)=O)C)Cc2ccccc2C1=O 60028,CN1CCC(C(=O)NCC2(F)CCN(C(c3ncncc3Cl)=O)CC2)S1(=O)=O 60029,CC1(C)COC(CC(N2CCCCC2C2(NC(=O)CNC(N)=O)CC2)=O)C1 60030,N1(C(CC2CCCN(C(C(CC=C)C(C)C)=O)CC2)=O)CCC2(CNC(=O)C2)C1 60031,C1(C(=O)NCC2C3N(C(Cc4nnc(C)s4)=O)C(CC3)C2)CCc2ccnn2C1 60032,C1(NC(c2cc(OC)n[nH]2)=O)C2CC1CN(C(=O)CCc1csc(=N)[nH]1)C2 60033,C12(CNC(c3c(C)cc[nH]3)=O)CC(NC(=O)C(C)C(F)(F)F)(C1)C1(CCOCC1)O2 60034,c1(C(N(CCNC(C2CCC2OC(C)(C)C)=O)CC)=O)cc(C2CC2)n(C)n1 60035,c1(C(N2CCC(CN(C)C(C3(O)CC(F)(F)C3)=O)C2)=O)cnc2[nH]nnc2c1 60036,CCC(CNC(=O)CCP(C)(C)=O)(CC)C(=O)NC1CCC1(C)C 60037,C1(N(C(=O)Cc2ccsc2)C)CN(C(c2ccc(CO)o2)=O)CC12CC2 60038,N1(C(CC2(OC)CCCC2)=O)CCC(C2(NC(=O)CCC(C)SC)CC2)CC1 60039,N1(CCCNC(C(CC)O)=O)CCN(C(=O)CSC2CCCCO2)CC1=O 60040,N1(C(CC2OCCN(C(COC(CC)CC)=O)C2)=O)CCOC(C2CC2)(CC)C1 60041,C(=O)(C(CN(C)C)C(C)C)NCc1c(C(=O)NC(CCC)c2ccco2)occ1 60042,c1(C(=O)NCCC2C(C)CN(C(C3CCCC3)=O)C2)c(F)ccc2cnn(C)c12 60043,N1(C(=O)Nc2cc(OCC)c(Cl)cc2)CC2CC(C)N(C(=O)C3CC3)C2C1 60044,C#CC1(C(=O)NCCC(C)OC)CCN(C(c2cc(OC)no2)=O)C1 60045,C1(NC(c2cncc(Br)c2)=O)CC2(C1)CC(C(=O)NCc1cnco1)C2 60046,c1(C(=O)NCC(C)N(C(=O)CC2CCC(=O)NC2)CC)cc(C)cc(C)c1C 60047,N1(C(C2(CNC(C(CCC)C(C)C)=O)CCCO2)=O)CCc2nnnn2CC1 60048,C1(C(N2C(CNC(C(CC(C)C)(C)C)=O)C=CC2)=O)CCc2ccccc2CC1 60049,c1(NC(C2CNCCN2Cc2ncccc2[N+](=O)[O-])=O)cc(Cl)c(O)c(Cl)c1 60050,N1(C(C(C(CC)(C)C)=O)=O)CCC2(CC1)CC(NC(=O)C(F)CC1CC1)C2 60051,C(C(COC)CC(=O)N1CCC(CCC(=O)NC(C)CS(C)=O)C1)OC 60052,c1(C(=O)NCCOC2CC(NC(C=CC(C)(C)SC)=O)C2)cc(C#N)ccc1O 60053,c1(NC(C2CC(F)CN(Cc3cc(Br)ccc3I)C2)=O)cnc2ccc(F)cn12 60054,CCC(C(=O)OC)C(=O)N1CC(O)(CNC(=O)C=C(C)CCc2ccccc2)C1 60055,c1(CC)ccc(C(=O)NC(C)C(C)(C)NC(=O)COCC2CCCC2)[nH]1 60056,c1(C(=O)Nc2ccc(C)nc2)cc2c(nc1N)CCC2 60057,C1(C(=O)NC(C)CCN(C(=O)CCSC(F)(F)F)C)C2CC3C(C2=O)C13 60058,C1(CNC(c2scc(C)c2C)=O)CN(C)CCN1C(=O)C(C)OCCN(C)C 60059,N1(c2n(CC=C)c(-c3ccccc3F)nn2)CC2CC1CN2C(=O)C(C)O 60060,C(C)(C(=O)N(C)CCN(C(=O)CCN)S(C)(=O)=O)NC(=O)OC.C(C)C 60061,C1(NC(=O)NCc2n(C)c(Br)nn2)C2CC3CC1CC(O)(C3)C2 60062,c1(NS(C)(=O)=O)c(C(=O)NC2CCC2CNC(=O)C=NOC)cccc1Cl 60063,C#CC1(C(=O)NCC2CC(C(=O)N3CCS(=O)(=O)CC3)=NO2)CCCCC1 60064,C1(N(C(=O)C(O)CC2CC2)C)CCN(C(=O)C(C)(C)c2ccccn2)CC1 60065,c1(CC(=O)OCC)cnnc(NC(C2CC2CNC(=O)C=C(C)C2CC2)=O)c1 60066,c1(C(=O)NC(CCC)CNC(=O)C(N2CCCC2)C2CC2)cn(C(C)(C)C)nc1C 60067,C1(C(=O)NCCCCCn2cc(CCC3CCCCO3)nn2)NC(=O)C2CCC12 60068,N1(C(C(N)=O)=O)Cc2[nH][nH]c(=NC(=O)c3ccc(-c4cccs4)o3)c2C1 60069,N1(C(C(C=C)(C)O)=O)CCC2(CC1)OCCC2NC(=O)C(C)CCOC 60070,N1(C(C=CCC)=O)CC2CC1CN(C(=O)Cc1cc(C)[nH]n1)C2 60071,N1(C(C(C)Cc2ccccc2)=O)CCC2CCC(C1)N2C(=O)CCC(F)F 60072,N1(C=O)CCC(C)(O)C(NC(C23CCC(OC)(CC2)C3)=O)C1.C1(C(=O)N)CC12CC2 60073,CCC(C)CCC(=O)NC1CC2C(NC(c3occc3C)=O)C2C1 60074,N1(C(C(CCCC)NC(N)=O)=O)CCN(C(=O)C=Cc2ccsc2)CCC1C 60075,Cc1cc(Cl)cc(C(=O)N(C)CCNC(c2ncc(Cl)cc2Cl)=O)c1N 60076,C(=O)(C(C)C(C)S(C)(=O)=O)NCC1(CNC(CCOCCC)=O)CCCC1 60077,Cc1nccnc1C(=O)NC1COCC1NC(C1CC(C)(C)CO1)=O 60078,C(C)(C(O)C(=O)NC1CCC1CNC(=O)C(C)(C)Oc1ccccc1)SC 60079,c1(NC(Cc2cccc(OC)c2OC)C)cc(Cl)c(Br)cc1F 60080,c1(OC)ncc(Br)cc1CN1CCCN(C(c2ccnn2CC(F)(F)F)=O)CC1 60081,N1(C(c2ncc(C)nc2)=O)CCC2(CC1)CC2(CO)CNC(c1cocn1)=O 60082,C1(C(=O)NC(c2nccs2)C)CCC(NCc2sccc2Cl)CC1 60083,C1(CC)C(C(N2CCCC2)=O)CCN1C(=O)Cn1cccnc1=O 60084,c1(OCCC)cccc(C(=O)NC(c2cnsn2)C)c1 60085,C12CCCN1C2.c1(CCC(=O)NCC2N(C(C(C)SCC)=O)CC2)ccccc1 60086,c1(C(=O)NC(C(C)NC(c2csc(CO)n2)=O)C)ccccc1Br 60087,C(CCC(C)(C)NC(c1nc(C)n(C)n1)=O)NC(CN(C(COC)=O)C)=O 60088,C(=O)(CC(C)(C)CC(F)F)N(C1CC2N(C(C(C=C)(C)O)=O)C(CC2)C1)C 60089,N1(C(C2C(C(=O)OC)C2)=O)CC(C)(C)OCC1CNC(c1cnc2cccnn12)=O 60090,C1(CCCNC(c2c(C)occ2)=O)CN(C(=O)CN2CCOC2=O)CCO1 60091,c1(C(F)(F)F)cc(CCN(c2cccnn2)C2CC2)ccc1Cl 60092,Cc1ncc(C(=O)N(C2CCN(C(C3C(C)C3C)=O)CC2)CCO)cn1 60093,C1(C(=O)NC2CCCN(C(=O)CC3COCCO3)C2)CC2(CCCO2)C1 60094,N1(c2nccc(OCCC)n2)CC2(CCC(NC(c3ccc(O)nc3)=O)CC2)C1 60095,N1(C(c2ccc(F)c(C)c2Cl)=O)CC2CCCC(NC(=O)CC(O)C3CC3)C2C1 60096,N1(C(c2c(C)ccs2)=O)CC2CCN(C(=O)C(c3ccc(Cl)cc3)O)CCC2C1 60097,CS(=O)(=O)c1cccc(-c2nc(-c3n[nH]cc3Cl)n(CCc3ccncc3)n2)c1 60098,C1(CNC(C(F)OC)=O)C2CC2CN1C(c1cncc(Cl)c1)=O 60099,c1(OC)ccc(O)c(NC(=O)CCC2CCCN2C(=O)CCCC(=O)N(C)C)c1 60100,C1(CC)C(C(=O)NC(c2cccnc2C)C)CCN1C(c1cc(OC)ncn1)=O 60101,c1(OC)cc(F)c(Br)cc1C(=O)NCC(O)CNC(=O)C=Cc1cnc[nH]1 60102,Cc1c(C(N2CC(O)(SCC(N3CC(C(N)=O)C3)=O)C2)=O)ccn1C 60103,N1(C(CCn2c(C)ncc2)=O)CC(C(N2CCN(C)CC2)=O)C(C2CC2)C1 60104,CC1CCN(CCC(=O)NC(C)(C)C2(C3CCCN3C(CC(C)(C)C)=O)CC2)CC1 60105,C=CCN=C(NCC(=C)Cl)NCc1csc(COCC)n1 60106,CC1CCN(C(c2scnc2C2CC2)=O)CC1CNC(=O)CC1(CO)CCCC1 60107,C(=O)(C1=C(C2CC2)N(CC(F)F)C(=S)NC1c1cn2ccsc2n1)OC 60108,c1(C(N(CCNC(C(C(CC)O)C)=O)CC)=O)cc2ccc(Cl)cc2[nH]1 60109,c1(C(N2CC(CNC(c3nc(C)oc3)=O)C(C)C2)=O)cccc2occc12 60110,N1(C(c2c(CC)cno2)=O)CC2CCC(NC(=O)Cn3nccn3)CC2C1 60111,C=CC1(CC(=O)NC2CCC(C(C)C)CC2)CN(C(C2CC2Cl)=O)C1 60112,C(N=c1nc2sccc2c(NCCOC(F)F)[nH]1)C1C(c2ccn(C)n2)CC1 60113,C1(CC(=O)NCC(N2CCCCCC2)=O)CC(O)CN1C(=O)C(O)CC1CCCC1 60114,C1(NC(CC2CC(=C)C2)=O)CCC(C(=O)NC2(COC)CC(F)C2)CC1 60115,Cc1c(C=CC(N2CCCCC2C2CCN(c3ncccn3)C2)=O)cnn1C 60116,c1(CN(C(CCN2CCCCC2)C(N)=O)C(C)C)ccc(Cl)c(F)c1 60117,c1(COC)[nH]nc(C(N2CCCC(c3n[nH]c(C4CC4)n3)C2)=O)c1[N+](=O)[O-] 60118,C(CCN(C)OC)NC(CCC1CC(NC(CCCOC)=O)C1)=O 60119,CN1CCN(C(c2c(F)ccnc2F)=O)CC1CNC(C1(NC2CC2)CCC1)=O 60120,c1(C(N2CCC(NC(CNC(CC(C)C)=O)=O)C2)=O)ccc(C(C)O)cc1 60121,c1(CNC(CCCC#CC)=O)ccc2c(c1)CN(C(c1cccc(Cl)c1C)=O)C2 60122,C1(C)(C(N(CC)Cc2cncn2C)=O)CC(O)CN1C(=O)CC1CCCC2CC12 60123,CCC(Cc1ccccc1)CC(=O)NC(CNC(=O)CC1(O)CCOCC1)CC 60124,C1(C(C2CC2)NCC(CNC(c2csc(-c3cccnc3)n2)=O)O)SCCCS1 60125,C1(=O)CC(C)(C)CO1.C1(OC(C2CCCCO2)C)CCCC1CN=[N+]=[N-] 60126,c1(CNC(C2(CNC(C3C(C(=O)OCC)C3)=O)CCCO2)=O)cc(Cl)ccc1C 60127,C(CNC(=O)COc1ccc(F)c(C(F)(F)F)c1)(CC(F)(F)F)NC(C=CC)=O 60128,N1(C(C2OCC3CCCC23)=O)CCC2(CCN(C(c3cc(Br)n[nH]3)=O)C2)C1 60129,C(=O)(C1CCCc2sccc21)NCC(C)NC(c1cn(C(C)C)nc1C1CC1)=O 60130,c1(C(=O)NCCN(CCO)CC)ccc(C(=O)NC)cc1 60131,Cc1c(C(N2CC=CC2(C)C(=O)NOC(C)C)=O)cccc1C#N 60132,C1(NC(CSC)=O)CC2(CCN(c3ccc([N+](=O)[O-])c(SC)c3)CC2)C1 60133,C=CCCCC(C(=O)NCC(CC)(CC)CO)NC(C1CCC1C(=O)OC)=O 60134,C(C(C)(C)CNC(=O)CC(C)C1CCCC1)N(C(CSCC#C)=O)CCOC 60135,N1(C(c2cc(C)sn2)=O)CC(C(=O)NCC2(C)CC=CCC2)C2(CC2)C1 60136,C12(NC(CCCC)=O)CCCC1CN(C(c1ccc3c(c1)OCO3)=O)C2 60137,c1(CNC(C(c2cnc(C(C)C)s2)N(CC(CCC)C)C)=O)ccc(F)cc1 60138,N1(C(C(c2ccc(CC)[nH]2)=O)=O)CC(NC(=O)Cn2nc(C)cc2C)CC(O)C1 60139,c1(C(N(C(CNC(CC2C(C)=NNC2=O)=O)C)C)=O)ccc2c(c1)CCC2(C)C 60140,N1(C(C2CN(OC)C(=O)C2)=O)CCC2(CC1)OCCC2NC(c1ccc(F)s1)=O 60141,c1(C(=O)NC(CNC(C2CC3CCC2O3)=O)CO)cccc2c1CCO2 60142,c1(C(N(C(CCNC(CC2(C=C)CCCCC2)=O)C)C)=O)coc(S(N)(=O)=O)c1 60143,C1(CC)CCCCCCN1C(C1CCCC(NC(C2CC(=O)NC(C)C2)=O)CC1)=O 60144,c1(C(=O)NCC(C(C)C)NC(C(C=C=C)C)=O)nn(C)c2c1C(=O)CCC2 60145,c1(CNC(C2CC(F)CN(C(c3ccc(I)c(Cl)c3)=O)C2)=O)cccc(F)c1Cl 60146,C(C(=O)N1CCCC(C(=O)NCCOCCN(C)C)C1)(C(C)C)OC 60147,CC(C)CCC(=O)NCC(=O)NC1CCC(NC(c2nc(C3CC3)cs2)=O)C1 60148,CC1(CNC(=O)CCC(N)=O)CCN(C(=O)C(c2ccccc2)O)C1 60149,c1(C(=O)NCC(CNC(C2CCCC(=O)N2)=O)OC)cnc2n1CCCC2 60150,n1(CC)nc(C(=O)NC2CCN(C(=O)Cn3cc(C(=O)NC)nn3)C2C)c(C)n1 60151,Cc1nc(C(=O)NCC2CC2NC(c2cc(C(C)C)[nH]n2)=O)c(=O)[nH]c1C 60152,C(=O)(CS(C)(=O)=O)OC(C1C(NC(C(C)NC(C)(C)C)=O)CCC1)=O 60153,N1(C(C(C)(C2CCC2)NC(=O)Cc2ccsc2)=O)CC2CC(O)CC2C1 60154,CN1N=C(CC(=O)NC2(C)CCN(Cc3ccncc3Cl)C2)CC1=O 60155,c12ccc(s1)C(=O)NCC2.C1(c2c(C(=O)OC(C)=O)cco2)(NC)CCOC1 60156,C1(C(=O)NCC2N(C(C(COC)(F)F)=O)CC(O)C2)CC2(CCC2OC(C)=O)C1 60157,C1(NC(c2[nH]cc(CC)n2)=O)CCCN(C(c2cc[nH]c2C2CCC2)=O)C1C 60158,CCCC(C)C(C)NCC1CC1C(=O)OC(C)(C)C 60159,C1(NC(C(CCC)CNC(=O)C(CC)NC(N)=O)=O)C2CCCCCCC12 60160,Nc1cnc(C(=O)NCc2cc[nH]c2C(=O)NCC2CCC(CO)O2)cn1 60161,c1(C2N(CCc3cc(F)cc(F)c3)CCC2)ccc2[nH]ccc2c1 60162,c1(C(N2CC(OCCNC(c3cc(CCC)n(C)n3)=O)C2)=O)cnc(N)c(Cl)c1 60163,C1(OC)(CNC(=O)NCC2CN(Cc3ccccc3OC)CCO2)CCOCC1 60164,c1(C(C(=O)NCCC(=C)CNC(c2ccnc(OC)c2)=O)O)ccc(Cl)c(Cl)c1 60165,C(=O)(CCN(C(=O)C(C)NC(=O)CCOCC)C)OCC 60166,N1(C(C(c2cccc(C(N)=O)c2)C)=O)CC(NC(C2CCCN2C=O)=O)CC1(C)C 60167,C(=O)(CC(C(F)(F)F)c1ccco1)NC(CN(C(=O)CCc1cnnn1C)CC)C 60168,C=CCC(CNC(c1ccncc1Cl)=O)C(=O)N1CCC(C(F)F)CC1 60169,c12ncc(c(C)n1)C(=O)OC1CC(C1)C2.N1(C(C(=O)OC)C)CCNC1=N 60170,Cc1cn2c(n1)C(C(=O)N1CCC(C(C)NC(=O)C(=O)C(C)(C)C)CC1)CCC2 60171,c1(NCc2cnn(CCO)c2)cc(C(=O)NC(c2n(C)ccn2)CO)n(C)c1 60172,c1(C(=O)NCCN(C(C(C)NS(C)(=O)=O)=O)C2CC2)cnn2ccncc12 60173,c1(CS(N)(=O)=O)cccc(C(=O)NCC2(F)CC(NC(c3csnc3Cl)=O)C2)c1 60174,C(c1ccsc1)=CC(=O)NCC1CC1C(=O)NCC1CC(=C2CCC2)C1 60175,CC=C=CCCN=c1nc(SC)c2ncccc2[nH]1.CCCC(C)O 60176,c1(C(=O)NC2C(CNC(C3CC(=C)C3)=O)C2)cc2c(N(C)C)cccc2s1 60177,c1(CNC(c2c(C)nc(-c3ccccc3F)s2)=O)nc2ccsc2s1 60178,N1(C(c2c(CC)[nH]cc2)=O)CCCC(O)(CNC(C2(CO)CCOCC2)=O)CC1 60179,c1(NC(c2cnc(OCC)s2)=O)ccc2ccccc2c1O 60180,c1(C(N2CC(N(C)C(C3CC3F)=O)C2)=O)nc(OCC(F)(F)F)ccc1Cl 60181,C1(C(N2C(CC(=O)NC3(CF)CCC3)CCC2)=O)CCCC12CCC2 60182,c1(C(=O)NC2CCC(NC(Cn3c(C)c(Cl)cn3)=O)CC2)cc(O)cc(Cl)c1Cl 60183,N#CC1(C(=O)NCCC2CC(C(=O)N(C3CC3)Cc3ccoc3)C2)CCC1 60184,c1(NC(c2nnnn2CCCF)C(C2CCCCC2)C)ccc(S(N)(=O)=O)c(F)c1 60185,CS(=O)(=O)CCCNC(C1(NC(c2cc(N3CCCC3)ccn2)=O)CCC1)=O 60186,N1(C(c2cc(C)sc2C)=O)CC(F)(F)CC1C(=O)NC1(C)CCCC1(C)C 60187,C1(CC(=O)NCC(C)(C2CC2)NC(C(C)C2(O)CCC2)=O)CCC=CCC1 60188,c1(N(C)CC2CCCCO2)nc(=NC2CCCC(O)C2)[nH]c2c1COCC2 60189,c1(C(N(C2CCN(C(=O)C(O)C(C)OC)C2)CCC)=O)cn2nccc2nc1C 60190,N1(C(C2(COCC)CC2)=O)CCC2(CC1)C(NC(=O)CCS(C)=O)CS2(=O)=O 60191,C1(NC(c2ccc(N(C)C)cc2)=O)CC2CCC(C1)N2CCCc1ccccc1 60192,c1(C(N2CC=C(COC)CC2)=O)cn2nc(NC(CC(=C=C)C)=O)ccc2n1 60193,N1(C(CC=C)=O)CCC(NC(c2ccc(C3CC(F)(F)C3)cc2)=O)C(CO)CC1 60194,S(=O)(=O)(c1ccc(Br)cc1NCC1(C(C)(F)F)CC1)NCCCn1c(C)ncc1 60195,CC(C)(C)C(=O)C(=O)NCC1CCC(CC(=O)NCCCCCCF)CC1 60196,C1(C(=O)OCC)(NC(C2OCCC2C(C)C)=O)CC(O)C1(C)C 60197,C1(CCNC(C2(C)CC(F)C2)=O)CCCN(CC(=O)N)C1.c1(CN)ccccc1 60198,c1(CNC2(CC(=O)Nc3ccc(C)cc3O)CCC2)ccc2ccn(C)c2c1 60199,C1(NC(c2ccc(OC)c(F)c2)C)CNC2CCOCC2C1 60200,c1(COC)ncc(C(N2CCC(C(C)NC(=O)CC3CC=CCC3)C2)=O)s1 60201,N1(C(C(C)O)=O)CCc2[nH]nc(CNC(=O)CCC3CCOC3)c2C1 60202,S(=O)(=O)(c1csc(Cl)c1)Nc1cc(C(N(c2ccccc2Cl)CC)=O)c(C)o1 60203,C(=O)(CCC(C)C)NCC(CCOC)NC(=O)CN1CSCC1=O 60204,CC(C)C(CCC(=O)N1CC2CC3CC2C1C3)NC(c1nnn(C)c1N)=O 60205,C(CS(=O)(=O)CC(=O)N1CCC1CNC(=O)CCCC(C)(C)C#N)OC 60206,CC1(C(F)(F)F)CCCN1N1CCCC2(CCCNC2=O)C1 60207,N1(C(C(C)(C)C)=O)CC2CC(CNC(c3cc(C(C)(C)O)ccn3)=O)C2C1 60208,C12(C(N(CCC(=O)OC)C)=O)CCC(CC1)N(C(c1ccncc1N)=O)C2 60209,C(CC(=O)NC1CC(CCNC(=O)C(O)c2ccsc2)C1)N(CC#C)C 60210,CC(C(=O)NCCOCCNC(=O)COC1CC=CC1)c1ccsc1 60211,N1(C(C(C=C)NC(C)=O)=O)CC(C2CCCN(C(C3CC3(C)C)=O)C2)C1 60212,C1(SCCOC(C)C)CCC(C)(C)CC1 60213,c1(CC)cc(C(N2CCC(NC(=O)CCc3nc(O)n[nH]3)CC2C)=O)cc(C)c1 60214,C1(CN(C(=O)CN2CCCC2CO)C)CCCN(C(c2cccc(O)c2)=O)C1 60215,N1(C(CC(C)NC(C2CC3(CCO2)CC3)=O)=O)CC2(C1)CC(C)(O)C2 60216,c1(CCC(=O)NCC2COCCN2C(=O)Cc2ccccc2Cl)cccc(F)c1Cl 60217,n1(CC(=O)NCC2(F)CCCN(C(c3c(C)nns3)=O)C2)ccc2ccccc12 60218,CC1(NC(C2C=CCN2C(=O)CC2CC3CC3C2)=O)CC(F)C1 60219,N1(C(C2C(C)(C(C)C)C2)=O)CCOC(CNC(=O)CCCCN2CCOCC2)C1 60220,C(=O)(CC(C)n1ccc(C)n1)C1(CNC(COCCOCC)=O)CC1.C(C)S 60221,N1(C(C(=O)NC2CCC(CC)CC2)=O)CCC(Cc2ccc(C)cc2F)C(C)C1 60222,c1(OC)csc(C(=O)NC(C)CC(C)NC(=O)CC2(OC)CCCC2)c1 60223,c1(NC(C(=O)NCCC2CCCC(C)C2)=O)cc[nH]c2nccc1-2 60224,C1(C(N(Cc2c(C)nc[nH]2)CC2CCC2)=O)CCCC(=O)N1C.C12CN(C1)C2 60225,c1(-n2cc(CN(C(c3c(CC4CC4)cccc3)C)C)nn2)ccc2c[nH]nc2n1 60226,N1(C(c2nc(N(C)C)oc2)=O)CCOC2(CCN(C(C3CCCC(F)C3)=O)C2)C1 60227,Cc1c(C(=O)NC(CC(C)C)C(=O)NCC(C)(C)N(C)C)cccc1F 60228,c1(C(=O)NCC2N(C(CC(C(C)C)O)=O)CCCC2)ccn2ccnc2c1 60229,C1(NC(C2CC(C(=O)OCC)C2)=O)CC(=O)N(C2CC2)C1.C1C(O)C(=O)N1 60230,c1(C(=O)NCCN(C(c2cn(C)nc2-c2cccnc2)=O)CC)ccccc1F 60231,c1(C(=O)NCCC(C)NC(C(C(C)C)C#N)=O)c(C)oc2ncnc(O)c12 60232,C1(NC(C=CC(C)(C)NC(C)=O)=O)C2CC(NC(C3CCN(C)C3C)=O)CC12 60233,c1(COC(c2cccc(Cl)c2)CNS(C)(=O)=O)cc(Cl)c([N+](=O)[O-])[nH]1 60234,C(=O)(C1CC(=O)Nc2ncccc21)NC(C)(C)CCCNC(c1ccc(F)o1)=O 60235,c1(NC(CNC(C(CC)OC)=O)(C)C)cccc(C)c1.c12cncn1NC(=O)C2 60236,c1(C(N(CCCCCC)CCNC(=O)C(C)c2ccsn2)=O)ncc(N)cc1Cl 60237,c1(CNC(C(C(C)C)NC(C(CSC)O)=O)=O)cc(F)ccc1F 60238,C1(CNC(C2CCC(C)(C)C2)=O)CC(F)(F)CN1C(C1C2CCC(=O)C12)=O 60239,C(=O)(C(CNC(=O)CC1CCCN1C)N(C)C)N(CCN1CCCC1)CC 60240,C1(=O)C(CC(C)C)N(c2cc(C)co2)CC(=O)N1C.C1(N(CCC)C(C)C)CCCCCC1 60241,C1(C(=O)Nc2cccc(I)n2)C2CCCC1CN(C(c1ccc(O)cn1)=O)C2 60242,Cc1cc(C(=O)N(C)CCOCCNC(c2cnc(S)[nH]2)=O)c(C)c(C)c1 60243,c1(NC(=O)Nc2ccc(C#N)c(Cl)c2)cccc(C#CCO)c1 60244,C1(CC)CCN(N(C(CC2(NC(CN(CCC)C)=O)CCC2)=O)C2CC2)C1 60245,C1(C(=O)NCC(CN(C)C(c2ncccc2O)=O)(C)C)Cc2cccnc2C1 60246,CCC(CNC(=O)N(C(C)C)Cc1conc1C1CC1)CCl 60247,C1(C(=O)NCCN(C(CC2(C=C)CC2)=O)CCc2ccccc2)CN(C)CCO1 60248,CCCC(C(=O)OC)C(F)(F)C(=O)NCCC(O)CNC(c1coc(Cl)n1)=O 60249,CC(=O)CCCC(=O)N1CCN(C(=O)CC23COC(C(F)(F)F)(C2)C3)CC1C 60250,c1(C(=O)NC2CC(C)(CNC(C(CC=CC)C)=O)C2)ccc(F)c(C(=O)CC)c1 60251,N12CCCC(C1)C2.c1(CCC(=O)N(C(C)CC2CC2)C)ccccc1Cl 60252,c1(CNC(C2CN(C(N)=O)C2)=O)nocc1C(=O)N(CCF)C1CC1 60253,c1(SC)cccnc1C(=O)NC1CN(C(C2OCC2(C)C)=O)CC1SC 60254,c1(C(=O)NC2CN(C(c3c(Br)ccc(OCC)c3)=O)C2)c[nH]c2cccc(F)c12 60255,c1(C(N2C(CC(=O)OC)CC2)=O)cc(Br)ccc1C 60256,C1(CCCC)CN(C(c2n[nH]c(C)c2Br)=O)CCN1C(=O)CC(C)F 60257,C=C(F)C1(CC(N2CCC(CNC(=O)CSCC(=O)OC)(OC)C2)=O)CCC1 60258,S(=O)(=O)(c1ccc(F)cc1F)N(C1CC2CC1CN2)C(c1cc(C(C)C)no1)=O 60259,c1(CCOC)noc(CCC(=O)NC2CCN(C(=O)C(F)(F)C3CC3)C2)n1 60260,c1(C(=O)NC2CC(NC(Cc3nc(C)sc3)=O)C2)ncnc2sccc12 60261,C1(C(=O)NC2CCC(NC(c3cnn(-c4ccccc4)n3)=O)C2)CCC2(CCC2)C1 60262,CCC(C)C(C)(O)CNC(=O)CN(C(c1cnccc1C)=O)C(C)C 60263,CC(C)CCCC(=O)N(C1CCN(C(C2CCCCN2N=O)=O)C1)CC1CC1 60264,N1(C(C2(C)CCCN(C(c3n(COC)ncc3)=O)C2)=O)CCC2(CC=CCO2)C1 60265,c1(C(N(CC(C)(C)NC(C2=CCCC2C)=O)C)=O)cnc2ncnn2n1 60266,C(CN=c1c(C#N)c[nH]c2ccc(C)cc12)N(C(c1ccc(C)nc1)=O)C1CC1 60267,C(N=c1[nH]nc(C(F)F)s1)C1CC(NC(c2ccn(CC(C)C)n2)=O)C1 60268,c1(CNC(C2CCC(CC(CC)C(=O)OC)C2)=O)ccc2c(c1)CCN(C)C2 60269,c1(C(N2C(C)CC(NC(c3ccc(NC)cc3)=O)C2)=O)ccc(P(C)(C)=O)s1 60270,C1(CC)CN(Cc2ccsc2Br)CCN1Cc1ccccc1C(=O)O 60271,C1(C(=O)NCC(C2CC2)SC)CC2CN(C(=O)Cn3nnc(C)n3)CC2C1 60272,c12ccc(cc1)CC1(COC1)NC2=O.c1(NC(c2ccco2)=O)ccccc1 60273,CCCC(C)(C)CC(=O)NC(CCC(=O)N1CCC1C(N)=O)C(C)C 60274,C1(CC)(CNC(C2(NC(c3cc(OC)no3)=O)CC(O)C2)=O)CCOC1 60275,c1(CC)cc(C)nc(N2CCCC2CCCNC(C2(C3CC3)CCCO2)=O)n1 60276,Cc1ccc(C(=O)NC2(CS(N)(=O)=O)CC2)nc1C 60277,C(=O)(C(C)(CSC)NC(=O)C=Cc1ccoc1)NC(C#C)C 60278,C1(C(N2CC(c3onc(C)n3)C2)=O)CC(C)(C)CN1C(c1cnc(C)[nH]c1=N)=O.C1CC1 60279,C(C(C)(C)CNC(c1ncoc1C1CCC1)=O)N(C)C(c1coc(Br)n1)=O 60280,CC1C2CCCCC2CN1C(=O)CC(C(F)(F)F)NC(=O)CCC1CCC(=O)C1 60281,c1(CCCC(=O)NCC(C)N(CC2CC(OCC)C2)CC)ccc(F)cc1 60282,N1(C(Cc2ccc(C#C)cc2)=O)CCC2C(CCCN2C(c2cn(C)nn2)=O)C1 60283,C=CC1(C(=O)N(C)Cc2ncn(C)n2)CCN(C(=O)CCc2cccs2)C1 60284,CC1(C#CC(=O)NC2CC3CCC2N3C(c2cc(Cl)c(Cl)s2)=O)CC1 60285,C1(C(N(C2CCCC2)CCNC(=O)CCc2ccoc2)=O)CCC2CC12 60286,C1(NC(Cc2c(C)non2)=O)CN(C(C23CC2COC3(C)C)=O)C2(CCC2)C1 60287,c1(C(=O)NC(C2CCCN2C(=O)C(C)(C)C(=O)N(C)C)C)nccc(Cl)c1C 60288,C1(CCNC(COCC(=O)NC)=O)CCCN(C(c2cc(C)sc2C)=O)CC1 60289,C=CCC1CC(=O)N2CCC(CC2)COC(C)C(=O)N1.C1(SC)CC1 60290,C1(F)(CNC(C(CCC)(C)C)=O)CCCN(C(=O)CC2COC(=O)N2)CC1 60291,CC(CC(=O)NC(C1(O)CCCCC1)C(N1CC=CC(O)C1)=O)C(F)(F)F 60292,C(CCCCC(=O)NCC(C)(C)OCC(=O)NCC1CC(O)(C(C)C)C1)OC 60293,c1(OC)nc(C(=O)NCC2CCC(C)CN2C(=O)CC2CC(SC)C2)cc(O)n1 60294,C1(NC(C(C)(C)CF)=O)CCCC2CN(C(C3Cc4cccc(F)c4C3)=O)CC12 60295,CC1(C)CCCN(C(C2CCO2)=O)C1CNC(c1cnc2ccsc2c1)=O 60296,C1(NC(C(C=C=C)C)=O)CCCCN(C(c2cnc(OC)s2)=O)C1 60297,CC1(NC(=O)CC2CCCC23CC3)CCN(C(=O)Cn2nnc(=N)[nH]2)CC1 60298,CC#CCCCC(=O)N1CCC(C(=O)NCC(F)(F)C(F)F)(CC)CC1 60299,c1(OC)ccc(F)c(C(=O)NCCC(C)NC(C2CC(C)N(C)C2)=O)c1N 60300,C(C(C)C(C)C(=O)NCCN(C(=O)CNC(c1cccnc1)=O)C)OC.N1CC(OC)C1 60301,CC1CC(CC(=O)NO)CCO1.C1(=O)C(C)N1C 60302,C12(CNC(c3n(C)c(=O)ccc3)=O)CCC(CN(C(C3CCCC3CF)=O)C1)C2 60303,C1(CNC(c2cncc(OC)c2)=O)CCN(C(=O)CC(C)N(C)C)C12CCC2 60304,C1(NC(C2(OC)CCCCC2)=O)CC(C)CN(C(c2csc(=N)[nH]2)=O)C1 60305,C1(CCC)(NC(=O)CCc2cnoc2)CCN(C(c2ccc([N+](=O)[O-])s2)=O)CC1 60306,C1(OCC(=O)NCCC2(O)CCN(C(C(C(C)C)SC)=O)C2)CCC(F)(F)CC1 60307,N1(C(c2cn(CCC=C)nn2)=O)CCN(CCCNC(c2n[nH]cc2Cl)=O)CC1 60308,CCC(C)(C)CC(=O)N1CC(N2CC(NC(=O)CC(C)N3CCCC3=O)CC2=O)C1 60309,C#CC1CCN(C(C2COCCN2C(=O)C(C)=C2CCCC2)=O)CC1 60310,CC1(C(=O)NC2CN(C(c3cccc[n+]3[O-])=O)CC2CO)CCC(O)CC1 60311,c1(C(=O)Nc2nc(C)c(-c3ccccc3)s2)n[nH]c2cc(Br)ccc12 60312,c1(C(=O)NC2CC3CN(c4ncc(C#N)nc4)CC32)nnn2c1COCC2 60313,C12(C(=O)NC(COC)CC(=O)N3CC(c4ncc[nH]4)C3)CCC(C1)OC2C 60314,C1(C(N2CCC(C)C2)=O)(C(C)C)CCN(C(C2CC3CCC2O3)=O)C1 60315,C=Cc1cccc(-c2cccc(NC(=O)C(N3CCCC(C)CC3)C)c2)c1 60316,C1(CC)CN(C(c2c(Cl)cccc2I)=O)CCN1Cc1cc(C)cc(Br)c1 60317,c1(C(C(=O)NC(C(=O)OC)C)N(C(C)CCO)C)ccc(OC)c(Br)c1 60318,CCCCC(O)C(C)C(=O)N1CCC(CNC(c2ncccc2C)=O)(OC)CC1 60319,c1(C(N(CCC)CCNC(C2CC2C(C)(F)F)=O)=O)cnc(CC)nc1 60320,CC(CC(C)(C)C)C(=O)NCC(C)(CO)NC(=O)CCCn1cncn1 60321,c1(C(N2CC(F)(F)CC2CNC(=O)C(F)(F)C(O)C2CC2)=O)cccc(=S)n1O 60322,c1(OC)ccccc1NCC(N1CCCC(C(C)NC(=O)CCF)C1)=O 60323,Nc1cccnc1S(=O)(=O)NC1CC(=O)NC1c1ccccc1 60324,c1(C(N2CCCCCC(NC(c3nc(C)oc3)=O)C2)=O)cccc2c1OCCC2 60325,c1(C(=O)NC2C(C)CN(C(=O)CN3CCOCC3)C2)cc(N)c(Br)c(F)c1 60326,N1(C(C2CCCN(C)C2)=O)CC2CCC(C(=O)NC3C(OC)CCC3)(C2)C1 60327,C=C(C)C1OCCCC1C(N1CCC2(C1)CN(C(c1cc(O)n(CC)n1)=O)C2)=O 60328,C1(NC(C=C(C)c2ccsc2)=O)CCC2(CC1)CN(C(=O)C(C)S(C)(=O)=O)C2 60329,CN1CCNC(=O)C12CCCN(CC(c1cnc3ccc(Cl)nn13)=O)C2 60330,C1(OCC)CCN(C(=O)CNC(C2CC2c2ccc(C)o2)=O)CC1 60331,C(c1ccc(C)cc1)=CCC(N1CC2C(CNC(C(CCC)OC)=O)(C2)C1)=O 60332,CN1C(=O)CCC1CC(=O)N(C1CCN(C(=O)C=CC2CCC2)CC1)CC1CC1 60333,c1(C(N2C(C(N3CC(CC)N(C)CC3)=O)CNC(=O)C2)=O)ccc2[nH]ccc2n1 60334,C1(OC)CCC2(C(=O)N(CCCCC(=O)N(C)Cc3cnco3)C)CC12 60335,Cc1cc(Br)cnc1C(C(=O)NC1CCOC1)N(CC(C)OC(F)F)C 60336,C(CN=c1nc2c(ncn2C)c(NCC2CCN(C)C2=O)[nH]1)N(CC)CC 60337,c1(C(=O)NCC(CC(F)(F)F)NC(=O)C(O)C2CCC2)cc2ccc(F)cc2o1 60338,C1(NC(c2c(CC)nc[nH]2)=O)CC2(CCN(C(=O)C(C)CCCOC)C2)C1 60339,C(CCC(O)C(=O)N(C1CCOC(C)(C)C1)C)NC(C=CCN(C)CC)=O 60340,N1(C(CCCc2onc(C)n2)=O)CCC2(NC(c3ccncc3)=O)CC2C1 60341,N1(C(CCCCN(C)C)=O)CC2CCN(C(c3snc(Cl)c3Cl)=O)CC2C1 60342,Cc1cnc(C)c(C(=O)NCC(C)CNC(=O)C(C)Sc2ccc(F)cc2F)c1 60343,c1(C(=O)NC2C(NC(C(CC)(C)C#N)=O)CC2)cc2c(cc1F)OCC(=O)N2 60344,N1(C(C)=O)CCCC(C(=O)NC(C)(CNC(=O)C(O)CC2CC2)CO)C1 60345,c1(SC)cc(C)c(C(=O)NCC=CCNC(c2ncsc2C2CC2)=O)s1 60346,C(=O)(C(C)C(C)(C)C)N(C1(CC(=O)NC(C#C)C(C)OC)CC1)C 60347,c1(C(N2C(C3CCCN(C(C4CCC=CCC4)=O)C3)CCC2)=O)cc(Cl)cnc1O 60348,c1(OC)cnc(Cl)nc1N1CCCC(C(C)NC(c2cnn(C)c2C2CC2)=O)C1 60349,C1(NC(=O)Cc2cc[nH]n2)COC2CN(C(=O)C(C3CCOCC3)F)CC12 60350,c1(C(CC)C)nc(-c2ccc(CCOC(C)(C)C)nc2)nn1C1CSC1 60351,Cc1ncnc(C)c1C(=O)NCCCN(C(=O)C1=NOC(C(C)(C)C)C1)C 60352,C1(C(N2CCC(N(C(C3(C4CC4)CC=CC3)=O)CC)CC2)=O)(OC)CCS(=O)(=O)C1 60353,c1(-c2cn(C(c3ccccc3)CC)nn2)cc(OC(C)C)nc(Cl)c1 60354,N12CCC(C1C(C)C)C(=O)N(C)C1(CC1)CC2=O.O(C(F)F)OCC 60355,N1(C(C(CO)OC)=O)CCC(C2CCN(C=O)CC2)C1.c1(C2C(N)C2)ccccc1 60356,N1(C(C=CCOC)=O)CCCC2C1CCCN2C(c1ccoc1C(C)C)=O 60357,C1(C(=O)Nc2cccc(Cl)c2Br)CCC2(CCN(C(c3[nH]nnc3CO)=O)C2)O1 60358,C(C(C(=O)NC1CC(C)(NC(=O)C(O)CN2CCCC2)C1)N(C)C)OC 60359,c1(OC(C)C)cncc(C(=O)NC2CCCC2NC(=O)COc2nccs2)c1 60360,C1(NC(=O)CN2CC3CC3C2)CC2CN(C(=O)CNC(N)=O)CC12 60361,c1(OC)ccc(C=CC(=O)NCCCCCNC(=O)C(C)(C)C2CC2)cc1 60362,C(CC)(CC)(CCNC(=O)CCCCCn1cnnn1)NC(C(CC)SC)=O 60363,c1(C(=O)NC(CN(C(C2CCCN2C)=O)CC)C)c[nH]c2c(C#N)cccc12 60364,C12(NC(c3c(C)cccc3)=O)CCCC(CN(C(=O)C=CC3(C)CCOCC3)C1)C2 60365,CCC(C)(F)C(=O)NCC1CCC(NC(c2ccccc2NCC(N)=O)=O)C1 60366,C#CCC(CC(F)F)C(=O)NC1CC=C(C(=O)Nc2ccccc2C2CC2)C1 60367,C1(CC(=O)NCCCCC2C(=O)NC(=O)N2)C2CCCC2N1C(C1C=CCC1)=O 60368,c1(C(N(CCN(C(=O)C(O)C(C)C)CC)CC)=O)sc2cc(C)ccc2c1C 60369,Cc1ccc2[nH]c(C)c(CC(N3CCC(C)C(NC(=O)C(C)(C)F)C3)=O)c2c1 60370,N1(C(C)=O)CCC(C)(C(N2CC(O)(CNC(c3[nH]cnc3C#N)=O)C2)=O)C1 60371,c1(C(=O)NC2CN(C(C(CC=C)C(C)C)=O)C2)[nH]c2c(F)cc(F)cc2c1C 60372,CCC(C)C(O)C(C)C(=O)NCC1(C(N2CCC3OCCCC3C2)=O)CC1 60373,C1(NC(CCOCCSC)=O)CN(C(c2snc(C)c2N)=O)CC1O 60374,C1(C(=O)NCCNC(C2CC(C)(CC)C2)=O)CCC(=O)N(c2cnn(C)c2)C1 60375,C1(NC(C(C=C)CC)=O)CN(C(=O)CNC(=O)CCC)CC1C1CC1 60376,Cc1c(C(=O)NCC2CCCCC2NC(=O)COc2ccon2)cccc1O 60377,c1(CC(=O)NCCOCCn2cc(-c3ccc(C(F)(F)F)s3)nn2)cncnc1 60378,N1(C(C(C)NC(=O)NC)=O)CCN(C(C2CN(C)CCO2)=O)C2CCCC2C1 60379,N1(C(C(C)OCc2cccc(C)c2)=O)CC2CC(NC(=O)CC(C)C)C2C1 60380,N1(C(C(C)O)=O)CCC2CN(C(c3ccncc3N)=O)CC12 60381,c1(NCC(C)C)ccc(C(=O)NC(C)CNC(=O)C(c2ccccc2Cl)C)cc1 60382,C(C(COC)CC(=O)NCCCNC(c1sc(C)nc1C1CCCO1)=O)OC 60383,C=CCC(C)(C)CNC(=O)CC1CCCC1NC(=O)C(c1cccnc1)O 60384,N1(C(C2CN(C(C)=O)C2)=O)CC(NC(c2cc([N+](=O)[O-])c[nH]2)=O)C2(CCCC2)C1 60385,C(c1ccc(Cl)cc1F)=CC(=O)NC1CC(F)(CNC(C23CC(C)C2C3)=O)C1 60386,N1(C(CC2(C)CCCC2)=O)CC(CNC(c2cccc(F)c2Cl)=O)CC12CCC2 60387,N1(C(c2nc(CC)oc2)=O)CC(C)(C(=O)NC(C)CC(C)(C)OC)CC1(C)C 60388,c1(C(=O)NC(C(C)NC(C2=C(C)OCCC2)=O)C(C)C)ccc2nc(O)[nH]c2n1 60389,c1(C(N2CCC(O)(C(C)NC(c3ccncn3)=O)C2)=O)nccc2n[nH]cc12 60390,c1(CC(=O)NCC2CCC(NC(c3cnc(OC)s3)=O)C2)cc(C)ccc1OC 60391,N1(C(C(CCC)C)=O)CC2(C1)CN(C(C1CCC(F)(F)C1)=O)CCO2 60392,C1(C(=O)NC(COCC)C)CCC(O)CN1C(C1CCCN(CC)C1)=O 60393,N1(C(C2(C)CC(=C)C2)=O)CCN(C(c2ccc(N)cc2OC)=O)CC(C)(C)C1 60394,Cc1nc(O)c2c(n1)CCN(C(c1ccsc1S(C)(=O)=O)=O)C2 60395,N1(C(C2C(CCC)CCC2)=O)CCOC(CCNC(=O)CP(C)(C)=O)C1 60396,C(=O)(C(=O)N=S(C)(C)=O)NC1C(C)CN(C(c2ccc(C(C)(F)F)cn2)=O)CC1 60397,C1(O)(C(C)NC(=O)C(c2cncnc2)C)CCN(C(c2nnn(C)c2N)=O)CC1 60398,c1(C(N2C(CCCNC(CSC)=O)CCC2)=O)ccc(F)cc1N 60399,CN1CC=C(CC(=O)NC(C)(CNC(C23CCCC2OCC3)=O)C2CCC2)CC1 60400,c1(C(=O)NCC2CCCN(C(CN3CC(C)(OC)C3)=O)C2)cn2c(n1)SCC2 60401,N1CCCCC1C.c1(C2N(C(C=C(C)C#N)=O)CC2)cccn1C 60402,C1(CNC(C2C(=C)C2)=O)CCCN(C(C2(CC=C)CCCC2)=O)CC1 60403,C(N=c1[nH]cnc2cc(F)c(F)cc12)NC(=NCC(C)C)NCC(C)OC(F)F 60404,N1(C(c2ccc(C#C)o2)=O)CCC(CNC(c2ccc(Cl)nc2C)=O)C12CC2 60405,c1(C(N2CCC(CCN(C(CCC(=C)Br)=O)C)CC2)=O)ccc(C)c(CO)c1 60406,c1(C(C)=O)cc(C(=O)NCCCNC(c2cn[nH]c2)=O)ccc1C 60407,N1(C(c2n[nH]c(CC)c2C)=O)CC(C)N(C(c2cccs2)=O)CC1C 60408,C1(C(C(=O)N)=O)CC(c2ccccc2)=NO1.C(CC(C)OCCOCC)N(C)C 60409,C1(CCNC(=O)C=CC2CCOC2)(OC)CN(C(=O)CCOCCOC)C1 60410,c1(COC)c(C(N2CCCC(N(C(=O)CN(C)C)C)C2)=O)oc2ccccc12 60411,c1(C(=O)NCC2(O)CCCN(C(C(CC=C)N(C)C)=O)C2)cc2ccccn2c1 60412,c1(CC)[nH]nc(C(N2C(C(=O)OC(CCC#N)c3ccccc3)CCCC2)=O)c1C 60413,C(CN=c1[nH]c(=NCC2CCS2)c2c(F)cccc2[nH]1)C1C(C)(C)CCCO1 60414,C1(CCC)CN(C(c2cc(C)c(C)s2)=O)CC1C(=O)NCc1cccs1 60415,CC(CC(F)F)C(=O)N1CC(CNC(=O)Cc2ccccc2)(CC)C1 60416,N1(C(C2C(C=C)C2)=O)C(CNC(=O)Cc2ccc(OC)c(F)c2)CC2CCCC12 60417,CON1CCC(CC(=O)NC(C(C)NC(=O)CCNC(=O)C=CCl)C(C)C)CC1 60418,Cc1ccnc(O)c1CN1CCOCC1.N12CCN(CC1)C1CC(C1)C2=O 60419,C1(NC(C2(C)CCN(C)C2)=O)CN(C(c2cn3c(n2)SCC3)=O)C(C)(C)C1 60420,n1(CC(C)C(=O)NC2CCSC23CN(C(=O)C(Cl)=CCl)C3)cnc2ccccc12 60421,C1(C(C)NC(CCSCC)=O)CC2CCC(C1)N2C(=O)CCOC1CCCCC1 60422,C1(CNC(CCC=C=C)=O)CN(C(c2cnc(C)[nH]c2=N)=O)C2(CCC2)C1 60423,Cc1nn(CC(N2CCC(NC(C3C=CCC3)=O)C(C)C2)=O)c2ncccc12 60424,C1(C2(C(N(C)CCC3(c4cc[nH]n4)CCC3)=O)CC2)CSCCO1 60425,c1(C(=O)NCC2(C)CCCN2C(C2C3CCC23)=O)ccc(F)c2cccnc12 60426,c1(CNC(C2(CC=C)CCCCC2)=O)cnn2c1CN(CC#CCOC)CC2 60427,C1(NC(C2(CC(C)C)CCC2)=O)CCCC(NC(=O)CSCc2ccccn2)C1 60428,n1(CCC(=O)NC(CC)CN(C)C(C2CC2C(N)=O)=O)ncc2c1CCCC2 60429,N1(C(C(C)NC(COC)=O)=O)CCN(C)CC1CNC(c1scnc1C)=O 60430,Cc1ccc(F)cc1C(=O)NCCCOCCN(C)C(C12CCCC(CO1)C2)=O 60431,C1(C(=O)NC2(CCC)CCC2)CCN(C(C2C3CCC(C3)C2C)=O)C12CC2 60432,C(=O)(C(C#N)C(C)(C)C)NC(C)(C)CC(=O)CNC(=O)CNCCO 60433,CS(=O)CCC(O)C(=O)NC1CCCCC1NC(c1cc(O)cc(Cl)c1Cl)=O 60434,N1(C(CC(C)(C)OC)=O)CCC2CCCC12CNC(C1(CC)CCCC1)=O 60435,C1(C(N2CCN(C(CN(C(C3CC(OC)C3)=O)C)=O)CC2)=O)CC(F)C(=O)N1C 60436,Cc1cnc(C)c(NC(C2(NC(c3cc(C)[nH]n3)=O)CCSC2)=O)c1 60437,c1(C(=O)NC2CCN(C(C(CCC)(C)C)=O)C2C)cn2cc(C)sc2n1 60438,N1(CCC(=O)NCCNS(CCC)(=O)=O)CCN(C)CC1.C12OCCC1C(=O)N2 60439,N1(CC(=O)NCCN(C2CCCCC2)C(=O)C(O)c2ccsc2)CCCCS1(=O)=O 60440,CCC(COCCC(=O)NC)C(=O)N1CC(OCCC(C)N(C)CC)C1 60441,C(=O)(CC(CC1CC1)NC(C)=O)N(CCCC)C1CC1.C1(=O)CC2(CC2)N1 60442,N1(C(C2CC23CCOC3)C(=O)NCC)CC(N(C)CC)Cc2cc(OC)ccc21 60443,c1(C(=O)NC(C)CNC(c2n[nH]c(C3CC3)n2)=O)cc(Cl)cc2c1OCC2 60444,N1(C(c2cnc(C(C)O)s2)C(=O)NCCCSC)CCC(C)(CO)C1 60445,c1(C(=O)OC)cc(=NCC(C)CNC(c2cc(C(F)F)on2)=O)[nH]c(Cl)n1 60446,Cc1nc(C2CCC2)ccc1-c1nc(C2CC2)nn1CC(C)C 60447,N1(C(=O)COCC2CCCO2)CCCCC(C(=O)Nc2cncnc2O)C1 60448,N1(C(C2ON=C(C)C2)=O)CCC(C)C1CNC(c1ccnn1C(F)F)=O 60449,c1(C(=O)NCC(C)(C2CCC2)NC(C(CC#C)O)=O)cc([N+](=O)[O-])n[nH]1 60450,C1(NC(C2CCCN(CC)C2)=O)CCN(C(C2(C(F)F)CCC2)=O)C12CCCC2 60451,N1(C(C=CCCC)=O)CC(NC(c2cc(F)cc3nccnc23)=O)C2CCCCC12 60452,C12(CNC(CN(C(C)C)C)=O)CCCC1CN(C(C13CCC(CC1)CC3)=O)C2 60453,N1(C(c2c(C)nc(C)s2)=O)CCC(CNC(c2coc(Br)c2)=O)C12CC2 60454,Cc1nnc(COC)s1.C(CCC(C)N)NC(=O)CCCC1CCC1.C1C(=O)N1 60455,C1(N(C)C)(CNC(=O)C(CC2CCC2)NC(C2(O)CCOC2)=O)CCCC1 60456,C1(SC)CN(C(c2ccc(F)cn2)=O)CC1n1cc(CO)nn1.[nH]1ccnn1 60457,N1(C(CC=CC=C)=O)CCC2CC1C(=O)NCC2.C1(C(O)CO)(OC)CC1 60458,c1c(Cl)ccc(F)c1O.C1(CC)NCCC1N 60459,CCC(C(=O)N1CCC(NC(=O)C(n2nccc2C)C)C(C)(C)C1)C(C)(C)CC 60460,C1(S(C)(=O)=O)(C(N(C2CCN(C(C3CC(=C)C3)=O)CC2)C)=O)CCOCC1 60461,c1(C(CNC(=O)CCCCN(C)C)NC(CCOC)=O)ccc(F)cc1 60462,C12(C(=O)NC(CCC)CCCNC(=O)Cc3cccnc3)CC1COC21CCC1 60463,C1(C)(C(N2C(CCNC(CC3ON=C(C)C3)=O)CCC2)=O)CS(=O)(=O)C1 60464,N1(C(C(CC(=O)OCC)C)=O)CC(C(=O)NCc2cn(C)nc2C)C2(CCC2)C1 60465,O=C(C1=CCSC1)NCC(c1ccccc1)CNC(c1ccc(Cl)cc1)=O 60466,C1(CC)(NC(c2nnc(C)s2)=O)CCN(C(=O)Cc2cccc(OC)n2)CC1 60467,N(C1CCCOc2ccc(Br)cc21)C(c1c(C)scn1)=O 60468,C1(NC(Cc2cncc(C)c2)=O)CC2CN(C(c3csc(Cl)c3Cl)=O)CC2C1 60469,CC1(C)CC(NC(c2cc(C(F)(F)F)no2)=O)CN1C(C1CC12CCSCC2)=O 60470,CC1CCSCCN1C(=O)N(CCC(c1ncnn1C)C1CC1)CCN(C)C 60471,C(C)(CNC(c1ncccc1Cl)=O)(CC(C)C)NC(C(CC)OC)=O 60472,C1(NC(c2n[nH]c3c2CCC3)=O)COC2C(NC(C3CCCOC3)=O)COC12 60473,N1(C(C=CC(=O)N(C)C)=O)CCC(CC(=O)NCC2CCSC2)C1C 60474,N1(C(Cn2c(C)ccn2)=O)CC(F)(F)CC1C(N1CCCC1C(=O)N(C)C)=O 60475,C1(N(CCOC)CCc2ccnc(Cl)c2)CCN(C(=O)C(C)C2CCOC2)CC1 60476,c1(SCC(=O)NC2C(CNC(C3(CCC)CC3)=O)C2)ccccc1F 60477,N1(CC(C)S(C)=O)CC(=O)N(Cc2ncccc2CN(C)C)C1=O 60478,C1(OCC(=O)N(C(CNC(C2(n3cncn3)CC2)=O)C2CC2)C)CCCCC1C 60479,N1(C(C(C)C(F)F)=O)CC(NC(c2ccc(F)c(F)c2F)=O)C(C2CC2)C1 60480,N1(C(c2ccn(CC)n2)=O)CCCC(N(C)C(c2cc(CO)[nH]n2)=O)CC1 60481,n1(CCCF)nnnc1C(c1ccccn1)NCC(C)(C)SC1CCC1 60482,CC(CCC(C)(C)C)NC(=O)CC1CC(O)CN1C(c1cc(F)cnc1O)=O 60483,c1(N(CC(N2CC(CNC(=O)OC(C)(C)C)C2)=O)C)ccc(C#N)cc1F 60484,c1(N(CCOCC=C)C)nc(=NC(C)c2ccc(F)c(C)c2)[nH]c2c1CSC2 60485,C1(C(=O)NC23C(CN(C(C(C4CCC4)OCC)=O)C2)C3)CCOC(=O)CC1 60486,O=S1CCC(Nc2ccc(CN3CCCC3)nn2)c2ccccc21 60487,c1(C(N(C)CC2CN(C(=O)CC(C)(O)C3CC3)CCO2)=O)cc(O)nc(O)n1 60488,C1(NC)CCCCN1C(c1ocnc1C(N1CCCC1C(N)=O)=O)=O 60489,Cc1ccc(C=CC(N2CCC(NC(=O)C(C)Oc3cccc(Cl)c3)C2)=O)cn1 60490,N1(C(c2cn(CCC)nc2)=O)CCCC2(NC(=O)CC3C=CS(=O)(=O)C3)CC2C1 60491,Cc1ccc(OCCCC(=O)N(C)CCNC(=O)C(C)N2CC(C)C2)cc1 60492,c1(C(=O)NCCN(C(=O)CCC(C)OCC)CCC)c[nH]c2c(CC)cccc12 60493,c1(OCCC(=O)NC2CCC(CCNC(C=NOC)=O)C2)ccc(OC)cc1 60494,CC1(C)CC=C(C(=O)N2CCOCC2)CC1.C12CN(CC(=O)N1)CCO2 60495,N1(CC(=O)NCC(CCCC)NC(=O)Cc2occc2C)C(=O)CN(C)C1=O 60496,CCCCCCN(C(=O)Cn1ccc(C)n1)CCN(C(C1CCCC1C)=O)CC 60497,Cc1cc(NC(c2ccc(S(C)(=O)=O)o2)c2nnnn2C(C)(C)C)cc(C)c1F 60498,c1(C(C)C)sc(Cl)nc1C(=O)NCC=CCNC(=O)CC(C)F 60499,C1(C(=O)NC2CCC(NC(CCn3c(C)ccc3C)=O)CC2)CC12CCSCC2 60500,c1(C(=O)NC2CC3CC(NC(=O)C=Cc4ccsc4)C3C2)c[nH]c2ccc(Cl)cc12 60501,c1(C(=O)NC(CNC(CCC2OCC(C)(C)C2)=O)C2CC2)cc(Cl)ccc1Cl 60502,c1(C(=O)NCC2CCN2C(c2cnco2)=O)cnn(CC2CCCC2)c1 60503,C(CCC(=O)NC1(C(=O)NCC(c2cccs2)C)CCC1)NC(C)=O 60504,C(=O)(C#CC1(C)CC1)N(C)CC1CCCN1C(c1cn(C)c(C(F)F)n1)=O 60505,CCCCCC(C)CC(=O)N1CCC(C)C(CNC(c2sccc2C(F)F)=O)C1 60506,Cc1cc(C(N2CCCCC2CC(=O)NC2(c3ccccn3)CC2)=O)sc1C 60507,c1(C(C)(C(=O)NCc2ccccc2)N(C2CC(F)(F)C2)c2nn[nH]n2)ccc(Br)cn1 60508,c1(C(C(N2CC(OC)C(NC(C3(F)CCOC3)=O)C2)=O)(F)F)ccc(F)c(F)c1 60509,c1(C(=O)NCC(CNC(C2C(C=C)C2)=O)C)cnn(-c2ccccc2)c1C 60510,c1(CNC(c2n(CC#C)ccc2)=O)ccc(CNC(=O)CNC(=O)C(C)C)cc1F 60511,CC1=C(C)CC(C(N2CC(C)(CCC(N3CCCC(C)C3C(N)=O)=O)C2)=O)CC1 60512,C1(C(=O)NC(CN(C(=O)C(C)n2cnnn2)CC)C)CCC(=O)N1C 60513,C1(C)(C(=O)NCCC(C)n2cccn2)CC(O)(C#N)C1 60514,CCC(F)(F)CC(=O)N1CCCC(C2CCCCN2C(C23CSCC2C3)=O)C1 60515,C1(NC(C(=O)NC(C)C)=O)CC2CN(C(=O)COc3ccc(O)cc3)CC2C1 60516,N1(C(C2(C)CC(C)C2)=O)CCC(NC(=O)C=CSc2nc[nH]n2)C(O)C1 60517,CC1(C)C(CC(N2CCOC3CC23)=O)CCN1C(=O)Cc1ccon1 60518,C1(NC(CNC(C2C(C)C2)=O)=O)C=CC(C(=O)N(CCN=[N+]=[N-])C)C1 60519,c1(C(N(C)CC2CCCN(C(C3CCC3(F)F)=O)C2)=O)cc2nc[nH]c2cc1F 60520,CC1(CNC(C2C=CCN(C(c3nc(Cl)cs3)=O)C2)=O)CC2CCC1C2 60521,N1(C(c2c(C)nco2)=O)CCc2c(CNC(=O)C(C)(C)C3CCC3)cccc2C1 60522,c1(C(C)(F)F)cccc(C(=O)NC2CC2NC(=O)CC2C=CS(=O)(=O)C2)c1 60523,N1(C(c2cc(C)c(C)[nH]2)=O)CC=C(CC(=O)NCc2cccc(O)c2)CC1 60524,N1(C(C2CC23CC3)=O)CCN(C(=O)C(F)CC2CC2)C2(CCC2)C1 60525,c1(CC(=O)NC2CCN(C(C=C(C)C(C)C)=O)C2C)cc(C(F)(F)F)c(O)nn1 60526,C(C1CCCCC1)=C(C(=O)NCCCC(C)NC(C1(C)CC=CCO1)=O)F 60527,N1(c2nnc(OCC)s2)CCC(C)C(NC(c2cnn(C)c2C)=O)C1C 60528,N1(C(C(C)Cc2ccc(Cl)cc2)=O)CCOC2(C1)CN(C(=O)C(O)C1CC1)C2 60529,Cn1cc2c(n1)CCCC2C(=O)N1CCCCC1CNC(=O)CC#N 60530,C(N=c1[nH]c(N2CC(C#N)C3(CCC3)C2)nc2c1CSC2)c1c(C)nc(CC)o1 60531,C1(C(C)CO)CCCCN1C(c1coc(CNC(c2ccc(CO)o2)=O)c1)=O 60532,C1(NC(C(C)CC2CCCC2)=O)CC2CC1N(C(c1nc(Br)c[nH]1)=O)C2 60533,C(CCCCCNC(C1OCCC1(C)C)=O)NC(C(C1CC1)SC)=O 60534,CCCC(C(O)C(=O)NC1CCN(C2CC2)C1)NC(C1(n2cccc2)CC1)=O 60535,c1(C(=O)NC(c2cccc(F)n2)C)ccc(S(C)(=O)=O)cc1 60536,C(C1c2ccccc2CN1C(C1C2(CC2)C12CC2)=O)NC(C(C)OCC(C)C)=O 60537,N(C1CCCn2ncnc21)C(C(CCSC)NC(=O)CC(C)C(F)(F)F)=O 60538,Cc1nc(CN(CCNC(C2CCCN2C2CCCCC2)=O)C(C)C)cc(O)n1 60539,C=CCCCC(C(=O)N1CC(C(N)=O)C2(CC2)C1)NC(C1C2CCCCCC12)=O 60540,C1(NC(c2cc[n+]([O-])cc2)=O)CCCC12CN(c1nc(Cl)ncc1Br)C2 60541,C1(C)(C(=O)NCC(C)(C)OCCNC(c2cc(Br)no2)=O)C=CCCC1 60542,N1(C(c2cccnc2NCC(=O)OC)=O)CCC2(CCN(C(=O)N(C)C)C2)C1 60543,c12cc3c(s1)CCN(C3)C2=O.c1(NC(CCCC(C)C)=O)ncc(C#N)cc1I 60544,CON1CCC(CC(=O)NCCOCCN(C)C(C2(C)CCCS2(=O)=O)=O)CC1 60545,C1(N(C(C(C)=C2CC2)=O)C)CC2CCC(C1)N2C(=O)CSCc1cccs1 60546,C1(CC(C)NC(c2ccc(N)cn2)=O)CCN(C(=O)Cc2cncs2)CC1 60547,CC(C)(C)C(=O)C(=O)N1CCCOC(CNC(=O)C=Cc2cnc[nH]2)C1 60548,c1(C(N2CC3(c4cn(CC(F)(F)CO)nn4)CCCC23)=O)cnn2c1CCCC2 60549,c12ccccc1NC2=O.C(=O)(C(C)CF)NCCCN(C(C)=O)CC 60550,c1(OC)cccc(C(N2CCC2C(=O)Nc2c[nH]nc2I)=O)c1OC(F)F 60551,c1(C(N2CC3C(CNC(C4(CC)CCCO4)=O)(C3)C2)=O)cccc(C#N)c1 60552,N1(C(CCN(C)C)=O)CCCCC1CCC1CCCN1C(C1CCCC(F)C1)=O 60553,N1(C(C2CCC(OCC)CC2)=O)CCCN(C(c2cnn[nH]2)=O)CCC1 60554,CCCCC(O)C(=O)NC1CCCCN(C(C2(Cn3cccn3)CC2)=O)C1 60555,C1(C(=O)NCC(CC)NC(=O)C(C)OCCN(C)C)CCC(F)(F)C1O 60556,N(C(=NCCCF)N1CCC2C(C1)NC(=O)N2C)CCc1c(C)nns1 60557,C1(CC=C)(NC(c2csc(CC(C)C)n2)=O)CN(C(=O)C(CC)NC(C)=O)C1 60558,c1(C(C)C)ccc(C(CNC(=O)CSC2CCOC2=O)NC(=O)C(N)=O)cc1 60559,CC1CN(C(C2CC(C)(F)C2)=O)CCC1NC(=O)CCN(c1ccncc1)C 60560,C=C(C)CC(C)C(=O)NCC(C)(C)NC(c1ccsc1C)=O 60561,c1(CC)ccc(C(=O)N(C2CN(C(=O)CC3CC(CC)C3)CC2(C)C)C)c(O)c1 60562,N1(CC(=O)NC(CNC(c2cc(O)ccc2F)=O)CO)Cc2ccccc2C1 60563,N1(C(Cc2ccc(C)cc2)=O)CCC(O)C(N(C(=O)C(O)C2CCC2)C)C1 60564,N1(C(c2ccc(C(=O)OCC)o2)=O)CC2CCC(NC(=O)C(C)C3(O)CCC3)(C2)C1 60565,C1(NC(C2C(C)C2)=O)CCC(C)(NC(=O)Cc2c[nH]ccc2=O)CC1 60566,Cc1ccc(C(C)C(N2CC(O)(CCNC(=O)OC(C)(C)C)C2)=O)o1 60567,C1(C2(NC(C3C(CCC)C3)=O)CC2)CCCCN1C(c1cnsn1)=O 60568,c1(C(=O)NC2CCCN(C(CS(=O)(=O)NC)=O)C2)ncc(C)cc1OC 60569,CC1C(NC(c2c[nH]cc(F)c2=O)=O)CCCN1C(c1ccccc1F)=O 60570,C1(C(F)(F)F)(C(=O)OCC)CCCN(CC(O)C(C)(C)F)C1 60571,c1(CN=C(NC(C=C)C)NCc2cnsn2)cn2cc(F)ccc2n1 60572,C(=O)(CCCS(N)(=O)=O)NCC1(COC)CCN(C(=O)C(F)(F)C(O)C2CC2)C1 60573,N1(C(C2N(C=O)CCC2)=O)CCC2C1CCCN2C(c1ncccc1Cl)=O 60574,C(=O)(CC1OCCc2ccccc21)N1C2CC(NC(C3CC3(F)F)=O)CC1CCC2 60575,C1(CC(=O)NCC2C(NC(COCC(C)C)=O)CCC2)SC(=N)NC1=O 60576,c1(C(=O)NC2(CCOC)CCN(C(COC)=O)CC2)ccc2cccc(C)c2n1 60577,c1(OC)ccc2ccccc2c1-c1ccnc(C(=O)Nc2cc(C)c(C)cc2Br)c1 60578,CC(C(O)CC(=O)NC1(CC(C)(C)C)CCC1)C1CC1 60579,c1(C(N(C2CN(C(CCC(=O)N(C(C)C)C)=O)C2)C)=O)cnn2c1NCCC2 60580,N1(C(C2CN(C)C2)=O)CC2CS(=O)(=O)CC2(CNC(=O)CCC(C)(C)F)C1 60581,C1(N(C(c2cccc(CC)n2)=O)C)CCCCN(C(=O)C(=O)Nc2ncc[nH]2)C1 60582,N1(C(COC2(C)CN(C(=O)CC3CSCCO3)C2)=O)CC(CO)C(C)(C)C1 60583,N1(C(CC2ON=C(CC)C2)=O)CCC(C(=O)NCC(=O)OC(C)C)C(C)C1 60584,c1(C(=O)OC)cnccc1C(=O)NC1CC1CNC(C1CCC(C)C1)=O 60585,C(C(COC)C(=O)N1CCCC1CCC1CCCCN1C(c1ccsn1)=O)OC 60586,CC1CCCc2cc(C(=O)NCC3(NC(=O)CCN4CCCC4)CCOC3)nn21 60587,CC1(C2CCN(C(C3CCN(C(=O)COCc4nc[nH]n4)CC3O)=O)C2)CC1 60588,C1(OC)CC(CCNC(=O)CCn2ccnc2)N(C(=O)CCc2ccc(C)s2)C1 60589,S(=O)(=O)(c1cc(Cl)ccc1F)NC1C(c2ccccc2)(CC)CC1 60590,c1(C(=O)NC2CC(C)(NC(C3C(C)OC(=O)N3)=O)C2)cnc(S(C)(=O)=O)s1 60591,c1(C(N(C)CC2CCCN2C(c2ncoc2C2CCCO2)=O)=O)nc(=O)n(C)[nH]1 60592,C123CCC(CC1)N(C2)c1nc(cc(C)n1)NC1(CC1)C(=O)N3.C(COC)SCC 60593,C1(C(=O)NC2C=CCN(C(c3c(C)[nH]nc3Cl)=O)C2)CCc2ccccc2O1 60594,C1(NC(C2OCCN(C(CC(COC)COC)=O)C2)=O)CC2CC1CC21CC1 60595,c1(CC(=O)N(CCC(C)NC(c2cc3scnc3[nH]2)=O)C)cnn2c1OCCC2 60596,c1(C(N(CCNC(=O)C(C2CCOCC2)F)CC)=O)ccc(C)cc1O 60597,C(N=c1[nH]c2cnc(Cl)cc2s1)c1cccc(C(=O)NC2(C=C)CCOCC2)c1 60598,C(=O)(CC(C)C(C)C)NCCC1(CNC(C2N(CC)CCC2)=O)CCC1 60599,N1(C(C2N(C(C(C)SCC)=O)CC(O)C2)=O)CCC(F)(C#N)C1 60600,c1(C(=O)NCCCC(c2ccccc2)NC(C(C)O)=O)cccc(=O)o1 60601,C(CC(C)(C)CC(=O)NC(C1(O)CN(C(=O)CC(C)c2cccnc2)C1)C)OC 60602,C1(NC(=O)NCc2nnc(CC)o2)(CSC)CCCCCCC1 60603,N1(C(c2n[nH]c(CC)c2C)=O)CCC2CCCC12C(N1CC=CC1)=O 60604,C1(CC)CN(C(=O)CC2CCC(=O)N2C)CC1NC(C1(C2CCCO2)CCC1)=O 60605,C=C(C)CC(C(=O)NCC1(C)CCCS1)NC(=O)CCOCCOC 60606,c1(C(N2C(C(N3CCCC(C)(O)C3)=O)C3CCC2C3)=O)n[nH]c2ccc(F)cc12 60607,CCC(CCC(=O)N1CCCCC1CN(C(=O)CN1CC(C)(OC)C1)C)OC 60608,N1(C(c2ccn(CCNC(C(C)SC)=O)c2)=O)CCN(C)C(=O)C1CC 60609,CC1CN(C(c2c[nH]c(C(F)(F)F)c2)=O)CC1NC(C1CCC(=O)N1)=O 60610,c1(CC(=O)NCC2CC2)ccc([N+](=O)[O-])cc1C(N1CC(C(C)(C)O)(CC)C1)=O 60611,Cc1cc(C(N2CC3CC(C2)N3C(=O)C(C2CCOCC2)=O)=O)ccc1C#N 60612,C(CC1CCCC1)(C(=O)N(C)CCn1cncn1)NC(C(c1cnn(C)c1)C)=O 60613,c1(C(N2CC(NC(C3(COC)CCC3)=O)C(C)CC2)=O)cc(Cl)c(OC)cc1Cl 60614,c1(NC(CN2CCC(N)C(F)C2)=O)nc2n(n1)CC(c1ccccc1)CC2 60615,c1(CC)cc(C(=O)N(CC(C)N(C(=O)C=Cc2nc(C)cs2)C)C)ccc1OC 60616,CC1CCN(C(=O)CCNC(N)=O)CC1CC(=O)NCc1cc(F)cc(F)c1 60617,CC(C)C(O)C(C)(C)C(=O)N1CCC(C(=O)NCCC2(C)CC2)O1 60618,c1(CC)n[nH]c(=NC2CCN(C(c3cnn(C4CCC4)c3C)=O)C(C)C2)s1 60619,N1(CC)CCN(c2ccnc(N3CCCC3)n2)CC1.c12nc(no1)CNCCS2 60620,C=CCCCC(C(=O)NCc1cc(Br)c(F)cc1OC)OC 60621,c1(CCCC(=O)NCC2(NC(c3cnn(CC)n3)=O)CC2)ccccc1OC(F)F 60622,C1(C(=O)NCC2CC(C(=O)NCCC(O)C3CC3)C2)CCCN1C=O 60623,Cn1nnc2cc(C(N3CC4CCC4(NC(c4csc([N+](=O)[O-])c4)=O)C3)=O)sc12 60624,C1(CC(=O)NC(CN(C(c2cnc(O)n2CC)=O)CC)C)CCCCC1(C)C 60625,C(C1c2ccsc2CCN1C(C1COC1)=O)NC(C(=O)NCC)=O 60626,Cc1cc(C(N2CCCCC2CS(N)(=O)=O)=O)ccc1Br 60627,S(=O)(=O)(c1cc(C)cnc1Cl)N1CCC(C(=O)Nc2cccc(CCC)n2)C1 60628,C(=O)(C(=O)CCC(C)C)NCCCC(CCC)c1ccccc1C(=O)OC 60629,C#Cc1ccnc(C(=O)NCC2C(CNC(=O)CC(CN(C)C)CC)C2(F)F)c1 60630,Cc1cc(C(N2CC=CC2C(N2CC(C(=O)N(C)C(C)C)C2)=O)=O)oc1C 60631,c1(OC)cccc(-c2cn(C3CCC(C(=O)NCC4COCC4O)C3)nn2)c1F 60632,c1(C(=O)NCCN(CC(C)O)C(c2ccccc2Cl)=O)cc2ccccc2cn1 60633,C=CC1(C(=O)NCCCN2CC=CC2)CCN(C(=O)C(C2CCCCC2)C)CC1 60634,c1(C(=O)NC(CCCNC(c2c(NCC)scn2)=O)C)cnc2c(c1)CCOC2 60635,c1(C(C)C)cnn(C)c1C(N1CC(NC(=O)C(O)CN(C)C)C(O)C1)=O 60636,c1(OC)c(C)csc1C(=O)NCCOCCCNC(=O)C=CCc1ccncc1 60637,c1(-c2cc(OC)c(F)cc2C#N)cnc2[nH]cc(C(=O)NC(C)CF)c2c1 60638,c1(C(=O)NC(C)Cc2ccc(CNC(C3CC3C)=O)cc2)ccc(N)cc1F 60639,C1(CNC(C(n2cc(Cl)cn2)C)=O)CC2(CCC2)CN1C(C1CCCC12CC2)=O 60640,Cc1ccc(O)c(NC(c2nnnn2-c2ccccc2)c2cnoc2)c1 60641,C1(NC(C2CS(=O)(=O)C2)=O)CC(O)CN(C(=O)CN2CCCCCC2)C1 60642,CC(c1ccsc1)=CC(=O)NCCCC(C)NC(c1ccc(CO)s1)=O 60643,C(c1cccnc1)=CC(=O)NCC1CCC(NC(=O)Cc2cc[nH]n2)C1 60644,c1(C(=O)NC2(CCNC(=O)CCn3cc(Cl)cn3)CC2)cc(O)nc(O)n1 60645,Cc1cc(C(=O)NC2CCC2NC(c2[nH]nnc2C(F)F)=O)cc(C)c1Cl 60646,C1(NC(c2c(COC)ncs2)=O)CC(=O)N(C2CN(C(=O)Cc3cncs3)C2)C1 60647,C1(CNC(C(CC=C)N(C)C)=O)COCCN(C(c2ccncc2COC)=O)C1 60648,C1(CN(C)C(C2CCCN2C)=O)CCCN1C(C1(C2CCCO2)CC1)=O 60649,C1(C(=O)NC(C2CCOC2)C#C)(CNC(c2ccns2)=O)CCCC1 60650,c1(C(N2CCC(F)(CNC(CC(C)C3CC3)=O)C2)=O)ccc2c(n1)COCC2 60651,c1(NC(C)=O)cnccc1C(=O)N(CCNC(C1CC1(C)C(C)C)=O)C1CC1 60652,c1(C(N2CCC(O)(CNC(C(C(C)C)SC)=O)CC2)=O)ncnc2c(C)csc12 60653,Cc1ccc(C(C)(C)C(N2CCCC(C(=O)NC3CN(S(C)(=O)=O)C3)C2)=O)cc1 60654,c1(C(=O)NCC2N(C(=O)CN3CCC3)CC=C2)cccc(-n2cccn2)n1 60655,C1(C(=O)NC(CC=C)(C)C)CC2(CCN1C(C1CCCC(C#N)C1)=O)CC2 60656,C(c1cccc(Cl)c1)=CC(=O)N(C1CCN(C(c2c(C)coc2)=O)C1)CCO 60657,C1(CC(=O)NCC(CO)NC(C(C)SSC)=O)CCN(CCF)CC1 60658,C1(C(=O)NCCOCCN(C(C(C(C)C)O)=O)C)CN2CCN1C(C)C2 60659,C(N=c1[nH]c(=NCC(C(C)(C)C)OC)[nH]c2c1COCC2)C1C(CCC)C1 60660,N1(C(C2CCC(CC)CC2)=O)CCC2(CO)CN(C(=O)CC3(C)CC3)CC2C1 60661,Cc1nc(Cl)[nH]c(=NCC2C3COC(C)(C)C23)c1F 60662,C(=O)(C(O)C(CCC)NC(=O)CN1CCSCC1)NC(CC#CC)CO 60663,C12(CNC(C(CC=C)C)=O)CCC(CNC(c3cc(C#N)on3)=O)(CC1)CO2 60664,c1(C(=O)NC23CC(NC(c4nccc(C=C)c4)=O)(C2)C3)cccn2ccnc12 60665,CC(Cc1cccnc1)C(=O)NC1CC(NC(=O)C(O)Cc2ccco2)C1 60666,N1(C(CCC(F)(F)F)=O)CC(n2cc(C3(C)CCCO3)nn2)C(O)C1.C=CCCNC 60667,C1(c2nc(C(CC)(CSc3ccccc3)CC)on2)CN2CCCN1CC2 60668,C12(CNC(NCC3CCCC(COC)C3)=NCC(C)C)CC3CC(CC(C3)O1)C2 60669,N1(C(Cc2c(C)ccnc2)=O)CC(C)CN(C(=O)C2=CSCCO2)C(C)C1 60670,[N-]=[N+]=NC1CC2(C(N3CC(O)(CCNC(C4(Cl)CC45CCC5)=O)C3)=O)CC12 60671,N1(C(C(C)CS(C)=O)=O)CCC(C(C)(C)C(=O)N2CC(N3CCCC3)C2)CC1 60672,c1(C(C(=O)NCCCF)N(c2ccsc2)CCC)ccc(OCC)cc1 60673,C=Cc1ccc(C(=O)NC(Cc2cccnc2)C(N2CC3(COC3)C2)=O)cc1 60674,C(=O)(C1CCCn2cnnc21)NCC1C2CN(C(=O)OC(C)(C)C)CC21 60675,O=CN1CCCC1C(N1CC(O)CC1CNC(=O)C(O)c1ccco1)=O 60676,Cc1nc(CC(N2CCC(C(C)(C)NC(=O)CCC3CSCCS3)C2)=O)cs1 60677,c1(OC)ccc(S(=O)(=O)Nc2ccccc2Cl)cc1C(N1CC(S(C)(=O)=O)C1)=O 60678,Cc1cnc(C)c(C(N2CCC(CO)(CNC(C34CCC(C3)C4)=O)CC2)=O)c1 60679,C1(NC(c2cnc(C)o2)=O)CCN(C(C2CC3C(C2)C3(C)C)=O)C1(C)C 60680,S(=O)(=O)(c1ccc(Br)cc1NC(c1cc(Cl)ccc1F)C)N(CCC)CC 60681,N1(C(C2C(C)C2C)=O)CC(NC(c2cc(N)nc(Cl)c2)=O)CC(C)(C)C1 60682,c1(OC)ccc(CNC2CC(C(=O)NCc3cnc(Br)s3)C2)nc1Br 60683,C1(C(N(CCCNC(CC(C)n2ccnc2)=O)C)=O)CC2(C1)CC2F 60684,C=CC(C)(O)C(=O)NC(C1CN(C(c2ccnc(CC)c2)=O)CCO1)C 60685,N1(C(COCC(=O)NC)=O)CC2CC1C2CNC(c1c(C)ccn1C)=O 60686,CN1CC2CCN(C(=O)CC3CCCN3C(=O)CNC(N)=O)CC2C1 60687,CN1CCCC(CCC(N2CC=CC(NC(=O)Cn3ncnn3)C2)=O)C1 60688,c1(CC(=O)NC(C2CCCCN2C(=O)Cc2ccco2)C)cn2ccsc2n1 60689,c1(C(=O)NC(CC=C)CNC(=O)C(O)CC(N)=O)cc2cc(Cl)sc2[nH]1 60690,C1(NC(C2(COC)CCC2)=O)CCN(C(=O)CNC(N)=O)CCC1CO 60691,N1(C(COCCCC)=O)CC(C(N2CCCC(C(C)(C)C)C2)=O)CC1(C)C 60692,CCCCS(=O)(=O)N(C(C)C(=O)NCCCNC(=O)CC1(C(F)F)CC1)CC 60693,c1(CNC(=O)NCc2c(CS(=O)(=O)NC)cccc2)cnc(Cl)cc1Cl 60694,c1(C(N(CCNC(c2ccnnc2S)=O)CC)=O)cc(Br)cnc1OC 60695,C=Cc1cncc(C(N2CCC(C(=O)N(CCCO)CCC)C2C)=O)c1 60696,C1(CNC(C(C)OCCC=C)=O)CC(C(N2CC(N3CCCCC3)C2)=O)CO1 60697,c1(C(N2CCC(C)N(C(c3cnns3)=O)CC2)=O)ncnc2ccccc12 60698,CCC(C(=O)NCCC1CC(F)(F)CN1C(c1nc(O)sc1C)=O)C(C)(C)CC 60699,C(CC(C(=O)NCCCN(C)C(C)=O)NC(=O)CN(C)C1CC1)=CC 60700,O=C(C1=CCCOC1)NC(CNC(C1(F)CC1c1ccccc1)=O)CO 60701,CC1CCC(C(=O)Nc2cc(C3CC3)no2)CN1C(c1cc(=O)n(C)cn1)=O 60702,CCC(C)C(O)C(C)C(=O)N1CC2CCC1CN2C(=O)CN1C(=O)CNC1=O 60703,Cc1nc2cc(F)cc(C(N3CCCC3c3ccccc3I)=O)c2nc1C 60704,N1(C(C(C)CC2CCCC2)=O)CC2CC1CC2NC(C1CC1(C)C)=O 60705,C(=O)(C(=O)N=S(C)(C)=O)N1C(CNC(C(CC)NC(c2ccco2)=O)=O)CC(O)C1 60706,c1(CN2CC3N(C(C4CC4c4ccc(F)cc4)=O)C(C3)C2)cc(Br)cc(Cl)c1F 60707,C1(NC(c2n[nH]c(C3CC3)c2Br)=O)CCCCN(C(=O)CC2CCCC2)C1 60708,N1(C(=O)C=Cc2cccc(Cl)c2)CCCC2C1CCN2c1nccc(Br)n1 60709,C1(CS(=O)(=O)NCCCSC(F)F)CCS(=O)(=O)C1 60710,CCC(CC(=O)NC1CC(CCNC(c2cnc(CO)nc2C)=O)C1)C(C)(C)C 60711,N1(C(C(C)SC)=O)CCCC1C1CCN(C(C2(c3ccccc3)CCCO2)=O)C1 60712,c1(CC(C(=O)NCCC2(O)CN(C(C(COC)N(C)C)=O)C2)C)cccc(F)c1 60713,CCCCCC(O)C(=O)N1CC(C(F)(F)F)C1.c12ccc(nc1)[nH]c2=O 60714,N1(C(C(=Cc2cccs2)C)=O)CC2CC(NC(=O)Cc3cnn(C)n3)CC(C2)C1 60715,C(C(=O)NNC(=O)C(F)(F)F)N(CC)Cc1coc(C)n1 60716,Cc1nc(C)n(CCCC(=O)NC2COCCC2NC(=O)CN(C)C)n1 60717,N#Cc1ccc(NC(=O)CSc2ncc(-c3ccc(F)cc3)[nH]2)cc1I 60718,C(=O)(C(C)(C)C(=O)NCC(C)NC(c1ccc(SC(F)(F)F)s1)=O)OCC 60719,c1(C(=O)NC(C2CC(=O)NC2=O)C(N2C(COC)C=CC2)=O)cncc(F)c1C 60720,N1(C(c2sccc2F)=O)CC2(C1)CN(C(c1ccc(O)cc1F)=O)C2 60721,Cc1cc(CC(=O)N(CC(C)(C)CNC(c2nccn2C)=O)C)nn1C 60722,C(=O)(C(F)CC(C)(C)NC(c1ccccc1)=O)N1C(C)(CC)CC1 60723,C(CC(C)(C)NC(c1cnco1)=O)NCCSC 60724,C1(NC(c2n(C)nc(O)c2)=O)CCN(Cc2cccc(C(F)(F)F)c2O)CC1F 60725,C1(NC(COc2ccc(C#N)cc2)=O)CN(C(=O)CCC2CC2)C2(CCCC2)C1 60726,C(=O)(C(C)(C)C)NC(C)C(=O)NCC1(CNC(=O)Cc2ccsn2)CCCO1 60727,Cn1c(O)nc(NC2CCCCC2NC(C2(CO)CCOCC2)=O)cc1=O 60728,c1(OC(C)=O)ccc(Br)cc1C(N1CCN(C(C2(CF)CCC2)=O)C(CO)C1)=O 60729,n1(CC)c(-c2ccoc2C)n[nH]c1=NC(=O)NC(c1cc2ccccc2s1)C 60730,C1(NC(CS(=O)(=O)NC)=O)CCN(C(=O)C(n2cc(Cl)cn2)C)CC1O 60731,c1(CC(=O)NCC(CNC(Cn2c(C)c(Cl)cn2)=O)F)cc(C(F)(F)F)cc(F)c1 60732,C1(NC(COCc2ncc(C)o2)=O)CCC(C)(CNC(=O)C(C)(C)N(C)C)C1 60733,c1(C(N2CCC(CN(C(c3cn(CC)nc3)=O)C)C2)=O)cccc2c1CCCC2 60734,N1(C(=O)COCc2ccccc2)CCN(CC(c2ccccc2)(F)F)CC1 60735,c1(C(=O)NC2CCCC(NC(C3CCCS3)=O)C2)cnc2ncc(Cl)cn12 60736,C1(C2CCN(C(=O)Cc3cc(Cl)ccc3Cl)CC2)(NC(C2CNC(=O)N2)=O)CC1 60737,C1(NC(c2sc(CC)c(C)c2)=O)CC2CC1N(C(C1CC1COCC)=O)C2 60738,c1(OC(C)C)ccccc1CC(N1CC(N(C)C(c2cscn2)=O)C(F)C1)=O 60739,O=C(CC1COc2ccccc21)NC1CC(NC(=O)C(F)(F)c2cscn2)C1 60740,C(=O)(CC(C(F)F)C(C)(C)C)N1CCC(CCNC(C2=C(C)CCC2)=O)CC1 60741,c1(C(C2CCN(C(=O)C=C(C)C(C)C)CC2)NC(C(C)SC)=O)ccc(F)cc1C 60742,N1(CC)CCC(NC(CC2(OC)CN(C(=O)CCC(C)OC(C)C)C2)=O)CC1 60743,C(=O)(C(O)C(F)(F)F)N1CC(NC(C)C(=O)NCC(c2ccccc2)N(C)C)C1 60744,CCC(CC(=O)N1CCCC(CN(C(=O)Cc2cnccc2OC)C)C1)SC 60745,C1(C(C)NC(=O)CCC2CCN(C(c3cscn3)=O)C2)CCN(C(N)=O)CC1 60746,N1(C(CNC(=O)OC)=O)CCC(CO)C(NC(=O)CN2CCC(C)(C)C2)C1 60747,Cc1cc(C#N)c(N2CCCC3CC23)nc1C 60748,c1(OC)cc(C(=O)NC2CC(NC(=O)CC(C)(C)SC)C(O)C2)cc(C)c1 60749,c1(CC)c(C(=O)NC(C)CCCNC(c2conc2C2CCC2)=O)cccc1C 60750,C1(CNS(CCOCC)(=O)=O)CC(C(=O)OC)C1(C)C.C(=O)CCCNC 60751,C(CC(C)C)(C(=O)N1CCC(CNC(c2nnn(C(C)(C)C)n2)=O)C1(C)C)OC 60752,CC(C)CCC(C)N=c1[nH]c(=NCC2CCC=CO2)[nH]c2c1COC2 60753,CC1(CNC(=O)CC2CCCC(C)(C)O2)CCC(NC(=O)CSC2CC2)CC1 60754,c1(C2CCCC(C)CC2)csc(=Nc2ccccc2)n1CC1CC(OC(F)F)C1 60755,C1(C(N)=O)CN(C(C2CSCCS2)=O)CCN1C(c1cc[n+]([O-])cc1)=O 60756,C1(CNC(C(=O)NC)=O)(CNC(=O)Cn2cnc([N+](=O)[O-])n2)CC2CCCC2C1 60757,c1(OCC(=O)N(C(CSC)C(=O)N2CCCC2CF)C)cccc(C)c1 60758,C1(CNC(C(C)OCC=C)=O)CC(C)N(C(c2cc(C(N)=O)no2)=O)C1 60759,c1(C(=O)NCCC2CN(C(C3CC(CC(F)F)C3)=O)C2)csc(C2CCCO2)c1 60760,C12(NC(=O)NCCCCC(C)c3ccccc3)CC1CS(=O)(=O)C2 60761,N#Cc1sc(=NC23CCCC2CN(C(c2cnnc(Cl)c2)=O)C3)[nH]c1Cl 60762,C1(NC(C2OCCN(C)C2)=O)CC2(CCN(C(c3ccc(C#N)cc3O)=O)C2)C1 60763,c1(CNC(C2C(CC)(CC)C2)=O)cc(-c2c[nH]nn2)n(C)n1.C1CC1 60764,N1(C(c2cnn(CC)n2)=O)CC(CNC(=O)Cc2nnc(C)s2)OC2CCCC12 60765,c1(N(CC(N2CCCC(COCCNC)C2)=O)C)ccccc1[N+](=O)[O-].C1(C)CC1 60766,CC(C)C(O)C(=O)N(CCCNC(=O)CCN1CCCCCC1)C 60767,c1(C(N2CCC(CNC(C(CCC)O)=O)C2(C)C)=O)nccc2cccnc12 60768,Cc1noc(-c2cn(CC(=O)N(C)CCN(C(c3ccon3)=O)C(C)C)cn2)n1 60769,C1(CCNC(=O)CN2CCCC2)CSCCN1c1nccc(CCO)n1 60770,CS(C)(=O)=Nc1ccc(C(N2CC3CCCC3(CNC(c3cnn[nH]3)=O)C2)=O)cc1 60771,Cn1cnc(C(=O)N(CCC(N2CC(O)CC2(C)CO)=O)CC2CC2)cc1=O 60772,N1(C(=O)NC2(c3ccc(C)o3)CC2)CCn2c(C)nnc2C1C 60773,C=CCC(C(=O)OCC)NC(=O)CCN(C(C1CCC1C)=O)CC1CC1 60774,C(=O)(CCC(C)C#N)NCC1CCC(NC(c2c(C)coc2C(C)(C)C)=O)C1 60775,c1(C(=O)NCC2(OC)CCN(C(=O)C=CC3CCCO3)C2)cc(C)c(C)cn1 60776,[N-]=[N+]=NC1CN(Cc2ccns2)CC1C(=O)Nc1ccccc1 60777,Cc1[nH]nc2c(C(N3CCC(CO)(NC(C4CNC(=O)C4)=O)CC3)=O)cccc12 60778,N1(C(C2CN(C(CNC(=O)OC)=O)CC(F)(F)C2)=O)CCC2(CCOC2)CC1 60779,C(=O)(CCCCCC(C)C)NC1C(CO)CCN(C(CCCC#C)=O)C1 60780,C(C1CCC(C)CC1)=C(C)C(=O)NC1CCCCC1NC(=O)CC1CC2CC2C1 60781,c1(OCC)ccc(CC(N2CCC(NC(=O)C=CSc3ccccc3)C2)=O)cc1 60782,C1(NC(N(CC(O)C(=O)OC(C)(C)C)C)=O)CCCCCCC1 60783,C1(NC(C2CN(CC)C(=O)C2)=O)CCC12CN(C(c1cn(CC(N)=O)nn1)=O)C2 60784,CC1(C)C(CNC(=O)Cn2ncnn2)CCN1C(=O)COc1ccsn1 60785,C12(NC(Cc3cnc(C)o3)=O)CCN(C(c3ccns3)=O)CC1C2 60786,c12cc(ncn1)N2.c1(C(CO)N(c2ncc(Br)cn2)C)ccc(C(C)(C)C)cc1 60787,c1(C(=O)NCC(C)NC(=O)C(F)CC2CC2)ccc(Br)cc1 60788,c1(COC)nn(C)c(Cl)c1C(=O)NCCCCNC(C1(C2CCCO2)CCC1)=O 60789,Cc1nn(C(F)(F)F)c(C)c1C(N1CCC(O)(CC2CCOCC2)C1)=O 60790,CC1CN(C(=O)NC2CC2c2ccccc2)CCN1C(=O)C(C)n1ccnc1 60791,c1(C(=O)NCC(C(=O)N(C(CC)CC)C)(C)CC)ccc2nccn2c1 60792,C1(NC(=O)NCC2(CC)CCCO2)CC2CC1CC2C(N)=O 60793,C1(NC(c2c(C)nccc2)=O)CN(C(c2ccnc(Cl)c2I)=O)CC1C#N 60794,N1(C(CCCOCCOCC)=O)CCCCC1CNC(C1NC(=O)OC1C)=O 60795,N1(C(C#C)(C)C)CCN(C(=O)NC2C3CCC(F)C23)CC1 60796,C(=O)(CS(=O)(=O)Cc1cncn1C)OC(c1ccc(Cl)cc1)C(C)C 60797,CC1CC(C)N(C(c2cccc3oncc23)=O)CCN1C(c1ccco1)=O 60798,N1(C(C2C(C=C)OCC2)=O)CCN(C(c2c(C(C)C)nn(C)c2Cl)=O)CC1CC 60799,C1(NC(C2CCC(C)O2)=O)CCC2CN(C(=O)C(c3ccccc3)C)CCC2C1 60800,c1(-n2ncc(NCC3(C(N)=O)CN(C(=O)CO)C3)n2)cccc(Br)c1 60801,N1(C2CCC(NC(COCC(C)(C)C)=O)C2)CCN(C(=O)C(Cl)=CCl)CC1 60802,CC(C)=C=CC(=O)NCC(O)CNCC(=O)N(C1CC1)CC.C(C(N)=O)O 60803,C1(NC(C(=O)NC(C)C)=O)CCN(C(c2cc(C(C)C)cnc2O)=O)C12CC2 60804,N1(C(C(N)=O)=O)CC(NC(=O)CNC(=O)CC2CCCCC2)CC12CCC2 60805,C(=O)(C(C)S(C)(=O)=O)NC1C(CC)N(C(=O)CCn2ccnc2)CC1 60806,N(C1CCCc2cc(C#N)ccc21)Cc1cc(NC(=O)OC(C)(C)C)cc(Br)c1 60807,C(C(C)C(F)C(=O)NC1CC(C)(C)C1C(=O)OC)NC(C1CC(C#C)(O)C1)=O 60808,C(=O)(C1=CC2CCCC12)N1CCCC(C)(NC(c2c(C)oc(C(C)C)c2)=O)C1 60809,Cc1oc(C2CC2)nc1C(=O)NC1CCC(NC(C2(C)CCNC2=O)=O)C1 60810,Cc1ccc(=O)n(CC(=O)NCCCCNC(=O)C(c2ccc(F)cc2)(C)F)n1 60811,CCC(C)(C)C(C)CNCCNc1c(OC)cccc1Br 60812,C1(CC)C(C(N2CCOCC2CCNC(=O)CNS(=O)(=O)CC)=O)CCN1C 60813,CC(CCN=c1[nH]c(=NCC2CC(=O)N(CC)C2=O)c2ccccc2[nH]1)CC(C)(C)C 60814,CCCC(C)(O)CC(=O)NC1CCC(CNC(=O)CCn2cnccc2=O)CC1 60815,C1(Cl)(C(=O)NCCNC(c2cnc(C(F)F)s2)=O)CC12CCOCC2 60816,C12(CNC(C3(OCC)CCC3)=O)CCCCC1CN(C(c1ccc(SC)s1)=O)C2 60817,Cc1nc(C=CC(N2CC(F)(CNC(=O)CC3CC(=O)NC3=O)C2)=O)[nH]c1C 60818,c1(C(=O)OC)cc(CC(=O)N(C)C(c2cnn(CCF)c2)=O)c[nH]1 60819,c1(C(N2C(C)CN(C(c3ccc(SC)s3)=O)C(C)C2)=O)ccc2c(c1)N(C)CC2 60820,C1(C(=O)NCC(CC2CC2)CO)(NC(c2c(CC)n[nH]c2)=O)CCCCC1 60821,C(=O)(N=c1ccn(-c2ccc(F)cc2)[nH]1)c1nc(C)nc(N2CC3CCCC3C2)c1 60822,CCC(C)C(C(=O)NC1CC(F)(F)C1)N1CCC(CNC2CCCO2)CC1 60823,C1(C(=O)NCCC2CCN(C(c3ccccc3O)=O)C2)CCC2C(CC1)C2(F)F 60824,Cc1nc2cc(C(=O)NC(C)CCN=[N+]=[N-])cnc2s1 60825,C12(CNC(C(C(CC)C)OC)=O)CCC(CC1)N(C(=O)Cc1cccnc1F)C2 60826,c1(C(N(C)CCOCCCNC(=O)C(O)C2CCC2)=O)cc(P(C)(C)=O)cs1 60827,c1(C(NCC2(NC(c3snc(Cl)c3Cl)=O)COC2)C2CC2)c[nH]c2ccc(F)cc12 60828,c1(C(N2CC(CNC(CC(CCC)O)=O)CC2(C)C)=O)ccc(N)cc1[N+](=O)[O-] 60829,C1(NC(C(C(C)C)O)=O)CCC(C)(CNC(c2nn(C)cc2Br)=O)CC1 60830,CC(C)C(C)C(=O)NCc1cc(C(=O)NOCC2CCOC2)on1 60831,Cc1ccc(C(=O)NCC(c2ccccc2)CNC(=O)CC#N)c(F)c1 60832,n1(CCC)cc(Cl)c(C(=O)NC2CCC(C)(CNC(C3CN(C(C)=O)C3)=O)C2)n1 60833,C1(CC2C(=O)N2)CCC(C)(C)O1.c1(CC(C)N(C2CC2)CC2CCOC2)cccs1 60834,Cc1ccccc1C=CC(N1CCC(C(N2CC3(CC3)CC2CO)=O)(C(C)C)C1)=O 60835,c1(C(=O)NC2CC(NC(C3(C)CCCCO3)=O)C2)cc2sc(Cl)cc2s1 60836,N1(C(CCc2cc(OC)no2)=O)CC(NC(=O)C#CC(C)C)C(C)C1 60837,C(c1cc[nH]n1)=CC(=O)NCC(C)(C)OCCNC(C1CCCC1O)=O 60838,Cc1cccc2c1CC(C(N1CCC(NC(c3csc(Cl)c3Cl)=O)C(F)C1)=O)N2 60839,CC(C)(CS(C)(=O)=O)C(=O)NC(CNC(=O)CC1CCCNC(=O)C1)CO 60840,C#CCC(C(=O)N(C1(C(N2CCOCC2)=O)CC1)CCC=C)NC(=O)COC 60841,C1(P(C)(C)=O)(C(=O)NC(CN(C(c2nonc2CC)=O)CC)C)CC1 60842,c1(CN2CC3C(CNC(c4c(C)ccc(C)c4)=O)C3C2)ccc2c(c1)CCC2 60843,CC1(C)OC2(Cn3cc(CCNC(c4cncc(N)n4)=O)nn3)CCC1C2 60844,C(=O)(C(CCC)C(C)C)N1CCC(N2CCN(C(C(CCC)=CCC)=O)CC2)C1 60845,N1(C(C(C(C)(C)C)OC)=O)CC2(CC(NC(=O)CSCc3ccccc3)CO2)C1 60846,C(C)(CNC(=O)CCc1cccnc1Cl)(C(C)C)NC(C1N(C(C)=O)CCC1)=O 60847,c1(C(=O)NCC2CCC(NC(C3=C(C)OCC3)=O)C2)c[nH]c2c(Br)cccc12 60848,CCCC(C)(CC)C(=O)N1CCC(C(C)NC(=O)C(C)=CC(C)(C)C)CC1 60849,CC1(C)CN(C(c2sc(C#N)cc2Cl)=O)CC(CNC(c2n[nH]cc2F)=O)O1 60850,Cc1c(C(=O)NC2(CNC(=O)C(C)OCC3CC3)CCOCC2)cncc1Cl 60851,C(C(=O)NC1CCCCC1(F)F)(C(C)(C)C)NC(c1cccc(CC)c1)=O 60852,N1(C(c2c(C)c[nH]n2)=O)CCOC(C)(CNC(C2CN(C(N)=O)C2)=O)C1 60853,Cc1cc2c(C(=O)N(C(C)CCNC(C3CCNC(=O)C3)=O)C)cccc2o1 60854,c1(NCC2CC(N(C)C)C2)cc2oc(-c3ccccc3)cc2[nH]1 60855,c1(C(=O)NC(C(C)(C)NC(CCNC(=O)OC)=O)C)cc(C)nc2cc(C)nn12 60856,C1(CC(=O)N(C2CCN(C(C=CC3N(C)CCC3)=O)CC2)C)CCC2(CC2)CO1 60857,c1(C(=O)NC2C(NC(C(C(=O)OC)C)=O)CC2)cnc2cc[nH]c2c1 60858,C(=O)(C1=NOC(C)C1C)NCC#CC(=O)Nc1n(C=C)ncc1 60859,C1(NC(CN2CCN(C)CC2)=O)C2CCC1N(C(C1(C3(C)OCCO3)CC1)=O)C2 60860,C#Cc1cncc(C(=O)NCC(O)CNC(c2cnc(C(F)(F)F)c(C)c2)=O)c1 60861,Cc1cc(C(=O)NCCCN(C(c2ccc(C(F)F)s2)=O)C2CC2)[nH]c1C 60862,C1(CC(N2CC(O)(C(C(=O)NCC(C=C)C)F)C2)=O)CC2(CCC2)C1 60863,C1(NC(c2ccc(N(C)C)cc2)=O)CC2CC1CN(C(c1cc(Cl)no1)=O)C2 60864,c1(C(=O)NCCC2N(C(c3n(C)cnn3)=O)CCC2)ncsc1S(N)(=O)=O 60865,CCS(=O)CC(=O)NCC1CCCC(CNC(C2(n3cnnn3)CC2)=O)C1 60866,C(=O)(C1CCc2cccnc21)NCC(CCNC(c1ncn(C)n1)=O)O 60867,C=C(Cl)CCC(=O)N1CCCC(N(C(=O)CC(=O)NCC)CC2CC2)C1 60868,N1(C(c2cc(C)n(C)c2)=O)CC2(CCN(C(c3ccc4occc4n3)=O)CC2)C1 60869,C#CCCCC(=O)N1CCN(c2ccccc2C(N2CCCC2CO)=O)CC1 60870,Cc1ccc([N+](=O)[O-])cc1CN1CCNCC1C(=O)Nc1c(O)cccc1Cl 60871,c1(NC(C23C(CN(C(Cc4cc(C)no4)=O)C2)C3)=O)c(F)cc(F)cc1[N+](=O)[O-] 60872,C(C)(CCC(=O)NC(CCC1CCC1)C(=O)NCCc1ncccc1F)OCC 60873,CC1(C)CC(CC(=O)NC2(CF)CCN(C(=O)C(=O)C(C)(C)C)C2)C(=O)O1 60874,c1(SC)ccc(C(N2CCCC(C)C2N(C)C)C(=O)NCCOC)cc1SC 60875,c1(-c2scc(C(C)(C)C)n2)oc2ccccc2c1OC(F)F 60876,N1(C(CN2CC(C)(C)C2)=O)CCC2(CC2)CC1C(=O)Nc1cnc(Cl)nc1 60877,c1(C(=O)NC(CNC(C(CCCC#C)C)=O)C)cnc2[nH]c(C)nc2c1 60878,c1(CNC(CCNC(c2c(CC)n[nH]c2)=O)=O)nc2cc(C)ccc2n1C(C)C 60879,CCC(CC)C(C(=O)N1CC2(C)CC1(C(N1CCCCC1CC(C)C)=O)C2)OC 60880,C=CC(C)(CC)C(=O)NCC1=CCN(C(=O)C(C)c2cc[nH]n2)CC1 60881,CCCCC(C(=O)N(C)CC1(O)CCCN(C(c2cnn(CC)c2)=O)C1)N(C)C 60882,C1(NC(C(CCC)NC(N)=O)=O)CC2CC1CN(C(=O)CCCCC(C)C)C2 60883,CC1(C)C(c2cccc(F)c2)CCN1C(=O)NCC(=O)OC(c1cccnc1)=O 60884,C=CCC(CC=C)C(=O)N1CCCCC1C(C)NC(=O)CCCC(=O)NCCC 60885,CC(C)(CC1CCOCC1)C(=O)NCC1CCN1C(C1CC1(C)C)=O 60886,c1(C(C(=O)NC2C(COC(C=CC(=O)OCC)=O)C2)O)ccccc1Br 60887,C1(C(N2CCC(C)(NC(C3CN(C4CCC4)C3)=O)C2)=O)CN2CCC1(C)CC2 60888,CC1CN(C(C2CCC(C(F)(F)F)C2)=O)CCC1CNC(c1nscc1N)=O 60889,C(=O)(C#CC(C)(C)CNC(=O)CC1(COC)CC1)NC(CCCC=C)C1CC1 60890,C1(O)(C(C)NC(CCC(=O)c2ccc(C)s2)=O)CCN(C(C2CCC(C)O2)=O)CC1 60891,N1(CCNC(=O)CC2CCCC23CC3)CCN(C(=O)CN2CCCNC2=O)CC1 60892,c1(C(N(C2CCCN(C(=O)CCc3nccs3)C2)C)=O)cnc2c(Cl)cccn12 60893,S(=O)(=O)(CCC(=O)NCC1CC(C(=O)NCc2cc(C)cnc2F)=NO1)NC 60894,c1(C(N2CCC(N(CCO)C(C3CCSC3)=O)C2)=O)ccc2c(c1)NS(=O)(=O)C2 60895,N1(C(c2cc(C(=O)OC)sc2C)=O)CC(NC(C2CC2C2CCC2)=O)C(C)(C)C1 60896,c1(C(=O)NCCNC(C2(C)CCCNS2(=O)=O)=O)cccc2c1OCCCO2 60897,N1(C(c2ccon2)=O)CCCC2(C1)CN(C(c1cnc(O)s1)=O)CCO2 60898,Cc1nc2c(C(=O)NC(C3(CNC(c4sncc4C)=O)CC3)C)cccc2o1 60899,N1(C(=O)Nc2c(OC(F)(F)F)cccc2F)CCC2(CC1)CC(O)(C(F)(F)F)C2 60900,CCC(CC(=O)C(=O)CC1CC(C(F)(F)F)C1)N(C(=O)C(C)CC1CC1)C.OC 60901,Cc1oc(C)c(C(=O)NCC(O)CN(C(=O)Cn2cc(F)ccc2=O)C)c1C 60902,Cc1cc(OC(c2ccc(OC(=O)NC3(C)CCC3)cc2)=O)ccc1[N+](=O)[O-] 60903,C(C)(CCC(=O)NC(C)(CNC(=O)C(N1CCC(C)C1)=O)CO)OCC 60904,CCCCC(C)(F)C(=O)NC1CCN(C(c2ccc(COC)o2)=O)CC1CC 60905,C1(CCC(=O)NC(CNC(C2(COC)CCC2)=O)(C)C)C(=O)ON=C1C 60906,c1(NC(C)=O)cc(F)c(NC(=O)NC2CC(N(C)C)C(C#N)C2)c(F)c1 60907,C(=O)(C1COc2ccccc21)NC(c1ccc(N(C)C)cc1)CNC(=O)CO 60908,C(=O)(C1=CCCCC1C)NC1(CNC(C2CCN(CC(C)C)C2)=O)CC(F)(F)C1 60909,C1(COC)CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CCN1C(C12CCC(F)(CC1)C2)=O 60910,CC(C)CC(CNC=O)CC(=O)NCC(C)N(C)C(c1cccc2nonc12)=O 60911,N1(C(CCOC(C)=O)=O)CCCC2(NC(C3CN4CCC3(C)CC4)=O)CC2C1 60912,C1(CNC(CC(CC)SC)=O)CC2(CC2)CN1C(c1ccc(Cl)c(OC)c1)=O 60913,C1(CC(=O)NC(C2CCOC2)CN(C(=O)C=Cc2cocn2)CC)(OC)CCCCC1 60914,C12(NC(c3nccc(C)c3F)=O)CCCC1N(C(C1CC13CC(C)(C)C3)=O)CC2 60915,C1(NC(CCCOCC=C)=O)CCCCN(C(=O)Cn2cc(C)ccc2=O)CC1 60916,CCCCC(C(=O)NCC1(CC2CC2)CCC1)NC(=O)C1=CC(C)(C)C1 60917,c1(OC)ccc(C(N2CC(NC(C3CC(CN(C)C)C3)=O)CC2C)=O)nc1Cl 60918,Cc1ncc(Cl)cc1C(=O)NC1(CNC(C2(F)CCOC2)=O)CCCC1 60919,N1(Cc2cc(C)sc2C)CCCC(CO)(NC(=O)C(C)C2CCCO2)C1 60920,N1(C(c2c(OCC)nccc2)=O)CC(NC(=O)CCNC(=O)CC)CC(F)(F)C1 60921,Cc1ccnnc1C(N1CCC(Cn2cc(-c3ccc(Cl)s3)nn2)C1)=O 60922,C(CC(=O)NCC(C)S(N)(=O)=O)(C(F)F)NC(C(N1CC(C)C1)C)=O 60923,C(=O)(CC(C(F)(F)F)n1ccnc1)NCC(C)N(C(CCC(=C)C)=O)C 60924,CCC(C)CCC(=O)N1CC(CNC(c2c(NC(C)=O)c[nH]c2C)=O)C1 60925,N1(C(CCOCCCNC(C2CC(CC)OCC2)=O)=O)CC2(CCC(=O)N2)C1 60926,c1(OC)cc(CCOC)ccc1Cl.N1(C(C(=O)NCCN)=O)CC(C)(OC)C1 60927,c1(C(=O)NCC2(NC(C(C)NS(C)(=O)=O)=O)CC2)ccc(C2CC2)nc1 60928,C12(NC(C3CCCN(C)C3)=O)CCCC(NC(C3CC4CC4C3)=O)(C1)C2 60929,C1(NC(C(C)=CC2CC2)=O)C2COCC1CN(C(c1nnc(O)nc1O)=O)C2 60930,N12CCOC3(CCN(CC3)Cc3c[nH]c(c3)C1=O)C2.C(=O)(CC(C)(C)C)OC 60931,CC(C)C(CNC(=O)Cc1ccc(F)nc1)C(=O)NC1CCCC(O)C1 60932,CCCCC(=O)C(=O)N(C(C)CCNC(C1(c2cccc(Cl)c2)CCCC1)=O)C 60933,CC1=C(C(=O)N2CCCCC(CNC(C3CCC3)=O)C2)CCC1 60934,C(=O)(C(N)CCCCCc1ccccc1)N(S(=O)(=O)Cc1ccc(I)cc1)C1CC1 60935,C1(C(=O)NCC23C(CN(C(c4cnc(SC)[nH]4)=O)C2)C3)CCc2nnnn2C1 60936,n1(CC(=O)NC2=NC(Br)(Br)C(Br)=N2)ccc(=NC(=O)c2ccc(F)c(O)c2)nc1O 60937,Cc1noc(C)c1C(C)NC(C(=O)NCc1cn(C)nc1OC)=O 60938,Cc1conc1C(N1CCCC1C1(C(=O)NCCn2nccc2C)CC1)=O 60939,C1(CNC(CC(=O)NC)=O)CCN(C(c2cc(Cl)nc(=N)[nH]2)=O)CC1C 60940,C1(CN2CC(NC)C2)CCC2(CCCCC2)N1 60941,C1(C(N2CC3C(NC(c4n(C)c(Cl)cn4)=O)(CC3)C2)=O)CC(C)(C)SC(C)(C)C1 60942,c1(OC)cc(OC)c(N(CCNC(=O)O)Cc2nnc(-c3cccs3)o2)c(OC)c1 60943,c1(NS(CCC)(=O)=O)cccc(C(=O)N(C)CCNC(=O)CCN2CCCC2)c1 60944,CC1(C)CCN(C(C2CC3(CCC3)C2)=O)C(C(=O)NCC2(C)CCCO2)C1 60945,c1(C2(C)CC2C(=O)NC2CC(NC(C3(c4cc[nH]n4)CC3)=O)C2)c(F)cccc1F 60946,c1(C(N2CCCC(CN(C(=O)C(C)SC)CC)C2)=O)cnc2cc(C)ccn12 60947,C(C(C(=O)NC(CC)C1CC1)NC(c1cc(CO)[nH]n1)=O)OCC 60948,C1(CN(C(C2C(C(C)(C)C)C2)=O)CCO)C=CCC(C(=O)NCCc2nccs2)C1 60949,N1(C(=O)NCC(=O)OCCCC)CCOC(CCNC(=O)C(C(C)C)SCC)C1 60950,C=CC1(C(=O)N(C)Cc2ccoc2)CCN(C(c2ccncc2O)=O)C1 60951,C(=O)(C(CCC1CCCC1)N(C(C)C(C1CC1)Sc1ccccc1)CC)NCC 60952,N1(C(c2n(CCC)ccc2)=O)CC(NC(=O)Cc2cnn(CC)c2)C(C)C1 60953,c1(C(N(CC(C)NC(c2nocc2Br)=O)C)=O)cccc(Cl)n1 60954,c1(CC)nc(C)n(C)c1C(=O)NC1C2CCN(C(c3csnn3)=O)CC12 60955,C(=O)(CCC(=O)C1CC1)N1CC(CC)(CN)C1 60956,c1(NC(=O)NCc2cn(C)nn2)c[nH]c2cccc(Br)c12 60957,C1(O)(CN(C)C(c2cc(Cl)cc(Cl)c2)=O)CCN(C(c2cn(C)c(O)n2)=O)CC1 60958,c1(CC)cc(Cl)ccc1C(=O)N(C(CNC(C1CCO1)=O)C1CC1)C 60959,Cc1cc(C(N2CC(C3(NC(=O)CCC4(C)CC4)CC3)C2)=O)cnc1C(F)(F)F 60960,C1(C#N)(SC)CN(C(=O)C=CCN(C(=O)C(C)=C2CC2)C)C1 60961,N1(C(c2c(C)nccc2)=O)CCN(C(=O)C(C)SC(F)(F)F)CC(C)(C)C1.C(N)=O 60962,C1(O)(CN(C(C2C(OC)CCC2)=O)C)CCCN(C(c2ccncc2Cl)=O)C1 60963,C#CC1(C(N2CCC3C(O)CC23)=O)CN(C(c2ccn(C)c2CC)=O)C1 60964,c1(C(=O)OC(CC)C(=O)Nc2nccs2)cccc(C2(C(F)(F)F)CC2)c1 60965,C1(C(C(=O)NC2CC(=O)C2)N(C(c2cccc(F)c2)C)C)CCC(F)(F)CC1 60966,C1(NC(c2occ3c2CCC3)=O)COC2(C1)CN(C(=O)C1=CCCC1)C2 60967,C(=O)(CC(C)P(C)(C)=O)NCC1C2N(C(c3c(C)scc3)=O)C(CC2)C1 60968,c1(C(=O)NC2CCC(CCNC(CC(C)(C)OC)=O)C2)ccc2c[nH]nc2c1 60969,CC1CC2(CCO1)CCN(C(c1ccc([N+](=O)[O-])cc1OC(F)F)=O)C2 60970,C1(C(=O)NCC(C)(C)N2CCCC2)CCN(C(C2CC(=O)C23CCC3)=O)C12CCC2 60971,N1(Cc2nc(C)oc2)CC(=O)N(Cc2cc(C#N)cn2C)C1=O 60972,CCC(CC)CC(=O)NC1CC(CNC(c2ccc(C)nc2N)=O)C1 60973,C1(C2CCCCC2)(C(=O)NC(CNC(C(COCC)(C)C)=O)(CC)CC)CC1 60974,c1(N(CC(C)C)C)nccc(N2CCCC(c3nc(CNCC(F)F)no3)C2)n1 60975,C1(CN(C(c2c(C)scc2)=O)C)CCCCN1C(=O)C(c1ccncc1)C 60976,C1(C(=O)NCCC(=O)NC(CC)C)CC(O)(CNC(C2CCCCS2)=O)C1 60977,c1(C(N2CCC(N(C(CC=CCC)=O)C)C2)=O)cc(Cl)c(C)cn1 60978,c1(C(=O)NCC2(CO)CCN(C(CC=CC=C)=O)CC2)cc(F)cc2cc[nH]c12 60979,N1(C(C=CC=CC)=O)CC2CC(NC(c3ccnn3CCOCC)=O)CC(C2)C1 60980,CC(C)C(CN1CCCC1)NCC1CC2CC1C2 60981,c1(C(N2CC(NC(C(C=C)(F)F)=O)C(C)CC2)=O)cc(S(=O)(=O)NC)c[nH]1 60982,C1(CN(C)C(c2c[nH]c(C#N)c2)=O)CN(C(=O)COCc2nc[nH]n2)CCO1 60983,C(c1ccccc1)=C(C)C(N1CCCC1CCC(=O)N(C)Cc1ccnn1C)=O 60984,C(CN=c1nc(N2CCC(C)C(F)(F)C2)c2c([nH]1)COC2)NC(=O)OCC 60985,C1(NC(CCNC(C)=O)=O)CCCC(C(=O)NCC23CC(CCO2)C3)C1 60986,c1(C(N2CCC(NC(C(C)NC(COC)=O)=O)C2CC)=O)cc(O)cc(N)c1Cl 60987,C(=O)(C(C)(C)C(F)c1ccccc1)N1CCC(NC(c2c(Cl)cn(C)n2)=O)C1 60988,c1(C(N2C(C)CN(C(=O)CC3(CO)CC3)CC2)=O)cnc(O)n(C2CC2)c1=O 60989,c1(C(=O)NC(C(C)NC(=O)Cc2cc[nH]c2)(C)C)cc(Br)cc2c1OCC2 60990,CCC(O)CC(=O)NC(c1ccc(-c2ccc(N3CCNCC3)cn2)nc1)C 60991,c1(OCCOCCOC)ccc(C(=O)NC(C)C(C)CC2CC2)cc1 60992,CC(C)(C)CC(O)C(=O)N1CCC(O)(CNC(C2CC(n3cnnc3)C2)=O)C1 60993,C(C)(C)(CCCC(=O)NCc1ncc[nH]c1=O)NC(CC(C)CN(C)C)=O 60994,C1(C(N(C)CCn2ccnc2)=O)CC(O)CN1C(=O)Cc1cccnc1 60995,C1(N(C(Cc2c(CC)con2)=O)C)CCC(NC(=O)CSCC(F)(F)F)CC1 60996,c1(OC)nscc1CNC(=O)CCCC1(NC(c2ccn(CCF)n2)=O)CCC1 60997,Cc1ccc(C(F)F)c(C(N2CC(O)(CCNC(=O)Cc3cocn3)C2)=O)c1 60998,N1(C(C2(COC)CC2)=O)CCC2(CCN(C(=O)Cc3ccsc3)CC2)C(C)C1 60999,N1(C(C(C)c2ccco2)=O)Cc2[nH]nc(C(N3CC(CNC(N)=O)C3)=O)c2C1 61000,CCC(C#N)(CC)C(=O)N1CCC(SC2CCN(C(C34COCC3C4)=O)CC2)C1 61001,CC(C)(CN=C(NCC1CCCO1)NCC1CCOC1)Oc1cccc(Br)c1 61002,C(CC(C(=O)NCCC(C(C)C)N1CCOCC1)NC(c1ccn(C)n1)=O)SC 61003,C1(CCC(=O)NCCN(C(C=CC(CC)C)=O)C)NC(=O)NC1=O 61004,c1(CC)cc(C(=O)Nc2ccc(NC(=O)Cn3cnnc3O)c(C)c2)ccc1Cl 61005,N1(C(Cc2cccc(C)c2)=O)CC2OCCN(C(=O)C3=CCCCCC3)C2C1 61006,C(=O)(C(CC(C)C)OC)N1CC(CCC)C(C(N2CCCC2CC)=O)C1 61007,c1(C(=O)NCC(CC)N(C)C(c2c(C)n[nH]c2C)=O)ccc(N)c(O)c1 61008,N1(C(CC(CCC)O)=O)CC2CCC1CN2C(c1cn(CC(F)F)cn1)=O 61009,N1(C(c2ncc(OC)nc2)=O)CCC(NC(c2c[nH]c(=N)s2)=O)C(O)C1 61010,N1(C(COCc2c(C)ncs2)=O)CC(NC(c2cnn(CC(C)C)c2)=O)C(O)C1 61011,N1(C(c2c(NC(C3(C(=O)OC)CC3)=O)cnn2C)=O)c2ccccc2CC1C 61012,c12ccc(cc1)CNC(=O)C2.C1(CC)C(CC(=O)NCC2CC2C2CC2)C1(F)F 61013,c1(COC(c2cnn(Cc3ccccc3I)c2)=O)c(F)cccc1F 61014,CCCCCCC(C)(c1nnnn1C(C)CC)NCc1nsc(C(=O)OCC)n1 61015,CC1(NC(c2n[nH]c3c2COC3)=O)CCC(NC(C2(C)CCCCO2)=O)CC1 61016,C(C(C)(O)CC(C)C)NC(C1C2CN(C(c3c(COC)cco3)=O)CC21)=O 61017,CC12COCC1CN(C(=O)CCc1nnc(C3CC3)o1)C2 61018,CCC(=O)NNC(=O)C(C)(C)CCCCNC(=O)CNC(C1=CS(C)=N1)=O 61019,C(=O)(C1=NN(C)C(=O)CC1)NC1CCC(N(C(c2c(C)c(N)cnc2)=O)C)C1 61020,n1(CC)cnc2c(N3CCCC(C#N)C3)[nH]c(=NCc3nn(C)cc3C)nc12 61021,C1(C(=O)NCC(CCOC)NC(c2ccc(Cl)s2)=O)CC2(C1)NC(=O)NC2=O 61022,c1(NC(c2ccc(F)cc2F)=O)ccc2c(-c3cncs3)n[nH]c2c1 61023,C1(F)(CNC(C2C(C(=O)OC)C2)=O)CC(NC(=O)COCCF)C1 61024,C(C)(CCN=c1[nH]c(=NCCSC)[nH]c2c1CCC2)CC 61025,N1(C(Cc2c(C)ccs2)=O)CCC2C(CCN2C(c2ccc([N+](=O)[O-])cn2)=O)C1 61026,C1(C)(C(=O)NCCCC(C)CO)CN(C(c2ncc3ccccn23)=O)C(C)(C)C1 61027,N1(C(c2cc(C(C)(C)C)n[nH]2)=O)CCC(C)(C)C1C(=O)NCC(F)F 61028,N1(C(C=CC(C)=O)=O)CC=C(CNC(=O)Nc2ncccc2C)CC1 61029,c1(CNC(C2CCC(CNC(=O)CCn3cnnn3)C2)=O)cnccc1Cl 61030,N1(C(C2CC(C)SCC2)=O)C2CCC1CC(C(=O)N(CCO)CC1CC1)C2 61031,Cc1cccc(C(=O)N(CCCNC(=O)C(c2cnccn2)C)C2CC2)c1Cl 61032,c1(CC(=O)NCC2C(NC(c3c(C)n[nH]c3)=O)C2)c(F)cccc1Br 61033,C(CC(C)C)(C(=O)N(C)CCOCCCN(C)C(c1ncc(C)cc1F)=O)OC 61034,N1(CCNC(CC2C(C)(C)C2)=O)CCN(C(=O)C(c2cscn2)N(C)C)CC1 61035,c1(SC(C)C(=O)N(C(C)CCNC(=O)CCN2CCC(F)C2)C)ccccn1 61036,C(=O)(CC(C(C)C)NC(c1cnncc1C)=O)N1CCC(CC)(CC)C1 61037,c1(C(=O)NC2CCC(NC(c3nc(C)sc3)=O)CC2)c(C(C)C)cccc1F 61038,N(C1CCc2cccc(Cl)c21)c1c(C)c(NCCC2CCCCC2O)ncn1 61039,c1(C(=O)NC(CNC(c2cnc(OC)s2)=O)C)sc(F)cc1Cl 61040,C1(C(=O)OCC)CC(OC)CN(C(C(=O)Nc2ccc(F)cc2)C2CCOC2)C1 61041,N1(C(c2cc(OC)ns2)=O)CCC(NCC(C)(C2CC2)OC)C(C)(C)C1 61042,N1(C(c2cnn(C(C)C)c2Cl)=O)CCN(C(=O)CCc2cc[nH]n2)CC1C(F)F 61043,c1(C(N(CC(C)NC(C(C2CCOCC2)OCC)=O)C)=O)[nH]cnc1C#N 61044,N1(C(c2c(C)nc(O)[nH]2)=O)C2CCC1C(C)C(NC(C1CC(C)(C)CN1C)=O)C2 61045,CC(C)C(C)(C)COC(=O)CC(F)(F)c1nccs1 61046,C1(C(=O)NCC(c2nnc(C)s2)NC(C=CCC)=O)CC2CCC1C2 61047,c1(C(=O)NC2CCOCC2C(=O)NCc2nccs2)c[nH]c2cccnc12 61048,c1(C(N2CC=CC(NC(Cn3c(C(C)C)ncc3)=O)C2)=O)ccc2ocnc2c1 61049,N1(C(C(CC#C)CC#C)=O)CC2CCCC(C1)N2C(=O)CC1CCC1 61050,Cc1cc(=NC(=O)c2cc(-c3ccc(-c4cnn(C)c4)cc3)[nH]n2)[nH]n1C 61051,C1(OCC(N2CC(CNC(C3(n4cnnn4)CC3)=O)C2)=O)CCOCC1 61052,CC(C)CC(C)C(=O)N(CCNC(C1CC2CCC1C2)=O)Cc1ccccc1 61053,C1(NC(c2cc(C)n(C3CC3)n2)=O)CCN(C(=O)C(C)C)C12CC2 61054,n1(C(C(=O)NCCN(C(C2(Cl)CC2(F)F)=O)CC)C)cc(C)cn1 61055,c1(C(N(CC(C(=O)NC(CC#C)C)C)C)=O)cc(C)n(C)n1 61056,c1(C(N2CC3CCN(C(CC(C)SC)=O)C3C2)=O)ccnc2ncccc12 61057,C1(NC(c2ccc(CCF)cc2)=O)CCC2CN(C(C3CCCO3)=O)CC2C1 61058,c1(NC(CCNC(C=C(CCC)CCC)=O)C(C)C)cc(SC)ncn1 61059,C(N=c1[nH]c2c(F)cccc2o1)C1(CNC(c2on(C)c(=O)c2)=O)CC1 61060,CCC(CCC(=O)Nc1ccc(SC)nc1)NC(=O)CC(C)c1ccco1 61061,C1(C(=O)NCCCCCN(C)C(C23CC2CCC3(F)F)=O)(OC)CCC(C)CC1 61062,c1(C(=O)NCCC2(CNC(C3(COC)CC3)=O)CC2)n[nH]c2c1CN(C)CC2 61063,CCCC(C)(O)C(=O)N1CCOCC(NC(=O)C(C(C)C)c2ccccc2)C1 61064,C1(NC(C=CC)=O)CC2CCC1N(C(c1cnn(CC(F)F)n1)=O)C2 61065,C(CCCCCNC(c1ccccc1)=O)N(C(=O)C(O)c1ccco1)C 61066,c1(C(N2CC(C)C(NC(c3nc(Br)c[nH]3)=O)C2)=O)ccc2c(c1)C(=O)NCC2 61067,C1(C(N2CC(NC(C=Cc3ccn(C)c3)=O)(CO)C2)=O)CCc2ccnn2C1 61068,C1(C(=O)NCCc2cc(C)no2)(CO)CCN(C(=O)COC2CCCCC2)C1 61069,C1(CNC(C(CO)NC(N)=O)=O)CCN(C(C2(CF)CC2)=O)CC1(F)F 61070,CC1CC(C(=O)NCCN2CCN(CC(F)(F)F)CC2)CCS1 61071,C1(C(N2C(C)C(NC(c3ncoc3C3CC3)=O)CC2)=O)CC2(CC(=O)C2)C1 61072,C(C(C)(C)C(=O)NC1CC(N(C(=O)CCc2cc(C)on2)C)C1)OC 61073,N1(C(c2nc(C(C)OC)sc2)=O)CCC2CN(C(c3cc(N)ccn3)=O)CCC12 61074,Cc1cc(NC(C2(C)CN(C(=O)CCc3ccccn3)C2)=O)cnc1F 61075,c1(C(CNC(C2CC(c3cccc(O)c3)(O)C2)=O)N(C)C)cccc(F)c1F 61076,C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CN(C(=O)C=Cc1ccccc1Cl)C)(C)C 61077,C(=O)(C1CN(C(C2C3CCC(F)(F)C23)=O)c2c(C)cccc21)OCC 61078,N(C(=NCC1CC1(F)F)NC)S(C)(=O)=O.c1(C2(C(=O)NCCN)CC2)ccsc1 61079,C1(CNC(C2(OCC)CC2)=O)(NC(=O)C2=COCCC2)CCCCC1C 61080,C1(C(=O)OC)CC(n2cc(CCO)nn2)CN1C(=O)Cn1cc(C2CC2)cn1 61081,N1(C(c2nncc(OC)c2)=O)CC(O)CCC1C(=O)NCC1(Cl)CC1(F)F 61082,Cc1oc(C(N2CCCCC2CNC(c2ccc(C(F)(F)F)[nH]2)=O)=O)cc1Br 61083,Cc1cnc(C(N2CC3CC2C3CNC(=O)C(C)Cc2ccccc2)=O)nc1 61084,N1(C(C(F)=CCC)=O)CCN(C(C2CCCCC2(C)C)=O)CC1C(C)(C)C 61085,c1(C2(C(=O)NCC(CC)(C)NC(c3conc3C)=O)CC2)ccnc(Cl)c1 61086,C(=O)(C1=C(Cl)CCC(C)C1)NCC(CCCC)NC(c1ccc(Cl)o1)=O 61087,c1(CNC(c2c(C)coc2C)=O)cc(O)nc(CNC(=O)CC(O)C(C)C)n1 61088,C(C(F)(F)C(=O)NCC1(NC(=O)C(n2cc(C)cn2)C)CCCCC1)OC 61089,CC(C)CC(CNC(c1sccc1Cl)=O)C(=O)Nc1ccc2nc[nH]c2c1 61090,CCC(C)(C(=O)NCC1(F)CC(NC(=O)C(c2cnn(C)c2)O)C1)C(F)F 61091,c1(OC)cc[n+]([O-])c(C(=O)NC(C2CN(C(=O)C(C)CSC)C2)C)c1 61092,N1CC(C(N)=O)CCC1(C)C.Cc1ccc(C2CC2C(N)C=O)cc1 61093,C(=O)(CC1=Cc2ccccc2C1)N1CC(CNC(C2CC=CCC2)=O)OCCC1 61094,C=C(C)CCCC(=O)N(C(CNC(c1ccc(OCCC)c(N)c1)=O)C1CC1)C 61095,C#Cc1ccc(C(N2CC(C3(NC(=O)C(C)C4CCOC4)CC3)C2)=O)cn1 61096,N1(C(C2=C(C)OCC2)=O)CC(NC(=O)C(F)CC2CCCC2)CC2(CCC2)C1 61097,Cc1cn2cc(C(N3CCC(N(C)C(C4(O)CCOCC4)=O)C3)=O)sc2n1 61098,N1(C(C2CCN(CC)C2)=O)CC2CCC(C1)N2C(=O)C=Cc1sccc1C 61099,N1(C(C(c2ccccc2)NC(=O)CC(C)(F)F)=O)CCC(CCOC)(OC)CC1 61100,N1(C(C=CC=CC)=O)CCC2CN(C(c3cn(CC4CCOC4)nn3)=O)C2C1 61101,C#Cc1nc(C(N2CCN(CCN(C)C(C3CCCC(OC)C3)=O)CC2)=O)cs1 61102,C(=O)(C1=CCC(C)(C)CC1)NCC1CCN(C(C(CC)OC2CCCC2)=O)C1(C)C 61103,C1(NC(C(C(C)C)C#N)=O)CN(C(C2CC3(CSC3)C2)=O)CC2(CCC2)C1 61104,c1(CNC(c2ccc(F)cc2)C(CC)C)ncc(OC)cn1 61105,C(C)(C(O)C(=O)NCC1CCCCC1C(=O)NC(C1CC2(CCC2)C1)C)SC 61106,C(CCCCCNC(C1CC1c1ccon1)=O)CCO.C1(=O)COCCN1C1CC1 61107,C(=O)(C(Cc1ccccc1)N1CCCC1c1ccsc1)OCC.c12ccnn1N2 61108,C1(CNC(c2c(CC)cco2)=O)CC2CCC1N2C(=O)CNC(c1ccoc1C)=O 61109,N1(C(C(C)NC(C)=O)=O)CCN(CCC2CCCN2C(C23CC(C)C2C3)=O)CC1 61110,N1(C(C(C)SC(C)C)=O)CCC(C(O)CNC(=O)C(C)n2cncn2)CC1 61111,c1(-c2cnc(NC(c3ccc(C#N)cc3)=O)c(O)c2)cnc2ccc(F)cc2c1 61112,CC(C)CC(O)C(=O)NCC1CC1NC(=O)C(c1ccc(Cl)cc1)(F)F 61113,C1(C(=O)Nc2ccccc2-n2cccn2)CC2CC2N1CCOc1ccccc1 61114,N1(C(C(CNC(=O)C(O)Cn2cncn2)OCC)=O)CCCCC1C 61115,c1(OC)ccnc(F)c1C(=O)NCC12CC(CN1C(=O)C(C(C)C)OC)C2 61116,C1(n2cc(CCOC(C)=O)nn2)CCCN(C(c2csc(C(F)F)c2)=O)C1 61117,c1(C(=O)NCC(C)NC(c2ccnc(OC(C)C)c2F)=O)cc2ncccn2n1 61118,Cc1ccc(C(N2CCCC(NC(C3(C4CCCO4)CC3)=O)C2)=O)c(F)c1C 61119,c1(C(=O)NC(CCCNC(c2c(C)scc2)=O)C)ccc(=N)[nH]c1Cl 61120,Cc1cc2c(C(=O)NCCCCCCN(C)C(C3CCCC3F)=O)cccc2o1 61121,C(CN=c1[nH]c(=NCCN2CC3CCCC2C3)[nH]c2c1COC2)c1c(C)n[nH]c1 61122,CCC(C)(C)C(=O)N1CCC(C(=O)Nn2ccnn2)O1.C1(C=O)(CC)CCCC1 61123,C#CCCC(O)CCN(C(C(O)CC)c1ccccc1)CC 61124,CC(C)C(C(=O)OCC(=O)NC(c1nncs1)C)n1cc(Br)cn1 61125,Cc1ccc(C(N2CCCC(C(N3CC(=O)NC(=O)C3)=O)C2C)=O)cc1C 61126,C1(C(N(CCC(N(C(C)C)CCn2cccn2)=O)C)=O)CC2CCC1NC2=O 61127,Cc1nc(CC(N2CC(C)(NC(=O)C(C)NC(c3ccccc3)=O)C2)=O)co1 61128,CCC(C)CC(=O)NC1CCCCC1N(C(=O)CNC(c1ccccc1F)=O)C 61129,CC(C)CC(F)(F)C(=O)N1CCOC(CCNC(=O)CSc2nc[nH]n2)C1 61130,n1(CCCC)nnnc1C(c1c[nH]nc1-c1ccnn1C)NC(c1nnc(C)s1)C 61131,c1(C(=O)NCCCN(C(=O)C(F)(F)COC)CC)cccc2c1NC(=O)CC2 61132,C1(NCCC2CC(OCC)C2)CCS(=O)C1 61133,C(=O)(C(F)C1CCOC1)NC(CN(C(C1(CC#C)CC1)=O)C)C 61134,Cc1c(C(=O)NCC(C)CN(C(=O)C=C2CCC(C)C2)C)ncn1C 61135,C(=O)(CCC(=O)N(C)CCOC1CCCCC1C)OCC 61136,C1(C(N(CCCCCCC)C)=O)CC2(CCN1C(=O)C(CC1CC1)OC)CC2 61137,c1(CC)ncncc1C(=O)NCC(C)NC(=O)Cc1cc(Cl)cs1 61138,Cc1nc(C)c([N+](=O)[O-])c(C)c1C(=O)NC1CCC(NC(=O)C(C)(F)F)C1 61139,C1(C(=O)NCC2N(C)CCCC2)CCN(C(c2cn(C)nn2)=O)C(C)(C)C1 61140,N1(C(c2cc3sccc3[nH]2)=O)CC2CCN(C(=O)CC34CCC(CC3)C4)C2C1 61141,c1(C(N(CC(C)NC(c2n[nH]c3c2COC3)=O)C)=O)cc(Cl)c(Cl)cc1N 61142,C1(NC(=O)CC(CC2CC2)NC(c2cn(CCO)nn2)=O)CCCC(C(N)=O)C1 61143,C(CCCCCNC(=O)C(N1CCCC1)C1CC1)NC(=O)CCCn1ccnc1 61144,C12(CNC(CC(C)N(C(C3C(C(=O)OC)CC3)=O)C)=O)CCCC(CO1)C2 61145,Cc1nc(C#N)c(NNC(=O)N2CC(CSc3ccccc3)OC(C)C2)o1 61146,C1(C(=O)CCN2CCCC2)CCC(=O)N1.C1(C(N(C)C(C2CC2)C2CC2)=O)CC(CCN)C1 61147,C1(C(=O)NC(c2ccc(C(=O)OC(C)(C)C)o2)C)CC(C(=O)O)C12CCC2 61148,N1(C(CC(=O)N(C)C)=O)CC2(CCCC(CNC(c3n[nH]c4c3CCC4)=O)O2)C1 61149,CC(C(=O)N1CC(O)CC1CNC(c1ccc(CCN(C)C)cc1)=O)C(C)(C)C 61150,c1(C(=O)NCCC(C)CCNC(C2CCCOC2)=O)ccc2c(c1)C(=O)NC2 61151,Cc1ncc(C(=O)NC(C2(CNC(=O)CCN3CCCCC3C)CC2)C)c(=N)[nH]1 61152,CCC(CC)CCC(=O)N1CC2CC2(NC(C2(C)C=CCC2)=O)C1 61153,N1(C(C(C)OCC2CCCO2)=O)CC=CC1CNC(=O)Cn1cc(C2CC2)cn1 61154,c1(COC)nc(SCC2(c3nncn3CC)CCC2)no1 61155,C(=O)(C1=C(Cl)CCOC1)N1CCC(N(C(=O)CSCc2ccccc2)C)CC1 61156,C1(NC(c2ccccc2Sc2cccnc2)=O)CCN(C(c2cscn2)=O)CC1F 61157,N1(C(c2cnc(C)[nH]2)=O)CC(NC(c2cc(C(C)(C)C)nn2C)=O)C(C)C1 61158,C(=O)(N1CC(O)CCO1)c1cc(CNC(C(=CC2CCC2)C)=O)nn1C 61159,N1(Cc2cccc(C(C(=O)OC)OC)c2)CCN(Cc2cnc(C)s2)CC1C 61160,C1(C(=O)NCc2n(C)ncc2)CC12CCN(C(c1cnc(Cl)c(Br)c1)=O)C2 61161,C1(NC(C)CC(=O)NS(=O)(=O)Cc2cccnc2)CN(C(=O)C(F)F)CCC1(C)C 61162,N1(C(C=C(C)Cl)=O)CC2(CCCCN(C(=O)Cn3nnc(=O)[nH]3)C2)C1 61163,C(CCC(CC)CC)NC(=NCC=C)NCC(C)(C)CN1CCOCC1 61164,N(C(=NCC(F)(F)C(F)F)NCCSc1ccccc1)C1CCC(OCC)CC1 61165,C12CCCN(C1)C2=O.c1(C2C(NC(C=CC=CC)=O)C2)ccncc1F 61166,c1(C(=O)NCC2CCN(C(c3c(OC)ccs3)=O)CC2C)cnc2ccoc2c1 61167,N1(CC)CCC(CNC(C2C(C)CCN2C(C2CC=C(C)CC2)=O)=O)CC1 61168,c1(C(C)CC)ccccc1OCCNC(=O)C(=O)NC1COCCOC1 61169,N1(C(CC=C)=O)CC2CN(C(=O)CCC3(CO)CC3)CCC2(CO)C1 61170,c1(C(N2CCC(NC(CN(c3ccncc3)C)=O)C2)=O)ccnc(Cl)c1O 61171,c1(-c2onc(-c3ccc(CC)cc3Cl)n2)c[nH]c2c(C)c(Cl)ccc2c1=O 61172,c1(C(N(C(C)CNC(=O)CSCC(F)(F)F)C)=O)csc(C(F)(F)F)n1 61173,C1(C(N2CCC(N(C(c3c(C(C)C)con3)=O)C)C2)=O)CC2(C1)CC(F)C2 61174,C12CCCN(C1)C(=O)CC2.C1(CC=C)CCN(C(c2ccc(C(F)F)o2)=O)C1 61175,n1(CC(=O)NCC2=CCN(C(=O)CC3C=CCCC3)CC2)nc2n(c1=O)CCCC2 61176,CC1CCCCCN1C(=O)C=CCN(C)C(C1COCC1(C)C)=O 61177,C=CCC(C(=O)OCC)NC(=O)CC1C=CC(NC(=O)C(C)C=C)C1 61178,c1(C(=O)NCC2CN(C(CCOC(C)=O)=O)C2)ccnc(S)c1 61179,C1(CC)CN(C(=O)CCOCCCOC)CC1NC(c1sccc1-n1cnnn1)=O 61180,CCC(C(=O)NC1(C)CCCN(C(c2ccn(C)c2CC)=O)C1)C(C)(C)CC 61181,N1(C(CCCC(N)=O)=O)C2CCCC1CN(C(=O)COCCCF)CC2 61182,Cc1cc(C(N2CCC(C)CC2C(N2CC3(CCOC3)C2)=O)=O)cnc1C 61183,C(=O)(C(C)(O)CC(C)C)N1CCCC(C(N2CC(CC)C2)=O)C1 61184,N1(C(C2CCC(NC(c3ccccc3)=O)C2)=O)CCCCCC1C(=O)O 61185,c1(C(N(CC(C)NC(=O)Cn2cnc(=N)[nH]2)CC)=O)ccc(CO)cc1 61186,C1(C2CCOCC2)(C(N2CCN(C(c3c(C)[nH]cc3)=O)CC2C)=O)CC1(F)F 61187,n1(C(C(=O)NC(C(=O)NC(COC)C2(C)CC2)C)C)ccc(C)n1 61188,Cc1nsc(C)c1NC(C1(NC(=O)C(C2CCOCC2)F)CC(F)C1)=O 61189,N1(C(CCC(=O)NC)=O)CCC2C(C1)NC(=O)CN2C(=O)COC1CCCOC1 61190,c1(C(N(C)CC2(NC(c3cnn(C)c3C(F)F)=O)CC2)=O)cnc(P(C)(C)=O)cn1 61191,C1(CC(N2CC(NC(c3ccc(OC)s3)=O)C(C(F)F)C2)=O)C(=O)N(C)N=C1C 61192,C1(C(=O)NC(CCNC(c2c(CC=C)cccc2)=O)(C)C)CS(=O)(=O)CCO1 61193,c1(C(N(C(C)CNC(c2cnsc2)=O)CC)=O)ncoc1C 61194,CC1(CNC(c2coc(C(F)F)n2)=O)CCC(NC(c2cc[nH]c2C2CC2)=O)C1 61195,N1(C(c2c(NCC)ccc(Cl)c2)=O)CCC(C)(C)C(NC(=O)CCC2CC2C)C1 61196,N1(C(CCC)=O)CC2CCC(NC(=O)CCC(C)c3ccc(Br)cc3)CC2C1 61197,C1(NC(C2CCCN(C(C)C)C2)=O)CCN(C(C2(C)CC2)=O)CCC1CO 61198,N1(C(Cc2c(C)ccs2)=O)CCC(NC(C2CCOC2C)=O)C(F)C1 61199,c1(C(=O)NCCC2(O)CN(C(C(C)=O)=O)C2)ccc2c(c1)nc(C)n2C 61200,C(=O)(C1CCCc2nc[nH]c21)C(NN(Cc1c(C)n(CC(F)(F)F)nc1)C)=O 61201,N1(C(C(CC)(F)F)=O)CCC12CN(C(=O)CCC(C)c1ccccc1)C2 61202,CC(C)(C)CCCCNC(C1C(CNC(=O)CCc2ccccn2)C1(C)C)=O 61203,C(=O)(C(O)P(C)(C)=O)NCC(C)CN(C)C(c1cncc2c1CCC2)=O 61204,Cc1c(C(N2CC(CNC(=O)CC3CC3C(F)(F)F)C(F)(F)C2)=O)[nH]ccc1=O 61205,c1(OCC)ccc(Cl)c(C(N2CCCC(CNC(=O)C=CS(C)=O)C2)=O)n1 61206,c1c(F)cc(Br)c(F)c1F.n1(CC(=O)NCC2CCCCO2)cc(COC)nn1 61207,NS(=O)(=O)C1(C(=O)NCCN(C2CCCCC2)C(C2CC(F)(F)CS2)=O)CC1 61208,C(=O)(C(F)C(C)(C)O)NCC1C(NC(c2ccc(CC(C)C)nc2)=O)C1 61209,CC(CCCCNC(C1CCC(=O)N1C)=O)NC(c1ccn(CCF)n1)=O 61210,c1(C(=O)NC2(C(=O)O)CCN(C)C2)ccc2cc(Br)ccc2n1 61211,C(=O)(C(C1CCCO1)C1(C(=O)CCN(CC(=O)NCC2CCCC2)C)CC1)OCC 61212,Cc1cccn(CC(=O)NC2CC(F)CN(C(=O)Cc3ccsn3)C2)c1=O 61213,N1(C(=O)CNC(C23CSCC2C3)=O)CC2(CCOC2)C1 61214,C(=O)(CCCCC(C)C)N1CCC(CC#C)(NC(=O)COCCSC)C1 61215,C12(C(=O)NCCCN(CCCNC(CC(C(C)C)O)=O)C)CCCC(C)(C1)OC2 61216,Cc1cc(=NCCN2CCCC(C)C2)[nH]c(NC(C)CCO)n1 61217,c1(CCCc2n(-c3cn(C)nc3)nc(C(F)F)n2)ccc2cnn(C)c2c1 61218,c1(C(N2CC(C(C)NC(C3(CC=C)CC3)=O)C2)=O)nc(C)ccc1C 61219,CC1(C)COC(CCNc2ccc(C3(C)CC3(F)F)cc2)CO1 61220,c1(C(C)C)nc(C(=O)NCCN(C(C2CC3CC3C2)=O)CC2CC2)cs1 61221,N12CCC(C1)C(C)(C)C(=O)NCC1CC1C2=O.C(CCF)OCCS.CC(C)(C)O 61222,N1(C(C=CC(C)C)=O)CCc2nc(CNC(C3(C)CC(C)OC(C)C3)=O)sc2C1 61223,C(=O)(C(C)(C)CS(C)(=O)=O)N(CCNC(c1c(C)ncn1O)=O)C 61224,N1(C(C(CCC)OCC)=O)CCC(C2CC2)C1C(=O)NC1CCCC1COC 61225,C1(C(N(C(c2cccc(-c3nn[nH]n3)c2)C)CC)=O)CC2CCC1O2 61226,C1(NC(=O)Cn2cc3ccccc3n2)CC2CN(C(=O)CC3CC3)CCN2C1=O 61227,C1(NC(CCNC(COC)=O)=O)CN(C(=O)CC2CC(C)=NO2)C(C)(C)C1 61228,N1(C(CN(C(=O)C=C(C2CC2)C2CC2)CC#C)=O)CCC(N(C)C)C1CC 61229,N1(C(c2c(C)ncs2)=O)CCOCC1CNC(=O)CC12COCC(C1)C2 61230,C1(CNC(c2cnn(CC)n2)=O)CC(C)N(C(=O)CCCN(C)C(C)=O)C1 61231,C12(CCCC1)C(=O)NC2.c1(C(N2CC(CCCCOC)C2)=O)nsnc1O.C 61232,c1(N(c2ccccc2)C(C(=O)Nc2ccccc2)=O)ccc2c(c1)S(=O)(=O)C=C2 61233,N1(C(C(CC)(CC)CO)=O)CCC2(CCC2NC(c2cnc[nH]2)=O)CC1 61234,c1(C(C(=O)Nc2cccc(-c3cn(C(C)C)nn3)c2)(C)N)cccc([N+](=O)[O-])c1 61235,C12(NC(c3c(SC)csc3)=O)CCC(NC(=O)CC3CCOC3(C)C)(CC1)C2 61236,C1(CC(=O)NCC(C)N(C)C(C2CNC(=O)CC2C)=O)CC(C)(C)CCO1 61237,C(=O)(C(C)(C)S(C)(=O)=O)NC1C(c2n(C)ncc2)CN(C(C2CCOC2)=O)C1 61238,CC(C)(C)C(O)C(=O)NC1CCC(CNC(c2cn(C3CC3)cn2)=O)CC1 61239,C(=O)(C1=CCCC1C)NCC1(C(=O)NCc2cn(CC)nn2)CCCO1 61240,c1(C(C)NC(=O)CSc2ncc(C(F)(F)F)[nH]2)cc(Cl)cc(Cl)c1F 61241,C(=O)(CCCCN1CCCCC1)C1C(CN(CCCN)C(C)C)=CC=CC1 61242,N1(C(C2(OC)CCC(C)(C)C2)=O)CCCN(C=O)CC1 61243,Cc1cc(F)c(N)cc1C(=O)NCC(CC(C)C)NC(=O)CC(O)C1CC1 61244,N1(C(CNC(C2(C)N(C)CCC2)=O)=O)CCC(C2CC2)C1 61245,c1(OC)cccc(F)c1C(=O)NC1CCC1NC(c1ccc(C)s1)=O 61246,c1(OC)ccccc1C=CC(N1CCCC1C(C)(C)CNC(=O)CC)=O 61247,N(C1c2ccccc2OC1(C)C)Cc1ccc(OC(F)F)nc1 61248,C#CCCCC(=O)NCCCC(CO)NC(c1ccncn1)=O 61249,N1(C(c2ccc(CC)c(N)c2)=O)CC2CCN(C(c3ccc(CO)nc3)=O)CC12 61250,N1(C(C(C(CC)(C)C)=O)=O)CC2(C=C(C(=O)NCCC(C)O)CO2)C1 61251,C(N=c1nc(N(C)Cc2ccnc(CO)c2)cc(C)[nH]1)C1C(CC)OCCC1 61252,C1(CNC(c2c(C)n[nH]c2)=O)CC2(CC2)CN1C(=O)C(C)CSc1ccccc1 61253,CCCCCC(F)C(=O)N1CCC=CC1C(=O)N(Cc1cn(CC)nn1)OC 61254,C1(N(C(C(C)=CC)=O)C)CS(=O)(=O)C12CCN(C(C1(CC)CCCO1)=O)CC2 61255,C12(C(=O)NCCOC(C(C)C)C)CNCC1(C(F)(F)F)C2 61256,c1(C(=O)Nc2c(OC)ccc(C#N)c2)cccc2c1CCC2NC(=O)OC(C)(C)C 61257,c1(C(N2CCCC(CN(C(c3nc(CC)sc3N)=O)C)C2)=O)cc2occc2s1 61258,C1(NC(=O)CN2CCS(=O)CC2)CCC2(CC1)CN(C(C1CC(F)C1)=O)CCO2 61259,c1(C(N(CC(O)CN(C)C(c2cc(O)ncn2)=O)C)=O)cc2c(=O)cc[nH]c2s1 61260,n1(CC(N2CCC(CN(C)C(C3CCC4CC34)=O)C2)=O)cc(Br)c(O)nc1=O 61261,C1(OC)(CNC(c2nnnn2CC(F)F)CC2CC2)CC2CCCC12.C(CCOC)S 61262,C(=O)(CC1COc2cc(OC)ccc21)NCC(CN(C(=O)C(N)=O)CC)(C)C 61263,C(=O)(CCCCC(N)=O)N1C(C(C)N(C2CCCC2)CCCCCO)CCC1 61264,CN1CC(O)CCC1C(N1CCCCCC1CC(=O)NOCc1nc[nH]n1)=O 61265,C(=O)(CC(F)(F)C(=O)O)NC1CC(C(N2CC(c3cccc(Br)c3)C2)=O)C1 61266,CC(C)CC(F)C(=O)NCCC1(O)CCN(C(c2cc(CCCO)on2)=O)C1 61267,C1(C(C)NC(CN(C(C)C)C)=O)CCN(C(=O)Cc2cnn(C)c2)CC1 61268,C(C)(CNC(=O)Cc1ccc(C)cn1)(CC(C)C)NC(C(C)OCC=C)=O 61269,Cc1c(C(=O)NC2(C)CN(C(=O)CCC3CC4CCC3C4)C2)cncc1Cl 61270,C12(OC)CCC(C(=O)NC3CCC(CC(=O)NC4CC45CCCC5)C3)(CC1)C2 61271,C(C(C)(C)CN(C(=O)CCc1ccon1)C)NC(CC=CC=C)=O 61272,C1(NC(CCc2c(OC)cccc2)=O)CCN(C(c2ncoc2C)=O)C12CC2 61273,C=CCC(CNC(=O)CCCF)C(=O)N(C)CCn1cccn1 61274,Cc1cc(C(=O)NC2CN(C(c3cccc4c3OCO4)=O)C2)c2c(C)noc2n1 61275,N1(C(C(N)C2CC2)=O)CCCCC1C(=O)NC1CCCC1CC1CCOC1 61276,N1(C(C2(C)CCN(C)C2=O)=O)CC2CCC1C(CNC(=O)C=Cc1cc[nH]c1)C2 61277,c1(C(N2CC(NC(CS(CC)=O)=O)C(O)C2)=O)cc(Cl)c(Cl)[nH]c1=N 61278,C(CN=C(NCc1ncccc1C)N1CCC(F)(c2ccccc2F)C1)OC 61279,c1(C(NOCC(=O)NCC2(CC3CC3)CC2)=O)ccncc1F 61280,C(c1nc(C)c(C)[nH]1)=CC(=O)NC(C(C(C)C)NC(c1c(CC)scn1)=O)C 61281,N1(C(CCC)=O)CCCN(C(c2cccc(N3CC=CC3)c2)=O)CC1CO 61282,n1(C2CC(C(N(CC=C)C)=O)C2)cc(-c2ncoc2C)nn1 61283,c1(C(N2CCN(CCNC(CCC(=C)Cl)=O)CC2)=O)coc2ccc(Cl)cc12 61284,N1(C(c2nc(C(N)=O)sc2)=O)CC2CN(C(=O)CC(O)c3ccccc3)CC2C1 61285,C(=O)(C(O)CC(F)(F)F)NCC(N(C)C(C1CCS(=O)(=O)CC1)=O)C1CC1 61286,C(C1=CCN(C)C1)NC(C(C1CCN(C(C2(F)CC2)=O)CC1)C)=O 61287,n1(C(CC)CC)nccc1C(=O)N(C)Cc1cc(C(=O)O)ns1 61288,n1(CC(=O)NCCNC(CSCc2ccc(C)cc2)=O)c([N+](=O)[O-])cnc1C 61289,C1(CNC(CCOC)=O)CC2(CC2)CN1C(=O)C(c1cccc(C(F)(F)F)c1)C 61290,C1(NC(Cn2ncc(CC)c2)=O)C2CC3C(C2)C13C(=O)NC(CC1CC1)CC 61291,c1(CC)ccc([N+](=O)[O-])[nH]1.C12CCN(C1)C(=O)C1CCCN1N(C1CC1)C2=O 61292,c1(CC(=O)N(CCn2cc(-c3cc(C)nn3C)nn2)C)ccc(Br)c2nsnc12 61293,c1(CCCC)ccc(C(=O)OC(C)C(C#N)CC)cc1C(F)(F)F 61294,c1(C(=O)NCC(CNC(C2(CC#C)CCOC2)=O)O)cc(O)cc(F)c1F 61295,c1(C(N2CC(NC(c3ncc(C)cn3)=O)C(C)CC2)=O)cccc2scnc12 61296,C1(CC)CN(C(=O)C(C)CC2CCCO2)CCC1NC(=O)CC1COCC1(C)C 61297,Cc1nc2cc(C(=O)NCC34CCCC3CCN4C(c3cocn3)=O)ccc2o1 61298,Cc1c(C(=O)NCCC(C)N(C(=O)C(F)=CC2CC2)C)nn2ccccc12 61299,C(=O)(CCCC(C)(C)CC)NC1CN(C(c2c(CC)noc2)=O)CC1C(F)(F)F 61300,c1(OC)cc(F)c(CNC2CC2C(=O)Nc2cc(Br)c(F)cc2Br)cc1F 61301,N1(C(NNC(=O)C2N(CC#C)CCC2)=O)CCC(O)C(F)(F)C1 61302,c1(C(N2CC(C(=O)NCCCc3ncc[nH]3)(SC)C2)=O)cc(C)nnc1C 61303,C1(CNC(c2n(CCCC)ncc2)=O)CN(C(=O)C2=CCCC2)CCC1C 61304,n1(CC(=O)NCC(C2CCC2)NC(C(CC=C)(F)F)=O)cc([N+](=O)[O-])nc1C 61305,Cc1nncc(CNC(C2CCCCC2(C)NC(c2ccc(CO)o2)=O)=O)c1C 61306,c1(CC)cc(C(=O)NC2CCCC2NC(C2CCC(=O)N(C)C2)=O)ccc1O 61307,N(C(=NCCF)NCC(CC)C(C)C)CCOCC=C 61308,C1(C(N2CC(C#N)C2)=O)CC(F)(F)CN1C(c1cccc(O)n1)=O 61309,c1(C(=O)NC2CC(CNC(C(C)OCC#C)=O)C2)cnn(C)c1F 61310,c1(C(=O)NC2CCCN(C(c3c(C)cccc3O)=O)CC2)ccc2ccsc2c1 61311,CC(C)C(C)CC(=O)NC1CCCC(Nc2cc(O)ncn2)C1 61312,c1(OC)cccc(C(N2CCN(C(=O)Cc3cccc(C)c3)C3CC23)=O)c1C 61313,C1(C(N2CCCC(c3ccccn3)C2)=O)COC2(CCC2)CN1 61314,c1(OC)ccc2[nH]cc(C(=O)N(c3nc(Cl)c(C(=O)OC)s3)C3CC(N)C3)c2c1 61315,c1(N2C(C)C(NC(=O)C(C)(F)F)CC2)nc(Cl)nc2ccc(Cl)nc12 61316,CON=C(C(=O)N1CCCC(C)(CNC(=O)C=Cc2ccsc2)C1)c1ccco1 61317,C#CCC(CC#C)C(=O)N1CCC2(C1)CN(C(C1CC(O)(C#C)C1)=O)C2 61318,N1(C(C(CSC)C)=O)CCC2(CC1)OCCC2NC(=O)C1=NOC2COCC12 61319,c1(C2(C(N(CC(CNC(Cn3ccc(C)n3)=O)O)C)=O)CC2)ccccc1Cl 61320,C(=O)(C1=NOC(c2ccccc2)C1)NCCN(C)C(C1CCCN1C1CCCC1)=O 61321,c1(C(=O)NCC(C)(C)NC(=O)C(c2cccc(F)c2)F)cncc(F)c1Cl 61322,CC1CN(C(C2CCS(=O)(=O)CC2)=O)CCC1NC(=O)CC=CC(C)(C)C 61323,C(C)(C)(CC(=O)NC(C)C(C)(C)CO)N(C(c1cc(C(C)C)on1)=O)C.C1CC1 61324,N1(C(C(C)N(C)Cc2ccccc2)=O)CC(NC(=O)CC(C)(O)C2CC2)C(C)(C)C1 61325,c1(OC(CC)C)ccccc1C(=O)NC(CNC(C1CCC(C)S1)=O)C(C)C 61326,Cc1nnc2c(C(N3CC(NC(=O)Cc4cncs4)CC34CCC4)=O)cccn12 61327,C1(CC(=O)NCC(C)(C)CNC(=O)Cc2ccsn2)CCCCCO1 61328,CCC(CCCC(=O)NCCC(C)C)NC(=O)CN1CCCC1C 61329,c1(C(=O)NC2(CNC(C3N(C)CC3)=O)CCCC2)cc(Cl)sc1S(N)(=O)=O 61330,C1(CNC(C=C(C)c2cccs2)=O)CN(C)CCN1C(=O)C=Cc1ccccc1 61331,[N-]=[N+]=NCC(F)(F)CCC(=O)N1CC(NC(C2CCNC2=O)=O)CC(O)C1 61332,Cc1oc(C(F)(F)F)nc1C(=O)NCC(C(C)C)NC(c1ncn(C)n1)=O 61333,c1(CNC2C(C(N(CC)Cc3cccc(Br)c3)=O)C2)c[nH]c2cc(Br)ccc12 61334,O(NC(=O)C(CCF)NC(c1ccncc1OCC)=O)C(C=C)C 61335,CC1CN(C(=O)CCc2ccccc2F)CCC1NC(c1ncc(F)cc1F)=O 61336,C1(C(=O)NCC(CC)NC(c2cc(CCO)on2)=O)CCC(O)CN1C 61337,Cc1ccc(C(N2CCN(C(=O)CCc3ccncn3)C(C(C)C)C2)=O)c(O)n1 61338,N1(C(=O)CSC2N(C(CCC)=O)CSC2)C2CCC1CC(CCCN)C2 61339,C1(C(N2CC3(NC(C(CC)C)=O)CC2(COC)C3)=O)CCc2nc[nH]c2C1 61340,Cc1nccnc1C1C(=O)N1.C1(CCCCNC(=O)OC(C)(C)C)C=CCC1 61341,C1(CC(=O)Nc2cn(CCOC)nc2)CCCCC1(F)F.C1C(=O)NCCS1 61342,C1(C(N2CC(CNC(c3c(C)nc(C4CC4)[nH]3)=O)OCC2)=O)CC12CC(F)(F)C2 61343,C(=O)(C1=CCC(C)(C)CC1)NC1(CCC)CCCN(C(c2ccc(=O)oc2)=O)C1 61344,CC1CC(NC(=O)C=CCO)CN1c1nnc(-c2ccoc2)o1 61345,C1(C(C(=O)NC(C(=O)NC)CC2CC2)C)CCCN(C(=O)C=C(C)C(C)(C)C)C1 61346,c1(C(=O)NC(C)CCCCNC(C2CCCN(S(C)(=O)=O)C2)=O)n[nH]cc1[N+](=O)[O-] 61347,CC(CC1CC1)C(=O)NCCc1ccc(Cl)s1 61348,c1(N(CC(=O)NCC(C)NC(=O)C(F)(F)c2nccs2)C)ccccc1 61349,C#Cc1cncc(C(=O)NC2CC(NC(=O)C(c3ccccc3)OC(C)=O)C2)c1 61350,CCC(C)C(CC(=O)OCC1CC(C2CC2)C1)NC(=O)COC1CCC1 61351,c1(C(C)(C(=O)NC2CC2NC(=O)CCn2cccc2)OC)ccccc1C 61352,CC(Cc1cnn(C)c1)C(=O)NC1CCC1CNC(=O)CCn1cc(Cl)cn1 61353,N1(C(C(C)(OC)NC(C)=O)=O)CCC(CCNC(=O)C(C)CC2CCCC2)CC1 61354,c1(N(CC(c2ccccc2)CC)C)nc(=N)nc(N(C)C(C)C)[nH]1.C1(N(C)C)CC(S)C1 61355,C(CC(C(=O)N1CCCC(OC)C1)NC(C1(OC)CCCC1)=O)OCC 61356,N1(C(CCOC(C)C)=O)CC2CCCC(CNC(=O)CC3COCC3O)C2C1 61357,C1(C(N(CCCC(C)C)C)=O)CC(NC(=O)CCC2CCOC2)CCO1 61358,C1(C(=O)NCC(N2CC(N(c3ccccc3)C)C2)=O)CCCCCN1C 61359,C1(NC(C(C)c2ccco2)=O)CC(NC(C2CCC(=O)N(C)C2)=O)CC1O 61360,C#CCC(CC(=O)OC)NC(C1CCC(O)CN1C(C1CC2(C1)CC(O)C2)=O)=O 61361,C#CC1CN(C(=O)CC2CCC2(C)C)CCN1C(=O)CCOC1CCCC1 61362,n1(CC)cc(CNC(=NCCF)NCc2ccccc2Cl)c(O)nc1=O 61363,Cc1ccc(F)c(C(=O)NCC(C(=O)N2CCC(C(C)C)CC2)C(C)C)c1 61364,N1(C(C2C(CCOC)C2)=O)CCC(F)C(NC(c2cscc2C)=O)C1 61365,C1(CC)(NC(c2ccc(F)s2)=O)CCN(C(=O)CN2CCC2C)CC1 61366,C(=O)(CC(=O)NCCn1cc(CC(C)O)nn1)OC 61367,C1(C)(CNC(CC2CCC(NC(Cn3c(C)csc3=O)=O)C2)=O)NC(=O)NC1=O 61368,Cc1cc2ncc1S(=O)(=O)N2.N1(CCCN(C)C(C)C2CC2)CC=CCC1 61369,CC1(C)CCC(C)(C(=O)NCCOCCNC(=O)Cc2ccccc2O)CC1 61370,CCCCCC(O)C(=O)NCCN(C(=O)CC1CC(=O)NC1=O)C 61371,C(=O)(CCCC(=O)NCCC1CCCN(C(C2CC3C=CC2C3)=O)C1)N(C)C 61372,c1(C(=O)NC(CN(C(C(COC)(C)O)=O)C)C)coc2c(F)cccc12 61373,c1(C(N2CCCC(F)(CNC(C(C)=C3CC3)=O)C2)=O)cccn2nccc12 61374,N1(CC(C)Oc2cccc(OC)c2)CCSC2COCCC12 61375,c12ccc(cc1)[nH]c2=O.C12CCN1C2=O.C1(C2(NC(N)=O)CC2)CCCO1 61376,C12(CN(C(=O)CN(c3ccccc3)C)CC#C)CC3CC(CC(C3)C1=O)C2 61377,c1(CC(N2CCC(OCCNC(C(C)S(N)(=O)=O)=O)C2)=O)cc2cc[nH]c2cn1 61378,c1(C(=O)NC2CC(N(C(c3ncn(C(C)C)c3)=O)C)C2)c[nH]c2ccccc2c1=N 61379,N1(C(c2ccc(C(C)=O)nn2)=O)CCC2CN(C(=O)C=Cc3ccoc3)CC12 61380,c1(C(CC)C)nc(C)cc(=NCC2CN(C(c3cnc(C(C)O)s3)=O)CC2C)[nH]1 61381,c1(C(=O)NC(CCNC(C(CC)SC)=O)C)c[nH]nc1S(N)(=O)=O 61382,CC1C2CCCN1C2=O.c1(N(CCC#N)C(=O)C2CC2)cccc(N(C)C)c1 61383,C(=O)(C1=CC(O)C(NC(c2ccc(C)cc2C)=O)C1)NCCOCC(=O)OC 61384,C(=O)(C1=CCCCCC1)NCc1c(C(N2CCCN(CC=C)CC2)=O)[nH]cc1 61385,C1(C(=O)NCCN(C(=O)C(C)(F)c2ccon2)CC)CC(C)CCO1 61386,C(C(O)C(=O)NC1CCC(CCC(=O)NCCN(CCCF)C)C1)=CC 61387,N1(C(C(C)O)=O)CCCC(NC(C2CC3C=CC2C3)=O)CC1 61388,CN1N=C(CC(=O)N2CC3CCN(C(=O)CSC4CC4)C3C2)CC1=O 61389,Cc1cc(C(=O)NC(C2(O)CCCCC2)C(=O)NCC2(F)CC2)n(C)n1 61390,c1(OC)ccc(CS(CC2(OC(C)C)CCCC2)(=O)=O)cc1Br 61391,c1(OCC)cnc(C(=O)NC2CCCC(NC(c3cc(C)cs3)=O)C2)c(Cl)c1 61392,Cc1cc(CC(=O)NCc2occc2C(=O)O)ccc1Br 61393,C1(NC(C2CC(SC)C2)=O)CCCCCCC1NC(=O)CC(C)C(F)F 61394,C1(CCNC(C2(OC(C)C)CCOC2)=O)CN(C(c2nccn2C)=O)CC1C 61395,N1(Cc2ccc(-c3ccc(CS(C)(=O)=O)cc3)o2)C(=O)C2COCCN2C1=O 61396,C1(NC(C2CCN(C(C(CC)n3cncn3)=O)C2)=O)CC(=O)N(O)C1 61397,c1(C(N2CCCN(C(CSCCC)=O)C(C)C2)=O)cccc(P(C)(C)=O)n1 61398,C(=O)(C(F)CC(C)(C)NC(=O)CCC(C)(C)N(C)C)N1CCN(CCC#C)CC1 61399,c1(C(C)C(=O)NCC2CCN2C(=O)COC2(C)CCC2)c(F)cccc1F 61400,C12(C(=O)NCC(C)(Cl)Cl)COC(C1)C(NC(=O)CCC1CCOC1)C2 61401,C(C)(CC(C(=O)NC1CCN(C(C)=O)CC1)N1CCOC(CCC(C)C)C1)SC 61402,N(C(=NCCN1CCCC1)NCC1C(OCC)C1)CC12CC(C#N)(CO1)C2 61403,c1(C(C(=O)NC)N(CC(=O)N(CCO)CCO)C)cc(Cl)cc(Cl)c1.C(C(C)C)N 61404,C#Cc1cncc(C(=O)N(C(C(=O)NC(C#C)Cc2ccco2)C2CC2)C)c1 61405,CC(C)CC(C(=O)N1CC(NC(=O)CCOCC2CC2)C1)C(C)C 61406,CC(C)C(CNC(c1cn[nH]c1)=O)NC(C1(c2cccnc2)CCCC1)=O 61407,N1(C(C(CCCNC(c2c(F)ccc(C)n2)=O)(C)C)=O)CCC2CCC(O)C1C2 61408,C1(NC(COCCOC)=O)CC2(CCCN(C(=O)CC3CCC(F)(F)CO3)C2)C1 61409,CCC(O)C(C)C(=O)NCC1CC(NC(=O)C=Cc2cccs2)C1 61410,c1(CNC(C2(OC)CC2)=O)ccc(C(=O)NCc2nc(C(C)C)n[nH]2)s1 61411,C=CCCC(C(=O)NC1COCC1F)NC(C1CCCN1C=O)=O 61412,n1(CCOC)nccc1C(=O)NCC1(F)CN(C(=O)C(O)CC2CCCCC2)C1 61413,C1(C(=O)OC)CCC(C(=O)NCC2CCN(C(=O)CNS(=O)(=O)C3CC3)C2)C1 61414,C1(CNC(c2c(CC)ocn2)=O)CCN(C(c2occ(C)c2C)=O)C12CC2 61415,c1(C(=O)NC(CN(C)C(C2COC(=O)C2)=O)Cc2ccccc2)ccc(F)cn1 61416,N1(C(C23OCC(CC)(C2)C3)=O)CCC2(C1)CN(C(=O)C(n1cc(C)cn1)C)C2 61417,Cn1cnc([N+](=O)[O-])c1NC(=O)C(N1CCC(N2CCCC2C(=O)NC)CC1)=O 61418,CC1CC(C(=O)NC2(CC3CCC3)CC2)CN(C(c2ccn(CCF)n2)=O)C1 61419,C1(NC(c2nc(C)c(C)[nH]2)=O)CCCC2CN(C(c3cnc(Cl)s3)=O)CC12 61420,Cc1noc(COCC(N2CC(C(C)NC(c3ncsc3C)=O)C2)=O)n1 61421,c1(C(N2CCCC(C)(CNC(C(C(C)C)F)=O)C2)=O)cc2cc(Cl)c(Cl)cc2[nH]1 61422,N1(C(C2(OC)CCOC2)=O)CCC(F)(C(=O)NCC2CCCC(=O)C2)CC1 61423,C1(CCNC(C=C(C)Cl)=O)CN(C(=O)CCCc2ccsc2)CCS1(=O)=O 61424,c1(CC(=O)NCC2CC(C)N(C(=O)Cc3cnns3)C2)cccc(S(C)(=O)=O)c1 61425,c1(C(C(=O)NC2(C(N(CCSC)C)=O)CCC2)F)ccccc1 61426,N1(CC2(NC(CC3(C)CCC3)=O)CC2)CCN(C(C2CC3CC3C2)=O)CC1 61427,c1(C(=O)OCC(N2CCSCC2)=O)cccc2sncc12 61428,CC1CCCC(C)N(C(C2CCC(CNC(c3cccnc3)=O)O2)=O)C1 61429,c1(C(N(CC(C)N(C)C(C2CCCS(=O)(=O)C2)=O)C)=O)ccc2ncccc2c1 61430,CN1CCN(C)C(C(=O)NC2CCC2NC(c2ccc(N)c(F)n2)=O)C1 61431,CC(C)C(Cc1ccccc1)C(=O)NCC1CN(C(c2cccnn2)=O)C1 61432,C1(C(N2C(C(C)C)CC(F)(F)C2)=O)CN(C(=O)CC2CCCC2)CCC1(C)C 61433,Cc1ccc(C(=O)N(CCCNC(=O)CC2(C)CC2(F)Cl)C(C)C)c(O)c1 61434,Cc1nn(-c2ccc(Cl)cc2)cc1CN1CCCCC1C 61435,n1(CC)nccc1CNC(=O)CC1(CNC(=O)C(O)Cn2cncn2)CC1 61436,CC(=O)C(C)CC(C)C(=O)N1CCCCCC(NC(=O)CC(C)(C)CN(C)C)C1 61437,Cc1nn(C)c(C)c1CC(=O)NCC1CCC(C)CN1C(=O)CCc1cnc[nH]1 61438,CCC(C(=O)NC(CCCNC(C1CC1c1nc[nH]n1)=O)c1ccccc1)SC 61439,c1(CC)ncc(C(N2CC(O)(CCNC(=O)CNS(=O)(=O)CC)C2)=O)s1 61440,Cc1ccc(C(N2CC(NC(c3cc(C)n(C(C)(C)C)n3)=O)C3CC23)=O)cc1C 61441,c1(C(N2CCC(CNC(C3(CC)CCCC3)=O)C(C)C2)=O)c(C)ncn(C)c1=O 61442,C(=O)(CCCC(=O)NCC1(C)CCN(C(c2cc(OC)ccc2N)=O)C1)NCC 61443,C(=O)(C1Cc2ccccc21)NC1CCC(CNC(c2nccc3nn[nH]c23)=O)C1 61444,c1(C(=O)NC2CC(C(C)NC(c3ccc(C)o3)=O)C2)cc(Cl)ccc1O 61445,C(=O)(CN=c1cc[nH]cc1)N1C(CNC(C2C(C)SCCC2)=O)CCCC1 61446,C1(NC(=O)Nc2c(C)ccnc2)CCC(C)(C)CO1.C12CCC(CC1)C(=O)NC2=O 61447,C(CC(CNC(C1CC1F)=O)NC(=O)CSc1csc(C)n1)OC 61448,N1(C(C2(C)CCCN(C(=O)CCCCCBr)C2)=O)CC2CCNCC2C1 61449,C=CCC(CC)C(=O)NC1CCC(N2CCN(C(=O)CC(C)C(F)F)CC2)CC1 61450,CC1CC(CCNC(=O)C(C)(C)C)CCN1C(=O)CC1(CO)CCCC1 61451,N1(C(c2c(CC)c[nH]n2)=O)CC(C2CCCCN(C(C3(F)CCOC3C)=O)C2)C1 61452,CC#CCCCC(=O)N1CCC(C(=O)NC2(CSC)CC2)C1 61453,C(CN=c1cc(C)nc(N2CCC(N(C)CCO)C2)[nH]1)(C1CC1)OC 61454,C1(CNC(C2(N(C)C)CCCC2)=O)CN(C(=O)CCC2CC(C)(C)CO2)CCO1 61455,N1(C(COC(C)=O)=O)CCCC1C1CCCN1C(c1cncc(Cl)c1)=O 61456,S(=O)(=O)(c1cccc(F)c1)N1C2CN(Cc3ccc(-c4cccc(C)c4)s3)CC21 61457,C(=O)(CP(C)(C)=O)NCC(C)CN(C(=O)C(C)(C)Oc1ccc(Cl)cc1)C 61458,CCCC(O)C(CO)NC(C1CCCC(NC(=O)CCCSC)C1)=O 61459,C(=O)(N=c1[nH]nc(CC(C)C)s1)C1(CC=C)CCCCN1CC1CC1 61460,n1(CCC(=O)NC(CNC(c2[nH]c(CC)c(Cl)n2)=O)C2CC2)cnc(C)cc1=O 61461,c1(OC)ccc(F)c(OC)c1C(=O)NCC(C)NC(=O)CCCNC(C)=O 61462,c1(C(=O)NCC(C)(CO)NC(c2ccc(COC)cc2)=O)cncc2c1CCC2 61463,C1(NC(C=CC)=O)CCC2CCN(C(=O)CCc3cc(C)cc(F)c3)C12 61464,CC1(C)CCN(CC(N2CC(C(N)=O)(CNC(C3CC=CCO3)=O)C2)=O)CC1 61465,c1(CC(=O)NC2CCN(C(C34CC(C3)C4)=O)CC2F)ccc(O)c(Cl)c1 61466,c1(CC)ncnc(N2CC=C(CNC(C3(C)CCC(=O)N3)=O)CC2)c1F 61467,C1(F)(CNC(C2(C)CCC2)=O)CCCN(C(=O)CC2(C)CCOCC2)C1 61468,C1(NC(C(COC)N(C)C)=O)CC2CC1CN(C(c1nccc(C(F)F)n1)=O)C2 61469,C1(C(N(C)CCNC(c2cc(C(F)(F)F)on2)=O)=O)CCCN(CP(C)(C)=O)C1 61470,c1(C(N2C(COC)CN(C(C3CCN(C)C3C)=O)CC2)=O)cc(C)c(C)nc1C 61471,C1(O)(COCC)CCN(S(=O)(=O)Cc2[nH]nnc2C)C1 61472,c1(C(=O)NC(C(C)NC(c2ccc(CCO)cc2)=O)(C)C)cnn2ccncc12 61473,C(=O)(C(CCCC(=O)OC)N1CCC2(CCSC2)C1)N(CC(=C)C)CC 61474,C1(F)(C(N(CC(CC)O)C)=O)CCN(C(=O)C(C)CC(C)C)CC1 61475,S(=O)(=O)(c1nc(NC2CCC2C)ccc1Br)N1CC(C)NC(=O)C1 61476,CC(C)(Cc1cnn[nH]1)C(=O)NC1CC1NC(C1CC(C)(C)C1)=O 61477,N1(C(c2cc(CCC)[nH]n2)=O)CCN(C)C(C(=O)NC2CCC3CC2CO3)C1 61478,c1(C(N2CC(O)(CNC(c3cnc(OC)s3)=O)C2)=O)ccccc1C(=O)NCCO 61479,c1(OC)noc(C)c1C(=O)N(C)CC1(O)CCN(C(=O)C(c2nc(C)cs2)C)C1 61480,Cc1ccc(CC(=O)N(CC(C)NC(=O)C(C(C)C)N(C)C)C)cn1 61481,C1(CCNCCN(C)C(=O)OC(C)(C)C)CC(=O)OC1(C)C.C12(CCC1)C(=O)N2 61482,c1(NC(=O)NC(C(c2ccccc2)OC)C)n[nH]c(C(=O)OC(C)(C)C)n1 61483,C1(COC)CN(C(c2cnn(C)c2N)=O)CCN1C(c1ncccc1Br)=O 61484,c1(OC)cc(CNCc2ccncc2C(F)(F)F)cc2cc(C)oc12 61485,c1(C(=O)NCC2(F)CCN(C(C3(C)C(CC)CCC3)=O)C2)ccn2c1CCCC2 61486,N1(C(CCSCC=C)=O)CCCC(NC(=O)CNC(=O)NC)C1 61487,C1(COC)COCCN(C(=O)C(CC2CCCCC2)OC)C1.C12(O)CN(C1)C2=O 61488,C(=O)(C(C)CC(C)C)N1CC(C(=O)N(C)Cc2cnccn2)(COC)C1 61489,C(C(=O)N1CC(O)(CNC(=O)CC2CCSCC2)C1)(C(C)(C)C)NC(C)=O 61490,C12(C(=O)NC3(C)CN(C(c4cc[nH]n4)=O)C3)CCCC1CS(=O)(=O)C2 61491,C1(=O)CCC(C)(C)C(=O)NCC2(F)CCN1CC2.C1(CC)OCCC1C(=O)OC 61492,C(=O)(C(C)(CCNC(=O)OC(C)(C)C)C(F)(F)F)NC(CNC(C1(CC)CC1)=O)C 61493,N1(C(C(N2CCCS2(=O)=O)C)=O)CCCCC1CNC(c1ccncc1F)=O 61494,c1(C(C(=O)NC2CC(NC(=O)CSc3ccccn3)C2)OC)ccccc1O 61495,CN1CCN(C(=O)C(C(C)(C)C)NC(=O)Cc2cscn2)CC1(C)C 61496,c1(OC)cc(C(N2CC(NC(C3CCOC3(C)C)=O)C(O)C2)=O)cc(N)c1O 61497,Cc1ccncc1CC(N1CCC1CNC(c1cc(C)n(C(C)(C)C)n1)=O)=O 61498,c1(NC(C)CCC2(C)CCOC2)cc(F)cc(Cl)c1 61499,N1(C(CC2C(NC(C3CCC(=O)O3)=O)CC2O)=O)CCCOCC1 61500,c1(-c2cc(C(N3CC4CC4(Nc4cnccc4Br)C3)=O)on2)cccc(F)c1F 61501,N1(C(C(C)C(C)(C)C)=O)CCC2(CCCN(C(C3CCS(=O)(=O)C3)=O)C2)C1 61502,c1(C(N(CCNC(CC(CC)C2CC2)=O)CC)=O)cc2c(OC)c(F)ccc2[nH]1 61503,S(=O)(=O)(c1ccn(C2CC2)n1)N1CC(C)(NC(=O)CN)OCC1 61504,C1(C(CNC(=O)CSCC(F)F)(C)O)CCCN(C(=O)C(F)F)C1 61505,N1(CS(C)(=O)=O)CCN(C(C2CCN(C(=O)CCc3cnc[nH]3)C2C)=O)CC1 61506,n1(CC)nnc(C)c1CNC(C1(CCCO)CCCC1)=O 61507,C12(C(=O)NCC(CN(C)C(C3(C(F)F)CCC3)=O)O)COCC1C2(F)F 61508,c1(NC(=O)OCC)cccc(C(=O)NCC(CO)NC(=O)CC2(O)CCOC2)c1 61509,c1(NC(C(C)C)=O)ccccc1C(=O)NC1CN(C(c2ncccn2)=O)CCC1 61510,C1(O)(CNC(C2(OC)CC2)=O)CCN(C(=O)C(C)(CO)OC(C)=O)C1 61511,N1(C(C2CCC(N(C)C)CC2)=O)CC2CC1CN2C(=O)CN(CC(C)(C)C)C 61512,c1(C(=O)NCC2C(C(=O)NCC(COC)C)CCO2)nccc2cc[nH]c12 61513,C(=O)(C(F)C(CC)CC)NC(CN(C(C(C)OCC=C)=O)C)C 61514,N1(C(C(C2CCC(=O)N2)C)=O)CCC(C)(NC(c2ncccc2N)=O)CC1 61515,C1(C(=O)NCC2CN(C(CC(C=C)C)=O)C(C)(C)C2)CC2CCC1C21CC1 61516,Cc1cn2c(n1)C(C(=O)NC1CCCCC1NC(c1cnc[nH]1)=O)CCC2 61517,C1(CC(=O)NC2CCC(CCNC(C3(C=C)CCC3)=O)C2)(C(F)(F)F)CNC(=O)C1 61518,C1(C(=O)NCCOC)CCC12CN(C(c1ccc(NC(C3CC3(C)C)=O)cc1)=O)C2 61519,c1(-n2cc(C(CC)(C)O)nn2)cc(C(=O)NC(CO)CC(F)F)ccn1 61520,C1(CNC(c2c(C)ncn2O)=O)CCCCN(C(C2(C)CC=CCO2)=O)C1 61521,C1(NC(c2c(C)c(F)ccc2)=O)CC2CC(NC(c3nnccc3C)=O)CC2C1 61522,C1(C(N(C(C)CCNC(C2CCCC2)=O)C)=O)CCCC(F)(F)CC1 61523,c1(OC)cc(C(=O)NCC(C(C)C(C)C)NC(=O)C(C)SC)cc(N)c1 61524,N1(C(CCC)=O)CCC(C(=O)NCC2CC(C(C)(C)C)C2)=C(F)C1 61525,CCC(F)(F)CC(=O)N1CC2CC2(CNC(=O)C2=C(C)OCC2)C1 61526,c1(C(=O)NCC(C2(O)CCN(C(CC3(C=C)CC3)=O)C2)C)cc(OC)cc(Cl)c1 61527,c1(C(=O)NCC(C2CCOC2)NC(c2occ(C)c2)=O)cc2c(ncn2C)s1 61528,C1(C(=O)NC2(C)CCC(NC(C(CCC)(C)C)=O)CC2)CCc2cnnn2C1 61529,c1(C(N(C(C(=O)OC)C)C)=O)ccc(CNC(=O)CC2C=CCCC2)s1 61530,c1(OCC)ccc(C(=O)NCCCN(C(=O)CCn2ncn(C)c2=O)CC)cc1 61531,C1(NC(c2ccc(SCC3CC3)cc2)=O)CC2CC1N(C(c1n[nH]cc1Cl)=O)C2 61532,CC1(C)CC1(Cl)C(=O)NC1(C2CCCN2C(c2cscc2Br)=O)CC1 61533,C(C(C)C(=O)NCC(C)N(C(=O)Cc1[nH]cnc1C)C)OCC 61534,c1(C(N2C3C(NC(c4nc(C)sc4C)=O)CC(C3)C2)=O)coc2c1C(O)CCC2 61535,S(=O)(=O)(c1c[nH]c(C(N2CCN(C(C3(C#N)CCCO3)=O)CCC2C)=O)c1)NC 61536,N1(C(=O)Cn2nnc(-c3ccccc3)n2)CCN(C(C2CC2)=O)CC1CCO 61537,c1(CN(C(C2CCC(F)CC2)C(=O)NCCC)C2CC2)cccc(Br)n1 61538,n1(CCC(=O)N(C(C(=O)N(C)CC)C)C)cc(CN(C)C(=O)C2CC2)nn1 61539,C1(CN(C)C(c2c[nH]c(C(F)(F)F)c2)=O)CCN(C(C23CC(CO2)C3)=O)CC1 61540,C(C)(C)(CCCNC(=O)C(C)OC1CCCC1)NC(C=C(C)C1CC1)=O 61541,c12ccc([nH]1)C(=O)NCC1(CC1)CNC2=O.c1(COC)ccccc1 61542,C(=O)(C(C)CCCC(C)C)NC1C(CC)CN(C(c2cc(C(C)C)[nH]n2)=O)CC1 61543,C12CCCN1C(=O)CNC2=O.c1(C(C2CC2)C2CC2)nn[nH]n1 61544,c1(NC)ccc(C(N2CCCC2C(C)(C)NC(=O)C(F)=CCCF)=O)nc1 61545,Cc1cc(NC(=O)CCCCCN(C(=O)C(C)S(N)(=O)=O)C)cc(Cl)c1 61546,C1(NC(=O)Cn2nccn2)CC2(C1)CN(C(c1ccc(C(F)F)cc1F)=O)C2 61547,CC1CCC(C)C(CN)N1C(=O)NC(c1nccn1C1CC1)=O 61548,c1(C(N(C)CC2(NC(C(c3ccc(Cl)cc3)C)=O)CC2)=O)csc2c1CCCC2 61549,C1(CN(C(C(C)=C2CC2)=O)C)CCCCN1C(=O)C(c1ccccc1Cl)C 61550,c1(CCC(=O)N(CC(N2CCN(C(=O)CN(C)C)CC2)=O)C)nnc(S)nc1O 61551,C(=O)(C1=NN(CC(C)C)C(=O)CC1)N1CC2CN(C(CCOC)=O)C2C1 61552,C1(NC(N(c2ccc(Cl)cc2)CC#C)=O)CCc2nnc(C)n2C1 61553,C1(CCC(=O)Nc2cn(CC)nc2)CCCN(C(=O)CCC(=O)C2CCCC2)C1 61554,N1(C(c2ccc(C)cc2)=O)C2CCC1C(C)C(NC(=O)CCCc1ccsc1)C2 61555,C12C3CN(CC13)C(=O)CCNC2.N1(C(=O)C2CC2)CCC1.c1(C=O)cccs1 61556,c1(OC)cc(C(=O)NC(C)C(C)NC(c2cnc(C(C)C)o2)=O)cc(F)c1F 61557,c1(NC(=O)CC2CCC(NC(c3cncc(F)c3)=O)C2)cnc(I)cn1 61558,N1(C(C(CCC)(C)C)=O)CCC2OCCN(C(c3ccc(S(N)(=O)=O)o3)=O)C2C1 61559,c1(CNC(CN(S(C)(=O)=O)C)=O)ccc(CCNC(C2CCCC2F)=O)cc1 61560,C1(CCC(=O)NC(CC)Cc2nn[nH]n2)CCCCC1 61561,c1(OC)cc(N)c(F)cc1C(N1CC2CCC1CN2C(=O)Cc1cnns1)=O 61562,c1(CCNC(C(n2cc(CCCSC)nn2)C)=O)ccc(O)cc1C 61563,C1(C(N(C2CN(C(c3ncccc3Br)=O)CC2O)C)=O)CC2(CCCC2)CO1 61564,C1(C)(C(=O)NCC(CNC(C2C(C(C)(C)C)CC2)=O)(C)O)COCCO1 61565,C1(=CC(=O)NCCCN(C(C(C)OCC=C)=O)CCC)CCC(C(C)(C)C)CC1 61566,C(C(CC)(CC)C(N)=O)NC(=O)Nc1cncc(C(CSC)(C)C)c1 61567,C1(NC(c2n(C)ccn2)=O)CC2(CCN(C(=O)C#CC3CCCCO3)CC2)C1 61568,c1(C(=O)NCC(CNC(Cc2cncc(C)c2)=O)(C)O)cn2cccc(Cl)c2n1 61569,Cc1cnc(C(=O)NCC(C)(F)CNC(c2c[nH]nc2C2CC2)=O)cc1Br 61570,C1(F)(C(=O)NC(C)Cn2cccn2)CCN(C(=O)C(C)N(C)C2CC2)C1 61571,C(C(CC1CCCC1)C(=O)N1CCC(C(N)=O)C1)NC(C(OC)OC)=O 61572,c1(CCC)ccc(C(N2CC(NC(=O)CC(C)(F)F)C3(CC3)C2)=O)cc1[N+](=O)[O-] 61573,CCN=c1cc(C(N2CC(NC(c3cnncc3C)=O)C3(CCC3)C2)=O)cc[nH]1 61574,C(c1ccccc1C)=CC(N1CCC(CC(=O)N(C2CCN(C)C2)CC)CC1)=O 61575,n1(CC(=O)NCC(C2CCOC2)NC(=O)Cc2cccs2)cc(Cl)cn1 61576,c1(OCCCC(=O)NCCN(C(C2(C)CC2C)=O)CC)ccc(Cl)cc1C 61577,c1(C(=O)OC)ccc(CNC(=O)C(F)C(F)(F)F)cc1F.C12(C)CCCN1C2 61578,c1(N2CC(C)CN(C)CC2)[nH]c(=NCCS(C)=O)nc2scnc12 61579,C1(CCC)CCCC1C(=O)NC1CCN(C(C)=O)C1.C12(CCCC1)C(=O)N2 61580,C(=O)(CCC(F)(F)C(F)F)NC(C)CCCCNC(C1C(SC)CCC1)=O 61581,C(=O)(C1=CC2CCCC12)NCCOCCN(C)C(c1cnn(C)c1Cl)=O 61582,N1(CCC)CCC(C(C)NC(CONC(=O)C2(COC)CC2)=O)CC1 61583,C1(NC(c2cccc(C)c2F)=O)CN(C(=O)CC(O)C(C)C)C2(CCCCC2)C1 61584,c1(C(=O)NC(CC)(C)CNC(=O)Cc2cncs2)cnc(C)c(C#N)c1 61585,C12(CNC(c3c(C)nn(C)c3)=O)CCC(C1)N(C(C1CCC3CC1CO3)=O)C2 61586,c1(C(=O)NCC(C)N(C)C(c2c[nH]c(=O)cn2)=O)cnc(C(F)F)cn1 61587,C1(NC(c2c(CC)csc2)=O)CC=C(C(=O)NCCc2ccon2)C1 61588,n1(CC)cnc2c(NCc3cnn(CC)c3)[nH]c(=NCC(C(C)(C)C)SC)nc12 61589,C12(NC(CC3(C=C)CCCCC3)=O)CCCC1N(C(c1ccc(F)o1)=O)CCC2 61590,CC12CCN(C1)NC2=O.C1(C)CC(=O)N(c2ccccc2F)C1.c1ccccc1F 61591,C12(C(N3CC(C(N)=O)(CNC(c4cccc(CC)n4)=O)C3)=O)CCCC1CCC2 61592,N1(C(c2noc(CC)c2C)=O)CCC2CCN(C(c3c(Br)nnn3C)=O)CC12 61593,CC1(C)CC(NC(c2snnc2C2CC2)=O)CCN(C(=O)Cc2ccsc2)C1 61594,C#Cc1ccc(CC(N2CC(NC(=O)CCC3CCCOC3)C(CC)C2)=O)cc1 61595,n1(CCC(N2C(C(C)(F)F)CCC2)=O)nc(O)c2c1CCCC2 61596,c1(OC(C(=O)OC(CCCCC)C)C)cc(F)ccc1C.C12=CC=C(C=C1)C2=O 61597,c1(NC2C(CO)CCCCC2)nc2ccccc2nc1NC1CC2CCC1O2 61598,C1(C(N2C(CC)CC2)=O)CCN(C(=O)Cc2nccn2C)C1(C)C 61599,c1(NC(C(CC2(NC(=O)OC)CCC2)F)=O)cccc2c1oc1ccccc21 61600,Cn1c(O)nc2cc(C(=O)NCCC3CCN(C(C4CC(C)(O)C4)=O)C3)cnc12 61601,CN(C)S(C)(=O)=Nc1nc(C(=O)NC2CN(C(c3csc(C4CC4)n3)=O)C2)cs1 61602,c1(NCC(C)S(C)=O)[nH]c(=NCc2nc(Br)n(C)n2)nc2c1cnn2C 61603,N1(C(CCCOCC=C)=O)CCN(C(=O)C(C)c2ccco2)CC1c1cn[nH]c1 61604,C(c1cccnc1)=CC(N1CCC(OCCN(C(c2onc(C)n2)=O)C2CC2)C1)=O 61605,N1(C(C2CC3CCCC3C2)=O)CC2CCCN(C(=O)CSC(F)(F)F)C2C1 61606,C(CS(=O)(=O)CC(=O)N1CCC(C2CC2)C1C(N(C)C[Si](C)(C)C)=O)OC 61607,C1(CC#C)CCCN(S(=O)(=O)CC2(C(=O)OCC)CCS(=O)(=O)C2)CC1 61608,C1(NC(=O)NCc2c(OC(F)F)cc(C)c(F)c2)CCCn2cncc2C1 61609,C(=O)(N1CC(C)(O)CO1)C1CN(C(C(C)NC=O)=O)CC1C 61610,C(CC(O)CNC(=O)C(C)N(C(=O)CN1CCNC1=O)C1CC1)OC 61611,c1(CN2CCC(C(=O)NCc3ccc(Cl)cc3F)C(O)C2)cc(Cl)c(O)c(Cl)c1 61612,N(C)(C1CCc2c(F)cccc21)C(C(C(CC)C)C)=O 61613,C1(C(N(CCCCCCNC(c2cccc(Cl)c2)=O)C)=O)CCCCC(=O)N1 61614,CC1(C)C(C(N2CCCC(CCO)C2)=O)CCN1C(C1CSC1)=O 61615,N1(C(CN(S(C)(=O)=O)C)=O)CC(NC(=O)CCSCC(N)=O)C(C)(C)C1 61616,C1(CNC(=O)Nc2c(OC)ccc(F)c2)(CO)COCC2CCCCN12 61617,c1(C(=O)NCC(C2CC2)OC)n[nH]c2c1CN(C(=O)C(C)CC1CCCC1)C2 61618,C1(NC(C(CCC)OCC)=O)COC2(C1)CN(C(c1cc3c([nH]1)CCCC3)=O)C2 61619,c1(CC(=O)NCC(C)(C)NC(C2CCC2n2cccn2)=O)cccc(Cl)c1 61620,c1(C(=O)OC)ccc(CC(N2CCN(C(c3cccc(Br)c3)=O)CC2)=O)cc1F 61621,CC(CN=c1nc(C(F)(F)F)[nH]c2ccccc12)N1CCN(CC2CC2)CC1 61622,C1(CNC(=O)CCc2ccc(Cl)s2)CCN(C(c2nnc(O)nc2O)=O)C12CC2 61623,c1(NC(CCC(C)(C)NC(=O)CCN=[N+]=[N-])=O)cncc2ccccc12 61624,c1(CCNC(C(=O)NC(C2CCCN2)CC)=O)ccc(C2CC2)s1 61625,c1(C(=O)NC(CNC(C=CC2C(C)CCC2)=O)(C)C2CC2)nc(F)ccc1Cl 61626,C1(CCC(=O)NCC(=C)CCNC(=O)C(O)c2ccsc2)CCCC(=O)N1 61627,c1(-n2c(C(C3CC3)OC)nc(CC(C)C)n2)nc2ccccc2c(=O)n1C 61628,C(=O)(C(C)(C)CN=c1[nH]c(=NCCC2CC(C)C2)[nH]c2ccccc12)NCC 61629,C1(CCC)CN(C(c2ccccc2Cl)=O)CC1C(=O)N(C)Cc1cc(=O)cc[nH]1 61630,C1(C(N)=O)CC(OC(c2cnccc2Cl)=O)C(=O)N1Cc1ccccc1 61631,Cc1cc(=NCCC2CCCN2Cc2cc(C(=O)O)c(F)c(F)c2)[nH]cc1S(C)(=O)=O 61632,CON(C)S(=O)(=O)c1cccc(C(N2CC3CC2C3NC(C2CC(F)C2)=O)=O)c1 61633,Cc1cc(C(=O)NCc2cccc(C(=O)NC(C)C(F)(F)Cl)n2)c(C)s1 61634,CC1(C)CCN(C(C2CSCCS2)=O)CC1NC(c1coc(Cl)n1)=O 61635,C(N=c1ccc(C#N)c[nH]1)C1(C(=O)NC(C)C(=O)NC2CC2)CCOC1 61636,Fc1ccc2c(c1)C(Nc1cc(NC3CC4CCC3CC4)ncn1)CC2 61637,Cc1ccc(C(N2CC3CC2C3NC(C2(C(c3ccccc3)=O)CC2)=O)=O)c(F)c1 61638,c1(CC(=O)NCC(CCNC(CCC=CC)=O)(C)C)coc2c(F)c(F)ccc12 61639,C(C(C)C(F)(F)F)NC(CC1C(NC(C2(C=C)CCC2)=O)CC1O)=O 61640,c1(C(=O)NCC(CC)N(C(=O)CC2CCOCC2)C)cnsc1C 61641,CCN=C(NCCS(=O)(=O)c1ccccc1C)N1CCC2(CCCC2)C1 61642,CC(=O)n1ncc2c(C(=O)NC3CCS(=N)(=O)CC3)cc(C3CC3)nc12 61643,CN1CCN(C(C2CNC(=O)N2)=O)CC1CNC(c1ccc(-c2ccco2)o1)=O 61644,Cc1oc(S(N)(=O)=O)cc1C(N1CCCN(C(C2CC23CCCC3)=O)CCC1)=O 61645,CCS(=O)(=O)c1cnc(O)c(C(=O)NCCCCCN(C)C(C2CC2(F)F)=O)c1 61646,C(=O)(C(C(C)(C)C)NC(CCC(O)C1CCCC1)=O)N(C)CC1CNC(=O)C1 61647,C1(C(N(CCNC(CCOCCOC)=O)C)=O)C(CCCCSC)C1(F)F 61648,c1(C(=O)NC23CCCC(NC(CCCC(=C)C)=O)(C2)C3)cc(F)c(F)c(C#N)c1 61649,c1(C(=O)NC2(CO)CN(C(CC3CNC(=O)O3)=O)C2)cc2n(n1)CCO2 61650,S(=O)(=O)(C1CCCC1(F)F)N1CCC(C)C(C(=O)O)C1 61651,c1(N(C(=O)CP(C)(C)=O)C2(c3ccccc3)CC(NC(C)=O)C2)ccc(F)c(F)c1 61652,c1(OC)cccc(C2(CNC(=O)NC3CC3C3CC=CCC3C)CC2)n1 61653,c1(OC)ncc(NC(c2ccc(OCc3ccc(F)cc3)cn2)=O)cn1 61654,C1(C(=O)NCC2(F)CN(C(C(C3CC3)SC)=O)C2)CCN(CC(C)C)CC1 61655,c1(C(N2CCC(CCCNC(c3ccn(C)c3)=O)CC2)=O)ccc2c(c1)OCO2 61656,CCC(CC(=O)N1C(CNC(=O)CCc2cnn(C)n2)CC2CCCC12)C(C)C 61657,c1(C(=O)NCCC23C(CN(C(C(C)(C)C(F)F)=O)C2)CC3)cnc2occc2c1 61658,C1(C(N(CCOC)Cc2ccccc2)=O)CC(c2ccccc2)CN1 61659,CCCCC(C(=O)NCCC1CCCCN1C(=O)CSCCOC)C(C)C 61660,c1(CC(=O)NCC(C)NS(CCCC)(=O)=O)nc(Br)n2c1CCCC2 61661,N1(C(C(COC)OC)=O)CC2CCC2(CNC(c2cnccc2OC)=O)C1 61662,C1(CC#C)(C(=O)NC2CC(CCNC(c3cncn3C)=O)C2)CCCO1 61663,C1(OC)CC(CNC(=O)C(F)Cc2ccccc2)N(C(=O)CCC2OCCO2)C1 61664,n1(CCC(=O)NC(CC=C)CNC(=O)C(F)(F)C(C)O)nc(O)c2ccccc12 61665,N1(Cc2nc(C(=O)OCC)sc2)CCCC(CO)(NC(=O)C(C)C(C)(F)F)C1 61666,N#Cc1cc(C(N2CC(NC(C3CCCOC3)=O)CC(F)C2)=O)ccc1F 61667,n1(CC(=O)NC(C2CN(C(=O)C(O)CC3CCOCC3)CCO2)C)ncccc1=O 61668,CC1(C)CCOC1C(=O)NCC1(C(=O)Nc2cncc(Cl)c2)CC1 61669,C(CCCC(O)C(=O)NC1(c2nn[nH]n2)CCOCC1)NC(C1CC(C)(C)C1)=O 61670,N1(C(c2cn(CCNC(C3CC3Cl)=O)nc2)=O)CCn2cncc2C1 61671,c1(CC(N2CC(COC)(CNC(=O)CC3CCCC3(F)F)C2)=O)ccc(F)cc1Cl 61672,c1(C(=O)NC(C(C)C)CNC(=O)CCc2cncnc2)cccnc1O 61673,C(=O)(C(O)C1=CCCCC1)NC(C(=O)NCC(C#C)OC)CC(=C)Cl 61674,c1(C(N2CC(NC(C=CCOC)=O)(CO)C2)=O)ccnc(N2CCC(C)CC2)c1 61675,CC(CC(C)NC(c1cnn2ccccc12)=O)N=c1[nH]c(Cl)nc2c1SCC2 61676,CC(C)C(C)CC(=O)NC1(C2CCCN2C(=O)CN2C(=O)CCCC2=O)CC1 61677,c1(N(CC(c2ccc(Cl)cn2)OCC)C)ccc(S(=O)(=O)NCCSC)c(Br)c1 61678,C1(C)(OCC)CN(N2CCCC(c3nc(C)c(C)[nH]3)C2)C1 61679,C(C(C)(C)CN(C(=O)CN1CCCC1CO)C)NC(C(C1CC1)OCC)=O 61680,C1(OCC)CCC(C(=O)OCCSC)CC1.N12CCCC1c1cscc1C2=O 61681,c1(NC(=O)NC(C2CC(F)(F)C2)CC)cc(O)ncc1Cl.C1(S)CC1 61682,C12(NC(c3c(CC)csc3)=O)CCCC1CN(C(=O)Cc1ccc(CC)s1)C2 61683,N1(C(C(C(CC)C)N)=O)CCC2CN(C(=O)Cc3cccc([N+](=O)[O-])c3)CC12 61684,C=C(Br)CN=C(NCCOc1ccc(F)c(F)c1)NCC1CC(C)(C)C1 61685,N1(C(CC2CC(OC)C2)=O)CCCC(C)(NC(=O)C(=O)C(C)C)C1 61686,c1(OC)ccc(CN(C(c2ccccc2OC)C(=O)NC2CCCC2)C)nn1 61687,CCC(C(=O)OC)C(=O)NC1CCC1NC(c1cn(C(C)C)nn1)=O 61688,c1(C2CN(C(CCC3CC(NC(C=CC(C)(C)SC)=O)C3)=O)C2)cc(O)n[nH]1 61689,O(NC(=O)CCC(CC)NC(=O)C(CSC)CC1CCCC1)CCC#C 61690,N1(C(c2c(N)ccc(C)c2)=O)CCC2(CCN(C(C3(C(N)=O)CC3)=O)C2)C1 61691,C1(CN(C(C(C)(C)NC(=O)NCCC)=O)C)CCCCN1C(C1C(C)C1C)=O 61692,CC1(CNC(C23CCCC2CCC3)=O)CCCN(C(c2cc(N)c(F)cn2)=O)C1 61693,c1(C(N(CCOC)CCNC(=O)CO)=O)c(C)nc(C(C)C)nc1O 61694,C1(C)(NC(C2CC(=C)C2)=O)CCN(C(=O)CCn2c(-c3cccs3)nnc2S)CC1 61695,n1(C(C=C)C)nc(C2CCOCC2)nc1Cc1ccccc1Cl.[nH]1ncn(C)c1=O 61696,CC(C)CC(C(=O)N1CCC(C(=O)NCc2cocn2)CC1)N(C)C 61697,CC1N(C(=O)CC2N(C(C3CCCSC3)=O)CCC2(C)C)CCOC1(C)C 61698,C=C(C)C(CC(=O)N1CCC(F)(CNC(=O)CCCC2CCCCC2)C1)OCC 61699,c1(C(=O)NC(C2CCN(C(c3csc(C(N)=O)n3)=O)C2)C)cccc2sccc12 61700,C1(C)(NC(CCSCCCC)=O)CN(C(c2scnc2C(C)C)=O)C1.OCC 61701,Cc1cc2ncnc(NC3CC4CN(C(=O)Cc5c(Cl)cnn5C)CC34)c2[nH]1 61702,C(C(CNC(C1C2(CC2)C12CC2)=O)S(C)(=O)=O)NC(C(c1c(C)cccc1)C)=O 61703,c1(C(N(CC(C)NC(c2c(C)cc[nH]2)=O)C)=O)cc2ncn(C)c2cn1 61704,N1(C(c2cc3cccnc3o2)C(=O)NCCCC)CCNC(=O)C(F)(F)C1 61705,C1(CC)(CC)CC(NC(=O)C(O)Cc2ccccc2)CN1C(c1cnc(Cl)[nH]1)=O 61706,c1(C(=O)NCC(CNC(=O)C=Cc2cn[nH]c2)O)cccc(F)c1[N+](=O)[O-] 61707,C1(C(N(C2CCCCC2)CCNC(C2CC2C2CCC2)=O)=O)Cc2nncn2C1 61708,C1(c2nc(C)c(C)[nH]2)CCCN1N1Cc2ccccc2C(C)C1 61709,C1(C(=O)OC)CC=CCC1C(N1CC(C(N2CCN(CCO)CC2)=O)C(F)C1)=O 61710,C1(O)(C(N2CC(OCC(F)F)C2)=O)CCN(C(c2cc(Cl)n[nH]2)=O)C1 61711,C1(NC(=O)NCCSC)CN(C(C2(C)SCCCS2)=O)Cc2cccn2C1 61712,O=C(C(F)(F)C(F)(F)C(F)(F)C(F)(F)Cl)N1CCC(C(O)C(F)(F)F)CC1 61713,c1(CNC(=O)CSC2CCCCO2)ccc(CNC(=O)CCc2cnc[nH]2)cc1 61714,CC(O)C(F)(F)C(=O)N1CC=CC(NC(c2ccc(C(O)CF)cc2)=O)C1 61715,c1(CC(=O)NCC2CCC2NC(C2CCC3CC3CC2)=O)c[nH]c2cccc(F)c12 61716,c1(NC2N(C(=O)OC(C)(C)C)CSC2)nc(F)ccc1Br 61717,c1(C(=O)NCCn2cc(CNC(COCCC)=O)nn2)cc(F)ncc1OC 61718,C12(N(CC(N3CC(C)C(C(O)C(F)(F)F)CC3)=O)C)CC3CC(C1)C(=O)C(C3)C2 61719,c1(N2CC(=C(CNC(C3(OC)CCC3)=O)F)C2)ncnn2c(Br)ccc12 61720,c1(CCC(=O)NC2(CCO)CC2)c[nH]c(C(=O)NCCC2(N)CC2)c1.CC 61721,c1(C(=O)NC2CCCN(c3nc(O)n[nH]3)C2)c(Cl)cc(F)cc1Br 61722,Cc1nsc(N(C)CCOCCNC(C2CCC(C)O2)=O)c1C#N 61723,N1(C(C(C2CC2)OCC)=O)CCC(C(C)(C)C)(CNC(c2ccnnc2S)=O)C1 61724,c1(CC(=O)N(CCN(C(CCC=C)=O)C)C(C)C)ccc(C(F)(F)F)nc1 61725,CC1CC(=O)NCC1C(N1CCC(C)(CC(=O)N(C)Cc2ccn(C)n2)C1)=O 61726,C1(C(=O)NCCCC(=C)Cl)CCN(C(C2CCN(C)C(=O)C2)=O)CCO1 61727,c1(C(=O)NC2CN(C(COCCc3noc(COC)n3)=O)C2)cncn(C)c1=O 61728,N1(C(Cc2cn(CC)nc2)=O)CCCC(C(N2CCN(C(=O)C(C)(C)O)CC2)=O)C1 61729,N1(C(C(C)SC)=O)CCCC(C)(C)C1C(=O)N(C)CCC1CCCN1C 61730,CN1C(=O)OC2CN(C(=O)C(c3ccccc3)NC(C3CCCC(C)CC3)=O)CC12 61731,c1(CNC(=O)C(=O)NCC2CCCCO2)c(F)ccc(F)c1O 61732,CCCCCCC(=O)NC(C1CCCC1)CNC(c1ccncc1C(F)F)=O 61733,Cc1cc(C(=O)NCC(N2CCN(C3CC4(C3)CN(C)C4)CC2)=O)c(N)cc1F 61734,C(=O)(C1=CCS(=O)(=O)C1)NCCN1CCC(NC(c2nn(C)c(Cl)c2)=O)CC1 61735,C(=O)(C1=CCCC1)NC(CC)CN(C(=O)C(c1ccccc1)OC)C 61736,c1(C(=O)NC(C(C)C)CC(=O)NCCc2ccn(C)n2)cccc2cc[nH]c12 61737,C1(C(N2C(C3(NC(Cc4n(C)cnc4)=O)CC3)CCC2)=O)OCCOC12CCC2 61738,C1(CC(N2CCCC(CNC(=O)C3CC3)C2)=O)Oc2ccccc2NC1=O 61739,N1(C(C2CC(=C)CN2C(=O)CCCSC)=O)CC2(C)CC1CCO2 61740,c1(OC)cc(C(=O)N(C2CC(NC(c3sccc3C)=O)C2)C)cnc1OC 61741,c1(CC)c(C(N2CCC(Cn3cc(CCC(C)O)nn3)C(O)C2)=O)csc1C 61742,c1(CNC(c2c(F)cccc2F)CCOC)ccc(OC(F)F)c(F)c1 61743,C1(C)(NC(CC(=O)NC(C)C)=O)CCN(C(=O)CC23CCCC2C3)C1 61744,N1(C(C2CCC(Nc3ncnc4ccccc34)CC2)C)CCC2(CCCOC2)C1 61745,CN1CCN(C2C(=O)NC3CC23)C(c2ncc[nH]2)C1.C1(COC)CCCO1 61746,C(=O)(CCCCC(C)(C)C)N(C1C2CCCC12)C 61747,C1(C)(C(N2CC(=C(CNC(CC(C)C3CCCO3)=O)F)C2)=O)CCOC(C)C1 61748,Cn1cc(S(=O)(=O)NCc2ccc(-n3ccccc3=O)cc2)c2ccc(Br)cc12 61749,c1(OCC)cccc2cc(C(=O)OCCc3csc(C(C)OC)n3)c(=O)oc12 61750,N1(C(=O)CCN2C(=O)CCC2=O)CCC2CCN(C(c3cncc(Cl)c3)=O)C2C1 61751,C(=O)(C#CC1(C)CC1)N1CCC(C)(CCNC(C2CN(C)C2)=O)C1 61752,c1(CCC(=O)NCC2CC2NC(=O)CC2CNC(=O)C2)cccnc1Br 61753,CCCCCCCCC(=O)Nc1cccc(S(=O)(=O)N(C(C)(C)C)C(C)C2CC2)c1 61754,C(=O)(CC(C(F)(F)F)NC(=O)Cc1cccnc1O)NCCSCC#C 61755,C#CCC(C)(C(=O)N1CCCC1CN(C)CC)NC(C1CC1CC)=O 61756,C1(C(=O)NC(CC2CN(C(C(C#C)(C)C)=O)C2)C)CC(c2cnn(C)c2)=NO1 61757,c1(C(=O)NC2C=CC(CNC(C(CC)(C)COC)=O)C2)ccc(C)c(F)c1F 61758,Cc1cccc2c(NCC3CCCN(C(C45CC4CNC5=O)=O)C3)ncnc12 61759,C(C(C)(O)C(=O)NCC(C)(C)Cn1cc(C2CC(C3CCOCC3)C2)nn1)OC 61760,C1(NC(C2CC3(CCC3)C2)=O)CC(CO)N(C(=O)CC2COC(=O)C2)C1 61761,N1(C(CC(CN(C)C)NC(=O)CC(O)C2CCCC2)=O)CC2(CNC(=O)OC2)C1 61762,C1(C(C)C)CCc2sc(C(=O)OCCC3CN(C(=O)OC(C)(C)C)C3)cc2C1 61763,n1(CC(=C)C)nc(C2CCC2)nc1-c1nn(C)cc1Cl 61764,C1(CC)CC(C(=O)NCCN(C(=O)C(C)NC(=O)OCCCSC)C)C1 61765,C(c1ncc[nH]1)=CC(=O)NCC(CO)NC(=O)C=CC1CCOC1 61766,CC1CNC(=O)CN1C(=O)C=CC1CCN(C(=O)CCCc2ncco2)CC1 61767,Cc1cc(C)c2[nH]nc(C(=O)NC3CCCCN(C(=O)C4=CCOCC4)C3)c2c1 61768,N1(Cc2c(C)cc(C)s2)CCC(Nc2ccccc2)C(O)C1.n1(C)ccnc1 61769,C(CCC(CCC)NC(=O)C=Cc1cncc(F)c1)NC(C=C)COC 61770,CC1(C)COC(CC(=O)NC2CC(NC(=O)C=C3CCC3)C2)CO1 61771,C(=O)(C1=CNS(=O)(=O)N=C1C)N1CC(CC(C)NC(C=C(COC)C)=O)C1 61772,CCC(C)(C)C(O)C(=O)N1CCC2CC1CN2C(c1ccc(CO)c(OC)c1)=O 61773,N1(C(c2c(C(=O)OC)cccn2)=O)CCC2(CC1)CN(C(=O)Cn1cc(Cl)cn1)C2 61774,C1(CNC(=O)Cc2cncc(F)c2)COCCN1C(=O)CSCCO.C1(C)CC1 61775,C1(C(N2CCC(O)(CO)C2)=O)(CNC(=O)CCc2cn[nH]c2)CC(F)(F)C1 61776,CC1(C)CC(NC2CCCN(c3ccncc3)C2=O)CCS1(=O)=O 61777,c1(CC)ncc(C(=O)NCC#CCNC(=O)C(c2cnn(C)c2)C)s1 61778,N1(CC(=O)NC2CCCCC2)CCN(CC2(CNc3cccc(I)c3)CC2)CC1 61779,CCCCC(O)CC(=O)N1CCN(C)CC1C(=O)NC(CCC)C1CCCC1 61780,c1(C(N2CCC(N(C(C(C)NC(=O)OC)=O)C)C2)=O)ccc(O)nc1C 61781,C1(CNC(CC2CCC(C)C2)=O)CN(C(c2cc(O)n(C)n2)=O)CCCO1 61782,N1(C(C2(OCC)CC2)=O)CCC(C(=O)CC2CC(CNC3SCCC3C)C2)CC1 61783,C1(NC(COC(CC)(C)C)=O)CN(C(=O)C=Cc2ccccc2C)C2CCCC12 61784,N1(C(C=COCC)=O)CCC2(CC1)CCN2C(c1cccc2[nH]ncc12)=O 61785,C1(C(=O)NCC(C2CCN(C(C(C)n3cccn3)=O)CC2)O)CC(=O)NC(=O)N1 61786,c1(C(=O)NC(C2CCN(C(c3coc(CN(C)C)n3)=O)C2)C)ncc(Cl)s1 61787,c1(C(N(CCOCCNC(CC2CC(=C)C2)=O)C)=O)c(C)ccn1C 61788,C(CC(CNC(=O)CC1(C)CCC1)NC(c1cnnn1-c1ccccc1)=O)OC 61789,Cc1cnc2cc(C(=O)NC3(C)CCN(C(=O)CCN4CCC(F)C4)C3)nn2c1 61790,Cc1nn(CCO)cc1C(=O)NC1CC(NC(=O)C(C)(O)C2CCOCC2)C1 61791,c1(SC)nc(N2CCOC(C(C)NC(c3csc(C(C)C)n3)=O)C2)ncc1C 61792,CC(C(=O)NCC1(NC(=O)CC2CCCC(F)(F)C2)CCCC1)S(C)(=O)=O 61793,Cc1csc(C=CC(=O)NCC2CCCN2C(C2CCC(F)(F)C2)=O)n1 61794,c1(OC)cccc(OC(F)(F)F)c1Cn1cc(CN(C(=O)C(N)=O)C)nn1 61795,Cc1cc(C)c(OCCNC(C2(C#N)CC3CCC2C3)=O)c(Br)c1 61796,Cc1cccc(N)c1C(=O)NCC1CCCN(C(c2cscc2CO)=O)C1 61797,C1(CC=C)(NC(c2cccc(C(F)F)c2)=O)CCN(C(=O)CCCCSC)C1 61798,Cc1cccc(C)c1CCN=C(NCc1cc(C#N)cs1)NCC1CC1(F)F 61799,c1(C(=O)NC23CC(NC(c4csc(C(F)F)c4)=O)(C2)C3)cc(Cl)c2n[nH]cc2c1 61800,C(=O)(CC(C)C(C)(C)C)NCCN(C(C1C(C(C)C)CCO1)=O)C 61801,c1(C(=O)OCC)nc(=NC(C)CNC(=O)CC2CCC=CCC2)cc(CC)[nH]1 61802,c1(OC)cc(C(=O)NCCC(C)NC(C2CNC(=O)C2)=O)cc2c(C)c(C)[nH]c12 61803,N1(C(c2cc(OC)ns2)=O)CC(NC(C2CC3(CC3)CO2)=O)C(F)C1 61804,c1(C(C)=O)ccc(C(=O)NC2(CNC(C34CCCC3C4(F)F)=O)CC2)c(C#N)c1 61805,CC1CN(C(c2cc3n(n2)CCO3)=O)CC(C)N(C(=O)COC2CCCOC2)C1 61806,c1(C(N2C(C)C(NC(=O)Cc3cncnc3O)CC2)=O)cn2c(n1)SCC2 61807,C#CCCCC(C)C(=O)NCCCOCCCNC(c1cc2cnccc2[nH]1)=O 61808,C12(CNC(CC3N(C)CCC3)=O)CC1CN(C(=O)CCNC(=O)CO)C2 61809,N#Cc1cccc(C(N2CC(NS(=O)(=O)c3cn[nH]c3)C2)=O)c1[N+](=O)[O-] 61810,N1(C(C(c2ccc(F)cc2)OC)=O)CCCCC1CC(=O)NCCCn1ccnn1 61811,Cn1cc(C(N2CCC(C(F)CNC(=O)CCS(C)=O)CC2)=O)c(Cl)n1 61812,c1(C(=O)NC(C2CCN(CCSc3nnnn3C)C2)C)cccc2cnccc12 61813,C(=O)(CCCCCC#N)NC(CC#C)C(=O)N(C(C)C(C)(C)C)C 61814,CC(C)(C)C(CC(=O)NCc1cccc(NC(=O)CC=CC(C)(C)C)c1)C(F)F 61815,Cc1ncc(Cl)c(C(=O)NC2CC23CCN(C(c2ccncn2)=O)C3)n1 61816,C1(C(=O)NCC2(CNC(COCC(C)C)=O)CCCC2)CC(=O)N(C)C(=O)N1 61817,Cc1cc(C(N2CCOC(C(N3CC(C)C(O)C3)=O)C2)=O)cnc1Cl 61818,Cc1ccc(-c2ccsc2C(=O)NCCCNC(=O)COC(F)(F)F)cc1 61819,C1(C(N2CC(C(=O)NCC3CNC(=O)O3)(CC)C2)=O)C2CC3C(C2)C13 61820,c1(CNC(c2nccc(=N)[nH]2)c2ccc(Cl)cc2)ccc(F)c(Cl)c1 61821,C(=O)(C(C)(C)CC(C)(C)C)NCC(C)NC(c1onc2ccccc12)=O 61822,C(=O)(CCCC(=O)NC1COCCC1NC(c1cnc(C(C)(C)C)nc1)=O)OC 61823,c1(NC(C)=O)cc(NC(C2NCC(O)C23CC3)=O)cc(N(C)C)c1 61824,c1(C(=O)NCC(C(C)C)(C)NC(c2cccc(Cl)c2Cl)=O)nccc(C#N)c1F 61825,N1(C(COCCC=C)=O)CCC2CCN(C(=O)C(c3ncccc3C)(F)F)CC12 61826,CC(C)(C(=O)NCCC1CCCN(C(C2(O)CCOC2)=O)C1)S(C)(=O)=O 61827,CCCCC(C(=O)Nc1ccc(N(C)C)cc1)NC(=O)CC1CCCCN1C 61828,C1(NC(C(C=C)c2ccccc2)=O)C2CC1N(C(C1(S(C)(=O)=O)CC1)=O)C2 61829,c1(OC)cc(NC(C2CCCN(C(c3cc(Cl)ccn3)=O)C2)=O)cc(F)c1F 61830,N1(C(C=CCOC)=O)CCOC(C)(CNC(c2ccn(C(C)C)c2C)=O)C1 61831,c1(CCNC(=O)NCC(C2CCOCO2)(C)C)ccc(CO)cc1 61832,c1(C(N(C(CCNC(c2c(C)[nH]nc2Cl)=O)C)C)=O)ccc(S(C)=O)cc1 61833,C1(CNC(C=CC)=O)CC2(CCC2)CN1C(C1(c2ccccc2)CCCO1)=O 61834,C1(CC#C)(C(=O)NCCC(C)CCNC(c2c[nH]cc2C)=O)CCOCC1 61835,c1(C(=O)NC2CC(N(C(C3OCCN(C(C)=O)C3)=O)C(C)C)C2)cncc(Cl)c1C 61836,C(=O)(C(C)(O)C(F)(F)F)N(C1CCCN(C(C23CC4CC2C3C4)=O)CC1)CC 61837,Cc1cc(C)c(C(=O)N(C)CC2CCCN2C(C2CC2C(C)O)=O)cc1N 61838,N1(C(CCCSC)=O)CCC(C(=O)NC(C)CC(F)(F)F)C12CC2 61839,Cc1ccc(N)c(C(=O)NC2(C)CC(NC(=O)C(C)C3CCOC3)C2)c1 61840,CCCC(C)(CCC)C(=O)NCCOC1CCN(C(=O)CC2CCC2C)C1 61841,C#Cc1cc(C(=O)N(CC(C)NC(c2ccc(OCCF)cc2)=O)C)cc(F)c1 61842,C#CC12CC(CN1C(C1(COC)CN(C(=O)C(C)CC(C)C)C1)=O)C2 61843,C(C(=O)Nn1nnc2c1CCCC2)C1N(C(Cc2c(C)n[nH]c2)=O)CC1 61844,C1(C(=O)NCCOCC(=O)N(C(CF)CF)C)CCOC1C1CC1 61845,c1(C(N(C2CCN(S(=O)(=O)CCCN3CCOCC3)C2)CC)=O)ccnc(F)c1 61846,c1(OC)cc(C=CC(N2CC(C)CCC2C)=O)ccc1F.c1ncc(F)c(O)n1 61847,c1(C(N2C(C(=O)NC(CC)CC)CC(C)C2)=O)cc(OC)cc(C(F)(F)F)c1 61848,c1(C(N2CC(OC)NCC2)=O)cc(Cc2ccccc2)ccc1F 61849,C1(c2n(CC)nnn2)(NCc2nn(C)cc2Cl)CCC(=O)N(C)C1 61850,C1(NC(C(C)CF)=O)CCSC12CN(C(C1CCCCC1CC(F)(F)F)=O)C2 61851,C1(NC(C2CN(C)C2)=O)CCN(C(c2cn(C)c(=O)cn2)=O)CC1O 61852,C1(C(=O)NCC(CC(C)C)NC(=O)C(C)n2cccn2)CC(S(C)(=O)=O)C1 61853,C1(F)(CNC(C(CC)c2ccccc2)=O)CCN(C(c2sccc2C)=O)C1 61854,N1(CCNC(c2c(CC)nccn2)=O)CCCN(C(c2ccc(C)nn2)=O)CC1 61855,c1(COC)ccc(C(=O)NC(CN(C(=O)CCOCCCC(C)C)C)CC)cc1 61856,C#CC1CCCN(C(c2ccc(C(=O)OC)nc2C)C(=O)NCCOC)C1 61857,c1(C(N(C2CN(C(=O)CN(C)S(N)(=O)=O)C2)C)=O)cc(F)ccc1O 61858,N1(C(C2C(C=C)OCC2)=O)CC(CC(N2CCC(C)(NC(C)=O)C2)=O)CC1(C)C 61859,c1(C(C(=O)NC)N(C)C(c2ccccc2F)C)cc(Cl)c2c(c1)OCCCO2 61860,c1(C(=O)OC)ccc(C(=O)NCCCC(C)NC(=O)C=Cc2cc[nH]n2)o1 61861,N1(C(c2cn(CC=C)nn2)=O)CC(CNC(c2c(C3CC3)cnn2C)=O)C(C)C1 61862,c1(C(N(CCC(F)(F)F)CC)=O)cccnc1CNC(=O)C(C1CC1)SC 61863,C1(OCC)CN(C(=O)CC2(C(=C)F)CCC2)CC1CNC(=O)C=C1CCC1 61864,C(N=c1[nH]cnc(Cl)c1C)C1(CNC(c2c(N)ncc(C)c2)=O)CCCC1 61865,c1(C(=O)NCC(CC)(CC)NC(c2coc(C3CC3)n2)=O)ccnn(C)c1=O 61866,CCCC(CNC(=O)C(C)=CCOC)NC(c1cn(C(F)F)cn1)=O 61867,c12ncc(C#N)c(n1)N2C1(C#N)CCNC1.C#Cc1ccccc1COC 61868,Cc1cc(=NC(=O)CSCCCNC(=O)CSCCCCCN)[nH]o1 61869,N1(C(C=CCC)=O)CC2CC1CN2C(c1cccc(-c2cnn(C)c2)n1)=O 61870,C1(NC(C2CC(C)CN2C(C2CC2c2ccccc2)=O)=O)CC(C)N(C)CC1C 61871,CC(CCN=c1[nH]cnc2cccnc12)NC(=O)CCC1CCCOC1 61872,CC1(C)CN(C(=O)CC2OCCCO2)CCC1NC(c1cncc(C(F)F)c1)=O 61873,N12CCC(CC1)C2.N1(CC)CCCCCC1.C1(c2ncco2)C(=O)N1CC(C)C 61874,C(CC(C(C)(C)C)NC(C1CCC(C)(C)C1)=O)N(C(C1(CCCC)CC1)=O)C 61875,c1(CNC(N(c2ccc(OCOC)cc2)CC)=O)cc(C)c2c[nH]nc2c1 61876,C(=O)(C(C)C(C)c1ccco1)NCCCN(C(CC(=O)NCC)=O)C 61877,N1(C(C(C(C)C)C)=O)CCN(C(c2ccc([N+](=O)[O-])s2)=O)CC(CO)C1 61878,C#Cc1ccc(C)c(NC(C2CC(C)(NC(=O)CC3CCC(=O)N3C)C2)=O)c1 61879,CC1CN(Cc2cnccc2C(F)(F)F)CCN1C(=O)C(C)O 61880,c1(C(=O)NCCNC(c2ccoc2)=O)cc(C(=O)O)sc1Br 61881,Cc1[nH]nc(C(N2CCOCC2CN(C(=O)C(F)(F)c2nccn2C)C)=O)c1N 61882,C12(CNC(C3(CCOCC)CC3)=O)CCN(CC1)CC2.C1(=O)CCN1 61883,c1(NCCN(N(C)C)CC)ccc(S(=O)(=O)NCCC2CC2)cc1C#N 61884,c1(C(=O)NCC2(O)CN(C(C(C)=C(CC)C)=O)C2)sc(Cl)nc1C 61885,c1(C(=O)NCCN(C(c2ncc(C)c(Cl)c2)=O)C2CC2)cc2n(c1)CCSC2 61886,c1(C(=O)NCC2(CCNC(c3ccc(C)s3)=O)CC2)ccc(Cl)nc1N 61887,c1(C(=O)NCC2CC(F)CN2Cc2cccc(C(=O)O)c2)nc2ccccc2o1 61888,C1(NC(Cc2nc(C)sc2)=O)CCC(N(C)C(C2CCN2S(C)(=O)=O)=O)CC1 61889,C1(C(=O)NC(C#C)C)(NC(=O)C(COC)N(C)C)CC1(C)C 61890,C1(CNC(C(CC)NC(C)=O)=O)CC2CCC1N2C(=O)CCCCN(C)C 61891,C1(NC(=O)C(F)CC2CC2)CC(Nc2cc(O)ncn2)C12CCC2 61892,C12COC3(CCC3)C1NC2.c1(CCC(=O)OC)cnc(C2CCCN2CC)nc1 61893,C1(c2nnnn2Cc2ccco2)(N2CC(c3nc(C)[nH]n3)C2)CCCCCC1F 61894,N1(CC)CC(CC)(NC(c2csc(C)n2)c2nnnn2C2CCOC2)CCC1=O 61895,C1(C(=O)NCC(CC(C)C)NC(c2cc(Br)c[nH]2)=O)CNC(=O)CC12CCC2 61896,C1(CNC(C(F)=CC)=O)CCCC1NC(c1cc(C(=O)NC)[nH]n1)=O 61897,C1(CNC(C(CC)CC)=O)CCN(C(C2CC3CC(=O)C2O3)=O)C12CCC2 61898,C(=O)(C(O)C(C)(C)C)NCC(C)(C(C)C)NC(C1(C(=O)OCC)CCC1)=O 61899,C(=O)(CCCC(C)C)N(C)CC1CCN(C(C(C)OC)=O)C1 61900,c1(CN(CC)CC)ccc(C(=O)NC2CC(C(=O)OC)CC(C)O2)c(Cl)c1 61901,CC(C)(C)CC(=O)NC(C)(C)CNC(=O)C(F)OC.N12CCC(CC1)OCCC2=O 61902,C(CCC)(CCCNC(=O)C1=C(C)OCCS1)NC(CNC(=O)OC)=O 61903,N1(C(Cn2c(C)ncc2)=O)CCC2(CCCC2NC(=O)Cc2n[nH]cc2Br)C1 61904,CN1CCCC(C(N2CCCC2CC(=O)Nc2cncc(N3CCCC3)n2)=O)C1 61905,C(=O)(CCCC(C)(C)C#N)NCCOCCN(C)C(C1OCC2CCCC12)=O 61906,N1(C(c2c(OCC)cccc2)=O)CC2COCCC2(NC(=O)CC(C)C2CC2)C1 61907,n1(CC(=O)NCC2C3N(C(CCSC)=O)C(CC3)C2)nc2ccccn2c1=O 61908,C1(C(=O)NC(C)(C)C=CC(=O)NC(C2CCOC2)(C)C)C2CCC(F)C12 61909,C1(O)(CC(=O)NCC2(OCC)CN(C3CCC(=O)NC3=O)C2)CCCN(C)C1 61910,c1(C(=O)NCC(CNC(=O)C(C(CCC#CC)=O)CC)CO)cc(N)ncc1Cl 61911,c1(CC)cc(C(=O)NC2C3CC2N(C(c2oc(C)nc2C)=O)C3)ccc1C 61912,CCC(CNC(=O)CC(C)CNC(c1ncc(C)cn1)=O)(CC)OC 61913,c1(CC)cc(C(=O)NCC(O)CNC(c2cnc(C(C)(C)C)o2)=O)nn1C 61914,N1(C(C(C)CF)=O)CCCC(N2CCN(C(c3n[nH]c(=N)s3)=O)CC2)C1 61915,c1(C(=O)NCC(CCNC(C2(CC)COC2)=O)O)nc2n(c1C(C)C)CCCC2 61916,c1(C(=O)NC(CNC(C(C)c2ccsc2)=O)(C)CO)cc2c(s1)CC(C)(C)C2 61917,n1(CC)nc(C(=O)NC(C2CCN(C(C3CCCCS3)=O)CC2)C(C)C)cc1C 61918,c1(N(C)C)nc(C(=O)NCCC2(O)CCN(C(C34CC(F)C3C4)=O)C2)ccn1 61919,C1(NC(c2c(CC)noc2)=O)CCN(C(c2ccccc2C(C)(C)C)=O)CC1C 61920,N1(C(=O)Cc2nnc(O)s2)CCC(Oc2ccc(Cl)cn2)CC1 61921,c1(C(N2CC(CCC)C(NC(=O)CC(C)OC)C2)=O)cc(C)nc(C)n1 61922,c1(C(CC)NC(=O)NCCCCC2CC(NC)C2)ccccc1OC 61923,C(=O)(CCCC(=O)N(CCCCNC(=O)Cc1ccccc1NC(C)=O)C)OC 61924,C1(NC(C(CC=C)CC=C)=O)CCCC2CN(C(=O)C(C#N)CCC)CC12 61925,CCN=C(NCCC1CCCCC1O)N1CCc2c(Br)cccc2C1 61926,C1(O)(C(C)NC(=O)CC(C)c2ccco2)CCN(C(c2ncc(Cl)s2)=O)CC1 61927,c1(C(N(CC(C)CO)C)=O)coc(CNC(C2(O)CCOC2)=O)n1 61928,c1(NC)c(C(=O)NC(C2CCN(C(C3CC4CCCC34)=O)C2)C)cccc1N 61929,C(=O)(C(C)CCCc1ccccc1)N1CCC(N(C(C=CC)=O)CC)C1 61930,C1(C)(N(N2CCCC2)C(CSCC)=O)CC(OC)CN1C(=O)CC(C)n1cccn1 61931,C1(NC(=O)C(O)Cc2ccccc2)CC2CC1CN(C(C1CCC3(CC3)C1)=O)C2 61932,C12(C(=O)NCC3(N(C(C)C(=O)NS(C)(=O)=O)C4CC4)CC3)CCCN(CCC1)C2 61933,N1(C(C=C2CCN(C)CC2)=O)CCCN(C(c2ccc(Cl)nc2N)=O)CC1 61934,CN1CC(C)(C(=O)NCC2(O)CC(CNC(c3nnn4c3CCC4)=O)C2)CC1=O 61935,C1(NC(CCCCSC)=O)COC2(CCN(C(=O)Cn3ccc([N+](=O)[O-])n3)C2)C1 61936,c1(CNC(C(C)(C)c2ccc(Cl)s2)=O)ccccc1-c1nn[nH]n1 61937,C1(NC(=O)NCC(COC)C)CCN(Cc2nnnn2C(C)(C)C)CC1C 61938,c1(C(c2nnnn2CCCOCC2CC2)NCCCCCC)cccc2c1CCO2 61939,c1(CC(=O)NC(C(=O)NC2CCN(CC)C(C)C2)C2CC2)csc2nc(C)cn12 61940,Cc1cc(N)cnc1C(=O)NCC1CN(C(=O)C(C2CCCCC2)F)CCCO1 61941,c1(C(=O)NC2CC(NS(=O)(=O)c3ccc(Cl)nc3)C2)cc(Cl)nc(Cl)c1F 61942,c1(COCC(=O)Nc2ncccc2Br)c(Br)c(O)c(Br)cc1Br 61943,n1(CC(=O)NCc2onc(-c3cccc(C)c3)n2)c(C(C)C)nc2ccccc12 61944,C1(OC)CC(C)CN(C(C2(C)CCCN2C(=O)NCCCl)=O)C1 61945,N1(C(c2c(OC)cnc(F)c2)=O)CCCCC(NC(c2ccncc2C)=O)CC1 61946,n1(CC(=O)NCC(C)(O)CNC(C2(CC(F)F)CC2)=O)cnc2c(N)ncnc12 61947,C#CC(C)(C)C(=O)N1CC(CNC(C2CCCC(C)C2)=O)C(C)C1 61948,C1(NC(CCC=C(C)C)=O)COC2(C1)CN(C(=O)C1=NNC(=O)C1)C2 61949,N1(C(C2N(C)C(=O)CCC2)=O)CC2CC(NC(C3C=CCC3)=O)CC1C2 61950,C1(NC(C=CC(C)NC(c2n(CCC)ncc2)=O)=O)CCN(C)CC1C 61951,N1(C(CSC2C(=O)OCC2)=O)C2CCCC1CN(C(c1csc(S)n1)=O)C2 61952,c1(C(=O)NCCOCCNC(c2c(C)nc(N)cn2)=O)cccc2scnc12 61953,c1(C(=O)NCC2N(C(c3cc(SC)oc3)=O)CCCC2C)n[nH]c2c1CSCC2 61954,CC1CCCC(C(N2CC3C(CN(C(=O)C=Cc4cnn(C)c4)C)C3C2)=O)C1 61955,Cc1ccc([N+](=O)[O-])c(C(=O)NCC2CC3CCC2N(C(C2CCOC2)=O)C3)c1 61956,CC1CC(=O)NC(C(=O)NC(C)(C)C(C)NC(=O)CSc2ccccc2Cl)C1 61957,N1(C(C(C)=CC2CC2)=O)CCCCC2(CCN(C(=O)C3=C(C)CCCC3)C2)C1 61958,CC(O)(C(=O)N1CC2CC(C(=O)NCCN=[N+]=[N-])CC2C1)C(F)(F)F 61959,C1(CNC(=O)CCn2cncn2)CC(F)CN1C(=O)C(C1CCCCC1)=O 61960,c1(CC)cc(F)ccc1C(=O)N(C1CCN(C(c2c(CC)nn(C)c2C)=O)C1)C 61961,C12(CCN3CCN(C(c4ccc(OC)cn4)=O)CC3)CCC(CC1)C2(C)C 61962,c1(C(C(C(=O)NCC(C(=O)OC)Sc2ccc(F)cc2)C)C)c(C)noc1C 61963,C1(C(=O)NCC(CC=C)NC(=O)CCC2(C)CC2)C(C)(C)CCCC1(C)C 61964,Cc1nc(C(=O)NC2(C(N3CCC(CCF)CC3)=O)CCCC2C)c(C)o1 61965,c12cccn1CC2.C1(OC(NOCC(=O)NC2C(NC(C)=O)CC2)=O)CCCCC1 61966,C(C(O)C(F)(F)F)NC(c1cncc(OCCN2CCCCC2)c1)=O 61967,N1(CC(=O)NCC2N(C(CCCSC)=O)CCC2C)CCN(C)C(=O)C1 61968,C1(NC(C(C)OC2CN(C(C3(COCC(F)(F)F)CC3)=O)C2)=O)COCCOC1 61969,c1(C(=O)NCCCC(C)NC(C2C(OC)CCC2)=O)ccc(NC=O)cc1 61970,N1(C(C2(C)CC2Br)=O)CC(NC(c2csc(C(F)F)n2)=O)C(O)C1 61971,C1(CNC(C(C)NS(CC)(=O)=O)=O)CN(C(=O)Cc2ccoc2C)C(C)(C)C1 61972,CC1CC2(CCN(C(=O)CCc3cnc[nH]3)CC2)CN1C(c1ccc(S(C)=O)o1)=O 61973,C=CC(C)(C)CC(=O)N(C(C)CNC(=O)CCC1CCCCO1)C 61974,c1(C(=O)NC2C(NC(C(CC(C)C)F)=O)COC2)cc2n(n1)CCNS2(=O)=O 61975,CC1(CNC(=O)C(C#N)C2CC2)CCCN1C(c1cnc(S)[nH]1)=O 61976,c1(C(=O)OCC)sc2ccncc2c1NC(=O)CNCc1scc(Br)c1Br 61977,Cc1ccc(C(=O)N(C(C)CCNC(c2cnn(C)c2)=O)C)nc1 61978,N1(N(C(C(CC(C)C)NC=O)=O)c2ccc(Cl)cc2)CCC2C(CCC2(F)F)C1 61979,C1(NC(C=C(C)C(C)C)=O)(CNC(=O)Cc2nc(C)cs2)CCCCC1C 61980,c1(C(=O)NC(CCC)C(=O)N2CCNCC2CCO)cccc([N+](=O)[O-])c1 61981,C1(C(=O)NCCN(C(=O)C=CCF)CC)CCCC1SC 61982,OCC(F)(F)CCCCN=C(NCc1ccon1)NC1CCC1 61983,Cc1cc(Cl)ncc1NC(=O)C(C)C(C)NC(c1ccn(CO)c1C)=O 61984,C1(CC(=O)NCC2C(NC(C=C(C)C(F)F)=O)C2)CC(C2CC2)C1 61985,Cc1cc(=O)oc(C)c1C(=O)NCCC1CN(C(c2cnc3n2CCCC3)=O)C1 61986,C=CC(CCC)CC(=O)N1CCCC1CCCNC(c1cc2n(n1)CC(F)C2)=O 61987,Cc1nc(N(C)C)sc1C(=O)NC(C)C(C)NC(=O)CCF 61988,CCCCN=C(NCCc1cccc(F)c1F)NC1CN(C2CC2)C1 61989,C1(C(=O)NC2(CC=C)CCOC2)CC2CCC1N2C(=O)C(C)(C)CCOC 61990,C1(CNC(CCN(C(=O)CNC(=O)CN(C)C)C)=O)CCNC(=O)C1 61991,CCCC(C(=O)OC)C(=O)NCC1(C2(O)CN(C(=O)C=Cc3cnc[nH]3)C2)CC1 61992,c1(N(CCC)C)nnc(CCC2CC(=O)N(c3cccc(F)c3)C2)n1CC1CC1 61993,Cc1nc(C=CC(=O)NCC(O)CNC(=O)CCOC2CCOCC2)cs1 61994,c1(C(N2CC3C(CNC(=O)OC)C3C2)=O)cc2c(OC)ccc(C)c2[nH]1 61995,C#Cc1ccc(F)cc1C(=O)NC1CN(C(c2ccc(F)cc2C#N)=O)CC1C 61996,N1(C(CC(C)(C)CNC(=O)C=CCN2CCCC2)=O)CCC(C2(O)CC2)CC1 61997,N1(C(COC(c2c(CC)nccc2)=O)=O)CC(C)(C)C(O)C1(C)C 61998,C1(C)(C(=O)NCC(C)(C(C)C)NC(C(CCC)=CCC)=O)CCCCC1(F)F 61999,c1(N(CCC(C)NC(C2N(CC)CCC2)=O)C)cc(C)c(C#N)cn1 62000,N1(C(C2(CC(C)C)CC2)=O)CCC(C(=O)N(CC(C)C(C)C)C)(CO)C1 62001,C1(NC(c2c(CC)cncc2)=O)CCC2CCN(C(c3ccc(O)nn3)=O)C1C2 62002,CCC(F)(F)CC(=O)N1CCN(C(c2ncsc2Br)=O)C(CCO)C1 62003,N1(C(C=Cc2occ(C)n2)=O)CC2CN(C(=O)CN(C)C)CCC2(CO)C1 62004,C(C1CCCN1C(C1(C(N)=O)CCC1)=O)=CC(NOCC1(C)CCC1)=O 62005,C(CCC(=O)NCCCOCCC(=O)N(C(CC1CC1)CC)C(C)C)=CC 62006,c1(C(N2C(C(=O)Nc3c(Br)ncc(OC)c3)CC(F)C2)=O)ccc(C#N)cc1O 62007,C(=O)(N=c1cccn[nH]1)NCc1ccc(N2CC(C)OCC2)cc1 62008,c1(CCC(=O)NCC2CCN2C(c2ncccc2Cl)=O)ccc2c(c1)CCO2 62009,C12CN(CCC1(F)F)C2.c1(NC(C(COC(C)C)NC(C)=O)=O)ccn(C)c1C 62010,N1(CC)C(=O)NC2CN(C(=O)C(CC(C)C)OC)CCC12 62011,N1(C(CCC)=O)CC2CCC1C(CNC(=O)CCN1CCC(O)CC1)C2 62012,N1(C(=O)Cn2cc(Cl)cn2)CCCC1C(C)(C)CNC(=O)CCOCC1CCC1 62013,S(=O)(=O)(c1ccc(C(N2CCC(CO)(NC(C3COC(=O)C3)=O)C2)=O)o1)N(C)C 62014,C(=O)(C1=CNC2=NCCC2=C1)NC1CCN(C(CSc2c(C)ccc(C)c2)=O)C1 62015,CC1CCCN(S(=O)(=O)NC(C(=O)NC2CCCC2)C(C)O)C1 62016,c1(C2C(C(=O)NCCNC(Cc3nnc(CC(C)C)o3)=O)C2)cc(Br)ccn1 62017,c12cnc(nc1)CNC2=O.c1(C(CO)NC(=O)CC2CCCO2)nc[nH]n1 62018,C1(CNC(C(C(C)C)OC)=O)CC2CCC1N(C(C13CCCCC1C3)=O)C2 62019,c1(C(=O)NC2CC(NC(c3c(C)nc(CCC)s3)=O)C2)csc2ncnc(O)c12 62020,C(CC(C(=O)N1CC(OCCNC(=O)C=CSC)C1)NC(N)=O)SC.C(C)(=O)N 62021,c1(NC)cncc(C(=O)NC(C)CCCCNC(=O)CC2(C)CC2(Cl)Cl)c1 62022,C(=O)(CCCCC(F)(F)F)NCC12CCC(NC(CC3(C)CCC3)=O)(C1)CO2 62023,CCCC(C(O)C(=O)Nc1ccc(O)nc1)NC(=O)COCC1CC1 62024,n1(CC)c(C)nn(CC(=O)NCCCNC(c2ccc(C(N)=O)cc2)=O)c1=O 62025,C(=O)(C(F)(F)C(F)F)NC1CN(C(c2c(C(C)C)nns2)=O)C(C)C1 62026,CCC(CN1CC(=O)NCC1C(C)C)(CC)C(=O)OCC 62027,N#Cc1c(C(N2CCC3CCCC23C(=O)NC2C3CC4C(C3)C24)=O)cccc1F 62028,Cc1nc2sc(C(N3CCC(CNC(=O)C(C)CN4CCCC4)C3)=O)cn2c1C 62029,C1(O)(C(N2CC(O)(C(C(=O)NCCN(C)S(N)(=O)=O)F)C2)=O)CCSCC1 62030,C1(NC(=O)CCC2CC2(F)F)CCN(C(c2ccnnc2O)=O)CC12CCC2 62031,CC(C)CC(CC(=O)NC1(CO)CCC(C)C1)NC(C1CC2(CCC2)C1)=O 62032,c1(C(C)(C)C(=O)NC(CNC(=O)CC2CC3CC3C2)CO)ccc2c(c1)OCO2 62033,CC1CCC(OCCNC(=O)C(C)C(C)OC2CCOC2)CC1 62034,c1(OC)ccc(C(=O)N(C)CCNC(C2(C)CCCC2(F)F)=O)c(N)c1F 62035,C1(CNC(C2CC(C)C(C)CC2)=O)C(C2CC2)CCN1C(=O)CSC1CCOC1=O 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62054,c1(N2CCC(C3(C(C#CC(C)(C)C)=O)CC3)C2)cc2c(cn1)C(=O)CCC2 62055,c1(C(=O)NCCCCN(C(C(C)n2cnnn2)=O)C)ncccc1N 62056,c1(-c2cn(C(Cc3ccc(F)cc3)OC)nn2)cc(F)c(F)c(F)c1 62057,Cc1cc(F)c(CC(=O)NCCCCCCNC(C2COCCC2C)=O)cc1F 62058,c1(C(N(CCCNC(=O)C(C)C2CC2)CC)=O)sc(C)cc1C 62059,c1(NC(c2ccccc2-c2nn[nH]n2)=O)cc([N+](=O)[O-])ccc1C(=O)NC1CC1 62060,C1(CSC)CN(C(=O)CCCC(=O)OC(C)(C)C)CCN1C(C1CCC(=O)N1)=O 62061,c1(C(=O)OC)ccnc(Nc2cncc(-c3cnc(=N)[nH]c3)c2)c1F 62062,CCC(CC(=O)NCCn1cc(C(=O)Nc2ccc(C)c(O)c2)nn1)C(C)C 62063,N(C1CS(=O)(=O)N(C)c2ccccc21)C(=O)NC(c1cccnc1)CC 62064,Cc1[nH]c2ccccc2c1NC(c1ccc(C(=O)N=c2nc[nH]s2)cc1C)=O 62065,CC1(C)CC(C(N2CCN(C(=O)CC3(C#N)CCC3)CC2C2CC2)=O)CCO1 62066,N1(C(C2C(C)(C(F)(F)F)C2)=O)CC(CNC(=O)C(C)(C)C(N)=O)C2(CC2)C1 62067,Cc1c(Cl)ccc(NC(C2CCN(Cc3cc4sccc4s3)CCC2O)=O)c1F 62068,c1(C(=O)NC(C)CNC(=O)C(CO)c2ccccc2)cccc2c1OCCN2 62069,c1(C(=O)NCC2CCC2NC(c2ccccc2O)=O)ccc2nc(CO)[nH]c2c1 62070,C1(NC(C2CCCCO2)=O)CCN(C(=O)CCc2ccccc2Cl)C12CCCC2 62071,C1(C(N2CC(NC(c3c(C)cn(C)n3)=O)C(C)C2)=O)CC2CCC(C1)C2 62072,C(C1c2ccccc2CN1C(=O)OC(C)(C)C)NC1(CC=C)CN(C)C1 62073,N1(C(CC=C)=O)CC(NC(c2cn(C)nc2-c2cnn(CCC)c2)=O)C(F)C1 62074,N1(C(CC(=O)NCC2CCCC2)=O)CCc2nc(S)[nH]c2C1 62075,c1(SC)ncc(C(N2CCN(C(c3cnc(=N)[nH]c3)=O)C(CO)C2)=O)c(O)n1 62076,N1(C(C#CC(C)C)=O)CC2COCCC2(NC(c2nccnc2N)=O)C1 62077,C1(C(=O)NC2CC(NC(c3cnn4ncccc34)=O)C2)CC2CCC(C1)C2(F)F 62078,CC(C)C(O)C(F)(F)C(=O)NC1CC(C)N(C(C2CC23CC(C)(C)C3)=O)C1 62079,Cc1cc(C(=O)NCC(C)(C)CNC(=O)C(O)Cc2ccc(F)cc2)cc(C)c1 62080,C(=O)(C(C)(C)CCCF)NCCC1CC(NC(C(c2n(C)ncc2)O)=O)C1 62081,C1(CCNC(C(C)SC)=O)CCN(C(=O)CSCC(F)F)C1 62082,c1(C(N2CCN(C(Cc3c(C)non3)=O)C(CF)C2)=O)cn2c(n1)CCC(C)C2 62083,C1(N(C)C)CN(C(=O)NC2(CNC(C)(C)C)CCC2)C1 62084,CC1(C(=O)NC2CCC(NC(c3ncoc3-c3ccco3)=O)C2)CCC(=O)NC1 62085,c1(C(N2CC3C(CNC(c4cnc(C(C)C)[nH]4)=O)(C3)C2)=O)ccc(C(N)=O)c(Cl)c1 62086,Cc1ccc(C(=O)NCCC(C)NC(c2cnc(C(N)=O)s2)=O)c(N)n1 62087,CC(CCCCNC(C1CCC(N(C)C)C1)=O)NC(C1CC1c1cnc[nH]1)=O 62088,CCCCS(=O)(=O)CC(=O)N1CCC(NC(c2n[nH]c(CC)c2F)=O)C1(C)C 62089,CC1(NC(c2ccc(N3CCCC3)nc2)=O)CCN(S(=O)(=O)CCCCl)C1 62090,C(=O)(C(C)CCC(C)(C)C)NC(CC)(CNC(c1sc(OC)nc1Cl)=O)CC 62091,N1(C(C2CCCN(CCC)C2)=O)CC(CNC(=O)CCc2ccco2)C(C)(C)C1 62092,c1(N2CC(C)(C)C(NC(C3CC3(C)C)=O)C2)ccc([N+](=O)[O-])cc1-n1cnnn1 62093,CN=C(NCCCCCCN1CCCC1)N1CCC(S(=O)(=O)N2CCCC2)C1 62094,c1(OC)cc(C2CC2)ccc1C(=O)NC1(C)CC(NC(=O)Cc2ccon2)C1 62095,Cc1nn(CCO)cc1C(N1CC(CNC(C2(C3CCCO3)CCCC2)=O)C1)=O 62096,C1(C(=O)NCC(C(C)C)OC(C)(C)C)CC12CN(C(=O)OC(C)(C)C)C2 62097,Cc1nc(=NC(=O)CSCC(F)(F)F)n(-c2ccc([N+](=O)[O-])cc2F)[nH]1 62098,Cn1ccnc1C(F)(F)C(=O)NCCOC1CN(C(=O)C(F)(F)C2(O)CCC2)C1 62099,c1(C(=O)NC(CC)CN(C(C23CSCC2C3)=O)CC)cc(C2(Cl)CC2)n(C)n1 62100,C1(C(N(C)CC2CC2=C)=O)COCC1NC(=O)Cn1ccnc1 62101,N1(C(c2ccc(C)c(C)c2)=O)CC(C2CN(C(c3csc(Br)c3C)=O)C2)C1 62102,C1(NC(C2C3C(NC(C45CC(CO)(C4)C5)=O)C4C(C3)C42)=O)CCC2(CCCC2)C1 62103,C1(C(N2C(C(N)=O)CC2)=O)CSCN1C(c1ccsc1)=O 62104,c1(CC(=O)NCC2(OC)CCN(C(C(=O)NCC)=O)C2)ccc2c(c1)CC2 62105,C1(CC(=O)NCC(C)(C2CC2)NC(=O)CCCC2CCCO2)CNC(=O)O1 62106,C1(F)(C(=O)NC2COCCN(c3nccc(Br)n3)C2)CCCCC1(F)F 62107,CCC(C)(C)CCCC(=O)NCCCC(=O)NCC1CCCC(C)CC1 62108,CN(C)NC(=O)CCC(=O)NC1CC2CN(C(c3ccc(=O)n(C4CC4)c3)=O)CC2C1 62109,Cc1cnc(C(=O)NC(CNC(c2cn(C)nc2C(N)=O)=O)CC(C)C)c(F)c1 62110,Cc1cc(C(N2CCC(NC(=O)Cc3ccco3)C23CC3)=O)cc([N+](=O)[O-])c1Cl 62111,N1(C(=O)OC)CC2CCN(C(C)(C)Nc3cc4ncccc4s3)C2C1 62112,CC1CCC2CN1C(=O)CNC(=O)C1(CC1)C(=O)N2.c1(NC(N)=O)ccccc1 62113,c1(C(N2CC(S(C)(=O)=O)C2)=O)cccc2ccc(Br)nc12 62114,Cc1ccc(C(C)(F)F)cc1NC(=O)CCC(C)N(C)C.N12CC3CC1C3C2=O 62115,C1(NC(c2c(C(C)C)ccs2)=O)CCC2CCN(c3ncnc4sccc34)C1C2 62116,O=NN1CCCCC1C(=O)NCCc1ccc(CNC(C2(O)COC2)=O)cc1 62117,N1(C(C2CC2c2ccc(F)cc2)=O)CCC12C1CC3CC(C1)CC2C3 62118,C1(C(=O)NCCC2N(C(Cc3c(C)nccc3)=O)CCSC2)CCn2cncc2C1 62119,C1(OC)CC(C)CN(C(C2CN(C(=O)CC3NC(=O)NC3=O)CCO2)=O)C1 62120,Cc1[nH]c2ccc(Cl)cc2c1C(N1CC(NC(C2(O)CCOC2)=O)CC(O)C1)=O 62121,N1(C(Cc2c(OC)nccc2)=O)CCC2CN(C(c3ccnnc3C)=O)CC2C1 62122,CCCCC(CC)C(C(=O)Nc1ccc(F)cc1)N1CCCC1C1(C)CC1 62123,Cc1nc(Br)sc1NC(N1CCC(CC(=O)NC2CCOC2)CC1)=O 62124,C1(O)(CN(C(=O)C(O)Cc2ccccc2)C)CCN(C(=O)Cn2cccc2)C1 62125,N1(C(C2C(C)(NC(C(=O)N(C)C)=O)CCCC2)=O)CCOC2(CCCC2)C1 62126,S(=O)(=O)(c1cccc(=NC2CCOCC2)[nH]1)N(N1c2c(cccc2)CC(C)C1)C1CC1 62127,C1(C(=O)NC(C(C)(C)C)CNC(=O)CCc2cnc(O)[nH]2)CCC2CC1CO2 62128,Cc1nsc2ncc(C(N3CC(CC(C)NC(=O)Cc4ccon4)C3)=O)cc12 62129,N1(C(C(CCCC)=O)=O)CCC2(CCOC2)C(CNC(C2CCSC(C)C2)=O)C1 62130,C1(C(C)NC(C2(C(F)(F)F)CCCC2)=O)CCCN(C(=O)Cc2cnns2)C1 62131,C1(CNC(c2ccc(CC)cc2C)=O)CC2COCC2N1C(C1(F)CCC1)=O 62132,C1(N(C(=O)CC2CC(N)C2)CC)CCCCC1.C(=O)(C(C)c1ncco1)C(=O)CNC 62133,C1(C(=O)Nc2c(CC)ncs2)CC(F)(F)CN1Cc1ccn(C)n1 62134,c1(C(=O)NC2(CNC(c3ccn(C4CCCC4)n3)=O)CCC2)ccc(C(F)(F)F)o1 62135,C(=O)(C(CSC(C)(C)C)NC(c1cnn(CC)n1)=O)NC(c1ccccc1)C=C 62136,N1(C(CCCOCC=C)=O)CC2CC1CN2C(c1ncccc1C(=O)OC)=O 62137,c1(OC)cc([N+](=O)[O-])ccc1C(=O)NC1(CO)CCN(C(C2OCCO2)=O)C1 62138,C1(CC#C)(C(=O)NC2CC(CCNC(=O)COC(C)CC)C2)CCC1 62139,C=C(C)C(C)(O)C(=O)NC1CCN(C(C2Cc3ccccc3S2)=O)CC1 62140,C1(C=O)NCCOC1(C)C.C1(COC)CN2CC1C1CCCN21 62141,c1(C(=O)NC(CCNC(C(C)CO)=O)Cc2ccccc2)ncn2cccnc12 62142,CC1(CC(=O)O)CN(C(c2ccoc2CC(=O)NC)=O)C1.n1(CC2CCC2)ccnc1 62143,c1(OC)c(C(=O)NCC(C)(C2CC2)NC(c2ccc(CO)s2)=O)csc1C 62144,C1(C(=O)NCC(CC)NC(=O)CCOC2CCCC2)CC2(CC2)CO1 62145,C=CCC(C)(C(=O)NC1(CCNC(=O)Cc2ccc(F)cn2)CCCC1)N(C)C 62146,Cn1nc(C(=O)NCC23CC2CN(C(c2cc(C4CCC4)[nH]n2)=O)C3)cc1C#N 62147,C1(CNC(c2c(C)cn(C)n2)=O)CCN(C(=O)CCCC2CCC2)C12CC2 62148,C1(C(=O)NC(C)Cn2cccn2)C=CCN(C(C2CCCC(=O)C2)=O)C1 62149,N1(C(C2(C)COC2)=O)CCN(C(C2CCCC2n2cccc2)=O)C(CCO)C1 62150,c1(C(c2n(CCCC)nnn2)NCC(C(C)(C)C)SC)cccc2nonc12 62151,C(=O)(C1CCCc2nn[nH]c21)N1CC(O)(CCNC(c2nc(C)nc(O)c2)=O)C1 62152,N1(CC2N(C(CN(C)C)=O)CCCC2)CCN(C(=O)CCS(N)(=O)=O)CC1=O 62153,C1(CC(=O)NC2(CN(C)C(C3(C)C=CCCC3)=O)CC2)CCCC(=O)C1 62154,N1(C(COCCOCC)=O)CC2(C1)CN(C(C1CCCS1(=O)=O)=O)CC(C)(C)O2 62155,CCCC(O)CCNC(C1CCN(C(C2C3CC4C(C3)C24)=O)C1)=O 62156,CC(C(F)(F)C(F)(F)F)=CC(=O)NCCC1CCCN(C(C2CCCN2C)=O)CC1 62157,C1(C(=O)NC(C#CC)(C)C)CN(C(=O)CCS(C)(=O)=O)CC(C)O1 62158,C1(C)(C(N2CC(C(C)C)N(C(c3n[nH]c(O)n3)=O)CC2)=O)CCCNS1(=O)=O 62159,N1(C(C(C)(CO)OC)=O)CC(C(N2CCC(N3CCC3)CC2)=O)C2(CC2)C1 62160,C1(C(=O)NC)Cc2ccccc2N1C(c1ccc2c(c1)CNC2=O)=O 62161,c1(C(=O)NC(CN(C)C(C2CC2C(N)=O)=O)(C)C)ccc(Br)cc1F 62162,c1(CN(CCCCC)C2CCCC2)cc(C(F)F)cc(Cl)n1 62163,c1(C(=O)NCC(CO)NC(c2ccc3c(c2)CC3)=O)cc2n(n1)CCC2 62164,N1(C(c2cc(CC)no2)=O)CCCC2(CCN(C(=O)C(C)S)C2)C1.CO 62165,Cc1cc(Cl)c(C(N2CC(CNC(=O)CC3(CO)CCCCC3)CC2C)=O)cc1C 62166,C(c1ccccc1)=C(CC)C(=O)NCC12CC(N)(C1)C2.C12(CC1)C(=O)N2 62167,C1(COC)(NC(c2sccc2F)=O)CCN(C(=O)CC2(O)CCOCC2)C1 62168,N1(C(C)C(=O)Nc2ccc(CCN)cc2)CCC2CCCC12 62169,N1(C(COC(C)(C)C)=O)CCCN(C(=O)CS(=O)(=O)Cc2cccs2)CCC1 62170,C1(C)(C(=O)NCC(CCNC(C2(CCOCC)CCCC2)=O)O)CCCC1(F)F 62171,CC1CCCC(n2nccc2NC(=O)N(C)CC2CC2(C)C)C1 62172,Cc1cc(C(N2CCC3CC23C(=O)Nc2cccc(C3CC3)c2)=O)nc(C)n1 62173,c1(C(=O)NCC(=O)N(CC)CC)cc2cc(-c3cc(C)cs3)cnc2[nH]1 62174,c1(N(CCCNC(c2c[nH]cc2C(=O)OC)=O)CC)cc(Cl)nc(SC)n1 62175,c1(CC)cnc(C(N2CCC(C(N3CCC3(CO)CO)=O)(CO)C2)=O)nc1 62176,CC1(C)C2CCN1C(=O)c1cccc(c1)C(=O)NC2.c1(C(=O)NC)ccncc1Cl 62177,CC1C(C(=O)Nc2cnn(CCF)c2)CCCN1C(=O)CCCN1CCCC1 62178,c1(CCC)cc(C(=O)NC2CC(F)(CNC(=O)COCCC(C)C)C2)n[nH]1 62179,C1(n2nc(C)n(-c3ccccc3)c2=O)CC2CCCC2N1CC(F)F 62180,C1(C(N2CCC(NC(c3cncc(C)c3)=O)C2C)=O)CCOCC1(C)C 62181,c1(CC)ccc(C(N2CCC(O)(C(=O)N(CC(C)C)CC)CC2)=O)cc1Br 62182,CC(C)(F)CCC(=O)NCCCNC(c1cc(-c2ccc(Cl)cc2)ns1)=O 62183,C(=O)(C(O)C(CCC)NC(c1cc(O)n(C)n1)=O)NCCC(CCC)O 62184,c1(OC)ccc2[nH]c(C(N3CCSC(C(=O)NCC(C)O)C3)=O)cc2c1 62185,N1(C(CC2C=CC(NC(c3nc(C)n(C)c3)=O)C2)=O)CC2CC(CO)C(C2)C1 62186,C1(CNC(=O)COCCF)(CO)CC1(F)F.C12(CC1)C(=O)N2 62187,N1(C(C(CCC)C(C)C)=O)CC(NC(=O)C(C)(C)CS(C)(=O)=O)CC12CCCC2 62188,C1(NC(CNC(C(C)(C)C)=O)=O)CCN(C(=O)CN2CCCC2)CC1(C)C 62189,C(=O)(CCC(F)(F)CN=[N+]=[N-])N1CC(O)(C(C)NC(c2ccc(C(N)=O)o2)=O)C1 62190,O=C(CCCC(=O)N1CCN(C(=O)C(O)C2CC2)CC1)c1cccs1 62191,c1(C(=O)NC2C(C)CN(C(=O)C(F)F)CC2)nc2ccc(Br)cn2n1 62192,C1(C(=O)NCC(C)(C)NC(C2CCC(F)CC2)=O)CCc2nncn2C1 62193,c1(CNC(=NCC)NCC2COC(C)(C)C2)nn(C)c2cccnc12 62194,CCCCC(C(=O)N1CCC(F)C(NC(c2cocc2C)=O)C1)ON=C(C)C 62195,C(=O)(CCCNC(c1cnn(CC2CC2)c1)=O)N1C(CN=[N+]=[N-])CC1 62196,N1(C(C2CCN(C(C(C)C#N)=O)CC2O)=O)CCC2C(O)C(C)(C)C12 62197,Nc1sc2c(c1C(N1CCC(C3CC3)(NC(=O)CCC3CCCO3)C1)=O)CCC2 62198,C(=O)C(C1=CCSC1)N1CCC12CCCSC2.Cc1ccccc1 62199,N1(C(c2cc(C)[nH]n2)=O)CCCCC1CCC(=O)NC1CCCC=C1Br 62200,Cc1cccc(C)c1CCN=C(NCF)NC1CCCCN(C(=O)OC(C)(C)C)C1 62201,C1(C(N2CC(CC(C)NC)C2)=O)(CSCc2ccccc2)CCCO1 62202,c1(C(=O)NCC(CNC(C2CCC3CC23)=O)OC)ccc(=NCC2CC2)[nH]c1 62203,Cc1cc(N)ccc1C(=O)NCCN(C)C(C1(C2CCCO2)CCCC1)=O 62204,N1(C(c2c(SC)cn(C)n2)=O)CCC(C)(C)C(CNC(=O)C(C)=CC2CC2)C1 62205,c12cccc3oc(nc13)c1nc(no1)c1nc2no1.c12ccc-1o2.CCCCC 62206,N1(C(C(CCF)NC(c2n(CC)ccn2)=O)=O)CCSC(C)(C)C1 62207,C1(NC(=O)Cc2cc(C3CC3)no2)CCC(CNC(c2ocnc2C2CC2)=O)CC1 62208,c1(C(N(CCOCCN(C(C(F)OC)=O)C)C)=O)cc(-c2ccc(C)s2)[nH]n1 62209,c1(C(N2C(CNC(C(CC=C)OC)=O)C(C)(C)CC2)=O)cc(C)c(N)cc1Cl 62210,c1(OC)cccc(I)c1C(=O)OCC1CCN(S(=O)(=O)C(F)(F)F)C1 62211,c1(-c2scc(C)n2)nc(-c2ccc(C(C)C)o2)n(CCN(C)C)n1 62212,C(CCCCCC(=O)N1CC(CNC(C2OCCC2C)=O)CC1C)NC(C)=O 62213,c1(SCC(=O)NC(CNC(C(COC(C)=O)C)=O)C2CC2)c(C)n[nH]c1C 62214,c1(C(=O)NC2CC(CNC(C(C3CCCOCC3)OC)=O)C2)ccc([N+](=O)[O-])s1 62215,C1(CC(C)C)C(=O)NC2(CC(=O)NO1)CC2.N1(CC)CCCCC1C(=O)OC 62216,C1(NC(C2CC(C)N(C)CC2)=O)CC2CCC1CN2C(c1sccc1CC#N)=O 62217,N1(C(C2CCN(C)C2=O)=O)CC2CC(NC(C3(CCF)CC3)=O)C1C2 62218,C1(CNC(c2cn(CC=C)nc2)=O)CCCCN1C(c1c[nH]ccc1=O)=O 62219,C1(C(N(Cc2cccc(C(=O)F)c2)CC2CCC2)=O)CCC(N)C(O)C1 62220,C1(C(=O)NCCCC2(NC(CN(C)C(c3ccsc3)=O)=O)CC2)CC(F)(F)C1 62221,c1(C(=O)NC2C(CNC(C(C)(C)NS(C)(=O)=O)=O)CCC2)ccc2nccn2n1 62222,CC(C)(C)C(O)C(=O)N1CC(F)(F)CC1CCNC(C1CCNC1=O)=O 62223,C1(n2c(C(C)CO)nc(-c3cccs3)n2)CC2CCC1(C)C2(C)C 62224,C1(C(N2CC(CNC(CC(C)(C)C)=O)C(C)(C)C2)=O)CC2(O)C1OC21CCC1 62225,c1(N2CCC(C)(CN(C(c3cccnc3)=O)CC)CC2)cc(C)nc2nc(C)nn12 62226,N1(C(C(CCSC)N)=O)CCOC(C#N)C1.C(=O)(CCS)C(C)C 62227,c1(C(C)NCC(C)N(C)C)cn(C)nc1OC.c1ccccc1 62228,C(C(CC1CC1)C(=O)NCCCC1CCCCO1)NC(c1c(C)occ1)=O 62229,C1(C(=O)NC(C#C)CC2CCCO2)(CC#C)CCN(C(C2COCCN2C)=O)CC1 62230,C1(C(N2CC(C3(C)CC3)OCC2)=O)C2CCC(C2)N1C(C12CC(C#N)(C1)C2)=O 62231,Cc1cc(CC(=O)NCC(C2CCOC2)NC(c2c[nH]nc2C2CCC2)=O)no1 62232,N1(CCCCNC(c2c[nH]c(=N)o2)=O)CCN(C(c2cccnc2)=O)CC1 62233,C1(CC)CN(C(c2ccc(C(F)(F)F)o2)=O)CCC1NC(c1n[nH]c(C)c1Cl)=O 62234,C(C)(C(COC)C(C)C)NC(c1n(CCCSC)nnn1)c1cnc(OC)s1 62235,c1(C(=O)NC(C2CCN(C(=O)CC3(C#N)CCC3)C2)C)ccc2c(c1)CC2 62236,C1(C(N2CCC(CCCCCNC(CSSC)=O)CC2)=O)CCCCN(C)C1=O 62237,C12(N(C)C)CCC(C(=O)NC3C4CN(C(C5(C#N)CCCO5)=O)CC34)(CC1)CC2 62238,N1(C(C(C)n2cccn2)=O)C2CCC1CC(N(C)C(c1cnn(C)c1F)=O)C2 62239,Cc1ccc(Br)c(CN2CC(NC(c3cnc(Cl)s3)=O)C3(CC3)C2)c1F 62240,C1(OCC(=O)NCCN2CCN(C(C3CC3(F)Cl)=O)CC2)CCC(F)(F)CC1 62241,C1(C(=O)NCC2(C)CCC2)CCN(C(=O)Cc2ccncc2F)CC1(C)C 62242,Cc1cccc(CSCCC(C)CCO)c1C 62243,CCC(C)CC(C)C(=O)NCC1(C(N)=O)CN(C(c2ccc(OC)c(Cl)n2)=O)C1 62244,N(C1c2ccccc2CC1NC(=O)CNS(C)(=O)=O)C(C1CN(C)C(=O)C1)=O 62245,C1(C(=O)NC(c2nnnn2-c2ccccc2)CC)CCCN(c2cc(C)[nH]n2)C1 62246,c1(C(=O)OC(COC(C(c2c(C)cc(Br)cc2)(C)C)=O)C)ccc2occc2c1 62247,N1(CC)CC(NC(=O)NC2CC2C2CCCC2)CCC1=O 62248,Cc1ccc(-c2cnc(NC(=O)CNC(c3ccccc3C)=O)c(F)c2)cc1Cl 62249,c1(C(=O)NCC(CC=C)NC(c2ccc(NC)cn2)=O)ncccc1OC 62250,C1(CNC(C2CC(C)SCC2)=O)CN(C)CCN1C(c1cccnc1N)=O 62251,C1(C)(C(N(C2CSC2)C)=O)CCCN(CCC2NC(=O)NC2=O)C1 62252,c1(C(=O)NC(C(=O)NC(C)CF)Cn2cncn2)cc(O)ncn1 62253,C=CCC(C)(CC=C)NC(C1CC(OC)CCO1)=O 62254,C(=O)(C(C)COC(C)=O)NC(C=CC(=O)NC1(CC(=O)NC)CC1)C 62255,C(=O)(C1=CCC(C)CC1)N1CCC(CNC(C2CCCC(OC)C2)=O)CC1 62256,c1(C(C)(C)C)nc(C(=O)NCC2CN(C(c3cc[nH]n3)=O)C2)n[nH]1 62257,C1(NC(C(c2c(C)noc2C)C)=O)CCC2CN(C(c3ns[nH]c3=O)=O)CC2C1 62258,c1(NC(C(c2ccc(OC)cc2)N2CCCC2CCO)=O)cccc([N+](=O)[O-])c1 62259,n1(CC(=O)NC(C2CN(C(=O)CC(C)n3cccn3)C2)C)cc(C(F)(F)F)nn1 62260,c1(CC(=O)NCC2(NC(C(C)n3cccn3)=O)CCCC2)cccc(C(F)F)c1 62261,Cc1[nH]c(C(=O)NCC(O)CO)c(C)c1C(N1CCCC(N(C(C)CO)C)C1)=O 62262,Cc1csc(=NCC(=O)NCC2CC(C)N(C(c3cscc3F)=O)C2)[nH]1 62263,C1(NC(=O)CN2CC=CC2)CCC2(CCCN2C(=O)CS(=O)(=O)C2CCCC2)CC1 62264,CC1CCC(C(=O)NC(c2ncccn2)C)N1C(C12CC(C(=O)O)(C1)C2)=O 62265,C#CCC(C)(CC)C(=O)N1CCC(c2ccncc2)C1.N1(CC(=O)NCS)CCCC1=O 62266,C1(CCC)CCCC1C(=O)N(C(C)CCNC(=O)C(C)OCc1ccccc1)C 62267,c1(OC)cccc2c(OC(c3ccc(N4CCCCC4=O)cc3)=O)c(C)cnc12 62268,c1(OC)ccc(C(=O)NC2CC2C(=O)NCC2COCC2O)cc1F 62269,Cc1cnc(N(CC(C)NC(c2snnc2C)=O)C)nc1O 62270,N1(C(CS(=O)(=O)NC)=O)CC(C)(C)CC1C(N1CCC(c2cnn[nH]2)C1)=O 62271,Cc1noc(Cl)c1CC(=O)NC1CCN(C(=O)CC2C=CS(=O)(=O)C2)C1C 62272,N#Cc1ccc(CN2CCOC(CNC(=O)C=Cc3ccccc3F)C2)c(Cl)c1 62273,N1(C(CC=C)=O)CC=C(CC(=O)NC2CCCC2CN(C)C)CC1 62274,c1(CNC(c2ccc(C#C)o2)=O)nc2ccccc2s1.N12CCN(CC1)CC2=O 62275,CC1CC2(CO1)CN(C(=O)CCC1CCN(C(=O)CCc3ccsc3)C1)C2 62276,C1(C(N(CC(C)N(C)C(C23CC(F)(C2)C3)=O)C)=O)CCCCS1 62277,c1(C(=O)NC(CC=C)CNC(C2CCCC23CCC3)=O)ccnc2c1cnn2C 62278,N1(C(c2c(OCC)oc(C)n2)=O)CCC(NC(C2CC=CCO2)=O)C(C)C1 62279,C12(NC(c3sc(C)c(O)n3)=O)CC(C)(C1)OC21CN(C(C2CCC(F)C2)=O)C1 62280,Cc1cc(CNC(=O)CCN(C(=O)CC2CCC3CC23)CCO)sn1 62281,N1(C(C2CCN(C(Cn3nc(C)oc3=O)=O)CC2)=O)CC(C)OCC1C 62282,N12CCC3(CCN1CC3)C2.Cc1nn(CC(C)C)c(=O)o1.C(=O)CCS 62283,C(=O)(CC1=CCCC1)N(C1CCC(NC(c2c(C)noc2C(C)C)=O)C1)C 62284,C1(C(=O)NCc2cn(C)nn2)CC(C)(C)CCN1C(=O)CCc1ccccc1 62285,Cc1cc(=O)oc(C)c1C(=O)N(C)CC1(NC(=O)C2=CC3CCC2C3)CC1 62286,C12(C(=O)NCCCCC(C)NC(C(COC)O)=O)CCC(N=[N+]=[N-])C1C2 62287,N1(C(C(COC)C)=O)CC(N(C)C(c2[nH]nc(C(F)(F)F)c2C)=O)C(O)C1 62288,c1(CNC(C2N(C(CC)=O)C(C3CC3)CC2)=O)nn(C)c(=O)n1C 62289,c1(C(=O)NCC(N(C)C(c2cccc3[nH]ncc23)=O)C2CC2)coc2c1COC2 62290,CCC(C)(CC(=O)N(CCCN(C)C(c1ccc(O)c(C)c1C)=O)C)C(=O)OC 62291,N1(C(c2c(C)nc(CNC(CSCCC)=O)o2)=O)CCC2CN(C)CC2C1 62292,Cc1[nH]nc2c1CC(C(N1CCN(C(=O)CC(C)(F)F)C(CC(F)F)C1)=O)CC2 62293,c1(C(=O)NCCN(C)C(C2CC2(Cl)C(N)=O)=O)ccc2c(c1)NCCC2=O 62294,C(CC(N)=O)(C(=O)NCc1noc(C2CC2)n1)NC(CCCC#C)=O 62295,N1(C(C(=O)N2CC(CCNC(C(CC)SC)=O)C2)(C)C)CCN(C(C)C)CC1 62296,C1(CN(C)C(C2CCCCC2)=O)CCCN1C(=O)CCCn1ccnc1 62297,c1(C(=O)NC2CCCC(NC(C3CCC(F)(F)C3)=O)C2)cc(F)ccc1C1CC1 62298,N1(C(CCC(C)OC)=O)CCC2(CC1)CCN(C(C1(S(N)(=O)=O)CCCC1)=O)C2 62299,C(=O)(C(F)CC(C)(C)NC(C1CC2CCC2C1)=O)NCC(C(C)C)(C)O 62300,Cc1ccc(C(=O)NCC(C)(C)OCCNC(=O)CC2CC(=O)NC2=O)cc1F 62301,C1(C(=O)NCCCNC(Cc2c(C(=O)OCC)scn2)=O)CC(=O)N(CCOC)C1 62302,n1(CC)ncc2c1CCCC2Cc1nc(C(F)F)nn1-c1cccnc1 62303,C1(NC(C2C(C(=O)NCCCOC3CC3)CC=CC2)=O)CCCCC12CCC2 62304,CCCCC(C(=O)NCCC(C)(O)CC)NC(=O)CC1OCCC1C 62305,c1(C(=O)NC2CC(C)(CNC(C3(c4ccncc4)CC3)=O)C2)ccc(O)nn1 62306,O=[N+]([O-])c1cc(Cl)ccc1CN1CCC(N2CCCC2)C(F)C1 62307,c1(C(N2CCC(CN(C(C(CC#C)O)=O)C)CC2)=O)cccn2nnnc12 62308,CC(c1ccsc1)=CC(=O)NC(C)(C)C(C)NC(=O)CC(C)n1ccnc1 62309,c1(C(C)C)nc2cccc(C(N3CCSCC3CCNC(=O)CC(C)O)=O)c2[nH]1 62310,c1(C(=O)NC(CC(=O)NC)C(=O)O)nn(Cc2ccccc2)c2ccc(Br)cc12 62311,Cc1cc(F)ccc1NC(=O)C(CC1CC1)NC(c1ccccc1F)=O 62312,c1(C(=O)OC(C)C(=O)Nc2ccc(N(C)C)cc2)cc(Br)c2occc2c1 62313,N1(C(c2c(CC)nn[nH]2)=O)CC2CC2(CNC(=O)Cc2cncs2)C1 62314,c1(CC)cc(C(N2CCCC2CNC(=O)Cc2cc(C)[nH]n2)=O)ns1 62315,c1(C(=O)NC(CC)CN(C)C(C2(CC(=O)OC)CC2)=O)cnc(O)c(F)c1 62316,CC1CN(C(=O)CCC2(C)CCCN2C(C23C(=O)C4CC2C3C4)=O)CC1(C)C 62317,c1(C2(C(=O)NC(CCCN(CC)Cc3nccs3)C)CC2)cccc(C(F)(F)F)c1 62318,C1(NC(C2(CC=C)CC2)=O)CCC2(CC1)CN(C(=O)C(c1ccc(Br)cc1)=O)C2 62319,Cn1cc(C(N)=O)n(C)c1=O.C12CCCC1C(=O)N1CCCC1CC(=O)NC2 62320,CC1C(NC(C2(NC(C3(C)CC3(F)F)=O)CC2)=O)CC2CCC1N2C(N)=O 62321,N1(C(C(C)Sc2nncs2)=O)CCn2c(C3CC3)nnc2C1 62322,C1(CNC(C=CC=CC)=O)CC(O)CN1C(c1scc(C(F)(F)F)c1C)=O 62323,Cc1ccccc1-c1cc(COC(=O)C=CCCC(C)C)nn1C 62324,Cc1c(N2C(C(=O)NC(=O)CCc3cn(C)cn3)CCC2C(C)C)cccc1CO 62325,c1(OC)cc(C)ccc1CNC(=O)C(F)C1CC(NC(=O)C2=CCCC2)C1 62326,Cc1ccc([N+](=O)[O-])c(NCC(=O)N(CC(C)CO)CCN)c1 62327,C1(SCC2(CNC(N(CCOC)C)=O)CC2)CCCOC1 62328,c1(CNC(c2cc(C)[nH]n2)=O)ccc(C(=O)NC2CCC2CN(C)C)nc1 62329,N1(C(C2ON=C(C)C2)=O)CCN(C)C(CNC(=O)CC=Cc2ccccc2F)C1 62330,C1(C(=O)NC(CC=C)CNC(=O)C(c2cncn2C)O)CCCCC1O 62331,C1(NC(C2(CNC(c3c(CC)cccc3)=O)CCCO2)=O)CN(C)CC12CC2 62332,O=S(=O)(c1ccccc1)C1CCN(c2nc3c(F)cc(Cl)cc3s2)C1 62333,c1(C(N(C(CNC(c2nc(C(=O)OC)sc2)=O)C)C)=O)ccc2cncn2c1C 62334,N1(C(C2CN(C)C(=O)C2)=O)CC(O)(C2(CNC(=O)C(F)CC3CCC3)CC2)C1 62335,C1(NC(C=CC(C)(C)NC(C(CSC)O)=O)=O)CCCCC12CC2 62336,c1(N(C)CC2CCCS2)cc(N2CCCN(CCCO)CC2)nc(CN(C)C)n1 62337,c1(C(=O)NC(C(C)N(C(c2ccc(OC)cc2)=O)CC)C)cccc2nncn12 62338,c1(C(=O)NC(CCNC(c2c(CC)[nH]c(=N)s2)=O)(C)C)cc2occc2[nH]1 62339,C1(NC(Cc2cn(CC)nc2)=O)CCC(C)N(C(c2cc(F)n[nH]2)=O)C1 62340,C1(NC(c2c(N)ccc(Cl)n2)=O)CC12CCN(C(c1ncccc1Cl)=O)CC2 62341,CCC(CC(F)F)C(=O)NC(C1CCN(C(=O)Cn2cc(C)cn2)CC1)(C)C 62342,CCCCCC(C(=O)NCCC1CN(C(=O)C=Cc2ncc[nH]2)CC1C)C(C)C 62343,C1(OCC(=O)NCC2(F)CCN(C(C(C)n3cccn3)=O)C2)CCC(F)(F)CC1 62344,c1(CC)cc(C)c(C(N2CCC(N(C)C(c3cscc3Cl)=O)C2)=O)o1 62345,Cn1c(C(=O)NCCC2CCC(NC(c3cnc(CC4CC4)s3)=O)C2)cnc1Cl 62346,c1(C(CC(=O)NCCCOC)NC(c2nccn2C)=O)ccc(C#N)cc1 62347,CC1CN(CC(=O)NCc2cnn(CC(F)(F)F)n2)CC2(CCC2)O1 62348,c1(Cc2ncc(-c3nc(C)c(CNC)s3)cn2)ccc(O)c(Cl)c1 62349,C(N=c1nc(N2CCC(C(N)=O)C2)c2c([nH]1)CCS2)C1CN(CC(F)F)C1 62350,C1(c2n(CC)ncc2)CCN(C(C2(C(=O)NC)CCCN2C)=O)CC1 62351,C(=O)(CCC(=O)NC1CC1)NCC(C(=O)NCCCn1ccnc1)OC.C(C)(=O)O 62352,C1(O)(C(=O)NCCCc2n(C)nnn2)CCN(C(c2ccn(C3CC3)n2)=O)CC1 62353,c1(C(N2CC(O)(CN(C(CC3C(C)C3)=O)C3CC3)C2)=O)snc(Cl)c1Cl 62354,C1(NC(CC(C)(C)OC)=O)CCN(C(C2CCCN2C=O)=O)CC1(C)C 62355,C1(OC)CC(CNC(C2(C(F)F)CC(O)C2)=O)N(C(c2cc[nH]c2)=O)C1 62356,c1(C(=O)NC(CC(C)C)CNC(C2(C#N)CCC2)=O)cc(Cl)cc2ccncc12 62357,N1(C(c2ccc(OC)cc2F)=O)CCC2C(C1)CN2C(=O)CSC1CCCCO1 62358,C=C1CC2CCC(C1)N2C(C1CCC(C)CN1C(=O)CC1CC(OCC)C1)=O 62359,N1(C(c2c(C)snn2)=O)CCC(C2CCN(C(=O)CC(C)(C)C)C2)CC1 62360,C1(C(=O)NC(C(CC)C)C)CCC(NC(=O)NC)CCC1 62361,n1(NC(=O)OC)cc(-c2sccc2C(=O)NC(C2(C(=O)NC)CCC2)=O)nn1 62362,C=CCS(=O)(=O)CCNCC(=O)N(C)Cc1nnc(-c2ccccc2Br)o1 62363,CC(C)CCC(O)C(=O)NCC(F)CNC(c1cc(C2(C)CC2)on1)=O 62364,C1(C(N2CCC(OC)CC2)=O)C(C)OCCN1C(C1CCC1C)=O 62365,C1(CCC)CN(C(=O)CCCOC(C)=O)CC1NC(C1CCS(=O)CC1)=O 62366,CC(C)(C)C(CNC(=O)CC1CC2CC2C1)NC(c1cccc(C(F)(F)F)c1)=O 62367,c1(C(=O)NCCC2CC(Nc3nc(SC)c(C)cn3)C2)cnn2c1C(=O)NCC2 62368,N1(C(C2N(C(COC(C)=O)=O)CC=CC2)=O)CC(C)(C2CCC2)C1 62369,c1(C(=O)NC(CCCC)CNC(=O)C(C)(C)n2cnnn2)nc(OC)ccc1C 62370,C1(C(N2CCC(NC(C3CCCC3)=O)C2)=O)COc2ccc(F)cc2C1 62371,c1(CCNC(=O)NCCCCCl)cc(O)nc(O)n1 62372,c1(C(N2CCC(N(C)C(c3ccc[nH]3)=O)C2)=O)cnc(CC2CCC2)nc1O 62373,c1(CC)cnc(O)c(C(N2CCC(N(C(=O)C(O)C3CC3)C)C(C)C2)=O)c1 62374,C1(C(=O)NCCCN(C(C2CCCC(F)(F)C2)=O)C2CC2)CCC2(CCC2)CO1 62375,Cc1cc(Br)cc(CNc2ccc3ccoc3c2)c1O.N12CC3CC1C3C2=O 62376,Cc1cccc2[nH]c(C(N3CC4CC(NC(=O)Cc5csc(S)n5)C3C4)=O)cc12 62377,N1(C(C(CC)(C)CO)=O)CCC2C(C1)NC(=O)CN2C(=O)C(CO)N(C)C 62378,c1(NC(CC2CCC(NC(C(C)(C)F)=O)C2)=O)ccc2c(c1)CCCC2 62379,CN1CCC(O)(C2(C(N3CCCC3C3CCN(C(=O)CS(C)(=O)=O)C3)=O)CC2)CC1 62380,Cc1nc(CNC(c2ccc(CNC(c3csc(F)c3)=O)nc2)=O)sc1C 62381,CC1CN(C(c2cc3ccccc3o2)=O)CCCN1C(=O)CSC1CC1 62382,N1(C(CCCCC#C)=O)CCCC2C(NC(=O)CCC3CCCCC3)CCCC12 62383,C1(N(C(COCC#C)=O)C)CCCCN(C(=O)CSCCC)C1 62384,C(=O)(C(CCS(C)(=O)=O)c1cn(C2CC2)nn1)N(C(C)(C)CSC)C1CCCC1 62385,N1(C(C2CCO2)Cn2cc(CC(=O)OC)nn2)CCOCC1Cl 62386,N1(C(c2c(CC)non2)=O)CCC12CN(C(c1c(C(F)F)cccc1N)=O)C2 62387,c1(OCC)ccc(C(=O)NC2(CF)CCN(C(=O)C(C(C)C)OC(C)C)C2)cn1 62388,N1(C(C2CCCC(=O)O2)=O)CCOC2CCN(C(c3cc(Cl)ccc3Cl)=O)CC12 62389,C1(O)(CNC(C(CC)OCC)=O)CCN(C(C2(c3ccnc(Cl)c3)CC2)=O)C1 62390,C1(COC)CN(C(=O)C(C)(COC)OC)CCN1CC(C1CC(=O)N(OC)C1)=O 62391,c1(COC(COCCC(C)C)=O)ccc(C2CC2)cc1 62392,N1(C(C2(CCN3CCN(C(COC)=O)CC3)CCC2)=O)CCN(CCO)C(=O)C1 62393,S(=O)(=O)(c1cc(Br)cnc1N)N1CCN(C(C)C2CC2)CC1 62394,Cc1cc(F)cnc1C(N1CCCC(CNC(c2cn(C)ccc2=O)=O)CC1)=O 62395,CC1CC(CNC(=O)C(C)(C)c2ccccc2)CN1C(=O)CCOCC(F)(F)F 62396,c1(C(=O)NC2C(OC)CN(C(=O)C(C)c3ccco3)C2)cc(F)c(SC)cc1N 62397,C(CCCC(=O)N1C(CNC(C2CC2F)=O)CC2CC12)OCCC=C 62398,C1(NC(COCCCC)=O)CCCCC12CCCN(C(c1n[nH]c(CC)n1)=O)C2 62399,c1(SC)ccc(C)c(C(N2CC3(CCN(C(=O)C(c4cnn(C)c4)C)C3)C2)=O)c1 62400,C#Cc1ccccc1NC(C1CC(O)CN1C(=O)Cc1ccc(Cl)cc1)=O 62401,N12CC3C(C3C1)C2=O.c1(C)cc(C#N)cs1.c12ccc(nn1)n2NC(C)=O.N(C)C 62402,O=C1CCc2c(C(N3CCC(CCNC(C4(CCO)CC4)=O)C3)=O)cccc2N1 62403,C(=O)(C(C)(O)CC(C)C)N(C1CCCN(CC=CC)C1)CCC 62404,Cc1cc(C(=O)NC(C(C)NC(=O)C=CSc2nc[nH]n2)C(C)C)c(O)nc1C 62405,C1(CC=C)(NC(=O)C(C)OC)CCN(C(c2csc(C(C)NCCCC)n2)=O)C1 62406,C(=O)(CCCC(F)(F)F)NCCC1N(c2cc(C(=O)OC)ncn2)CCCC1 62407,C(=O)(C(C)(C)CCF)NCC1OCCN(C(COc2ccc(C)cc2)=O)C1 62408,c1(C(=O)NC2C(CNC(c3cnn(CC)n3)=O)CC2)ccc(Cl)cn1 62409,c1(OC)ccc(CC(O)C(=O)NCC(C)(C)CNC(C2(C)CC2(C)C)=O)cc1 62410,C(=O)(CCCS(C)(=O)=O)N(CCN(C(CC(c1ccccc1)NC(C)=O)=O)C)C 62411,N1(C(C2=NNC(=O)CC2)=O)CCC2C(CCN2C(=O)C(CC(F)F)C2CCC2)C1 62412,C1(C(=O)NC2CCC(N(C(=O)C3=CCCSC3)C)C2)(OCC)CCCCCC1 62413,C1(C(=O)NCCCOCCCNC(C(n2ccc(C)n2)C)=O)CCCCCCC1 62414,c1(CC(=O)NCCN(CCC)C(C2CCCCC2C)=O)ccc(O)cc1 62415,c1(NC(C2CC(=C)CN2C(c2ccncc2Br)=O)=O)ccc(OC)nc1Br 62416,n1(CC=C)cc(C(=O)NCCCCCNC(=O)C(C)(C2CCOCC2)OC)nn1 62417,c1(CC)c(NC(C2CCN(C(c3ccn(CCN(C)C)n3)=O)C2)=O)ncnc1Cl 62418,N1(C(CC(CCC)O)=O)CC2CC1CCC2NC(=O)CCc1nnc(C)n1C 62419,c1(CC)cccc(C(=O)NCCOCCCN(C)C(c2cccc(C)n2)=O)c1F 62420,C(=O)(C1=CCC(NC(C2(C)COC(=O)N2)=O)C1)NC(c1nnc(C)o1)C 62421,C=CCC(CNC(=O)CCn1cnnn1)C(=O)NCC1CCCCCCC1 62422,C1(NC(N2C3C(C(=O)OC(C)(C)C)C(CC3O)C2)=O)CCc2nnn(C)c2C1 62423,c1(C(N(C(CCNC2C3CCCCCC23)C(C)C)CC)=O)ccnc2ccsc12 62424,N1(C(c2cccc(CSC)c2)=O)CC(NC(C2C=C2C)=O)C2(CCC2)C1 62425,N1(CC2C(C)CCCC2)C(=O)CN(CCn2cncn2)C1=O 62426,N1(C(CCC#C)=O)CCCC(NC(C2CCCN2C(=O)OC)=O)C1 62427,c1(N(C)CC2CCCC2Cl)nc(C(F)(F)F)ns1 62428,N1(C(C2(C=C)CCN(C(c3ccncc3)C)C2)=O)CC2CCC(OC)C2C1 62429,CCC(O)C(F)(F)C(=O)NCC1C2CN(C(C3(C(=O)N(C)C(C)C)CC3)=O)CC12 62430,c1(C(=O)NC2(CNC(c3c(CC)nns3)=O)CCCC2)cc2c(cn1)CCCC2 62431,C1(C(=O)NC(CNC(C2(CC)CCCO2)=O)CC(F)(F)F)CN2CCN1CC2C 62432,N1(C(C2C(C)(CC)C2)=O)CC=C(C(=O)N2CCCOCC2C)CC1 62433,N1(C(Cc2n(C)ccc2)=O)CCC2C(CCCN2C(c2cnn3c2CCC3)=O)C1 62434,C=CCCCCCCC(=O)N1CCC(CNC(=O)C(F)(F)c2cccnc2)CC1C 62435,C1(C(=O)NC2CCC(NC(CC3(C)CC3F)=O)CC2)CCCCCCC1 62436,C(=O)(CC1NC(=O)c2ccccc21)N(C1CCCN(C(C2(O)CCC2)=O)CC1)C 62437,CC1CN(C(c2cccc[n+]2[O-])=O)CCC1CNC(=O)COc1ccc(F)cn1 62438,c1(C(N(C2CCN(C(c3cc(O)cc(F)c3F)=O)C2)C)=O)csc(S(N)(=O)=O)c1 62439,S(=O)(=O)(c1c[nH]c(C(=O)NC2CCN(C(c3cc(Cl)cnc3O)=O)C2)c1)N(C)C 62440,C1(CNC(c2cc(C)sc2C)=O)N(C(C2CCOCC2(C)C)=O)CCCC1(C)C 62441,N1(C(c2cscc2F)=O)CCCC2(C1)CN(C(C1CC(O)C13CCC3)=O)CCO2 62442,S(=O)(=O)(c1ccc(N2CC(CO)C3(CCC3)C2)cc1Cl)NCC1(CC(C)C)CC1 62443,CC1CC(C#N)(C(N2CCC(CNC(=O)CC3CCN(C)C3=O)CC2)=O)C1 62444,c1(C(C)=O)cc(=NCC2CC(NC(c3cc(Br)co3)=O)C2)[nH]cn1 62445,Cc1ccc(Cl)c(C(N2CCC(CCNC(C3CCCCO3)=O)C2)=O)c1N 62446,C1(C2CCN(C(c3ccc4cncn4c3)=O)C2)(NC(C=CCC)=O)CC1 62447,C1(O)(CNC(c2cnc(C(C)=O)s2)=O)CCN(C(=O)CN2CCCCC2C)CC1 62448,c1(N2CC(CO)OCC2)[nH]c(=NCCC(O)C2CC2)nc2sccc12 62449,C1(CNC(c2nccc(C)c2)=O)COC(C)(C)CN1C(C1CC(F)C1)=O 62450,Cc1cc(C(=O)NCC(O)CCNC(=O)C(C)C2CCC2)c2c(n1)CCCC2=O 62451,C1(CCNC(Cc2c(C)n[nH]c2)=O)CN(C(=O)CCCC(=O)N(C)C)CC(C)O1 62452,C1(CC(N2C(CNC(c3ncccc3Cl)=O)CC2)=O)CC2(CCC2)CCO1 62453,c1(C(N(CCCNC(c2ocnc2C)=O)CC)=O)cc2cc(Cl)ccc2o1 62454,C(=O)(C(F)C(C)C)NCCC1N(C(c2nc(C(=O)NCC(=C)C)sc2)=O)CCC1 62455,CC1CCc2ncc(C(=O)NC3(C(F)F)CC(NC(=O)CC4(C)CC4(F)F)C3)n2C1 62456,c1(CC(=O)N(CC(C)NC(c2cnc(O)c(F)c2)=O)CC)cnn2c1OCCC2 62457,CCC(CC)(CCNC(C1CC2(CCO1)CC2)=O)NC(C1C(C)(C)C1(F)F)=O 62458,S(=O)(=O)(c1ccncc1)NC1CCC(NC(c2ccccc2Cl)=O)C1 62459,C1(C#N)(NC(Cc2c(SC)cccc2)=O)CCN(Cc2ccnn2C)C1 62460,C1(C(N2CCC(CC(=O)Nc3cscc3Cl)C2)=O)(COC)CCOC1 62461,N1(C(COC)=O)CCCCC1C1CCCN1CC(=O)OC.N12CCC(CC1)C2=O 62462,c1(C(=O)NCC2OCCN(C(C(CCC)C)=O)C2)c(C)nn(C)c1-n1ccnc1C 62463,C1(NC(CC(C)F)=O)CC(F)CN(C(c2cccc(-c3cccs3)n2)=O)C1 62464,c1(C(=O)NCCSCC(=O)N(C(CC)C2CC2)C)ccncc1Cl 62465,C(CCN(C)C)(C(=O)NC(C)(C)CCCO)NC(Cn1c(C)ncc1)=O 62466,CC(C)C(C(=O)NCCOC1CN(C(c2ccc(O)nc2)=O)C1)N(C)C 62467,N1(C(C2N(C(c3ccc(C)s3)=O)C(C3CC3)CC2)=O)CC2(CCOCC2)C1 62468,C(=O)(C1CCCc2nc[nH]c21)NCCCNC(c1c(C)n(C2CC2)cc1)=O 62469,c1(OCCOC)cnc(C(=O)N(C)CC2CN(C(=O)C(C)CF)CCO2)cn1 62470,CC1CCCCN1CC(=O)N(CCCCNC(c1cccc(SC2CC2)c1)=O)C 62471,N1(C(C(CC=CC)C)=O)CCN(C(=O)COc2ccc(SC)cc2)CC1C(C)C 62472,Cc1nc(O)nc(O)c1CCC(=O)N(C(C)CNC(=O)CSCCC#N)C 62473,c1(C(N(C2CCCC2)CCNC(C(C)NC(CC)(C)C)=O)=O)sccc1Br 62474,c1(OC)ncc(C(=O)NCCCn2cc(-c3cccnc3O)nn2)c(C)c1Br 62475,c1(C(N(CC(=O)N(CC(=O)N(C)C)C)CC)=O)ccc(C#N)n1C 62476,N1(C(c2cnn(C)c2Cl)=O)C2CCC(C2)C1CNC(C1(C#N)CCCCC1)=O 62477,CC(C(=O)NN1CCCC1C(=O)N(CCN=[N+]=[N-])CC)=CC1CC1 62478,Cc1cc(C(=O)NC2CS(=O)(=O)CC2NC(=O)C(C(C)C)N(C)C)cc(C)n1 62479,CC(C)(O)C(F)C(=O)N1CC=CC1CNC(C1(c2cc[nH]n2)CCC1)=O 62480,CCCCCCC(=O)N1CCCCC1CNC(c1c(Cl)cncc1Cl)=O 62481,N1(C(C)C)CCC2C1CCCN2C(=O)CCCCn1cc(C(C)N(C)C)nn1 62482,c1(OC)ccc(C(N2CCCC(NC(=O)CCC(C)N(C)C)C2C)=O)c(C)n1 62483,c1(C(=O)OCC)cnc(NC2(O)CCN(C(=O)CCCc3nncn3C)C2)cn1 62484,CC(C)C(O)C(=O)NCC(CC(C)C)NC(=O)CCCc1ccccc1N 62485,C1(C(=O)NC2C(C(=O)Nc3cncc(OC)c3)CCC2)Cc2ccccc2C1 62486,CC(C)(C)CC(F)C(=O)NC1CN(C(c2ncc(F)cn2)=O)C(C)(C)C1 62487,N1(C(CCCc2scc(C)n2)=O)CCN(C(=O)CCCCC2CC2)C(C(C)C)C1 62488,N1(C(C(C)SC)=O)CCCC(C2CCN(C(=O)C(C3CCC(=O)N3)C)C2)C1 62489,c1(C(N2CCC(CCCCNC(C(CCC)C)=O)CC2)=O)cn2c(n1)SCC2 62490,C1(CC=C)(NC(=O)C(c2cnn(C)c2)C)CN(C(C2CC(OC(F)(F)F)C2)=O)C1 62491,CCC(CC)C(C)C(=O)NC1CCC(F)(CNC(c2n[nH]c(C)n2)=O)C1 62492,C1(CCC(=O)N(CC(C)(C)C)CC)CCCCN1C(=O)CN(C)C1CC1.C(N)=O 62493,c1(C(=O)NC(CCCNC(C(CC)C(C)O)=O)C)cc(C)c2nc(C)cn2n1 62494,NS(=O)(=O)c1ccc(C(=O)NC2C3CCN(C(=O)Cc4c[nH]nc4O)CC23)cc1 62495,C1(CN(C)C(c2cc[nH]n2)=O)CC(O)CN1C(C1CCC(Cc2ccco2)O1)=O 62496,C#CC1(O)CCCN(C(C2(N(C)C(C3CCCC(C#N)C3)=O)CC2)=O)C1 62497,C1(CNC(CCC(C)O)=O)CCCC12CCN(C(=O)C(=O)C(C)(C)C)CC2 62498,Cc1cnn(C)c1CNC(C1CC1C#N)=O.C12(CCCC1)CC(=O)N2C 62499,C1(NC(c2cc(C)sn2)=O)C2CC1N(C(c1cccc(N)c1Br)=O)C2C 62500,C1(=CC(N2C(C)CCC(NC(CCN(CC)CC)=O)C2)=O)CCCCCC1(F)F 62501,C=CCCCC(C(=O)N1CC(n2cnnn2)C1)c1ccccc1 62502,C1(C(=O)NCCCC(C)NC(CCn2c(C)nc(C)n2)=O)COCC2(CCC2)O1 62503,Cc1cc(C(=O)NCC2CN(C(=O)CC3CC(F)(F)C3)C2)cc(S(C)(=O)=O)c1F 62504,N1(C(=O)CCC2CC2(F)F)CCN(C(=O)C2CC2)C(c2cn[nH]c2)C1 62505,N1(C(c2cc(OC)no2)=O)CCC(O)C(NC(=O)Cc2ccc(C)cc2Cl)C1 62506,c1(C(N2CC(C)C(NC(c3c[nH]nc3C(F)(F)F)=O)C2)=O)ccc(Cl)c(F)c1 62507,C(CN=C(NCc1cnco1)NCC1CCCCC1C)OC(C)CC 62508,C#Cc1ccc(C(=O)NC2(C)CCCCC2C(N2CC(F)(F)CC2C)=O)cc1 62509,C(=O)(C(O)CC(C)C)N1CC2C(NC(c3n[nH]c(C)c3Cl)=O)(C2)C1 62510,c1(NC(c2c(CC)cccc2)c2nnnn2C(C)C)cc(C)cc(Br)c1 62511,C(=O)(C1CCc2c[nH]nc21)NC1(C2CCN(C(COC)=O)C2)CC1 62512,CCCCC(=O)C(=O)N1CC(CNC(C2(CO)CCOCC2)=O)C(C)(C)C1 62513,N1(C(C(C2CCCN(C(c3c(C)scn3)=O)C2)(C)C)=O)CC2C(C1)C2(C)C 62514,C1(NC(CCC)=O)C(CNC(c2nc(C)ccc2F)=O)CCC12CCC2 62515,N1(C(CCN(C(C)=O)C)=O)CC2CCC1CN2C(c1csc(C(C)C)n1)=O 62516,N1(C(Cc2c(C)occ2)=O)C2CCC1CC(NC(C1CC(=O)N(C3CC3)C1)=O)C2 62517,C1(NC(c2cccn3ncnc23)=O)CN(C(=O)CC2OCCO2)C2(CCCC2)C1 62518,C(C(=O)N1CCC(C(N2C3CCC2CC3)=O)O1)c1c(=N)[nH][nH]c1 62519,C(C)(CC(=O)NCC(C)CNC(C1(CCN=[N+]=[N-])CC1)=O)OC 62520,c1(C(=O)NCC2(C)N(C(C(F)=CCC)=O)CC(OC)C2)cc(C)c(O)c(C)c1 62521,c1(C(N2CC(C)CC(C(N(CCC)CC)=O)C2)=O)c[nH]c2ccccc12 62522,c1(-c2nc(OCCCOC)on2)cccc(-c2csnn2)c1 62523,N1(C(C(C)CN2CCOCC2)=O)C(C)C2CC1C2NC(=O)C(C)(C)N(C)C 62524,CC(CC(=O)N1CCC(C2CCCN2C(c2ccc(CO)cn2)=O)C1)C(F)F 62525,C1(COC)(CNC(=O)C(Cc2ccccc2F)c2c[nH]nn2)CCCCC1.C(C)(=O)O 62526,CCC(CCCC(=O)N(CCCn1ccnc1)C)NC(=O)C(C)N1CCCC1 62527,n1(CCOC)nc(C)c(S(=O)(=O)Nc2ccccc2-n2nc(C)cc2C)c1C 62528,c1(CCC)nc(C(=O)N(CCO)CCO)cs1 62529,n1(CCC)nccc1C(=O)NCC(CC)N(C(=O)C(C)SCC)CC 62530,C(C(C)(C)CN(C)C)NC(CN(C(=O)CCc1ncco1)C(C)C)=O 62531,CC(CCCCNC(=O)CC1NC(=O)NC1=O)NC(=O)CSc1cccc[n+]1[O-] 62532,Cc1ccc(C2(SC3CC3)CC2)c(F)c1.c12ccccc1C(=O)NC(C)CNC2=O 62533,S(=O)(=O)(CC(=O)NCC(F)CNC(=O)C(N1CCOCC1=O)C)NC 62534,CCC(F)(F)CC(=O)NC(C)CN(C(=O)CCc1cccn(C)c1=O)C 62535,C(C(=O)N1CC(O)C(O)CO1)C1CCCN(C(CCC#CC)=O)C1C(F)(F)F 62536,c1(NC(C2CCC2)=O)nc(Cl)ccc1F.CC(C1CC1)=C(F)C(=O)NC1CC1 62537,Cn1ccc2ccc(C(N3CC4(CC(CNC(=O)CNC=O)C4)C3)=O)cc12 62538,C1(C(=O)NCCCNC(C2C(C)CC2C)=O)CCCCNC1=O 62539,c1(N(c2cnn3c2CNCC3)C(c2c(C)cnnc2)=O)ncnc2c1cnn2C 62540,c1(CCC)nnsc1C(=O)NCC#CCNC(c1ccnn1CCOC)=O 62541,CS(=O)(=O)c1ccc(CN2CC3C(Nc4ncc(I)cn4)C3C2)c(F)c1 62542,N1(C(CNC(NC)=S)=O)CC2CCCC2(N=c2cncc(Cl)[nH]2)C1 62543,c1(C(N2CC(CCCCCCNC(=O)C#CC3CC3)C2)=O)ccc2cccnn12 62544,Cc1oc(-c2ccco2)nc1CC(=O)NC1CCN(C(=O)COC2CCC2)C1 62545,N1(CC)N=C(C(=O)NC2CCC(NC(=O)C=CC(C)(C)C)C2)CCC1=O 62546,c1(OC)cccnc1C(F)(F)C(=O)NCC1CCCN(C(=O)C(CO)N(C)C)C1 62547,N#Cc1cccc(C(=O)NCC(CNC(=O)CC2CCC(=O)N2)C(F)(F)F)c1 62548,c1(C(=O)NC2CC(CNC(C3(C)CC(C)OCC3)=O)C2)cc2c(=O)cc[nH]c2s1 62549,C1(C(=O)NCCN(C(c2nocc2C(C)(C)C)=O)CC)CC=CCO1 62550,Cc1cc(CCC(=O)N(C)CC2CN(c3nccc(CO)n3)CCO2)cc(C)n1 62551,c1(C(=O)NCC(CC)NC(=O)CN(c2ccon2)C)c(C)c(Cl)cc(C)c1N 62552,C1(NC(c2cc(OC)no2)=O)CC2CC1CC2C(=O)Nc1cnn(C2CC2)c1 62553,N12CCCC(CC1)N2C.C(=O)(C(C)c1ccsc1)NC1CC(C=O)C1.C(C)(C)(C)O 62554,N1(C(C=CC(CC)C)=O)CC(N(C(=O)C=Cc2ccc(C(N)=O)cc2)C)C2(CC2)C1 62555,CCC(C)C(=O)NCC(=O)NCCCC(c1ccccc1)NC(=O)C(CC)SC 62556,C(=O)(C1CCOc2ccccc21)NC(C)C(C)(C)NC(c1scnc1Cl)=O 62557,C12(C(=O)NCCCN(C(=O)CC3CCCC34CC4)CC)CCC(F)(CC1)CC2 62558,C1(C(=O)NCC(CC)OC)CC2(CCC2O)C1.c12cc(nc(C(=O)OC)c1)NC2=O 62559,N1(C(=O)NCC(C)OC(F)F)CCC(C(=O)Nc2ccc(O)cc2F)C(C)C1 62560,N1(C(C(C)(C)OC)=O)CCC2(CCCC2NC(=O)C=Cc2sc(Cl)nc2Cl)C1 62561,C1(NC(Cc2ccc(C)cc2C)=O)CCCC12CCN(C(=O)Cc1cocn1)C2 62562,c1(-c2cc(C(N(CCC)CCNC(=O)C(F)OC)=O)sn2)cccc(Cl)c1 62563,c1(C(C(=O)NC2CC2)N(C2CC2)CC)cc(Cl)cc2cccnc12 62564,c1(CC(=O)NCC2CCC(NC(CN(C)C)=O)CC2)coc2ccccc12 62565,C1(N(C(CNC(C(CC)C)=O)=O)C)CCCN(C(c2ccnc(S)c2)=O)C1 62566,N1(C(CNC=O)=O)CCCC(NC(c2ncc(Br)cc2F)=O)C(F)C1 62567,c1(C(=O)NC2CC(NC(c3ccc(Cl)nc3O)=O)C2)cc2nn[nH]c2cc1F 62568,C1(O)(CNC(C2C(C)OCC2)=O)CCCN(Cc2cc(F)cc(Br)c2)C1 62569,C=CCC(C)C(=O)NCC(O)CNC(C1CC1c1ccccc1)=O 62570,C=CCC(C(=O)NCCCCC(C)NC(=O)COC1(C)CCC1)OC 62571,N1(C(=O)C(F)(F)Cc2ccccc2)CCCC(NC(C23CCCC2CC3)=O)CC1 62572,C(N=c1[nH]c2ccc(Cl)cc2s1)C1CCC(NC(=O)C(F)(F)C(F)(F)F)C1 62573,c1(C(=O)NCC(CCOC)NC(=O)Cc2ccc(Cl)nc2O)c[nH]cc(C)c1=O 62574,C1(CC(=O)N(C)C)CCN(C(=O)C(C2CCOCC2)F)C1.c1ccc(Cl)s1 62575,C(=O)(C(CNC(=O)C=C(C)C(C)C)CC(C)C)NCC(CC)(C)O 62576,c1(C(=O)NCCN(C(=O)C(O)Cc2ccc(F)cc2)C)coc2c1C(O)CCC2 62577,c1(C(N2CC(COC)(NC(c3cnc(COC)s3)=O)C2)=O)nc(C(C)C)oc1C 62578,Cc1ccc2cccnc2c1CNC(C1CC(=O)N(C)C1)=O 62579,Cc1cc(C(N2CC(CC(C)NC(=O)CC3CC4CC3C4)C2)=O)cc(C)c1C 62580,C1(CN(C(=O)CC2C=CCCC2)C)CCN(C(=O)CC2C=CCC2)CC1 62581,N1(C(c2c(OC)nccc2)=O)C2CCC1CC(C(=O)NC1CC(C)(C)C13CC3)C2 62582,c1(SC)ncc(C(=O)NCC2(C3CCOCC3)CC2)s1.C12(CC1)C(=O)NC2 62583,Cc1c(NC2(N)CCCC2)cccc1COc1ccc(C#N)nc1 62584,Cc1cnc(C(N2CC3C(CNC(c4ccccc4OCF)=O)C3C2)=O)c(C)c1 62585,O=C(C(O)C(F)F)NC(C1CCCC1)CNC(=O)CCc1nnc(C(F)F)o1 62586,Cc1[nH]nc2c(C(N3CC(NC(c4cn(C)c(O)n4)=O)CC3C)=O)cccc12 62587,c1(C(N(CC(C)NC(C2CC3CCC2C3)=O)C)=O)cnc2c(c1)N(C)CCO2 62588,C(=O)(C(C)C(=O)N1CCC=CC1C(=O)N(CC(O)CO)C)OC 62589,C1(NC(c2c(C)snc2)=O)CCCCC1CNC(=O)CCc1ccc(Cl)s1 62590,C(=O)(C(O)COC(C)=O)NCCC1(C(N(CC(COC)C)C)=O)CC1 62591,c1(C(N(C2CC(NC(C(COC)OC)=O)C2)C)=O)cnn2c1C(C)CCC2 62592,C(C)(C(=O)N1CC(CC(N2CCN(C3CC3)CC2)=O)C2(CC2)C1)(C(C)C)OC 62593,c1(C(N2CC(C)C(C)(CO)C2)=O)c(F)ccc(N)c1F 62594,Cc1ccc(CCC(=O)NC(CNC(=O)Cc2ccn(C)n2)CO)c(Br)c1 62595,O=C1CNC(=O)C(CC(N2CC(NC(C34CCC(C3)C4)=O)C3(CC3)C2)=O)N1 62596,N1(C(C(CC=CC)C)=O)CCN(C(c2n[nH]c(C)c2C)=O)CC1CC(=O)NC 62597,C1(NC(CC(=C)C)=O)COC2CN(C(c3sccc3OCC)=O)CC12 62598,C1(C(=O)NCCC2(OC)CN(C(C(C=C)(F)F)=O)C2)CCC2CCC(=O)N12 62599,c1(C(=O)NCC2OCCN(C(C=CC)=O)C2)cc(C(C)C)cc(Br)c1 62600,c1(C(=O)NCCN=c2[nH]nc(SCC)s2)cc2cccc(NC(N)=O)c2o1 62601,C(=O)(C(C)(C)C(C)(F)F)NCC1N(C(CNC(=O)OCC=C)=O)CCOC1 62602,c1(CNC(NC(CC)CC)=NCc2ccc(C)c(O)c2)nc2ccccc2o1 62603,c1(NC2CC(C(=O)Nc3cccc(C(C)(C)O)c3)C2)cc(C(F)(F)F)cc(Cl)c1 62604,CCC(CC(=O)NCc1ccoc1C(N1CCC(OC2CC2)CC1)=O)OC 62605,c1(C(=O)NCC2OCCN(CC(=O)N(C)C3CC3)C2)cc(F)ccc1O 62606,c1(OC(C)C)ccccc1.C1(C2CC3(CC3)NC(C)C(=O)N2)CCCCC1 62607,C1(NC(=O)C2=CCCS2)CCC2(CC1)CN(C(C1(n3cccn3)CCC1)=O)C2 62608,N1(C(C=C(COC)C)=O)CCCC1CN(C(=O)C(C)C1CCCC1)C1CCCC1 62609,c1(CC)ccc(F)cc1C(N1CC(NC(=O)CCOCC2CCC2)CC(F)C1)=O 62610,C(=O)(C(C)CC(C)(F)F)N1CCC(C(C)NC(c2ccc(C3CC3)[nH]2)=O)CC1 62611,C1(C(=O)NC(CN(CCCC)C)C)COCCC1NC(=O)C(C)(C)C#N 62612,c1(C(N2CCN(C(C(C=C)O)=O)C(CO)C2)=O)c(F)cc(F)cc1Br 62613,C1(CC(=O)NC2(CCNC(Cc3cc(C)sc3C)=O)CCC2)CC(O)C12CCC2 62614,CC1(NC(=O)C(F)C2CCOC2)CCCN(C(=O)C=CI)C1 62615,N1(C(C(CNC(C(CC=C)C)=O)N(C)C)=O)CCS(=N)(=O)CC1 62616,N1(C(C2=CCN(C(C3(C(=O)NC)CCC3)=O)C2)=O)CC2C3CCC(C3)C12 62617,C1(C(=O)NC2C3C(C)N(C(Cc4ccc(C)cn4)=O)C2C3)CC2(CCCO2)C1 62618,CC(O)CCCCCC(=O)NCc1ncccc1Cn1ccnc1 62619,N12CCCCC3(CCN(C3)c3nnc(n3CC3CC3)C1)C2.CC1CCN(C2CC2)C1 62620,CC(C)CCC(=O)NCCC(=O)NCC(C1CCC1)NC(c1ccc(=O)oc1)=O 62621,c1(C(=O)NCC2CC(C)N(C(=O)C=Cc3cncs3)C2)cccc2sccc12 62622,c1(C(=O)NCC2(CNC(c3c(OCC)nccc3)=O)CC2)ncc(N)nc1C 62623,C1(C(=O)NC(CCOC)(C)C)CN(C(=O)C(C)C(C)(C)C)C2(CCC2)C1 62624,C1(NC(=O)Cn2ccc(C(F)F)n2)CCCCN(C(C2OCCO2)=O)C1 62625,C(=O)(CCCC(=O)N(C)C)NCC(C)(CO)NC(C(CNC(C)=O)C)=O 62626,N1(C(CCSCCC)=O)CCC(NC(c2n[nH]c3c2CC2CC32)=O)C(F)(F)CC1 62627,C1(CN(C(=O)C(F)C2CCC2)C)CCCN(C(=O)COCC2CCCC2)C1 62628,C(CCC(C)(C)C(=O)NCC1CC1(C)C)NC(C(CC(=O)OC)C)=O 62629,Cc1cc(C(N2CCC(CNC(=O)Cc3sccc3C)C23CC3)=O)cc(N)c1 62630,c1(NC(=O)NC(C(=O)O)c2nccs2)cc2c(s1)CCCC2 62631,N1(C(C(C2CCCCC2)NC(C(CN(C)C)O)=O)=O)CC(O)C(O)C1 62632,c1(CC(=O)OC)ccc(NC(c2ccc(F)cn2)c2nnnn2C(C)C)cn1 62633,C1(OC)CN(C(=O)C(=O)NCC(F)(F)F)CC1C(=O)NCC1(OC)CCOC1 62634,Cc1ccc(C(F)(F)F)cc1C(=O)NC1CN(C(=O)C(O)CNC(N)=O)C1 62635,C1(OC)CCCC12CCCN(C(=O)CN(C)C(C1CCC3(CC3)C1)=O)C2 62636,C1(CN(C2CCN(C(=O)OC(C)(C)C)C2)C)CCC(N=[N+]=[N-])C1 62637,c1(C(N2C3CN(C(C=CS(CC)(=O)=O)=O)CC2CCC3)=O)cc2ccc(Cl)cc2s1 62638,c1(C(=O)NCC(C)CN(C(=O)CNC(N)=O)C)cc2ccccc2nn1 62639,C1(NC(C(C)OCC=C)=O)CC2CCC1C(NC(c1ccoc1CC)=O)C2 62640,c1(C(N2CC(CNC(CNS(NC)(=O)=O)=O)C(C)C2)=O)ccc(Cl)c(Cl)c1 62641,CCCCC#CC(C)(C)NC(=O)CC1COCCN1C(C1CC1(Cl)Cl)=O 62642,C1(C(N(CCNC(=O)C#CC2CCCCO2)CC)=O)CCCN1S(=N)(=O)N(C)C 62643,c1(C(=O)NC2CC3(CN(C(C(COC)OC)=O)C3)C2)nccc(C#N)c1F 62644,C(=O)(C(CC)C(=O)NC1(C(C)C)CCCN(C(C2C(N)CC2)=O)C1)OCC 62645,C(C(=O)N1CC(NC(C2(c3nccs3)CC2)=O)C(C(F)F)C1)(C(C)C)NC(C)=O 62646,C1(NC(C(COC)C2CCOCC2)=O)CN(C(c2ccc(=N)[nH]c2)=O)CC1(C)C 62647,Cc1ccc2c(c1)C=C(C(=O)N(C)CC1(CNC(=O)CCCC(N)=O)CC1)CO2 62648,c1(CNC(C2(COC)CC2)=O)cccc(NC(=O)CCN2CCCCCC2)c1F 62649,C1(C(=O)NCCNC2CCN(Cc3cccs3)CC2)CC2C=CC1O2 62650,C(=O)(C(O)C(C)(C)C)NC(C)CC1CN(C(=O)C(F)=C2CCC2)C1 62651,C1(C(=O)NCC(C2(O)CN(C(C=CCC)=O)C2)(C)C)CC2(CCCCC2)C1 62652,C1(CC)CN(C(C23CC4CC2C3C4)=O)CCC1NC(C1(C(F)F)CCOCC1)=O 62653,C(=O)(CCC(C)Cc1ccccc1)NCCC(C)N(C(C(OC)OC)=O)C 62654,Cc1cccc(OCC(=O)NC(C)C(C)(C)NC(c2cccnc2N)=O)c1F 62655,C=CC(CC)C(=O)N1CCC(C(=O)NC2(CO)CC2)C1C 62656,C1(N(C)C(C2CCCS2)=O)CN(C(c2c[nH]c(C#N)c2)=O)CC12CC2 62657,N1(C(C2(OC)CCCC2)=O)CC(CNC(c2scnc2Cl)=O)OC(C)(C)C1 62658,C1(CNC(COCCCCC)=O)CC2CC1CN2C(=O)C(c1cccc(C)c1)=O 62659,N1(C(Cc2c(C)noc2)=O)CC(C)N(C(=O)CN(C)C2CCC2)CC1C 62660,C1(c2nnnn2CCCOCC2CC2)(NC2(CCC)CC2)CC2CCOC12 62661,c1(CN2C(COC(C3CCOCC3)=O)CCC2)cc(=O)n2ncsc2n1 62662,c1(C(=O)NCC(C)N(C(CCC)=O)C)cc2cccc(C(F)(F)F)c2nc1O 62663,N1(C(C(C#C)(C)C)=O)CCC(C)(C)C(CNC(=O)COc2ccc(OC)cc2)C1 62664,C1(C(N2CCC(CC#C)C2)=O)CC2(CCN1C(=O)C(CC)OC)CC2 62665,c1(CC(=O)N(C(C)CCNC(=O)CO)C)cc(F)c(N)cc1F 62666,C1(NC(C(C)SC(C)C)=O)CCCCC12CCN(C(c1n[nH]cc1C1CC1)=O)CC2 62667,CC(C)(C)CC(O)C(=O)NC12CCCCC(NC(C3CSCCS3)=O)(C1)C2 62668,O=C(N=c1cc(Br)[nH][nH]1)C(=O)Nc1c(F)cccc1Br 62669,Cc1nc2cccc(N(CC3=CC(=O)N=N3)C(C)(C(C)C)c3nnnn3C)n2n1 62670,c1(C(N(CCNC(=O)CC2CCC(C)(C)C2)CC)=O)c(F)ccc(N)c1F 62671,C(=O)(C(CC)C(F)(F)F)N1CCC(n2cc(CNC(C(C=C)CC)=O)nn2)CC1 62672,CC(CC(F)F)C(=O)NC1(CNC(=O)CC2CN3CCN2CC3)CCCC1 62673,C1(C(=O)NCC(C)(C2CCC2)NC(c2ccc(SC)o2)=O)CCCCC1N(C)C 62674,C(CCC1CCC1)(C(=O)N(C1(CNC(C(=Cc2ccco2)C)=O)CC1)C)N(C)C 62675,Nc1cc(F)cc(Cl)c1C(=O)NC1COCC1NC(C1CC1C(F)F)=O 62676,C1(C(=O)NCCCn2cc(C(O)Cc3ccccc3)nn2)CCn2ncnc2C1 62677,O=C(C#CC1CCOC1)NC(C1CCCC1)CNC(c1ccc(CS(C)(=O)=O)o1)=O 62678,N1(C(C2(C)CC(C)OCC2)=O)CC2(CO)CC1(C(=O)NC(c1cncs1)C)C2 62679,N1(C(c2c(O)ccc(C)c2)=O)CCCN(C(=O)C(O)Cc2cnc[nH]2)C(C)C1 62680,N1(C(c2c(C)cco2)=O)CC2(CC(C(N3CCOC(CCCCCl)C3)=O)CO2)C1 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62854,c1(CC(N2CCN(C(=O)C(O)C(F)(F)F)C(CO)C2)=O)c(F)cccc1F 62855,C1(CC)CCCC1C(=O)NC1(CC=CC(=O)NCCCCc2cnc[nH]2)CCC1 62856,c1(C2(C(=O)NC(C(CO)NC(c3nnc(C)s3)=O)C)CC2)cc(F)ccc1F 62857,c1(C(=O)NCC2CC(NC(C(C3CCCC3)OCC)=O)C2)ccn2nncc2c1 62858,c1(C(=O)NC2(C)CN(C(=O)CN3CCNC3=O)C2)scc(Cl)c1Cl 62859,c1(C(=O)NCC2(C)CC3CCC2O3)n[nH]c2c1CC(C(=O)O)CC2 62860,C(=O)(C(C)C(C)(C)c1ccccc1)N(CC(CNC(CC(COC)C)=O)C)C 62861,C1(NC(C=CSC)=O)CC(OC)CN(C(c2nc(-c3cnn(C)c3)oc2C)=O)C1 62862,C1(NC(c2ccc(C)c(C)n2)=O)COC2(C1)CN(C(C1C3C=CSC13)=O)C2 62863,Cn1cc2cc(C(=O)NCCC(C)(C)CNC(c3c[nH]c(=N)o3)=O)ccc2n1 62864,C1(CNC(CC2(C=C)CC2)=O)C2CCC(C2)N1C(c1cccc(NC(=O)NC)c1)=O 62865,c1(CN2CCN(C(C3(CNC(C(COC)(C)O)=O)CC3)=O)CC2)cc(Cl)c(C)cn1 62866,C(=O)(CC1C(=O)Nc2ccc(F)cc21)NC(C)CNC(=O)Cc1ccc(O)nc1 62867,c1(C(=O)NCC(=C)CCNC(=O)C(CC)NC(=O)C(F)(F)F)cc2sccc2s1 62868,C1(C(=O)NC(C(=O)NC(C#C)COC)CC2CC2)CCCC(O)C1 62869,c1(Cn2cc(CC3N(C(Cn4c(C)ccn4)=O)CCC3)nn2)c(Cl)cccc1Cl 62870,C#CCCCCCC(=O)N(C1CCCN(C(=O)C(c2ccc(O)cc2)(C)C)C1)C 62871,c1(N(C(C(CC)C)C)CC)nc(N2CCC(N3CCOC3=O)C2)nc2c1ncn2C 62872,N1(C(CC(CC)OC)=O)CC(NC(c2cn(C)nc2SC)=O)CC12CCOCC2 62873,N1(C(c2c[nH]c(=N)o2)=O)CCC2(C1)CN(C(c1cscc1Br)=O)CCO2 62874,N#Cc1c[nH]c(C(N2CCC(CNC(c3cn(C4CC4)nn3)=O)CC2)=O)c1 62875,Cc1ccc(C=CC(=O)N(CCCNC(c2nn[nH]c2Cl)=O)CC2CCCC2)o1 62876,N1(C(C(C(C)C)OC)=O)CC(C(=O)NCc2nscc2O)C(C2CC2)C1 62877,N1(C(CCCOCC)=O)CC2CCCCC2(NC(C2CC(N(C)C)C(O)C2)=O)C1 62878,C#CC(CC(C)C)NC(=O)C(C)(C)NC(C1CCC1CCOC)=O 62879,C1(C(N2C(C#C)CC2)=O)C2CCC(C2)N1C(=O)Cn1c(C)ccc1C 62880,Cc1ccc(C=CC(N2CCC(C(O)CNC(c3cnc[nH]3)=O)CC2)=O)o1 62881,C(CCCCC(=O)NCC1=CCCC1)N(C(=O)C(F)CC1CCOC1)C 62882,CCCC(C)(C)CC(=O)N1CCC(C)(CNC(c2ccnn2COC)=O)C1 62883,CC(C)CCC(F)C(=O)NC1CCCN(C(=O)COc2ccc(O)cc2)CC1 62884,C(C)(C(=O)N(O)Cc1cn(Cc2nnc(C)o2)nn1)CCCCC 62885,c1(CNC(CCC2CC(NC(CCN(C)CC)=O)C2)=O)nc(C)sc1C 62886,N1(C(c2c(C)nc(Br)cc2)=O)CC2(CCN(Cc3cccc4[nH]ccc34)CC2)C1 62887,c1(OCC)cccc2c1C(C(=O)N1CC(NC(C3(F)CC4(CCC4)C3)=O)C1)CC2 62888,N1(C(c2cnc(CC)[nH]2)=O)CCCC(CCNC(=O)C(C)OCCC(C)C)C1 62889,C(=O)(CCCCO)N1CC(O)(CNC(C2N(C(C)=O)CSC2)=O)C1 62890,Cc1ccc(F)c(C(=O)NC2CC(C(=O)NC(c3ncc[nH]3)C)C23CCC3)c1 62891,c1(OC)cnc(C(N2CCCC2CCCNC(=O)CC(C)O)=O)c(F)c1 62892,CCC(C)(C)C(O)C(=O)N1CC(CNC(=O)Cn2nc(C)n(C)c2=O)C(C)(C)C1 62893,c1(OCC)cc(C(=O)NCC(C2CC2)N(C)C(c2ccsc2C)=O)ccc1C 62894,N1(C(C2(COC)CC=CCC2)=O)CCCC(N(C(=O)COC(F)F)C)CC1 62895,c1(NC(C2CC2NCc2cccc(Br)c2F)=O)ccc2[nH]nc(O)c2c1 62896,C12(CCNC(c3cc(C)ncc3)=O)CCC(C1)N(C(=O)CCc1n[nH]c(=N)s1)C2 62897,c1(C(=O)NC2C(NC(=O)CNS(C)(=O)=O)CCC2)nccc(Cl)c1Cl 62898,c1(OC)ccc(C(N2CC(C)CC2C(N2CC(NS(C)(=O)=O)C2)=O)=O)cn1 62899,C1(C(C)C)CN(C)CCN1C(C1CC(O)CN1C(=O)CCC1CCCC1)=O 62900,c1(OC)ccccc1CC(CNC(=O)CC(C)CN(C)C)C(=O)O 62901,c1(N2CCC(NC(C(C)OCCCc3ccccc3)=O)C2)ncccc1C#N 62902,N1(C(CCCC)=O)CC2ON=C(CNC(c3cn(-c4cncc(F)c4)nn3)=O)C2C1 62903,C1(NC(c2cc(C(N)=O)oc2)=O)CC2CC(C1)N(C(c1ncc(Cl)s1)=O)C2 62904,O=C(C(F)C(F)(F)F)NC1CC2(C1)CN(C(=O)CCc1ccc(Cl)cc1)C2 62905,N1(C(CC(=O)C(F)C(F)(F)F)=O)CC2CCCC2(Oc2ccc(C)cc2C)C1 62906,N1(C(C2C(C)(C(C)C)C2)=O)CC2C(CNC(C3CCC=CCC3)=O)C2C1 62907,CC1N(C(=O)C(C2CCNCC2)F)CCCC1(C)C 62908,c1(C(C)C)ncc(Br)c(=NC2CC2C(=O)NCCn2ccnn2)[nH]1 62909,N1(C(C(C)OC2CCCC2)=O)CCC2(CC2)CC1C(N1CCn2nncc2C1)=O 62910,Cc1cnc(C(=O)NC2(C)CCCN(C(C3CCOC(=O)CC3)=O)C2)c(Br)c1 62911,C1(OC)CC(NC(=O)Cc2cccc(Cl)c2)C12CCN(C(=O)CCSC(C)C)CC2 62912,C1(CC(C)=O)(NCCn2cc(NS(C)(=O)=O)nn2)CCCC1.N12CCCC1C2=O 62913,N#Cc1cccc(C(O)C(=O)NCc2ccnc(OC3CCCCC3)c2)c1 62914,O=C(C1=CC2C=CC(C1)C2)NCCCC(O)C(=O)NCCCC(F)F 62915,Cc1cncc(C)c1C(=O)NCC(O)CNC(=O)C(c1ccccc1)F 62916,C12(C(=O)NC3CC(C)N(C(c4ccc(CC5CC5)s4)=O)C3)CCC(NC)(CC1)C2 62917,C(CNC(c1cnc(Br)s1)=O)(CC(C)C)NC(CCNC(=O)NC)=O 62918,C1(C)(C(N2CCC(C(=O)NCC(=O)N(C)CC)CC2)=O)CCC2CC2C1 62919,C(CCC)(C(=O)NC(C)(CNC(c1c(C)n[nH]c1C)=O)C1CC1)=CCC 62920,c1(C(=O)NC(CN(C)C(C2(COC)CCCO2)=O)(C)C)nnc2ccccn12 62921,c1(SC)c(C(N2CC3(C2)CN(C(c2ncoc2C)=O)C3)=O)cccc1Br 62922,c1(CCNC(c2nnnn2CCCC2CC2)(COCCOC)C)ccncc1Br 62923,N1(C(C(C)(C)NC(=O)NCC)=O)CCN(CCNC(C2COCC(C)O2)=O)CC1 62924,N1(C(C(C(CC)C)O)=O)CC2CCC(NC(=O)C=Cc3cccs3)C2C1 62925,CCN1C(=O)C(NNC(=O)Cc2c(C)cccc2F)Cc2ccccc21 62926,N1(C(C(C2(O)CCC2)NC(c2nc(CC)oc2C)=O)=O)CCc2nnnn2CC1 62927,C1(C(N(C)Cc2ncc[nH]2)=O)CN(C(C2CC(F)(CF)C2)=O)CC1F 62928,C(=O)(C1COc2ccccc21)N1CCC2(CC(NC(=O)C=Cc3ncco3)C2)C1 62929,C(=O)(C(F)C(C)CC(C)(C)C)NCC1CCC(N(C(COCCCC)=O)C)CC1 62930,Cc1ccc(-n2cnc(CNC(N3CCN(c4cccc(Cl)c4)CC3)=O)c2)cc1 62931,C(CNC(=O)CC1CC(F)(F)C1)(CC(=O)N(c1nccs1)C(C)C)OC 62932,c1(C(N2CC(CCNC(C3(C)CC3(Cl)Cl)=O)C2)=O)cnc(N)c(N)c1 62933,CC1CS(=O)CCN1C(=O)C(Cc1cnc[nH]1)NC(=O)CC1CCC(C)(C)O1 62934,N1(C(CCC(C(C)C)C)=O)CCCC1(C)C(=O)NOCCC(C)O 62935,C1(C(=O)NC(CN(C(c2sc(CO)nc2C)=O)CC)C)CCC2(CCOCC2)O1 62936,C1(NC(CCS(C)=O)=O)CC2CC(NC(=O)CNS(N)(=O)=O)CC12 62937,Cc1nccc(C(=O)NC2CC(CNC(c3cc(C(C)C)on3)=O)C2)c1C 62938,Cc1nc2ccccc2cc1C(=O)NCC(CO)NC(=O)C(O)CC[S+](C)C 62939,CC1(C)CC(F)(F)CN1.c1(Cc2ccccc2)nc(-c2ccc(Cl)s2)no1 62940,C1(C(N2CC(OCC(=O)NC)C2)=O)CCCCN1C(=O)C(F)C1CCC1 62941,C(=O)(C1CCCn2cc(C(F)(F)F)nc21)OCCCNC(=O)C1CC1 62942,Cc1cc(C2(C(=O)Nc3sc(C)cc3Br)CC2)n(C)n1 62943,C1(OC)CC(C(N2CC3CCCC(C2)N3Cc2ccccc2)C=O)C12CCOCC2 62944,CC1CCC(C(N2CC(S(C)(=N)=O)C2)=O)CN1C(c1ccc(C(N)=O)o1)=O 62945,c1(C(=O)NCC2CC(NC(c3ccc([N+](=O)[O-])s3)=O)C2)ccc2nc(O)oc2c1 62946,C1(C(=O)NC2C=C(C)CCC2)C(C)OCCN1C(c1cccnc1CO)=O 62947,c1(C(N2CCC(C(CNC(CCCC#C)=O)(C)O)CC2)=O)ccc2c(c1)CC2 62948,c1(C(=O)NCCN(C)C(c2cn(C)[nH]c2=N)=O)cc(Cl)cc2c1CCC2 62949,N1(C(C2CCC(CNC(CSC)=O)C2)=O)CC2OC(=O)N(C)C2C1 62950,C1(NC(CCSc2n(C)nnn2)=O)CCN(C(=O)CC2C=CCC2)C12CC2 62951,C1(NC(C(CC)F)=O)CC(F)CN(C(c2ccccc2C2CCCC2)=O)C1 62952,CC(C)CC(O)C(=O)NC(C)C(=O)NCc1ncn(CCF)n1 62953,c1(CC)n[nH]c(CC)c1CC(=O)NC1CN(C(=O)COC(C)(C)C)CC1CC1CC1 62954,C1(C2(SC(C)(C)C)CC2)CN(c2cnc(C(N)=O)cn2)CCO1 62955,N1(C(CSc2nnc(C)s2)=O)CC(NC(=O)COCCCF)CCC1C 62956,C1(C(N(C(C)CNC(C2CC2C(F)(F)F)=O)C)=O)CCC2(CCC2)CC1 62957,c1(CCC2CC3CC(NC(CC(CC=C)(C)C)=O)CC23)ccc2c(c1)OCCO2 62958,N1(C(CC(C)(C)OC)=O)Cc2nccn2CC(NC(C2(F)CCCOC2)=O)C1 62959,O=C1CC(C(=O)N2CCOCC(CNC(c3cc[nH]n3)=O)C2)c2ccccc2N1 62960,c1(C(=O)NCC2(OCC)CN(C(=O)CCC3CCC(C)O3)C2)ccnc(C)n1 62961,N1(C(CC=C)=O)CC2(CCCC2NC(=O)CCc2cc(C)sc2C)C1 62962,CC1(C)C=C(C(=O)NCC(C(C)(C)C)c2ccccc2)C1 62963,Cn1c(CNc2ncc(F)cc2-c2ccccc2)nc2cc(Cl)ccc12 62964,c1(CCC(=O)NCC=CCNC(c2sc(N3CCCC3)nc2Cl)=O)ccc(Cl)nc1 62965,C(=O)(CCCCC(F)F)N(CC(C)(C)NC(C1C(C2CC2)C1(F)F)=O)C 62966,C1(NC(c2ccc(C)s2)=O)C=CCN(C(c2cnnn2C)=O)C1 62967,C(=O)(C1=CC2(CCOCC2)C1)NCC1(C)CCN(C(=O)CCn2cccn2)C1 62968,CC1(C)C(NC(=O)Cc2cc(F)ccc2F)CCN1c1ncns1 62969,c1(CC(=O)NCC2CCCN(S(=O)(=O)C(F)(F)F)C2)cncnc1O 62970,c1(C(N2CCC(C(C)NC(=O)CC3(O)CCC3)C2)=O)ncc(F)cc1N 62971,C1(NC(COCC(=C)C)=O)CC(CO)N(C(c2sccc2OC)=O)C1 62972,C1(C(N2CCC(NC(c3c(OC)cncn3)=O)C2)=O)CC2(CCOC2)C1 62973,c1(CC)nc(-n2cccc2)sc1C(=O)NCC(O)CNC(c1cnccc1Cl)=O 62974,N1(C(c2c(C(=O)OCC)c[nH]c2)=O)CCC(C)C(CN(C(=O)C(N)=O)CC)C1 62975,c1(OC)cc(C(=O)NCC(CO)NC(=O)CC2CC=CCC2)cc([N+](=O)[O-])c1Cl 62976,Cc1c(N)ccc(C(=O)NCC(C)CNC(=O)CN2OC(C)(C)CC2=O)c1C 62977,c1(C(C)C)nc(NCCC2CC2)cc(=NC(C)C2CCC2)[nH]1.c1(SC)ccccc1C 62978,N1(C(c2n(CC)ncn2)=O)CC(NC(=O)C(c2ccccc2OC)(C)C)CC1C 62979,c1(C(N2CCC(CCNC(c3c(CCC)occ3)=O)C2)=O)cccc(F)c1Br 62980,CCC(C)(C(=O)N1CCC(CNC2CCN(C(=O)C(C)(Cl)Cl)C2)CC1)OC 62981,C1(NC(C=CCOC)=O)CC2CC1N(C(=O)C(F)C(C)(C)O)C2 62982,N(C(=NCC(OC(F)F)C1CC1)NCc1ncnn1C(C)C)C(C)C 62983,C#CCCCC(C)C(=O)NC(COCC=C)C(=O)NC(c1ncccn1)C 62984,c1(OC)cc2cc(COc3ncnc(C)c3F)[nH]c2cc1C(=O)OC 62985,C(CC(F)F)(C(=O)NC1CCCN(C(C)C)C1)NC(c1cn(CC=C)nn1)=O 62986,N1(C(C(C)CO)=O)CCCCC(C2CN(C(C3CC34CCC4)=O)C2)C1 62987,Cn1ccc2ccc(C(=O)NCC3CCC(NC(C4CCCCO4)=O)CC3)cc12 62988,N1(C(C2C(C)(C)OCC2)=O)CC2(CCCC2)C1n1cc(COC2CS(=O)(=O)C2)nn1 62989,n1(CC)ncn(NC(=O)C(F)C(C)CNC(=O)C(C)(CO)OC)c1=O 62990,c1(C(=O)OC)ncccc1C(=O)Nc1ccc(CO)nc1.N12CCC(F)(C1)C2=O 62991,c1(C(N2C(CN(C(c3ccc(Cl)cc3F)C)C)CCC2)=O)c(O)ccc(Cl)c1O 62992,CCCC(C)(CC)C(=O)N1CC(NC(=O)C(CC(C)C)N(C)C)C(C)(C)C1 62993,C1(NC(C=C(C)C)=O)CC2CCC1N2C(c1c(C)nn(C)c1-n1cc(C)cn1)=O 62994,C(CC(C(=O)N1CCCCC1CNC(c1cc(C(F)F)cs1)=O)NC=O)SC 62995,N1(C(Cc2cc(OC)ncc2Cl)=O)CC2CN(C(c3cnccc3N)=O)CC2C1 62996,N1(C(c2c(C)scn2)=O)CCC2(C1)CN(C(c1nc(C(C)C)no1)C)CC(C)O2 62997,C#Cc1ccc(C(=O)N(C(C)C(N2CCCC(F)CC2)=O)CCC)cc1C 62998,CN(C)NC(=O)CCC(=O)N1CCC2(C(N3CCCC(CCO)C3)=O)CC2C1 62999,CN1CCC(C(=O)NCC2CC2NC(c2cc(C#N)c[nH]2)=O)CC1 63000,N1(C(C(C=C)O)=O)CC2CC(NC(=O)Cn3c(C)cc(O)cc3=O)CC2C1 63001,N1(C(c2c(C)scn2)=O)CCC(CCNC(C2(C(F)(F)F)CC(C)(C)C2)=O)CC1 63002,Cc1cccc2cc(C(=O)NC(C)CCN(C)C(C3(O)CCOCC3)=O)nnc12 63003,CCCCCC(CC)C(=O)N1CC(NC(=O)CC(F)(F)F)C(C)(C)C1 63004,C1(CC=C)(NC(=O)C2=NOCC2)CCCN(C(=O)COCC(C)=O)C1 63005,C1(CNC(c2c(CC)nco2)=O)CN(C(C2(C#N)CC23CCC3)=O)CCC1(F)F 63006,C1(C(N2CC(CNC(=O)Cc3cn[nH]c3)C(F)(F)C2)=O)C2(CCC2)C12CCC2 63007,c1(C(N2CC(CC(=O)NC(C=C)C3CCC3)C(C)CC2)=O)cc2ncccc2[nH]1 63008,CN(CCc1nc2ccccc2s1)N1CCCC(C(=O)OCC2CCCO2)C1 63009,CN1CC(C)(C)CC1C(N1CCCC(c2cn(CCCF)nn2)C1)=O 63010,c1(CNC(C2CC3CCC2N3C(c2ccnc(O)c2F)=O)=O)cc(F)ccc1O 63011,CCCCCS(=O)(=O)CC(=O)NCC(C(C)(C)C)NC(=O)CCN(CCC(C)(C)C)C 63012,c1(C(=O)NCC2N(C(C(CC=C)CC)=O)CCCC2)ccc2c(c1)nnn2C 63013,N1(C(COCCSC)=O)CCC(F)CC1C(=O)NCC1CC(F)(F)CO1 63014,N1(C(=O)CCCn2cncn2)CC2CC(C1)N(C(=O)Cc1n[nH]cc1C1CC1)C2 63015,c1(C(=O)NC(C(C)NC(c2snc(C)c2N)=O)C)nc2c(s1)COCC2 63016,Cn1c(C(N2CC(NC(c3ccc(C(C)(F)F)cn3)=O)C2)=O)cnc1[N+](=O)[O-] 63017,N1(C(C(F)=CC)=O)C2CCCC1CC(n1cc(-c3cc(N)ccc3C(=O)O)nn1)C2 63018,C1(=O)C(=O)NOCC(=O)NCCN1.c1(C(N2CCCCC2)C)ccc(F)cc1 63019,C(=O)(CCCCCCn1cc(-c2ccc(Cl)nc2)nn1)NC(CC)CC(C)O 63020,CC(C)CC(CC(=O)NCCN(C(=O)CC(C)Sc1ccccc1)C)CC(N)=O 63021,c1(C(N(CCCNC(C23CCC2C3)=O)C)=O)cc2c(s1)CCCCC2 63022,C(C)(C(=O)N(C)OC)NC(c1cccc(OC2CC2)c1)c1n(CC)nnn1 63023,N1(C(c2ccc(NC(C)=O)s2)=O)CCC2CN(C(C3OCCC3C)=O)CC2C1 63024,O=C(CCS(=O)(=O)c1ccccc1)NC1CCC2(CNC2)c2ccccc21 63025,N1(c2sc(C(C)=O)c(Cl)n2)CCCC2(CC(NC(c3snnc3C)=O)C2)C1 63026,c1(C(=O)NC2C=CCN(C(=O)COCC3CCCCO3)C2)n[nH]c2cccnc12 63027,N1(C(C2CCC3N(C(c4c(C)ccnn4)=O)C2CC3)=O)CCc2ccncc2C1 63028,c1(C(=O)OCC)nn(C)c(C)c1CNC(C1CCCSC1)=O 63029,C1(C(=O)NCC(=O)NC(C=C)C2CCC2)CC(C)CC(=O)N1 63030,N1(C(C(CCSC)O)=O)CC(CNC(c2cn(C)c(=O)n2C)=O)OC2(CCC2)C1 63031,C1(NC(CC(C)CNC(c2cccc[n+]2[O-])=O)=O)COCCC1(F)F 63032,C1(NC(C2CC(OC)C2)=O)(CO)CCN(C(c2cn(C(C)C)nc2Br)=O)C1 63033,Cc1[nH]nc(C(=O)NC2CCCCC2CC(=O)NOCCCN(C)C)c1C 63034,Cc1ccc(F)cc1C(N1CC(CNC(=O)Cc2cn(C)nc2C)CCC1C)=O 63035,N1(C(=O)CC2CCN(Cc3ccc(O)c(Cl)c3)C2)CCN2CCOCC2C1 63036,Cn1ncc([N+](=O)[O-])c1C(=O)NC1C2CN(C(=O)C(=O)NCC(F)(F)F)CC12 63037,N1(C(C2OCC(=O)C2)=O)CC2CCCC(NC(=O)C(=O)C(F)(F)F)C2C1 63038,N1(C(c2cncc(OC)c2)=O)CCCC2(NC(=O)COc3ccon3)CC2C1 63039,C1(NC(c2csc(Br)n2)=O)CCCC(O)C1 63040,C1(CCCNC(C(C)=C(C)C)=O)CCCN1C(c1cnc(N(C)C)o1)=O 63041,C12(C(N3CCC(CCNC(=O)CCC=CBr)C3)=O)CCCC1CCC2 63042,CCCCCCCc1cn(CC(C)NC(c2cc(C)co2)=O)nn1 63043,N1(C(=O)C2=CCSC2)CC(C2CCCN(C(c3cccc4c3OCCO4)=O)C2)C1 63044,C1(CNC(C(C)OC)=O)CN(C(c2cc3ccoc3cc2F)=O)CC(C)(C)O1 63045,c1(CC(=O)NC23CC(NC(CN(CCC)C)=O)(C2)C3)c(F)cccc1Br 63046,Cc1ccc2c(c1)CC(C(=O)NCC(O)CNC(C1(C(F)F)CCC1)=O)O2 63047,C1(NC(CCOCC#C)=O)CC2CC(NC(=O)C=Cc3cccc(C)c3)CC2C1 63048,c1(OC)ccc(O)c(C(N2CCOC(CNC(=O)C(O)CC(N)=O)C2)=O)c1 63049,C(CN=c1cc(C)nc(-c2cc(F)ccc2OC)[nH]1)NC(CN(CCC)C)=O 63050,c1(C(=O)NCC2C(CNC(C3CC(n4cnnc4)C3)=O)C2(F)F)c[nH]c(=O)cn1 63051,C1(C(N(C2CCCCCC2)C)=O)(NC(c2ccncc2N)=O)CCOCC1 63052,c1(CN2C(C(=O)NCCCCCCN(C)C)CC2)cc(Cl)cc(Cl)c1 63053,N(C1CCOc2ccc(SC)cc21)C(c1occ(C(=O)OC)n1)C 63054,N1(C(C(C)NC(CCC(=O)NC(CC)(C)C)=O)=O)CCC(CO)C(C)(C)C1 63055,C1(C)(NC(=O)Cn2cnc(=N)[nH]2)CC2(CCC2)C1.C12CC1C(=O)NC2C 63056,C(C(CC)(CC)C(=O)NC1CC2(CCC2)C1OC)NC(CSCC=C)=O 63057,c1(C(=O)NC2C(C)CN(C(c3scnc3C3CC3)=O)CC2)ccc(S(N)(=O)=O)[nH]1 63058,Cc1oc(Cl)nc1C(=O)NC1(C(=O)N(C)Cc2cnn(C)c2)CCSC1 63059,c1(C(=O)NC(C)CNC(C2CCOC2C)=O)ccc2[nH]c(=N)oc2c1 63060,N1(C(Cn2ccc(C)n2)=O)CCC(C(=O)NCCCC2(C)CC2)C1C(C)C 63061,N1(C(COC2(C)CCOCC2)=O)CC2COCC2(NC(C2CCCN2C2CC2)=O)C1 63062,N1(C(C(Cc2c(C)nc[nH]2)O)=O)CCCC2CN(C(=O)CCNS(C)(=O)=O)CC12 63063,N1(C(C2(CC)CCCC2O)=O)CCOC(C)(CNC(C2CN(CC)CCO2)=O)C1 63064,c1(C(=O)NC2CCC(NC(=O)CSCC(F)(F)F)C2)ccccc1[N+](=O)[O-] 63065,c1(C(=O)NCCC(CC)(CC)NC(C(CC)O)=O)cc2nccnc2[nH]1 63066,c1(CCNC2(NC(=O)CC3CCCC3)CC2)ccc2c(c1)OCO2 63067,C1(OC)(CNC(c2snc(Cl)c2Cl)=O)CCN(C(C2CCCCC2)=O)C1 63068,c1(CC(N2CC(CNC(C3C(=C)C3)=O)C(C)(C)C2)=O)nc2ncccn2n1 63069,c1(C(N2CCC(N(C)C(C34CC(CC(F)F)(C3)C4)=O)C2)=O)cccc2[nH]ccc12 63070,C(=O)(C1=C(Cl)CCOC1)NC1CN(C(C(C)OCCOCC)=O)C(C)C1 63071,C(=O)(C(C)(O)C(F)(F)F)Nc1cccc(NC(c2ccc(OC)c(Cl)n2)=O)c1 63072,c1(C(N(C(CNC(C2CCC(C)(C)O2)=O)C2CC2)C)=O)cc2ccc(Cl)cc2o1 63073,c1(NC(=O)NCCC2C(C)CCC2)ccc(N2CCCC2)cc1Cl 63074,C(C(CC(C)C)C(=O)NCC1(F)CCN(C(c2nccc3occc23)=O)C1)OC 63075,N1(C(c2n(C(CC)(C)C)ncc2)=O)CC2CC1C2NC(c1ncccc1OC)=O 63076,C12CC(CN1S(C)(=O)=O)N2.N1(C(C)=O)CCCC1C(=O)N(C(C)(C)CN(C)C)C 63077,c1(OC)cnc(F)c(C(=O)NCC(C)N(C(=O)CSc2nc[nH]n2)C)c1 63078,N1(C(CCC2CCC(=O)NC2)=O)C2CCC(C2)C1CNC(c1ccc(O)nc1)=O 63079,Cc1cnc(NCc2cc(C)no2)c(S(=O)(=O)NCC2(CO)CC(C)C2)c1 63080,CCCC(C)(O)C(=O)N1CC(CCNC(=O)C(c2ccccc2F)C)(OC)C1 63081,C#Cc1cc(C(=O)NC2CCC(NC(=O)C(C)O)CC2)cc(N)c1 63082,c1(C(=O)NC2CN(C(c3c(C(C)C)ccs3)=O)CC2O)c(Cl)nc2ccccn12 63083,C1(NCc2c(OC)c[nH]n2)CCC(CNC(=O)C(c2cncn2C)N(C)C)CC1 63084,c1(CNC2C(C(N3CCC(C#N)C3)=O)C2)c[nH]c2nc(Cl)ccc12 63085,C(C(C(=O)NC1CCC1NC(c1cccc2nsnc12)=O)C(C)(C)C)OCC=C 63086,Cc1cccc2[nH]c(=NCCN(C(=O)C(C)CSC(F)(F)F)C3CC3)oc12 63087,N1(C(COCC)=O)CCC(NC(=O)C(C)(C)CCCOC)C(CO)CC1.CO 63088,Cc1ccc(C(N2CC=CC2C(=O)NCC2CN(C3CC3)C2)=O)cc1 63089,c1(CNCC2N(C(CC=C)=O)CCOC2)cc(F)c(Cl)cc1Cl 63090,N1(C(CSCCOC)=O)CCCC(CCC(=O)NCC(=O)NO)C1 63091,C1(C(=O)NCc2nc(C3CC3)no2)CCCCCCN1C(=O)CCC1CC1 63092,C(=O)(C(F)CCC(C)C)N1CC(N(C(c2cn(CCC(C)C)nn2)=O)C)C(O)C1 63093,c1(C(=O)OC)ccc(N2CC(CCN(C(=O)NC(C)(C)C)C(C)C)C(O)C2)nc1 63094,N1(C(c2c(C)n[nH]c2)=O)CCCC(CC(=O)NCc2cc(Cl)cs2)C1 63095,C(=O)(C1CCOc2ccccc21)NC(C)CN(C)C(c1c(N)cnn1C)=O 63096,N1(C(C(CC)N(C)C)=O)CCOCC(NC(=O)CC2(OCC)CC2)C1 63097,CCC(C)C(O)C(C)C(=O)NCc1cc(C)c(C(=O)N(C2CCOC2=O)C)o1 63098,N1(C(C(CC(F)F)N(C)C(c2ccn(C3CC3)n2)=O)=O)CCCC2CNC(=O)C12 63099,C1(O)(CCNC(C2(CC#C)CCCC2)=O)CCN(C(c2ccnn2C(C)C)=O)C1 63100,C1(C#N)(C(=O)NCCC(C)NC(C(C)N2CCCC2)=O)CCSCC1 63101,N1(C(CCC2(C)N(C(c3c(C)c[nH]n3)=O)CCC2)=O)CCOCC2(CC2)C1 63102,Cc1cn2nc(C(=O)NC(C)(C)CN(C(=O)CC3CSC3)C)cc(C)c2n1 63103,C1(C(C(=O)NC(CCOC)CNC(c2cnccn2)=O)C)CCN(CC(F)F)CC1 63104,Cn1cnc(NC2CCC(NC(=O)CCc3ccncc3)CC2)cc1=O 63105,C1(CCc2n[nH]c(COC)n2)CCN(NC(C(CCC)NC(N)=O)=O)CC1C 63106,N1(C(C)=O)CCCCC1C(N1CCC(CNC(=O)CCCc2csc(C)n2)C1)=O 63107,C=CC1CN(C(=O)CC2CNC(=O)C2)CC1NC(=O)CSc1cn[nH]c1 63108,CC(C)(CC=CC(=O)N1CCC1)N(N1CCCC1=O)C(=O)CCN1CCOC1=O 63109,C(=O)(C#CC1(CC)COC1)N(CCNC(c1cc(CO)oc1C)=O)CC 63110,C(CN=C(NCC1CC1)N(C)Cc1ccnc(F)c1)NC(C1CCCC1)=O 63111,C1(N)NC(=O)CC1C(F)(F)F.c1(C(=O)NCCN(CCC(=O)COC)CC)cnn[nH]1 63112,c1(C(c2nnnn2C2CC2)NCc2cn(C)nc2Cl)cc(S(C)(=O)=O)cs1 63113,CC1OC2(C(=O)NCC3CCN(C(c4cncc(Cl)n4)=O)CC3)CCC1C2 63114,CCC1=C(C(=O)N2CC3CC2CCC3NC(c2ccnc(F)c2)=O)CCCO1 63115,C1(C2CCC2)(C(=O)NCC(C)N(C(=O)CC(C)(C)C)CC)CC1(F)F 63116,C1(C(=O)NCCNC(CC)=O)C2Cc3c(Br)cccc3C12 63117,c1(C(=O)NCC(CC)N(CC(=O)Nc2cccs2)C)ccccc1N=NN(C)C 63118,n1(CCC(=O)NCCCN(C)C(C2CC2F)=O)c(-c2cccs2)nnc1S 63119,C1(CNC(c2c[nH]c(=O)cn2)=O)CN(C(C2CCCO2)=O)CCC12CCC2 63120,C12(C(=O)NC3CN(C(Cn4c(C)ccn4)=O)CC3C(F)F)CC1COC2(C)C 63121,c1(C(N2CC3CC2CN3C(c2cc(F)ccc2F)=O)=O)cccc(F)c1O 63122,c1(C(=O)NC2CC(NC(c3ccccc3-n3ccnc3)=O)C2)cc(F)ccc1Cl 63123,c1(C(=O)NCC2(C)CN(C3CCN(C(=O)CC#N)CC3)C2=O)cc(F)ccc1N 63124,Cc1cccc(C(N2CC3(NC(c4sncc4C)=O)CCC2C3)=O)c1Cl 63125,c1(CC(=O)NC2C(CNC(COCCC#C)=O)CC2)coc2c(C)c(C)ccc12 63126,c1(C(=O)NCC(C)NC(C2N(CCC)C(=O)CC2)=O)cccc2cccc(O)c12 63127,N1(C(CN(C(COC)=O)C)=O)CC(NC(=O)C(C)(C)C2CCC2)C(O)C1 63128,N1(C(C(C)(O)Cc2ccccc2)=O)CC(F)(F)CC1C(N1CCC(CO)C(O)C1)=O 63129,C(=O)(C1CCCc2ncnn21)NC1CC(CCNC(c2cc(CC)nn2C)=O)C1 63130,c1(C(=O)NCCCN(C)C(c2cnc(S)[nH]2)=O)nc(C(C2CC2)C2CC2)ncc1Br 63131,C(=O)(C1=CCC(F)(F)CC1)N1CCC(CCNC(CCC(C)OC)=O)C(F)(F)C1 63132,N1(C(c2c(C)[nH]cc2)=O)C(CC(N2CCC(C)(CO)C2)=O)C2CCCC12 63133,C1(CC)CCN(C(=O)CCc2cn(C)cn2)C1C(=O)NCCCCOC 63134,C(=O)(CCC(C)CN(C)C)NC1CN(C(COCc2onc(C)n2)=O)C(C)C1 63135,C1(C(C)C(=O)NCC(c2ccccc2)F)CCN(C(c2ccoc2Cl)=O)CC1 63136,c1(Sc2cccc(NC3C(CC)CCO3)c2)cccc(C)c1OC 63137,C=CC(CC)C(=O)N1CCC(=CC)CC1.C(=O)(CC)NCCSCC 63138,c1(CC)ccc(C(N2CCCC2CCNC(C2C(Cl)(Cl)C23CC3)=O)=O)cc1Cl 63139,CC1=C(C)CC(C(=O)NCC(C(=O)N(CC(C)C#N)C2CC2)C(C)C)CC1 63140,N1(C(CC2CCCN(C)C2)=O)CCN(C)CC1CNC(=O)C(=O)NC1CC1 63141,Cc1cc(CNC(C2COC(CNC(c3sccc3C)=O)C2)=O)cc(C)c1 63142,c1(-c2ccc(C(=O)NCC3N(C(C(COCC)C)=O)CCC3)o2)ccccc1F 63143,Cc1cccc(C2(C(=O)NCCCC(C)NC(=O)C(O)C(F)F)CC2)c1 63144,N1(C(CCCC(C)NC(C(C)(C2(C)CC2)OC)=O)=O)CC2COC(=O)C2C1 63145,C1(C(=O)NCC(=O)N(CC)CC)CC(F)(F)CN1C(=O)CC1COCCOC1 63146,C1(NC(CC2CC(=C)C2)=O)CCC(C)N(C(c2ccc(N)c(OCCO)c2)=O)C1 63147,c1(-c2cn(CC(N3CC(C)C3NS(C)(=O)=O)=O)nn2)ccc2ccn(C)c2c1 63148,c1(CC)ccc(C)c(C(N2CCC(N(C(=O)C(c3cccnc3)O)C)C2)=O)c1 63149,CC(CCCC(=O)NC(C)(C)CC1CCOC1)NC(c1cc(Cl)no1)=O 63150,c1(C(=O)N)ccc[n+]([O-])c1.C12CN(C1)C(=O)CC1(CCC1)C2C1CC1.CCCCC.CCC 63151,C1(N(C(c2cc(COC)on2)=O)C)CC2CC1N(C(=O)CC1CSCCS1)C2 63152,Cc1nc(C(=O)NC2CN(C(C3CCC3c3nc[nH]n3)=O)C2)cn(C)c1=O 63153,c1(C(=O)OCC)cc(C(C)C)c(N(C(=O)CCCc2ccccc2)CC)[nH]1 63154,c1(CC(=O)NCC(CNC(=O)CC2CC(CF)C2)OC)ccc2c(c1)OCCO2 63155,c1(CNC(c2ccc(CC)o2)=O)c(C)nn2c1CN(C(C1(C)CC1F)=O)CC2 63156,N1(C(C2C(Nc3c4cccc(C)c4ncn3)C2)=O)CCc2ncc(Br)cc2C1 63157,c1(C(=O)NC2(CCNC(CCCOCC)=O)CCC2)ccc(N)c(Cl)n1 63158,C=CCC(F)(F)C(=O)NC1CCC(NC(c2ncccc2CSC)=O)C1 63159,O=S(=O)(CCO)CCSC1CCCCCCC1 63160,c1(C(N(C)CC2N(C(CSCC#C)=O)CC(F)C2)=O)cc2n(n1)CCC2 63161,c1(C(=O)NC2CN(C(c3c(C)ocn3)=O)CC3C2C3)ccnc2ncccc12 63162,c1(OCC(N2C(CNC(=O)CCF)CCC(C)C2)=O)cccc(S(C)(=O)=O)c1 63163,c1(C(=O)NC(C(C)NC(c2c(OC)ccc(F)c2)=O)C)cccn2ccnc12 63164,C1(N(C(C(C)NS(CC)(=O)=O)=O)C)CCCCC1N(C)C(c1cccc(C)c1)=O 63165,N1(CCN(C(C2CC(C)OC2)=O)C)CCN(CC(O)C(C)c2ccccc2)CC1 63166,C12(C(=O)NCC3(C)CCN(C(CC(C(=C)C)O)=O)CC3)C3CC(CC13)C2(F)F 63167,C(=O)(C(C)CC)NC(C(=O)NCC(CSCC)O)c1ccoc1 63168,c1(N2C(CNC(c3cc(CCC)[nH]n3)=O)CC(F)(F)C2)ccc(S(C)(=O)=O)cn1 63169,C1(C(=O)NCc2cc(C(=O)Nc3ccc(Cl)cc3)n[nH]2)CC2(CCC2O)C1 63170,CN=c1cc(C(=O)N(C(C)C(N2CCCC(C)(N(C)C)C2)=O)C)cc[nH]1 63171,c1(CC(=O)N(CC(C)NC(=O)CC2CCCS2)C)cccc2c1CCC2 63172,CC(CC(=O)N1CCC(NC(c2cc3n(n2)CCOC3)=O)C1)CC(F)(F)F 63173,c1(NCCCCSC)ncccc1S(=O)(=O)NC1COC2(CCC2)C1 63174,C(C(C)(C)C(=O)N1CCC(C(C)NC(=O)CC=Cc2ccccc2)C1)OC 63175,c1(C(N2CC(N(C(C(CC)C#N)=O)C)C3(C2)CC3)=O)c(F)cc(OC)c(F)c1F 63176,C1(C(=O)NC2CN(C(c3c(CCC)nsc3N)=O)C2)CC2(CCCC2)CO1 63177,C1(OC)Cc2ccc(NCC(=O)NCC(c3ccccn3)(F)F)cc2C1 63178,C12(C(=O)NCCOCCSC)CC(NC(=O)CCc3cccnc3)(C1)C2 63179,N#Cc1ccnc(C(=O)NC(C2CCOC2)CNC(=O)CC2CSC2)c1F 63180,C(=O)(CCCCC(F)(F)F)NCC(n1cc(CNC(C)=O)nn1)(C)C 63181,C=CC(C)(O)C(=O)N1CCOCC1CC(=O)NCCOc1ccccc1F 63182,C12(NC(Cc3n(C)ncc3)=O)CCN(C(c3cc4sccc4s3)=O)CC1C2 63183,N1(C(Cn2cnc(=N)[nH]2)=O)CCN(C(=O)Cn2cc(C3CC3)nn2)CC1CCO 63184,Cc1cc(C)c2[nH]c(C(=O)NC3CC3NC(=O)CNS(=O)(=O)C3CC3)cc2c1 63185,c1(OCC)cc(NC(C)CCNC(=O)C(O)c2ccsc2)ccc1[N+](=O)[O-] 63186,Cc1cc(O)ncc1C(=O)NC1CC(O)CN(C(c2ccnc(C(C)C)n2)=O)C1 63187,N1(C(C2OCC(C)C2)=O)CCN(C)C(CNC(c2ccn(C(C)(C)C)n2)=O)C1 63188,Cc1csc(C(=O)NCCNC(c2c(C3CC3)noc2C(C)C)=O)c1C 63189,C1(C(C)N(C23CC(N(C)C)(C2)C3)C(=O)CCOC(C2CCN(C)CC2)=O)C2CCCC12 63190,C1(C(C)C)CN1C(C1CCN1C(C1(CCNC(N)=O)CC1)=O)=O 63191,c12cc(C(=O)OC)c(OC)cc1OC2=O.N1(CCSCC=C)CC(F)(F)C1 63192,Cc1cc(C(=O)N(C(C)CCNC(=O)C(F)(F)c2cnn(C)c2)C)c(C)cn1 63193,O=C(CNC(C1(F)CCOC1)=O)NN1CCCC1C(=O)NC12CCC(CO1)C2 63194,C1(C)(NC(CCC)=O)CCC(NC(c2ccc(C(F)(F)F)c(Cl)c2)=O)CC1 63195,CC(C)(F)CCC(=O)N1CCCCC1CNC(c1c(N)cccc1F)=O 63196,NS(=O)(=O)c1ccc(C(N2CC(NC(=O)Cc3cncnc3O)C(O)C2)=O)nc1 63197,N1(C(Cc2cc(C)sc2)=O)CC(CNC(=O)CCOC2CCC2)C2(CC2)C1 63198,N1(C(C(C)SCCCC)=O)CCC(NC(c2cc(C(C)=O)cs2)=O)C(C)C1 63199,C1(NC(CC=C)=O)CCCN(C(=O)C(CO)NC(=O)OC(C)(C)C)CC1 63200,c1(C2C(C(c3nnnn3CCCF)(C)NCCCCOC)C2)ccccc1 63201,C(=O)(C(C(C)C)C(C)C)N1CCOCC(C(=O)NCC(COCC)O)C1 63202,C(=O)(C1=NOC(C)C1C)NC(c1occ(C(=O)NC2CC(=C)C2)n1)C 63203,CCC(CC(C)C)C(=O)N(C(C)C(=O)N(C)CCOC)C1CC1.CC(C)O 63204,c1(C(=O)NCC2N(C(C(CCC)(C)C)=O)CCCC2)cc2n(n1)CC(C)NC2=O 63205,c1(C(N2CC(N(C(C3C(C(C)C)C3)=O)C)C2)=O)cc(N)cc2ccccc12 63206,c1(C(=O)OC)ccc(C)nc1N1CCCCC(NC(=O)CCCCSC)C1 63207,CC(CC(=O)NCCN(C(=O)Cc1ccccc1)C1CC1)n1ccnc1 63208,C12(N(CCCN(C)C)C(C3CCOC3)=O)CC(n3cc(C4CC4)nn3)C1C2 63209,Cc1csc(=O)n1CC(=O)NC1(CO)CN(C(C2CC3CC2C3)=O)C1 63210,Cc1c(C2(C(=O)NCCC3(NC(c4ncccc4O)=O)CC3)CC2)cccc1F 63211,C1(C(=O)NC2CC(CCNC(c3c(CC)ocn3)=O)C2)CCCC(C)(C)O1 63212,CCC(F)(F)CC(=O)N1CCOCCC1C(=O)NC(C)CCF 63213,C1(C)(OC)CC2CC1CC2NC(=NCCN(S(=O)(=O)CCC(=O)OC)C)NC(C)C 63214,c1(OC)cc2nc(NC(=O)CC(C)SC)[nH]c(=N)c2cc1Br 63215,Cc1ccc(C(N2CCCC(C)(NC(=O)CC(C)c3ccncc3)C2)=O)c(N)c1 63216,C1(NC(C2(CC)CCCN2C(=O)C(F)C2CCCC2)=O)CCC2CC1CO2 63217,Cc1cc(Nc2nccc(C(C)C)n2)nn1C(c1ccccc1)C(=O)OC.C(=O)N(C)C 63218,C1(C)(n2cc(CN(C(=O)CCC(=O)OC(C)(C)C)C(C)C)nn2)CCCCC1C 63219,c1(C(N(C2CCNC2)CC)=O)c(F)ccc2c1OCO2 63220,C(CC)(CC(=O)NC(C)CC1CCCO1)N(C(C(CC)=CC)=O)C 63221,C1(NC(c2c(CC)cno2)=O)CC2CC1CN(C(=O)Cc1ccsc1C)C2 63222,CC(CC(=O)NC1CCC1NC(=O)CC(=O)N(C)C)P(C)(C)=O 63223,Cc1ccc(NC(C2CCCCN2c2ncnc3occc23)=O)c(F)c1F 63224,C1(CNC(C(CC)N(C)C)=O)CC(C)CN(C(=O)CCNc2cccnc2)C1 63225,c1(C(N2C(C(=O)NCCC#C)CC3(CC3)C2)=O)cccc2c1CCC2 63226,C1(CC(=O)OC(C(C)(C)C)=O)COC2(CCC2)CN1N1C2CCCC1CC2 63227,CCCCCC(O)C(C)C(=O)N1CCCC(CNC(C2(COC)CC2)=O)CC1 63228,C(C1CCC(C)CC1)=C(C)C(=O)Nc1ccc(C(N2CCOCC2)=O)cc1 63229,CC1(CNC(=O)N(CCCn2ccc(C(F)(F)F)c2)Cc2ccccc2)CCCCO1 63230,C1(CC(=O)NCC(C)CNC(=O)C(F)(F)c2csc(=N)[nH]2)CC(=O)NC1=O 63231,C1(C(=O)NCC2(F)CC(NC(CCNC(C)=O)=O)C2)CCCC(O)C1 63232,CC1CN(C(=O)Cc2cnn(C)c2)CCC1C(=O)NC(C)CC1CCCC1 63233,C1(C)(C(N(CCN(C(C(CCCC)O)=O)C)C(C)C)=O)CCCCCCC1 63234,c1(C(=O)OC)ccc2ncnn2c1.c1(N2C(C(=O)O)(CO)CCC2)c(C)ccn1C 63235,C(=O)(C(F)C(F)(F)F)NC1C(CNC(CC2CC(OC(c3ccccc3)C)C2)=O)C1 63236,CC1CCCC1(C(=O)NCc1nncn1C)NC(=O)CSC1CC1 63237,C12(CNC(c3n(CC)ncn3)=O)CN(C(=O)Cn3ccccc3=O)CC1CCO2 63238,C1(NC(CCc2cn(C)nn2)=O)CN(C(C2(O)CCOC2)=O)CC(C)(C)C1 63239,N1(C(CNC(CN(C)C)=O)=O)CCN(C(=O)CCc2cncn2C)CC1C1CC1 63240,C1(CNC(C2C(C)CCCC2)=O)CC(C)CN(C(c2ccnn2CC2CC2)=O)C1 63241,N1(C(C=CCCC=CC)=O)CCC(C)(C)C(CNC(C2CCCC3(CC3)C2)=O)C1 63242,N1(C(C(c2cnn(C)c2)N(C(CCOC)C)C)=O)CC(NC(=O)OC)CC1C 63243,CN1CCc2cc(C(=O)NCC(C3CCC3)NC(=O)C(O)CC(N)=O)ccc2C1 63244,C#CCCC(C(=O)NCCCC(=C)Cl)NC(=O)C(C)O 63245,C(CN=C(NCC1CCC1)N1CC2CCOCC2C1)C1CC(CF)C1 63246,N1(C(CSCCCC)=O)CC(C)(CNC(=O)CCc2ccnc(C)n2)CC1(C)C 63247,c1(C(=O)NCC=CCNC(CCC(C)C#N)=O)cc2n(n1)CCCN2 63248,C(=O)(CC1=CCOCC1)NCC1N(C(CCn2cnc(=N)[nH]2)=O)CCOC1 63249,C(CCCN=c1[nH]cnc(COC)c1F)(c1ccccc1)NC(CC1(C=C)CC1)=O 63250,Cc1ccc(CCC(=O)NC2(CNC(=O)Cc3ccc(O)nc3)CC2)cc1C 63251,c1(COC)nc(NN2CCC3(CCN(C)C3)C2)cc(=NCC(C2CC2)SC)[nH]1 63252,N1(C(Cc2c(C)noc2C)=O)CCC2(CCN(Cc3cc(Br)ccc3Cl)C2)C1 63253,Cc1cc(=NC2CC2C2CCN(C(=O)Cn3ncn(C)c3=O)CC2)[nH]c(Cl)n1 63254,N1(C(=O)CN2CCN(C3CC3)CC2)CCN(C(C2(F)CC=CC2)=O)CC1C1CC1 63255,C1(C)(CC)CCC(C(N2CC(NC(c3cscn3)=O)C2)=O)O1 63256,C12(NC(C(CC)C)=O)CCC(C(N3CC(O)(C(C)NC(=O)COC)C3)=O)(CC1)C2 63257,N1(C(C2C(CC)(CC)C2)=O)CC(C2(NC(C3CCN(C(N)=O)CC3)=O)CC2)C1 63258,O=C1NCc2c1ccnc2C(=O)Nc1nc2c(O)nc(=O)n(C3CC3)c2[nH]1 63259,N1(C(=O)NC)CCN(C(=O)C(=O)NCCCC2CCCC(C)C2)CC1 63260,C12(C(=O)NCC(=O)NC3CN(C(=O)C4CC4)C3)CC(CC(F)F)(C1)C2 63261,N1(C(C2CC(OC)C2)=O)CC(NC(c2c[nH]c(Br)c2)=O)CC(F)(F)C1 63262,C1(O)(C(=O)NCC2CCCN(C(C(C)C3CCCO3)=O)CC2)CCC(C)(C)CC1 63263,C1(C2(O)CN(C(C3CCc4n[nH]cc4C3)=O)C2)(CNC(C2CC(C)(O)C2)=O)CC1 63264,c1(CC)[nH]nc(C(=O)N(C)CCN(C)CC)c1Br.C12CC1N2.C(=O)O 63265,C#CCCCCCC(=O)N1CC(NC(c2nn(CC)nc2C)=O)C(F)C1 63266,N1(C(COC(C)C)=O)CCCC(C)(C)C1C(=O)NC(CC1CCCC1)CO 63267,N1(C(CNC(C(C)(C)c2cscn2)=O)C(F)F)CCCS1(=O)=O 63268,c1(C(=O)NC(CC2CN(C(CCCC#C)=O)C2)C)cnn2c1CC(C)CC2 63269,C1(C(C)NC(C2(CC3CC3)CC2)=O)CCN(C(=O)C(F)(F)C2CC2)C1 63270,C12(C(=O)NCC3CCN(C(c4ccncc4)=O)C34CC4)CC3CC(CC1C3)C2 63271,c1(CC)nnc(CNC(=O)C(O)CC2CCNCC2)s1 63272,C1(C(N)=O)(NC(c2ccc(F)c(F)c2)C)CCCCCC1 63273,CC(CC(F)(F)F)C(=O)NC1CN(C(=O)CC2CC(n3cnnc3)C2)CCC1O 63274,Cc1csc(C(N2CCC(C(=O)NCC(F)(F)CO)C2)=O)c1 63275,c1(-n2cc(C(=O)NC)nn2)cccc(NC(c2ccoc2)C)c1 63276,CCC(CC#N)N=c1ccc(Br)c(S(=O)(=O)N(C)CC)[nH]1.C1CS(=O)(=O)N1C 63277,C(C(=O)NCC(C)CNC(c1c(NC(C)=O)c[nH]c1C)=O)(C(C)C)OC 63278,N1(C(c2ccc(OC)c(Cl)c2)=O)CCN(C(C2CC=CC2)=O)CC(C)(F)C1 63279,N1(C(=O)C(=Cc2cccnc2)F)CCC2CCN(c3nc(Cl)ncc3F)CC2C1 63280,c1(C(=O)NC(CN(C(C2(CCC=C)CCCC2)=O)C)C)nccc(Cl)c1O 63281,c1(C(=O)OC)cc(Cl)c(F)cc1S(=O)(=O)NCCNS(=O)(=O)C(F)(F)F 63282,CCCCC(CC)C(=O)NCC(C)(CO)NC(C1CC2(C1)CC(C)C2)=O 63283,N1(CCC(=O)NC2CCC(NC(c3cc(=O)cc[nH]3)=O)CC2)C(=O)CCC1=O 63284,Cc1cc(N2CC(CNC(C3CCC3F)=O)C2)nc(=N)[nH]1 63285,c1(CC(N2C(C)(NC(=O)Nc3c(C)nn(C)c3)CC2)=O)ccc(F)cc1F 63286,C(=O)(CC(C)(C)C(F)F)N1CCCCC(NC(CCC=C=C)=O)C1 63287,C1(NC(CCC(=C)Cl)=O)CN(C(=O)COc2cc(Cl)ccc2C)CC12CCC2 63288,CC1CC=CCC1C(N1CCN(CC2(O)CN(C(=O)CCC3CCC3)C2)CC1)=O 63289,C1(C(=O)OC)CN(C(=NCCSc2ccccc2)NC(C2CCCO2)C)CCC1O 63290,N1(C(CCC(C)OC)=O)CCCC2(NC(=O)CN3C(C)CCC3C)CCCC12 63291,c1(C(=O)Nc2ccc(NC(C(CCC)CC)=O)cc2C)cnc2c(c1)NCC(=O)N2 63292,N1(C(CNS(NC)(=O)=O)=O)CCCN(C(C2CC(O)C2)=O)C(C(C)C)C1 63293,C1(N(C(CCOCCN(C(C=CCC)=O)C)=O)C)CCCCN(C)C1 63294,c1(C(=O)NCCC(C)NC(C(c2ccccc2)C)=O)ncsc1Br.C12CC1C2 63295,C12(NC(c3nc(CCCC)sc3)=O)COCCC1CN(C(=O)Cc1cccs1)C2 63296,C1(C(N(C)CCNC(=O)C(C)(C)n2cnnn2)=O)CCC(=O)NC1 63297,C1(C(=O)NCCCCC(=O)OC)CCC2(CC2)N1C(c1cn(C(C)C)nn1)=O 63298,Cn1c(C(=O)NCC2CCCCN2C(=O)CCn2cncn2)ccc1C1CCCO1 63299,c1(C(N2CC(CC=C)(NC(c3ccc(C)s3)=O)C2)=O)ccc(F)cc1 63300,C=C(CC(C(=O)NCC1CC1)N1CC(OC)CC(OC)C1)C(C)(C)C.c1(CS)nccs1 63301,c1(-c2ncc(C(=O)Nc3cc(C)c(F)nc3)nc2)ccc2c(c1)C(=O)CC2 63302,N1(Cc2scc(C(=O)N(C)C)n2)CCC(NC(Cn2c(C(C)C)nnn2)=O)CC1 63303,N1(C(Cc2nc(C)sc2C)=O)CCC2(CC1)CC2CNC(C1(C#N)CCOC1)=O 63304,N1(C(CC(C)(C)C)=O)CCN(C(=O)C=CC2CC2)C(CC2CC2)C1 63305,C(=O)(C(CC(C)C)N(C)C)NCc1nc(Cn2cc(C(C)(C)OC)nn2)sc1 63306,CC1CCN(C(c2ccccc2C(F)F)=O)CCN1C(=O)CC1CCC(=O)N1C 63307,Cc1nccn1CCCC(=O)NCCCC(=O)NCCC1(CO)CCC1 63308,C(=O)(CC(C)(O)C(F)(F)F)N1CCCC(C(C)NC(C2(SC)CC2)=O)CC1 63309,c1(N(C(=O)NC(C(=O)NC(c2cccnc2Br)CC)C)C)cccc(OC)c1 63310,C1(NC(c2c(C)nn(C)n2)=O)CN(C(c2ccc(F)c(CO)c2)=O)CC1N=[N+]=[N-] 63311,c1(NC(C2CC(C)(NC(CCCC#C)=O)C2)=O)cc(C)nc(OC(C)=O)n1 63312,CC1(C)CN(C(c2csnc2Cl)=O)CCC1CNC(C1CCC(C)(C)CO1)=O 63313,C(=O)(CCC(C)(C)C(=O)N1CCC(F)C(O)C1)OC(C)(C)C 63314,c1(C(=O)NCC=CCNC(C2CC(C)N(C)C2)=O)cnn2cccc(Cl)c12 63315,C1(C(=O)NCCC(F)Cn2cc(CNC3CCCCO3)nn2)CC2CCC1O2 63316,C(=O)(C(F)CC(C)(C)C)NCc1cc(C(N(C(C)C(C)C)CC)=O)on1 63317,N1(C(C(C)(C)OC)=O)CCN(C(c2ccc(C#N)c(F)c2)=O)CC(C)C1 63318,C(=O)(C(C)(O)C(C)(C)C)NC1CC(NC(c2ccc(CC)nc2C)=O)C1 63319,C12(NC(c3ccc(Cl)cc3F)=O)COCCC1CN(C(c1ccns1)=O)C2 63320,c1(C(C(=O)NCc2cccs2)N(C2(C#N)CC2)C)cc(-c2ccccc2)nn1C 63321,c1(C(=O)CC23CC(CNC(C4(NC(C)=O)CCC4)=O)(C2)C3)cccc2c1OCC2 63322,Cc1cncc(CCC(=O)NC(C2CCN(C(c3cnncc3O)=O)CC2)C)n1 63323,N1(C(C2=NOC(C)C2)=O)CCN(C(C2(C3CCCCC3)CC2)=O)CCC1C 63324,Cc1c(Cl)cccc1S(=O)(=O)N1CCC(C(=O)NCC2(C)CCCC2)CC1 63325,c1(OC)ccc(-c2ccccc2)cc1CCNC1CNC(=O)OC1=O 63326,C12(OC)CCC(Cn3cc(CC4CCOC4(C)C)nn3)(CC1)C2 63327,c1(C(=O)NCC(C2CCCN(C(C=C(C)C)=O)C2)(C)C)ccc(C(F)F)nc1 63328,c1(C(=O)NC2C(CNC(C3CCC(C)CC3)=O)CCC2)cccc2cncn12 63329,N1(C(Cc2c(C)scc2)=O)CCC(NC(=O)C=Cc2ccoc2)C(C)C1 63330,c1(NC(C(CC)N(C)C(C2CCSC(C)C2)=O)=O)cc(C)cc([N+](=O)[O-])c1 63331,C(=O)(C(F)C(C)(F)F)NCC1(C)C(=O)N1.c1(COC)nc(C2CC2)no1 63332,c1(C(=O)NC2CC3CN(C(C4(NC(N)=O)CC4)=O)C2C3)c(Cl)cc(Cl)nc1N 63333,C(=O)(C(C)(C)CCCO)N1CC(C)N(C(c2coc3c2CSC3)=O)CC1 63334,N1(CC(=O)NCC)C(=O)CCC1=O.N1(CC)CCOCC1CC=O.n12nccc1C2 63335,c1(CC(=O)NCCNC(=O)C=CCF)c[nH]c2ccc(Cl)cc12 63336,O=C(C1CCCc2scnc21)NC1CCN(C(=O)CCOCC(F)(F)F)C12CC2 63337,C1(CC(=O)N(Cc2scc(C(=O)NCCc3c(C)ocn3)c2)CC)CCCNC1=O 63338,C1(N(C(=O)COCP(C)(C)=O)C)CN(C(C2CCN(CC(F)(F)F)C2)=O)CC12CC2 63339,C12(C(=O)OC)C3C4C1C1C2C3C41C(=O)NCCC(CN)OC(C)C 63340,C1(NC(C2N(CC)CCOC2)=O)CCN(C(=O)Cc2cccs2)CC1C 63341,N1(C(C(C)(C)F)=O)CCCCC(NC(c2ccsc2Br)=O)CC1 63342,Cc1c(C(N2CCCN(C(C3CCCO3)=O)CC2)=O)[nH]c2cc(F)ccc12 63343,C(=O)(CCC(=O)NCCCCN(C)C(C1CCCC(F)C1)=O)N(CCC)CCC 63344,C1(CNC(COCCCC#C)=O)CC(C)CN(C(c2occc2CC)=O)C1 63345,C1(NC(c2n(C)ccn2)=O)CN(C(C2CC2C(C)(F)F)=O)C(C)(C)C1 63346,c1(C(=O)NCC2(OC)CN(C(c3c(C)nc(CC)s3)=O)C2)ccc2c(n1)NCC2 63347,N1(C(C=C(CCC)C)=O)CCC(N(C(=O)Cc2c(C)nc(C)nc2O)C)C2(CC2)C1 63348,C1(NC(c2n(C=C)nnc2)=O)(CC)CCN(C(=O)C(C2CCC(=O)N2C)C)CC1 63349,C1(NC(C2(C(N)=O)CCC2)=O)CCC(NC(c2cnc(Br)s2)=O)C1 63350,c1(CC)c(C(=O)N(C2CCCN(C(=O)CCn3cncn3)C2)C)cccc1Br 63351,c1(C(=O)NC2C(CNC(c3c(C)coc3)=O)CCC2)c(C)nn(CC(C)C)c1Cl 63352,Cc1nsc(CCC(=O)NCC2(NC(C3CCCOC3)=O)CCOC2)n1 63353,N1(C(c2[nH]cc(C)c2)=O)CC(N)C2(CCOCC2)C1 63354,C1(NC(c2nc(C)c(C)s2)=O)CCCN(C(=O)CN2C(C)CCC2C)CC1 63355,S(=O)(=O)(c1ccc(=NCCC2CCOC2)[nH]c1)NC1CC(C)(C)S(=O)(=O)CC1 63356,Cc1cc(C(=O)NCC2COC(CNC(=O)Cc3n[nH]c(C)n3)C2)nc(O)n1 63357,CC1C(NC(=O)CC2CSCCS2)CCN1C(=O)CCCc1ccccc1 63358,C=C(C)CC(C(=O)NCC1CCN(C(c2ncccc2F)=O)CC1C)NC(C)=O 63359,N1(C(COCCC(C)C)=O)CCC(F)(C(=O)NCCN2CCCCC2)C1 63360,c1(C(=O)NCC(O)CNC(c2cc(-c3ccccc3)co2)=O)cc(Br)cnn1 63361,N1(C(C2(COC)CCC2)=O)CC(CNC(c2cc(OC)nc(F)c2)=O)C(C)(C)C1 63362,c12cccc(F)c1C(=O)O2.c1(NC(=O)NC)ccc(SCSC)cc1 63363,CC1(O)CCCN(C(C2CCCCN(C(=O)CCc3ccc[nH]3)C2)=O)C1 63364,CC(C)C(O)C(=O)NC(C)(CNC(c1ccc(C(C)(C)C)s1)=O)C(C)C 63365,Cc1conc1C(=O)NC(C)C(c1ccccc1)NC(C1CSC1)=O 63366,CC1(C)CN(C(=O)Cc2nc[nH]n2)CC(CNC(C2COC3(CO)CC2C3)=O)O1 63367,C1(C)(C(N2CCC(O)(C(C)NC(c3ccc(C(F)(F)F)o3)=O)C2)=O)CCC2CC2C1 63368,c1(C(=O)NCCS(=O)(=O)N(CC)CC)ccc(S(N)(=O)=O)cc1.N12CCC(C1)C2 63369,C1(OC)CC(NC(=O)CCNC(=O)CN2CCNC2=O)C12CCC2 63370,C12(C(=O)NCC(C)(C)CNC(C3(C)CCOC3)=O)CCC(CC1)C2(C)C 63371,CC1CCC(O)CN1C(=O)CCC1CC(NC(c2cccc(Cl)c2O)=O)C1 63372,N1(C(C(CCSC)O)=O)CC(C(=O)NC2CCCC2N=[N+]=[N-])CC(C)(C)C1 63373,c1(SCC=C)cnc(Cl)cc1OC(C1CC2CC2N1c1nccc(OCC)n1)=O 63374,c1(C(N(C2CCCC(NC(CCC=CC(C)C)=O)C2)C)=O)cc(Cl)cc(F)c1F 63375,c1(CNC(C(=O)NC(c2nc(C3CCCCC3)no2)C)=O)cccc(F)c1 63376,N1(CN(C2C(OCC)(OC)C(OC)C2)CC(F)(F)F)CCC2(CC1)CN(C)C2 63377,Cn1c(C(N2CCN(Cc3cn4ccccc4n3)C3CC23)=O)cc2ccccc12 63378,N1(c2ncc(C)c(C)n2)CCC(NC(=O)C(C)S(N)(=O)=O)C(C)(C)C1 63379,CCCCCCCCC(C)CC(=O)N1CC(NC(=O)CCNC(=O)OC)C(C)C1 63380,CN1CCN(c2cc(N(C)Cc3ccc(Cl)cc3)nc(C(F)(F)F)n2)CCC1=O 63381,C1(=CC(=O)NCC2CCC(NC(C(C=C)C)=O)C2)CCC(C)CC1 63382,C(CCCCCC(=O)N1CC2CC1CN2C(c1cnn2ccn(C)c12)=O)SC 63383,N1(CC)CCCC(C(=O)NCC2CN(C(=O)COC)CC2C(F)(F)F)C1 63384,Cc1noc(C(C)C)c1C(=O)NCC(C)(C)CCNC(C1CCCN1C1CC1)=O 63385,c1(C(N(C)Cc2ccccc2-c2nncn2C)=O)ccc(I)c(OC(F)(F)F)c1 63386,c1(CC)ccc(Cl)c(C(N2CCC(CO)C(NC(c3ccc(OC)o3)=O)C2)=O)c1 63387,C1(C(=O)NCC2N(C(C(C(CC)C)OC)=O)CC2)CC2CCCCCC12 63388,N1(C(C(C(CC)O)C)=O)C(CNC(=O)Cc2cccn2C)CC2CCCC12 63389,C1(CNC(c2c(C)nc(C(C)C)o2)=O)CN(C(C23CC(CO2)C3)=O)CCC1(F)F 63390,Cc1cc(C(=O)NCCC2CCCN(C(C3CC3c3ccccc3)=O)C2)n(C)n1 63391,N1(C(C2(C)C(C)(C)C2)=O)CC2CC(CNC(C3CC4(CC4)CO3)=O)C2C1 63392,C1(NC(N2C(C(=O)NCC)CCC2c2ccccc2)=O)CCC(OC)CC1 63393,Cc1nc(=N)[nH]c(=NCCCCNC(=O)C(C)(C)NS(C)(=O)=O)[nH]1 63394,c1(COC)nc(N2CCC(C)C2CNC(=O)CSc2cccc(Cl)c2)cc(Cl)n1 63395,c1(CNC(=O)N(c2ccc(Cl)cc2)c2ccccc2)cc(C(=O)C(F)F)ccc1F 63396,N1(C(C(C=C)(C)CC)=O)CC(C2CCCN(C(c3ncn4ccccc34)=O)C2)C1 63397,c1(C(=O)NCc2cccc(NC(c3c(C)ccs3)=O)c2)cnc2[nH]cncc1-2 63398,C(=O)(C1=NOC2(CCOC2)C1)N1CCC(CN(C(=O)CNS(C)(=O)=O)C)C1 63399,CCCCCC(O)C(=O)NCC1CC(CNC(=O)CC(F)(F)CC)C1 63400,c1(CC)cnc(C(=O)N(CCCCN(C(=O)CC2COCCO2)C)C)nc1 63401,c1(C(c2n(CC(=C)C)nnn2)Nc2ccsc2)cccc(OC)c1Cl 63402,C1(CNC(c2cncs2)=O)CN(C(=O)CN2C(=O)CCC2=O)CCC12CCOC2 63403,CCC(CCOC)C(=O)NCC(CNC(=O)Cn1ccnc1C)OC 63404,c1(COC)nc(CC(CC(F)F)C2CC2)n(-c2ccc(Cl)cc2)n1 63405,C(=O)(C(F)(F)C(C)O)N(CCCNC(C1CCCC1(F)F)=O)C(C)C 63406,c1(COCC(=O)NCC)ccc(F)c(C)c1.C1(C2CC2C)CCN(C(=O)CO)CC1 63407,c1(OC)cccc2c1OC(C(=O)NC1C3CCC1N(C(C1(CF)CCC1)=O)C3)C2 63408,CCCC(CNC(C1CCCSC1)=O)NC(c1cnc(CC(C)C)s1)=O 63409,C(=O)(C(C)C(C)(C)C)N1CCC(C(C(=O)NCc2n(CC)ccn2)(C)C)C1 63410,Cc1noc(CO)c1C(=O)NCCN(C(=O)CCN(CCC(C)(C)C)C)C(C)C 63411,c1(C(CCO)OC)ccc(C(C)C)cc1.n1(CC)nnnc1C1C(C2CCCC2)N1 63412,C1(NC(CCC(C)NC(c2c(C)scc2)=O)=O)C2C3CCC(C3)C12 63413,S(=O)(=O)(c1cccc(N2CC3CC2C(F)(F)C3)n1)NC1(CC)CCC1 63414,C1(NC(=O)Cc2ccsc2)CC(F)(F)CC1NC(C1(O)CCC1)=O 63415,CC(C)C(CN(C)C)C(=O)N1CCC1CN(C1CCN1)C(C1CCC1)=O 63416,C1(C(=O)Nc2cccc(NC(=O)Cc3nc[nH]n3)c2)CC2CCC(C1)C2F 63417,C1(C(=O)NCC2(OC)CN(C(C(CC=C)(C)C)=O)C2)CC2COCC(C1)C2 63418,c1(OC)ccc(C(=O)NCC2(CNC(C3CCC(C(C)C)CC3)=O)CCC2)cc1 63419,C(=O)(C1=CCC(NC(=O)C(C)(C)CO)C1)NCC(CSC)OC 63420,N1(C(CCC#C)=O)CCC2(CC1)C(NC(=O)C(N1CCC(C)C1)=O)CS2(=O)=O 63421,C(=O)(CCC(C)(C)NC1(CC(N2CCC(C)C(C)C2)=O)CC1)NC 63422,C1(COC)(NC(=O)CC2CCC(C)(C)C2)CCN(C(c2cscn2)=O)C1 63423,C(C)(C)(CCC(=O)N1CCC(OCC(=O)N(CC(C)(C)O)C)C1)OC 63424,C(c1cccc(F)c1)=CC(=O)N(CC(C)O)CCNC(CN(C)CC)=O 63425,C1(NC(=O)CN2CCCCCC2)COCCN(C(C2(n3ncnn3)CC2)=O)C1 63426,Cc1cc(=O)c2cc(NC(=O)NC3(c4ccc(F)cc4F)CC3)ccc2[nH]1 63427,CC1(C#CC(=O)N2CC3CN(C(c4cncc(Cl)c4)=O)CCC23)CCCO1 63428,C1(CNC(C2CC(C)(C)C2)=O)COCCN1C(C1SCCS1)=O 63429,C1(CC)CCN(C(=O)CC(C)C2CCCO2)C1CNC(C1C2CCCCC12)=O 63430,C1(C(=O)NC2COCCN(C(c3c(C(C)C)ocn3)=O)C2)CS(=O)(=O)CC12CC2 63431,C1(CNC(CC2N(C)CCC2)=O)(CO)CCN(C(C23CCCC(CO2)C3)=O)CC1 63432,O=C(N=c1cc(Cl)nc[nH]1)c1cc2c(s1)CCN(C(=O)Cc1ccccc1Br)C2 63433,Cc1cc(C#N)c[nH]c1=NCC1CC2(CC(NC(C3CCCC3)=O)C2)C1 63434,C1(CC(=O)NC(C2CCCN2C(=O)C(C)(C)n2cnnn2)C)CC(=O)NC1=O 63435,N1(C(c2cnc(S)n2C2CC2)=O)CC2(CCCCN2C(C2CC2F)=O)C1 63436,C(CC(C)C(=O)NC(C)CN(C)C(c1ccc(CCCCCC)o1)=O)=CCC 63437,c1(C(N2CC(O)(CNC(CC(=C)Br)=O)C2)=O)nc2cc(O)ccc2[nH]1 63438,C12C(CCCN1C(=O)CC1CC(=O)NC1=O)NC2=O.C1(CC)CCCCO1 63439,C1(NC(COCCC#C)=O)CC2CCC1N2C(C1CCN(C2CC2)C1=O)=O 63440,C(=O)(CC(C)C(=O)NCC(C)CNC(c1coc(Br)c1)=O)OCC 63441,CC1(C)CN(C(=O)C(C2CC2)NC(=O)C(C2CCCCC2)F)CCC1O 63442,CP(C)(=O)COCC(N1CCC(n2cc(CNC(c3ncccn3)=O)nn2)C1)=O 63443,C1(NC(C2CCCCC2)=O)CC2CCC1N(C(c1ccn(C3CC3)n1)=O)C2 63444,C(=O)(C(C)(C)CSC)NCC1CC(NC(C(C=C)c2ccccc2)=O)C1 63445,N#Cc1ccc(F)cc1C(N1CC(C(=O)NC)CC1c1nc(C(F)(F)F)no1)=O 63446,c1(C(C)=O)cc(NC(c2csc(NC(=O)Nc3cnc(C)nc3)n2)=O)ccc1O 63447,CON=C1CN(C(c2ccc(C(N)=O)o2)C(=O)NCc2ccc(F)cc2)C1 63448,C1(CC#C)CCCCN1C(=O)C(C)CNC(c1cc(Cl)c[nH]1)=O 63449,C1(NC(c2scnc2C2CC2)=O)CN(C(=O)CC2OCCCO2)Cc2nccn2C1 63450,C(=O)(C(C)CNC(=O)C(CNC(c1nc[nH]n1)=O)N(C)C)OC 63451,CC1C(C(=O)NCC2CC(F)(F)C2)CCN1C(=O)CCC1CC1(F)F 63452,C1(NC(C2CC(N3CCN(C)CC3)C2)=O)CCN(C(=O)CC2CCOC2)CC1F 63453,c1(OCC)nc(N(CCCN(C)C(c2cscn2)=O)C)ncc1C 63454,C1(NC(c2c(C)onc2C(F)(F)F)=O)CN(C(=O)Cc2cccn2C)CC12CC2 63455,C1(NC(C(C)C)=O)CCN(C(c2ccc(C(=O)NC3CC3)o2)=O)CC1 63456,C1(N(C(CS(=O)(=O)NC)=O)C)CCCCN(C(c2nnc(S)n2C)=O)C1 63457,CCC(CCCC(=O)N(C)CCc1cnccn1)NC(=O)Cc1cnn(C)c1 63458,C(CCCCC(=O)N1CC(NC(C2(F)CCCCC2)=O)C2(CC2)C1)NC(C)=O 63459,c1(C(=O)OC)cc(C)sc1NC(C1CN(C(=O)C(C)Cc2c(C)noc2C)C1)=O 63460,C1(NC(C2CC23CCC3)=O)CCN(C(c2cc3c(s2)CCCC3)=O)C12CCC2 63461,N1(C(c2c(Cl)cn(CC)n2)=O)CCN(C(=O)Cc2c[nH]nc2O)C(CO)C1 63462,N1(C(CCN(C)C(C2(C(N3CCCC3)=O)CCOC2)=O)=O)CC2(CNC(=O)N2C)C1 63463,CC(CC(=O)NC(CNC(=O)C(N)=O)C(C)(C)C)S(=O)(=O)c1ccc(F)cc1 63464,CCCCC(CNC(c1cncc(F)c1)=O)NC(=O)Cn1ccnn1 63465,CC(CN(C)C)CCC(=O)NC(C)(C(=O)N1CC(CC(N)=O)C1)C1CCC1 63466,C12(C(N3CCC(NC(=O)OC)CC3)=O)CN(c3ccc(Cl)nn3)CC1CCO2 63467,c1(C(=O)NC(C(=O)NC(C(=O)N(CC)CC)C)C(C)O)ccc2c(c1)CC2 63468,N#CC1CN(C(=O)CC2CCCN2C(c2cnn(CCCCO)c2)=O)CC12CCC2 63469,C(=O)(CC(C)CCC=C(C)C)NCC1C=CC(NC(c2c(O)ccc(OC)c2)=O)C1 63470,c1(COCC(N2C(c3ccc(C(=O)O)o3)CCC2)=O)ccc(F)cc1 63471,C1(C(N(CCO)CC)=O)CC(O)CCN1C(=O)C1=NOC(C)C1 63472,CC1(C)CN(C(c2cc[nH]n2)=O)CC1NCCCc1cccc(Cl)n1 63473,CCCS(=O)(=O)CC(=O)NCCC(O)CNC(c1cc(OC)cs1)=O 63474,c1(C(CC(=O)O)C(=O)Nc2ccccc2F)cccc(OC2CCC2)c1 63475,N1(C(C(CCC)NC(N)=O)=O)CCC(NC(c2ccc(C)cc2F)=O)C12CC2 63476,N1(C(CC(C(C)C)C)=O)CCCCC(C2CN(C(C3(C(F)(F)F)CC3)=O)C2)C1 63477,c1(C(N(CC)Cc2cn(-c3cc(O)ccc3Cl)nn2)=O)cc2c(F)cccc2[nH]1 63478,c1(C(c2nnnn2CCC)NC2(CC=C)CCCCCC2)cc(C)c(C)cc1C 63479,CC(C(=O)NC1(CC(=O)NCCC2CC2C)CC1)C1CCC1 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63498,C1(CCNC(c2c(COC)cccn2)=O)CC2CCC(C1)N2C(=O)CCSC 63499,n1(C(C)C)ccc(C(=O)NC2CC(CNC(=O)C(C)NC(C3CCC3)=O)C2)n1 63500,c1(CSCCN(C)C)csc(=NC(CCO)C2CC2)[nH]1 63501,N1(C(c2ccc(OC)c(I)c2)=O)CC(NC(c2cnsn2)=O)CC(F)(F)C1 63502,CC(CC(=O)NC1(C)CCN(C(c2cnn(CCF)c2)=O)C1)C(F)F 63503,c1(OC)ncc(C(N2CC3(C2)CN(C(C2COCC(C)O2)=O)C3)=O)cc1C 63504,Cc1ccc2c(=NCCC3CC=CC3)[nH]c(=NC(C)c3ccccc3)[nH]c2c1 63505,C1(NC(C(N2CCCCC2=O)C)=O)CN(C(=O)CSC(F)(F)F)CCC1CO 63506,c1(C(CNC(C=CSC)=O)(C)NC(c2coc(O)n2)=O)ccccc1C(F)(F)F 63507,Cc1cc(C(N2CCN(C(c3cnc(O)c(Br)c3)=O)C(C)C2)=O)nnc1Br 63508,c1(C(=O)NCC(COC)NC(=O)CN2CCCCC2=O)nnc(S)nc1C 63509,N1(C(c2c(OCC)ocn2)=O)CC(N2CCOCC2)C2(CC2)C1 63510,N1(C(C2(C)CCCO2)=O)CCCC(F)(CNC(=O)COc2ccsn2)C1 63511,CC(C)(O)C(F)C(=O)NCC1CC(F)(F)CN1C(=O)CCCn1ccnc1 63512,c1(C(N2C(CNC(C34OCCC(C)(C3)C4)=O)CCC2)=O)cccc2c1COCC2 63513,c1(CC(CC)OC)nc(-c2cccc(N)n2)nn1C1(C)CCOCC1 63514,N1(C(c2nn(C)c(O)c2)=O)CCC2(CCCN2c2nnc(C3CC3)o2)CC1 63515,C1(NC(C2N(C(C)=O)CCC2)=O)CCC(CN(C)C(c2cnnn2C)=O)CC1 63516,C1(CCC)(NC(c2ccc(F)c(CC)c2)=O)CCCN(C(=O)COC)C1 63517,c1(C(=O)NC2CCN(C(c3ccnc(OC)n3)=O)C2)cccn2ccnc12 63518,c1(NC(C2CCN(Cc3ccncc3O)CC2O)=O)cnc(Cl)cc1[N+](=O)[O-] 63519,C(CNC(c1n[nH]c2c1COC2)=O)(CC(F)(F)F)NC(C1(CC#C)CCC1)=O 63520,c1(C(N(CCC(=O)N2CCC2)C)=O)ccc(S(=O)(=O)N2CCCCC2)cc1.CN 63521,c1(CC(=O)NC(c2ccccn2)CC)csc(C(c2ccccc2)C)n1 63522,Cc1cc(C)n(C(C)C)n1.C1(C)(C(=O)COC(=O)CN(C)C)CCC1 63523,CCC(F)(F)C(=O)NC(C)CNC(=O)C(C)(O)C1CCC1 63524,C(=O)(CCCCCC(C)(C)C)NC(C(=O)OCCCC)(C)C(C)C 63525,C1(F)(C(=O)NCC(COC)F)CCN(C(C2COCCC2C)=O)CC1 63526,C(=O)(CC1CCOc2ccccc21)N1CC(C)C(NC(=O)C=CBr)C1 63527,Cc1cccc(NCC(N2CCC(CC(N)=O)(NC(=O)CC(C)(F)F)CC2)=O)c1F 63528,N1(C(C(C)SCC)=O)CCCC2CN(C(c3ccc(CC(C)C)s3)=O)CC12 63529,Cc1ccc(C(=O)NC(C)(C)CNC(=O)Cc2ncn3c2CCC3)cc1CO 63530,c1(C(N2CCC(Cc3cn(-c4ncc(Br)cn4)nn3)C2)=O)cccc2oc(O)nc12 63531,c1(CNC(Cc2c(C)nsc2)=O)ccc(C(=O)NC(c2ccccc2)C(N)=O)cn1 63532,Cc1cc(Cl)cnc1C(N1CCC(C(=O)NCCc2nn[nH]n2)C(O)C1)=O 63533,S(=O)(=O)(CCC(=O)NC1(CO)CN(C(c2sc(C)cc2OCC2CC2)=O)C1)NCC 63534,c1(C(C(=O)N(CCCNC(=O)COCC2CCCCC2)CC)O)cccc(Cl)c1 63535,C1(C(N(C2(CCO)CC2)C)=O)OCCC1NC(c1cnn(C(F)F)c1)=O 63536,CC1CCN(C(c2cnc(CN(C)C)s2)=O)CC1Cn1cc(C(C)(C)C)nn1 63537,C1(N(C)C)CN(C(=O)C(CCF)NC(=O)CC2CC(=O)NC2=O)CC12CC2 63538,C(CC(C)C(=O)NC(CNC(C1(c2cc[nH]n2)CCC1)=O)C(C)C)=CCC 63539,CCCCCC(F)C(=O)N1CC(CNC(=O)CN2CCOC2=O)CC(C)C1 63540,C1(NC(C(C)SC2CC2)=O)CCOC(NC(=O)CC2(O)CCOCC2)C1 63541,c1(NC(CC(N)Cc2ccc(F)c(Cl)c2)=O)cc(N2CCCC2=O)ccc1Cl 63542,C1(C(=O)Nc2scc(-c3c(C)cc(C#N)cc3)n2)CCC2(CC1)OCCO2 63543,C12(C=O)CCC(CC1)N(C(=O)CCCN=[N+]=[N-])C2.C1(C(C#C)OC)CCOC1 63544,Cc1nn(C)cc1C(=O)NC1CCCC1C(=O)NCC(O)C1(C)CC1 63545,C1(C(=O)NC(C(N2CCCC(CCC=C)C2)=O)CCC)CCC(O)CN1C 63546,C1(OC)CCC(C(N2CCCC(NC(c3cnn(C)c3Br)=O)C2)=O)CC1 63547,CC1CCC(C)(C(=O)NCC(C)CNC(C2CCOC2)=O)CC1 63548,C(C)(C(=O)NC(C)Cc1cccnc1)(C1CC1)OC 63549,Cc1cccn2cc(CC(=O)NC(C)C(CO)NC(=O)C(C3CC3)C3CC3)nc12 63550,Cc1nc(NC(C)(C)CN(C(=O)CSC(F)F)C)cc(Cl)n1 63551,c1(C(=O)NC(CNC(=O)NC(C)=O)C(C)C(C)C)cc(Cl)cc(Cl)c1Cl 63552,Cc1cnc(C)c(NC(C2(F)CC=CC2)=O)c1 63553,C1(C(=O)NCCCC(=C)C)CC2CCC1N2C(=O)C=C=C(C)C 63554,N1(C(CSCC#C)=O)CC2CCCC(C(=O)NC3CCC(=O)NC3C)C2C1 63555,CCN=c1[nH]c(C)c(C(N2CCCCC(NC(=O)C(F)=CCCF)C2)=O)s1 63556,c1(NC(C2CC2C(N2CCC3(CCO3)C2)=O)=O)ccc(Br)c(CO)c1 63557,Cc1scc(C(=O)NC2CN(C(c3cc(O)ncn3)=O)CC2C(N)=O)c1C 63558,CC(C)C(C(=O)NCC1C2CCCOC12)C(C)NC(c1cc(C#N)ccc1N)=O 63559,N1(C(C(COC(C)C)NC(C)=O)=O)CC(NC(=O)C=C2CC2)C(O)C1 63560,C(=O)(C1=Cc2cc(Cl)ccc2OC1)NC(C)CN(C)C(C1C(C)C1C)=O 63561,c1(OC)cccc(CNCCNC(c2ccnc(OC3CCOC3)c2)=O)c1 63562,N1(C(CSCCC)=O)CC2CCCCC2(CNC(=O)C=C2CCCCC2(C)C)C1 63563,c1(OC)cc(Cl)ccc1C(N1CCC(O)C(F)C1)C(=O)NCc1cccc(Br)c1 63564,Cc1nccnc1C(N1CCC(C(=O)NCC2(N(C)C)CC2)C1)=O 63565,C1(CC(NOCC#C)=O)CC(C(=O)N(C)C)C1(C)C.C12CCN1C2 63566,C1(C(C(=O)NCCCOC=C)NC(=O)CCn2cccc2)CC=CCC1 63567,c1(CC(=O)N(CC(CNC(COCC=C)=O)(C)C)C)cc(Cl)cc(Cl)c1 63568,C1(C(N2CC(CCC)C(NC(c3cc[nH]n3)=O)C2)=O)CSc2ccccc2O1 63569,N1(C(=O)Nc2c(C)cc(N3CCOCC3)cc2)CCN2CCOCC2C1 63570,Cc1ccc(F)c(C(=O)NCC2CCN(C(C3(CC4CC4)CC3)=O)CC2)c1F 63571,C1(NC(c2c(CC)nn[nH]2)=O)CCCCC1C(=O)NC1CC(CCSC)C1 63572,N1(C(c2n(CC)ncc2)=O)CC(C(=O)N(CC(C)OC)CC)CC12CCC2 63573,C1(CC=C)(C(=O)NCCCCN(C(=O)CCc2cccn2C)C)CCCCC1 63574,c1(C(N2CCC3(CN(C(c4cc(C)ns4)=O)C3)C2)=O)cn2cccc(F)c2n1 63575,O=C(C1=Cc2cccc(Br)c2OC1)OCC(C1(F)CCOC1)=O 63576,C(=O)(CC1CCOc2ccccc21)N1CC(NC(C(COC)C)=O)C(C)C1 63577,C1(C(=O)NCC2CCCN(C(=O)CCC3CC3C)C2)(OC)CS(=O)(=O)C1 63578,C(c1ccc(F)c(F)c1)=CC(N1CC(C)C(NC(=O)CN2CSCC2=O)C1)=O 63579,CP(C)(=O)CCC(=O)NC1CC(F)(CNC(=O)CCn2cncn2)C1 63580,CC1CC(C(N2CCC(CCCCCNC(C3CC3C)=O)CC2)=O)CCS1 63581,C=CCCCC(C1CC1)NC(=O)C=C(C)CNC(=O)Cc1ccc(C)o1 63582,CN1CC(NCc2ccc(-c3ccccn3)nc2)Cc2ccccc21 63583,CCC(C(=O)NCC1(NC(=O)COC2CCCOC2)CCC1)C(C)(C)CC 63584,c1(NC2(CSC)CC2)cc(=NC2(c3nnnn3C(C)C)CC(C)SC(C)C2)[nH]n1C 63585,c1(OC)cc(CN2CC(NC(c3ccc(C(F)(F)F)nc3Br)=O)C2)ccc1O 63586,c1(C(c2nnnn2C)NC2CC2)ccc(COC(C)CC2CC2)cc1 63587,S(=O)(=O)(C1CCN(C(=NCCSc2ccc(F)cc2)NC2CSC2(C)C)C1)NC 63588,N1(C(C=C(CC)CC)=O)CCC2CCCC12C(N1CCCC1CSC)=O 63589,C1(C(C)C)CN(C(c2c(Cl)cccc2I)=O)CCN1C(=O)Cc1cnn(C)c1 63590,C(=O)(CCCCCN(C)C(C1CC(C)(F)C1)=O)NCCCOCCCC 63591,c1(OC)ccc(C(=O)N(CC(O)CN(C(=O)C(O)CCN(C)C)C)C)c(OC)c1C 63592,C1(C)(C(=O)NC(COC)(C)C)CC12CCN(C(=O)C(O)C(C)(C)C)CC2 63593,Cc1c(C(N2CCC(N(C)C(c3cccc(F)c3Cl)=O)C2)=O)ccc2c1CCC2 63594,c1(C(N2CC3C(CNC(CCCOCC=C)=O)(C3)C2)=O)ccc(OC)nc1Cl 63595,CC1CN(C(C2CC23CCSCC3)=O)CCN1C(=O)CCCC1CCCCC1 63596,C=CC(CC(=O)NC(C)CCCCNC(=O)Nc1nccc(C)n1)c1ccccc1 63597,C1(CNC(=O)C(F)C2CCCC2)CCN(C(=O)C=Cc2cscn2)C12CCC2 63598,N1(C(c2nc(CC)oc2)=O)CC(C(=O)Nc2cc(C#N)ccc2O)C2(CCC2)C1 63599,C=CCCC(CC(C)C)C(=O)N(CCNC(=O)C(C(C)C)NC(=O)OC)CC 63600,C1(CCN(C(=O)C(F)OC)CCCC)CCN(C(C2(CF)CC2)=O)CC1 63601,C1(N(C(=O)CC2(C#N)CCC2)C)CC2CCC(C1)N2C(c1cnn2c1OCC2)=O 63602,Cc1n[nH]cc1CC(=O)N(C1(C(=O)NOCCCC2CC2)CCC1)CC1CC1 63603,C1(C(C)C)CN(C(c2cc(C3CC3)cnc2Cl)=O)CCN1C(C1CCCCO1)=O 63604,C(=O)(C(O)C1=CCCCC1)NCCOCCCN(C)C(C1COCC(C)(C)O1)=O 63605,c1(NC(CC)CSC)cc(=NCC(Cc2ccccc2F)CO)[nH]c(C)n1 63606,CC1CC(C)C(C(=O)NC(C)CCNC(c2cc(C(C)(C)C)no2)=O)O1 63607,C1(CNC(c2ccc(C)o2)=O)CCCC2(CCN(C(=O)CC(C)C(C)C)CC2)O1 63608,n1(CC(=O)NC2C(C)CN(C(=O)CN3CC=CC3)C2)ccc([N+](=O)[O-])n1 63609,Cc1ccc(C(=O)NCCC(C)NC(c2cnn(CC(F)F)c2)=O)cc1F 63610,CN1CCC2(CCN2)C1.c1(-c2cn(C3CC4(C=O)C3C4)nn2)ccc(Cl)cn1 63611,N1(C(c2cc3c(cc2Cl)OCO3)C(=O)NCC=C)Cc2ccccc2CC1CC 63612,Cc1cnc(C(=O)NC2CCN(Cc3cc(Cl)ccc3Cl)CC2C)c(C)c1 63613,CN1CCC(NC(=O)CC(C)(C)C)C12CCCN(C(C1(O)CCCCCC1)=O)C2 63614,C1(NC(CCNC(C)=O)=O)CCOC12CCN(C(=O)CC1CCC(=O)C1)CC2 63615,c1(CNCC(CCCC)CCC)nc2cc(F)ccc2s1 63616,N1(C(c2ccn(CCC)n2)=O)CC2(CCC2)CC1CNC(c1cc(C)c(C)o1)=O 63617,c1(N(CC(C)=O)C(C)C)ccc(F)cc1C(=O)N(C1CCCOC1)C1CCNCC1 63618,c1(C(N2CC(COC)(CNC(=O)CCCF)C2)=O)cnn2ccncc12 63619,CCC(C)(C)C(=O)N1CC(NC(=O)C(c2cccc(OC)c2)OC)C(C(F)F)C1 63620,N1(C(CC2(OC)CC2)=O)CC(CNC(=O)CSC2CC2)C2(CC2)C1 63621,c1(OC)ccc2c(CC(N3CCC(CCNC(=O)CCCSC)C3)=O)coc2c1 63622,N1(C(CSCC(=O)OC)=O)CC2CC1(CN(C1CCCC1)C(c1cncnc1)=O)C2 63623,c1(OC)ncc(Br)cc1C(N1CC2(C1)CN(C(c1cc[nH]c(=N)c1)=O)C2)=O 63624,c1(CC(=O)NC2CN(C(C3CCCC4CC34)=O)C2)ccc2c(c1)OCCO2 63625,C1(NC(C2CC(=C)C2)=O)CCN(C(c2cc(OCCC)cc(SC)c2)=O)C12CC2 63626,C(=O)(CC(C)(C)N(C)C)NCC1N(C(CCOCCOCC)=O)CC=C1 63627,C=Cc1ccc(C(N2CCC(C(CO)NC(=O)Cc3cc[nH]c3)CC2)=O)cc1 63628,c1(C(C(C)NC(C2(CC)CN(C(c3c[nH]nc3CN)=O)C2)=O)O)ccc(Cl)cc1 63629,N1(C(C2N(C(c3cc(C)ncn3)=O)CCC2O)=O)CC2CCC(O)C2C1 63630,C1(C)(CNC(CCOC(C)C)=O)CCCN1C(=O)Cc1cn(C)nn1 63631,c1(C(N2CC(N(C(C=CCOC)=O)C)C2)=O)[nH]c(-c2cccc(C)c2)nc1C 63632,C(c1ccc(F)c(F)c1)=C(C(N1C2CN(C(C3(OC)CC3)=O)C(C2)C1)=O)C 63633,N1(CC(COC(=O)Cc2cc3c(s2)CCC3)O)CC2CCCC2C1c1nn[nH]n1 63634,N1(C(C(C)NS(CC)(=O)=O)=O)CCC2(CC1)CCN(C(C1C(C)C1C)=O)CC2 63635,S(=O)(=O)(c1c[nH]c2ncccc12)N1CCC(NC(=O)OC(C)(C)C)C(C)(C)C1 63636,N1(C(C(C)S(N)(=O)=O)=O)Cc2ccccc2C1CNC(C1CC2(C1)CC(O)C2)=O 63637,N1(C(CCOC)=O)CCCC(c2cc(O)n[nH]2)C1.C#CCS 63638,C1(C(N2C(CN(C)C(c3ncn4c3CCC4)=O)CCC2)=O)C2CCC(C2)C1C 63639,c1(C(=O)NCC(C2(O)CCN(C(C=CC=CC)=O)C2)C)cc(Cl)ncc1N 63640,C1(CCNC(c2c(C)snn2)=O)CN(C(c2ccnnc2O)=O)CCCO1 63641,c1(C(=O)OCC)cnc2n1CCN(C(C1(O)CCN(Cc3ccccc3)C1)=O)C2 63642,c1(OC)ccc(F)c(F)c1.c1(C2(C(=O)NCC3C(=O)N3)CC2)ccc(CO)cc1 63643,C1(C(NOCCCC=C)=O)CC2(CCN1C(=O)C(C)C(C)(C)C)CC2 63644,C1(C(N2CCC(C(=O)NCC(CC)(C)CO)C2)=O)CC2CC(=O)C1O2 63645,C1(C(=O)NC2CCN(C(CNC(c3n(C)ncc3)=O)=O)C2)CC2(C1)CC2F 63646,C1(NC(c2ccc(OCC)s2)=O)CN(C(=O)Cc2cnsc2)CC12CC2 63647,CN1CCC(C(N2CC(F)(CO)C2)=O)(NC(C23CCCC2C3)=O)C1 63648,CCC(CC(=O)NCCC1CCOC1(C)C)NC(=O)C(n1cc(C)cn1)C 63649,c1(C(=O)NC2CN(C(C(C)NC(C)(C)C)=O)C2)ccc(-c2ccccc2)[nH]1 63650,N1(C(C2CN(CC)C(=O)C2)=O)CC2(CCC2)CC1CNC(C1C=CC=CC=C1)=O 63651,c1(C(=O)NCCC2(CNC(c3n(CC)ccn3)=O)CC2)cc2n(n1)CC(F)C2 63652,n1(CCC(=O)NCC2N(C(C3CC(=O)C3)=O)CCC2)cnc([N+](=O)[O-])c1 63653,C=C1CCC(C(=O)N(C)CCOCCCNC(C23CCC2C3)=O)CC1 63654,c1(C(C(=O)NCCOC)N(C(=O)OC)C)cnc(C(C)(C)C)[nH]1.c1(CC)ccccn1 63655,CCCCC(C)(F)C(=O)NCC1CC2CCC1N(C(=O)C(C)CC)C2 63656,c1(C(N2CCC(N(C(C(CC)O)=O)C)C3(C2)CC3)=O)cc2cccnc2cc1F 63657,N1(C(Cc2c(OC)cc(F)cc2)=O)CCCC12CN(Cc1cc(Cl)cnc1F)C2 63658,c1(C(N(CC(CN(C(Cc2c(C)occ2)=O)C)O)C)=O)ccc2c(c1)CCC=C2 63659,Cc1ncc(CCC(N2CC3CC(NC(c4ncccn4)=O)C3C2)=O)c(O)n1 63660,c1(C(N2C(CCNC(CC3(C)CC3(Cl)Cl)=O)CCC2)=O)c[nH]ccc1=N 63661,N1(C(CNC(c2c(C)occ2)=O)=O)CCC2CN(C(=O)C(C)CN(C)C)C2C1 63662,c1(CN2C(C(=O)NCCc3cccc(C)n3)C=CC2)cc(C)ccc1O 63663,CC1(C)CN(C(=O)Cc2ccccc2O)C(CNC(=O)CCc2nccs2)CO1 63664,C1(CNC(c2ccc(SC)s2)=O)CC(NC(c2nncn2CC2CC2)=O)C1(C)C 63665,N1(C(C(C=C)C)=O)CCC(C)(CC(=O)NC(C)CS(N)(=O)=O)C1 63666,c1(C(N2CC(CNC(c3ccncc3O)=O)C3C2C3)=O)ccc2snnc2c1 63667,C1(C(=O)NC(C2CN(C(c3c(CC)onc3C)=O)C2)C)CCC2(CCOCC2)C1 63668,C12(NC(C3CN(C(C4C5CC6C(C5)C46)=O)CC3F)=O)CCC(CC1)CC2 63669,C(=O)(CC(C)C)NC1CC(C(C(=O)N(C(CCC)C)CC)F)C1 63670,c1(CC(=O)NC(C(C)(C)NC(C(CC)C#N)=O)C)ccc(Br)c(OC)c1 63671,N1(C(C2C(C(N)=O)COC2)=O)CC2CCCC2(NC(=O)CCOCC(F)F)C1 63672,c1(C(=O)N(C(=O)CCCC(c2ccccc2)O)CCCO)ccccc1Cl.NC1CC1 63673,C=CC1(CC(=O)NCC2CCCN2C2CCC(C)(C)CC2)CCCCC1 63674,C1(C(=O)NCC2C(C(=O)NC(C(C)C)CO)CC2)CC2C(C1)C2(F)F 63675,C1(NC(c2cn(CC3CC3)nn2)=O)CCCCN(C(C2C3CC4C(C3)C24)=O)C1 63676,C1(NC(C(C)C2CC2)=O)C=CCC(C(=O)NCCOc2cccnc2)C1.C1CO1 63677,Cc1cn2cc(C(N3CC(NC(=O)COCCc4cccs4)C4CC34)=O)sc2n1 63678,c1(C(N2CCN(C(C3(O)C(C)(C)C3)=O)CC2)=O)ccnc2[nH]c(O)nc12 63679,c1(C(N2C(CN(C)C(c3ccns3)=O)COCC2)=O)cc2n(n1)CCC2 63680,N1(C(C2C(=O)NCC2)=O)CCC(C(=O)NCC23CC4CC2C3C4)(CF)C1 63681,C(C)(CC(=O)NCC(CO)NC(c1ccc(CC2CC2)cc1)=O)(C(F)F)N(C)C 63682,C(=O)(CC(C)CC(C)(C)C)NCCC1N(C(c2sc(C)c(O)n2)=O)CCSC1 63683,c1(CC)cc(N)ccc1C(=O)NC1CC2CC1N(C(=O)CCOCCOC)C2 63684,N1(C(C(CCCC)N2CCCCC2)=O)CCC(C)N(C(c2cnsc2)=O)CC1 63685,C1(NC(c2cc(-c3nc(C)sc3)sc2)=O)CCC(NC(C2(C)CCCS2)=O)CC1 63686,C1(NC(C2CCCC(O)C2)=O)CN(C(=O)COC2COC2)CC2(CCC2)C1 63687,c1(NC(C(=O)NC(COCC)CO)=O)ccc(C)c(O)c1 63688,C#Cc1cccc(OCC(=O)NC(CNC(=O)CCc2nccs2)CC(C)C)c1 63689,C(=O)(C#CC1CCOCC1)NC1CCC(NC(C2CCc3nnnn3CC2)=O)C1 63690,c1(C(N2CC3(C(NC(c4cn5c(n4)CCC5)=O)CC3)C2)=O)c(F)ccc(F)c1Cl 63691,C1(CC(=O)NCC(C)Cc2ccncc2)CCN(C(=O)CCC2CCCO2)C1(C)C 63692,C(C(C(=O)NCC(F)(F)F)N1CCC(OC)CC1)(C1COC1)OCC.C1CCC1 63693,c1(C(C)C)nc(NCCCCSC(C)(C)C)cc(=NCCn2ccnn2)[nH]1 63694,c1(CC(=O)NCC2N(C(C3C(C)C3C)=O)CC=C2)ccc2[nH]ccc2c1 63695,C#CCC(CC(=O)NC1CCC(C)(CC)CC1)NC(=O)CNC(C1CC1C)=O 63696,N1(C(CCC2(NC(c3c(CC)cco3)=O)CCCC2)=O)CCCC1(C)COC 63697,C1(CNC(c2nc(C)n(C)c2)=O)COCCN(C(C2CC2(C)C(F)F)=O)C1 63698,C1(CC(=O)Nc2ccnc(C(C)(C)C)n2)CCCNC(=O)C1.C1CCN1CCO 63699,c1(C(C(=O)NCC=C)NC)ccc(OC)nn1.C12CC(C1)OC2=O.CCC 63700,C1(C(N2CCN(CC(C)O)CC2)=O)(OC)CCN(C(=O)Cc2cccn2C)C1 63701,N1(C(C(CN(C)C)N(C)C)=O)CC(c2cn(C3CCCC3(C)O)nn2)CC1(C)C 63702,C1(N(C(c2cc(CC)no2)=O)CC2CC2)CCN(C(C23CCCCC2C3)=O)CC1 63703,c1(C(=O)NCC(C)CN(c2cnc(C#N)cn2)C)ccc(-c2cccs2)cc1F 63704,N1(C(C(=O)NCC)C)CC(CNCCN(C)C)(OC(C)(C)C)C1 63705,N1(C(C=C(CC)C)=O)CCC2CCC12CNC(c1ccnn1C)=O 63706,C1(NC(C(CC)O)=O)CC=C(C(=O)N2CC(n3cnnn3)C2)C1 63707,c1(C(=O)NC2CN(C(C3(OC)CC(C(F)(F)F)C3)=O)C2)cccc(Cl)c1 63708,c1(C(N2CC3(CC3C(N3CCn4nccc4C3)=O)C2)=O)cccc2occc12 63709,CCC(F)(F)CC(=O)NC1CN(C(=O)C=CCF)CC1C(F)F 63710,N1(C(C(CCC)CNC(c2cc(CO)on2)=O)=O)CCOCC(F)(F)C1 63711,C=CC(CC)CC(=O)N1C2CCC1C(NC(=O)CS(C)(=O)=O)C2 63712,C1(NC(C(COC)N(C)C)=O)(COC)CCN(C(c2nc(C)nn2C)=O)C1 63713,N#Cc1nc(Br)cnc1NC(C1(C(F)(F)F)CCC1)=O 63714,Cc1ccc(F)cc1CC(=O)NCC(C(C)C)NC(C1(C#N)CC12CCC2)=O 63715,CC1CCN(C(=O)COC(C)(C)C)CC1CNC(c1ccc(F)c(Cl)n1)=O 63716,c1(C(=O)NC(CN(C(CN(CC)CC)=O)C)C)cc2c(s1)CC(C)(C)C2 63717,C1(C(=O)NC2C(NC(c3ccoc3)=O)COC2)CCCOC1c1ccncc1 63718,c1(C(=O)NC2CN(C(C3C(CC)OCCC3)=O)C2)ccn2cc(C)nc2c1 63719,c12ccc(cc1)N(C(=O)C1CC1)N2C.c1(CC)ccccc1OCOC.C1CCN1 63720,c1(C(=O)NC2CCCC(NC(c3c(C)ccnc3)=O)C2)c(C)cccc1F 63721,c1(C(N(CCOC)CCNC(=O)CCCCF)=O)cc2c(s1)CCC(C)C2 63722,N1(C(CCOC)=O)CCN(CC2CCN(C(=O)CCC3C(=O)ON=C3C)C2)CC1 63723,c1(C(N2CC(SC)C(NC(=O)Cc3cccn3C)C2)=O)n[nH]c2ccc(Cl)cc12 63724,C(=O)(C1=CCS(=O)(=O)C1)N1CCCC(N(C(CN2CC(CC)C2)=O)CC)CC1 63725,c1(CC)nc2n(n1)CC(NC(=O)Nc1cccc(C(F)F)n1)CC2 63726,C(=O)(CC(C(C)C)c1ccccc1)N(CCCNC(c1[nH]cc(C)c1)=O)C 63727,N1(C(CN2CCC(OC)C2)=O)CC=C(C(=O)N2CC(CS(C)=O)C2)C1 63728,C1(C2(O)CCOCC2)(C(N2C(CNC(C3(C)CC=C(C)CC3)=O)CCC2)=O)CC1 63729,C12(C(=O)NCC3N(C(=O)CC4CC4)CC=C3)CC3CC(C1)CC(O)(C3)C2 63730,c1(C(=O)NC(C2(O)CCN(C(=O)C3=CSCS3)C2)C)cn2cc(F)ccc2n1 63731,Cc1nc(-c2ccccc2)[nH]c1C(=O)N(CCCNC(c1ccsc1)=O)CCO 63732,c1(C(N(CCOC)CCNC(=O)C(C)SC(F)(F)F)=O)ccoc1Cl 63733,C(=O)(C1=CC2C=CC(C1)C2)N1C(C(=O)Nc2cccc(C(C)F)c2)CC1 63734,C(=O)(CC1COc2cc(O)ccc21)N(CC(C)NC(=O)CCC(=O)NN(C)C)C 63735,C1(C)(NC(C(CC=C)NC(c2cc3occc3[nH]2)=O)=O)C(C)(C)C1(C)C 63736,N1(C(c2ccc(OC)s2)=O)CCC2C(NC(C3CCCCC3C)=O)CCC12 63737,c1(C(N2CC(CCO)(NC(CNC(C)=O)=O)C2)=O)ccn2cnnc2c1 63738,N#CC1(C(=O)NC2(CO)CCN(C(=O)CCCc3ccccn3)C2)CCOCC1 63739,c1(NCC=CS(C)(=O)=O)ccc(O)c(CO)c1 63740,N1(C(Cc2ccn(C(C)C)n2)=O)CCN2C(=O)C(NC(c3cnn[nH]3)=O)CC2C1 63741,C1(C(=O)NCC(CC)(C)NC(c2csc(=N)[nH]2)=O)CC2CCC1O2 63742,C=CC(CC)CC(=O)NCCC1CC(OC)CN1C(=O)Cc1cc[nH]c1 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63899,C1(CC(C)(C)C)CN(C(=O)CSC2CCCO2)CC1NC(c1cn[nH]c1)=O 63900,Cc1cc(C(=O)NC2C3CCN(C(=O)Cc4ccc(O)c(C)c4)C23)ccc1F 63901,N1(C(c2c(CC)n(C)nn2)=O)CCCCC(CNC(=O)C(=O)NCC2CC2)C1 63902,N1(C(C(CC)NC(N)=O)=O)CCC12CN(C(=O)CC1CCCOC1)C2 63903,C1(C(CCC)C)Cc2ccccc2CN1CC(=O)Nc1cnc2c(c1)ncn2C 63904,C1(C(=O)N(c2cccc(Cn3ccnc3)c2)CCl)Cc2cc(C(F)(F)F)ccc2O1 63905,c1(C(=O)NCC2(NC(c3n(C)ncn3)=O)CCCCC2)cccc(S(N)(=O)=O)c1 63906,C1(CNC(C2C(OC)CCC2)=O)CN2CCC1C1CN(C(=O)OC(C)(C)C)CC21 63907,c1(C(=O)NCC2(OC)CCN(C(=O)CCCC3CC3)C2)ccn2c(O)nnc2c1 63908,C1(N(C(c2csc(-c3cccs3)c2)C(=O)NC2CCC2)C)CCN(CCO)CC1 63909,C(CNC(=O)CCCSC)(CC(F)(F)F)NC(c1ccc(OC(CC)C)cc1)=O 63910,C1(C(=O)NC(C)CN(C(=O)Cc2nc[nH]n2)C)CN2CCCCC2CO1 63911,Cc1cccc(C(=O)NC2(C)CCN(C(C3CCCCC3C(F)(F)F)=O)C2)c1N 63912,C=CCCCC(C(=O)NCc1ccncc1CC)NC(=O)C(CC)N(C)C 63913,c1(NC)scnc1C(=O)NC(COC)C(=O)NCCCc1cccnc1 63914,C1(CNC(=O)C(=O)C2CC2)CCCCN1C(c1ccccc1N1CCCCC1)=O 63915,C(=O)(C(CC(C)C)NC(=O)C(C)CCOC)N(CC(CCC=C)O)C 63916,C1(NC(=O)CCc2cc(Cl)cs2)CC2(C1)CC2NC(c1cc(C2CC2)[nH]n1)=O 63917,C12(CNC(C=CCCC)=O)CN(C(=O)C=Cc3ccc(C)s3)CC(F)(C1)C2 63918,C1(S(N)(=O)=O)(C(=O)NC2CC(NC(c3cnn(C)c3C(C)(F)F)=O)C2)CCCC1 63919,N1(C(CS(CCCC)(=O)=O)=O)CC(C2CCCCN(C(c3cc(C)sn3)=O)C2)C1 63920,c1(C(=O)NC(CC)CNC(c2ccc(C)cc2F)=O)cccc2cccc(Cl)c12 63921,c1(NC(CCNC)(C)C)nc2cc[nH]c2c(=NC(C)c2ncccc2F)[nH]1 63922,c1(CC)cc(Br)ccc1C(=O)NC1CC(NC(c2csc(C3CC3)n2)=O)C1 63923,N1(C(C(C)CC2CCC2)=O)CC2CCC1CN2C(c1noc2c1COCC2)=O 63924,C1(NC(CC(C)c2cccnc2)=O)CC12CCN(C(=O)C(C)(C)CCC#N)CC2 63925,C(=O)(CC1C(=O)Nc2c(F)cccc21)NCCC1CN(C(C(CC)C)=O)C1 63926,C1(CC)CN(C(C2CCC(C)O2)=O)CCN1C(c1ncnn1CC)=O 63927,C(=O)(CCCCC(=O)NC(C)(C)CCCC(=O)NCCC1CC(=O)NC1=O)OC 63928,C(=O)(C(C)(CC)C(=O)N(C)CCNC(=O)C(C(C)C)OCC1CC1)OCC 63929,N1(C(CC2C(C)=NOC2=O)=O)CC(NC(c2n[nH]cc2Cl)=O)C2CCCCC12 63930,C(CCCCC(=O)NCc1ccc(CNC(c2cc(C)ccc2F)=O)cc1)SC 63931,c1(OC)cc(SCC(N2CC(CNC(C3CCC(C)(C)CO3)=O)C2)=O)cc(F)c1 63932,CC(Cc1ccc(Cl)cc1)CC(=O)NC(C)(CNC(=O)C=Cc1nccs1)CO 63933,CC(CCC(C)(C)C)C(=O)N1CCN(CCN(C)C(c2cc(Cl)ccn2)=O)CC1 63934,c1(C(N2CC3C(CN(C)C(C4(N(C)C)CCC4)=O)C3C2)=O)ccn(C)c(=O)c1 63935,CC1CCCC(CNC(c2cc(CNC(c3cc(Cl)n[nH]3)=O)nn2C)=O)CC1 63936,C1(C(=O)NCC(=C)F)CSCCN1C(=O)C(O)C1CCC1 63937,N1(C(Cc2cc(C)sc2)=O)CC=C(C(C)(C)C(=O)N2CCCCC2C(C)CO)C1 63938,c1(CC)ccc(C(=O)N(CCCn2cc(C3(F)COC3)nn2)C(C)C)c(Br)c1 63939,N1(C(c2ccc(OC)o2)=O)CCCC(C2CCCCN2C(C2CCCOC2)=O)C1 63940,CC1(C)C(NC(=O)CCOc2cccc(F)c2)CC1NC(=O)CCC1CCCO1 63941,CCCC(F)F.C(=O)(C(C)n1cccn1)N(CCC)CC 63942,c1(C(=O)NC(C(=O)NCc2cc(C)c(C)s2)COC(C)C)ccc(F)c(F)c1 63943,C(=O)(C(CC(C)(C)C)NC(c1ccc(F)cn1)=O)N(CCCCCC=C)C 63944,N1(S(CC)(=O)=O)CCOCC(C(=O)NC(C)CNC2(O)CCCCC2)C1 63945,Cc1nn(C)cc1CCC(=O)NCC(C1CC1)NC(=O)C(=CC1CCCCC1)F 63946,C12(NC(c3cc(O)ncn3)=O)COC(C1)C(NC(c1scnc1Cl)=O)C2 63947,N1(C(CCC(=O)NC(C)C)=O)CC2CCCC2(NCC2CN(C3CCOC3)C2)C1 63948,C1(C)(CC)CCC(C(=O)NC2C=CCN(C(=O)C=CCN(C)C)C2)O1 63949,C(=O)(C(C(F)(F)F)C(F)(F)F)NC(CNC(c1cn(C)nc1C1CC1)=O)C1CC1 63950,C1(CNC(C2N(C(N)=O)CC(O)C2)=O)CC2CCC1N(C(=O)Cc1ccon1)C2 63951,C#CCCCCCNC(=O)CC1(C=C)CN(C(c2cc(CO)ccn2)=O)C1 63952,c1(C(=O)NCC(C(C)C)NC(C2CCO2)=O)cnc(N)cn1 63953,c1(C(=O)NCCN(C2CCCC2)C(=O)C=CC2CC2)ccc2c(c1)C(=O)CCN2 63954,N1(C2(C)CC2)CC(C(N2CCCC2CNC(c2ccnnc2O)=O)=O)CC1=O 63955,C(CC(CC)CC)(n1nnnc1)Nc1cccc(-n2nc(C)cc2C)c1.C=CC 63956,c1(C(=O)NCC2C(NC(CNC(CC)=O)=O)CCCC2)ncc2[nH]ncc2n1 63957,N1(C(C(CC)SC)=O)CCC(CN(C(=O)Cc2cc(CC3CC3)nn2C)C)CC1 63958,C12(NC(COCC#C)=O)CC3CCC(C1C2)N3C(c1cccc(C)c1F)=O 63959,Cc1cccc2c(CN3CCC(NC(c4ccc(I)cc4O)=O)C(F)C3)c[nH]c12 63960,C(c1nc(C)c(C)[nH]1)=CC(N1CCC(n2cc(CSCC)nn2)C1)=O 63961,C1(CNC(c2ncncc2Cl)=O)C2CCC(C2)N1C(C12CC3CC1C2C3O)=O 63962,Cc1cc(=NCC(C)C2CC2)[nH]c(N2CCN(CC(F)F)CC2)n1 63963,CCCC(CCC)C(=O)NC1CCCC(NC(c2cc(CCCO)on2)=O)C1 63964,CC1CCCCC1(C)C(=O)NCCOCCN(C)C(=O)COc1cncc(Cl)n1 63965,c1(C(=O)NCC2OCCCN(C(C3(C)COC3)=O)C2)ncnc2c1CCCC2 63966,C1(C(=O)NCC(CC)CCO)CN(C(C2CN(C3CCC3)C2)=O)CC1(C)C 63967,N#Cc1cc(C(N2CCC2CNC(C2CC3(CSC3)C2)=O)=O)c2ccccc2c1 63968,c1(N2CC3CN(C(c4cc(C)nc(C)c4)=O)C3C2)ncnc2n[nH]cc12 63969,c1(OC)cccc(CN2CCCC(CNC(=O)C=Cc3ccoc3)C2)c1C 63970,Nc1c(F)cc(SCCC(=O)Nc2n[nH]c3ccccc23)cc1F 63971,c1(NC(C2(CNC(c3ccc(C(N)=O)nc3)=O)CC2)=O)ncc(Cl)nc1Br 63972,C1(NC(c2cc(CC)[nH]n2)=O)CCN(C(c2cc(C)ccc2N)=O)C(C2CC2)C1 63973,c1(C(N2C(C(N3CC(c4cc(C)no4)C3)=O)CCCC2)=O)c(F)cc(F)cc1Br 63974,c1(C(=O)Nc2c(C)nccc2)c[nH]c2cc(-c3ccsc3C)cnc12 63975,c1(CC(=O)NCC(CC=C)NC(c2cc(Cl)no2)=O)cn2ccsc2n1 63976,c1(C(N2CCC(N(C(CN(CC)CC)=O)C)C2)=O)nnc(O)c(Br)c1O 63977,C(=O)(C1c2ccccc2C2CC1C2)N(C1CCOC1(C)C)C 63978,C1(C(=O)NC2(C)CN(C(C(c3cscn3)N(C)C)=O)C2)CC2CCC(C1)C2(F)F 63979,c1(C(=O)NCC(CC=C)NC(=O)CC)cnc2cccc(C)n12 63980,n1(CC)ccc(CC(=O)NCC(CNC(C2CC=CCC2)=O)OC)n1 63981,N1(C(C(C=C)C)=O)CCN(C(C)CNC(c2cn(C)nn2)=O)CC1 63982,Cc1cnn(C)c1CC(=O)NCC1CCC(NC(c2ccc(N(C)C)nn2)=O)C1 63983,c1(C(=O)NC2(CCNC(C(C(C)(C)C)SC)=O)CCCC2)cc(C)c(N)cc1Cl 63984,c1(NCCC2CCN(C(C(CC)(F)F)=O)C2)ncnc2sc3c(c12)CCC3 63985,N1(C(C2CCC(CNC(CC3(SC)CC3)=O)C2)=O)CCCNC(=O)C12CC2 63986,c1(NC(C2(C)CCN(Cc3nccc(C(=O)OC)c3)C2)=O)cc(Cl)c(Cl)cc1O 63987,c1(C(=O)NCC(CCCC)NC(C23CCCC2CCC3)=O)cc(C#N)ccc1F 63988,C(=O)(C(COC)COC)N1C(CC(=O)NC2(COC)CCCC2)CCC1 63989,C1(C(N(C2CN(C(C3CCN(C(C)=O)C3)=O)C2)C)=O)CCCCN1C(=O)C(C)C 63990,C1(C(C)NC(CN(C2CC2)CC)=O)CCCCN1C(=O)CC1CCOC1(C)C 63991,N1(C(C(CSC)OC)=O)CCC2(CCC(NC(c3[nH]c(O)nc3C)=O)CC2)CC1 63992,C(CCCCN(C(=O)C(C)NC(=O)Nc1ccccc1)C)NC(C=CCC)=O 63993,Cc1nn(C)c(C)c1CCC(=O)NC1CCC(F)(CNC(C23COCC2C3)=O)C1 63994,c1(COC)nc(NCCc2cnn(C(C)(C)C)c2)cc(=NC(C)C2CCCO2)[nH]1 63995,C(=O)(CC1=CCCCC1)NCCOC(C)(C)CNC(=O)CCNC(C1CCC1)=O 63996,C1(NC(c2cc3c([nH]2)CCCC3)=O)CCN(C(C2(O)COC2)=O)CC12CCC2 63997,C1(NC(COC(CCC)C)=O)CC2CCC(C1C)N2C(c1cnn(CCO)c1)=O 63998,C(N=c1[nH]c2ccc(F)cc2o1)C1C(C)CN(C(c2occ3c2CCOC3)=O)C1 63999,CCC(CC(=O)NCC1C=CCN1C(c1cc(OC)cs1)=O)C(C)C 64000,Cc1nc(C(=O)NCCCC2CCCCN2C(=O)Cn2nnc(=O)[nH]2)c(C)s1 64001,C1(C(N2CCC(NC(C3CCOCC3)=O)C2)=O)(OCC)CCOCC1 64002,CCC(F)(F)C(C)(C)NC(C1CCC(C2CC2)N1C(=O)CCC1(C#N)CCC1)=O 64003,c1(C(=O)NC2C(NC(c3cc(C)c(C)s3)=O)CCOC2)ccc2ncccc2c1 64004,Cc1cncc(C(=O)NCCC2(C)CCN(C(=O)C(O)P(C)(C)=O)C2)c1C 64005,c1(C(=O)NCCC(C)(C)NC(C2C(C)OCC2)=O)ccc(C(F)(F)F)cn1 64006,CC1(C)CCCN(C(=O)Cc2n[nH]cc2Br)C1CNC(c1scnc1Cl)=O 64007,CCC(CN(C)C)CC(=O)N1CCC(OCCNC(=O)Cc2ccoc2C)C1 64008,c1(C(CNC(C2CC2F)=O)NC(C2CCCC(CF)C2)=O)ccc2ccccc2c1 64009,C1(NC(C2CN(C(C)=O)C2)=O)CCC2CCN(C(c3csnc3C)=O)C1C2 64010,N1(C(C(C)CN(C(=O)C(c2ccccc2)C2CC2)C)=O)CCCCC(SC)C1 64011,N1(C(Cc2c(CC)cccc2)=O)CC2(CCCC2)C1C(=O)NCCC(O)COC 64012,C(C1CN(C(C2(C)CCCC2O)=O)CC1C(=O)NCC(C1CCCC1)OC)=CC 64013,C(=O)(C(C)(C)COCCN(C)C(C1CC(N(C)C)C1)=O)NC(C=C)CO 64014,C1(NC(CCOCCCOC)=O)CCN(C(c2cnn(C)c2N)=O)CC1C 64015,N1(C(C)=O)CC2(C1)CN(C(C1CSCN1C(C1CCOC(=O)CC1)=O)=O)C2 64016,C1(NC(C=CC)=O)CC2CN(C(=O)CCc3c(C)nn(C)c3C)CCN2C1=O 64017,N1(C(Cc2nnc(C)o2)=O)CC2(CO)CC1(C(=O)NCCSC(C)C)C2 64018,C1(F)(CNC(C2N(C)CCC2)=O)CCN(C(c2ccc(-c3ccncc3)o2)=O)C1 64019,C1(CNC(=O)CC2CCC3CC3C2)CC2COCC2N1C(c1ccc(F)s1)=O 64020,c1(C(N2CC(C(C)NC(=O)CC(O)C3CC3)OCC2)=O)ccc2nc(O)[nH]c2c1 64021,N1(C(C)C)CCCCC1C(=O)NCCCN(C(=O)C(C1CCOCC1)C)C 64022,C(=O)(C(F)C(C)(F)F)NCC1(C(N2C(C)(CC)CC2)=O)CCCC1 64023,N1(C(c2cc(C)oc2C)=O)CCCOC(CNC(=O)Cc2cocn2)C1 64024,C(=O)(CC1=CCCCC1)N1C(CCNC(CCC(=O)N(C(C)C)C)=O)CSCC1 64025,CCC(CC)C(O)CNC(=O)C(C1(O)CN(C(c2ccn(C)c2C2CC2)=O)C1)F 64026,C12(NC(CC3CCC(=O)N3)=O)CCCC1CN(C(c1c(O)cc(Cl)cc1F)=O)C2 64027,Cc1cc(C=CC(=O)NCC(O)CN(C(=O)C(C)c2ccsc2)C)c[nH]c1=N 64028,C(=O)(C(O)CCNC(=O)Cn1cnnc1O)NC1CC(C=C)C1 64029,c1(C(=O)NC(CN(C(C2(OC)CCCCC2)=O)C)C)ccccc1CC(C)(C)C 64030,N1(C(C(C)(C)F)=O)CCCC1C=CC(=O)NC(C(N)=O)C1CCCC1 64031,N1(C(C(CC2CCC2)NC(c2c(C)oc(CO)c2)=O)=O)CCCC(C)C1C(C)C 64032,c1(C(C)NC(N(C(C(=O)NCCOCCC=C)C)CC)=O)cc(Cl)ccn1 64033,c1(Cn2ncc(NC(C3(c4ccccc4)CCC3)=O)c2)cc(Br)cc2[nH]ncc12 64034,C(=O)(CC(CC)C(C)C)N1CCN(C(CCC=CC)=O)C(CCOC)C1 64035,N(C1CC(C)n2ncnc21)CC(C)N(C(=O)CCc1ccccc1)C 64036,C(CCCC(=O)NC1CCCC1NC(=O)Cc1ccc(C)s1)OC 64037,c1(C(C)C)nc(NC(=O)C(CC)NC(=O)NCC(F)(F)F)cc(Cl)n1 64038,CN1C(=O)OCC1C(=O)NCC12CC1CN(C(=O)CC1CC1C(F)(F)F)C2 64039,C(C(CNC(=O)C1=CCCC1)C(F)(F)F)NC(c1c(CC)oc(C)c1)=O 64040,C(c1cocn1)=CC(=O)NC1(CC(=O)N(CCOC)C)CCC1.C1(C)CC1 64041,c1(CC)cc(C(=O)NCC(=C2CN(C(c3cnn(C)n3)=O)C2)F)c2c(c1)CCO2 64042,c1(N(CC(N2CC(N(C)C(C3CC3F)=O)C2)=O)C)ccccc1 64043,c1(C(=O)NC2C(C(C)(C)C)N(C(=O)C(C)NC=O)CC2)nnn2c1CCCC2 64044,C(N=c1[nH]c2ccc(N)cc2s1)C1CCCCN(C(c2nn(CC)c(C)c2)=O)C1 64045,c12cc(C)c(cn1)C(=O)N(CCOC)CCNC(=O)C(C1CCC1)O2.O(C)OC.S.CC 64046,c1(OC)c(Br)cc(CN2C(C(=O)NCCc3ccc(I)cc3)CC3CC23)cc1Br 64047,C(C(C(C)C)NC(=O)C(C#N)=C1CCC1)NC(C=CCOCCOC)=O 64048,CC(C)(C(=O)NCC1CCC(NC(=O)CN2CCCC2=O)C1)c1cc[nH]n1 64049,c1(N2CCCCC(CC3CC(C)NC3)C2)ncnc2c(F)cc(F)cc12 64050,c1(C(N2CCCC(C(C)NC(c3cc(C)sn3)=O)C2)=O)n[nH]c2cc(Cl)ccc12 64051,Cc1cnn(CCC(N2C(C=O)CC2C)=O)c1.N1(C(CNC(C)C)=O)CCCC1 64052,C1(CNC(CC=C)=O)CC(C(=O)N2CC(O)(C3CC3)C2)=NO1 64053,C1(CNC(c2cc(CC)oc2C)=O)CN(C(=O)COCC(C)C)CC2(CCC2)O1 64054,CC1(C)CCN(C(c2csnc2Cl)=O)C1CNC(c1cc(C2CCCC2)no1)=O 64055,c1(CC(C(=O)N(CCNC(C2(C)CCCO2)=O)CC)O)cccc(C(F)(F)F)c1 64056,C1(NC(c2nc(C)oc2C)=O)CCN(C(=O)C(C)Cc2cnn(C)c2)CC1F 64057,CCC(CC(=O)N1CC2CCCC2(NC(=O)COC(C)(C)C(F)(F)F)C1)C(C)(C)C 64058,C(CO)(CCCCNC(c1cnn[nH]1)=O)NC(=O)Cc1cc(Br)cs1 64059,c1(C(=O)Nc2ccc(O)c(F)c2)cn2c(n1)CN(Cc1cc(I)cnc1Cl)CC2 64060,Cn1cc(C#CCN=C(NCC2CCSC2)NC(C2CC2)C2CC2)cn1 64061,C1(NC(C(CC)N(C)C)=O)CN(C(=O)OC(C)(C)C)CC1C 64062,C12(NC(CCCC3C(C)C3)=O)CCOC(CNC(=O)Cn3cc(Br)cn3)(C1)C2 64063,c1(C(=O)NC(C(C)(C)C)CNC(C2CC3CC3C2)=O)cc(F)cc(Cl)c1O 64064,C1(C(N(C2CCN(C3CC3)C2)C)=O)(NC(=O)COc2ccccc2)CCCC1 64065,C1(N(C(C(C)N(C(c2cn(CC)cn2)=O)CC)=O)C)CCCCC1C 64066,C(=O)(CCC(C(=O)N1CC(C)N(C(=O)C=CSC)CC1)N(C)C)OC 64067,N1(C(C2(NC(C3C(CC)C3)=O)CCN(C)C2)=O)CC(OC)C2(CC2)C1 64068,O=C1NCC2(CCCN(C(c3ccnc4ccccc34)=O)C2)O1 64069,C1(NC(c2cccc(O)c2)=O)CCN(C(=O)C(F)(F)C2CCCC2)CC1CO 64070,c1(C(C(=O)NC)N(CC(C)C)C2CC2)ccc(C#N)c(Cl)c1 64071,C1(C(N2CCC(NC(C(CCC)CC)=O)C2C)=O)Cc2ccncc2N1 64072,C1(C(N(CCNC(C2CC2F)=O)CC)=O)CC2C=CC1CCC2 64073,Cc1[nH]c(C(=O)NCCC2CN(C(CC(F)(F)F)=O)CCO2)c(C)c1C(=O)O 64074,C#CC(CC)(CC)NC(=O)C(CC=C)NC(c1nnsc1C)=O 64075,C12(C(=O)NC(CN(C(C3=NOC(C)C3C)=O)C)C)CC(C)(C1)OC21CCC1 64076,c12nc(cc(N(C)CC3CCCSCC3)n1)N2.C(CC(=O)N(C)C)OC(C)C 64077,C(N=c1[nH]c(=NC(CCO)C(F)F)[nH]c2c1CSC2)C1(OC)CCCC1 64078,N1(C(C(C)NC(C)=O)=O)CCN(C(c2sc(C(F)(F)F)nc2C)=O)C(C)C1C 64079,N1(C(C(CC)n2cncn2)=O)CCN(C(CNC(C2CC2C)=O)C(F)(F)F)CC1 64080,C1(CC(=O)NCC2CCCC2NC(c2cc(F)c[nH]2)=O)CC2(CCC2)CCO1 64081,c1(CSCC(=O)NCCCNC(C(C)CO)=O)nc(=O)c2ccccc2n1C 64082,C(C(C)(CNC(=O)CCn1cc(C)cn1)OC)NC(C(C)OCC=C)=O 64083,C1(COC(C2(SC)CC2)=O)COCC2(CCN(C(=O)OC(C)(C)C)C2)O1 64084,C(=O)(C(F)CCC(C)(C)C)NC(C)CCCNC(c1cccnc1O)=O 64085,c1(C(=O)NC2CC3(CNC(c4c(C)ncs4)=O)C2C3)cccn2cnnc12 64086,CCC(CC(C)C)C(=O)N1CC2C(CC(=O)NCC3CC3CC)C2C1 64087,C12(C(N(C)CC3CC(F)CN3C(=O)CCC34CCC(CC3)C4)=O)CCN(CC1)C2 64088,N1(C(CC(C)(C)CC(F)F)=O)CC2CCN(C(c3ncccc3Cl)=O)CCC2C1 64089,N1(S(CCC)(=O)=O)CC(CC)CC(CNC(=O)CCOc2cc(C)cc(C)c2)C1 64090,C(=O)(C1=NOC2(CCC2)C1)Nc1c(C(=O)OCC)ncc(Cl)n1 64091,C12CN(CC1C)C(=O)c1cn2nn1.c1(CN(C(C)=O)C)sccc1C 64092,c1(NC(CNC(CC(CCC)C)=O)C)ncccc1[N+](=O)[O-] 64093,c1(CC)onc(C)c1C(N1CCCCC1CN(C(=O)CCN(C)CC)C)=O 64094,C(=O)(CC(F)(F)CC(=O)OC)NC1CN(C(CCOCCOCC)=O)C2C1C2 64095,Cc1ccc(C)n1CC(=O)Nc1cc(C(=O)NCC2CN(C)CCO2)n(C)c1 64096,CN=C(NCC1CCCN(C(=O)OC)C1)N1CCS(=O)(=O)CC1 64097,c1(NC(C2N(CC34OCC(C)C(C3)C4)CCCC2)=O)ccc([N+](=O)[O-])cc1Cl 64098,c1(Nc2c(C)cncc2)cc(S(=O)(=O)N2CC(C3CCCCC3)C2)ccc1C#N 64099,C1(NC(c2nc(COC)sc2)=O)CCN(C(=O)CCNC(N)=O)CC(C)(C)C1 64100,C(C)(c1cccnc1)=CC(=O)NCC1(O)CC(NC(CCCC#C)=O)C1 64101,c1(COC)ccnc(C(N2CC3(NC(C4CC4C)=O)CC2C3)=O)c1 64102,CN=c1nc(N(CC(=O)NCC(C)C)C)[nH]c(=NCc2ccc(Cl)c(F)c2F)[nH]1 64103,c1(C(=O)NCCC2(CNC(c3nc(OCC)oc3)=O)CC2)cnn(C)c1C(F)(F)F 64104,c1(OC)ccc2c(c1)CCCC2N(C(c1cnn(C2CCOCC2)c1)=O)C(N)=O 64105,C1(NC(CC)=O)CN(C(c2ccc(NC)cc2)=O)Cc2nccn2C1 64106,N1(C(c2nc(OCC)oc2)=O)CC2CCCC2(CNC(=O)CC(C)(O)CCC)C1 64107,C1(C(=O)NCC2CCC(NC(C3C(C)(C)C3)=O)C2)CCCC(O)C1 64108,c1(C(N2CCCC(COC)C2)=O)cnc(O)cc1OC.c12cc([nH]n1)C(=O)N2C 64109,c1(C(N(CC(=O)N(CC=C)CCOC)CC2CC2)=O)cc(O)ccc1C 64110,c1(C(=O)NCC2C=CCN2Cc2cc(Br)c[nH]2)cccnc1N1CCCC1 64111,C1(NC(Cc2nc(C)sc2)=O)CN(C(C2CCC=CCC2)=O)C2(CCOCC2)C1 64112,N1(C(C(COCCO)NC(C)=O)=O)CCOCC(C)(NC(c2ccc(C)nn2)=O)C1 64113,c1(C(C2C(C=C)CN(S(C)(=O)=O)C2)c2nnnn2CCCF)cccc2cncn12 64114,N1(C(C(OC)OC)=O)CCOCC(NC(c2cnnc(C)c2)=O)C1 64115,C1(OC)CC(C(N2C(C(=O)OC)CC2C)=O)N(C(=O)CCC2CCCOC2)C1 64116,C1(C)(C(=O)NC(C(C)C)CNC(C2(F)CC2C)=O)CCS(=O)(=O)CC1 64117,c1(C(=O)NC(CC)CN(C(=O)CN(C)C(C)C)C)ccc(F)c(OC)c1F 64118,N1(C(c2c(C)con2)=O)CC2CCC(NC(=O)Cc3cccc(F)c3)C2C1 64119,c1(C(C)=O)cc(C(=O)NC2CC(NC(=O)CCOC(C)CC(C)C)C2)n[nH]1.C1CO1 64120,c1(OC(C(=O)NC)C)ccc(C)cc1OC.C(C=O)NC(=O)NC.C12(CC1)CC2 64121,c1(NCCC2CCC(NC(CCC(=C)C)=O)C2)ncnc2c1COC2 64122,CC(=O)CCCC(=O)NCC1(O)CCN(C(=O)C(C)OC2CCCCCC2)CC1 64123,C1(O)(C(=O)NC2C(CC(C)(C)C)C2)CCN(C(=O)CSC(F)F)CC1 64124,N1(C(CCN(C(=O)CC(Cl)Cl)C(C)C)=O)CCC(C)C(O)C1 64125,CC(C)C(C(=O)NC(C)CC(C)NC(c1cccnc1C(F)F)=O)NC(N)=O 64126,N1(C(C(C=C)(F)F)=O)CCCCCC(NC(c2oc(CC)cc2C)=O)C1 64127,N1(C(C2CC(C)NC(=O)C2)=O)CCC2(CC1)CCN(C(=O)CC1OCCO1)C2 64128,CC(CC(=O)N(CCCN(C)C(C1(Cc2ccccc2)CC1)=O)C)C(F)F 64129,N1(C(c2c(CNC(C(C)OC3CCCC3)=O)n[nH]c2)=O)CCC(C2CC2)C1 64130,C1(CC(=O)NC(CC)CN2CCCC2)CC(F)CN1C(c1cnc(NC)s1)=O 64131,C1(C(=O)Nc2c[nH]nc2C2CC2)CC(=O)N(C2CN(CC3CCCCS3)C2)C1 64132,N1(C(C(CC2CCCC2)NC(c2c(CC)[nH]cc2)=O)=O)C2CCC1CC2 64133,N1(C(c2csc(O)n2)=O)CCC2CCN(C(c3nc[nH]c3C(F)(F)F)=O)CC2C1 64134,N1(C(C(CC)NC(C)=O)=O)CC(O)CC1C(=O)Nc1ccsc1 64135,C=CCC(C)(C)CC(=O)NC(c1ccc(F)cc1)CNC(=O)Cc1nccn1C 64136,c1(C(N2C(C)COC(CC(=O)O)C2)=O)cc(Cl)c2ccc(Br)nc2c1 64137,c1(OC)ncccc1CN1CC(F)CC1C(=O)NCC(c1cccc(Br)c1)O 64138,C1(CNC(C(=O)NCC)=O)CN(C(=O)CCC2C(=O)ON=C2C)C2(CCC2)C1 64139,c1(C(N2CCCC(F)C2)C(=O)N(c2cn(C)nc2)C2CCCC2)ccc2nsnc2c1 64140,c1(OC)ccc(CC(=O)NCC(C(C)(C)C)NC(C2(F)CC2C)=O)cc1[N+](=O)[O-] 64141,Cc1cccc(C=CC(=O)N(C2CCN(C(c3cnc(C(C)(F)F)s3)=O)C2)C)c1 64142,c1(C2C(=O)N2C(C)(C)C)ccoc1C.C(CCSC(C)(C)C)OC 64143,CS(=O)(=O)c1cnn(CC(N2CC(OCCNC(C3CC3C(F)(F)F)=O)C2)=O)c1 64144,c1(SCC(N2CC3C(CNC(C(C)NC(N)=O)=O)(C3)C2)=O)ccc(F)cc1F 64145,C12(C(N(C3CN(C)C3)C)=O)CCC1CN(C(c1ccc(Cl)cc1Br)=O)C2 64146,C1(CNC(C(C)CN(C)C)=O)CC2COCC2N1C(=O)CC1CCC(O)C1 64147,c1(C(=O)NCCN(C(c2nc(C(C)C)sc2)=O)CC2CC2)ncccc1O 64148,N1(C(=O)CCOCCCOc2cccc(Cl)n2)CCC12CCC2 64149,c1(C(=O)NCC2(NC(C3C(CC)CCCC3)=O)CCOCC2)c(F)ccnc1F 64150,[N-]=[N+]=NC1CCOC1OC(C1CCN(CCN2CCC2)CC1)=O 64151,C12(NC(CC(=O)NCC)=O)CC3CCC(C1C2)N3C(=O)C(C(C)(C)C)OC(C)C 64152,c1(C(=O)NC(CNC(c2ccc(OC(C)C)nc2)=O)(C)C)[nH]nc([N+](=O)[O-])c1Cl 64153,C1(CNC(CSS(C)(=O)=O)=O)CC2CC1CN(C(=O)C(C)(F)c1ccccc1)C2 64154,Cc1ccc(OCCC(=O)NC(C)CCNC(c2c(C)cnn2C)=O)c(C)c1 64155,c1(-c2ccc(C(=O)NC(CCC=C)C(=O)NC)cc2)ccc2nonc2c1 64156,c1(-c2cn(CCN(C)C(c3cccc(C(F)(F)F)c3F)=O)nn2)c(F)cccc1Cl 64157,c1(CNC(c2c(CC)cc[nH]2)=O)cccc(C(=O)NCC(Cl)Cl)n1 64158,c1(C(N(C2CC2)CC2CCCN(C(CCCSC)=O)C2)=O)cc(Cl)cnc1C 64159,c1(OC)ccc(NC(C2CC3CC3N2C(c2cnc(O)[nH]2)=O)=O)cc1F 64160,c1(CCC(C)NC(=O)CCOC2CC2)ccccc1F 64161,Cc1ncnc(O)c1C(=O)NC1CCN(C(=O)Cn2cncn2)C1(C)C 64162,C1(NC(C2N(C(c3cccc(OC)n3)=O)CCCCC2)=O)CCn2ncnc2C1 64163,C1(CNC(C2N(C(CCCOCCOC)=O)CC2C)=O)CC12CCOC2 64164,C12(NCc3nc(CCC)on3)CCC(CN(C(c3cc(C)cc(F)c3)=O)C1)C2 64165,C=CCC(C(=O)NCCCN(C(=O)CC(C)O)C1CC1)OC 64166,c1(-c2cc(OC)cc(NC)c2)cnc2c(C(=O)Nc3cccnc3Cl)cccn12 64167,n1(C(C)C)cc(C(N2CC(CNC(=O)C(C)(C)C(C)C)C3(CC3)C2)=O)ccc1=O 64168,C(=O)(C(C)(C)CC(C)(C)C)NC1C(CNC(c2c(CSC)cccn2)=O)COC1 64169,N1(C(CC(C)OC)=O)CCCCC1C1(NC(=O)CN2CCCCC2)CCOCC1 64170,c1(C(N(C(C)CNC(=O)C=CCOC)CC)=O)c(Cl)cccc1Br 64171,C1CCC(=O)N1.c1(C(CNC(C=CCC2(OC(C)=O)CCC2)=O)C)ccccn1 64172,C=CC(C)(CC)C(=O)N1CC(OC)C(NC(=O)C(F)(F)c2cscn2)C1 64173,O=C(CS(=O)(=O)NC1CCOC1C(F)(F)F)NCCC1CCCCN1CC1CC1 64174,c1(NC(c2c(OCC)nn(C)c2)=O)cn(C)c(=O)cn1.C1(=O)C(C)C(C)N1 64175,C(CCC1CC1)(C(=O)NC(C)C)NC(CSC)=O.N12CC(C1)C2=O 64176,Cc1cc(O)c(F)cc1CC(N1CCOC(c2cn(CC3(O)CCC3)nn2)C1)=O 64177,C1(C)(C(=O)NCC(CC(=O)N(CCNC(C(C)C)=O)C)C)CCC(=O)NC1 64178,c1(C(N(C2CCN(CC3CCOCC3)CC2)CC#C)=O)csc2c1CCCC2 64179,C(=O)(N=c1ccc(Cl)n[nH]1)C12CC(NC(c3nc(Br)cs3)=O)(C1)C2 64180,C#CC1(C(=O)N(C)Cc2nccs2)CN(C(c2cc[nH]c2)=O)C1 64181,C1(F)(CNC(C2(C)CC2)=O)CCCN(C(C2(n3cnnn3)CC2)=O)C1 64182,C1(NC(CC(C)OC)=O)CN(C(c2cc(C)c(C)nn2)=O)CC2(CCOCC2)C1 64183,C1(NC(C(C)C)=O)CN(C(=O)C(F)C2CCC2)C2(CCOCC2)C1 64184,CC1(C)NC(=O)N(CC(N2CC3CN(C(=O)C(F)=C4CCCC4)CC3C2)=O)C1=O 64185,c1(C(=O)OC)cc2cc(CN(C3(C)COC3)C)ccc2o1 64186,CCC(C)CC(=O)C(=O)N1CCC2(CC2)CC1C(=O)NCCN1CCCOC1=O 64187,C1(C)(CNC(C2(F)CN(C(C(CCSC)O)=O)C2)=O)CC2(CCC2)C1 64188,CCC(C(=O)N1CCCC1C(C)(C)NC(c1ccc[nH]1)=O)OC 64189,N12CCOC(C)(C1)C2.c1(CNC(C(C)NC(=O)Nc2ccco2)=O)ccoc1C 64190,CN1CCN(C(C2CCC(O)C2)=O)c2cc(C(F)(F)F)ccc21 64191,c1(OCC(=O)NC(C)CN(C)C(c2cocn2)=O)ccccc1Br 64192,C(C(CC)NC(=O)CCc1cc[nH]n1)N(C(C=CCOCCOC)=O)C 64193,C1(CC(=O)N(CC(CN(C(C(CC)=CC)=O)C)O)C)CCCC(C)(C)CC1 64194,c1(NCCc2n(C(CC)C)nnn2)cnc(C(F)(F)F)nc1.C1(C(=O)N)(CF)CC1 64195,C1(C(=O)NC(C(=O)N(CCCCO)C=O)CC2CCCC2)CCC2(CC1)CC2 64196,C1(CC(=O)NCCCN2C(C)CCCC2)CCC2(CCC2)CC1 64197,Cc1cc(C)c(C(=O)N(C(CNC(=O)C(C)(C)C(=O)C2CC2)C2CC2)C)c(O)n1 64198,Cc1cnc2ccccc2c1C(=O)NC1CC1NC(=O)Cc1ccno1 64199,C1(CN(C(C2C(C)C2)=O)C)CN(C(=O)CCOc2cc(Cl)ccc2Cl)CC12CC2 64200,c1(CC(C)NCCN(C(=O)O)Cc2ccccc2)cccc(SC)c1.C(F)(F)F.CO 64201,C1(NC(C2C(C)C2)=O)CN(c2nc(Cl)nc3[nH]cnc23)CC12CCOCC2 64202,N1(C(c2cccc(NCC)c2)=O)CC2CC(NC(=O)C=CCF)CC2C1 64203,C(=O)(C1CCc2ccccc21)NCC1CN(C(C#CC2(C)CCCO2)=O)C1 64204,CC1CCCC=C1C(=O)NC(COC(C)C)C(N1CC(O)C(O)C1)=O 64205,N1(C(c2ccc(OC)cc2)=O)CCCC12CN(C(=O)CCn1nc(C)cc1C)C2 64206,C1(C(N2C(C)C(NC(c3ncnn3C)=O)CCC2)=O)CCc2nncn2C1 64207,c1(OC)cccc2sc(C(=O)N(C)CCNC(=O)C(C)N(CC(F)(F)F)C)cc12 64208,c1(CC(=O)N(C2CCCN(C(CCC=CC)=O)C2)CCO)c(Cl)cccc1Cl 64209,CCCC(C(=O)N1C2CCC1CN(C(c1nncn1CC)=O)C2)C(C)C 64210,c1(C(C)=O)ccc(C(=O)NC2CC2C(N2CCOCC2c2ccccc2)=O)nc1 64211,CCCC(C)CC(=O)NCc1cc[nH]c1C(=O)N(C)CC1CC1(F)F 64212,CC(C)(O)CCC(=O)NCCCCC(=O)NCCC1CCCC1 64213,N1(C(c2csc(C)c2C)=O)CC2CCN(C(c3cc(Br)c(Cl)cc3F)=O)C2C1 64214,CC1C(C(=O)NC(C2CCOC2)CO)CCCN1C(c1cnn(C)c1N)=O 64215,c1(C(=O)NC(C(=O)NC(COCC)C(C)C)c2ccoc2)cnc(O)c(F)c1 64216,Cc1cc(C(=O)NC(C(=O)NC(C2CSC2)C)C(C)O)cc(O)c1 64217,c1(CC#N)ccccc1C(=O)NCCC1CCN(C(=O)CC2C=CCC2)CC1 64218,Cc1ncncc1C(=O)NC1CCCC1C(=O)NCC1(CO)CC1(C)C 64219,C1(NC(C(C)SC)=O)CCOC12CCN(C(c1cc(Cl)c(F)cc1N)=O)CC2 64220,C(=O)(N=c1c(C)c[nH]cc1Br)C1C2(CN(Cc3c[nH]c4ccc(OC)cc43)C2)C1 64221,N1(C(CC2(C)CCCC2)=O)CC(NC(c2coc(Cl)n2)=O)CC(O)C1 64222,C1(NC(CSCCC)=O)CC(C)CN(C(=O)C(O)C(C)CC)C1 64223,Cc1ccc(CC(=O)NC2CN(Cc3ccon3)CCC2C)c(C)c1 64224,C12(CCNC(=O)Cc3ccsn3)CCC1CN(C(=O)CCc1cscn1)C2 64225,c1(C(N2CCC=C(F)C2)C(=O)NCc2ccccc2)ccc2cccnc2n1 64226,c1(C(C)=O)ccc(C(=O)NC(C)C(C)NC(=O)C(CN(C)C)C(C)C)cc1C 64227,Cc1cnc(C(=O)NC2CCC(N(C(=O)CCc3cn(C)nn3)C)C2)nc1 64228,c1(C(=O)NCc2c(C)ccnc2)cc2ncccc2[nH]1 64229,S(=O)(=O)(c1csc2ccccc12)N1C2CN(C(COC)=O)C(CC2)C1 64230,c1(C(CO)NC(=O)OC(C)(C)C)ncc(C2CC(C(=O)NC(C)(C)C)C2)cn1 64231,C1(C#N)(C(=O)NCc2c(F)cc(OC)cc2F)CC2CCC(C2)C1 64232,C(=O)(CC(C(F)(F)F)NC(c1nn(C)cc1Cl)=O)N1CC(N(C)C)C2(C1)CC2 64233,Cc1ccc(OCCC(=O)NC2CN(C(=O)Cn3ccnn3)CC2(F)F)c(C)c1 64234,Cn1ccc2nc(N3CCN(C(=O)COCC4CCCO4)CC3)nc(Cl)c12.OC 64235,c1(NC(C2(C)N(C(c3ccc(OC)c(Br)c3)=O)CC2)=O)cc(Cl)cc(Cl)c1O 64236,N1(c2c(S(=O)(=O)NCC3CCC4CC34)cccn2)CCc2ncnc(O)c2CC1 64237,C1(CN(C(C2=NOC(SCC)C2)=O)C)CCC2(CCC2)CO1 64238,c1(C(=O)NCC(C)(C)NC(=O)CCc2ccc(Br)s2)ncncc1Cl 64239,C1(NC(CCCN=[N+]=[N-])=O)CC2CN(C(c3ccc(F)s3)=O)CCN2C1=O 64240,C1(N(C(C2(CC)CC(C)(C)C2)=O)C)CC2CC1N(C(=O)CCc1cnco1)C2 64241,c1(CC)cc(C(=O)NCCN(CCOC)C(C2CCS2(=O)=O)=O)c(C)nn1 64242,C(=O)(CC(C)CC(=O)OC)NC(CCC)C(=O)N(CC(C)C#N)C1CC1 64243,C1(C(N(CC(C(=O)OC)C)C)=O)C2CC3C(C2NC(=O)C(C(C)C)C2CCC2)C13 64244,N1(C(C(=O)NC)CCc2ccc(Cl)cc2)CCCN(C(C)CO)CC1 64245,c1(C(=O)OC)cncc(C(N2CC(F)CC2CNC(=O)CCC=C(C)C)=O)c1 64246,CCC(C(=O)NCC1(CCNC(c2sc(C)nc2C)=O)CC1)C(C)C 64247,C#CCCCCCCC(=O)NC1CC1NC(=O)CC1CCOC(C)(C)C1 64248,C1(CCNC(C#CC(C)C)=O)CN(C(c2c[nH]c3cnccc23)=O)CCS1(=O)=O 64249,c1(C(=O)NC(CNC(c2cc(C)n(C)n2)=O)(C)C(C)C)cnc2c(C)cccn12 64250,c1(C(N2CCN(C(CS(=O)(=O)NCC)=O)C(C)C2)=O)cc(Cl)cc(C)c1O 64251,c1(C(N2CCCC(NC(CNC(CC)=O)=O)(CO)C2)=O)cc2c(C)cccn2c1 64252,C(=O)(CC(C)CC(C)(C)C)Nc1c(C)c(NNC(=O)c2ccc(Cl)cc2)ccc1 64253,C1(C)(CC(=O)N(CC#C)Cc2ccccc2)CCCN1C(=O)Cc1ccn(C)n1 64254,C=C1CCN(C(c2nocc2CC)=O)C(C(N2CCCC(O)C2C)=O)C1 64255,C(=O)(CC(F)(F)C(F)F)NC1CCCN(C(c2cn(CCCOC)nc2C)=O)C1 64256,N1(C(C2C(NC(CCCC3C(C)C3)=O)COC2)=O)CCCC(C2CCC2)C1 64257,Cn1cc(N)c(-c2nc(CCc3ccccc3)nn2-c2ccccc2)n1 64258,c1(C(c2nncn2C)NC(C(CC)(C)C)C)ccc2c(c1)CCC2 64259,Cc1ccc(Br)c(NC(c2nc(-c3cnn(CCCO)c3)cs2)=O)n1 64260,C1(NC(C(c2ccccc2)OCC)=O)CCN(C(c2cnc(Cl)nc2)=O)CC1 64261,C1(F)(CNC(CSC)=O)CCCN(C(=O)Cc2ccc(CC(C)C)cc2)C1 64262,c1(C(C)C)cc(C(N2CCC(CNC(c3ccnc(Cl)c3N)=O)C2)=O)cc(O)n1 64263,c1(OCC)ccc(Cl)cc1C(=O)NCCCNC(=O)C(O)C(C)C.C(CC(C)C)O 64264,c1(OCC)c(NC(=O)NC2CCCC(c3ccncc3)C2)cccc1F 64265,N1(C(CN(C)CC)=O)CCC(CNC(=O)C(COC)COC)C(C)C1 64266,N#Cc1ccnc(N2CCN(CC(=O)NCC(c3cccc(Cl)n3)(F)F)CC2)c1 64267,C(=O)(CC(CC)SC)NCC(CC=C)NC(=O)Cc1coc(C)n1 64268,Cc1ccc(C=CC(=O)NC2(C)CCN(C(c3cc(C(C)(F)F)on3)=O)C2)nc1 64269,N1(C(=O)NC(CCCC(=O)NC2CCOC2)OC)CCc2ccc(Cl)cc2C1 64270,c1(NCC2(F)CC(NC(CC(C)C3CCCO3)=O)C2)ncnc(N(C)C)c1[N+](=O)[O-] 64271,C(=O)(C1=CCOCC1)NCC1C(NC(Cc2ccc(C(=O)OC)s2)=O)CCCC1 64272,N1(C(c2cc(CC(C)C)on2)=O)CC(CNC(c2nsnc2O)=O)CC1(C)C 64273,Cn1c(=O)n(C)c2c(C(N3CC(CO)(NC(=O)COCCF)C3)=O)cccc12 64274,N1(C(CC(CC)C)=O)CC(C2CCCCN(C(c3cccc4ncoc34)=O)C2)C1 64275,CC1CC(C#N)CN1.C1(C(=O)N)CC2C(C1)C2(C)C.C12(CC)CC(n3cc(C)nn3)C1C2 64276,N1(C(c2c(COC)scc2)=O)CCCC12CCC(NC(=O)C(C)(C)C(C)C)CC2 64277,c1(C(=O)NCC(C)(C2CC2)NC(c2nc(OC)oc2)=O)cncc(Cl)c1Cl 64278,C1(NC(=O)COC2CCCC2)COC2(C1)CN(C(=O)C=CBr)C2 64279,C(CC(F)(F)F)N(C(=O)CCn1cccn1)CC.C1=CC(=O)NC1(C)C 64280,C1(N(C(c2ccc(CC)s2)=O)CC)CCCN(C(=O)CCc2ccccn2)C1 64281,N1(C(c2cccc([N+](=O)[O-])c2)=O)CCC2(CC1)CCN2C(c1ccc(F)nc1F)=O 64282,C1(C(=O)NCC2C(NC(c3c(CC)ncs3)=O)CC2)CCCCN1N=O 64283,C(c1ccc(Cl)s1)=CC(=O)NC(CNC(C=CCN(C)CC)=O)(C)CO 64284,c1(C(N(CCNC(c2ccc[n+]([O-])c2)=O)CC)=O)cccc2c[nH]nc12 64285,C1(NC(c2coc(CO)c2)=O)COC2CN(C(c3nccc4occc34)=O)CC12 64286,c1(OC)ccccc1C(F)(F)C(=O)NCC1C=CCN1C(c1cc(Cl)c[nH]1)=O 64287,CN1CCC(=CC(N2CC(NC(c3ncccc3C(F)(F)F)=O)C(O)C2)=O)CC1 64288,CC1(C)CC(C(=O)N2CCC(NC(c3ccc(C(F)(F)F)nn3)=O)C2)=NO1 64289,c1(N2CCC(C)(C)CC2)nc2c(c(=NCCc3cc(F)c(F)c(F)c3)[nH]1)COC2 64290,C1(N(CCC#N)CCn2cc(CCC#N)nn2)(CC)CC2(CC(F)C2)C1 64291,Cc1nc(CCC(=O)NCC2CC2NC(=O)CNC(=O)CCSC(F)(F)F)[nH]c1C 64292,Cc1cc(Cl)cc(C)c1NC(C1(C(C#N)N(C2CCCCC2)CC=O)CC1)=O 64293,CCS(=O)CC(=O)NCC(N1CCN(C(C2(C)CC2)=O)CC1)C 64294,N1(CCN(C)C)CCN(C(=O)CNC(CCOCCNC(N)=O)=O)CC1 64295,c1(CCC)noc(CCCC(=O)NC(C)CN(C(=O)CC#N)CC)n1 64296,CC1(C=CC(=O)NCC2CN(C(C3CC3C(F)F)=O)CC2(F)F)CCOCC1 64297,CCCC(C(=O)N1CCC(C(C)C)(CNC(=O)C(C)C(C)COC)C1)S(N)(=O)=O 64298,C(=O)(C(c1ccco1)NC(C1CC=CC1)=O)N(C)CC1CCOC1 64299,N1(C(CN(CCC)C)=O)CCC(OCC(=O)N(C)CCc2cccs2)C1 64300,C(C1=CCN(C(=O)CCN2CCC(O)CC2)CC1)NC(C(C(C)C)NC(C)=O)=O 64301,N1(C(C(CC)C)=O)CCCC(C)(NC(=O)CCc2cccnc2Cl)C1 64302,N1(C(C)C)CCc2cc(NC(=O)Nc3ccccc3C(F)(F)F)ccc21 64303,C(=O)(CC(O)C(Cl)(Cl)Cl)NCC=CCNC(C(C(=C)C)(C)O)=O 64304,C1(C)(CC)CCCC1NC(=O)C(C1CN(C(C2CC3(CSC3)C2)=O)C1)OC 64305,C1(C(N2CC(Cn3cc(C4CC(F)(F)C4)nn3)C(O)C2)=O)CCCC2CCCN12 64306,c1(OC)ccc(C=CC(=O)NC2(C)CCN(C(C3C=CCCC3)=O)C2)cc1 64307,CON(C(=O)C1C2CC3C(C2NC(=O)COC2CCCOC2)C13)C1CCOCC1 64308,c1(C(=O)Oc2ccc(OC3CCCCC3)cn2)cnn2cccnc12 64309,C(=O)(C(C(C)C)n1cnc(C)c1)N1CCC(CN(C(C2CC2C#N)=O)CC)C1 64310,C1(NC(CCOCCCNC(c2c(C)nn[nH]2)=O)=O)CN2CCCC1C2 64311,C1(N(C)C)CC(S(C)(=O)=NC(=O)C23CC2CN(C(=O)OC(C)(C)C)C3)C1 64312,Cc1ccnc(C(=O)NC(CN(C(=O)C(N)=O)C)Cc2ccccc2)n1 64313,c1(CN2CCC(NCC(=O)NC(CC)C(=O)OC)C2)cc(C#N)[nH]c1C 64314,C(=O)(C1=CC2C=CC(C1)C2)N1CC(NC(c2n(CC)ccn2)=O)C(N=[N+]=[N-])C1 64315,C12(NC(C(C)=CC)=O)CCC1CN(C(=O)Cc1sc(C)nc1C)C2 64316,C(=O)(C(C)(C)C1=CCSCC1)NCC1N(C)CCN(C(c2csc(O)n2)=O)C1 64317,c1(C(=O)NCC2CCC(NC(c3c(SC)cnn3C)=O)C2)cc(C)c(O)c(N)c1 64318,Cc1nc2ncccn2c1NC(C1CC12CN(C(=O)C(C)n1cccc1)C2)=O 64319,c1(CC)cnoc1C(=O)N(CCC(C)NC(=O)Cc1cscc1Br)C 64320,c1(N(C)C)ccc(C(=O)NC2(C(F)F)CCN(c3nc(C4CCC4)ns3)C2)cc1 64321,c1(OC)cccc(CC(=O)NCCCC2COCCN2C(c2cnco2)=O)c1 64322,N12CC3CC(C3C1)NC(=O)CN2C.C1(C)(C=O)C=CCCC1.c1(C(=O)N)ccsc1 64323,N12CCC13CCC(CC3)C2=O.c1(OCC=C)ccc(C(C(F)(F)F)NC)cc1 64324,C(=O)(CC(C)(O)C(F)(F)F)NCC(C)(C(C)C)NC(c1c(C)n(C(C)C)nc1)=O 64325,N1(C(CNC(CC)=O)=O)CCC2(NC(=O)CCc3ncnn3C)CCCCCC12 64326,N1(C(=O)OC)CCN(C(C2CCC2CNC(c2cnc(C)s2)=O)=O)CC1(C)C 64327,C1(COC)(NC(=O)C(C)c2cccs2)CCN(C(C2CN(C3CCOC3)C2)=O)C1 64328,C1(NC(C(C)N(CC)CC)=O)CN(C(c2cc(C(F)F)[nH]n2)=O)C2CCCC12 64329,CC1CC(CN(C=O)Cc2ccccc2CO)C1(C)C 64330,C(=O)(CC(O)CC(C)C)NC12C(NC(c3ccc(C)c(N)c3)=O)CC(CC1)C2 64331,N1(C(c2cccc(SC)c2)=O)CC(C)CN(C(=O)C=Cc2cnc[nH]2)CC1C 64332,c1(N(CC(CN(C(C(c2ccccc2)SC)=O)C)O)C)ccc([N+](=O)[O-])c(C)c1 64333,C1(C(=O)NC2COCCN(C(=O)C3=CCCC3)C2)CCn2nnnc2C1 64334,CCCC(C)C(=O)NC(CN(C)C(C1CCC1OC)=O)(CO)CO 64335,c1(OC)ccc(C(N2CC(OC)CC2CNC(=O)C(F)=C2CCC2)=O)c(O)c1F 64336,CC(C)CC(CC(=O)O)NC(=O)NCCC1CCN(Cc2ccccc2)C1 64337,c1(C(N(CC(CC)NC(C2CC(CF)C2)=O)CC)=O)cc(C)ccc1C 64338,c1(C(=O)NCC2CN(C(C3(C)CC(=C)C3)=O)C2)sc(C)cc1OC(F)F 64339,c1(C(C(=O)NCCC)N(CC(=O)OC(C)C)C)cc(OC)ccc1Br 64340,c1(C(N2CCC(C(C(=O)NC(n3ccnc3)C)C)CC2)=O)c(F)ccc(Cl)c1Cl 64341,c1(C(N2CC(C)N(C(C3CCCC4(CC4)C3)=O)CC2)=O)ncc(C#N)cc1F 64342,C1(C(=O)NCC(CC)CCO)CC12CCN(C(C1CC(=O)C1(C)C)=O)CC2 64343,O=C(C1=CC2CCC(C1)C2)OCC(N1CCCCC12CCOC2)=O 64344,C1(C(C(=O)NCC(COCCOC)C)(C)C)CCC(C(=O)OC)CC1 64345,N1(C(C2C(C)(C)OC(COC)CO2)=O)CCc2cccnc2C1 64346,C1(NC(C2N(C)CCC2)=O)CCC(NC(C2(C)CC=CCO2)=O)CC1 64347,C1(COCC(=O)NC2(CNC(C3CCSCC3)=O)CC2)CCCOCC1 64348,CC1CCC(CNC2CC3(CCC3)C2)C(=O)N1.c1ccccc1 64349,c1(C(=O)NCC=CCOc2ncc(C(=O)OC)cn2)c[nH]c2ncc(OC)cc12 64350,C(=O)(CC(F)(F)F)N(C(CCCc1onc(C)n1)=O)CC1CCN(CC(F)(F)F)C1 64351,C(=O)(CS(C)(=O)=O)NCc1c(CCNC(CC(C)F)=O)ocn1 64352,CC(CCCNC(=O)C=CSc1ccccc1)N(C1(Cl)CC1(F)F)C(=O)OC(C)(C)C 64353,c1(CCCOC)nc(-c2ccnc(C)c2)n(-c2cccc(OC)c2)n1 64354,C1(C(=O)NCC(C2CCC2)NC(=O)CCOCC2CC2)(OCC)CCCCC1 64355,N(C1c2cccc(Br)c2CC1(F)F)C(c1n(CCC)nnn1)(C)CSC 64356,c1(C(=O)NCC(C)N(C(C2CC2c2ccccc2)=O)CC)cc(F)cc(=O)o1 64357,c1(-c2c(C(=O)NC3C(NC(C4CC(C)(F)C4)=O)C3)c[nH]c2)ccc(F)cc1 64358,N#Cc1ccc(C(=O)NC2COCC2NC(=O)CCc2ccncc2)cc1F 64359,c1(N(C(C2CCOC2)CO)C(=O)Nc2cn(C3CC3)cn2)c(F)cncc1Cl 64360,C1(=CC(=O)N(CC(CNC(C(n2c(C)ncc2)C)=O)(C)C)C)CCCCC1(C)C 64361,C1(CC(=O)NC2(C(C)C)CCC2)CCC(C)CO1.C12CCCC1NC2=O 64362,C1(N(C(=O)CCOCC2CC2)C)CCN(C(=O)C(F)C2CCC2)CC1 64363,CCC(C)CC(C)C(=O)N1CC(CNC(C2CC3CCCC23)=O)C2(CCC2)C1 64364,N1(C(C2CC(CC)C2)=O)CCOC2(CCN(C(C3(SC)CCOCC3)=O)CC2)C1 64365,C1(C(N2C(CNC(C3C4CC5C(C4)C35)=O)CCC2)=O)CC2CCC(C1)C2=O 64366,N1(C(CC=CC)=O)C(C(=O)NC(c2ccn(C)n2)(C)C)CCC12CC2 64367,c1(SCC)ccc(CN=C(NCC(C)(C)CO)NC2CCCCC2)cc1 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64525,C1(NC(=O)CC2CC3(CC3)C2)CCN(C(=O)CS(=O)(=O)CC2CCCO2)CC1F 64526,C(c1cncc(OC)c1)=CC(=O)NC(CC=C)CNC(C1CCCN(C)C1)=O 64527,C1(CNC(C2CC2C2CCCC2)=O)CCCN(C(=O)CCc2cncs2)CC1 64528,Cc1ccc(CCN=C(NCC(C)(C)C2CCCC2)NCSc2cccs2)c(O)c1 64529,c1(C(N(CCNC(C2CCC(F)(F)C2)=O)CC)=O)nc2sccn2c1C 64530,c1(C(=O)NC2COCCN(C(C(C)c3ccsn3)=O)C2)cccc2cnsc12 64531,N1(C(Cc2nc(C)sc2)=O)CC(O)CC1CNC(C1(C(=O)N(C)C)CC1)=O 64532,Cc1ccc(C(N2CC(NC(=O)C(C(C)C)NC(=O)NC(C)C)C2)=O)c(C)c1 64533,Cn1ncc2c1CN(C(=O)C1=CCCN(C(C3CCOCC3)=O)C1)C2=O 64534,C1(C(N(CCOC)CC2CCCC2)=O)CC(N(C)C)C1.C12CC(C1)NC(=O)C2 64535,C1(C(=O)NC(c2ccc(F)cc2)CC)CC(O)CCN1C(c1sc(C)cc1C)=O 64536,C1(C(=O)NC(CCC(C)C)C)CC1C1CN(C(C2(O)CCCC2)=O)C1 64537,CCC(C(=O)NC1CCN(C(c2ccsc2COC)=O)C1)N(C)C 64538,c1(C(=O)NC2C(C)(C)S(=O)(=O)C2)ccc2nc(C(C)(C)C)[nH]c2c1 64539,c1(C(N2C(C(C)(C)C(=O)NCc3ccccc3)CCC2)=O)cc2ncccc2[nH]1 64540,C1(CN(C[Si](C)(C)C)CC)CCCN(S(N)(=O)=O)C1 64541,CC1=C(C)CC(C)(C(=O)NCC(C)NC(c2c[nH]cc(C)c2=O)=O)CC1 64542,N1(C(C(CC)(C)CC)=O)CCC2CN(C(C3(C#N)CC3)=O)CCC2C1 64543,N1(C(=O)CC2CCCN2C(c2ccn3cncc3c2)=O)CCC2(CCNC2=O)CC1 64544,c1(CC(N2CCC(N(C)C(c3cnn(CC4CC4)c3)=O)C2)=O)cc(F)ccc1F 64545,N1(C(=O)C=Cc2ccccc2)CCC2(CC2NC(=O)CC23CCCC2C3)C1 64546,c1(C(=O)Nc2ccc(F)c(C3CC3)c2)noc2c1CCCCC2 64547,c1(C(N(CC(C)N(C(COCc2ccc(C)s2)=O)C)C)=O)nccc(F)c1Cl 64548,C=C(C)C1CN(C(=O)N(CCCCCC)C(C)COCC)CCO1 64549,Cc1ncsc1COC(C(=O)NC1(C(C)(C)O)CN(C(=O)CO)C1)OC1CC1 64550,N1(Cc2n(CC(=C)C)nnn2)CCCC(NC(c2cc(CC)nn2C)=O)C1C 64551,C(=O)(C(C)(C)C(=O)N(C)C)N(CCN(C(c1c(OCC)cncc1)=O)C)C 64552,c1(CCC)sc(C(=O)NC(C)C(C)NC(c2ccc(CO)cc2)=O)cc1Br 64553,c1(NC(C)=O)ccc([N+](=O)[O-])c(C(=O)NC2CCCC2NC(=O)CC2(C)CC2)c1 64554,C1(C(=O)NCC2(C(N)=O)CN(C(c3cc(CCC)on3)=O)C2)CCCC(F)C1 64555,CC(CC(=O)N1CC(F)(CF)C1)C(C)(C)NC(=O)C(c1ccccc1)C 64556,C1(CN(C(C=C(C)C(C)(C)C)=O)C)CC(F)CN1C(=O)COCC(F)F 64557,C1(C(=O)NC(c2ccccc2O)CNC(=O)CSc2ccsc2)CC1C1CCC1 64558,c1(N(C(=O)C(=O)Nc2ccccc2OC2CCCC2)CCC)ccc(C)cc1CC 64559,C1(CNC(C=Cc2ccc(CC)o2)=O)CC(F)(F)CN1C(=O)CC1C=CCCC1 64560,N1(C(C(CN(CC)CC)F)=O)CC(NC(=O)CN2CCCC2=O)CC1CO 64561,C(CC(=O)NC(C)(C)CCNC(=O)COc1ccc(Cl)c(F)c1)(C(F)(F)F)OC 64562,CCC(C)(C)C(C)(NC(c1csc(Br)c1)c1nnnn1C)Cc1ccccc1 64563,C(c1ccccn1)=C(C)C(=O)NC(C)(C)C(C)NC(c1cc(C)c(C)[nH]1)=O 64564,C1(C(=O)NC(C(=O)NCCOCC)Cc2cn(C)nn2)(OC)CCC(C)C1 64565,N1(C(c2c(C(=O)OC)n(C)nc2)=O)CC(NC(C2CNC(=O)C2)=O)CC2(CC2)C1 64566,c1(Oc2ccccc2)n[nH]cc1C(=O)NCC(Cc1cn[nH]c1)CO 64567,c12csc(c1)CNC(=O)CNC2=O.CC(C)C(=O)NCC(=O)N.C1(C)CC1 64568,c1(C(=O)NC(CC(C)NC(c2cc(OC)ns2)=O)C)cccc(C(C)(F)F)n1 64569,N1(C(C2CCC(NC(c3cn4c(n3)CCC4)=O)C2)=O)CC2(CNC(=O)N2)C1 64570,N1(C(C2CCC(CNC(C34C(C)(C)C(CC3)C4)=O)O2)=O)CC2CCC(C1)C(=O)O2 64571,C1(C)(CNC(c2cc(C)on2)=O)CCCN1C(=O)C(c1cccnc1)C 64572,C1(C(N2CCC(OC(C)=O)C2)=O)CCN(C(=O)CC2CCCS2)C(C)C1.C(=O)C(C)C 64573,N1(C(c2c(C)n(CC(C)C)nc2)=O)CCN(C(c2coc(C#N)c2)=O)CC1CF 64574,C(=O)(C(O)CC[S+](C)C)NCC1CC(OC)CN1C(c1cccc(Cl)c1O)=O 64575,N1(C(CC2(C=C)CC2)=O)CCc2c(CNC(=O)CCCC3CC3)cccc2C1 64576,CON(C(=O)C1CC(=O)N(C)C1c1ccnn1C)C(C)O 64577,C1(C(=O)OCC)(N(CC(C)C(=O)OCc2ccccc2)C)CC2(CCCC2)C1 64578,C(=O)(C(C)(F)C(C)(C)F)NCC1N(C(CCCC(=C)C)=O)CCN(C)C1 64579,C1(NC(CCN(CCC)C)=O)CCCCCC1(C)C.C12CC1CNC2=O 64580,Cc1ccc(-c2ccc(N(CC(O)CO)C)cc2)cc1F 64581,C1(C(=O)NCC2(OCC)CC2)CCCCN1C(C1(C)CCC(=O)N1)=O 64582,c1(C(N(CCCCNC(CC2C(OC)CC2)=O)C)=O)cnn(CCC#N)c1C 64583,c1(CNC(C2C=CCS2)=O)ccc(C(=O)N(CC(N)=O)CCO)s1 64584,C12CCC(CC1)C(=O)N2C.c1(C(N(C(C)CC2CC2)CC)=O)sccc1Cl 64585,n1(CCC(=O)NCC2(C)OCCN(C(C(CC)C)=O)C2)ccc2cc(Cl)ccc12 64586,c1(CCNC(=O)NCC(C2CCCCC2)OC)nccc(=O)n1C 64587,CC1CC=C(C(=O)N2CCC(F)(F)C(CNC(=O)CCC3CCCO3)C2)CC1 64588,N1(CCN2C(C(=O)N)CCC(F)C2)C(=O)C(=O)N(CCCCO)C1=O.C1CCCO1 64589,CC1(C)CC(C)(CN2CC(C(=O)O)CC23CC3)CN1 64590,Cc1cn(C)c(C(c2nnnn2CC(F)F)NCCCCCCC2CC2)n1 64591,C1(CC#C)CCN(C(=O)CS(N)(=O)=O)CC1.C(=O)(C(F)=C(C)C1CC1)N 64592,N1(CC(=O)NCC2(F)CC(NC(CCC(C)C)=O)C2)C(=O)C2CCCCC2C1=O 64593,N1(C(CCOCCC)=O)CC(NC(c2[nH]nnc2CC)=O)CC1(C)COC 64594,Cn1cc(Cl)c(CC(=O)NCc2ocnc2C(=O)NCC(O)C(N)=O)n1 64595,c1(C(CN(C(C(=O)NC(C)CC2(O)CCC2)=O)C2CC2)O)ccc(Cl)cc1 64596,Cc1ccc(NC(=O)NCC(CO)NC(C2CCCN(C(=O)N(C)C)C2)=O)cc1 64597,C1(NC(CC2(C)CC2)=O)CCCCC1CNC(C1(C)CCNC1=O)=O 64598,C1(CC(=O)NCC(CC=C)(C)C)CCCN(C(C2CCCN(CC)C2)=O)CC1 64599,C(C)(c1cnn(C)c1)=CCNC(C(C)Oc1ccc(CC)cc1)=O 64600,c1(N)c(Br)cccc1[N+](=O)[O-].C1(C(=O)O)CC2(CCN(Cc3cnc(Br)s3)CC2)CO1 64601,CC(C(C)C(=O)N1CCOC(CNC(C2CC23CC(C)(C)C3)=O)C1)S(C)(=O)=O 64602,CC1(C(=O)NC2CC2NC(=O)CCc2nc(-c3cccs3)no2)C=CCC1 64603,c1(CC(=O)NCCC2N(C(c3c(OC)n[nH]c3)=O)CCC2)ccc(Cl)cc1F 64604,C1(C(=O)NCCCOC)CN(C(=O)CC2(O)CCOCC2)CC(C)O1 64605,C1(C(=O)NCCN2CCOCC2)CN(C(=O)C=Cc2ccncc2)CCO1 64606,C(=O)(CC(C)CC(C)C)N1CC2(CN(C(c3c(C)ccc(O)n3)=O)C2)C1 64607,Cc1c(C(N2CCCC(NC(=O)C(CO)N(C)C)C2)=O)cc([N+](=O)[O-])cc1Br 64608,c1(C(CC)(C)C)nocc1Cn1cc(C2(C)CN(C(=O)CC(C3CC3)OC)C2)nn1 64609,n1(CC)cnc2nc(=NCC3(COC)CCC3)[nH]c(N(C)CC3CC3Cl)c12 64610,N1(C(CCOCC#C)=O)CCCC12CCN(C(=O)C(c1c(C)noc1C)C)C2 64611,Cc1nc([N+](=O)[O-])cn1CC(N1CCCC(c2ncco2)C1)=O 64612,CC(=O)CC(C)(C)CC(=O)N1CCC(NC(=O)C(CN(C)C)CN=[N+]=[N-])C1 64613,Cc1cn2c(n1)CCC(NC(c1cnccn1)c1nnnn1CCOCC1CC1)C2 64614,c1(C(=O)NC2CC(CNC(C(C#C)(C)C)=O)C23CCC3)cccc2sccc12 64615,c1(C(=O)NC(C=CC(=O)NC(CCC)(C)CC)C)ccc2cccnn12 64616,c1(NC2CC3(CC(C)C3)C2)nccc(=NCCCCc2cnn(C)c2)[nH]1 64617,C1(NC(C(C(C)C)S)=O)CCC2(CC1)CCN(C(C1CCC(=O)N1)=O)CC2 64618,N1(C(CN(CCC)C)=O)CC(NC(c2cc(C)oc2C)=O)C2CCCCC12 64619,CC1CCC(CC(N2CCC(C(C)(C)NC(=O)Cn3ccc(C4CC4)n3)C2)=O)C1 64620,c1(C(=O)OC)conc1C(=O)NCCOCCNC(C1(OC)CC1)=O 64621,N1(C(c2c(C)n(C3CCOCC3)nc2)=O)CCCC(NC(=O)C2=CCSC2)CC1 64622,S(=O)(=O)(c1cccc(-c2ccc3ccccc3c2)c1)N1CCN(CCOC)CC1 64623,C1(NC(C2(N(C(C=C(C)C3CC3)=O)C)CC2)=O)CC2CC1C(O)C2O 64624,Cc1ccnc(C(N2CCCC2C(C)(C)CNC(c2cnsc2)=O)=O)n1 64625,N1(C(C2C3(CCN(C(C4N(C)CC(F)C4)=O)C3)C2)=O)Cc2ccc(O)cc2C1 64626,CC(F)(F)C(C)(C)CS(=O)(=O)NCCc1cncc(Br)c1 64627,c1(CCNC(=O)Nc2cnn(C(C)C)n2)cccc(OCC(F)(F)F)c1C(N)=O 64628,c1(SC)cc(C(=O)NCCCN(C(=O)CCC2(C)CCC(=O)N2)C(C)C)oc1C 64629,c1(C(=O)O)n[nH]c(CNCCCc2ccc(SC(F)(F)F)cc2)c1Br 64630,Cc1nc(C)n(CCC(N2CCC(CO)(CNC(c3c[nH]c(=N)s3)=O)C2)=O)n1 64631,N1(C(Cn2cnc(=N)[nH]2)=O)CCCC(CNC(=O)CCc2ccc(O)nc2)CC1 64632,CC1CN(CC(=O)NCc2ccc(OC(F)F)nc2)Cc2nncn21 64633,CC1OC(C)(C)OC1(C)C(=O)NCc1ncoc1CCNC(=O)CCCC(F)(F)F 64634,c1(N(CC)CC2CCN(C(C3CC34CC4)=O)CC2)cc(C)nc(C(F)(F)F)n1 64635,Cc1ccc(C(=O)N(CCNC(c2cncc(C3CC3)c2)=O)C2CC2)c(CO)n1 64636,C=CC(C)(O)CC(=O)NC1CCC(NC(=O)CS(=O)(=O)NC)C1 64637,N1(C(C2C(OC)CN(C(c3cc(C)ccc3O)=O)C2)=O)CCC(N=[N+]=[N-])CC1 64638,N1(C(C(C)NC(CC)=O)=O)CCC2(CC1)CC2(C)C(N1CCNC(=O)CC1C)=O 64639,C1(CNC(C(CCC)OCC)=O)CC2(CCN(C(=O)CC3CCC(C)CC3)C2)CO1 64640,c1(CN(C(C(c2ccccc2Cl)(C)C)=O)Cc2ncco2)cccc(Cl)c1 64641,N1(C(C2(OC)CC2)=O)C(C(=O)NCC2CC23CCCCC3)C2CC(O)C1C2 64642,C1(C)(c2cn(CC3N(C(CCCc4nc(C)sc4)=O)CCC3)nn2)CCC(C)C1 64643,Cc1cnc(C(=O)NC(CNC(c2cnc(=N)[nH]c2)=O)C(C)C)c(F)c1 64644,c1(N(CCC)C)nc2ccc(S(=O)(=O)N3CCC4(CCSC4)C3)cc2s1 64645,N1(C(CCSCC)=O)CCC(CNC(=O)COc2ccc(Br)cc2)C1(C)C 64646,c1(SC(C2CCCCO2)CC)cc(C#N)ccn1.C12CCC(C1)NC(=O)N2 64647,c1(C(=O)OC)ccc2c(n1)CCCN2C(c1ccc(-c2cnnn2C)cc1)=O 64648,c1(C(=O)NCC2COC(CNC(=O)C(F)n3ccnc3)C2)ccnc2[nH]ncc12 64649,N1(C(CNC(COC)=O)=O)CCCOC(CO)C1.c12ccccc1CC(=O)N2 64650,N1(C(C(C)S(N)(=O)=O)=O)CC2(CCC(CNC(C3CC(S(C)(=O)=O)C3)=O)O2)C1 64651,c1(NC2C(CC)CN(C(=O)Cn3ncnn3)CC2)c([N+](=O)[O-])c(C)nn1C(C)C 64652,N1(C(=O)CCN2CCOC2=O)CCC2CN(C(c3ccc(C(=O)OC)[nH]3)=O)C2C1 64653,C(=O)(C(CO)C(C)(C)C)N1CCN(C(CNC(c2c(COC)cco2)=O)C)CC1 64654,O=C(C#CC1CCOC1)NCC1CC2CCC1N(C(=O)CC1CCC(F)(F)C1)C2 64655,c1(NC(C2N(C(C)C(C)(C)C)CCOC2)=O)ccc2nncn2n1 64656,C(=O)(C#CC1CCCOC1)NC1CC(CNC(C2(SC)CCCCC2)=O)OCC1 64657,c1(SC)cc(C(=O)NCCC(C)NC(=O)C(C)NC(c2cccs2)=O)ccc1F 64658,CC(CC(=O)N(C1(C(N2CCOC(C#N)C2)=O)CC1)C)C(F)F 64659,C(C)(CO)(CC(F)F)N(C(c1ccc(SC(F)(F)F)cn1)C(=O)NCC=C)C 64660,c1(NC2CC(OCC)C2)nccc(=NC(CC)CC#N)[nH]1 64661,C#CC1CN(C(=O)C(C)C2CCC2)CCN1C(=O)C(C)OCCN(C)C 64662,c1(Sc2nc(C(=O)OCC)on2)nc(N=c2cncc[nH]2)c(F)cc1COC 64663,c1(C(=O)NCCOCCN(C)C(C2CC2F)=O)ccc2cc(C#N)ccc2c1 64664,CC(C(=O)N1CC(NC(c2ccc(CO)c(Cl)c2)=O)C2(CC2)C1)C(C)(F)F 64665,c1(CNC(=O)CNC(=O)CC2CCCN2C(C2CC(F)(F)CS2)=O)cccc(O)c1 64666,S(=O)(=O)(c1c(C)cc(Cl)cc1C)NCc1oc(C(=O)OC)c(C)c1 64667,N1(C(c2c(SC)cccc2)=O)CC2(CCN(C(C3(C#N)CC(C)C3)=O)CC2)C1 64668,CC(C)CCCC(=O)N1CCC(O)(CCNC(C2(O)CCSC2)=O)CC1 64669,c1(C(=O)NCC2(O)CN(C(C3C4C5CCC(C5)C34)=O)C2)cccc2c1CCCN2 64670,C#CCCCC(C)C(=O)NCC1CN(C(c2ccc(F)o2)=O)C1 64671,c1(C(N(CCCNC(=O)CC(O)C2CCCC2)CC)=O)ncccc1OC 64672,c1(OC)ccnc(NC(c2ccsc2C(=O)NOC2CCN(C(C)C)C2=O)=O)c1 64673,CC1(C)CC(CNC(=O)CN2C(=O)CNC2=O)CN1C(C1CCC1C#N)=O 64674,N1(C(CC(CC)C)=O)CC2(CCN(C(c3cc(C(F)(F)F)ccc3N)=O)C2)C1 64675,c1(OC)cc(OC)c(C(=O)NCCCNC(=O)C(C)Sc2ccccn2)cc1Cl 64676,CC1CC(NC(c2cc(F)ccc2F)=O)CN(C(=O)Cc2cccc(F)c2F)C1 64677,c1(C(=O)NC2(CF)CCN(C(C=C(C)C(C)(C)C)=O)C2)nccc2ccsc12 64678,C#CCC(CC(=O)N1CCC(C)(O)C1)NC(c1cnsc1)=O 64679,C1(C(=O)NC2(COC)CCCC2)(CO)C=CCN1C(=O)C(CSC)O.C1(C)CC1 64680,C=CCCC(C(=O)NCC(O)CC(C)C)NC(c1cccnc1O)=O 64681,C1(F)(C(=O)NCC(C)(C)CNC(C2(c3ccccc3F)CCC2)=O)CCCOC1 64682,c1(C(=O)NC(CC=C)CNC(=O)Cc2cncn2C)cccnc1C(F)F 64683,N=c1[nH]c2cc(C(=O)NCCNC(=O)CSc3nnc(S)s3)ccc2o1 64684,c1(C(=O)NC2CCN(C(=O)CS(=O)(=O)Br)C2c2ccccc2)c(F)cccc1Cl 64685,c1(C(=O)NC2CC(NC(=O)C=CCN3CCC3)C2)csc(C(F)F)c1 64686,C(C1=CCCCC1)(c1nnnn1C1CCCC1)Nc1ccc(C#C)cc1 64687,c1(CCNC(c2n(CC)nnn2)c2ccco2)cccc(F)c1 64688,CC1(NC(c2ccc(C3CC3)s2)=O)CCN(C(C2(C)CCOC2)=O)C1 64689,C1(C(N(CC(O)CO)C(C)C)=O)CC(F)CN(CCc2c(OC)cccc2O)C1 64690,Cc1n[nH]c(C)c1C(C)C(=O)NCC(C(C)C)NC(=O)C=Cc1cncs1 64691,c1(N(C2CN(C(=O)CCc3ccc(F)cc3)C2)C)ccc(Br)cc1[N+](=O)[O-] 64692,C(CCN=c1[nH]c(=NC)[nH]c(=NC2CCc3n[nH]c(C)c3C2)[nH]1)(C1CCC1)OC 64693,c1(C(=O)NC(CNC(c2cc(OC)no2)=O)C2CC2)cc(Cl)c(Br)[nH]1 64694,CC1CCN(C(c2cnsc2)=O)CC1NC(c1cc(CF)on1)=O 64695,C(CNC(c1cc(O)nc(C2CC2)n1)=O)(CC(F)(F)F)NC(C1CCC(=O)C1)=O 64696,c1(CC(=O)NC2C(CNC(Cn3c(C)ncc3)=O)CC2)nc2c([nH]1)CCCC2 64697,C1(C(=O)NC(CN(C(C2CCC2C2CCCC2)=O)CC)C)CCCN(C(N)=O)C1 64698,C1(C2CCCN(C(=O)C(C)C#N)C2)(NC(c2ccn(C(C)C)c(=O)c2)=O)CC1 64699,C(CN1C(=O)Cc2ccccc21)N(C)C(=O)Nc1c2cc(Br)ccc2nn1C 64700,C1(NC(c2cc(C(=O)OC)no2)=O)CN(C(c2c(C)ncn2C)=O)CC1F 64701,Cc1oc(C)c(C(=O)N(C)CC2CCN(C(=O)Cc3nnc(O)s3)C2)c1C 64702,c1(C(N2C(C(CNC(c3c(C)csc3)=O)(C)C)CCC2)=O)ncnc2c1cnn2C 64703,C1(CNC(c2c(CC)nc(C)[nH]2)=O)CC2(C1)CN(C(=O)Cn1nc(C)cc1C)C2 64704,C=CCN=C(NCC1CCC2(COC2)O1)N1CCC(C)(C)C2(CCC2)C1 64705,N1(C(C=CC)=O)CCC(C2OCCC2C(=O)NCCn2ccnc2C)CC1 64706,CCC(C(O)C(C)C)NC(=O)NC(C)CCc1ccc(Br)cc1 64707,C12(O)CCN(C1)C(=O)Cc1ccc(cc1)N(CC)CC(=O)N1CC2C1.CCOC 64708,c1(C(=O)N(CCN(C(C(C)OC(C)(C)C)=O)C)C(C)C)ccc(Br)cc1 64709,C#CCC(CC(=O)N(C1CCCC(C)(C)C1)C)NC(=O)C(O)c1ccsc1 64710,C=CCCCC(=O)N1CC2C(NC(c3c[nH]cc3C(C)(C)C)=O)C2C1 64711,N1(C(c2c(CC)noc2)=O)CCCCC1CCN(C)C(c1c[nH]c(=O)cn1)=O 64712,C1(OC)CCC12CC(C(=O)NC1(C3CCCN3C(=O)CC(C)(C)C)CC1)C2 64713,CN1CC(C(=O)NCC2CCC(CNC(c3cnn(C4CC4)c3)=O)CC2)CC1=O 64714,c1(CC)nn(C)cc1C(=O)N(C1CCC(=O)N1)CC 64715,CCC(C)C(C(=O)NCC1=CCN(C(C2CC2c2ccc(F)cc2)=O)CC1)OC 64716,C1(NC(C2(OC)CCN(C(C3CN4CCC3CC4)=O)C2)=O)CN(C)CC1(F)F 64717,c1(C(=O)OCC)cccc(C(N2CC(NC(=O)CC3COCCO3)C(F)C2)=O)c1 64718,c1(OC)ccc(CN2CC(O)CC2C(N2CCCC(O)C2C)=O)c(C(F)(F)F)c1 64719,N1(C(C2(COC)CC2)=O)CCOC(C2CN(C(C3CN(C(C)=O)C3)=O)C2)C1 64720,c1(C(=O)OC(C(=O)Nc2c(C)ncc(C)n2)C(C)C)cc(C)ccc1[N+](=O)[O-] 64721,c1(C(=O)NCC(=C)CCNC(c2c(C)nn(C)c2C)=O)sccc1S(=O)(=O)NC 64722,N1(C(CN(C)CC)=O)CCCC(C)(NC(=O)COc2ccccc2C(F)(F)F)C1 64723,n1(CC(=O)NC(COC)CNC(=O)Cc2cn(C)nc2C)cccc(C)c1=O 64724,C=CCC(CC)C(=O)NCc1cccc(NC(C2CC(NC(=O)C(C)C)C2)=O)c1 64725,C(=O)(CCCNC(=O)CSC(C)(C)C)N(C)CC1(C#N)CC1 64726,C1(C(=O)NCC(CC)NC(=O)CN2CCCC2CO)(COC)CCOCC1 64727,CCC1c2ccsc2CCN1C(c1cnc(OCC)c(Br)c1)=O 64728,C(CNC(=O)CCc1nc[nH]n1)(C(=O)N(C)CC1(C)CCC1)OC 64729,CC1(CNC(c2cc(C(=O)C3CC3)on2)=O)CCCN1C(=O)CNC1CCCC1 64730,C(C(C(=O)N(C(C)CC(C)C)C)NC(=O)Cn1cc(C)cn1)OCC 64731,c1(CCC(=O)NC2C(C)(CC)C2)nc(C(C)OC)no1 64732,C1(CC)(CO)CCN(C(C2(C)CCCN2C(c2nccnc2N)=O)=O)CC1 64733,CC1C(C)N(C(=O)CNC(=O)CN(C)C)CCN1C(c1cc(S(C)(=O)=O)co1)=O 64734,CC(C)C(O)CC(=O)N1CCN(C)C(CNC(=O)C=Cc2cccnc2)C1 64735,c12cnn(C)c1NC(=O)C(COCC)NC2=O.C1(CCNC)CCCC(C)C1 64736,N1(C(c2c(C)nc(O)cc2)=O)CCCCCCC1C(=O)NC1C(O)C2CCOC12 64737,C1(NC(c2cc(C(C)C)no2)=O)CCCCCN(C(=O)C(=Cc2c[nH]cn2)F)C1 64738,c1(CN2CC(C(N(C3CCC3)CC)=O)C(O)CC2)ccc(C#N)cc1 64739,c1(C(=O)NCCCCNC(c2cc(C)c(N)cn2)=O)cccc2nonc12 64740,C1(NC(CSCCC)=O)CC2(C1)CN(C(c1csc(C3CC3)n1)=O)C2 64741,S(=O)(=O)(c1c(F)cccc1F)NCC(C(=O)O)Cc1ccc(I)cc1F 64742,CS(=O)(=O)c1ccc(S(=O)(=O)NCC(N2CC3CC3(NC(=O)C(N)=O)C2)=O)cc1 64743,c1(CNC(c2ccc(Br)cc2)C)ccc(NC2=NCC(c3ccc(Br)cc3)C2)cn1 64744,c1(CC)cnc(C(c2nnnn2C(C)C)NC(c2ccncc2)C)[nH]1 64745,C=CCC(CC(=O)Nc1cnc(O)c(F)c1)NC(C12CSCC1C2)=O 64746,c1(C(=O)NC(C(CO)NC(C(CCCOC)C)=O)C)nnc(O)c2ccccc12 64747,C(=O)(CC(C)P(C)(C)=O)N1CCC(CCNC(c2cc(C)nc(O)c2)=O)C1 64748,Cn1c(C(=O)NCC2CC(NC(=O)CC3CCCC(=O)C3)C2)cnc1O 64749,C1(C(N(C2CCN(C(=O)COc3ccsn3)C2)C)=O)CC(O)CN1C 64750,n1(CCC)ncc(C(N2CCCCC2CCNC(C2CCS(=O)CC2)=O)=O)c1Cl 64751,C1(CNC(CC(C=C)CC)=O)CC2(CCN(C(=O)C(C)C(F)(F)F)CC2)CO1 64752,COn1cnc(C)c1C(=O)NCC(c1cc(F)cc(Cl)c1)NC(=O)C(F)=C1CCC1 64753,c1(C(N(CCNC(CCN(CCC)C)=O)CCC)=O)cc(S(C)(=O)=O)oc1C 64754,C#Cc1cccc(C2CC2C(=O)NC(C)C(C)NC(=O)CC#N)c1 64755,N1(C(c2c(CC)nco2)=O)CC(NC(C2CCCC2CF)=O)C(O)C1 64756,c1(CN2CC3C(C(N4CCC(=C)CC4)=O)(C3)C2)c(C)cccc1C 64757,c1(C(=O)NCCOCCCNC(C(C)NCCCC)=O)cc(Cl)ncc1O 64758,c1(C(N2CCC(F)(CNC(C(C)(C)CO)=O)C2)=O)cc(Cl)c2ccccc2c1O 64759,CCC(C)CC(=O)N(C1CC(NC(=O)Cc2sc(C)nc2C)C1)C 64760,C(=O)(CC1=CCCCC1)N1CC2CC(C)C1C2 64761,n1(CC(=O)NC2C(CC)CN(C(=O)C=C3CCC3)C2)nc(C)c(F)c1C 64762,N1(C(c2c(C)nccc2)=O)CCC2CC2(C(=O)NCC2(O)CC=CC2)CC1 64763,Cc1[nH][nH]c(=N)c1C(N1CCC(C(C)CNC(c2cnc(C(C)C)[nH]2)=O)C1)=O 64764,N1(C(C(N2C(C#C)CCC2)=O)=O)CCN(C)CC1C 64765,C1(C(=O)N(C)CC2CCN(C(=O)C(C)C(C)O)CC2)(CC)CCC(O)CC1 64766,C1(CC=C)CCCCN1C(=O)CC=CCN(C(=O)CC(O)C1CC1)CC 64767,c1(C(N2C(CNC(c3ccc(C(C)C)s3)=O)CC2)=O)occ2c1CCOC2 64768,CCC(C(=O)NC(CC1CCC1)C(=O)NCCCCCN(C)C(C)C)OC 64769,c1(CCNCC)cc(N(C(c2nncn2C)(C)C)C2CC2)c(Cl)cc1[N+](=O)[O-] 64770,C1CC(=O)NOCCCN1C(CCOC)=O.C(CCNC1CC1)O.N(C)C 64771,Cc1cc(C(=O)N(C(C)CNC(=O)C(O)c2ccsc2)C)c(C)n1C(C)C 64772,n1(CC)nc(C(=O)NC2CN(C(=O)C(C3CC3)N(C)C)CC2C)cc1C(F)(F)F 64773,c1(C(COC)NC(CNCC)=O)ccc(C(=O)OC)cc1.C(C(=O)OC)N 64774,C(=O)(C#CC(C)(C)CNC(C1(C)CCCC1O)=O)NC(C(=O)N(C)CC)C 64775,C(=O)(C(C)C(F)(F)C(F)F)N1CCN(C(C=CC=CC)=O)CC1COC(C)(C)C 64776,C1(C(=O)NCCNC(C2CC(=C3CCC3)C2)=O)CCC([N+](=O)[O-])CC1 64777,c1(OC(C2CCC(C)(N(C)C)C2(C)C)=O)cccc2c1COC(=O)N2 64778,c1(C(N2C(CC(C)C)CCCC2)C(=O)NC2COC2)cccn2ccnc12 64779,N1(C(C(CC)F)=O)CC2(C)CC1(C(=O)NCCCCCO)C2 64780,N1(C(C(CCC)C)=O)CCN(C(=O)CSCC(C)C)CC1C 64781,N1(C(C2C=CCCC2)=O)CCN(C2CCOC2)CC1.O=C1COCCN1 64782,C1(C(C)(C)O)(CNC(CC=C)=O)CN(C(=O)CC2(COC)CC2)C1 64783,N1(C(c2cc(CC)on2)=O)CCN(C(=O)C=Cc2ccc(CC)cc2)C(CF)C1 64784,c1(C(=O)OCC)ccc(CC(=O)NC2CCN(C(=O)C=Cc3ncco3)C2)cc1 64785,c1(C(COC)NC(N2C(CN(C)C(=O)OC(C)(C)C)CCC2)=O)ncccc1F 64786,N1(C(C(C)OCC(F)(F)F)=O)CCN(C(=O)C=Cc2cccnc2)C2CCC12 64787,Cc1ccn2ncc(C(N3CCC(CC(C)NC(=O)C(F)C4CC4)CC3)=O)c2n1 64788,Cn1c(C(N2CCN(C(=O)C(F)C(C)(C)O)C(CCO)C2)=O)cccc1=O 64789,CC1(NC(C2C3CCCCCC23)=O)CCCCCC1.c12ccc(nc1)c(=O)[nH]2 64790,C1(C)(C(=O)NC2(CCC)CCC2)CC(OCCSC)CN1C(=O)CCC(C)C 64791,Cc1cc(CNC(=O)CC(CC#N)NC(=O)OC(C)(C)C)c(C)n1-c1ccon1 64792,C1(C(=O)NCC=C)CCN(c2nnnn2CCC2(O)CCCOC2)CC1 64793,C1(C(n2cc(C(CC(=O)O)SC)nn2)C2CC2)COC(C)(C)C1.CCC1C(=O)N1 64794,c1(C(N2CCN(C(C3(CF)CC(=C)C3)=O)CC2CF)=O)cc(F)c2cn[nH]c2c1 64795,c1(C(=O)NC(C(=O)NCCNS(CC)(=O)=O)C(C)C)ccc(C)nc1O 64796,C1(C(N(C(C)C)CCNC(C2CCC2C)=O)=O)CCCN(c2ccnc(Cl)n2)C1 64797,C(C(F)(F)C(=O)OC(C)(C)C)OCC.c1(C(CO)N(C)C)cc(-c2ccco2)on1 64798,Cn1ccc(=O)c(C(=O)NC2CCCC(NC(C3CCS(=O)(=O)CC3)=O)C2)c1 64799,C1(NC(C2C3CN(C(C(N4C(=O)CCC4=O)C)=O)CC32)=O)CCCOC12CCC2 64800,c1(C(N2C(C)CCC(CNC(=O)Cc3cccs3)C2)=O)cncc2c1CCC2 64801,N1(C(C(C)=CC2CC2)=O)CCCC(CO)(NC(c2cncc(Cl)c2)=O)C1 64802,C#CC1CN(C(C23CC(CN(C(=O)Cc4cncnc4)C2)C3)=O)CCO1 64803,c1(C(=O)NCC2C(C)CCN(C(CCCC#C)=O)C2)cccc2c1COC2 64804,C1(NC(Cc2ccc(C)c(Br)c2)=O)CC2(CCC(NC(=O)C(F)=CCCF)CC2)C1 64805,C(CCC(C)(C)C(=O)N1CC(O)CO1)NC(c1c(C)cns1)=O 64806,Cn1[nH]c([N+](=O)[O-])nc1=NCC(c1ccccc1F)NC(=O)C=C(Cl)Cl 64807,N1(C(C2N(C(CCSCCCC)=O)C3(CC2)CC3)=O)CCC2(COC(C)C2)C1 64808,N1(C(C2CN(C(C)=O)C2)=O)CC2CC2(C(N2CCCC2C)=O)C1 64809,c1(C(C)NC(=O)C(N2CCC3(CCO3)C2)=O)ccc(-c2cccs2)cc1F 64810,c1(OC)cc(C(N2CC(O)CC2CNC(C23CC(C2)C3)=O)=O)c2c(c1)CCO2 64811,C1(C(=O)NCCOCC(=O)NC2(CCC=C)CC2)CCOC1C1CC1 64812,N1(C(C=C(C)Cl)=O)CC2CC1CN(C(c1cc(C)ccc1Cl)=O)C2 64813,CCC(C(=O)NCC1CCN(C(C2CCN(CC)C2)=O)C1)n1cncn1 64814,c1(C(=O)NC(COCC#C)=O)ccc(C2COCCN2C(c2ccsc2Cl)=O)n1C 64815,C1(C(N2CC(NC(C3(CC)COC3)=O)C2)=O)CCOC(C)C1 64816,CN1CCOC(C(=O)NC2CN(C(c3cc(-c4ccccc4)ns3)=O)CC2O)C1 64817,N1(C(C2C(=C)CC2)=O)CCN(C(=O)C=Cc2cncc(OC)c2)CC1CCOC 64818,C1(COC)CN(C(=O)NC2CCN(S(C)(=O)=O)CC2)CC1O 64819,c1(CC)occc1C(=O)NC(CNC(c1cnc(C)s1)=O)CCOC 64820,C1(OCCOCCN(C(CN2CCC(CC)C2)=O)CC)CCC2CC2C1 64821,N1(Cc2nnc(C3OCC(C4C(C)C4)C3)o2)CCC(n2ccnc2O)CC1 64822,C(=O)(CC(O)Cc1ccccc1)N1CC(CCNC(CN(C2CCCC2)C)=O)C1 64823,n1(CCCN=C(NCC(=C)C)NC2COC(C)C2)nnc2ccccc2c1=O 64824,c1(C(=O)NCCN(C(=O)CSC)CC)cc2cc(Cl)ccc2n1C 64825,c1(NC(C2CCCN(C(C3CCC(C(F)(F)F)CC3)=O)C2)C)ncc(I)cn1 64826,c1(CC)cccc(C(N2CC(F)CC2CNC(c2ccc(F)s2)=O)=O)c1O 64827,c1(CNC2CC(NC(=O)NC3CCOCC3)C2)cc2cccc(Cl)c2nc1Cl 64828,c1(C(CC(N2CCOC(CC(F)(F)F)C2)=O)SC(F)F)cccc(F)c1 64829,C1(CNC(C2N(C)C(=O)OC2)=O)CN(C(=O)CSc2ccncc2)CCC1(F)F 64830,c1(CC)cc(Cl)cnc1-c1c[nH]nc1C(=O)NC(c1cc(F)ccc1F)C 64831,c1(NC(=O)OC)cc(C)sc1NCCc1nnc(-c2ccc(OC)cc2)s1 64832,C1(C(=O)NC(C2CCCCC2)C(=O)N(C2CC(N(C)C)C2)C)CN2CCC1C2 64833,C(CCC(C)C(=O)N1CC(O)(CN(C(=O)Cc2cc(C(F)(F)F)n[nH]2)C)C1)OC 64834,C1(NC(C2(NC(C3C(=C)C3)=O)CC(O)C2)=O)CCCNC1=O 64835,C1(NC(c2cn[nH]c2)=O)C2CN(C(=O)CCCOC3CCOCC3)CC12 64836,c1(C(=O)NC2CN(C(C(CC(C)C)OC)=O)CC(C)C2)scc2c1OCCO2 64837,c1(C(N2CC(C)N(C(=O)C=CC3CCOC3)CC2)=O)cc(Cl)c(F)c(Cl)c1 64838,CC1N(N(C)Cc2ccn(C(F)(F)F)n2)C2(CCCC2)C1=O 64839,C12(COC)CN(Cc3cc(Br)nn3Cc3ccccc3)C(C)(CO1)C2 64840,C1(NC(C(=O)OCC)=O)CCCC1C#N.c12conc1C1CN(C1)C2=O 64841,N1(C(c2ccc(C#N)o2)=O)CC2CCC1C(Nc1ncnc(Cl)c1Br)C2 64842,C(C(CC)(CC)CC)(c1n(CCOC)nnn1)NCC1CC(C2CCC2)C1 64843,c1(C(=O)NC(C(=O)NCCc2cnc(C)[nH]2)Cc2ccoc2)cnc(Cl)n1C 64844,Cc1nnc(C(=O)N(C(C)CCNC(C2CC2(C)C(F)(F)F)=O)C)s1 64845,C1(CNC(CC2(N(C)C)CCCC2)=O)CCCCCN1C(=O)CCc1ccoc1 64846,Cc1ccc(C(N2CCN(C(=O)C=CC(C)(C)C)CC2CCO)=O)c(=O)n1C 64847,N1(C(c2ncc(F)cn2)=O)CC2CCC1CN2C(c1ccc(Cl)cc1)=O 64848,N1(C(c2c(CC)onc2)=O)CC2(NC(=O)C=Cc3sccc3C)CCC1C2 64849,Cc1ccc2c(=NCC(C)CN(C)C)[nH]c(NCC3CC4(CC4)C3)nc2c1 64850,c1(NC2CCN(CC)CC2)cc(N2CCC(CCO)(CO)C2)nc(C)n1 64851,C=CC1(CNC(C2CCCC2CNC(=O)C(=CC2CCCC2)C)=O)CCC1 64852,c1(NC(=O)NC2CN(c3ccc(C)cc3)C(=O)C2)cccc2c(C)cc(C)nc12.C1CC1 64853,c1(C(=O)NCCC(C)N(C(C2CC(CCC)C2)=O)C)cn2cc(Cl)cnc2n1 64854,N1(C(C(C)SC)=O)CC(C)CN(C(c2cnn(CCN(C)C)c2C)=O)CC1C 64855,c1(C(C(=O)NC2C(C(=O)NCC=CCCC)CCC2)(C)C)cccc(Br)c1 64856,C(=O)(C1CCc2nccn21)NC1(CNC(C2CC(C)OCC2)=O)CCCCC1 64857,[N-]=[N+]=NCCCCC(=O)N1Cc2occ(C(=O)NC3C4CCCC34)c2C1 64858,C1(CC)CC(C(=O)NCC2CC(NC(C3(C(=O)N(C)C)CC3)=O)C2)C1 64859,c1(NC)cccc(C(=O)N(CCCNC(c2ncccc2C)=O)C(C)C)n1 64860,N1(C(CCC(=O)NC)=O)CC(=O)NCC1C(=O)NOC(C)(C)CC1CC1 64861,c1(CNc2c(CCC(=O)NCC#C)cccc2)c(Cl)cc(Br)cc1Cl 64862,C1(CCOC)CCCCN1C(C1CCN(C(c2cc(C)no2)=O)C1)=O 64863,c1(Cc2nc(CNC(c3ccccc3)=O)on2)cccc2c(Br)cccc12 64864,N1(CC(=O)NCCC2(OC)CN(C(CC3CCC(C)C3)=O)C2)CCCNS1(=O)=O 64865,C(CC(C)(C)C(=O)NCCC(C)N(C)C(c1cccc(OC)c1Cl)=O)OC 64866,CN(C[Si](C)(C)C)C(=O)CC1CCCCN1C(=O)CCc1cnco1 64867,C(=O)(C1Cc2ccc(F)cc21)N1CCCC(N(C)C(C2C(C#N)C2(C)C)=O)CC1 64868,c1(OC)ccc(C)nc1C(=O)NC1CCCC(NC(C2CC3(C2)CC(O)C3)=O)C1 64869,CC1CCCCC1OCC(=O)NCC1CC(NC(C2(CC(F)F)CCC2)=O)C1 64870,Cc1cc([N+](=O)[O-])cnc1N1CC(CNC(C2(Cl)CC2)=O)OC2(CCC2)C1 64871,C(=O)(C1=CC(C)(CC)C1)NCC1(C)N(C(c2cnc(OCC)s2)=O)CCC1 64872,CC1(C)C(CNC(=O)Cc2cc(C(F)(F)F)co2)CCN1C(=O)CCc1cnoc1 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65029,Cc1cccc([N+](=O)[O-])c1C(=O)NCCC(C)NC(C1CC2(C1)CC(F)(F)C2)=O 65030,N1(C(c2c(CC)[nH]cc2)=O)CCCOC(CNC(C2(c3cc[nH]n3)CCC2)=O)C1 65031,C1(C)(NC(CC2(NC(C)=O)CC2)=O)CCN(C(c2c[nH]nc2C(F)(F)F)=O)C1 65032,c1(OC)cccc(C(N2CC(NC(=O)CSc3n[nH]c(C)n3)CC2C)=O)c1OC 65033,n1(CCCSCC)nnnc1C(c1cccnc1)NCc1cccn1C1CC1 65034,c1(C(=O)NCC2CCC(NC(c3n(C)c(S)nn3)=O)C2)cc2ccoc2cc1F 65035,CCCC(Cc1ccccc1)C(=O)NC(=O)C(c1cc(C(F)(F)F)ccn1)=O 65036,c1(C(c2nnnn2C2CC2)NCC(CC(=O)NC)C)nc2ncccn2n1 65037,c1(CN(C)C)ccc(C(=O)NCCCNC(=O)CC2CC3CCC2O3)cc1 65038,C1(C#N)(C(N(CC(=O)N(CC(CC)NC(=O)C(F)(F)F)C)C2CC2)=O)CCOC1 65039,c1(CC(=O)NC(C)CCCNC(c2cnoc2C2CCC2)=O)cccc(C#N)c1 65040,c1(-c2cn(CCC)nc2)ccc(C(CC(=O)O)NC(=O)Sc2cnn(C)c2)cc1 65041,c1(C(=O)NC2CC(C(=O)Nc3cnn(C4CC4)c3)C2)cccc(O)c1F 65042,c1(C(=O)NC(C(=O)NCCCCN(CC)CC)CC2CCC2)cc(C)cc(F)c1 65043,CC1CCOCCN1C(C1CCC2(CC2)N1C(=O)C(C)(C)N=[N+]=[N-])=O 65044,C1(C(N2CCCC(CCNC(=O)CC3CCCCCO3)C2)=O)CC2CCC1CC2 65045,c1(OC)cncc(C=CC(=O)NCC23CCC(CC2)N3C(C2CCSCC2)=O)c1 65046,C(=O)(C#CC1(C)CCCO1)NC1CCC(C)(NC(CCN(CCC)C)=O)CC1 65047,C12(CN(C)C(C3C=CCN(C(=O)Cc4cccs4)C3)=O)CCC(CC1)C2 65048,c1(C(N2CCC(N(C)C(C34CC5CC3C4C5)=O)C2)=O)cc(O)c2ccccc2c1 65049,C(=O)(C(CC(=O)OC(C)=O)C(C)=O)NC12CC(NC(c3c(C)ccc(C)n3)=O)(C1)C2 65050,Cc1c(C(N2CCCCCC2)C(=O)NC2CC(C(N)=O)C2)n[nH]c1C1CC1 65051,c1(N(C)C)cccc(NC(C2CN(C(=O)CSCc3cccs3)CCO2)=O)c1 65052,C1(C(N(CCCCCC)C(=O)N)C2CC2)CC(OCC2CC2)C1(C)C 65053,c1(C(=O)NCC(CC=C)NC(=O)C(C(C)(C)C)OC)cc2c(cc1Cl)OCO2 65054,C1(N(C)CC)CCCCC1(C)C.c12cn(nn1)C1CC(C1)C(=O)OC2 65055,c1(OC2CCC(CC3C(C)CCCC3)CC2)nc2ccccc2[nH]1 65056,C(=O)(C1=CCC(C)(C)CC1)NCCC(C(=O)NC1CCOCC1C)OC 65057,C12(C)CCC(CO)(CC1)CC2.C1(CCN2CC2)COC1.CO 65058,C=CC(C)(CC)C(=O)NCc1cc(C)c(C(=O)N(CC(O)CO)C(C)C)o1 65059,CCC(CNC(=O)CC1CCCC1O)(CC)C(=O)N1CC(N2CC(O)C2)C1 65060,CCC(CC(=O)NC1(CC)CCCN(C(=O)CCSC)C1)CC(F)(F)F 65061,N1(C(c2c(COC)occ2)=O)CC2CC2(CNC(=O)CCCc2ccccc2)C1 65062,c1(C(N2C(CNc3cc(COC)ncn3)CCC2)=O)ccc(Br)c2ncccc12 65063,N(C(=NCCC(C)=O)NCCC1CCSC1)Cc1n(CCC)ncn1 65064,C(=O)(C1=C(C#N)CCC1)NC(C=C)CC(=O)N1CCC1COC 65065,C(C(C)(C)CCNC(C1COCCO1)=O)NC(C(C1CC1)OCC)=O 65066,N1(C(C2C(C(=O)OC)C2)=O)CC(NC(c2ccc(OC)cc2Cl)=O)C2(CCC2)C1 65067,c1(C(=O)NCC2(F)CC(CNC(c3c(C)ocn3)=O)C2)cc(O)ccc1Br 65068,CCCCCCCCCC(O)C(=O)N(CC(C)CNC(c1nccnc1C)=O)C 65069,C12(C(=O)NCc3nc(C)c(C(=O)NCC4CC(CF)C4)o3)CCCC1C2(F)F 65070,C1(NC(c2cn(CCC)nc2)=O)CCN(C(=O)CCCCC(N)=O)CCC1(F)F 65071,CC(C)CC(C)CNC(=O)C(O)CNC(=O)CSC(F)(F)F 65072,N1(C(C(C(C)C)SC)=O)CC(CNC(=O)C(C)NC(=O)C2CC2)C2(CC2)C1 65073,N1(C(c2ccc(C(F)F)[nH]2)=O)CCC2(C1)CN(C(C1(F)CCCOC1)=O)CCO2 65074,c1(CC2N(C(CC(c3onc(OC)n3)N)=O)CCC2)cccc(C)c1 65075,C1(NC(Cc2c(C)con2)=O)CC(C)N(C(=O)C(C)CSc2ccccc2)C1 65076,CS(=O)c1ccccc1C(N1CC2(C1)CN(C(c1cnc(C(F)F)nc1)=O)C2)=O 65077,C1(C(N2C(CCNC(c3ccnc(C)n3)=O)CSCC2)=O)CCCC(C)(C)C1 65078,Cn1cnc(C(=O)NC2CC(C(=O)NCC(CSC3CC3)CO)C2)c1 65079,c1(C(=O)NC(C)CN(C)C(C2CCCN2c2cnccn2)=O)ccc(Cl)cc1O 65080,CCCS(=O)(=O)C(C)C(=O)NC1CCCC1NC(c1cnc2n1CCCC2)=O 65081,C1(C(=O)NC(CNC(=O)Cc2sccc2Cl)C2CC2)CC=CC(O)C1 65082,C1(CC(=O)Nc2ncn(CCC)c2)CCN(C(c2cccc(OC)c2)=O)C1(C)C 65083,C(C1=CCN(C(=O)C(C)S(C)(=O)=O)CC1)NC(CCCc1scc(C)n1)=O 65084,N1(C(Cc2n(C)ncc2)=O)CC(=O)NCC1C(=O)NCCC(=O)NC1CC1 65085,C1(C(N(CC=C)CC2CC2)=O)CCOCC1NC(=O)CCC1CC1C 65086,C1(NC(C2CCC(C(=O)OC)C2)=O)C2CC1CN(C(c1ccc(F)c(F)c1)=O)C2 65087,C1(CC)C(C)CCN1C(=O)CN(CC(C)C)C(c1ccn(CCF)n1)=O 65088,C1(CNC(C2CC(OC)C2)=O)N(C(c2ccc(Cl)cc2Cl)=O)CCCC1(C)C 65089,c1(NCCCN2C(C)CCC2)cc(NCCNS(=O)(=O)C2CC2)ncn1 65090,C1(NC(C(C)NC(COC)=O)=O)CN(C(C2CC(C)(C)C2)=O)CCC1C(F)(F)F 65091,CC(O)C(C(=O)NCCNC(=O)C(=O)NC(N)=O)NC(C12CC(C)(CO1)C2)=O 65092,C#CCC(C)(CC)C(=O)NCC(C(=O)N(C)Cc1nc(C)ns1)C(C)C 65093,N1(C(c2cn(CC)nc2)=O)CCCC1(C)CNC(=O)CCSCc1ccccn1 65094,CCC(F)(F)C(C)(C)C(=O)NCCN(C)C.c1(CC=O)ccc2ncccc2c1 65095,C(C)(C(=O)N[SH](CCCC)CCSC)N(CC(=O)N(C(C)C)C(C)C)C 65096,C1(CNC(CCCC)=O)CCCC2(CN(c3ccc([N+](=O)[O-])c(Br)c3)C2)O1 65097,c1(C(=O)NC2CN(C(C3CCC3(F)F)=O)CC2CC2CC2)ccc(F)cc1F 65098,C1(NC(C2C(C=C)OCC2)=O)CCN(C(=O)CCC2CC(C)C2)CC1O 65099,C1(NC(CC=C)=O)CN(C(=O)Cc2cnc(Cl)cc2C)CCC1C(F)(F)F 65100,CC(C)(CC(=O)N1CC=CC(NC(c2cccc(-n3cccn3)n2)=O)C1)C1CC1 65101,c1(C(=O)NCC2CCN(C(C(C(C)C)OCC)=O)C2)cccc2nc[nH]c12 65102,C1(C)C(CC(C)C)CNC(=NCc2n(C=C)ncc2)N1.C1(C)CCC1.CO 65103,c1(NC(c2cnn(C)c2S(N)(=O)=O)c2n(CCC)nnn2)cc(Br)cc(C#N)c1 65104,N1(C(C2(CNC(CC(C)(C)C#N)=O)CCCO2)=O)CCC(O)C12CCC2 65105,c1(CC(C(C)C)NC(=O)NCC2CC(F)CN2)ccccc1C(F)(F)F 65106,C(=O)(C1=COCCO1)NC1CCC(N(C)C(c2cn(CCCF)nn2)=O)CC1 65107,C1(NC(C(N2CC(NC(C)=O)OCC2)C)=O)Cc2ccccc2C1OC 65108,c1(OCC)cc(C(=O)NC2CCC2CNC(=O)C(C)N2CC(C)C2)ccn1 65109,C1(C)(CNC(C2C(=C)CC2)=O)CC(F)(F)CN1C(=O)C=Cc1ccc(F)nc1 65110,C1(O)(CN(C(Cc2cc(C)sc2)=O)C)CCN(C(=O)CC(C)N(C)C)CC1 65111,Cc1cc(N(C)C)ccc1NC(=O)CC(=O)N(C(=O)CN1CCCC(C)C1)C(C)C 65112,C(=O)(CC(O)CNC(=O)CC1CSCCO1)N(C)Cc1scc(C)n1 65113,c1(C(CCO)NC(=O)CO)ccccc1OCc1ccc(F)cc1 65114,C=C(Cl)CC(C(=O)NC1CCCC1CN=[N+]=[N-])NC(=O)CC1CNC(=O)O1 65115,C=CC(C)CC(=O)NCCN(CCOC)C(c1ccn(C)c1)=O 65116,N1(C(c2c(COC)ccs2)=O)CC2C(CN(C)C(C3CCOC(C)C3)=O)C2C1 65117,c1(C(=O)NC2C3CN(C(C4=CC=CC(N)=CC4)=O)CC2C3)cnc2c(n1)CCCC2 65118,C1(CCNC(c2nc(C)oc2)c2nnnn2C(C)(C)C)CN(C)CCO1 65119,C#CC1(C(=O)NCCCc2ccccn2)CCN(C(c2ccc(Cl)cn2)=O)C1 65120,C=CCC(F)(F)C(=O)NC1CN(C(C2CC3CC2C3)=O)CC1OC 65121,CC(CC(=O)N1CCCCC1c1n[nH]cc1N(C=O)NC=O)C(C)(C)C.CCO 65122,C1(CCC(=O)N(CCCc2cnccn2)C)CCCCN1C(=O)Cc1ccc[nH]1 65123,C1(C(F)(F)F)(C(=O)NC)CCN(C(CCCn2cncn2)=O)C1 65124,N1(C(c2c(Cl)nn(C)c2Cl)=O)CCC2CN(C(=O)C3=COCCC3)CCC2C1 65125,C(=O)(C(CC)(CC)CO)N1C(C(NOCCOCC)=O)C(C)OCC1 65126,CN1CCN(C(C2C=CCCN2C(=O)C(C2(O)CCCC2)F)=O)CCC1=O 65127,C1(C(N(CCCNC(C(C)OC(C)(C)C)=O)C)=O)CCC(O)C1 65128,N(C1CCSc2ccc(Cl)cc21)CCCn1c(C)nnc1 65129,C(CCCCC(=O)N(C1CCN(C(=O)C(C2CCCCC2)N(C)C)C1)CC)=CC 65130,c1(C(=O)NCC2C3N(C(C4C(C#C)C4)=O)C(CC3)C2)ccc2nonc2c1 65131,c1(C(N2CCC(N(C(c3nccnc3N)=O)CC)CC2)=O)cccc(N)c1C 65132,C1(NC(CSCc2ccc(C)cc2)=O)CC(NC(C2(C3CC3)CC2)=O)C12CCC2 65133,c1(C(=O)NCC2C(CNC(c3ccc(C)cc3C)=O)C2)ccccc1P(C)(C)=O 65134,c1(C(N2C(CNC(CC(=O)NC)=O)CC(F)(F)C2)=O)c(C)nc2ncnn2c1C 65135,c1(OC)ccc(C(N2CCC3CCC23)C(=O)NCCc2ccccc2)c(Cl)c1O 65136,C(C(C)(C)C(=O)NC(c1ccco1)CNC(=O)CN1CC(C)C1)OC 65137,N1(C(c2cc(C(N)=O)[nH]c2)=O)CC2(C=C(C(=O)N3CC=CC3CN(C)C)CO2)C1 65138,c1(C(=O)NC(COC)CCO)cnc(CNC(c2cnn(C(F)F)c2)=O)nc1 65139,c1(C(=O)NCC2(O)CCN(C(=O)Cc3ccccc3)C2)ccc(Cl)c(Cl)c1 65140,c1(C(C)C)cccc(C(N2CCC(CCNC(C3CCC3CF)=O)CC2)=O)c1F 65141,C(=O)(C(C#N)C(C)C)NC(C1OCCN(C(c2cn(CC)nn2)=O)C1)C 65142,N1(C(c2c(CC)ocn2)=O)CCCC(N(C(=O)CC2(O)CCCCC2)CCO)C1 65143,Cc1cc(=NCC2(F)CC(CO)C2)[nH]c(=NCc2ccc(C#N)cn2)[nH]1 65144,CC(C)(C)S(=O)(=O)CC(=O)N(C1CCCCC1)CCNC(=O)C(F)C(F)(F)F 65145,C1(NC(C2CC3C=CC2N(C(c2cnc(Cl)s2)=O)C3)=O)CN2CCC1(F)CC2 65146,C(=O)(C(C(C)NC(=O)Cc1csnn1)C(C)C)NCC(=O)OCC 65147,Cc1cnc(C(=O)NC2CC3CC2N(C(c2nc(Cl)ccc2N)=O)C3)cc1C 65148,N1(C(C2C(C)(C)NC(=O)C2)=O)Cc2[nH]nc(C(=O)NC3(C)CC=CCC3)c2C1 65149,CC(C)(C)C(CNC(=O)C(F)(F)c1cccnc1)NC(C1CC2CC2C1)=O 65150,c1(C(N2C(CNC(c3scc(C(N)=O)n3)=O)CC3CC32)=O)nc(Cl)ccc1Cl 65151,CCCCC(C(=O)NC(C(N1CC2(CCC(=O)NC2)C1)=O)C(C)OC)C(C)C 65152,CCC(CC(=O)NOCC(=O)NC1CCC(OC)CC1)CC(C)C 65153,c1(OC)cc(CSCC(=O)N(C)O)cc(Cl)c1OC 65154,c1(NC(C(N2CCC(C)(C)C2)=O)=O)ccc(F)c(S(=O)(=O)N(C)C)c1 65155,CCC1=NOC(CNC(C2CCC(NC(c3c[nH]nc3OC)=O)CC2)=O)C1 65156,N1(C(COC(C)C)=O)CC2CCN(C(=O)CCCF)CC12 65157,C#CC(CNC(=O)CC1CCN1C(=O)CCc1cscn1)CC 65158,c1(C2(C(N(C3CN(C(c4c(C)[nH]cc4)=O)CC3F)C)=O)CC2)ccc(Cl)c(F)c1 65159,N1(C(c2cc(CCC)[nH]n2)=O)CCC(C2CC2)C1CNC(=O)CSC(C)C 65160,c1(C(N(CC(CC)NC(c2occc2C)=O)C)=O)sccc1Cl 65161,c1(C(N2CC3(C2)CN(C(C2CCOC2c2ccncc2)=O)C3)=O)ncnc(O)c1F 65162,c1(C(N2CCN(CC(=O)N(CCCCOC)C)CC2)=O)cccc(F)c1O 65163,c1(C(=O)NC(CC(C)C)(C)CNC(C2COC2)=O)ccc(S(=O)(=O)NCCO)s1 65164,Cc1oc2cc(C(N3CCC(C)N(C(=O)CC4(C)CCCO4)CC3)=O)[nH]c2c1C 65165,N1(C(C(CC2CCOCC2)NC(CC2CCCC(=O)N2)=O)=O)C2CC1CC1(CC1)C2 65166,N1(C(C(F)OC)=O)CCN(C(c2cc3n(n2)CCNC3=O)=O)CC(C)(F)C1 65167,c1(C(N2CCCCC2C(C)C)C(=O)NCC(=C)C)cccc2ccnn12 65168,C1(CNC(C2=CC(C)CC2)=O)CCC(C)(C)CN1C(c1nccc2ccsc12)=O 65169,c1(CC(=O)NC(CN(C(C(COCC)C)=O)C)(C)C)cc(F)c(N)cc1F 65170,CC(C(C)C(=O)N(C1CCCC1)C)NC(C1CN(C)CCO1)=O 65171,c1(C(N2CCC(C)C2CNC(c2ccc(O)nc2)=O)=O)n[nH]cc1[N+](=O)[O-] 65172,C1(COC)CN(C(C2C=CCN2C(=O)C(=CC2CCCC2)C)=O)CCO1 65173,C12(C(=O)NCC(CC)NC(c3cc4sccc4cn3)=O)C3CC(CC13)C2(F)F 65174,c1(C(NOC(C(C)C)CO)=O)ccnc(NC(=O)CCc2ncccc2F)c1 65175,N1(C(CC2OCCN(C(c3ccc(C)c(O)c3)=O)C2)=O)CC(C)C12CCOCC2 65176,Cc1cc(C(N2CCCC(CNC(=O)C=CC3CC3)C2)=O)cc(S(C)(=O)=O)c1F 65177,C(C1CN(C(=O)CSC2CC2)CC1C(=O)NC1CCCC1(F)F)=CC 65178,c1(CC(N2CCC(O)(CNC(CCS(C)=O)=O)C2)=O)ccc2c(c1)OCO2 65179,CCN=c1[nH]c(C(=O)NC(C2CCN(C(=O)CNC(C)=O)C2)C)cs1 65180,CC1CN2CCN1CC2C(=O)NCC1CCCCN1C(c1cnc(C(C)O)s1)=O 65181,C(C)(CCC(=O)N(CC(c1cn(C)nn1)=O)C)OCC.C1C(=O)N1 65182,c1(CCNCCNCC(C2CC2)OCC)ccsc1 65183,C(=O)(C(C(C)NC(=O)C(C)=CC1CC1)C(C)C)N1CC(OCC)(CO)C1 65184,c1(C(N(C2CCN(C(C3CC(SC)C3)=O)C2)C)=O)cn(C)nc1C(F)F 65185,c1(C(C(N2CCCC(NC(C(CCC)NC(C)=O)=O)C2)=O)=O)cc(Cl)cc(Cl)c1 65186,C(N=c1[nH]c2c(c(=NC3CCN(CC4CC4)CC3)[nH]1)CSC2)c1c(CC)nn(C)c1 65187,Cc1cnc(C(N2CCC3(CC3NC(=O)CCC(=O)N(C)C(C)C)C2)=O)c(C)c1 65188,N1(C(CCSCCC)=O)CC(CNC(=O)C(C)Cc2ccco2)(COC)C1 65189,c1(CN(C(c2cc(F)c(CO)c(F)c2)=O)CC)ncccc1S(C)(=O)=O 65190,C(C)(C(C)(C)C(=O)N(CC(Cl)Cl)C)NC(Cc1nc(C)oc1)=O 65191,C1(CC(=O)NC(C(=O)N(CC(C)(C)O)CC)CC2CCC2)CC(=O)NC1=O 65192,n1(CC(=O)N(C2(C3CC(F)C3)CC2)CC)c(=O)n(C)c(=O)c2ccccc12 65193,c1(OC)c(C(=O)NC(C)(CNC(c2ccc(C3CC3)o2)=O)C(C)C)csc1Cl 65194,CC1(O)CCC(C(=O)NCCN(C23CC(F)(C2)C3)C(c2ccc(Cl)nc2)=O)CC1 65195,CNS(=O)(=O)N1CCN(CC(N2CCCCC2c2ccc(OC)nc2)=O)CC1 65196,N1(C(CCC(=O)NCC)=O)Cc2occ(C(=O)NC3CCCC(F)(F)C3)c2C1 65197,c1(CC)cccc2c(C(=O)NCC3CCC3NC(=O)C(C)(CC)CO)c[nH]c12 65198,c1(C(=O)NC2(OC)CC3CCC2CC3)c(OC)c(O)nc2ccccc12 65199,CC(C)C(CO)C(=O)N1CCCCC1CNC(=O)CCn1cnccc1=O 65200,C1(NC(CCN2CCN(C)CC2)=O)COCCN(C(C2CCCCN2C)=O)C1 65201,N1(C(CC2(C#N)CCC2)=O)CCCC(N(C(=O)COC(F)F)CCF)C1 65202,CN1CC=C(CC(=O)N2C3CCCC2CC(NC(=O)Cc2ccccc2)C3)CC1 65203,CCC(C)(C)C(O)C(=O)N1CCC(C(F)F)(CNC(C2CC3(CCCO3)C2)=O)C1 65204,C1(COC)(CO)CCCN1C(C1CCN(C(C2(CCN=[N+]=[N-])CC2)=O)C1)=O 65205,c1(C(N2C(CNC(c3cccc(F)n3)=O)CC2)=O)ccc2cc[nH]c2c1 65206,C1(C(=O)NC(CNC(c2cc(COC)on2)=O)C2CC2)(CO)CCCNS1(=O)=O 65207,c1(C(=O)NCC2(F)CC(CNC(C(CC#C)C)=O)C2)n[nH]c2ccc(F)cc12 65208,N1(C(Cn2ncc(C)c2)=O)C(C(=O)NC2CC(=O)NC2=O)CCC12CC2 65209,N1(C(=O)C=Cc2ccoc2)CCC2C(CCN2CC(O)CCc2ccccc2)C1 65210,C1(CNC(c2csnc2Cl)=O)CN2CCCCC2CN1C(=O)CCN1CCCC1 65211,C1(C(N(CCCNC(=O)C(C2CCCCCC2)O)C(C)C)=O)CCS(=O)(=O)CC1 65212,Cc1cc(C(=O)NC(C2CCOC2)CNC(c2cc(CO)n(C)n2)=O)ccn1 65213,C(C)(C)(CC(=O)NOC1CCCC1)N(C(CC(C)CN(C)C)=O)C 65214,Cc1cc(C)c(C#N)c(NC(=O)Cc2csc(C)n2)n1 65215,C1(C(C)(C)C)CC(C(=O)N2CCC(CO)(CNC(=O)Cc3cnoc3)CC2)=NO1 65216,CCC(C(=O)N(C(C)CN(C)C(c1cnn(CC)c1)=O)C)NC 65217,Cc1sncc1C(=O)NCCCN(C)C(C1CC1(C)C)=O 65218,N1(C(C(CCC)C)=O)CC(NC(=O)C#CC2(CC)COC2)C2CCCCC12 65219,C1(C(=O)Nc2ccc(O)nc2)(CC)CCN(C(=O)CCCC2CCCO2)CC1 65220,c1(CCC(=O)NC2C(OC)CCC2)cnc2n1CCCC2 65221,CC1C(NC(c2nn(C(F)F)cc2Cl)=O)CCCN1C(=O)C(C)Cc1cnc[nH]1 65222,S(=O)(=O)(CC(=O)N1CCC(C)C1CNC(c1cccc(NS(N)(=O)=O)n1)=O)NC 65223,c1(C(N(CC(C)NC(=O)C2=C(Cl)CCC2)C)=O)ccc2c(c1)CCCC2=O 65224,c1(C(=O)NC2CC(C)(CNC(C3CCN(CC)C3)=O)C2)cc2cncn2c(O)n1 65225,N1(C(C(N2CCOCC2)C)=O)CCCC(O)(CNC(=O)C2=CSCCO2)C1 65226,CC1CC(CNC(=O)CCOCC2CC2)CN(C(C2(C(C)C)CCC2)=O)C1 65227,CC(C)C(CCNC(C1CCCN1N=O)=O)N=c1nc(C2CCOCC2)[nH]s1 65228,N1(C(CCC(C)N(C)C)=O)CC2(CCCN2C(c2sccc2CN(C)C)=O)C1 65229,c1(CCC)nsc(N(C2CC2)CC2CCCN2C(=O)CC2CCCCO2)n1 65230,c1(CC)nc(C)c(C(N2CCCCC2CNC(=O)Cn2cnnc2O)=O)c(C)n1 65231,N12CCCCC(C1)C2=O.c1(OCC)nccc(N2CC(c3ccc(O)cc3)C2)n1 65232,C(N=c1ccc(C(N2CCCC(Br)C2)=O)c[nH]1)c1ccc(N(C)C)cc1F 65233,N1(C)C(=O)CNC1=O.N1(C(C(=O)OC2CC(CCC(=O)OC)C2)C2CC2)CCCCC1 65234,N1(C(c2ncsc2C(=O)NCCC2(CC)CC2)=O)CCN(C)CC1C 65235,n1(CC#C)c(C)cc(C(=O)NCCN(CC(CC)NC(=O)C2CC2)C(C)=O)c1C 65236,N1(CC)CC(C(=O)N(C(CC)CC(=O)NCC2(COC)CCCC2)C)CC1=O 65237,N1(C(c2c(C)nn(CC)c2C)=O)CC(NC(c2n[nH]c(C)c2C)=O)C2(CCC2)C1 65238,Cn1cc(C2CC2C(N2CC(C)(NC(=O)COc3nc[nH]n3)C2)=O)cn1 65239,N1(C(CCCCC)=O)CCC(C2CCN(C(C3CNC(=O)N3C)=O)CC2)C1 65240,C1(CCC)CN(C(=O)Cn2cc(Cl)cn2)CCN1C(=O)CN1CCC(C)(C)C1 65241,CCC(CC)C(CNC(=O)C(=O)NC(c1cccc(F)c1F)C)N1CCOCC1 65242,N1(C(C=C(C)c2ccccc2F)=O)CCCCC2(CCN(C(C3CCO3)=O)C2)C1 65243,c1(NC(C23CC(NC(C4(C)CCN(C)CC4)=O)C2C3)=O)n[nH]c2c1COCC2 65244,CC1=NOC2(CCN(c3cc(C(F)(F)F)ccc3[N+](=O)[O-])CC2)C1 65245,C1(Nc2ccc(C(=O)OC)cn2)(CNC(=O)Cn2cnnc2)CCCCC1C 65246,c1(C(n2ccnc2)CNC(=O)NC(c2ccccc2)COC)cc(Cl)ccc1Cl 65247,c1(C(N2CC(O)(CCNC(CC(c3ccccc3F)C)=O)C2)=O)ncc(F)cn1 65248,C(CNC(C1CCOC2(CCC2)C1)(C)C)(CCS(C)(=O)=O)OCC 65249,C=CCCN=C(NCCC(=C)C)NC1CC(CCC(=O)OC)C1 65250,C1(NC(c2cnc(C3CC3)nc2)=O)CCCCC12CCN(C(=O)C=CI)C2 65251,c1(C(N(C2CCCC2)CCNC(c2ccsn2)=O)=O)ccc(O)nn1 65252,C=CCC(C)(C)CC(C(=O)NC1CC(F)(F)C1)NC(CCC)C(C)(C)C 65253,C(=O)(CCCCN(C)C(C1CCC1)=O)NCCNC(CC1CN(C(C)=O)C1)=O 65254,C1(CNC(C2N(CC#C)CCC2)=O)CN(C(c2csc(COC)n2)=O)CCN1C 65255,c1(NC(C2CCC2)=O)ccnc(CCn2cc(CC3CCCNC3)nn2)c1 65256,N1(C(C(CCC)OCC)=O)C2CCC1CN(Cc1nc(Cl)sc1Cl)CC2 65257,N1(C(c2cc(C)sc2)=O)C2CCC(C(=O)NCc3cncc(Cl)c3)C1CC2 65258,c1(C(=O)NC2CC(CNC(C(CC)(C)O)=O)C2(C)C)ccc(OC(F)F)c(Cl)c1 65259,CC1CC(NC(=O)CCP(C)(C)=O)CN(C(=O)COc2ccc(Cl)nc2)C1 65260,N1(C(C2CC2NCc2cc(Cl)cc(Cl)c2)=O)CCN2CCOCC2C1 65261,c1(NC(c2nnc(N(CCN(C(C)C)C(C)C)C)s2)=O)ccccc1C1CC1(F)F 65262,N1(C(C(CSC)O)=O)CC2(CCCC2NC(=O)Cc2ccnc(F)c2F)C1 65263,CC(C)C(C)(C)C(=O)NC1CC(CNC(C2(C)CC3CCC2C3)=O)C1 65264,Cc1nccc(Cl)c1C(=O)NCCNC(=O)CC1(O)CCC1 65265,CON1CC(C(=O)NCCC(=O)OCCF)CC1=O.C(C)(C)C 65266,CON(CCC(=O)NC1CC(N2CCOCC2)C1)C(=O)COc1ccc(O)cc1 65267,C1(NC(C(C)OCCOCC)=O)CC2CN(C(c3nc(Cl)sc3C)=O)CC2C1 65268,C1(C(N(CC(C)(O)C2CC2)C)=O)CCCC1NC(=O)CC(=O)NC1CC1 65269,O=C1NC(=O)C2(CCC(C(=O)NC(N3C4C(NC(=O)C(Cl)(Cl)Cl)C(C4)C3)=O)CC2)N1 65270,c1(OC)cccc(C(C(N2CC(N(C(c3sc(C)cc3Cl)=O)C3CC3)C2)=O)OC)c1 65271,N1(C(CC2CCC(NC(c3[nH]cc(C)c3)=O)C2)=O)CC(S(C)(=N)=O)C1 65272,c1(C(=O)NC2CCC(CCNC(CS(=O)(=O)NC)=O)C2)cc2ccc(C)cc2o1 65273,c1(C(C)C)ccc(C(N2CCC(C(=O)O)C2(C)C)=O)c(N2CCC(=O)NC2=O)c1 65274,c1(OC)ccc(C=CC(=O)NC2(CO)CN(C(=O)Cc3cnc[nH]3)C2)c(OC)c1 65275,C(CC(=O)NC1CC(CSC)C1)N(C(=O)CC1CC1(C)C)CC 65276,c1(OC)ccc(C(=O)NCC2CC(C)N(C(=O)Cc3ccnc(NC)c3)C2)cc1 65277,CC(C)C(C(C)NC(=O)CCC(F)F)NC(=O)C(=C1CCCCC1)F 65278,Cc1cc(O)ncc1C(N1CC(C(=O)NC(c2cccs2)C)CCC1C)=O 65279,Cc1ccc(C(=O)OCCOC2CC(C(F)(F)F)N2)c([N+](=O)[O-])c1 65280,C1(NC(c2ccc(CC)s2)=O)CCC2(CC1)CN(C(=O)CNc1ccccn1)C2 65281,c1(COC)nc(NCCC2CC(F)C2)cc(=NC2CCN(S(C)(=O)=O)CC2)[nH]1 65282,N#Cc1cncc(CNC(C2CCN2C(=O)CC2CC3CCC2CC3)=O)c1 65283,N1(C(C2(C(=O)N(C)CCc3nccs3)CC2)=O)CC2CC2(CN)C1 65284,C1(C(=O)Nc2cccc(NC(C(CC)(C)CC)=O)c2)CC2CCCCN2C1 65285,C1(CNC(c2cnn(CC)n2)=O)CN(C(=O)C(C)CC(F)F)C2CCCC2O1 65286,C1(NC(C(C)C)=O)CCCC1(C)CN(C(=O)CCSCC(N)=O)C 65287,c1(CC(=O)NC2CC(N(C(c3c[nH]c(=NC)o3)=O)C)C2)c(OC)cccc1Cl 65288,C1(C(=O)Nc2cn(CC(C)C)nc2)CC2(CCN1C(c1ccsn1)=O)CC2 65289,C1(C(=O)NCC(CN(C(CSCC(=O)OC)=O)C2CC2)O)CNC(=O)N1 65290,N1(C(c2ccc(NC=O)cc2)=O)CCC(CNC(=O)C(F)C2CCC2)C12CCC2 65291,C#CC1(O)CCCN(C(C2CC3(CC(NC(c4cc[n+]([O-])cc4)=O)C3)C2)=O)C1 65292,C(=O)(C#CC1CCCCO1)NCCCC1OCCN(C(c2c(C)nc(O)[nH]2)=O)C1 65293,CC1(C)C(C(=O)NCC(O)CNC(C2(C)CCC(=O)N2)=O)CCS1(=O)=O 65294,[N-]=[N+]=NCCC(=O)NC(c1cccnc1)C(N1CC(CO)CCC1)=O 65295,Cc1cnncc1C(N1CC(C(N)=O)(CNC(C2(C)CCCCO2)=O)C1)=O 65296,Cc1ccc(C(N2CC(N(C)C(c3ncn4c3CCCC4)=O)C2)=O)c2c1CCC2 65297,c1(NC(C2(C)CCN(C(c3ccc(OC)nn3)=O)C2)=O)cccc(F)c1O 65298,C(CC(=O)NOCC1CCCO1)(C1CC1)NC(C1(CC#C)CCCO1)=O 65299,N1(C(c2onc(CC)c2C)=O)CCCC2C(CCCN2C(c2ncsc2C)=O)C1 65300,C1(NC(C(C)OCC)=O)CCN(C(=O)C(C)(C)Oc2ccccc2)C12CCC2 65301,N1(C(C2(C)CC=CC2)=O)CC2(CC2)CC1CNC(=O)CC1CC2(CCC2)CO1 65302,Cc1cc(C(=O)N(CCC(c2cccs2)NC(=O)CCC(F)F)C)c(Cl)cn1 65303,c1(CNC(c2ccn(CC(F)(F)F)n2)=O)csc(CNC(C2CC2Cl)=O)n1 65304,C=CCC(CC=C)C(=O)NCCC1CCCN(C(C2(OC)CS(=O)(=O)C2)=O)CC1 65305,C(=O)(C1CCCc2nncn21)NC1CC(NC(C2(C)CCSCC2)=O)C1 65306,N1(C(C(COC)(F)F)=O)CCN2C(=O)C(NC(c3cc(C)ncn3)=O)CC2C1 65307,O=C1CC(CC(=O)N2CC(O)(Nc3ncc(I)cn3)C2)c2ccccc2N1 65308,c1(C(=O)NC(CNC(CNS(CC)(=O)=O)=O)(C)C)ccccc1 65309,C(=O)(CC1NCc2ccccc21)OC(=O)C(F)(F)C(C(C)C)CC 65310,c1(C(=O)NC2CC(CCNC(C(C=CCCC)O)=O)C2)cccc2nccn12 65311,C(c1cnc2ccccc2n1)=CC(=O)NC1CN(C(CCOC)=O)C2(C1)CCC2 65312,c1(NC)cc(C(N2CCN(CCNC(=O)CC3CC(OC)C3)CC2)=O)cc(Cl)n1 65313,CCC(=O)CCC(=O)N1CCOCC1CCNC(=O)CCc1cccc(C)c1 65314,C1(C(N2CCC(C(C)(C)O)C2)=O)(CC)CN(C(=O)Cc2ccccc2)C1 65315,Cc1ccc(C(N2CCC3CCCC23CNC(c2nc(Cl)cs2)=O)=O)c(=O)n1C 65316,CC1CN(C)CC(C(=O)NCCCNC(c2cn(C)nc2I)=O)O1 65317,c1(CCC)n[nH]c(=NCC(C)(C)NC(c2cnc(F)c(F)c2)=O)s1 65318,Cc1ncsc1C=CC(N1CCCC1(C)CNC(=O)CC1CCCCN1C)=O 65319,N1(CC(C)NC(=O)C(=O)N(c2ncnn2C)C)CCc2ccccc2C1 65320,N1(C(C(C)SC(F)(F)F)=O)CC(C2(NC(=O)CCc3ccc(Cl)s3)CC2)C1 65321,S(=O)(=O)(c1cc(F)cc(Br)c1)NC1CC(C(=O)NCC2CCCCC2)C1 65322,Cc1ccc2nc(C(=O)NC(C)(C)CN(C(=O)C(C)C#N)C)ccc2c1 65323,N1(CC)CCOC(C(N2CCC(CNC(c3cc(C)sn3)=O)C2)=O)C1 65324,N1(C(c2c(C)cccc2Cl)=O)CC2(CCN(C(=O)CC(C)(F)F)CC2CO)C1 65325,C1(NC(C(C)=CC)=O)C2CCC1N(C(c1ccc(OC)c(OCC3CC3)c1)=O)C2 65326,C(=O)(C(C)(F)C(=O)N1CCCC(CNC(c2nc(OC)ccc2C)=O)C1)OC 65327,CS(=O)(=O)C1(C(=O)NCC2(NC(C3CC(=C(F)F)C3)=O)CCOC2)CC1 65328,c1(NC(CNC(N2C(C)CCOC2)=O)=O)cccc(Cl)c1F 65329,C(=O)(C(C)(C)C)NC1CC(N(C(=O)OC)CC2CC=CCC2)C1 65330,N1(C(C2CN(C(Cc3c(C)ocn3)=O)C(C)CO2)=O)CCN(C)C2(CC2)C1 65331,N1(C(=O)C=CC2CCCO2)CCOCC(NC(=O)C(F)(F)Cl)C1 65332,C(=O)(CC(C)(C)CC(F)F)N1CC2(C(NC(C(C)=CC3CC3)=O)CCC2)C1 65333,C1(OC)CCCCCN(C(CC2CC(F)(F)C2)C(=O)NCC2CCOCC2)C1 65334,c1(C(N2C(CNC(=O)Cc3cncnc3)CC2)=O)ccc2c(c1)NCCC2 65335,C1(C)(CC)C=C(C(=O)NC2CCCN(C(c3ccc(CN(C)C)o3)=O)C2CC)C1 65336,Cc1n[nH]c(C)c1CC(N1CCC(c2ccccc2)(NC(C2CC23CC3)=O)C1)=O 65337,N1(C(CON(c2cc(C)nn2C)C)=O)CCCN(C(C2CCCC23CC3)=O)CC1 65338,CCCC(C(O)C(=O)N1CCOCC1C(C)C)NC(c1c(F)cncc1F)=O 65339,N1(C(CCCC#C)=O)CCCCCC1CNC(c1cc(C)nnc1CC)=O 65340,N1(C(C2(NC(c3scc(C)c3C)=O)CC(CO)C2)=O)CCCC(C)(O)C1 65341,N1(C(=O)NC2CCCC2(F)F)CCC2CCC(C1)O2 65342,C(=O)(C1=CC2(CCOCC2)C1)NCC1(C(N)=O)CN(C(C(CC)(C)F)=O)C1 65343,c1(C(=O)NC2C(C)CN(C(c3cccnc3)=O)CC2)c(Cl)ccc(Cl)c1O 65344,c1(C(=O)NC(C2CC2NC2CCCCCC2)C)cccc(CNC(=O)C2CC2)c1F 65345,C1(CNC(c2cn(C3CCC3O)nn2)=O)CCCCN(C(C2CC2C2CC2)=O)C1 65346,Cn1ccnc1C(C1CCCC1)NC(=O)C(N)CC1CCOC1 65347,C(=O)(C(C)CC(F)(F)F)NC(CC(C)C)CNC(=O)CCc1cscn1 65348,N#Cc1c(F)cc(NCC(O)CN2CCN(CCCc3nccs3)CC2)cc1Br 65349,CC1C(C(=O)NCCCCCCF)CCCN1C(C1CCCC(=O)N1C)=O 65350,CC1CC(NC(=O)Nc2ccccc2COCCO)CCN1CC(N)=O 65351,C1(CC=C)(C(=O)NCC2CCC(C)C2)CN(C(=O)C(C2CCCC2)OC)C1 65352,CON1CC(C(=O)NC(C(N2CCC(C)(C(C)C)C2)=O)c2ccco2)CC1=O 65353,C(=O)(C(C)(O)CCN(C)C)N1CC(C(C(=O)NCCC(C)(C)OC)O)C1 65354,c1(C(=O)NC2CN(C(C3C(C(=O)OCC)C3)=O)C2)ccccc1Br 65355,N1(C(C2(COCC)CC2)=O)CCCCC(N(C)C(C2CCCC2(F)F)=O)C1 65356,c1(C(=O)NCC2(CO)CCN(C(C3(C)ON=C(C)C3)=O)C2)c(Cl)ccc(F)c1N 65357,CC(CCCCNC(=O)C(C)CCOC)NC(C1(c2cccc(Cl)c2)CC1)=O 65358,C#Cc1ccc(CNC(C2C(O)CCN2C(=O)CC(F)(F)F)=O)cc1 65359,Cc1ccc(C=CC(N2CCC(C(C(N3CC(NC(=O)C4CC4)C3)=O)O)CC2)=O)o1 65360,C1(NC(c2c(C#C)c[nH]n2)=O)CC2CN(C(=O)COCC(F)(F)F)CC12 65361,c1(C(N(C(C)CNC(c2cc(O)nc(O)c2)=O)C)=O)ccc(F)c2ccncc12 65362,Cc1cc(Cl)c(Br)cc1S(=O)(=O)NCC1(CN)CCCCCC1 65363,c1(C(=O)NCCN(C(=O)C(F)(F)c2ccccc2)CC)cccc(F)c1N 65364,C1(C(=O)NCc2cn(C)nc2)CC(NC(c2cnccn2)=O)C1(C)C 65365,CC1CCCC1CC(=O)NCC(C)(F)CNC(=O)Cc1cccs1 65366,C(CS(=O)(=O)CC(=O)N(CC(C)O)CCNC(c1c(C)ncn1O)=O)OC 65367,C(=O)(CCCCNC(N)=O)NC(C(=O)NC)C1CN(C(C2(CSC)CC2)=O)C1 65368,c1(NC(C(=O)NCCC(OCC)OCC)=O)cc(C)n(-c2ccc(Cl)cc2)c1C 65369,c1(OC)ccc(C(C)C(=O)NCCCCCNC(=O)CSC2CC2)c(C)c1 65370,c1(C(N2CCN(C3N(C(=O)CCC45CC(C4)C5)CC3)CC2)=O)ccc2nc[nH]c2n1 65371,C(=O)(C(C)(O)C(C)C)NCC(C(N1CC(CC#C)OCC1)=O)Cc1cnn(C)c1 65372,c1(C(N(C(C)CNC(=O)C=Cc2ccnn2C)CC)=O)ccc(C(C)C)cn1 65373,C12CCCN(C1)C(=O)CO2.C(C)(C)(C(=O)NC1CC1CSCc1cccs1)OCC.OC 65374,CCC(CC(=O)NC1CC2CCC1CC2NC(c1cn(CC)nn1)=O)C(C)C 65375,Fc1c(I)c(-c2cc(=NCC3(CO)CCOC3)[nH]cn2)cc2ccccc12 65376,c1(C(=O)NCCN(C(c2ncccc2N)=O)CC)cnn(C)c1F 65377,CN1CCC(F)(CNC(=O)C=CCN(C(=O)C(c2cnn(C)c2)O)C)C1 65378,CC1OC2(C(=O)NCC3CC(O)(CNC(C4(C)COC(=O)C4)=O)C3)CC1C2 65379,C1(NC(=O)COC2CC(F)(F)C2)(CF)CCN(C(=O)CC2CCC(=O)O2)C1 65380,Nc1ccc(-c2nc(C(N3CCCC3C3CCC3)=O)cs2)nc1 65381,CCCC(C(=O)NC1CC2(CCCN(C(=O)C(C)(C)S(C)(=O)=O)C2)C1)S(N)(=O)=O 65382,c1(C(=O)NC2CC(NC(C(CCC)OCC)=O)C(O)C2)ccc(C2CC2)c(C)c1 65383,C=CCCCCCCC(=O)NC(C1CCN(C(=O)CCC(=C)C)C1)(C)C 65384,c1(C(=O)NC(C(C)NC(C(C)OCCOC)=O)C)cccc2c1CC(=O)N2 65385,C1(C(=O)NCC(C)(C2CC2)NC(c2cccc(CC#N)c2)=O)(CO)CCCCC1 65386,N1(CC(=O)NCC2(F)CCCN(C(=O)CCc3ccsc3)C2)CCC(=O)NC1=O 65387,C1(C(C(=O)CCN(CC(F)F)C(C2CC2C2CCCO2)=O)=O)CCS1(=O)=O.NC 65388,CN1CCc2[nH]c(=NCC3(C(=O)Nc4ccnn4C)CC3)c(C#N)cc2C1 65389,c1(OCC(=O)NCC(C)N(C)C(C2CCC(CN(C)C)O2)=O)ccc(Br)cc1 65390,N1(C(c2c(OC)cccc2)=O)CC2CN(C(C3CC4(CCC4)CN3C)=O)CC2C1 65391,N1(C(C(C(C)C)C#N)=O)CCc2nc(CNC(=O)CCn3ccnn3)sc2C1 65392,c1(C(=O)N)cncc2ccsc12.c1(CNC(C)=O)ccc(C(=O)NCC2(C)CC2)o1 65393,Cn1cnc2[nH]c(C(N3CC(NC(C4SCCCS4)=O)CC(F)C3)=O)cc12 65394,C1(NC(C)=O)CCN(C(C2COCC2NC(=O)C(=CC2CCCC2)C)=O)C1 65395,c1(C(N2CCC(C(C)NC(CCC=C(C)C)=O)C2)=O)cc(C)c(N)cc1F 65396,C1(C(=O)NCCC2CCOC2)CC2(CC2)CN1C(=O)C=CC(F)F 65397,C=CCC(C)(C)CC(=O)NC(C)(C)C(C)NC(c1cn(C)c(C(F)F)n1)=O 65398,Cc1nnc(C(c2nnnn2CC2CCOC2)NCC(Cl)Cl)n1C 65399,N1(C(CS(CCC)(=O)=O)=O)CCC2CCN(C(C3CC4CCC3C43CC3)=O)C2C1 65400,c1(C(N(CCCOCCN(C(C=CC(CC)C)=O)C)C)=O)cn(C)nc1Cl 65401,C1(Cc2cn(CC(=C)O)nn2)CCCCN1C(c1scnc1C(F)F)=O 65402,c1(C(N2CC(CNC(C3(OC)CC3)=O)CC2(C)C)=O)ccc2nonc2c1 65403,N1(C(C(C2CCCC2)NC(CCCCC)=O)=O)CC2(CCC(=O)NC2)C1 65404,c1(C(N2C3CN(C(C(C=C)(C)C)=O)CC2CC3)=O)c(Cl)c([N+](=O)[O-])nn1C 65405,CC1=NOC(C(=O)NC(CNC(C2CC(NS(C)(=O)=O)C2)=O)C(C)(C)C)C1C 65406,N1(C(c2c(C)nc(COC)s2)=O)CCC(C2CC2)C1CNC(C1CC1C(C)O)=O 65407,c1(CCC(=O)NCC(CN(C(c2nc(CCC)sc2)=O)C)O)nnc(S)nc1O 65408,C(=O)(N=c1[nH]c(=NCCc2ccc(C#N)cc2)[nH]cc1Br)c1nn(C)c(Cl)c1 65409,N1(C(c2ncc(-c3cn(CCN4CCOCC4)nn3)s2)=O)CCCCC1CF 65410,c1(C(N2CC3CCCN(C(=O)CC4CCOC4)C3C2)=O)ccc2c(c1F)CCC2 65411,CCC(C)(C#N)C(=O)NC1CC(NC(c2cc(Cl)ccc2OC)=O)C1 65412,c1(CNC2C(c3c(C)ccc(C)c3)CCC2)ccccc1S(=O)(=O)N1CCOCC1 65413,N1(C(CC(C)OC)=O)CC(NC(=O)CC23CCCN2CCC3)CCC1C 65414,N1(C(=O)C(C2CCC2)C2CC2)C(C(=O)NCc2nccs2)CCC1C1CC1 65415,C1(C(=O)NC2(CC=C)CN(C(c3cc(C(=O)OC)no3)=O)C2)CC(C)OC1C 65416,c1(CC)cc(C(=O)NC2CC2NC(=O)C(C)OCc2cccc(C)c2)c(C)o1 65417,C1(C(=O)NC(C(CC)C)CO)CC(C)(C)CCN1C(c1cc(O)nn1C)=O 65418,c1(C(=O)NCCCN(C(C2C(C)COCC2)=O)C)ccc(F)c(Br)c1F 65419,C1(CCC)(CO)CCCN1C(C1CN(C(c2coc(C)n2)=O)CC1F)=O 65420,c1(C(N2CC(CC(C)=O)C2)=O)nn(C)c(N)c1C 65421,C(CC(=O)N1CC2(CNC(=O)N2)C1)(C(F)(F)F)NC(C(=Cc1ccccc1)C)=O 65422,Nc1ccnn1CC(=O)NCC1CC1NC(c1occc1-c1ccccc1)=O 65423,c1(C(N(CCCN(C(=O)Cc2ccc(F)c(Cl)c2)C)C)=O)nc2cnccc2s1 65424,CN=c1[nH]c(NC(=O)NC2CCCC2Cc2ccccc2)ncc1Cl 65425,N1(C(CC2C(=O)OCC2)=O)CC2(CC(C(=O)NCC34CCC(CC3)CC4)CO2)C1 65426,Cc1cc(Br)c(F)cc1C(=O)NC1CC(NC(=O)CCOC(C)C)C1 65427,C1(OCC)CC2(C1)CC2C(N1CC(OCC)C1)=O.N1(CC(=O)NCCS)CCC1C 65428,C#CC1(C(N2CCOCCC2C)=O)CCN(C(=O)CCCn2cccc2)C1 65429,CC1CCCC(CC(=O)NCCC2CCN(C(=O)COc3cn[nH]c3)CC2)O1 65430,c1(CNC(N(CC(c2ccccc2)COC)C)=O)cc(C2CC2C)on1 65431,C(C(CNC(=O)Cc1ncccc1F)C(F)(F)F)NC(c1ccc(COC)o1)=O 65432,C1(F)(CNC(CC(C)NC(C)=O)=O)CCN(C(=O)C(C)C(C)(C)C)CC1 65433,C1(NC(C=CC=CCC)=O)CC12CCN(C(=O)C(COC)COC)C2 65434,CN=c1cc(C(=O)NC2CC(C)N(C(C3CCC(OC)CC3)=O)C2)cc[nH]1 65435,N1(C(=O)CCc2cccnc2)CC2(C1)CN(C(C1(CCO)CC1)=O)CCO2 65436,c1(C(c2nnnn2C2(C)CC2)NC(C=C)C2CCC2)cn(C)nc1C(F)F 65437,CCC(C(=O)Nc1ccc(C(C)C)c(Cl)c1)C(C)C 65438,C1(C(N2CC(N(C)C(c3ccc(F)cc3F)=O)C2)=O)CCc2cncn2C1 65439,Cc1ccc(NCC(c2nnnn2C2CC2)(C)NC(=O)Nc2ccncc2)cc1 65440,C1(NC(C=CC(C)(C)SC)=O)COCCC1NC(=O)C(C)(O)C1CC1 65441,C1(OCC(N2CCC3CNCC23)=O)CCCC2(CCOCC2)O1.c1c[nH]c2cnccc12 65442,C1(NC2(C(=O)NC(CSC)CSC)CCCC2)CCN(C(=O)OC(C)(C)C)CC1 65443,C1(CNC(C(CC)N(C)C)=O)CCC2(CN(C(c3cc(C)c(Br)s3)=O)C2)O1 65444,CC1=CCC(NC(=O)CN(C(=O)C(C)C)C)CC1.C1(C(C)C)C(=O)N1 65445,C1(C(N2CC(C(=O)NC3CCCC(SC)C3)(COC)C2)=O)CCCS(=O)(=O)C1 65446,Cc1ncncc1C(=O)NC(C1CC=CCC1)C(=O)N(C1CCN(C2CC2)C1)C 65447,C1(CC(=O)N(C2CCC2)C)CCN(C(=O)CCc2ccn(C)n2)CC1 65448,C(=O)(C(C)=NOCC#N)NCC(CC)N(C(=O)C(O)CN(C)C)C 65449,N1(Cc2cn(C)nc2C2(CO)CCCC2)CC(=O)N(CCCC2CCOC2)C1=O 65450,N1(C(CC(=O)NCC)=O)CCCC1(C)C(=O)NC(C1(OC)CCC1)C 65451,Cc1cc(=O)oc(C)c1C(=O)NCC1CC1NC(=O)Cc1ccccc1Br 65452,C1(F)(C(N2CCC(C)(CCNC(C3(C#C)CCC3)=O)C2)=O)CCCN(C)C1 65453,c1(C(=O)NCCCN(C(=O)C(C)(O)C2CCOC2)CC)scnc1Cl 65454,c1(NC(=O)NC(COC)C(=O)Nc2cccc(NC(C)=O)c2)cnc(Cl)cc1Cl 65455,CCCC(CCC)C(=O)N1CCC(C(=O)N(C(C)CC(C)C)C)O1 65456,C1(CCNC(C2CC(=O)NC2)=O)CCCCN1C(=O)CCNc1cncnc1 65457,c1(OC(C)C(=O)N(C2CC2)CC2CC(F)CN2C(=O)C2=CCC2)cccc(Cl)c1 65458,c1(OCC(=O)NC2C(NC(=O)OC(C)(C)C)C2)ccc(F)c(C=O)c1 65459,N1(C(C(C)O)=O)CCCC(C2CCCN(C(=O)C(N3CCN(C)CC3)C)C2)C1 65460,C(CC(F)F)(C(=O)NCCCN1CCCCC1)N(C)C(c1cncs1)=O 65461,c1(C(=O)NCC(CCOC)NC(c2oc(C)nc2C)=O)ccc(C(C)C)nc1O 65462,N1(C(c2nnc(C)s2)C)CCC(NC(c2cccc(F)c2Cl)=O)C(C)C1 65463,C(CNC(c1cncnc1)=O)(CC(F)(F)F)NC(c1cnc(CC(C)C)s1)=O 65464,C=CC(C)(CC)C(=O)N(CCNC(c1ccc(CS(C)(=O)=O)o1)=O)CCOC 65465,n1(CC(n2cc(C3(F)CCN(C(C(C)C4CC4)=O)C3)nn2)=O)cc(Br)ccc1=O 65466,c1(C(N(CC(C)NC(C2C3CCCCCC23)=O)C)=O)cccc2c1COC2 65467,c1(C(=O)NCCC2(NC(C3CC(C)C3)=O)CCCC2)cc2n(c1)CCOC2 65468,C1(CNS(=O)(=O)CC2CCC2)CC2(C1)CN(Cc1cc(O)ncc1Br)C2 65469,C(=O)(C(CC)C(C)(C)CC)NCC(CNC(C(C)OCC#C)=O)OC 65470,C1(SC)CN(C(c2cncnc2)=O)CC1NC(c1ccc(-c2ccon2)cc1)=O 65471,C1(OCCCOC)CCN(C(C2CC(NC(C(c3cccnc3)OC)=O)C2)=O)C1 65472,Cc1cc(Cl)ccc1CC(=O)NCc1ccc(O)cc1F 65473,CCC(C)CC(C)C(=O)NCC(C(C)C)NC(c1n[nH]c(C)c1Cl)=O 65474,c1(NC(c2c(CC(=O)OCCN(C)C)nc(C)o2)=O)ccc(F)c(C)c1 65475,Cc1cnc2n1CC(C(=O)NCC(F)CNC(c1csc(Br)c1)=O)CC2 65476,C(=O)(CCP(C)(C)=O)NCCN(C(C1CCCC(OC(F)(F)F)C1)=O)CC 65477,c1(N(C)C)ccc(Cl)c(C(=O)NC(CNC(=O)OC(C)(C)C)C(C)(C)C)n1 65478,c1(OC)cccc(Br)c1CNCc1ccc(C(=O)NC2CC2)cn1 65479,C(=O)(CCC(O)C(C)(C)C)NC(CN(C)C(c1csc(S)n1)=O)(C)C 65480,Cc1cc(C)c(C(N2CCCC2CNC(N)=O)C(=O)NC2CCCO2)cc1C 65481,N1(C(C(C)OCC(F)(F)F)=O)CCN(CCCNC(=O)C2=C(Cl)CC2)CC1 65482,N1(C(c2cc(CC)nnc2C)=O)CCCC12CCN(C(c1cc(Cl)c(Cl)[nH]1)=O)C2 65483,Cc1ncnc(C)c1OCC(=O)N(C1CCN(C(C2CCOC(C)(C)C2)=O)C1)C 65484,c1(C(N(C2CCN(C(C3(CO)CCC3)=O)CC2)CCCC)=O)nnc(O)nc1O 65485,CC1CCCC1N(C(=O)CNC(=O)C=CC(=O)NCC(N)=O)C1CC1 65486,Cc1nc2ccnn2c(C)c1C(=O)NCC1(O)CCN(C(=O)CCS(C)=O)C1 65487,c1(C(N(CCN(C(C2(CCOC)CCCC2)=O)C)C)=O)ccc(F)cn1 65488,C(c1ccc(C)c(Cl)c1)=CC(=O)NCC1CN(C(COCCCC)=O)CC1(F)F 65489,Cc1cccc(CC(=O)NCCCNC(=O)CN2CCNC2=O)c1Cl 65490,C(=O)(C(CCC)CC(C)C)N1CC2C(C(N3C(OCC#C)CC(F)C3)=O)(C2)C1 65491,C(=O)(C1CCCc2n[nH]cc21)N1CCC(COC)(NC(c2c(C)ncn2O)=O)C1 65492,C1(C(=O)NCC(C2N(C(C=CC(=O)N(C)C)=O)CCC2)(C)C)C(C=C(C)C)C1(C)C 65493,c1(C(=O)NC(c2ccccc2)CNC(C=C(C)C(F)F)=O)ccc(Cl)c(C)c1Cl 65494,CC(N=c1[nH]c(=NC2CN(N3CCC3)CC2C)[nH]c2c1CSC2)c1nc(=N)[nH][nH]1 65495,N1(C(CC(=O)NCC#C)=O)CCC(NC(=O)C(C)CC(F)F)C2(CCC2)C1 65496,CCC(CC(F)(F)F)N=c1nc(N2CCC(F)(C#N)C2)c2c([nH]1)CCC(C)C2 65497,N1(C(c2n(CC)ccn2)=O)CCC(C(=O)NCC2(OC)CCOC2)(CO)C1 65498,N1(C(C(C(C)C)(C)O)=O)CCC2(CCCN(C(=O)CCn3cc(Cl)cn3)C2)CC1 65499,C1(C(N2CC(OCC(=O)NC)C2)=O)CC(F)CCN1C(=O)CCCN=[N+]=[N-] 65500,CC1(C)C2CCC1(COC(=O)C(c1ccccc1F)(C)F)C2 65501,c1(CCC(=O)NC(C)C(c2cccc(F)c2)C)ccc2cccnc2c1Br 65502,Cc1cc(C#N)ccc1C(N1CCCC(NC(C2CN(C3CCC3)C2)=O)CC1)=O 65503,C(C1=NOC2OCCC12)NC(C1CS(=O)(=O)CC12CC2)=O 65504,n1(CC(=O)NCC2(OC)CN(C(=O)CC3NC(=O)NC3=O)C2)c(C)c(C)sc1=O 65505,c1(C(N2CCC(NC(c3c(CC)ocn3)=O)C(C)C2)=O)nccn2cc(C)nc12 65506,c1(NC)cnc(C(N2CCC(O)(CCNC(C3CC3C3CC3)=O)C2)=O)cn1 65507,c1(OC)ncc(C(N2CCC(NC(=O)C(C)CSC)C3CC23)=O)cc1Br 65508,N1(C(C2C(C(C)C)C2)=O)CCCC1CNC(=O)CCn1cc(Cl)cn1 65509,c1(C(=O)NC2CCC(C)N(C(=O)C=CCF)C2)ccc2nnn(C(C)(C)C)c2c1 65510,c1(C(N2C(C(N(CCCC)CCO)=O)CC3CC32)=O)ccc([N+](=O)[O-])cc1O 65511,c1(C(=O)NCC2(F)CCC(CNC(C(CSC)C)=O)C2)cccc2nc(C)[nH]c12 65512,N1(C(CN(C)CCC2CCC2)=O)CCCCC1C1(NC(c2ccncc2)=O)CC1 65513,C1(C)CC(=O)OCC(=O)N1C.CC1CC1CO 65514,C1(CNC(C(c2cccs2)NC(C(C)NC(=O)NC)=O)=O)CNC(=O)C1 65515,Cc1cc(CN=C(NCC(F)F)NCC2(N(C)C)CCC2)cc(C)n1 65516,c1(C(=O)NCC2(F)CC(NC(c3c(CC)onc3)=O)C2)[nH]c(O)nc1C 65517,CCCC(C(=O)N1CCC1CC(=O)NC(CC)CCO)OCC 65518,N1(C(C(c2ccoc2)NC(=O)CC(C2CC2)C2CC2)=O)C2C=CCC1CC2 65519,c1(C(N2CCC(O)C(C)C2)=O)cc(Cl)cnc1-c1cccc(C2(CC)CC2)c1 65520,C1(C(N(CCN(C(C2(F)CCCCC2)=O)CC)CC)=O)CCC(C)CC1 65521,N1(C(C(C)(C)CC#N)=O)CCCC2CN(C(c3cnc4sccn4c3=O)=O)CCC12 65522,C12(N(C)C)CCC(C(=O)NCCC(C)(C)NC(=O)Cc3cnnn3C)(CC1)CC2 65523,C1(C(N2CC(N(C)C(C3(C)CCOC3)=O)C2)=O)CCCCC(C)(C)C1 65524,c1(C(=O)NCC2N(C(c3nn(CC)c(O)c3)=O)CC2)cc[nH]c2nccc1-2 65525,C1(F)(CNC(c2cc(Cl)c[nH]2)=O)CN(C(C2CCCSC2)=O)C1 65526,c1(CC(=O)NC2C(CC(=O)NCCC(C)C)OCC2)ccnc(O)c1 65527,CCC(CC(=O)NCC1CN(C(=O)C(c2cnn(C)c2)=O)C(C)(C)C1)C(C)(C)C 65528,c1(C(=O)OCC)cnc(NC(C2CC3(CCO2)CC3)=O)c(N)c1 65529,C1(CC)CC(NC(N2CCC(O)(CC(C)C)C2)=O)CCO1 65530,c1(C(=O)NCC(C2CCCN2C(c2cc(Br)n[nH]2)=O)(C)C)nc(Br)c[nH]1 65531,C(C(C)CC(=O)NC1CC(NC(=O)C=Cc2ccc(Cc3ccccc3)o2)C1)OC 65532,C(=O)(CS(=O)(=O)C1CCCC1)NCCC(C)CCNC(=O)CSc1ccccc1 65533,C12C3CN(CC13)C2=O.CC1(C(N2CCC(F)C2)=O)CCCN1 65534,c1(C(=O)NC(CC)CN(C(C2(Cl)CCCC2)=O)CC)cc[n+]([O-])cc1 65535,C1(CNC(CC(C)SC)=O)CC(F)(F)CN1C(=O)C=C(C)C1CC1 65536,CC(c1ccc(F)cc1F)=CC(=O)NC(C)C(C)NC(=O)C(C)(C)C(C)O 65537,C1(N(C(C)=O)C2CC2)CCC12CCN(C(=O)Cc1ccc3nn(C)cc3c1)CC2 65538,N1(C(C2(COCC)CC2)=O)CCC2(CCCN(C(=O)C(C3CCC(=O)N3)C)C2)C1 65539,N1(C(c2cc(OC)n(C)n2)=O)CC(NC(=O)Cc2sccc2Cl)C2CCCC2C1 65540,c1(OC)cc(=O)n(C)cc1C(N1CC(NC(=O)C#CC2CCCC2)CC1C)=O 65541,N1(C(Cc2cccc(CC)c2)=O)CCCCC12CC(NC(c1ccc(C)nn1)=O)C2 65542,CCC(CC(=O)NC1(CNC(=O)C(C)Oc2ccc(C)cc2)CCCCC1)SC 65543,C1(C(=O)Nc2ccccc2Nc2ccccn2)CCC2(CC1)CS(=O)(=O)C2 65544,c1(C(N2CC(Cn3cc(-c4ccc(Cl)c(F)c4)nn3)C2)=O)cc2n(n1)CCCC2 65545,c1(OC)c(C(=O)NC2CC2CNC(C2(C)CC3CC3C2)=O)ccc(Cl)c1Cl 65546,C1(CN(C)C(C2(NC(=O)COc3ccsc3)CC(F)C2)=O)CC2(CC2)C1 65547,C1(CNC(c2c(CC)cccn2)=O)CCN(c2nc(Cl)ncc2Cl)CCC1(F)F 65548,N1(C(CC(=O)OCC)=O)CC2(CC2)CC1C(N1CCC(CC(C)C)C1)=O 65549,C12(NC(C=Cc3c(C)cccn3)=O)CCCN(C(=O)C=CC3CCOC3)CC1C2 65550,C(=O)(CCCCC(C)=O)N1CC(C(C)NC(CC(CC)(C)C)=O)OCC1 65551,CC(C)(CNC(=O)CCN(C(c1nc(=N)cc[nH]1)=O)C1CC1)C(N)=O 65552,C1(C(NOC(C)(C)C)=O)CCOC1CCNC(=O)C(F)F 65553,c1(C(N2C(C)(CC)CC(NC(=O)CCSC)C2)=O)cc2nc(C)cc(C)n2n1 65554,Cc1ocnc1C(N1CCCC1C(C)(C)CNC(=O)CC1CNC(=O)C1)=O 65555,N1(C(C=Cc2n(CC)ncc2)=O)CCC(NC(=O)CCSC(F)(F)F)C(O)C1 65556,C(F)(F)(C(F)(F)F)OCC(=O)NCC(CN(C(c1ccc(C)o1)=O)C)C 65557,C1(N(C)C(C2CNC(=O)N2)=O)CCN(C(C2(N(C)C)CCCOC2)=O)CC1 65558,Cc1cscc1C(C(=O)NCCCC1CC1)NN(CCN(C)C)Cc1ccccc1 65559,c1(-c2cc(N3CCCC(C#C)C3)ncn2)cc(C)cc(OC)c1O 65560,C1(C(=O)NC(C#C)CC2CCC2)(CC)CCCN(C(C2CC2C(C)(C)C)=O)C1 65561,N1(C(c2nnn(CC)c2C)=O)CCC(C2CC(NC(C3(CC)CCC3)=O)C2)CC1 65562,CC1CC(C)CN(C(=O)CN(C2CCN(C(=O)CCC3CCC3)CC2)C)C1 65563,c1(C(N2CCC(NC(CCCC=C)=O)C2C2CC2)=O)ncc(P(C)(C)=O)cn1 65564,CCC(C)C(=O)N(C(C)CCNC(c1ccn(C2CCC2)n1)=O)C 65565,c1(C(=O)NCC(CC=C)NC(=O)C=CC(F)(F)F)ccccc1OC 65566,CCCC(CCNC(=O)C(C)N(C(c1cncc(OC)c1)=O)C1CC1)C1CC1 65567,C1(CNC(CC2CC(CC)C2)=O)CC2CCC1N(C(C1(CO)CCCCO1)=O)C2 65568,N12CCCC(C1)C2=O.c1(C(C)C)cc(C(=O)NC)n[nH]1.C1(NC)CCC2CC12 65569,C1(NC(c2cc(C)n(C)n2)=O)C2CC(CN(C(C3CCCC3)=O)C2)C1CO 65570,C1(C(N(C2(C(=O)NC3CC3F)CC2)C)=O)CC(=O)CC12CCC2 65571,N1(C(COCC(=C)C)=O)CC2CCCC2(CNC(c2cc(CCC)n(C)n2)=O)C1 65572,c1(C(=O)NCC2(C)CCN(C(CC(C)n3cccc3)=O)C2)n[nH]c2c1CSCC2 65573,CN1CCN(C(c2ccccc2CC#N)=O)CC1CNC(=O)C(C)(C)C(N)=O 65574,c1(CC(=O)NCCN(C(c2ccc(C)s2)=O)C)ccc(C)c(Br)c1 65575,C(=O)(C(O)CC(C)C)N(CCCNC(c1ccccc1COC(C)C)=O)CC 65576,N1(C(C23C(C)OC(C)(C2)C3)=O)CC2(CC(NC(=O)CCS(C)(=O)=O)CO2)C1 65577,C(CCC(C)C)(C(=O)NCCN1CCCCC1=O)NC(CC(CCC)C)=O 65578,N1(C(=O)CNC(=O)NCc2ccc(F)cc2)CCC2(NC(C(C)SC)=O)CC2C1 65579,C1(NC(CC2CC(=C)C2)=O)CN(C(C2(CCCC)CCC2)=O)CC2(CCC2)C1 65580,C12(C(=O)Nc3cc(C(F)F)ncn3)CCCCCC1N(C(=O)COC(F)F)CC2 65581,C1(NC(=O)COCCn2cncn2)CCC2CC1CN2C(=O)Cc1ccccc1 65582,C1(C(N(C(CNC(c2ncnc(C)c2C)=O)C)C)=O)CC12CCc1ccccc12 65583,C1(C(C)(C)C)(CNC(c2scc(OC)c2)=O)CCN(C(C2(CO)CCCO2)=O)C1 65584,C(=O)(CCC(C)(C)[N+](=O)[O-])N1C(CNC(c2c(C)oc(C)c2C)=O)CC(O)C1 65585,CC(C(=O)NCCC1CCCN(C(C23COCC(C2)C3)=O)C1)C(F)(F)F 65586,CC1CC2CCC(C(=O)NC(C3CN(C(c4cc(Cl)cc(Cl)c4)=O)C3)C)CN2C1 65587,N1(C(c2ccc(CCC)cc2)=O)CCN(C(C2C(C)(C)C2(F)F)=O)CCC1C 65588,C=CCC(C)(C)CC(=O)NCCN(C(=O)CC1CCC(=O)NC1)C1CC1 65589,C1(N(C(C2(C)C(C)CCC2)=O)C)CCCCN(C(c2cnccc2Br)=O)C1 65590,C1(C(=O)NCCCCCC2CCCN2C(C2CCOC2)=O)CCC2(CC2)C1 65591,c1(Nc2scc(C(=O)Nc3c[nH]c4ncccc34)n2)cc2c(Cl)nccc2s1 65592,C1(C(=O)NC2(CC=C)CN(C(=O)COCC(F)(F)F)C2)CCc2nncn2C1 65593,c1(C(=O)NC2(CCCNC(Cn3ncc(CC)c3)=O)CC2)ccc(N)cn1 65594,C12(C(N3CC(C(=O)O)C(c4ccccc4)C3)=O)CC(C1)C(c1ccccc1)O2 65595,C1(NC(=O)CCCc2ccccc2)CC12CCN(C(=O)CCC1OCCO1)CC2 65596,CCCS(=O)(=O)C(C)C(=O)NCCN(C)C(c1ccc(Br)c(OC)c1)=O 65597,c1(C(=O)NC(CNC(COCCC#C)=O)C2CCC2)c(C)cnnc1O 65598,c1(C(C)=O)c[nH]ccc1=NC(=O)c1cccc(F)c1-c1ccc2c(c1)C(=O)NC2 65599,CCC(C(C)(C)O)NC(=O)C(CC1CCC1)NC(=O)CCC(=O)N(C)C 65600,CC1CCC(CC(=O)NCc2cc(C(=O)Nc3cnn(C(F)F)c3)n[nH]2)C1 65601,C1(C(=O)NCCC(O)C2CCCC2)CCCCC1NC(C1(C2CC2)CC1)=O 65602,O=S(=O)(c1ccc2nc(O)oc2c1)Nc1nc(-c2cc(O)ncc2Br)cs1 65603,C(=O)(C(C)(C)CC(C)(C)C)NC1CN(C(CC(CC)CC)=O)CC(C)C1 65604,N1(CC=CC(=O)NC(C)CN(C)C(C2(C)CC2Br)=O)CCOCC1 65605,C123CC(C1)N(C2)C3=O.c1(C(=O)NCCCc2ccccc2)cccnc1O 65606,N1(C(c2ccc(CSC)cc2)=O)CC2CC(NC(=O)CCC3CCCO3)CC1C2 65607,C1(C(N(C2(n3cccn3)CC2)C)=O)COCCC1NC(=O)CC1COCCO1 65608,C1(COC)(CNC(C2CC(SC)C2)=O)CCN(C(=O)Cc2ccc(Cl)s2)C1 65609,C(=O)(CCC(C)(C)C)NCC(C)NC(C1(c2ccc(O)cc2)CCOCC1)=O 65610,N1(C(c2ccc(OC)nc2)=O)CC(NC(=O)C=Cc2ccccc2)C(C)(C)C1 65611,c1(N2CCC(N(C(C=C(CC)CC)=O)C)CC2)cc(C)nc2nc(C)nn12 65612,N1(C(c2ccc(Br)cc2Cl)=O)CC(NCCOCC(C)O)C2(CCC2)C1 65613,Cc1cc(C(=O)NCC(O)CNC(C2NC(=O)OC2C)=O)ccc1C1CC1 65614,N1(C(=O)NC2CC(NC(CC3CCN(C(C)(C)C)C3)=O)C2)CCc2sccc2C1 65615,N1(C(CC(C)SC)=O)CCC(NC(=O)CCc2ccc(F)cc2F)C2(CCC2)C1 65616,C1(CC=C)(NC(c2cnn(C(C)C)c2Br)c2nnnn2C)CCN(CC)C1 65617,C(=O)(CCC(C)(C)C)NC(C1(O)CCN(C(Cn2c(C)csc2=O)=O)C1)C 65618,N1(C(c2n(CC)ncc2Cl)=O)CC2CCC2(NC(=O)CCc2cnn(C)n2)C1 65619,c1(C(=O)NCC(CCOC)NC(C23CC4CC2C3C4)=O)nn(C)c(C)c1Br 65620,c1(C(=O)NCC(C2CCC2)NC(c2nccc(CC)c2)=O)cnc2n1CCC2 65621,c1(CN2CCC(NC(c3c(C)nc(OC)s3)=O)C(F)C2)ccc([N+](=O)[O-])cn1 65622,Cc1ccc(C)n1CC(N1CC=CC1CNC(C1CC(=O)N(C2CC2)C1)=O)=O 65623,CCC(C)(COC)C(=O)NC(C)CCCNC(c1ccn(C(C)C)n1)=O 65624,C1(C(=O)NC(C2CCCN2C(c2n[nH]cc2-c2ccccc2)=O)C)CS(=O)(=O)C1 65625,C1(C)(SC(C)=NCCF)N(C)N=CC=C1 65626,Cc1cc2c(CC(N3CC(CN4CC(C(=O)NC5CC5)C4)CC3C)=O)csc2s1 65627,C=CCC(CC(=O)N(CCCF)C)NC(c1coc(N(C)C)n1)=O 65628,C12(OC)CCCCC(C(N3CCC(NC(=O)CCCF)C(CO)C3)=O)(C1)C2 65629,C1(CCC(=O)NC(CNC(c2c(C)cno2)=O)C2CC2)CCC(=O)NC1 65630,N1(C(C(c2ccnn2C)NC(C=C(C)C)=O)=O)CCC(F)(C#N)C1 65631,C1(C(=O)NCCCN(C)C(C2(F)CCCC2)=O)Cc2cccc(OC(F)F)c2O1 65632,c1(C(N(C)CC2COCCN2C(C2CC23CCC3)=O)=O)cc2c(nn1)CCCO2 65633,c1(C(N(C)CCNC(=O)CC2C=CCCC2)=O)nn(CCF)cc1Br 65634,c1(C(=O)NCCC2(OC)CN(C(=O)CO)C2)cc(N(S(C)(=O)=O)C(C)C)ccc1C 65635,CC1=C(C(=O)NCC2CC3COCC3N2C(=O)Cc2csc(Cl)c2)CCS1(=O)=O 65636,c1(C(=O)NC2(CCCNC(=O)CC(=O)Nc3nccs3)CC2)cc([N+](=O)[O-])c[nH]1 65637,C(=O)(C1=COc2ccccc2O1)N1CCC(N(C(C(C)(C)SC)=O)C)C(C)C1 65638,C12(NC(=O)CC3CCC=CCC3)CCCN(C(c3cc(Cl)sc3Cl)=O)CC1C2 65639,c1(OC)ccc(Cl)cc1CC(=O)NC1CCN(C(c2ccon2)=O)C1(C)C 65640,C1(C(=O)NCCN(CC(C)O)C(=O)C=Cc2ccccc2)CCN2CCOCC12 65641,C=CCCC(F)(F)C(=O)N1CCC2(CC1)CC2NC(=O)C1=CC(C)(CC)C1 65642,c1(C(=O)NCC2CC(NC(c3cc(F)ccc3Cl)=O)C2)cc2n(n1)CCCO2 65643,N1(C(=O)C=Cc2cncc(O)c2)CC2CCC1CN2C(C1CC1(CC)CCF)=O 65644,Cn1c(CC(N2CCOC(Cn3cc(-c4cncs4)nn3)C2)=O)cccc1=O 65645,N1(C(C2CCCN(C)C2)C(=O)NC2CCCCCC2)CCCCC2(CCC2)C1 65646,C1(NC(C(C)NC(c2ccoc2)=O)=O)CC2CC1N(C(=O)NC1CCC1)C2 65647,N1(C(C(=C(C)C2CC2)F)=O)CCC(NC(c2cnn(C3CC3)c2)=O)C(F)C1 65648,Cc1c(C=CC(=O)NC2CC(CNC(c3cncs3)=O)C23CCC3)cnn1C 65649,[N-]=[N+]=NC1CN(C(=O)CC2CCCCC23CC3)CC1NC(=O)Cc1cccnc1Cl 65650,C(CC(C)(O)CNC(=O)C(CCC1CCC1)NC(=O)C=CCO)OC 65651,N1(C(C(CC)OCC)=O)CCC(C)(CCNC(c2cnc(C)[nH]2)=O)C1 65652,Cc1cocc1C(N1CC(CCCCNC(C2(CC3CC3CF)CCCC2)=O)C1)=O 65653,C(C)(CCC(=O)N1CCCCC1CN(C)C(C1SCCCS1)=O)OC 65654,c1(C(=O)Nc2n(C)c(C3CC3(C)C)nn2)ccc(Cl)c(F)c1F 65655,N1(C(c2c(CC)ncs2)=O)CCC(C2CC2)(CNC(=O)C(C)CO)C1 65656,C(C)(C(C)C(=O)N1CCOC(C(C)(C)C)C1)NC(c1ncn(CC)c1)=O 65657,c1(C(N(C2CCN(C(=O)CC3CCNC3=O)C2)CCC)=O)ccc(CO)s1 65658,c1(C(N2CCC(C(C)NC(c3ncccn3)=O)C2)=O)sc2sccc2c1Cl 65659,C(=O)(CCCCCCCCC1CC1)N1CCCC(NC(C(C)CC(N)=O)=O)CC1 65660,C#CCCCCC(=O)NCC(CC1CC1)C(=O)NCCCCC(=C)C 65661,N1(C(C23C(CN(C(c4c(CC)noc4)=O)C2)C3)=O)CCC(C#N)CC12CC2 65662,N(C(=NCCc1ccc(OC(F)F)cc1)NC1CC(C(N)=O)C1)C(C=C)C 65663,N1(C(c2c(CCC)ocn2)=O)CC(C)CN(C(=O)C=CC(F)(F)F)C(C)C1 65664,C(=O)(C1CCCc2ncccc21)N1CCC(N(C(CC)=O)CCO)CC1 65665,C1(CNC(C2C(NC(C(C)OCc3cccnc3)=O)CCC2)=O)CC(=O)N(C)C1 65666,N1(C(C2CC(CNC(C(C(C)C)=O)=O)C2)=O)CCN(C)C(C(C)C)C1 65667,c1(OC)cnn2c1C(=O)NCC2.c1(NCC(c2ccccc2)OCC)nc(C)sc1C 65668,N1(C(C2(CC)CC2)=O)C2CCC1CC(NC(=O)CN1CC(C)(C)C1)C2 65669,C(=O)(CCCCCC(C)C)N(CCOC)CCNC(=O)C#CC1CCOC1 65670,C(CS(C)(=O)=O)N(C)C(C1CCC1CNC(=O)CCN(C)C)=O 65671,c1(C(=O)NC(C)CCCNC(=O)C=Cc2ccc[nH]2)cccc(Br)c1 65672,CCC1=NOC(C(N2CCCC(N(CCF)C(c3cn(C)cn3)=O)C2)=O)C1 65673,N1(C(c2c(C)nn(C(C)C)c2)=O)CCC(CNC(=O)COC2(C)CCC2)C(C)C1 65674,c1(OC)cc(C(=O)N(C)CCN(C)C(c2cc(N)ccn2)=O)cc2cnn(C)c12 65675,c1(CC(=O)NCC2CCN(Cc3cc(O)cc(Br)c3)C2)ccc2c(c1)C(=O)CC2 65676,CONC(=O)CNC(C1(F)CN(C(C2CC=CCC2)=O)C1)=O 65677,C1(C(=O)NC2CN(C(CC(=C)C)=O)CC2(C)C)CC2CCCC(C1)C2 65678,CC(C)CC(=O)C(=O)NC1CCCC(CC(N2CCCC2C(=O)N(C)C)=O)C1 65679,c1(C(N(CC(=O)NN(C2CC2)CC2CC(=C)C2)C)=O)n[nH]c2c1COC2 65680,C1(C(=O)NC(CC)COCC2CC2)CN(C(=O)C(C#N)C(C)C)CCN1C 65681,CC1CC(NC(c2nccnc2Cl)=O)CN(Cc2ncccc2C(F)(F)F)C1 65682,CCC(CC)C(C)C(=O)NCC1CCCN1C(=O)CNC(c1cccc(C)c1)=O 65683,CC(C)C(C(=O)NC(CCC(=O)O)c1ccc(Br)cc1)C1CCC1 65684,c1(SC)cc(C(=O)NC(C)C(C)NC(c2conc2-c2ccccc2)=O)c(C)o1 65685,Cc1ccc2nc(C(=O)NCc3ccc(C(F)F)cn3)[nH]c2c1 65686,CC(C)(CNC(=O)Cc1cccnc1)CC(=O)NCC(O)CC1CCC1 65687,C(C(C)(O)C(=O)NCC1(CNC(=O)CC(F)F)CC1)OC 65688,c1(C(=O)NCC(C2CCCCC2)NC(C(C)NC(N)=O)=O)cc2scc(Cl)c2[nH]1 65689,C1(OC)CN(C(=O)CN2CSCC2=O)CC1NC(=O)C(C1CCN(C)CC1)F 65690,c1(C(N2CCC(C(N(CC(C)N(C(C)=O)C)C)=O)C2)=O)cccc(Br)c1Br 65691,CN1CCn2cc(C(=O)NCC3CCCN(C(C4CCSC4)=O)CC3)nc2C1=O 65692,C1(CCC(=O)NCc2cc(C(N)=O)no2)CCCN(C(c2ccccc2F)=O)C1 65693,c1(C(C(=O)NC2CC(C(=O)OC)C2)N(CCC)C)csc(C(C)(C)C)n1 65694,C(C(C(C)(C)C)NC(=O)Cc1cc(C)ns1)NC(Cc1ccc(C)o1)=O 65695,CCC(C)C(O)C(=O)N1CCN(C(=O)C(c2ccccc2C)C)CC1C1CCCC1 65696,CCCCCCC(CC)n1nc(Cn2cncn2)nc1-c1cccc(CC)c1 65697,N1(C(C2CCC(OC)CC2)=O)CC(NC(C2CCOC(C)(C)C2)=O)C(C)(C)C1 65698,N1(C(=O)OCC)CC2(CCN2C(C2CCC(=O)C(OCC)C2)=O)C1 65699,Cc1[nH]c(C)c(CNC(=O)CC2(O)CCCCCC2)c1C 65700,CC1=NS(=O)(=O)NC=C1C(=O)N1CC2CC1C2NC(=O)CC(O)C(C)C 65701,C(=O)(CC(C)(O)COC)N(CC(CC)NC(=O)C=Cc1sccc1C)C 65702,N1(C(COCC=C)=O)CCN(C(=O)C(C)NS(C)(=O)=O)C(C(C)C)C1 65703,CC(CC(=O)N1CC2CCC1CC2NC(C1(C)CCCCO1)=O)P(C)(C)=O 65704,c1(OC)ccc(I)c(C(=O)NC2CCC(NC(=O)Cc3cc(F)ccc3O)C2)c1 65705,C(=O)(C(C)(O)C(F)(F)F)N1CCCC(OCC(=O)NCc2c(OC)cccc2)C1 65706,C1(CC)CCCC1NC(C1CCC(CNC(=O)CCc2ccco2)O1)=O 65707,CC1CC(CNCC2CCC(=C3CCC3)CC2)CN(C(=O)OC(C)(C)C)C1 65708,n1(CCC)cc(C(=O)N(C(C)(C)CC=CC(=O)NC(C)C2CC2)C)nn1 65709,CCC(O)C(C)C(=O)NCCCN(C1CCCC1)C(c1cnc(C2CC2)[nH]1)=O 65710,N1(C(C=NOC)=O)CCCC1C1CCCN1C(=O)Cc1c(OC)cccc1F 65711,N1(C(C2(F)CCN(C(c3cccc(C(F)(F)F)c3)=O)C2)=O)CCC2(CC1)OCCO2 65712,c1(CS(C)(=O)=O)cn(C2CCN(C(c3cn(C4CC4)nn3)=O)C2)nn1 65713,c1(N(C)C)cnc(F)c(C(=O)NCC2CCCN2C(c2cncc(F)c2Cl)=O)c1 65714,N1(C(CC(C(=O)OC)C)=O)CCC(C)(C)CC1C(=O)NC(C1CCOC1)CO 65715,c1(-c2cn(-c3ccc(NC(CSCCC)=O)cc3)nn2)c(Cl)cccc1Cl 65716,C1(NC(C2CCC(C)S2)=O)(CNC(c2cncc(F)c2Cl)=O)CC2CCC1CC2 65717,c1(NC(C2N(C(C(CSC)O)=O)CC(F)C2)=O)ccc(O)cc1C 65718,Cc1cc(CC(N2CC(NC(C3CCS(=O)CC3)=O)CC2C)=O)cc(C)c1 65719,C(=O)(CC(O)C(C)C)NCCS.n1(C(C(C)O)C)cc(COCC2CC2)nn1 65720,N1(C(C2CC(=C)C2)=O)CCC(C)C1CNC(c1cnc(C2CC2)nc1)=O 65721,Cc1ccc(C(=O)NCC(CC(C)C)NC(C2(C3CC3)CCC2)=O)cc1C 65722,c1(C(N2CCC(N(C)Cc3c(F)cccc3F)C2)=O)ccc2nnc(Br)n2c1 65723,N1(C(c2c(N(C)C)ccc(Cl)n2)=O)CCN(C(C2CCCCO2)=O)CC(O)C1 65724,C1(C(N(CC(COCC)O)C)=O)COCC1NC(C1(CSC)CC1)=O 65725,C(=O)(C(C)(F)C(=O)NC1CN(C(c2ccc(SC(F)(F)F)cn2)=O)C1)OCC 65726,CC(C)C1=CCC(NC(C2(NC(=O)C=CC3CC3)CCN(C)C2)=O)CC1 65727,C(=O)(CC#CC(C)(C)O)N1CC(C(N)=O)(CNC(C(CC(C)C)F)=O)C1 65728,C1(NC(CCc2cc(C)nc(C)c2)=O)CC2(CN1C(=O)C(C)C)CC2(F)F 65729,C(=O)(CCC(C)(C)F)N(CCCNC(=O)CC1CCCC1(F)F)C 65730,n1(CC)ncc(CSCCOC)c1C.N12CCN(CC1)C(=O)NCC2 65731,N1(C(c2cccn(C)c2=O)=O)CCC2(NC(C3CCc4nc[nH]c4C3)=O)CCCC12 65732,N1(C(c2c(OC)scc2)=O)CC(NC(c2ccc(Cl)c(F)c2N)=O)C2(CCC2)C1 65733,N1(C(C(N2CCOCC2)C)=O)CCCCC(NC(=O)C=C(C2CC2)C2CC2)C1 65734,CC1CC(C(=O)NCC2CCC(NC(C3(C4CC4)CC=CC3)=O)C2)CCC1C 65735,N1(C(C(C)OCCCC)=O)CCN(C(c2ccc(C(F)(F)F)s2)=O)CC1CCO 65736,C1(C#N)(C(N2CCC(C(C)NC(c3cncc(CO)c3)=O)C2)=O)CCN(C)CC1 65737,c1(OCC#C)ccc(CNC(=NC)NCC23CC(C)C2C3)cc1 65738,C(=O)(C(c1ccoc1)N(C(=O)C(C)N1CC(C)C1)C1CC1)NCCCSCC 65739,NS(=O)(=O)N1CCCC(C(=O)NCC(O)CNC(c2c[nH]c(C(=O)C(N)=O)c2)=O)C1 65740,c1(NCC)scnc1C(=O)N(CCCC(=O)NCC1(O)CCSC1)C 65741,CCCCC(O)C(=O)NCC=CCNC(c1cn(-c2ccc(F)c(F)c2)nn1)=O 65742,Cc1ccccc1C=CC(=O)NC(C)CCN(C)C(C1CC2CC2C1)=O 65743,c1(C(N2CCC(NC(CN(CC)CC)=O)C(O)C2)=O)cccc2c1OCCO2 65744,c1(SC)cc(C)c(C(N2CC(CNC(C3(C)CCOC3C)=O)C(O)C2)=O)o1 65745,CC1N(C(=O)C(CC(C)(C)C)NC(c2cccnc2)=O)CCOC1(C)C 65746,CCCCC(C(=O)NCC(CC(N1CC(CO)CC(C)(C)C1)=O)OC)C(C)C 65747,C(C)(CC(=O)NCC(C)(C)CNC(c1cc(N)c(F)cc1F)=O)(C(F)F)N(C)C 65748,C1(CNC(CCOC)=O)CC2(CCOCC2)CN1C(=O)CCC1CC2CCC1C2 65749,C1(NC(C(C(C)C)O)=O)CCC(O)CN(C(=O)CCOc2ccc(F)cc2F)C1 65750,n1(C2CCN(C(c3cc(C)cc(F)c3)=O)C2=O)ncc2c1CCCC2 65751,C1(NC(CC)=O)CCCC(C(=O)Oc2ccc(Br)cn2)C1 65752,CC1(C)CN(C(C2CCCCN2C(c2cc3cccnn3c2)=O)=O)C2CCCC12 65753,N1(C(C2C(C)(CC)C2)=O)CCC2(CC1)CCN(C(c1csc(C)c1C)=O)C2 65754,c1(SC)ccc(Cl)c(C(=O)Nc2ncc(SC)s2)c1 65755,Cn1cnc(S(N)(=O)=O)c1C(=O)NC1CC(CNC(c2cncn2C)=O)C1 65756,C=CCC(CC(F)F)C(=O)N1CC(CNC(=O)CSCc2cccs2)CC1(C)C 65757,C12(C(N(C)CC3CCNC3)=O)CC3CC(C(=O)N1)C2C3.n1(CC=O)cnnc1O 65758,c1(N(C(CCCN(C(C=CCC)=O)C)=O)CC)ccc(F)c(C)c1 65759,C(=O)(NNc1nccnc1C(F)(F)F)NC(C(=O)Nc1ccc2onc(C)c2c1)C 65760,c1(OC)ncccc1C(N1CC(CNC(c2cc(C3CC3)on2)=O)CC1C)=O 65761,Cc1cccc(C)c1OCCNC(C1COCCN1C(C1CC(C2CC2)C1)=O)=O 65762,C1(C(=O)NCC2(COC)CN(C(c3occc3C)=O)C2)CCc2nnn(C)c2C1 65763,c1(C(N2CCC(C(=O)OC)CC2(C)C)=O)cc(C)cc2c1OCC2.CO 65764,C#CCC(C)(CC)C(=O)NC1COCCC1C(N1CCOC(C)C1)=O 65765,CCC(CC(=O)NCCN(C(=O)C(C)(C)CF)C1CCCCC1)C1CCC1 65766,c1(CNC(C2(C)CCN(C)C2=O)=O)nc2c(s1)CN(C(C1(CO)CC1)=O)CC2 65767,c1(CCC(=O)NC2CC2CNC(C2(F)C3CCCC23)=O)ccc2ncccc2c1 65768,CC1(C)CCOC(CC(=O)NC2CCCN(C(c3ccsc3C#N)=O)CC2)C1 65769,O=C(CCC1CC1CC1CC1)NC1(CCF)CC1 65770,c1(CN(C(C2CCN(C(c3cn(CC)nn3)=O)CC2)=O)C)ccc(C)c(C)c1 65771,C12(C(=O)NCCC(C)(C)CNC(C3C4CC5C(C4)C35)=O)CCCCC1OCC2 65772,C1(C(=O)NC(COCC)C)(NC(c2nccn2C)=O)CCC(C)CC1 65773,C(CC(C)(C)CC(=O)NCCC1(O)CCN(C(C2(O)CC(CF)C2)=O)C1)OC 65774,C1(NC(=NCC)NCCc2cccnc2O)CCc2ccccc2C1 65775,C1(CCNC(Cn2cnc(CC)n2)=O)CN(C(=O)COC2CC=CC2)CC1C 65776,C1(NC(C(C)(C)CF)=O)CCN(C(=O)CC2NC(=O)NC2=O)CC1CO 65777,c1(C(N(C)CC2CCCCN2C(=O)CC2(CO)CC2)=O)cnc2ccccc2n1 65778,C1(C(C)C)CN(C(=O)C=Cc2ccco2)CCN1Cc1nc(Cl)ccc1Cl 65779,C(CCOCC)(C(=O)N(C)CCN1CCCC1)NC(C(CC)n1ccnc1)=O 65780,c1(OC)cc(CO)ccc1C(N1CCCC(C)C1CNC(C1CC(C#N)C1)=O)=O 65781,Cc1cc(=O)oc(C)c1C(=O)NC1COCC1NC(c1ncn(C)n1)=O 65782,C1(O)(CNC(C2(C)CC(=C)C2)=O)CCCN(C(c2ccc(Br)c(C)c2)=O)C1 65783,c1(OCC)cc(C(=O)NC(CCNC(=O)CCC2(C)N=N2)C(C)(C)C)oc(=O)c1 65784,N12CCCC(C1C)C1CCN(C1)C2=O.C=CC(C)OC 65785,c1(C(N(CC(C)CC)NC(=O)C(=O)N(C)C)=O)ccc2c(c1)C(=O)OC2(C)C 65786,c1(C(N2CCC(NC(c3cncc(C(C)(F)F)c3)=O)CC2)=O)nnn2c1CCC2 65787,c1(CC2C(=O)NC(=O)C2)cnn(C)c1O.C1(C2C(C)CC2)CNC(=O)C1 65788,Cn1cc(C(=O)NC2C3CC(NC(=O)CCC4CCCC4)CC23)ncc1=O 65789,c1(OCC)ncccc1C(=O)NCC1CCN(C(C2(n3nccn3)CC2)=O)C1 65790,C(=O)(C1=CCCCC1C)NCC(C)(C1CCC1)NC(c1occ(C)c1)=O 65791,Cc1nc(Cl)ccc1S(=O)(=O)N1CC2CN(C(c3ccc(C#N)s3)=O)CC12 65792,c1(-c2c(CNC)ccc(F)c2)ccc2c(c1)CN(C(=O)C(C)(C)O)CC2 65793,Cc1cc(F)c(Cl)cc1C(=O)NCC(C)CN(C)C(c1ccc(C#N)nc1O)=O 65794,c1(C(N2CC(CC(=O)NCC3(CCOC)CCC3)C2)=O)cc(C#N)ccc1C 65795,N1(C(C=CCC)=O)CCN(C(c2cnn(CC)c2C(C)C)=O)C(CC)C1 65796,c1(C(=O)NC2CCN(C(=O)C(C3CCCCC3)F)CC2F)ccc2nnnn2c1 65797,C1(C(=O)NCCc2cn(Cc3occ(C(=O)O)n3)nn2)CCC2CC1CO2 65798,CN1CC(CC(=O)N(CC(N2CC(OCCCO)C2)=O)CC2CCCC2)C1 65799,C1(NC(CC)=O)(CO)CCCN(C(c2oc(-c3ccc(C#N)cc3)nc2C)=O)C1 65800,c1(OC)cc(C#N)ccc1CNC(c1ccc(C)cc1-c1ccc(F)nc1C)=O 65801,C(=O)(C1CCc2snnc21)N(C(C)C)CCNC(c1cnn(C(F)F)c1)=O 65802,c1(-c2ccn(CCOC)n2)nc(-c2cnn(C)c2)nn1C(c1cccc(O)c1)C 65803,C1(C(C)NC(Cc2nc(C)sc2)=O)CCCCN1C(C1SCCS1)=O 65804,C1(O)(CCNC(C2(F)CCOC2)=O)CCN(C(=O)COCC2CCCO2)CC1 65805,Cn1cc(C(=O)NCC2CN(C(=O)Cc3ccsn3)CC(C)(C)C2)c(O)nc1=O 65806,C1(COC)(NC(=O)Cc2csc(=N)[nH]2)CCN(C(C2CCS(=O)CC2)=O)C1 65807,N1(C(C(C)NC(CC)=O)=O)CC2(C(=O)NCCC=CC3CCCC3)CC1CO2 65808,C=CC(C(=O)NC(CNC(C1CCN(CC)C1)=O)C(C)C)OC 65809,C1(CNC(C(C)NC(CC)=O)=O)CCC(F)(CNC(c2cnc(CC)s2)=O)CC1 65810,N1C2=NCCCN1CC1(C(F)(F)F)CCN2C1.C1(CS(C)(=O)=O)CCOC1.CC 65811,C12(NC(c3cc(COC)cn3C)=O)CCC(C1)N(C(=O)CC1CCCC(=O)N1)C2 65812,N1(C(c2cc(CC)oc2C)=O)CCN2CCN(C(c3cc(F)cs3)=O)CC2C1 65813,CC(=O)CCC(=O)NC(=O)C(C(C)C)NC(c1ccccc1)(C)CO 65814,c1(NC(C2CN(Cc3cncc(OC)c3)C2)=O)ccc(F)cc1I 65815,Cc1ccsc1C=CC(N1CCC(C(C)NC(=O)CCC(C)C)C1)=O 65816,C(=O)(C(=O)N=S(C)(C)=O)N1CC(NC(CC2CCC(C)CC2)=O)C(C)CC1 65817,Cn1nc(COc2ccc(C#N)cc2CO)c(C(=O)O)c1C#N 65818,N1(C(CCCC#C)=O)CCC(NC(c2cccc(N)c2F)=O)C(F)(F)CC1 65819,N1(C(C(C)=CC)=O)CC(C(=O)NCc2csc(CC)n2)C2(CCS(=O)(=O)CC2)C1 65820,N1(C(=O)CC2CCOC2)CCC(OCC(F)F)CC1 65821,N1(C(C)C)CCCC1C(=O)N(C(C)CNC(C1(C)CC1C)=O)C 65822,CC1CN(C(C2(O)CCSC2)=O)CC1CNC(c1cc(-c2cnn(C)c2)on1)=O 65823,c1(C(=O)OCc2ccn(C)n2)ccccc1NC1N(c2ccc(F)cc2)CCC1 65824,N(C1CCc2cc(C(F)(F)F)ccc21)CC(C1CCCSC1)=O 65825,C1(C(=O)NCc2cn(CC(=O)NCC(O)C(F)(F)F)nn2)CC2C(C1)C2(F)F 65826,C1(NC(C(=O)N(CC(CC)OC)C)=O)CCN(C(=O)C(F)(F)C2CC2)CC1 65827,c1(CC(C(=O)N(C(C)CNC(C2CC2F)=O)C)C)ccc([N+](=O)[O-])cc1 65828,Cc1cccc2[nH]cc(C(=O)NC34CC3CN(C(C3CCC3)=O)C4)c12 65829,C(=O)(C1=NOC(C)C1C)N(C1(CC(=O)NCC(CC)(C)OC)CCCCC1)C1CC1 65830,C1(C(=O)NC(C(C)C)C2CCC2)CCN(C(=O)CC(=O)NC2CC2)CC1O 65831,C1(C(=O)NC2(C)CCN(C(c3n[nH]c(=N)s3)=O)CC2)CSc2ccccc2O1 65832,c1(CC(=O)NCC(CNC(CC2(C)CC2)=O)O)ccc(C(N)=O)cc1 65833,N1(C(c2c(CC)cc[nH]2)=O)CCN(C(=O)Cn2c(C)csc2=O)C(CC(F)F)C1 65834,c1(SC)nccc(=NC(CNC(c2n[nH]cc2C2CCC2)=O)C(C)C(C)C)[nH]1 65835,CC(=O)CCN=C(NCC(Cl)C(F)(F)F)NC1CC(F)(F)C1 65836,c1(CN(C(C(=C)C)C)CC#CC)cccc2ccccc12 65837,C#CCC(CC(F)F)C(=O)NC1COCCC1N1CCCC1 65838,Cc1nc(C(C)(C)C)sc1C(N1CC(NC(=O)C(O)C2CCC2)C1)=O 65839,c1(C(=O)NC(CNC(C(CC=C)(C)N(C)C)=O)C)ccc2c(c1)C(CC)C(=O)N2 65840,C(=O)(C1=CCCSC1)NC1C(NC(CCc2ccc(OC(C)C)cc2)=O)CCC1 65841,C1(NC(c2ccnc(OCC3CC3)c2)=O)CCOCC1F 65842,CCC(C)CC(=O)NCC(=O)NC1CCCN(CC(F)F)C1 65843,N1(C(CCCc2c(C)ccs2)=O)C(CNC(C2CCC(C(N)=O)O2)=O)CC2CC12 65844,C#Cc1ccc(C(=O)N(C)CCOCCNC(=O)Cc2n[nH]c(=NC)s2)cc1 65845,C12(NC(=O)CN3CCCCC3)CCC(CC1)N(C(C1CC3C=CC1C31CC1)=O)C2 65846,C1(CN(C(CC(=C)C)=O)C)CN(C(c2ccn(C)c2)=O)CCO1 65847,C1(NC(C2CC(CC=CC(=O)NCC3CC(N(C)C)C3)C2)=O)CCC(C#N)C1 65848,CCC(C(=O)N(CCCCCCNC(c1nccnc1C)=O)C)C(C)O 65849,C(=O)(C(F)CCC(C)(C)C)N(C1(C(N2CCC(C(=O)NC)C2C)=O)CC1)C 65850,C1(CC(=O)NCC(CNC(CC=CC=C)=O)C)CCCC1C 65851,Cc1nnc(O)c(C(=O)NC2CN(Cc3cccs3)C2)c1C 65852,C1(NC(CN(C(C)(C)CCNC(=O)C=CC2CCOC2)C)=O)CCCN1N=O 65853,c1(C(=O)NCC2(N(C(=O)COC3=NCCN3)CC)CCCC2C)ncc(F)cc1N 65854,C1(C(=O)OC)(C(=O)N(CCCCN(C)C(C2CC2F)=O)C)CCO1 65855,N1(C(C(C=C)(C)CC)=O)CCOC2(CCN(C(c3cccnc3)=O)C2)C1 65856,N1(C(c2c(C)onc2-c2ccccn2)=O)CC2CC1CN2C(c1coc(Cl)c1)=O 65857,N1(C(CCSC)=O)CCC(C(=O)Nc2ccc(C3CC3)nc2)C1C1CC1 65858,N1(C(C(C)CN(C)C)=O)CCN(C(c2cc(F)n[nH]2)=O)CC1c1ccccc1Cl 65859,C12CCN(CC1(C)C)Cc1cnc(nc1)N2.c1(CC)cc(C)cnc1Cl 65860,C1(C2(O)CCN(C(c3csc(O)n3)=O)CC2)(NC(=O)CCOC2COC2)CC1 65861,C1(C(=O)Nc2cnc(-c3ncccn3)s2)CCCN(C(C2CCCCC2O)=O)C1 65862,N1(C(c2c(C)nc[nH]2)=O)C2CCC1CN(C(=O)CCc1ccc(O)c(O)c1)C2 65863,c1(C(=O)OC)ccnc(N(C)C(=S)Nc2ccc(F)cc2)c1 65864,N1(C(CC2C=NN(C)C2=O)=O)CC(NC(=O)CCCn2c(O)nnc2O)CC(F)C1 65865,c1(N(C)C)c(F)cc(C(=O)NC2CC2C(=O)NCc2nc(Br)cs2)cc1F 65866,CCCCC(O)CC(=O)N1CC(C)(C)CC1C(=O)NC1CCCC1N=[N+]=[N-] 65867,N1(CC(=O)NC(CNC(c2cccc(OC)n2)=O)(C)C(C)C)CCC(=O)NC1=O 65868,c1(NC(C2N(S(CCC)(=O)=O)CCC2)=O)cc(C(=O)OC)cc(C(F)(F)F)c1 65869,C(CCC(O)C(=O)NC1CC1)NC(=O)C(F)F.C12CCC1C(=O)N2 65870,S(=O)(=O)(c1cccnc1NC(CO)C1CC1)NC(C(C)(C)C)c1ncccn1 65871,C1(NC(C2(C=C)CCC2)=O)CCCN(C(c2ocnc2-c2ccccc2)=O)C1 65872,C(C(C)(C)C#CC(=O)N(C)Cc1ccoc1)NC(c1scc(C)c1)=O 65873,c1(C(N2CCC(C(C)NC(C(C)NC(=O)NC)=O)C2)=O)cccc2c1CCCC2 65874,C(=O)(C(F)C1=CCCCC1)NCCN(C(C(Cc1c(C)cccc1)C)=O)C(C)C 65875,N1(C(C2C(C(C)C)(CC)C2)=O)CC(NC(c2cc(=O)cc[nH]2)=O)CC1CO 65876,N1(C(c2c(C)onc2CO)=O)CC(N(C(=O)Cc2ccoc2)C)C2(CC2)C1 65877,c1(C(N2CCCC(C(=O)NC(c3cnc(C)s3)C)CC2)=O)cc(C)cc(C#N)c1 65878,c1(C(N2C(C(N(C(C)CC3CC3)CC)=O)CCC2)=O)cccc(C(F)(F)F)n1 65879,N1(C(c2ccc(OC)cn2)=O)CC=C(C(=O)NC2CC2C2CC2C)C1 65880,c1(CNC(N2C(c3cc(=N)[nH]cc3)CCC2)=O)nc2ncccc2o1 65881,c1(C(=O)NCC(C)(C2CC2)NC(CCS(=O)(=O)NC)=O)ccc(C(C)C)cc1C 65882,Cc1n[nH]cc1C(=O)NCCCC1(CO)CCCC1.C1(C(=O)N)CCC(C(N)=O)C1 65883,CC(C)C(CC(=O)NCCCC(=O)OC(C)(C)C)NC(=O)NC12CCCCC1C2 65884,c1(CC)nc(C#N)cc(=NCC2(NC(C3(C)CC(F)C3)=O)CCCC2)[nH]1 65885,Cc1nc(C)c(C(=O)NC2CCCC(NC(c3cnc[nH]c3=N)=O)C2)o1 65886,Cc1n[nH]c2nc(O)c(C(N3CC(O)(C(C)NC(=O)C=C4CCC4)C3)=O)cc12 65887,N1(C(C2(CNC(C3CCC(C)(C)CC3)=O)CC(=C)C2)=O)CC(F)(F)CCC1C 65888,N1(C(CSS(C)(=O)=O)=O)CC(O)C(O)C1CNC(C1CC(=C(F)F)C1)=O 65889,N1(C(C2(COC)CC2)=O)CCCC1C(=O)OC 65890,CC1(C)CN(C(=O)C(C2CCOCC2)O)CC1CNC(c1ccc(F)c(F)c1)=O 65891,C1(NC(C2N(CCC)CCCC2)=O)CC2CCC(C1)N2C(c1c[nH]c(=NC)s1)=O 65892,c1(NC(=O)NC(c2ccc(C)cc2)c2ccco2)cnc(Br)c(C)c1 65893,c1(OC)ccc(C(=O)N(C2CCCN(C(C3CC(C)(C)C3)=O)C2)CCF)c(Cl)c1 65894,c1(C(N(CCCOCCNC(c2c(C)ocn2)=O)C)=O)sc2ccccc2c1Cl 65895,CC1C(NC(=O)CC(C)(C)C(F)F)C(C)CCN1C(=O)CCOCC(F)F 65896,CC1CC(NC(c2ccnn2CCC(F)(F)F)=O)CN1C(c1ncc(F)cn1)=O 65897,c1(C(=O)NC2C(OC)CN(C(=O)C=CBr)C2)nc(C)c(C)[nH]c1=O 65898,N1(CC(=O)N(C)Cc2cc(Br)cs2)CC(C)(C)OC2(CCCOC2)C1 65899,N1(CC(=O)NCC2C(C(=O)NC(CCSC)C)C2)CCCC1C 65900,C1(NC)CCN(C(C2(CC)CC(C(=O)NCCc3cc(Br)ccc3O)C2)=O)CC1O 65901,C1(CC)CN(C(C2(F)CC=CC2)=O)CCC1NC(C1CCC(CC#N)CC1)=O 65902,c1(NC(=O)C(N2CCCC(Cc3ccccc3)C2)=O)cc(Cl)cnc1Br 65903,C1(C(CC)C)CCCN(C(c2cncc(CNC(=O)C=CC(F)(F)F)c2)=O)C1 65904,C(N=c1[nH]cnc2c1SCCC2)C1C(C)(C)CN(C(c2cnc(C3CC3)s2)=O)C1 65905,C(C(O)CCNC(c1csc(-c2nc[nH]n2)n1)=O)NC(=O)CCc1cnn[nH]1 65906,c1(C(=O)NC(C2CCCN(C(c3cc(C)n(CO)n3)=O)C2)C)ccc(C#N)n1C 65907,C1(C(C)NC(=O)Cc2nnc(O)s2)CN(C(c2ccc(C(F)F)o2)=O)CCO1 65908,c1(C(=O)NC2C(NC(CCN(CC)CC)=O)CC2)cnc(O)cc1O 65909,c1(CC(=O)N(CCCNC(c2nn(C)c(O)c2)=O)CC2CC2)c(F)cccc1C#N 65910,Cc1ccnc(C(N2CC(O)(CN(C)C(C3CC(N(C)C)C3)=O)C2)=O)n1 65911,C12(C(C)NC(C(CC)NC(=O)C=Cc3ccnn3C)=O)CCC(CO1)C2 65912,N1(C(C(CCSC)(C)C)=O)CCC=C(C(=O)N(C)CC2C(C)(C)C2(C)C)C1 65913,c1(NC(C2CN(C(c3n(C)c(S)nn3)=O)CC2F)=O)cccc2c1CCO2 65914,C1(C(CNC(C2C(CCC)C2)=O)O)CCN(C(c2csc(C(C)OC)n2)=O)CC1 65915,C12(C(=O)NC3(CO)CN(c4snc(C(C)(C)OC)n4)C3)CCC(CO)(CC1)CC2 65916,c1(C(N(CC(CC2CC2)C(=O)NC2CC(O)C(O)C2)C)=O)ccc(C#N)cn1 65917,c1(C(N(C)CCOCCCNC(C2CCNC(=O)C2)=O)=O)n[nH]c2c1CSCC2 65918,C(CO)(C(=O)NC(C)C(=O)NCC(O)Cn1cccn1)OC 65919,c1(C(=O)NC2CCCN(C(=O)CSCC(F)(F)F)C2)ccc2c(c1)B(O)OC2 65920,N1(C(CCC#C)=O)CCC(CN(C)C(c2cnc(O)n2C)=O)CC1 65921,CC1CN(C(c2cc(CNC(c3ccoc3C(C)C)=O)[nH]n2)=O)CCC1O 65922,C1(CNC(C=C=C(C)C)=O)CCCCCN1C(=O)CN(C)Cc1ccccc1 65923,C1(C(=O)NCC2(CCNC(c3cc(OC)n[nH]3)=O)CC2)CCCC1S(C)(=O)=O 65924,N1(C(CCOC)=O)CC(NC(c2ccc(F)c(C(C)(C)C)c2)=O)CC2(CC2)C1 65925,C(C(F)C(=O)NCC(O)CCNC(C1(C#N)CCC1)=O)N(CC)CC 65926,C1(CC(=O)NCC2(C(F)(F)F)CCN(C(=O)CC3CC4(CC4)C3)C2)CC2C=CC1C2 65927,C(=O)(C(C)(C)COC)N1CC(C)(C(N(CCCCC=C)C)=O)C1 65928,C1(C(=O)NC(C)CNC(c2cncc(Cl)c2)=O)CCC2(CC1)CC2(F)F 65929,N1(C(C(c2cccc(C)c2)O)=O)CC2CC(C1)C2NC(C1CC1C)=O 65930,c1(C(N2CC(COC)(CNC(C3CCC=CCC3)=O)C2)=O)ncnc2ccsc12 65931,C1(C(=O)NCC2C(CNC(=O)C=Cc3ccncc3)C2)CCC2(CCC2)O1 65932,c1(NC(C2CCCCC2NCc2nc(Cl)ccc2F)=O)cc(Cl)cc(Cl)c1Cl 65933,C1(CC=C)(NC(C2CNC2(C)C)=O)CCN(C(c2ccccc2)=O)C1 65934,N1(C(COc2ccc(C#N)cc2)=O)C2CCC1CC(NC(=O)C(CO)N(C)C)C2 65935,C1(C(N2C(CNC(c3ccc(C(N4CCCC4)=O)s3)=O)C=CC2)=O)C2CC3C(C2)C13 65936,N1(C(CC2CCN(C)C2=O)=O)C2CCC1C(F)C(NC(c1ccc(Cl)cn1)=O)C2 65937,CCC(CC(=O)N1CCCC(N(C)C)C1)NC(C1CC(=C2CCC2)C1)=O 65938,N1(C(CCOC(C)C)=O)CC(CNC(=O)CNC(=O)C(F)(F)F)CC1C 65939,c1(C(=O)NC2CN(C(c3c(C)c[nH]n3)=O)C2)ccccc1N(S(C)(=O)=O)C 65940,C1(C(=O)NCCn2ccc(C(=O)NC(CC=C)(C)C)c2)OCCCC1(C)C 65941,C1(CC)COC(=O)N1.c12coc(n1)CNC(=O)CC1CC(C1)CNC2=O 65942,C1(C(C)C)CN(C(C2CCC3(CCC3)C2)=O)CCN1C(c1cncs1)=O 65943,Cc1noc(N)c1C(=O)N(C(CNC(c1ccc(C2CC2C)o1)=O)C1CC1)C 65944,C(CC(C)C(=O)N1CCC(NC(=O)CC2CC(SC)C2)C1CC)=CC 65945,N1(C(=O)CCc2nncs2)CCCC2CN(C(C34CCCCC3C4)=O)CC12 65946,Cn1nc(C(=O)NC(C(=O)NCC2=NOCC2)C2CCOC2)cc1F 65947,N1(CCN(CC(=O)O)C(c2ccc(F)cc2)=O)C(=O)NC2(CCOC2)C1=O 65948,N1(C(CC=C=C)=O)CCCC12CCN(C(=O)Cn1cc3ccccc3n1)CC2 65949,CC(C)(C)C(C#N)C(=O)NC1COCCC1NC(c1cnc(S)n1C1CC1)=O 65950,C1(C(C)(C)O)CC(Cc2ccc(C(=O)O)cc2)N(CC)C1.C(F)(F)CF 65951,C(=O)(C1=NOC(C)C1)NCCC1(C(=O)NC(c2nc(C)sc2)C)CCC1 65952,n1(CC(N2CCC(O)(C(C)NC(c3cocn3)=O)C2)=O)cnc2sccc2c1=O 65953,N1(C(c2c(CC)cccc2)=O)CC(C(N2CC3CC3(C)C2)=O)C(C)(C)C1 65954,N1(C(=O)NCC(O)Cn2ccnc2)CC2CCC(C1)N2Cc1ccc(O)nc1 65955,N1(C(c2c(C)ocn2)=O)CC2(CCN(C(=O)C(C)(C)Oc3ccc(O)cc3)C2)C1 65956,N1(C(c2cc(C)c(O)cc2)=O)CCCC12CN(C(c1ocnc1C)=O)C2 65957,CC1COc2c(C(=O)NCCCCNC(C3C=CCCC3)=O)cccc21 65958,C1(C(=O)NCC(CO)NC(c2c(COC)nn[nH]2)=O)CC2C(C1)C2(F)F 65959,c1(OC(C(=O)NC(C2(O)CN(C(CC#C)=O)C2)C)C)ccccc1Br 65960,C(N=c1[nH]c(N(C)Cc2ccoc2)nc(=N)[nH]1)C1(C)CC1Br 65961,CC#CCCCC(=O)NC(COC(C)C)C(=O)NC(c1scnc1C)C 65962,N1(C(CN(CCC#C)C)=O)CC(NC(=O)C(c2cccc(F)n2)(F)F)C(C(F)F)C1 65963,C1(NC(CNS(NC)(=O)=O)=O)CC2CCC(C1)C2NC(c1ncoc1C)=O 65964,c1(OCC)ccc(C(C)NCC2OCC2(C)C)c(Br)c1OC 65965,c1(NC2CCCC(CC(=O)NCc3cn(C(C)C)nc3)C2)cncc(C#N)c1 65966,c1(C(=O)NCCN(CCC)C(C23CC(C)C2C3)=O)cnn(-c2nccs2)c1 65967,c1(NC(C2C3CN(C(Cc4c(C)noc4C)=O)C2C3)=O)cnc(C#N)nc1 65968,c1(CC)nc(C)cc(=NC2CC(NC(=O)CC3CC4CCC3C4)C2)[nH]1 65969,C1(C(N(CCC(=O)NC)C)=O)CCCN(C(=O)CCc2cnn(C)c2)CC1 65970,N1(Cc2[nH]nc(C(=O)OC)n2)c2cccc(O)c2CCC1C 65971,N1(C(c2[nH]cc(CC)c2)=O)C2CCC1CN(C(=O)CCc1ccc(C)cc1)C2 65972,Cc1[nH]nc2c1CC(C(N1CCC(CO)(NC(c3cnn(C)c3)=O)CC1)=O)CC2 65973,n1(CC=C)nnnc1C(CC(C)C)NC(C)CC(=O)Nc1ccccc1 65974,C12(CNC(C3C(CNC(C(C)=CC(C)(C)C)=O)C3)=O)CC=CC(C1)OC2 65975,c1(CC(C(=O)N(CCCNC(C2C(OCC)C2)=O)CC)O)ccccc1Cl 65976,c1(CC)ncc(Cl)c(C(N2C3CCC2C(NC(=O)COc2ccccc2)C3)=O)n1 65977,C1(n2cc(CNC3(OC)CCCC(C)(C)C3)nn2)Cc2ccccc2C1C 65978,CCCC(CC)CCC(=O)N1CCC(N(C)C(c2cc(N)ccc2O)=O)C1 65979,c1(C(=O)NC2C(C)N(C(c3cnc4sccn34)=O)CC2)ccc([N+](=O)[O-])s1 65980,CC1CC2CCC(C(=O)NCCC(C)NC(c3ncc(Cl)n3C)=O)CN2C1 65981,c1(C(N2C(C)CCC(NC(=O)CC=C(Cl)Cl)C2)=O)ccn2nccc2n1 65982,c1(C(=O)OCc2cccc(Br)c2)cnc2c(cnn2Cc2ccc3c(c2)OCO3)c1 65983,c1(CN2CC3C(CC)(CC3)C2)cnc2c(c1)NCC(=O)N2 65984,c1(CC(=O)NCC2C(NC(c3cncc(C)c3Cl)=O)C2)cccc2nsnc12 65985,N1(C(C(C2CC(F)(F)C2)OCC)=O)C2CCC1CC(CNC(c1ccsc1)=O)C2 65986,CC1CN(C(c2ncn(C)n2)=O)CCC1CNC(c1cnn(C2CC2(F)F)c1)=O 65987,C1(NC(C2N(C(C(C)N(C(C)=O)C)=O)CCCC2)=O)CCc2ncnn2C1 65988,N1(C(C(F)=C(C)C)=O)CCC(C(F)(F)F)C(NC(=O)C=C2CCN(C)C2)C1 65989,Cc1cnccc1C=CCN(CCCNC(C1CCOC(C)(C)C1)=O)C1CC1 65990,Cc1cc(C(=O)NC2(C)CC(NC(c3cc(Cl)no3)=O)C2)nc(O)n1 65991,C(=O)(C1=C(C)CCC1)NC(C(N1CC(CCC#C)C1)=O)C1CC1 65992,C1(N(C)C(C23CC(CO2)C3)=O)CCC(NC(C2CCCN2C(=O)N(C)C)=O)CC1 65993,C12(C(=O)NCC(CCOC)NC(C3OCCCO3)=O)CCCN(C1)S(=O)(=O)C2 65994,C1(C(N(CCNC(=O)C=CCO)CCOC)=O)CC2CCN(C(C)C)CC12.CC 65995,C1(C#N)(C(=O)NCC2N(C(CCC(CC)OC)=O)CCC2)CC2C=CC1C2 65996,C1(C(N(C2CCN(C(C34CCC(C)(CC3)O4)=O)CC2)C)=O)CC12CCCOC2 65997,C1(C)(C(=O)NC(CN(C(c2ccccc2SC)=O)CC)C)CC(OC)CN1C 65998,c1(-n2cc(CC3CCN(C(C4CC(C)(C)SC4)=O)C3)nn2)cccc2c1CCC2 65999,CN1CCCCN(C(c2cnc(Cl)n2C)C(=O)NC2CCOCC2)CC1 66000,C1(CCCNC(C(C)c2ccco2)=O)CCCCN1C(=O)CSc1nncs1 66001,N1(C(c2nc(CC)sc2)=O)CCC2CCN(C(C3(C)CCOC3)=O)CC12 66002,C#Cc1cccc(C(=O)NC(CNC(=O)CCC2CCC(=O)N2)(CC)CC)c1F 66003,c1(C(=O)NCCN(C(=O)C(C2CCOCC2)O)C(C)C)ccc(Cl)s1 66004,c1(C(=O)NC2CC(F)(CNC(CC=C)=O)C2)cnc(C(F)(F)F)c(F)c1 66005,C1(NC(C=C(C)C2CC2)=O)CN(C(c2cncc(N)c2C)=O)CC1(C)C 66006,c1(C(N2CCC(CSC)C2)C(=O)NCC(C)C)cc(F)c(F)cc1F 66007,CC#CCCC(=O)NC(C)(CNC(=O)CSCC1CCCO1)C(C)C 66008,C(=O)(CCCCN=[N+]=[N-])NC1(C(=O)NCC(C(C)C)(C)O)CCOCC1 66009,CCC(O)C(F)(F)C(=O)NCC(CCNC(C1(n2cc(C)cn2)CC1)=O)OC 66010,C1(OCC)CCCC(NC(c2cc(NC(c3cc(COC)sn3)=O)no2)=O)C1 66011,N(C(=NCCCN(C)C(C)C)N1CCCC(Cc2cnco2)C1)C(C)C 66012,CCCC(C)CCCC(=O)N(CCNC(C1(c2cncnc2)CCCC1)=O)C1CC1 66013,C1(CNC(CC(CC)NC(c2cnc(=N)[nH]c2)=O)=O)OC(=O)CC1(C)C 66014,C1(NC(C2(C)C=CCC2)=O)CC2(C1)CC2NC(c1cnn(CC(F)F)n1)=O 66015,C=C=CCN=c1[nH]c(=NCC2CCS(=O)(=O)C2(C)C)[nH]c2c1SCC2 66016,c1(C(=O)NC2CCN(C(c3c(C)[nH]cc3)=O)C2(C)C)ccc(Br)c(F)c1F 66017,c1(C(=O)NCC2(C)C(NC(c3c(OC)csc3)=O)CCC2)cc2c(Cl)cncc2o1 66018,c1(CN)cccc2c1CN(C(c1cc3n(n1)CC(O)CO3)=O)CC2 66019,n1(CC(=O)NC(CNC(CC(=O)OCC)=O)C(C)C(C)C)ccc2ccc(F)cc12 66020,CC1CC(C)(C(N2CCC(N(C(=O)Cn3ccccc3=O)C)C2)=O)CC(C)O1 66021,c1(C(N(C2CCN(C(C(CCC)C)=O)CC2)C)=O)ccc2nc(C)n(C)c2c1 66022,C(=O)(CCCCC(=O)NC(CNc1nn2cc(C)nc2s1)C1CC1)NC 66023,N1(C(C(C)OC)=O)CCC(F)(CNC(=O)Cc2cncc(C#N)c2)CC1 66024,CCC(C)C(O)C(=O)N1CCC1CC(=O)NC(CCO)C(C)C 66025,C(=O)(C1=CCCOC1)NCCCOCCCNC(c1n(CC)ncc1)=O 66026,C1(NC(CC2(C=C)CN(C(=O)CC(=O)N(C)C)C2)=O)COC2(CCC2)C1 66027,n1(C(C)C)ccc(CC(=O)NCC(C)NC(=O)CC(C)C2CCCCC2)n1 66028,c1(C(N2C(CC)CN(C(C3(CO)CCOC3)=O)CC2)=O)cc([N+](=O)[O-])oc1C 66029,c1(CCC)cc(C(=O)NC2CC(N(C)C(C3(OC)CCC3)=O)C2)cc(O)n1 66030,N1(C(c2cccc(C(C)=O)c2)=O)CCN(C(=O)C(c2ccccc2)C)C(CCO)C1 66031,N1(C(C2(Oc3cn(C)nc3)CC2)=O)CCCCC1NC(=O)CC(O)C1CCCC1 66032,C1(C(=O)NCCC2CC(NC(c3cc(C(=O)OC)no3)=O)C2)CCCC12CCC2 66033,N1(C(CC(C)C)=O)CC(C(=O)NC(C)Cc2cn[nH]c2)OC(C)C1 66034,c1(C(N2C(C)CC2CNC(=O)C(F)OC(F)(F)F)=O)cccc(=O)n1C 66035,C1(CNC(C(COC)C)=O)CCCCCN1C(c1nc(C)ncc1Br)=O 66036,c1(CN(CC)CC)nnc(N2CCC(O)(c3ccccc3C)C2)n1CC 66037,C(=O)(C(F)(F)C(O)C1CC1)N1CCN(C(C2CC(C)C2(C)C)=O)CC1 66038,C1(COC)(NC(=O)C=CCO)CCN(C(C2(CN(C)C)CC2)=O)CC1 66039,c1(NC2CC3CN(C(C(C)n4cncn4)=O)CC32)c(C#N)cccc1[N+](=O)[O-] 66040,C(=O)(C1=CCOCC1)NCC1(C(C)NC(c2cc(Br)cn2C)=O)CC1 66041,C1(NC(=O)CCCC2CCCCC2)CCCN(C(C2CC23CCCC3)=O)CC1 66042,C1(C(=O)NCC(C)C(=O)NCC(C)(C)CSC)(OC)CCOC1 66043,CCC(CCCC(=O)NCc1cnn2ccccc12)NC(=O)CSC 66044,CN1CC2CCN(C(=O)CC3CC3CNC(=O)C=CCN3CCOCC3)C2C1 66045,C(=O)(C(CC(F)(F)F)OC)OC(CCC)CCOC(C(C)(C)C)=O 66046,C1(=O)N=C2C=C(N(C)N2)NCC12CCC2.C(COC)(OC)OCC1CCCO1 66047,C1(C(=O)NC(c2cn(-c3c(C)ccc(C)c3)nn2)C)CCc2nc(C)sc2C1 66048,c1(C(=O)NC2C(NC(=O)CC3C=CCCC3)CCC2)ccc2c(c1)CC(=O)NC2 66049,Cc1cc(C(N2CCOC(C(C)NC(c3cn(C4CCC4)nn3)=O)C2)=O)ccn1 66050,CCCCCC(=O)NC(C1CCN(C(=O)CC(C)Cc2cccc(F)c2)C1)(C)C 66051,CCCCCCC(F)C(=O)NCC(C)(C(C)C)NC(c1cc2ncccn2n1)=O 66052,C1(C(=O)NC2CC2)CNC(=O)CN1C(=O)COCC1CCOC1.CCC1CC(=O)N1 66053,Cc1ccc(CC(N2CCCC(N(C(=O)C(C)CO)C)CC2)=O)c(C)c1 66054,Cc1cccc2[nH]cc(C(N3CCCC(CC(=O)NCc4ccccc4)C3)=O)c12 66055,CCCC(CCC)CC(=O)N1CC(CCNC(=O)C(C)=C2CCC2)S(=O)(=O)CC1 66056,C(C(C)(C)C(=O)N1CCC(C)(CNC(C2(c3cnn(C)c3)CCCO2)=O)C1)OC 66057,c1(C(=O)NCC(C(C)(C)C)NC(C2(C)CCCOC2)=O)cnc(Cl)c(Cl)c1 66058,CC1(C)CC(=O)CCC1C(N1CCCC(C)(NC(=O)CCCCC2CC2)C1)=O 66059,N1(C(Cc2ccn(C(C)C)n2)=O)CC(NC(c2cc(C(N)=O)no2)=O)CCC1C 66060,C1(NC(=O)CCc2cccnc2F)CN(C(C2CCC(O)C2)=O)C2(CCCC2)C1 66061,C(=O)(C(CC)C(=O)NCC1C(C(N2CC(C)(CC)C2)=O)CCN1C)OCC 66062,Cc1ccc(C)c(OCC(=O)NCCN(C(=O)C(C(C)(C)C)c2cc[nH]n2)C)c1 66063,c1(CC(=O)NC2CCN(C(c3ccc(OC)s3)=O)CC2O)ccc2c(c1)COC2 66064,C1(NC(C(C)OCCOCC)=O)CC(OC)CN(C(=O)Cc2ccon2)C1 66065,CCCCC(F)C(=O)NCC1CCC(NC(c2cnoc2)=O)CC1 66066,c1(CC)nn(C)c(Cl)c1C(=O)NCCCC1(NC(c2cnc(O)c(F)c2)=O)CC1 66067,N1(C(c2cnn(C3CCCCC3)c2)=O)CCOC2(CCN(Cc3cncs3)C2)C1 66068,C1(N(C(CC(=O)OCC)=O)C(C2CCN(C)C2)C)C2CCC1CNC2 66069,c1(C(N2C3CN(Cc4ccc(OC)cc4OC)CC32)=O)cc(Br)cc([N+](=O)[O-])c1 66070,c1(C(N2C(C(C)NC(=O)Cc3ccon3)CCC2)=O)cccc(-c2ncon2)c1 66071,N1(C(c2cccc(OC)c2OC)=O)CC2C3CCC(C2C1)N(C(C)C)C3 66072,N1(C(c2ncc(F)cn2)=O)CC2(CCCN(C(c3ccnc4c3CCC4)=O)C2)C1 66073,C1(NC(NCCC(C)=O)=NCCCCC2CC2)Cc2n[nH]cc2C(C(F)(F)F)C1 66074,C(CC(=O)NNC(=O)OC(C)=O)c1cn(C(C(=O)NCCCC)C)nn1 66075,c1(C(=O)NCCCc2onc(C)n2)coc2c1CN(C(=O)CCc1cnco1)C2 66076,c1(CC(=O)N(C)CC2CC(F)CN2C(c2cc(CO)on2)=O)cnn2ccccc12 66077,C1(NC(C2CC(C)(CNC(CCN(C)CCO)=O)C2)=O)CCc2nncn2C1 66078,N1(C(C(CC)C(C)O)=O)CC(CNC(c2cc(S(N)(=O)=O)c[nH]2)=O)OC(C)(C)C1 66079,C1(CNC(c2c(CC)nn(C)c2)=O)CCN(C(c2ccon2)=O)C1(C)C 66080,Cc1cn(C)nc1C(=O)NCC1CN(C(c2cc(CO)on2)=O)CC1C(F)(F)F 66081,C1(NC(CC)=O)COC2(C1)CN(C(=O)CC1(C)CC1(F)F)C2 66082,Cc1cc(F)c2ncc(C(N3CCC(NC(=O)CC(C)O)C34CC4)=O)cc2c1 66083,C1(F)(CNC(CCSCC(C)C)=O)CCCN(C(=O)C(C)Oc2ccccc2)C1 66084,C1(C)(CNC(CSCC#C)=O)CCCN(C(c2cc(F)ccc2OC(F)F)=O)C1 66085,C1(C(=O)OCCC2OCCC(C)(C)C2)CC12CCc1ccccc12 66086,c1(OC)ccc(CC(N2CCC(NC(C3(C)CS(=O)(=O)C3)=O)C(F)C2)=O)cc1F 66087,c1(CN2CCCC(C)(C(=O)NCCC3CCOCC3)C2)ccc2c(c1)CNC2=O 66088,C1(CCOC)CN(C(c2cc[nH]c2)=O)CCN1C(=O)CC1CCCC(C)(C)C1 66089,c1(CC(=O)NCc2c(F)ccc(C(=O)OC)n2)cc(C)c(Br)c(C)c1 66090,C1(NC(c2cn(C)n(C)c2=O)=O)CN(C(=O)Cc2cc[nH]n2)CC(C)(C)C1 66091,c1(C(=O)NC2CCC(CNC(C3(CO)CC(F)(F)C3)=O)C2)sc2ncccc2c1Cl 66092,N1(C(c2c(Cl)ccc(CC)c2)=O)CCC2(CCN(Cc3ccc(F)c(I)c3)C2)C1 66093,c1(SCCC(c2ccccc2)O)cccnc1Cl.c12ccc(cc1)c(=O)[nH]c2=O 66094,c1(CNC(C(C)n2cccn2)=O)ccoc1C(N1CC(OC(C)=O)C1)=O 66095,N1(C(C2(CC)COC2)=O)CC2C(C(N3CCCC(CS(C)(=O)=O)C3)=O)C2C1 66096,c1(C(=O)NC2CC3CCC2N3C(=O)CCN2CCCC2=O)cnc2ccccn12 66097,c1(CO)ccc(C(=O)NC2C=CC(CNC(C(C)OCCOC)=O)C2)nc1 66098,S(=O)(=O)(c1ccc(Cl)c(C2OCCO2)c1)NC(C#C)Cc1cccc(C)n1 66099,N1(C(C2(C#N)C(C)C2)=O)CC=C(C(=O)NCc2cnc[nH]2)C1 66100,N#Cc1ccc([N+](=O)[O-])cc1CN1CCCC(CNCc2c(Cl)cccc2Br)C1 66101,c1(CCC(N2CCN(C(C3C(=C)C3)=O)CC2C)=O)cccc2oc(C)nc12 66102,C1(NC(CCOc2c(OC)cccc2)=O)C(C)CN(C(=O)Cn2ccnn2)CC1C 66103,N1(C(c2c(C)nc(C)[nH]2)=O)CCCC(O)(CCNC(c2coc(Cl)c2)=O)C1 66104,CCC(C(=O)N1CCC1CC(=O)N(C)CC1CCC1)SC 66105,N1(C(C(C)Nc2ncccn2)=O)CC(O)(C(C)NC(CCOCCC)=O)C1 66106,CCC(C(=O)N(C1CCCC1)CCNC(=O)CC(C(C)C)c1ccccc1)C(C)O 66107,c1(NC2CCN(C(=O)NC)CC2)nc2ccccc2nc1NCc1ncnn1C 66108,c1(-n2cc(C34CN(C3)C4=O)nn2)c(F)cc(Cl)cc1F.CN(C)C1CC1 66109,C(c1ccco1)=C(C)C(=O)NCC1CC1NC(=O)CNC(c1nscc1C)=O 66110,C(N=c1[nH]c(=NC)[nH]c(=NC2CC2C2CCOCC2)[nH]1)C1C(CCC)C1 66111,C(=O)(C(F)C(C)(F)F)N(CCCOCCNC(=O)CCc1nc(O)n[nH]1)C 66112,CC1COc2c(NC(N3CCc4cc(Br)ccc43)=O)cnn2C1 66113,N1(C(CC=CC=C)=O)CC2CCN(C(C3CC(=O)N(O)C3)=O)CC(C2)C1 66114,CC(C(=O)NCC1(NC(c2cc(N)c(Cl)cn2)=O)CCCCC1)C(C)C(C)(C)C 66115,c1(CC(C)(CO)NC(C2(c3cccc(Cl)c3)CC(N)C2)=O)ccc(F)cc1 66116,n1(CC)nccc1C=CC(=O)NCC(C)(C)CNC(c1cc(=O)cc[nH]1)=O 66117,C(CC(C)CC)(C(=O)N1CC2C(CO)C2C1)NC(C(CC)OC)=O 66118,n1(C(C(=O)NCCOC(CC)C)C)cc(CC(O)C(C)C)nn1 66119,c1(CCC(=O)N(CC(C)N(C(C(C)O)=O)C)C)ccc(Cl)cc1Cl 66120,CCC(C)(C)C(O)C(=O)N(C(C)CNC(C1CCN(C(c2cccs2)=O)C1)=O)C 66121,N1(C(C(CC)NC)=O)CCc2c(ncn2C)C1C 66122,C1(CC(=O)NCCCN(C(=O)CCC2CCCO2)C(C)C)CCCOCC1 66123,c1(C(=O)OC)cc2c([nH]1)CCN(C(=O)C(c1ccc(N)cc1)(C1CC1)OC)C2 66124,C1(NC(=O)CCC2OCCO2)CCSC12CN(C(=O)C=Cc1cncnc1O)C2 66125,C12(C(=O)NCc3n(CCC)ccn3)CC(CN1C(c1cc(O)cs1)=O)C2 66126,C1(C(=O)NCC(CCOC)OC)CCCCN1C(C1C=C(C)CS1)=O 66127,N1(CCC)CC(C(=O)N(CC(C)NC(=O)C(C)(C)C2CCCO2)C)CC1=O 66128,C=C(C)CCCC(=O)NC(CNC(C1CCCN(CCC)C1)=O)CC 66129,C1(C(N2CC(CNC(C3CC(CN(C)C)C3)=O)C2)=O)CC2(CCC2)C1 66130,C(=O)(C(C(C)C)N1CCCS1(=O)=O)NCC(CC)NC(C1(C)CCNC1=O)=O 66131,c1(C(=O)NCC(CNC(C2(N(C)C)CCCOC2)=O)O)ccc2c(n1)NCC2 66132,CC1CC(C)(C(=O)NCc2cccc(NS(C)(=O)=O)c2)CC(C)O1 66133,N1(C(CCCC)=O)CCC(NC(=O)CCc2ccccn2)C1C(C)(C)C 66134,Cc1ccc(C2CC2)c(NC2CCC3CCC2O3)c1 66135,c1(C(N(C2CN(C(CCS(C)=O)=O)C2)CC2CCCC2)=O)cc2scc(Cl)c2[nH]1 66136,C1(CC=CC)CCCCN1C(c1cn(C(C)C)cn1)=O 66137,c1(C2C(C(N(CCCCNC(=O)CCF)C)=O)C2)nccc2ccccc12 66138,C1(C)(CCNC(c2cc(SC)c(C)o2)=O)CCN(C(c2cnc(OCC)s2)=O)C1 66139,CC1C(NC(=O)C=Cc2cccc(F)c2)C(C)CCN1C(c1ncc(Br)cn1)=O 66140,N1(C(CCC#CC)=O)CCCCC1C1CCCN1C(=O)CCC1CCCCCC1 66141,C#CCC(CC#C)C(=O)N1CCCCC(CNC(=O)COCc2ccccn2)C1 66142,C1(CC(=O)NCCC2CN(C(C3(Cl)CC3)=O)C2)SC2=NCCN2C1=O 66143,C1(C(N2CC(C)(C)C(Nc3ncnc4sccc34)C2)=O)CCCC(F)(F)CC1 66144,N(C1CCCc2ccnc(O)c21)C(C(C(C1CCOCC1)C1CC1)C1CC1)C 66145,C1(C(=O)NCc2n(CCC)ncn2)CC(N=[N+]=[N-])CN1C(=O)C(C)C1CCCC1 66146,C12(CN(C(C3N(C(CNC=O)=O)CSC3)=O)C3CC3)CCN(CC1)CC2 66147,CC1CCC(C)(NC(=O)Cn2ccccc2=O)C1.C12(C)CCN(C1)n1cc2nn1 66148,c1(CNC(=O)CC2OCCO2)cccc(C(=O)NCCC2CCC3CC23)n1 66149,C(C)(C(CC(=O)NCC1(C)CC(C)(C)C1)NC(=O)C(C)C(F)(F)F)OC 66150,CC1CN(C(c2ccc(Br)o2)=O)CC1NC(c1cn(C(C)(C)C)nn1)=O 66151,C1(NC(c2cccc(C)c2)=O)CC2CCC(C1)N2CC1OC(=O)NC1(C)C 66152,N12CC(CC13CCCOC3)NC(=O)CCCSCC2=O.C=C(C)COC 66153,N1(C(c2n(CC=C)ccc2)=O)CC(O)CC1CNC(=O)CNC(=O)NC1CC1 66154,c1(C(c2cnc(C(C(=O)NCC)N3CCCC3)[nH]2)C(=O)NC2CC2)ccccc1Br 66155,C12(N(C(=O)C(=O)NCC(F)F)C)COCCC1CN(C(=O)CS(N)(=O)=O)C2 66156,N1(C(C(=O)NC2CC2)=O)CCC(C(N2CCC(n3ccnn3)C2)=O)(CF)C1 66157,c1(OC)cc2ccccc2cc1C(N1CC2CC(C(=O)NC3CCCC3)C1C2)=O 66158,Cc1n[nH]c2cnc(C(N3CC=CC3CO)=O)cc12 66159,N1(C(C2CN(CC)C2)=O)CCC(NC(=O)NC)C1.C1(N2CC2=O)CC(C#N)C1 66160,c1(C(N(CC(C)NC(C2(CC#C)CC2)=O)C)=O)cnc2c(cnn2C)c1N 66161,c1(C(N2CCC(CCNC(c3cnc(C(N)=O)s3)=O)C2)=O)cnc2n1CCS2 66162,C1(C(=O)NC(CC)Cn2cncn2)CCN(C(c2cccc(F)c2)=O)CC1C 66163,C1(CC)C(NC(=O)CN(CC(C)(C)C)C)CCCN1C(=O)C(C)CC(N)=O 66164,N1(CC(=O)NCCCCCCNC(=O)CC2CC(C(F)F)C2)CCC(=O)NC1=O 66165,N1(CC)CCN(CC(=O)NC2CN(C(C3CC4CC3CO4)=O)CC2O)C(=O)C1=O 66166,c1(CC)ncccc1NC(=O)C(C1CCN(C(=O)CCC2CCCCO2)CC1)C 66167,C1(C)(C(N(CCCCNC(=O)CCc2ccncc2)C)=O)COC(=O)OC1 66168,CCC1=C(C(=O)NCC2C=CC(NC(=O)CC3=CCOCC3)C2)CCCO1 66169,C1(NC(c2c(CC)non2)=O)CCC2CCN(C(c3cnc(Cl)cc3Cl)=O)C1C2 66170,CCCCCCN(CC(=O)NC1CC(CNC(C23CC(C2)C3)=O)(OC)C1)C 66171,c1(C(N(CCCN(C(C2CC(SC)C2)=O)C)C)=O)c[nH]c2cccc(F)c12 66172,C1(NC(C2C(C)CC2)=O)CCC(N(C)C(c2cnsc2)=O)CC1 66173,CCC(=O)CCC(=O)N1C(CC(=O)NCCCC2CCOCC2)C2CCCC12 66174,N1(C(C(CC2CCC2)OC)=O)CC2CCCC(C1)N2C(=O)CN1CCCCC1 66175,c1(CC2C(C(=O)NC(C)CC3CCC3)C2)ccccc1 66176,N1(C(C)=O)CCCC(C(=O)N(C)CC2CN(C(c3ncccc3F)=O)CCO2)C1 66177,N1(C(CC2(C)CC2(Cl)Cl)=O)CC(NC(c2ccnc(N(C)C)c2)=O)CC1CO 66178,C1(N(C(CCNC(COC)=O)=O)C)CN(C(c2ccc(C#N)[nH]2)=O)CC12CC2 66179,c1(C(=O)NCCC2CCC(NC(C=C(CCC)C)=O)C2)ccc2occc2n1 66180,C(=O)(C(O)C(F)(F)F)N(C(C1CCC2CC12)C(=O)NCC1CCOCC1)C(C)C 66181,C12(C(=O)NC(C)Cc3nc[nH]n3)CC(CN(C(=O)C(O)CN3CCCC3)C1)C2 66182,N(C(=N)N1CCC(C(c2ccccc2)O)C1)C(C)C 66183,c1(OC)cnc(C(N2CCCC(N(C(=O)CC3CC3C3CC3)C)C2)=O)cn1 66184,Cc1cccc(C)c1C(N1CCCC(N(c2cc(Cl)ncn2)C)C1)=O 66185,C(CC(C)C(=O)N(C1CCCCC1NC(=O)Cc1ccsc1Br)C)=CC 66186,N1(C(c2c(COC)nccc2)=O)CCCC(n2cc(CC3CCC3)nn2)CC1 66187,C1(CCC(=O)NC(CC)CN(C)C(C2(c3cc[nH]n3)CCC2)=O)CC(C)(C)CO1 66188,CC1CN(C(=O)C(C)(C)F)CCC1Nc1ncnc(=N)[nH]1 66189,c1(SCC)cc(C)ccc1C(=O)NCCC1(NC(c2ccn(CC)n2)=O)CCC1 66190,Cc1cc(CN)nc(NC(C2CSCN2C)=O)n1 66191,N1(C(C2C(C)C2)=O)Cc2nccn2CC(NC(=O)Cc2ccnc(Br)c2)C1 66192,c1(C(N(CCCNC(=O)C2=COCC2)CCO)=O)ccc2nn[nH]c2c1 66193,N1(C(CC=CCCCCC)=O)CCCC1C=CC(=O)NC(c1nnc(C)o1)C 66194,C1(CC(=O)NC2(CNC(=O)Cc3cccc(Cl)c3)CCOC2)CCCC1(F)F 66195,C1(NCC)CCN(C)CC1C#N.c1(-c2cn(C3(C=O)CC3)nn2)cnc(N)cn1 66196,c1(C(=O)NCCC2CCN(C(CCOCC)=O)C2)scc(C)c1OC 66197,C1(NC(C2CCCNS2(=O)=O)=O)CCC2CC1CN2C(c1ccncc1)=O 66198,n1(CC(N2CC(SC)C(NC(C3(C)CCCO3)=O)C2)=O)cnc([N+](=O)[O-])c1 66199,CC1(C)CCCCC1C(=O)NCC1CCC1NC(=O)CN(C1CCC1)C 66200,N1(C(=O)NCC(c2scc(C)n2)C)CC=CCC1C(F)(F)F 66201,Cc1[nH]nc(CO)c1C(=O)NCC(C(C)(C)C)NC(C1CN(c2cnn(C)c2)C1)=O 66202,C1(F)(C(=O)NCC(C2CC2)SC)CCN(C(=O)C(C)(C)C2CCCO2)CC1 66203,C(=O)(C(C)(C)CCC#N)N(C1CCCN(C(=O)CN2CCC(C)(O)C2)C1)CC 66204,N(C1CCc2ccccc21)C(C1(C)N(C(C2CN(C(C)=O)C2)=O)CC(O)C1)=O 66205,c1(C(N2CC(OCCOCCC(=O)NC3CC3)C2)=O)nc2cc(F)ccc2s1 66206,N1(C(C(C(C)C)SC)=O)CC2(C1)CN(C(C1CCC(=O)N1C)=O)CC2CO 66207,C1(C(N2CC(C(N(c3ccccc3)C)=O)C(O)CC2)=O)CCn2nncc2C1 66208,Cc1cccc(C(CNC(=O)NCCN2CC3CC3C2)CO)c1 66209,Cn1cnc2c(NC(C3C4CN(C(c5nc[nH]n5)=O)CC34)=O)ncnc12 66210,c1(CC(N2CCC(NC(CSCCOC)=O)C2)=O)cccnc1OC(C)C 66211,Cc1ccc(CN(C)CCN(C)C(C2CC(c3ccccc3)CO2)=O)cc1 66212,N1(C(COCc2c(C)cccc2)=O)C2CCC1CC(NC(C13CC(C1)C3)=O)C2 66213,C(=O)(CCN=c1cc[nH]c2ccc(C#N)cc12)NC(C)CC.C1COCCOCCO1 66214,N1(CC)N=C(C(=O)NCC(C)NC(c2cc(C)nc(N(C)C)n2)=O)CCC1=O 66215,c1(C(=O)NCC2(NC(C3C(OCC)C3)=O)CCC2)cc2ccc(Cl)cc2c(O)n1 66216,C(=O)(C(CC(C)C)N(C(=O)CCCCCN(C)C)C)NC1(COC)CC1 66217,c1(C(N(CCCNC(C2CC2F)=O)C2CC2)=O)cc(-c2cccs2)on1 66218,CCCCC(C)(F)C(=O)NC(C)CCCC(=O)NCc1cnc(C(C)C)s1 66219,c1(C(=O)NC(CC(F)F)C(=O)NCC(Cl)=CCl)ccc2n[nH]cc2c1 66220,c1(CC(=O)NCC(C)CN(C(=O)C(C)(C)C2CCCC2)C)ccn(C(F)F)n1 66221,N1(c2nnc(CC(=O)O)s2)CC(O)C(O)C1CF 66222,N1(C(C(CC)(C)O)=O)CCCCC(CNC(=O)CCc2csc(=N)[nH]2)C1 66223,N1(C(=O)OCC)CCN(C(=O)NC2CCN(S(C)(=O)=O)C2)CC(O)C1 66224,Cn1cccc(C(=O)NC2CC(CCNC(C3CC3(C)C(F)F)=O)C2)c1=O 66225,C#Cc1cccc(CC(=O)NC(CCC=C)C(=O)NC2CC(=O)NC(=O)C2)c1 66226,Cc1ccccc1-n1nc(CO)nc1CC(c1nc(-c2ccccc2)n[nH]1)(C)C 66227,c1(-c2c(OC)ccc(CN3CCC(CF)CC3)c2)ccc2c(c1)C(=O)NCC2 66228,C(=O)(C1=NOC2COCC12)N1CCC(C)(CC(=O)NCc2c(C)oc(C)c2C)C1 66229,N1(C(CCCCC=C)=O)C(CNC(=O)C(C)NS(=O)(=O)CC)CC2CCCC12 66230,c1(C(N(CC(CN(C(C2(CC(C)C)CCC2)=O)C)O)C)=O)ccc(Cl)nn1 66231,C(=O)(CCC(C)(C)N(C)C)NCC.CC1Cc2cn(nn2)CC2CCN(C1=O)C2 66232,c1(C(N(C(CCNC(c2cc(C(C)C)[nH]n2)=O)C)C)=O)cc2cccn2c(O)n1 66233,C1(CNC(Cc2ccn(CC(C)C)n2)=O)CCN(C(=O)COCCCF)C1(C)C 66234,CCC(C)C(C)(O)CNC(=O)C(C)(CNC(c1ccc(C)c(C)n1)=O)CC 66235,N1(C(C(CC(C)C)C(C)C)=O)CCCC2CN(c3nnc(C(F)(F)F)s3)CCC12 66236,C(=O)(C1=C(C(F)Cl)N(c2cc(C)no2)C(=O)NC1c1ccsc1)OCC 66237,c1(CC)nccc(C(=O)NC2CC=CCC2C(=O)NCCCCC2CC2C)n1 66238,c1(C(N2CCC(N(C)C(C3(C)CCCCO3)=O)C2)=O)ccc(F)c(F)c1F 66239,S(=O)(=O)(c1cccnc1N1CCc2ocnc2C1)NCC=CCCC 66240,c1(C(=O)OC)nccc(=NC2CCCCC2NC(c2nn(C)cc2C)=O)[nH]1 66241,CC(F)(F)CN=c1[nH]c(=NCC2(CCO)CCOC2)[nH]c2c1CSC2 66242,c1(C(=O)NCC(C)NC(=O)CN2CCC(O)CC2)cccc(NS(C)(=O)=O)n1 66243,c1(CC(N2C(CNC(C3CCCOC3)=O)C=CC2)=O)c[nH]c2ccc(Cl)cc12 66244,N1(C(C)=O)CCCC2CN(C(=O)C=CSCc3ccco3)CC12 66245,c1(C(=O)NCC(C)(CO)NC(c2cn(CC=C)nc2)=O)cc2cccnc2s1 66246,c1(C(C)C)ccc(C(=O)NCC(C)N(C)C(c2c(Br)nnn2C)=O)c(O)n1 66247,N1(C(C2C(C)C2)=O)CC(CNC(=O)C=Cc2nccs2)OC(C(F)(F)F)C1 66248,C1(C(N2CC(CNC(c3ccc(C(N(C)C)=O)cc3)=O)C2)=O)CCC(N=[N+]=[N-])C1 66249,N1(c2cccc(C)c2)CCN(C(=NCC(=O)N(C)C)NCCOCCF)CC1(F)F 66250,c1(CNC(CC2(C=C)CN(C(=O)C(C)(O)CC)C2)=O)cn2ccsc2n1 66251,C(=O)(C(CCOC)NC(=O)Cc1cccc(O)c1)NCCC(=O)NCCC 66252,c1(C(CCC(=O)NC(C)CCCOC(C)(C)C)C)ccc(C(C)(C)C)cc1 66253,CC1=CCSC1C(=O)N(C1(CC(=O)NCC2CCCCO2)CC1)C 66254,c1(C(=O)NC(CC=C)CNC(=O)COCC2CCC2)cc(F)c(OC)c(F)c1 66255,C1(CNC(CC2N(C(C(CC)NC(C)=O)=O)CCC2)=O)OC(=O)CC1(C)C 66256,N1(C(CC(C)N(C)C)=O)CCC(C)(C(=O)NCCCC(N)=O)CC1 66257,N1(C(COCC=C)=O)CCC(C(C)(C)NC(=O)C(C2CC2)NC2CCOC2)CC1 66258,N1(C(C2C(NC(C(C=C)OC)=O)CCOC2)=O)C2CCCC1CN(C)C2 66259,c1(C(=O)NC2CCC(C(N3CCCC(F)(CO)C3)=O)C2)cc2ccccc2o1 66260,C1(C2CC2)(CNC(c2n(CC)ncc2Br)=O)CCN(C(c2cc[nH]n2)=O)C1 66261,Cc1ccc(F)cc1C(N1CC2CCC2(CNC(c2nnn(C(C)C)c2C)=O)C1)=O 66262,N1(C(c2c(CC)n(C)nn2)=O)CCC(NC(C2(c3nccs3)CC2)=O)C(F)C1 66263,c1(C(=O)NCC2CC(NC(C3(C#N)CCCOC3)=O)C2)coc2c1C(=O)NCC2 66264,c1(C(N2CCC(C(C)NC(CCC(=C)Cl)=O)C2)=O)cncc(Cl)c1C 66265,c1(N2CCC(CCOC)C2)nc(NCC(C)CCOC)nc2c1ncn2C 66266,CC(CCC(=O)NC(c1ccccc1)(C)C)NC(C1CNC(=O)C1)=O 66267,C(c1cccnc1)=CC(=O)NCCN(CCCN(C)C)C(c1c(C)c[nH]n1)=O 66268,c1(NC(=O)CCCn2cc(CC3CCCOC3)nn2)cncc(C(F)F)c1 66269,C=C1CC2CCCC(C1)N2C(Cc1cnc[nH]1)CC 66270,N12CCc3ccccc3C1CN2.c1(C(N2C(CC)CCC2)=O)c(C)ccnc1Cl 66271,c1(C(N2CC(C(=O)Nc3ccc(OC)nc3)C(O)CC2)=O)ccc(C#N)c(F)c1 66272,C1(NC(C(C(C)C)O)=O)CN(C(c2cnc(=N)[nH]c2)=O)C(C)(C)C1 66273,C12(NC(COCCC)=O)CCOC(CNC(c3cn(C)nn3)=O)(C1)C2 66274,Cc1ccc(OCC(=O)NCC2CC(NC(c3cncc(Cl)c3)=O)C2)cc1 66275,C(=O)(CCCCc1ccc(F)cc1)NCC(C)(CO)NC(=O)CCc1ccco1 66276,C(=O)(CS(=O)(=O)C1CC1)N1CCOCC(NC(C(C2CCC(=O)N2)C)=O)C1 66277,C=CC1OCCC1C(N1CCC(C(C)C(=O)NCc2ocnc2C)C1)=O 66278,CC1(C)CCCCC1=CC(=O)NCC1(C)CCN(C(C2OCCOC2(C)C)=O)C1 66279,C1(C(N2CC(C)(NC(C3(CF)CCNC3=O)=O)C2)=O)CC2C=CCC(C1)C2 66280,c1(CNC(C(COCC)NC(=O)C(F)F)=O)cccc(C)n1 66281,C(=O)(C(C(C)(C)C)NC(C1C=CCC1)=O)NC1(CCCC)CC1 66282,C1(Nc2ncc(C#N)nc2)CC12CCN(C(C1(N3CCCC3)CCC1)=O)CC2 66283,CC(C)C1=NOC(C)(C(=O)NC(C)(C)CCNC(=O)C(C#N)CC2CC2)C1 66284,N1(C(CC(C)SC)=O)CCC(O)C(N(C)C(C2SC3C=CC2CC3)=O)C1 66285,N1(C(C(CC2CCC2)OC)=O)CCS(=N)(=O)C(C)C1 66286,C1(O)(C(C)NC(=O)C=Cc2cc[nH]n2)CCN(C(c2nncs2)=O)C1 66287,C1(NC(C2OCCC(C)C2)=O)COCCN(C(C2CCCN2C=O)=O)C1 66288,Cc1cc(CC(=O)NC2CCN(C(=O)CC3CC(C)(C)C3)CC2C)cc(F)c1 66289,C1(C(CO)NC(c2n(C(CC)CC)ncc2)=O)CCN(C(C2CCC(C)O2)=O)CC1 66290,C(=O)(C(C(C)(C)C)NC(=O)C(C)=CC1CC1)NCc1cc(CC)on1 66291,c1(CNC2C(CCC)CN(C(=O)Cn3cccn3)C2)ccc(F)nc1C 66292,C#CCCCC(=O)N1CCCC1C(=O)N(CC1(Cc2ccc[nH]2)CC12CCC2)CC 66293,C(=O)(C(C(C)(C)C)n1cc(COCC)nn1)OCC.C12CN(C1)C(=O)N2 66294,C1(CCC=C)(CNC(=O)Cc2sccc2C)CN(C(=O)CCn2ccnn2)C1 66295,CCC(CC(=O)N(C1CCCN(C(=O)CCC(F)F)C1)CC)SC 66296,C1(C(=O)OC)C2CC(NC(COc3c(COC)cccc3)=O)CC12 66297,C1(N(C=O)Cc2cc(C)ns2)CCc2ccccc2NC1 66298,CC(C)C(C(=O)NCC1CN(C(N2CCCCC2=O)=O)CC1O)N1CCCCC1 66299,C1(C=O)CC=C(C)CC1.C1(=O)CC(C)N1.C12CC(C1)N(C)C(=O)CO2.CO 66300,c1(C(=O)NCCC2(O)CN(C(c3c(C)coc3C)=O)C2)ccc2sc(=N)[nH]c2c1 66301,c1(CC(C(=O)C(C2CC(N(C(=O)Cn3nccn3)CCO)C2)=O)O)c(F)cccc1F.N 66302,C1(CC)CCC(C(=O)NC2(C(=O)NCC(F)C3CCC3)CSC2)O1 66303,c1(OC)cc(Cl)ccc1C(N1CCCCC1CN(C)C(C1(CO)CC1)=O)=O 66304,N1(C(C2C=C(C)CS2)=O)CCCCC(N(C(=O)CSc2nccn2C)C)C1 66305,Cc1sc2ncc(C(=O)NCC3(O)CN(C(=O)C(C)(C)C(N)=O)C3)n2c1C 66306,C=C(C)C1OCCC1C(N1CCCC(C)(CNC(c2cn(CCO)nn2)=O)C1)=O 66307,c1(C(N2CCCC(O)(CCNC(CCS(N)(=O)=O)=O)C2)=O)ccc(F)c(O)c1F 66308,CCC1=C(C(=O)NC(CNC(c2cn(C(F)F)c(C)n2)=O)CC(F)(F)F)SCCO1 66309,c1(CC(=O)NC2CN(C(C(CC)(C)O)=O)CC2C2CC2)cn2cc(F)ccc2n1 66310,C12(NC(C(C)n3cnnn3)=O)CCCCC1N(C(=O)COC1CCOCC1)CC2 66311,c1(-n2c(C3COC(=O)C3)nc(CC3(C)CC3)n2)ccc(Br)c(F)c1 66312,Cc1cc(C(N2CC(C(N(C3CCCC3)CCO)=O)C3(CC3)C2)=O)nnc1O 66313,Nc1cc(C(N2CCC(=CCNC(c3cccc[n+]3[O-])=O)CC2)=O)cnc1N 66314,N1(C(C(C)Cc2ccccc2)=O)CC2(CCC2NC(c2cc(Cl)no2)=O)C1 66315,C1(C(=O)NC(C2(CO)CC2)C)(NC(c2cc(CCCO)on2)=O)CCC(C)(C)C1 66316,C1(NC(C=CC)=O)CN(C(c2ccc3cncn3c2)=O)CC(C)(C)C1 66317,c1(OC)cc(NC(=O)C(=O)N(C(C)C)Cc2cccnc2)cc(Br)c1.C1C(=O)O1 66318,N1(C(C2CC(CCC)C2)=O)CCC(O)(C(=O)N(CCNC(=O)CC)CC)C1 66319,c1(CC)scnc1C(=O)NC1CCC1NC(=O)CNC(c1ccoc1)=O 66320,c1(C(=O)NC2C(NC(C(CCC)(F)F)=O)CC2)ccc(OC)c(OC)c1C 66321,N1(C(C=CCCC)=O)CCC(C)C(CNC(C2(COC)CCCO2)=O)C1 66322,CCCCCCC(C)(C)C(=O)N1CCCC12CCN(C(C1CC3(CC3)CO1)=O)C2 66323,N1(C(C(COCC)C)=O)CCC2C(NC(=O)CCc3cc(C)on3)C2C1 66324,N1(C(C(CC)CC)=O)CCC(C2CCN(C(=O)C(C)OC)CC2)CC1 66325,N1(C(C2C(C)(CC)C2)=O)CC2CC(C(=O)NCC(C)OC)(C2)C1 66326,n1(CC(=O)NCC2N(C(C3C(CC(C)C)C3)=O)CCCC2)cccc(N)c1=O 66327,N1(C(C2(CC#C)CCOCC2)=O)CC2CCC2(CNC(=O)Cc2cnn(C)c2)C1 66328,C(=O)(C1=CCCOC1)N1C(C(=O)NCC(CC)(C)O)CCCC1 66329,C1(C(=O)Nc2c(CC)c(Cl)ncn2)CN(C(=O)CC(C)(C)O)Cc2ccnn2C1 66330,c1(CSCC(CN(C(=O)C(C)N(C)C)CC)O)coc2c(C)cc(COC)cc12 66331,c1(CC(=O)NCC2CC(NC(=O)CC3(O)CCOCC3)C2)cncnc1O 66332,CC1CN(C(C2CCCC2(F)F)=O)CC(C)N(C(=O)CCc2cc(Cl)cs2)C1 66333,c1(CNC(C2CC(=C)CN2Cc2cccc(C)c2O)=O)cn2cc(Cl)ccc2n1 66334,C(=O)(CCCC(N)=O)NC1CN(C(CSC)=O)C(C)C1 66335,C1(C(N(C(CC)COC)C)=O)CSCN1C(=O)C(C)CSC 66336,C1(OC)CN(C(c2n[nH]c(C)c2Cl)=O)CC1NC(=O)CCc1nc(C(C)C)no1 66337,C1(O)(C(=O)NCC(C)C)CCCN(C(c2cccc(C(N)=O)n2)=O)C1 66338,C(=O)(C(CCC(N)=O)NC(C)=O)NCC1CN(C(CN(C(C)=O)C)=O)CC1C 66339,N1(C(C=CC(CC)C)=O)CCC(O)(CCNC(C2CCC=CCC2)=O)C1 66340,N1(C(Cc2nc(C)sc2)=O)CC(NC(=O)CCC(=O)c2ccc(O)cc2)C(C)C1 66341,c1(COCC)cnc(N2CCOC(CNC(=O)C(F)C3CCOC3)C2)nc1 66342,Cc1cnn(CCCN2CC(CCOC(C)(C)C)C2)c1.C1(=O)C(CN(C)C)N1 66343,c1(C(N2CCC(NC(C=C(CCC)C)=O)(CC)CC2)=O)cccc2c1C(=O)NC2 66344,C12(C(=O)NC(C(C)C)(C)CNC(=O)C(C)(C)N3CCCC3)CCCC1CC(=O)C2 66345,CC1CC(C(=O)OC(C)(C)C)CN1C(=O)Oc1c(C(=O)NC)cccc1 66346,C#CCC(CC(=O)N(C1CCC1)C1CC1)NC(=O)C(COC)CC 66347,c1(C(N(CCC)CCNC(C2CCN(C)C2C)=O)=O)c(OC)ccc(Cl)c1Cl 66348,c1(C(N(C)CC2(NC(Cc3c(C)nc(C)s3)=O)CC2)=O)ccc2oc(O)nc2n1 66349,c1(C(N2C(CNC(c3ccc(OCC)s3)=O)CC2)=O)cn(C)c(C(F)F)n1 66350,c1(C(=O)NCC2(CO)CN(C(C3(COC)C=CCC3)=O)C2)cnc2cccnn12 66351,N1(CC)CCN(CCNC(=O)C(C)NC(c2cc(COC)ccn2)=O)CC1 66352,C(=O)(C(C)(CO)N(CC(F)(F)F)C)N(CC(C)NC(=O)Cc1cc(Cl)cs1)C 66353,CC(C(=O)NC1CC(F)(NC(=O)COCP(C)(C)=O)C1)C(=O)OC(C)(C)C 66354,CCC(CC(=O)N1CC(CNC)CC1C)CNC(C1CC12CCC2)=O 66355,c1(NC(C2C(C)C2c2cc[nH]n2)=O)ccccc1C1CC1 66356,c1(C(=O)NCC(C2CC2)NC(C(CC)N(C)C)=O)cnn(C)c1S(C)(=O)=O 66357,C1(NC(C(C2CCC2)OCC)=O)CN(C(=O)Cc2cc(C)cc(C)c2)CC1(C)C 66358,CCC(C)CC(=O)N1CC(NC(c2cc(CSC3CC3)on2)=O)C(CO)C1 66359,Cc1ccc(C(=O)NC(CNC(c2nc(F)ccc2Cl)=O)C(C)C)c([N+](=O)[O-])c1 66360,c1(C(=O)NCCN(C(=O)C(O)CCC(C)C)CCC)ccc2oc(=N)[nH]c2c1 66361,c1(C(N2CC(N(C(C3C(CC(C)C)C3)=O)C)C(F)C2)=O)ccc(C(F)F)c(Cl)c1 66362,C(CCC(C)(C)N)N(C)C(=O)OC(C)(C)C.n1(CCO)cc(C(O)CO)cn1 66363,C1(N(C(C(C)OCCOC)=O)C)CCCC2CN(C(=O)CCc3cccs3)CC12 66364,C1(CC)C(NC(c2c[nH]c(=N)s2)=O)CCN1C(=O)CC1CCC12CCC2 66365,N1(C(CC23CC(C)(OC2)C3)=O)CCCCCC(NC(c2scnc2C2CC2)=O)C1 66366,C1(OC)CCCN(C(C2CCN(C(c3c[nH]c(=NC)o3)=O)C(C)C2)=O)CC1 66367,C(CC(CC)C(=O)NC12CCC1CN(C(=O)Cc1ccc(OC)nc1Cl)C2)=CC 66368,N1(C(C2(C)C(C(=O)OC)CC2)=O)CCN(C(c2cnns2)=O)C(CCO)C1 66369,Cc1cccc(C(=O)NCC(C2CCN(C(=O)C(O)C(C)C)CC2)(C)C)n1 66370,N1(C(C(N2C(Cc3c(C)cncn3)CCC2)=O)=O)CCC(O)(C(F)(F)F)CC1 66371,C1(CNC(C(C)NC(N)=O)=O)CN(C(=O)CC2(C#N)CC2)CCC12CCOCC2 66372,C12(CNC(CCOCCOC)=O)CSC(C1)C2 66373,c1(C(=O)NC(CCNC(COCCC#C)=O)C)cc(Cl)cc2ccccc12 66374,C(C)(C(=O)OC(C1(C)C(CNC(C2(C(N)=O)CSC2)=O)C1)=O)N(C1CC1)CC 66375,Cc1nc[nH]c1CC(O)C(=O)NCC(F)CNC(c1cn(CC(F)(F)F)nn1)=O 66376,C1(NC(c2ccc(C)cn2)=O)CC2CCC(C1C)N2c1ncnc2c1CCCC2 66377,c1(NC(C2(C)CCN(c3cccnn3)C2)=O)ccc(Br)nc1Br 66378,N1(CC(N2CCCC(CCC(=O)OC)C2)=O)CC(=O)CCC1=O 66379,c1(COC)ccoc1C(=O)NCC(CNC(=O)Cn1[nH]cnc1=N)CO 66380,C1(C)(CCC)CCN(C(C2CC(C)CCN2C(=O)C(COC)CC)=O)CC1 66381,C1(CNC(CN(C(c2cnc(C(=O)OC)cn2)=O)CC)=O)CC(CO)C1(C)C 66382,C1(CNC(CC2CCCC(C)C2)=O)CC(C)(C)CN1C(=O)CC1C=CCC1 66383,N1(C(CC2CC(=C)C2)=O)CCN(C)CC1C(N1CC(CCOC)C1)=O 66384,c1(OCCC(N2Cc3nnsc3C2)=O)cc(Br)cc(F)c1F 66385,C(=O)(CC(C(F)(F)F)c1ccon1)NC1(CCCNC(C2=NOC(C)C2)=O)CC1 66386,c1(CC)[nH]nc(C(N2CC(OC)C(NC(c3ccc(CC)[nH]3)=O)C2)=O)c1[N+](=O)[O-] 66387,c1(C(=O)NC2C(C)CN(C(c3cc(CCO)on3)=O)C2)ccc2c(c1)CC2 66388,CC1CCOC(C2CCOCC2)C1.C1C(c2ccccc2)C(=O)NCCO1 66389,C1(CNC(C(C)NS(CC)(=O)=O)=O)CCC(F)(CNC(=O)CCCSC)CC1 66390,C1(C(N2CCC(C)(O)C2)=O)CC2(CCN(Cc3cc(F)c(F)cc3Cl)CC2)CO1 66391,c1(C(=O)NC2C(C)N(C(=O)COC(F)(F)F)CCC2)c[nH]c2cccc(C#N)c12 66392,C(CNC(=O)Cc1cc(C)nn1C)(CC(=O)NCC1CCOC1=O)OC 66393,C(=O)(C(C)CCCC(C)C)N1C(CN(C(C2CC(=O)NC(=O)N2)=O)CC)CCCC1 66394,CC(C)CS(=O)(=O)N1CC(NC(c2ccc(Cl)nc2)=O)C(O)C1 66395,N1(C(c2cccc(NC(C)=O)c2)=O)C2CCC1CN(C(=O)C1=CC(C)(C)C1)CC2 66396,O=C(C1=CCCC1)NC1CC(NC(c2cc(C3CCC3)[nH]n2)=O)C1 66397,C12(C(N(C)CC3COC(=O)N3)=O)CCC(CC1)N(C(=O)CN1CC3CC3C1)C2 66398,C1(CC(=O)N(CCN(C(C(=O)NCC2(CNC(C)=O)CC2)=O)C)C)CCCCC1 66399,Cc1ccc(C)c(C(=O)NCC2(C(N3CC4(CC4)C3)=O)CC(C)(C)C2)c1 66400,C1(CNC(CC(C(C)C)C)=O)COC(C)(C)CN1C(c1cc(O)cc(O)n1)=O 66401,C1(C(N(CCCC)C2CC2)=O)CCC(C)(C)N(C(=O)CCOC(C)=O)C1 66402,Cc1ccn2cc(C(N3CC(C)N(C(c4cnns4)=O)CC3C)=O)nc2c1 66403,c1(C(C)(C)C)cc(CNC(c2ccc(F)c(N(C)C)c2)=O)cc(F)c1 66404,S(=O)(=O)(c1cc(C)cc(Br)c1)NCc1ccc(NC2CCN(C(C)=O)CC2)cc1 66405,C#Cc1cnn(C)c1C(N1CCCC(CC(=O)NCCC(C)CCO)CC1)=O 66406,C1(C)(CC)CC(NC(C23CC2CCN3C(c2cc(C)[nH]n2)=O)=O)CCO1 66407,c1(C(N(CCNC(c2cc(CC)ncn2)=O)CC2CC2)=O)sccc1S(C)(=O)=O 66408,N1(C(C2(CCC)CC2)=O)CCN(C(=O)CC)CC1C1CCCC1.CC=CC 66409,C1(NC(c2c(OC)n[nH]c2)=O)CN(C(c2cnsn2)=O)CC1O 66410,C1(C(=O)NCC#CCNC(=O)C(F)(F)C2(O)CCC2)CCc2nc[nH]c2C1 66411,C1(NC(C=CC(=O)OCC)=O)CC(C(F)C(=O)NC2(C)CC2)C1 66412,N1(C(C(CC)O)=O)CCCC(CNC(=O)Cc2ccc(OCC(F)(F)F)cc2)C1 66413,C1(NC(C2CN(C)C(=O)CC2)=O)CCN(C(=O)CCc2cnc[nH]2)CC12CCC2 66414,C1(NC(c2ccnc(Cl)c2)=O)CN(Cc2cccnc2O)CC1(F)F 66415,c1(OCC)ccc2cc1-c1ccc(o1)NC2.C1(C(=O)O)(CO)CCC1 66416,CCCCC(CNC(c1ccccc1)=O)NC(C1CC(=O)N(CCC(C)C)C1)=O 66417,c1(C(=O)NC2CCN(Cc3cncc(Cl)n3)CC2F)ccc2ncsc2c1 66418,C1(NC(c2cccc(OC)c2)=O)CC(F)CN(C(=O)Cc2cccc(O)c2)C1 66419,Cc1cc(Cl)ccc1NC(=O)NC12CC(CCC(=O)NC(C)CO)(C1)C2 66420,C1(NC(CC2(NC(Cc3cn(CC)nn3)=O)CC2)=O)CN(C)NC1=O 66421,Cc1c(C(=O)NC2CCC(Cn3cc(-c4cncs4)nn3)CC2)cccc1CO 66422,Cn1cc(C(N2CCC(C)(CNC(c3nsnc3O)=O)C2)=O)ncc1=O 66423,N1(C(CC2CCCC(C)(C)C2)=O)CC2(CNC(C3(C)CC3(F)F)=O)CCC1CC2 66424,C(=O)(C(=O)N=S(C)(C)=O)NCC1CCC(NC(C(C)Cc2ccccc2)=O)C1 66425,CC1(C)CCCCC(NC(c2cnoc2-c2ccc(Cl)s2)=O)C1 66426,C1(C(N2CCCC2c2ccccn2)=O)CCCC2CC12 66427,Cc1cc(C(N2CCOC(CNC(C3CCN(C)C3C)=O)C2)=O)c(C)n1CC1CC1 66428,C(=O)(CCCCN=[N+]=[N-])N1CC(CNC(c2ccc(C)s2)=O)N(C)CC1 66429,N1(C(C2(C)CCC(C)C2)=O)CC(C(=O)NC(C)(C)C(F)F)C2(CCC2)C1 66430,C1(S(C)(=O)=O)(C(=O)NCC2CCN(C(C(CC=CC)C)=O)CC2O)CCOCC1 66431,Cc1cnc(O)c(-c2cccc(CN)c2)c1.N12CCC(C1)OCC2 66432,c1(N(C2CCCN(C(c3cncn(C)c3=O)=O)C2)C)ncc([N+](=O)[O-])cc1Br 66433,C1(NC(Cc2nc(C)oc2)=O)C=CCN(C(=O)C(C)Oc2cccc(O)c2)C1 66434,N1(CCC)CC(C(=O)N(CCCCNC(c2ccc(C(=O)OC)[nH]2)=O)C)CC1=O 66435,c1(N(C)C)ccc(CNc2cccnc2I)cc1 66436,N1(C(C(CC)OCC)=O)CC2CCC1C(CNC(c1cc(C3CC3)[nH]n1)=O)C2 66437,CCC(CC)CC(=O)N1CCN(C(c2csc(-c3ccccc3)n2)=O)C2CC12 66438,c1(C(N2CCC(O)(CN(C)C(C3CC3C(N)=O)=O)CC2)=O)cc2ccncc2s1 66439,N1(C(C(C)(C)SC)=O)CC(NC(c2csnn2)=O)C(c2nccn2C)C1 66440,C1(S(N)(=O)=O)(CN(C)C(=O)NC(c2ccccc2F)c2ccccc2)CC1 66441,C1(NC(C(CCSC)NC(C2(N(C)C)CCCC2)=O)=O)CCn2ncnc2C1 66442,C1(NC(CC2C(C)C2)=O)CCC(NC(c2ccnc(OCCO)c2)=O)CC1 66443,c1(N2CC3CN(CC)CC3C2)nc2c(c(=NC3C=C(C)CCC3)[nH]1)COC2 66444,c1(OC)ccc(Cl)c(C(N2CCOC3CCC23)C(=O)NCCCF)c1F 66445,n1(CC(=O)NCC(CCNC(C2(CC)CC(C)(C)C2)=O)O)nnc2c1CCCC2 66446,N1(C(C(C2CC2)NC(c2c(C)cco2)=O)=O)CCCNC(=O)C1 66447,c1(C(N2CCN(C(C(CC)C)=O)CC2COC)=O)cnc2ncnc(O)c2c1 66448,c1(C(=O)NCC2CC(CNC(c3n(C)nnc3)=O)OC2)ccc2nc(S)[nH]c2c1 66449,Cc1cc(N)cnc1C(=O)NCCCCN(C)C(C1CC(C)(C)C1)=O 66450,CC1SCCN(C(=O)C=CCC2(C(=O)NCc3ncc[nH]3)CCC2)C1C 66451,C=CCC(C)(C)C(=O)NCc1cccc(NC(=O)CNC2CCC3CC3CC2)c1 66452,C1(C(=O)NCC(C)NC(C2(CC#C)CCCCC2)=O)CC2(CC(=C)C2)C1 66453,C1(C(N(CC2N(CC)CCC2)CC)=O)CN(C(=O)C2=COCCC2)CC(C)(C)C1 66454,c1(OC)cc(-c2cccc(C(=O)Nc3cnn(C4CC4)c3)n2)ccn1 66455,CCCC(C(=O)OC)C(=O)NC(C)CN(C(=O)C(c1cccc(C)c1)C)C 66456,N1(C(C2CCC(CCC)N2C(c2cc(CC)[nH]n2)=O)=O)CCC(N(C)OC)CC1 66457,N1(C(C(COCC)(C)C)=O)CC(CNC(C23CC(C)(CO2)C3)=O)CC(C)(C)C1 66458,C1(O)(C(N)=O)CCCN(C(C2CCCCN2C(C2(F)CCCCC2)=O)=O)C1 66459,CC1(C)C(NC(=O)CCn2cncn2)CC1C(=O)NCC#CC(F)(F)F 66460,Cc1cc(CCC(N2CC3(C)CC2C3NC(c2cncc(Cl)c2)=O)=O)cc(C)c1 66461,C(C(C)C)(C(O)C(=O)NC1CCCC(CC(N2CCC(O)C2(C)C)=O)C1)OC 66462,c1(OCC=C)ccc(Cl)nc1C(=O)NC1(CN(C(=O)C(C)O)C)CC1 66463,C1(NC(C(C)OC(=O)OCC)=O)CN(C(=O)CO)CC2(CCC2)C1 66464,N1(CC(=O)NC(C=CC(=O)NC(c2ccnc(O)c2)C)(C)C)C(=O)CNC1=O 66465,C1(NC(C2CCCC23CC3)=O)CCN(C(C2CC3(CCC3)CO2)=O)CC1F 66466,c1(CC(N2CC(CCNc3c(OC)cccc3)OCC2)=O)c[nH]c2ccncc12 66467,C1(NC(c2ccc(C=C)cc2)=O)CCN(c2ncc(C(F)F)cn2)C12CCC2 66468,N1(C(c2n(C)c(C#N)cc2)=O)CCC2(CC(NC(=O)C(C)(C)c3cnsc3)C2)C1 66469,N1(C(C(C)(C)NC(=O)CN=[N+]=[N-])=O)CCCC(c2ccncc2)CC1 66470,c1(C(N2CC(NC(CNC3(CCOC)CCC3)=O)(CO)C2)=O)ccc(C)cc1 66471,c1(C(N2CCC(C(=O)NCc3ncccn3)C2)=O)ccc(I)c(Cl)c1 66472,C(C(C)(C)C(=O)N(C)CC1CCN(C(C2CN(C(C)C)CCO2)=O)C1)OC 66473,N1(C(C(C=CCCC)O)=O)CCN(C(C2(COC)CC2)=O)CC1C(F)F 66474,c1(NC2CN(C(C34CCC(F)(CC3)CC4)=O)CC2C(F)F)nc2ccccc2o1 66475,CCC(CC(=O)NCc1ccc(CNC(=O)C(O)CCSC)cc1)C(C)(C)C 66476,c1(C(=O)NC2(CC)CN(C(c3ncn(CC)c3)=O)C2)ccc2cccnn12 66477,c1(C(c2n(CCCC)nnn2)NC23CC(C2)C3)ccc(OC)c(C)c1 66478,CON(C)CCNC(C1(C2CCCN2C(c2n[nH]cc2Cl)=O)CC1)=O 66479,C(=O)(N=c1[nH]c(Cl)ncc1O)c1n[nH]c2cccc(-c3c(C)cc(F)c(C#N)c3)c21 66480,N#Cc1ccc(CCC(=O)NC2(C(F)(F)F)CCCNC2)cc1 66481,c1(C(C)NC(=O)Cc2csc(C(=O)OC(C)(C)C)c2)ccc(N2CCOC2=O)cc1 66482,Cc1cc(C)c(N(C2CCOCC2)C(C(=O)NC(C)(C)C)c2cc[nH]n2)c(C)c1 66483,c1(C(=O)NCC2(F)CC(NC(c3c(OC)c[nH]n3)=O)C2)ccc(C)c(Cl)c1 66484,c1(C(=O)NCc2cc(C(=O)NCCCCCC=C)sc2)cncn(C)c1=O 66485,CC(C)CC(C(=O)OC(=O)C(C)NC(N)=O)N(C(=O)C(CO)NC)C 66486,C1(C)(NC(CN(CCC)C)=O)CCN(C(C23CC(C(=O)OC)(C2)C3)=O)CC1 66487,N1(C(c2cc(OC)cc(C)n2)=O)CCC(C)N(C(C2CCCC(=O)CC2)=O)CC1 66488,C12(CNC(=O)CCN3CCCC3)CCC(C1)N(C(=O)CCC(=O)C1CC1)C2 66489,C(C(C(=O)N(CCC(N1CC=C(C)C1)=O)C1CC1)OC)OC 66490,C(=O)(C1=CCS(=O)(=O)C1)N1CC(NC(C(C=C)c2ccccc2)=O)C1 66491,c1(NC(C2CC(C(=O)Nc3ccsn3)C2)=O)nccc(-n2ccnc2)n1 66492,Cc1nc(C2CCC2)oc1C(=O)NC(C)(C)CNC(C1(C#N)CC1C)=O 66493,CC1(C)C(NC(=O)C(C)(C2CCC2)NC(=O)COC2CCCOC2)C1(C)C 66494,N1(C(C2=CC(O)C(NC(c3nncc(OC)c3)=O)C2)=O)CCCC(C2(C)CC2)C1 66495,C1(O)(C(N2CCCC(c3c(C(N(C)C)=O)nco3)C2)=O)CN2CCC1CC2 66496,CCC(C)CC(=O)C(=O)NC(C)C(=O)NCc1cccnc1 66497,Cc1nnc(=NCC2(CC(C(=O)C(C)C(C)C(F)(F)F)=O)CC2)[nH]c1C.N 66498,c1(NC(c2c(CNC(COC(CC)(C)C)=O)ocn2)=O)cc(N(C)C)ccc1F 66499,N1(C(C(C)=C(C)C)=O)CCC(F)(F)C(CNC(c2cnoc2-c2ccco2)=O)C1 66500,CCC(C(C)(C)O)NC(=O)C(C)CNC(c1ncn(C)c1C)=O 66501,C1(C(N2CC(N(C)C3CC3)C2)=O)CN(C(C2(F)C(C)(C)C2(C)C)=O)CC1C1CC1 66502,n1(CC)nc(C(=O)NCc2nc(C(N3CCN(C(C)CO)CC3)=O)co2)cc1C 66503,N1(C(c2c(C)ncnc2C)=O)CC2(CC(NC(=O)CC3CC3)c3nccn32)C1 66504,N(C(=NCCF)N1CCC2(O)CCOCC2C1)CCC1(C)CCCCC1 66505,CC1CCCCN1C(=O)C(=O)N(CC(c1ccc(Cl)cc1)C)CCO 66506,c1(C(N2CC(OCCCOC)C2)=O)ccc(C)cc1.c1(C(=O)N)cnn(C)c1C 66507,c1(C(=O)NC2CCCN(C(C(n3cc(Cl)cn3)C)=O)C2)c(Cl)cccc1[N+](=O)[O-] 66508,C1(NC(c2nc(CC)oc2)=O)CCC2CCN(C(c3cnoc3C3CC3)=O)C1C2 66509,CC1CCC(NC(=O)C=Cc2ccc(C(N)=O)o2)CN1C(c1nnn(C)c1N)=O 66510,c1(C(=O)NCC2C(CNC(C3C(C)(C)C3)=O)C2)cc(Br)c(C2CC2)s1 66511,C1(CNC(c2cc(C(F)(F)F)n[nH]2)=O)CC2C(O)CC2O1 66512,CC12CCCC1N(C(c1cnc(C(F)F)nc1)=O)CCN(C(c1ccsc1Cl)=O)C2 66513,Cc1cc(C(=O)NC2CCN(c3nnc(C(N)=O)s3)CC2)nc2[nH]nc(O)c12 66514,C1(C)(C(=O)NCC2C(C(=O)NCC(C3CCCCC3)C)CC2)CC(F)C1 66515,C#Cc1cccc(CC(=O)NC2(C(N3CC(N4CCCC4)C3)=O)CC(CO)C2)c1 66516,C1(NC(c2ccc(C)cc2)=O)COC2(CCN(C(C3(C)C(C)(C)C3(C)C)=O)C2)C1 66517,c1(C(=O)NCCCNC(C(C)CN(C)C)=O)ccc(C2CCC2)cc1 66518,Cc1c(C(=O)NC2(CNC(c3cnc4n3CCS4)=O)CC2)oc2ccc(Br)cc12 66519,N1(C(c2c(C)[nH]cc2C(F)(F)F)=O)CCCC(NC(c2csc(O)n2)=O)C1C 66520,c1(C(N2CC(CNC(C=CC)=O)N(C)CC2)=O)cc2cccn2cn1 66521,N1(c2ccnc(C)n2)CC(CNC(c2nc(C)cc(C)n2)=O)OC2COCC12 66522,c1(C(N2C(C)C(NC(=O)Cc3ccno3)CC2)=O)ccc(Cl)cc1N 66523,C1(C(CC2(CC(=O)NC(CCC)=O)CC2)(C)O)CCN(C(=O)C#CC2CC2)CC1 66524,c1(CCC(N2C(C)(C(=O)NCc3cc(Br)co3)CC2)=O)cccc(F)c1Br 66525,c1(CC(C(=O)NCC(CO)NC(C2(C)CC=CCC2)=O)OC)ccccc1F 66526,c1(CC)nc(=N)[nH]cc1C(=O)NC1CCN(C(=O)C(F)C(C)(F)F)C1 66527,CC(CC(F)F)C(=O)NC1CC2(C1)CN(C(=O)C(C)Cc1ccncc1)C2 66528,Cc1cc(C(N2Cc3ccccc3C2)=O)c2c(c1)CCCN2 66529,C1(NC(C2C(CCOC)C2)=O)(CO)CCN(C(=O)C=Cc2ccc(C)nc2)CC1 66530,C(=O)(CCCC(C)NC(c1ccncn1)=O)N1CC(CCn2c(C)ncc2)C1 66531,C1(C(=O)NCCCCNC(C2SCCS2)=O)C2(CCC2)C12CCC2 66532,N1(C(C(C(C)C)F)=O)CC2(CNC(c3ccc4c(c3)OCO4)=O)CCC1CC2 66533,c1(C(=O)NCC2CC(OC)CN2C(C2CC(SC)C2)=O)ccc2nc(C)nn2c1 66534,CC(O)CC(C)(C)CNC(C1(CO)CCN(C(c2cc[nH]n2)=O)C1)=O 66535,c1(C(N2CC(N(C(Cc3cnc(C)o3)=O)C)C2)=O)cc2nn[nH]c2cc1F 66536,N1(C(=O)NC2CCN(Cc3ccccc3)C2)CCC(C#CBr)CC1 66537,C1(NC(c2cc(C(F)(F)F)on2)=O)CC2CCC(C1)N2C(c1cccc[n+]1[O-])=O 66538,Cc1cc(C(N2CSCC2C(=O)NCc2cc(Cl)ccc2O)=O)cc(O)n1 66539,C1(OC)CC(C(N(C2CCN(C(C3(CCCC)CCC3)=O)CC2)C)=O)C12CCC2 66540,C1(NC(c2nnn(C(C)(C)C)n2)=O)C(C)CCN(C(=O)CSC(F)F)C1C 66541,C1(OC)(CNC(c2cc(C(C)(F)F)ccn2)=O)CCN(C(C2(C)C=CCC2)=O)C1 66542,N1(C(c2c(-n3cc(CC(=O)O)nn3)cccc2)=O)CC2CC3CCCN3C2C1 66543,C(=O)(C1=CN=C2N=CNN2C1)N(C1CCCN(C(C(C)(C)OC(C)C)=O)C1)C 66544,N1(C(C=CCC(C)(C)NC(CCN(C)C2CC2)=O)=O)CCC2CN(C)CC2C1 66545,c1(OC)cccc(C)c1CN1CC(c2ocnc2CNC(=O)C(O)C(C)(C)C)C1 66546,Cc1cncc2cc(C(N3CCN(C(=O)C(F)C(F)(F)F)C4CCCC34)=O)sc12 66547,CC1(C)C(C(=O)NC(C2(NC(=O)CSC(F)F)CC2)=O)CC1CN1CCCC1 66548,n1(C(c2cn(CCC3=CCCCC3)nn2)C)c(S)nc2c(Br)cccc2c1=O 66549,N1(C(c2c(C)noc2N)=O)CCCCC(NC(c2cnc(N(C)C)o2)=O)C1 66550,c1(CNC(C(C2(OC)CCOCC2)(F)F)=O)ccc2c(c1)NCCCN2 66551,C(=O)(CC(C(F)(F)F)OC)NC(CCNC(C1CN(CC)C(=O)CC1)=O)(C)C 66552,Cc1cc(NC2CC(NC(c3ccc(O)nc3)=O)C23CCC3)c([N+](=O)[O-])c(C)n1 66553,C(=O)(CC(O)CC1CC1)NC(CNC(C=C(C)Cl)=O)(C)Cn1cccn1 66554,C12(C(N3CC(CNC(c4ccc(F)cc4)=O)C3)=O)CCCC1CCC2 66555,Cc1noc(C)c1CCNC(=O)C(Cc1cn[nH]c1)NC(=O)C(C)c1ccsc1 66556,CC1(C)CCC(C(=O)NCC2(O)CCN(C(c3cccc(F)c3)=O)C2)CO1 66557,c1(Cn2cc(C(CC)CO)nn2)cc([N+](=O)[O-])ccc1Br 66558,CC(C)(C)C(C(=O)N1CCC(CNC(=O)CC2CC2)CC1)NS(C)(=O)=O 66559,C1(NCCOC(C(C)(C)C)=O)CN(N2CCC(OC(F)(F)F)C2)C1 66560,c1(C2C(=O)NCCN2N2CCCC2)ccc2cccnc2c1F.C(CCF)SC 66561,Cc1nc2cccc(C(N3C(CNC(C4(O)COC4)=O)CC4COCC34)=O)c2[nH]1 66562,C1(C(=O)NC(Cc2cc[nH]n2)C(=O)NCC2C=CCOC2)CC2(CCC2)CO1 66563,N1(C(C2CCC(C)CC2)=O)CC2(C1)CN(C(C1(Cl)CC1(C)C)=O)C2 66564,N1(C(c2cnc(C)s2)=O)CC2CC(NC(C3CCCC(F)(F)C3)=O)CC1C2 66565,CC1(C)CC(C(=O)NC2(C(=O)NC3(CC4CCC4)CC3)CC2)=NO1 66566,N1(C(Cc2nn(C)c(=O)o2)=O)CCCC(C)(C(=O)NCC2(C3CC3)CCCO2)C1 66567,C(=O)(CC(C(C)(C)C)NC(=O)Cc1cnnn1C)NC(c1cccs1)CC 66568,C1(CC=C)(NC(C(=O)C=CC(=O)NC(C(C)N)C)=O)CCCC1.N1(C)CCOCC1 66569,C1(C(=O)NC(C)CCNC(=O)C(O)C2CCC2)C(c2ccncc2)C1(C)C 66570,c1(NC(C2CN(C(=O)Cc3ccnc(F)c3)C2)=O)ccc2scnc2c1 66571,c1(N(c2cc(Cl)cc(Cl)c2)C(C2CC(F)CN2[SH](=O)=O)=O)ncc(F)cc1Br 66572,C12(CNC(CSC)=O)CCCC(C1)OC2.C12CCN(CC1)C(=O)c1cn2nn1 66573,C1(NC(c2c(CC)scc2)=O)CCN(C(c2ccccn2)=O)C(C)C1 66574,c1(C(=O)NCCCC(C)(C)OC)cc(Cl)c(Br)cc1F 66575,c1(C(N2CCC(NC(CC3CCCCC(=O)N3)=O)C2)=O)ccc(F)c2ccsc12 66576,S(=O)(=O)(c1ccc(C2OCCO2)cc1)C(=O)NCC(C1CC1)NC(=O)OC(C)(C)C 66577,C12(C(=O)NC3(COC)CCCN(C(CCC)=O)C3)CCCC(=O)N1CCC2 66578,C(=O)(C(C(C)Cc1ccccc1)N(CCCOC)C)NCC 66579,CCCCCS(=O)(=O)CC(=O)N1CCCC(O)(Cn2cc(CO)nn2)CC1 66580,c1(CC)cc(F)ccc1C(=O)NC12CCN(C(C3(n4cncn4)CC3)=O)CC1C2 66581,C(=O)(CC(C)(C)CCOC)N(C1CN(C(C(CC)NC(C)(C)C)=O)C1)C 66582,C=C(C)C(C)(C)C(=O)N1CC(N(c2c[nH]nc2-c2cccnc2)C(C2CC2F)=O)C1 66583,CC1(C(=O)NCC(C2CC2)NC(c2ccc(F)cc2)=O)CC2CCC(C1)S2 66584,c1(NCCc2c(F)cncc2F)ccnc2c(Cl)cnn12 66585,CC(C)(CNC(c1cc([N+](=O)[O-])c[nH]1)=O)CC(=O)NCCCOCC1CCC1 66586,C1(CC(=O)NCC(C)N(C(C)=O)C)CC2(CCC2)CN1C(=O)C=Cc1cocn1 66587,c1(C(=O)NCC(CNC(Cc2c(C)cccc2Br)=O)O)cc(F)cc(C)c1O 66588,C12(NC(C(C)SC(C)C)=O)CCC(C1)N(C(=O)CCCC(=O)N(C)C)C2 66589,Cc1ccc2c(C(=O)NC(C3CN(C(=O)Cn4c(C)ccc4C)C3)C)coc2c1 66590,CC1CC(C(=O)N2CCC(CNC(c3ccn(C)c3)=O)C2)c2ccccc2N1 66591,c1(CCC(=O)NCCC2CCCN(C(C(CC)F)=O)C2)nc2cnccc2[nH]1 66592,c1(OC)ccc(CN2CCOC(CC(=O)Nc3nccnc3Br)C2)cc1[N+](=O)[O-] 66593,C1(NC(C2(C(=O)OCC)CC2)=O)CCN(C(c2ccc(OC)nc2)=O)C1C 66594,N1(C(c2ccc(CC)cc2)=O)CC(NC(c2nc(C)nn2C)=O)C(C)(C)C1 66595,c1(C(=O)NC2C(CNC(c3ccc4scnc4c3)=O)C2)cc2ccccc2o1 66596,c1(C(=O)NC2C(C=C)CN(C(C3CCCCNC3=O)=O)C2)ccc(N=[N+]=[N-])cc1 66597,c1(C(C(=O)NCCSC)N(CC(=O)OCC)CC(F)F)ccc(Br)c(F)c1 66598,Cn1ncc(Cl)c1C(=O)NC1C2CN(C(C3CC3Cc3ccccc3)=O)CC12 66599,C(C)(CC(C)(C)O)NC(C(C)N(C(=O)C(c1ccnn1C)C)CCC)=O 66600,N1(C(c2c(C(C)C)onc2)=O)CCCC(CN2CCN(C(=O)C(C)O)CC2)C1 66601,N1(C(CNC(C(CC)CC)=O)=O)CC2CCCCN2CC1CNC(=O)C(=O)NC 66602,C(C(O)CC(=O)N(C1CC1C)C)NC(c1c(C)ocn1)=O 66603,c1(C(=O)NCC2CCC(NC(C(C(C)C)SC)=O)C2)ccc(C2CC2)nc1C 66604,CC(C)C(C(=O)N(CCCCN(C(=O)C(C)C)C)C)ONC(=O)OC(C)(C)C 66605,C(CC(C)C(=O)NCCCC1CCCN1C(=O)C(=O)NCC(F)F)=CC 66606,N1(C(C2C=CCS2)=O)CCC2CN(C(=O)CCSC3CCCC3)C2C1 66607,C1(CNC(c2nnc(C)s2)=O)CCCC2CN(C(=O)C(C)OCC(C)C)CC12 66608,Cn1cc(CC(=O)NCC2CC(NC(c3c[nH]nc3Br)=O)C2)cn1 66609,c1(OC)ccccc1CN(CCCO)C(C1CCC(n2cc(C3(O)COC3)nn2)C1)=O 66610,C1(C)(C(N(CC(COC)O)C)=O)CCCN(C(c2cnc(C)n2C)=O)C1 66611,c1(OC)cc(C(=O)NC2(C)CN(C(c3ccc(F)cc3C)=O)C2)cc([N+](=O)[O-])c1 66612,Cc1cccc(O)c1C(N1CCCC(CN(S(=O)(=O)CCCl)C)C1)=O 66613,CC1CN(C(=O)CC#N)CC(C)N(C(c2ccnc3c2ccn3C)=O)C1 66614,C1(C(=O)NC2C(OC)CC2)CCOCC1NC(C1CC2(CSC2)C1)=O 66615,c1(C(N2C(C(=O)NCCCOC)C3C(C2)C3(C)C)=O)cccc([N+](=O)[O-])c1C 66616,CC1CN(C(C2CCCN2C(C23CCCN2CCC3)=O)=O)CCCO1 66617,N1(C(C(C)(C2CCC2)NC(C(C)N2CCCC2)=O)=O)CCCC(F)(CO)C1 66618,C(=O)(C1=CCCCC1C)N1CC(NC(c2c(C)nc(-c3cccs3)o2)=O)C1 66619,c1(CNS(C)(=O)=O)ccccc1NC(C(=O)OCCC1CCOC1)=O 66620,N1(C(c2c(C)nc(COC)s2)=O)CC2(CCCC2NC(C2CCCN2C=O)=O)C1 66621,Cc1cc(CC(=O)NC23CC2CN(C(=O)Cc2ncc(C)s2)C3)cc(C)c1 66622,C(=O)(CC(C(C)C)NC(=O)Cn1c(C)ccc1C)NC(C(=O)OCC)C1CC1 66623,C1(NC(C2CCN(C(C)=O)CC2)=O)CC2C1CCN2C(=O)CNc1ccccn1 66624,Cc1nc(C(=O)NC2CCC(NC(=O)C(C)C3CCC3)C2)sc1C 66625,CCCC(CC)C(=O)N1CCC(CN(C2CCCN(CC3CC3)C2=O)C)CC1 66626,Cc1cc(=NCCNC(C2CC(C)OC(C)C2)=O)[nH]c(-c2ccc(CO)cc2)n1 66627,c1(C(=O)NC(CSCC#C)C)c(OC)nsc1OC(C)(C)C 66628,CC(C)CC(O)CC(=O)NC1(Cc2ncc(F)cn2)CC1 66629,C12(OC)CCC1CN(C(C1CCN(C(=O)CCC(=O)C3CC3)C1(C)C)=O)C2 66630,Cc1c(C(=O)NC(C)CN(C(=O)C(C)C)C)c(=O)n(-c2ccccc2)n1C 66631,N1(C(C2(C(=O)NCC(CNC(C)=O)OC)CCC2)=O)CC(SC)C(C2CC2)C1 66632,c1(CC(=O)N(C2CCN(C(=O)Cc3cnco3)C2)CC)nocc1C 66633,c1(C(=O)NCCC2CCN(C(CCSC)=O)C2)cc(Br)cc(C)c1F 66634,O=C(CC(O)C(Cl)(Cl)Cl)NC(C1CCN(C(=O)CC2C=CCC2)CC1)CO 66635,N1(C(CCCC#C)=O)CCC(C2CCCN(C(=O)CCC(=O)C(C)(C)C)C2)CC1 66636,N1(C(CC2CCC(=O)NC2)=O)CCN(C(c2cccc(Cl)c2F)=O)CC(CO)C1 66637,Cc1cccn(CC(=O)NCCCCc2ccccc2Br)c1=O 66638,CN(C)S(=O)(=O)N1CC(NC(=O)C(=O)N(C)C)C1.C12CC3CCC1C3C(=O)O2 66639,O=C(C#Cc1ccccc1)N1CC2C(C1)N2C(C1(c2ccccc2)CC1)=O 66640,c1(NC(C2CC23CN(C(c2c(F)ccc(Cl)c2Cl)=O)C3)=O)nccc2[nH]ccc12 66641,CCCCCC(O)C(=O)N(C)CC1(CC(=O)NC2CN(C(=O)CC)CCO2)CC1 66642,C1(C(N(C)C)=O)CCC(C)(C(=O)NCCNC(=O)CSCCC#N)C1(C)C 66643,C1(NC(N(C2CCN(C(C3(C)COC3)=O)C2)CC2CC2)=O)CCC(=O)N1 66644,C1(C(C)NC(C(C)CF)=O)CCN(C(C2(F)CC2(Cl)Cl)=O)CC1 66645,S(=O)(=O)(c1cccnc1)N1C(CC)CN(C(=O)NCCNc2ccccc2)CC1 66646,N1(C(C(CC)C)C(=O)NCCCOC)CCC2(O)CCOCC2(C)CC1 66647,c1(NCC2(CCCC)CCC2)cc(NCC2(CC3CCC3)CC2)ncn1 66648,CC(CC(N)=O)(c1ccsc1)NC(c1ocnc1C1CC1)=O 66649,c1(-n2c(C3(NC(C)C=C(Cl)Cl)CCCOCC3)nnn2)ccc2c(c1)OCCO2 66650,N1(C(CCCCOCC)=O)C2CCC1CN(C(c1cc(C)n(C(F)F)n1)=O)CC2 66651,N1(C(c2ccc(SC)s2)=O)CC2CCN(C(=O)C(c3cccc(F)c3)O)CC2C1 66652,N1(C(CCc2nnc(C)o2)=O)CCc2cc(Br)c(F)cc2C1 66653,C1(CNC(c2nncc(OC)c2)=O)CC2(CO1)CN(C(=O)CCc1cnc[nH]1)C2 66654,N1(C(COCC(C)(C)C)=O)CCCN(C(c2cnc(Cl)c(N)c2)=O)C(C)C1 66655,Cc1nc(C=CC(=O)NC2CC(NC(c3occc3-c3cnn(C)c3)=O)C2)cs1 66656,CN1CCCCC1CC(N1CCC1CNC(C1CC(C(F)F)C1)=O)=O 66657,c1(OCC)ccc(C(=O)NC(C2(CNC(c3cc(C#N)c[nH]3)=O)CC2)C)nc1 66658,C1(CNC(CC(=O)NCC#C)=O)CCCCN(c2nnc(C(=O)OC)s2)C1 66659,C1(C(=O)NCCNC(C2(OCC)CC2)=O)CC12CCOCC2 66660,C(=O)(C1=NOC2COCC12)NC(C(=O)N(CCOCC#C)C)Cc1cn[nH]c1 66661,c1(OCC(C2CN(C(=O)C(n3cnc(C#N)n3)C)C2)N)ccc(C(CF)N)cc1 66662,C1(NC(C2C(OC)CCCC2)=O)CCC2(CC1)CN(C(=O)CS(=O)(=O)C1CC1)C2 66663,Cc1cc2occ(C(=O)NC(c3ccccn3)C(F)F)c2cc1C 66664,Cc1cc(C(=O)NCC2CN(C(C3CC3C(F)(F)F)=O)CC2(C)C)c(Cl)cn1 66665,n1(CCCC)cc(C(N2CCC(CNC(C3CC(n4cnnc4)C3)=O)C2)=O)nn1 66666,N1(C(c2c(CC)occ2)=O)CCC(C)(C(=O)N(CCC(N)=O)C)C1 66667,C(=O)(NNC(=O)c1cncc(N(C)C)n1)Nc1nc(C(C)(C)C)sc1 66668,c1(COC(C2CS(=O)(=O)CC(=O)N2)=O)ccc2ncccc2n1 66669,C(CC(=O)NCCCC(C)(F)F)(C(F)F)NC(CC(C)c1ccco1)=O 66670,C1(C)(C(C)N(C(C(=O)NCCC(C)(C)C)C2CCOC2)C2CC2)CC(=O)C1 66671,C1(CNC(C(c2ccccn2)=O)=O)CCCN(C(=O)Cc2cc(C3CC3)on2)C1 66672,Cc1nccc(C(=O)NCCCNC(=O)CCCNc2ccc(F)c(Cl)c2)c1C 66673,C(=O)(C1=CC2CCCCCC12)NCC1C2CN(C(CC(CCC)C)=O)CC21 66674,CC(CC(F)F)C(=O)N(CC(O)CNC(c1ccnc(CO)c1)=O)C 66675,N1(C(c2c(C)nc3ccccc3n2)=O)CCC2CC(C)CCC12 66676,N1(CC(=O)NCC2(O)CN(C(C3CCC(=O)O3)=O)C2)CCCCCC1 66677,N1(C(CC(C)SC)=O)CCC2(CC1)CC(NC(c1sc(F)cc1Cl)=O)CO2 66678,C1(O)(C(C)NC(=O)Cc2cnoc2)CCN(C(=O)CCCN2C(=O)CCC2=O)C1 66679,CC1CCN(C(c2ccccc2)Cc2cc(CC(F)(F)F)co2)C1CO 66680,n1(C(C)C)ncc(C(=O)NCC2CN(C(=O)C(C)(C)c3ncco3)C2)c1F 66681,N1(C(C=C(CC)CC)=O)CC(C(N2CCCC2(C)C2CC2)=O)C(F)(F)C1 66682,n1(CCOC)nnnc1C(c1c[nH]nc1C)NCC(C1CCC1)OCCO 66683,CC(C)C(O)CNC(=O)C(c1cccs1)NC(c1ncc[nH]1)=O 66684,C1(C(=O)NCC(CCO)OC)(C(C)C)CCCN1C(C1CC(N=[N+]=[N-])C1)=O 66685,Cc1cnc2c(C(=O)NCC(CO)NC(=O)C(c3ccc(C)o3)C)c(C)nn2c1 66686,N1(C(CCc2cc(OC)c(O)cc2)=O)CCCC12CCN(C(C1SCCS1)=O)C2 66687,c1(C(=O)NCC2(OC)CN(C(=O)CCNC(=O)CO)C2)cnccc1C 66688,c1(N2CC(CN(C(C(c3c(OC)cccc3)C)=O)C)C2)ncnc2c1CCC2 66689,C1(C(N(CC(C)(C)C)C)=O)CCCN(C(=O)Cc2cnn(C)c2)CC1 66690,CC(CC(F)F)C(=O)N1CC(NC(C2CCC2c2ccc(F)c(F)c2)=O)C1 66691,c1(CN(C2(C)CCN2CCOc2cccc(Br)c2)CC)ccc2cccc(Cl)c2n1 66692,c1(N(C(C2CC2NCCN2CCN(C)CC2)=O)CC)c(F)cc(C(F)F)cc1F 66693,CCCCCC(c1nnnn1CCOCC(N)=O)NC.c1(CSC)cccc(OC)c1 66694,CN1CC2CN(c3ccnc(NCCOC4CCOC4)n3)CCN2C1=O 66695,N1(C(Cc2cc(CC)no2)=O)CCC2(CC1)CN(c1ccc(C#N)nc1)CCO2 66696,c1(NC(C2C(C(=O)OC)C2)=O)ccc(C(=O)Nc2cc(Cl)ncc2F)cc1C 66697,Cc1ccc(CN2CC(F)CC2C(=O)Nc2ccnc(-c3cccnc3)c2)cc1 66698,Cc1cnc(C(=O)NC2CCCCC2NC(=O)CCF)c(Br)c1 66699,C1(C)(C(=O)NCCCNC(C2(NC(C)C)CC2)=O)CCOC1 66700,n1(CC)ccc(C(=O)N(CCNC(C2(CC3CC3)CC2)=O)CCOC)n1 66701,C1(NC(C(C)(CO)NC(c2c(C)nc(C)s2)=O)=O)CCOCC12CCC2 66702,c1(CNC(C)=O)ccc(OCC(N)=O)c(Cl)c1.C1(COCC#N)C(=O)N1 66703,C1(NC(C(C)CC2CCCC2)=O)CC(NC(c2cccn2C2CC2)=O)CC1O 66704,N1(C(C2CCCN(C)C2)=O)CCC2(CC(NC(=O)CC3(C)CCC3)C2)C1 66705,C1(CCCC)CN(C(C)(C)C)CCN1C(c1ccnn1C)C(=O)OC(C1(C)CC1)=O 66706,c1(C(=O)NC(CCCNC(Cc2c(C)cco2)=O)C)sc(N2CCCC2)nc1Cl 66707,CCCCCCC(C)(C)C(=O)NCC(=O)C(C)(C)[N+](=O)[O-] 66708,N1(C(=O)Cn2cccn2)C(CNC(C2(CF)CC2(F)F)=O)CC2COCC12 66709,C1(C(N2CC(CC)N(C(=O)Cc3c[nH]nc3O)CC2)=O)CC12CCC1(CC1)CC2 66710,c1(OC)c(CNCC2CCCN2C(=O)CCC(N)=O)cc(F)cc1F 66711,CC1CC=C(C(=O)NC2C3CN(C(C4C(C5CC5)C4(F)F)=O)CC23)CC1 66712,C(=O)(C(C(C)(C)C)OC)N(CC(C)NC(C12CC(c3ccccc3)(C1)C2)=O)CC 66713,N1(C(CN2CC(=O)NCCC2)=O)CC2CC(F)(F)CC2C1 66714,C#Cc1cccc(C(=O)NC(COC)C(=O)NOCC2CCOCC2)c1 66715,c1(C(=O)NC23C(CN(C(C4(C(F)(F)F)CC(=C)C4)=O)C2)C3)cnc([N+](=O)[O-])n1C 66716,C1(C(=O)NCC(c2ccc(OCCC#N)cc2)N(C)C)CC2C(C1)C2(F)F 66717,Cc1cc(C)n(CC(N2CCN(C(=O)CC(C)c3ccncc3)C(C)C2)=O)c(=O)n1 66718,Cc1nc(C#N)ccc1C(=O)N(CC(O)CN(C)C(c1ccnn1C1CC1)=O)C 66719,c1(C(=O)NCC(COC)NC(=O)C(O)c2ccsc2)conc1C1CCCC1 66720,N1(C(C(c2cccc(Cl)c2)C)=O)CCC2C(C1)CN2C(C1CCCN1C)=O 66721,C1(NC(c2ccc(Br)o2)=O)CCC(CNC(c2cccn2C(F)F)=O)C1 66722,C1(O)(CCNC(CCOCC)=O)CN(C(c2ccc(C(F)F)o2)=O)C1 66723,C1(CC(=O)NCC(C)N(C)C(c2cc(C(N)=O)c[nH]2)=O)COc2ccccc2O1 66724,C1(C(N2C(CCCNC(CC=C=C)=O)CCC2)=O)CC12CCSCC2 66725,C1(NC(c2cc(C)c(-c3ccccc3)s2)=O)C2CC1N(C(C1CCOC1)=O)C2C 66726,c1(OC)c(C(=O)NCCCCNC(c2cnn(C(C)C)c2C2CC2)=O)csc1C 66727,C(=O)(C#CC1CCOCC1)N1C(n2cc(-c3ccc(C#N)cc3)nn2)C(O)CC1 66728,Cc1csc(C(N2CCOC(C(C)NC(=O)CN(CC(C)(C)C)C)C2)=O)c1Cl 66729,c1(C(N2CCC(C)(C)C2CNC(c2csc(S)n2)=O)=O)cc2ccc(Cl)cc2[nH]1 66730,CCCCCC(C(=O)NC1CCC(F)(F)CC1)N(CCC(C)(C)c1ccccc1)C 66731,N1(C(c2nc(C)oc2C)=O)CC2CC(NC(c3cc(Cl)cc(Cl)c3)=O)C(C2)C1 66732,C1(C)(C(N(CCC(C(C)C)N(C)C)C)=O)CCN(C(=O)C(CO)N(C)C)CC1 66733,CCC(C#N)C(=O)N1CC(COC)(NC(=O)CCOCC(C)(C)C)C1 66734,CCCC(CC)C(=O)N(CCN(C(C1CC2CCC(C1)S2)=O)CC)CC 66735,O=C1CN(CCC(N2CC(O)CC3(CCCC3)C2)=O)c2ccccc2N1 66736,c1(C(=O)NC2C(C)CN(C(=O)CC3CCN(C)C3=O)C2)ccc2c(c1)C(C)CN2 66737,N1(C(C2CC(=C)C2)C(=O)NC(=O)Nc2ccccc2)CCOCC1c1nccn1C 66738,N1(C(C=CCCC=C(C)C)=O)CCC12CN(C(c1cc(C)c(Cl)cn1)=O)C2 66739,C1(CC)CC(C(=O)N(CC(C)CNC(c2nn(C)c(C)c2Cl)=O)C)CCC1=O 66740,C(=O)(CCCCCc1cccs1)NCC1CN(C(c2nc(CC)oc2)=O)CC1C 66741,c1(C(N2CCC(n3ccnn3)C2)C(=O)NCC2CCC2)ccc(C(F)(F)F)o1 66742,N1(C(C23C(C)(C)OCC2C3)=O)CC(C2CCN(C(=O)C3=NNC(=O)CC3)CC2)C1 66743,C1(NC(c2ccc(C(C)=O)cn2)=O)CCCCN(c2ncc(C(C)(C)O)cn2)C1 66744,Cc1cnc(CCC(=O)N(CCCN(C(=O)CCc2ncc[nH]2)C)C)[nH]1 66745,CCC(CC(=O)NC1CC2CC1N(C(c1c(F)cccc1F)=O)C2)C(F)F 66746,C1(COC)=NC2=CC(=NC3CCC(CC3)N2)N1.c1(COC)cncn1C1CC1 66747,c1(C(=O)NCC(=C)CCNC(C2(CC)CCNC2=O)=O)cc([N+](=O)[O-])ccc1Cl 66748,c1(C(N(C(C)CNC(c2onc(C)c2C)=O)CC)=O)cc(CO)ccn1 66749,C1(CNC(C(COCC)C)=O)CN(C(=O)CCCF)CCC1(C)C 66750,C(=O)(C1=CCCC1C)NCCCC(=O)NC(C(=O)NCCC)CC 66751,c1(NC(=O)CC2C(NC(C3CCCC(O)CC3)=O)CC2O)n[nH]c2c1COC2 66752,c1(C(N2C(CNC(c3cc(OC)ncc3)=O)CC2)=O)cc(S(N)(=O)=O)cs1 66753,N1(C(C2C(C)OC(C)C2)=O)CCC2(CNC(=O)CC3CSC3)CCCC12 66754,N1(C(CNC(=O)NC)=O)CCC(C(=O)NCC2CN(C3COC3)C2)C1 66755,N1(C(C2N(C(Cc3c(C)scc3)=O)CC=CC2)=O)CCC2CCCC2C1 66756,c1(NC(N(C)C)=O)ccc(-c2ccccc2F)n1C 66757,N1(C(c2c(CC)ncs2)=O)CC2CC(NC(c3cn4c(n3)COCC4)=O)C(C2)C1 66758,C1(C(=O)NCCC(=O)NC(CSC)(C)C)CCS(=O)CC1 66759,N1(C(CCC=CC)=O)CC2CN(C(=O)CCCC(=O)N(C)C)CC(F)(F)C2C1 66760,C(C(N=c1[nH]c(=NCC(C(C)C)OC)[nH]c2ncn(C)c12)c1ccco1)OC 66761,N1(C(C2C(OC)CN(C(C3(CO)CCCCC3)=O)C2)=O)Cc2cnn(C)c2C1 66762,C1(C(C(=O)NCC2(C=C)CCC2)(C)C)CCCN(C(=O)C(CCOC)OC)C1 66763,N1(C(c2c(CCC)n(C)nn2)=O)CC2CC1CN2C(C1CC1(F)F)=O 66764,C12(NC(c3cc(OC)no3)=O)CC1CN(C(c1[nH]nc(OC)c1Cl)=O)C2 66765,C1(N(C(=O)CNc2ccccc2Cl)C)CCCCN(C(C2CC3(CC3)CO2)=O)C1 66766,c1(C(=O)NC(C(C(=O)NCCOCCC)C)C)cccc(F)c1C 66767,NC(=O)CCC(C(=O)NCc1cncnc1)n1cc(-c2ccnn2CC(F)F)nn1 66768,N1(C(C(CCOC)OC)=O)CC2(CCN(C(C3CCOC(C)(C)C3)=O)C2)C1 66769,C1(CC(=O)N(C2CCCC(NC(C3(CC#C)CCC3)=O)C2)C)CN2CCN1CC2 66770,N1(C(C(=O)C(c2cc(-c3ccccc3)co2)C)=O)CCC(CCO)(C(=O)O)C1.N 66771,N=c1[nH]c2ccccc2cc1C(N1CC(F)C1)=O 66772,C1(NC(c2ccc(C)nn2)=O)CC1C1CCCN(C(C2CC=CCO2)=O)C1 66773,CC1(CNC(c2ncoc2CNC(c2ccc(N)c(F)n2)=O)=O)CCCCC1O 66774,N1(C(C23CC(OC)C2C3)=O)CC2CC3CC2C1C3NC(c1cnc(S)nc1)=O 66775,c1(CC(=O)Nc2nc(-c3ccccc3C(F)(F)F)cs2)ccncc1Cl 66776,C(C(F)(F)C(F)F)NCCC(=O)NCC(c1ccccc1F)(C)C 66777,C12(NC(=O)CO)CCCC1N(C(=O)Cc1cnns1)CC2 66778,N1(C(C2(F)CCC(C)CC2)=O)CCOC2(C1)CN(C(C1(C)CCOCC1)=O)C2 66779,C(=O)(C1=NNC(=O)C1)N(CC1CC(C(=O)NC(=O)C(CO)N(C)C)C1)C1CC1 66780,N12CCCC(C)(C)C1CNC(=O)CN(C)CC2=O.c1(C=O)ccccc1.CN 66781,C1(CC)CC(C(=O)NCC(C)CNC(C2C=CCC2)=O)CC(=O)N1 66782,N1(C(c2cc(CC)c(O)cc2)=O)CC2CCN(C(c3snnc3CC)=O)C2C1 66783,c1(C(C)C)cccc(NC(C2CN(C(c3coc(C4CC4)n3)=O)CC2C)=O)c1 66784,c1(C(=O)OC)cc(C(=O)NC2CCCCC2NC(=O)CCS(C)=O)n(C)n1 66785,N1(C(c2ccc(C(=O)NCC)n2C)C(=O)NCCC)CCCC(C2(C)CC2)C1 66786,C(C)(C(=O)N1CC(NC(=O)C(C)Oc2cccc(C)c2)CC(C)C1)(C(C)C)OC 66787,N1(C(c2c(C)noc2)=O)CCN(C(=O)CNC(=O)Cc2ccccc2)C2CC12 66788,C(=O)(C(CC1(C)CC1)NC(C1CCCS1)=O)NC1(CC)CCCN1 66789,CCC(C)CC(C)C(=O)N1CC(NC(=O)CCNc2ccccc2Cl)C1 66790,C1(C(=O)Nc2ccc(C)cc2F)CN(C(=O)CCc2ccncc2)CC12CCC2 66791,c1(C(C)NCC2(F)CC3CCC(C2)N3)cc(F)c(F)c(F)c1F 66792,N1(C(c2cccc(C)c2)=O)CCCCC(NC(c2nnsc2C(F)F)=O)C1 66793,C12COCCN1C2.C(=O)(CN(C(=O)C=CC=CC)CCC)NCCC 66794,NS(=O)(=O)CCC(=O)NCC1CCN(C(C2(F)CCCOC2)=O)C1 66795,C(CC(=O)NOC1CCCC1)(C(C)(C)C)NC(C1CC(CC)C1)=O 66796,C(=O)(C#CC1CC(F)(F)C1)N1CC2C(CNC(C3OCCN(C)C3)=O)(C2)C1 66797,c1(CNC(C(C)NC(CC)=O)=O)n[nH]c2c1CN(C(C1CN(C)C(=O)N1)=O)CC2 66798,C1(C(=O)NCCCCCNC(C2C(C3C(C)C3)C2)=O)CCc2ccnn2C1 66799,CC1(C)CCCC(CC(=O)NC2(C)CCN(C(C3(O)CC3)=O)CC2)O1 66800,C1(C#N)(C(=O)NC2(C)CN(C(Cc3ccc(NC(C)=O)cc3)=O)C2)CCCOC1 66801,C1(NC(CCN(C(C(C=C)O)=O)C(C)C)=O)CCNC(=O)CC1 66802,N1(C(CC(CC)C)=O)CCN(C(C23CCC(CO)(CC2)C3)=O)CC1CF 66803,c1(NC(C(CCNC(=O)CCCn2cncn2)O)=O)ccc(O)c(F)c1 66804,Nc1cc(Cl)cc(F)c1C(=O)NCCCN(C(=O)CCCC1CCC1)CCO 66805,c1(C(=O)NCCN(C(C)C)C(C2CCCN2N=O)=O)cc(Cl)cc(F)c1Br 66806,S(=O)(=O)(c1cncn1C)N(C)Cc1ncco1 66807,C1(NC(C2C3CNC(=O)C32)=O)CCCCCN(C(C2(C(F)(F)F)CC2)=O)C1 66808,C1(NC(CC(=O)NCC#C)=O)CS(=O)(=O)CC1NC(c1nccc(N)c1Cl)=O 66809,c1(C(=O)NCC2C(NC(CCCN(C(C)=O)C)=O)C2)c(Cl)nsc1Cl 66810,C(=O)(CCCCCC(C)C)N1CC2C(NC(c3ccc(OC)c(N)c3)=O)(C2)C1 66811,c1(N2CCC(C(C)NC(C3N(C(C)=O)CCC3)=O)CC2)ncn(C)c(=O)c1Br 66812,c1(CNC(C=C(CC)C)=O)cc(CCNC(=O)C(O)C2(C)N=N2)no1 66813,C=C(CC)CN=C(NCC1CC1)N(C)Cc1ccccn1 66814,C1(NC(C2(C)CCC(=O)N2)=O)CCC(O)CN(C(=O)Cn2ccc([N+](=O)[O-])n2)C1 66815,C(C(CC(=O)N(c1cnn(C)c1)C)NC(c1csnc1C)=O)OC 66816,O=C(CN=c1[nH]c(=NCc2csc(O)n2)[nH]c2c1CSC2)N1CCCC1 66817,c1(C(N2CCC(C(C)NC(C(CC(C)C)(C)C)=O)C2)=O)csc2ccc(F)cc12 66818,C(=O)(C#CC(C)(C)C(F)F)N(C)CCNC(C1CCCN1c1nccs1)=O 66819,C1(CNC(=O)CCF)CN(C(=O)Cc2sccc2Cl)CCO1 66820,Cc1ncc(Cl)c(NC(CCCCN)C)n1.c1(NCC(=O)N)ncccn1.C1C(=O)N1 66821,N1(C(N2CC(C(=O)Nc3cccnc3Br)OCC2)=O)CCC(C(=O)N(C)C)CC1 66822,C1(CC)CCN(C(=O)Cc2ccsc2C)C(CNC(=O)CC2CCC2)C1 66823,C1(C(C)(C)OCC)CCN(Cc2nccc(N(C)C)n2)CC1.C12CC1C(=O)N2 66824,C(=O)(C(CCCCCCC1CC1)N1CC(CO)CC1CS(C)(=O)=O)NCC 66825,C=CCC(C)(O)C(=O)NCc1cccc(CNC(=O)CN2C(=O)CCC2=O)c1 66826,N1(C(C(C)c2ccco2)=O)CCCC(NC(c2ncc(Cl)nc2Cl)=O)C1C 66827,Cc1ncnc(C)c1CC(N1CCCC(NC(=O)CCC2CCCN(C)C2)C1)=O 66828,c1(NC(C2OCCN(C(C3CCC(C)O3)=O)C2)=O)cc(F)cnc1Br 66829,N1(C(COC(CC)(C)C)=O)CCCC2(C1)CN(C(=O)CN1CC=CC1)C2 66830,c1(C(C)C)noc(CCC(=O)NC2CC(N(C)C(=O)OC(C)(C)C)C2)n1 66831,c1(C(=O)NCC)ccc(C(N2CCSC(C)C2)C(=O)NCCC)cc1.OCC 66832,Cc1cccc(Cl)c1C(N1CC2C(CNC(=O)C(C)OC3CCCC3)C2C1)=O 66833,C12CNC(=O)CN1C(=O)C(C1CCOC1)NC2=O.C1(CC)CCCC1.CC 66834,CCC(CC(=O)NCC1(C(C)(C)C)CCN(C(=O)Cn2cnnc2)C1)C1CCC1 66835,C1(NC(CN(CC(C)(C)C)C)=O)CCCC(CNC(c2cnco2)=O)C1 66836,c1(C(N2CC(C)C(NC(C3CCCC(CF)C3)=O)C2)=O)nn(C)c(Cl)c1Cl 66837,N#Cc1ccc(CCCCC(=O)N2CCCC2C2CCN(C(=O)CCF)C2)cc1 66838,C(C(=O)NCCC1CCN(C(=O)C(C)N(C)C)C1)(C(C)C)NC(C)=O 66839,CCC(CCOC)C(=O)NC(C)CCCC(=O)N1CC(F)(C2CC2)C1 66840,N1(C(CCNC(=O)OC)=O)CCN(C(=O)CCCc2ccc(C)cc2)C2CC12 66841,c1(OCCC(=O)N(C2CCN(C(C34COCC3C4)=O)CC2)CC)ccccc1O 66842,C#Cc1ccc(C(=O)NCC2CC2CNC(C2CC(C)(F)C2)=O)c(F)c1 66843,C(c1ccc(=N)[nH]c1C)=CC(N1CC(COC)(NC(=O)CC(C)C)C1)=O 66844,CC1(C(=O)NCc2cc(C(=O)NCc3ccccn3)on2)CCOC1 66845,C1(C(=O)NC(CNC(c2scnc2C(F)F)=O)C2CC2)CCCNS1(=O)=O 66846,N1(C(CC(C=C)(C)O)=O)CC2CC(NC(c3cncc(C)c3Cl)=O)C(C2)C1 66847,N1(C(CSCC(C)C)=O)CC2CCCC1(CNC(c1coc3c1COC3)=O)C2 66848,C(=O)(C#CC1(C)CCCO1)NCC1C(NC(CN(CCC)C)=O)CCC1 66849,C1(NC(Cc2c(C)cc(C)s2)=O)CCN(C(c2cnc(C(C)C)s2)=O)C12CC2 66850,C1(CNC(C(CCCOC)C)=O)CC2(CCN(C(c3nc(=O)n(C)[nH]3)=O)C2)CO1 66851,c1(C(=O)NC2CCCN(Cc3c(C)nccc3)CC2)c[nH]c2ncccc12 66852,Cc1ncc(C(=O)NCCCCOCCNC(=O)NCCC2CC2F)cn1 66853,c1(CN2CC(C#N)C(NC(c3cc(Br)c[nH]3)=O)C2)cc2cc(F)ccc2s1 66854,C1(OC)CN(C(c2cc(Br)n3c2CCC3)=O)CC2(CC2)C1 66855,c1(C(=O)NCC23CCCC2N(C(C2CC2(Cl)Cl)=O)CC3)cnn2c1C(=O)NCC2 66856,N1(C(c2cc(OC)c(F)cc2)=O)CC2CCC1CC2NC(=O)CC(C)(C)C#N 66857,O(N1CCC(NC(=O)CC2CCC(NC(=O)C(C)N=[N+]=[N-])C2)CC1)CC 66858,CC1CCC(NC(c2ccn(CC(F)F)n2)=O)CN1C(=O)CC1COC2CC1C2 66859,c1(CCC(=O)N(C2CN(C(C3(C45CC(C4)C5)CCCC3)=O)C2)C)ccc(F)cc1 66860,N1(C(c2cc(C(C)=O)[nH]n2)=O)CCOC2CN(Cc3c(C)cc(Br)cc3C)CC12 66861,CC1(C)C(=O)NC2CCC(C(=O)Nc3ccc(SCc4cnc[nH]4)cc3)CC12 66862,C12CCN(C13CC3)C2=O.C(CC(C)SC)NC(C1(C(=O)OCC)CC1)=O 66863,c1(CS(C)(=O)=O)ccc(CO)cc1.CC(O)CC(=O)N1CCC(CN(C(=O)C)C)C1 66864,C1(OC)(OC)CC(C)(C(N2CCC(NC(c3n[nH]c(C)c3Cl)=O)C2)=O)C1 66865,CC(C)(CC(=O)NCC1CC12CCC2)NC(C1CCC=CCC1)=O 66866,c1(C(CCN(C(CC2CC(OC)C2)=O)C)NC(=O)C(N)=O)ccc(C)cc1 66867,N1(C(c2nn(C)c(=O)cc2)=O)CC2(CCC2)CC1CNC(=O)C(F)C1CCOC1 66868,S(=O)(=O)(c1ccc(C#N)cc1)NC(c1c(CC)nn(C)c1)=O 66869,C1(CNC(C(=C(C)C2CC2)F)=O)CN(C(=O)C(C)CF)CCC12CCC2 66870,C1(NC(CCC(C)OC)=O)CN(C(=O)CC(n2nc(C)cc2C)C)CC2CC12 66871,C1(NC(CCc2c(C)n(C)nc2)=O)CCCN(C(=O)CCc2ccco2)C1C 66872,c1(NCc2cn(C3CCN(C(C)=O)C3)nn2)cc(N)cc(S(C)(=O)=O)c1 66873,N12CCCC(C1)NC2=O.c1(NC(N)=O)nnc(C(C(C)C)SCCCC)o1 66874,N1(C(c2c(CC)csc2)=O)CC(NC(c2cnc(C)s2)=O)C2CC12 66875,c1(NC(C2(C)CC(NC(c3cc(C)nc(O)c3)=O)C2)=O)cncc([N+](=O)[O-])c1 66876,CN1C(=O)CN(C(C2C3CN(C(C4CC(C)(C)CN4C)=O)CC23)=O)CC1=O 66877,c1(C(N(CCNC(=O)C=CC2(C)CCOCC2)CC)=O)ccc2ncncc2c1 66878,C(=O)(CC(C)C(=O)OC)NCCN(C(=O)Cc1cc(F)ccc1F)CCOC 66879,C1(O)(CCNC(C2(CCCC)CCC2)=O)CN(C(=O)C(C)OCC2CCCO2)C1 66880,C(=O)(C(C(C)(C)SC)C1CCCCO1)NC1C(CC)CN(C(=O)OC(C)(C)C)C1 66881,c1(CC)[nH]c(=N)sc1C(=O)NCC(O)CN(C)C(c1ccno1)=O 66882,c12ccc(cc1)S(=O)(=O)N(C)C1CCCN(C1)C(=O)C2C.C1(NC=O)CCC1 66883,N1(C(Cc2ccc(C)s2)=O)CC(C(N2CCC(C(F)F)CC2)=O)CC(C)C1 66884,c1(C(=O)NC(C2CCN(C(C(C(C)C)OCC)=O)C2)(C)C)ccc(C)c(O)c1 66885,Cc1c(Br)ccc(NC(=O)COCC(=O)NC(C)C)c1I 66886,Cc1cc2cc(C(=O)NCCCC(C)NC(=O)C(C)OCCC=C(Cl)Cl)ccc2cn1 66887,C1(C(=O)NC2CCC(C(=O)N(CC(O)C3CCC3)C)C2)(OC)CCOC1 66888,C(=O)(CC(CC1CC1)NC(=O)C(F)OC(F)(F)F)N1C(CCC)CCC1 66889,N1(C(C(C)OCCC=C)=O)CC2(C1)C(NC(c1cc(C)on1)=O)CCS2(=O)=O 66890,C1(C)(OC)CCN(C(C2SCCS2)=O)CC1.C12(C(=O)OCC)C(NC=O)C3CC1C2C3 66891,Cc1nc(CNC(=O)COC(C)(C)C)sc1C(=O)NOCC1CCOC1 66892,N1(C(C2Cc3c[nH]nc3C2)=O)CCCCC2(C1)CN(C(=O)CCn1cnnn1)C2 66893,C1(C(C(=O)N(CC=C)CCOC)NC(c2cnco2)=O)CC=CCC1 66894,c1(CC(=O)NCC#CCNC(c2c[nH]nc2[N+](=O)[O-])=O)ccc2ccccc2c1 66895,N1(C(C(C)OCOC)=O)CC(NC(=O)C=CCCC(C)C)CCC1C 66896,c1(-n2ccc(C(N(C(CO)C(=O)O)C(CC)(C)C)=O)n2)ccccc1C 66897,Cc1nc2cccc(C(=O)NC3COCC3CNC(C34CCC3CC4)=O)c2[nH]1 66898,c1(C2C(NC(C3(F)CCN(C(c4cnc(Cl)nc4)=O)C3)=O)C2)ccc(F)cc1 66899,c1(C(N2CCCC(CN(c3nc(SC)nc(O)c3)C)C2)=O)ccc2c(c1)CCO2 66900,C1(F)(CNC(C2C(OC)(OC)CC2)=O)CCN(C(c2c(C)coc2C)=O)C1 66901,C1(CC(=O)N(C)CC2N(C(C(F)=CCC)=O)CCC2)COC2CC1C2 66902,c1(OC(C(C)N(C(C)C)CC2CCN(C)C2)=O)ccccc1Cl 66903,N1(C(C=NOC)=O)CCC2(CC1)CC(NC(=O)C(CO)NC(N)=O)C2 66904,S(=O)(=O)(CCCCCS(=O)(=O)C(F)(F)F)NCc1ccc(COC)s1 66905,C12(C(=O)NCC3C(C)CCN(C(C4(CC(F)F)CC4)=O)C3)CCC(CC1)C2(C)C 66906,C=C1Cn2c(C(=O)NCC3CC4CN(C(=O)C=CSC)CC34)nnc2S1 66907,C1(NC(c2cc(OC)ncc2Cl)=O)COC2(CCN(C(C3CC3C#N)=O)CC2)C1 66908,N1(C(C#CC(OCC)OCC)=O)CC(C)N(C(=O)CC(F)(F)C(C)C)CC1C 66909,CC1C(NC(=O)COCC2CCCC2)CCCN1c1ccc(C#N)nc1 66910,N1(C(CC(=O)OCC)=O)CC2(CC(CC(=O)NC3(C#N)CC3)C2)C1 66911,N(C(=NCCCCC(C)(F)F)NC(c1cnnn1C)C)C(CC)CC 66912,C1(C(c2ccccc2)NC(NCC(CC)(C)c2ccccc2)=NC)CC(C2CC2)=NO1 66913,Cc1cc(C#N)ccc1NC(c1ccc(I)cc1F)=O 66914,c1(OCC)ccc(Cl)c(NC(C2CCN2CC2CCCC2)=O)n1 66915,N(C1CN(C(=O)C2=CCSC2)Cc2ccccc21)C(=O)C=CC1CCCO1 66916,CC1CCCC(CC(=O)NCC(C2CCCCC2)NC(C2CC(F)C2)=O)C1 66917,CC(C(=O)N1CCOC(CCCNC(c2ccc(F)c(N)c2)=O)C1)C(F)(F)F 66918,c1(N2CCC(NC(C(COC)NC(C)=O)=O)C(O)C2)cc(C#N)nc(SC)n1 66919,c1(C(N2CCC(C)(CNC(c3ccccc3F)=O)C2)=O)cc2ccc(F)cc2o1 66920,C1(c2cn(C(C)C)nc2)CN(C(=O)C(c2cnn(C3CC3)c2Cl)=O)CCO1 66921,C1(NC(=O)C(F)=CC2CC2)CN(C(c2ccccn2)=O)C2(CCCOC2)C1 66922,C(=O)(CCN(C)C(C1CC1Cl)=O)N(CC1C(C(=O)NC)C1)C1CC1 66923,C1(CCC)CN(C(c2cnc(=N)[nH]c2)=O)CC1C(=O)NC1(C)CCSC1 66924,C1(C(N(C)CCF)=O)(CNC(c2coc(C(F)F)c2)=O)CC12CCC2 66925,Cc1cccnc1C(C(=O)NC(C1CCOC1)C)NC(=O)OC(C)(C)C 66926,C(C)(CCCC(=O)N(CCCC(C)O)C)NC(Cc1c(C)scc1)=O 66927,C1(NC(C2C(CC)CCN2C(c2nccnc2N)=O)=O)CCCC(C)(C)C1 66928,N1(C(CNC(CCC(C)C)=O)=O)CCC(NC(=O)CC2CNC(=O)C2)C12CCC2 66929,c1(C(=O)NCC2CN(C(COCCC=C)=O)C2)c(N)cccc1Cl 66930,N1(C(Cc2c(C)occ2)=O)CC2CN(C(=O)COc3ccc(F)cc3)CC2(C)C1 66931,c1(C(=O)NC2CC(CNC(C3CCCC3(F)F)=O)C2)ccc2nc(S)oc2c1 66932,C1(C(=O)NC(CC#C)CC(F)F)CCN(C(c2cnn(C(F)F)c2)=O)C12CCC2 66933,C1(=CC(=O)NCC(CN(C(C(CC)O)=O)C)O)CC2CCC(C1)N2C 66934,N(C(=NCCCN(CC(C)C)C)NCC1CCCCS1(=O)=O)CC(C)C 66935,CC1=C(C(=O)NC2CC3CC(NC(c4cc(O)nc(C)n4)=O)CC23)CCCC1 66936,CC1CCCN(Cc2c(NCC3(C)CCCC3)cccc2)C1 66937,c1(C(=O)OC)c[nH]c(C)cc1=NC1CN(C(=O)OC(C)(C)C)CC1C(N)=O 66938,Cc1c(C(N2CC3(CC3)CC2CNC(=O)CCOC(C)C)=O)sc2ccccc12 66939,C(CC(C(=O)N1CC(O)C(O)C1)NC(=O)CC1CCCN1C)SC 66940,c1(CNC(C(C)N(C(CC)C)C)=O)nc(SC(F)F)n[nH]1 66941,C1(C)(CNC(CC2C=NN(C)C2=O)=O)CN(CCc2ccccn2)CCO1 66942,CC1CCN(C(=O)CCc2c(Cl)cncc2Cl)CC1NC(=O)C=CC1CC1 66943,c1(CC(=O)NCC(C)NC(=O)Cc2cncs2)ccnc(O)c1 66944,C1(CCC)CCCC1C(=O)N(CCCC(=O)NCCCc1ccnn1C)CC 66945,c1(N(C)C(C23CCC(C(=O)Nc4nccs4)(CC2)C3)=O)ccc(F)cc1[N+](=O)[O-] 66946,c1(C(=O)NC(C(C)NC(CC(C)C)=O)C)cc2c(cc1[N+](=O)[O-])OCCCO2 66947,C1(CNC(CC=CC)=O)CC(NC(c2cn(C)cn2)=O)C12CCC2 66948,N1(C(C2CCOCC2)=O)CCC(NC(C2(C3CCCO3)CC2CO)=O)C(F)C1 66949,C(=O)(C1=CCCOCC1)N1CCCCC(CNC(C23CCC(C)(C2)CO3)=O)C1 66950,N1(c2nnc(C(C)(C)C)s2)CCCC2(CC(NC(=O)Cc3ccc(O)nc3)C2)C1 66951,C1(C(=O)NC(CC)CN2CCCC(C)C2)COCCC1(F)F 66952,c1(SCc2nc(C(C)OCC)nn2-c2ccc(SC)cc2)cc(Cl)ccc1Br 66953,C(=O)(C(F)C(CC)CC)N1CCN(CC(C)NC(c2nc(CCC)oc2)=O)CC1 66954,C(=O)(C1=CS(=O)(=O)CCC1)N(CC(C)NC(=O)COc1cccc(O)c1)CC 66955,n1(CC)cnc2nc(N3CCN(C)C4(CCC4)C3)nc(N(CC(F)(F)Br)C)c12 66956,CCC(CCCC(=O)N1CCOC(CC)CC1)NC(C1CCN1CC)=O 66957,CCS(=O)(=O)CC(=O)N(CC(C)N(C(=O)CCCC(=O)c1ccccc1)C)C 66958,CCC(CNC(=O)CCN(C(C1CC12CCOC2)=O)CC1CC1)C(C)C 66959,C1(CNC(C(C)(O)CCc2ccccc2)=O)CC2CCC1N(C(=O)CCF)C2 66960,C1(C(=O)NC2(C(=O)OC)CCC2)CCCN(C(c2cccnc2F)=O)CC1 66961,C1(C(=O)NCCN(CCO)CC)(NC(=O)Cc2cncc(F)c2)CCN(C)C1 66962,c1(C(N2CCCC(C)(NC(=O)CCC3CCCOC3)C2)=O)ccnc2c1CCN2 66963,C(=O)(CN=c1[nH]c2ccccc2s1)NCC1CCC(NC(C(C)(C)O)=O)C1 66964,N1(C2CN(C(=O)NCC3CC3c3ccco3)C2)CCCS1(=O)=O 66965,c1(NC(=O)CNC2CCOC2C(F)F)ccc(C2CC2)cc1Cl 66966,C1(CCC)CN(C(=O)CC(C)C)CC1C(=O)NCC(F)C1CCC1 66967,C1(C(C)C)CN(C(=O)CC(C)c2cnn(C)c2)CCN1C(c1ccoc1Cl)=O 66968,C1(C(N(CC(C)NC(C2COC(=O)N2)=O)C)=O)CCCN1C(c1ccccc1)=O 66969,C(=O)(C(F)C(C)(C)O)N(CC(CC)NC(c1nnc(C)s1)=O)CC 66970,CN1CCC(C(=O)NC2(CCNC(C3CCC(F)C3)=O)CCC2)CC1=O 66971,N1(C(C(C)(C)Cc2n(C)cnc2)S(C)(=O)=O)CC(C#N)(S(C)(=O)=O)C1 66972,C(c1ccc(F)nc1)=CC(=O)NCC(CNC(c1c(C)nc(N(C)C)s1)=O)C 66973,C1(N(C(c2ccc(CNC(C)=O)s2)=O)C)CCCN(C(C2COC(=O)O2)=O)CC1 66974,C(=O)(CC(C)(C)CNC(c1cc(Cl)n[nH]1)=O)NCC(C)CC1CCC1 66975,C(=O)(C(C)(O)C(F)(F)F)N1C(CCNC(C2CCCCC2)=O)CC(OC)C1 66976,C(CCC(CCC)N(C(C=CCC)=O)C(C)C)NC(c1n[nH]c2c1CCC2)=O 66977,C1(C(=O)NC(COC(C)C)CO)(CC)CCCN(C(C2CCCN2C(C)=O)=O)C1 66978,C(=O)(CC1=CCOCC1)NC(C1CCN(C(c2nc(C)n(C)c2)=O)C1)(C)C 66979,Cn1ccc(=O)c(C(=O)NCCCN2CCN(C(C3CCS(=O)(=O)C3)=O)CC2)c1 66980,Cc1cc2ccccc2nc1C(N1CC2CCN(c3nncs3)CC2C1)=O 66981,C(CCCCC(=O)N1CC(NC(=O)CSC)CC(C)C1)OCC 66982,c1(C(N2CCCCC2c2cn(CC(F)(F)F)nn2)=O)cc2n(n1)CCC2 66983,CC1(C)CC(C(=O)N(C2CCCCCC2)CCC2(C3CC3)CCCO2)CO1.C(=O)(N)CCC 66984,N1(C(C=C(CC)C)=O)CCC2(CC1)CCN(C(c1cncc(N(C)C)c1)=O)CC2 66985,c1(C(=O)OC)cc(NC(c2sc(NC(C3(C)CCC3)=O)cc2C)=O)c(C)cc1Br 66986,c1(CC(N2CC(C)C(n3cc(C(C)(C)C)nn3)C2)=O)cc(C#N)ccc1F 66987,c1(NC2(COC)CCN(C(CC3ON=C(CC)C3)=O)C2)cc(C)nc2ccnn12 66988,N1(C(c2c(C)nco2)=O)CCCC(O)(CN(C(=O)C(C)CN2CCCCC2)C)C1 66989,C1(C(=O)NC(C(=O)NC2CC2O)c2ccco2)CN2CCCC1C2 66990,CC(CN1CCOCC1)N=c1[nH]c(=NC(C)c2nc[nH]n2)[nH]c2c1CCCCC2 66991,Cn1ccc(-n2cc(CC3CCCN3C(c3nccs3)=O)nn2)cc1=O 66992,C1(C(c2n(C(C(=O)OC)C)nnn2)NCc2ccoc2)CCOC1(C)C 66993,c1(C(=O)NCc2c(OC)cccc2O)nsc2cc(Br)ccc12 66994,C1(CN(CC(CN(C(CC(C)c2ccco2)=O)C)O)C)CC(=O)c2ccccc2O1 66995,c1(CN2CC3CN(C(=O)CCc4ccccn4)CC32)ccc(I)c(F)c1F 66996,C(=O)(C#CC1CCCOC1)NCCOCCN(C(CC(C(=O)OC)C)=O)C 66997,CCC(C)C(C)(O)CNC(C1(CCNC(=O)C(CC(C)C)OC)CCC1)=O 66998,CC1CCCC(O)(CNC(c2conc2CNC(=O)Cn2ncccc2=O)=O)C1 66999,N1(C(C(CCC)O)=O)CCCC(C)(NC(=O)Cn2ncc(O)nc2=O)C1 67000,c1(SCC)ncccc1C(=O)NCC(C)(C)NC(=O)C(C)NC(C)(C)C 67001,N1(C(c2c(CC)ocn2)=O)CC(NC(c2cc(N)ccc2F)=O)C2CCCC2C1 67002,Cc1ccc(Cl)c(C(=O)NCC2CCN(C(C3(n4cnc(O)n4)CC3)=O)C2)c1N 67003,C1(OC)CC(CN)N(C(=O)CC(C)c2cccnc2)C1.C(=O)(CC(C)(C)C)C(=O)CS 67004,CCCC(O)C(CO)NC(C1(CNC(=O)C(C)COC)CC=CC1)=O 67005,C(=O)(C(F)C(C)(C)O)N(C1CCN(C(=O)CCSCC(C)(C)C)C1)CC 67006,N1(CCC)CCCCC1C(=O)N(C)CC1CCCCN1C(c1cn(C)cc1C)=O 67007,N(C(=NCc1cccs1)NC1CC12CCCC2)C(CC)C1CC1 67008,CCCC(CCO)NC(=O)CNC(C1(CC(=O)OC)CC1)=O 67009,c1(OC)cc(C(=O)NCCc2ccccc2O)cc(C)c1 67010,c1(CC(N2CC(OC)C(CNC(=O)CC(C)OC)C2)=O)ccc(Cl)cc1Cl 67011,C12(NCC(C(C)O)O)CC(NC(=O)OC(C)(C)C)(C1)C1(CCOCC1)O2 67012,N#CC1CN(C(c2cccc(N3CCOCC3)c2)=O)CC1NC(=O)CC(F)(F)F 67013,C1(NC(=O)Cn2cncn2)(CO)CCN(C(=O)CCc2cccc(F)c2)C1 67014,N1(C(COC(C)=O)=O)CCCC(C2CCCN(C(C3Cc4nccnc4C3)=O)C2)C1 67015,N1(C(CP(C)(C)=O)=O)CCOCC(NC(c2ccccc2Cl)=O)C1 67016,N(C(=NCCC1CC(F)C1)NCc1ccco1)CC(N1CCCCC1)=O 67017,CS(=O)(=O)c1cnn(CC(=O)NC2CCCC(NC(c3cnco3)=O)CC2)c1 67018,c1(C(N2CC(Nc3ccccc3)(CO)C2)=O)cncc(Cl)n1.O=C1CCN1 67019,C1(C(=O)NC2C(CC)N(C(=O)C=C(C)c3ccco3)CC2)CC(F)(F)C12CCC2 67020,Cc1cc(CO)cc(Cn2cc(C3CN(C(=O)CCn4ccnc4C)C3)nn2)c1 67021,CCCC(CC)CC(=O)N1CC2CCC(C1)N2C(c1nc(Br)c[nH]1)=O 67022,C1(C(N(CCOCC)CC)=O)CN(C(=O)C(CC)n2cccn2)CC1F 67023,N1(C(CCC(CC)OC)=O)CCC2(N(C(=O)Cc3csc(S)n3)CC)CCCC12 67024,C1(NC(c2nccc(OC)c2)=O)CN(C(=O)C(C)(C)N(C)C)CCC1C(F)(F)F 67025,C1(COC)CC(CNC(C2CC2C(C)(F)F)=O)N(C(=O)CCOCC(C)C)C1 67026,c1(NC(CSCC=C)=O)ccccc1NCC(N1CCC(N2CCCC2)C1)=O 67027,c1(C(=O)NC2(CNC(C3(CC#C)CCCO3)=O)CCC2)nnn2c1C(=O)NCC2 67028,C(=O)(C(C)(C)C(C)(C)C)NC1CN(C(CC2C(C(=O)OCC)C2)=O)C1 67029,Nc1ncc(Br)cc1C(=O)Nc1ccc(Cl)cc1NC1CCOCC1 67030,c1(C(=O)NC(CNC(CC2CC(=C)C2)=O)C2CCC2)nccc(N)c1Cl 67031,c1(CN2CCN(C(=O)OCC)C(CC)C2)cc(F)cc2nccnc12 67032,Cc1c(NC(=O)C(C2CCCN(C(=O)C(C)n3cccc3)C2)(C)C)cnn1C1CC1 67033,C1(CC(=O)NCC2(C#N)CCC2)(NC(=O)C(=O)NCC2CC2)CCSC1 67034,C(=O)(C(C)(C)CNC(C1CCCCO1)=O)N(CCO)CC 67035,C1(CNC(c2ccc(OC)s2)=O)CCC(CNC(=O)C(O)C2CC2)CC1 67036,Cc1cc(Cl)c(Cl)cc1C(N1CCCCC1CNC(c1cn(C2CC2)nn1)=O)=O 67037,C1(C(N(C(C)CNC(=O)CC(C)(C)C2CCCCC2)CC)=O)CC(C2CCC2)C1 67038,c1(CC)ccoc1C(=O)N(C)CCOCCC(=O)NCC(=O)NC1CC1 67039,Cc1[nH]c2ccccc2c1C(N1CCC2(C1)CN(C(C1C(F)(F)C13CC3)=O)C2)=O 67040,C=CCC(C(=O)N1CC(CNC(c2cc(Br)cnc2C)=O)(OC)C1)C(C)C 67041,c1(CNC2CN(C(CCc3c(C)noc3C)=O)CC2C)cc(F)cc(C#N)c1 67042,c1(NC(C2C(C(N(CCOC)C(C)C)=O)C2)=O)cc(SC)nc(C)n1 67043,N1(C(C(C)N2CCC2)=O)CCCCC(C(=O)N(Cc2ncccn2)CC2CC2)C1 67044,N1(C(C(COC)C)=O)CC(NC(c2cc(Br)ccc2OC(F)F)=O)C2(CC2)C1 67045,C1(N(C(c2cc(OC)ns2)=O)C)CCN(C(c2cccc(C)c2N)=O)CC12CC2 67046,C1(CNC(C2(OCC)CCOC2)=O)(CNC(=O)CC(F)F)CC12CCC2 67047,C(CCC(C)(C)C(=O)NCCCc1cnn[nH]1)NC(c1cc(=O)cc(C)[nH]1)=O 67048,N1(C(c2ccc(C(C)=O)o2)=O)CCCC(N(C(=O)C2=CCOC2)C)C1 67049,c1(C(CC)OC2CC(c3nccc(Cc4ccccc4)n3)C2)ccccc1OC 67050,CC(C)CCC(C(=O)Nc1cccc(F)c1C)NC(c1cnn[nH]1)=O 67051,CC1CN(C(C2(O)CCOC2)=O)CC1NC(c1cc(C2CCC2)nn1C)=O 67052,c1(C(=O)NC2CCN(C(C3CC(C#N)C3)=O)CC2O)cccc2c1OCCO2 67053,N1(C(CCOC(C)C)=O)CCC2CCN(C(c3cc(C(F)(F)F)n(C)n3)=O)C2C1 67054,c1(N(C(=O)Cc2cccc(C3CCC3)c2)CCO)ncc([N+](=O)[O-])cn1 67055,c1(OC)cccc(C(N2CCC(CSC)C2)C(=O)Nc2csc(C)n2)n1 67056,c1(C(=O)NCC(C)(C2CC2)NC(=O)CCNC(=O)C=CCl)ccc(CCF)cc1 67057,n1(CC(=O)NCC2(C)CCN(C(C3CC(S(C)(=O)=O)C3)=O)C2)ncc(O)nc1=O 67058,C(CCN(C)C(c1cnn(COC)c1)=O)(C(C)C)NC(c1ccc(CCC)[nH]1)=O 67059,Cc1csc2ccc(CC(=O)NC(C)CCCNC(C3CCC(O)C3)=O)cc12 67060,C(N=c1ccc2nnc(Sc3ccccn3)n2[nH]1)c1scc(CSC)n1 67061,C1(C(=O)NC2C3CCN(C(CCOC)=O)C32)COc2ccc(F)cc2C1 67062,C1(C(=O)NCC2(C(=O)NCCCOCC)CC2)CC=CCC1 67063,C(CC(C(C)(C)C)NC(c1ccnc(CO)c1)=O)N(C)C(c1cnc(N)cn1)=O 67064,N1(C(C(C)SCCCC)=O)CC2(CCCN(C(=O)CC3CC(=O)NC(=O)C3)C2)C1 67065,Cc1ccc(C(N)=O)cc1NC(=O)NCC1CC(NC(=O)C(C)CC(N)=O)C1 67066,Cc1nc(C(N2CCC(CCC(C)(C)C)(NC(C3C4CCC34)=O)C2)=O)oc1C 67067,C#Cc1ccc(C(=O)NCCC(CNC(=O)CN2CCC(=O)CC2)OC)cc1 67068,C1(OC)CCC(C(=O)NCCn2cc(C(N3CC(C(C)(C)Cl)C3)=O)nn2)CC1 67069,Cc1cc(F)c(F)cc1C(N1CC2CC1C2C(=O)Nc1ncc(Br)nc1Cl)=O 67070,c1(C(N(CCCN(C(=O)C(F)C2CCOC2)C)C)=O)cc([N+](=O)[O-])ccc1N.CN 67071,C1(C(C)C)CN(C(=O)Cn2cnnn2)CCC1NC(=O)C(F)(F)c1cccnc1 67072,N1(C(CS(=O)(=O)N(C)C)=O)CCOC2(C1)CN(C(C1(Cl)CC1(C)C)=O)C2 67073,c1(C(N(CC(O)CN(C)C(C2CCCN2N=O)=O)C)=O)ccn(C)c(=O)c1O 67074,C1(CC(=O)NCC(CO)NC(C2CC2Cc2ccccc2)=O)CCCCCC1 67075,Cc1cccc(CNC(=O)CC2COCCN2C(c2ncc(Br)cc2Cl)=O)c1F 67076,C1(C(=O)OCC)CC2(CCCN2C(=O)C(=O)N(C)CC2CCCS2)C1 67077,N1(C(CN(C)C(N)=O)=O)CCC2(CCCCN(C(C3(Cl)CC3(C)C)=O)C2)C1 67078,N1(C(c2c(C)ncs2)C(=O)NC(C)(C)C)CC(C)(C)OC2(CCOC2)C1 67079,c1(C(N2CC3CN(C(C(C)(C)C(F)F)=O)CC3C2)=O)nc2ccc(Cl)nn2n1 67080,N1(C(c2c(SC)csc2)=O)CC2CS(=O)(=O)CC2(NC(c2ccc(=N)[nH]c2)=O)C1 67081,N1(C(C2C(C)OCC2)=O)C2CCC1CN(C(=O)C(c1ccccn1)C)C2 67082,c1(OC)c(C(=O)NCC2C3CN(C(c4n[nH]cc4F)=O)CC23)cccc1Cl 67083,C1(NC(c2c(C)nnn2C)=O)CC2CC(C1)N(C(=O)CCc1cncc(F)c1)C2 67084,Cc1cc(C(F)(F)C(=O)NCC(O)CNC(=O)CCC2CCC(C)O2)cc(C)c1 67085,C1(C(=O)NC2CC3CC(NC(c4cc(C)oc4)=O)C3C2)CCC(=C(F)F)CC1 67086,c1(C(=O)NS(CC2CC(OC)C2)(=O)=O)nccc2[nH]ccc12 67087,c1(NC(C2CC(F)CN2C(C2CCOC2)=O)=O)cnc(Br)nc1 67088,c1(C(=O)NC2CC(C(F)F)(NC(Cc3cn(C)nc3)=O)C2)cnc2[nH]ccc2n1 67089,C(CN=C(NCC(c1cnccn1)C)NCCN1CCCC1)C1(OC)CC1 67090,C1(CCNC(C(Cc2ccccc2)N(C)C)=O)CN(C(C2SCCS2)=O)CCO1 67091,CC(C)C(C)C(CNC(=O)COCCF)NC(c1cc(C#N)on1)=O 67092,c1(NC)cccc(C(=O)NCCCCOC)n1.N12CC(O)(C1)C(F)C2=O 67093,C(C(N=c1[nH]ccn2nnnc12)c1ccco1)OC 67094,c1(C(N2CC(OC)C(F)C2)C(=O)NCCC#N)cc(C)cc(Br)c1F 67095,c1(NC(C2(C(=O)C3CC3c3ccccn3)CC2)=O)cnc(O)c2ccccc12 67096,C1(NC(C2N=C(C)SC2)=O)CC(C)N(C(=O)C=Cc2ccsc2C(F)(F)F)C1 67097,c1(NC(C(=O)N(C2CCN(C)CC2)c2ccccc2)=O)c(C#N)cnn1C(C)(C)C 67098,c1(C(N(CCCOCCN(C(c2c(C#C)c[nH]n2)=O)C)C)=O)cccc(Cl)c1F 67099,C1(C)(CC)CC(C(N2CC(c3cc[nH]n3)C2)=O)C1.C1C(C)(C)OCC(=O)N1 67100,c1(CC(N2CC(C)C(NC(c3nc(=O)n(C)[nH]3)=O)C2)=O)ccc2sccc2c1 67101,N1(C(c2c(CC)cns2)=O)CC2=C(C1)CN(C(c1cc(C)c(C)[nH]1)=O)C2 67102,CC(CCO)C(=O)N1CCCCC1Cc1cn(-c2cccc(F)n2)nn1 67103,C1(CC(=O)NCC2C(C(N(CC(F)(F)Cl)C)=O)C2)CCCCO1 67104,N1(C(C2C=CCN(C(C3C=C(C)CS3)=O)C2)=O)CC2CCCCC2C1 67105,C1(C(=O)N(C2(C(=O)NC3CCCC(CC(C)C)C3)CC2)C)(OC)CCCCC1 67106,c1(Cn2ncc(C(=O)NC(C)C(CO)NC(CC(F)(F)F)=O)c2)ccc(O)cc1 67107,N1(C(CSCCOC)=O)CC2CCN(C(c3ccc4nonc4c3)=O)CC2C1 67108,O=C(C1=NOC2(CCC2)C1)N1CC(C2CN(C(=O)C(C3CCCCC3)F)C2)C1 67109,c1(C(N2CCCC(NC(=O)CC3CCCCC3O)C2)=O)ccc2nc(S)[nH]c2c1 67110,C(c1cncc2ccccc12)=CC(=O)N(C(C)C(=O)N1CCCC1)C 67111,C1(NC(c2nc(CCC)oc2)=O)CC(N=c2[nH]c3cccnc3s2)C1 67112,C12(CC(=O)NC(C(=O)N(CC(F)Cl)C)Cc3cn[nH]c3)CCC(CC1)C2 67113,CCS(=O)c1ccccc1C(=O)N(C(C)CNC(c1cc(OC)n[nH]1)=O)C 67114,c1(C(N2CCC(CNC(C(c3cccc(Cl)c3)CC)=O)C2)=O)ccc(F)c(N)c1 67115,c1(CC(N2CCCC(NC(C(C)OCC)=O)C2)=O)ccc2nsnc2c1 67116,Cc1ccc(CNC(C2CCN(C(=O)CN3CCCCC3)CC2)=O)c(F)c1F 67117,C=CCC(C)C(=O)NCC=CC(=O)NCC1(CO)CCCO1 67118,CCC(O)C(C)(C)C(=O)NCC1(O)CC(C(=O)N(CCC(F)(F)F)C)C1 67119,C(=O)(CC(C)(C)C(F)F)NCC1N(C(c2c(Cl)cn(CCC)n2)=O)CCN(C)C1 67120,Cc1c(C(=O)NCC2CN(C(=O)C=CC3CC3)CC2C)noc1-c1ccccc1 67121,C1(C(N2C(C(N3CCC(NC(CC)=O)C3)=O)CC(O)C2)=O)CC2(CCO1)CC2 67122,c1(C(=O)NCC23CC(NC(C(C)OCC4CC4)=O)(C2)C3)ccc2nccn2c1 67123,C12CCCN1NC(=O)C1CN(CC1F)C2=O.CCC(CC)OC(C)=O 67124,c1(CC(=O)NC(C)(C)CCNC(C23CCCC2C3(F)F)=O)c[nH]c2cnccc12 67125,N1(C(c2c(NC)cccc2)=O)CCC2C(CCCN2C(C2(C)CCCC2)=O)C1 67126,CC1(F)CCC(C(=O)NOCc2cn(CC3CCC(F)(F)CC3)nn2)CC1 67127,C1(C(=O)NCCN2c3c(cc(C)cc3)C2=O)CCC2C1C2(F)F.CCCOC 67128,CC1CN(C(c2cnccn2)=O)C(C)CN1C(C1OCC2CCCCC12)=O 67129,N1(C(c2sccc2Cl)C(=O)NCC)CCC(C)(C(=O)OC)C1.C(C)(C)(C)OC(=O)N 67130,c1(N(C(=O)C(=O)NC2CCC(CC#N)CC2)CC#C)ccc(F)c(Cl)c1 67131,C1(NC(C(CN(C)C)(C)C)=O)CN(C(c2ccc(Cl)cn2)=O)CCC1CO 67132,C(=O)(C1CCCc2cc(O)ccc21)NCC(C)NC(C1CCN(CC(C)C)C1)=O 67133,N1(C2C(c3n(C)nnc3)C2)CCN(Cc2ccsc2C(F)(F)F)CC1 67134,C1(CC)CN(C(=O)CSc2nncn2C)CCC1NC(c1cc(Cl)cs1)=O 67135,c1(NCCC(=O)OC(C)(C)C)ccc2[nH]c(C)c(C(=O)OCC)c2c1.C1CS1 67136,N1(C(CNC(CC)=O)=O)CCC(C(C)C)CC1CNC(=O)C=CBr 67137,C(=O)(CCCCC(C)(C)C)NCCCC(C(=O)Nc1c(C)ccs1)N.C1CC1 67138,C=CCC(CC)C(=O)NCC1(O)CC(C(=O)NCCC(O)CO)C1 67139,C1(CC(C)NC(C23CSC(C2)C3)=O)CCN(C(=O)CN2CC(=O)NC2=O)CC1 67140,CN1CCC2CCN(C(=O)C(O)CCCNC(c3ccc(F)c(F)c3)=O)C2C1 67141,N1(C(Cn2cc(CCCC=C)nn2)=O)CCC(O)C1C(C)(C)C 67142,C(C)(C)(CC(C)(C)O)NC(C1N(C(C=C=C(C)C)=O)CCC1)=O 67143,C=CCCCCC(=O)NC(CNC(C1CCCC(C)(C)O1)=O)CO 67144,C(C(=O)N1CC(F)(F)C1C1CC1C(=O)O)(C(C)(C)C)NC(c1c(C)nccc1)=O 67145,Cc1c(Br)ccc(F)c1C(=O)NC(C)CCNC(=O)CC1C=CCC1 67146,N1(C(C2=NNC(=O)C2)=O)CC(NC(=O)CC2CCC(=O)NC2)CC(F)(F)C1 67147,O=C1CNC(=O)C(CC(N2CC3CN(C(=O)CC4CC5CC4C5)CC23)=O)N1 67148,C1(C)(C(N2CC(SC)C(n3cc(CC4CCOC4)nn3)C2)=O)CCCCNC1=O 67149,C(C1c2ccsc2CCN1C(=O)CSCC(N)=O)NC(c1n(C)cnc1)=O 67150,C1(C(=O)NCC2C(C)CN(C(c3cc(Cl)on3)=O)CC2)CN2CCCN1CC2 67151,N1(C(CCN(C)C(c2ccc(CO)c(F)c2)=O)=O)CCCC2CCCC12 67152,c1(NC(c2nc(NC(C)=O)sc2)=O)ccc2nc(Br)sc2c1.C12CC1CNC2=O 67153,C(=O)(C(F)C(C)(F)F)NC(C)CC1CCC(=O)C1.c12ccc(s1)CNC2=O 67154,C1(NC(C)=O)C2CC3C1C3C2C(=O)NC1C(F)(F)C12CC2 67155,C1(C(=O)OC)CCCC(C(N2CCC(F)(C(N3CCOC(CO)C3)=O)C2)=O)C1 67156,C12(CC(N3CCC4CC34)=O)CCC1CN(C(c1cccc(CO)n1)=O)C2 67157,C1(C)(C(=O)NCC2(O)CC(C)(C)C2)CCCN(C(=O)Cn2cnc(C#N)n2)C1 67158,c1(NCC(C)Oc2nccc(Cl)c2C(F)(F)F)c(F)cccc1Cl 67159,C(=O)(C(F)(F)Cn1cc(Br)cn1)N1CC(C(=O)NCc2ccc(C(F)F)nc2)C1 67160,C(=O)(CN=c1ccc(Cl)n[nH]1)N1CC(CNC(c2nn(C)c(O)c2)=O)C(F)(F)C1 67161,CCC(C)C(C(=O)NCCc1cnc(C)o1)N(C(=O)CCCC1CC1C)C 67162,C#CCC1(C)C(=O)N(C2CC(=O)NC2=O)CC2(CC(=O)N1)CC2.C1CC1.SCC 67163,C(C(N=[N+]=[N-])C(=O)NCC(C)(C)NC(C1CC(=O)N1)=O)OCC 67164,C1(C2CCN(C(=O)CCCN3CCCC3)C2)(NC(c2cccc(CC)n2)=O)CC1 67165,C1(CNC(CCCC=C)=O)CN(C(=O)CN2CCC(=O)NC2=O)CC1(C)C 67166,c1(C(N(CCCNC(C2CC2(C)C)=O)C(C)C)=O)cnc(CCC(F)(F)F)s1 67167,C1(C(=O)NC2CCC(NC(C3CC34CCC4)=O)CC2)CC2CSCC(C1)C2 67168,N(C(=NCCc1ccc(Cl)c(C)c1)NCC1CC2CC1CC2O)C(CC)CC 67169,C#CC1CN(C(=O)C(c2c(C)cccc2Br)NC(=O)CCCC=C)CCO1 67170,Cc1c(Br)noc1C(N1CCC(C)C1CNC(=O)CN1CC2CC2C1)=O 67171,C(=O)(C1=CC2CCC(C1)C2)N1CC(C(N(C)CC2(C)CC2)=O)C(F)(F)C1 67172,c1(C(=O)NCC(CN(C(c2cc(CCC)nn2C)=O)C)(C)C)cc2occc2[nH]1 67173,N1(C(C(C)CC(N)=O)=O)CCCCCC(Nc2ncnc(C(C)(C)C)n2)C1 67174,N1(C(CCC#C)=O)CCCC(CCCCNC(C2(Cl)CC2(F)F)=O)C1 67175,c1(C(N2C(CC(=O)NC(C#C)C)CCC2)=O)c(NC)cccc1F 67176,c1(C(N(C(CNC(c2cc(C)c(C)o2)=O)C2CC2)C)=O)ccn2nccc2n1 67177,CC(=O)C(C)(C)CC(=O)N1CCCC1C(=O)N(C1CC(O)C1(C)C)C 67178,c1(NCC(C2CC2)NC(C2(OCC)CCCCC2)=O)ncc(Cl)c(C)c1C#N 67179,c1(N2CCCC(N(C)CCO)C2)ccc(S(=O)(=O)NC(C)=O)c(Cl)c1.CCCCO 67180,CC(C)(C)C#CC(=O)NCCCC1CCCCN1C(=O)CC1CCC(=O)O1 67181,N1(C(C(CCC)OC)=O)CC2CCCC1(CNC(c1cn(C)nc1C)=O)C2 67182,N1(C(c2cccc(Cl)c2O)=O)CC2(C1)CN(C(C13CC(O)C1C3)=O)CC2CO 67183,Nc1c(C(=O)NC2CC2NC(C2CCC(N(C)C)CC2)=O)cccc1[N+](=O)[O-] 67184,c1(CC)c(C)nn2c(=O)cc(C(=O)N(C(C)CCNC(C3(C)COC3)=O)C)[nH]c12 67185,C=C(C)C(O)CC(=O)NCCC1CN(C(=O)CCCc2nc(CC)no2)CCO1 67186,c1(C(=O)NCC(CC)(CC)NC(C2C(=C)CC2)=O)cc2n(n1)CCNS2(=O)=O 67187,c1(CCC(=O)NCC2CCCN(C(C(CC)(C)O)=O)CC2)nc2ncccn2n1 67188,c1(NC(C2C3(CN(C(c4cncc(C)n4)=O)C3)C2)=O)cc(C(F)(F)F)ccc1I 67189,C(=O)(CC(CC)CCCC)NC(CCC#C)C(=O)NC(C)Cc1ncn(C)n1 67190,C(=O)(C(F)Cc1ccccc1)NC1(CN(C)C(C2CC(=O)C2)=O)CC1 67191,C#CCC(CC(F)F)C(=O)NC(C(=O)NCC1=C(C)CCOC1)C(C)CC 67192,N1(C(CC2CC(=C)C2)=O)C(CNC(c2sncc2C)=O)CC2CC12 67193,CN(C(=NCc1cccs1)NCC1CCCN1C)CCc1ccsc1 67194,c1(C(=O)NC(CC)(CNC(=O)C(C2CC2)OC)CC)n[nH]c2c(C)cccc12 67195,c1(C(=O)NC2CN(C(=O)C3=CCCOC3)CC23CC3)[nH]nc2ncnc(O)c12 67196,c1(CC(=O)NCCC(C)NC(c2c(F)ccc(CC)c2)=O)cnn2c1CCCC2 67197,C(=O)(C(CCSC(C)C)NC(=O)NOCC=C(C)C)NC 67198,CC1=C(C(=O)NC(C)(CNC(C2(C)CNC(=O)N2)=O)C2CCC2)SCCO1 67199,c1(NCCC2CC(NC(c3n(CCC)nnn3)C3CC3)C2)nc(C)c(C)s1 67200,N(C(=NCCOCC1CCOC1)NCCn1cccnc1=O)CC(C)C 67201,Cc1cccc(C)c1NC(N1CCOCC(NC(c2nc(C3CC3)cs2)=O)C1)=O 67202,Cc1ccccc1-n1cc(C(=O)NCC2CC2NC(C2CC(C)(C)CO2)=O)nn1 67203,c1(-c2n(CC=C)c(N(C)CC3CCCC3O)nn2)cnc2c(C)nsc2c1 67204,Cc1cccc(N2CCC(NC(=O)Cn3cc(-c4cnn(C)c4N)nn3)C2=O)c1 67205,C(F)(c1ccccc1)=CC(=O)NCCC(C)(C)NC(C1CCC(F)(F)C1)=O 67206,c1(C(C(N2C(CN(C(c3c(CC)ocn3)=O)C)CCC2)=O)C)ccncc1C 67207,N1(C(CC(CC)C2CC2)=O)CC2CC(NC(=O)C3=CCCCCC3)CC1C2 67208,CC(C)C(C)(C)C(=O)NCCN(C(C1CC(S(C)(=O)=O)C1)=O)C1CC1 67209,C(CN=c1cc[nH]c(C(N)=O)c1)SCC(=O)SC1CCN(C(C(CC)O)=O)CC1 67210,c1(C(N(C(C)CCNC(=O)C(C(C)O)NC(N)=O)C)=O)cnc(N)c(Cl)c1 67211,C=CC(CCC)CC(=O)NCCN1CCC(NC(c2sccc2OC)=O)CC1 67212,C(=O)(C1=NOCC1)N(CCCNC(c1occc1SCc1cccs1)=O)C1CC1 67213,c1(C(N(CCC(=O)NC(C2CCOC2)C#C)CC)=O)cccc(C#N)c1 67214,CCC(C#N)C(=O)N1CCC(CCNC(c2c(C)noc2C)=O)C1 67215,C12(C(=O)NC)CCCC(CNC(=O)N(N3CCOCC3(C)CC)C)(C1)OC2 67216,C(CCS(C)(=O)=O)(C(=O)NCCCN(C(c1ncccc1O)=O)C1CC1)OC 67217,C12(NC(CCNC(=O)OC)=O)CCCC1CN(C(=O)C(C)CN1CCOCC1)C2 67218,Cc1ccccc1CCC1CCCN(C(=O)NCCCCc2cncnc2)C1 67219,C1(OC)(CNC(c2cc(C3CC3)on2)=O)CCN(C(C2CCCCS2)=O)CC1 67220,Cc1ccc(C)c(C(N2CCCC(C)(C(=O)NCC3CCC(O)CN3C)C2)=O)n1 67221,C1(CC)COC(C)(C)CN1C(=O)CC1(C)CC(NC(c2ncc(F)cc2F)=O)C1 67222,Cc1cccc2cc(C(=O)NC(COC(F)(F)F)C(C)(C)C)oc12 67223,c1(C(=O)NC2(C)CC(NC(C=C3CCC(C)CC3)=O)C2)cccc2c1CCN2 67224,n1(CC(N2CCC(CC(N3CCC(C(=O)NC)C3)=O)C2)=O)nc(C)oc1=O 67225,c1(C(=O)NCC(COC)NC(C2(C)CCOCC2)=O)cc(C)c(OC(C)C)c(C)c1 67226,C(=O)(CCCCCOC)NCC1(C(=O)NC(C#C)CCC)CCCO1 67227,Cc1cc(CC(=O)NC(C)CCCNC(C2CCC2Cc2ccccc2)=O)on1 67228,N1(C(C(F)=CC)=O)CCC(COC)(NC(C2CCCC2)=O)C1 67229,C1(CN(CC(=O)N(CC(=O)N(CC(C)OC)C(C)C)C)C(=O)C2CC2)COC1 67230,CCCCS(=O)(=O)CC(=O)N(C1CCN(C(=O)C(CO)N(C)C)CC1)C 67231,C1(C(=O)NCC(C)N(C(Cc2scc(C)c2)=O)C)C(C)(C)C1(F)F 67232,c1(SC(CCC=C)C)nc2ccccc2s1.C(=O)(CCS)N1CC(=O)NCC1 67233,C(=O)(CC(C(C)OC)NC(=O)C(F)C1CCC1)N1CC(C(CC)CC)C1 67234,c1(N2C(CN(C)C(c3ncccn3)=O)CC(F)C2)nc2cc(F)cc(F)c2o1 67235,C1(C(N(CCNC(C2(CF)CC2)=O)CC)=O)CC2C(C1)C2(F)F 67236,CCCC(O)C(=O)NC(CNC(c1sccc1COC)=O)CC 67237,n1(CC#C)c(C)cc(C(N2CC(CCNC(c3cc(C(C)C)no3)=O)C2)=O)c1C 67238,C1(NC(c2ccc(S(N)(=O)=O)[nH]2)=O)CN(C(c2ccc(Cl)s2)=O)C2CCCCC12 67239,c1(C(C)NC(=O)NC2(C(=O)O)CCCC2(C)C)ccc(Br)cc1O 67240,C(c1ccc(C(C)(C)C)cc1)=CC(=O)NCC1(CO)CN(C(C(CSC)OC)=O)C1 67241,c1(C(N(C2CCN(C(CC3CC(C)(C)C3)=O)C2)CCO)=O)ccncc1Br 67242,CCC(CC)C(C)C(=O)N(CCC(=O)NCc1csc(C)c1)CCCO 67243,N1(C(C=CCN(C)CC)=O)CCCC(N(C(=O)C(N2CCCC(O)C2)C)C)C1 67244,C(CS(=O)(=O)CC(=O)N1CC(NC(c2cc(C)sn2)=O)CC12CCC2)OC 67245,C1(CCNC(c2ccc(CO)s2)=O)(OC)CN(C(=O)Cc2cnc(C)s2)C1 67246,c1(C(C2CC23CC3)NC(=O)NC2CCSCC2)nnc2n1CCC2 67247,CC1CCCC(C)N1C(=O)C(N1CCC(CN(C)C(c2cc(Br)n[nH]2)=O)CC1)=O 67248,C12(C(NOCC=C)=O)CCCC1CN(C(c1ccc(CO)cc1)=O)C2 67249,c1(CCC(N2CC(O)(C(C)NC(C(C)OCCCC)=O)C2)=O)ccnc(C)n1 67250,c1(C(=O)OC(C)(C)C)cccc(Cl)c1SCc1ccccc1.C1(=O)C(CC(C)C)O1 67251,C1(CNC(c2c(Br)sc(C)c2C)=O)C(C)CCCN1C(=O)Cn1cccn1 67252,c1(CC(=O)NC2C(NC(CCCC#C)=O)CCCC2)csc2nc(C)cn12 67253,c1(CNC(=O)C(O)C2CCC2)ccnn1C(C1CC1)C1CC1 67254,CC(C(C)(C)Nc1ccccc1)NC(=O)CN(C(=O)COCC1CCOC1)C 67255,c12nnc(n1CCCC1CCCC1)CO2.c1(C(C)C)ncn(C)n1 67256,C(=O)(C1=CCCCC1P(C)(C)=O)NCCCNC(CC(C)c1cnn(C)c1)=O 67257,c1(C(=O)NC2C(NC(C3(CC)COC3)=O)C2)ccc2ccn(C)c2c1 67258,N1(C(CSCC#C)=O)CC(NC(c2cnc3cc[nH]c3c2)=O)C(C2CC2)C1 67259,C1(NC(COCc2nc(C)oc2)=O)C2CC1N(C(=O)Cc1c[nH]nc1C)C2 67260,Cn1nnc2c1CCN(C(C1CCN(C(=O)C(C)(F)C(C)(C)F)C1)=O)C2 67261,Cc1c(C(=O)NCC(C)NC(C23CC2COC3(C)C)=O)cncc1Cl 67262,C12C(C)CCN1C2=O.C1(CC)CC(NC(=O)C(C)(C2CC2)OC)CCO1 67263,C1(C(=O)NC2CC(N(C)C(C3CC(O)C3)=O)C2)CCc2cnn(C)c2C1 67264,c1(N(C(=O)NCC(C(C)C)c2ccccc2)C)cccc(Br)c1 67265,N1(C(N)=O)CCC(C(=O)NCC(O)CNC(=O)Cc2ncc(Cl)s2)CC1 67266,C(CCCCCC(=O)N1CCC(F)C(O)C1)NC(C(C)SCCCC)=O 67267,c1(C(=O)NC2CC(C(C)NC(C3CC(CCC)OCC3)=O)C2)ccc([N+](=O)[O-])s1 67268,N1(C(C(CCN(C)C)O)=O)CC2CCN(C(c3cccc(Cl)c3N)=O)CCC2C1 67269,C1(NC(c2c(OC)n[nH]c2)=O)CCN(C(=O)CCN2CCOC2=O)CC1O 67270,C1(C(N(N(C)C)Cc2onc(C)n2)=O)CC(C)CN1C(c1ccc(C(N)=O)o1)=O 67271,C1(CNC(C(CC)N(CC)CC)=O)CN(C(=O)CCc2ccccn2)CCC1(C)C 67272,c1(SC(C)C(=O)NC2CC(NC(=O)C=Cc3cscn3)C2)ccccc1Cl 67273,c1(-n2ncc(C)c2)cccc(C(=O)NCCNC(c2oc(C(C)C)nc2C)=O)c1 67274,C(CCCCCCC)NC(C(Cc1cc[nH]n1)NC(C1CCC(=C)CC1)=O)=O 67275,c1(C(=O)NC2(CCNC(c3ccc(C)nc3C)=O)CC2)cc(C)cc(C)c1N 67276,C#CCC(CC(=O)NC1CCC(NC(=O)C=CC(C)(C)C)C1)c1ccccc1 67277,C(=O)(CCCC(C)(C)C)N1CC(OC)(CNC(=O)Cn2ncn(C)c2=O)C1 67278,c1(C(=O)NCCN(C(c2c(O)cc(C)nn2)=O)C2CC2)c(C)nc2ccccn12 67279,CCCCC(O)C(=O)N1CCC(C(F)F)(CNC(c2ccc(OC)s2)=O)C1 67280,CC1CCCC(CNC(c2cc(CNC(C3(O)CC3)=O)no2)=O)C1 67281,c1(NC(=O)C(N2CCCCC(CO)C2)=O)cc(N2CCCC2)cc(F)c1 67282,N1(C(CC(C)(C)OC)=O)CC(C)N(C(C2(C)CC3CCC2O3)=O)C(C)C1 67283,C1(C)(CNC(CCc2cn(C)nn2)=O)CCC(NC(=O)COCc2ccnn2C)C1 67284,c1(SC)ccc(Cl)c(NC(=O)C(C)N(C(c2oc(C(F)F)cc2C)=O)C(C)C)c1 67285,c1(OC)cc(OC)cc(CC(C)NCc2cnc(C3CCCCC3)s2)c1 67286,C1(NC(C(c2cccc(Cl)c2)C)=O)CN(C(c2cc(F)n[nH]2)=O)CCC1O 67287,CC1(CO)C=CCN1C(=O)CCC1CCN(C(=O)CN2CC=CC2)C1 67288,c1(CC(N2CCC(C)(CNC(c3cn[nH]c3)=O)C2)=O)cnc(O)nc1O 67289,C1(C)(C=O)CC2C=CC1C2.Cc1cccnc1OCC1CCC(C(=O)NC)CC1 67290,c1(C(=O)NCCCN(C)C(c2csc(Cl)n2)=O)nccc2c1NCCC2 67291,CCC(CC)(CCNC(=O)CN(C)C(C)=O)NC(=O)CC1CCCOC1C(C)C 67292,CCC(F)(F)CC(=O)N1CCCC1CCNC(c1cnn(CCOC)c1)=O 67293,N1(C(C(C(C)C)c2cccnc2)=O)CCOCC(NC(c2cccnc2)=O)C1 67294,C1(C(N2CC(c3ccccc3)(NC(CC(C)OC)=O)C2)=O)CCCCC1(C)C 67295,c1(N2CC(C)C=C(C)C2)nc(N2CCCC3(CCOC3)C2)c2c(n1)CCS2 67296,Cc1nc(C(=O)N(CCCOCCCCOCCN(C(=O)C)C)C)cs1.N(C)(C)CC 67297,c1(C(=O)N(c2ccccc2F)Cc2cccs2)ccc2nc[nH]c2c1F 67298,C1(C(N(CCCC)C(C)CC)=O)CCN(C(=O)CCCc2cccs2)C1 67299,C(C(F)(F)C(C)(C)O)NC(C1(C(C)NC(C2CC3(CSC3)C2)=O)CC1)=O 67300,CC(O)(C(=O)NCC12CC(CNC(=O)CN3CCCNS3(=O)=O)(CO1)C2)C(F)(F)F 67301,CCCCCCCC(=O)NCCCC(C)NC(C1CCCC1CC)=O 67302,CCCCCC(F)C(=O)NC(C)(C)CCNC(=O)Cc1cnn(C)c1C 67303,CN1CCCC2CN(Cc3cccnc3-c3ccccc3Cl)CCC12 67304,N1(C(C(CC)F)=O)C2CCCC1CN(C(c1c([N+](=O)[O-])c(CC)nn1C)=O)CC2 67305,CC1(C)CC(C(N2CC3(CCC3O)C2)=O)CN1C(c1ccco1)=O 67306,CCC(O)C(C)(C)C(=O)NCC(CC(=O)N(CC(C)(CC)OC)C)OC 67307,n1(N2C(C)CC(N)CC2)ncc2cc([N+](=O)[O-])ccc2c1=O 67308,c1(C(=O)NC(C2CCN(C(C(C(C)O)C)=O)CC2)CO)cn2cc(Cl)cnc2n1 67309,C1(COC)(NC(c2[nH]ccc(=O)c2C)=O)CCN(C(C2CC3(CC3)CO2)=O)CC1 67310,C1(C(=O)NCCCC(C)NC(=O)CCC#N)(CO)CCCCO1 67311,Cc1csc(C)c1C(N1CCC(C2CCCN2C(C2CC(n3ccnc3)C2)=O)C1)=O 67312,CC#CCC(C(=O)Nc1cnccc1OC)NC(=O)CCC1CC(OC)C1 67313,O=C(CC=C(Cl)Cl)NC1CCCC1CNC(=O)C=Cc1cc[nH]n1 67314,c1(CN(C)CC2CCC(F)CC2)cc2ccsc2n1C 67315,N1(C(C2C(C)CC(=O)NC2)=O)CCC(NC(=O)CCCS(C)(=O)=O)C12CCC2 67316,N1(C(CCC)=O)CCC(C)C1CNC(=O)CCc1ncc(Br)cn1 67317,C1(C)(C(=O)NCC(C)N(C(=O)CC2CCCC2)CC)CCCC1O 67318,S(=O)(=O)(c1ccc(NCCN2CCC(O)C2)cc1Br)NCc1c(C(C)C)cccc1 67319,c1(OC(C(=O)NC(CNC(Cc2cnn(CC)n2)=O)CO)C)cccc(Cl)c1 67320,C(Cn1cc(-c2c(C)cnn2C)nn1)(C(C)C(C)C)NC(CCCC=C)=O 67321,C#CC1(C(=O)NC(C)Cc2ccncc2)CCN(C(c2cscn2)=O)C1 67322,C1(C(=O)NC2C(CC(=O)NCC(C)N(C)C3CC3)CCC2)CC2CCCC2C1 67323,Cc1ccc(C#CC(=O)NCCC2CCOCO2)cc1 67324,C1(NC(c2cncc(OC)c2)=O)CN(C(C2CCSC2)=O)C2CCCC12 67325,C12(C(N(CC(C)CNC(=O)CC3CC3(Cl)Cl)C)=O)CC(C)(C1)OC2C 67326,O=C(C1=NOC2(CCOC2)C1)N1CCC2CCN(C(=O)C(F)F)CC12 67327,c1(C(=O)NCC2CN(C(Cc3cnc(C)[nH]3)=O)C(C)C2)ccc(Br)c(F)c1 67328,c1(CNC(CSCCC)=O)cnn2c1CN(C(c1[nH]nnc1C)=O)CC2 67329,N1(C(=O)COCC(F)(F)C(F)(F)F)CC(NC(=O)C(F)(F)CO)CCC(O)C1 67330,c1(-c2c(SC)cccc2)nc(=NC2CC(NC(c3cccnc3)=O)C2)s[nH]1 67331,Cc1c(Cl)sc(Cl)c1C(=O)OCCC1C=CCC1 67332,C1(CC(N2CCC(OCC)C2)=O)CC2CCC1CC2.CC(C=CC=O)N(C)C 67333,N1(C(c2c(CNC(c3cc(OCC)n[nH]3)=O)ccs2)=O)CCCC(C(N)=O)C1 67334,C1(C(C)(C)C)(CNC(CC=C=C)=O)CCN(C(=O)CCN2CCNC(=O)C2)C1 67335,c1(N(CCCNC(Cc2c(C)ncnc2C)=O)C2CC2)cc(=O)n(C(C)C)c(O)n1 67336,N1(C(CN(CC)CC)=O)CC(CNC(=O)CCc2ccc(SC)cc2)C2(CC2)C1 67337,N1(C(CC(C)CN(C)C)=O)C2CC1CN(C(=O)COCCc1ccccc1)C2 67338,C1(C(N2CC(C(C)C)OCC2)=O)COCCN(Cc2c(N)c(C)nn2C)C1 67339,CC1CCOC(C(=O)NC2CC3C(NC(=O)C(N4CCOCC4=O)C)C3C2)C1 67340,C1(N(C(=O)C=Cc2nc[nH]n2)C)CCCN(C(c2ccnc(OC(F)F)c2)=O)C1 67341,C1(C(=O)NCC2CCC(C)C2)(OC)CCN(C(=O)C=NOC)C1 67342,N1(C(c2cc(C(F)F)[nH]n2)=O)CC(CNC(C2(CC(F)F)CCC2)=O)CC1(C)C 67343,C(=O)(CCCCN(C)C)NC(CC)CNC(=O)CNC(=O)Nc1ccccc1 67344,N1(C(c2c(COC)nn(C)c2)=O)CCN(C(=O)C(C)C(F)(F)F)C(CCO)C1 67345,N1(C(CC2C(C)CCO2)=O)CC2(C=C(C(=O)N(C)CP(C)(C)=O)CO2)C1 67346,N1(CC(=O)N(C2CCCN(C(C3CNC(=O)N3)=O)C2)C)CCCNC1=O 67347,c1(-c2n(CC=C)nc(-c3ccc(SC)cc3)n2)c(C)cccc1Cl 67348,c1(C(N(CC(O)CNC(=O)C(F)CC2CCCC2)C)=O)ccc(C#N)cc1 67349,C1(NC(C2N(C)CCC2)=O)CC2(CCCCN2C(=O)CCC(N)=O)C1 67350,N1(C(CSCCC)=O)CCC2(CCCN(C(C3CCN(C(N)=O)CC3)=O)C2)C1 67351,CCC(C)C(=O)N(CCCOCCN(C(=O)C(C)(C)c1ccccc1)CC)C 67352,c1(OC)ccc(C(=O)NCC2(C)CCN(C(C3CC(=C4CC4)C3)=O)C2)c(O)c1 67353,C(=O)(C(C(C)(C)O)NC(=O)CC1COCCO1)N(C)CC1(C#N)CC1 67354,N1(C(C)=O)CCOCC1C(=O)NC1CN(C(C2CC(F)(F)CS2)=O)C1 67355,N12C(=O)CCC1CC(=O)NCC2.C(=O)(CP(C)(C)=O)N1CC(CC)(OC)C1 67356,c1ccc2c(c1)nc(CN1CCOC(c3cccnc3)C1)n2CCc1nn[nH]n1 67357,C1(CC(=O)NC(CC=CC)CO)CN(C(=O)CNC(=O)OC)CC1(C)C 67358,N1(C(c2c(OC)ccc(C)c2)=O)CCCCC(CNC(C2CCCC2O)=O)CC1 67359,c1(C(=O)NC2CN(C(c3c(C)snc3)=O)CC2O)cn(CCO)c(=O)nc1O 67360,c1(NC(N(C)C)=O)cccc(C(N2CCOC(C(C)(C)C)C2)=O)n1 67361,S(=O)(=O)(c1cc(F)c(F)cc1F)NC(Cc1ccc(C)c(F)c1)C(=O)O 67362,C1(NC(Cc2n(C(C)C)cnn2)=O)CCC(C)N(C(=O)CC2(C)OCCO2)C1 67363,N1(C(c2cc(CC)[nH]n2)=O)CCC(NC(c2ccc(C(C)C)s2)=O)C(C(C)C)C1 67364,CC1=C(C(=O)N2C(C)CCC2(C)C)C(C)n2nnnc2N1C 67365,CCCCCCC(C)NC(=O)C(C)=CCNC(c1coc(C2CC2)n1)=O 67366,N1(C(CC2CC(OC(C)(C)C)C2)=O)CCCC(CNC(c2n[nH]c(=N)[nH]2)=O)CC1 67367,c1(C(N2CC3CCCN(C(C(C)OC)=O)C3C2)=O)ccc2c(Cl)nccc2c1 67368,C(=O)(CCC(F)(F)C(F)F)NC1CN(C(c2ccn(CCC)n2)=O)CC(O)C1 67369,c1(CC(=O)N(C(CNC(C(C)OCCC=C)=O)C)C)ccc(C)nc1 67370,c1(NC)ccc(C(N2CC(O)(C3CCCN3C(=O)CCOC)C2)=O)cn1 67371,C12(C(=O)NCC3CCCN(C(C(C)S(N)(=O)=O)=O)CC3)CCCCC(F)(C1)C2 67372,c1(C(=O)NC2C(C)N(C(=O)C3=CCCCO3)CCC2)nn2c(c1Br)CCC2 67373,c1(C(N2C(CC(N3CC(C)C(N)C3)=O)CCC2)=O)cc2ccccc2cc1O 67374,C12(C(=O)NCC3CN(C(c4ccc(F)cn4)=O)CC3O)CCC(F)(CC1)CC2 67375,C(=O)(C1CC(=O)c2ccccc21)N(CC(C)C(=O)OC(C)(C)C)C 67376,C1(NC(C2(Cl)C(C(C)=O)C2)=O)C=CC(CC(=O)NCc2cncnc2)C1 67377,c1(OC)ccc(C(N2CC(NC(c3ccc[nH]3)=O)CC(C)C2)=O)c(F)c1 67378,C1(NC(CC(COC)C)=O)CCC2CN(c3cc4nnc(C)n4cn3)CCC2C1 67379,c1(OC)cc(C(=O)Nc2ncccc2CNC(C2CCC2CF)=O)ccn1 67380,C(CC(=O)Nc1cccc(Cl)c1O)(C(C)(C)C)NC(c1cnc(C)o1)=O 67381,CC(C)CC1COC(=O)C1.C1(C(=O)NOC(C)(C)C)CCCC(C)(C)CC1 67382,CCC(O)(C(=O)NCCN(C(=O)CC(C)(O)c1ccccc1)C)c1ccccc1 67383,C(CC(=O)NCC(O)C1CC1)NC(C=C(COC)C)=O 67384,Cc1c(C(N2CCCC(C3CCCN3c3ncccn3)C2)=O)cccc1Cl 67385,CN(C1CCc2c(F)cccc21)C(=O)C(=O)NC12CCCC1CCC2 67386,c1(C(=O)OC)cccc2nc(CCCOC(F)(F)F)cn12.c1(C(=O)O)ncccc1C 67387,N1(C(CC=CO)=O)CCC(NC(=O)CS)C(CO)CC1.C(CC(C)C)N(C(C)=O)C 67388,N1(C(c2ccc(C(C)C)cn2)=O)CC(CNC(=O)CP(C)(C)=O)C2(CCC2)C1 67389,c1(CN(C(c2csc(C(F)(F)F)c2)C(=O)NCCOC)C)ccc(OC)c(Cl)c1 67390,C1(C(=O)NC(c2nc[nH]n2)CC)CCCN1C(=O)CC1CCSC1 67391,N1(C(C2(C)CCC(=O)N2)=O)CCC2CC(NC(c3ccc(F)cc3)=O)CCC2C1 67392,C1(NC(C2CCC(F)(F)CC2)=O)CN(C(C2CC2(Cl)Cl)=O)C2(CCOCC2)C1 67393,c1(C(N(C2CN(C(c3cccc(O)c3)=O)C2)C)=O)ccnn(C)c1=O 67394,C1(NC(C=CC(=O)N(C)C)=O)CCCCC1C(=O)N(C)CCC1CC1 67395,c1(SC(C)C(=O)NCC(C)(O)CNC(c2ccn(C)c2)=O)ccccn1 67396,n1(CC(=O)NCC(N2CCN(C(C3CCC3Br)=O)CC2)C)ncc2ccccc12 67397,N1(C(C2CN(C(c3cc(C(C)C)[nH]n3)=O)CC(F)C2)=O)Cc2ccccc2C1 67398,C1(C(=O)NC2CCCN(C(c3ccc(C(C)C)s3)=O)CC2)CC2(CCCC2)CO1 67399,Nc1cc(Cl)cc(Cl)c1C(N1CCCN(C(C2CCSC2)=O)CC1)=O 67400,CC1CN(C(=O)CSc2ccc(C=O)o2)c2cnccc21 67401,C1(CN(C(=O)CN2CC(=O)NC2=O)C)COCCN1C(C1(C)CC1(F)F)=O 67402,C(=O)(C(C)S(N)(=O)=O)NCC(N1CCN(C(C2COCCN2C=O)=O)CC1)C 67403,N1(C(Cn2ccc(C)n2)=O)CCC12CCCN(C(c1n[nH]c(C)c1C)=O)C2 67404,c1(C(=O)NCCOC2CCN(C(CC(C)SC)=O)CC2)ccc(C)cc1[N+](=O)[O-] 67405,c1(C(=O)NCCCCN(C)C(C2CC(F)C2)=O)cc(N)cc(F)c1 67406,CCC(C)CCCC(=O)N1CC2CCC(C1)N2C(c1cnsn1)=O 67407,c1(Cc2scc(OCC)n2)nc(C)c(C(CC)C(=O)OC)s1 67408,C(=O)(C(CS(=O)(=O)Oc1cccc(OC(F)(F)F)c1)OC)OCCOC 67409,C(C)(CC(=O)NCC1CC(F)CN1C(=O)CCc1ccccc1F)(C(F)F)N(C)C 67410,N1(C(C(C)=CC=C)=O)CCN(CC=CC(N2CCC(N3CCCC3)C2)=O)CC1 67411,N#CC1(C(N2CCC(NC(C3CCCC(C(N)=O)C3)=O)C2)=O)CCCO1 67412,N1(C(C2(OC)CC2)=O)CCC(O)(C2(NC(=O)CC34CCCC3C4)CC2)CC1 67413,CN1CCCCCC1C(=O)Nc1ccc(Oc2cccc(C#N)c2)cc1 67414,c1(C(C)=O)ccnc(CNC(CC2CCCC2)Cc2ccc(F)cc2)c1 67415,C#CC1(C(=O)NCC(C)S(N)(=O)=O)CCN(C(=O)CC2CC2C2CC2)C1 67416,C1(NC(C(=O)NC)C2CCC2)CCOCC1(C)C 67417,C1(CC(=O)NCCCC2N(C(C3CC(=C)C3)=O)CCC2)CCCC12CC2 67418,CC1CN(C(=O)C2=COCC2)CC1CCNC(C1OCCC1c1ccccc1)=O 67419,c1(C(N(CCCCNC(C2COCC(C)O2)=O)C)=O)ccnc(C(F)(F)F)c1F 67420,c1(C(=O)NCC(CC=C)NC(c2cc(C3CC3)nn2C)=O)nnn(C)c1N 67421,N1(CC(=O)NCCC(C)N(C(=O)C=Cc2cscn2)C)CCC(C(F)(F)F)CC1 67422,C12(NC(C(CCCC)OC)=O)CC3CCC(C1C2)N3C(C12CCOC(C)(C1)C2)=O 67423,C1(OC)=CC(C2CCC2)=CC=CC=C1.C(=O)(C(C)NC(C)=O)NC1C(NC=O)C1 67424,Cc1nccn1CC(=O)NNC(=O)NS(=O)(=O)Cc1cc(F)cc(F)c1 67425,c1(C(=O)NC(C)CCNC(=O)C(c2ccc(F)cc2)F)ccc(C#N)nc1 67426,C#Cc1cccc(CC(N2CC3CC(N(C)C(c4cc[nH]n4)=O)C2C3)=O)c1 67427,C1(CNC(CC(C)SC)=O)CCN(C(c2cn(C)[nH]c2=N)=O)C12CC2 67428,c1(SCC)c(OC)ccnc1Br.N12CCCC1C1(O)CN(C1)C(CC)C2=O 67429,N1(Cc2nc(C)sc2C)CCC(NC(c2cccc([N+](=O)[O-])c2)=O)CC(C)(C)C1 67430,C(CCN=C(NC1(C(=O)NC)CCCC1)N1CCSC(C(F)(F)F)C1)OCC 67431,C12(C(=O)NCC(C)CN(C)C(c3conc3C(C)(C)C)=O)CCCCC1C2(F)F 67432,N1(C(C2(C(F)F)CC(=C)C2)=O)CC2(CC(CNC(=O)CCc3nc(C)no3)C2)C1 67433,N1(C(Cc2cc(C)[nH]n2)=O)CC(C)CN(C(c2ccc(N(C)C)nc2)=O)CC1C 67434,C1(C(=O)Nc2ccc(C(c3ccccn3)C(C)C)cc2)CCC(F)(F)CC1 67435,c1(-c2n(CCCC)nc(-c3ccc(OC)nc3)n2)ccc(C)c(C)c1 67436,c1(N2CCN(C(C)=O)CC2)nc(N2CCC3(CCCN3C)C2)nc2c1CSC2 67437,c1(C(N2CC(CNC(Cc3c(C)ncs3)=O)C2)=O)cc(C)c(C)o1 67438,C1(CNC(Cn2ncc(CC)c2)=O)CN(C(=O)CSC(F)F)CCC1C 67439,CC1(C)C(CCN2CC(C)(C(=O)Nc3ccnc(F)n3)C2)CC1O 67440,C(=O)(CC(C)CCC(=O)NC1CCN(C(C23CCCC2C3)=O)CC1)OC(C)(C)C 67441,CCC(C)C(=O)C(=O)N1CC(C(=O)NC2CCN(C3CC3)C2=O)C(F)(F)C1 67442,C1(NC(CCC)=O)(COC)CCCN(C(=O)CC2CCC(F)(F)C2)C1 67443,c1(OCC)ccc(O)c(C(N2CCN(C(=O)Cc3cccc(Cl)n3)CC2C)=O)c1 67444,C(CCN=c1[nH]cnc(C)c1C#N)N(C1CC2CCCC12)CC 67445,C#CCCC(C(=O)N1CCC1c1cn(C(c2cc(F)ccc2OC)C)nn1)N(C)C 67446,c1(CC(N2CCC(F)(C(=O)Nc3cccc(Br)c3)C2)=O)ccc(Br)c(F)c1 67447,C=CCC(CC(=O)N1CCN(C)C(CC)C1)NC(=O)C(C)n1ccnn1 67448,N1(C(C2CCN(C(C3(CCN)CCCC3)=O)C2)=O)CCC(CC(C)O)CC1.COC 67449,C1(C(N(C)CC2CN(C(c3cnn(C)c3N)=O)CCO2)=O)CCN2CCOCC12 67450,C1(NC(C2C(C)OCC2)=O)COC2(C1)CN(C(c1c[nH]c(C#N)c1)=O)C2 67451,N1(C(CNC=O)=O)CCN(C(CNC(=O)CC2CCC(=O)N2)C(F)F)CC1 67452,C1(C(=O)NCCC(C)O)CCCN(C(C2CCN(C)C2=O)=O)CC1 67453,CC1CCCCC1(CNC(=O)COCCN(C)C)NC(=O)C=Cc1cn(C)cn1 67454,Cc1nnc2n1CC(C(=O)NCCCOCCNC(c1ccncn1)=O)C2 67455,C1(NC(c2c(NC(CC)=O)ccc(N3CCCCC3)c2)=O)Cc2ccc(F)cc2C1 67456,C1(NC(CCc2n(C)ccn2)=O)CCCCC1NC(=O)CN1C(=O)CCC1=O 67457,c1(CC)nn(C)c(C(N2C3CCC(C3)C2CNC(C2CC3C=CC2C3)=O)=O)c1Cl 67458,c1(C(=O)NCC(C(=O)NCC(COC)O)C)cnn2ccccc12 67459,N1(C(CC2ON=C(CC)C2)=O)CC(CNC(c2ccc(Cl)cc2)=O)C2(CCC2)C1 67460,C1(COC)(CNC(=O)C=CC(C)C)CCCN1C(=O)CCc1nnc(C(F)F)o1 67461,Cc1ccc(C(=O)NCC2(C)CN(C(C3(C(C)C)CC3)=O)CCO2)cc1[N+](=O)[O-] 67462,c1(C(N2C(C)CC(CNC(=O)CCc3cnn(C)n3)C2)=O)cc2ncccc2o1 67463,N1(C(CNC(C(CC)CC)=O)=O)CCC(NC(c2coc(O)n2)=O)C(C)C1 67464,c1(C(=O)NCCN(C(CCSC)=O)CCCN(C)C)ccn2cc(C3CC3)nc2c1 67465,N1(C(C(CCOC)OC)=O)CCN(C)CC1C(=O)NCc1ccnc(O)c1 67466,c1(C(N2CC(NC(c3cc(COC)cn3C)=O)C2)=O)c(F)c(N)cc(Cl)c1F 67467,C=CC(C)(CCOC)C(=O)N1CC(CNC(=O)CC(O)CCCC)CCC1C 67468,N1(C(Cc2ccn(CC)n2)=O)CCCC(C)(C)C1C(=O)NCC1CCCC1(C)C 67469,CCS(=O)CCNC(=O)CC1(N(C)C(c2cccn2C2CC2)=O)CC1 67470,c1(C(N2C(CC)CCC(C(=O)OC)C2)=O)c(F)cc(I)cc1F 67471,Cc1coc(C(C)C)c1C(=O)NCC(c1cccnc1)NC(=O)C(=O)NC1CC1 67472,N1(C(C(=O)N(C2CCCC2c2ccncc2)C)=O)CCC(NS(C)(=O)=O)CC1 67473,N(C1CCCOc2ccc(Br)cc21)C(CC(CC)(F)F)=O 67474,Cc1[nH]c(=NCCC2CCC(NC(c3cc4ccncc4s3)=O)C2)ccc1C#N 67475,N1(C(C2C(CN(C)C)C2)=O)CCC(=CCNC(=O)CCCCN2CCCC2)CC1 67476,N1(C(c2cc(C)c(C)o2)=O)CC2OCCN(C(=O)CCN3CCCCCC3)C2C1 67477,C1(C(=O)NCC(C(=O)NC2CC(O)C2)O)Cc2nccn2C1 67478,Cn1nnc2c1CCN(c1nnnn1C1CCN(CC3CCCCO3)C1)C2 67479,C1(NC(C(F)=CC)=O)CCN(C(c2ccc(C)cc2C(C)=O)=O)CCC1CO 67480,c1(C(C(=O)OC2CCN(c3ncc(Br)s3)C2)O)ccc(F)c(Br)c1.c1(O)ccccc1 67481,N1(C(c2cnc(OC)s2)=O)CCC(C(C)NC(C2CCCOCC2)=O)CC1 67482,c1(C(=O)NCCCCCN(C(c2ccc(CC)cc2)=O)C)cc2occc2n1C 67483,C1(C(=O)NC(c2ccncn2)C)CN(C(=O)CCC2CCCOC2)C2(CCC2)C1 67484,C(C(=O)N1CC(=O)C(NC(=O)C(C)NCC(=O)NC)C1)(C(C)C)SCC 67485,CC1(C)OC(=O)NC1C(N1CCCOC(CNC(C2(C)CCCO2)=O)C1)=O 67486,CC(CCC(=O)NC1CC1)NC(C1CCCN1C=O)=O 67487,N1(C(Cn2cc[n+](C)c2)=O)CC2CC2(NC(=O)C=C2CCSCC2)C1 67488,C(=O)(C=CS(F)(F)(F)(F)F)NCCN(C(CC(CC)(C)C)=O)C 67489,C1(NC(C2C(C)C2C)=O)CN(C(C2CCC(C(N)=O)C2)=O)C2CCCC12 67490,N(C(=NCCc1cnccn1)N)C(C)C.c1(C2CCCC2)ccc(=N)[nH]c1 67491,C1(CC(=O)NC(C2CCCN2C(=O)CSCC(F)(F)F)C)CCC2CC12 67492,N1(C(C(c2ccc(C)o2)C)=O)C(C)CN(C(C2C3CCC(F)(F)C23)=O)CC1C 67493,C(C)(CCC(F)(F)F)NC(CCN(CCCO)C(c1n(CC)nnc1)=O)=O 67494,c1(NC(C2N(C(C(C#C)(C)C)=O)C3C(C2)C3)=O)c(C(=O)OCC)ccc(Cl)c1Cl 67495,CCN(OC)C(=O)C(C1CCCC1)N(C(c1scc(C)c1C)=O)CC 67496,c1(OC(C)C)ccc(C(=O)NCC2C=CCN2C(=O)C(F)C(C)C)nc1 67497,c1(N(CC(C)C)C(=O)NCC2CCN(CC(C)C)CC2)cc(O)cc(O)c1 67498,C(=O)(C(C)(C)C(C)(F)F)N(C1CC2CCC(C1)N2C(C1CCS1(=O)=O)=O)C 67499,Cc1[nH]ccc(=NC(=O)C2CC3CC3N2C(c2ccno2)=O)c1F 67500,c1(C(N2CC(C)N(C(=O)CC3(C)CCCO3)CCC2)=O)ccc2c(c1)NC(=O)C2 67501,CCCC(C)(C(=O)O)NC(C1CCC(OC)CC1)=O 67502,CC1CN(C(C2CC2F)=O)CC1CNC(=O)C(c1ccccc1)C1CC(F)(F)C1 67503,N1(C(c2ccc(N3CCCC3)cc2)=O)CCN(Cc2ccc(I)c(O)c2)C2CC12 67504,c1(C(N2CCC(N(C(=O)CCn3ccnc3C)CC)C2)=O)cc(Cl)cc(F)c1N 67505,c1(C(=O)Nn2cc(Cl)cn2)cnc(C2CC2)nc1.C12CC(CN1)C(CC)NC2=O 67506,C(=O)(CCCCC(N)=O)NC1CCC(C)N(C(c2cnc3[nH]cnc3c2)=O)C1 67507,C1(CNC(c2ccc(C(C(=O)NCCC)N(C)C)cc2)=O)OCCNC(=O)C1O 67508,C1(NC(c2cc(C(CC)C)no2)=O)CC(CO)N(C(C2CCC(F)(F)C2)=O)C1 67509,c1(CC2C(Cn3cc(C4(NC(C(CC)F)=O)CC4)nn3)C2)nnc(C)n1C 67510,c1(C(N2C(CNC(COCC#C)=O)C=CC2)=O)nn(CC)cc1[N+](=O)[O-] 67511,CC1C(NC(=O)C2=C(Cl)CC2)CCCN1C(C1CCC(C(F)(F)F)O1)=O 67512,N1(C(CNCCNS(C)(=O)=O)=O)CCCC(n2cc(CC3(C)CCC3)nn2)C1 67513,n1(CC(C)C)cc(C(=O)NCCC2CCC(NC(c3cc(CO)c[nH]3)=O)C2)cn1 67514,C(CC(=O)NCC(F)CNC(c1cc(C)ccn1)=O)(C(C)C)OCC 67515,C1(N(C(=O)CCCN2CCCCC2)C)CC2(C1)CC2c1nn[nH]n1 67516,N1(C(c2cnccc2Cl)=O)CCCC12CN(Cc1ccc(Cl)nc1Cl)C2 67517,C1(C(C)C)CN(C(=O)CCCn2ccnc2)CCCN1C(=O)CS(C)(=O)=O 67518,c1(NCCCOCCOC)ccc(S(=O)(=O)NC(C)CCC2CCCC2)c(Cl)c1 67519,c1(C(N(CCNC(c2cnc(C)nc2O)=O)CC)=O)cc(C)c2nc(C)cn2n1 67520,C1(NC(c2c(CCC)n[nH]c2)=O)CCCC(NC(=O)C(C)CC)C1 67521,c1(CNC(CCCCOC)=O)cccc(O)c1C.C12CCCN1C(=O)CC2 67522,N1(C(COC)=O)CCC2(CCN(C(c3ccc(C(=O)OC)s3)=O)CC2)C1 67523,N1(C(C(CC(=C)C)NC(=O)C(F)COC(C)(C)C)=O)CCCC12CCOCC2 67524,O=C(CCCC(F)(F)F)N1CCC(OCCNC(C2C3CCCCC23)=O)C1 67525,CC(O)C(C)(C)CNC(=O)C(c1cccs1)NC(=O)C(O)CCN(C)C 67526,c1(C(N2CC(OCCNC(=O)CCCn3cccn3)C2)=O)ccnnc1Cl 67527,C1(C)(CNC(c2c(CC)noc2)=O)CCN(C(=O)CC2CC2(Cl)Cl)C1 67528,CC(C)(C)C(=O)N1CCCC1C(=O)N(C(Cc1ccccc1)C(=O)O)CC(=O)O 67529,CCCCCCC(C)C(=O)NCCCN(C(c1cn2c(n1)CCC2)=O)C1CC1 67530,c1(C(N2C(CNC(CC=C(C)C)=O)C=CC2)=O)ccc(C)c(S(C)(=O)=O)c1 67531,C1(F)(CNC(CC(CC)SC)=O)COCCN(C(=O)CSc2ccccc2)C1 67532,Cc1cc(Br)cc(Cl)c1NC(=O)NCc1nccn1C 67533,c1(C(=O)NCC(C(=O)OC)CC2CCCN(C)C2)ccc(Cl)c(C)c1 67534,c1(CN2CC(CNC(C3(CC)CC3)=O)C2)cc(Cl)ccc1Cl 67535,N1(C(C(C)CC2CCCC2)=O)CCCCCC(NC(c2cn(C3CC3)nn2)=O)C1 67536,N1(C(C(C2(O)CN(C(CSCCOC)=O)C2)F)=O)CCCCC(N(C)C)C1 67537,C(=O)(CC(C)(C)CNC(c1scc(C)c1C)=O)N1C(C(N)=O)CC(OC)C1 67538,CC1(CNC(C2CCNC2=O)=O)CCN(C(C2SCCCS2)=O)C1 67539,CCC(C)CCCCC(=O)NCCCCCN(C)C(C1(OC)CCC(C)(C)C1)=O 67540,C(=O)(C1=NN(c2ccccc2F)C(=O)CC1)NC(C)CS(C)=O 67541,N1(C(c2c(CC)snn2)=O)Cc2[nH]nc(C(N3C(CC)CCC3C)=O)c2C1 67542,C1(C(N2C(CNC(CCNC(COC)=O)=O)CC(OC)C2)=O)CC2(C1)CC2F 67543,c1(OC)ccc(OC)c(CCC(=O)N2CCC2CNC(C2Cc3nccn3C2)=O)c1 67544,C12(C(N3CC(C(C)NC(=O)Cc4cccs4)C3)=O)CC3CC(C1)C(=O)C(C3)C2 67545,C1(N(C)CC)CN(c2nnc(Cc3cc[nH]n3)n2CC2CC2)CC1C 67546,N1(C(Cc2n(CCC)cnn2)=O)CCCC12CN(C(C13CC(C(=O)OC)(C1)C3)=O)C2 67547,Cc1noc(N)c1C(N1CCC1CNC(=O)CC(O)C1CCCC1)=O 67548,N1(C(CNC(COC(C)=O)=O)=O)CC2CC1CCN2C(c1ncc[nH]1)=O 67549,c1(C(=O)O)cnc(-c2cn(CC(N3CC4(CC4)C3)=O)nn2)cn1 67550,C1(CCNC(CCCC)=O)CCCCN1C(=O)Cc1nc(C(C)OCC)no1 67551,CCC(CC)C(C(=O)N1CCC(C(=O)N(CCCP(C)(C)=O)CC)(CC)CC1)OC 67552,CC1CCN(C(c2ccncc2C(N)=O)=O)CC1NC(C1CC(F)(CO)C1)=O 67553,c1(C(N2CCCC2CCNC(C2CC(O)C2)=O)=O)cc(Cl)c2[nH]c(O)nc2c1 67554,c1(C(N(C)Cc2c(C)cco2)=O)ccnc(CNC(=O)COc2ccsn2)c1 67555,c1(C(c2n(C3(C)CC3)nnn2)NCC2CCC3(CC3)C2)cccc2sccc12 67556,c1(CC(=O)NCCC(C)N(C(=O)CSCc2nccn2C)C)ncc(Cl)s1 67557,c1(NC(=O)C(N2CC(O)(NCCCSC(F)(F)F)C2)=O)cc(F)ccc1F 67558,c1(C(=O)NCC(COC)NC(C)=O)cnn(C)c1S(C)(=O)=O 67559,C1(C(=O)NC2(C)CN(C(=O)CO)C2)C2Cc3ccccc3C12 67560,c1(OC)noc(C(=O)NCCOCC(=O)O)c1Br.n12cc(nn1)COCC2 67561,CC(CC(=O)NC1COCC1C(=O)NCC1CCCSC1)N(C)C 67562,CCCC(CCC)C(=O)N(C1CCN(C(C2(CCOC)CCCC2)=O)C1)C 67563,c1(OC)ccc(C(N2CCC(NC(=O)C(O)CSC)C2(C)C)=O)cc1OC(F)F 67564,c1(C(N2CCC(NC(C(CC)=CC)=O)CC2C)=O)cc2c(cc1OC)OCO2 67565,C1(NC(c2n(CCN(C)C)ccc2)=O)CN(C(c2cnn(C)c2)=O)C(C)(C)C1 67566,CC(C)C(C)(O)CNC(c1sccc1CNC(=O)C=Cc1cccnc1)=O 67567,Cc1nc2c(s1)CCCC2COC.C1(C(C)(C)C)C(=O)N2CCC2c2cn1nn2 67568,C1(C(=O)NCCCN(CCCNC(c2ccc(F)s2)=O)C)CCCCC12CC2(F)F 67569,C#Cc1cn(C)nc1C(N1CCC1CNC(c1cccc(O)c1C)=O)=O 67570,c1(C(=O)NC(CNC(c2c[nH]c(=NC)o2)=O)C)cc(-c2ccccc2)cnc1O 67571,n1(CC(N2CC(C)(NC(C(F)=C(C)C)=O)C2)=O)cc(C)c(O)nc1=O 67572,C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C(=O)NCC(CC(C)O)(C)C)(C)CO 67573,C(=O)(CCCCC(C)C)N1C(CNC(=O)Cc2cnsc2)CC(COC)C1 67574,N1(Cc2ccc(SCC)s2)CCN(C(=O)C(c2nnc(C)n2C)(F)F)CC12CC2 67575,C1(NC(CNC(C(COC)C)=O)=O)CCN(C(=O)COCC(C)C)C12CCCC2 67576,C=CC1CCCN(C(=O)CC2(N(C)C(c3ccc(C#N)[nH]3)=O)CC2)C1 67577,CCCCC(C)(F)C(=O)N1CC(CC(F)C(=O)Nc2cn(CCOC)nn2)C1 67578,N1(C(c2ccc(CSC)o2)=O)CC(C(=O)NCC(c2ccccn2)C)C2(CC2)C1 67579,Cc1cc(N(C(=O)CC2(NC(c3cnc(S)nc3)=O)CC2)C)cc(C)c1 67580,c1(C(N2CC(CNC(C3CC(O)C3)=O)C(O)C2)=O)cc(F)c(CO)c(F)c1 67581,C=CCC(CC)C(=O)NCCC(O)CNC(C1CC(=O)CC(=O)N1)=O 67582,C12CC3CC(CC13)C(=O)N2.Cc1ccc(C)n1CC(=O)O 67583,CCCC(CC(=O)NC(C)(C)C(=O)NC)NC(c1ccc(F)s1)=O 67584,n1(CC(=O)NC2C(NC(C(F)OC)=O)C2)nnc(-c2ccccc2)n1 67585,CC(Cc1cnc[nH]1)C(=O)N(C1CCN(C(C2CC(F)(F)C2)=O)C1)C 67586,c1(OC)ccc(CN(C2CN(C(=O)CC(C)(C)CN(C)C)C2)C)cc1F 67587,c1(C(=O)NCCCN(C(C(C)OCCC#C)=O)C)c(OC)ccc(F)c1Br 67588,CC1(C)OCCC1C(N1CC(OC2CC2)C1)=O.C12CCN(CC1)C(=O)C(=O)N2 67589,c1(C(N(CCCNC(=O)CC2(C)CC2F)CC)=O)cnc(CO)nc1O 67590,N1(C(c2c(SC)cccc2)=O)CCCC(C)C1CNC(=O)CC1CC(F)(F)C1 67591,C1(CNC(c2nc(CCC)sc2)=O)CN(C(c2nocc2Cl)=O)CCC12CCC2 67592,C1(C(=O)NCC=CCNC(COC(C)C)=O)CCCC(C2CC2)O1 67593,N1(C(c2c(OC)n[nH]c2)=O)CCOC(C(N2CCCC(O)(C(N)=O)C2)=O)CC1 67594,c1(C(N2CCN(CCOC)CC2)=O)cccc(C)c1O.C12CC1NC2=O 67595,C(CC(=O)NC1CC=CCC1)(C(F)(F)F)NC(C1(CCC=C)CC1)=O 67596,C(C1CCCN1C)=CC(=O)NCC(C)C(=O)N1CCCCC1.N12CCC(C1)C2=O 67597,c1(C(N2CCC3CN(C(C4CCCO4)=O)CCC23)=O)ccc2ccc(Br)cc2n1 67598,N1(C(C2C(C)OCC2)=O)CCC(CNC(C2(c3ccno3)CC2)=O)C(O)C1 67599,C(CCCC(=O)N1CCOC(CCO)C1)NC(C(C=C)O)=O 67600,c1(CC(=O)NC2C(CNC(c3[nH]cc(CC)c3)=O)C2)ccnc(F)c1F 67601,C1(CNC(c2cc(CF)on2)=O)CCC(NC(C2CCS2(=O)=O)=O)C1 67602,c1(C(CC(=O)O)NC(c2cccn(COC)c2=O)=O)cccc(Cl)c1Cl 67603,S(=O)(=O)(c1cccs1)NC(C)C(N1CCOC(C(=O)NC2CC(N(C)C)C2)C1)=O 67604,C1(CNC(Cc2scc(C)n2)=O)CN(C(=O)C(F)(F)C(F)F)CCC1(C)C 67605,C1(OC)COCCC1CC(=O)NCC(C)(C)CNC(c1scc(C)c1Cl)=O 67606,C1(NC(COC(C)(C)C)=O)COC2(C1)CN(C(c1ccc3c(c1)COC3)=O)C2 67607,CC(CN(C)C)CC(=O)N(CCCC(=O)NC1CC(=O)N(C(C)C)C1)C 67608,C1(NC(c2ccc(Cl)o2)=O)C2CN(C(=O)Cc3ccccn3)CC12 67609,c1c2ccc(cc2)c1.c1(CC)nocc1C(=O)NC1CCN(S(=O)(=O)CC)C1 67610,N1(C(CN(CCCCCC)C)=O)CC2CC1C2CNC(=O)CC(C)(C)O 67611,c1(OCC)nc(C(=O)NC2(C(=O)NC3CC(C(N)=O)C3)CC2(C)C)co1 67612,CC(C)C(CNC(c1ccnn1C)=O)NC(c1cc(-c2ccco2)[nH]n1)=O 67613,N1(C(C2=CC(C)(CC)C2)=O)Cc2ccccc2C(NC(C2(F)CCCC2)=O)C1 67614,CC1CN(C2CCCN(c3ccccc3OC(F)F)C2=O)S(=O)(=O)C1 67615,N(C)(C1=CCC2CC2C1)C(C1CN(C(c2cn(CC)nc2)=O)CC12CC2)=O 67616,C1(C(N2C(C)(CCC)CC2)=O)CCCN(C(=O)C(C)(F)c2ccon2)C1 67617,c1(C(N(CC(C)N(C)C(C2CC2C(F)F)=O)C)=O)ccc2c(c1)C(=O)CCS2 67618,C1(C2CC2)(CNC(CC2C(C)(C)CO2)=O)CCN(C(c2ccc(Cl)cc2O)=O)C1 67619,C1(NC(c2ccn(CCCC)n2)=O)CN(C(=O)CCn2cccnc2=O)CC1O 67620,c1(C(N2CC(O)CC2C2CC2)C(=O)NCCCSC)ccccc1Br 67621,c1(CN2C(CNC(c3nc(C(F)(F)F)ccc3Br)=O)CCC2)ccc(Br)cc1O 67622,C12(CNC(C3C(C=C)CC3)=O)CCC(CC1)N(C(C1(n3ccnc3)CCCC1)=O)C2 67623,C(=O)(CC1CCc2ccccc21)NC1CC(CNC(c2cc(C)nc(O)c2)=O)C1 67624,C1(C(=O)NCCF)CC2CC2N1C(C1C=CCC1)=O 67625,c1(C(=O)NC2C(NC(C3(CCC)CC3)=O)C2)cccc(Br)c1 67626,C(=O)(CCP(C)(C)=O)NC(C(=O)NC(c1cncn1C)CC)CC1CCC1 67627,c1(NC(c2n(C)ncc2Cl)=O)ncnc(Cl)c1CO.C12CCCCC1NCC2 67628,N1(C(C=CCC=C)CCCC)CCN(C(=O)CNS(C)(=O)=O)CC1CC=CCl 67629,c1(NC2C(NC(C(C)SCC)=O)CCCC2)ncnc2cnccc12 67630,c1(C(N(CCO)Cc2ccc(C)o2)=O)ccc(-c2nn[nH]n2)nc1 67631,C1(CC=C)(NC(=O)C(c2cccc(Cl)c2)O)CCCN(C(c2cocc2C)=O)C1 67632,C1(C(=O)NC2(C)N(C(C34OCC(C)(C3)C4)=O)CCC2)CC2CCC(C1)N2C1CC1 67633,c1(N2C(CN(C)C(C3CCCN3C)=O)CCC2)ncccc1S(C)(=O)=O 67634,Cc1nccc(C(N2CCCC(N(C)C(C3CCC(=O)N3)=O)CC2)=O)c1N 67635,C(C(=O)NC)(C(C)OC)NC1C(NC(CNS(CCC)(=O)=O)=O)CCC1 67636,c1(C(=O)NCC2CC(O)(CNC(C(C(C)C)O)=O)C2)cscc1S(C)(=O)=O 67637,C(C)(C(C)(C)C(=O)NC1C(C)(C)C1(C)C)NC(c1ccc(CC)[nH]1)=O 67638,N1(C(c2c(C)snc2)=O)CCC2CCN(C(c3cc4n(c3)CCCC4)=O)C2C1 67639,CC1Cc2cccc(C(N3CC4(NC(c5cncc(Cl)c5)=O)CC3C4)=O)c2O1 67640,C1(C(=O)NCC(C)N(C)C(c2ccc(OCCF)nc2)=O)CC(O)CN1C 67641,C1(NC(C2CC2Cc2ccccc2)=O)C=CCN(C(=O)C2=COCC2)C1 67642,C(CN=c1[nH]c(=NC(C)c2cc(C)on2)[nH]c2c1SCC2)SCCOC 67643,CCC(O)CC(=O)N1CC(NC(=O)C(C)Oc2cccc(C(F)(F)F)c2)C1 67644,N1(C(c2n[nH]c(C)c2C)=O)CCCC12CCCN(C(C1CCCCC1(F)F)=O)C2 67645,C1(NC(c2c(C)nc(N(C)C)s2)=O)CN(C(=O)C=CC(=O)N(C)C)CC1C1CC1 67646,C(=O)(CCC(C)(C)c1ccccc1)N(C1CCCC(O)C1)C 67647,c1(C(N2C(C)CN(C(CSCCC)=O)C(C)C2)=O)cnc(O)c([N+](=O)[O-])c1 67648,C(=O)(C1=CC(O)C(Nc2nc(N3CCS(=O)CC(C)C3)cc(C)n2)C1)OC 67649,c1(C(=O)NC(CCNC(CCSC)=O)(C)C)cn(C)c(-c2ccccn2)n1 67650,C(CC(=O)NC(C1CC(O)C1)C)N(C(=O)COCCCOC)CC 67651,N=c1nc2c(C(N3CCC(CNC(C4CC=CCC4)=O)C34CC4)=O)cccn2[nH]1 67652,N1(C(c2c(SC)ccs2)=O)CC(NC(c2ccn3c2CCCC3)=O)C2(CCC2)C1 67653,CCS(=O)C1CCCC(NC(=O)C(=O)Nc2cc3ccccc3n2C)C1 67654,N1(C(CCC#CC)=O)CCN(C(=O)C=CC(F)(F)F)CC2CCCCC12 67655,N1(C(c2cn(CC=C)nc2)=O)CCC2(CCN(C(=O)C(F)=C3CCCC3)C2)C1 67656,C1(C(=O)NC(CC(=O)NC)C)CN(C(c2sccc2CO)=O)CC12CCC2 67657,C(=O)(C(F)(F)c1ncc[nH]1)NC(C1CCN(C(c2c[nH]nc2C2CC2)=O)C1)C 67658,c1(CN2CC(n3cc(Nc4c(F)cccc4)nn3)C2)ccc(Br)c(Cl)c1F 67659,c1(C(=O)NCC(CC(=O)NCC2CC(C)(O)C2)OC)cccc(C)c1O 67660,c1(CCCn2cc(C(CC)NC(C3(C)CNC(=O)C3)=O)nn2)cc(F)ccc1F 67661,C1(C(=O)NC(C(=O)NCC(C(C)C)(C)F)CC2CCC2)CC2(CCC2O)C1 67662,C(=O)(CC1=CCCCC1)N1CC(C)CC(NC(C2N(CCC)CCC2)=O)C1 67663,N#Cc1ccc(CN2CC3CN(C(c4ccn(C(F)(F)F)n4)=O)CC3C2)c(Br)c1 67664,c1(C(N(C2CCN(C(C3CC3(F)Cl)=O)CC2)CC)=O)cc(Cl)cc(Cl)c1N 67665,C1(NC(c2scc(OC)c2)=O)CC2(C1)CN(C(c1ccn(CCOC)n1)=O)C2 67666,c1(C(N2C3(CNC(c4ccnc(O)c4)=O)CCC3CC2)=O)cnc2nccn2c1 67667,C(C(C(=O)N(C)CC1(F)CCCC1)N(C)C)NC(C(C)n1cccn1)=O 67668,c1(C(=O)NCc2c(C([N+]3([O-])CCC(C)(C)C3)=O)c[nH]n2)n[nH]c2ccccc12 67669,CC1CCC(NC(c2nc(Cl)ccc2F)=O)CN1c1ncccc1F 67670,CCCCCCC(CC)(CC)C(=O)NCC1CCCN1C(=O)C(F)C(C)(F)F 67671,N1(C(c2ncn(CCNC(C3CC(C(C)C)C3)=O)c2)=O)CC(S(N)(=O)=O)C1 67672,CC(=O)N1C(=O)CSc2cc(C(=O)NCC(c3ccc(F)cc3)O)ccc21 67673,c1(C(=O)NCC(CNC(c2nc(C)sc2C)=O)C)cc(N)cc(O)c1C 67674,C(=O)(C1=Cc2ccc(Cl)cc2OC1)NCCNC(C12CCC(=O)CC1CCC2)=O 67675,c1(NC2(c3n(CCOC)nnn3)CCOC(SC)C2)ccc2c(c1)CCNC2=O 67676,C(=O)(CC(O)CC(C)(C)C)N(C)CC1(O)CCN(C(C(C=C)(C)C)=O)CC1 67677,C(=O)(Nn1cnnc1C)C1N(CCC)CCCC1.C1CCC(=O)O1 67678,CCC(C)CCCCC(=O)NC(C)(CNC(=O)CNC1CC2CCC1C2)C1CC1 67679,C1(C(=O)NCC(C)Cn2ccnc2)CC(=O)CN1C(C1OCCC1(C)C)=O 67680,N1(C(CCCOCCC)=O)CCC(CNC(=O)CCCN=[N+]=[N-])C(C)C1 67681,c1(CC(=O)OC)cn(C)nc1C(F)(F)F.C(C(C)C(C)C)CCC(=O)N1CC1(C)C 67682,N1(C(CSCC#C)=O)CC2CC(NC(C3CN4CCN3CC4)=O)C(C2)C1 67683,c1(-n2cc(CNC(CC=C)Cc3ccccc3)nn2)cc(C(F)(F)F)ccc1Cl 67684,C1(C)(C(=O)NCC2(COC)CCN(C(=O)CC3CCC(=O)N3)C2)CCC(=O)CC1 67685,C(=O)(CC(C(F)F)NC(=O)Cc1ccns1)NCC(C)SC 67686,Cc1ccc(-c2cc(C(=O)NCCCCC(C)NC(=O)CC(C)(C)F)on2)cc1 67687,c1(OCCC=C)cccc(CC(=O)NCC2CC2CNC(=O)CCOC)c1 67688,Cn1cncc1CC(N1CC(O)(C(C)(C)CNC(C2CC2F)=O)C1)=O 67689,c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)CC2C)cncn(C)c1=O 67690,C1(C(=O)NC(CC)(C)CNC(=O)CSCC(C)C)CCN(C2CC2)S1(=O)=O 67691,c1(C(=O)NCC(CNC(C(F)=C(C)C)=O)(C)O)c[nH]nc1[N+](=O)[O-] 67692,CCCC(C)(C)C(=O)NC1CCCC(CC(=O)NC2(C(=O)N(C)C)CC2)C1 67693,c1(C(CNC(c2c(C)snc2)=O)NC(=O)CC2CC(C)(C)C2)ccc(F)cc1F 67694,Cc1cc(C(N2CCCC2c2nc(-c3ccccn3)cs2)=O)c(C)n1C(C)C 67695,CC(C)C(F)C(=O)NCC12CC1CN(C(=O)Cn1cnc(Br)c1)C2 67696,N1(C(C2(CCC)CC2)=O)CCN(C(C2C=CCC2)=O)C(Cc2ccccc2F)C1 67697,c1(CN(CC2CCC(CC)O2)CC2CC2)ccc(SC)nc1 67698,C1(NC(C(C(C)C)c2cccnc2)=O)CCN(C(c2n[nH]cc2F)=O)CC(O)C1 67699,C1(C(=O)NCCCCNC(=O)C(C)OCCOCCO)(CC)CCCC1 67700,C(=O)(C#Cc1ccc(Cl)cc1)N1CCC(C#N)(C#N)CC1 67701,c1(OC)cc(C)c(CN2CC(C(=O)NCC3CCCO3)CC2CO)cc1OC 67702,C1(NC(=O)Cc2cnoc2)CCC2CCN(C(c3coc(Br)c3)=O)C12 67703,CC1=C(CNC(C2CN(CC(F)F)C2)=O)SCCO1 67704,c1(CC)cc(C)ccc1C(=O)NC(C)CC(C)NC(=O)Cc1ccsc1Cl 67705,c1(C(=O)NCC2C(CNC(C(C)N3CCC3)=O)C2)ccc(O)cc1[N+](=O)[O-] 67706,N1(C(Cn2c(C)nnn2)=O)CCN(C(=O)COc2ccc(O)cc2)C(CCO)C1 67707,C1(C(=O)NCC(=O)OCCCC)CC(O)CN1C(c1ccn(C(F)F)n1)=O 67708,C(=O)(C(C)(c1ccccc1)NC(=O)C1CC1)NCC(C)NC(c1n[nH]cc1Cl)=O 67709,N1(c2cccc(OC)c2)C(=S)NC(c2cn(C(C)C)nn2)C2=C1CCN(C)C2=O 67710,CC1CN(C(=O)CCCN(C)C(C)C)CC1(C)CNC(c1ccc(CF)cc1)=O 67711,C12(OCC)CCC(C(N3CCC(CF)(NC(=O)CSCC(N)=O)C3)=O)(CC1)C2 67712,N1(C(CC(C)C2CC2)=O)CC(=O)NCC1C(N1CC=CC(O)C1)=O 67713,N1(C(C2C=C(C)CS2)=O)CCCC12CCCN(C(C1CCCCC1O)=O)C2 67714,c1(C(N2CCC(CCNC(CC(C)SC)=O)CC2)=O)n[nH]c2c1CCCCC2 67715,c12ccc(cc1)c(=O)[nH]2.c1(CC(=O)N(CCCC)C)cnn(C(C)C)c1 67716,C1(CNC(=O)C=CI)C2CCCC1N(C(C1C3CC4C(C3)C14)=O)C2 67717,c1(CC(=O)N(C2CCN(C(=O)CN3CCC3C)CC2)CCC)ccc(O)c(F)c1 67718,C12(NC(CN3CCN(C(C(C)(C)C4CCCO4)=O)CC3)=O)CC1COC2(C)C 67719,Cc1nn2cc(C(=O)NCC3CN(C(=O)C(O)CN4CCCC4)C(C)(C)C3)nc2s1 67720,C1(O)(CC)CCN(C(C2C(NC(=O)Cc3cc[nH]c3)C2(C)C)=O)CC1 67721,C1(C(N2CC(C(C)C)C2)=O)CCN(C(C2CC23CCOCC3)=O)C12CCC2 67722,C1(NC(=O)OC)CCCN(C(=O)Nc2cc(C)oc2C)C1.N12CCCC1C2=O 67723,C(CC(=O)NCCS(C)(=N)=O)(CC(C)C)NC(c1c(C)cc(C)nc1)=O 67724,C(=O)(CC(C)C(C)(C)C)NC(C(N1CCC(F)(C(C)C)CC1)=O)Cc1cc[nH]n1 67725,C=CCC(CC)C(=O)NCC1(C(C)(C)C)CCN(C(=O)CC2(O)CCCOC2)C1 67726,c1(C(=O)NCC2(C)CCC(NC(C=C(C)C(C)C)=O)C2)ccc2cc[nH]c2n1 67727,CCC(C(=O)N(CCNC(c1cc(O)cs1)=O)CCc1ccccc1)OC 67728,C(=O)(C(C)(C)N(C)C)N1C(C(N(C(C=C)C2CC2)C)=O)CC1 67729,N1(C(C2C(C)CC2)=O)CCC(n2cccn2)(CNC(C2CC(CF)C2)=O)CC1 67730,N1(C(CC2CC(OCC)C2)=O)CC(NC(=O)Cn2cc([N+](=O)[O-])cn2)C2(CC2)C1 67731,C1(CNC(C=CC(C)NC(C=CC(C)(C)SC)=O)=O)CCOC(C)C1 67732,C(=O)(C1=CC2(CCOC2)C1)NC(C(C)NC(C(=O)Nc1ccc(C)cc1)=O)CO 67733,N1(Cc2c(Br)ccc(OC)c2)CC2CCNC2C1.c1(C(=O)OC)cc(CO)cc(Br)c1 67734,c1(C(N2C(C)CCC(NC(c3csc(C#N)c3)=O)C2)=O)ccn2nccc2c1 67735,c1(OC)cc(OC)c(N)c(C(N2CCC(CCNC(c3ncccn3)=O)C2)=O)c1 67736,C1(C(C)C)CN(C(=O)C(C2CCCN(C(c3sccc3Cl)=O)C2)(C)C)CCCO1 67737,Cc1cnc(C)c(C(=O)NCCC(C)CCNC(=O)C(N2CCC(O)CC2)C)c1 67738,N1(C(C)=O)CCCN(C(c2ccc(-c3csc(C)n3)s2)=O)CC1 67739,Cc1ccncc1C(N1CCC(C(=O)NCC(N2CCC(CO)CC2)=O)C1)=O 67740,c1(OC)ccc2c(c1)OCC(C(=O)NC(CNC(c1ccc(C)s1)=O)CO)C2 67741,CC(C)CN=C(NCc1cccnc1-n1cccn1)N1CCC(C)C1 67742,n1(CCC(=O)N(C(C)CNC(=O)Cc2cnsc2)C)cnccc1=O 67743,c1(C(N(CCCCN(C(CSCC)=O)C)C)=O)cc(N)ccc1S(C)(=O)=O 67744,CCC(C(=O)NCC1(NC(=O)CNc2cccnc2)CC1)C(C)C 67745,C1(CC(=O)N(CCCC#C)C)N(C(=O)C2=C(C)OCC2)CCC1(C)C 67746,C(=O)(CCC(C)(C)C#N)NCC=CCNC(c1nc(C)sc1)=O 67747,c1(CC)ccc(C(=O)NC(CN(C)C(C2CC2(Cl)Cl)=O)CC)cc1[N+](=O)[O-] 67748,c1(OC)cccc2c1C(C(=O)NCC(O)CNC(=O)CSc1nnc(S)s1)CC2 67749,CC(C(=O)N1CC(=C(F)CNC(=O)C=Cc2cnc(C(C)(C)C)s2)C1)S(N)(=O)=O 67750,C(=O)(CCCCC(OC)OC)N(CCNC(C(c1ccc(Cl)c(Cl)c1)CC)=O)C 67751,CC1(C(=O)NCC2CCN2C(C2CCCCS2)=O)CC2(CCC2)C1 67752,O=C1CCC(O)CN1CCN1CCCC(C(=O)NCCO)CC1 67753,CCC(C)CC(C(=O)NCCn1cccnc1=O)NC(c1cnc2n1CCC2)=O 67754,C(N=c1[nH]cnc(Cl)c1Br)C1(CNC(CCCC(C)C)=O)CC12CCC2 67755,C12(NC(c3ccccc3)=O)CCCN(C(c3cc4cccnc4[nH]3)=O)CC1C2 67756,N1(C(C(c2ccc(Cl)cc2Cl)C)=O)CCC12CN(C(=O)Cc1nncn1C)C2 67757,CC(C)CC(O)CC(=O)NCC1(O)CC(CNC(c2ncn(C(C)(C)C)n2)=O)C1 67758,C1(C(=O)NCC(C)(C)NC(=O)CSCC(N)=O)CC2(C1)CC21CCC1 67759,N1(C(C(C(C)C)O)=O)CC2(C1)SCCC2NC(c1ccc(-n2cncn2)nc1)=O 67760,C1(C(N(C)CC2(CNC(=O)Cc3sccc3Cl)CC2)=O)(N(C)C)CCCCC1C 67761,CCC(C(=O)NCCCOCCCNC(=O)C(C1CCCCC1)OC)OC 67762,C1(CNC(=O)CCN2CCCC2)CC(O)CN1C(=O)Cc1ccno1 67763,C1(C(=O)NCC(CCCC)NC(=O)C(CCC)N(C)C)CCCCC12OCCO2 67764,CCC(O)C(=O)NCC1CCN(C(=O)CCSCCC(=O)OC(C)(C)C)C1 67765,C(=O)(C(C)CN(C)C)N1CC(C(C)NC(c2cnn(CC(F)F)c2)=O)C1 67766,c1(CC(=O)NCC(C)NC(c2c(CCC)n[nH]c2)=O)ccnc(C(=O)NC)c1 67767,N1(C(Cc2cnn(C)n2)=O)CCC2CCCN(C(=O)C=CC3CCC3)C2C1 67768,N12CCC(C3(CC3)C1=O)CC2.C12(CN3CC(C=C)COCC3)CCOC(C)(C1)C2.OCC 67769,C=C(C)C1OCCC1N=c1nc2c(ncn2C)c(NCC2CCCC2)[nH]1 67770,c1(C(=O)NCC(c2ccccc2F)NC(CC=C=C)=O)cn(C)nc1C(F)F 67771,c1(OC)ccc(C(=O)NC2CC2CNC(=O)Cc2sccc2Cl)nc1OC 67772,C=C1CCN(C(c2cccs2)=O)C(C(=O)NCc2cc(C)ccc2O)C1 67773,C#CCC(C)C(=O)NC(CN(C)C(c1cn(-c2cccc(F)c2)nc1C)=O)CC 67774,c1(OC)cc(Cl)ccc1C(N1CCN(C)C(CNC(=O)C(C)(O)COC)C1)=O 67775,c1(C(=O)NCCCNC(CN(CCCC)C2CC2)=O)cc([N+](=O)[O-])c(NC)cc1O 67776,C#CCC(O)C(=O)N1CC(C(=O)NCCc2ccn(C)n2)C(CC)C1 67777,CCCCC(CC(=O)NCC(C)(O)C(C)CC)NC(c1ccccn1)=O 67778,C1(O)(CNC(=O)CCCn2ccnn2)CCCN(C(c2cc(O)nc(O)n2)=O)C1 67779,N1(C(C2CC=C(C)CC2)=O)CCCC(O)(CNC(c2c[nH]c(=N)nc2C)=O)C1 67780,c1(CCC(N2CC(N(C(CC=C=C)=O)C)C(O)C2)=O)ccc(F)cc1Br 67781,c1(C(=O)NCCC(C)CCNC(=O)COCP(C)(C)=O)cc(Cl)c(F)cc1O 67782,c1(C(N2CCCC(NC(c3c(OC)oc(C)n3)=O)C2)=O)c(C)cc(C)cc1C 67783,CC1(CNC(c2cc(C#N)c[nH]2)=O)COCCN(C(=O)CN2CSCCSC2)C1 67784,c1(C(C(=O)NC2COC2)N(C(CC)C(=O)OC)C)cnc2ccnn2c1 67785,c1(C(=O)NC(C(C)C)CNC(=O)Cc2ccccc2F)ccc2[nH]ccc2n1 67786,CC1(C)CCCCC1(C)NC(C1CCCN1C(=O)CSc1nc[nH]n1)=O 67787,C1(C(N2CCC(NC(c3c(C)nn(C)c3)=O)C(C)C2)=O)CCC(C2CCCO2)O1 67788,C1(NC(COc2c(CC)cccc2)=O)CCN(C(=O)CCC2CCOC2)CC1C 67789,C1(c2n(C(CC)C)nnn2)(NCC2(COC)CCCO2)COCCOC1 67790,c1(C(N(CC(CNC(CCC2CC(C)C2)=O)O)C)=O)ccc(=O)n(C)n1 67791,Cn1[nH]c(=NC(=O)C2CC23CCN(C(c2cc([N+](=O)[O-])ccn2)=O)C3)s1 67792,C1(NC(Cc2scc(C)n2)=O)CC(NC(=O)Cc2ccnn2C)C12CCOCC2 67793,c1(C(=O)NC(c2ccccc2F)CNC(=O)CCC2CCC2)ccc([N+](=O)[O-])o1 67794,N1(C(CCC2(C)CC2(F)F)=O)CCC12CCNC2=O 67795,c1(C(C(C)C)N(C(c2cccc(Cl)c2)C(=O)NCC)C)ccccc1I 67796,C1(C2CCN(C(=O)Cc3cccnc3N)C2)(NC(c2c(C)ncs2)=O)CC1 67797,C1(C)(C(=O)NC2CC(OC(C)C)C2)CCCN(C(c2cc(C3(C)CC3)on2)=O)C1 67798,Cc1ccc(C(CNC(C2CCC(C)O2)=O)NC(C2(F)CC2)=O)c(Br)c1 67799,C1(CC(=O)N(CCCC(=O)OC)CCC=C)CC2(CC2)CN1C(c1cscn1)=O 67800,C(N=c1[nH]c(N2CCC3CC3C2)nc(=N)[nH]1)C1(SC)CC1 67801,C(=O)(C1=Cc2ccccc2C1)NC1C2(CCN(C(CCCCSC)=O)C2)C1 67802,C(c1ccc(C(F)(F)F)cc1)=C(C(=O)NCC12CC(NC(C(C=C)O)=O)(C1)C2)F 67803,C(=O)(C1CCCc2ncccc21)N1CC=C(CNC(c2cc(Cl)no2)=O)CC1 67804,C1(NC(c2occ3c2CCCC3)=O)CCN(C(C2CC=CCO2)=O)CCC1(F)F 67805,N1(C(C(C(C)C)OC)=O)CC(CN=c2cc(Cl)nc[nH]2)C2(CCOCC2)C1 67806,C=CCC(C)(C)CC(=O)N1CCN(C(c2cn(CO)nn2)=O)CC1CC(F)(F)F 67807,C(N=c1[nH]c(=NCCC2CCC2)c2ncccc2[nH]1)c1cccc(CC(F)(F)F)c1 67808,CC1(C(=O)NCCNC2CCCC2)CCN(C(=O)C2=CCCSC2)CC1 67809,C1(CCC)CN(C(=O)CC(C)(C)SC)CCN1C(=O)CC1C=CCCC1 67810,N1(C(COCCOCC)=O)C2CCC(NC(=O)CC(C)(O)C3CC3)CC1C2 67811,C1(CN(C(C(CC)C)=O)C)CCCN(C(C2CC3(COC3)C2)=O)C1 67812,C(CC)(C(=O)NC(C)CN(c1ccc(CC(C)C)s1)CC)OCC 67813,N1(C(CC(CC#C)NC(=O)C(C#N)C(C)C)=O)CCn2nccc2C1 67814,N#Cc1ccccc1C=CC(N1CC(NC(=O)CCc2ncc[nH]2)C(O)C1)=O 67815,Cn1nc2c(c1NC(C1CSCCN1Cc1cc(F)ccc1F)=O)CCC2 67816,N1(C(C(C2CCC2)OC)=O)CC(O)(C2(CNC(C3CCCO3)=O)CC2)C1 67817,C(=O)(C1=CC(C)(CC)C1)NCC(CN(C(=O)Cn1cc(C)cn1)CC)(C)C 67818,C1(C(=O)NC(C)C(C)(C)NC(=O)CCc2ccnc(Cl)c2)CCCC1C1CC1 67819,C1(O)(CCNC(c2nc(N(C)C)oc2)=O)CCN(C(C2CCCOCC2)=O)CC1 67820,C1(CNC(CC(C=C)CC)=O)CC2CCC1N(C(c1cnn[nH]1)=O)C2 67821,C(=O)(CCCC(F)F)N1CC2C(N(C(=O)CCCN3C(=O)CCC3=O)C)C2C1 67822,C1(NC(CC2C(C)(C)N(C(c3cc(Cl)ns3)=O)CC2)=O)CCCOC12CCC2 67823,C(c1cccnc1)=CC(N1CCCC1(C)CNC(C12COCC1C2)=O)=O 67824,S(=O)(=O)(c1[nH]c(=NCC(C2CCCO2)OC)ccc1Br)NCC(COCC)(C)C 67825,C(=O)(CC(=O)N1CCC(NC(=O)C(=O)NC2CCCC2)C1)N(CC#C)C 67826,C(=O)(CN=c1ccc(C#N)c[nH]1)N1CCCC(N(C(C(CCC)C)=O)C)C1 67827,C(=O)(CC(F)(F)C(F)(F)F)N1C(CCCNC(c2cncs2)=O)CCC1 67828,CCC(CC(=O)NC1CC(CNC(c2cnns2)=O)C12CCC2)CC(C)C 67829,CC(CCNC(C1CC=CCC1NC(c1cc(Cl)ns1)=O)=O)CC(C)(C)C 67830,CCCCC(C)CCC(=O)NCC1CCC(C(=O)NCCc2ccco2)O1 67831,C12(C(N(C3CN(C(C4CCCS4(=O)=O)=O)C3)C)=O)CCC(CO)(CC1)CC2 67832,C1(F)(CNC(C2(C)C(C)C2)=O)CCC(NC(=O)CCc2ncc(F)cn2)C1 67833,N1(C(C2(COC)CC2)=O)CC=CC(C(N2CCC2C(N)=O)=O)C1 67834,Cc1c(COC(=O)CC2(NC(C)(C)C)CCN(C)C2)nnn1C 67835,C(CC(C)C)(C(=O)NC1CCN(C(c2cnc(C#N)s2)=O)C1C(C)C)OC 67836,C1(CCC)(NC(c2ccc(C(F)F)o2)=O)CCCN(C(c2cccc(C)n2)=O)C1 67837,C1(C(N)=O)CCN(C(=O)CNC(c2ccoc2C2CC2)=O)C1NC(N1CCCC1)=O 67838,c1(NC(C23N(C(c4cc(CC)[nH]n4)=O)C(CC2)CC3)=O)ccc2ncccc2c1 67839,C(C(CNC(=O)CSCC(C)C)OC)NC(C1C(=C)C1)=O 67840,N1(C(C(Cc2cc[nH]n2)NC(=O)Cc2cccs2)=O)CCC(CCCO)CC1 67841,C1(C)(C(=O)NC(c2ccccc2F)CN(C)C)CCN(Cc2ccc[nH]2)CC1 67842,CC(C)C(CCN(C(=O)CC1CCC1)C)NC(=O)C(C(C)O)c1ccsn1 67843,CC1CN(C(C2(F)CCOCC2)=O)CCC1N=c1[nH]c(Cl)ncc1Br 67844,c1(C(N(C2CC(NC(c3cnc(=N)[nH]c3)=O)C2)C)=O)cccc(F)c1C1CC1 67845,C1(NC(CCN(CC#C)C(C2CC(C)(F)C2)=O)=O)CC2(CC2)C1 67846,C1(F)(C(N2CCCC(CN(C(CCCOCC)=O)C)C2)=O)CCC(C)CC1 67847,c1(C(C(N2CCC(CNC(c3sccc3F)=O)C2)=O)OCC)ccccc1F 67848,CC1=C(C)CC(C)(C(N2CC(NC(c3cscn3)=O)C(O)C2)=O)CC1 67849,Cc1nc2c(N3CCN(C(c4c(F)cncc4F)=O)C4CC34)ncnc2[nH]1 67850,N(C1CCc2ccccc21)C(CCCCNC(CC=C)=O)=O 67851,c1(C(N2CCCC(C(=O)NC3C=C(C)CCC3)C2)=O)cc(C#N)n(C)n1 67852,c1(C(N2C(CC(C)O)CCC2)=O)cccc(S(=O)(=O)NCCc2cc(O)no2)c1 67853,c1(C(=O)OCC)nc(C(N2CCC(C(C)NC(=O)CC3CCC3)C2)=O)cs1 67854,c1(C(=O)NC2(C)CC(C)C2)nn(C)nc1CSc1ccnc(Cl)c1 67855,c1(C(=O)NC2CCN(C(C3CCC(F)(F)C3)=O)CC2F)ccc2nccc(Cl)c2c1 67856,N1(CCCC)CCN(C(c2c(C)cnn2COC)C(=O)NC)CC1 67857,Cc1c[nH]cc1C(=O)NCCC(=O)NC1COCC1F 67858,N1(C(C(=O)Nc2c(OC(C)(C)C)cccc2)=O)CCc2ccc(Br)cc2C1C 67859,c1(OC)c(C)csc1C(N1CCCC1CCNC(=O)CCCc1cccs1)=O 67860,c1(C(=O)NC2C(NC(c3c(CC)scc3)=O)CCC2)cccc2cccnc12 67861,c1(C(=O)NC(C)CC2CN(C(=O)C(O)C3CC3)C2)ccc(C#N)c([N+](=O)[O-])c1 67862,C1(NC(C2(C)CC(=C)C2)=O)CCC2(CC1)CN(C(=O)CCc1ncccn1)C2 67863,C1(CNC(c2nc(C(C)C)oc2)=O)CCC(C)N(C(c2ccc(CO)nc2)=O)C1 67864,CCC(C(=O)OC)C(=O)NC(C)(C)CN(C(=O)C(COC)OC)C 67865,c1(N(C(=O)COCC2CCCCN2C(C)=O)CC)ccc(C(F)(F)F)c(F)c1C 67866,C(=O)(CC(CNC(C1C=CCCC1)=O)C1CCC1)NCCCC#C 67867,C12(C(=O)NC3CCC(NC(CCCC#N)=O)C3)CC3CC1(CO)CC3C2 67868,c1(C(=O)NCC(C)(C2CC2)NC(c2cc(C(F)(F)F)c[nH]2)=O)ncc(F)cn1 67869,N1(C(CCC=C)=O)CCC2CCN(C(c3cc(N)ccc3SC)=O)CC2C1 67870,C12(C(N(C(C)C)CCNC(=O)CCNC(N)=O)=O)CC(C)C1C2 67871,c1(OC)cnc(F)cc1C(N1CCC(NC(=O)CN2CC3C=CC2C3)C(O)C1)=O 67872,C1(NC(COC)=O)CN(C(=O)C=CC(C)(C)C)CC1F.C12CCC(C1)N2 67873,C1(O)(C(C(=O)NC2C(O)CC2O)NC(N)=O)CCCCC1 67874,C(=O)(CCCC(F)(F)F)NC(C)CCCNC(c1cnc(-n2cccn2)cn1)=O 67875,CC(CCCNC(c1csc(O)n1)=O)NC(c1csc(O)n1)=O 67876,c1(C(=O)NCC(=C)CCNC(=O)CCC2CCCOC2)ccccc1SC 67877,C1(C(=O)NCC2CC(C)N(C(=O)CN3CCCC3=O)C2)(OC)CCC(F)(F)CC1 67878,C(CCC(C)CC(=O)NC1CN(C(=O)Cc2cnn(C)c2C)C1)=C(C)C 67879,N1(C(C(C)(Cl)Cl)=O)CCC2(NC(=O)CSC(F)F)CC2C1 67880,c1(C(C)NC(c2n(CCCC)ncc2)=O)ccc(CNC(=O)CS(C)(=O)=O)cc1 67881,C1(C(=O)NC(CNC(=O)CC2(O)CCC2)C2CCC2)(CC)CCCCC1 67882,C(=O)(C1c2c[nH]nc2CCC1C)NC1C(S(CC)=O)CCC1 67883,CN1CC(NC(=O)C(c2cccc(I)c2)O)Cc2ccccc21 67884,C(=O)(C(O)C(CCC)NC(=O)Cc1ccn(C)c1)N(CCCCC=C)C 67885,n1(C(CC)CC)nc(C(=O)NC(C)C(C)NC(=O)C=Cc2csc(C)n2)cc1C 67886,C(=O)(C(F)C(C)CNC(=O)C(C)(C)C(F)F)NCCc1c(C)ncs1 67887,c1(CNC2CCC(C(=O)Nc3cncc(C)n3)OC2)csc2ccc(Br)cc12 67888,c1(NC(C2C(NC(c3ccccc3CO)=O)C2)=O)nc(Cl)c(Br)cc1O 67889,c1(N2CCC(N(C(CCC(C)SC)=O)C)C2)snc(C)c1C#N 67890,C1(NC(C2CCOCC2)=O)CN(C(=O)Cc2cocc2Br)CC12CC2 67891,c1(CNC(=O)CC2CC(C(N3CCC(F)C(F)(F)C3)=O)C2)ccc2c(c1)CCC2 67892,c1(OC2CCN(C(N(c3cc(F)ccc3Cl)CC)=O)CC2)cccc2[nH]ccc12 67893,Cc1c(CN(CC(C)NC(c2ccccc2C(F)(F)F)=O)C)cccc1O 67894,C(N=c1[nH]c(=NC2CCCC(F)(F)C2)[nH]c2c1COCC2)C1CC2C(F)(F)C2C1 67895,c1(N(CCCNC(=O)C(C)CN2CCOCC2)C(C)C)ncc2ncn(C)c2n1 67896,C1(NC(c2c(C)ocn2)=O)(CNC(=O)CCn2ccnn2)CC2CCC1C2 67897,C1(C(C)C)CN(C(C2(n3cncn3)CC2)=O)CCN1C(=O)C(C)c1ccsc1 67898,C1(C(=O)NCC(n2cccn2)C)CCOCCN1C(c1ccc(C#N)o1)=O 67899,c1(C(=O)NC2C(NC(C3(C)C=CCCC3)=O)CCCC2)cc(F)c(F)c(O)c1F 67900,c1(C(=O)NC2CC(NC(c3[nH]nnc3C3CC3)=O)C2)coc(OCC(F)(F)F)n1 67901,C=Cc1cc(C(=O)NCC2(C)CCN(C(c3ccnc(OC)c3)=O)C2)cc(F)c1 67902,c1(COC)nn(C)c(Cl)c1C(N1CCCC1CCNC(C1CC(C)(C)C1)=O)=O 67903,Cc1ccc(C=CC(=O)NCC(C)CNC(=O)Cn2ncc(C#N)c2N)cc1Cl 67904,C1(CCC(=O)NCC(CC)C(C)C)CCN(C(=O)CC2CCC(=O)C2)C1(C)C 67905,c1(-n2c(CCC(CCC)O)nc(C3CCCO3)n2)cc(CC)cc2cccnc12 67906,N1(C(C(C)SC)=O)Cc2ccccc2C(CNC(c2cnc(NC(C)=O)o2)=O)C1 67907,C1(CNC(C=C(C)C(C)(C)C)=O)CC2CN(C(C3(C#N)CC4CC4C3)=O)CC12 67908,CCC(CC(=O)NC(C)(C)CC(F)C(=O)N(CC(=O)NC)C)CC(C)C 67909,N1(C(=O)Cn2cnc(Br)c2)CCC2CCCC(C1)N2C(C1C2COCC12)=O 67910,CS(=O)(=O)c1cnc(CCNC(=O)C(=O)NC2CCC(=O)NC2=O)nc1 67911,C1(NC(c2cn(C)c(=O)nc2O)=O)CC(C2CCN(C(=O)CC3CC3)C2)C1 67912,CC(C)(O)C(F)C(=O)N1CCOC(C2CN(C(c3cncc(N)n3)=O)C2)C1 67913,N1(C(c2ccc(OCCOC)cc2)=O)CCC(C2(NC(C3CC3F)=O)CC2)C1 67914,CC1(C)CN(C(c2ccoc2)=O)CC1NC(C1CC1c1cccc(O)c1)=O 67915,CCCCS(=O)(=O)N1CCCC1C(=O)NCCCN(C(c1cnccn1)=O)CC 67916,N1(C(CCCCCC)=O)CC2(CCC2)CC1CNC(=O)C(c1cccc(C)c1)F 67917,C1(NC(C(CSC)(C)C)=O)CCCN(C(c2cc3sccc3s2)=O)CC1 67918,CN1CCC(C(=O)NCCOCC(=O)NC(CSC=O)C(C)(C)C)CC1.C(C)(C)(C)O 67919,C1(C2CCN(C)CC2)(C(N(CCC(C)NC(C(C2CC2)OC)=O)C)=O)CC1 67920,CC1CCCC(OCCN(C(=O)C(=O)Nc2ccsc2Br)Cc2ccccc2)C1 67921,CC1(C(=O)NCc2cccc(Cl)c2F)CCCN(Cc2nccs2)C1 67922,c1(CC(=O)NCCNC(CCCN(CCOC)C)=O)ccc(OC(F)F)c(F)c1 67923,c1(NC(c2cn(CCC=C)nn2)=O)cccc2c1CN(S(C)(=O)=O)C2 67924,c1(C(N2CCC(C(=O)Nc3cncc(I)c3)C2)=O)nc(Cl)ccc1F 67925,N1(C(c2n[nH]cc2C(F)(F)F)=O)CC(N=c2[nH]nc(CO)s2)C2(CCC2)C1 67926,N1(C(C)=O)CCCC(O)(C(N2CC(O)(CNC(=O)CSc3cccs3)C2)=O)C1 67927,CCC(CC)CC(=O)NCC1CN(C)CCN1C(c1cc(C)nn1C(F)F)=O 67928,n1(COC)nccc1C(N1CCC(OCC(=O)NC(C)Cc2ccnn2C)C1)=O 67929,N1(C(CC(C)(C)C)=O)CC2(CCC2)CC1CNC(c1ccnc2c1CCC2)=O 67930,C(=O)(CC(=O)NCC1CC(NC(c2c[nH]nc2C(C)(F)F)=O)C1)N(C)C 67931,N1(C(C)=O)CCN(C(=O)CCCn2cc(C(O)C3CC3)nn2)CC1 67932,Cc1nn(C)c(C)c1C(N1CC(NC(=O)CCN2CCCS2(=O)=O)CC(O)C1)=O 67933,N=c1[nH]cc(C(=O)NCC(F)CNC(c2cscc2F)=O)c2cc[nH]c12 67934,C1(C(N(CCN(C)C(c2cnncc2C(F)(F)F)=O)C)=O)CCC(O)CN1C 67935,N1(C(C#CCNC(=O)C=CC(=O)NC2CC2)=O)CC2(CCC1CO)CC2 67936,c1(C(N(CCCNC(c2cnsc2C)=O)CC)=O)cc(=O)n(C)c2ccccc12 67937,c1(C(=O)NCCC(C)(C)NC(C2C(OCC)C2)=O)snc(C)c1N 67938,c1(-c2cn(NC(CC3CCC(NC(CC)=O)C3)=O)nn2)ccc(C#N)cc1[N+](=O)[O-] 67939,C1(C2(O)CCOCC2)(CS(N2C(C(=O)OC(C)(C)C)C(O)CC2)(=O)=O)CC1 67940,c1(OC(C)=O)cccc(C=CC(=O)NC(C)CNC(=O)Cc2c(C)noc2C)c1 67941,c1(C(=O)NCC2C(C(=O)NCC=C)CC2)cccc(-n2ccnc2)c1 67942,Cc1cnc(C(C)NC(=O)C(C2CCCCC2)C)s1 67943,N(C(=NCc1ccccc1)N1CCC(F)(C(F)(F)F)C1)CCc1[nH]nc(N(C)C)n1 67944,C(=O)(C(C)(CC)CO)NCC(CCCC)NC(c1n[nH]cc1[N+](=O)[O-])=O 67945,CC1(C#CC(=O)NC2CCCC(NC(=O)CCc3nc(=N)[nH][nH]3)C2)CC1 67946,C(=O)(C(O)C(C)(C)C)N1CC(C)C(NC(=O)Cc2ccncc2Cl)C1 67947,C#CC1(C)CCN(C(C2CC3(CCN(C(C4CCC(C)C4)=O)C3)C2)=O)CC1 67948,C(c1ccc2occc2c1)=CC(=O)NC1CN(C(C=CSC)=O)C(C)C1 67949,C(=O)(CC(C)(C)C(F)(F)F)N1C(CCNC(C(C)SC(F)(F)F)=O)CCC1 67950,CCC(CC)(CCO)NC(c1cncn1C(C)(C)C)c1nnnn1C 67951,C1(COCC(=O)NCC(=O)NC(CCCN(C)C)C2CC2)COCC1C(F)(F)F 67952,c1(C(=O)NCC2C(NC(C(C(=O)OC)C)=O)C2)ccc2c(c1)C(=O)OC2(C)C 67953,C(CNC(=O)CCc1cnn(C)n1)(CCOC)NC(C(C)NC(CC)=O)=O 67954,c1(C(N2CCC(C(=O)NCC)CC2)=O)ccc(F)c(-c2c(C)cccc2F)n1 67955,C(=O)(C1=CCCSC1)NC(C(C)C)CNC(=O)COC1CCCOC1 67956,C1(NC(c2nc(CC)oc2C)=O)CN(C(C2CC2F)=O)CC1N=[N+]=[N-] 67957,c1(NC(CCCNC(C(C)SC)=O)=O)cc(C)nn1C 67958,N(C(=NCc1noc(C2CC2)n1)N1CC(c2ccccc2)C2(CCC2)C1)C(C)C 67959,Cc1cc(C)n2nc(C(C)NCCOc3cccc(Br)c3)nc2n1 67960,c1(SCC)ccc(Cl)cc1C(=O)N(CC(CC)NC(=O)C(F)CC1CCC1)C 67961,C1(CN=C(NCc2ccc(OC)nn2)NC2CC2)CCC(F)(F)CC1 67962,c1(C(=O)NC2CC(NC(c3nc(C)sc3C)=O)C2)ccc2nn[nH]c2c1O 67963,c1(C(N2CC(CC#C)(C(=O)NCC)C2)=O)cc(Br)cnc1CC.C1(C)C(=O)O1 67964,C1(NC(C(C)C)=O)CCN(C(c2csc(C(C)(C)C)c2)=O)CC1CO 67965,C#CCCCCCC(=O)NCC1(F)CN(C(c2c(C)csc2C)=O)C1 67966,C12(CNC(C3N(C)CCC3)=O)CCCC(CN(C(=O)C(F)C3CCC3)C1)C2 67967,O=S(=O)(c1cccc(NCCF)c1)N(CCCC(F)(F)F)CCF 67968,c1(C(=O)NCC2N(C(Cn3c(=O)sc(C)c3C)=O)CC2)c(F)ccc2c1OCO2 67969,C12(CNC(C=CCOC)=O)CC1CN(C(C1CC(C)(F)C1)=O)C2 67970,C(=O)(CCCCCOC)NCC1C(C(N2CCC(=C)C2)=O)C1 67971,c1(C(=O)NC(C(C)C)C(C)NC(=O)Cc2cn[nH]c2)cc(=O)c2ccccc2[nH]1 67972,C1(NC(C(N(C)C)C2CC2)=O)COCC1NC(c1ccoc1I)=O 67973,CC(CNC(=O)C(F)F)(C(F)F)NC(c1ccc(C2(C#N)CCC2)cc1)=O 67974,c1(C(=O)NC(C2(O)CN(C(CC(C=C)C)=O)C2)C)n[nH]c2c1CS(=O)(=O)CC2 67975,c1(C(N2CCCC(CNC(CCC3CC(C)C3)=O)C2)=O)cn(C)c(=O)n(C)c1=O 67976,N1(C(Cn2c(C)ncc2)=O)CCC(O)(CNC(=O)CCc2cccnc2)C1 67977,c1(Cc2nnnn2C2COC2)cc(CNC(C)CCC#N)ccc1C#N.CC 67978,C#CC1CCC(C(N2CC(OC(F)F)C2)=O)CC1.c1(N)ccccc1 67979,CC(C)(C)C(CNC(c1ccn(C(F)F)n1)=O)C(=O)NCC1CCC1 67980,C1(NC(CC2CN(C)C2)=O)CN(C(c2cncn2C2CCOCC2)=O)CCC1O 67981,[N-]=[N+]=NCC(C(=O)NCC1C2CCCC12)NC(C1CC1C(N)=O)=O 67982,C1(CNC(C2CC(C)OCC2)=O)CC2(CCN(C(=O)COC3CCOC3)C2)CO1 67983,Cc1ccc(F)c(C(=O)NCC2=CCN(C(=O)CC3(C)CCCO3)CC2)c1F 67984,C1(CNC(CS(=O)(=O)NC)=O)CCC2(CCC2)CN1C(c1cncn(C)c1=O)=O 67985,C1(C(C)NC(CCOCCCOC)=O)CN(C(=O)CC2CS(=O)(=O)C2)CCO1 67986,c1(OC)cc(C(=O)NC2CC(C)CN(C(=O)OC(C)(C)C)C2)ccc1C 67987,N1(C(C(CCOC)OC)=O)Cc2ccccc2CC1C(=O)NC1CCOC1 67988,c1(CC(=O)NC(Cn2cc(C=CC)nn2)C)ccc(C#N)cc1F 67989,Cc1noc(C2CC2)c1C(=O)NC(CNC(c1csc(C2CC2)n1)=O)CO 67990,C1(C(N2CC3(N(C(C(C(C)(F)F)F)=O)CC3)C2)=O)CCc2nccn2C1 67991,c1(CC)oc(C(N2CCC(NC(=O)CCC3CCC(=O)NC3)C2)=O)cc1C 67992,C1(COC)(CNC(=O)CCc2cc(C)no2)CCCN1C(C1CCCC1)=O 67993,c1(CC(=O)NCC(CNC(c2cc(CC)on2)=O)O)c(C)n[nH]c1C 67994,C1(CNC(C(CO)N(C)C)=O)CC2(C1)CN(C(C1(C(C)(C)O)CC1)=O)C2 67995,N1(C(CSc2c(C)n[nH]c2C)=O)CCN(C(C2(C)COC(=O)C2)=O)CC1C(F)F 67996,c1(CC)nccc2c1CCN(Cc1ncsc1Br)C2 67997,C(C)(C)(CCCNC(C1CCC(O)C1)=O)NC(c1c(C(C)C)ncs1)=O 67998,C1(CC(=O)OCC)CCCN(C(=O)C=CC(C)(C)NC(=O)CCC(C)C)C1 67999,N1(C(C(C=C)(C)O)=O)CC(NC(C2CC3(CCOCC3)C2)=O)CC2(CCC2)C1 68000,C1(NC(C=C(C)C(C)C)=O)CCN(C(C23CC(C)(CCO2)C3)=O)CC1C(C)C 68001,Cc1cc(NCCC(C)NC(=O)C(c2cccnc2)O)c(Br)cc1[N+](=O)[O-] 68002,c1(N2C(CC(=O)Nc3cc(CCC)no3)COCC2)ncc2cccc(Br)c2n1 68003,C1(C)(C(=O)NCc2cccc(CC)c2)CC12CCN(C(c1[nH]ccc1C)=O)CC2 68004,c1(C(N(C(CNC(C(C)CC2CCC2)=O)C)C)=O)c[nH]c2nccc-2c1 68005,C1(CNC(c2ccn(CC)n2)=O)CC(NC(=O)C(O)Cc2ccccc2)C(O)C1 68006,N1(C(CCOCC)=O)CCN(C(C23CC(C2)S(=O)(=O)C3)=O)CC1C 68007,c1(C(=O)NC(C2CN(C(=O)C3=NNC(=O)CC3)C2)C)cc(F)c2cn[nH]c2c1 68008,Cc1nc(CC(=O)NC2(C(=O)NC3CCC3)CSC2)cs1 68009,N1(C(C2(CC)CCNCC2)=O)CCC(C#N)(OCC)C1 68010,c1(C(=O)NC(C2CCCCN(C(=O)Cc3nccn3C)C2)C)cc(N)nc(Cl)c1 68011,N1(C(CNC(CCC(C)C)=O)=O)CCC(C(=O)N(C)Cc2ccsc2)C(C)(C)C1 68012,CC1(CO)CCCN(C(=O)C(c2ccco2)NC(c2cn[nH]c2)=O)C1 68013,c1(C(=O)NC(CNC(C2(OC)CCC2)=O)(C)C)cnc(OC)c(C(=O)NC)c1 68014,C(=O)(C1=C(Cl)CCCC1)NC1(O)CCN(C(CCOC(CC(C)C)C)=O)CC1 68015,CCC(CC)C(C)C(=O)NCC(C)(CC)NC(=O)CSc1nncn1C1CCCC1 68016,c1(CN(C(CN(C)CC)=O)C)ccc(CC2(C(=O)NC)CC2)cc1 68017,N1(C(c2scc(C)c2C)=O)CCC(CNC(=O)CCC2CCC(C)O2)C(F)(F)C1 68018,c1(C(N2CC(c3cn(C4(C(=O)OC)CC4)nn3)(C)C2)=O)ccnnc1C 68019,C(CC1CC1)(C(=O)N1OC2CCC1C2)NC(c1cc(CC)n(C)n1)=O 68020,N1(C(c2cnc(CC(C)C)s2)=O)CC2CC(NC(=O)CC3=NNC(=O)C3)CC1C2 68021,CCCC(C)(CC)C(=O)N1CC(C2(NC(=O)C(C)CCOC)CC2)C1 68022,O=C(C1=COCC1)NCCC1CN(C(C2(Sc3cccc(F)c3)CC2)=O)CCO1 68023,C12(CCOCC1)C(=O)N(C)CCN(C)C2.c1(NC(=O)C(C)(C)F)ccccc1 68024,C1(OC)CCC(C(=O)NCC2CCN(C(=O)CCSc3ccc(C)cc3)C2)CC1 68025,C12(C(=O)NCC3C4CN(C(C(C)(C)N(C)C)=O)CC43)CCC(C)(C(=O)O1)C2(C)C 68026,Cc1nc(N2CCC3(CCN(C(=O)C(C)c4cccs4)C3)C2)c2sccc2n1 68027,c1(SC)cccnc1C(=O)N(C(C)CNC(=O)C(CO)NC(N)=O)C1CC1 68028,CC1CC(NC(=O)CC2CCC(=O)N2C)CCN1CCc1cncs1 68029,C1(C(=O)NC2CC(F)(CNC(=O)CN3CCCS3(=O)=O)C2)CC12CC(F)(F)C2 68030,N1(Cc2cn(CC)nc2)C(C(N2CCC(C)C2C)=O)CC2CC12 68031,C1(NC(c2ccc(N(C)C)nc2)=O)CN(C(C2CC2C(F)(F)F)=O)CC1C1CC1 68032,C(=O)(C(O)CCC(F)(F)F)N1CCC(OCCNC(C(COC)(C)C)=O)C1 68033,c1(NC(C2CN(c3ncc(C)cn3)CC2(C)C)=O)c(C)nc2ccc(Br)cn12 68034,C(=O)(C1Cc2ccc(F)cc21)N(C)CCNC(c1cscc1C1CC1)=O 68035,N1(C(c2n(C)c(Cl)nc2)=O)CCC(O)C(C(=O)N(CC#N)CC#N)C1 68036,c1(NC(CNC(C2(NC(CSC(C)(C)C)=O)CCC2)=O)=O)c(F)cccc1F 68037,Cc1ccc(C=CC(N2CCCN(C(=O)CCCC3CC3)CC2CO)=O)cc1Cl 68038,C1(N(C)C(c2cnncc2O)=O)CCCN(C(C2(Nc3ccccc3)CC2)=O)C1 68039,CCCCC(CC)CC(=O)N1CC(F)CC1CN(C(=O)CC(C)(C)C(F)F)C 68040,C1(NC(C2C(C)CN(C(c3cnc(O)n3C)=O)C2)=O)CCN(C)CC1C#N 68041,C(CC(C(=O)NCCN(C(=O)C=Cc1cocn1)C1CC1)N(C)C)SC.C(C=C)=C 68042,C(=O)(CCN=c1ccc(C)c[nH]1)NC1CC(NC(C(COCC)(C)C)=O)C1 68043,O=C(C#CC1CCOC1)NCC1CCN(C(c2ccc(CO)o2)=O)CC1O 68044,C=CC1(CC(=O)NCCc2nc[nH]n2)CN(C(=O)CC(CC)SC)C1 68045,C(CC(=O)NCC(C)(C)N1CCCC1)(C(F)F)NC(C(COC(C)C)(C)C)=O 68046,C1(c2n(CC(=C)C)nnn2)(NC(C)C)CC(C)N(C)C1.c1(C)ccccc1COC 68047,c1(C(=O)NCC(C(=O)NCC(COCC)C)O)ccc2[nH]ccc2c1 68048,Cc1cscc1C(=O)NCCCCC1CN(C(=O)CCc2cncnc2)C1 68049,c1(N(CC(=O)NC2CCC2)C(c2c(CC)cco2)=O)ccc(O)c(OC)c1 68050,C1(CNC(CN2CCC(C)CC2)=O)CN(C(=O)Cc2cn(C)nn2)C(C)(C)C1 68051,c1(OCCC2(OC)CCOC2)c(C)ncn1O.N12CC(C1)NC(=O)CC=CC2=O 68052,C(=O)(C(C(=O)NCC12CC1CN(C(C1CCC1OC)=O)C2)C(C)C)OCC 68053,c1(C(=O)NCCOCCn2cc(-c3nn[nH]n3)cn2)cccc(=O)n1O 68054,C1(CNC(C=CCCC=C(C)C)=O)COCCN(C(C2CCCN(C)C2)=O)C1 68055,c1(C(=O)NC2C(C)CCN(C(C(C(C)C)(C)C)=O)C2)cc2c(nc1N)CCC2 68056,c1(C(N2CCC(NC(C=C(CC)C)=O)C(F)C2)=O)cnc2c(N)cccc2c1 68057,N1(C(C)C)CC(C(N2CC(CCNC(=O)C(C)NC(N)=O)C2)=O)CC1=O 68058,C1(C(=O)NCC(C2CCCCC2)C)CCCN(C(c2nccnc2N)=O)C1 68059,C1(C(C(=O)N(C2C(C)CC2)C)C)CCCN(C(=O)Cn2cccc2C=O)C1 68060,C(C(O)C(=O)NC1CC(F)(CNC(c2csnn2)=O)C1)SC 68061,C1(NC(C2(c3cc(C)no3)CC2)=O)CCN(C(c2cccnc2)=O)CCC1(F)F 68062,C(=O)(C(C)(C)CS(N)(=O)=O)NCC1(F)CC(NC(CC(=O)NCC#C)=O)C1 68063,C(=O)(CC1=CCN(C(C2OCCC2(C)C)=O)CC1)N(C(CSC)C)C 68064,Cc1cccc2nc(C(=O)NCC(O)CNC(C34CCCCC3C4)=O)cn12 68065,C1(F)(CNC(C2C(OC)C2)=O)CC(CNC(C2CC2OC)=O)C1 68066,c1(C(=O)NCCC(=C)CNC(=O)C(c2ccnn2C)O)cc(F)cc(F)c1 68067,c1(C(N(C2CCN(C(C3CC(F)CN3C)=O)C2)CCC)=O)nccnc1N 68068,CC1CCN(C(C2CC3CC3C2)=O)CC1C.c12cc(nn1C)CNC2=O 68069,c1(C(C)C)nn(C)c(C(=O)N(C(C)CNC(=O)C(O)CF)C)c1Cl 68070,N1(C(=O)OC)CCN(C(C2CCCN2Cc2csc(C(C)=O)c2)=O)CC1 68071,CCC(C)C(CC(=O)N1CCn2nncc2C1)NC(=O)CSCC(F)F 68072,c1(NC(=O)NC2C(CC(=O)OC)COCC2)ccc(F)c(F)c1 68073,C(=O)(CCCCNC(C1(C)CCNC1=O)=O)NCC(C)(C)CN1CCCC1 68074,C1(NC(=O)C2=CC(O)CCC2)CCC2(CC1)CN(C(=O)C(F)C(F)(F)F)C2 68075,C=CC(C)CC(=O)NC(CNC(=O)CC1CNC(=O)O1)C(C)C 68076,C1(CC(=O)NC(C2CCCN(C(c3cocn3)=O)C2)(C)C)CC(=O)NC(=O)C1 68077,N1(N(C(=O)C=C2CCCCC2)C)CCCC(CCC(F)(F)F)C1 68078,Cc1ccc(CN2CC(NC(C3(C4CCOC4C)CC3)=O)CC2C)cc1 68079,c1(NCC(=O)NC(c2cn(C)c3ccccc23)C)ncnc2[nH]cc(C(N)=O)c12 68080,c1(C(=O)NCC(CNC(C(CC)c2cccnc2)=O)C)ccc(Cl)nc1O 68081,c1(C(N(C)CC2CN(C(CS(=O)(=O)NCC)=O)C2)=O)ccc(SC)cc1C 68082,C1(C(=O)NC2(CO)CN(C(C(=Cc3cnc[nH]3)C)=O)C2)CCS(=O)(=O)N1 68083,c1(CN(C)C(c2cn(C3(NC(C4CC(O)C4)=O)CC3)nn2)=O)ccc(F)cn1 68084,CCC(F)(C(=O)OC)C(=O)N1CCCC1CNC(c1ccc(F)c(OC)c1F)=O 68085,N1(C(C(C)CCN(C)C)=O)CCC(C2CC2)C1C(=O)N(CC1CCC(O)CC1)CC 68086,Cc1noc(C)c1C(C)C(=O)N(CCNC(=O)Cc1ccc(C(N)=O)nc1)C1CC1 68087,C12(COC)CCC(C(=O)N(C)CCNC(C3(C#N)CCCO3)=O)(CC1)CO2 68088,CN1CC(C)(C(N2CC=CC(NC(c3sccc3Cl)=O)C2)=O)CC1=O 68089,C1(NC(C2C(NC(C3CCCN3CC(F)F)=O)C2)=O)CCCCCCC1O 68090,c1(CCOC(CC(C)CC2CCC2)=O)ccccc1[N+](=O)[O-] 68091,C1(C(N2CCC(CC(O)C3CC3)CC2)=O)COC2(CNC2)C1 68092,C12(NC(c3cn(C4CC4)nn3)=O)CC3CCC(C1C2)N3Cc1c(CC)cccc1 68093,N1(C(C)=O)CCC(C)(C(N2C3CC2CN(C(C2C=CCS2)=O)C3)=O)CC1 68094,CN1CCCC1C1CC1CNC(C1CC(N(C(=O)Cn2[nH]cnc2=N)C)C1)=O 68095,C(N=c1[nH]cnc(Cl)c1CO)C1CCC(NC(c2ccc(C(=O)NC)nc2)=O)C1 68096,n1(C(C(=O)N(CC(CC)NC(=O)C(O)C2CCCC2)C)C)nc(C)cc1C 68097,N1(C(CCCC#C)=O)CCCC2C(NC(c3cc(O)cc(C#N)c3)=O)C(C)(C)C12 68098,C=CCCC(=O)NCCCCCNC(=O)CC1(NC(C)=O)CC1 68099,c1(C(N2C(C)CC(NC(c3ccc(OC)cc3F)=O)C2)=O)cccc2[nH]ncc12 68100,c1(C(N(CCC)CCNC(C2(CCF)CCC2)=O)=O)cc(Cl)cc(Cl)n1 68101,c1(CC(=O)NC2CN(C(c3c(OC)nsc3)=O)C3C2C3)cc2ccccc2o1 68102,c1(C(=O)NC2COCCN(C(C3CC(CC)OCC3)=O)C2)cn2ccccc2n1 68103,N1(C(C2C(C)CCO2)=O)CC2C(CNC(=O)C(F)(F)Oc3ccccc3)C2C1 68104,C(=O)(C(C(C)(C)C)NC(=O)Cc1cncs1)NCCc1c(C)ncs1 68105,c1(C(=O)NCCC(C)N(C)C(C2(CO)CCCO2)=O)cnn2c1OCCCC2 68106,C(CNC=O)(CCSC)OC.n1(C2(n3nccn3)CC2)cc(CN2CCSCC2)nn1 68107,CCC(C)C(C)N(C(C=CCNC(=O)CSC)=O)CC 68108,c1(C(N(C)CC2CN(C(C3C(C(=O)OC)CCC3)=O)C2)=O)c(C)cccc1O 68109,C1(CNC(C(C2CC2)NC(c2ccsn2)=O)=O)CCCN1C1CC1 68110,C(C(=O)NCCC)(C1=Cc2cc(Br)ccc2OC1)N(CC(CC)C)C 68111,Cc1c(C)n(C)c2ccc(C(=O)NCC3CN(C(=O)C(C)(F)F)CCC3C)cc12 68112,C1(OC)CC(CNC(=O)C(C)(C)n2cnnn2)N(C(=O)CC2CS(=O)(=O)C2)C1 68113,N1(C(CCSCC(C)C)=O)C2CCCC1CN(C(=O)C(c1ccccc1)F)C2 68114,Cc1cncc(CCC(=O)NCC2CC(C)N(C(=O)CSC(F)(F)F)C2)c1 68115,C(=O)(CCC(CC)NC(=O)CCCCOC)N1C(C=C)CCC1 68116,C1(NC(CC(=O)NCC(C2C(C)(C)C2(F)F)(C)C)C2CC2)CC(=O)N(CCl)CC1 68117,C1(NC(Cn2nc(C)c(Br)c2)=O)CN(C(c2cnc(N)cn2)=O)CC1(C)C 68118,CCC(C(=O)NCC(C)(C)NC(C1CC1c1cncn1C)=O)SC 68119,C1(C(N2CCC(CC(=O)NC)C2)=O)CCCN1NC(=O)C(=O)C1CCOCC1 68120,Cc1ccc(F)cc1C(=O)N(C(C)C(=O)NCc1cnc(C)cn1)C1CC1 68121,c1(C(N2C(CN(C(COC(CC)C)=O)C)CCCC2)=O)ccnc2ncsc12 68122,C(=O)(CN=c1[nH]cnc2c(Br)cccc12)NC(c1ccccc1)C(C)C 68123,C1(NC(CCCC)=O)CCC2(CC1)CC2NC(=O)CC1CCC(=O)N1C 68124,C(=O)(CCCCCOC)NCCN(C(C1N(S(CCCC)(=O)=O)CCCC1)=O)C 68125,C#CC1CN(C(c2n(CC)ccc2)=O)CCN1C(=O)Cc1sccc1C 68126,C1(NC(=O)Cc2cscn2)CN(C(C2COCC2C(F)(F)F)=O)CC1O 68127,CC(C)(C)CCN=c1[nH]c(=NCc2csc(C(F)F)n2)[nH]c2cc[nH]c12 68128,N1(C(c2ccc(F)cc2)C)CCC2(CCCN(C(=O)CCc3ccccn3)C2)C1 68129,C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CCN(C(c2n(C)nnc2)=O)C2C1C2 68130,C1(O)(CCNC(Cc2ccc(C)nc2)=O)CCN(C(=O)C(C)(C)CC#N)CC1 68131,N1(C(c2cc(Cl)c(Br)c(Cl)c2)=O)CCC2C(CCN2Cc2cc(I)cnc2Cl)C1 68132,C1(C(=O)NC2C3CN(C(CC(CC)CC)=O)C2CC3)CCc2nnnn2C1 68133,Cc1nn(CC(=O)NC(C)(CNC(=O)C=CS(C)=O)C(C)C)c(=O)o1 68134,n1(CCCc2cccc(SC)c2)nnc2ccccc12 68135,C=CCC(C)C(=O)NC(C)Cc1ccc(CNC(c2cnncc2C)=O)cc1 68136,c1(C(N(C)CC2(NC(C(F)=CCC)=O)CC2)=O)cn2c(n1)CCC2 68137,C1(NC(C(CNC(C)=O)C)=O)C2CC1N(C(=O)CC(=O)NCC(F)(F)F)C2 68138,C1(CCC)CCC(NC(Cc2cn(-c3ccn(C)n3)nn2)CC(=O)O)CC1 68139,C1(C(N2CCN(C(c3c(CC)nccc3)=O)C(C)C2)=O)CC2CC(O)C(C1)C2 68140,Cc1cnc(CNC(C2CCC2CNC2(c3ccccc3F)CC2)=O)cn1 68141,Cc1cncc(C(N2CCCC2CCCNC(=O)C(C)OCC2CC2)=O)c1C 68142,Cc1ccc(Cl)cc1NC(=O)C(C)(C)C1CCCN1C(=O)CC(C)N(C)C 68143,c1(CCCC(=O)NCCOCCN(C(C=CCC)=O)C)cccc(Cl)n1 68144,c1(CC(=O)NCC=CCNC(C2C(COC)C2)=O)ccc(F)c(Cl)c1 68145,N1(C(C(CCC)NC(c2cc(C)nn2C)=O)=O)CCC2(CCCOC2)C1 68146,Cc1nc(NCC(F)(F)Br)cc(N2CCCC(N3CCC3)C2)n1 68147,C1(C(N(CC(C)CNC(c2cnccc2Cl)=O)C)=O)CCN(C)S1(=O)=O 68148,c1(C(N2CCC(NC(CSCC#C)=O)CC2C)=O)cc2nc[nH]c2cc1F 68149,C(=O)(C(C)S(C)(=O)=O)NC1CCCC(NC(CSC(C)C)=O)C1 68150,C1(OC)CC(C)(C)C1CNC(c1conc1C)c1nnnn1CC1CCOC1 68151,N1(C(=O)NCc2cn(CC(=O)OCC)nc2C)CC(=O)N2CCCCC2C1 68152,C1(C(=O)NCC2(Cl)CC2(F)F)COC2(C1)CN(C(=O)CCSC1CCC1)C2 68153,c1(C(N2CC3CC(NC(CC=CC=C)=O)CC3C2)=O)csc(N=S(C)(C)=O)n1 68154,C#Cc1ccc(C(N2CCC3CC23C(=O)NC(c2cnn(C)c2)C)=O)nc1 68155,CCCCCCCCC(=O)NC1CCC(NC(=O)Cc2csc3ccccc23)C1 68156,N1(C(C=CCC)=O)CCCC(O)(CCNC(=O)CN(c2cccc(Cl)c2)CC)C1 68157,c1(NCC2C3CN(C(C=CS(CC)(=O)=O)=O)CC32)ncc2ncn(C)c2n1 68158,c1(C(N2C(CNC(C3CC(C)=C(C)CC3)=O)COCC2)=O)cc(C)cc(Cl)c1N 68159,C1(C(=O)NC)CC(OC)CN1C(=O)Cc1cnn(C)c1OC 68160,Cc1cccnc1CC(=O)NC(CN(C)C(C1CCC(CO)CC1)=O)(CO)CO 68161,c1(-c2c(OC)ccc(-c3nccn3CC(O)CO)c2)cc2cccc(OC)c2o1 68162,C(CC(C(=O)NCC1(F)CC(NC(=O)C(F)=C2CCC2)C1)OC)OC 68163,c1(CC)ccccc1CC(N1CC2CC1C2NC(C1CCOC1C(=O)OC)=O)=O 68164,N1(C(Cc2c(OC)nccc2)=O)CCN(C(=O)CC=C(C)C)CC1C1CCCC1 68165,C(CCCCCCC(=O)NCCOCCN(C)C(C1C2COCC12)=O)SC 68166,C1(CNC(CC(CC)C)=O)CC2(CN(C(=O)CCS(C)=O)C1)CC2 68167,C1(NC(C(C)n2cncn2)=O)C=CCC(C(=O)NC2CC2c2cncs2)C1 68168,Cc1ccc2ccccc2c1C(=O)NCC(C)N(C)C(c1nnc(S)n1C)=O 68169,n1(CC(=O)NCC(C)(C(C)C)NC(C(c2cccnc2)SC)=O)nc(C)c(C)c1C 68170,C1(CCC)CN(C(c2cnn[nH]2)=O)CC1C(=O)Nc1c(C)nsc1C 68171,N1(C(CCCCCOC)=O)CC2CCOC2(CNC(=O)Cc2nc(C)oc2C)C1 68172,c1(OC)ccc(C2(CO)CC2)cc1C(N1CCC(C(C)N=c2[nH]ncs2)C1)=O 68173,c1(CC(=O)NC2CC(CNC(Cc3c(C)ncs3)=O)C2)sc(O)nc1O 68174,N12CCCCCCC1C2=O.CCC(C)CC(=O)N(C1CCCCCC1)C 68175,c1(CNC(N(C)C)=O)ccc(NC(=O)CC(c2ccccn2)N(C)C)cc1 68176,CC(CC(C)(F)F)C(=O)N1CCN(CCNC(c2cnc(N)c(CO)c2)=O)CC1 68177,Cc1cnncc1C(=O)NC(Cc1cccs1)CC(=O)NCC(N1CCOCC1)=O 68178,C1(C(N(CC)CC2CC2)=O)Cc2nccnc2CN1C(c1sc(Br)cc1I)=O 68179,c1(C(=O)OC)cc(Cl)c(OC)nc1C.c12cc(cc(C)c1)CN2 68180,c12cc(CCOC)ccc1O2.O(NC(=O)NCC1CC1)CC(=C)C 68181,c1(C(C(=O)NCC(CCOC)NC(c2sccc2C)=O)(F)F)ccc(C)cc1 68182,N1(C(C(CCC)C(=O)OC)=O)CCOC2(C1)CN(C(=O)CCc1cc(C)on1)C2 68183,c1ncc(Br)cc1Cl.N12CCSCC1c1cnc(s1)C2=O.C1CC1 68184,c1(OC)cc(OC)c(F)c(C(=O)NC2CC(F)CN(C(C3CCCS3)=O)C2)c1 68185,c1(C(=O)NC(CC=C)CNC(C2CCCN2C)=O)cnnc(O)c1 68186,Cc1nc2ncnn2cc1C(=O)NC1CCCCC1NC(=O)Cc1cccnc1 68187,C1(NC(CN2CC(=O)NCC2)=O)CCCC12CCN(C(=O)Cc1cccs1)CC2 68188,c1(C(N(C)CC2CCN(C(=O)C(C3CC3)C3CC3)CC2)=O)ccc(S(N)(=O)=O)s1 68189,C1(CC=C)(NC(=O)C(C)C(C)(F)F)CCN(C(=O)C(C)Cc2ccncc2)CC1 68190,C1(CNC(C2C(CC)CCCC2)=O)CN(C(c2cc3[nH]ccc3s2)=O)CCN1C 68191,C1(COC)CN(C(c2ccccc2Br)C(=O)Nc2ccccn2)CCO1 68192,C(C(O)C(=O)NC1(C)CC(NC(c2cc(C3CCC3)[nH]n2)=O)C1)=CCCC 68193,c1(OCCC)cncc(C(N2CC(NC(=O)C(C)n3cncn3)C(CC)C2)=O)c1 68194,CC1CCc2[nH]c(C(N3CCOC(CCNC(c4ccnnc4)=O)C3)=O)cc2C1 68195,c1(C(N2C(C(N3C(C)C(O)CCC3)=O)CC(C)C2)=O)ccc([N+](=O)C2CC2)cc1F 68196,c1(C(=O)NC2CC(C(C(=O)NC(CC)C(C)(F)F)F)C2)ccn(C)c(=O)c1 68197,CC(C)C(CC(=O)NCC1CC2CCC1CC2)NC(C1CC2(CCO1)CC2)=O 68198,c1(C(=O)NCCN(C(c2n[nH]cc2C)=O)CC)c(F)ccc(O)c1Br 68199,C1(C(C)C)CN(C(c2cc(-c3cccnc3)no2)=O)CCN1C(=O)CC(F)F 68200,C(=O)(C1=C(Cl)CCCC1)NC(CCN(C(c1cc(CC)c(C)cc1)=O)C)C 68201,C(=O)(CCCN=[N+]=[N-])NC(CNC(c1c(C)nncc1)=O)C1CCC1 68202,c1(C(N)=O)ccc(CN(CCCCCN)CCO)cc1.c1(=O)c(=O)[nH]1 68203,C(CC(C)CC)(C(=O)NC1COC1)N(C(CCC)CCC)CC 68204,c1(CC)nc(CC(=O)NCC(O)CNC(=O)C(F)=CCCN2CCOCC2)cs1 68205,N1(C(C2(CC=C)CN(C(c3coc(C(=O)OC)n3)=O)C2)=O)CC2CC(C)C2C1 68206,C(=O)(N1CC2COCC2O1)c1cc(CNC(C(CC)OC)=O)oc1C 68207,c1(OC)ccccc1C1(C(=O)NC2CCC2NC(c2nocc2C)=O)CCC1 68208,C(C1=NOC2CN(C(=O)C=C3CCC3)CC12)NC(C=Cc1cc(OC)ns1)=O 68209,C1(CCC)(NC(c2cncn2C)=O)CCN(C(C2CC23CC(F)(F)C3)=O)CC1 68210,C(C(C)(C)C(=O)OC)(c1n(CCC)nnn1)NCC1(c2ccccc2)CC1Br 68211,c1(C(N2CCC(C)(C(=O)NC(C(F)F)C3CC3)C2)=O)cc2ncccc2[nH]1 68212,C1(NC(C(C)(C)OCC)=O)C2CCC(C2)C1C(=O)NCC(O)C(=O)NC 68213,c1(C(=O)NCC2CC(CNC(C3(Cl)C(C)(C)C3)=O)C2)cc2cn[nH]c2cn1 68214,c12cc(ncn1)N(CC)C(=O)CC1CCN2C1.C(=O)(C(C)CSC)OCC#C 68215,c1(CN(C)Cc2oc(C(N3CCN(CC4CC4)CC3)=O)cc2C)ccc(C)nc1O 68216,C1(C)(NC(C(C2CCCCC2)NC(c2c(C)snc2)=O)=O)CCC2(CC1)CC2 68217,C1(C(N(C2CCC(NC(c3cncs3)=O)CC2)C)=O)COCCN1CC(F)(F)F 68218,C1(C(=O)O)CN(C(c2cc(Br)cc(Cl)c2F)=O)CC12CN(Cc1ccc(Cl)o1)C2 68219,C=C1CC2CC1CN2C(=O)C(C1(O)CN(C(=O)C(F)F)C1)F 68220,c1(SCC(=O)NCC(CNC(c2cccc(N)c2)=O)OC)cccc(F)c1 68221,C(CC(=O)N1CCCC1)NC(COCC(=O)N(CCOC)CC)=O 68222,C(c1cnc[nH]1)=CC(=O)NCC(CN(C(=O)Cc1ccno1)C)O 68223,N1(C(CC2(C)CCN(C(C(C(C)(C)C)OC)=O)C2)=O)CC2(CCNC2=O)C1 68224,c1(C(=O)NCC(CC)NC(C2CCCCC2C(N)=O)=O)ccnc(OC)n1 68225,N1(N2CCC(OCC#C)C2)CC2CCCC1C2C(=O)OC(=O)OC(C)(C)C 68226,N(C1CCc2ccc(F)c(F)c21)C(c1ccc(C)c(Br)c1C)=O 68227,N1(C(C2(CC#C)CCCO2)=O)CC(CNC(c2cc(C)ncn2)=O)C(O)C1 68228,Cc1nc2n(c1CC(N1CCC(Oc3c(C)cccc3Cl)CC1)=O)CCCC2 68229,c1(C(=O)NC2CN(C(Cc3nn(C)c(Cl)c3)=O)CC2F)cccc2c1CCCO2 68230,Cc1nnc(O)c(C(=O)NC(C2(O)CN(C(C3OCCC3C(C)C)=O)C2)C)c1C 68231,N1(C(C(C)=C(CC)C)=O)CC2CCC(CNC(C3(Cl)CC34CCOCC4)=O)(C2)C1 68232,C(=O)(C(C(C)(C)C)N(C)C)NCCC(C)N(C)C(c1ccc(F)c(C(F)F)c1)=O 68233,C1(N(C)C(C2CC(N(C)C)C2)=O)CCCN(C(=O)CCCN2C(=O)CCC2=O)C1 68234,C1(C(N2CC(C)(CNC(=O)Cc3ccon3)OCC2)=O)COc2ccccc2C1 68235,N1(C(C(CC2CCOCC2)NC(=O)Cc2cncs2)=O)CC2COCC2C1 68236,N#CC1(C(N2CC3(CCC3CNC(=O)CCCC3CCCC3)C2)=O)CCOCC1 68237,C=C(C)CCC(=O)N1CCC(N(C(=O)C(=Cc2cnc[nH]2)C)C)CC1 68238,C#Cc1cccc(C(N2CC(C(N3CC(CCO)(CC)C3)=O)C(F)C2)=O)c1 68239,C1(F)(CNC(COC(CC)C)=O)CCN(C(C2CCCCCCC2)=O)CC1 68240,N1(CC(N2C(CN(C(CC)=O)C)CCCC2)=O)C(=O)C(=O)N(C)C1=O 68241,N1(SCc2scc(CC(=O)NCC3(C(C)C)C(C(=O)OC)C3)n2)CCN(C)CC1 68242,C1(C(C)NC(=O)N(CCO)CCO)CCCC(C(F)(F)F)C1 68243,c1(OC)ncc(C(=O)NCC(C)N(C(=O)Cc2cncnc2O)C2CC2)cc1Cl 68244,c1(C(N2CCCCC(CNC(C3CN(C)C3)=O)C2)=O)cccc2c1CC(C)(C)C2 68245,Cc1ccc(Cl)c(OCC(N2CCC(=CCNC(=O)C3=NNC(=O)C3)CC2)=O)c1 68246,C1(CC)CN(C(C2CC23CCCCC3)=O)CCN1C(=O)CCC(C)(C)F 68247,C1(C(=O)NCC2(C)CCCN2C(C2(F)CCC2)=O)Cc2ccccc2S1(=O)=O 68248,N1(C(C(=O)NC2CCN(c3ccc(F)cc3F)C2)=O)CC2CCCCCC2C1 68249,C1(NC(C(C)CC2CCC2)=O)CCCC12CN(C(c1sc(F)cc1Cl)=O)C2 68250,C(=O)(CC(C(=O)NC(C)CC1CN(C(C2CC=C(C)CC2)=O)C1)NC(C)=O)OC 68251,c1(NC(c2ccccc2C)c2n(C(CC)C)nnn2)cncc(NC(=O)OC)c1 68252,Cc1cc2[nH]c(C(N3CC4=C(C3)CN(C(C3(C)CCCCN3C)=O)C4)=O)cc2s1 68253,c1(C(=O)NCC(C)CN(C(=O)CC2COC(=O)N2)C)ncc(Cl)nc1Cl 68254,Cc1cccc2c1CC(C(=O)NC1CC1)N(CC(O)CN1CCCC1)C2 68255,CCCC(O)C(CO)NC(=O)CC1(CNC(c2[nH]cc(C)c2C)=O)CC1 68256,C(=O)(C1=NNC(=O)CC1)N(C(C)CNC(c1cnc2n1CCS2)=O)C 68257,C=CCC(C(=O)N1CC(OCCNC(C2CC(CC)C2)=O)C1)c1ccccc1 68258,N1(C(=O)CCC2CCC2)CCCCC(C(=O)NC2(C3CC3)CCCC2)C1 68259,N1(C(C2(CC)CC2)=O)C2CCC1C(C(=O)NC(c1ncnn1C)C)C2 68260,C1(C(N(C2CN(C(C3(F)CC3)=O)CCC2O)C)=O)CCc2ccnn2C1 68261,Cc1csc(=NCC(=O)NC2CN(C(C3CS(=O)(=O)CC(=O)N3)=O)CC2(C)C)[nH]1 68262,N1(C(=O)Cc2cscn2)CCN(C(C2CC3(CCC3)CO2)=O)C(c2cn[nH]c2)C1 68263,N1(C(C2CC(C)(O)C2)=O)C2CCC1CC(F)(F)C2.c12ccc(cc1)Nc1noc-2n1 68264,c1(NC2CN(C(COC)=O)C2)[nH]c(=NC(C)c2nc(C)cs2)nc2sccc12 68265,Cc1cc(C(N2CC3OCC(NC(C4CCCN(C)C4)=O)C3C2)=O)c(Cl)cc1F 68266,C1(C(=O)NCc2c(CNC(C3(SCC)CC3)=O)c[nH]n2)CCC12CCCO2 68267,c1(N2C(C)(C)C(NC(=O)Cn3cncn3)CC2)cc(C#N)ccc1[N+](=O)[O-] 68268,N1(C(c2ccn(COC)n2)=O)CCN(C(c2cc(COC)on2)=O)CC1CF 68269,C(C)(CC(C)NC(c1ccnn1C1CCCC1)=O)NC(COCCOCC#C)=O 68270,c1(C(N2CCCC(C(C)NC(C3(SC)CCC3)=O)C2)=O)cc(C)nc(O)c1 68271,C12(C(=O)NCc3cn(C)nn3)CC1CCN2C(=O)Cc1cnn(C)c1 68272,Cc1ccc(F)c(NC(C2C3CC2N(C(n2nc(Cl)ccc2=O)=O)C3)=O)c1 68273,Cc1[nH]c(C(=O)NC(c2cc[nH]n2)C)c(C)c1C(=O)NC(C1CCCO1)C 68274,C1(C(N2C(CNC(Cn3c(C)c(Cl)cn3)=O)COCC2)=O)CCn2cnnc2C1 68275,N1(C(c2cc(C)c(C)[nH]2)=O)C2CCCC1CC(NC(=O)CC1C=CCCC1)C2 68276,N1(C(C(CC)O)=O)CC2(CCC2)CC1CNC(c1ccnc(-c2ncc[nH]2)c1)=O 68277,Cc1cc(C)n(CC(=O)NCC(C2(O)CCN(C(c3[nH]c(O)nc3C)=O)C2)C)n1 68278,C1(C(=O)NCC2(CC)CC2)C=CCN(C(=O)CC23CCC(CC2)C3)C1 68279,N1(C(CC(C)=C(C)C)=O)CCCC(C)(C(=O)Nc2cccc(Cl)c2)C1 68280,C(CC)(CC)(CCNC(c1c[nH]cc1-c1cc(C)no1)=O)NC(CCOC)=O 68281,C1(C(=O)NCC(=O)OCC)CN(C(c2ccc(N3CCNCC3)cc2)=O)CC1F 68282,Cc1cccc2c(=O)n(CC(=O)NCCCOCCNC(=O)CC3CC3)cnc12 68283,CCC(F)(C(=O)OC)C(=O)NCCCCNC(c1c(Cl)ccc(F)c1C)=O 68284,Cc1cncc(C(N2CCC(CCNC(c3nncs3)=O)C2)=O)c1 68285,C1(NC(c2c(C(C)C)ocn2)=O)CCN(C(=O)C=Cc2cnccn2)CC1C 68286,c1(C(N2CCC(NC(C(C)NC(N)=O)=O)C2C)=O)cc(N)cc(F)c1 68287,CCCCC(O)CC(=O)N1CC2C(CNC(=O)C=C(Cl)Cl)C2C1 68288,Cc1ccc(F)c(C(NC(=O)OC(C)(C)C)CC2(N3CCC3)CCOCC2)c1F 68289,C1(NC(=O)COCCc2ccccc2)CCN(C(c2cscn2)=O)CCC1CO 68290,c1(C(=O)NC2(NC(CC3(C(=O)OC)CC3)=O)CCC2)ccc(N(C)C)cc1F 68291,N1(C(C2C(C)CC2)=O)CCCC2CCN(C(=O)C=Cc3nccs3)CC12 68292,C1(NC(COCc2c(C)ncs2)=O)CCCN(C(c2cccc(F)c2F)=O)C1C 68293,C1(NC(C2(c3ccc(Br)cc3)CCCC2)C)CCSC2(C1)CC(C(N)=O)C2 68294,C(=O)(C1CCc2cccnc21)NC1(CNC(Cn2cc(CC)nn2)=O)CCOC1 68295,Cn1cc(C(=O)NCC2(NC(=O)CC3=CCOCC3)CC2)c2ccccc12 68296,CC(c1ccccc1F)=CC(=O)NCC(C(C)C)NC(C1COCCN1C)=O 68297,C1(N(C)C)CNCC(C(=O)NCCCOC2CC(F)(F)C2)C1 68298,N1(C(CCCOC(C)=O)=O)CC2CCC1CC2NC(=O)CC1CCCSC1 68299,C1(C(CO)NC(C2(NC(=O)COCC3CCC3)CC2)=O)CCCCC1 68300,c1(C(N(C)C)=O)ccc(CNC2(c3ccncc3)CNC2)cc1[N+](=O)[O-] 68301,C1(CC(=O)NC2CN(C(C=CCC)=O)CC2C(F)F)CC2CCC(C1)N2C 68302,c1(CCC(N2CC(C(C)NC(=O)C(CC)N3CCCC3=O)C2)=O)c(C)noc1C 68303,C1(NC(=O)CC2(O)CCC2)CC2CCC1CN2C(C1CNC(=O)N1)=O 68304,C#CCCCCCCCC(=O)NCC1(C)CCCN1C(c1cc(C)[nH]c(=NC)n1)=O 68305,C(=O)(CC(C)CC(C)(C)C)N(C(CC(=O)NCCc1ncc(C)cn1)(C)C)C 68306,Cc1ccc(C(=O)NC2CCOCC2NC(C23CC(F)(C2)C3)=O)c(F)c1F 68307,N1(C(C(C(C)NC(=O)C(N2CCNC2=O)C)(C)C)=O)CCC2CCCC2CC1 68308,C1(C(=O)NC23C(CN(C(C4(CC(=O)OC)CC4)=O)C2)C3)CCc2nc(C)[nH]c2C1 68309,Cc1nc(C(=O)NCC2C3CN(C(=O)CC(c4ccccc4F)C)CC23)oc1C 68310,c1(C(=O)NC)snc(C)c1N.CCCC1CC(C)C(=O)N1 68311,CN1CCC(NC(=O)C(C2CCC2)NC(c2cc3ccccc3o2)=O)C(C#N)C1 68312,C(=O)(C(C(C)O)NC(c1ccsc1)=O)N(CCNC(CCC)=O)CCOCCO 68313,c1(NC(CC2CCN(c3ncc(C)c(C)n3)CC2)=O)c(F)cc([N+](=O)[O-])cc1Br 68314,c1(C(N2CCCC(CCNC(C(C)=CC)=O)C2)=O)cccc2c1OC(C)C2 68315,CCC(C)(C(=O)N1CC(CCNC(=O)C(C)(C)C2CCCCC2)(OC)C1)OC 68316,N1(C(c2c(COC)ncs2)=O)CC(NC(=O)C=Cc2cccc(F)c2)CC1(C)CC 68317,CC(C(C)(C)NC(=O)CCC1CC1(F)F)NC(=O)C=CCN(C)C 68318,c1(C(=O)NCC2(F)CN(C(c3cc(C)[nH]n3)=O)C2)cc2sccc2s1 68319,O=C(C#CC1CCOC1)NCC1=CCCN(CC23CCC(CC2)CC3)C1 68320,N1(C(C(C)N(C(=O)CC2(C)OCCO2)C2CC2)=O)CCCC(C)(C)C1C 68321,N1(C(C)C)CC2CCC1CN2C(=O)CC1CC(NC(=O)OC(C)(C)C)CCO1 68322,N1(C(C2(CC=C)CCN(C(=O)C(C)OCCC(C)C)C2)=O)CCC(O)CC(C)C1 68323,N1(CC)CCN(C(C2CCN(C(=O)CCC(C)(N)Cl)C(C)C2)=O)C(C)C1 68324,c1(COC(=O)NC2CCCC(NC(=O)NC)C2)ccc(C#N)cc1 68325,N1(C(COCCC)=O)CC(NC(=O)C(C(C)(C)C)c2cn[nH]c2)CC1(C)C 68326,CCCCCCOCC(=O)NCC1(NC(=O)CCc2cnc(O)[nH]2)CCOC1 68327,CN1CCC(C(N2CCC(N3CC=CC3)CC2)C(=O)NCc2ccco2)CC1 68328,c1(C(=O)NCC(CC)(CC)NC(=O)CC2CCCN2C)c[nH]cc(F)c1=O 68329,C1(NC(c2cncc(F)c2)=O)CN(C(=O)C#CC2CCCO2)C2(CCC2)C1 68330,C1(CN(C(=O)C=CC(F)(F)F)CC)CCCN1C(=O)C(F)OC 68331,C1(C2CC2)(CNC(COCCC)=O)CCN(c2ncnc(Cl)c2C(=O)OC)C1 68332,c1(C(=O)NC2CCC(NC(CCOCC#C)=O)CC2)cc2ccc(Cl)c(F)c2[nH]1 68333,N1(C(CCS(C)=O)=O)CCCC2CN(C(C3CCc4c(nnn4C)C3)=O)CCC12 68334,C1(C#CC(=O)N2CC(O)(NCC3CC4(NCc5ccccc5)C3C4)C2)(CC)COC1 68335,N1(C(c2nn(C(CC)C)c(C)c2)=O)CC(NC(=O)C=CS(C)(=O)=O)CC2(CC2)C1 68336,Cc1cccc(C)c1NC(=O)C(C)NC1CCC(NC(=O)CC(C)(C)C)C1 68337,c1(CC(N2CC(CC(=O)O)C(NC(=O)C(F)(F)F)CC2)=O)c[nH]c2nccc(Cl)c12 68338,Cn1c(O)nc2cc(C(N3CCN(C(C4(C)CCCO4)=O)CC(O)C3)=O)cnc12 68339,Cc1noc2ncc(C(=O)NC3CC4CC3N(C(c3ncccn3)=O)C4)cc12 68340,CC1(C)CC(C)(CNC(c2nn[nH]c2Cl)=O)CN1C(=O)CN1CC2CC2C1 68341,c1(NC(c2c(C)cccc2)C)cc(Br)ccc1S(=O)(=O)N(C)CCC1CCCC1 68342,Cc1cc(Cl)ncc1CC(N1CCC(CNC(C2CCC2C)=O)C(C)C1)=O 68343,C(=O)(CC(C)CC(C)(C)C)N(C(C1ON=C(C(C)C)C1)=O)CC1CCN(C)CC1 68344,Cc1cc(C(=O)N(C(C)CNC(=O)CC2COC3CC2C3)C)oc1Br 68345,C(=O)(C1=CC2C=CC1C2)N1CCC(C)CC1CNC(c1cccc2c1OCC2)=O 68346,C1(NC(COC(C)=O)=O)CCC(C)(CNC(=O)Cc2csnc2C)C1 68347,C1(=CC(N2CCC(NC(C(CCC)CC)=O)C2)=O)CC2CCC(C1)N2C 68348,C#CCCCCCCC(=O)NCC1(C)CN(C(c2ocnc2C(C)C)=O)CCO1 68349,N1(C(C(=O)NCC)=O)CCN(C(=O)C(C)CC(N)=O)C2CCCC2(C)C1 68350,C(=O)(C1=CS(=O)CCC1)NC12CCC(n3cc(N(C)C)nn3)(CC1)C2.C12CC1C2 68351,c1(OCC(=O)NCC2COCCN2C(=O)COC(F)F)ccc(Cl)cc1Br 68352,c1(C(N(C)CC2(CNC(=O)CCC3CCCC3)CC2)=O)ccnc(Cl)c1Cl 68353,c1(C2(ON)COC2)cccc(OCCCOC(c2cccc(Cl)c2)=O)c1 68354,N1(C(c2cc(CNC(c3c(C)c[nH]n3)=O)no2)=O)CC(O)C(O)C1 68355,C1(CCOC)CN(C(c2cnnc(C)c2)=O)CCN1C(=O)C(O)C(C)(C)C 68356,c1(C(=O)O)ccc(F)c(C(=O)NCC2CN(S(=O)(=O)CC3CC3)C2)c1 68357,c1(C2(CNC(=N)NC(c3cccc(F)c3)CF)CC2)ccc(F)c(F)c1 68358,c1(CC(N2CC(F)(CNC(C3(CCOC)CCCC3)=O)C2)=O)cc(F)ccc1C 68359,C1(NC(=O)NC(CSC)(C)CO)C(=O)NCCC1C 68360,C1(C2CC2)(C(N2CC(n3nc(C)oc3=O)C2)=O)CN(C(=O)C)C1.Cc1nonc1 68361,c1(C(=O)NC2(C)CC(NC(=O)CC3CCC(F)(F)CC3)C2)ccc2nonc2c1 68362,CC(C)(C)CC(O)CC(=O)NC1CCCCC1NC(c1cc2cccnn2c1)=O 68363,C(C)(N=c1ccnc(NCC2CC2(C)C)[nH]1)c1ccc(SC)cc1 68364,CCC(C)CCC(=O)NCC(C)(CNC(c1ccc(F)cn1)=O)OC 68365,CCC(CC(=O)NCC(O)C(=O)NCc1ccncn1)C(F)F 68366,C(=O)(C#CC(C)(C)CNC(=O)CSC(C)(C)C)NC(CCC)CC 68367,C(=O)(C1=C(Cl)CCC1)N1C(C(C)NC(=O)CCOCC(F)F)CCC1 68368,C1(N2C(=O)CC(N(C)C(c3ccc(Br)o3)=O)C2)CCN(CC2CCCC2)CC1 68369,CCCCC(C(=O)NCC1(CC(C)C)CCC1)NC(c1cn(C)nn1)=O 68370,CC(C)CCCC(C)CNC(C1CCCCC1(C)NC(=O)CC(C)C)=O 68371,N1(C(CN(C2CCC2)C)=O)CCN(C(C2CC23CCOC3)=O)CC(O)C1 68372,Cc1c(C(=O)NCC2C3CC2N(C(C2CCCN2N=O)=O)C3)cncc1N 68373,C=CCCCCCC(=O)NC1(C2CC2)CCN(C(c2ccc[n+]([O-])c2)=O)C1 68374,N1(C(c2c(C)ccc(=N)[nH]2)=O)CC2CCCC2(NC(c2csc(C)c2C)=O)C1 68375,C1(CC(=O)N(C2CCN(C(=O)CCC(C)SC)C2)CC)C(C)(C)C1(C)C 68376,N1(CC(=O)NC2CN(C(C3(F)CCCOC3)=O)CC23CC3)CCS(=O)(=O)CC1 68377,C1(CC(=O)NC2C(NC(=O)C(c3cn[nH]c3)=O)C2)COCCN1CC(F)(F)F 68378,Cc1cc(=N)[nH]cc1C(=O)NCC1(CNC(=O)C(C)(C)C(C)C)CCC1 68379,c1(CC)nc(C(=O)NCC2(C(C)(C)O)CN(C(c3csc(O)n3)=O)C2)c(C)o1 68380,N1(C(C(C(C)C)OCC(C)C)=O)CCC(NC(c2cncc(F)c2Cl)=O)C(C)C1 68381,C(C1=NOC2CN(C(=O)CCCc3ccccc3)CC12)NC(CCC=CC)=O 68382,N1(C(CC2C(=O)OCC2)=O)CC(O)(C2CCN(C(=O)CCC3CC3)CC2)C1 68383,C(C(C)(O)C(=O)N1CCCC(CN(C(=O)C=C2CCOCC2)C)C1)OC 68384,C1(CN(C)C(C2CCO2)=O)CN(C(=O)CCCNC(C2CCCC2)=O)CC12CC2 68385,N1(C(c2c(OC)ccs2)=O)CC2=C(C1)CN(C(=O)CC1C=NN(C)C1=O)C2 68386,c1(NC(=O)Nc2cc(C)sn2)cccc(CC2CC2)c1 68387,C1(N(C(C2(C(N(OC)C)=O)CC2)=O)C2CC2)CN(C(=O)Cc2ccc[nH]2)CC1F 68388,C1(C)(CNC(CC(C)CF)=O)CCCN(C(c2cc(NS(C)(=O)=O)ccc2O)=O)C1 68389,c1(OC)cc(NC(C2(F)CCN(C(c3ccc(Br)c(Cl)n3)=O)CC2)=O)nc(Br)c1 68390,C12(CNC(C=CCC(C)(C)NC(c3ccc(CO)nc3)=O)=O)CC(C)(CCO1)C2 68391,c1(C(=O)NC2CC(NC(CNS(CCC)(=O)=O)=O)C2)cc([N+](=O)[O-])ccc1O 68392,C(=O)(C#CC1CCCC1)NCCN(C(C(CCC)(F)F)=O)CC 68393,C(C(C)(C)CC(=O)N(C)CCc1ccccc1)NC(C(OC)OC)=O 68394,C#CC(C(C)C)NC(=O)C(C)N(C(=O)C(N)=O)C 68395,C1(CNC(c2c(CC)nn(C)c2)=O)CCN(C(C2C3COCC23)=O)C1(C)C 68396,N1(C(C(CC)SC)=O)CC2CC(NC(=O)Cc3ncc(F)cc3F)C2C1 68397,c1(C(=O)NCC(CCCC)NC(C=CCC)=O)ccc(P(C)(C)=O)cn1 68398,Cc1nn(C)c(C)c1NC(C1CCN(C(c2ccc(C(F)(F)F)cc2I)=O)C1)=O 68399,C1(NC(C(C2CC2)NC(CCNC(N)=O)=O)=O)CN2CCC1(C)CC2 68400,N1(C(CCC(CCCC)O)=O)CCc2sccc2C1CNC(=O)C=CCOC 68401,CC1CN(C(=O)C(C)NC(C2(O)CCOCC2)=O)CC(=O)N1 68402,c1(C(=O)NCCN(C(c2c(CO)noc2C)=O)CC)cc2n(n1)CCCC2 68403,N1(C(CCC2(NC(CSCCC(C)C)=O)CCC2)=O)CCOC(C(C)(C)C)CC1 68404,c1(C(=O)NC2(CNC(c3c(C)[nH]cc3)=O)CCOC2)cc(C)n(CC(F)F)c1C 68405,C(=O)(C1=NOC(CN)C1)NC1CC(N(C(=O)CC(C)(C)c2ccc(F)cc2)C)C1 68406,C1(C(N2CCN(c3cncc(C4CC4)n3)CC2)=O)CC2OC1C1CC21 68407,Cc1cccc(C(N2CCN(Cc3ccc(F)c(F)c3)C(C)C2)=O)c1C 68408,c1(OC)cc(CN(C2CCN(C(C3CN(C)C3)=O)C2)C)c([N+](=O)[O-])cc1O 68409,C(C(C(=O)N1CC(C(O)C(=O)NCCNC(=O)CO)C1)C(C)(C)C)NC(C)=O 68410,C1(NC(c2cccc(C3CC3)c2)=O)CC1C1CCCN(C(c2cccnn2)=O)C1 68411,c1(OCC(=O)NC2C(NC(c3cc(CC)on3)=O)COC2)ccc(Cl)cc1C 68412,C1(OC)CC(CNC(=O)CN2CCCOC2=O)N(C(=O)CN2C(=O)CNC2=O)C1 68413,N1(C(C=CCOC)=O)CC2CCCC2(CNC(=O)CCCCNC(N)=O)C1 68414,c1(C(C2CCCN(C(C3(C(=O)NC4CC4)CCC3)=O)CC2)=O)nc2ncccn2n1 68415,N1(C(CC(=C)C)=O)CCC(CNC(c2cncc(NS(C)(=O)=O)c2)=O)CC1C 68416,c1(OC)ccc2oc(C(N3CC4CC3C4C(=O)Nc3cccnc3C)=O)cc2c1 68417,c1(C2CCCN(C(=O)NCC(C(C)(C)C)CO)C2)ccccc1[N+](=O)[O-] 68418,N12CCn3cc(nc3C1)C2=O.C1(NCC)CCCCC1NC(C)=O 68419,CC1CC(CNC(=O)C(=O)N(C)CCO)CN1C(=O)Cn1cnc(C#N)n1 68420,O=Cc1ccc2cc(-c3nc(CCCF)no3)[nH]c2c1 68421,C1(C(=O)NC(C(=O)NCC2CC=CC2)c2cccs2)(C2CC2)CCCO1 68422,c1(CS(=O)(=O)NC(c2nncs2)CC)cccc(F)c1 68423,N1(C(=O)NC(C)CCC(=O)O)CC(C)(C)C(O)C1 68424,C12(NC(CC3C(C)=NNC3=O)=O)CCC(CC1NC(c1ncccc1Cl)=O)C2 68425,C1(NC(CC2N(CC)CCOC2)=O)CCN(C(=O)C2=CCSC2)CC(C)(C)C1 68426,C1(OC)(NC(=O)C(c2ccc(C)cc2)OC)CS(=O)(=O)C1 68427,c1(CN2CCC(NC(c3cccc(-c4nc[nH]n4)c3)=O)CC2)c(Cl)cc(Cl)cc1Cl 68428,C(=O)(C1=NOC2COCC12)N1C2C(NC(CCNC(N)=O)=O)CC(C2)C1 68429,c1(CNC(CSCC(C)C)=O)nc(CNC(=O)C(C)(C)c2cncs2)cs1 68430,CC1CCN(C(C2CCCC2(C)C)=O)CCN1C(c1cnco1)=O 68431,CCCCC(C(=O)NCCC1CCCCN1C(=O)CN(C)C)C(C)C 68432,n1(CC(=O)N(C(c2ccccc2)CNC(c2cnnn2C)=O)C)nnc(C2CC2)n1 68433,C(CCCCCNC(c1c(Br)nnn1C)=O)NC(CC1ON=C(C)C1)=O 68434,C(CCCC(=O)OC)(C(=O)NC1CC1)N1CCCC(COC)C1 68435,C1(C(N2CCC(F)(CNC(CCC(C)C)=O)C2)=O)CCn2ncnc2C1 68436,Cc1cc(C(N2CC3C(C(=O)Nc4ccnc5c4OCO5)C3C2)=O)c(C)cc1F 68437,C(=O)(C1=CC2C=CC(C1)C2)N(C1CCN(C(c2ncoc2CC)=O)C1)CCC 68438,N1(C(c2cc3ncccc3o2)=O)CCC2(CCCN2C(c2c[nH]c(=O)cn2)=O)C1 68439,S(=O)(=O)(c1cn(C2CCCCC2)nc1OC1CNC1)N(C1CCC1)C 68440,C(=O)(C(O)CC(C)(C)C)N(C1CCN(C(C2CCC2CF)=O)CC1)CCOC 68441,C1(C(N(CCC(=O)OCC)C)=O)CCOCC1NC(C1OC2CCC1C2)=O 68442,c1(C(=O)NCC2CN(C(CC3(C)CC3F)=O)C2)ccn2c(O)nnc2c1 68443,C(C(COC)C(=O)NC(CO)C(=O)NC1CC(C(C)(C)O)C1)OC 68444,c1(C(=O)NC2CC(NC(c3cc(Cl)ccn3)=O)C2)ccc(Cl)cc1F 68445,C12(COC)CC(CSC3CCC3)(CN1C(c1ccc(Cl)c(C)c1)=O)C2.C1C(=O)N1 68446,C1(NC(C2(CCNC(C(CC)(C)C)=O)CC2)=O)CC2CC1C(O)C2O 68447,C1(NC(COCCOCC)=O)CN(C(c2ccn3ccccc23)=O)CC12CCCC2 68448,N1(C(c2ccc(C3CC3)nc2O)=O)CC2CCCN(C(c3cccnc3)=O)C2C1 68449,Cc1cc(C(=O)N(CC(C)CNC(c2c(C(F)F)cnn2C)=O)C)sc1C 68450,C(C(=O)N1CC(NC(=O)CCC2CCCC2)C(C)C1)(C(C)(C)C)NC(C)=O 68451,N1(C(C2(COC)CC2)=O)CCCCN(C(c2ccnc(C)c2)=O)CC1 68452,c1(-c2occ(CC(=O)NCCN(C(c3c(CC)nco3)=O)C)n2)ccc(O)cc1 68453,Cc1cc(CC(=O)NC2CCCC2n2cc(C3CC34CC4)nn2)cc(C)c1Br 68454,n1(C)cc(Cl)cn1.c1(C(C2CC2)NCC(C)SC)nnnn1C1COC1 68455,c1(C(=O)NC2C(NC(c3sc(CC)c(C)c3)=O)CC2)ccc(F)c(F)c1C 68456,C1(C(=O)NCCNC(CN2CCN(CC)CC2)=O)CC(C2CCCC2)C1 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68565,C1(C2CCCCO2)(CN(C)CC2CC2)CCCO1 68566,C1(CC)CCCC1C(=O)NC(C)CC1CN(C(c2cc(-c3ccco3)c[nH]2)=O)C1 68567,C1(NC(=O)C=CCN2CCCC2)CCN(C(c2c(C(=O)NCCO)csc2)=O)C1 68568,c1(OC)ccnc(C(N2CC(NC(c3cn(CCO)nc3C)=O)C(C)C2)=O)c1O 68569,C(=O)(CCCC(C)SC)NCCN(C(CC1(OC)CCCC1)=O)CCCN(C)C 68570,c1(NC(c2cccc(C)c2)CNC(C2CCC3CC3C2)=O)cc(C)nc(C)n1 68571,N1(C(CCC=CCC=C)=O)CCOCC(CNC(=O)C(C)SC(F)(F)F)C1 68572,c1(C2(C(F)(F)F)CC(=O)C2)ccc(C(N2CCCC2c2ccccc2F)=O)cc1 68573,C1(CC(=O)NCCC(C(C)C)NC(=O)C(C)(C)CO)SC2=NCCN2C1=O 68574,c1(NCCCN(C(CCc2onc(COC)n2)=O)C)ncnc(O)c1Br 68575,c1(CC(N2CCC(CCCNC(C=C(CC)C)=O)CC2)=O)ccc(F)cc1F 68576,C(=O)(CC(C)(O)C(F)(F)F)N1C(C)CN(C(C2CC(O)C2)=O)CCC1 68577,c1(NC(CC2N(C(c3cc(C)[nH]c3)=O)CCC2)=O)ccccc1C(C)(C)C 68578,c1(N(CCC)CCOC(c2csc(CC(C)C)n2)=O)ncnc2c1ncn2C 68579,C=CCC(CC(C)C)C(=O)N1CC2(C1)CN(C(C1CCCCC1CC)=O)C2 68580,C12(C(N3C(CN(C)C(c4cnc(Br)s4)=O)CCC3)=O)CCC(C)(C1)OC2 68581,N1(C(C(CCSC)OC)=O)CCCC(C)C1CNC(=O)CCOC1CCCCC1 68582,c1(CN(c2cccc(F)c2)C(CCSC2CCC(C)CC2)=O)c(F)cccc1F 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68600,C12(C(=O)NCCC3(CNC(C(C4CC4)OCC)=O)CC3)CC(C)(C1)OC2C 68601,C12(C(=O)NCC3OCCN(C(CS(N)(=O)=O)=O)C3)CCCC(=O)N1CCC2 68602,C1(NC(C2(CC(C)=O)CC2)=O)CC2CCC(C1)N2C(C1CCCCC1(C)C)=O 68603,N1(C(CC(CCC)C)=O)CC(C)N(C(=O)CC(C)(C)C(F)F)C(C)C1 68604,C1(C(=O)NC2(CF)CCN(C(C3N(C(=O)NC)CCC3)=O)C2)CC2C(C1)C2(F)F 68605,C1(NC(C(CCC)NC(N)=O)=O)CC(OC)CN(C(c2c(O)cccc2F)=O)C1 68606,C1(C(C(=O)NCC(CC)O)F)CCN(C(=O)CSC2CC2)C1 68607,Cc1cnc(NC(C2CCN(Cc3ccc(Cl)cn3)CC2O)=O)nc1Cl 68608,c1(CN=[N+]=[N-])ccc(CNC(C2(CCN)CCCC2)=O)cc1 68609,c1(C(=O)NC(CC)CNC(c2nncs2)=O)ccccc1NC 68610,CC(C)CC(CC(C)C)C(=O)N1CC2(CCCC2NC(c2ccc(=N)[nH]n2)=O)C1 68611,c1(CC)cc(NC(C2CCCN(CC3(CC(=O)OC)CC3)C2)=O)cnc1C 68612,c12nncn1NC(=O)N(CC#C)C2.C1(CC)CCNCC1Oc1ccccc1 68613,N1(CC)CC(NC(C2C(CNC(c3ccc(=N)[nH]n3)=O)C2(C)C)=O)CC1=O 68614,Cc1ccc(C(=O)NCCOC2CCN(C(=O)C3=CCCO3)CC2)nc1F 68615,N1(C(CCc2c(C)noc2)=O)CCC(CF)(NC(=O)Cc2nccn2C)C1 68616,C(=O)CCCC(F)(F)F.C12(CCn3cc(C(N4CCCC4)C)nn3)CCCCC1C2 68617,N1(C(c2cn(CCOC)nc2)=O)CC2CCC1CN2C(=O)C(=O)NCC(F)(F)F 68618,N1(C(C(C(C)C)=O)=O)C(C(=O)N(C)CCc2cnc[nH]2)CCC12CC2 68619,c1(C(=O)NC(C(C)C)C(=O)N2CC(O)CC2CO)ncn2ccccc12 68620,c1(CC(N2C(CCNC(=O)C=Cc3cocn3)CCC2)=O)cccc2c1CCC2 68621,c1(OC)ncc(C(=O)N(C2CCC(NC(c3scc(C)c3C)=O)C2)C)cc1Br 68622,N1(C(C2(C(C)C)CCC2)=O)CC=C(CC(=O)NCC2CCNC(=O)C2)CC1 68623,N1(C(C=Cc2c(C)noc2C)=O)CC2CC(O)C1C2NC(C1CCSCC1)=O 68624,C=CC(F)(F)C(=O)NCC=CCNC(=O)C=CCN(C1CC1)CC 68625,C1(O)(CC(=O)NCCNC(C2(CN(C(C)C)C)CC2)=O)CCCC1 68626,C1(NC(=O)COC2CCCOC2)CC2CC(NC(=O)Cc3cnoc3)CC12 68627,C=CCCC(F)(F)C(=O)NCCNCCCCNC(c1cn2cc(C)nc2s1)=O 68628,CC1c2c[nH]nc2CCC1C(=O)NCCNC(c1scnc1Cl)=O 68629,C1(C(=O)NC(COC)(C)C)CCN(C(=O)C(C)COC)O1 68630,C=CCCCCCCC(=O)NC1CCC(CNC(c2ccnc3ccnn23)=O)C1 68631,N1(C(c2cc(CN3CCCC3)c[nH]2)=O)CC2(C1)CN(C(C1CC(O)C1)=O)C2 68632,C(C(C)(C)CC(=O)NC(C)CCO)NC(Cn1c(C)nc(C)n1)=O 68633,c1(CC(C)C)cccc(NC(C2COCC2NC(=O)CCc2ccn(C)c2)=O)c1 68634,N1(CC)CCCC(C(=O)NCCC2CC(C(=O)NC(C)(C)C(F)(F)F)C2)C1 68635,S(=O)(=O)(c1c[nH]c(=NCCC#CBr)cc1C)NC(CC)C1CC1 68636,Cn1c(=O)[nH]c(NCC23CC(CNC(=O)CNC=O)(CO2)C3)c(C#N)c1=O 68637,C1(C(=O)NCC(C(C)C)NC(=O)CCCC2CC2)CCC(C(=O)N(C)C)CC1 68638,CC(C)(C)C#CC(=O)NCC(CC(=O)NCC1OC(=O)CC1(C)C)OC 68639,c1(CNC(=O)NC2CC3(CC(C)OC3)OC2)ccc2c(c1)CN=S2(C)=O 68640,c1(C(N2CCC(O)(CNC(C3CCCN(C(C)=O)C3)=O)C2)=O)c(C)cc(C)nc1O 68641,C1(CC)(NC(C2CCCCC2NC(=O)C(C)C(C)(C)C)=O)CCCCCC1 68642,C12(CNC(=O)CCCc3cc[nH]n3)CCC(CC1)N2C(=O)CN1CCCCCC1 68643,c1(CC(=O)N(CC(C)NC(c2csc(COC)n2)=O)CC)ccccc1C 68644,C1(CC(c2ccccc2)N(C(=O)CCCOc2ccccc2)C)CCCC2CC12 68645,N1(C(C(C)n2cncn2)=O)CCOCC(NC(C2C3C4CCC(C4)C23)=O)C1 68646,c1(CC=C)cccc(C(N2CCC(O)(CCNC(=O)C(F)=C(C)C3CC3)C2)=O)c1 68647,C(C)(C)(CCCNC(C1(CC)CCC1)=O)NC(C(CC)n1cncn1)=O 68648,C1(C)(C(=O)NCCSC(C)C)CCCN(CC2(CC(=O)O)COC2)C1 68649,C1(NC(c2ccc(-c3ncc[nH]3)nc2)=O)C2CC1N(C(=O)Cc1cnc[nH]1)C2 68650,Cc1cc(OCC(N2CC=CC(NC(c3snnc3C)=O)C2)=O)ccc1F 68651,c1(CC(=O)NC2CCCN(C(Cn3ccc(C)n3)=O)C2)c(F)c(F)cc(F)c1F 68652,C(CC(C)C)(CC(C)C)NC(CCNC(=O)OCC)=O.C(=O)(CC)N(C)CCS 68653,C(=O)(C(CC(C)C)C(N)=O)NC1N(C(C(CC#C)C2CCCCC2)=O)CCOC1C 68654,N1(C(C(COCCOC)F)=O)CCCC(N2CCN(C(c3nccs3)=O)CC2)C1 68655,N1(C(Cc2cc(C)nn2C)=O)CCC2CN(C(=O)CCS(N)(=O)=O)C(C)C12 68656,c1(NCc2n(C)nnc2Br)ccc2c(c1)C(C)(C)CC2(C)C 68657,CCCCCCC(C)CC(=O)NC1(C)CN(C(c2c[nH]nc2CC)=O)C1 68658,C1(C(N(C(C)C(N)=O)C)=O)CC12CCN(C(=O)Cc1cnsc1)CC2 68659,CC(C)(C)CCC(=O)NC1(CC(N)=O)CCN(C(=O)CC2COCC2(C)C)CC1 68660,c1(C(N(C2CCC(NC(c3ns[nH]c3=O)=O)C2)C)=O)cc(Br)cs1 68661,CC(c1ccc(F)cc1F)=CC(=O)N(CCCCNC(C1CC2CC2C1)=O)C 68662,C#CC1(C(N2CCC(C(C)O)CC2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)C1 68663,C(CN=[N+]=[N-])N(C(C1(C(C)NC(=O)C=C(C)C)CC1)=O)CC 68664,c1(C(CC)(C)C)cccc(N(C(=O)C(N2CCCC(C(O)OC)C2)=O)C)c1 68665,c1(C(N2CC(OC)CC2(C)CNC(C2CCC2)=O)=O)cccc2[nH]cc(Cl)c12 68666,CCC(C)C(CC(=O)N(C1CCC(=O)N(C)C1)C)NC(c1ccncc1C)=O 68667,N1(C(C(C(C)(C)C)OC)=O)CCC2(CC1)CC2C(=O)NCCN1CC2CC2C1 68668,c1(OC)ccccc1C1C(=O)N1.C1(O)(C(N2CC(F)(c3nn[nH]n3)C2)=O)CCOC1 68669,C1(CNC(C=CC(C)C)=O)CC2(CCN(C(=O)CCOc3ccccc3)C2)CO1 68670,C=CCC(C(=O)NCC(CC(C)C)NC(C1(c2ccc(F)cc2Cl)CC1)=O)C(C)C 68671,N1(C(C=CC)=O)CCC(O)(C(C)NC(c2c[nH]c(C)cc2=O)=O)CC1 68672,C(C(O)C(F)(F)F)N(C(C1C(CNC(c2cc(C)[nH]c2)=O)C1(C)C)=O)C(C)C 68673,c1(OCC)cc(C(=O)NCC(CNC(=O)CCC(C)OC)CO)ccc1C 68674,CC#CCS(=O)(=O)c1cccc(C(=O)NC2(CNC(=O)CSC)CCOCC2)c1 68675,C1(=O)CCCCCCO1.C(C(F)(F)F)(C1CCCC1)NC(C)(C)C 68676,C1(NC(c2c(CC)noc2)=O)CCCC12CN(C(=O)CCc1cnco1)C2 68677,C(=O)(C(CNC(C1CC1C(F)(F)F)=O)CC(C)C)NC(c1nc[nH]n1)CC 68678,Cc1ccc(Cc2c(Cl)cn(Cc3nc(C)ccc3C)n2)c(F)c1 68679,N1(C(C(C(=O)OCC)OC)=O)CC(C(N2CCN(C(C)C)CC2)=O)C2(CCC2)C1 68680,Cc1nc(O)sc1C(=O)NCCC1CC(C(=O)NC(C)C)C1.C12(CC1)C(=O)N2 68681,CC1CN(CCO)CC1N.c1(C(=O)NS(C)(=O)=O)ccccc1N(CCO)CCO 68682,c1(C2C(=O)NCCN2C)ccc([Si](C)(C)C)s1.N1(CC2CC2)CCCC1 68683,C1(C(=O)NC(C)CCCNC(=O)COCC2CC2)C(C(F)(F)F)C1[N+](=O)[O-] 68684,N1(C(C2N(C(c3c(CC)nn[nH]3)=O)CCC2)=O)CCC(C)(C2CC2)C1 68685,C=CC(C)(O)CC(=O)NC(CNC(=O)C(C)Sc1ccccn1)CC 68686,N1(CCNC(C(CC)CC2CCCC2)=O)CCN(CC2(C)CCNC2)CC1=O 68687,CCN=C(NCC1(CC)CCC(=O)N1)N1CCC2(C1)CC2(F)F 68688,C1(Nc2cc(N(CCC(C)CCO)c3ccccc3)ncn2)CC2CCCC(C1)C2 68689,C(C)(C)(CCC(=O)N1CCC(C)(C(=O)NCC2(C)CCC2)C1)N(C)C 68690,C=CC1COCC1NC(C1CSCN1C(=O)C(C(=O)OC)OC)=O 68691,C1(NC(C=Cc2scc(C)n2)=O)CCCC12CCN(C(=O)Cn1nnnc1C)C2 68692,N1(C(C(=O)NCC2CC2)=O)CCC2CC12C(N1CCN(CCF)CC1)=O 68693,c1(C(C)=O)ccc(C(=O)NC(C2CCCN2C(=O)Cc2cc(C)no2)C)cc1 68694,C1(C(=O)NC2CCN(C(C3COC(=O)O3)=O)CC2)CCc2ncncc2C1 68695,C1(CNC(C(c2cn(CC)nc2)(F)F)=O)CC(C)N(C(=O)CSCC(N)=O)C1 68696,C1(C(=O)NC(C2N(C(C(=CC3CCCC3)C)=O)CCC2)C)CCCCCS1(=O)=O 68697,C1(SC)CC(N=c2cc(C)nc(N3CC=CCC(C)(C)C3)[nH]2)C1 68698,N1(C(c2c(C)cc[nH]2)=O)C2CCC(C2)C1CC(=O)NCCNC(=O)C(F)(F)F 68699,c1(C(=O)NCc2cn(C)nc2)ccc(Cl)cc1NCc1cn(CC(=O)O)nn1 68700,c1(C(=O)NCCCC2(NC(CC(=C=C)C)=O)CC2)cccc2c(C)[nH]nc12 68701,C1(C(=O)NC(C2(O)CCCCC2)CC)CCCN(C(c2ccc(Br)nc2C)=O)CC1 68702,C(=O)(C1=NN(CCOC)C(=O)CC1)N1CCC(O)(CN(C(CSCC=C)=O)C)C1 68703,C1(NC(C(CNC(C)=O)(C)C)=O)CN(C(=O)C(C)(C)CO)CCC1CO 68704,N1(C(C(=O)N(CC(F)F)C)=O)CCC(C(=O)N(C)C)(C(F)F)C1 68705,CCCC(C(O)C(=O)N(C)CC1(C)CC1)NC(=O)C(C)N1CC(C)C1 68706,N1(CCNC(CC2CC(NC(C=CC=CCC)=O)C2)=O)CCOC1=O 68707,C12(NC(C(c3nccc(C)c3)(F)F)=O)CCC(CNC(=O)C(C)O)(C1)OC2 68708,C1(C(CNC(Cc2c(C)ocn2)=O)(C)C)CCN(C(C2(O)CCC2)=O)CC1 68709,N1(C(C=Cc2c(C)n(C)nc2)=O)CCCC(NC(=O)Cc2cncn2C)C(F)C1 68710,C1(C)(Nc2cc(CN(C(=O)CCSCC(N)=O)C)oc2)CCCCCC1 68711,c1(C(=O)NCCN(C(=O)CC2(C)CCCC2)CCC)ncc(C(C)(C)C)o1 68712,C1(CC(=O)N(CCCOC)C)CCN(Cc2cn(C)nn2)C1 68713,CCCCCCC(=O)N(CC(=O)NC(CC)C(=O)OCC)CC1CC1 68714,c1(C(C)C)c[nH]nc1C(=O)NCC(C1CC1)NC(=O)CCN1CCC(F)C1 68715,Cc1ncc(CCC(=O)N(CC(O)CNC(c2sccc2C2CC2)=O)C)s1 68716,CC1C(C(N2CCC(C)(N(C)C)C2)=O)CCCN1C(C1CC2CCC(C1)O2)=O 68717,C1(CNC(c2c(C)n[nH]c2C)=O)CCN(C(C2CC2c2cnnn2C)=O)CC1C 68718,C1(CC(N2C(C)C(NC(=O)CC3(CO)CC3)CC2)=O)CSc2ccccc2O1 68719,C1(F)(CNC(c2nc(C(C)=O)sc2)=O)CCC(CNC(=O)Cc2cnoc2)CC1 68720,C1(COC)CCCCCN1C(C(=O)NC1CC1)C1CC1(Br)Br 68721,c1(CCC(=O)NCC(C)NC(Cc2ccc(C#C)cc2)=O)ccc2c(c1)CCO2 68722,N1(C(C(C)NC(=O)NC)=O)CCCCC(NC(=O)CNc2ccc(Cl)cc2)C1 68723,C1(C(=O)NCCC(C(=O)OC)C)CC(C)(C)CN1C(c1ccn(C(F)F)n1)=O 68724,C(CCC(C)CC(=O)N1CC(NC(C2(C)CCC2)=O)C2CC2C1)=C(C)C 68725,C1(CCNC(c2c(CC)occ2)=O)CN(C(=O)C(c2cccc(C)c2)O)CC1C 68726,C1(Cn2cc(CC3(SCC)CC3)nn2)CN(C(=O)CCc2ccccc2C)CCO1 68727,N1(C(c2c(CC)ccc(F)c2)=O)CC2(CCCC(CNC(=O)OC(C)(C)C)O2)C1 68728,C1(NC(C2(C)CC(C)(C)C2)=O)CCN(C(=O)CC2CCC(C)(C)O2)CC1O 68729,C1(C(F)(F)F)(NC(C2CCN(C(c3cc(Cl)nc(Cl)c3)=O)C2)=O)CCCCCC1 68730,CSC1=C(C(=O)NCC2CN(C(=O)Cc3nonc3C)CC(C)(C)C2)CCCC1 68731,c1(N2CCC(CC=C)(NC(C3CCC=CO3)=O)C2)nc(Cl)nc(C)c1[N+](=O)[O-] 68732,C1(CN(C(=O)CC2(O)CCCOC2)C)COCCN1C(C1CCN(C)CC1)=O 68733,C1(c2cn(C)nc2)C(C(=O)NOCC(N2CC(C3CC3)C2C2CC2)=O)CC(=O)N1C 68734,N1(C(CCNCc2ncc[nH]2)=O)CC(CC(=O)OC(C)C)CC1(C)C 68735,c1(CN2C(C(=O)NCc3ccc(Br)s3)CSCC2)c[nH]c2ncc(Cl)cc12 68736,C1(NC(c2cn3ccnc3s2)=O)CN(C(C2CC(F)(F)C2)=O)C2(CCCOC2)C1 68737,C(=O)(C=C1SCC(=O)N1C)NC12CCCN(C(CC(C)C3CCCC3)=O)CC1C2 68738,C(=O)(C(C)(C)CC(F)F)N(C(CNC(CCCC(=O)NCCC)=O)C1CC1)C 68739,C1(NC(C(C)(C)Cc2cccc(Cl)c2)=O)CC2CC(C1)N(C(=O)CCC1CC1)C2 68740,c1(C(C)C)ccc(C(=O)O)cc1.C1(C(=O)O)(CN2CC2=O)CCOC1 68741,c1(C(=O)NC2CCCC(NC(CCN(C)CCO)=O)C2)cc(Cl)c(F)cc1F 68742,N1(CC)CCOC(C(=O)NCC#CCNC(=O)CCc2cncc(OC)c2)C1 68743,C1(O)(CNC(c2ccc(Cl)cn2)=O)CCN(C(C2CCC2C(F)F)=O)CC1 68744,Cc1cc(=NC2CC(C)N(C(=O)CCN(C)C)C2)[nH]c(CC(C)(C)C)n1 68745,CC1(C)CN(C(=O)C(F)F)CCC1C1CC(c2cn(-c3cccnc3)nn2)C1 68746,C1(C(N(C2CCN(C(C3(NC(C)=O)CC3)=O)C2)CC)=O)CCCC1n1cccc1 68747,CN(C)NC(=O)CCC(=O)N1CC=CC(NC(=O)CC2C=CS(=O)(=O)C2)C1 68748,c1(NC(C2C3CN(C(c4c(OC)cccn4)=O)CC32)=O)ccc(Cl)c(F)c1 68749,c1(C(=O)NCC2OCC(=O)NC2)ccc2c(c1)CCCO2 68750,C(C(C(C)C(C)C)NC(C1(C(F)(F)F)CC(F)(F)C1)=O)NC(CCOCC#C)=O 68751,CCC(C)CCC(=O)NCC(O)C(=O)NC1(CC)CCOCC1 68752,c1(Nc2cnn(C)c2C2CC2)cccc2c1C1CCC2O1 68753,C(=O)(C1CCc2ccccc21)N1CCC(C)(CNC(CCC(C)(C)O)=O)CC1 68754,C12(CNC(c3c(COC)scc3)=O)CCCC1CN(C(=O)CCC(C)(C)F)C2 68755,Cc1cccnc1C(=O)NC(c1ccccc1F)CNC(=O)C=Cc1cncs1 68756,N12CC3CCC1C(C3)C2=O.N1(C(=O)OC(C)(C)C)CCCC(O)(CNC2CCC2)C1 68757,C(=O)(C(C#N)C(C)(C)C)N1CC(CC)N(C(c2occc2Cl)=O)CC1 68758,C1(NC(C(N2C(CNC(CCNC(C)=O)=O)CCCC2)=O)=O)CCOCC1(C)C 68759,N1(C(C(CC)C)=O)CCC2(CCCN(C(=O)Cc3ccc(OC)c(OC)c3)C2)C1 68760,Cc1nccc(C(N2CCCC(NC(C3CC(C4CCC4)C3)=O)C2)=O)c1N 68761,c1(CN2CCC(C(N3CC4(CCC4)C3)=O)C2)c(O)cccc1F 68762,N#CCCCCC(=O)NC1CCN(C(C2C3CC4C(C3)C24)=O)CC1 68763,C#CCC1CC(=O)N1.c1(C(=O)OC)cncc(OC)c1.C12CC1C(=O)NC2 68764,C1(NC(C(C)OCCN(C)C)=O)CCCN(C(=O)C(F)(F)c2ncccn2)CC1 68765,c1(C(N(CC(C)NC(c2cncc(OC)c2)=O)C)=O)cn2nccc2nc1C 68766,c1(C(N2CCC(C(=O)NC3(C)CCCC3(F)F)C2(C)C)=O)cc(C#N)ccc1N 68767,CON=C(C(=O)N1CCOC(c2ccc([N+](=O)[O-])cc2)C1)c1ccco1 68768,c1(OC)ccc(C)cc1C(N1CCC(C(C)NC(=O)C(C)n2cccn2)C1)=O 68769,c1(C(N2CC(CCCCNC(C3C(=C)C3)=O)C2)=O)ccc(=O)n(CCOC)c1 68770,Cc1[nH]c2ncnc(N3CCC(C(C)(C)C)(CNC(C4(C#N)CCC4)=O)C3)c2c1C 68771,c1(C(C)C(=O)NC2CCC(NC(=O)COC(C)(C)C)C2)ccc2c(c1)OCO2 68772,c1(C(=O)NC2(CF)CCN(C(Cc3nn(C)c(Cl)c3)=O)C2)cc(N)cnc1Cl 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68808,C1(CNC(C2CCC(=C)CC2)c2n(C(C(=O)OC)C)nnn2)CCCCCC1 68809,CC1(C)CCN(C(=O)CC2CCSC2)C1CC(=O)NC1(C)CC2(CC2)C1 68810,Cc1cc(C)c(C(N2CC(C)C(NC(C3(N(C)C)CCC3)=O)C(C)C2)=O)c(C)c1 68811,C1(NC(C(c2ccc(OC)cc2)=O)=O)CC2CC1CN(C(C1CN(C)C1)=O)C2 68812,N1(C(C(CCOC)C)=O)CCC(CCNC(=O)Cc2nc[nH]n2)(OC)CC1 68813,Cc1nc(C)c(C(=O)NC(C2CN(C(c3cocc3C)=O)C2)C)[nH]1 68814,N1(C(c2cc(COC(C)=O)no2)=O)CCC(N(C(C2CC2C)=O)CC)C1 68815,c1(C(N2C(C)(CC(N3CC(F)(CO)C3)=O)CC2)=O)ccc(=N)[nH]c1 68816,c1(Cc2nc(-c3cncc(C(=O)O)c3)on2)cnc(O)nc1O 68817,C(C(CC1CCCC1)C(=O)NCCC1CC=CC1)NC(CC1N(C)CCC1)=O 68818,CC1(CC(=O)NOC(C2CC2)C2CC2)CN(C(=O)C(Cc2ccoc2)NC=O)C1 68819,C1(NC(C(c2c(OC)cccc2)=O)=O)CC2CCC1N2C(C1CC=CCC1)=O 68820,Cc1ccc(Cl)c(C(=O)NC2CCC(NC(=O)COc3ccc(F)cc3O)C2)c1 68821,c1(CC(=O)NC(CC)CCCC(=O)OC)nc2sc(C)cn2c1CC 68822,N12CC(Oc3ccccc31)C2.c1(-c2cn(C(C)C)nn2)ccc2c(c1)OCO2 68823,N#Cc1ccccc1CC(=O)NCC1(O)CCN(C(c2ccc(CO)o2)=O)C1 68824,C1(C(N2CCC(C(C)NC(c3cnc(C(F)(F)F)s3)=O)C2)=O)CCS(=O)(=O)N1 68825,C1(CC)CN(C(=O)CCOCC2CC2)CCC1NC(=O)CC1CCC=CCC1 68826,Cc1ccc(C)c(C(Cc2ccc(Cl)cc2Cl)NCc2cc(C)c(O)cn2)c1 68827,N1(C(C2CN(CC)C(=O)C2)=O)CC(C(=O)NCCCOC2CC2)CC12CCC2 68828,N1(C(C2(C)CCCO2)=O)CC2(CC(CC(N3CCCC3CCCO)=O)C2)C1 68829,c1(CC(N2C(CCNC(c3ccncc3O)=O)CSCC2)=O)cc(F)cc(Cl)c1 68830,C1(CNC(=O)CCn2ccnn2)CCC(C(=O)NCC2(Cl)CC2(F)F)CC1 68831,C(C)(C)(C(=O)N(C)CC1(CNC(C2CSCCS2)=O)CC1)OCC 68832,C(C)(C(=O)NC1CCOC1c1nc[nH]n1)(C(C)C)COC(C)=O 68833,c1(C(C)(C)C)nocc1C(=O)NC1CCCC1NC(=O)CC(C1CCC1)C1CC1 68834,c1(OC(C)C)ccc(Cl)cc1CNC(N1CCC1)=O.c1(C(=O)OC)cc(CO)on1 68835,Cc1nc2ccccc2nc1NC(C1CC1C(N1CCOC(C)(C)C1C)=O)=O 68836,C(=O)(C(C)CC(F)(F)F)Nc1ccnc(C2(C(=O)NCCCOCC)CCC2)n1 68837,c1(C(=O)OC)cnc(NC(=O)CC2CC(O)CN2C(=O)C2=COCCC2)nc1C 68838,N1(C(C2CCCCC(=O)N2)=O)CC(N=c2ccn3ccnc3[nH]2)CC2(CCC2)C1 68839,C1(c2nnnn2CCN(C)C)(NCCCC(C)(C)C)CCCC(C(F)(F)F)C1 68840,c1(C(=O)Nc2ccc(F)c(C)n2)ccc(F)c(Cl)c1F.C12CC1CN(CC)C2=O 68841,C12CCCC(C1)N(C)CN1CCCC(C1)CC(=O)N(C)C2=O.N1(C(C)C)CCN(C)CC1 68842,C(=O)(CCC(C)(C)C#N)C(C(COC)NC(=O)CCc1ccc(C)cc1)=O.NC 68843,C(CC1=CCOCC1)C(=O)NC(CNC(=O)CCn1cnnn1)C1CCC1 68844,Cc1ccn2cc(C(=O)NC3CN(C(C4CCC(N=[N+]=[N-])C4)=O)CC3(C)C)nc2c1 68845,N1(C(CCN(C)C(=O)OC(C)(C)C)=O)CCN(C(C2CC2F)=O)C2CCC12 68846,CC1CS(=O)(=O)CCN1CCn1cncn1 68847,C1(NC(=O)C(N)=O)CCC2(CCC2)C1CNC(CCCCCNC(C)=O)=O 68848,C(=O)(C1=CCOCC1)N(CCC(=O)OCCC12CC(C)(C1)C2)CC 68849,c1(C(=O)Nc2ncc(CCNC(C(N3C(=O)CCC3=O)C)=O)s2)ncccc1F 68850,C1(CCNC(CCCC#C)=O)CN(c2cc(C(=O)NC)nc(Cl)n2)CC(C)O1 68851,c1(CNC2CN(C(c3ccc(F)c(F)c3)=O)CC(F)C2)cc(Cl)c2cn[nH]c2c1 68852,c1(COC(c2c(CO)ncn2-c2ccccc2)=O)c(F)cccc1Cl 68853,c1(CCC)ccccc1C(=O)NCC(C(C)C)NC(=O)C(N1CCN(C)CC1)C 68854,c1(C(=O)NCCNC(C(C(C)C)c2ccn(C)n2)=O)csc(S(C)(=O)=O)c1 68855,N1C(=NCCc2cccs2)NCc2c(nccc2)C1.N1(CCF)CCCCC1 68856,c1(OC)c(F)cc(-c2nc(C(=O)NCCOc3nccs3)cs2)cc1F 68857,c1(CC(=O)NCC2C(C)CCN(C(Cc3ncc(C)o3)=O)C2)cc(F)cc(F)c1F 68858,N1(CC(c2ccc(C)c(F)c2)=O)CCN2CCOCC2C1 68859,C(=O)(C(=O)CC(C)CC)NCC1(CC(=O)N(C2CC(=C)C2)C)CC1 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69105,CON1CC(C(=O)NC2CCN(C(=O)CCc3cncc(C)n3)C2(C)C)CC1=O 69106,c1(C(Cc2ncccc2F)NC(C(=O)NC2CCC(=O)N2)=O)ccccc1F 69107,O=S(=O)(C1CCOCC1)C(F)(F)F.NC(=NCCSC)N1CCC(F)(F)CC1 69108,c1(C(=O)NCC2CC(NC(CCCC=C)=O)CC2O)cc2occc2s1 69109,C(N=c1nc2c(ncn2C)c(NC2CCSC2)[nH]1)c1cnn(CCCC)c1C 69110,C1(C(=O)NCC2N(C(C(c3cc(F)cc(Cl)c3)C)=O)CC2)CC(=O)NC(=O)N1 69111,C1(OC)CN(C(=O)C=Cc2cnccc2C)CCC1NC(=O)CCC(F)(F)F 69112,C1(NC(=O)Nc2ccc(C)cc2)CC12CCC(N)CC2 69113,Cn1c(O)nc(N2CC3(CN(C(=O)CCN4CCCCC4=O)C3)C2)cc1=O 69114,C12(C(N3CCN(C(CCC(=O)OCC(F)(F)F)=O)CC3)=O)CC3CC1C2C3O 69115,N1(C(C2(C(=O)NC)CC2)=O)CCN(C(C2CCN(C(=O)CC3CC3)CC2)=O)CC1 69116,N1(C(c2c(CC)cccc2C)=O)CC2CCC(C1)N2C(=O)COCC(F)(F)F 69117,C(=O)(CCCC(C)(C)CC)NCC(C(=O)NCC(=O)NCC#C)(C)C 69118,CCCCCCCNC(=O)C(CCN(C)C)NC(c1cc(C2CC2)on1)=O 69119,C12(NC(c3ncn(C)c3)=O)CN(C(=O)C3=CCS(=O)(=O)C3)CC1CS(=O)(=O)C2 69120,c1(N(C)C)ccc(CCC(=O)NCCC2CCC(Nc3cc(F)c[nH]3)C2)cn1 69121,N1(C(c2c(OC)scc2)=O)CCCC2CN(C(C34CC(C#N)(C3)C4)=O)CC12 69122,N1(C(C2N(C(C)=O)CCCC2)=O)CCC(NC(c2ccc([N+](=O)[O-])o2)=O)C12CCC2 69123,C1(C(N(CCN(C)C)C)=O)C2CC(F)C(C2)N1C(C1C=CC(=O)N=N1)=O 69124,C(=O)(C(F)CC(C)(C)C)N(CCN(C(CCOCC)=O)C)CCOC 69125,c1(C(N2CC(CNC(C(CC)C)=O)C2)=O)cc(F)cc(Br)c1 69126,Cc1nc(CC2CCCO2)ncc1NCc1nnnn1CCCOC.c1(C)ccccc1 69127,N1(C(C2N(C(CNc3c(C)cno3)=O)CC2)=O)CCN(C2CCC2)C(C)C1 69128,CCCC(C)CC(=O)NCC12CCC1CCN2C(c1ccc(=N)[nH]c1)=O 69129,N1C(=NCCCc2ccc(Cl)cc2)NCCC2CC12.c1cccc(Cl)c1Cl.CO 69130,O=C(CCCCn1ccnn1)N1CC(CC(N2CCC(c3ccccn3)C2)=O)C1 69131,N1(C(C=C(CC)CC)=O)C2CCC1C(C(=O)NCc1cc(Cl)cc(Cl)c1)C2 69132,C=CCCC(O)CN(C)C(C1CSCCN1C(c1ccncc1Cl)=O)=O 69133,C=CCC(CC=C)C(=O)NC1CCOCC1NC(C1(O)CCC1)=O 69134,N1(C(C2(CC#C)CCOCC2)=O)CCCCCC(NC(c2ccoc2C)=O)C1 69135,c1(C(=O)NC(C)CCCNC(c2cc(C3CC3)ns2)=O)cc(C(C)(C)C)n(C)n1 69136,c1(CN(C(C(C2(O)CCC2)NC(C2C(C(=O)OC)C2)=O)=O)C)ccc(O)cc1 69137,C(=O)(C(F)(F)C(F)(F)C(F)F)NC(C1CCN(C(C2CC23CCOCC3)=O)C1)C 69138,C1(CNC(CC(C)(C)C)=O)CCC2(CCC2)C1NC(=O)CC1=NNC(=O)C1 69139,Cc1cc(=NC(C)C(c2ccccc2)NC(c2cnn(C(C)C)c2C)=O)[nH]n1C1CC1 69140,O=C(N=c1[nH]nc(Cl)cc1Br)c1n[nH]c2c1CN(C(c1cc(Cl)ccn1)=O)C2 69141,C1(C(=O)NCCCCn2cc(C(C)OCC)nn2)C[Si](C)(C)CN1 69142,N1(C(CCSCC(C)C)=O)CC(NC(C2CCCC(=O)C2)=O)C(C)C1 69143,CCCCC(C)CCC(=O)NC(C)CNC(c1ccc(O)c(C)c1)=O 69144,C1(c2n(CC=C)c(SCCC(=O)OC)nn2)(OC)CCS(=O)(=O)C1 69145,C(=O)(CC1C(=O)Nc2c(F)cccc21)N1CCN(C(CSCC)=O)C(C)C1 69146,C(=O)(C(C(C)(C)O)NC(C1CC12CCCCC2)=O)N(CC)Cc1ccoc1 69147,N12CCC(C)C(C1)N(C(=O)C(F)=CC1CC1)CC2=O.C(CCOC)OC 69148,c1(C(=O)NC(CC=C)CNC(=O)Cc2ccccc2)ccc(NC(C)=O)cc1Cl 69149,CCCC(C(=O)OC)C(=O)N1CCOCC1CCNC(=O)CC(C1CC1)C1CC1 69150,Cc1ccc(CNC(C2CCCCN(C)C2=O)=O)c([N+](=O)[O-])c1 69151,C1(C(=O)NCCC(=C)CNC(c2cnnn2C(C)C)=O)CCCC(C)(C)O1 69152,c1(NC2CC(=C)C2)cc(=NC(C)c2ccn(C)n2)[nH]c(COC(C)C)n1 69153,Cc1cc(C(=O)NC2CC2NC(=O)C2=C(Cl)CCC2)cc(O)n1 69154,N1(C(CN(C(=O)Cc2cnn(C)c2)C)=O)CCCC(C(=O)Nc2c(C)onc2)C1 69155,CC1CCOC1C(=O)NC1(C(=O)NCC2CC(Cl)(Cl)C2)CCC1 69156,c1(C(=O)NCC2CCCCN2C(c2csnn2)=O)ccn2cccc2c1 69157,Cn1ccnc1C(N1CCC(CNC(=O)CCOc2cccnc2)C1)=O 69158,C1(CCCC)CN(C(c2nc(O)sc2C)=O)CCN1C(=O)C(CSC)OC 69159,C1(CC=C)(C(=O)NCC(CNC(=O)CC2(O)CCOC2)CO)CCCC1 69160,CCC(CNC(C1CC1(F)Cl)=O)(CC)C(=O)NCCS(=O)CC 69161,C(C(CC(C)C)NC(c1cnc(C)s1)=O)NC(c1n(CC=C)ccc1)=O 69162,CC(F)(F)CCC(=O)N1C2CCC1C(CNC(c1ccnn1CC1CCC1)=O)C2 69163,N1(C(C)C(N2Cc3[nH]nc(O)c3C2)=O)CCC(C)C2OC(C)(C)OC12 69164,c1(CN(CCCCOC2CC2)C)csc(-c2cnn(C)c2)n1 69165,CC1CN(C(=O)CCn2ccnc2)CCC1NC(c1cn(C)ccc1=O)=O 69166,C1(NC(c2nc(C)sc2C)=O)CCN(C(c2nc(C)ncc2Cl)=O)CC1C(C)C 69167,C1(NC(CN(CC)CC)=O)CC2(C1)CC(C(=O)NC1CCC3CCC13)C2 69168,N1(OC(=O)CC=CC(C)(C)C)CCC(F)(F)C(O)C1.CC1CC12C(=O)N2 69169,N1(C(CCNC(=O)NC)=O)CC2CCC2(CC(=O)NC2CC(C(=O)OC)N(C)C2)C1 69170,C1(O)(CCNC(COCc2nnc(C)s2)=O)CCN(C(c2cnc(O)o2)=O)C1 69171,Cc1cc(C(N2C(C(N3CCC(F)(F)C3)=O)CC3CC23)=O)c(C)cc1Br 69172,C(=O)(C1CCCc2scnc21)N1C(C)(C)CC(NC(=O)CC2CCC(O)C2)C1 69173,C1(CC(=O)NCC=CC(=O)NCCNC(=O)OC)CCC(CC2CCCC2)CC1 69174,CC1CC(C(=O)NCC2(O)COC2)N(C(c2cnc(Br)s2)=O)C1 69175,c12ccccc1[nH]c(=O)c(=O)[nH]2.C(=O)(CC(F)(F)F)N(C(C)CC#N)C1CC1 69176,N1(C(COc2cccc(CC)c2)=O)CCC2(NC(=O)C(C)(F)F)CC2C1 69177,c1(NC(c2cn(CC=C)nn2)=O)cccc(CNC(=O)CC2CC2C2CC2)c1 69178,C#CCC(C)(C(=O)NC1CCC2CC12)NC(C1CC2(CC(=O)C2)C1)=O 69179,N1(C(C2CCC(OCC)CC2)=O)CC2CC1CCC2NC(c1cncc(F)n1)=O 69180,N1(C(Cc2c(C)ocn2)=O)C2CCCC1CN(C(C1CCCOC1)=O)CC2 69181,N1(C(=O)NC(C2CCO2)C2CCC2)CCN(N2CCC2)CC1 69182,c1(NC(C(c2cc(C)oc2C)C)=O)nc(C)nc(Br)c1F 69183,c1(C(=O)NC(CNC(c2c(C)ccnc2O)=O)C(C)(C)C)ccc2c(c1)OCC2 69184,C12(CCCO1)C(=O)NC2.c1(C(=O)NOCCC(F)F)cnn(CCF)c1 69185,N1(C(CCC2CCN(C(c3c(C#N)scc3)=O)C2)=O)CCCNC(=O)C1 69186,CC1Cc2cc(CCN=C(NCC(F)F)NC(C)Cc3ccccc3)ccc2O1 69187,C1(NC(C=CC)=O)CC2CN(C(c3[nH]nnc3COC)=O)CC12 69188,N(C(=NCCCC1C=CCC1)N1CC=C(c2cccs2)CC1)CCOC 69189,C(=O)(C1=NOC2(CCOC2)C1)NC(CC=C)CNC(c1cnc(Br)s1)=O 69190,C=CC1CN(C(C2CC(=O)CC(=O)C2)=O)CC1NC(C1CCCOC1)=O 69191,CCC(CC(=O)NC1CCC12CN(C(=O)CNc1ccc(C)c(C)c1)C2)C(F)F 69192,c1(CC)cnc(C(=O)NCC(C)CNC(c2n[nH]c(C(C)(C)C)n2)=O)nc1 69193,S(=O)(=O)(c1ccc(NCC2CCCC23CCC3)c(Cl)c1)NC(c1ccsc1)CC 69194,N1(C(C=C)=O)CCCC(NC(c2nc(C)n(-c3nc[nH]n3)n2)=O)C1C 69195,C(CCC(=O)NCCC1(NC(=O)CCF)CCCC1)=CC 69196,S(=O)(=O)(c1cnc(NCC2CCC2(F)F)c(Cl)c1)NCC(C(CC)CC)O 69197,N1(C(C(C2CC2)OC)=O)CC(CNC(=O)CSc2ccccn2)C2(CC2)C1 69198,CC1CCCCC1CCNC(=O)CC(c1cccc(Br)c1)C 69199,Cc1ccc(F)c(CN2CC(C(=O)NCc3cccc(-c4ccsc4)c3)C2)c1F 69200,C(=O)(C(CNC(C1(C(C)C)COC1)=O)CC1CC1)N(CCC)CC 69201,CC1CCC(NC(=O)CC2CCCO2)CN1C(c1cccc(Cl)c1N)=O 69202,N1(C(C=Cc2ccc(SC)s2)=O)CCN(C(C2C3C4CCC(C4)C23)=O)C(C)C1 69203,CC1(C(=O)NCC2(O)CCN(C(=O)CCCn3cccc3)C2)CCCNS1(=O)=O 69204,N1(CCCCOC(C)C)CC(NCCO)C(C)C1 69205,c1(C(N(C)CC2(O)CN(C(c3ccc(SC)o3)=O)C2)=O)cc(C)nc(C)c1 69206,c1(C(=O)NCC2N(C(C3CCN(C)C3)=O)CCOC2)cncc2c(F)cccc12 69207,c1(C(=O)NC2(C)CN(C(C(CCC)(C)C)=O)C2)n[nH]c2c(C)cccc12 69208,Cc1cccc(OCCCC(N2CC(CNC(=O)C#CC(C)C)C(O)C2)=O)c1 69209,C(=O)(CC1=CCCC1)NCC(C)CNC(c1conc1C(F)(F)F)=O 69210,c1(C(=O)NCCCCC(C)NC(=O)C(N2CCCC2)C2CC2)ccn2nccc2c1 69211,C1(NC(c2cc3c(s2)COCC3)=O)CCOC2(CCOC2)C1 69212,CCC(F)(F)CC(=O)N1C2CCC1C(CNC(c1ccc(OC)c(C)c1)=O)C2 69213,N1(OCCC)CC2CCCCC12.c1(C(=O)OC)cc(OC)cc(C(=O)OC)c1 69214,C1(NC(=O)COC2CCCCC2)CC2CCC1N(C(=O)CO)C2 69215,C(=O)(C(C)(C)CNC(C1CCN1C(C1CCCC(O)C1)=O)=O)NCC 69216,Cc1nc(=N)[nH]c(C)c1C(=O)N(C)CCNC(c1cc(F)ccc1C(F)F)=O 69217,C(C(=O)N1CCC(C(C)NC(=O)Cc2cccs2)C1)(C(C)C)SC 69218,N#Cc1cnn(CC(=O)NC2CC(CNC(c3cccnc3Cl)=O)C2)c1 69219,Cc1nc2ccccn2c1C(=O)NC(CNC(c1ccnc(Cl)c1)=O)C(C)(C)C 69220,C1(NCC(N)Cc2ccccn2)CCc2ncsc2C1 69221,CN1CCN(C(c2ccc(O)nn2)=O)CC1C(N1CC(c2cc[nH]n2)C1)=O 69222,c1(CC)cc(N)c(C(=O)NCC2CCN(C(=O)CCC(CC)SC)C2)cc1F 69223,C1(C(=O)NC(C(N2CC(C)(COC)C2)=O)C2CCCO2)CCC(=O)CC1 69224,c1(CC)ncsc1C(=O)NCC1(CC(=O)NC(C)CCO)CCC1 69225,C(CCCCC(C(=O)NCC1CCCO1)N1CCN(C(C)(C)C(N)=O)CC1)OC 69226,S(=O)(=O)(c1cc(C)cnc1NCC(O)C(C)C)NC(c1scc(CC)n1)C 69227,c1(OC)cc(C)sc1C(=O)NC1CC(NC(c2cc(Br)n(C)c2)=O)C1 69228,C1(N(C)CC)CCN(C(C2C3CC2N(C(=O)C(C)(COC)OC)C3)=O)CC1 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69282,Cn1cccc(C(=O)N(C2CCN(C(C3(CC(F)F)CCC3)=O)C2)CCO)c1=O 69283,N1(C(C(CCC)N(C)C)=O)CCC(C2CN(C(C3(OC)CCOC3)=O)C2)CC1 69284,C1(CC(=O)NCC(n2cc(-c3c(C(=O)OC)n[nH]c3)nn2)C)CCCC(C)(C)C1 69285,N1(C(c2ccc(C(C)=O)o2)=O)CC(CNC(=O)CC2CCCO2)OC2(CCC2)C1 69286,C(CC(CNC(c1cnn(C(C)C)c1)=O)NC(=O)CSCCC(C)C)OC 69287,N1(C(C(CC(N)=O)O)=O)CCCC2CN(C(c3scc4c3CCCC4)=O)CCC12 69288,C12(NC(C=CCN(CC)CC)=O)CCC(CC1)N(C(=O)C(C)CC1CCCO1)C2 69289,CC1N(C(=O)Cn2cc(C3(O)CCC3)nn2)CCC1(C)C 69290,c1(CC(=O)NCc2ccc(C(=O)OC)n2C)noc2ccc(Br)cc12 69291,c1(CCNC(CC2C(C)CN(C(=O)CC3CNC(=O)O3)C2)=O)cnc2n1CCC2 69292,C1(CC(=O)N(CC(C)(C)C)C)CCCN1C(=O)CC1CC(F)(F)C1 69293,N1(C(CCC=C)=O)CCCC(C(C)(C)C(=O)N(CCC)CCN(C)C)C1 69294,c1(CC(=O)NCC2(C(C)(C)O)CN(C(C(CO)OC)=O)C2)c(C)cc(C)cc1C 69295,c1(C(=O)NC2C(CNC(C3CC(SC)C3)=O)C2)cc(C#N)oc1C 69296,N1(C(c2ncc(C)c(Cl)c2)=O)CC2CCN(C(C3CCCC3)=O)CC12 69297,Cc1cccc2cc(C(=O)NCC3CCN(C(=O)C=CC(C)C)CC3(F)F)nn12 69298,C(=O)(C1=NN2CCCN=C2N1)N1CC(O)CC(NC(C(CC)C(=O)OC)=O)C1 69299,Cc1nc(C(=O)N(CC(C)NC(=O)CCN2CCNC(=O)C2)C)cc(O)n1 69300,c1(C2N(C(c3c(I)ccc(OC)c3)=O)CCC2)cccc2ncccc12 69301,CC1CN(C(=O)CC2CC3CC3C2)CC(C(=O)NCc2cc(C(F)F)no2)O1 69302,c1(NC(COC2CCN(C(C(CC)(CO)OC)=O)C2)=O)[nH]nc2ncccc12 69303,Cc1ccc(O)c(C(N2C3CCC2C(CNC(C2CC=CCC2)=O)C3)=O)n1 69304,C(=O)(C1=NNC(=O)CC1)N(C1CN(C(CSCC=C)=O)CC12CC2)C 69305,c1(C2(C(=O)NCC(C)CN(C)C(C3CC=CC(O)C3)=O)CCC2)cccc(F)c1 69306,C1(C(N2CCN(C(=O)CC3NC(=O)NC3=O)CC2)=O)C2C3CCC(C3)C12 69307,C(=O)(N=c1cc2ccccn2[nH]1)C(=O)NCc1nc(CC2CCOC2C(=O)O)co1 69308,N1(C(C(c2ccccc2)NC(C2CCC(CC)O2)=O)=O)CCC2(CCN(C)CC2)C1 69309,c1(C(N(C2CCC(NC(C3(C4CC4)CCCO3)=O)C2)C)=O)cccc(F)c1O 69310,S(=O)(=O)(c1cc(Cl)ccc1F)N1CCN(C(c2cc(F)c(Cl)cc2Cl)=O)C2C1C2 69311,CC(O)CC(C)(C)CNC(C1(C)CC(NC(=O)CC2CC2(C)C)C1)=O 69312,C1(OC)CCCC(CC(N2CC(F)CC2CNC(=O)CCSCC(N)=O)=O)C1 69313,c1(C(=O)NCC(CNC(c2cccc(C)c2)=O)C)ccc2nnc(C3CC3)n2c1 69314,c1(C(=O)NCCOCCN(C(COc2cn(C)nc2)=O)C)nccc(Cl)c1F 69315,C1(C(N2CCC(C)(CNC(=O)C=CBr)C2)=O)CCOC(=O)CC1 69316,C1(N(C(C(CSC)C)=O)CCO)CCN(C(c2cncc(C(C)(C)C)c2)=O)CC1 69317,C1(C(=O)NCC2(CNC(C=CC(C)(C)SC)=O)CCC2)C(F)(F)C12CCC2 69318,Cc1cccc(-c2nc(-c3cccc(Cl)c3)nn2CCC(F)(F)F)n1 69319,Cc1c(CNC(=O)CC2(F)CN(C(c3cc(C(N)=O)[nH]n3)=O)C2)nnn1C 69320,C1(C)(NC(c2ccnc(C)n2)=O)CCN(C(c2sccc2C)=O)CC1 69321,C(=O)(C(C)(C)C1=CCSCC1)NC(CCCC)CNC(c1cccnc1OC)=O 69322,CC(O)(CC(=O)N1CCCC2(C1)CN(C(=O)CCOCC1CC1)C2)C(F)(F)F 69323,N1(C(=O)OC(C)(C)C)CC2CC(Nc3nccnc3Cl)C(C2)C1 69324,N1(C(C2ON=C(C)C2)=O)CCC(CNC(c2ccnc(C3CC3)c2)=O)C1(C)C 69325,C1(C(C)NC(=O)CCC2CCCO2)CCCN1C(c1n[nH]c(C2CC2)n1)=O 69326,CC(C)C(O)C(F)(F)C(=O)N1CCN(C(C2(C)CC2(Cl)Cl)=O)CC(C)C1 69327,C1(C(N(CC(CC)NC(c2c[nH]c(C(=O)NC)c2)=O)CC)=O)CCCCC1C(N)=O 69328,C1(CC)CC2CC(C1)N(Cc1ccccc1OC(C)C)C2 69329,C(=O)(C(=O)N=S(C)(C)=O)N1C(CCOC)CN(C(c2coc(C(F)F)c2)=O)CC1 69330,N1(C(c2cn(CCOC)nn2)=O)CC2(CC(NC(c3csc4nccn34)=O)C2)C1 69331,CC1CN(C(C2CC3(CCC3)C2)=O)CC(C)N(C(C2CC(=O)N2)=O)C1 69332,NC1(CNC(C2CCC(CC(=O)CNC(=O)NC3CC3)C2)=O)CCOC1 69333,C1(CNC(CC=C)=O)CC(O)CN1C(C1CCN(c2nc(C)cs2)CC1)=O 69334,c1(C(=O)NC(CNC(c2n(CC)ccn2)=O)C)cc2ccc(Cl)cc2o1 69335,Cn1cc(C(N2CCC(CNC(c3cccc4c3OCC4)=O)C2)=O)c(O)nc1=O 69336,N1(c2cc(C(=O)OC)ncn2)CCC2CCC(NC(c3ccc(F)c(Cl)n3)=O)C1C2 69337,CCC(C)C(C(=O)NC1CC(C(=O)NCc2c(F)cccc2F)CC1O)N(C)C 69338,C12(C(=O)NCC(C)(C)CC3CCS(=O)(=O)C3)CC(C(F)(F)F)(CO1)C2 69339,CN1CC(O)CC1C(=O)NC1CCN(C(C2C=CCC2)=O)C1 69340,C12(C(=O)NC3(CNC(C(C)C4CC4)=O)CCOCC3)CC3CC(C1)CC(C)(C3)C2 69341,c1(SCC(=O)N(C2CCOC2)CCC#N)ccc(Cl)c(Cl)c1 69342,c1(C(N(C2CN(C(C3(C)CC=CC3)=O)CC2F)C)=O)ccnc(C(F)(F)F)c1N 69343,Cc1nc2cc(C(=O)NCCCCNC(=O)CC3CCCNC(=O)C3)cnc2s1 69344,c1(CCNc2cccc(NC(C)=O)c2)cccc2cncc(C(C)(C)C)c12 69345,c1(CCC(=O)NC(C2CCN(C(C3CC(CC)(CC)C3)=O)C2)C)ncc(F)cn1 69346,C=CC1OCCC1C(=O)NCc1cccc(CNC(C2CN3CCN2CC3)=O)c1 69347,CC1(C)CN(C(C2(F)CC2)=O)CC1NC(C1CCC=CCC1)=O 69348,CCC(C)C(C)C(=O)N(CCCNC(=O)CCc1scnc1C)C 69349,C(C1CCCCC1)=C(C(=O)NCC(C)NC(C=CC(CC)C)=O)F 69350,CC1(C)CC(C)(CNC(=O)CC2(C#N)CC2)CN1C(c1cc2ccccc2o1)=O 69351,CC1(C)CCC(C)(C(N2CCC3(NC(=O)CC4(O)CCC4)CC3C2)=O)CC1 69352,C(CN=c1[nH]c(=N)[nH]c(=NCc2coc(C)c2)[nH]1)c1c(OC)ccc(OC)c1 69353,C1(CCNC(c2cn(CC)nc2)=O)CCN(C(c2ccc(C)cc2F)=O)C(C)C1 69354,N1(C(CCc2ncn(C)c2)=O)CCC(CNC(C2CC23CCC3)=O)C(O)C1 69355,C(=O)(N=c1cc(C)[nH][nH]1)c1nccc(NC(c2cc(OC)c(C(F)(F)F)cc2)=O)c1 69356,c1(N(C)C)ccccc1NC(=O)C(O)CCNC(C1(C)C=CCC1)=O 69357,c1(C(N2CCC(NC(=O)C=C(Cl)Cl)C(O)C2)=O)cc(F)c2ccccc2c1 69358,c1(C(=O)NC(CC)CNC(c2cnc(O)s2)=O)cc(OC(F)F)ccc1C 69359,C1(CCNC(=O)CCC2CCC2)(NC(CCSCC(N)=O)=O)CCOCC1 69360,C(=O)(C#CC(=O)N1CCCC(CNC(c2[nH]ccc2C2CC2)=O)C1)N(C)C 69361,N1(Cc2n(C)ncc2)CCC2CN(C(c3ncc(C(F)(F)F)cn3)=O)CCC12 69362,C1(C(=O)NC(C)(CNC(C2CCC(C(F)(F)F)CC2)=O)CO)COC2(CCC2)C1 69363,c1(OC2CCN(c3n(CCC)nnn3)C3(C2)CC3)c(F)cc(Cl)cc1Cl 69364,C1(NC(c2sccc2F)=O)CCN(Cc2cc(Br)cc(F)c2)CC1F 69365,c1(C(C)NCc2cnc(O)nc2O)nnc2n1CCC2 69366,C(=O)(C1=NOC(C(N2CC(C)(NC(=O)Cc3ccc(Cl)s3)C2)=O)C1)OC 69367,C1(N(C(CC2(OC)CN(C(C3CCCC3C(C)C)=O)C2)=O)C)CCOCC1C 69368,c1(C(N2CCC(CNC(CC(=C=C)C)=O)C(C)C2)=O)ccc(N)c(F)c1F 69369,CC12CN(C(C3CC4(CCC4)CO3)=O)C(C(=O)NOCC3CCOCC3)(C1)C2 69370,N1(C(C2(C#N)C(C)C2)=O)Cc2occ(C(N3CC4(CCC(=O)O4)C3)=O)c2C1 69371,C(CN=c1nc(O)c(Cl)c[nH]1)C1CCC(NC(c2cn(CC)nc2C2CC2)=O)C1 69372,N1(c2ncc(C(N(C3CCNCC3F)C)=O)cn2)CCN2CCCC2C1 69373,C(c1cn(C)cn1)=CC(=O)N(CC(C)CNC(=O)CCN1CCCC1)C 69374,CC(C)(C)CCC(F)C(=O)N1CCOC(C2CN(C(c3ccc(C4CC4)s3)=O)C2)C1 69375,N1(C(C2CCSC2(C)C)C(=O)NCCOC)CCC2CCC(C1)N2C(=O)NCC1CC1 69376,c1(C(=O)NC2CC3CCC2O3)cc(Br)cc2nc(O)[nH]c12 69377,C1(NC(c2onc(C)c2C)=O)CC2CC1N(C(c1cnco1)=O)C2 69378,Cc1nc(C)n(CC(N2CCCCC2C(=O)NCCCOC(F)(F)F)=O)n1 69379,N1(C(C(C)OCC)=O)CC(NC(C2CCOC(C)C2)=O)C(c2cccc(F)c2)C1 69380,C(CCC(O)C(=O)N(CCCC)CCO)NC(C(CC#C)C1CC1)=O 69381,C1(C(=O)NCC2(F)CC(NC(C3(CCCC)CC3)=O)C2)COC2(CCC2)CO1 69382,C(CN=c1[nH]c(NC2CCC2)nc2cc[nH]c12)C1CC(O)C1 69383,c1(OC)cc(C)sc1C(N1CC(CCNC(=O)C(O)Cc2cnc[nH]2)(OC)C1)=O 69384,N(C1CCc2cccnc21)C(C1C(O)CCN(C(c2c(C)c(Cl)ccc2)=O)C1)=O 69385,N1(C(c2nc(OCC)oc2)=O)CCC2(CC1)CC(NC(=O)CCC(N)=O)CCO2 69386,C1(C(C(=O)NCCNC(Cc2ccc(C(C)=O)s2)=O)C)CCCCCC1 69387,CC1(CCNC(C2(C)CCCCC2)=O)CCN(C(=O)C=C2CCCCC2)C1 69388,Cc1cc(Br)cc(S(=O)(=O)N(C2(C)CCOCC2)C2CC3CC2CN3)c1 69389,c1(C(C(=O)NCC2COC2)N(CC(=C)Br)C)cc(OC)ccc1Br 69390,c1(NC(=O)OC(C)(C)C)ccc(NC(C2(CS(C)(=O)=O)CCOC2)=O)cc1 69391,c1(OCC)cc(C(=O)NCC23CC(NC(=O)CC4CC(C)=NO4)(C2)C3)ccn1 69392,C1(C(N(CC2(OCC)CCC2)CC)=O)CC(C)(C)CN1C(=O)C(=O)NOC 69393,C1(OCC)(CNC(=O)CC(C)n2cccn2)CN(C(c2cnc[nH]2)=O)C1 69394,C1(NC(c2cn(C(COC)C)nc2C)=O)CN(C(C2CC23CC3)=O)CC2CC12 69395,CCC(C)(CNC(C1CC1(F)Cl)=O)C(=O)N(CC(C)(C)OC)C 69396,N12CCCC(C1)CC(=O)N2.C1(C(N2CC(CC)(OC)C2)=O)COCCN1C1CCC1 69397,c1(OCC(N2CCC(NCCO)C2)=O)nc(O)nc(O)n1.C1(C=O)C2CC3C(C2)C13 69398,Cc1cccc2c1CC(C(=O)NCC1(C)CCCN1C(C1CN3CCC1CC3)=O)O2 69399,c1(C(N(C(C)CNC(C2CCC(C)(C)CO2)=O)CC)=O)onc2c1CCCC2 69400,C(=O)(C(C(=O)N1CCOC(CC2CC2)C1)OC)OC.C12(CC(F)C1)C(=O)N2 69401,C(=O)(CC(C)C(=O)NC(CC1CC1)C(=O)NCC1COCC1N(C)C)OCC 69402,C1(O)(CC(N2CCC(OCC(=O)NCC3ON=C(C)C3)C2)=O)CCCOC1 69403,Cc1cc(C(N2CCC(C)C2C(=O)NC(C)(C)CCCO)=O)[nH]c1C 69404,C1(OC)CN(C(=O)C(F)(F)n2ccnn2)CC1NC(c1cnn(C)c1C1CC1)=O 69405,c1(C(=O)NC2CCCN(C(c3nccc(C)c3)=O)C2C)cc2cc(Cl)ccc2[nH]1 69406,Cc1cc(C(=O)NC2(CF)CN(C(C3CC4CC(=O)C3C4)=O)C2)nc(C2CC2)n1 69407,C1(F)(C(=O)NCC2(C)CC(NC(c3c(C)ncn3C)=O)C2)CCCCCC1 69408,C(=O)(CC(C)P(C)(C)=O)N1C(CNC(c2c(C)non2)=O)CC(O)C1 69409,c1(O)cc(Cl)cc(Cl)c1[N+](=O)[O-].O(NC(=O)NCCC)CCCN 69410,CC(C)(C)CC(O)C(=O)NC(CNC(c1cc(C(N)=O)[nH]n1)=O)CO 69411,N1(C(C2(OCC)CCOC2)=O)CCC(C2(NC(=O)C(n3ccc(C)n3)C)CC2)C1 69412,CN1CCCC(CCC(=O)NC2(C3CN(C(C4(C#N)CC4)=O)CCO3)CC2)C1 69413,C1(CCNC(C(COC)C)=O)CSCCN1C(=O)C(C1(O)CCCC1)F 69414,C1(F)(C(N(CC(C)N(C(=O)CC2CCN(C)CC2)C)C)=O)CC=CCC1 69415,CC1(CC(N2CCC3C(NC(=O)CSc4nncs4)C23)=O)CCOCC1 69416,n1(CC(N2CCCCC(NC(C3(O)CC(C)(C)C3)=O)C2)=O)cnc2ccccc12 69417,C(=O)(C(O)CC(N)=O)NC1CN(C(CCOc2cccc(OC)c2)=O)C2C1C2 69418,c1(C(=O)NC2CC(C)CN(C(c3csc(C#N)c3)=O)C2)cnc2ccccn12 69419,C1(NC(C(CC#C)CC#C)=O)CC2CN(C(=O)C(C)(C)CO)CCN2C1=O 69420,C1(CNC(COCCC(C)C)=O)CN(C)CCN1C(=O)C(C)Cn1ccnc1 69421,C12CC3CN(CC3C1)C2=O.c1(CNC(C2(SC)CCC2)=O)cccc(C#N)c1 69422,N1(C(C(CC)N(C)C)=O)CCN(C(C2(C)CC3CCC(C2)S3)=O)CCC1C 69423,O=C(C(Cl)=CCl)NCCCC1CCCN1C(C1(c2ccncc2)CC1)=O 69424,C1(C(=O)NC(C2CCCC2)C)CCCN1C(=O)CCc1ncnn1C 69425,C1(C(=O)NC2(COC)CCCC2)C2CCC(C2)N1C(C1C=CC=CC=C1)=O 69426,c1(C(=O)NC2C(NC(C=Cc3ccc(C)s3)=O)CCCC2)ncc(F)cc1N 69427,CC1(C)CN(C(c2cncc(Cl)c2)=O)CCN1C(C1CN(S(C)(=O)=O)C1)=O 69428,N1(C(C2C(C=C)C2)=O)CCC2(CC1)CC2CNC(=O)C=Cc1ccc(Cl)cc1 69429,CCS(=O)(=O)CCN=c1[nH]c(N2CCOCC(COCC)C2)nc2c1CSC2 69430,CC1COCC1N=c1[nH]c(N2CCN(C(=O)C3CC3)CC2)nc2c1CCCCC2 69431,C(CS(=O)(=O)CC(=O)NC1COCC1C(=O)NOCC1(C)CC1)OC 69432,C(=O)(C(CCC(C)C)NC(C1COCCC1C)=O)NC(CCC)C(N)=O 69433,C12(NC(CCCC=C)=O)CC(CNC(c3cc(C)n(C)n3)=O)(C1)OC2C 69434,C12(NC(c3ccc(F)c(O)c3)=O)CCC(C(N3CCC3CO)=O)(CC1)C2 69435,C(CC(C)(C)CNC(=O)Cn1ncc(Br)n1)NC(C(=O)NC(C)C)=O 69436,c1(C(N(CC(CNC(COC(C)=O)=O)C)C)=O)ccc(N2CCOC2=O)cc1 69437,C1(NC(CCOC)=O)C2CN(C(=O)COC3CCCOC3)CC12 69438,C1(CN(CCCNC(Cc2cn(C(C)C)nc2)=O)C)CC2(CCC2)CO1 69439,C(c1ccc(=N)[nH]c1)=CC(=O)NC(C)CCCNC(=O)COc1ccc(Cl)cc1 69440,Cn1cc(S(=O)(=O)NC2CCN(C(C3(c4ccc(F)cc4)CCCC3)=O)CC2)cn1 69441,C1(C(=O)NCC2(NC(C3CC(C)(CC)C3)=O)CCC2)CCCCN1C(C)C 69442,N1(C(C2(CCC=C)CC2)=O)CC(N(C)C)C(CNC(c2cnccn2)=O)C1 69443,c1(CC)cccc(C(=O)NC2(CNC(=O)Cc3cncnc3)CCOCC2)c1O 69444,N1(CC(=O)NCC2(CNC(=O)CCN3CCC(F)C3)CCC2)CCCC(O)C1 69445,C1(C)(C(=O)NCc2cccc(CNC(CC3CC(C)(C)C3)=O)c2)CCCNC1=O 69446,C1(NC(C=CCC)=O)CC(=O)N(C2CN(C(=O)C(c3cccs3)SC)C2)C1 69447,c1(CNC(C=C(C)C(C)C)=O)cccc(CNC(C2(C)CC3CC3C2)=O)c1 69448,CCCCCCC(O)CCC(=O)NCC1CC2CCC1N(C(=O)C(C)(C)CF)C2 69449,c1(C(=O)NC2C(NC(c3c(Cl)cccc3Cl)=O)CCCC2)cnc2ccsc2c1 69450,c1(OCCC(=O)C(N(CCN)CC)=O)cc(Br)c(C)nc1NC(=O)OC(C)(C)C 69451,c1(NC(C2CC3(CCC3)C2)C)cnc2ccccc2n1 69452,c1(CC(N2CCC(CN(C(c3nnc(C)s3)=O)C)C2)=O)ccc2nn(C)cc2c1 69453,N1(CCCC)CCC(N=c2cccc(S(=O)(=O)NCC3CCN(CC)C3)[nH]2)CC1 69454,N1(C(c2cnc[nH]2)=O)CCCC(Cn2cc(CN3CCCC3)nn2)C1 69455,c1(C(C(=O)NC(CC)C)N(C(C)CN(C)C(C)=O)C)ccn2nccc2c1 69456,c1(CC)noc(CNC(C2CC(CNC(=O)CCOC3CCC3)C2)=O)n1 69457,C#CCC(CC#C)C(=O)NC1CC(CNC(c2ccc(C)c(Br)c2F)=O)C1 69458,N1(C(C(C)C2(O)CCC2)=O)CCC(C2CC2)(CNC(C2C=CCC2)=O)C1 69459,N1(CC)CC(C(=O)NCCCn2cc(Cc3cccc(C)c3)nn2)NC1=O 69460,C1(C(=O)NC2(C)CN(C(C3C(=C)CC3)=O)C2)CCCC1C1CCOCC1 69461,c1(CCC(=O)NCC23CC2CN(C(c2ccncc2Cl)=O)C3)ccc(O)c(Cl)c1 69462,N1(C(C(c2scc(C)n2)C)=O)CCC(NC(C23CCC(CC2)OC3)=O)CC1C 69463,Cc1ccc(CC(=O)NCCC23CCC2CN(C(=O)CSC2CC2)C3)c(F)c1F 69464,CCC(C)CC(=O)N(CC(C)NC(=O)CCOCCN(C)C)C 69465,N1(Cc2nc(NC(CCc3n(C)ccn3)=O)sc2)CCC(F)(CO)C1 69466,N1(C(CC2N(C)CCC2)=O)CCC(OCCNC(C2CCSC2)=O)CC1 69467,C1(CO)(CO)CCN(C(=O)CC2(C)CC2)C1.C1(=CC(=O)NC2CC3CC3C2)CCCCC1 69468,c1(C(N2CCC3CC(C(=O)NCC=C)C3C2)=O)nc2nc(C)c(Cl)cn2n1 69469,CCC(C)(C)C(C)CC(=O)NC1CC12CCN(C(=O)CC(F)(F)F)CC2 69470,C(C(=O)NOCc1ncccc1C)(C1CCCC1)NC(CCn1ccc(C)n1)=O 69471,CC1(C)C(CNC(=O)Cc2csc(S)n2)CCN1C(=O)C(C1CC1)C1CC1 69472,C1(OC)(OC)CN(C(=O)CC2CCC(=O)O2)C1 69473,C(=O)(C1=CSCCO1)N(C1CN(C(c2csc(C(N)=O)n2)=O)CC1(C)C)C 69474,C(=O)(CCS(C)(=O)=O)NC1CC(CNC(C(C)OCC2CCCCO2)=O)C1 69475,CC1(C)CN(C(c2ccsn2)=O)CCC1NC(c1cc2ccccn2n1)=O 69476,c1(C(N2C(C)CN(C(=O)COc3cccnc3Cl)CC2)=O)ccc(S(N)(=O)=O)o1 69477,S(=O)(=O)(c1cc(C(=O)NC2(CNC(c3cccn3C)=O)CCC2)co1)NC 69478,C(CN=[N+]=[N-])(C(=O)NCC1C(CO)C1(F)F)NC(C(C=C)CC)=O 69479,C#CCC(C)(CNCc1cc(C)ccc1N1CCCC1)CO 69480,c1(C(=O)NCC2(C(=O)NC3(CC)CC3)CCCCCC2)ccc2nc(C)oc2c1 69481,c1(CC(N2CC(N(C)C(c3cc(Cl)ccc3Cl)=O)C(O)C2)=O)cc(F)cc(F)c1F 69482,C#Cc1cccc(C(=O)NCC2CCC(C)CN2C(=O)C=CCOC2CC2)c1Cl 69483,Cc1cccn2cc(C(=O)N(C3CCN(Cc4ccnn4C)C3)C)nc12 69484,c1(C(N(C(CN(C(CCSCC=C)=O)C)C)C)=O)c(C)cc(OC)cc1C 69485,C1(NC(Cc2n(C)ccn2)=O)CCC2CN(CCCCc3ccccc3)CC2C1 69486,c1(C(=O)NCCCCNC(c2nccc(C(N)=O)c2)=O)ccc2n[nH]cc2n1 69487,CCC(C(=O)NC1(CF)CN(C(C2CCSC2)=O)C1)C(C)(C)CC 69488,c1(C(=O)NC(c2cccc(C#N)c2)CC(=O)OC)ccc2nc(C)n(C)c2c1 69489,c1(OC)ccc(NC(=O)C(=O)NCCCc2ccsc2)cc1OC 69490,C(C(=O)NC(C)CCCNC(=O)COC1CC(F)(F)C1)(C(C)C)NC(C)=O 69491,Cc1cnccc1N1CCN(C(CCC2CCCOC2)C(=O)NC2COC2)CC1 69492,N1(C(c2cc(C)oc2C)=O)CC(NC(c2cc(C)nc(O)c2)=O)CC12CCCC2 69493,CCC(CC1CCCC1)CC(=O)NC1CC(C(C)NC(=O)CCCc2nccs2)C1 69494,CC1=NN(C)C(=O)C1CC(=O)N(C1CCC=C1Br)C1CC1 69495,CC(C)(C)CC(F)C(=O)NCC(C)(CO)NC(C1C(C)(C)C1(C)C)=O 69496,C1(NC(c2c(C)nn(C)c2)=O)C2CCC(C2)C1C(=O)NCc1ccc(C(N)=O)o1 69497,C1(C(=O)NC(C=CC(=O)NC(C)Cc2ccncc2)C)CCC(C)(C)O1 69498,C=CC(C)(C)CC(=O)N1CCOCC(C(N(C)C[Si](C)(C)C)=O)C1 69499,C1(CC(=O)NC(c2ccc(Cl)cn2)C)CCCN(C(=O)C=C2CCCC2)C1 69500,C1(OC)CC(C(=O)NC(C)C(CO)NC(C2CC(OC)(OC)C2)=O)N(CC)C1 69501,CC1CC(NC(ONC(=O)C2CC2c2ccccc2)=O)C(C)CN1C 69502,C1(NC(c2c(C)ncnc2)=O)CCCN(C(c2cn3cccnc3n2)=O)CCC1 69503,C1(CNCC(C2CC(F)(F)C2)OCC)CCCCN1C1CCCC1 69504,CN1CCN(C2CCCC2C(N2CC3C(C(=O)NCCN(C)C4CC4)C3C2)=O)CC1 69505,C1(CN(C)CC2CN(C(=O)CS(=O)(=O)Nc3ccccc3)C2)CC(=O)NC(=O)C1 69506,CC1(C)CCCN(C(c2c[nH]nc2F)=O)C1CNC(=O)CCc1ncccn1 69507,c1(NC(=O)NC(C2CCCCCC2)C)ccc2c(c1)N(C)CCO2 69508,N1(c2nnc(-c3cccc(C)n3)n2CCC#N)C2CCCC1CC(O)C2 69509,O=CCC(C)(c1ccccc1)SCC(C1CC1)NC(C1CC(O)C(F)C1)=O.C1CC1 69510,C(CCCC(=O)N1CCC(N(C)C(C2CC3C=CC2C3)=O)C1)SC 69511,O=S(=O)(c1cncc(Br)c1)NCCC1CC(NCCc2ncc[nH]2)C1 69512,C(=O)(CCC(C)S(C)(=O)=O)NCC(CCOC)NC(=O)CCc1c(C)n[nH]c1C 69513,Cn1cc([N+](=O)[O-])c(-c2nnc(-c3ccn(C)n3)o2)n1 69514,c1(CC(=O)NCCNC(c2nn(CC)c(C(F)(F)F)c2)=O)ccc(C)c(F)c1F 69515,N1(c2ncc(CCC)cn2)CCC2(CCN(S(=O)(=O)c3cncc(Br)c3)C2)C1 69516,N1(C(=O)C(O)Cc2cnc[nH]2)CCC2C(CCCN2C(c2cscn2)=O)C1 69517,c1(NC(c2n(C(C)C)ncc2)=O)ccc(Br)c(OCF)c1 69518,C(=O)(C(=O)N=c1cc(C(C)(C)C)o[nH]1)Nc1cccc(CC(=O)OC)c1 69519,N1(C(CN2CC(C(=O)NCCC=C)C2)=O)CC2CCC1CN2C(C)=O 69520,Cc1ccc2cc(C(=O)NCCC3CN(C(=O)C(N)=O)CC3C)[nH]c2c1 69521,C(=O)(CCCCCF)N(C(C(=O)NC1CCCN(CC)C1)C)C 69522,n1(CCC)nnnc1C(C)(CC1CCC1)NC(c1nc(C)cs1)C 69523,CC1C=C(C(=O)N2CCCCC2CNC(=O)C=Cc2ccc(F)cc2)CC1 69524,N1(C(CC(C)OC)=O)CCCC12CCN(C(C1CCN(C)CC1)=O)C2 69525,c1(C(=O)NC(CNC(C(C=C)(C)CCOC)=O)CO)[nH]c(C)c(S(N)(=O)=O)c1C 69526,c1(C(N(CCNC(C2CCC(C)(CC)O2)=O)C)=O)cnn2c1NCC(C)C2 69527,n1(CC(=O)NC(C2CN(CC=C(Cl)Cl)C2)=O)ncc2cc(Br)ccc2c1=O 69528,Cc1cc(NCC(C)N(C)C(c2nnc(O)nc2O)=O)cc(C#N)c1[N+](=O)[O-] 69529,C(=O)(CCCC(C)(C)C)N(CC(C)(C)CNC(=O)CCCOC(=O)CCF)CC 69530,N1(C(C2N(C(CSCCOC)=O)CCOCC2)=O)CCCN(C)CC1C 69531,c1(C(=O)NC(C(C(C)C)Nc2nnccc2C#N)C)c(Cl)cccc1Cl 69532,C1(CNC(=O)C(F)C2CCC2)CCN(C(C2CC3CC2C3)=O)CC1 69533,Cc1n[nH]c(C)c1CCC(=O)NC(C)CNC(=O)CC1CC1C(F)(F)F 69534,C(CC(C(C)(C)C)NC(c1cccc[n+]1[O-])=O)N(C)C(c1cnc(Cl)cc1N)=O 69535,c1(CC)ccc(C(=O)NCC=CCOC)cc1NC1CC1c1ccco1 69536,N1(C(C(N(C(=O)Cc2ccnc(O)c2)C)C2CC2)=O)CC2(C1)NC(=O)NC2=O 69537,C1(CC(=O)NC2C(CNC(CP(C)(C)=O)=O)COC2)CCC2(CCC2)O1 69538,Cc1ncc2n1CCC(C(=O)NC1COC3C(NC(=O)CNC=O)COC13)C2=O 69539,CCC(C(=O)NCC1CC(O)CN1C(=O)C1=CCCS1)C(C)(C)CC 69540,c1(C(=O)OC)ccc2c(n1)N(c1ccc(OC)nn1)CCO2 69541,N1(C(COC(CC(CC)C)CO)=O)C2CCC1CC(N(c1cc(C)nc(C)n1)C)C2 69542,C=CCCC(C(=O)NCC(C)CC(=O)OC)NC(C1CN(C(C)C)C1)=O 69543,C1(NC(CCN(CC#C)C(C2C=C(C)CS2)=O)=O)CC(O)C1(C)C 69544,C(=O)(CS(=O)C(F)(F)F)NC(CC(=O)N(C)C)C(F)F 69545,CC1(C2CC2)CCN(C(C23CC(CO)(CN2C(C2CC4CCC2O4)=O)C3)=O)C1 69546,N1(CC(=O)N(C2CCC(CNC(=O)CC3COCC3O)CC2)C)CCCNC1=O 69547,C1(NC(CCSCCCC)=O)CC1C1CCN(C(=O)Cc2cncc(C)c2)CC1 69548,c1(C(=O)NC(CC)(C)CN(C)C(c2cc(Cl)no2)=O)cncc(C(=O)NC)c1 69549,CCCC(C(O)C(=O)NCc1ccc(F)nc1C)NC(c1cc(N)cc(F)c1)=O 69550,N1(C(C(C)=CC)=O)CC(NC(=O)CCOc2cccnc2)C2(CCOCC2)C1 69551,CC(C)CC(C)(CNC(=O)C(F)=CCCF)NC(c1cc(C(F)F)cc(F)c1)=O 69552,c12nn(C)cc1NC2=O.c1(C(C(=O)N(CCCC2CC2)C)(F)F)ccc(F)cn1 69553,C1(NC(C2(C)CC(C)C2)=O)CCN(C(c2ccnc(F)c2)=O)CC1(C)C 69554,CCC(CC)CCCC(=O)NCC(O)CC(N1CCc2c(ccn2C)C1)=O 69555,N1(C(CC2N(C(c3c(OCC)cccc3)=O)CCC2)=O)CC2OCC(CO)C2C1 69556,C12(NCC(C)C)CCCN(CC1)C2.C1(CO)C(=O)O1 69557,N1(C(C(CCC)C)=O)CCC(O)CC1C(=O)Nc1ccc(OC)cc1OC(F)F 69558,N1(C(C(C)(C)SC)=O)CCCCC2(CCN(C(C3(C)CCCNS3(=O)=O)=O)C2)C1 69559,c1(CN(C(C2CN(C(C3NC(=O)CC3C)=O)C2)C)C)cc(C(C)(C)C)ccn1 69560,N1(C(C(CO)OC)=O)CCCCC(C(=O)NCCc2cnco2)C1 69561,c1(C(=O)OCCN(C(CC(C=C)CCC)=O)CC)ccc(N=NC(N)=O)cc1 69562,C1(NC(C=CCCC)=O)CCCCC12CCN(C(=O)Cc1ncc(C)s1)C2 69563,C1(C(N2CC(F)(F)C2C2CC2)=O)CN(C(=O)CC2CCC3CC23)CC12CC2 69564,c1(NC(c2c(CC)c(Br)ccc2)=O)cn2c(n1)CN(C(C)=O)CC2 69565,C(C)(CCC(C)C)(c1nnnn1CC1CCCO1)Nc1nc(C)c(C)s1 69566,Cc1nn(CC(=O)NCC(C)(O)CNC(=O)C(C)(C)CC2CC2)c(=O)o1 69567,CC1(C)C(NC(C2CC3CCCC23)=O)C2CCCN(C(=O)CCC3CC3(F)F)C12 69568,N1(C(CSCC)=O)CCC(CC(=O)N(CC)Cc2nnc(C)o2)C1 69569,C1(NC(CSCCOC)=O)CC(C(=O)Nc2cc(C)cc(F)c2)C12CCC2 69570,c1(C(=O)NC2(CCNC(C(C(CC)O)C)=O)CC2)cc2oc(Br)cc2s1 69571,C(CCCN=c1nc2c(ncn2C)c(N2CCCC2C2CC2)[nH]1)c1n(C)ccn1 69572,C(C)(C(=O)N1CC2CC1CN2C(=O)CO[Si](C)(C)C)(C(C)C)NC(C)=O 69573,c1(C(N2CC(NC(C3(C=C)CCCCC3)=O)C(C)C2)=O)cccc2nccn12 69574,CC1CN(C(C2(c3ccno3)CC2)=O)CCCN1C(=O)CC(C)(C)C#N 69575,CC1=NC(C)(CNC(C2(CO)CCN(C(c3ccc(C(F)F)o3)=O)C2)=O)CS1 69576,c1(OC)ccc(C(=O)NC(C2CN(C(c3sccc3F)=O)C2)C)c(OC)n1 69577,C1(N(C(=O)CC(=O)N2CCCC2)C)CN(C(=O)CC2(O)CC2)CC1(C)C 69578,C1(NC(C(C(C)C)O)=O)CCN(C(c2cnn(C)c2)=O)C12CC2 69579,C12(C(=O)NC(C)CCNC(=O)CCN3CCC3)CCCC(CCC1)C2O 69580,c1(NC2CC(F)(CNC(CC(C(C)C)C)=O)C2)cc(O)nc(=O)n1C 69581,C1(OC)CCC(CC(=O)NCCCCC(C)NC(=O)CCc2ncccn2)CC1 69582,c1(OCC)ccccc1-c1nc(C2COCCO2)n(C2CCOC2)n1 69583,C1(CCOC)(NC(c2ccnn2C)=O)CCN(C(C2(C)CCC(=O)C2)=O)C1 69584,c1(CC)cc(Cl)ccc1C(=O)NCC1(CO)CC(NC(=O)COC2CC2)C1.COC 69585,c1(C(=O)NC2CCN(Cc3cccc(I)c3)CC2)cc2ccsc2[nH]1 69586,c1(CN2CC(NC(c3scc(C)c3)=O)C(O)C2)cccc(S(C)(=O)=O)n1 69587,N1(C(C2N(S(C)(=O)=O)CC2)=O)CCCC(C)(NC(c2cc(C3CC3)ccn2)=O)C1 69588,N1(C(c2c(CC)oc(C)c2)=O)CC2CN(c3nnc(C(N)=O)s3)CC(C1)O2 69589,C1(NC(Cc2nc(C)sc2)=O)CCCCN(C(C2C3CCOCC23)=O)CC1 69590,C1(CC=C)(C(N2CCC(CNC(C)=O)C2)=O)CCN(C(c2ccnnc2O)=O)C1 69591,n1(C(C(=O)NC(C)COC(C)(C)C)(C)C)cc(C2(n3nccn3)CC2)nn1 69592,C#CCC(CC(F)F)C(=O)NCC(F)(C(=O)N(C(C)CN(C)C)C)C(C)C 69593,Cc1cc(NC2CCCN(C(c3ccnc4c3ncn4C)=O)C2)ncc1[N+](=O)[O-] 69594,n1(CC(=O)N(C(C2CC2)C2(C3CCOC3)CC2)C)cc(C(c2ccc(Br)o2)O)nn1 69595,C(C(C)C)(C(O)C(=O)N(C(CC(F)F)C(N1CC(C2CCCC2)C1)=O)C)OC 69596,c1(CC(N2CC(CC(C)NC(C3CC(F)CN3C)=O)C2)=O)ccc(Cl)nc1 69597,CC1CC(=O)OC(=O)N1.C(C)(C)(C)OC(=O)OCC=C 69598,c1(OC)cccc(=NC(=O)CN2CCC(CN=c3[nH]c(C)c(C#N)s3)CC2)[nH]1 69599,N1(C(c2ccc(OC)cc2)=O)CC(NC(=O)CN2CCN(C)CC2)CC(C)C1 69600,Cn1nnc2c(C(N3CCC(O)(CCNC(C4CC4(F)Cl)=O)CC3)=O)cccc12 69601,C(C(CC(C)C)C(=O)N(C)CC1CCN(C)C1)NC(C(C=C)(C)CC)=O 69602,Cc1n[nH]c(C)c1C(=O)NC1(CNC(C2CN(CC(C)C)C2)=O)CCOC1 69603,C1(N(C(C2C3CCCC23)=O)C2CC2)CN(C(C2(N(C)C)CCC2)=O)C(C)(C)C1 69604,c1(CC(=O)NC(COC)CNC(=O)CCOCC2CCCO2)ccc(F)c(Cl)c1 69605,N1(C(c2c(C)ncs2)=O)CCN(C(C2C=CC=CC=C2)=O)CC1c1cccnc1 69606,C=CCCCC(C1CC1)NC(=O)C(C)C(C)CNC(=O)C=CC(=O)OC 69607,c1(C(=O)NC2CCN(C(C(CCC)C)=O)CC2)sc2ccccc2c1Cl 69608,C1(NC(c2nn(C)c(F)c2)=O)CN(C(c2csc(Cl)c2)=O)CC2CCCC12 69609,c1(OC)ccc(SCC(=O)NC(C)CN(C)C(c2cn(CC(N)=O)nn2)=O)cc1 69610,N1(Cc2ccc(CC)o2)CCC(F)(C#N)C1 69611,N1(C(c2c(C)c(Br)cnc2)C(=O)Nc2ccc(F)cc2)CC(C#N)C2(CCC2)C1 69612,c1(C(=O)NC2CCN(C(c3ccc(OC)c(O)c3)=O)CC2F)c(F)ccc(F)c1Cl 69613,C(=O)(CCS(=O)(=O)C(F)(F)F)N(CC(C)O)CCNC(C1CCCCO1)=O 69614,c1(OC(C(=O)NCC(CC)NC(C2CC(O)C2)=O)C)ccc(Br)cc1 69615,c1(C(=O)NCC(CC)NC(c2coc(C3CCCC3)n2)=O)ccn2ncnc2c1 69616,c1(C(=O)NCCCCCCNC(CCCC)=O)c(Cl)ccc2ccoc12 69617,c1(N2CCN(C(=O)Nc3cc(C(=O)OC)sc3)CC2)ccc2oc(N)cc2c1 69618,c1(CC(=O)NCC2CCCN(C(c3ccc(N)cc3)=O)C2)cccc([N+](=O)[O-])c1 69619,c1(NCCC2CC(NC(C(C=CC)O)=O)C2)ccc([N+](=O)[O-])cc1S(C)(=O)=O 69620,C1(NC(c2c(C)nn(C(C)C)c2)=O)CC2(C1)CN(C(=O)C(C)C(C)C)C2 69621,C12(NC(=O)CNC(C3CC4C=CC3C4)=O)CCC(C1)C(O)C2O 69622,N1(C(C(C#C)(C)C)=O)CCC(NC(=O)CC2CCC(=O)N2CC)C(C)(C)C1 69623,S(=O)(=O)(c1cccc(C(=O)NC2CN(C(C3C(C)C3(F)F)=O)CC2C)c1)NC 69624,C1(NC(c2c(NCC)scn2)=O)CCCCC1CNC(=O)C(C)(C)C 69625,C1(C(=O)NCc2cc(CC)on2)CN(C(c2cc(C)nn2C)=O)CC12CC2 69626,C1(CC(=O)NCC2(NC(CCN(C(CCC)C)C)=O)CC2)CCCCC1 69627,c1(C(N2CC(NC(=O)CC3NC(=O)NC3=O)CC(C)C2)=O)c(F)ccc(Cl)c1N 69628,C1(NC(c2cnc(Cl)c(Cl)c2)=O)CN(C(=O)C(F)=CC2CC2)Cc2nccn2C1 69629,c1(OC)cc(C(N2CCC3CC23CNC(=O)CCCCOC)=O)cc(F)c1 69630,C1(CC(=O)N(CCCNC(=O)C(C)NC(N)=O)CC)COCCOC1 69631,CC1=C(C(=O)NC23CC(c4cccc(OC(F)F)n4)(C2)C3)CCO1 69632,C1(CNC(Cc2c(C)cc(C)s2)=O)CCC(C)CN1C(=O)CCCCC1CC1 69633,C12(NC(Cc3cc(C)n(C)n3)=O)CCC1CN(C(=O)C(C1CCC1)C1CCC1)C2 69634,CCC(CC)(CC)C(=O)NCC1CC(F)(CNC(c2ccc(C#N)c(Cl)c2)=O)C1 69635,Cc1cc2[nH]c(=O)c(C(=O)NC(C)CN(C)C(C3CCCC(C)CC3)=O)cn2n1 69636,C1(C(N2CCC(CN(C(C3(C=C)CC3)=O)C)C2)=O)CN2CCC1CC2 69637,CC(C(=O)N(C)Cc1ccc(CNC(C2CC2C(N)=O)=O)cc1)C(F)F 69638,C12(C(N3CCC(O)(C(C)CNC(C4(C)CCCC4)=O)C3)=O)CCN(C1)S(=O)(=O)C2 69639,c1(OC(C)C)cccc2c1CCN2c1cc(NCC2C3CCC3CCC2)ncn1 69640,N1(C(C(C)OCC(C)C)=O)CC(NC(=O)CCNC(c2ccoc2)=O)CC(O)C1 69641,Cc1nc(C(=O)NCC2CC2NC(=O)CCC=CBr)cn1C(F)F 69642,C=C=CCCC(=O)NC1CCC(C)(CNC(=O)CCN(CCCCC)C(C)C)C1 69643,C#CCC(O)C(=O)NCC1COCCN1C(=O)CCc1ccccc1O 69644,c1(CC(=O)NCCOC2CCOCC2)c[nH]c2ccc(F)cc12.CC1CCN1C 69645,c12cccc(c1)C(=O)NC2.CC1(CN2CCSCC2)CCCC1 69646,N1(C(C(C)=CC(C)(C)C)=O)CC(=O)NCC1C(=O)NCCc1ccc(F)nc1 69647,CC(N=c1[nH]nc(C2CC2)s1)C1CCN(C(c2ncnc3sccc23)=O)CC1 69648,C(CC(C)(C)C)(C(=O)NCC1CCC1)N(CC(CCCC)CC)C 69649,c1(CNC(C2CC(=O)OC2)=O)ccc2c(c1)CCC2NC(=O)C=CC(F)(F)F 69650,C(=O)(C1CCCc2cccnc21)NC1CCCN(C(c2ccc(C)o2)=O)CC1 69651,C(=O)(C(CCC)c1ccccc1)NC(CC)CN(C)C(C1CC1C)=O 69652,c1(OCC(=O)NC(c2ccccc2)C(C)NC(=O)C=CCF)cccc(Cl)c1F 69653,N1(CC(C)NC(Cc2cn(CC)nc2)=O)CCN(C(C2(COC)CCCO2)=O)CC1 69654,c1(C(=O)NCCCC2CN(C(=O)Cn3cnnc3)CCO2)cc(F)c(Cl)cc1Cl 69655,N#Cc1ccnc(C(=O)NCC2CC(NC(c3ccc(C(F)(F)F)o3)=O)C2)c1 69656,C1(CC(=O)NCCCN(C(C2CC2C(C)(F)F)=O)CC)CC2CCC1O2 69657,C(CS(=O)(=O)NCC(=O)OC(C)(C)C)C(c1nncs1)C 69658,Cc1c(C(=O)NC2CCC2NC(c2csc3nccn23)=O)oc2ccc(F)cc12 69659,C1(NC(Cc2cc(CC)nn2C)=O)CCN(C(=O)C(C)=CC2CC2)CC1(C)C 69660,C1(CC)CCC(CCNC(N2CC(NC(=O)OC(C)(C)C)C(C)C2)=O)CC1 69661,C1(CNC(C2CC2(F)F)=O)CC2(CCC2)CO1.C12CC(C1)C(=O)NC2 69662,S(=O)(=O)(c1cccc([N+](=O)[O-])c1)N(CCCC)C.C1(=O)C(CC2CC2)N1 69663,N1(C(c2c(C)onc2)=O)CCC(NC(=O)C=CCN2CCCCC2)C(CO)CC1 69664,N1(CC2(C(=O)NC)CCN(C(CN(CCC)C)=O)C2)CC(C)=CC(C)C1 69665,c1(CCC(=O)NC(C2CC=CCC2)C(=O)NCC(CSC)OC)nccn1C 69666,c1(C(N(C)CC2N(C(C3C(C)CCCC3)=O)CCCC2)=O)cnc(F)c(Cl)c1 69667,CC(F)(F)CCCNC(N1CCOC(c2cccc(F)c2)C1)=O 69668,C1(OCC(=O)OC(C)(C)C)CC2(CCC(C(=O)Oc3ccc(I)cc3)OC2)C1 69669,C1(CC)CN(C(c2cn(CC)nc2C)=O)CCO1 69670,N=c1nc(Cc2noc(C3CCCC3)n2)cc[nH]1 69671,c1(C(=O)NCCN(C)C(C2CCC3COCCC3C2)=O)cnc2c(Cl)cccn12 69672,c1(C(=O)NCC(CO)NC(=O)C(O)CF)ccnc2c(F)cccc12 69673,CCCC(CCCNC(=O)C(C)C)NC(C1(n2cccn2)CC1)=O 69674,c1(C(=O)NCC23C(CN(C(CCS(N)(=O)=O)=O)C2)C3)ccc2ccnc(Cl)c2n1 69675,c1(C(=O)NCC(CNC(C2(OC)CCSC2)=O)O)cc2c(ccn2C)[nH]1 69676,Cc1cc(N2CCC(CC(C)NC(c3ccc4c(c3)CC4)=O)CC2)nc(Cl)n1 69677,C1(CCNC(CSCC)=O)CN(C(=O)C(C2CC(F)(F)C2)OOCC)CCCO1 69678,Cn1nc(C(N2CCC(CCNC(c3cncc(Cl)c3)=O)C2)=O)c2c1CCSC2 69679,NC1(CC(=O)Nc2ncc(Br)n2Cc2ccccc2)CCS(=O)(=O)C1 69680,Cc1ccc(C(=O)NC23CCCN(C(c4ccco4)=O)C2C3)cc1C 69681,CC1(NC(=O)Cn2cnnn2)CCC(C(N2CC3CCC2C3)=O)CC1 69682,C(CCCNC(=O)NCCC(C)(CO)C1CCOC1)OC(C)C 69683,CC(C)CC(C)(O)CNC(=O)Cc1cn(OCC2CC3CC3C2)nn1 69684,C1(C(=O)NCc2c(CC)nccn2)CCCCCCN1C(C1CC=CCC1)=O 69685,N1(C(c2c(C)cco2)=O)CCc2ccccc2C(N(C)C(=O)CCOC2CC2)C1 69686,C(=O)(C1=CC2C=CC1C2)N1CC(NC(=O)Cc2nc([N+](=O)[O-])n[nH]2)C(F)C1 69687,Cc1ccc(CC(N2CC(NC(C3(F)CC=CCC3)=O)C(C(F)(F)F)C2)=O)cc1 69688,c1(C(c2ccc(F)cc2)O)cn(C2c3ccccc3CC2CC)nn1 69689,c1(C(N2CC(C(=O)Nc3ccc(C)c(I)c3)C2)=O)cnn2cccc(F)c12 69690,c1(COCC)nc(C)c(C(=O)NCCCC(C)NC(C2CCC(CC)O2)=O)s1 69691,C1(C(=O)NC)CCC(OC)(NC(=O)C(c2cc(C)ccc2F)(C)C)CC1 69692,Cn1cc2c(C(N3CC4CCCN(C(=O)Cc5cc[nH]n5)C4C3)=O)cccc2n1 69693,C(C(N=c1ccc2nnnn2[nH]1)C(C)C(C)C)NC(c1c(C)ncn1C)=O 69694,C1(NC(C=C(CC)C)=O)CCCC(NC(=O)C(c2cn(C)nc2C)(C)C)CC1 69695,N1(C(Cc2c(C)nc(SCC)s2)=O)CCC(NC(c2nocc2C)=O)C(F)C1 69696,O1NC(=O)CC2CCN12.C1CCN(C(=O)C(Cl)Cl)C1.CC(C)C 69697,CCCCCCC(F)C(=O)N(C(C)CN(C(=O)CCOc1ccccc1C)C)C 69698,C#CCC(CC(=O)NC(C)C(=O)NC)NC(C1CN(C)C1)=O 69699,c1(OCC(=O)NCC2C3CN(C(=O)CNc4cccnc4)CC23)ccccc1O 69700,c1(C(N2CC(N(C(CCCCN(C)C)=O)C)C(F)C2)=O)ccc(F)c(N)c1 69701,Cc1ccc(C(=O)NC2(Cc3ccc(Br)cc3)CC2)c(O)n1 69702,c1(C(N2C(C(=O)Nc3cc(Cl)ccc3CO)C=CC2)=O)cc(Br)cc2[nH]ncc12 69703,CCCC(CC)CCC(=O)NC12CC1CN(C(c1nnc(O)nc1O)=O)C2 69704,c1(C(N2CC(CC)(NC(=O)CCC3CCCC3)C2)=O)cnn(C(C)C)c1Br 69705,C1(Nc2nc(C)nc(N3CCC(OCCO)C3)c2)COC2(CCCCC2)C1 69706,Cc1ncccc1C(c1nnnn1C1CCC1)NCCCCOC(C)C 69707,c1(N2CC(C)(C)OC(CC(=O)O)C2)nccc(S(C)(=O)=O)n1 69708,C1(C(=O)NC(C(C)NC(c2cc[nH]n2)=O)C)CC(=O)N(Cc2ccccc2)C1 69709,CCC(C(=O)N1CC(CCNC(=O)C(CC)NC(=O)OC)C1)SC 69710,CCCCC(CNC(=O)Cn1cc(C#N)cn1)NC(=O)CN(C)C(C)C 69711,c1(CC(=O)NCCCN(C(=O)CC2CCCCN2C)C(C)C)ccc(F)c(F)c1 69712,c1(C(=O)NCC(CC)NC(C2CCCC2C(F)(F)F)=O)ccccc1C(=O)NC 69713,C12(CCCCC1)C(=O)N2C1CC1.C1(C)CCCC(F)C1.CC(C(=O)NC)=CC1CC1 69714,CCCCCC(C(C)(C)C)Nc1cc(NC2CCN(C)C2)ncn1 69715,N1(C(c2c(C)oc(Br)c2)=O)CCC2(CC(NC(=O)C=CSC)C2)C1 69716,C1(NC(CCCC#C)=O)CCC(O)CN(C(c2cc(-c3ccccn3)no2)=O)C1 69717,N1(C(c2c(OC)scc2)=O)CC2CC2(NC(C2(n3ccnn3)CC2)=O)C1 69718,C(=O)(C1CCCc2sccc21)NC(CNC(C(C(C)(C)O)(F)F)=O)C1CC1 69719,C(c1ccc(F)cc1)=CCC(=O)NCC1N(C(CN2CCC(OC)C2)=O)CC=C1 69720,C(=O)(C(C)(C)C(N)=O)NCC1(COC)CCN(C(c2ccc(SC)cc2)=O)C1 69721,NS(=O)(=O)CCC(=O)NCCC1COCCN1C(=O)C(O)C(F)F 69722,c1(C(=O)NCC(=O)NC(c2ccncc2)C2CC2)n[nH]c2c1COC2 69723,c1(C(N2CCC(N(C(CC(C=C)CC)=O)CCC)C2)=O)cn2nccc2nc1C 69724,N1(C(CC(COC)C)=O)CCN(C(C2CC(O)CN2C(C)=O)=O)C2(CC2)C1 69725,c1(C(=O)NCC2(OC)CCN(C(=O)C(F)C3CCOC3)C2)ccc(Cl)c(C)c1 69726,C(c1nc2ccccc2o1)=CC(=O)N(C(C)CNC(c1ncnc(O)c1F)=O)C 69727,C(CC(C(=O)NCc1nn[nH]n1)NC(c1csc(Cl)n1)=O)=CC 69728,C1(NC(C(c2cnc(CCC(C)C)s2)N(CCCOC)CC)=O)CCCOC1 69729,CC(C)C(CC(=O)NCc1nccs1)NC(c1ccn(C)c1)=O 69730,CCC(C)(C)C(O)C(=O)NC1(C2CCN(C(=O)CC(C)C3CCCO3)C2)CC1 69731,Cc1cc(C)c(C(=O)NC2CN(CCCC3CCOC3)CCC2C)c(C)n1 69732,C1(NC(C2CS(=O)(=O)C2)=O)CC2CC1N(C(c1csc(-c3ncc[nH]3)n1)=O)C2 69733,c1(Cc2c(C(N(C(CNC(C3(CCC)CC3)=O)C)C)=O)cno2)cccc(F)c1 69734,C=CCC(CC=C)C(=O)N1C2CCC1C(C(=O)NC1(C)CCCOC1)C2 69735,CCC(C(=O)NC(C)CCC(=O)NCCN(C1CC1)CC1CC1)C(F)(F)F 69736,CC(C(=O)NC(CC1CCC1)C(=O)NCCc1cnco1)C(F)(F)F 69737,c1(CNC(CCC=C(C)C)=O)ccnc(C(=O)NCCN2CCCC(O)C2)c1 69738,N1(C(C(=O)Nc2c(NC(C)=O)c(Cl)ccc2)=O)CCC2(C=Cc3ccccc3O2)C1 69739,C1(C(=O)NCCSC)CC(Nc2cscn2)CN1C(=O)OC(C)(C)C 69740,N1(C(C2(C)CN(C(c3c(CC)n(C)cc3)=O)C2)=O)CCC2(CCC(O)C2)C1 69741,N(C1CCOc2ccccc21)(C(=O)CC1CC1(F)F)CCCO 69742,n1(CC(C)NC(C2CC(c3ccnnc3)C2)=O)cc(CCCCCC2CC2)nn1 69743,N(C(=NCCC(C)(C)C)N(C)C1CCCC1)Cc1c(OC)ccc([N+](=O)[O-])c1 69744,c1(C(=O)NCC2C(C)CN(C(c3c[nH]ccc3=N)=O)C2)nncc2c1CCCC2 69745,C12(C(=O)NCC(C3CCCO3)OC)CC(CN1C(=O)C(C)CC1CCCC1)C2 69746,n1(CC)cc(Cl)c(=NC(=O)N2CCNC(C)(C)C2)[nH]1 69747,CCC(CCCC(=O)NCC1Cc2nccn2C1)NC(C1CCC(C)O1)=O 69748,c1(CSC(C)(F)F)csc(CNC(=O)CO)n1.C12CC1C(=O)N2.C1(N)CCC1 69749,CCCC(CC)C(=O)NC1CCC(NC(=O)CNC(=O)C=Cc2ccccc2)CC1 69750,c1(C(=O)NCCCN(C(C(n2ccc(C)n2)C)=O)C2CC2)cccc(C)c1C 69751,N1(C(CC(C)CN(C)C)=O)CCOC2(C1)CN(C(c1ccc(CO)nc1)=O)C2 69752,C(=O)(C(O)CC(N)=O)NC(CCC1N(C(c2c(CC)[nH]cc2)=O)CCCC1)(C)C 69753,N1(C(=O)CN2CCNCC2)CCOC2(C1)CC2(F)F 69754,CCS(=O)(=O)c1cnc(O)c(C(=O)NC2C3CN(C(=O)C(C)C4CCC4)CC23)c1 69755,C(=O)(C#CCC(C)C)NCCN(C(=O)CCC(C)OC)CC 69756,C(C(=O)NC1CCCCC1CC(=O)NCC1(C(=O)NC)CCCC1)(C(C)C)OCC 69757,CC1CCN(C(=O)C2=NOCC2)C(CNC(=O)CSCC(F)F)C1 69758,N1(C(C(CCCC)F)=O)CCC2CN(CCC3CC3C(C)C)CC2CC1 69759,Cn1nccc1CCNC(=O)CCC1(NC(C2CC2c2ccoc2)=O)CCCC1 69760,C(C)(C)(CC(F)C(=O)NC1CCCOC1)NC(C(C)SCC)=O 69761,c1(OC)ccccc1C(C)CC(=O)N1CCC(CNC(=O)Cc2csc(C)c2)C1 69762,c1(C(=O)NC2CC(N(C(C3C(C)C3C)=O)C)C2)cccc2c1nnn2C 69763,CC1CN(C(=O)CCc2nc(-c3ccsc3)no2)CCC1NC(=O)C=C1CCCC1 69764,c1(C(=O)NCC2CCCCN(C(C(CC)F)=O)C2)ccc(S(N)(=O)=O)o1 69765,Cc1cc(=NC(=O)CC2CCCCN2C(=O)C(c2ccccc2F)O)cc(C)[nH]1 69766,CCCCCC(C)Oc1ccccc1C(=O)Nc1ncccn1 69767,N1(C(C(C(CC)O)C)=O)CCCC2(C1)CN(C(=O)CCc1ccccn1)CCO2 69768,c1(C(N2C(C)(CNC(CCSCC)=O)CCC2)=O)coc(S(=O)(=O)CCOC)c1 69769,c1(NC2(CNC(CCCS(N)(=O)=O)=O)CCC2)cc2nn[nH]c2cc1[N+](=O)[O-] 69770,C(=O)(C(C)(O)CC(F)F)NCCCOCCNC(c1ccc(C(C)C)o1)=O 69771,c1(C(N(CC(CN(C(=O)C(=O)C2CC2)C)O)C)=O)coc(-c2ccccc2)n1 69772,O=C1Cc2cccc(C(=O)NC3CN(Cc4c(F)cc(I)cc4F)CC3O)c21 69773,C(=O)(N(CCC(N)=O)OC)C1CN(C(=O)C(C)=C(C)C)CC(CC)C1 69774,N1(C(C(OC)OC)=O)C2CCC1C(CNC(C1(c3cccnc3Cl)CC1)=O)C2 69775,N1(C(C(CN(C)C)O)=O)CCC(C(=O)O)(CNC(=O)C=Cc2ccoc2)C1 69776,c1(C(=O)NCC(C2CCCC2)NC(c2csnn2)=O)cccc2c1OCCO2 69777,c1(N2C(CC)CN(C(=O)C=C(C)C(=O)O)CC2)ncc2cc(C)ncc2n1 69778,c1(C(N2C(CN(C)C(C3CCCOCC3)=O)COCC2)=O)cnn2ccncc12 69779,CCC(C(=O)NCCOCCN(C(=O)CC1CCC(O)C1)C)C(C)C 69780,c12cnn(c1)C(=O)N1CCC(CC1)N(CCC)C2=O.C=CCC=O.C(C)(C)(C)O 69781,C(=O)(C1=C(Cl)CCCC1)N(C1CCCN(C(c2cc(Cl)cn2C)=O)CC1)C 69782,C1(O)(CN(C(Cc2cc(CC)on2)=O)C)CCN(C(=O)C(C)(C)C(F)F)CC1 69783,N1(C(CNC(C2(F)CC3(CCC3)C2)C)=O)CC2CC(C1)N(C(=O)OC(C)(C)C)C2 69784,N1(C(C(C)CC2CCC2)C(=O)Nc2ccccc2Cl)CCc2c(C(=O)O)n[nH]c2C1 69785,C(CC(C)C(=O)N1CCC(O)(CNC(c2nn(C)cc2SC)=O)C1)=CC 69786,N#Cc1ccccc1C=CC(=O)NC1CCCCN(C(=O)CC2CCC(O)C2)C1 69787,C(=O)(C(C)CC(C)(F)F)NCCCCCN(C(C1CC=C(C)CC1)=O)C 69788,C1(C(C)C)CNc2ccccc2C1CNC(=O)CCC(C)(C)c1nn[nH]n1 69789,Cc1ccc(C(N2CCC(CCNC(C34CCCC3OCC4)=O)C2)=O)c(F)c1F 69790,c1(CC(=O)C(CN(C(=O)CCN2CCC(F)C2)CCC)=O)ccccc1F.NC 69791,C(=O)(C=CS(=O)(=O)CC)NCC1(CNC(C2C(=C)CC2)=O)CCC1 69792,c1(C(C(=O)NCC)N(C2CC2)Cc2ccc(C)cc2)cc(C)cc(Br)c1F 69793,c1(SCC#C)cccc(C(=O)NC(CNC(=O)C(c2cccs2)SC)CO)c1 69794,c1(-c2n(C)c(I)nc2Cl)nc(C2CSc3ccccc32)no1 69795,N1(C(C2CN(C(C)C)C2)=O)CCN2CCN(C(C3CCC(=O)O3)=O)CC2C1 69796,C1(CNC(C(CC)F)=O)CCC2CN(C(c3cc4n(n3)CC(F)C4)=O)CCC2C1 69797,N1(C(C)C)CC2CN(CC34CCCC3C4)CCC12 69798,C(C(C(=O)N(CCCSC)C)C(C)(C)C)NC(C1N(CC)CCOC1)=O 69799,c1(OCC)nc(C(=O)NC2CC(NC(C3CCCC3c3nc[nH]n3)=O)C2)co1 69800,C1(C(C)O)CC(C)(C)CN1C(=O)Cc1cccc(F)c1.C12CC(C1)NC2=O 69801,C1(OC)=CC(C#N)=CC=NC(COC2C(C(=O)NCC3CC(CO)CO3)C2)=N1 69802,Cc1nnc(O)c(C(=O)NCC(C)N(C(=O)C(C)Cn2cccn2)C)c1C 69803,N1(C(C(N2CCCC(C)C2)=O)=O)CCC(NC(C2COC(=O)C2)=O)C1(C)C 69804,c1(CN(CCC(=O)NCC(C(C)(C)C)NC(C2C(C)C2)=O)C)ccc(Cl)cc1F 69805,c1(C(=O)OCC)cc(Br)c(F)cc1NC(C1CCN1Cc1cc(F)cc(Br)c1F)=O 69806,c1(CC)cc(=NC(=O)C2(F)CN(C(=O)CC3CC(O)C34CCC4)C2)[nH]n1C 69807,C1(C(=O)NCCCN(C(=O)C#CC2(C(F)(F)F)CC2)C(C)C)Cc2nncn2C1 69808,C12(C(=O)NC3(C4N(C(CC5(OC)CC5)=O)CCC4)CC3)CCN(CC1)C2 69809,c1(C(N2C(C(N3CCC(OC)CC3)=O)CC2)=O)c[nH]c2cccc(F)c12 69810,c1(C(N2CCC(NC(C(C)SC)=O)C(C)C2)=O)cccc2c1NCC2 69811,C(=O)(C(C(C)CC1CCOCC1)N(C1CCCN(C)C1)S(=O)(=O)CC)NCC=C 69812,C(=O)(C1=CC2(CCOCC2)C1)N1CCCC(C)(NC(=O)C2=CS(=O)CCC2)C1 69813,Cc1nnccc1C(N1CCC(CNC(=O)CN2CCCNC2=O)C1)=O 69814,N1(C(Cn2cc(C(C)O)nn2)=O)CC(NC(=O)CC(C)(F)F)CC1C 69815,C1(C(N2CCC3CN(Cc4ccccc4)CC23)=O)CCC(=C(F)F)CC1 69816,C12(C(=O)NCCCCC3CCCN(C(C(C(C)C)C)=O)C3)CC(C)(C1)OC2(C)C 69817,C1(C(=O)NC(CNC(c2cc(OCC)ncc2)=O)(C)C2CC2)CC2(C1)CC(F)C2 69818,C1(CC)CN(C(c2cc(CNC(C)=O)n(CCO)n2)=O)CCN1C(C)=O 69819,C1(C(N(C)CCS)=O)C2CN(C(=O)C(F)CC3CCOC3)CC12.Cc1cc(CC2CC2)on1 69820,C1(CNC(CCOCCCOC)=O)CN(C(C2OC3CCC2CC3)=O)CCN1C 69821,CC1CCN(C(=O)C=CC(=O)NC(C)(C)C(C)NC(=O)CCc2ccon2)CC1 69822,C1(CC(=O)N(CCNC(C(C(C)C)OCC)=O)CC2CC2)CCCC2(CCC2)O1 69823,C1(C(=O)OC)CCC(NC(c2ccsc2CNC(C2(C)COC2)=O)=O)C1 69824,C1(C(N(CCN(C(C)C)C(c2ccoc2Br)=O)C)=O)C(C(C)C)C1[N+](=O)[O-] 69825,c1(C(=O)NC2CC(C)(NC(CC(C)CF)=O)C2)nc[nH]c2ncnc1-2 69826,CC(CC(=O)NC(c1ccccc1)CNC(c1csc(CO)n1)=O)n1cccn1 69827,C1(NC(C2C(CC)C2)=O)CN(C(c2csnc2C)=O)CCC1C(F)(F)F 69828,c1(NS(=O)(=O)Cc2ccccc2I)ccccc1N1CCCCC1 69829,C=CC(C)(O)C(=O)NCCCC1(NC(=O)CSc2cccs2)CC1 69830,C1(NC(c2cccc(C3CCC3)c2)=O)C2CCN(C(C3CC=CCC3)=O)C12 69831,Cc1cc([N+](=O)[O-])cnc1C(=O)NC1CC2(C1)CC2NC(C1CCC(=O)C1)=O 69832,Cc1cc(C)c(C(=O)NCc2cc(C(=O)NC(C)C3CC3)n[nH]2)s1 69833,c1(C(=O)NCC(C)(C)OCCNC(C(CC(C)C)OC)=O)c(C)ccc(C)c1C 69834,c1(C(=O)NCCCN(C(c2cccnc2)=O)CC)cccc2scnc12 69835,C1(NC(CN(C)CC)=O)CC2CC(NC(=O)CSc3n[nH]c(=N)s3)C2C1 69836,C(=O)(CC(F)(F)F)NCC(=O)NCCNC(Cn1c(C)ccn1)=O 69837,C1(C(N2CCC(C(C)NC(=O)C(C)(C)C(N)=O)C2)=O)CNc2ccnn2C1 69838,C1(C(=O)NCCN(C(=O)C(=O)Nc2ccccc2)CC)COCCN1C 69839,CCCC(CC(=O)NC1(C(C)(F)F)CCC1)NC(=O)C(CC)N(CC)CC 69840,C(CC#CC)(C(=O)N1CCCC(O)C1)NC(C(C=C)C)=O 69841,C1(C)(C(N(CCCCO)CC)=O)CC12CCN(Cc1cc(C(F)(F)F)no1)CC2 69842,C1(C(=O)Nc2ccc(CC)nc2)CC2(CCC2)CN1C(c1cc[nH]c1)=O 69843,N1(C(C(=Cc2cccs2)C)=O)CCC2CN(C(=O)COc3ccon3)CC2C1 69844,CCCCCCC(C)(CC)C(=O)NC1CCC(NC(=O)CCc2nncs2)C1 69845,c1(C(N(C)CC2(NC(c3c[nH]c(=N)o3)=O)CCOC2)=O)cc(Cl)c(Br)[nH]1 69846,N1(C(C(=O)NC(CC)C)CC2C=CCC2)Cc2ccc(Br)cc2CC1C 69847,C(C(=O)N1OC2CCC1C2)C1CCN(C(C(N=S(C)(C)=O)=O)=O)C1 69848,C1(C2CC2)(CNC(CSC)=O)CCN(C(=O)C(C)(C)C(=O)OCC(C)(C)C)C1 69849,C(=O)(CC(C)C(C)C(C)C)NC1(CNC(c2nc(C)oc2)=O)CCOCC1 69850,C12CCCCN1C(=O)c1c[nH]nc12.c1(C(C(=O)NC2CC(O)C2)O)ccc(F)cc1 69851,c1(CNC(c2c(C)ncnc2)=O)nc(CNC(C2(CO)CC(C)(C)C2)=O)cc(O)n1 69852,C(=O)(C1=Cc2ccccc2C1)N1CC(F)(CNC(=O)C2=CC3(CCOC3)C2)C1 69853,CCS(=O)(=O)CC(=O)N(C1CN(C(=O)C=Cc2cnc[nH]2)CC1F)C 69854,CCCC(F)C(=O)NC1(CC(N2CC(F)(C#N)C2)=O)CCC1 69855,C(=O)(C1=CS(=O)CCC1)NC(C1CCCN(CCc2cn(CC(N)=O)nn2)C1)C 69856,C(CCNC(=O)CC1CC=CCN1C)(C(C)(C)C)NC(C1(C(=O)NC(C)C)CC1)=O 69857,C1(O)(CNC(C(C)N(C(C2(CCC=C)CC2)=O)C)=O)CCCCCC1 69858,N1(C(C2(CC)CCC2)=O)CCCN(C(c2ccc(OC(C)(C)C)nc2)=O)CCC1 69859,N1(C(c2ccno2)=O)CC(C2CCCN(C(C3(CO)CC3)=O)C2)C1 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69931,c1(CC)cc(=NCC2(O)CCN(C(=O)C=CCOC3CCOCC3)CC2)[nH]cn1 69932,c1(C(N2CC(NC(CCOC)=O)CC(C)(C)C2)=O)ccccc1C#CC1CC1 69933,C1(NC(c2sc(C)c(O)n2)=O)COC2(CCC2)C1.C12CCCC(C1)CNC2=O 69934,c1(C(=O)NCC2N(C(C(F)=CCC)=O)CCCC2)cncc2n[nH]c(C(C)C)c12 69935,CCCCCC(O)CC(=O)NCCC1(C(=O)Nc2cccc(C#N)c2F)CC1 69936,N1(CC(=O)NCC2N(C(CCOCCN(C)C)=O)CCC2)CCNC(=O)C1 69937,CC(CN1CCCCC1)C(=O)NC(C)CCNC(c1nn[nH]c1Cl)=O 69938,c1(CN(C)C(CCCCNS(C)(=O)=O)=O)ccc2cnccc2c1 69939,C#CC1(C(=O)NCCOCCOCC)CC(F)(F)C1.C12CC(C1(C)C)C(=O)NC2 69940,c1(NC(N(C(C)Cc2ccc(F)cc2F)C)=O)cccc2c1CCC(=O)N2 69941,C12CCCC(C1)C(=O)N2.C(CC(=O)C(CCNC1CC1)=O)NC(=O)NN1CCCC1.O 69942,c1(C2CC2)ccccc1F.C12(OC)CN(C1)C(=O)C1CC(C1)CNC(=O)C2 69943,N1(C(C2CCCN(CC)C2)=O)CC2(CC(CC(=O)NC3(CCF)CC3)C2)C1 69944,N1(C(c2c(C)ncc(Cl)c2)=O)CCCC2CN(C(c3cncnc3C)=O)CCC12 69945,c1(C(c2n(CCC)nnn2)NCCS(=O)(=O)CCOC)ccc2nonc2c1 69946,N1(C(CCc2ccc(OC)nc2)=O)CCCC(C2CN(C(C3(CO)CC3)=O)C2)C1 69947,C(=O)(CCC(C)(C)OC)NC(CC)(C)CNC(=O)C(C)N(C)C 69948,C1(=CC(N2CC(CNC(CC3(C#N)CCC3)=O)C3C2C3)=O)CCCCC1(C)C 69949,C(=O)(C(F)C(F)(F)F)N(CCCC1OCCN(C(C2C(C(C)=O)C2(C)C)=O)C1)CC 69950,N1(C(C(CCC)NC(C)=O)=O)CC2CCC(C(=O)NCC(C)CC3CC3)C2C1 69951,N1(C(CC(C2CC2)NC(c2cn(CCC)nn2)=O)=O)CC2CC2(CC)C1 69952,N1(C(c2cc(C#N)c(N)cc2O)=O)CCC2CCN(C(=O)COCCO)CC2C1 69953,C1(F)(C(=O)NC(C(C)C)CCN(C(=O)C=Cc2nnn(C)n2)C)CC2(CCC2)C1 69954,c1(NC(c2ccc(OC)c(OC)c2)C#N)cccc2c1OCCC2O 69955,N1(C(c2n(CC)ncn2)=O)CCC(O)C(NC(C2CC3(CCCO3)C2)=O)C1 69956,CCCC(O)C(CO)NC(=O)C1=CCN(C(c2cc(C3CC3)[nH]n2)=O)C1 69957,C1(NC(c2cn(-c3cccc(F)c3N)nn2)CC)CC2(CCC(C)(OC)CC2)C1 69958,c1(CCCC)cccc(CN2CCC(Cn3nc(C)cc3C)C2)c1 69959,C(=O)(C(C(C)C)n1ccc(C2CC2)n1)NCCCN(C(CSCCCC)=O)C 69960,C12(C(=O)NC(C)CN(C(=O)CC3CCN(CC(F)(F)F)C3)C)CCCC(CO1)C2 69961,N1(C(C2(CC)CNC(=O)C2)=O)CCC(C)C(CNC(c2cc(C)ccn2)=O)C1 69962,CCCCC(=O)C(=O)NC12CCC(CNC(c3nn(C)cc3C)=O)(C1)OC2 69963,C1(NC(C2C3CNC(=O)C32)=O)CN(C(c2cc(Cl)ccc2Cl)=O)CC1C1CC1 69964,N(C(=S)N1CCC(Oc2ccc(F)c(F)c2)C1)C(C)C 69965,c1(N2CCN(C(=O)NC3CC3)CC2)ncnc2ccccc12 69966,C(=O)(C=C=C(C)C)N1C(C(=O)NCCC2(COC)CC2)CC1C 69967,CCCC(C(=O)OC)C(=O)N1CCC2CC12C(=O)NCc1ccco1 69968,N1(C(Cn2c(CCC)ncc2)=O)CCC(O)C(N(C(=O)Cc2ccon2)C)C1 69969,Cc1cc(O)cc(O)c1CN1CC(NS(=O)(=O)Cc2ccccc2)C(C)C1 69970,C#CC1CCC(C(N2CCOC(C(C)NC(=O)COc3cn[nH]c3)C2)=O)CC1 69971,c1(CCC(N2CCC(O)(CNC(C3(O)CCCC3)=O)C2)=O)ccc(F)c(F)c1F 69972,C(=O)(C1CC(=O)Nc2cc(F)ccc21)N1CC(NC(C2(C3CC3)CC2)=O)C(F)C1 69973,C(C(C)(O)C(=O)NCCC1CC(NC(=O)CCNC(c2cccc(F)c2)=O)C1)OC 69974,CCC(C)(C)C(=O)C(=O)NC1(CO)CCCN(C(=O)C(c2ccc(C)cc2)O)C1 69975,c1(C(=O)NCC2(C)CCCN2C(C2CCSCC2)=O)cccn2cnnc12 69976,CC(C(=O)NCCC1C(NC(c2cccs2)=O)CC1)NC(=O)CCOCCSC 69977,c1(C(=O)NC(C(C)NC(c2cnn(C(F)(F)F)c2)=O)C)cc(Cl)n(C)n1 69978,C1(C(=O)NC2C(F)CCCC2)Cc2nc3ccccc3n2C1 69979,C1(CCC(C)C)CCN(CC(=O)NCCC2CCCCC2)CC1 69980,c1(C(=O)NC(CN(C(=O)CCn2cccn2)CC)C)cccc2nonc12 69981,c1(OC(C(=O)NCC2CN(C(CC3C(C)C3)=O)C2)C)cccc(Br)c1 69982,Cc1cc(C=CC(N2CCN(C(=O)C(C(C)C)N(C)C)CC2C)=O)c[nH]c1=N 69983,C1(C(=O)NCC(C)(C)OC(C)C)CCC2CCC1N2C(C1CC2(C1)CC21CC1)=O 69984,Nc1sc2c(c1C(N1CC(O)(CNC(C3C4CCCC34)=O)C1)=O)CCC2 69985,CCC(CNC(C12CC(C)(C1)C2)=O)(CC)NC(=O)CCn1cccn1 69986,C(=O)(CS(=O)(=O)CCOC)NCC1OCCN(CC)C1.C1(=O)C2=CCC(C2)N1 69987,C1(CCNC(C23CC(CC)(C2)C3)=O)CN(C(C2CCS(=O)(=O)N2)=O)CC1C 69988,c1(C(=O)NC2COC3CN(C(c4c[nH]ccc4=O)=O)CC23)cnc2[nH]ncc2c1 69989,C1(OC)(CNC(=O)CC2(C)CCN2C(=O)C(C)OCC(C)C)CCOC1 69990,N1(C(C2(C)CC2)=O)CCC2(CCOCC2)C(NC(c2cc(C(N)=O)nc(Cl)c2)=O)C1 69991,C1(C(=O)NCC2CC(NC(c3ccnnc3O)=O)C2)OCC2CCCCC12 69992,C1(CC)CCC(CC)CN1C(c1ccc(-c2ccccc2)[nH]1)=O 69993,C1(C(=O)NCCCCOC)CN2CCC1CC2.C1(OC)C(=O)N2CC1C2 69994,C1(CNC(CC2CCC(=O)N2)=O)CC2(CC2)CN1C(c1nc(C2CC2)ncc1Cl)=O 69995,C(=O)(C(F)(CNC(=O)C(CCC)N(C)C)C(C)C)NCCCCCC 69996,C1(C)(CC(=O)NCCOCC#C)CCN1C(=O)C(c1cncnc1)C 69997,c1(C(=O)NCCCCC(=O)NC2(CC=C)CN(C(C)=O)C2)c[nH]cc(C)c1=O 69998,c1(Cn2c(C(=O)NC(C)C)ccc2)cc(Cl)ccc1C(F)(F)F 69999,N1(C(C(C)Oc2ccc(C)cc2F)=O)CCC2(CCC(NC(=O)CO)CC2)CC1 70000,N1(C(c2nc(CC)oc2)=O)CCC(NC(=O)Nc2ccc(C)cc2OC)C(O)C1 70001,c1(C(C)C)ccc(OCCCC(=O)NC(C)CNC(c2cnsc2)=O)cc1 70002,C=CCCCCCC(=O)N1CCN(C(c2ccc(C(F)(F)F)nn2)=O)C(C)C1C 70003,CCS(=O)CC(=O)NC1(CNC(=O)COCc2ccc(OC)nc2)CCOC1 70004,C1(CNC(=O)CN2CC3CC3C2)CCCCN1C(C1(C2CCC2)CC1)=O 70005,C(=O)(CC(CC(N)=O)c1ccccc1)NC(C=CC(=O)OC(C)C)C 70006,c1(C(=O)NC2CCC(NC(C3(C=C)CC3)=O)C2)ccnc2c1CCO2 70007,c1(C(N(C)CC2OCCN(C(c3cn(CC)nn3)=O)C2)=O)ncccc1N=[N+]=[N-] 70008,C1(NC(CCCC(C)C)c2nnnn2C2CCC2)Cc2cccnc2C1 70009,c1(CCCC(=O)NCC(C)N(C(C(C)OCC2CC2)=O)C)cccc(Cl)c1 70010,C1(C)(NC(C2N(C(=O)CC(C)SC)CCC(=C)C2)=O)CC(C)(C)OC1=O 70011,C(=O)(C(O)CC[S+](C)C)N1CCC(OCCNC(COC(CC)(C)C)=O)C1 70012,CCC(C)CCCCC(=O)N1CCC(N(C)C(c2ccc3oc(O)nc3c2)=O)C1 70013,C(c1ccc(OC)c(F)c1)=CC(=O)NC(C(=O)OC)CC1CCCC1 70014,c1(CC(=O)NC(C2(CNC(C(C)OCC=C)=O)CC2)C)ccc2ccn(C)c2c1 70015,O=S(=O)(c1cc(F)cc(F)c1)Nc1ccc(Br)c(Cl)c1F 70016,c1(C(N(CCNC(c2ccc(=NC)[nH]c2)=O)CC)=O)ccn2nnnc2c1 70017,C1(c2n(CC)nnn2)(NCCOCCF)CC(C(=O)OC)(OC)C1 70018,C1(C(=O)Nc2cccc(CF)c2)C2CCC1CN(C(C1C3CCC(=O)C13)=O)C2 70019,C=C1CCN(C(=O)CC2CC2(C)C)C(C(=O)NC2C(O)CC2O)C1 70020,c1(CC)nc(-c2cc(C(F)F)no2)n(CC(N2CCCCCC2)=O)n1 70021,C(C(=O)NCCCN1CCN(C(=O)C=C(Cl)Cl)CC1)(C(C)(C)C)OCC 70022,Cc1ncc(NC(C2(CCNC(C3(C(=O)N)CC3)=O)CCC2)=O)c(C)c1C.C1CC1 70023,c1(C(=O)NCC23CC(NC(CC4C(C)CCO4)=O)(C2)C3)c(Cl)csc1Cl 70024,CN1CCCCC1C(=O)N(CCc1cccc(NCCO)c1)C1CC1 70025,CC(C)CC(C(=O)N1C2CCCC1CC(NC(c1cn(C)cn1)=O)C2)C(C)C 70026,C1(C(=O)NCC(C)N(C(c2ccc(F)cc2F)=O)CC)CN(CP(C)(C)=O)C1 70027,N1(C(c2c(CC)cc[nH]2)=O)C2CCC1C(CNC(=O)CCC(=O)N(C)C(C)C)C2 70028,c1(C(C)NC(=O)NC(C(=O)OC)C)cccc(F)c1 70029,C(C(CC(=O)NCCC(Cc1ccccc1)OC(=O)C1CC1)c1ccccc1)OC 70030,C#CCCCCCC(=O)NCC(C)C(=O)NC(c1ccnn1C)COC 70031,CCCCCC(O)CC(=O)NCC1CCCN1C(c1cnn(C)c1C(F)(F)F)=O 70032,C(CSC)(CC(=O)NC(c1ncc[nH]1)C1CC1)NC(C=C(CCC)C)=O 70033,CCC(CC(=O)NC1COCCOC1)NC(=O)C(C)C1(O)CCC1 70034,C#CCCC(C(=O)N(C(CO)C(C)C)C)NC(=O)C(C)NC(C)(C)CC 70035,C1(C(=O)NCCC(=O)NC(CC)C)CCN(C(C2CC2F)=O)C12CC2 70036,C1(C(=O)NCC=CCNC(C2(CC=C)CCCC2)=O)Cc2nnc(C)n2C1 70037,C1(NC(CCOCC(C)C)=O)CCC(C(N2CCC2CC2CC2)=O)C1 70038,c1(C(=O)NCCC(C)NC(=O)CCC(C)CN(C)C)cc2n(n1)CCCC2O 70039,C1(NC(=O)C2=CC3CCCC23)CCN(C(c2n[nH]c3c2CSCC3)=O)CC12CCC2 70040,c1(-c2cncc(OC(C)C)c2)ccc(F)c(CNC(=O)CCCc2cccs2)c1 70041,c1(C(N2CC(NC(c3cn(CCC)nc3C)=O)C2)=O)ccc([N+](=O)[O-])cc1F 70042,C12(C(=O)NC(C)CCCNC(C3NC(=O)CC3C)=O)CCCCC(=O)N1CCC2 70043,N1(C(C(CC)c2ccccc2)=O)CCC(NC(c2cnc(C)cn2)=O)C(C)(C)C1 70044,Cc1cc(C(N2CC3CC(NC(c4nnc(C(C)C)s4)=O)C2C3)=O)c(C)cc1Cl 70045,C1(CNC(C(C)OCCC=C)=O)CCC(NC(c2cn(CC(N)=O)nn2)=O)CC1 70046,N1(C(C(C)c2cc[nH]n2)=O)CC(CNC(c2cc(C(N)=O)no2)=O)C2(CC2)C1 70047,C1(C)(C(N2CC(CC(NOC(CC)C)=O)OCC2)=O)CC2C=CC1C2 70048,C12(CC(=O)NCC=CCSC)CCC1CN(C(=O)CCc1cccn1C)C2 70049,c1(C(N2CC(C)C(CNC(C3CC(C)(O)C3)=O)CC2)=O)ccc2c(c1)CCC=C2 70050,CC#CCC(C(=O)NCCS(N)(=O)=O)NC(C1CC(CCC(N)=O)C1)=O 70051,c1(CNC(C(n2cc(-c3cc(C)ncc3)nn2)C)=O)c(C)ccnc1O 70052,C1(CNC(CC(C(=C)C)OCC)=O)CC2CCC1N(C(C1(Cl)CC1)=O)C2 70053,c1(C(=O)NCCC2(OC)CN(C(=O)C(C)N(C)C(C)=O)C2)cccc2ccsc12 70054,N1(Cc2n(C)cc(Br)n2)CCC2(CC(C(=O)Nc3cccc4nc[nH]c34)=NO2)C1 70055,C1(NC(=O)NC2CCN(C(C)C)CC2)CC2CC(Nc3ccc(F)c(F)c3)CC12 70056,N1(C(CC(COC)C)=O)CCC2(CCCN2C(=O)CCc2nc(=N)[nH][nH]2)CC1 70057,c1(C(=O)NCCCOCCCNC(CC2(CC)CC2)=O)cnc2ncnc(O)c2c1 70058,C(=O)(C1=NNC(=O)CC1)N(C(=O)Cc1nnn(C(C)(C)C)n1)C.C12CCCN(C1)C2 70059,N1(C(C(=O)NCCCCCC)CCC2CCCO2)CCCC(CCO)CC1 70060,Cc1nc(NC2C3CCC(C3)C2C(F)(F)F)c2sccc2n1 70061,Cc1ccc(F)c(C(=O)NC(c2ccnn2C)C(=O)NCc2ncn(C)n2)n1 70062,C12(NC(CCSC)=O)CN(C(c3nc(C)n(C)c3C)=O)C(COC)(C1)C2 70063,c1(CN(C2CCCC(NC(CC3CC(OC)C3)=O)C2)C)cn2nc(C)sc2n1 70064,C1(C(N(C(C(=O)NCCN(CCOC)C)C2CC2)C)=O)COCCN1C 70065,C1(C(N2CC3C(CNC(C4CCCC4)=O)(C3)C2)=O)CCN(CCO)C(=O)C1 70066,CCC(CC(=O)N1CCC2CC12C(=O)NCC(C)(C)CN=[N+]=[N-])C(F)F 70067,CCCCCCCCCC(=O)NCC1CN(C(=O)C2=NNC(=O)CC2)CCO1 70068,c1(N2CCCC(CC(C)(C)C)C2)nc(=N)[nH]c(=NCc2nccs2)[nH]1.CC(F)F 70069,C(C(COC)CC(=O)NCCCC(=O)NCC1COCC1O)OC 70070,c1(C(N2CCC(C(F)F)(CNC(C(CC)(C)O)=O)C2)=O)ncnc2ccsc12 70071,C1(C(N2CCC(C(=O)N(C)CCC3CC3)(CF)C2)=O)(OC)CCCOC1 70072,C(=O)(C(C)(C)C(C)O)N1CCCC(CN(C(c2c(C)oc(Cl)n2)=O)C)C1 70073,c1(C(N2CC(NC(c3ncc(OCC)nc3)=O)C(C)C2)=O)cc(C)nc(Cl)c1N 70074,Cc1nc(CC(N2CCCC2C=CC(=O)NCCCc2ccccn2)=O)sc1C 70075,C1(C2CC2)(CNC(C(CO)OC)=O)CCN(C(=O)Cc2n[nH]c(C)n2)C1 70076,c1(CC(C)NC(CC)=O)cccc2c1CCCN2C(=O)C=CCOC(C)=O 70077,C1(CNC(C(C=C)O)=O)CCCC2CN(C(=O)CCCCC(=O)NC)CC12 70078,c1(C(N2C(CNC(CC(CCC)(C)O)=O)CC2)=O)cc(F)cc2nccnc12 70079,C1(NC(c2c(C)cc(C)o2)=O)CS(=O)(=O)CC1NC(c1nc(C)n(C)n1)=O 70080,C#Cc1cncc(C(N2CCN(C)CC2CNC(=O)C(C)n2cccn2)=O)c1 70081,C1(N(C(=O)C(=O)N(C2(C)CCCC2)CC)CC#C)C(C)CCCC1C 70082,C(=O)(C(O)C(F)(F)F)NCCSCC(=O)NCCc1csnn1 70083,c1(C(N(C(CN(C(C(COCC)C)=O)C)C)C)=O)cc2n(n1)CCCC2 70084,N1(C(c2nc(CNC(c3ccc(C)n3C)=O)oc2C)=O)CCc2cccc(F)c21 70085,C(CN=c1[nH]c(Cl)ncc1CO)C1CCC(NC(C2OCCN(C)C2)=O)C1 70086,C=CCC(C(=O)NCC1CC(F)(F)CN1C(=O)Cc1ccc(F)nc1)C(C)C 70087,c1(C(=O)NCCCNC(C2CC(O)(C(F)(F)F)C2)=O)ncn2c1CCCC2 70088,C1(NC(CCc2cnc(C)o2)=O)CN(C(C2(C(F)F)CCCC2)=O)CC1C1CC1 70089,N1(c2ncc(OCC)cn2)CCC(C2CN(Cc3nc(Cl)ccc3F)C2)CC1 70090,N1(C(=O)CC2CC3CC3C2)CCN(C(=O)CCCS)C(C(F)F)C1.C1(C=O)CCCC1 70091,C1(CNC(c2csc(Cl)n2)=O)COCCN(C(C2C3CCCC23)=O)C1 70092,N1(C(=O)CC2CCC2)CCC2C(C1)CN2C(C1CCOCC1)=O 70093,c1(-c2cn(CC(C)NC(c3ccc(OC)c(N)c3)=O)nn2)noc2c1CCCC2 70094,Cc1nc(C(C)C)oc1C(=O)N(C)CC1CCCCN1C(c1ccccn1)=O 70095,C12(NC(C3N(C(c4c(OC)scc4)=O)CC(O)C3)=O)CCCN(CC1)C2 70096,C=CCC(C)C(=O)N(C1CCC(NC(C2(OC)CCOCC2)=O)CC1)C 70097,c1(CNC(CC2CC(SC)C2)=O)ccc(Cl)cn1.C12(CCO)CN(C1)C2=O 70098,C1(C2CC2)(NC(c2c(C(C)C)ccs2)=O)CCN(C(=O)CNC(N)=O)C1 70099,N1(C(C2(CC)CCN(C(c3c(C)cccc3F)=O)C2)=O)CCC2(CCCCC2)C1 70100,c1(CNC(CN(C(=O)CN2CC3CC3C2)C)=O)cncnc1 70101,C1(CC(=O)N(C)C(C2(CO)CCCCC2)=O)CCCN(C(=O)C=Cc2cc[nH]c2)C1 70102,CC1C(=O)NC(=O)CN1C(C1(F)CCN(C(c2c[nH]c(=S)cn2)=O)C1)=O 70103,C(C(CO)C(F)(F)F)NC(C12C(CN(C(C3OCCN(C)C3)=O)C1)C2)=O 70104,CCC(CO)C(=O)N1CCC(n2cc(CNC(=O)Cn3nccn3)nn2)CC1 70105,C1(CC)CCN(C(C2CC23CCC3)=O)C1C(=O)NCC(=O)NC(C)C 70106,CC(CC=Cc1ccccc1)C(=O)N1CCC(NC(C2CC2CF)=O)C1 70107,C(C)(CCCC(=O)NCC1OCC2CCC1C2)NC(CCCOC(C)=O)=O 70108,C12(NC(CN=S(C)(C)=O)=O)CCOCC1CN(C(c1ccncc1)=O)C2 70109,C(=O)(C1CCCn2ccnc21)N1CCC(N(C(CCCS(N)(=O)=O)=O)CCO)CC1 70110,c1(C(=O)NCCOCCN(C)C(C2(C)CCNC2=O)=O)ccc2c(n1)CCO2 70111,C(N=c1nc(OC)c2nc[nH]c2[nH]1)C1OCCN(C(C2(SCC)CC2)=O)C1 70112,C(c1ccc(C(N)=O)o1)=CC(=O)N(CCNC(C(CO)OC)=O)C 70113,CC(CNC(=O)CN1CCC(=O)CC1)CC(=O)N(C)Cc1nnc(O)o1 70114,C1(NC(C(C)NC(=O)C(C)(C)C)=O)CC(O)CN(C(=O)CSC(F)(F)F)C1 70115,c1(C(N2CC(CNC(C=C(C)C(F)F)=O)N(C)CC2)=O)cccc2nc[nH]c12 70116,C=C(Cl)CC(C(=O)NCCCC(N)=O)NC(c1coc(SC)c1)=O 70117,C1(C(=O)NC(C2(C)CC2)CO)CCCCN(C(C2(O)CCOC2(C)C)=O)C1 70118,C1(N(C(C)C(=O)OC)C(C2COC2)=O)CC2C(NC(c3ccccc3)C)C2C1 70119,N1(C(C(CC)c2ccccc2)=O)CC2CN(C(=O)Cc3cnc(Cl)c(C)c3)CC12 70120,Cn1nnc2c1CCC(C(=O)NC1CCC(n3cc(-c4cn[nH]c4)nn3)CC1)C2 70121,N1(C(CC(CCC)(C)O)=O)C2CCC1C(C)C(NC(C1CCC(F)(F)CC1)=O)C2 70122,c1(NC(CC2OCCN(Cc3cnc(C(C)C)s3)C2)=O)cc(Cl)ccc1I 70123,N1(CCCC)CCCCC1C(=O)N(CCCCNC(C1(C(C)(F)F)CC1)=O)C 70124,CC(C)CC(CNC(C12CC1CN(C(c1scnc1Cl)=O)C2)=O)CO 70125,C1(NC(=O)Cc2cc(C(F)(F)F)n[nH]2)CC1C1CCCN(C(=O)C=CI)C1 70126,C1(CC(=O)NCCC(=O)NCCC)CN(C(c2cn(C3CC3)nn2)=O)C(C)(C)C1 70127,C(=O)(C#CC1(C)CCCO1)N(C)Cc1cccc(CNC(c2ccnn2C)=O)c1 70128,CCCC(O)C(=O)N(C)CC1COCCN1C(=O)CC12COCC(C1)C2 70129,Nc1cc(C(=O)NCCOC2CN(C(=O)CCc3ccncn3)C2)cc(Cl)n1 70130,C1(C(N2CCC(Cn3ccnc3)CC2)=O)Cc2ccc(O)cc2CN1 70131,C1(C(N2CCC(C(=O)NCCCc3cn(C)nc3)CC2)=O)CCC(C)(C)OC1 70132,c1(C(=O)NC(=O)CN(CCC2CC2)CCCC2CC2)ccoc1I 70133,c1(CC(=O)NC(C)(C)CN2CCN(C(c3csnn3)=O)CC2)cc(Cl)cc(Cl)c1 70134,C12(C(=O)Nn3cc(C#N)cn3)CCC(C=O)(CO1)C2.C12(C(=O)OC)CC(C1)C2 70135,c1(OCCCOC)cc(NC(N2CC(CC#N)C(C)C2)=O)ccc1OC 70136,C#Cc1ccc(F)cc1C(=O)NC1CN(C(=O)CC(C)F)CC1c1ccccc1 70137,C(=O)(C(C)C(CC)CC)N1C(C(=O)NCC(=C)Br)CC(=O)C1 70138,c1(C(=O)NCC(CN(C(COCC)=O)C)O)cc2sccc2n1CC1CC1 70139,C(CNC(c1cnc(C#N)s1)=O)(C(C)(C)C)NC(C1(COC)CC1)=O 70140,C=C(C)C(C)(C)C(=O)NC1CN(C(=O)C(C)OCC2CCC2)CCC1C(F)(F)F 70141,c1(C(=O)OC2C(OC)CN(c3ncc(Cl)c(O)n3)CC2)ccc2ccnc(Cl)c2n1 70142,c1(C(=O)NC2CCC(NC(c3ccc(Cl)s3)=O)C2)n[nH]c2c1CCC2 70143,C#CCC(C)(C)C(=O)N1CC(C(=O)N(c2cccc(N(C)C)c2)C)C(CC)C1 70144,C(=O)(CCCCCSC)NCCCC1CCN(C(C2C(=C)CC2)=O)C1 70145,C1(C(=O)NC2C(NC(c3c(Cl)cn(CCC)n3)=O)CCC2)CCc2nncn2C1 70146,C1(CC(=O)NCCC(=O)NC2CCN(C(c3ccoc3)=O)C2)CC(C2CC2)C1 70147,c1(C(N2CC3C(CNC(CC(=C=C)C)=O)C3C2)=O)cc[nH]c2nccc1-2 70148,CC(C)C1=NOC(C(N2CCC(C(C)NC(C3CC(=O)C3)=O)C2)=O)C1 70149,C=C=CCCC(=O)NCCC1CCC(NC(=O)CCS(C)=O)C1 70150,C1(NC(CCCc2ccc(C)s2)=O)CN(C(C2CC3COCC3C2)=O)CC12CC2 70151,C1(NC(C=CC(C)(C)SC)=O)CCCC1NC(=O)C(C)CC1CCC1 70152,N1(C(c2scc(C)c2C)=O)CCC2CC2(C(N2CCN(C(C)(C)C)CC2)=O)CC1 70153,c1(C(=O)NCc2c(C#N)cc(F)cc2)ncncc1C1=CCOCC1 70154,c1(C(N2CC3C(NC(CC4CC(OC)C4)=O)C3C2)=O)c(C)nn2ccccc12 70155,N1(C(CCN(CC(C)(C)O)C2CC2)=O)CCCC(C2CCN(C(=O)CC#N)CC2)C1 70156,c1(C(=O)NCC2(NC(CCCOCC=C)=O)CCCC2)ccc(OCC)c(F)c1 70157,c1(OC)ccccc1CCCNC(=O)C(C(C)C)N1CCOCC1 70158,C(=O)(C(O)C(C)(C)C)NC(CC)C(=O)NC1(C)CC(C)(C)C1 70159,C1(NC(=O)C(CO)c2ccccc2)CC2CC1CN2C(=O)C1=COCCC1 70160,N1(C(C2C=C(C)CS2)=O)CC2(CC(CNC(=O)C=CCF)CO2)C1 70161,c1(CC)ccc(C(N2CCCC2CNC(c2coc(C)n2)=O)=O)cc1 70162,C(CC(=O)NCC1CC(C)N(C(=O)CN2CC3CC3C2)C1)(C1=CCCC1)OCC 70163,C1(F)(NC(C2(OC)CCC2)=O)CCCN(C(=O)CCO)C1.C1(NC=O)COC1 70164,C(=O)(CCCCC(=O)NOC(C)(C)C)NC1C(NC(C(CC)=CCCC)=O)CCC1 70165,c1(OC)cc(C)cnc1C(N1CCC(O)(CCNC(C2C(C)C2C)=O)CC1)=O 70166,CC1(C)C(=O)NCC1C(c1cc(C(F)(F)F)ccc1O)N1CC(F)(F)C1 70167,C(=O)(CCC(=O)NCC1CCCN1C(=O)CC1CC1c1cccc(F)c1)NCC 70168,C1(N(C(=O)CC2CC(O)C2)C)CCCC(NC(C2CC(F)(F)CS2)=O)C1 70169,C(=O)(CCCC(=O)NC(C)C)N1CCC(O)(C(C)NC(c2c(NC)snc2C)=O)C1 70170,N1(C(C(CCC)N(C)C)=O)CCC2(CC(NC(c3c(C)cc(Cl)cc3C)=O)C2)C1 70171,N1(C(c2cncc(NC)c2)=O)CC(O)C(O)C1CNC(C1CC1OC)=O 70172,N1(C(c2nn(CC)c(O)c2)=O)CCN(C(=O)C(C)(C2CC2)OC)CC(C)C1 70173,C(=O)(C(C(C)(C)C)N(C)C)N(CCC1(NC(C(c2ncccn2)CC)=O)CC1)CC 70174,C(=O)(C(CO)C(C)(C)C)N1C(c2n(C)ncc2)CN(C(=O)CCSC(=N)N)CC1 70175,CCCCS(=O)(=O)N(C(C(=O)N1CCC(COC)(OC)C1)C(C)C)CC 70176,C1(C(=O)NC(CNC(C2CN(C3COC3)C2)=O)CO)CCCN2CCCCC12 70177,c1(SC)ccc(C(F)(F)F)cc1S(=O)(=O)NC(c1ccc(C(C)(C)C)cc1)C 70178,C1(C(=O)NCCOC2CN(C(CCc3cnc(C)s3)=O)C2)CN(C)CCO1 70179,C=CCC(F)(F)C(=O)N1CC(NC(=O)C(C)Cc2ccco2)C2(CC2)C1 70180,N1(c2n(CCOC)c(CC3(S(C)(=O)=O)CC3)nn2)CC2CN2C=NC=CC1 70181,Cc1cc(C(=O)NC(CO)C(C)NC(C2(C3CCCCO3)CCC2)=O)nn1C 70182,c1(C(N(C(CCNC(c2cccc(CC)c2)=O)C)C)=O)ccc2snnc2c1 70183,CN(C)NC(=O)CCC(=O)OC(c1ccnn1CC1CCC(F)(F)CC1)=O 70184,CC1(C)CNCC1N(C(C1CC1c1ccccc1)=O)CCC(F)(F)F 70185,C1(NC(c2c(C)cc(CNC(C(C)=CC(C)(C)C)=O)o2)=O)CCCC1C1CC1 70186,C1(C(C)NC(c2ccccc2)=O)CCCN(C(=O)Cn2cnc(=N)[nH]2)CC1 70187,c1(C(N2C(CCNC(C3(CC#C)CCCO3)=O)CCCC2)=O)cnc(F)c(Cl)c1 70188,c1(-c2c(CN3CCCC(C)(C)C3)c[nH]n2)cc(F)c(F)c(F)c1 70189,c1(C2CCN(C(=O)CC3CCN(Cc4occc4Br)C3)CC2)ccc(F)cc1F 70190,C1(C(=O)OC)CCN(C(c2cnnn2C)C(=O)NCCNCCCC2CC2)CC1 70191,C(=O)(CC(C)C(F)F)NCC1(O)CCN(C(c2nc(C)oc2C)=O)C1 70192,Cc1cc(C(=O)NC2CCCCC2NC(c2cccs2)=O)nn1CC(F)(F)F 70193,c1(C(N2CCN(CC(C)(C)NC(CC=CC)=O)CC2)=O)cnc(C)c(C#N)c1 70194,C1(CC)CCN(C(=O)CSCc2nc[nH]n2)C(C(=O)N)C1.C12CC(=O)N(C1=O)C2.CC 70195,n1(CC(N2CC(CNC(COc3cccc(C)c3)=O)C2)=O)cc(P(C)(C)=O)cn1 70196,c1(C(N2CCN(C(c3ccnnc3S)=O)C3CC23)=O)c(OC(C)=O)cccc1C 70197,N1(C(CC2(C#N)CC2)=O)C2CCC1CN(C(C1Cc3ccccc3S1)=O)C2 70198,CC1(C)OC2CC(COc3ccccc3)(C2)O1.C12CC3(C1)CC3CNC(=O)N2 70199,Cc1ccc(-c2cc(C(N3CCC3C#N)=O)nn2C)c(C)n1 70200,n1(CC(N2C(C)CC(CNC(=O)CC3(CN(C)C)CC3)C2)=O)ccc(O)nc1=O 70201,c1(NC)ccc(Cl)c(C(=O)NC2CC(NC(=O)C=C(Cl)Cl)C23CCC3)c1 70202,C1(C(N2CCC=C(CNC(c3c(CC)ocn3)=O)C2)=O)CC1C1CCCCC1 70203,N1(C(CCC=C)=O)CCC(NC(=O)COc2ccc(F)nc2)CC1C 70204,C1(C(=O)NCC2CCC(NC(C3CC(=C)C3)=O)CC2)CN(CP(C)(C)=O)C1 70205,N1(C(c2c(N)ccc(Cl)c2)=O)CCCN(C(C2(C(F)(F)F)CCCC2)=O)CC1CO 70206,c1(OC)cccc(CNC(=O)NCCc2cc(-c3cccs3)on2)n1 70207,CC(O)C(F)(F)C(=O)NC1CCN(CCCNC(c2ccccc2F)=O)C1 70208,C1(CC(=O)N(C(C)CNC(C2CCC(N(C)C)CC2)=O)CC)CCS(=O)(=O)C1 70209,c1(C(=O)NCCN(C(=O)CC2CC(F)C2)C)cn(C)cc1C(F)(F)F 70210,c1(C(N(C(C(=O)NCc2c(NC)ccnc2)=O)C)C)ccc(F)c(F)c1 70211,Cc1cc(C(=O)NC2CCCC(NC(=O)CCNS(C)(=O)=O)C2)cc(C)c1 70212,c1(CCC)nc(C)c(C(N2CCC(NC(C3CC3C)=O)C2C)=O)s1 70213,c1(C(=O)OCC2CC3(CCC3)C2)ccc([N+](=O)[O-])c(O)c1 70214,Cc1c(Br)ccc(O)c1C(=O)NCCOc1ccc(C#N)cc1 70215,C1(CC)CC(C(N2CCC(F)(CNC(c3cc(F)n(C)n3)=O)C2)=O)CC(=O)N1 70216,O=C(C(=O)C(F)(F)F)N1CCC(CCNC(C2CCCCC2O)=O)C1 70217,C1(C)(CNC(C2(OC)CC2)=O)CCC(NC(c2cc(CCO)on2)=O)C1 70218,C(=O)(CCS(C)=O)N1CC(O)(C(C)(C)CNC(=O)C(C)(C)c2ccccn2)C1 70219,C1(NC(CC(C)C2CC2)=O)CCCC12CCN(C(=O)CC1CC3(CC3)CO1)CC2 70220,C12CCN(CC1)C2=O.n1(CC2N(C(n3ncc(Br)n3)=O)CCC2)ccccc1=O 70221,N1(C(CCCNC(=O)OC)=O)CCN(C(=O)CC(C)(C)c2cccs2)C(CF)C1 70222,C1(C(=O)NCCN(C(=O)CCOC2COC2)C)(CC2CCC2)CCOC1 70223,C1(C(C)O)CCCCN1C.C(=O)(CN)NCCN(CCC)CCOCCO 70224,N1(C(C(C)=CC)=O)CC23CCCC2(C1)CN(C(c1cc[n+]([O-])cc1)=O)C3 70225,C1(NC(C2(F)C(C)C2)=O)CCC(C)N(C(=O)Cc2ccc(C(F)F)cc2)C1 70226,CC(C)C(C)C(CNC(C1(O)CCCC1)=O)NC(=O)CCc1ccc(CO)cc1 70227,c1(CCC(=O)NC2CCC(CNC(CC(=C)C)=O)CC2)cc(C)ccc1C(N)=O 70228,C1(CNC(C2CN(C(C)=O)C2)=O)CC(NC(c2n[nH]cc2Br)=O)C1(C)C 70229,c1(OC)ncnc(Cl)c1C(N1CCCCC(Cn2cc(C(O)C3CC3)nn2)C1)=O 70230,C(C1c2ccccc2CCN1C(c1ccc(C(N)=O)c(Cl)c1)=O)NC(C(C)C)=O 70231,c1(OC)cccnc1C(N1CCCC(N)C1)C(=O)NCCC#N.N1(CCSC)CCCC1 70232,c1(CC)ccncc1OC(C1COC(CNC(c2c[nH]c(=NC)o2)=O)C1)=O 70233,N1(C(C2(OC(=O)C(C)CC(=O)NC(C)=O)CC2)=O)CCC12CCSCC2 70234,C1(NC(C(C)(C)N2CCCCC2)=O)CN(S(=O)(=O)CCCCl)CC1(F)F 70235,c1(CC(=O)NCCCC(C(=O)N2C(C(=O)OC)C=CC2)O)csc2nc(C)cn12 70236,c1(CN(C(=O)CC2CCN(C(=O)CCn3cnnn3)CC2)C)ccccc1Cl 70237,C1(C(N(C)C)=O)CCCC1CNC(=O)CC1(O)CCC1.C12CCN1C2=O 70238,c1(C(=O)NC2CN(C(C#CC3(CC)CC3)=O)C(C)CC2)cc2n(n1)CC(F)C2 70239,CC1CC(c2nnnn2CSc2ccccc2)(NCC(C)(C)CO)CC(C)O1 70240,N1(C(c2c(C)n(C)cn2)=O)CC(C(=O)NCC(c2cnn[nH]2)C)CC1(C)C 70241,C(C#Cc1cccnc1)NC(C1CCCN1C(c1cccn2cncc12)=O)=O 70242,N1(C(C(=O)NCCN(C)C(C2CC(OC(C)(C)C)C2)=O)C)CCCC(O)C1 70243,c1(CC(=O)N(CC(CNC(CC2CC(OCC)C2)=O)C)C)cc(C)on1 70244,N=c1ccnc(CNC(C2(CNC(c3nnsc3N)=O)CC23CCC3)=O)[nH]1 70245,C(C1=CCN(C(=O)CC2CCCS(=O)(=O)C2)CC1)NC(CC1CCC(C)CC1)=O 70246,N1(CC)CCC(N(C(c2nc(CO)cs2)C(=O)NCC2CC2)CC)C1 70247,C1(C)(C(N2CCC(N(C(C3C(C(=O)OCC)C3)=O)CCO)C2)=O)CCC2CC2C1 70248,C1(C(=O)NC(CC)(C)C)CCN(C(C2CNC(=O)N2)=O)C(C)(C)C1 70249,N1(CC(=O)NC(C2CN(C(C3CCOC(=O)CC3)=O)CCO2)C)CCSC(C)(C)C1 70250,C1(CNC(Cc2c(C)nsc2)=O)CCCCN(C(=O)CCc2cncn2C)C1 70251,N(C1CCCn2nccc21)C(C1(C=C)CCN(C(c2n[nH]c(C)c2O)=O)C1)=O 70252,Cc1ccc(C(C)CC(=O)NC(C)(CNC(=O)Cn2ccnn2)CO)cc1 70253,c1(OC)ccc(-c2nc(COc3ccc(F)cn3)cs2)cc1F 70254,c1(OC)ccc(CO)cc1C(=O)NC(CNC(=O)CN1CCCCC1=O)C1CC1 70255,c1(C(N(C2CCN(C(=O)CCCC#N)CC2)CC)=O)cc2ccsc2s1 70256,CCC(CC(=O)N(C(C(=O)NC1CCCC1C#N)C(C)CC)C)C(F)F 70257,C1(C(N2CCC(C(=O)NC3(CC#C)CCCCC3)CC2)=O)CCCC(C#N)C1 70258,N1(C(c2c(CC)cco2)=O)CCCN(CCNC(=O)Cn2cncn2)CC1 70259,Cc1c(CNCC2C3CN(C(=O)CC4CCC(F)(F)C4)CC23)cccc1O 70260,C#CCCCC(C)C(=O)N1CCOC(C(=O)NC2CCCC2N(C)C)C1 70261,C(=O)(CCCCC(C)(C)C)N1CC(CN(C(CN2CC(C)C2)=O)C)OCC1 70262,C#CC1(NC(=O)C(C)(C2CCC2)NC(c2ccc(F)s2)=O)CCOC1 70263,N1(C(C2C(C(N)=O)C2)=O)CCCC(C2CCCN(C(c3ccc[n+]([O-])c3)=O)C2)C1 70264,C1(NC(CN(C)S(N)(=O)=O)=O)CCCC12CN(C(=O)Cn1cc[nH]c(=O)c1=O)C2 70265,c1(C(c2nnnn2C2CC2)NC(c2c(F)cccc2F)C)cc(F)c(Br)c(F)c1 70266,C(=O)(C(C)CC(=O)N1CC(NC(c2ccc(OC(F)F)c(Cl)c2)=O)C(F)C1)OC 70267,C1(CNC(C2CCC(C)O2)=O)CC2CCC1N(C(c1cc3n(c1)CCCC3)=O)C2 70268,c1(C(=O)NC2CC(C(C)NC(C(c3ccc(C)o3)C)=O)C2)ccc2[nH]ccc2n1 70269,N1(C(c2n(C)nc(C(F)(F)F)c2)=O)CCC2(CC1)OCCC2NC(=O)CC1CC1 70270,c1(CN(C)C)ccc(C(N2CCC2CNC(c2csc(S)n2)=O)=O)[nH]1 70271,C#CCC(C)C(=O)N1CCC(C(C)NC(c2ccc(C3(C)CCO3)cc2)=O)CC1 70272,C1(NC(CCOC(CCC)C)=O)CCN(C(c2cccc(OC)c2O)=O)CC1C 70273,N1(C(c2c(C)coc2C(C)C)=O)CCC(CO)(CNC(=O)C(O)C(F)(F)F)CC1 70274,C12CCC(C1)NC2=O.c1(C(=O)NCCNC(C2(Br)CC2)=O)ccco1 70275,c1(C(=O)OC)ccc(CC(N2CCN(C(=O)CCn3cnnn3)C3CC23)=O)c(Cl)c1 70276,C(C)(C)(C=CC(=O)NCCC1CC(C(N2CCC2)=O)C1)SC 70277,C(CCC(C)CCC)N(C(CC(C)(C)N(C(C(C=C)(C)O)=O)C)=O)CC 70278,c1(C(=O)NC(CNC(C(C)c2cc[nH]n2)=O)C(C)(C)C)cc2occc2s1 70279,C1(C(N2C(CNC(c3n(C)cc(C#N)c3)=O)CC(F)C2)=O)CNC(=O)C(C)(C)C1 70280,C(C(=O)N1CC(CC(C)(C)CNC(c2nccc(C)n2)=O)C1)(C(C)(C)C)SC 70281,c1(-c2nc(C(C)OC)nn2CCc2cncc(F)c2)cc2c(OC)cccc2[nH]1 70282,C1(NC(c2c(C)ocn2)=O)CN(C(=O)C(C)OCC(C)C)CCC1F 70283,C(CCCCC(=O)NCCN(C(C1CCC(F)CC1)=O)CCOCCO)SC 70284,Cc1nn(C)c(N)c1C(=O)NCC(C)NC(c1cccc(C(N)=O)c1C)=O 70285,CC(C)C(C(=O)N1CC(CCCCNC(C2CC3C=CC2O3)=O)C1)NC=O 70286,C#CC1(NC(=O)CN(C(=O)C(C)OCCC=C)C2CCC2)CCOC1 70287,CCCCC(CNC(c1ccc(F)s1)=O)NC(=O)C(C)(C)n1ccnn1 70288,N1(C(CCC(C)C)=O)CCC12CN(C(=O)CC1CCCC(C)(C)O1)C2 70289,Cc1c(C(N2CCCCC2CCN(C)C(c2csc(=N)[nH]2)=O)=O)nc2sccn12 70290,c1(COCCNC(C=C(C)CNC(C2C=CCS2)=O)=O)nc[nH]n1 70291,n1(C(CC)C)nc(C(=O)NCCC(C)(C)NC(C2CC3C=CC2O3)=O)cc1C 70292,CC(C)C(C)(O)C(=O)NCC(c1ccccc1)CNC(c1cc(Cl)ncc1O)=O 70293,C1(N(C(=O)C(C)N(CC)CC2CC2)CCC)CCN(C(=O)Cc2cn[nH]c2)CC1 70294,c1(C(N2CCC(NC(CCOCC)=O)C(C)C2)=O)ccc(S(=O)(=O)C(F)F)cc1 70295,N1(SC)CC(C(N2CCCC(N(C(=O)C(C)Sc3ccncc3)C)C2)=O)CC1=O 70296,C(C)(CCS(C)(=O)=O)(c1n(CCSC)nnn1)NCC1(C)COC1 70297,CC(C)CC(C)C(=O)NCc1ccsc1C(=O)N(C1COCC1(C)C)C 70298,C1(NC(c2cn(C)nc2C(F)F)=O)CC(NC(=O)CNC=O)C12CCC2 70299,Cc1cc(C)c(C(N2CCN(C(=O)CC3COCCN3C)C(CO)C2)=O)c(C)c1 70300,c1(C(C(=O)NCCCSC)N(CC(=O)NCCC)C)nc(Br)ccc1OC 70301,C(=O)(CC(P(C)(C)=O)P(C)(C)=O)N(CC(=O)N(CCCC)CCCC)CCCC(C)O 70302,c1(C(=O)NC2C(C)(C)CN(C(=O)Cc3cncs3)C2)ccc2[nH]nc(Cl)c2c1 70303,c1(C(N2CC(C(CC)CC)C2)=O)ccc(C(N)=O)o1.c12ccn(n1)CCNC2C 70304,C(CC)(CCC(=O)NC(CC)CC)NC(CN(CC=C)C1CC1)=O 70305,C12(NC(c3cc4n(n3)CC(F)C4)=O)CCCC1CN(C(c1cc(O)ncn1)=O)C2 70306,C=CCC(F)(F)C(=O)NCC(F)CNC(c1ccc([N+](=O)[O-])o1)=O 70307,c1(C(=O)NC2CCN(C(c3ccc(OC)s3)=O)CC2F)ccc2nc(O)oc2c1 70308,Nc1ccc(C(=O)NCC(CO)NC(C2CCCN2C=O)=O)c(Cl)c1 70309,c1(CNC(C(=O)NCC)=O)cccc(CNC(C2CCC(F)C2)=O)c1 70310,N1(C(C=Cc2cn(C)nc2)=O)CC2COCCC2(NC(=O)C(F)=C2CCCC2)C1 70311,C1(CCCNC(C2(OC)CC2)=O)CCN(C(=O)CN2CCCCC2C)CC1 70312,c12ccc(nc1)C1CN(C1)C2=O.CC(C(=O)NC1CC1)=CC(C)(C)C 70313,CCCC(O)C(=O)N1CCC(OCCNC(c2coc(C#N)c2)=O)C1 70314,c1(C(N(C(CC(=O)NCC(CC=C)(C)C)(C)C)C)=O)cc(F)cnc1O 70315,c1(NC(=O)CN2CCC(NC(CO)CO)C2=O)noc2cc(Br)ccc12 70316,C(C(C)N=c1nc(OC)cc(OC)[nH]1)N(C(CCCCC(=O)NC)=O)C 70317,CC(C)C(C(=O)N1CC(NC(c2c[nH]nc2C2CCCCC2)=O)C(C)C1)NC=O 70318,CC1CN(C(C2CC(C)(C)CO2)=O)CC1C(=O)NC1C=CCC1 70319,C1(NC(c2c(Cl)cn(CC)n2)=O)CN(C(=O)CC2(CO)CC2)C2(CCCCC2)C1 70320,C(CC(C(=O)N(C1CCOC1)CCF)NC(=O)CC1CCC(=O)C1C)OC 70321,C(CCCCC(=O)NCc1cc(C(N2CCC(CCO)C2)=O)cs1)OC 70322,C=C=C(C)CC(=O)NC(C1CCCN1C(=O)CCSc1nccn1C)C 70323,C(=O)(C1=NN(CC)C(=O)CC1)NC(CC)CNC(C1CN(C(N)=O)C1)=O 70324,N1(C(CCCOCCOCC)=O)CCN(C(=O)CN2CSCCSC2)C2CCC12 70325,C1(CC=C)(NC(C2CC2C=C)=O)CN(C(C2CC(C)(O)C2)=O)C1 70326,c1(OC)ccc(C(C)NC(=O)N(C(C)Cc2ccc(F)cc2)C)cc1C 70327,N#CC1CN(C(CCC2CC(F)(F)C2)C(=O)Nc2ccccc2)CC12CCC2 70328,C1(C(N2CC(C(O)C(=O)NC3CC(C(F)(F)F)C3)C2)=O)CCCC(O)CC1 70329,CC(C)(CCCO)C(=O)N(C1CN(C2CC2)C1)C(C1CS(=O)(=O)C1)=O 70330,c1(C(N(CCCN(C)C(c2nc(=O)cc(N)[nH]2)=O)C)=O)[nH]c2ccccc2c1Cl 70331,CCCC(C(=O)NC(C)CC1CN(C(c2coc(C#N)c2)=O)C1)S(N)(=O)=O 70332,c1(CC(=O)NC2C(NC(c3n(CC)ncc3)=O)CC2)cc(Br)ccc1C 70333,c1(OC)cc(C)cnc1C(=O)NC(CNC(=O)CC1(n2cccn2)CC1)C(C)C 70334,C(N=c1[nH]c2cc(Cl)cc(Cl)c2o1)C1CCN(C(c2cc(C)c(C)s2)=O)CC1 70335,Cn1cnc2ccc(NC(C3CC4(CC(NCc5cccc(Cl)n5)C4)C3)=O)cc12 70336,Cn1ncc2c1CN(C(C1(C)CCN(C(c3cc(I)c(O)c(I)c3)=O)C1)=O)C2 70337,CP(C)(=O)c1ccc(C(=O)NCC(O)CCNC(c2nc(=N)cc[nH]2)=O)cc1 70338,CC(C)(CNC(C1CC2CC1CC2O)=O)CC(=O)NCCC1(CO)CC1 70339,N1(C(C=CCNC(=O)CCC2OCCO2)=O)CC(O)CC12CCC2 70340,N1(C(CC2CN(C)CC2O)=O)CC(NC(c2cc(C#N)c[nH]2)=O)C(C)(C)C1 70341,C(=O)(CC(C(=O)N(C1CCCCC1NC(=O)Cn1nnnc1C)C)N(C)C)OC 70342,C1(C(=O)N)C2CCC(C2)C1C.C1(O)(C(C)C)CCN(C(C2CC(CF)C2)=O)C1 70343,C1(C(=O)NC2C(CNC(C3(CC#C)CC3)=O)CCC2)C2CC3CC(C2)CC1C3 70344,Cc1c[nH]c(C(=O)NCC2CCCN(C(=O)Cc3ncc(C(F)(F)F)[nH]3)C2)c1C 70345,N1(C(C(=O)NC2C(NC(CCCC)=O)COC2)CC)C(=O)CCC1=O 70346,N1(C(C(CNC(c2ccccc2C)=O)OC)=O)CC(C)CC(C)C1 70347,C=CCC(CNC(=O)C(C)(C)SC)NC(=O)C(C)=C1CCCC1 70348,C(C(C)C(=O)N(CC(=O)NC(C)(C)C)C)NC(C(C)SCCCC)=O 70349,c1(C(=O)NCC2C(C)CCN2c2nnco2)cc(F)cc(Br)c1F 70350,C1(C(N(CCN(C(c2ccsc2)=O)CC)CC)=O)CC2(C1)CC(F)(F)C2 70351,c1(SC)ccccc1F.C1C(C)(NC(C2CC2C)=O)CNC(=O)C2(CC2)C(=O)N1 70352,C(=O)(C(CNC(=O)CC1CC=CCC1)C(C)(C)C)N1C(COC)CC1 70353,C1(OC)CC(CNC(=O)COC2CCCC(C)C2)N(C(=O)CCCSC)C1 70354,N1(C(CC2CC(OC)C2)=O)CCC2CN(C(=O)C=CI)C2C1 70355,N1(C(c2c(CCC)n(C)nn2)=O)C2CCC1CN(C(=O)CC(CC)CCC)CC2 70356,N1(C(c2c(C)c[nH]n2)=O)CCC(C2CC2)C1C(=O)NC1CS(=O)(=O)C1 70357,Cc1cccc(C(C(C)C)OC(C2(C3CC=CCC3)CC2)=O)c1 70358,c1(OC)cc(C)c(C2(CN(C(CCC(F)F)C(=O)O)C=O)CC2)cc1OC 70359,N1(C(CNC(C2CCC2)=O)=O)CC2CCC(C(=O)O)C2C1 70360,C(=O)(C1=CCCN(C(C2(COC)CCCO2)=O)C1)NC(CCCC)(C)C 70361,CCC(CC(=O)N1CCN(C(=O)CCn2cc[nH]c(=O)c2=O)CC1)CC(F)(F)F 70362,S(=O)(=O)(CC(=O)N1CCCC1CNC(C1C2CC2C2CC12)=O)NC(C)(C)C 70363,N1(C(C(CC)NC(N)=O)=O)CC2CCCC(NC(c3cc(Br)cs3)=O)(C2)C1 70364,C1(C(N2CC=CC(NC(C(C)Sc3nncn3C)=O)C2)=O)CC(=O)NC1(C)C 70365,C(=O)(C(C)S(N)(=O)=O)N.C1(C(C)(C)C)(N(C(C)CCC)C(C)=O)CCCCC1 70366,c1(C(=O)NC(CNC(C=CSC)=O)C2CCC2)cccnc1C 70367,c1(C(N(C(C)C(=O)NCCc2ncc[nH]2)CCC)=O)ccnn1CCOC 70368,C1(C(=O)NC2CON(CC)C2=O)CC(C)(C)CCN1C(C1CCC(=O)O1)=O 70369,C1(C(=O)OC)CN(C(C(=O)NCc2ccccc2)C2CCC2SC)C2(CCC2)C1 70370,c1(OCc2onc(-c3ccc(C(=O)OCC)cc3)n2)cc(Cl)cc2ccncc12 70371,c1(C(N2CC(NC(C3(C)CC4C=CC3C4)=O)C(F)CC2)=O)ccc2c[nH]nc2c1 70372,N1(C(CC(C)CF)=O)CC2(C)CC1(C(=O)N(C)CC1(C)CCCC1)C2 70373,C=CCC(C)C(=O)NCCCC1(NC(=O)C2=CCOC2)CC1 70374,CC(C)(CCC(=O)N1CC(C(=O)NCC(c2cnc[nH]2)O)C(F)C1)[N+](=O)[O-] 70375,c1(NC(C(CC=C)CNC(C2CC3CCC(C2)O3)=O)=O)cnc(C)c(C)c1C 70376,c1(CC(C)(C)C)ccccc1CC(N1CC(C)(NC(=O)CC2CC(F)(F)C2)C1)=O 70377,C=CC(C)C(=O)CCCONC(=O)CN1CCC(C)C1 70378,c1(C(=O)NC2(C)CCN(C(=O)CCc3cnoc3)C2)nccc2ccsc12 70379,C1(CNC(C(CC)O)=O)CCCCN(C(c2ccc(OC)cc2Cl)=O)C1 70380,C12(C(=O)NCc3nc(C)on3)CCCC1CCN2C(C1C=CC=CC=C1)=O 70381,CN1CCC(C)(C(=O)NCC2CCCCN2C(=O)C=Cc2cccc(F)c2)CC1 70382,c1(N(CC(=O)NCCC(O)CNC(=O)NC2CC23CC3)C)ncnc2[nH]cnc12 70383,CCC(O)C(C)(C)C(=O)N1CCOC(CC(=O)NC2(C)CCCC2)C1 70384,c1(NC2C(C)C2)ccc2c(c1)oc1ccccc21 70385,c1(C(=O)NCC2CCN(C(CC=C)=O)C23CCC3)ccc2nc(N(C)C)sc2c1 70386,C1(CNC(CC2(C)CCC2)=O)CCN(C(c2ccc(N)cn2)=O)C12CCC2 70387,CC1CN(C(c2cccc(CO)c2)=O)CC1NC(C1(C(C)(C)C)CCC1)=O 70388,C1(C)(C(=O)NC(c2cnc(C)s2)C)C=CCN1C(c1cnn(C)c1Cl)=O 70389,C(=O)(C(F)(F)C1=CCOCC1)NC12C(CN(C(c3ccnc4ccnn34)=O)C1)C2 70390,c1(C(N(CC(C)O)CCNC(C(C)OCC)=O)=O)cnc(CC(C)(C)C)o1 70391,C(c1ccc(F)cc1)=CC(=O)NCCC1CC(C(=O)Nc2ccc(F)c(F)c2)C1 70392,C(C(CO)(CO)NC(=O)C=Cc1cn[nH]c1)N(C(=O)CCC1(C)CCC(=O)N1)C 70393,CC(C#N)C(=O)NC(Cn1cccn1)C(=O)N(C)Cc1ccsc1 70394,C(=O)(CC(C)CC(C)C)N1CC(c2ccc(CC)cc2)N(C(=O)C(Cl)=CCl)CC1 70395,n1(CC(N2CCCC(C(C)C(=O)O)C2)=O)cc2ncccc2n1 70396,c1(NC(=O)NC2(CC(=O)OC)CCOC2)ccc(-c2nccs2)cc1 70397,C1(C2(C)CCN(C(CSc3cccc(OC)c3)=O)C2)CCC(F)(F)CC1 70398,C1(CNC(C(C)ONC(c2ncoc2C2CCCC2)=O)=O)Cc2ccccc2O1 70399,CC1C(NC(C2CCCO2)=O)CCN1C(=O)Cn1ccnn1 70400,C1(CC(N2C(CNC(c3c[nH]c(=N)o3)=O)CC2)=O)CC(C2CC2)C1 70401,c1(C(=O)OCCCCCS(C)(=O)=O)ccc2nc(Cl)sc2c1 70402,c1(C(c2n(CCOC)c(N3CC(F)(F)CCC3C)nn2)O)nc2c(s1)CCCC2 70403,N1(C2C(NC(C3CC3c3cccs3)=O)CCC2)CCN(C(C)(C)C2(CC)CC2)CC1 70404,CC(C(=O)NCC1(CNC(=O)CCn2cncn2)CC12CCC2)S(C)(=O)=O 70405,c1(C(=O)NCC2(F)CC(NC(C(C)CC3CCCO3)=O)C2)cnc2c[nH]nc2c1 70406,Cn1nc(C(N2CC(NC(=O)C(C)(C)C)C3CC23)=O)c2c1CCOC2 70407,c1(C(=O)NCC2N(C(C(CC)NC(C)=O)=O)CCCCC2)cccc2sncc12 70408,O=C(CC1=CCCCC1)NC1CCC(NC(C2(C(F)F)CC2)=O)C1 70409,C1(C(C)C)CN(C(C2NC(=O)OC2C)=O)CCN1C(c1cccc[n+]1[O-])=O 70410,C(=O)(CC(C)(C(F)(F)F)N(C)C)N1CCC(N(C(=O)C=CCCC)CCC)C1 70411,C1(C)(CC)C=C(C(=O)N(C)CC2(O)CN(C(=O)C(c3ccc(C)cc3)O)C2)C1 70412,C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NCC1C(NC(C2CCC(C)CC2)=O)CC1 70413,N1(C(c2cnn(C)n2)=O)CCC2OCCN(C(=O)C(O)C(F)F)C2C1 70414,C=C(Cl)C(C)(C)C(=O)NCC12CC1CN(C(=O)C(c1ccccc1OC)=O)C2 70415,Fc1cncc(Cl)c1CNCc1nc(C(F)(F)F)n[nH]1 70416,c1(CNC(C(=O)NC(C)Cn2cncn2)=O)ccc(CN2CCNC(=O)C2)cc1 70417,CC(CC(=O)NCC(CC(=O)N1CC(N2CC(F)C2)C1)C1CCC1)C(F)F 70418,C(=O)(C(C(C)C)C(C)C)NC1C(NC(c2c(Cl)c(C)n(C)n2)=O)CCCC1 70419,Cc1nscc1C(=O)NCC(C1CCCCC1)O.C12(CCC1)CC(=O)N2 70420,N1(C(c2c(F)ccc(C)n2)=O)CC(C(=O)NCC2OCCC2(C)C)C2(CCC2)C1 70421,C1(CNC)CC(C(F)(F)F)CN1C(C12CC(C)C1C2)=O.C1(CC=O)CC(C)(C)CO1 70422,C1(CNC(C2(N(C)C)CCCC2)=O)CCC(NC(=O)Cc2cnccn2)CC1 70423,c1(CC)c(C(=O)NCC2(OC)CCN(C(C3CCC(=O)N3CC)=O)C2)cnn1C 70424,CC1(C)C2CCC(C(=O)NCC3(O)CCN(C(=O)CNC=O)C3)C1C2 70425,C1(CNC(C2C(CC)C2)=O)COC(C)(C)CN1C(c1cc(N)ccc1C)=O 70426,c1(CC)cnc(C(=O)N(C)CCN2CCN(C(C3CCC(C4CC4)C3)=O)CC2)cn1 70427,c1(OC)nc(=NC(C)CCNC(C2(C)CC2(F)F)=O)[nH]c2ccccc12 70428,N1(C(C(C)OCC#C)=O)CC(NC(c2cnc(NC(C)C)nc2)=O)C(C)C1 70429,c1(C(=O)NCCOC2CCN(C(CC3C(C)C3)=O)C2)cc(C#N)ccc1F 70430,C1(CC(N2C(CO)CC2C)=O)(OC)CN(C(=O)C=Cc2ccoc2)C1 70431,c1(N2CC(C(C)NC(=O)Cn3nnnc3C3CC3)OCC2)ncnc2[nH]cnc12 70432,C1(c2n(CC=C)nnn2)(N(C2(CCO)CCOC2)C2CC2)CC2(C1)CC(C)(C#N)C2 70433,C1(CC)C(NC(=O)CCSC(C)CC(C)C)CCN1C(C1CN(C)C1)=O.C(C)C 70434,CC1(CC(=O)NC2CC2CNC(c2ncccc2C2CC2)=O)CCOCC1 70435,c1(C(N(C2CN(C(CCC=C)=O)C2)C)=O)cccc(OC)n1 70436,C#Cc1ccc(NC(=O)C#CC(C)(C)CNC(c2cncn(C)c2=O)=O)c(C)c1 70437,C(=O)(CCCC(=O)NC1CCOC(C(=O)NCCCc2cc[nH]n2)C1)N(C)C 70438,CN1CCC(C(=O)NC(C(=O)NCC2(C(C)(C)O)CC2)C2CCC2)C1=O 70439,c1(C(C(=O)NC2COC2)N(C(CC(=O)OC)C)C)ccccc1N1CCCC1 70440,c1(C(=O)NC(COC)C(C)C)ccccc1C(=O)NC1CCCC1N 70441,N1(C(C=C(CCC)C)=O)CCC(CCNC(c2cccnc2C)=O)CC1C 70442,C1(C)(CNC(C(CC)CCOC)=O)CN(C(C23CCC2CC3)=O)C(C)(C)C1 70443,N1(C(c2c(C)csc2)=O)CCC(n2cc(-c3cscn3)nn2)C(O)C1 70444,N1(C(c2cc(CC)n(C)n2)=O)CC(NC(=O)Cc2nccn2C)C(C)(C)C1 70445,N1(C(C)=O)CC2(CCN2C(=O)CCCOC(c2ccc(OC)cc2)=O)C1 70446,c1(C(N2CCCC(NC(C(C)OCC#C)=O)C2)=O)cc(S(C)(=O)=O)cc(F)c1Cl 70447,CC1(C)CC(NC(=O)C(=O)NCC(F)F)CN(C(=O)C(C)(C)S(C)(=O)=O)C1 70448,c1(C(=O)NCCOCCN(C(=O)C(C2CC2)C2CC2)C)ccc(Cl)s1 70449,C(=O)(CC(C)CNC(C1COCC(C)O1)=O)NCCc1nc(C)[nH]n1 70450,C1(CNC(c2c(CC)n[nH]c2)=O)CCCN(C(c2cn(CC(N)=O)nn2)=O)C1 70451,C1(C2CN(C(=O)CNc3ccccn3)C2)CN(C(c2ccc(CO)s2)=O)CCO1 70452,O=C1CCc2nc(NC3CCCC(NC(c4cc5ncccc5o4)=O)C3)ccc21 70453,N(C1CCc2cccnc21)C(C1CC2(CC2)CN1Cc1ccc2cc[nH]c2n1)=O 70454,c1(C(N2CC3CC3(C(=O)NC3CONC3=O)C2)=O)ccn2cncc2c1 70455,S(=O)(=O)(c1ccc(N(C)Cc2ccc(Cl)cc2)cc1Cl)NC(C)CCCO 70456,C1(C(=O)NC2(CCNC(c3c(C)nsc3)=O)CCC2)CC2CCC(C1)C2 70457,c1(C(=O)NC2(CN(C(=O)C3=CCCC3)C)CC2)cc(Br)c2c(c1)CCO2 70458,c1(CCC(=O)NCC(C2CCOC2)F)nc(C2CC2)no1.C12(CC1)C(=O)N2 70459,C1(CCN(C(=O)Cc2ccc(CO)cc2)C)CCCCN1C(=O)C=CCF 70460,C(=O)(C(O)C(F)(F)F)NC(C(=O)N(CCOCC(C)N(C)C)C)C(C)(C)C 70461,CCCC(C)CC(=O)N(C(c1ccccc1)CNC(c1cc(C)cnc1C)=O)C 70462,C1(O)(CCCCN(N)C(C=C(CCN(C)C)Cl)=O)CCN(C(=O)C=Cc2cscn2)C1 70463,N#Cc1ccccc1C(N1CC2CCC2(CCNC(=O)C=Cc2ccsc2)C1)=O 70464,c1(CN(C(=O)CC2CCCN2C(=O)CCC2CCC(=O)C2)C)cn(C)nn1 70465,C1(C2CC2)(C(=O)NC(CC(=O)OC)C2CC2)CN(C(C2C=CCC2)=O)C1 70466,C(=O)(CC(C)(O)C(F)(F)F)N(C1CCCCC1)CCNC(C=C1CCC(C)CC1)=O 70467,c1(C(=O)NCC2OCCN(C(c3cc(CO)[nH]n3)=O)C2)ccc(Cl)c([N+](=O)[O-])c1 70468,C1(C(C)(C)NC(=O)NC(c2nc[nH]n2)C)CCN(C(C2CC23CCOC3)=O)CC1 70469,c1(C(N2C(CO)CC(NC(C=C(C)C)=O)C2)=O)cc(O)c2ccccc2c1 70470,C1(C(=O)NCC(CC(C)C)NC(=O)C(C)(O)C(C)C)CCCCNC1=O 70471,c1(C(N2CC(NC(CCC#C)=O)C(CO)CC2)=O)cnc2c(c1)NC(=O)CS2 70472,Cc1cccc2cc(C(=O)N(CC(C)(C)NC(c3occc3Cl)=O)C)cnc12 70473,C=CC1(C(=O)N(CCCN(C(=O)C(C)Cc2ccncc2)C)C)CCC1 70474,c1(C(N(C2CN(C(c3nnsc3N)=O)C2)C)=O)ccc2cccnc2c1F 70475,O=C(C1=CCCCO1)NCCCOCCNC(C1COC2(CO)CC1C2)=O 70476,C1(CC#C)(C(=O)NC2CCOCC2C)CCN(C(c2csnn2)=O)C1 70477,CC1(C)CC(C(=O)NCC2CN(C(=O)C3CC3)CC23CC3)CCO1 70478,O(N(C)C(=O)CNC(C1CCC(CNC(C2CCCC(C)O2)=O)CC1)=O)CC 70479,C#CCCC(=O)NCCOCCOCCOCCN(CC)CC 70480,C1(NC(C=C(NC(C)=O)C)=O)CC2CCC(C1)N2C(=O)Cc1ccccc1O 70481,C(=O)(C(CO)C(C)(C)C)N1C(C(N2CCN(CCOC)CC2)=O)C2CCC1C2 70482,c1(C(N(C(C)C)CCNC(=O)CCCCc2cnn[nH]2)=O)ccnc2[nH]ncc12 70483,C1(NC(c2n(C)ncc2Cl)=O)CCC2(CCN(C(C3(C#N)CCCOC3)=O)C2)C1 70484,c1(CC(=O)NCC(CNC(CCSCC(N)=O)=O)O)ccc2nonc2c1 70485,N1(C(C(C)C)=O)C2CCC1CC(CNC(c1cc(Cl)ccc1OC(F)(F)F)=O)C2 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70504,N1(C(C(C)OCC2CCCO2)=O)CCC(NC(=O)CCCN(C)C)C(O)C1 70505,N1(C(=O)NCc2c(C)nc(Cl)cc2)CCC(F)(F)C2(CCOC2)C1 70506,Cn1ncc(C#N)c1C(=O)NCCCOCCCNC(C12COCC1C2)=O 70507,C1(C(=O)Nc2ncc(C#N)s2)C2CCC(C2)C1NC(c1ccc(F)cc1O)=O 70508,N1(C(C)(C)C)Cc2ccc(NC(=O)N(C(=O)C(C)Cc3ccco3)C3CC3)cc2C1 70509,C1(NC(C(=O)NC(c2noc(CC3CCCCC3)n2)C)=O)CCSCC1 70510,Cc1ccc(CCC(N2CCN(C(c3nnc(O)nc3O)=O)CC2)=O)cc1Cl 70511,CN1CC(=O)N(CC(=O)NC2CC(NC(=O)Cc3cn(C)cn3)C2)C1=O 70512,C1(C(N2C(CNC(c3cc(CC)ncn3)=O)CC2)=O)CCOCC12CCC2 70513,Cc1[nH]c2ncccc2c1C(N1CCN(C(=O)CC2CCCO2)C(CF)C1)=O 70514,N1(C(C(CCC)CNC(=O)C(C)(C)C2CC2)=O)CC2CN(C)CC2C1 70515,c1(CC(N2CCN(C(C3CC(OC)C3)=O)C(C)C2)=O)nc(C)nc2sc(C)c(C)c12 70516,c1(C(C(=O)NC2C(CNC(c3nccc(C(C)(C)C)c3)=O)C2)O)cc(Cl)cc(Cl)c1 70517,N1(C(C(=O)Nc2ccccc2)=O)CC2CCNCC12.c12ccc(cc1)OCC2 70518,c1(OC)cc2nn[nH]c2cc1C(=O)NCC(C1CCOC1)NC(=O)CCF 70519,C(=O)(CC1=CCCCC1)N1CCC(OCC)C1.N1(CC=O)CCC(CC)CC1C(F)(F)F 70520,Cc1cc(C(=O)NC2CCN(C(=O)C(C)(C)c3cnco3)C2)n(C2CC2)n1 70521,c1(CNS(CC)(=O)=O)cccc(NC2CCCC2C(=O)NC(C2CC2C)=O)c1 70522,C(=O)(C(C(C)(C)C)N(C)C)N(CC(C)NC(C1(Cl)CCC1)=O)C 70523,c1(C(=O)NC2C(C)CN(C(=O)C3=NOCC3)C2)cc(Cl)cc(Cl)c1Br 70524,C1(NC(C2C(CNC(CCC(=C)Cl)=O)OCC2)=O)C(=O)OC2CCCC12 70525,C=Cc1cnn(C)c1C(=O)NCCCCCN1CCN(C(=O)CCCCC)CC1 70526,c1(OC)cccc(CN(CC(C)C#N)C(N)=O)c1Br 70527,C1(NC(c2ccc(CCC)cc2)=O)CCN(C(c2cnc(N)c(O)c2)=O)CC1F 70528,C(=O)(C(CCSC)NC(c1c[nH][nH]c1=N)=O)NC(CC=C)C1CC1 70529,C1(N(C)C(C2CCN(c3ncccn3)C2)=O)CC1C1CC1 70530,C1(NC(C2(CC)CN(C(C(CCCC)C)=O)C2)=O)CCCCC12CCC2 70531,C1(NC(c2cc(OC)ns2)=O)CCC2CCN(C(=O)COc3ccccc3)C1C2 70532,N1(C(C(C)(C)OC(=O)NCC)=O)CCN(C(=O)C(C)c2ccco2)C(CCC)C1 70533,c1(C2CCN(CC(CC#C)C3CC3)C2)nc(C)ccc1Br 70534,c1(C(N2CCC(NC(c3c(OC)n[nH]c3)=O)CC2C)=O)cc(C)cc2ccoc12 70535,c1(C(=O)NCCC(CNC(C2(CCC)CCC2)=O)O)cc(Cl)c2[nH]c(O)nc2c1 70536,c1(C(=O)OCC)cc(C)n(C(C)(C)C)c1.C1(CNC(C2CC2(C)C(F)F)=O)(N)CCC1 70537,C1(C(=O)NC(C)CCNC(c2ccnc(Cl)c2N)=O)CC(C(C)(C)C)=NO1 70538,C(C(C)(C)C(=O)NCC(C)=CC(N1CCC(OCCCC2CC2)CC1)=O)NC(C)=O 70539,C(C(=O)N1CCOC(CC(N2CC(O)CC2C(N)=O)=O)C1)(C(C)C)SCC 70540,c1(CC)cccc(OCC(=O)NCCC(C)(C)NC(C2CCC(C)O2)=O)c1 70541,c1(CC)ccc(C(N2CCC(C)=C(Br)C2)C(=O)NCC(F)F)cc1C 70542,C(=O)(C(C(C)C)N(C)C)NC1C(NC(C2(CSC)CCC2)=O)CC1 70543,c1(C(=O)NCC2N(C(C(=O)NCC)=O)CC3(CC3)C2)cn2c(n1)CC(OC)CC2 70544,C(=O)(C(C)(C)CCCNC(=O)CCc1nccs1)NCCOCCN(C)C 70545,C(=O)(N=c1[nH]nc(CCOC)s1)N1CCC(CC)C1OCC(C)C 70546,C1(C(CNC(C(C)(C)n2cnnn2)=O)(C)O)CCN(C(C2CCCCC2)=O)CC1 70547,C(CC(CNC(=O)COC)OC(C)=O)NC(C(C)OCCC#C)=O 70548,CN1CC(NC(c2cc(CNC(=O)CN3CCCC3=O)ccn2)=O)CC12CCC2 70549,CCCCC(O)C(C)C(=O)N(C)CCN(C)C(c1nc(C)ncc1Cl)=O 70550,C#Cc1cc(C(=O)NC23CCC2CN(C(c2c(C)nn(C)c2F)=O)C3)ccc1Cl 70551,N1(C(C2(COC)CC=CC2)=O)CCC(F)(CNC(C2(COC)C=CCC2)=O)CC1 70552,c1(-c2cccc(CC(C)NCC(C3CCCO3)O)c2)cccc(C(=O)O)c1 70553,O=C(CCC[N+](=O)[O-])N1CCOCC(CNC(C2(c3ccccn3)CC2)=O)C1 70554,c1(CC(=O)NC(CC=C)C(N2CC(C(N)=O)C3(CC3)C2)=O)ccc(C#N)cc1 70555,CC1CCC(CCC(N2CC(O)(CN(C(=O)CC34CC(C3)C4)C)C2)=O)O1 70556,N1(C(c2c(C(C)C)con2)=O)CCCC(C)(C(=O)NC2COCC2CO)C1 70557,CCCCC(C(=O)N1CC(CCOC)(NC(c2nn(C)c(Cl)c2Cl)=O)C1)C(C)C 70558,c1(C(N(C)CC2CCN(C(C(CCC)O)=O)C2)=O)cnn2c1N(C)CC2 70559,c1(C(=O)NCCN(CCC)C(c2c[nH]nc2CC)=O)c(C)csc1Cl 70560,C1(CNC(c2cnco2)=O)CC2(CCC2)CN1C(c1ncoc1C1CCC1)=O 70561,C(=O)(CC(C)(C)C(=O)N1CC2CC(NC(c3cc(Br)cn3C)=O)CC2C1)OC 70562,N1(C(C=Cc2ccn(C)c2)=O)CC(NC(C2CC3(C2)CC3F)=O)CC(F)C1 70563,CC(C)CCC(F)C(=O)NC1CCC(CCC(N2CCN(C(C)C)C(C)C2)=O)C1 70564,c1(CN=C(NCC(CC)(C)OC)NC2CC2)cc2n(n1)CCCO2 70565,C12CC(C1(C)C)C(=O)NC2.c1(C2CC(c3cn(C(C)(C)C)nn3)C2)ccc(Cl)nc1 70566,CCC(CC)C(F)C(=O)NCC1(CNC(=O)C(CC)OC)CCCCC1 70567,C(CC1CC1)(C(=O)NCC=CCNC(c1cc(Br)co1)=O)OC 70568,C=C(C)C(CC(=O)NC(C)(CNC(c1cc(O)ccc1O)=O)C1CC1)OCC 70569,C1(C(=O)NCc2c(C3CN(C(c4c(CC)con4)=O)C3)ocn2)CCCN(C)C1 70570,C1(CC(=O)NCC(C(C)C)(C)NC(=O)CN2CCC(=O)CC2)CCCCC1(F)F 70571,C1(C(=O)NCC2C(NC(C3(CC#C)CCOC3)=O)CCCC2)C2CCC(C2)C1C 70572,c1(CCN(C(=O)NC2CC3OC(=O)CC23)C2CC2)nc([N+](=O)[O-])n[nH]1 70573,N1CCCN(C(=O)CC2CC(Cl)C2)CC1.CS(C)(=O)=O 70574,c1(C(=O)NCC2N(c3cn(C)nc3)CCC2)cc(Br)cnc1S 70575,CC(C)CC(O)C(=O)NCC=C1CCN(C(C2(C3CCCCO3)CC2)=O)CC1 70576,c1(OCC)ccc(NC(c2nnnn2C2COC2)C2CC2)c(F)c1 70577,c1(CN(C)C(C2CN(c3ccncc3)C2)=O)ccnn1C 70578,CCC(C)C(O)C(=O)NC1(CO)CN(C(=O)C(C)(O)C2CC2)C1 70579,CN1C(=O)OCC1C(N1CC=CCC1C(=O)NCC(N1CC=CC1)=O)=O 70580,N(C(=NCCC(C)C)NCC1CCCC(=O)N1)CCc1c(CC)cccc1 70581,Cc1cnn(C(C)C(=O)NC(c2cccnc2)C(=O)N(C2CCCC2)CC(C)C)c1 70582,N1(C(CC=CC=C)=O)CCN(C(c2ccc(CCCCC)o2)=O)CC1c1cn[nH]c1 70583,C(CO)(CCCCNCCc1ccc(C2CC2)cc1)NC(C=CC(C)(C)SC)=O 70584,c1(CNc2nccc(Cn3c(C)ncc3)c2)ncc2ccccc2n1 70585,Cc1cc(C(N2CCCN(C(=O)CC3CCN(C)C3)CC2C)=O)c(O)c(C)n1 70586,N12CCCC1C2=O.c1(NC(=O)NCC(C)(C)OCCO)cccc(-n2nccn2)c1 70587,C(C(C(=O)NCC(=O)OC)NC(=O)CCCOC(C)C)SC 70588,c1(OC)cc(C)cnc1C(=O)NCC1(OC)CN(C(c2coc(C(F)F)n2)=O)C1 70589,c1(CCC(=O)NCCC2(NC(CN(C)CCO)=O)CCC2)ccc(=N)[nH]c1 70590,Cc1cc(C)n(CC(N2CCC2CNC(c2cc(Cl)c(F)cc2N)=O)=O)c(=O)n1 70591,Cc1ncc(C(=O)NCCC2(NC(=O)C(C)OCCN(C)C)CC2)s1 70592,c1(N(C2CCC(F)C2)C(=O)NCCOCOC)cnc[nH]c1=N 70593,CCC(C(=O)NC1CC(C)N(C(=O)Cc2cc(C)n(C)n2)C1)C(C)(C)CC 70594,c1(C(C)(C)OC)ccnc(NCC2CCCC2NC(=O)CCCF)n1 70595,c1(N2CC(C(C)C)N(C)CC2)nc2cccc(F)c2c(=NCc2n[nH]c(=N)o2)[nH]1 70596,C1(CNC(C(C#C)(C)C)=O)CN(C(=O)Cc2cc(C)on2)CCCO1 70597,C1(C)(C(=O)NCC(CNC(C2CCCC2(C)C)=O)OC)CCCN(C)C1 70598,N=c1[nH]c2ccc(C(=O)NCC3CCN3C(C3CCn4cncc4C3)=O)cc2o1 70599,c1(-c2cn(C3CN(C(C4(COCC)CC4)=O)C3)nn2)ccc(C)cc1 70600,c1(CC)cccc(F)c1C(=O)NCCOC1CN(C(=O)CC2CCC(=O)O2)C1 70601,c1(CN(CC(=O)N(C(C)=O)Cc2cn(C)nn2)C)cc2ccccc2c(C)c1Cl 70602,O=C(C(F)(F)CO)N1CCC(OC2CN(C(=O)Cn3ccc(C4CC4)n3)C2)CC1 70603,CCCC(C)(C)C(=O)NCC(C)CNC(C1(c2ccc(OCC)cc2)CCC1)=O 70604,c1(NC(CC)=O)cncc(C(=O)NC2CC(CCNC(=O)C(C)n3ccnc3)C2)c1 70605,C(CC(=O)N(CC(C)CO)C)(C(C)CC)NC(C(CCC)N(C)C)=O 70606,C1(C(N2CCC(C(C)(C)C)C2)=O)COCCN1c1nnc(C(F)(F)F)s1 70607,C(C(=O)NCC1NC(=O)CC1(C)C)(C(C)(C)C)NC(C1CCC(C)CC1)=O 70608,c1(C(=O)NC2CN(C(CC(C(C)C)C)=O)CC2(C)C)c2c(nn1C)CCCC2 70609,c1(C(=O)NC2(CNc3cc(CC)nc(C)n3)COC2)ccc2oc(S)nc2c1 70610,c1(C(N2CCC(C)(CNC(=O)CC3CCC(=O)N3)C2)=O)cc2c(Cl)nccc2s1 70611,N1(C(C(C)OCC(C)C)=O)CC(C2CCCN(C(c3cc(CO)[nH]n3)=O)C2)C1 70612,c1(C(=O)NCc2cc(C(=O)NC(COC)(C)CO)n(C)n2)ncc(F)cc1N 70613,CC1CCCC1(C)NC(=O)C=CC(C)(C)NC(=O)Cc1ccsc1 70614,C1(CNC(c2cn(CC)nc2C)=O)CC(C)CN(C(c2cnsc2C2CC2)=O)C1 70615,c1(CN(CCCC)S(C)(=O)=O)ccccc1-c1ccc(NC(c2nc[nH]n2)=O)s1 70616,CC1CN(C(c2cc(Cl)ccn2)=O)CC(C)C1NC(c1cc(N)nc(Cl)c1)=O 70617,C(=O)(C#CC1CCOC1)NC(c1ccccc1F)CNC(=O)CCC1CNC(=O)N1 70618,Cc1ccc(-c2cn[nH]c2)s1.C1(=O)C(CC2CC2)N(c2cnn(C)c2)C(=O)C(=O)N1 70619,C1(NC(C2C(NC(c3c(C)ccnc3O)=O)COCC2)=O)CCCCCC1(C)C 70620,C(=O)(C(O)CC(C)(C)C)NC(C(=O)Nc1c(OC)cc(C)cc1)CC(F)F 70621,c1(C(=O)NC(CCNC(CC2(OC)CCCCC2)=O)C)ncn2cc(Cl)ccc12 70622,c1(OC)ccc(Br)c(CC(=O)NOC)c1.c1snc(Cl)c1Cl 70623,N(C)(C(=NCc1ccc(CO)s1)NC(C)C1CC1)CCCC(=O)OC(C)C 70624,C(CCCCCNC(c1sccc1CO)=O)N(C(C(C)=C(C)C)=O)C 70625,c1(C(N2CCN(C(C=CCOC)=O)C(C)CC2)=O)ccc2c(c1)C(C)CO2 70626,c1(C(=O)NCCN(C(C)C)C(C2CC2(Cl)Cl)=O)ccccc1S(=O)(=O)C(F)F 70627,CC1SCCN(C(=O)CCC2CCCCN2C(C2(C)CCCCCC2)=O)C1C 70628,N1(C(CC(=C)Br)=O)CCC2(CCN(C(c3cccc(C(C)C)n3)=O)C2)C1 70629,c1(C(=O)NC2(O)CCN(C(COCCN(C)C)=O)C2)cc(N(C)C)nc(Cl)c1 70630,n1(CC(=O)NCC(CC(C)C)NC(CSCCCC)=O)cc(F)ccc1=O 70631,C1(C2CCC2)(NC(C(C2CCN(C(c3csc(F)c3)=O)C2)C)=O)CC1 70632,c1(C(N(CC(CC)NC(=O)CN2CCNC(=O)C2)CC)=O)cnn2cccc2c1 70633,c12cccc(c1)C(C)NC2=O.c1(SCCCOCC(F)(F)F)ccccn1 70634,CCCCC(CNC(C1CCC(OCC)CC1)=O)OCN=N.C1(=O)CCCCN1 70635,C1(C(=O)OCC(=O)N)C=CC(NCCN(CCC)CC)C1.OC 70636,C1(C#CC(=O)NCc2cc(C(=O)NC(C)(C)CC(C)C)no2)(CC)COC1 70637,C(=O)(C1=Cc2cc(F)ccc2OC1)N(C(C)CN(C)C(C1CCCCCC1)=O)C 70638,C(=O)(CCC(=O)Nc1ccc(C(C)Nc2cn(-c3ccccn3)nn2)cc1)OC 70639,C1(NC(C2(C)N(C(C(C(C)C)F)=O)CCC2)=O)CCC2CCCC1O2 70640,N1(C(CC(=C)C)=O)CCC(Nc2ncc(Br)cn2)C(c2ccccc2)C1 70641,C1(CN(C(=O)CS(=O)(=O)N(C)C)CC)CCN(C(C2OCCOC2C)=O)CC1 70642,N1(c2nc(NN3C4CCC3CC(F)C4)cc(C)n2)Cc2ccc(F)cc2CC1C 70643,N1(C(C(=O)NC(C)C)=O)C2CCC1C(NC(C1(c3ccc(Cl)cc3)CCC1)=O)C2 70644,Cc1ccccc1C=CC(=O)NCC1CCC(NC(=O)C(c2cscn2)N(C)C)C1 70645,c1(OC)cc(CNc2ccccc2CN=c2nn[nH]n2C)cc(I)c1O 70646,CCCC(C)(CC)C(=O)N(CC(=O)NC1CCCC1C#N)C(C)C 70647,N1(C(c2ccc(COC)[nH]2)=O)CC(NC(c2cscc2OC)=O)CC1CO 70648,c1(CN(c2cc(C)c(O)nn2)CC)ccc([N+](=O)[O-])cc1C#N.C12CCN(CC1)C2 70649,C1(C(=O)NCC2(O)CC(CNC(=O)CC3C=CCCC3)C2)Cc2nccn2C1 70650,C1(NC(C2(NC(COC3(C#C)COC3)=O)CCCC2)=O)CCC(C2CC2)C1 70651,C1(CNC(C(COC)(C)OC)=O)CCC12CN(C(=O)Cn1ccc(=O)cc1C)C2 70652,N1(C(c2nc(C)oc2C)=O)CCc2sccc2C1CNC(C12CCC1C2)=O 70653,C(C(C)(O)CC(=O)NCCCCCCNC(C1CC1c1ccc(C)o1)=O)OC 70654,CC1(C)CN(C(c2sccc2CNC(C2C(C)(C)C2(F)F)=O)=O)CCC1CO 70655,c1(CC)ccc([N+](=O)[O-])cc1C(=O)NCC=CCNC(c1cnc(C)s1)=O 70656,C(CC(C)(C)C)(C(=O)NC1CCCCC1N=[N+]=[N-])NC(CC1C(C)C(=O)CC1)=O 70657,C1(C(=O)NCCN2CCC(CC(=O)C(C3CC(=C4CC4)C3)=O)C2)CC2(CCC2)C1 70658,Cc1cc(C(N2C(C(=O)N(CC(C)C(C)C)C)CC2C)=O)cn1C 70659,Cc1cc(Cl)ncc1CC(N1CCN(C(=O)CCC2(C)N=N2)C(C)C1)=O 70660,c1(OC)cc(C(N2CC(O)CC2CNC(C2CCCCN2N=O)=O)=O)cc(C)n1 70661,c1(C(=O)OCC)ccc(C2CCCN(C(=O)CSCCC(C)C)C2)cc1 70662,C1(N(C)C)CCC(NC(=O)CC(C)(C2CCC2)C2CCC2)CC1 70663,CC(C)C(C(=O)NCC1(NC(c2ccc(-n3cnnn3)cc2Cl)=O)CC1)C(C)C 70664,C1(C(N(C(C)Cc2ccccc2Cl)C)=O)CN(c2ccnc(CO)n2)CCC1O 70665,Cc1cc(F)c(C(=O)N(C)CC2CCN(C(c3cnc(O)c(Cl)c3)=O)C2)c(Br)c1 70666,CC(CC(=O)NCC(CC1CCCC1)C(=O)NC1CNC(=O)C12CC2)CC(C)(C)C 70667,c1(COC)cccc(CC(=O)NC2CCC(CNC(C3CC=CCC3C)=O)C2)c1 70668,C1(CCNC(CN(CC(F)(F)F)C)=O)C(C)CCCN1C(=O)C(C)NC(N)=O 70669,C1(CC(=O)NC2CC(NC(C(C3CC(F)(F)C3)OC)=O)C2)COc2ccccc2C1 70670,C(=O)(C(C)CC(F)(F)F)NCC(C(C)C)NC(c1c(C)c(Br)ccn1)=O 70671,C1(C(N2CCC(=CCNC(C3C(C=C)C3)=O)CC2)=O)CCC2(CCC2)CO1 70672,c1(C(N2C(CCOC)CN(C(=O)CC3CCC3)CC2)=O)coc(S(C)(=O)=O)c1 70673,c1(C(N2CCC3C(NC(C(C)(C)CC4CC4)=O)C3C2)=O)cc2cccc(Cl)c2o1 70674,CCC(CC)=CC(=O)NC1CN(C(=O)C=CCF)C1 70675,C(=O)(C1COc2ccccc21)NC1CCC(N(C(=O)Cc2cccc(Cl)c2)C)C1 70676,N1(C(CC2N(S(C)(=O)=O)CC2)=O)CCCC1CNC(c1sccc1C(=O)OC)=O 70677,c1(C(N2CCC(C(C)NC(C(C)OCC#C)=O)CC2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 70678,CC(C)CC(=O)N1CCC(C(=O)NCCCC2C=CCC2)C1 70679,c1(C(=O)NC(C)C(N2CCC(C)(C#N)C2)=O)cccc2[nH]ccc12 70680,N1(CC)CCN(C(=NCCc2ccccn2)NCC2COC2)CC1(C)C 70681,CC1(C(N2CCC(OCC3CC3)C2)=O)CCCN(C(c2nc(Cl)cs2)=O)C1 70682,N1(C(C2C(c3ccn(C)n3)C2)=O)CC(C(C)C)OC(CNC(=O)C(F)(F)C(F)F)C1 70683,C1(NC(Cc2c(C)ocn2)=O)C=CCN(C(=O)C(c2cccc(F)c2)(C)O)C1 70684,C12(C(=O)NC3(COCC)CC3)CCOCC1CN(C(=O)CS(C)(=O)=O)C2 70685,C1(NC(c2c(CCC)occ2)=O)CCC(C)N(C(c2cnn(C)c2Br)=O)C1 70686,N1(C(=O)C(O)CCN(C)C)CCCC(F)(C(=O)NCCOC2CCOC2)C1 70687,C#CCC(CC(F)F)C(=O)N1CC(CC(=O)NC2(CCF)CCOCC2)CC1C 70688,c1(SC)cc(C)c(C(N2CC(NC(c3cc(CCO)on3)=O)C(C)C2)=O)o1 70689,C1(C(N2C(C)(CC(=O)NC(C#C)(C)C3CCC3)CC2)=O)CCCC(=O)C1 70690,CS(=O)(=O)c1ccc(C(N)=O)cc1.c12cccc3c1CN(C3)Cc1ccc-2cc1 70691,N1(C(c2c(C)scc2)=O)CCCCCC1C(=O)NC(c1nn[nH]n1)C1CC1 70692,C#CC1(C(N2CCC(O)C2)=O)CCN(C(c2cncc(C#C)c2)=O)C1 70693,N1(C(C(C)OC)=O)CCOCC1CN(C(=O)Cc1ccn(C(C)C)n1)C 70694,c1(NCC(C(=O)NCC)(C)C)ncc(S(=O)(=O)N2CCC(C3CCC3)C2)cc1Cl 70695,C1(C(=O)NC(C2CCC(C)CC2)C)CC12CCN(C(=O)CN1CCOCC1)C2 70696,c1(N(CCN(CCN(C(COC)=O)C)C)C)nnc(-c2cccs2)o1 70697,c1(C(N2CC3C(CNc4ccc(C(=O)OC)c(Cl)c4)(C3)C2)=O)cc2ccoc2cn1 70698,CC1(CNC(C2CC(NC(=O)Cn3cccc3)CCO2)=O)NC(=O)NC1=O 70699,c1(C(=O)NCC23N(C(CCCC)=O)CCC2CCC3)ccc2c(c1)CCCO2 70700,c1(Cc2ccc(C=C)cc2)cc(=O)oc2cc(OC3CCN(CC)CC3)ccc12 70701,N1(C(CN(C2(C3CC3)CC2C(F)(F)F)S(C)(=O)=O)=O)CCOC(C(F)(F)F)C1 70702,c1(CC(=O)NC2CN(C(C3(CC#C)CCCCO3)=O)CC2F)ccc(C)c(F)c1 70703,c1(OC)ccc(Cl)c(C(N2CCC2CNC(C2CCn3nnnc3C2)=O)=O)c1N 70704,c1(C(=O)NCC(CO)NC(C2(F)CCOC2)=O)nc2cccnc2s1 70705,Cc1cc(OCC(N2CC3CCCC3(NC(=O)CNC=O)C2)=O)cc(C)c1Cl 70706,c1(CN2CCC(O)(C(=O)NC3CCC(=O)N3)C2)c[nH]c2ncc(Br)nc12 70707,CCC(C)C(C(=O)N1CCCN(Cc2ccc(C(C)C)cc2)CC1)OC 70708,c1(C(C(=O)N(C(C)CNC(=O)C(=O)N(C)C)C)C)ccc2c(c1)OCCO2 70709,CCC(C)(C)CC(c1nnnn1CCOC)NC(C)C(C(=O)NCC1CC1)SC 70710,c1(C(=O)NC(C2CCCC2)CNC(C2CC2C(N)=O)=O)ccoc1Br 70711,c1(OC)cc(CNC2CCN(C(c3ccccc3C(C)C)=O)CC2C)c(Br)cc1O 70712,Cc1nn(C)c(N2CCC(C(C)(C)C)(CN)C2)c1C#N 70713,N1(S(CCOC)(=O)=O)CCC(O)CC1C(=O)ON1CCCCC1 70714,Cc1c(C=CC(N2CCC(C(C)NC(C3CC4CC3CO4)=O)CC2)=O)cnn1C 70715,Cn1cc(C(=O)NCCCC(c2ccccc2)NC(C2(F)CC=CC2)=O)nn1 70716,N1(C(C2(CC(C)C)CCCC2)=O)CCN(C(=O)Cc2cncnc2)CC1CO 70717,c1(C(=O)NC2CC(N(C(Cn3c(C)ccc3C)=O)C)C2)ccc(P(C)(C)=O)nc1 70718,c1(C(=O)NC(CCNC(C(C)CS(C)=O)=O)(C)C)scc2c1OCCO2 70719,CC(CNC(C1(CN(C)C)CC1)=O)C(F)C(=O)Nc1cc(O)cc(F)c1 70720,c1(COC)ccc(C(N2CC(CC(F)C(=O)NCC3CC3C3CC3)C2)=O)o1 70721,N(C(=NCc1ccn(C)c1)NCc1cccc(OC(F)F)n1)CC(C1CC1)OC 70722,N1(C(C(C)SCC)=O)CCC2(CC1)CCN(C(c1cnncc1O)=O)C2 70723,c1(-c2nc(SC)sc2)nc(C2CCOC2)nn1C(C)C(F)(F)F 70724,N1(C(CNC(=O)OC)=O)CCCC(C)(C(=O)NC(c2ccncc2)C)C1 70725,c1(CN(C(C(C)N(C(C)=O)C)=O)C)ccc(CNC(=O)CC(C)(C)C2CC2)cc1 70726,Cc1nc2ccccc2n1CC(N1CC(C)(NC(c2ccnnc2O)=O)C1)=O 70727,CCC(C)(CC)C(=O)N1CC(C2(NC(=O)CCC3CCC(C)O3)CC2)C1 70728,C1(CCNC(Cc2n(C)ccn2)=O)CN(C(C2CCCC(=O)C2)=O)CCO1 70729,CCCCC(CNC(=O)C(C)(C)N1CCOCC1)NC(c1cnccc1N)=O 70730,N1(C(C(N2CCC(OC)CC2)=O)=O)CCc2cc(F)ccc2C1 70731,CCCCC(C)N=c1cc(NCCCCCOCC2CCC2)nc(C)[nH]1 70732,C1(CNC(c2n(C)ccn2)=O)C2CCCC1N(C(C1CC3(C1)CC3(F)F)=O)C2 70733,C1(CC)CN(C(c2cnn(C)c2Br)=O)CCC1NC(C1(C#N)CCSCC1)=O 70734,CC(C)CC(C)CNC(c1csc(-c2ccccn2)n1)=O 70735,N1(C(C(=O)NCC#CCNC(C2(c3ccc(C)s3)CC2)=O)C)CCCCC1=O 70736,C1(N)CC2C=CC1CC2.C1(CC)C(=O)N1CC.C(=O)(NOCC)C1(C)CC1 70737,CS(=O)(=O)C(C(=O)NCCCCCOCCNC(C1(C(F)(F)F)CCC1)=O)N(C)C 70738,c1(C(=O)NCC(C)(CO)NC(C(C2CC2)OC)=O)cccc(-n2cncn2)c1 70739,c1(CN(C(C(OC)OC)=O)CCCNC(C2(C)COC2)=O)ccccc1 70740,C(=O)(CCCC(C)(F)F)NC1(COC)CCN(C(=O)C(C)C2CCCC2)C1 70741,c1(CN2C3CN(C(=O)Nc4c(OC)nccc4I)CC32)ccc(C#N)cc1Cl 70742,C1(C(N2CCC(C#CC)C2)=O)CCC2CCC1N2C(c1coc(C)c1)=O 70743,C(=O)(C1=CCC2CCC1N2C(c1coc(CO)c1)=O)NCC(C)N(C)C1CC1 70744,C(=O)(C#CC1CCCO1)N1CCC(NC(C(C2CC(F)(F)C2)OC)=O)C1 70745,N1(C(CC(C)N(C)C(C2CC(=O)N(C)C2)=O)=O)CCc2cc(F)ccc21 70746,C#CCC(C(=O)NC1COCC1F)NC(c1ccnc(C)c1)=O 70747,c1(C(=O)NCC2(C(C)NC(C3COCC(C)(C)O3)=O)CC2)cc2c(s1)CCOC2 70748,C#CC(C)(C)C(=O)N1CCC(C(=O)N(CC)Cc2nncs2)O1 70749,c1(N(C)C)cc(C(=O)NC2CCC2C2CC2)nn1-c1ccc(Cl)cc1 70750,c1(CN(c2cccc(N)c2)C(N2CCC(C)(C(=O)NC(C)C)C2)=O)ccc(Cl)cc1 70751,C1(COC(C2CC(n3ccnn3)C2)=O)CCC=CO1 70752,c1(C(=O)NC2CCN(C(c3cc(OC)c(F)cc3)=O)C2)cn(C)cc(Br)c1=O 70753,C1(N(C(=O)CC2CCOC2)CCC)CCN(C(=O)Cc2cc[nH]n2)CC1 70754,C1(C(=O)NCC2CC(C)N(C(c3cnc[nH]c3=N)=O)C2)CCCC(C)(C)O1 70755,C1(C(N(CCN(C(=O)CC(C)n2cc(Br)cn2)C(C)C)C)=O)CNC(=O)C1 70756,Cc1sc(N)c(C(N2CC(CCNC(=O)COCC(C)(C)C)OC(C)C2)=O)c1C 70757,N1(C(C(C(C)C)OC)=O)CCC(O)(C2(NC(=O)CCC3CC3(Cl)Cl)CC2)CC1 70758,c1(SC(C(c2cccc(N3CCCS3(=O)=O)c2)=O)CN2CCC(O)C2)ccc(F)cc1 70759,CCC(C)C(C(=O)N1CCC(C(N2CCC(OC3CCC3)C2)=O)C1)OC 70760,C1(OC)CN(C(c2nncs2)=O)C(C)(CNC(=O)CC=Cc2ccccc2)C1 70761,c1(C(=O)NC2CCc3n(C)cnc3C2)ccc2c(=N)[nH]cnc2c1 70762,C1(C(=O)NC(C)(C)CN2CCN(C(c3c[nH]c(=N)o3)=O)CC2)CCCCC1(C)C 70763,C#Cc1ccnc(C(=O)NC(c2nocc2C(=O)NCC(N2CCCC2)=O)C)c1 70764,C1(NC(c2c(OC)nc(C)cc2)=O)CC2CC(C1)N(C(=O)Cc1scnc1C)C2 70765,C1(CC=C)CCCC(NC(=O)CNC(C2(CCNC(N)=O)CC2)=O)CC1 70766,c1(NC(COC(c2cccc(OC)c2)=O)=O)cc2cc(C)[nH]c2cc1Cl 70767,C(CC(C)CCNC(=O)C=CC1CC1)NC(C1N(C(C(C)C)=O)CCC1)=O 70768,C1(C(=O)NC(CCNC(c2c(CC)n(CC(C)C)nc2)=O)C)CCC(O)CN1C 70769,C1(C(=O)OCC)C2C=CC(CC2)C1C(N1CCC=CC1COC)=O 70770,C(C(C(F)(F)F)NC(=O)CNCc1ccnn1C)OC 70771,N1(C(C(COC)C)=O)CCOC2(CCCN(C(c3ccc(CN(C)C)o3)=O)C2)C1 70772,C(=O)(C(C)(C)CC(=O)NC1CCOCC1NC(C1CC12CC2)=O)OC 70773,C1(CNC(C2CC2Cl)=O)CCC(C(N2CCCC2)=O)C1 70774,Cc1cc(C)c(C(N2CCCC(NC(=O)C=Cc3cnn(C)c3)CC2)=O)c(S)n1 70775,C=CCCC(C(=O)NCC1CCOC1=O)N(C(=O)COCCCN=[N+]=[N-])C 70776,C1(NC(c2c(OC)nccc2)=O)CC(F)CN(C(C2CC(=C(F)F)C2)=O)C1 70777,C=CCC(C(=O)N1CCC1(C)CC(=O)NC1CC(C)C1O)NC(C)=O 70778,c1(-c2c(SC)scc2)ccc2c(CN3CC(O)CC(O)C3)nsc2c1 70779,C1(NC(C2(NC(C(CCSC)O)=O)CCSC2)=O)CCn2nccc2C1 70780,c1(CC)ncc(C(N2CCC(F)(C(N3CCCC3(C)CO)=O)C2)=O)cn1 70781,C1(NC(=O)CCCCO)C(CNC(c2ccc(OCF)cc2)=O)CCC12CCC2 70782,CCCC(C)(C)C(=O)N1CC(OC)CC(NC(c2cnc(OC)nc2)=O)C1 70783,C12(NC(C3CC(=C)C3)=O)CCCC1N(C(c1noc3c1CCCC3)=O)CCC2 70784,C12(C(=O)NC(C(=O)NCCC3CC4CCC3O4)C3CCCC3)CCCC1C2(F)F 70785,c1(C(N(CCN(C(C(CC)F)=O)C)C)=O)cnc(OC2CCOCC2)cn1 70786,c1(NC2CC3C(NC(C(CC(=O)OC)C)=O)C3C2)coc2cc(C)c(C)cc12 70787,C(=O)(CC(C)CC)NC1(C)CN(C(CSCC)=O)C1 70788,Cc1cc(-c2nn[nH]n2)ncc1NC(C1CCCN1C(=O)OC(C)(C)C)C 70789,C1(CNc2nc(COC)nc(N3CC4CC3C4)c2)CCC2(CCOCC2)C1O 70790,CC1CCN(C(C2CC23CC(O)C3)=O)CCN1C(=O)CCC1CC1(F)F 70791,N1(C(CCC2(C)CC2)=O)CCC2(CO)CN(C(C3C4CC5C(C4=O)C35)=O)CC2C1 70792,N1(C(c2ccn(CC)n2)=O)CCC(C(=O)NC(C)C(=O)OC)C(C)(C)C1 70793,CC1C(CNC(=O)COCC2CCOC2)CCCN1C(c1ccc(Cl)c(Cl)c1)=O 70794,N1(C(c2ccc(SC)o2)=O)CCCC(CC(=O)N(C)CCc2nn[nH]n2)C1 70795,C(=O)(CC1=CCCCC1)N1C(C)CC(CNC(c2c(CC)nccn2)=O)C1 70796,c1(C(=O)NC(CNC(c2ccc(N(CC)CC)cc2)=O)(C)C)nn(C)c(Cl)c1Cl 70797,CCCC(CC)CC(=O)N(C)CC1COCCN1C(=O)CN(C)C1CC1 70798,N1(C(CCc2ccc(C)cc2C)=O)CC2(NC(C3CC3C(F)F)=O)CCC1CC2 70799,N1(C(=O)C=C2CCC2)CCCC2C1CCCCN2C(=O)CCF 70800,C1(C2(O)CN(C(C3CC3C#N)=O)C2)(CNC(Cn2nc(C)c(Br)c2C)=O)CC1 70801,c1(C(=O)NCC(CC)NC(=O)Cc2ccn(C)n2)cnc2c(c1)NC(=O)CS2 70802,C1(NC(=O)CN2CCCCC2)C=CCN(C(C2CC(c3ccc(Cl)s3)C2)=O)C1 70803,C1(NC(c2cc(C)n(C)c2C)=O)CCC2(CC1)CC(NC(=O)C(F)(F)C(C)O)C2 70804,C(=O)(C#CC(C)(C)CNC(=O)CCc1cccnc1)Nc1c(C)nccn1 70805,c1(C(=O)NCC(CO)NC(CC(=O)NCC)=O)csc2c(Br)cccc12 70806,C1(C(C)C)CN(C(=O)C(C)(C)F)CCN1C(c1cnn(C)c1)=O 70807,N1(C(CC2(OC)CC2)=O)CC2(C1)CN(C(=O)CC1CCCN1C)CC(C)(C)O2 70808,Cc1scc(CN2CC(C(=O)O)CC2C(=O)O)c1C.C12=CC=C(N=C1)C2 70809,Cc1ncc(C(=O)NC(C)(C)CCNC(C2CC(C3CC3)=NO2)=O)cc1N 70810,C1(CC(N2CCC(NC(c3cc(C)c(C)s3)=O)(CF)C2)=O)OC(C)(C)OC1=O 70811,CCC(C(=O)OC)C(=O)N(CCC(N1CC(C)=CC(C)C1)=O)CCOC 70812,N1(C(c2nccs2)=O)CCOCC(C(N2CCCC(N3CCCCC3)C2)=O)C1 70813,C(=O)(CCCCCN(C(=O)CCN(C)C)C)N1C(C(C)C)CCC1 70814,C(C(F)(C(=O)NCC1CC(O)C1(C)C)C(C)C)NC(C1(OCC)CCC1)=O 70815,c1(OC)ccncc1C(=O)NC12CC(NC(=O)C(C)(C)CC3CCOCC3)(C1)C2 70816,CC(C)CCC(O)C(=O)NCCCCCC(=O)NCC(C)C1CCC1 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70853,CC1CCc2[nH]c(C(=O)NCCCN(C(=O)CC(C)(C)O)C3CCCC3)cc2C1 70854,N1(C(c2n(C)nc(O)c2)=O)C2CCC1CC(CNC(C1(C#N)CC13CCC3)=O)C2 70855,C1(C)(CNC(c2c(OC)nsc2)=O)CCN(C(=O)Cn2ccnn2)C1 70856,C1(C#N)(C(=O)NC(C(=O)NC2CN(CCC)C2)c2ccoc2)CC2CC2C1 70857,N1(C(C(C(C)C)SC)=O)CCc2cc(CNC(=O)CCN3CCC3)ccc2C1 70858,c1(C(=O)NC2C(NC(c3ccccn3)=O)CCCC2)ccc(O)nc1Cl 70859,N1(C(c2ccc(C)cc2)=O)CC2CCN(C(=O)CC(C)C(F)F)CC2C1 70860,C(C1C(C(=O)NCC2CN(C(=O)Cn3cnnc3)CCO2)C1(C)C)=C(C)C 70861,c1(C(=O)NC2(CNC(=O)CCc3ncc[nH]3)CCC2)cc(Cl)cc2ccncc12 70862,c1(C(N(C)CCOCCNC(=O)CC2C=CS(=O)(=O)C2)=O)ccc2cncn2c1 70863,C1(NC(c2ncc(Br)cc2O)=O)CCN(C(c2ccc[nH]2)=O)C12CC2 70864,c1(C(N2CC(CC(=O)N(CCCCO)C3CC3)OCC2)=O)cc(Br)cc(F)c1F 70865,C(C(C)(C)CC(=O)N1CC(CC(=O)NC(c2[nH]c(C)nc2C)C)C2(CC2)C1)OC 70866,c1(C(CCC(=O)NC(CNC(c2cncc(C)n2)=O)CO)=O)c(F)cccc1F 70867,N1(C(C2(CC=C)CCN(C(c3ccccc3C)=O)C2)=O)CCOCCC1C1CC1 70868,S(=O)(=O)(c1ccc(N(C)CCF)c(F)c1)NCC1OCC(C)C1 70869,C(=O)(C#CC1CCCOC1)NC1CCCCN(C(C=C(CCC)C)=O)C1 70870,C1(CC(=O)N(CC#CC)C)CCCCN1C(c1cn(C)nn1)=O 70871,c1(CNC(C(CC)C)=O)ncccc1CNC(c1cc(Br)nn1C)=O 70872,C1(O)(C(C)NC(C(C)OCC2CC2)=O)CCN(C(C2(C)CCCC2C)=O)CC1 70873,C12(C(=O)NCCN(C(C3(CF)CCCO3)=O)CC3CC3)CCC(CO)(CC1)CC2 70874,CC(C)(C)C(C(=O)N1CC(C)(CCO)C1)NC(=O)CCc1cn[nH]c1 70875,c1(C(=O)NC2(CO)CN(C(C3(F)CCCOC3)=O)C2)ccc2nccn2n1 70876,c1(C(=O)NCCCN(C(C)C)C(C2CCC3CC23)=O)ccc2c(c1)CCOC2 70877,CC(CCCNC(c1cccnn1)=O)NC(C1CCCC1c1nc[nH]n1)=O 70878,n1(CC)cccc1C(N1CC(OCCNC(C2CCC2C)=O)C1)=O 70879,C(=O)(C1=CC2CCCCCCC12)N1C2(CCN(C(C#CC(=O)O)=O)C2)CCC1 70880,N1(CCC)CCC(C(=O)N(CC(C)O)CCNC(=O)CCC2CCC2)CC1 70881,N1(C(C2C(CNC(C(C)NC(N)=O)=O)OCC2)=O)CCOCC(C(C)C)C1 70882,c1(C(N2C3CN(C(Cn4c(C)ncc4)=O)CC2CC3)=O)ccc2c(n1)CCC(C)C2 70883,N1(C(CCc2n(C)ccn2)=O)CCCCN(C(c2cccc(CC=CCO)c2)=O)C1 70884,N1(C(C2CC(=O)NC2)=O)CC(CNC(c2cc3ncccc3o2)=O)C2(CCC2)C1 70885,Cc1nnc2n1CCC(C(N1CCN(C(=O)C=C3CCCCCC3(F)F)CC1)=O)C2 70886,c1(N2CC(CC(C)NC(c3ccc(CO)nc3)=O)C2)ncc(O)cn1 70887,C1(OCC(=O)NCC2CCC2)CCN(C(C2COCOC2)=O)C1 70888,N1(C(CCN(C(C)=O)C)=O)CC2(CC(NC(=O)C(C)(C)C(C)O)CO2)C1 70889,C(=O)(C(C)Cc1cnco1)N(CCNC(OC(F)(F)F)=O)CC 70890,C12(N(c3ccc(C)cc3)CC(C)C)CCC(NC(=O)N(C)C)C1CC2 70891,C(=O)(C(O)C(F)(F)F)N(C(CCO)C(=O)NCC12CCC(CC1)C2)C 70892,CCCCC(CN(C)C(C1CC(NC(=O)CC2(COC)CC2)C(O)C1)=O)CC 70893,N1(Cc2c(OC)cccc2C)CCC2(CCN(C(=O)Cn3cc(Cl)cn3)C2)C1 70894,CCCC(CCC)CC(=O)N(CCCNC(C1(C#N)CCCO1)=O)CCO 70895,c1(C(N(CC(C(=O)CC(O)Cc2cccs2)CC)CC)=O)cccc(F)c1C.OC 70896,CN1N=C(C(=O)NC2COCCC2NC(C2COC(C)(C)CO2)=O)CCC1=O 70897,N1(C(c2[nH]nc(OC)c2Cl)=O)CC2(CCC2NC(c2ccc(CO)cc2)=O)C1 70898,C1(CNC(c2ncc(OC)c(C)n2)=O)CCOCC12CCC2 70899,c1(C(N2CC3C(C(NCc4c(C)ccc(Cl)c4)CCl)(C3)C2)=O)cc2cccnn2n1.C(=O)C 70900,N1(C(CC2CC(SC)C2)=O)CC2OCCN(C(=O)CCC(=O)N(C)C)C2C1 70901,C1(C(N2CC(C#N)C(NC(c3csc(Br)n3)=O)C2)=O)CCc2ccccc2C1 70902,C1(O)(CNC(c2cc(CCC)nn2C)=O)CCN(C(C2(Br)CC2)=O)CC1 70903,c1(CN2CCC(N(C(C(C)n3cncn3)=O)C)CC2)cccc2c1CCCC2 70904,C(=O)(C(C)(CC)CC)NCOC1(COC)CCN(C(=O)CC(C)OC2CCCC2)C1 70905,CC1CCCN(C(C2(C(N3CC(N(C)C)C3)=O)CCCC2)=O)C1.C1CCC(C)N1 70906,CCC(C)(C(=O)N1CCC(O)C(N(C(=O)Cc2ccc(C)nc2)C)C1)C(N)=O 70907,Cc1cc(C(=O)NC2C3CCC2N(C(C2CC(=C4CCC4)C2)=O)C3)ncc1CO 70908,c1(CC(N2CCC(F)(C(=O)NCC(C)(C)N(C)C)C2)=O)cc(Cl)cc(Cl)c1 70909,c1(C(C)NC(C)(C)C)nccn1C.CC1CCNC(=O)O1 70910,CCC(O)C(F)(F)C(=O)NCCCCc1c(CNC(=O)CNC(C)=O)nco1 70911,CCCCCS(=O)(=O)CC(=O)N1CCCC(NC(=O)Cn2cnnn2)C1C 70912,Cn1c(C(=O)Nc2cccc3c2NCCO3)cc2cc(Cl)ccc12 70913,N(C1CCCn2ncnc21)C(C(CNC(c1ccc(CC)[nH]1)=O)OC)=O 70914,Cc1ccc(Br)c(NC(=O)C2CC2)c1.C1C(=O)N1 70915,N1(C(C(C)Cn2cccn2)=O)CCN(C(c2ccc(Cl)cc2I)=O)CC12CC2 70916,c1(SCCNC2(c3n(C(CC)C)nnn3)CCC2)ccnc2c(Br)cccc12.C(C)(=O)O 70917,c1(C(=O)NCCNC(CN(CC)CC)=O)cc(OC)ccc1OC.C12CC1CN2 70918,c1(C(=O)NCC2(C)N(C(c3cc(OC)nn3C)=O)CCC2)cc(O)nc(O)c1 70919,C1(CNC(=O)NCCCCc2[nH]c(=N)sc2)CCCC12NC(=O)NC2=O 70920,C(C)(C)(C(C)CC(=O)N1CCC(CSC)CC1)NC(C(C=C)OC)=O 70921,C=CCCCCCN=c1nc2scnc2c(NC(C)Cc2cnccn2)[nH]1 70922,N1(Cc2cncc(C)c2)CCC(O)CC1C(=O)Nc1cccnc1CO 70923,C1(C(N2C(CNC(=O)C=CC(C)C)CC3CC23)=O)(COC)CC=CCC1 70924,c1(C(=O)NC2CN(C(c3c(C)nsc3C)=O)CC2C(F)F)cccn2ccnc12 70925,N1(C(Cc2c(C)nsc2)=O)CCC2CN(C(c3cnn(CCF)c3)=O)CC12 70926,C12CN(CC1O)C(=O)C1(CC1)SCC(=O)N2.N1(Cc2cccs2)CC2C=CC1C2 70927,Cc1cc(C(N2CCSCC2C(=O)N=c2cc[nH][nH]2)=O)ccc1F 70928,c1(C(N(C2C(C)CCN(C(c3c[nH]ccc3=O)=O)C2)C)=O)ccc(C#N)c(Cl)c1 70929,C1(C2CCN(C(=O)C3=CS(=O)CCC3)C2)(NC(Cc2nc(CC)sc2)=O)CC1 70930,N1(C(COCCC=C)=O)CC(O)(C(F)C(=O)NCc2cc(C(C)C)n[nH]2)C1 70931,CCCCCC(CC)C(=O)N1CC(C)CC1C(N1CCC1C1CCCCC1)=O 70932,c1(C(=O)NC)c[nH]c(C(N2CCC(OC(C(C)NC(CC)(C)C)=O)C2)=O)c1C 70933,C(=O)(C1CSc2ccccc21)N(C(C)C)CCN(C(=O)COC(F)F)C 70934,C1(C(C)C)CCCC1C(=O)NCCC1CCN(C(=O)CNc2ncccn2)C1 70935,C#CC1(C(=O)NC2CCS(=O)CC2)CCN(C(=O)C(F)C2CCC2)C1 70936,N1(c2n(CC=C)c(C(C3CC(F)(F)C3)F)nn2)CCC2(CCOCC2)C1 70937,Cc1ccc(C(=O)NC2CCCC2NC(c2scnc2C2CC2)=O)o1 70938,C1(NC(CCc2n(C)ccn2)=O)CC12CCN(C(=O)CC1CC(F)(F)C1)C2 70939,c1(C(N2CC(C3OCCN(C(c4c(C)nns4)=O)C3)C2)=O)cc(Cl)cc(Cl)n1 70940,N1(C(c2c(C)ncnc2)=O)CC(C2(NC(C3CC4(C3)CC(C)C4)=O)CC2)C1 70941,c1(-c2c(C)ccc(CO)c2)cnc2[nH]cc(C(=O)Nc3cccc(C(C)C)c3)c2c1 70942,CCC(C)C(O)C(=O)N1CCCC1CN(C(=O)C=CC=Cc1ccccc1)C 70943,C1(N(C(COC(CC)CC)=O)C)CCN(C(=O)C=CC2CCOCC2)CC1 70944,Cc1ccc(C(=O)NCC2C3CN(C(c4c(C)csc4Cl)=O)CC23)c(O)n1 70945,C12(C(N(C3CN(C(C4(O)CCC4)=O)CC34CC4)C)=O)CCC(C)(CC1)CO2 70946,c1(C(=O)NC(C(CO)NC(c2cc(C)no2)=O)C)cnc2n1CCC(C)C2 70947,C1(CNC(c2c(C)cc(C(F)(F)F)s2)=O)CCS(=O)(=O)C1(C)C 70948,Cc1cc2cc(C(=O)NC3CC4(C3)CC4C(=O)NC3CCOC3)oc2cc1C 70949,C(=O)(C#CC1CCCCO1)NC1CC(C)(C)CN(C(c2ccccn2)=O)C1 70950,c1(C(=O)NC2C(C(=O)NC(C=C)(C)CC)CCC2)ccc2cncn2c1 70951,C1(CC)(NC(=O)CSS(C)(=O)=O)CCCN(C(c2cncc(OC)c2)=O)C1 70952,C(C1CCCN1C(=O)CC1CC12CC2)=CC(=O)N(CCCN1CCC1)C 70953,N1(CNC(C2(CCCC)CC2)=O)CCCN(C(=O)CC2CC2CC)CC1 70954,c1(COC)nc(C)ncc1C(=O)N(C)CCNC(c1ccc(C2CC2)cc1)=O 70955,CC(C)(C(=O)NCC1CCN(C(C2(c3cccnc3)CCC2)=O)C1)C1CCCC1 70956,c1(NCC2(C)CCN(C(C3CC(CCC)OCC3)=O)C2)cc(C)nc(Cl)n1 70957,c1(CC2(NC3CCCCC(F)(F)C3)CCCCC2)cccc2c[nH]nc12 70958,c1(C(C)C)nnsc1C(C)NC(=O)NCCCCOC(C)(C)C 70959,N1(C(c2occ(S(C)(=O)=O)c2)=O)CC2CCCN(C(c3n[nH]c(=N)s3)=O)C2C1 70960,c1(CCC)cccc(C(=O)NCCC2CCCCN2C(=O)C(C)SC)c1 70961,CCCC(C)(O)C(=O)N1CCC(C)(CC(=O)NCCC2(O)CCCC2)C1 70962,N1(C(CNC(=O)OC(C)(C)C)=O)CC=CC1C(=O)NCC1C2COCC12 70963,C1(C(=O)NC2C(C)CN(C(=O)CCc3cncc(F)c3)C2)CCC2C(C1)C2(F)F 70964,CC(C)CC(O)C(C)C(=O)N1CC(F)(F)CC1C(=O)NC1C=CCCC1 70965,C1(C(=O)NCC2(NC(=O)COC3CCCOC3)CCC2)C(C(F)(F)F)C1[N+](=O)[O-] 70966,N1(C(=O)NCC2CCCN(CC=C)C2)CCc2c(Br)cccc2C1C 70967,c1(CC)c(C(N2CC(NC(C3(CC4CC4)CC3)=O)C2)=O)csc1C 70968,c1(C(=O)NC2CC(CNC(C3N(C)C(=O)CC3)=O)C2)cccc2c1nc(O)n2C 70969,C1(N)CC2CNCC12.C(=O)(CCCOC1CCOCC1)C(=O)CSc1nncs1 70970,CCCCCCCC(C)CNC(=O)NC(c1ccc(Cl)cc1)C(F)F 70971,C1(NC(C(CC=C)OC)=O)CCCC12CN(C(=O)Cc1cccc(CC#N)c1)C2 70972,c1(CC(=O)NC(CC)CN(C)C(C2SCCS2)=O)ccc(C)nc1 70973,c1(CC)ncnc(NC(c2cncc(-c3nn[nH]n3)c2)=O)c1F.N1(C)CC(N)CC1=O 70974,Nc1c(O)ccc(Cl)c1C(=O)NCC(CNC(=O)CN1CCCNC1=O)CO 70975,C1(C)(C(=O)NCCN(C(c2cn(CC(F)(F)F)cn2)=O)CC)CNC(=O)C1 70976,C(=O)(C(F)(F)C(F)(F)OC(F)(F)F)N1CC(CNC(c2snc(O)c2Cl)=O)C1 70977,Brc1ccc(C2CCN(CCCCc3nccs3)CC2)nc1 70978,O=C(C1=CCSC1)NCC1CC(F)CN1C(=O)Cc1ccc(Cl)cc1 70979,c1(C(N2C(CC)CN(C(=O)CC3(OC)CC3)CC2)=O)cnc2c(c1)NC(=O)CS2 70980,c1(C(N2CCC(NC(C3CCC(OC)CC3)=O)C2)=O)cnc2cc(C)nn2c1C 70981,C1(NC(Cc2c(C)nn(C)c2)=O)CC2CCC1N(C(c1nnc(O)nc1O)=O)C2 70982,Cn1nc(C(N2CCC(NC(=O)Cc3cnns3)C(F)C2)=O)c2c1CCSC2 70983,c1(C(N2CCCC(CNC(C(COC)C)=O)C2)=O)cccc2[nH]ccc12 70984,C1(C(=O)NC2(C(C)NC(=O)Cc3cccnc3C)CCC2)CCCCC1(C)C 70985,C(CC(C)C)(C(=O)NCC1CC1C1CCC1)N(C(CCC(C)SC)=O)C 70986,c1(OC)ncccc1S(=O)(=O)NC(=O)C(=C1CCCCC1(C)C)F 70987,N1(C(CCCNC(N)=O)=O)CC2CC1CCC2NC(C1C2C3CCC(C3)C12)=O 70988,Cc1cc(O)cc(=O)n1CC(=O)N(C)CC1CCN(C(C2C=CCC2)=O)C1 70989,n1(CC(=O)NCCC2CN(C(Cc3cn(CC)nc3)=O)C2)sc(=O)c2ccccc12 70990,C(=O)(C(F)(F)Sc1cnn(C)c1)N(CCN(C(=O)COCc1ccn(C)n1)C)C 70991,C(CCNC(C1(C)CS(=O)(=O)C1)=O)(C(C)C)NC(C(COC)O)=O 70992,c1(C(=O)NCCN2CCC(NC(C(CC)C)=O)CC2)ccc(Cl)c(Cl)c1F 70993,C(=O)(C(C(C)(C)C)NC(C1CC2CCC(C1)O2)=O)N1CCC(C)(C(=O)NC)C1 70994,C1(NC(c2ccc(-n3cncn3)cc2)=O)CCCC(C(=O)Nc2ncc(F)s2)C1 70995,Cc1csc2nc(NC3C(O)CCN(C(=O)N=c4ccc(Br)n[nH]4)C3)cc(=O)n12 70996,Cn1c(CNCC2(c3ccccc3)CC2(F)F)cnc1Cl 70997,c1(C(=O)NCc2cn(CCNC(C3C(OCC)C3)=O)nn2)ccc(OC)c(N)c1 70998,c1(C(=O)NCC2(O)CN(C(=O)Cc3cccc(Cl)c3)C2)cccc2oc(O)nc12 70999,N#CCCCCCC(=O)N1CCCC1CCC(=O)NCc1cn(C2CC2)nn1 71000,N1(C(C(C(C)C)NC(C)=O)=O)CCCC2CN(C(c3ccco3)C)CC12 71001,C(=O)(C(C)(C)C(N)=O)N1C(CN(C(CC(C)NC(=O)OC(C)(C)C)=O)C)CCC1 71002,C#CCC(C)(C(=O)NCCN1CCCC1)NC(=O)C1=CCCC1C 71003,C1(CCNC(COCC(C)(C)C)=O)CCC(NC(C2CC2CC(F)(F)F)=O)C1 71004,C1(NC(c2cccc(OC)c2)=O)CN(C(c2cc(C)ccc2N)=O)CC2(CC2)C1 71005,c1(C(N(CCNC(C2CCCC2n2cccc2)=O)CC)=O)ccc(Cl)c(Cl)c1 71006,N1(C(C2CC(N(C)C)C2(C)C)=O)CCNC(=O)CC12CCC2 71007,c1(C(N2CC(C(C)NC(C(C)OCCOC)=O)C2)=O)n[nH]c2c1CCCCC2 71008,c1(COCC)nc(C)c(C(=O)NC(C2(O)CCN(C(=O)C(C)C3CC3)C2)C)s1 71009,N1(C(c2cncc(C(C)C)c2)C(=O)Nc2c(C)cccc2)CCCN(C)C(=O)C1 71010,CC1CCSCCN1C(c1cccc(CC#N)n1)=O 71011,CC(C(=O)NCCC1CN(C(=O)CCc2nncn2C)CCO1)C(F)(F)C(F)F 71012,C1(CC(=O)OC)(NCC(C2CCN(CC(=O)OC(C)=O)CC2)C)CCCS(=O)(=O)C1 71013,C1(CNC(C2(CC(C)=O)CC2)=O)(CO)CC12CCC2.c1(CC=O)ccncn1 71014,CC(C)CC(C(=O)N1CCOCC1)NC(=O)CC1CC(C)OC1C 71015,C(=O)(C1=CCOC1)NC(C)CC1CN(C(=O)C(C)c2cccs2)C1 71016,C1(C(N2CC3N(C(C(C(CC)C)=O)=O)C(C3)C2)=O)C2CCC(C2)C1(C)C 71017,CC(CNC(=O)CC1CCC(=O)C1)(CO)NC(=O)C(F)=CCCN1CCCC1 71018,CC(C)(C)C1=NOC(C(=O)OCC(C)(C)NS(C)(=O)=O)C1 71019,CCCC(F)C(=O)N1CCC(CC(=O)NC2CC2N(C)C)CC1 71020,N1(C(CCc2cc(C)on2)=O)CCC2CCC(NC(=O)CCc3cncs3)C1C2 71021,N1(C(C(c2cccnc2)NC(=O)C=Cc2cc[nH]n2)=O)CCC(F)C(F)C1 71022,N1(C(=O)CCC(F)F)CCN(C(=O)CCn2ccnc2)C(c2cccnc2)C1 71023,C(=O)(C1=CC2CC(C1)CC2O)N1C2C(NC(c3cnc[nH]3)=O)C(CC2)C1 71024,C1(CC=C)(NC(=O)C(C)OC(C2CCCO2)(C)CC)CN(C(=O)Cc2csnc2C)C1 71025,C1(C(=O)NC(COCC)C)CC2(CCC2)CN1C(=O)C(C)=CC(C)(C)C 71026,C1(NC(C2CCN(C(CC)=O)C2)=O)CN(C(c2ccc(F)o2)=O)CC1F 71027,Cc1c(C(=O)NCC2CC(C)N(C(=O)Cc3cc[nH]n3)C2)cccc1C#N 71028,C1(CN(C(COCCOC)=O)C)CCCC(NC(=O)CC2CC(OC)C2(C)C)C1 71029,c1(C(N(C2CCCN(C(CCNC(COC)=O)=O)C2)C)=O)ccc(S(N)(=O)=O)[nH]1 71030,c1(OC)ccc(CC(N2CCC(CNC(=O)CC(=O)N(C)C)(OC)C2)=O)cc1O 71031,c1(C(N2CCC2C(N2CCOCC2c2ccccc2)=O)=O)c(O)cccc1[N+](=O)[O-] 71032,c1(NC(C2(CNC(c3c(NC)cncc3)=O)CCC2)=O)ccc(Cl)c(O)c1 71033,c1(C(=O)NCC2CCCCN2C(c2cc[nH]c2C2CCC2)=O)cc2sccc2s1 71034,C1(NC(c2c(OCC)ccs2)=O)CC(C)CN(c2nccc(C(=O)OC)n2)C1 71035,O=C1CCCCCN1Cc1cn(CC2C=CCN2C(C2CSCCS2)=O)nn1 71036,N1(C(C(CC)SC)=O)CC(OC)CC1NC(=O)CCCC#N 71037,c1(C(=O)NCC(CC)NC(=O)CC2CC(N(C)C)C2)[nH]nc(OC)c1Cl 71038,c1(OCC)cccc(OCCCNC(C2CC(F)(F)C2)C)c1 71039,CCCC(O)CC(=O)NCC1CCC(C)CN1C(C1CCCC1)=O 71040,N1(CC(CNC(=O)C(C)(C)C(N)=O)O)C2CCC1CC(CCOCCC(C)C)C2 71041,Cc1ccc(O)c(CNC(=O)CC=CCNC(C2CC3CC3C2)=O)c1 71042,N1(C(CN(CCOC)C)=O)CCN(C(=O)CC2CCC(C)O2)C(C2CCC2)C1 71043,N1(C(Cc2c(CC)noc2CC)=O)CCCC(C2(NC(CC(F)(F)F)=O)CC2)C1 71044,C1(O)(C(N2CCC(CNC(C(C)CC(F)F)=O)CC2)=O)CN2CCC1CC2 71045,N1(C(c2nc(COC)[nH]n2)=O)C2CCC1CC(NC(c1cc3n(n1)CCC3)=O)C2 71046,c1(-c2nc(C3CCCN(OC(C4CCC4)=O)C3)on2)cc(Br)ccc1OC(F)F 71047,C1(NC(CCC(C)(C)OC)=O)CC2CCC(C1)N2C(C)C 71048,C1(C(=O)NCCCC)(OC)CCN(C(C2CCCS2)=O)C1 71049,C#Cc1cn(C)nc1C(=O)NCC(CC)NC(c1ccc(N)cc1Cl)=O 71050,C1(COC)CCC(CC(N2CCCC(NC(=O)Cn3ccnc3C)C2)=O)CC1 71051,C1(CNC(c2nn[nH]c2Cl)=O)(CO)CCN(C(c2occc2C2CC2)=O)C1 71052,Cc1cccc2c1CCOC2C(=O)NC1CCCN(C(c2nn(C)cc2Cl)=O)C1 71053,c1(C(=O)NCCN(C(C)C)C(c2cccc(F)c2F)=O)ccc2c(c1)COCC2 71054,c1(OC)cnc(Br)c(NC(c2cc(C(F)(F)F)ccc2F)=O)c1 71055,c1(N(C)C)ccc(C(=O)NCC(c2ccccc2)CNC(=O)CP(C)(C)=O)cc1 71056,c1(C(=O)NC(CC)CN(C(=O)CC2CC2(C)C)C)cnc(-c2cccnc2)s1 71057,c1(C(=O)NC(C)CN(C)C(c2nocc2C2CC2)=O)ccc(P(C)(C)=O)o1 71058,C(C1CCN(C(=O)C(O)CC(C)C)CC1)=CC(=O)NCC(=O)OC 71059,CCC(O)(CNC(=O)C(N)Cc1cc(Cl)ccc1F)CCC(F)(F)F 71060,c1(-n2cc(C(CC)O)nn2)ccc(SC)cc1C#N.N12CCC(C(C)(C)C1)C2=O 71061,c12cccc(c1)C(=O)N2.c1(C(CC)CC)cc(CSc2ncccn2)on1 71062,N1(C(CCOCC(C)C)=O)CCN(C(c2ccc(CCN(C)C)cc2)=O)C(C)C1C 71063,N1(C(CCN(C(C2CCCC(OC)C2)=O)CCO)=O)CC2CCN(C)C2C1 71064,c1(N(CCNC(c2c3c(nn2C)CCCC3)=O)CC)ncnc2c1c(Br)nn2C 71065,c1(SC)nc(Cl)c(C)c(=NCC(C)(C)NC(=O)Cc2ccc3c(c2)CCC3)[nH]1 71066,C(c1ncco1)=CC(=O)NCCOC1CN(C(=O)C(c2ccccc2)F)C1 71067,C1(C(C)(C)C)(CNC(CCC(C)N(C)C)=O)CCN(C(C2CCCC(C)C2)=O)C1 71068,C1(C(=O)NCC2CC(NC(c3cnoc3-c3ccco3)=O)C2)C2CS(=O)(=O)CC12 71069,C12(CNC(C34CC(OC)C3C4)=O)CC1CN(C(c1ccc(CCO)cc1)=O)C2 71070,CS(=O)CC(=O)NCCCC(Cl)=CCl.c12cn(nn1)CC(=O)NC2 71071,C1(C(=O)NC2(C)CCN(C(C(C)OCC)=O)C2)CCc2nc(C)nn2C1 71072,C(=O)(CC(CC)C(C)(C)C)NC1C(C=C)CN(C(C2C=CC=CC=C2)=O)C1 71073,C1(C(C(=O)NCC(C(C)C)NC(C2(CO)COC2)=O)C)CCCC(F)(F)C1 71074,C1(CNC(=O)Nc2cccc(CN3CC(=O)NCC3)c2)CCN2CCCC2C1 71075,C12(CNC(N(C)Cc3cnn(C)c3)=O)CCCC1OCC2 71076,c1(CNC(=O)NC(C2COCCO2)CO)ccc(Br)cc1[N+](=O)[O-] 71077,n1(CC)cnnc1C(N1CC(NC(=O)C(C)NC(c2ccoc2)=O)C1)=O 71078,c1(SCC(N2CCC(C)(CNC(C(C3CC3)OCC)=O)C2)=O)ccc(F)c(F)c1 71079,C(=O)(CCP(C)(C)=O)NC(C(C)C)C(=O)NCCC1(C)CCCO1 71080,n1(CCCOC)nnnc1C(c1cc(C(C)(C)C)on1)NCC1(F)CCOC1 71081,c1(C(C(C)NC(C(=O)NC(c2nccn2C)COC)=O)C)ccccc1Cl 71082,C1(CNC(CCOCC#C)=O)C2CN(C(=O)C=Cc3cnccn3)CC12 71083,C1(NC(CC2C(CC)C2(F)F)=O)CN(C(c2cc(C)c(N)cn2)=O)CCC1O 71084,C1(C(=O)Nc2c(C)n(C(C)C)nc2)CCN(C(=O)CC2CCC(F)(F)C2)CC1O 71085,c1(OC)ccc(C(N)CC(=O)OC2CC3CNC2C3)cc1 71086,c1(NC(=O)Nc2c(C#N)cc3c(c2)COC3)ccc(S(=O)(=O)CCS(C)(=O)=O)cc1 71087,c1(OCC)cc(C(=O)NCC(c2cccc(Cl)c2)NC(=O)C2=CCSC2)ccn1 71088,Cc1cc(C(N2CC3CC2CN3C(=O)C(n2ccnc2C)C)=O)c2[nH]cnc2c1 71089,c1(C(=O)NCC2(NC(CCCC(C)=O)=O)CC2)c(C)nn2ccccc12 71090,CC(C)(CS(C)(=O)=O)C(=O)NCC1CCC(NC(c2cc3n(n2)CCCN3)=O)C1 71091,C=CC1CCCCN1C(=O)CC1(C)CCN(C(c2ccccc2C)=O)C1 71092,Cc1noc2ncc(C(=O)NC3CC(CNC(c4cccc[n+]4[O-])=O)C3)cc12 71093,C(=O)(C(C)(C)C(=O)NCCN(C(=O)C=Cc1ccc(C(N)=O)cc1)C1CC1)NC 71094,c1(OC)cc(C(c2nnnn2C2CCCC2)NCC(CO)OC)ccc1Cl 71095,c1(C(N(CCN(C(C(C(C=C)C)C)=O)C)C)=O)ccc2c(=N)[nH]cnc2c1 71096,Cc1cc(C(=O)NCC2(C)CCCN2C(=O)CCC2CCCC2)c(O)nn1 71097,CC1(C)CN(C(=O)CCCS(N)(=O)=O)CC(CNC(C2CC3(CSC3)C2)=O)O1 71098,CC1=CCC=CC1C(N1CCC(C(C)CNC(C2CCC(=O)N2)=O)CC1)=O 71099,N1(C(c2ccc(OC)o2)=O)CC(O)CC1CNC(=O)C(C)(C)C1CCCCO1 71100,c1(CC(=O)NCC2OCC(CNC(C3CCC(=O)N3)=O)C2)c[nH]ccc1=O 71101,C=C1CCN(C(=O)CCCCOC(CC)C(C)O)C(C(=O)NCC)C1 71102,C1(NC(C)=O)CN(C(=O)C(C2CCCCC2)c2cccs2)C2CCCCC12 71103,C1(C(N(C)CC2(CNC(c3c(C)scc3)=O)CC2)=O)CCc2nncn2CC1 71104,c1(CN2CCCC(C(C)NC(c3ccc(Br)c(Br)c3)=O)C2)ccc(F)c(F)c1Cl 71105,N1(C(C)C)CCCC1CC(=O)NC1CCCC1NC(=O)C(C)(C)c1ccnn1C 71106,N1(C(C(CC)n2cccn2)=O)CCCOC(CNC(=O)CN2C(=O)CNC2=O)C1 71107,CC1(C)CC(=O)NCC1C(N1CCC(OCCNC(C2CC(=O)N2)=O)C1)=O 71108,N1(C(C(c2ccccn2)C)=O)CC2CCC1CN2C(=O)CSc1cccc(Cl)c1 71109,N1(C(CC2ON=C(CC)C2)=O)CCCCCC1C(=O)NCCc1cnc(C)[nH]1 71110,C12(NC(Cc3ccc(C)nc3)=O)CC(CO)(C1)OC21CN(C(C2(C#N)CC2)=O)C1 71111,C(=O)(CC(C(F)(F)F)NC(C1CC2CC2C1)=O)N(CCCCOC)C 71112,N1(c2ncc(CCC)cn2)CCC(NC(C2CC=C(C)CC2)=O)C(C)(C)C1 71113,CC1CC(N(C(=O)CC2(N(C(=O)COCCCN=[N+]=[N-])C)CC2)C)CCO1 71114,N1(C(c2c(NC)cccc2OC)=O)CC2(CCCN2C(C2(C)CC2)=O)C1 71115,c1(NC(C2(NC(c3[nH]c(=NC)sc3)=O)CC2C)=O)ccc2c(c1)CCC2 71116,C1(NC(c2cc(C)cc(O)c2)=O)CN(C(=O)Cc2c[nH]nc2C)C2(CCC2)C1 71117,N1(C(CCC(C)(C)C)=O)CCC2(CCC2NC(c2csc(C(F)F)c2)=O)CC1 71118,C(=O)(C1CCCc2nncn21)NCC1CCCCN(C(CSCCCC)=O)CC1 71119,C1(C(=O)NCCCc2nc(C)c(C)[nH]2)COCCN(C(C2CCC(F)CC2)=O)C1 71120,n1(N(C2COCC2c2ccc(Br)cc2Br)C)cnc2c(N(C)CCO)ncnc12 71121,N1(C(c2cncc(C)c2)=O)CCC(C)C(N(C)C(c2cn(C3CC3)cn2)=O)C1 71122,Cc1cc(=NC2CCCc3n[nH]cc32)[nH]c(N2CCC(F)(CO)C2)n1 71123,N1(C(C2CCC(C)C2)=O)CC(NC(c2ccc(C(=O)OC)o2)=O)C(CC2CC2)C1 71124,C1(NC(C2CC(=O)OC2)=O)CCCN(C(c2nc(F)ccc2Cl)=O)CC1 71125,N1(C(C(C)OCC)=O)CCC(NC(C2CC=CCC2)=O)C1 71126,c1(OC)ccc(NCCCC(C2CC2)NC(=O)OC(C)(C)C)o1 71127,CCN=C(NCc1ccc(CO)o1)NCC1CCN(CCC)C1 71128,c1(CNC(CC(C(C)C)O)=O)cnn2c1CN(C(c1cncc(O)c1)=O)CC2 71129,C12CCC(CC1)C2NCC1(CF)CCCC1.c1(CC2CC2)nnnn1C 71130,C1(C)(CC=C)CN(C(=O)CCC2CCC(NC(=O)C(C)SCC)C2)C1 71131,c1(CC)nc(NC(=O)CC2CCN(C(=O)CCc3ccncc3)C2)c(Br)s1 71132,C1(N(C(=O)Cn2cc(C(F)(F)F)cn2)C)CCN(C(C2C3COCC23)=O)CC1 71133,C1(CNC(=O)CNC(C2CC23CCC3)=O)CC(C2CC2)=NO1 71134,Cc1cccc(Cl)c1C(N1CCC(CNC(c2cccc(OC(C)C)n2)=O)C1)=O 71135,c1(C(=O)NC2C(NC(=O)COCC3(F)CC3)CCOC2)ccnc2c1CCC2 71136,N1(C(C(c2n(C)ccc2)=O)=O)CC2CCC2(CC(=O)Nc2ccc(O)cc2Cl)C1 71137,c1(CN2CCC(C(N(CCC(=O)OC)C3CC3)=O)CC2)cc(Br)c(O)c(Br)c1 71138,Cc1ccccc1-n1nnnc1C(c1nnc(C2CC2)o1)NCCc1ccsc1 71139,C1(CC)C2CCC1CN(Cc1c(C)nn(CC)c1Cl)C2.c12cccc(c1)C(=O)NC2 71140,N1(C(C=C(CC)CC)=O)CCC(COC)(NC(=O)CC2C(=O)NN=C2C)C1 71141,c1(C(=O)NC)ccc(C(=O)NC2CC2NC(c2cccc(C)c2C)=O)cc1F 71142,[N-]=[N+]=NC1CCN(C(=O)C2=C(Cl)CCC2)C1C(=O)NCCS(N)(=O)=O 71143,C(c1ccc(F)cc1F)=CC(=O)NC(C(C)NC(=O)CC(C)(C)O)C 71144,c1(OC)ccc(C(CNC(C2CC3CC2C3)=O)NC(=O)C(O)CN(C)C)cc1 71145,Cn1nc(C(=O)NCC2(CCNC(c3cncc(Cl)c3)=O)CC2)cc1O 71146,C1(CC)(CC)CCN1C(CNC1(C)CC1)C=O.c1(COC)ccccc1 71147,c1(CC)nnc(=NCC2CCC(NC(c3cc4ccccc4[nH]3)=O)C2)[nH]c1CC 71148,c1(CN(C=O)Cc2c(OC)c(F)c(F)cc2)cccc2c1OC(C)(C)C2 71149,N1(C(CC2CCC(NC(CC(COC)C)=O)C2)=O)CC(=O)NCC12CC2 71150,C1(NC(C(C2CCC(=O)N2)C)=O)CCCCN(C(C23COC(CCO2)C3)=O)C1 71151,C1(COC)(NC(C2CCSC2)=O)CCN(C(=O)CCCSC)C1 71152,C1(C(=O)NC2CC(C)(C(=O)NC(CC#C)C(=O)OC)C2)CCCC2(CC2)C1 71153,C(=O)(CCC(=O)N1CCN(C(C2(C(F)F)CCC2)=O)CC1)NCCOC 71154,N1(C(CCN(CCOC)C(=O)SC2CC2C)=O)CC(=O)N(C)C(=O)C1 71155,C(c1sc2ccccc2c1Cl)=CC(=O)NCC(O)CN=[N+]=[N-] 71156,N1(C(CC2C(=O)NC(=O)N2)=O)CC2CCN(C(=O)Cc3cnoc3)C2C1 71157,C(=O)(CCC(C)C)NC12CC(CNC(C3(CC)CCCO3)=O)(C1)C2 71158,N1(C(CCCOC)=O)CC(C(=O)NCCC(F)(F)C(C)C)CC(C)C1 71159,C1(NC(C2(C)CC=C(C)CC2)=O)CN(C(C2(C)CCCS2)=O)Cc2nccn2C1 71160,Cc1cnc(N)c(C(=O)NC2CCC(C)N(C(c3coc(Br)c3)=O)C2)c1 71161,C=CC1(CC(=O)NCC2CN(C(=O)C(c3cccnc3)O)CC2O)CCCCC1 71162,C1(C(N2C(CN(C(CC3(CSC)CC3)=O)C)CCC2)=O)C2CCC3C(C2)CC13 71163,Cc1ccsc1CC(=O)NC1CCC(N(C(=O)Cc2nccn2C)C)C1 71164,CC1(N=c2[nH]c(Cl)ncc2[N+](=O)[O-])CC(NC(C2(C3CCCCO3)CC2)=O)C1 71165,CC1CC(NC(c2ccn(C3CC3)n2)=O)CN(C(C23CCC(CC2)CO3)=O)C1 71166,c1(OC)cc(N2CC3CC2CN3Cc2cccc(Br)c2Cl)nc(OC)n1 71167,N#CC1(CO)CC12CN(C(=O)CCc1ccc(N)cn1)CC2 71168,N1(C(CC(C)(C)N(C(CC(C)SC)=O)C)=O)CCCC(O)(CO)C1 71169,C1(CC=C)(NC(=O)CN2CCN(C)CC2)CCN(C(c2ccc(N)cn2)=O)CC1 71170,CCC(CN(C)C)CC(=O)NC(C1CCN(C(c2csc(C3CC3)n2)=O)C1)(C)C 71171,n1(CCC)ccc(C(=O)NCCC(=O)NCC2=CCCC2)n1 71172,c1(CNC(C(C)Cn2cccn2)=O)ncc(C(=O)NCC2(CO)CCC2)cn1 71173,Cc1c[nH]c2ncnc(Nc3nc(CC(=O)Nc4ccc(S(C)=O)cc4)cs3)c12 71174,CC(CC1CCC1)C(=O)NCc1cc(C(=O)N(CC(C)(C)C)C)cs1 71175,C1(CCNC(C2CC(=C)C2)=O)CCN(C(c2cn(C)nc2CC)=O)CC1(F)F 71176,n1(C2CCN(C(=O)C(O)CF)CC2)cnc2c1CCN(C(C1CC(F)C1)=O)C2 71177,C1(CNC(C(C)SC(F)(F)F)=O)CCN(C(C2COCCN2C)=O)CC1 71178,CCC(CC)C(=O)NC(CNC(C1CCC(Cc2ccccc2C)O1)=O)CO 71179,N1(C(C(CNC(C(C)=C2CCC2)=O)CC2CC2)=O)CCCC2COCC12 71180,C1(CC=C)(NC(CC=CC=C)=O)CCN(C(c2cnc(NC)cn2)=O)C1 71181,Cc1noc(C)c1C=CC(=O)NC1CCCN(C(c2ccn(C(F)F)n2)=O)C1 71182,C1(CCC)CCN(C(C2CC(C)(NC(=O)C(C)Cn3ccnc3)C2)=O)C1 71183,c1(C(=O)NCC=CCNC(c2ccc(C(C)C)s2)=O)cc([N+](=O)[O-])n[nH]1 71184,N1(C(C2C3CCC(C3)N2C(C2CCOCC2)=O)=O)CC23CCC2(COC3)C1 71185,C1(CC(=O)NC2CC(OC3CN(C(COC(C)(C)C)=O)C3)C2)CC(=O)NC1=O 71186,N1(C(C(CCCC)C)=O)CCCN(C(c2ccc(CN3CCCC3)o2)=O)CCC1 71187,CCCC(CCC)CC(=O)N1CC2(NC(c3cc(CF)on3)=O)CCC1CC2 71188,c1(CC)ccc(CN2CCC(F)(C(=O)Nc3c(Cl)cnn3C)C2)c(F)c1 71189,c1(C(=O)NCC2C3N(C(COCC#C)=O)C(CC3)C2)c(C)ccc(Cl)c1F 71190,CSC1=C(C(=O)NCCC(C)NC(C2(C#N)CC2(C)C)=O)CCCC1 71191,N1(C(C=C(CC)CC)=O)CCC=C(C(=O)N2CC(Cc3ccco3)C2)C1 71192,N1(CC)CCN(CC(N2CCSCC2C(=O)N(CC(C)O)C)=O)CC1 71193,c1(CCn2cc(C(=O)N)nn2)csc2nccn12.C1(C(=O)O)CC12CN(C(=O)C1CC1)C2 71194,C1(C(=O)Nc2c(OC)nsc2)CN(C(=O)C(C2CCC2)OC)CCO1 71195,Cc1nsc2ncc(C(N3CCC(CSc4cn(-c5nccs5)nn4)C3)=O)cc12 71196,C(C(C)(C)CC(=O)N1CC=CC(NC(=O)CNC(C2CCC2)=O)C1)OC 71197,C(=O)(C1=NN(c2ccccc2)C(=O)CC1)NCC1N(C(C2ON=C(C)C2)=O)CC1 71198,c1(OCC)cc(C(=O)N(C2(C)CCN(C(=O)COCC)C2)C(C)CC)oc(=O)c1 71199,N1(C(C(C)OC)=O)CCC(C)(NC(=O)CC(C)CNC(=O)OC(C)(C)C)CC1 71200,N1(C(C(CCCC)=O)=O)C(CO)CCC12CCC2.C1(C)C(C)C(=O)N1 71201,C(=O)(C(C)(C)CNC(C1(OC(C)C)CC1)=O)N1CCC(NC(C)=O)C1 71202,C1(CC(=O)NCC(C)C(=O)N(C2CCC2(C)C)C)C=NN(C)C1=O 71203,c1(CC(C(=O)NCC2(c3ccc(Cl)cc3)CC2)NC(C)=O)ccc(O)c(Cl)c1 71204,C(CC(C)(C)C(=O)N1CCC(O)(Cn2cc(-c3ccc(F)c(C)n3)nn2)C1)OC 71205,Cc1nc(S)nc(C)c1CC(=O)NC(CNC(C1CC(F)C1)=O)CC(C)C 71206,C(CCC(=O)N(C)Cc1cc[nH]n1)(C(C)C)NC(c1cc(OC)n[nH]1)=O 71207,c1(C2(C(N3CC(C)(NC(C4(CSC)CC4)=O)C3)=O)CCCC2)cccc(F)c1 71208,C12(C(=O)NCC(c3cccnc3)NC(=O)Cc3ccccc3)COCC1C2(F)F 71209,C(=O)(C(C)C(O)CC(C)C)N1CCC2(C(N(C3CC(=C)C3)C)=O)C(CC1)C2 71210,C12(CNC(C)=O)CC(C(N)=O)(C1)C1(CN(C(=O)CN(C3CCCC3)S(C)(=O)=O)C1)O2 71211,CCCCN=C(NCC1CCCc2sc(C)nc21)N1CC(C)N(C)C(C)C1 71212,c1(C(=O)NC(CC)CNC(C2(CO)CCCO2)=O)cc(C)cc2c1NCCC2 71213,O(NC(=O)C#CC(C)(C)CNC(c1cc(F)ccc1F)=O)C(C=C)C 71214,C=Cc1cc(C(N2CC3C(NC(c4cnc(S)n4C4CC4)=O)C3C2)=O)cc(F)c1 71215,n1(CCO)cnc2c(cnn2-c2ccccc2)c1=O.CCC1(C)COC(=O)NC1=O 71216,c1(CC)ncc(CNC(=O)CNC(=O)CNC(=O)CCc2cc[nH]n2)s1 71217,N1(C(c2ncccc2Br)=O)CC2CCC1CN2C(c1cccc2c1CCC2)=O 71218,c1(C(C(=O)NC2(c3nn[nH]n3)CC2)N(C)CC2CC2)cc(Cl)cc(Cl)c1 71219,Cc1noc(C)c1CC(=O)NC1CCC1NC(=O)CCC1COC(C)(C)O1 71220,C1(C(N(c2ccnc(CN(C)C)c2)C)=O)CCCC(NC(=O)C=CCF)CC1 71221,N1(C(c2ccc(C#C)nc2)=O)CC(C(=O)O)Nc2ccccc21 71222,C(=O)(C1Cc2ccccc21)NC1CCCCN(C(Cc2cc(C)cc(F)c2)=O)C1 71223,C1(C(=O)NCCCC2(C)CCCN2C(C2CCO2)=O)Cc2nccn2C1 71224,N1(C(c2cccs2)=O)CCCC2(C1)CN(C(c1ncnc3c1CCC3)=O)C2 71225,N1(C(c2c(C)cno2)=O)C2CCC1C(C)C(NC(=O)C(C)(C)C)C2 71226,C1(C)(NC(C(C)N(C(=O)CC2CCOC2)C2CC2)=O)CN2CCC1CC2 71227,c1(O)ccc(NC(N(C)CC)=O)cc1.C1(C(C)N)CCCN(CC(F)(F)F)C1 71228,C(=O)(C1(C)OCCc2ccccc21)NC1(CNC(CCSCC(C)C)=O)CCC1 71229,c1(C(N2CC(CC(=O)N(CCOC)C3CC3)C3(C2)CC3)=O)cc2cc[nH]c2cn1 71230,N1(C(c2cc(CC(C)C)on2)=O)CC(NC(=O)CC(C)n2cccn2)CC(C)C1 71231,Cc1cn(C)nc1C(=O)NCc1nc(C(=O)Nc2cncc(F)c2)c(C)o1 71232,N1(C(C(CSC)OC)=O)CCN(C(c2cc(Cl)cn2C)=O)CC(O)C1 71233,C(=O)(C(C(CC)CC)OCC)NC(CC=C)CC(=O)N1CCCC(CCCO)C1 71234,C1(C)(CC)NC(=O)N(CC(=O)NCCCNC(c2csc(C)c2)=O)C1=O 71235,N1(C(C2N(C)CSC2)=O)CC2(C1)CN(C(=O)CC(O)c1ccccc1)CC2CO 71236,CCCCC(O)C(C)C(=O)N1CC(O)(CNC(c2cc(Cl)c(C)cn2)=O)C1 71237,C(CCCCN=c1[nH]ccc(=NCCCc2ccnn2C)[nH]1)OC 71238,CC(CO)C(=O)NC12CC(CNC(=O)C(C)CNC(=O)OC(C)(C)C)(C1)C2 71239,c1(N2CCCC(NC(=O)CN3CCCNC3=O)CC2)nc2ccc(F)cc2s1 71240,N1(CCN(C(C(CC)O)=O)C)CCN(C(c2cnc(O)o2)=O)CC1 71241,C1(C)(OC)CC(C)(C)C1.CC1CC2(C1)C(=O)NCCOCC(=O)N2 71242,C=C(C(=O)NC1CC(NC(c2cc(Br)ccc2F)=O)C1)C(F)(F)F 71243,c1(C(C(=O)NCC2CC2SS(Cc2cnc(CC(OC)OC)[nH]2)=O)(C)O)ccc(C)cc1 71244,C1(C2CCN(C(c3ncnn3C3CC3)=O)C2)(NC(c2ncn(C)c(=O)c2)=O)CC1 71245,C1(C(N2CC(OC)C2)=O)CCC2(CC2)N1C(=O)CN1CCNC1=O 71246,C1(CNCc2c(C)sc(C(F)(F)F)n2)CC1C1CCOCC1 71247,Nc1cc(C(N2CC3CC2CC3CNC(C2CCCCS2)=O)=O)cnc1N 71248,C1(C(=O)NCCCOCCN(C(c2cnc(CC)s2)=O)C)CN2CCN1C(C)C2 71249,N1(C(c2cc(=O)cc[nH]2)=O)CCC2(CCCN2C(C2CC=CCO2)=O)C1 71250,c1(OCC(=O)NCCCC2CCCN2C(c2cnccn2)=O)ccc(Cl)cc1F 71251,C1(NC(C=C(C)Cl)=O)CC(F)CN(C(c2n[nH]c(=N)s2)=O)C1 71252,N1(C(C(C#C)(C)C)=O)CCN(C(c2cnn(CC)c2)=O)CC1 71253,Cc1ccc(Cl)cc1OCC(=O)NC1CCC(NC(C2(C)CC3(CC3)C2)=O)CC1 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71307,n1(CC(=O)NC2(CO)CCN(C(C3OCCN(CC)C3)=O)C2)ccc(=O)cc1C 71308,CCN(COc1ccc(C(F)(F)F)cc1)N1CCC(c2ncc[nH]2)C1 71309,C12CCN(CC1F)c1nc(ns1)C1CC21.N1(C(C2(C)CCCO2)=O)CC2CCC1C2 71310,c1(CC)ccc(C(N2CCOC(CCOC)CC2)C(=O)NCCSC)cc1F 71311,O([Si](C)(C)C(C)(C)C)CC1CN(C(CNC(C(C)(C)C)=O)=O)CC1F 71312,Cc1cc(C(=O)NCC2CCN(C(C3C4CCC3CC4)=O)CC2)cc2c1CCC2 71313,N1(CCC(N2CCC(CNC(c3ccsn3)=O)CC2)=O)C(=O)NC2(CCC2)C1=O 71314,c1(C(N2C(C3(NC(C(C(=C)Cl)(C)C)=O)CC3)CCCC2)=O)cccc2nn[nH]c12 71315,c1(C(=O)NCCC(CNC(c2ccc(C)nc2O)=O)O)cccc(C=C(F)F)c1 71316,c1(C(=O)NC(C)CNC(=O)Cn2ncnn2)nccc2c(Cl)cccc12 71317,C=CCC(CNC(=O)C(=Cc1ccccc1)C)C(=O)NC1(C(=O)NO)CC(C)C1 71318,c1(C(=O)NCC)ccccc1NC(=O)Cn1cccc1 71319,Cc1cccc(CC(=O)NC(C)CC2CN(C(=O)C3=CCOC3)C2)c1 71320,C(=O)(CC1=Cc2ccccc2C1)N1CCC(NC(c2ccc(F)cn2)=O)C(F)C1 71321,C(=O)(CCC(C)(C)C#N)N1C(CNC(C(c2n(C)nnc2)(F)F)=O)CCCC1 71322,c1(OC)cc(O)ccc1NC(C1CSCCN1C(=O)CCc1ccc[nH]1)=O 71323,C1(SC(C2(Oc3ccccc3Br)CCC2)=O)C2CCC1CC2 71324,C1(C)(C(N(CCCN(C(C2CCN(C)C2=O)=O)C)C)=O)CCS(=O)(=O)CC1 71325,N1(C(c2c(N(C)CC)nccc2)C(=O)NCCCC2CC2)CCNC(=O)C1(C)C 71326,C(=O)(CS(N)(=O)=O)NC(C)CN(C)C(c1ncnn1C1CCOCC1)=O 71327,N1(C(C2CN(C)C2)=O)CCC2CCC12CNC(c1ccoc1Br)=O 71328,N1(C(C(C)C)=O)CC2COCCC2(NC(C2(c3ccccc3Br)CC2)=O)C1 71329,C(=O)(C1=NN(C2CC2)C(=O)CC1)NCCCN(C(C1CC1C)=O)CC 71330,c1(CN(CCC)C(=O)NC23CC(NC(=O)C(Cl)(Cl)Cl)(C2)C3)ccccc1 71331,CC1CCC=C1C(=O)NC1COCCC1C(=O)NC1CCC12CCCC2 71332,N1(C(CNC(CC)=O)=O)CCC(C(=O)NCC2(C)CC3CC3C2)C(C)(C)C1 71333,C1(C(N(C)CC2N(C(C=CCC)=O)CCC2)=O)CCc2cnn(CC)c2C1 71334,N1(C(C2CC(NC(C(CCOC)OC)=O)C(O)C2)=O)CCOC2(CC2)C1 71335,c1(C(C(=O)NC2CCCC(NC(C(CC)(C)C)=O)C2)O)ccc(F)c(Cl)c1F 71336,CON(C(=O)CC1COCCN1C(=O)CC1CCC2(CNC2)CO1)C1CCCC1 71337,C(CCC(=O)NC1(C(N)=O)CN(C(=O)C(C)OCCC(C)C)C1)OCC=C 71338,c1(CC)cc(C(=O)N(CC#N)CCC2NC(=O)NC2)ns1 71339,N1(C(C(CC)(CC)CC)=O)CCC2(CC1)CCN(C(C1(C#N)CC1)=O)C2 71340,C#Cc1ccnc(C(=O)N(CCCNC(=O)CCn2ccnc2)CCC)c1 71341,C1(NC(C(CCC)C)=O)CCCC2CN(C(C3(CO)CCC3)=O)CC12 71342,C(C(C(=O)NOCCOC)SC1CC1)NC(=O)CSCC(=O)N(C)C 71343,C(=O)(C(C)NC(=O)NCC(C)NCCN(C)C)NCC 71344,Cc1cc(NCC(C)(CO)c2ccccc2)ncc1S(=O)(=O)N1CCC(C)(C#N)C1 71345,N1(C(C(C)Cc2ccccc2)=O)CC(NC(C2CC(CCO)C2)=O)CC(O)C1 71346,CN1CCC(OCCCC(=O)NC2CCCN(C(C3(C)CCCOC3)=O)C2)CC1 71347,CC(C)CC(C)CC(=O)NC1COCC1CNC(c1cccc2ncoc12)=O 71348,c1(C(=O)NCCC(=O)NC(CC)C)ccc(C=C2CCC(C)CC2)cc1 71349,C1(C)(C(=O)NCc2n(C)nnn2)CC(O)CN1C(C1CN2CCC1CC2)=O 71350,c12cc(N)ccc1C(=O)N2.C1(CC(=O)NCC2CC2CN(C)C)(COC)CC1 71351,c1(C(N(C2CCN(c3nnc(CC(F)(F)F)s3)CC2F)C)=O)cc(C)c(C)nc1O 71352,c1(C(N(CCCCC=C)C)=O)cc(F)ncc1NC(c1ncccc1CO)=O 71353,CC1CCCn2c(CC(N3CC(C4CCCN4C(c4ccsn4)=O)C3)=O)cnc21 71354,N1(C(C(CO)NC(=O)CC2CC=CC2)=O)CCC2CCC(C1)N2 71355,c1(OC)ccc(F)cc1C(C1=CCCCC1)NCc1ccc(Cl)o1 71356,C(C(CO)N=c1cc[nH]cc1S(=O)(=O)NCCN1CCC(C)(C)C1)OC 71357,c1(CC)ccncc1NC(=O)C(Cc1ccco1)NC(=O)C(C)OCCN(C)C 71358,Cc1cc(C(=O)NC2CC3CCC(C2)N3C(C2CN(C)CCO2)=O)cc(C)c1N 71359,c1(CC(=O)NCC2CCCN2C(C2CC2CSC2CC2)=O)ccc(Cl)nc1 71360,N1(C(C(C=C)(C)CC)=O)CCN(C(c2ccsn2)=O)CC2(CC2)C1 71361,C1(CCOC)CN(C(=O)Cc2ncoc2C)CCN1C(=O)C1=CCCCC1 71362,c1(-c2n(C(c3cccs3)C)nc(CC(F)(F)F)n2)nc2n(c1Cl)CCCC2 71363,c1(OC(C)C(=O)N(CC(C)(C)CNC2CC2(F)F)C)cccnc1 71364,c1(NCC)cccc(C(=O)N(CCC(C)NC(c2snnc2C)=O)C)c1 71365,C1(NC(=O)CCC2CCCO2)CC(=O)N(C2CN(C(=O)CCC3CCC(=O)N3)C2)C1 71366,c1(C(=O)NCCCCCNC(C(C)SCC(C)C)=O)oc2ccccc2c1CO 71367,S(=O)(=O)(c1ccc(C#N)cc1)NCCSC(C)C#N 71368,C1(OC)CCC2(CCN(C(=O)C=CCNC(=O)C(CC3CCC3)OC)C2)C1 71369,c1(C(C)CC(=O)NC2CC(F)(CNC(=O)Cn3ncnn3)C2)cncc(F)c1 71370,C(=O)(C(C)(C)C(F)(F)F)NC1CC(C)CN(C(=O)CCCN(C)C)C1 71371,C1(C(N2C(C(=O)N(C)CC3CCCC3)(CC)CCC2)=O)CC2C(C1)C2(F)F 71372,C1(CNC(CO)C(F)Cl)C2(CCC2)C12CCC2 71373,CCCCCC(C)(C)C(=O)N1CCOC(CNC(=O)CC(CC)OC)C1 71374,c1(NC(C(=O)NC(c2cccc(SC)c2)C)=O)cc(Cl)n2nccc2n1 71375,C1(NC(CC(COC)C)=O)C2CC3CN(C(=O)C=CCN4CCOCC4)C1C3C2 71376,C1(C(=O)NCC(=C)C(F)(F)F)CN(C(c2snnc2C)=O)CCC1O 71377,C(C(C)(C)OCC(=O)NC)SCC(=O)OC(C)(C)C.C(CCO)C1(OC(F)F)CC1 71378,Cc1cc(O)c(NC(C2CCC(NC(c3cnn4ccccc34)=O)C2)=O)cc1Br 71379,c1(OCC)ccc(S(=O)(=O)N(C2CCCCCC2O)C)cc1C(=O)N(C)C 71380,c1(C(C(N2CC(NC(CC3(CSC)CC3)=O)C3C2C3)=O)O)ccc(Cl)c(F)c1 71381,N(C1CCCc2c[nH]nc21)C(C(c1ccnn1C)NC(c1cc(CC)[nH]n1)=O)=O 71382,c1(NCCOC(CC)(C)C)cc(=NCC2(C)CCC(=O)N2)[nH]c(C(F)(F)F)n1 71383,C1(CC(=O)NCC2(OC)CCN(C(c3ccc(F)cn3)=O)C2)CC(O)C12CCC2 71384,N1(C2CCN(C(C(C)(C)N3CCCC3)=O)C2)CCN(C(=O)Cc2cccs2)CC1 71385,c1(CC(N2CCCCC(N(C(c3nc(C)sc3)=O)C)C2)=O)ccc2c(c1)CCO2 71386,N1(C(C(C)NC(=O)C2CC2)=O)CCC(C(=O)NCc2cnccc2Cl)CC1 71387,N1(C(C(CC(C)C)ONC(C2CC3C=CC2C3)=O)=O)CC2(CCOC(=O)N2)C1 71388,c1(CC(N2CC(C(C)NC(c3cccc(=O)o3)=O)OCC2)=O)ccc(O)c(F)c1 71389,CC1(C)CCCC1(N)C(N1CCCN(Cc2cc(Br)cs2)CC1)=O 71390,N1(C(c2n(CC)ncc2)=O)CCCC2CCN(C(c3cnsc3)=O)CC12 71391,CCCCC(C)CCC(=O)NC(C)C=CC(N1CCC(CCF)CC1)=O 71392,c1(-n2c(CC(C)C)nc(C(CC)O)n2)cc(C)ccc1C 71393,O=C1CC(CC(N2CCCC(CC(N3CCC(OCC4CC4)C3)=O)C2)=O)C(=O)N1 71394,N1(C(C(C=CC)O)=O)CC=C(CC(=O)NCCC(O)C2CCCC2)CC1 71395,CN1CC(NC(c2c[nH][nH]c2=N)=O)C(O)C1.C1(=O)C(CC2CC2)CN1C 71396,C(=O)(CCS(=O)(=O)N(C)C)N1CC(N(C(=O)CC2CC(O)C23CCC3)C)C1 71397,c1(C(C(=O)NCCC)Nc2ncnc3[nH]cc(I)c23)cccc2cc(C)cnc12 71398,C1(NC(C(c2n(C)ccc2)=O)=O)CCCC1(C)CNC(C12CCC(C1)C2)=O 71399,c1(C(N2CCN(C(C)C)CC2)=O)n[nH]c2c1CS(=O)(=O)C2.c12cnc(cn1)[nH]c2=O 71400,Cc1cncc(C(=O)NC2CCCC(CN(C)C(c3nc(C)n(C)n3)=O)C2)c1 71401,C1(CNC(c2cc(C)cc(F)c2)=O)CN(C(=O)CC2(C#N)CC2)CCC1(C)C 71402,c1(C(=O)NC2C(OC)CN(C(=O)C(C)O)C2)ccc2c(c1)nc(C)n2C(C)(C)C 71403,C(=O)(C(CCCC(=O)OC)N1CCN(C(C2CC=CC(O)C2)=O)CC1)NC 71404,Cc1cc(C=CC(=O)NCC2CC3(C2)CN(C(=O)C(C)CO)C3)ccc1F 71405,N1(C(C2CN(C)C(=O)C2)=O)CC(C(=O)NCCOCC2CCCC2)C2(CC2)C1 71406,N1(CC(=O)NCC(CCOC)NC(=O)Cc2nnc(O)s2)CCN(C)CC1 71407,c1(SC)ccnc(C(N2CCOC(CCNC(C3CC3(Cl)Cl)=O)C2)=O)n1 71408,C1(CNC(CC(C)(F)F)=O)CCCN(C(C2(C)CCC2)=O)CC1 71409,C1(CNC(C(c2cccs2)NC(CCC=CC)=O)=O)COC(C)(C)C1 71410,C(=O)(C=CS(C)=O)NCC1(NC(C2CCN(C(CCC)=O)C2)=O)CCC1 71411,N1(C(C(C)C)=O)CCN(C(C)C(=O)N(C(C)CC)CCO)CC1 71412,C(=O)(C1=CCC(NC(=O)C=Cc2cc[nH]c2)C1)N1CC(O)(COC)C1 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71794,C#CCC(C)(C(=O)N1CCC(C(=O)OC)O1)NC(=O)C(CC)CC=C 71795,C(CCC)(C(=O)NC(c1ccnn1C)C(=O)Nc1cccc(SC2CC2)c1)=CC 71796,CC12CC(C(N3CCN(C(=O)CCF)C(CO)C3)=O)(C1)C1(CCOCC1)O2 71797,C=CCC(CC)C(=O)N1CC2CC(C1)C2NC(C1C=CC=CC=C1)=O 71798,C#CC1CN(C(=O)CC2CC(C)=NO2)CCN1C(c1cc(CO)[nH]n1)=O 71799,C1(NC(c2c(C)coc2)=O)CC(C)CN(C(=O)C(C)OC2COC2)C1 71800,C12(NC(c3nc(CC(C)C)sc3)=O)CCC(CN(C(c3ccoc3)=O)C1)C2 71801,N1(C(CC(C=C)CC)=O)CC2(CCC2)CCC1CNC(=O)CN1CCOCC1 71802,CC1CC(C(=O)NCCOCCN(C(=O)CCC=Cc2ccccc2)C)C1(C)C 71803,c1(C(=O)NCc2ccc(Cl)cn2)cn2c(n1)CN(C(c1ccc(F)cn1)=O)CC2 71804,CN1CCOC(C(=O)N(C(C)(C)CC(=O)NCCc2cnccn2)C)C1 71805,N1(CC)CCC(C(=O)N(C2(C(=O)NC3COCC3SC)CCC2)C2CC2)C1 71806,C1(=O)C(CN=[N+]=[N-])N1.C(=O)(C(CC)n1cncn1)NCCN(CCC)CCC 71807,C1(C(=O)NC(C2CCCN(C(Cc3ccc(C)s3)=O)C2)C)CC2(C1)CC(F)(F)C2 71808,C=C(Cl)CCC(=O)N1CCOC(CN(C(=O)CCc2cccc(O)c2)C)C1 71809,C1(NC(CCCC#C)=O)CS(=O)(=O)C12CCN(C(=O)C(C)CS(C)(=O)=O)CC2 71810,c1(C(=O)NCC2(O)CN(C(Cc3ccn(CC)n3)=O)C2)cc(C)oc1C(F)(F)F 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71846,C12(CCC(C)CC1)C(c1n(CCC)nnn1)NC1(CC1)C(=O)O2.C(C)(C)(C)OC 71847,C1(C(=O)NC(C(=O)N(CC)CC)C)CC2CCN(C3CCOC3)CC12 71848,CC(C)CC(C(=O)N(C1CCCC1)CCNC(C12CCC1C2)=O)n1ccnc1 71849,C1(N(C)CC2(CS(C)(=O)=O)CC2)(CN(C)C)CCOC2(CCCCC2)C1 71850,N1(C(C2CC(O)CN2Cc2cccc(Cl)c2Cl)=O)CCC2(CCCO2)C1 71851,N1(C(CCCOC)=O)CCC2(CC1)CC2C(=O)NCc1ncc(C)s1 71852,N1(C(C(C)SC(F)(F)F)=O)CCCC(NC(c2ccc(N(C)C)nn2)=O)C1C 71853,C1(OC)CC(CC(=O)NC23CC(NC(c4cc(CF)on4)=O)(C2)C3)C1(C)C 71854,N1(C(C(C)NC(C)(C)C)=O)CCN(C(=O)C=Cc2cncc(F)c2)C(CF)C1 71855,c1(OC)c(C(=O)NCCC(C(C)C)NC(C2CC=CCO2)=O)c(C)nn1C 71856,C1(NC(c2ncc(Cl)s2)=O)CCN(C(c2ccn(C(F)F)n2)=O)CC1CO 71857,C1(C(C)NC(C2CCC3CC23)=O)CN(C(c2csc(C(C)(C)C)n2)=O)CCO1 71858,CC1CC(=O)NC1C(=O)N(CCCNC(=O)CCn1cccn1)C 71859,Cn1cc(Cl)c(CNC(=O)C(=O)OCCc2cccc(Oc3ccccc3)c2)n1 71860,N1(C(=O)OC)CCCC(C(N2CCC(C)(NC(c3ccn(CO)c3C)=O)C2)=O)C1 71861,c1(C(=O)NC23CC(C(=O)OC)(C2)C3)coc(C#C)c1.c12ccccc1CNC2=O 71862,Cc1ccn(C)c1C(=O)NCC(c1ccccc1)CNC(C1(n2cncn2)CC1)=O 71863,c1(OC)ccc(C(=O)NC(C)CNC(c2cc(C(O)C(F)(F)F)ccn2)=O)nc1 71864,CC1CC(C(=O)N(CCCCCCNC(C2CCCC3(CC3)C2)=O)C)=NO1 71865,N1(C(C(CN(CC)CC2CC2)F)=O)CCN(C(=O)CCOc2ccccc2)CC1 71866,Cc1c(Br)cnc(NC(C2C3CCC(C3)N2Cc2cc(C#N)cs2)=O)c1[N+](=O)[O-] 71867,Cc1nnsc1C(C)NC(=O)Cc1cnn(-c2nccs2)c1 71868,Cc1noc(C)c1CC(=O)NCC1(O)CCN(C(=O)C(C)NS(C)(=O)=O)C1 71869,n1(CC)cc(C(=O)NCC(O)CNC(=O)CCn2ccnc2)c(C(C)(C)C)n1 71870,N1(C(c2c(CC)[nH]cc2)=O)CCOCC(F)(CNC(=O)CC2CCNC(=O)C2)C1 71871,N1(C(C2CN(C(C)=O)C2)=O)CC2CCC1C(CNC(c1n[nH]cc1C)=O)C2 71872,C(=O)(CCCC(=O)Nc1cn(CC2CCC(=O)O2)nn1)NC1CCC(SC)C1 71873,Cc1ccc2sc(N3CCCC3C(C)(C)NC(=O)C(C)CF)nc2c1C 71874,c1(CC)ccc(CNC(C2C(C)CCN2C(=O)C(C)n2ccnc2)=O)cc1 71875,CCC(C)(C)CC(=O)NC1CC(F)(CNC(C2CCCCN2C2CCCC2)=O)C1 71876,C(=O)(CC(O)CN(C)C)NC(c1ccccc1)C(N1C(CC)CC1C)=O 71877,N1(C(CC(C)NC(N)=O)=O)CC(CNC(=O)CCc2nnc(S)nc2O)C2(CC2)C1 71878,C=Cc1ccc(C(N2CCC(F)(C(=O)NCc3ccc(F)cc3C)C2)=O)cc1 71879,C1(NC(c2ccccc2N2CCOCC2)=O)CCCN(C(=O)C(F)C2CCC2)C1 71880,c1(CN(C(=O)NCC(CC)(C)COC)C)cccc(Br)c1F 71881,CC1CCc2ccccc2C1NCc1cc(Cl)nc2n[nH]cc12 71882,c1(C(=O)NCC2(F)CCC(CNC(CSC(C)C)=O)C2)cccc(Cl)c1F 71883,c1(C(=O)NCC(C(C)C)NC(=O)C2=CCCC2C)cc(C(F)(F)F)cc(F)c1 71884,CCCCCCC(=O)N1CCC(CF)(NC(=O)Cc2ccc(Cl)nc2)C1 71885,C1(OCC2(CO)CCCO2)CCC(OC(=O)Cc2ccncc2)CC1 71886,N1(C(C(=O)NCCOc2cccc(CC)c2)=O)CC2CC2(CC)C1 71887,N1(C(C(C)SCC)=O)CC2CCC(C1)C(C(=O)NC(=O)C(C(C)C)C1CCC1)C2 71888,C(C)(CCC(F)(F)Oc1ccnc(C(F)(F)F)n1)NCC(COC)O 71889,C1(CCC)CCCC1C(=O)N(C(C)CCNC(=O)C(C1CCOCC1)O)C 71890,c1(Oc2c(C)cccc2)ccc2c(c1)C(C)(C)OC2(C)C.N12CCN(CC1)C2=O 71891,c1(C(=O)NC(CC)CNC(c2cnc([N+](=O)[O-])n2C)=O)c(Cl)nc2ccccn12 71892,N1(C(C(C2CC(F)(F)C2)OC)=O)CCCC2(NC(c3cnsc3C)=O)CC2C1 71893,CCC(F)(F)C(=O)N1CC2CC2(CNC(=O)CC(C2CCC2)OCC)C1 71894,Cc1ccnc(C(F)(F)C(=O)N2CC(CC(C)NC(=O)CC(C)NC(N)=O)C2)c1 71895,C1(C(=O)NC(C2CN(C(C3(c4ccccc4)CC3C)=O)C2)C)CCSCC1 71896,N1(C(c2ccc(C)cc2)=O)CC(C(=O)N(CC2CC2)CC2CC2)CC(C)(C)C1 71897,CN1CCN(C(C2(F)CCCOC2)=O)c2cnccc21 71898,C1(NC(c2ncccn2)=O)CCN(C(=O)CC23CCC(CC2)CC3)CC1F 71899,C1(COC(Cc2c([N+](=O)[O-])cn(CC)n2)=O)CCCC12CCOCC2 71900,Cc1c(Br)csc1S(=O)(=O)NCCc1sccc1Br 71901,c1(CC=CC)cc(C(=O)NCC2(C)CC(OC)CN2C(=O)CCC=CC)cc(C)c1 71902,c1(OC)c(C)cnc(NC(c2nnnn2NCc2cncc(Br)c2)C2CC2)c1C 71903,c1(C(N2C(CNC(C3C(=C)CC3)=O)CC(F)C2)=O)cc2c(CC)cccc2[nH]1 71904,C=CCCCC(C(=O)NCCC(F)(F)Cl)NC(C1CNC(=O)N1)=O 71905,C(=O)(C(CC(C)C)NC(C1CC(O)C1)=O)NC(COC)CCO 71906,CCCCCCC(CC)C(=O)N1CC(F)(F)CC1CNC(=O)C(C)C1CCOC1 71907,c1(C(N2CC(NC(=O)CSCc3ccccn3)C2)=O)ccnnc1S 71908,CC(=O)CCCC(=O)NC1CS(=O)(=O)CC1NC(=O)C1=NOCC1 71909,c1(C(N2C(CNC(CC3CCC(=O)N3)=O)CCCC2)=O)c[nH]nc1S(N)(=O)=O 71910,C(N=c1[nH]c(=NCC2CC2(F)F)[nH]c2c1CSC2)c1ccc(N(C)C)c(F)c1 71911,c1(CS(=O)(=O)N(N2CCOCC2)CC(N2CCCCC2)C)ccc(Cl)cc1 71912,C1(NC(COCC=C)=O)CCC(CSCC(C)(C)C)O1.C12CN(C1)C(=O)CO2 71913,C1(C(=O)OC)CCC(C)CC1CNCc1cc(-c2ccccc2)[nH]n1 71914,Cc1cc(C(N2CCN(C(C3CCC(CN)C3)=O)C(C3CCC3)C2)=O)cc(C)n1 71915,C1(C)(C(=O)NCC(CC=C)NC(=O)CCc2ncccc2C)CC(=O)N(C)C1 71916,N1(C(c2c(C)c[nH]c2)=O)CC(CC(=O)NC2CC3C=CC2C3)C2(CC2)C1 71917,N1(C(C(C(C)(C)C)O)=O)CCCC2(CCN(C(c3cc(F)c(F)cc3F)=O)C2)C1 71918,c1(C(=O)NCC(C2CC2)Nc2nccc(C3CC3)n2)ccc2ocnc2c1 71919,C(=O)(CC(F)(F)C(C)(F)F)N1CCCC(C)(CNC(C=CCCC)=O)C1 71920,C1(NC(C=CCOC)=O)CCC2(CC1)CC2NC(=O)Cn1c(C)c(C)sc1=O 71921,N1(C(C(CCC)O)=O)CC2(CO)CC1(C(=O)NC(c1cc[nH]n1)C)C2 71922,N1(C(CSC)=O)CC(CNC(C2CC3(C2)CC(C)(C)C3)=O)N2CCC1C2 71923,Cn1c(C(N2C3CCC2C(CNC(=O)C2=CCCCC2)C3)=O)cc(Cl)c1Cl 71924,CCC(C)C(=O)NC1CCCC1CNC(C1(C)CCC1)=O 71925,N1(C(C(CCC)C(C)C)=O)CCC2(CC1)CN(C(C1CC(C)CO1)=O)CCO2 71926,c1(SC)ncc(N)c(C(=O)N(CCNC(=O)CCc2nc[nH]n2)C2CC2)n1 71927,C1(NC(C(CSC)O)=O)CN(C(c2csc(Cl)n2)=O)CC2(CC2)C1 71928,N1(C(c2ccc(OC)c(Br)c2)=O)CC(NC(=O)C2=CCC2)C(C2CC2)C1 71929,N1(C(=O)Nc2ncc(Cl)cc2F)CCS(=O)(=O)c2ncc(Br)cc21 71930,C1(n2cc(CCC(C)O)nn2)CCC(C(N2CCC(n3cncn3)C2)=O)CC1 71931,C(=O)(C(C)(CC)C(N)=O)NCC1(C)CCN(C(c2nn(CC)nc2C)=O)CC1 71932,C1(C(=O)NCC2(COC)CCOC2)CC12CCN(C(=O)C(C)=CC(C)(C)C)CC2 71933,n1(CCC(=O)NC2CN(C(C3CC34CC4)=O)C2)c(=O)oc2cc(Cl)ccc12 71934,N1(C(c2c(C)nn(C)c2)=O)CC2(CC(C(=O)NCCN3CC(C)(O)C3)CO2)C1 71935,C1(NC(C(C)=C2CCCC2)=O)CC2CCC(C1C)N2C(c1cc2cscc2s1)=O 71936,C12(C(N3CC(C#N)(SC)C3)=O)CCCC1CCN2C(C1CC2CC(=O)C1O2)=O 71937,c1(OC)ccc(CNC2=CCN(C(=O)C(C)(C)C(=O)OC(C)(C)C)C2)c(OCC)c1 71938,C1(CC=C)(NC(=O)CCSC(F)(F)F)CCN(C(c2cc(CC)[nH]c2C)=O)CC1 71939,c1(C(=O)NC2CCN(C(c3c(C)cc(Cl)cc3N)=O)C2)cnc2c(c1)nnn2C 71940,c1(OC)cncnc1C(=O)NC1CC(O)(CNC(c2ccc(C3CC3)cc2)=O)C1 71941,Cc1ccc(C(=O)NCC2CCCN2C(c2c[nH]nc2OC(F)F)=O)c(Cl)c1 71942,C1(C2CCN(C(=O)COCCN(C)C)C2)(NC(CCCC)=O)CC1 71943,CCC(CCCC(F)(F)F)NC(=O)NC(c1ccc(C)cc1)CF 71944,c1(N2CC3C(C)C3C2)nc2c(c(=NC3CCc4ccc(F)cc4C3)[nH]1)SCC2 71945,C(=O)(C1=CCC(NC(=O)C#CC2CC2)C1)Nc1cccc(C(C)F)c1 71946,CC(C)(F)C(=O)NC1CCCC1CNC(c1cn(CCO)nn1)=O 71947,c1(C(=O)NC(CCC)CCCNC(=O)CC(C)(C)O)ccc(F)c(C)c1O 71948,Cc1ccc(OCCC(=O)NC2CCC(=O)NC2c2cnn(C)c2)c(Br)c1 71949,C(C(=O)NCCC(O)CNC(=O)CCCc1ncco1)(C(C)C)(C(C)C)OC 71950,C=CCCCCCCCCC(C(=O)NCCCF)N1C2CCCC1CC(O)C2 71951,Cc1cc(=NC2CCC(N3CCOCC3)C2)[nH]c(=NCC2COC(C)(C)C2)[nH]1 71952,CC(C)C(CC(=O)N1CCN(C(=O)C(C)(O)CC(C)(C)C)C2(CCC2)C1)C(C)C 71953,C(c1cccc(Cl)c1Cl)=CC(=O)NC1CCCN(C(=O)CC2CC23CC3)CCC1 71954,C1(CNC(c2nsnc2O)=O)CCN(C(c2ccc(Cl)c(O)c2)=O)C12CC2 71955,CC1CN(C(c2ccc(-c3cccc(Br)c3)n2C)=O)CCC1O 71956,c1(C(=O)NCC2CN(C(CCCC)=O)C(C)(C)C2)cc(C)cc([N+](=O)[O-])c1N 71957,c1(CC)cccc(C(=O)NCC(C(=O)N2CCC2C(=O)NC)OC)n1 71958,c1(C(C(=O)NC)N(C)Cc2ccc(-c3ccc(Br)cc3)s2)cc(C)oc1C 71959,c1(OC(C)C(=O)NC2CCC(F)(CNC(C34CC(C)(CO3)C4)=O)C2)cccc(F)c1 71960,c1(C(=O)NC(C2CN(C(CCCOCC)=O)C2)C)cncc(C)c1C 71961,C1(NC(c2c(OC)nsc2)=O)CC2(C1)CN(C(C1C=CCS1)=O)C2 71962,Cc1cccc(CNC(c2ccc(-n3cncn3)nc2)=O)c1C 71963,C(CCCCCN=[N+]=[N-])NC(CC1CC(NC(CC(C)O)=O)C1)=O 71964,C1(CC(=O)NCCN(C(c2ccc(OC)cc2F)=O)C)CCC2(CC1)CCC2O 71965,CCCC(C(O)C(=O)NCCCc1cccnc1)NC(C1CC(O)C1)=O 71966,C1(NC(C2CCN(CC)C2)=O)CC(=O)N(C2CN(C(=O)C=CC3CCCC3)C2)C1 71967,C1(n2cc(CSCCNC(CC)C(=O)N3CCOCC3)nn2)CCCC(CO)C1 71968,N1(C(C=C2CCN(C)C2)=O)CC2(C1)CN(C(=O)C(O)CCn1cncn1)C2 71969,c1(OC)ccc([N+](=O)[O-])c(N2CC(NC(=O)C(C)C(C)O)CC3(CCC3)C2)c1F 71970,C(CCC)(C(=O)NCC(C1CC1)NC(c1cnc(COC)cn1)=O)=CCC 71971,C(CCCOC)(C(=O)N1CC(c2nncs2)C1)NC(CCC=C)=O 71972,C1(C(=O)NCC2CCN(C(c3n(C)nc(O)c3)=O)CC2)CN2CCCC1CC2 71973,N1(C(C(C)Cc2ccccn2)=O)CCN(CCNC(=O)CC2CCCCC2)CC1 71974,n1(CCC(=O)NCC(COC)(C)OC(C)=O)cnc(C)cc1=O.C(C)(C)C 71975,c1(C(=O)NCC2CCN(C(C3(CF)CC3(F)F)=O)C2)ccc(CO)cc1 71976,C12(C(=O)NCCN(C(C(C3CCC3)OC)=O)CC(C)O)CCC(=O)N1CCS2 71977,c1(OC)ccc(C(=O)NCC(CNC(C2CC(F)(F)C2)=O)OC)c(C)n1 71978,c1(C(N(C2CN(C(c3c(SC)snn3)=O)CC2F)C)=O)cccc2c1OCCO2 71979,C(CCCCC(=O)NCCC(=O)NO)N(C(C(C)CN(C)C)=O)C.C 71980,Cc1ccc(C(=O)NC(CNC(=O)C(N2CCN(C)CC2)C)C2CCC2)n1C 71981,CC1(CNC(=O)C(O)C2CC2)CCCN(C(=O)CNc2cc(F)ccc2F)C1 71982,C1(CCC)CCCC1C(=O)NCC(CC)NC(c1cn(CCN(C)C)nn1)=O 71983,c1(CNC(c2c(C)coc2)=O)ccc2c(c1)CCC2NC(=O)C(O)CCC(C)C 71984,C(=O)(C(C)CC(C)(F)F)N1CCC(N(C(=O)Cn2nc(C)n(C)c2=O)CC)CC1 71985,C1(C(=O)NC2(C)CCN(C(c3cccc(C(=O)NC)n3)=O)C2)CC(O)C12CCC2 71986,c1(CS(=O)(=O)CCNC(=O)NC(C)CC(O)c2ccccc2)nn(C)cc1Br 71987,c1(C(N2CCCC(CCC)C2)=O)coc2c1CN(C(=O)CCC1CCCCO1)C2 71988,c1(-n2cc(C(N(C(C(CC)Oc3cccc(C)c3)=O)C)C)nn2)ncccc1C 71989,Cc1c(C(=O)N(C)CCNC(C2(C(=O)OC(C)(C)C)CCC2)=O)nnn1C 71990,C(=O)(C(C)CCC(C)(C)C)NC(CCCNC(c1ccc(SCC)nc1)=O)(C)C 71991,C1(C)(C(=O)NCC2CCC(CNC(c3c(C)cncc3)=O)CC2)CCN(C)C1=O 71992,C1(COC)(CNC(C2(C)C=CCC2)=O)CCCN1c1nccnc1F 71993,c1(C(=O)NC2CC3(C2)CN(C(C2CCC4CCC2O4)=O)C3)cccc2nonc12 71994,c1(CC)cccc(OCC(=O)NCC2CN(C(c3ncccn3)=O)CC2O)c1 71995,C=CC(C)(CCOC)C(=O)NCC=CCNC(=O)C(c1c(C)cccc1C)CC 71996,c1(CC)cc(C(=O)NC(C)CN(C(C2C(C)C2C)=O)CC)ccn1 71997,c1(CC(N2CCC(C(C)NC(c3nc(CC)oc3)=O)CC2)=O)c(F)cncc1Cl 71998,N1(C(C(O)NC(=O)OC(C)(C)C)=O)CCC2(CCCN2C(C2CC3CC3C2)=O)C1 71999,c1(C(=O)NCC2C=CC(NC(CCCC3C(C)C3)=O)C2)c(Cl)ccnc1F 72000,c1(SCC(=O)NC(c2ccccc2F)CNC(C(C)SC)=O)ccccc1Cl 72001,O=C1CC(CNC(=O)CCn2cc(CCCCO)nn2)C(=O)N1.c12cccc(c1)C2 72002,C(=O)(C(C)C(C)c1ccccc1Cl)OC.C1C(=O)N1.C1COCCN(C)CCO1.COC 72003,C1(NC(c2c(C)cc(CNC(=O)CC3(O)CCOC3)o2)=O)CCn2nnnc2C1 72004,C1(C(N(C)CC2CCCN2C(=O)C=Cc2cc[nH]c2)=O)CCCC2(C1)CC2(F)F 72005,N1(CC)N=C(C(=O)NCCCCNC(C2CCC(n3ccnc3)O2)=O)CCC1=O 72006,c1(C(N(CCC(=O)NC2CCCOC2)CCO)=O)n[nH]c2c1CCC2 72007,C12(C(N3CCC(N(C(=O)C=Cc4ccccc4)CC)C3)=O)CC3CC1C2C3(F)F 72008,N1(C(C(C2CCCC2)OCC)=O)CC(N(C(=O)C=CC=C(Cl)Cl)C)C2(CC2)C1 72009,C1(N(C(=O)Cn2cnnn2)C)CC2CCC(C1)N2C(c1cnc(N)c(Cl)c1)=O 72010,N1(C(=O)OC)CCN(C(=O)NC(CC(=O)Nc2ccccc2)C(C)C)CCC1C 72011,C1(NC(c2c(C)nc(C)o2)=O)CN(C(=O)CCc2ccsc2)CC1C1CC1 72012,CC(C)CC(CC(=O)N1CCC(C(C)(C)O)C1)NC(=O)CCC1CCCOC1 72013,c1(C(=O)OCC)nc(=NCC(C)CNC(=O)CCCc2cnn[nH]2)c(F)c(Cl)[nH]1 72014,C1(NC(C=CCOC)=O)CCC12CN(C(=O)CC1(O)CCCC1)C2 72015,c1(C(=O)NC2CN(Cc3ccc(Br)cc3Cl)CC2F)ccc2cccc(Br)c2n1 72016,C1(NC(C(CC=C)CNC(C2(CC3CC3)CCC2)=O)=O)CCn2nnnc2C1 72017,c1(N2CC(CNC(=O)NC3CCN(C(C(C)O)=O)C3)C2)ncc(F)cn1 72018,N1(C(C2(C=C)CCC2)=O)CC2CCCC2(NC(=O)CSCCOC)C1 72019,C(=O)(C(O)CCC(C)C)N1C(CNC(C2C(OC)CCCC2)=O)CC2CC21 72020,C1(C2(O)CCOCC2)(C(N2CC3(CC(NC(C4C(CC)CCC4)=O)C3)C2)=O)CC1 72021,CCCN=C(NCC1COCCN1CC)N1CCC2(C1)CC2(F)F 72022,c1(C(=O)NC2C(NC(CC(C)CF)=O)C2)cc2c(Cl)ccnc2s1 72023,N1(C(CCCCOC)=O)CC2CCN(C(=O)CC3(N(C)C)COC3)C2C1 72024,C=CCC(C(=O)NCc1cc[nH]c1C(N1CCOC(CO)C1)=O)OC 72025,c1(OCC(c2ccccc2)N(C)C(C2CC3CC2CCN3)=O)cc(F)ccc1F 72026,n1(CC)ncc2c1CCCC2N=c1[nH]c2c(c(=NCCCN(C)C)[nH]1)SCC2 72027,c1(CNC(C2C(=C)C2)=O)cc(NC(=O)COCCOC)no1.C1(CN)CC(O)C1 72028,C(C1c2ccsc2CCN1C(=O)C=C1CCC1)NC(C1CC2CCC2C1)=O 72029,N1(C(COc2ccn(C)n2)=O)CCC2C(C1)CN2C(c1cc2c(s1)CCCC2)=O 72030,N1(C(C2OCCN(C(C(N3CC4CC4C3)C)=O)C2)=O)CCC(O)C(N(C)C(=O)NC)C1 72031,c1(C(=O)NCCC2(NC(c3c(C)onc3Br)=O)CC2)cc2c(cn1)OCCO2 72032,C1(C(=O)NCC2(C(N3CCCC(C(=O)NC)C3)=O)CC2)CC(=O)N2CCCCC12 72033,N#Cc1c(O)nsc1SCCNC(=O)Nc1cccc(Cl)c1Br 72034,c1(C(N(CCOC)CCNC(C2(C(F)(F)F)CC2)=O)=O)cc([N+](=O)[O-])c[nH]1 72035,N1(C(C(CN(C2CC2)CC)F)=O)CCCC(C2CC2NC(C2CC(OC)C2)=O)C1 72036,c1(N(C(=O)C(N)C(=O)OCc2cccc(Cl)c2Cl)C)cnnc(O)c1Cl 72037,CC1(C(=O)NC2(CCNC(C3CCC(C(F)(F)F)C3)=O)CCCC2)CCCCC1 72038,C(=O)(C1OCCc2ccccc21)NC1CCN(C(C(C)SCC)=O)C(CC)C1 72039,c1(C(N2C(C)CCN(C(=O)C=Cc3cc[nH]n3)CC2)=O)ccc2c(c1)CCCC2 72040,C(C)(C)(CCC(=O)N1CCCC(C)C1CNC(=O)CN1CC2CC2C1)OC 72041,c1(OC)ncnc(C(N2CCC(C)(CCNC(C3CC3(F)F)=O)C2)=O)c1F 72042,C1(C(=O)OC)(C(=O)NC2CCC2CNC(=O)COC2CCCCC2)C2CCC12 72043,N1(C(=O)OC(C)(C)C)CCC(C2CCO2)CC1.C12(C)CCN1C(=O)C2C(C)C 72044,C(=O)(C(C(C)C)N1CCCCC1)NC1C(CNC(C(COC)OC)=O)CCC1 72045,c1(C(=O)NC2C(CC)CN(C(c3ccc(Cl)nc3C)=O)C2)cnn2c1NCCC2 72046,C1(C2CCN(C=O)C2)(N(C(=O)CCC2CCCOC2)C)CC1.C(C)(C)(C)OC(=O)N 72047,c1(C(=O)NCC(CN(C(C2C(C)C2C)=O)C)C)c[nH]c2nccc(Cl)c12 72048,c1(C(N(C(CCNC(CCCCNC(C)=O)=O)C)C)=O)n[nH]c2c1CN(C)CC2 72049,C1(CC(=O)NCc2cnc[nH]2)OCC2CCN(C(c3cnc(F)c(Br)c3)=O)CC12 72050,N1(C(C2CC(C#C)(O)C2)=O)CC(C)N(C(c2cnn(CC)c2C)=O)CC1C 72051,C(=O)(C(F)(CNC(C1CCCC1C(C)C)=O)C(C)C)NCCNC(=O)NC 72052,Cc1nc(C(=O)C(=O)NCC(CNC(=O)CCC2CCCO2)CO)cs1 72053,C#CCCC(N)C(=O)N1CCCC(C(=O)N(C(C2CCCC2)CC)C)C1 72054,C1(C(=O)NCC2C(NC(CCOC)=O)C2)C2CCC1(c1ccncc1)C2 72055,c1(C(=O)NC2(C)CCCN(C(C=C(C)C(F)F)=O)C2)cccn2c(C)nnc12 72056,C=CC1(C(=O)NCC(O)CC(F)(F)F)CCN(C(C2CCC(OC)CC2)=O)C1 72057,C(=O)(C1=CC2CCCCCC12)NCCC1(CNC(C(CC(C)(C)C)O)=O)CC1 72058,C1(OC)(CNC(C2(CO)CC2)=O)CCN(C(C2(C)CC3CC3C2)=O)CC1 72059,CC(C)CC(C(=O)NCc1cncc(Cl)c1)ONC(C1(CCO)CCC1)=O 72060,C(=O)(CCC(C)(C)N(C)C)N(C(CC)C(N)=O)CC12CCC(OC)C1C2 72061,C#CC1(NC(C2CCCCN2C(=O)C=CCF)=O)CCC(C)(C)C1 72062,c1(C(=O)NC2CC(C(=O)NCC3CC4CCC4C3)CC2O)cnc2n1CCC2 72063,CCC(C(=O)NCCOC(C)(C)CNC(c1ccc(F)cn1)=O)C(C)(F)F 72064,C#Cc1ccccc1CC(=O)NC(C)C=CC(N1CCC2(CSC2)C1)=O 72065,C1(C(N2CCCc3n[nH]cc32)C)CC2(C1)CS(=O)(=O)C2 72066,N1(C(c2c(CC)nn[nH]2)=O)CC(C2CCCN(C(=O)C(C(C)C)C(C)C)C2)C1 72067,C12(CNC(c3c(C)nccn3)=O)CCC(CN(C(=O)Cn3cnnc3O)C1)C2 72068,c1(CN2CCC(CC(=O)Nc3c(C(N)=O)occ3)C2)cc(O)ccc1F 72069,N1(C(C(n2c(C)cc(C)n2)C)=O)C(C(=O)NCCSC(F)F)C2CC(O)C1C2 72070,c1(C(=O)NC2C(NC(COCCN(C)C)=O)CCC2)cc2c(nn1)CCC2 72071,Cn1nc(C(N2CCCC2(C)C(=O)NCc2ccc(Cl)cc2)=O)cc1C#N 72072,C1(NC(c2c(C)nco2)=O)CCCCC1NC(=O)CC1CC=CCC1 72073,CC1CN(C(=O)CC2(N(C(=O)COCC3CCC3)C)CC2)C(C)(C)C1 72074,c1(SCCCC)ccc(C(=O)NCC#CCNC(C2CC(C#N)C2)=O)cc1 72075,c1(COC)ccc(C(=O)NC2CCCC(NC(=O)C(F)(F)C3CC3)C2)cc1 72076,N1(C(C(c2ccccc2)C)=O)CC(O)CC1C(c1ncccn1)=O 72077,C1(NC(C(C)SCCCC)=O)CCCCN(C(=O)Cc2nc(F)ccc2Cl)C1 72078,C1(C(=O)NCCCCCCNC(=O)CC2CCSC2)(CC)CCCC1O 72079,Cc1cc(C(=O)NCCC2CC(NC(c3[nH]cnc3C#N)=O)C2)cc(C)c1Cl 72080,N1(C(C(CC(N)=O)NC(C2COCC(C)O2)=O)=O)CCOC2C(O)CC12 72081,C123CCCC1N(CCC2)c1[nH]cnc2nc3cc1-2.CCCCCC(=O)N(C)C 72082,n1(-c2ccc(NC(C(CCc3ccccn3)OC)=O)cc2)ncc(Cl)c1C 72083,c1(C(=O)NCC2CC(NC(c3c(C)cccc3C)=O)C2)cnc2sc(C)c(C)n12 72084,CC1(C)CN(C(=O)COc2cccnc2)CCC1NC(C1CCc2nn[nH]c2C1)=O 72085,N1(CCC(=O)NCC(CC)NC(CCN(CCCCC)CC)=O)CCOCC1 72086,N1(C(COCCC(C)C)=O)CCN(C(=O)CN(C)C(C)C)CC2CCCCC12 72087,CCC(C)CCCCC(=O)N1CCC(F)C(NC(C2(O)CN3CCC2CC3)=O)C1 72088,c1(-c2c(NC(=O)NC3CC3CO)cccc2)cc(F)c(O)c(F)c1 72089,S(=O)(=O)(c1ccc2nc(Cl)[nH]c2c1)NC(c1ccc(OC)cn1)C 72090,c1(C(NC(C2(F)CCOCC2)c2n(CCOCC)nnn2)CC)cnc(C)n1C 72091,c1(C(=O)NCCC(=C)CNC(c2oc(CO)nc2C)=O)cnc(N)c(N)c1 72092,c1(C(=O)NCCOc2c(C)cccc2)ccc(=NC2CCN(CCF)C2)[nH]n1 72093,c1(C(=O)NCC23CC(C(=O)NC4C(C)CN(C)C4)(C2)C3)cc(C#N)ccc1F 72094,c1(SC)nc(O)nc(C)c1C(=O)NC1(CN(C(=O)CCCN2CCCC2)C)CC1 72095,N1(C(COC(CC)C)=O)CC2C(CNC(=O)C(C(C)C)NC(N)=O)C2C1 72096,C1(CNC(C(COC)(C)O)=O)CN(C(=O)CNC(=O)NC2CC2)CC2(CCC2)O1 72097,c1(OC)ccc(C=CC(=O)NC2CC3C2CCN3C(=O)C(C)C2CCCC2)nc1 72098,N1(CC(=O)N(C2CCN(C(c3cccc(O)n3)=O)CC2)C)CCCCCCC1=O 72099,C(CCC(C)CC(=O)N1CCN(C(c2cncc(C)c2)=O)CC1C(F)F)=C(C)C 72100,CC(C)C(CC1CCCCC1)C(=O)N1CCCN(C(C2CCC3CC23)=O)CC1 72101,CCCCCCC(C)CC(=O)N1CCN(C)C(CNC(c2cc(C)sc2N)=O)C1 72102,c1(C(=O)NCCC2(CNC(C(C)(C)SC)=O)CC2)ccn2ccccc12 72103,C(C1CCOCC1)=CC(=O)NC(CNC(c1n(C(C)C)nnc1)=O)(C)C 72104,C1(CCC(C)(C)NC(=O)OC(C)(C)C)CN(C(C(CCO)C2CC2)=O)CCO1 72105,c1(CNC(CNC(C(N)=O)C2CCOC2)=O)cn(CC(N)=O)nn1 72106,c1(OC)ccc(CC(=O)NCC(CO)NC(C2CCC2OC)=O)cc1 72107,S(=O)(=O)(c1ccc(N2CCc3nocc3C2)cc1Br)N1CC(O)CC(C)C1 72108,C12(OC)CCCC(C(=O)NC(CNC(=O)C3=C(Cl)CCC3)CC(C)C)(CC1)C2 72109,c1(-c2cccc(C(C)=O)c2)cc(C(N2CCOC(O)C2)=O)c2cn[nH]c2c1 72110,C1(C2CCCN(C(=O)C3=CCCCC3)C2)(NC(=O)CC2COC(=O)C2)CC1 72111,c1(C(=O)NC(C(=O)NCCC(F)(F)CO)c2ccoc2)cccc2c[nH]nc12 72112,C#Cc1ccc(C(=O)NC(CC)(CC)CCNC(c2ccc(CF)cc2)=O)cc1 72113,c1(CCc2cn(C3(C(N4CC(C#N)(CC)C4)=O)CC3)nn2)ccc(C)c(C#N)c1 72114,CC1CN(C(C2CC3C(C2)C3(C)C)=O)CCC1N(C(=O)CCN1CCOCC1)C 72115,C=CCC(C(=O)NC1(CNC(=O)Cn2cc([N+](=O)[O-])c(C)n2)CCC1)C(C)C 72116,c1(C(=O)NC2(CN(C)C(C3(C)CC(C)(C)C3)=O)CC2)cccc(CS(N)(=O)=O)c1 72117,c1(C(N(CC(C)O)CCNC(c2c(C)oc(Cl)n2)=O)=O)c[nH]c2ccc(Cl)cc12 72118,c1(C(=O)NCCN(C(C)C)C(CCC2=CCCCCC2)=O)ccc(S(C)=O)cc1 72119,C1(NC(C=CCN(CC)CC)=O)CN(C(c2ccnc(C)n2)=O)C2CC12 72120,c1(CCN2CC(=O)N(CCC(=O)NCC(F)(F)CO)C2=O)cccc([N+](=O)[O-])c1 72121,CCCCC(O)CC(=O)NC1C2CCC(C2)C1C(=O)N(CC(O)COCC)C 72122,N1(C(c2cc(C)nn2C)=O)Cc2ccccc2C(CNC(c2nccn2C)=O)C1 72123,C1(NC2CN(C(C(=O)Nc3c(C)c(Br)ccc3)=O)C2)C2CCC(F)(F)C12 72124,CC1CCN(C(=O)C(O)C2CCCC2)C(C)C1NC(=O)C(C)NS(C)(=O)=O 72125,c1(NCCCOCC)cc(NCC2(CCC)CC2)nc(C)n1 72126,c1(CN(C2CCSC2)Cc2c(OC)cccc2)cc2cccc(F)c2o1 72127,N1(C(CCOC)=O)CC(NC(=O)Cc2cccc(C(C)(C)C)c2)C(C)(C)C1 72128,C1(NC(c2c(C)nc(C3CC3)o2)=O)(CNC(C2(C)CC2(C)C)=O)CCC(C)(C)CC1 72129,c1(CC(=O)NCC(CC(C)C)NC(C2(OC)CCCOC2)=O)cc(C)ccc1F 72130,CC1CN(C(c2sccc2CN(C)C)=O)CC1CCNC(c1snc(Cl)c1Cl)=O 72131,C1(CC)CCC2(CCN(C(=O)NCC3CCC(=C4CCC4)CC3)C2)O1 72132,C1(NC(Cc2scc(C)c2)=O)CC=C(C(=O)NC2C(C)CCC2C)C1 72133,CC1(C#CC(=O)NC(c2cccc(F)c2)CNC(=O)Cc2cnoc2)CCCO1 72134,c1(C(C)O)ncc(C(=O)NC(C)(C)C(C)NC(=O)CCc2ccn(C)c2)s1 72135,C1(NC(CC2C(C)=NNC2=O)=O)CCN(C(=O)CNC(C2CCCC2)=O)C12CC2 72136,S(=O)(=O)(c1ccc(NCC23CCC(CC2)C3)c(F)c1)NCC1(C)CCOC1 72137,C(=O)(C(C)(C)C(=O)NC1CCC(CC(=O)N(C)Cc2ncnn2C)C1)NC 72138,N1(C(CCCOC)=O)CCCC2(C1)C(NC(c1nc(C)ncc1Cl)=O)CCN2C 72139,C(=O)(CC(C)(C)O)NCCCC(C)NC(=O)C(F)(F)c1ccccn1 72140,c1(CC(=O)NC(CN(C(c2c(CCC)n[nH]c2)=O)C)C)cccc(C)c1 72141,Cc1cc(C(C)(C)C(=O)N2CC(CC(C)NC(=O)C(C)CF)C2)cs1 72142,C1(NC(CC2CCN(C)C2)=O)CCCC(NC(=O)CC(C)(C)O)C1 72143,c1(C(=O)NCC(CNC(C(CN(C)C)(F)F)=O)CO)cc2nccnc2cc1F 72144,N1(C(c2c(CC)nc[nH]2)=O)CCC2CCN(C(=O)C#CC3CC3)CC2C1 72145,C1(NC(CN(CC)CC)=O)COCCC1NC(=O)C(CC)SC 72146,C1(C(N(CCC(=O)N(CCC=C)CC)CCN(C)C)=O)C2CC3C(C2)C13 72147,c1(C(C)NC(C2CC(NC(=O)C(C)CN3CCCC3)C2)=O)cc(Cl)c(Cl)c(Cl)c1 72148,C1(NC(C=CC(C)(C)SC)=O)C2CCC1N(C(=O)CCc1cn(C)nc1C)C2 72149,C(=O)(CC(C)(C)CC(F)(F)F)N(CC(O)CNC(C1(C2CC2)CC1)=O)C 72150,C(=O)(C1=COc2ccccc2O1)NC1CC(C)(C)N(C(=O)C=Cc2cncs2)C1 72151,Cc1sc(C(=O)N(C2CCN(C(=O)CCC3CCCCCC3)C2)CCO)nc1O 72152,Cc1cc(C#N)ccc1N1CCC(Cc2ccncc2)CC1 72153,CC1CC(C(N2CC(CN(C)C(C3(C(N)=O)CCC3)=O)C2)=O)CO1 72154,C(=O)(C(CC(F)F)c1ccccc1)Nc1cccc(NC(c2n(C)nnc2)=O)c1 72155,C(=O)(C1=CCCCC1)N(CCOC)CCNC(c1c(OC)noc1C)=O 72156,c1(C(CC)N(C(C(=O)OC(C)(C)C)c2ccsc2)C)ccc(Br)s1 72157,C1(NC(COc2cc(C)on2)=O)CC2CCC1N(C(c1cc(C)c(C)nn1)=O)C2 72158,N(C(=NCC1COCCO1)NCCNCC(F)(F)F)Cc1ccc(C(C)C)cc1 72159,CCC(O)C(C)(C)C(=O)N(CCCNC(C1CC(F)(F)CCC1(C)C)=O)C1CC1 72160,N1(C(C)C(=O)NCC(F)(F)F)CCN(C(C2CC=CC(O)C2)=O)CC1 72161,CCCC(C(=O)NC(C)Cn1cccn1)NC(=O)CN(C)CC1CCOC1 72162,N1(C(c2c(C)n(C(C)C)nc2)=O)CC2CC(C1)CN(C(C1CC(C)CO1)=O)C2 72163,N1(C(c2n(C(C)C)nc(C3CC3)c2)=O)C2CCC1CC(NC(=O)C(O)CF)C2 72164,N1(C(C(C)(C)OCC)=O)CCCC(CCNC(=O)CCC2(C)CCC(=O)N2)C1 72165,C1(C)(C(=O)NC2CN(C(CNc3ccn(C)n3)=O)C(CO)C2)CC2(CCC2)C1 72166,O=C(CC1=CCCCC1)NCCC12CCC1CN(C(C1CC(=O)NC(=O)N1)=O)C2 72167,C(CCCCNC(=O)CCN1CCOCC1)N(C(=O)Cc1nccn1C)C(C)C 72168,C(C(=O)NC(C(=O)NC1CC=CC1)C1CCC1)(C(C)C)OC 72169,c1(-c2cccc(CC)c2)ccc2c(c1)COC2.N12NN=NC1=NC(=O)C1(CC1)C2 72170,CC1CN(C(c2cc(C(N)=O)[nH]n2)=O)CCN1C(=O)Cc1ccccc1CC#N 72171,Cn1nc(CN2CCN(c3ccnc(NCCC(C)(C)C)n3)CC2)cc1COC 72172,N1(C(c2cccc(C)c2C)=O)CCC2CN(C(c3ccc(=N)[nH]c3)=O)CC12 72173,N1(C(CC2CC(C)(C)CN2C(c2ccc(C(N)=O)o2)=O)=O)CCOC2(CCC2)C1 72174,C(=O)(C(CC)C(=O)OCC)NCC1N(C(c2nn(CC)nc2C)CC)CC1 72175,C=CC(CC)CC(=O)N1CC(C(O)C(=O)NC(C)(C)CC2CCC2)C1 72176,c1(SC)sccc1C(=O)NCCN(C(c1cnoc1C1CCC1)=O)CC1CC1 72177,Cc1c(O)cc(C(N2CCC3(CC2)C(=O)N3)=O)cc1O.C1(CC2CC2)CC1C 72178,C=C1CCN(C(C2CCN(C(C)=O)CC2)=O)C(C(=O)NCC(C)(CO)CO)C1 72179,C1(CNC(Cc2cc(C)sc2C)=O)CC(C)(C)CCC1NC(=O)CCF 72180,N1(C(CC(C)N(C)C)=O)CCCC1(C)CNC(C1(C)CCOC1)=O 72181,N1(C(C2(OC)CCOC2)=O)CCN(C(=O)C=C(C2CC2)C2CC2)C(CC(F)F)C1 72182,C1(CNC(CC2(C(=C)F)CCC2)=O)CN(C(C2(CCC)CC2)=O)CCC1C 72183,C1(NC(C2C(C#C)C2)=O)CCN(C(=O)Cc2cccc(C)c2F)CC(C)(C)C1 72184,S(=O)(=O)(c1cc(C(=O)OC)c(Cl)cc1Cl)N1CC(C#C)(c2ccccc2)C1 72185,N1(C(c2c(OCC#C)nccc2)=O)CCN(C(c2csnc2Cl)=O)C(CCO)C1 72186,C1(NC(CCc2ccc(C)s2)=O)CCCN(C(c2cc(C)n(C(F)F)n2)=O)CC1 72187,CCC(C)CC(=O)NC1CCC1NC(=O)CC1(C)CC1 72188,C=CCCC(C(=O)NCC1CCN(C(c2ccc(=O)n(C)c2)=O)C1)c1ccccc1 72189,C1(C(=O)NCCc2nc(CC)[nH]n2)N(C(=O)C(O)CSC)CC12CCCC2 72190,N1(C(c2c(F)ncc(C)c2)=O)CC(N=c2[nH]nc(COC)s2)CC(C)(C)C1 72191,C(=O)(CCC(CC)CCC)NCC1C2CN(C(CC3(C=C)CC3)=O)CC21 72192,c1(CCC(N2C(C)(C3CC3)CCC2)=O)ccc(F)c(F)c1.c1cn(CCF)nn1 72193,c1(SCC(C)C2CC2)nccn1CCC1CCCCC1 72194,N1(C(c2cn(C)nc2)=O)CC(C)(C)CC1CNC(=O)C(O)C1CC1 72195,CC1(C)C(C(=O)NCc2ncc(C(F)(F)F)s2)CCN1CCF 72196,c1(C(=O)NCC23CC(NC(C(CCO)NC)=O)(C2)C3)n[nH]c(C)c1[N+](=O)[O-] 72197,N1(S(CCOC)(=O)=O)CCN(C(=O)Nc2cc(Cl)ccc2OC)C(C(F)(F)F)C1 72198,c1(C(=O)NCCCN2CCN(C(CCCOC)=O)CC2)cc2cccnc2[nH]1 72199,c1(C(=O)NC(C)CC2CC2)ccc(-c2ccoc2)c2cc[nH]c12 72200,C(=O)(C1=CCCC1C)NCCc1cc(C(N(CCn2c(C)ncc2)C)=O)no1 72201,C(CSC)(CN=c1[nH]c(C(=O)Nc2ccc(OCCN)nc2)cs1)OC 72202,N1(C(C2C(CCC)C2)=O)CCCCC1C(=O)NCC1(CC2CCC2)CCC1 72203,C1(C(C)C)C(NC(c2cc(C(F)F)cs2)=O)CCN1C(=O)C(C1CCCCCC1)C 72204,C1(CC=C)(NC(c2coc(Br)c2)=O)CN(C(=O)C2CC2)C1 72205,N1(C(CCCOC)=O)CCC2CCCC(C1)N2C(C1CCC2(CC2)C1)=O 72206,c1(C2CCN(c3cc(Nc4c(C)ncc(Br)c4)ncn3)C2)ccccc1[N+](=O)[O-] 72207,c1(C(=O)NC2CC(NC(C(C)OCCC=C)=O)C2)c(F)cncc1Cl 72208,c1(C(N2CCC(C)C(CO)C2)=O)cc(P(C)(C)=O)cs1 72209,N1(N2CCC2CC=O)CCN(C)C(CC)C1.c1(COCC)cc(C(=O)OC)no1 72210,C(=O)(CCCC(F)(F)F)NCCCCCCN(C(C(C)CC(F)F)=O)C 72211,c1(C(=O)NCC2N(C(C(n3c(C)cc(C)n3)C)=O)CCCC2)cn2ccsc2n1 72212,N1(C(c2c(C)noc2)=O)CC2CCC1C(C(=O)NC1CCCCC1(F)F)C2 72213,c1(C(N(C(CNC(COCCCCC)=O)CC)CC)=O)sc(COC)nc1C 72214,c1(C(N(CCCNC(c2cc(CC)sn2)=O)C(C)C)=O)ccn2ccnc2n1 72215,c1(C(=O)OC)cnc(=NCC2CCC(NC(C3CCNC(=O)C3)=O)C2)[nH]c1 72216,CC1CC(C(=O)NC2(C)CCN(c3ncccn3)C2)CCS1 72217,Cc1cc(C(=O)NC(CN(C)C)C(=O)NCc2ccccc2O)c(C)n1C 72218,c1(Nc2ccc(Cl)c(I)c2)cccc2c(Cl)ccnc12.c12ccccc1C(=O)S2 72219,CC(CC(=O)NOCCCCC(=O)NCCc1nccn1C)c1ccco1 72220,c1(C(=O)NCC2(F)CN(C(C3CC(CC)C3)=O)C2)cnn(CC(C)(C)O)c1C 72221,N1(C(c2cc(CC)ncc2)=O)CC2(CCCC2NC(C2CC2F)=O)C1 72222,c1(C(C2CC2)NC(=O)OC)c(C)cccc1C.N12CCC(CC1)CSCC2=O 72223,C(=O)(CC(C)C(=O)N1CCC(C(C)C(=O)N(C2(CC)COC2)C)C1)OCC 72224,C1(NC(=O)Cc2ccccc2)CN(C(c2cncc(Br)c2)=O)CC1C1CC1 72225,n1(CC(=O)NC(C(C)(C)C)CNC(=O)C(C)(C)c2cnco2)cc(F)ccc1=O 72226,C1(C)(C(=O)NCCCCCN(CC(C)C)Cc2ccsn2)CCCNC1=O 72227,Cc1oc(C)c(C(=O)NCC2CC(CNC(=O)COCCN(C)C)CO2)c1C 72228,Cc1ncc(Br)c(N(C2CCCNC2)C(c2ccc(O)cc2Br)=O)n1 72229,C12(NC(=O)COC3CCC3)CC(C(=O)NCCc3ccon3)(C1)C2 72230,c1(-c2c(C)cc(C)c(C)c2)nc2c(s1)CCN(C(=O)CC(C)O)C2 72231,C12(CNC(C3CC(C)C3)=O)CCC1CN(C(c1cc(C3CC3)ncn1)=O)C2 72232,CC(C(=O)N1CC(O)(CCNC(c2ccc(Cl)c(Cl)c2)=O)C1)S(C)(=O)=O 72233,c1(C(=O)NC2(CN(C)C(c3ccnnc3O)=O)CC2)cccc(CO)c1 72234,N1(C(C(CC=CC)CC)=O)CC2CN(C(c3ncc(Cl)n3C)=O)CC2C1 72235,C(=O)(C1CCc2cccnc21)NCCOC1CN(C(CS(CCCC)(=O)=O)=O)C1 72236,c1(C(N2CCC(O)(C(=O)NCc3ncccn3)C2)=O)ccc(C#CCO)cc1 72237,CCC(CNC(C1C(CC)CCN1C(=O)Cc1ccoc1C)=O)CC(C)C 72238,N1(C(COCC(C)C)=O)CCC(C2CC2)(NC(c2cnc(S)n2C)=O)C1 72239,N1(C(c2ccc(CCCC)cc2)=O)CC(C(=O)OC)Oc2c(C)cccc21 72240,c1(C(=O)NCc2ccc(C(=O)Nc3n(CC=C)ccn3)o2)ccnc(SC)c1 72241,C1(CC(=O)NCC2CCCN2C(=O)CNC(=O)C2CC2)NC(=O)CNC1=O 72242,C(CCN=C(NCC1(C)CCCCO1)NC1CC1)OC(CC)C 72243,CCC(CC(C)C)C(=O)NCC1=CCN(C(C2CC3CCCC(C2)C3)=O)CC1 72244,CCC(C)(COC)C(=O)NC1CCC(CCC(=O)NCC2(F)CC2)C1 72245,C(=O)(C1=NOC2(CCOC2)C1)NC1C(N(C(=O)CCCn2ccnc2)C)CCCC1 72246,c1(CN2CC(F)(C(N(C)C)=O)C2)ccc(CNc2ncccc2O)cc1 72247,C1(C)(NC(C(CC2CC2)OC)=O)CCN(C(C2CCC(C)(C)OC2)=O)CC1 72248,c1(N(CCN(C(C2CC23CCC3)=O)CC)C)nc2ccc(F)cc2s1 72249,C1(NC(C(CC)SC)=O)CC(C)(NC(=O)C(C)OC(C)=O)C1(C)C 72250,N1(C(=O)NCC2CC2)CCN(Cc2cccc(F)c2)C(CCO)C1 72251,N1(CC(C)C)CCNC(=O)C1C(=O)O.n12ccnc1C(=O)N1CCCC21 72252,CC(C(=O)N(CC(C)NC(=O)Cn1nnc(-c2ccco2)n1)C)S(N)(=O)=O 72253,N1(C(C2N(C(C3CCC(C)CC3)=O)CCCC2)=O)CCCC2(CCO2)C1 72254,c12ccccc1O2.C1(NC(CSCCCC)=O)CC(CNC(c2nc[nH]n2)=O)C1 72255,CC1CCCCC1CCNC(c1c(Oc2ccccc2)cnn1C)=O 72256,C1(NC(CCCOCC)=O)CCC(N(C)C(C2OCCC2C(C)C)=O)CC1 72257,C(CCCCCNC(=O)Cc1cccnc1O)N(C)C(C1(CO)CCCO1)=O 72258,CC(C(CO)NC(C1CCCC1)=O)NC(=O)CN(C(=O)CC1CCCO1)C1CC1.CC 72259,C1(NC(C2CCC(C)C2)=O)CN(C(=O)CCc2ccc(F)nc2)CC2(CC2)C1 72260,C(=O)(C(C)(CO)NC(=O)CCc1ccncc1)NCC(C)(C)OCCO 72261,C1(NC(C(C2CCC2)OCC)=O)C2CCCN(C(C3CCC(=O)N3)=O)C2C1(C)C 72262,C1(NC(c2ccc(Cl)[nH]2)=O)CCC(CCNC(c2ccnn2C2CCC2)=O)C1 72263,c1(C(N2CC(C)C(NC(c3cn(C)c(=O)cn3)=O)C2)=O)ccc2ncnn2n1 72264,c1(CCC(=O)NCC(CNC(CCC2CCN(C)CC2)=O)O)cccc(F)c1Cl 72265,N1(C(C=C(C)Cl)=O)CCC(C2CCOCC2)(CNC(C2CCCCNC2=O)=O)C1 72266,c1(C(N(C2CCN(C(=O)C(COC)COC)C2)CC)=O)nn(C)c(C)c1Cl 72267,c1(C(N(CCC)CCNC(=O)CC2CCCC(O)C2)=O)c(C)[nH]c(C)c1C 72268,S(=O)(=O)(c1ccccc1F)NCC1N(C(c2ccc(Cl)c(Br)c2)=O)CCC1 72269,c1(CC(=O)N(C2C3CCC2CNC3)c2cccc(Cl)n2)cc(F)cc(F)c1F 72270,C12(C(N3CC(CN4CCN(C(c5cncnc5)=O)CC4)C3)=O)CCCC1CCC2 72271,C1(CC(N2CC(N(C(=O)CC)C)C2)=O)NC(=O)NC1=O.CC(C)C(O)C1(CO)CC1 72272,C(=O)(CCP(C)(C)=O)NC1CC(NC(C(C)CN(C)C)=O)CC1O 72273,c1(C(=O)OCc2c(F)ccc(F)c2Br)cc(I)ccc1[N+](=O)[O-] 72274,n1(CC)nnnc1C1(NC(C2CSC2)C)CCC1CS(N)(=O)=O 72275,N1(C(C2CN(C(C(C)OCC(C)C)=O)CC2(C)C)=O)Cc2ccncc2C1 72276,Cc1cccc(CCC(=O)NCC2CC2CNC(C2CCCS2(=O)=O)=O)c1 72277,N1(C(CC2N(CC)C(=O)CC2)=O)CC2CC1CN2C(c1sc(COC)nc1C)=O 72278,N1(C(C(C)=CC)=O)CCC(CNC(=O)C=Cc2cccc(CO)c2)C(F)(F)CC1 72279,c1(C(=O)NCC2CCN(C(CCC3C(C)C3)=O)C2(C)C)ccc2c(c1)ncn2C 72280,Fc1cc2c(cc1CN1CCC1CC1CC1)OCCCO2 72281,c1(C(N2C(C)CC(NC(C(CC(C)C)NC(C)=O)=O)C2)=O)cc(C)nc(Cl)c1N 72282,Cn1cc(Br)nc1CN1CCSCC1C(=O)NC(c1ccc(F)cc1)CCO 72283,C(=O)(C(Cc1cn(CCC(F)F)nn1)CC(F)(F)F)N1CC(CCOC)OCC1 72284,c1(N2CCC(C)(CC)C2)nc(=N)nc(N2CCC(CCN(C)C)C2)[nH]1 72285,C(=O)(CC1=NN(C)C(=O)C1)N1CCC(C#C)(C(N2CCOC(CC(N)=O)C2)=O)C1 72286,N(C1CCc2ccc(Cl)cc21)S(CCCC)(=O)=O.c12cc(ncn1)N1CCCC1N2 72287,c1(C(=O)NC(C2(O)CN(C(c3ccccc3Cl)=O)C2)C)ccc([N+](=O)[O-])s1 72288,c1(C(=O)NCCC2(C(=O)Nc3c(C)cc(F)cc3)CCC2)cc(F)c(F)c(F)c1 72289,C1(CNC(C(F)=CCC)=O)CN(C(=O)C(F)C(C)C)CC1C(F)(F)F 72290,c1(C(N2CC(NC(CCNC(N)=O)=O)C3(C2)CC3)=O)cccc2c[nH]nc12 72291,CC1(C)CN(C(=O)CSc2ncccn2)CCN1C(c1ccnc(Cl)c1F)=O 72292,C1(CN(C(=O)COC(C)(C)C)C)CCN(C(=O)CCN2CCC(F)C2)CC1 72293,c1(CN2CCCC(NC(c3cccc(Br)n3)=O)CC2)c(Cl)cc(F)cc1Cl 72294,C(CCC(C)C(=O)NCc1cc(N)on1)N1CC(OCC(N)=O)C1.CO 72295,C1(NC(c2c(C)c(N)n(C)n2)=O)CN(C(=O)C(O)CC(C)C)CCC12CCC2 72296,N1(C(C(C(=O)OC)(C)F)=O)CC(NC(=O)COC(F)(F)F)C2CCCC12 72297,N1(C(COCCC(C)C)=O)CCN(C(C2CC2CCOC)=O)CC1CO 72298,C(=O)(C(C)(C)CCC(=O)OC)N(C(CC)C(=O)NCC(=O)NC)C 72299,c1(C(N(C)CC2CCN(C(c3c(C)occ3)=O)C2)=O)ncc2ccccc2c1O 72300,c1(C(=O)NCCN(CCOC)C(c2cc(F)n[nH]2)=O)c[nH]nc1S(N)(=O)=O 72301,N1(C(C2CC(N(C)C)C2)=O)CC2(C(N3CC(C(N)=O)C3)=O)CC1CO2 72302,N1(C(C2C(=C)C2)=O)CC2CN(C(=O)CN(C)S(N)(=O)=O)CC2(C)C1 72303,c1(C(=O)NC(C(C)C)CCN(C(=O)C(C)O)C)c[nH]c2c(Br)cccc12 72304,CCCCC(=O)NNC(=O)C(C)NC(=O)C(C)Oc1ccccc1 72305,CC(CC(=O)N1CCCC1(C(=O)O)Cc1cn(C2CCC(C)(C)CC2)nn1)C(F)(F)F 72306,C1(CNC(C2CC=CCO2)=O)CN(C(=O)C(c2ccc(F)cc2)(F)F)CC1(F)F 72307,CCN=c1[nH]c(C(=O)NCC(C2CCC2)NC(=O)Cc2nnnn2CC)cs1 72308,c1(CNC(CC=C)=O)ccnc(C(=O)NCC2C=CCCC2)c1 72309,C1(NC(c2cc3n(n2)CCC3)=O)CCC2(CC1)CN(C(=O)C(F)OC(F)(F)F)C2 72310,C1(CNC(c2c(CC)n(C)nc2)=O)CN(C(=O)C(C)c2ccsn2)C2(CCC2)C1 72311,C1(C(=O)NCCCOCCNC(C2CCS(=O)(=O)C2)=O)Cc2nncn2CC1 72312,C1(NC(C(c2cccc(C)c2)C)=O)CC(F)CN(C(c2cn(C(C)C)cc2C)=O)C1 72313,CCC1=NOC(C(=O)NCCCCN(C(=O)Cn2cncn2)C(C)C)C1 72314,c1(CC)cc(Cl)cc2cc(C(=O)NC3(c4nnnn4C)COCC(SC)C3)[nH]c12 72315,c1(C(=O)NCC(CC=C)NC(=O)CCCCC#N)ccc2c(c1)CCS2(=O)=O 72316,CC(CC(C)(C)NC(C1C2CC3C(C2)C13)=O)NC(=O)C=Cc1nccs1 72317,N1(C(CS(CC)=O)=O)CC2CC1CN(C(C1(Cc3ccccc3Cl)CCC1)=O)C2 72318,c1(C(=O)O)ccc(=NCC2CC2c2ccccc2)[nH]c1 72319,C1(CC(N2CCC(NC(c3c(N)ccc(C)c3)=O)C2C)=O)CCn2cncc2C1 72320,c1(C(N(CC(C)NC(C(CC)OC)=O)C)=O)cnc2c(c1)CNC2=O 72321,C1(CNC(CC(C)C)=O)CCN(C(=O)CCc2ccc(F)cc2)C1(C)C 72322,c1(C(CCC)NC(=O)NC(c2ccccc2)c2cc(C)[nH]n2)cccc(F)c1F 72323,C=CCCCCCC(=O)NC(C)(C)CNC(=O)C(c1ccc(Cl)s1)C 72324,N1(C(CCc2n(C)ncc2)=O)CCC2CCN(C(c3cn(C)c(=O)cn3)=O)C2C1 72325,C(=O)(C(C)(C)CC(=O)OC)NCC(CC(=O)NC(CC=C)C1CC1)OC 72326,c1(C(=O)NCC2C(NC(CC(C(C)(C)C)O)=O)CCC2)sc2ccccc2c1Cl 72327,CCC(C(=O)NCCCN(C(=O)CC1(C)CC1)C)C(F)(F)F 72328,CC1OC(C)CC1CC(N1CC(CC(C)NC(=O)CCC2CCOC2)C1)=O 72329,N1(C(C(=O)O)c2ncco2)CCN(C(C)=O)CC1(C)C.c1(OCCOC)ccccc1O 72330,c1(C(=O)NCCN(C(=O)C(F)C2CC2)CC(C)O)c[nH]c2cccc([N+](=O)[O-])c12 72331,CC(O)C(F)(F)C(=O)OC(C)(C)C.C1CCCN(C)CCN(C)CCC(=O)O1 72332,C(=O)(C1CCCc2cncn21)NC(C)(CNC(C1CCCC1)=O)C1CC1 72333,C(CN=c1[nH]c2c(c(=NC(C)CC(=O)NC(C)C)[nH]1)CCCC2)c1ccc(C)cc1 72334,N1(C(C2C(OC)CCC2)=O)CC(=O)Nc2ccccc21 72335,C1(C(=O)NCC2(C)CCN(C(C=C(COC)C)=O)CC2)COc2ccccc2O1 72336,N1(C(C(C)=CC)=O)CC2(CCN(C(c3ccc(=O)n(CCF)n3)=O)CC2)C1 72337,c1(CC)cc(F)c(C(=O)NCCC2(NC(c3ccccn3)=O)CCC2)cc1F 72338,N1(C(c2n(C)cc(C#N)c2)=O)CCCC(C2CN(C(C3CC34CC(O)C4)=O)C2)C1 72339,C1(C(N2C(C(C)NC(=O)COC3(C)CCC3)CCC2)=O)CCc2c[nH]nc2C1 72340,N1(C(C=Cc2scc(C)n2)=O)CCN(C(C2CCCO2)=O)CC2(CC2)C1 72341,N1(C(C(=O)NC(=O)NCC)C)CC2CCCN(C(c3oc(C)nc3C)=O)C2C1 72342,C(=O)(C(C(C)(C)C)c1cc[nH]n1)N(CC)CC1CCC(C(=O)O)C1.n12cc(nn1)C2 72343,C1(NC(C(n2c(C)ccn2)C)=O)CCN(C(c2c[nH]nc2C(F)F)=O)CC1 72344,c1(C(N2C3C(NC(C4(CN(C)C)CC4)=O)C(C3)C2)=O)cccc2occc12 72345,N(C(=NCNCc1cn(C)nc1C1CCC1)NCc1snnc1CC)C(C=C)C 72346,c1(CC)oc(C(=O)N(C)CC2COCCN2C(C23CC(F)C2C3)=O)cc1C 72347,S(=O)(=O)(c1ccc(C(=O)NCCC(O)CCO)cc1)N(CC=C)C 72348,N1(C(Cc2nc(C)sc2)=O)CCC(CO)(NC(C2CCC(C(C)(C)C)O2)=O)C1 72349,C(CC(=O)NOCCC(F)F)C(F)(F)F.CC1CC(C2CC(=O)N2)=N1 72350,N1(C(C=C(C)C2CC2)=O)CCN(C(=O)CC23CCC(CC2)C3)CC1C1CC1 72351,c1(C(=O)NCC2CCN(C(C(C)(C)C3CCOC3)=O)C2)cncc(P(C)(C)=O)c1 72352,CC1=NOC(C)(C(=O)NC2CCC(CCNC(=O)CCC=CBr)C2)C1 72353,c1(NC(CC2(C)CN(Cc3cccc(C(=O)O)c3)C2)=O)cncc(Cl)n1 72354,C(C#CCNC(C1(C(F)(F)F)CC1)=O)NC(COC(C)=O)=O 72355,N1(CCN(C)C)CCC(N=c2[nH]c(N3CC4CC3C(F)(F)C4)nc(=N)[nH]2)CC1 72356,C1(C2CCC2)(C(=O)NCCCCN(C(c2cnn(C(C)C)n2)=O)C)CCC1 72357,C1(CNC(C(Cn2ccc(C)n2)C)=O)CN(C(c2nnn(C)c2N)=O)CCO1 72358,N1(C(=O)NCC(CC#C)OC)CC(CC#C)N(C(=O)OC(C)(C)C)C(C)(C)C1 72359,c1(C(=O)NC(C)(C)CN2CCN(C(=O)C(Cl)=CCl)CC2)ccc(N)cc1.Cc1nc[nH]n1 72360,N1(Cc2cccc(CNC(=O)OC(C)(C)C)n2)CC(CO)CCC1(C)C 72361,C1(NC(C(C#C)(C)C)=O)C2CCN(C(=O)C(C)CC(=O)c3ccc(F)cc3)CC12 72362,C1(C(N(C2CC(NC(C(CC)COC)=O)C2)C)=O)CN2CCC1CC2 72363,c1(C(N2CCCC(N(C(CC(C)N(C)C)=O)C)CC2)=O)ccn2c1CCCC2 72364,CC1OCCOC1C(N1CCOCC1CC(=O)NCC1(C)CC1(F)F)=O 72365,C(C)(CCC(=O)N1CCCC1C(C)NC(C12CC(CCO1)C2)=O)OC 72366,N1(C(C2CC(Oc3ccccc3)C2)=O)CC2ON=C(C(F)F)C2C1 72367,CCC(C)C(C(=O)NCCCCCCNC(=O)CN(C)S(N)(=O)=O)NC(N)=O 72368,CCC(CC)(CO)C(=O)N1CCC(NC(C2CCn3cncc3C2)=O)CC(O)C1 72369,Cc1nccc(C(=O)NCc2ocnc2C(=O)NC(C)C(N)=O)c1N 72370,N1(C(C2(C)CC=CCC2)=O)CC2=C(C1)CN(C(=O)CCOCC1CC1)C2 72371,C(CC(C(=O)NC1(C)CCCC1C)NC(=O)C(F)C(C)C)OC 72372,C1(CC)CCN(C(=O)C=CC(=O)NCC=CCSC)C(C(=O)NC)C1 72373,c1(C(=O)NCC2OCCN(C(C(C)(C)Cc3ccccc3)=O)C2)cc2scnc2[nH]1 72374,C1(CNC(C(C(C)C)NC(N)=O)=O)C2CCC(C2)N1C(=O)C(C1CC(F)(F)C1)O 72375,C1(N(C(Cc2ncc(C)o2)=O)C)CN(C(=O)CC2CN(C)C2)CC1F 72376,CC1(C)OCCOC1C(N1CCC(CO)(CNC(=O)CC2SC(=N)NC2=O)C1)=O 72377,CS(=O)c1ccc(C(CO)NC(c2ccccc2)C2CCC2)cc1 72378,c1(CNC(C2(NC(C3CC3C(F)(F)F)=O)C(C)(C)C2)=O)ccccc1O 72379,CCC(CC(=O)N1CCC(NC(C23CC(C)(CO2)C3)=O)C1C)C1CCC1 72380,C1(C(C)NC(C2C(=C)C2)=O)CCN(C(=O)CC2CC3CCC2O3)CC1 72381,C(=O)(CCC1=CCCCC1)NCC12N(C(CCCC#CC)=O)CC(CC)(C1)C2 72382,c1(CC(=O)NCC(C)NC(=O)CCc2ccc(Cl)nc2)cccc(F)c1F 72383,C1(NC(C2CCCC23CC3)=O)CC12CCN(C(c1ncc3[nH]ncc3n1)=O)CC2 72384,c1(N(C)CC2CCCCN2C(C2CCOC(C)C2)=O)c(C#N)cccc1[N+](=O)[O-] 72385,C(c1cn(CC2CCCN2C(=O)CCNC(C2C(C)C2C)=O)nn1)=CC 72386,C1(CC)CCC(C)N1C(=O)C(C)N(C(c1cc(O)nn1C)=O)CC 72387,N1(C(COCCCOC)=O)CCCC(NC(=O)CCCc2cccc(Cl)c2)C1 72388,C1(NC(c2[nH]cc(C)c2)=O)CN(C(c2cccc(CC#N)c2)=O)C2CCCCC12 72389,C1(OC)CC(CO)N(C(=O)C(=O)NC2(C(=O)O)CCC(C)C2)C1 72390,N1(C(=O)OC(C)(C)C)CCC2C1CCCN2C(c1cc(Br)cc2nc[nH]c12)=O 72391,C(=O)(CC(C)C(=O)OC)NCCC1(O)CCN(C(C2(OCC)CCOCC2)=O)C1 72392,C1(C2CN(C(=O)C(C)(C)C3CCCC3)C2)(NC(Cc2c(C)n[nH]c2)=O)CC1 72393,C1(CN(C(=O)COCC2CCCCO2)C)CCCCN1C(c1cc[nH]n1)=O 72394,c1(C(=O)NC2(CCCNC(CCC(=O)OCC)=O)CC2)cnc(C)cc1Cl 72395,Cc1nn(C)cc1CCC(=O)NC(C1CCCN1C(=O)CC1CC2CCC1C2)C 72396,C1(NC(c2c(C)sc(Br)c2)=O)CC2CC1CN2C(=O)C=C1CCC1 72397,Cc1ncnc(O)c1CCC=O.C1(C(N(C(C)CNC(N)=O)C)=O)CCC2(CCC2)C1 72398,CCN=C(NC)N1CCC(C)(C(N)=O)C1.CC1CN(C(=O)OC(C)(C)C)CC(C)O1 72399,C(C)(C)(C(C)CC(=O)NC1CCN(C(C)=O)C1)NC(C=CC=CCC)=O 72400,c1(C(=O)NCC2(OC)CN(C(C3(CN4CCCCC4)CC3)=O)C2)nc(C)sc1C 72401,C(=O)(C(O)(C(F)(F)F)c1ccccc1)N1CCC(CCNC(C2(F)CC2)=O)C1 72402,C(=O)(C1CCCc2n[nH]cc21)NCCCC(C)NC(C1CC1(F)F)=O 72403,N1(C(C(C=C)O)=O)CCC(F)(F)C(CNC(c2cc(-c3ccco3)n(C)n2)=O)C1 72404,Cc1nnc(N(c2cnn(-c3cccc(Cl)c3)c2)C(C2CC2(F)F)=O)nc1C 72405,c1(N2CCN(C(CCC)=O)CC2)cc(C)nc(C)c1[N+](=O)[O-] 72406,C1(C(=O)NCC2(N(C)C)CCC2)CC2CN(C(c3ncn(C)n3)=O)CC2C1 72407,C1(C(=O)NCC(C)(C(C)C)NC(C2N(CC(C)C)CCC2)=O)CN(S(N)(=O)=O)C1 72408,N1(C(C#CC2(CC)CC2)=O)CCCC2CN(C(C3(CO)CCC3)=O)CC12 72409,S(=O)(=O)(C1CN(C(c2cc(CO)[nH]n2)=O)C1)N1CCN(C(CC(=O)OCC)=O)CC1 72410,Cc1c(C(=O)NC2CCOCC2NC(=O)Cc2cncnc2)c[nH]c2nccc1-2 72411,CCC(C)C(O)CC(=O)N1CCOC(CC(=O)NCC(C)(F)C(C)(C)F)C1 72412,c1(C(N2CCC(CNC(=O)CN3CCC(O)CC3)C2)=O)cccc(Cl)c1Cl 72413,N1(C(C(C=C)OC)=O)CCN(C(c2cc(C(C)=O)on2)=O)CC1C 72414,N1(C(C=CC=CC)=O)CCC(NC(c2cn(CC(F)(F)F)nc2C(C)C)=O)C1C 72415,c1(OC)nc(Cl)ccc1C(=O)OC(c1nc(-c2ccncc2)no1)C 72416,N1(C(CSCC#C)=O)CCCC(C(C)(C)C(=O)NCc2cnn(CCC)c2)C1 72417,C1(NC(C(CC)(F)F)=O)CCN(C(=O)C(c2ccc(Cl)cc2)=O)CC12CCC2 72418,C(=O)(C(F)(F)C(F)(F)F)N1CC(N(C(=O)Cn2ncc(O)nc2=O)C)C(F)C1 72419,C1(C(=O)NCC(C)C(=O)NCC(O)CN(C)C)CNC(=O)CC1C 72420,c1(C(N2C3(CN(C(Cc4c(C)noc4C)=O)C3)CC2)=O)ccc([N+](=O)[O-])c(F)c1 72421,n1(CCC(=O)NC2C=CCN(C(CN(C)CCO)=O)C2)nc(O)c2ccccc12 72422,C1(C(N2C(C)(CN(C)C)CCC2)=O)CC2CCCC2N1C(=O)C1=C(C#N)CCC1 72423,N1(C(C(C2CCCOC2)NC)=O)CCC(Cc2cn(C)nn2)CC1 72424,N1(C(Cc2nnc(C)o2)=O)CCN(Cc2cccc(C)c2O)C2CC12 72425,C(=O)(CCCC(=O)NCC1CCCCN1CC(F)F)NC.C12CN(CCO1)C2=O 72426,N1(C(c2nc(C)n(-c3nc[nH]n3)n2)=O)CC2CC1CN(C(C1CCC(=O)O1)=O)C2 72427,C(=O)(CS(N)(=O)=O)NC1CC(C(N2C(C(C)O)CC2)=O)C1 72428,N1(C(C(=O)NCCC(C)c2ccco2)=O)CCC(NCC(F)F)CC1 72429,C(C(CC)(CC)C(N)=O)NC(C(CC(=C)C)NC(=O)Cn1cnnc1)=O 72430,N1(C(C(C(C)C)SC)=O)CCCn2cc(Br)cc2C1 72431,c1(SC)cc(NNC(=O)NC2COC3(CCNCC3)C2)ncn1 72432,CCCC(CNC(=O)C=C(C)C(C)C)C(=O)NCC(Cl)=CCl 72433,n1(CCOC)nc(-c2cccc(COC(C)(C)C)c2)nc1C12CSC(C1)C2 72434,CCC(C)C(=O)C(=O)NCCN(C(C1CCCC1C)=O)C1CC1 72435,C1(NC(C(C)CO)=O)CCC2(CC1)CN(C(c1coc(C3CCOCC3)n1)=O)C2 72436,Cc1cc(C(N2CCCOC(CNC(=O)CC(C)(C)O)C2)=O)cc(C)c1F 72437,c1(CC(=O)NCC(CNC(C(C)OCC(C)C)=O)CO)ncc(F)cc1F 72438,C(=O)(C1=NOC2COCC12)N1CC(CC)C(NC(=O)Cc2ccc(Cl)cc2F)C1 72439,c1(NC)ccc(NC(=O)NCCc2ccccc2CS(C)(=O)=O)c(Cl)c1 72440,C1(C(=O)NCC2(C)OCCN(C(C=CC=CC)=O)C2)CCCCN(C)C1=O 72441,C1(C(=O)NC(CNC(c2c(SC)csc2)=O)C2CC2)CCCCCCC1 72442,N1(C(C=CCCC)=O)CCCC2(CC(NC(c3cc(Cl)ccc3NC)=O)CO2)C1 72443,C1(NC(CC=C)=O)CC2(CCN(C(c3cc4sccc4cn3)=O)CC2)C1 72444,N1(C(C(C)=CC)=O)CCCC1CNC(c1nc[nH]n1)=O 72445,N1(C(C2CC(O)(CC#C)C2)=O)CC(C2CN(C(c3nccc(Cl)c3F)=O)C2)C1 72446,N1(C(c2cc(C)cc(F)c2)=O)CCC2(CC2)CC1C(=O)NC(C)C(C)(C)O 72447,c1(C(=O)NCC(C)NC(Cc2c(C)cco2)=O)cc2c(n1C)CCOC2 72448,C(=O)(CC(CC(C)C)NC(c1cc[nH]c1C)=O)Nc1cn(CC#C)nc1 72449,N1(C(c2ccc(OC)cc2O)=O)CC(C2CC2)C(F)(C(=O)O)C1 72450,C1(C(N2CC(NC(c3c(CC(C)C)cccc3)=O)C(O)C2)=O)CCN(C)S1(=O)=O 72451,C1(CC(=O)NCCc2cocn2)CCCN(C(=O)C=CCN2CCCC2)CC1 72452,c1(C(=O)NCCN(C(c2c(C)cc(C)o2)=O)C)ccc2c(c1)NC(=O)CNC2=O 72453,C=C(C)C(C)(C)C(=O)NC1CCCC(CN(C)C(c2ccc(CC)[nH]2)=O)C1 72454,C1(CNC(CSS(C)(=O)=O)=O)CN(C(C2(C)CC(F)C2)=O)CC12CCC2 72455,C1(NC(C2C=CCN2)=O)CCNCC12CC2.c1(-c2ccccc2)cccc(SC)n1 72456,c1(C(=O)NCC2(F)CN(C(c3cn(CCC=C)nn3)=O)C2)nccc(Cl)c1C 72457,Cc1cnc(C(=O)NC2CC(N(C)C(c3cnc(C)[nH]c3=N)=O)C2)c(C)c1 72458,C1(CNC(CC2N(C(CC3C(CC(C)C)C3)=O)CC2)=O)OCCC1(C)C 72459,S(=O)(=O)(c1cccc(C(=O)OC)c1)N(C(CC)C(C)O)Cc1ncccn1 72460,c1(C(=O)NC2CC3(CN(C(Cc4c(C)noc4)=O)C3)C2)cc([N+](=O)[O-])ccn1 72461,N1(C(CCCC#C)=O)CCOCC(NC(=O)CC(C)Cc2ccc(F)cc2)C1 72462,C1(C(=O)NCC2(O)CN(C(CNC(C(CC)C)=O)=O)C2)CNC(=O)C(C)(C)C1 72463,CC(C)C(F)(CNC(=O)C=CC(C)(C)C)C(=O)NC(C)C(=O)NC1CC1 72464,C(=O)(C(C)(C(=O)N1CCCCC1c1cccc(Cl)c1Cl)CC)OCC 72465,c12ccc(c(N3CCOCC3)c1)s2.C(c1cnc(OC)s1)=C(CC)C 72466,c1(CC(C)C)ccc2c(N)c(C(=O)NCc3cc(C(C)(C)O)ccn3)sc2n1 72467,N(C1COc2cc(Br)cc(C)c21)C(=O)Nc1ccc(-n2ccc(C)n2)cc1N(C)C 72468,C=CCCC(C(=O)NC1CCCN(CC2CCC2)C1)CC 72469,N1(Cc2nc(CCC(=O)OC)on2)CCCC(n2cc(C(=O)O)nn2)CC1 72470,c1(C(=O)Nc2n(C)nc(CC)c2I)nn2c(C)cc(C)nc2c1C 72471,CC1C(C)N(C(C23CCC(CC2)OC3)=O)CCN1C(=O)CNC(=O)CN(C)C 72472,C1(N)(CNC(C2C(c3c(C)ccc(C)c3)C2)=O)CCCC(C)(C)CC1 72473,c1(C(=O)Nc2n(C)nnc2)cnn2cccc(-c3cc(OC(C)(C)C)ccc3F)c12 72474,c1(C(=O)NCCC2CC(NC(CC#N)=O)C2)ccc2c(c1)S(=O)(=O)NC2 72475,C(=O)(C(C)(C)CCC#N)OC1C(OC(C)(C)C)COC1 72476,c1(C(CCCN(C)Cc2cc(C3CCCCC3)on2)=O)ccc2c(c1)OCCCO2 72477,C(=O)(C(C)(C)CNC(=O)CC1(NC(=O)CSC)CN(C(=O)C(C)(C)C)C1)OC 72478,C1(C(C)C)CCC(C)CC1NC(=O)NCc1nncc(Cl)c1Cl 72479,C(=O)(NN1CCCC1C(=O)NC1(CF)CCC1)C1CC(OC)C1 72480,c1(OC)cc(C2(C(=O)NCC(C)(O)CNC(C3CC(F)C3)=O)CC2)ccc1C 72481,c1(C(=O)NCCCCCNC(c2ccc(SC(C)C)cc2)=O)ccnc(F)c1N 72482,N1(c2cncc(C(N)=O)c2)CCCCC(NC(c2ccco2)=O)CC1 72483,c1(CCC(=O)NC2CCC(CNC(C3(C)CC3)=O)C2)cc(Cl)ccc1Cl 72484,n1(CCC(=O)NC(C(C)C)c2ncc[nH]2)cc(CNS(N)(=O)=O)nn1 72485,CCC(C)(O)CCNC(C1(NC(C2C3CCCOC23)=O)CCSC1)=O 72486,Cc1ccc2ncc(C(N3CCCC(CNC(C4CCNC(=O)C4)=O)C3)=O)n2c1 72487,c1(CN2CC(O)(CC(=O)NC3CCCCO3)C2)cccc2c1oc1ccccc21 72488,C(=O)(CCCCCF)NC1C(C)CN(C(c2cnc(C(C)(C)C)[nH]2)=O)C1 72489,C1(C(N2CC3C(NC(Cc4c(C)n[nH]c4C)=O)(C3)C2)=O)CCCCCN1C 72490,CC12CN(C(=O)Cc3ncc(Cl)s3)CC1CN(C(c1coc(C(F)F)n1)=O)C2 72491,c1(C(C)NC(=O)NCc2n[nH]c(O)n2)cccc(-c2cnn(C)c2)c1 72492,C1(NC(c2c(OC)nsc2)=O)CCCC(CNC(=O)Cc2c[nH]nc2O)C1 72493,C(CNC(c1cncnc1)=O)(C(C)C(C)C)NC(CCCC=C)=O 72494,c1(CCCCC)cc(C(N2CC(CO)(NC(=O)C(C)CSC(F)(F)F)C2)=O)n[nH]1 72495,c1(N2CCCC(CNC(c3n(C)ncc3)=O)CC2)ncnc2c1ncn2C1CC1 72496,N1(C(C(C)=CC2CC2)=O)CCC2(NC(c3conc3C)=O)CC2C1 72497,C1(N(C(C)C)Cn2cncn2)CCN(C2CN(S(C)(=O)=O)C2)CC1 72498,c1(C(=O)NCC2(F)CC(CNC(C(CC(=C)C)C)=O)C2)cncc(S(C)(=O)=O)c1 72499,c1(C(=O)NCC2N(C(C3CCC(C)(C)CO3)=O)CC2)c(Cl)cccc1[N+](=O)[O-] 72500,c1(C(=O)NCCN(CCOC)C(C23OCCCC2C3(F)F)=O)cc(Cl)ccc1F 72501,N1(C(C2(CC=C)CCN(C(c3cnn(C)c3OC)=O)C2)=O)CCC(C2CC2)C1 72502,CC(C)CCCCCC(=O)NC1CC1C(=O)NC1(CO)CC(C)(C)C1 72503,C(=O)(C(C)(C)C1CCC1)N(C1CC(NC(CCSCCC)=O)C1)C 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72572,c1(C(N(CC(CC)NC(=O)CNC(C)=O)C)=O)cc(Br)cc(C)c1F 72573,C1(CNC(C2N(C(CSC)=O)CC=CC2)=O)CCCC2(CC2)C1 72574,C12(CNC(C=Cc3c(C)ccnc3)=O)CCC(CN(C(=O)C(O)CN(C)C)C1)C2 72575,C1(C(N2CC=C(C(=O)OC)C2)C(=O)NC2CC2)CCCCC1S(C)(=O)=O 72576,C1(C(=O)Nc2cccc(OC)n2)CCN(C(c2cncc(F)c2)=O)CC1O 72577,N1(C(C(CC)C#N)=O)CC(NC(=O)COc2cc(OC)ccc2F)CC(F)(F)C1 72578,CCC(O)CCNC(=O)COc1ccsn1 72579,C1(NC(C2C(C)C2)=O)CC12CCN(C(c1ccc(C(F)F)cn1)=O)C2 72580,N1(C(C2C(OC)CC2)=O)CCCC2(NC(c3coc(C(C)C)n3)=O)CC2C1 72581,c1(C(N2CCC(C)C2)=O)c(CNC(c2cc(Cl)cs2)=O)cnn1C 72582,c1(NC2CC2NC(=O)NCc2ccnc(NC(=O)OC)c2)nccc2cc[nH]c12 72583,c1(CNC2C(C)CN(C(c3cc(Cl)ncc3F)=O)C2)cccc(F)c1C#N 72584,C(C(CC)CC)(C1CCCOC1)NCc1cccc(OCC=C(C)C)c1 72585,C1(C(=O)NC(CCCNC(C(C)Cc2cnc[nH]2)=O)(C)C)CCCC(=O)N1C 72586,C(=O)(C1=CCC(NC(=O)CCCC2CCC2)C1)NC1C(CCOCC)C1 72587,C(=O)(C1CCOc2ccccc21)NC1C2CN(Cc3c(C)[nH]c(C)c3C)CC21 72588,c1(CN(c2ncccc2N)C)cn2c(n1)CN(Cc1cc(Cl)c(Cl)c(Cl)c1)CC2 72589,C(C)(C)(CC(=O)N1CC(C#N)(C(N)=O)C1)N(C(CC(C)n1cccn1)=O)C 72590,N1(CC(=O)N(C(C)CNC(C2CC23CCOC3)=O)C)CCS(=O)(=O)CC1 72591,N1(C(c2cnc(C)n2C)=O)CCN(C(=O)CCN2CCCC2)CC1CO 72592,CCC(CC)C(C)C(=O)NC(COC(C)C)C(=O)Nc1ccc(F)cc1C 72593,CN1CCC(C(=O)NC2CC2NC(=O)C=Cc2cccc(CO)c2)S1(=O)=O 72594,c1(C(=O)NCC2CCCN2C(=O)CN2CCCC2)ncncc1Cl 72595,N(C1CC2(CN(C(C3CC(C)N(C)C3)=O)C2)n2ccnc21)C(C(C(=C)C)(C)C)=O 72596,O=C1CCC(NC(C2CC=CCC2NC(C2CC3(CCC3O)C2)=O)=O)C(=O)N1 72597,N#CC1CCCC1NC(C1CCCN1C(=O)CCC1CCC(=O)C1)=O 72598,C(CCCCC(=O)N(C)C)NC(c1c(C)nccc1)c1nnnn1C1CCC1 72599,C1(NC(C(=C)F)=O)CCN(C(c2cc(Br)ccc2OC(F)(F)F)=O)CC1F 72600,Cc1nc(O)sc1C(=O)NCCC(C)N(C(=O)CC(C)N(C)C)C 72601,CN1C(=O)CN(CC(N2CCN(C3CN(C(=O)C4=C(Cl)CCC4)C3)CC2)=O)C1=O 72602,c1(NC(NN(C)CC2CC(N3CCOCC3)C2)=O)ccc(NC(=O)NC(N)=O)nc1 72603,S(=O)(=O)(CC(=O)OC(=O)Cc1ccc(C(F)F)o1)NCC 72604,c1(SC(C(NOC(CCC)CC)=O)C)cnc(N)c([N+](=O)[O-])c1 72605,Cc1c(C(=O)NCC2(NC(C3C(Cl)(Cl)C34CC4)=O)CC2)sc2ccsc12 72606,C(=O)(CCP(C)(C)=O)N1CCC(CC=C)(C(=O)NCCN(CCC2CC2)CC)C1 72607,N1(C(C2(CC)CCCCO2)=O)CCCC(CO)(NC(c2ccsc2OC)=O)C1 72608,C(CC(F)F)(C(=O)N(C)Cc1ccsc1)NC(C1C(C)C1)=O 72609,C1(C(N2CC(C)(CC)C2)=O)C(C2CC2)CCN1C(C1COCCC1C)=O 72610,C1(NC(CNC(=O)NC)=O)CCC2(CC1)CN(C(=O)C(C)(CC)CO)CCO2 72611,N1(C(CCC=C)=O)CCC(C(=O)NC2CN(CCC)C2)=C(F)C1 72612,O=C1NC(=O)C2(CCS(=O)(=NC(=O)C34CCCCC3CNC4)C2)N1 72613,C(=O)(C#CC(=O)N(C)C)NC(CC=C)CNC(C1CC(C)=NO1)=O 72614,c1(N2CCN(C)CC2CNC(c2ccc(O)nc2)=O)nc2ncc(Cl)cc2o1 72615,c1(C2(C(N3CC(C(C)NC(C4(CC)CCC4)=O)C3)=O)CC2)ccc(F)cc1 72616,c1(C(=O)NC(CC)CN(C(=O)C=C(CC)CC)C)ccnc(N2CCCC2)n1 72617,N1(C(c2cccc(NC(c3ccc(I)c(O)c3)=O)c2)=O)CCn2cccc2C1 72618,C1(CNC(C(C)OCC#C)=O)CCN(C(c2cc(C)nn2C2CC2)=O)CC1(F)F 72619,C(C(=O)NCCCCC(C)NC(=O)C(C)Cc1cnc[nH]1)(C(C)C)SC 72620,c1(C(C(=O)NC2CC(NC(c3ccc(C(=O)OC)o3)=O)C2)C)cccc(F)c1 72621,C=C(CNC(=O)CC(C)COC)c1ccccc1F 72622,C(C(C)(O)C(=O)N1CCC1(C)CC(=O)NCc1nnnn1C)OC 72623,C1(CNC(=O)C(O)C2CC2)CCCCCN1C(=O)CC1CC2(CCC2)CO1 72624,C1(C)(C(N2CC(CC=C)(NC(=O)CNC(=O)OC)C2)=O)CCNC1=O 72625,C1(CNC(c2ccc(Cl)s2)=O)CC(O)(CNC(C23CSCC2C3)=O)C1 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72677,CC1CCc2[nH]c(=NC(C)c3cn(C)cn3)[nH]c(=NCC3(CC4CC4)CC3)c2C1 72678,C(C)(C(=O)NOCC(=O)NC1CC1)(c1ccccc1)NC(C)=O 72679,C1(C(=O)NCCNC(C)=O)CC(O)CN1C(c1cc(C(=O)OC)c[nH]1)=O 72680,C1(OCC#C)CCN(C(=O)CCC2CC2C(=O)OC)C1 72681,C(=O)(CS(=O)(=O)N(C)C)NCC(C)CN(C(=O)Cc1ccc(C(F)F)cc1)C 72682,c1(C(N2C(C3N(C(C4CCN(C)CC4)=O)CCC3)C2)=O)cnc2ccnn2c1O 72683,Nc1ncc(Br)cc1C(N1CCC(NC(=O)CC2CC=CC2)C(O)C1)=O 72684,c1(N2C(CNC(c3cnc(SC)s3)=O)CCCC2)c(CO)c(C)nc2ncnn12 72685,C=CCC(C)(C)C(=O)NCC(CCNC(=O)CS(=O)(=O)CC)OC 72686,C1(NC(C(NOC)=O)=O)CC2CCC(C1C)N2c1cccc(F)c1C#N 72687,c1(C(=O)NC2(CO)CCCN(C(c3ncn(CC)c3)=O)C2)cc(C)c(C)nc1C 72688,c1(NC(N2CCN(C(c3cccc(C)n3)=O)C3CC23)=O)ccc2c(c1)OCO2 72689,C(=O)(C1=CCC2CCC1N2C(=O)C(CN(C)C)N(C)C)NC(C#C)(CC)CC 72690,N1(C(c2ccc(OCOC)cc2)=O)CCN(C(=O)CSC(=N)N)CC1C 72691,c1(N(CC(CC)C)C)[nH]c(=NCc2nnc(CN(C)C)s2)nc2scnc12 72692,N1(C(C(CC(=C)Cl)NC(=O)C(C)C(=O)OC)=O)CC(C)(C)C2COCC12 72693,C#CC1(C(=O)NCCCC2(O)CC2)CN(C(=O)CSC)C1 72694,C1(C(=O)NC(C2CCOC2)C#C)CN(C(=O)CCCC2CC2)CC1(F)F 72695,c1(NC(C2(C)CN(C(CC=C=C)=O)C2)=O)cc(O)ccc1OC 72696,CC1CC(c2ccccc2)CN(C(=O)C(N2CCCCC2=O)CN(C)C)C1 72697,C12(C(=O)NCC=CCNC(c3nc(N)c(Br)nc3)=O)OCCCC1C2(F)F 72698,C1(C)(CNC(C2(COC)CCC2)=O)CCCN1C(=O)CCc1cccc(OC)n1 72699,Cc1cc(Cl)cc(N)c1C(=O)NCC1(F)CCC(CNC(=O)C(CO)C(C)(C)C)C1 72700,N1(C(c2c(OC)ncc(COC)c2)=O)CCC2CN(C(=O)CNC=O)CC12 72701,C1(F)(CNC(C(C)(C)c2cscn2)=O)CCC(NC(=O)C(N)=O)C1 72702,c1(CC)ccc(CN2CC(OC)CC2C)c(O)c1.C(C)(C)(C)ON 72703,C(=O)(C(O)CC(C)C)NC(COC)CC(=O)N1CCOC(C(C)(C)C)C1 72704,c1(C(N2CCC(OCCNC(C3(C)CC(C)C3)=O)CC2)=O)cc2c([nH]1)CCCC2 72705,c1(NC(C)=O)ccc(C(=O)N(C2CCN(C(C3C(C)C3C)=O)C2)C)cc1 72706,C1(NC(=O)CC2(O)CCOC2)CCC2CC1CN2C(c1nc(F)ccc1Cl)=O 72707,c1(CC)oc(C(=O)NC(C)(CNC(c2cccc(C)c2)=O)C2CC2)cc1C 72708,c1(CC(N2CCC(C)(CCNC(c3ccc(C)cc3)=O)C2)=O)cccc(C#N)c1 72709,c1(-c2cn(CCNC(CCNC(CCC)C)=O)nn2)cccc(CC)c1 72710,c1(C(=O)NC2C3CN(C(c4[nH]c(=N)sc4)=O)C(C3)C2)cc2cc(F)c(F)cc2[nH]1 72711,N1(C(CC=CCC)=O)CC(CO)C2(CCN(C(=O)CC(C)CC)CC2)C1 72712,N1(CC)CCCCC1C(=O)NCCN(CC(C)SC)C(C1CNC(=O)N1)=O 72713,N1(C(c2n(CC)ncc2)=O)CCCC(CO)(NC(=O)CN(c2ccncc2)C)C1 72714,C1(NC(=O)NCC2CC2C(C)(F)F)CCCN(C(=O)Cc2ccccc2O)CC1 72715,N1(C(C(CC=CC)C)=O)CC(C2CC2)(C(=O)NC(C)CCCC)C1 72716,CC(CF)CC(=O)N1CCN(C(C2CC2C(=O)OCc2ccccc2)=O)CC1 72717,C(=O)(C(C)(C)CC#N)NCCCCC(C)NC(=O)COc1ccc(F)cn1 72718,c1(C(=O)NCC(C)CNC(=O)C(=O)NCCC(N)=O)ncccc1[N+](=O)[O-] 72719,Cc1nccc(Cl)c1C(=O)NC1CC(F)CN(C(c2cn(C)c(=O)n2C)=O)C1 72720,N1(C(C(CCC)CNC(=O)COCCCOC)=O)C(C)CC2CCCC12 72721,CC1CC(CC(=O)NC(C2CN(C(C3CCCCC3C)=O)CCO2)C)C(C)O1 72722,c1(C(N2C(COC)CN(C(C3CCC3)=O)CC2)=O)cccc2c1NCC(C)C2 72723,N1CCN(C)C(CNC(C=C(C)C2CC2)=O)C1.C1CCC(=C2CCC2)CC1 72724,CCCCC(C)(F)C(=O)NC1CC1C1CCOCC1 72725,c1(C(C)NC(=O)CC2CC(=O)NC2=O)cc(Cl)cc(Br)c1 72726,Cc1c(C(N2CCCC(C(C)(O)CNC(=O)C3CC3)C2)=O)nn2c1CCCC2 72727,C1(NC(=O)CCc2cccs2)CCCC1CNC(=O)Cc1ccoc1 72728,C(=O)(C(COC1C(CCC)C1)OC)OCC 72729,C1(CN(C2CCN(C(=O)C3CCCC3)C2)C(c2nsnc2O)=O)CC2C=CC1CC2 72730,N1(C(=O)Cc2nc[nH]n2)CC2C3CCC(C2C1)N(C(c1coc2c1CSC2)=O)C3 72731,C(=O)(CC1=CCOCC1)N(C1CC1)CC1CCCCC1NC(C1(C(=O)NC)CC1)=O 72732,Cc1cnc(N2CC(NC(=O)CC(=O)NCC(F)(F)F)CCC2C)nc1O 72733,c1(OCC)c(OC)cc(C(=O)NCC(C)CNC(C2(C)CC2(C)C)=O)cc1Cl 72734,N1(C(CSCC)=O)CCC(CNC(=O)Cc2cnns2)C1(C)C 72735,c1(C(N2C(CN(C(CCn3ncc(C)c3)=O)C)CCC2)=O)c(C)nsc1C 72736,C1(NC(C(C)SC(F)(F)F)=O)COCCN(C(c2c(Cl)csc2Cl)=O)C1 72737,N1(C(CN(C)C)=O)CC(NC(C2CC(=O)N(CCN(C)C)C2)=O)CC(C)(C)C1 72738,C(=O)(CC1OCCc2ccsc21)N(C)CCN(C(=O)C(C)(C)c1sccc1Cl)C 72739,Cc1nn(C2CCC2)cc1C(=O)NCC(C)(C1CC1)NC(c1nc(C2CC2)cs1)=O 72740,C#Cc1ccc(CC(=O)N(C(C)CO)C2CC2)cc1.c12nocc1C(=O)NC2 72741,[SH](=O)(=O)C1CCN(C(=O)CSCCOC)C1.C1(CNC(COCC)=O)CCOC1 72742,C(C1CCCN1C)=CC(=O)NCCN(C(C(C)=C1CCCC1)=O)C1CC1 72743,Cc1cccc(C2(C(=O)NC(C)CC(C)NC(=O)CCN3CCCC3)CC2)c1 72744,c1(C(=O)NCC2CN(C(CCCSC)=O)C3C2C3)cc(Cl)ccc1OC(C)C 72745,c1([SH](CC(=O)NCC2C=CCN2CC2COCCO2)NN2CCCC2=O)ccc(Cl)cc1 72746,C1(NC(C(CC)Cc2cccc(C)c2)=O)CN(C(=O)C(C)C)Cc2ccnn2C1 72747,C1(O)(C(C(=O)NC(C2CCCCC2)CNC(CCOC)=O)(F)F)CCOCC1 72748,Cc1cccc(C(CF)NC(c2cc(-c3ccncc3)[nH]n2)=O)c1 72749,c1(-c2cn(C)nn2)csc2cncn12.C1(N(CC(F)(F)F)C)CCN(C(=O)CS)C1 72750,c1(CCC(=O)NC(CNC(=O)C#CC2CC2)CO)cc(F)cc(Br)c1 72751,O=C(C1=CCCSC1)NCCN1CCN(C(=O)CSc2ccncc2)CC1 72752,C1(C(=O)NCC(C(C)C)O)CC12CCN(C(=O)COc1cccnc1)CC2.C1CN1 72753,C1(NC(C=C(Cc2c(OC)cccc2)C)=O)CC2CC(NC(=O)C=C(C)C)CC12 72754,N1(C(C(CCN(C)C)O)=O)CC2C=CC1C(C(N1CC(NC(N)=O)C1)=O)C2 72755,c1(CN2C(C(N3CCC3CO)=O)CC3CC32)cc(F)c(O)c(F)c1 72756,N1(c2cc(C(C)C)ncn2)CC2CC(NC(C3CCCC(C)(C)C3)=O)CC2C1 72757,N1(C(C(C2CCN(C(=O)C=CCF)C2)C)=O)CC2OC(=O)N(C)C2C1 72758,N1(C2CC34C(C2)C3CC(=O)c2ccc(nc2)N(C2CC2)C4=O)CCSCC1C(F)(F)F 72759,N1(C(C2CC2(F)Cl)=O)CC(n2cncn2)C1 72760,c1(CC)ncc(C(=O)NCCOCC(=O)NCC(Cl)=CCl)o1 72761,c1(C(=O)NCC(C(C)C)(C)C(C)O)cccc(N=c2cncc[nH]2)c1 72762,CC(C)(F)CCC(=O)NCC1CCCC1NC(c1cnoc1-c1ccccc1)=O 72763,CCCCCC(O)C(=O)N1CC2C(CNC(=O)Cn3cnc(Br)c3)C2C1 72764,CCC(CO)N(CCOC)CC1(Cl)CCC1 72765,c12cnc(O)n(c1=O)C1C(CC1)NC2=O.C(C(=O)OC)(C1CC1)OCC 72766,N1(C(Cc2c(C)noc2C)=O)CC2CCCC2(NC(c2cc(C(C)C)sn2)=O)C1 72767,N1(C(C(C)=C2CCCC2)=O)CC2CCC(CNC(=O)C(C3CCCCC3)C)C2C1 72768,N1(C(c2cc(C)no2)=O)CCC(CC(=O)NCc2cnn(C(C)C)c2)C1(C)C 72769,C1(C(N2CCC(OCCNC(C=C(CC)C)=O)C2)=O)CCN(C2CC2)S1(=O)=O 72770,Cc1cc(Cl)cc(Br)c1NC(C1C2CC1N(C(c1ncoc1C)=O)C2)=O 72771,CC(C)(C(=O)NCCc1cnn[nH]1)C1=CCN(C(=O)CC2(O)CCC2)C1 72772,C=CCC(CC(F)F)C(=O)N1CC2CC(NC(=O)CSC(F)F)CC2C1 72773,N1(C(c2c(CC)c(F)ccc2)C(=O)NCC2CCOC2)CCCC(C2CCC2)C1 72774,C1(COC)CN(C(c2cc(C)cc(O)c2)=O)CCN1C(c1coc(C(C)C)n1)=O 72775,S(=O)(=O)(c1ccc(C(F)(F)F)cc1Cl)C1C(COC)CN(c2cc[nH]c(=N)n2)C1 72776,C1(CNC(c2cc(C)c(O)nn2)=O)CC2CCC1N(C(=O)C1=C(C)OCCS1)C2 72777,CC1CN(C(c2cc3n(n2)CCCC3)=O)CCN(C(=O)COC(C)(C)C)C1 72778,CCC(CO)(C(=O)N1CC(CCNC(=O)Cc2ccon2)C1)OC 72779,c1(OC)cccc2ncnc(N3CCCN(CCNC(=O)C(O)C(C)C)CC3)c12 72780,CC1CC(CCC(=O)NCC#CCNC(=O)CCc2ccn(C)n2)C(C)N1C 72781,C1(C(=O)NCCN2CCC(NC(C3CC(=C)C3)=O)CC2)CCCCCN1C 72782,c1(C(N(CC(CC)NC(c2ccc(CO)s2)=O)C)=O)c[nH]nc1Br 72783,c1(C(=O)NCC2(CC3CC3)CC2)cc(S(=O)(=O)C(N(C)CC2CCC3CC23)=O)c[nH]1.N(C)C 72784,C1(C(N2CCC(CNC(c3ccn(CC(=O)OC)c3)=O)C2)=O)CCC2(CC1)CC2 72785,C(C(CC)(CC)C(N)=O)NC(CN(C(=O)C=CCN1CCC1)CCC)=O 72786,C=CCCCC(=O)NC1COCC1NC(C1CCCCC1CN1CCCCC1)=O 72787,C1(C(=O)NOCCC(C)C)(NCC(=O)N(C(C)CS(C)=O)C2CC2)CC12CCC2 72788,N1(C(c2nnc(C)s2)C(=O)NCc2cccs2)CCn2ncc(Cl)c21 72789,c1(C(CC)=O)ccccc1C(=O)NCC(C)CNC(C1CC1c1nccn1C)=O 72790,Cc1nc(C(c2nnnn2C(C)(C)C)NCCN2CCOCC2)cs1 72791,c1(C(=O)NCC(C2CC2)NC(C(C(=O)NC)(C)C)=O)ccc2nonc2c1 72792,n1(C(C)C)cc(C(N2CC3CC2C3CNC(=O)CS(=O)(=O)CC)=O)c(O)nc1=O 72793,c1(C(N(CCNC(C(Br)=C(C)C)=O)C(C)C)=O)ccc2occc2c1 72794,N1(C(C2C(C)(C)C2(F)F)=O)CCCC2(C1)OCC(O)C2O 72795,C1(CN(C(=O)CSc2cnn(C)c2)CC)CCCCN1C(=O)C=Cc1ccco1 72796,N1(C(C(CNC(C(C)SC)=O)CC2CC2)=O)C2CCC1CC(O)C2 72797,N1(C(C(F)=CCC)=O)CC(CNC(=O)COC(F)F)C2(CCC2)C1.C(C(=O)OC)S 72798,Cn1ncc(C2CCCN2C(=O)NCCCNC(c2nn[nH]n2)=O)c1F 72799,C(=O)(CC(O)CNC(C1(N(C)C)CC1)=O)N1CCC(OCC)C1 72800,C(C1CCCO1)=CC(=O)NCC1(CCNC(CC(C)c2ccncc2)=O)CC1.C1CC1 72801,c1(C(c2nnnn2C)NCC#CC)ccnc2[nH]c(C(F)F)nc12 72802,C1(CNC(c2cc(C)c(C(F)(F)F)nc2)=O)CCN(C(=O)C(C)(F)F)C12CCC2 72803,N1(C(Cc2nc(CC)sc2)=O)CCOC(C)(CNC(c2cc(C)cs2)=O)C1 72804,c1(CCNC(C2N(CC)CC2)=O)cc(C(=O)N(C)Cc2cncn2C)no1 72805,Cc1ccc(O)c(CN2CCC(C)(C(=O)NCc3cc(F)cc(Br)c3)C2)c1 72806,c1(CC)[nH]c(Cl)nc(=NCC2(NC(c3ccnn3C)=O)COC2)c1C#N 72807,c1(C(N(C(C)CCNC(=O)Cc2ccccc2CO)C)=O)ccc(N=[N+]=[N-])cc1 72808,C(CCC(C)C(=O)N1CCC(C2CCCCN2C(=O)CC(C)C2CC2)C1)OC 72809,N1(C(C=C(C)C)=O)CCC2OCCN(C(C3CC3(c3ccc(F)cc3)C)=O)C2C1 72810,Cc1c(C(=O)NCCNC(=O)C(C)Cc2cnc[nH]2)nnn1-c1ccccc1F 72811,N1(C(Cc2cc(C)cc(C)c2)=O)CCC(C2(NC(C3CC3CC(C)C)=O)CC2)C1 72812,Cc1ccc(C(=O)NCCCN(C(=O)C(O)CNc2[nH]cnc2C)CCO)cc1 72813,c1(C(CNC(c2cc[nH]c2)=O)CO)ccc(O)cc1 72814,c1(C(=O)NC2C3CN(S(=O)(=O)Cc4ccccc4)CC23)c[nH]c2cccnc12 72815,N1(Cc2c3ccc(C#N)cc3[nH]c2)CCC2CCN(C(=O)C(=O)NC3CC3)CC2C1 72816,C1(CC)(CC)CC(NC(=O)C(C)(CO)OC)CN1C(C1CC1CC)=O 72817,CC1(C)CCCN(C(C2CC(F)C2)=O)C1CNC(=O)CCN(c1ccncc1)C 72818,c1(OC)ccc(C(=O)NC2CN(C(C3COC4CC3C4)=O)CC2OC)cc1O 72819,c1(OCC(C)C)ccccc1C(N1CCC(C)(NC(c2ccc(=O)oc2)=O)C1)=O 72820,C(=O)(CC(=O)NCCOC(C)(C)CNC(=O)CCNS(C)(=O)=O)N(C)C.C1CC1 72821,C1(C(=O)NC2CC(NC(CS(CC)(=O)=O)=O)C2)CCCC2(CCC2)C1 72822,c1(CCNC(N2CC(C=C)OCC2)=O)cccc2ccccc12 72823,C1(NC(C2C(CC)CCC2)=O)CCCCN(C(c2ccc(N(C)C)nc2)=O)C1 72824,c1(C(=O)NCC(CO)NC(c2ccc(CCCCCC)s2)=O)cnn2ccoc12 72825,C(=O)(C(F)(F)C(C)O)NC(C(=O)NCc1nnn(CC)n1)Cc1cc[nH]n1 72826,c1(C(N(CC(=O)O)Cc2cn(C(C)C(=O)O)nn2)=O)ccnc2ccncc12 72827,Cc1ccc2c(C(=O)NC(C3CCCN(C(C4(C#N)CC4)=O)C3)C)csc2c1 72828,CC1(CNC(c2c[nH]c(C#N)c2)=O)CCCN1C(C1CCCN(CC(F)F)C1)=O 72829,C(=O)(C(C)(C)C(=O)N1CC(CNC(c2cnc(C)[nH]2)=O)C2(CC2)C1)NC 72830,C(C(C(C)C(C)C)NC(c1cc(C)n(C)c1C)=O)NC(COCC(=O)NC)=O 72831,C1(C(N2CC(NC(C3CCCN3C=O)=O)C2)=O)(OCC)CCCCCC1 72832,C=C=C(C)CC(=O)N(CC(C)O)CCNC(c1cn(C)nc1CC)=O 72833,c1(C(C)C)[nH]nc(C(=O)NC2CC2NC(=O)Cc2c[nH]nc2O)c1Br 72834,C=CCC(C)C(=O)N(C(C)CN(C)C(C1CCN(c2cc(=O)cc[nH]2)CC1)=O)C 72835,C1(NC(Cn2c(C)cc(C)n2)=O)C2CCN(C(c3sc(F)cc3C)=O)C2C1(C)C 72836,N1(C(c2csc(C)c2C)=O)CC2OCC(NC(C3(F)CC=CC3)=O)C2C1 72837,CCC(O)C(C)(C)C(=O)NCC(C)(C)CNC(=O)CCCCN(C)C(C)C 72838,N1(C(c2sccc2I)=O)CCC(C(N2CC(C)(C(F)(F)F)C2)=O)CC1 72839,C1(NC(C(COC)C)=O)CCCN(C(=O)C(C)(C)OCC(F)(F)F)C1 72840,c1(OC)ccc(Cl)cc1S(=O)(=O)NCc1cc(Br)ccc1N(C)C.C1(C)C(=O)O1 72841,c1(CC(C(=O)N(CCC(C)NC(c2cnsc2)=O)C)=O)cccc(Cl)c1 72842,N1(C(COCCOC)=O)CCCC1CC(=O)NCC1CCC(C(N)=O)C1 72843,N1(C(CCCC)=O)CC2CCCC2(C(=O)NC(C2CCCC2O)C)C1 72844,N1(C(C2=C(C)OCCS2)=O)CCCC2CN(C(C3(O)CCSCC3)=O)CCC12 72845,c1(C(=O)NCCCN(C(=O)CC(C)C)CC)cc(Cl)n[nH]1 72846,c1(C(=O)NC2CC(CNC(C3(O)CCCC3)=O)C2)ccc2cnccc2c1 72847,C1(Cc2cn(NC(C34CC(F)C3C4(F)F)=O)nn2)CC2(CCCC2)CO1 72848,C1(NC(C(CCC)OCC)=O)CCN(C(C2CCCC2O)=O)CC1C 72849,CC(C(CCc1ccccc1)NC(=O)CC1(C)CC1)NC(=O)Cn1cnnc1 72850,Cc1cnc(C(=O)NCC2CCCCN(C(=O)C=Cc3ncc(C)[nH]3)C2)c(F)c1 72851,C1(C(=O)NC2C(CNC(C3CC34CCOC4)=O)COC2)CCC=CCC1 72852,C1(C(N2CC3C(NC(C=C(C)C4CC4)=O)C3C2)=O)COC2(CCC2)CO1 72853,CC1CCC(C(c2ccccc2)=O)CN1C(=O)Nc1cccc(Cl)c1 72854,C1(C(N(C2CC3CCC2O3)C)=O)CCC(C)(C)N(C(c2c(O)cccc2F)=O)C1 72855,c1(C(=O)NC(CN(C(C2CC2CC(C)C)=O)CC)C)c(Br)ccc(F)c1N 72856,c1(OC)ccc(C(=O)N(C(CNC(=O)Cc2cncnc2O)C2CC2)C)c(F)n1 72857,CC(C)CC(C)CC(=O)NCC1(F)CCC(NC(C2(F)CCCC2)=O)C1 72858,C1(C(=O)Nc2ccc(OC)c(C(C)C)c2)CC12CCN(C(=O)C(C)(C)C#N)CC2 72859,c1(CN2CCC(O)(C(N3C(C(N)=O)CCC3)=O)C2)cc(I)ccc1F 72860,c1(C(C(=O)NCC2C(NC(=O)CCOCC3CC3)C2)O)cccc(O)c1 72861,C12(CNC(=O)Cc3csc(Cl)n3)CCC(CC1)N(C(c1cc(F)cnc1O)=O)C2 72862,C1(C(N2CC(n3cc(CNC(COC(C)=O)=O)nn3)C2)=O)CCCC(C)(C)CC1 72863,c1(CCC(=O)NCC(N2CCCC2CN(CC)CC)=O)c[nH]c2c(C)cccc12 72864,C(=O)(C1=COCCC1)NC1C(C(=O)NCCn2c(C)ncc2)CCOC1 72865,C12(NC(c3cccn4ccnc34)=O)CCCC1N(C(=O)C1=NOCC1)CC2 72866,N1(C(c2ccc(N)cc2F)=O)CC2CCC(C1)N2C(C1CCCCS1)=O 72867,c1(C(N(CCC(C)NC(=O)C(C)(C)N2CCCC2)C)=O)ccc2nn(C)cc2c1 72868,Cn1cncc1C=CC(=O)NCCCCNC(C1COC(=O)N1)=O 72869,N1(C(C(=O)Nc2cn(CC)nc2)=O)CC(C(N)=O)C(C(C)(C)CN)C1 72870,N1(Cc2cnn(CCC)c2C)CCC2CN(C(=O)C(C)Cn3cccn3)CCC12 72871,c1(CN(C(=O)NCC(N(OC)C)=O)C2CC2)cc(F)ccc1NS(N)(=O)=O 72872,N1(C(C(C=C=C)C)=O)CCC(CC=C)(C(N2CCC(c3ncco3)C2)=O)CC1 72873,N1(C(CC(C)C2CCCO2)=O)C2CCCC1CC(NC(=O)CN1CCN(C)CC1)C2 72874,C(=O)(C1=NOC2COCC12)NCC(CC(=O)Nc1ccc(C)nc1C)O 72875,C#CC1(C(=O)NCc2ccccc2Cl)CN(C(c2ccc(C)s2)=O)C1 72876,Cc1nc(C(=O)NCC2CCN(C(C3CCNC(=O)C3)=O)C2(C)C)ccc1C#N 72877,C1(NC(c2[nH]cc(CC)c2)=O)CCOC(C(=O)NCc2nncn2C)C1 72878,c1(C(=O)NCC(C)(CO)NC(c2c(OC)c(Cl)sc2)=O)ccc(F)c2[nH]ccc12 72879,CC1CC(N(C(=O)C(=O)N(C)C)CC(c2cccc(C(F)(F)F)c2)C)CCO1 72880,CCCC(C)(O)C(=O)NC1CCCC(C(N2CCC(O)CC2C)=O)CC1 72881,N12CCCC(C1)C2=O.C(=O)(C(CC)OCC)NCCOCCSC1(CCCC)CC1 72882,C1(C(=O)NC(CN(C(CN(C)CC)=O)CC)C)CC2OC(C)(C)OC2C1 72883,c1(C(N2C(CC=C)(NC(=O)C(C)OCC)CCC2)=O)ccn2cncc2c1 72884,N1(C(C(C)Cn2cccn2)=O)CC(NC(c2c(Cl)cnn2C2CC2)=O)C(O)C1 72885,c1(OC)ncccc1CC(=O)NC1CCN(C(=O)C(C2CC2)SC)C1C 72886,C1(C)(C(=O)OC)CCC1(C)C(=O)NCCCN(C)C(c1sc(F)cc1C)=O 72887,CC1(C(=O)NCC(C2CCCC2)NC(=O)CCCCN2CCCC2)CCCCO1 72888,N1(C(Cc2scc(C)c2)=O)CCCCCC(Nc2ccnc(C3CC3)n2)C1 72889,c1(CCCCCC)nc(CCCC(C)C)n(-c2cc(C)ccn2)n1 72890,C1(O)(CNC(C(CC)NC(C)=O)=O)CCCN(C(=O)NC2(C3CC3)CC2)CC1 72891,Cc1cccc(CCNC(c2nnnn2C)CCOc2ccccc2)c1 72892,c1(CC(N2CCCN(C(C(C)NC(C)=O)=O)CC2)=O)coc2ccccc12 72893,c1(NCc2cn(CCNC(C(C3CCCOC3)OC)=O)nn2)cc(C)ncn1 72894,c1(NC(=O)COC2(CCO)CN(C(CC(=O)NCC#C)=O)C2)cc(C)ccc1F 72895,C(=O)(CCCS(N)(=O)=O)N(CCC(C(C)C)NC(Cn1nc(C)n(C)c1=O)=O)C 72896,c1(C(N2CCC(C(C)NC(COCCC(C)C)=O)C2)=O)cccc2c1CNC2=O 72897,N1(C(C(C(=O)OCC)(C)C)=O)CCCCCC(NC(C2CC=CCC2C)=O)C1 72898,C1(C(=O)NC)(C(N2CCC(C(C)C(=O)N(C)CCOCC3CC3)C2)=O)CCCC1 72899,c1(C(CC(=O)NCCC2CCN(C(CCCOC(C)=O)=O)C2)O)ccc(Cl)cc1 72900,C1(C(N2CC(CC(C)NC(C3CCCCC3O)=O)C2)=O)C2CC3CC(C2)CC1C3 72901,C1(NC(CCN2C(CCCCCCC)CCC2)=O)CC=C(C(=O)NC)C1 72902,N1(C(C2C3(CC(OCC)C3)C2)=O)CC2CC(NC(=O)C(=O)C(C)(C)C)C1C2 72903,CC(C)(CCNC(=O)Cn1cnc(=N)[nH]1)NC(C1CCCSC1)=O 72904,c1(C(=O)NC(c2cc(Br)ccc2Cl)(C)C)cc2ccc(Cl)nc2s1 72905,c1(OC(C)C)ncncc1Nc1nnc(-c2ccc(Br)cc2)n1C 72906,c1(-c2nc(-c3c(C)scn3)n(C(C)C3CC3)n2)ccc(CC(F)(F)F)c(Cl)c1 72907,CCC(CC)(CC)C(=O)NCC(C(C)C(C)C)NC(c1ccc(S(N)(=O)=O)s1)=O 72908,c1(OC)ccc(NC(=O)C(C)Cc2ccc(C)cc2)c(O)c1OC 72909,c1(SC)nc(N2C(C(=O)Nc3cc([N+](=O)[O-])cs3)CC3CC23)ncc1Br 72910,CCCCC(C)(F)C(=O)N1CCC(C(=O)NCC(CSC)OC)C1 72911,C(CNC(=O)CC1CC1)(CC(=O)N(C1CC12CC2(F)F)CC(C)C)OC 72912,C1(C)(C(=O)NCC(C)(CNC(=O)C(C)=C(C)C)OC)CCC(C)C1 72913,CC(CC(F)(F)F)C(=O)N1CC(CC(=O)NC2(CCF)CC2)CC1(C)C 72914,c1(C(=O)OCC)c[nH]nc1S(=O)(=O)NCCOCC1CCCC1 72915,N12CCCC(C1)OCC2=O.C(CC)(C(=O)NCC(C)(C)OC)OCC.C1(C)CC1 72916,c1(C(=O)NC(C)CCCCNC(c2ccon2)=O)c(Cl)oc2ccccc12 72917,c1(OC)ncnc(C(=O)NCC2CCCCC2NC(=O)Cn2cnnc2O)c1F 72918,C(=O)(C(CO)C(C)(C)C)NCC1(C)OCCN(C(c2cnc(C(C)(F)F)[nH]2)=O)C1 72919,N1(C(c2nc(C(C)OCC)sc2)=O)CCC(C)(NC(=O)CS(=O)CC)CC1 72920,N#CCCCCCC(=O)NCCC1CN(C(=O)Cn2cc(CO)nn2)CCCO1 72921,c1(C(N)=O)cc(C(=O)NCCCCCCNC(C2CC(Cl)(Cl)C2)=O)ccc1O 72922,CC1CCCC(CC(=O)NCCCCc2ccc(Br)cc2)O1 72923,c1(C(=O)NC2C(CNC(C3C(=C)C3)=O)CCCC2)ccc(N)c(F)c1Br 72924,c1(C(C(=O)N(CC(CC)NC(C(C=CC)O)=O)C2CC2)=O)cc(Cl)cc(Cl)c1 72925,Cc1cccc(C(=O)NCCC2(NC(=O)CC(F)F)CC2)c1.c12cnn(c1)C2 72926,C(=O)(CCC(C)(C)[N+](=O)[O-])NCc1c(OC)ncnc1OC 72927,c12ccc(cc1)CO2.C1(O)(CC#C)CC(C(N2CCCC2CC(C)C)=O)C1 72928,N1(C(CCC(CC)C)=O)CCN(C(c2ccn3c2CCCC3)=O)C2(CC2)C1 72929,C#CC(C1CCc2ccccc21)NC(=NCCc1ccc(Cl)cc1)NCCC=C 72930,c1(C(C(=O)NC2CC2)N(CCN(C(CC)C)C)CCOC)ncnc2cc[nH]c12 72931,C1(CCCNC(C=C(C)C(C)C)=O)CCCCN1C(C1CN(C(=O)OC(C)C)C1)=O 72932,C(=O)(C1CCCc2scnc21)NCCCCNC(c1c[nH]c(=NCC)s1)=O 72933,CC1COCC(C(=O)NC2CCC(CC(N3CCC(CC4CC4)C3)=O)CC2)O1 72934,CCCC(C)CCCC(=O)NCC1(F)CCC(CNC(=O)C2=COCCO2)CC1 72935,C(=O)(C(C#N)(CC)CC)N(CCCNC(C1CCC(CN2CCCC2)CC1)=O)C 72936,c1(C(=O)NC2CC(NCc3cncc(O)c3)C2)cc2cc[nH]c2cc1F 72937,C1(NC(c2c(C)cno2)=O)CCC2(CC1)CN(C(c1ccccc1S(C)=O)=O)C2 72938,C1(C(=O)NCC#CC(=O)N2CC(c3nc(=O)o[nH]3)C2)C(F)(F)C12CC2 72939,c1(NC(CC=C)C)[nH]c(=NCC2(C)CC2)nc2c1cnn2C 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73218,Cc1noc(C)c1C(N1CC(CCNC(=O)CNC(CCC(F)(F)F)=O)C1)=O 73219,c1(OC)cccc2ncnc(N3CCC(CNC(c4nnc(O)nc4O)=O)C3)c12 73220,C#CCC(CC#C)C(=O)N1CC(NC(=O)C(CC)CC)C(C(F)(F)F)C1 73221,c1(C(N2CCC(NC(C3CC(C)(CC)C3)=O)C2)=O)c(C)nnn1CC 73222,Cc1nc2c([nH]1)C(Nc1cc(C)c(S(N)(=O)=O)c(C)c1)CCC2 73223,c1(Nc2ncc(COC)s2)cc(NC(c2cnc(F)c(C)c2)=O)ccc1[N+](=O)[O-] 73224,N1(C(C(C2CC2)OC)=O)CCCC(C(=O)NCC2CCC3(CC2)CC3)CC1 73225,C#Cc1cnn(CC(=O)NCC(C)(C(C)C)NC(c2nc(Cl)sc2C)=O)c1 73226,C12(NC(CCN(C(CCC)C)C)=O)CCCC1CN(C(=O)Cn1cnccc1=O)C2 73227,c1(C(=O)NC(CCCC)CNC(C2(SC)CCCC2)=O)nc2ccccc2[nH]1 73228,N1(C(C2CCC(=C)CC2)=O)CC=C(CC(=O)N2CC(C(N)=O)CC(C)C2)CC1 73229,C1(C(F)F)(CNC(COCCOC)=O)CCN(C(=O)Cc2c[nH]ccc2=O)C1 73230,C12(C(=O)NC(CC(C)NC(c3coc(-c4ccccc4)n3)=O)C)CC(C)(CO1)C2 73231,C(C(=O)N1CC(O)C(O)CO1)c1cc(C(N2CC3CCC(C2)O3)=O)n[nH]1 73232,C12(CNC(C(C)NS(CCCC)(=O)=O)=O)CN(C(=O)Cn3ccc(C)n3)C1CCO2 73233,CN1CCCCC(C(=O)N(CCCN(C)C)CCNC(=O)C(F)(F)CO)C1=O 73234,c1(C(=O)NC2CCN(C(=O)C(F)(F)C3CCCCC3)C2)nccc2[nH]ccc12 73235,Cc1c(C(N2CC(O)(CN(C)C(c3ccnn3CC3CC3)=O)C2)=O)cccc1Cl 73236,C(=O)(C1=NOCC1)N(CCCNC(C1CCCCN1C1CCCC1)=O)CCO 73237,C(=O)(C(O)C(F)(F)F)NC1(CO)CCN(C(C(N2CCOCC2)C)=O)C1 73238,C1(C(=O)NC2CCCN(C(c3ccc(C(F)F)nc3)=O)C2)CCc2nnnn2C1 73239,C1(C(=O)NCCCCCOCC(=O)NCC2CCCO2)CNc2ccccc2O1 73240,Cc1nc(NC2CCC(NC(=O)CC(C)n3ccnc3)CC2)cc(C#N)n1 73241,Cc1nc2ncccc2cc1C(=O)NC1CCC(NC(=O)C(C)CC(N)=O)CC1 73242,C#Cc1ccc(F)c(F)c1CNC(c1cccc(C(C)(C)O)c1)=O 73243,Cc1cccn2cc(CC(=O)NC3CC(CNC(=O)CSc4cn[nH]c4)C3)nc12 73244,c1(N2C(C(CC)C)CCC2)cc(C)c(C(=O)OC(C)(C)C)cn1 73245,c1(C(=O)NCC2C(NC(C3(SC)CCCC3)=O)C2)c(C)nn(C)c1Br 73246,c1(C(=O)NCC2C(NC(C(C)C3CCC3)=O)C2)cc(Cl)cnn1 73247,c1(OC)cccc(F)c1C(N1CC(O)(C(C)NC(=O)CCCCCF)C1)=O 73248,CC1(C(=O)NOCCCCCO)CCCN1C(=O)Cc1nc(=N)[nH][nH]1 73249,C=CC(CC)CC(=O)N1CCCC1C(=O)NC(CCOC)C(C)C 73250,N1(C(C(C)CNC(=O)CC(C2CC2)C2CC2)=O)CCCC2(CC(O)C2)C1 73251,c1(CC(=O)NCC2C(NC(CCN(CCCCC)C)=O)C2)cncnc1 73252,c1(OC)nccc(Br)c1NC(=O)C(C)C(C)(C)C 73253,CC(C)CCC(O)C(=O)NN1CCCC1C(=O)NC1(C)CCCC1C 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73395,c1(OC)c(C(=O)NC2CC(CNC(c3cnn(CCO)c3C)=O)C(O)C2)csc1C 73396,CN1CC(O)CC1(C)C(=O)NCCC1(CNC(C2CNC(=O)C2)=O)CC1 73397,C#CC1(O)CCCN(C(C(=O)NCCOCC)c2ccsn2)C1 73398,C1(OC)CC(F)CN(C(c2cnn(C3COC3)c2)C(=O)NC2CCOC2)C1 73399,CCCCC(CNC(C1CN(C(=O)C(F)CCC(C)C)C(C)(C)C1)=O)CCC 73400,N1(C(c2c(C)noc2C)=O)CC(C)(C)OC2(C1)CN(C(=O)CCc1nccs1)C2 73401,N1(C(C2C(CC)C2)=O)CCN(C(=O)C=Cc2cccc(F)c2Cl)C2CCC12 73402,CCC(C)C(O)C(=O)N1CC(C)C(C)(CNC(=O)CC2CCCC(C)(C)O2)C1 73403,C=CCC(CCC)NC(=O)C(C)N(CCC)C(C1(CO)CCOC1)=O 73404,C(=O)(CS(=O)(=O)CCOC)N1CC(CCOC)OCC1.C12CCCC1NC2=O 73405,N1(C(C2C(CC)C2(F)F)=O)CCC(NC(c2coc(OC)n2)=O)C(C)C1 73406,c1(C(=O)NC(CCOC)CNC(=O)C(C)NS(C)(=O)=O)c[nH]c(=S)cn1 73407,c1(CCC(=O)NC(C(=O)OC)C(C)O)nc2ccccc2c(=O)n1CC(C)C 73408,C1(C(=O)NC(CCC)c2nn[nH]n2)C=CCN(C(=O)CN(C)C(=O)OC)C1 73409,N1(C(C(CC(=C)C)NC(=O)Cc2ccon2)=O)CCN2C(=O)OCC2C1 73410,c1(CCCC(=O)NCC2CCN2Cc2ccccc2Br)ccccc1Cl 73411,c1(OCC#N)ccc(Cl)nc1C(=O)NC1CCN(c2ccccc2)C1 73412,C=C1CC2(C1)CC(C(=O)NC1(CF)CCN(C(c3cc(N)cc(F)c3)=O)C1)C2 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73467,c1(C(N2C(CNC(c3n(CC)cnn3)=O)CCC2)=O)cnn2c1S(=O)(=O)NCC2 73468,c1(C(=O)NC2CC2)ccc(C(=O)NC2CCN(C(=O)CN3CCC3)C2)cc1 73469,c1(CC(=O)NCC(C)N(C(c2ccsn2)=O)CC)nnc(C)o1 73470,C1(NC(COCCN(C)C)=O)CCCC(NC(=O)C2=COCCO2)CC1 73471,C1(C(=O)NCCC(C)N(C(c2cc(OC)n[nH]2)=O)C)CCCC2(CCCCC2)C1 73472,c1(OC)cccc(C(CNC(=O)C(Cl)=CCl)NC(c2c[nH]nc2F)=O)c1 73473,c1(C(N2C(CC)CN(C(c3ccc(=O)n(C)n3)=O)CC2)=O)ccc(C)c(F)c1F 73474,N1(C(C2CCN(C(CC)=O)C2)=O)CCC(F)(CNC(c2ccn(C(C)C)n2)=O)C1 73475,c1(C(=O)NCC(C)(CC(C)C)NC(CCOCC(C)C)=O)ccn2ccnc2n1 73476,c1(OC)cc(OC)cc(C(N2CC3CC(C2)N3C(c2snnc2C)=O)=O)c1 73477,c1(NC)cc(C(N2CCC(CNC(=O)CSCC(N)=O)C(C)C2)=O)cc(Cl)n1 73478,c1(CN2CC(C(=O)Nc3ccc(Cl)c(Br)c3)OCC2)ccc2c[nH]nc2c1 73479,N=S(=O)(CCNS(=O)(=O)c1cnc(-c2ccc(Cl)cc2)s1)c1cccs1 73480,C#CCCCCCC(=O)N(CCCCC(=O)N(C)Cc1ncnn1C)C 73481,CC1(C)COC(C(=O)NCCC2CN(C(=O)COC3CCCCCC3)C2)C1 73482,c1(C(CC(=O)NCCOCCCNC(c2cc(CC)[nH]n2)=O)C)ccccc1F 73483,c1(OC)cnc(C(=O)N(CCC(C)NC(c2sccc2C)=O)C)cn1 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73518,c1(C(=O)NCC(C(C)(C)C)NC(=O)CCc2cnc[nH]2)nnn2c1CCCC2 73519,C(=O)(CCCCCNC(=O)OC)N1CCC(CNC(CCC#CC)=O)(COC)C1 73520,c1(OCC)nc(C)ccc1C(=O)NCC1(CNC(=O)CCC(C)C)CCC1 73521,c1(C(N(C2CCC(NC(=O)CC34CCCC3C4)CC2)C)=O)ccc(CCO)cc1 73522,C1(CC(=O)NCc2c(C)csc2)CCN(Cc2csc(C(C)C)n2)CC1 73523,c1(C(N2C(CCNC(c3ccnc(C)n3)=O)CC(OC)C2)=O)ccc(N)cc1O 73524,C1(C)(C(N2C(C#C)CC2)=O)CCCN(C(c2cnncc2NCC)=O)C1 73525,N1(C(C=CCSC)=O)CCC(CCNC(=O)CN(c2ccc(Cl)cc2)C)CC1C 73526,C1(CC(=O)NCCCN2C(C)CCC2)CC(F)CN1C(=O)CCCOC(F)F 73527,N1(C(CCN(C)CC)=O)CCCCC(C(=O)NC2CCCC2)C1 73528,N1(CC)CC(NC(=O)C(CNC(=O)COC)OC2CC3CC(=O)C2C3)CCC1=O 73529,c1(Oc2c(NC(CC3(C(=C)F)CCC3)=O)cccc2)nc2ccc(Br)cc2s1 73530,c1(C(=O)NCC(CC)NC(C2OCCO2)=O)cc([N+](=O)[O-])cc2c1OCCO2 73531,C(=O)(CC(=O)NCCN(C(=O)CNC(c1ccccc1)=O)CC)NCC#C 73532,N1(C(C2C(C)SCCC2)=O)C2CCC(C(N3CCC3(CO)CO)=O)C1CC2 73533,N1(C(c2c(CC)nccn2)=O)CC(O)CC1(C)C(=O)N(C)Cc1nncs1 73534,C=CCC(C)(C)CC(=O)N1CCCCCC1C(=O)NC1(CC)CC1 73535,N1(C(C(C)(C)C2CCC2)=O)CCCCC1C(=O)NCCC(O)(C1CC1)C1CC1 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73554,CN=c1nc(N2CCC(Cn3cncn3)CC2)[nH]c(=NCCC2COCCO2)[nH]1 73555,Cc1ncc(C(=O)N(CC(C)(C)CNC(=O)CC2CCCC2O)C)cc1N 73556,C=C(Br)CCC(=O)NC1CN(C(c2cc(C(N)=O)ccn2)=O)C1 73557,C12(NC(CC3N(C)CCC3)=O)CCCCC1CN(C(=O)CSC1CC1)C2 73558,c1(C(=O)NCCC(C)CCNC(C=CC)=O)cc(Cl)cc(Cl)c1.c1ccncc1Cl 73559,C1(C2(O)CCOC2)(C(=O)NCCC(C)NC(=O)CCN2CCCC2=O)CC1 73560,C(C(C)(O)C(=O)NCC1(C)CCCN1C(C1CCC(C)C1)=O)OC 73561,c1(C(C(=O)NC2C(NC(CCCC)=O)CC2)(C)C)c[nH]c2ccccc12 73562,C1(N(C)C(c2cccc(O)n2)=O)CC2CCC(C1)N2C(c1ccc(CO)cc1)=O 73563,N(S(=O)(=O)N1CCC1c1cccnc1)(CC(C)C)CC 73564,N1(CC(=O)NC(CN(C(C2(C(=O)NC)CCC2)=O)C)(C)C)CCC(=O)NC1=O 73565,c1(C(=O)NCC2C(CNC(c3c(CC)c[nH]c3)=O)C2(F)F)cc(C)cnc1Cl 73566,C1(C)(COC)CCCN(C(=O)Nc2ccccc2Cn2ccnc2)C1 73567,N1(C(C(CO)OC)=O)CC(NC(=O)C(F)=C(C)C)CC12CCCCC2 73568,N1(CC)CCOC(C2CCCCC2)C1.C1(=O)C(C2CCN2C(=O)OC(C)(C)C)N1 73569,C1(CNC(c2cnc(C)[nH]2)=O)C2CN(C(=O)Cc3ccnc(Br)c3)CC12 73570,Cc1ccc(C(N)=O)cc1NC(C1C2CN(C(c3csnc3Br)=O)CC12)=O 73571,C(CCCS(=O)(=O)CCO)NC(c1cccc(CNC(N2CCCC2)=O)c1)=O 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73676,CC#CCC(C(=O)NC(CO)C1(C)CC1)NC(c1sccc1C#N)=O 73677,c1(CN(C(C2(C(=O)OCC)CC2c2cccnc2)=O)C)ccc(C#N)cc1C 73678,N1(C(C(c2ccc(C)s2)C)=O)CCN(c2cc(CNC(=O)C(N)=O)ccn2)CC1 73679,N1(C(Cc2ccc(CC(C)(C)C)cc2)=O)CCC(NC(C2COC2)=O)C(C)(C)C1 73680,N1(C(C2(CC=C)CCCN2C(c2nnn(CC)c2C)=O)=O)CCOC2CN(C)CC12 73681,c1(CCNC(c2scc(C(=O)OC3CCCCC3)c2)=O)cccc(Cl)c1 73682,C(=O)(CCCC(C)(F)F)N1CC(NC(CC2CC(OCC)C2)=O)C(C)(C)C1 73683,N1(C(c2ccc(Cl)nc2)=O)CC2CN(C(=O)C(O)C3CCCC3)CC2C1 73684,CC1C=C(C(=O)NC2CCN(C(c3cc(C(F)F)cs3)=O)C2)CC1 73685,N1(C(CC2(C)CCN(C(CC(C=C)C)=O)C2)=O)CCCCCCCCC1 73686,Cn1ccc2c(NC(c3cn(-c4ccc(Cl)cc4)nn3)=O)cccc2c1=O 73687,C#CCCC(=O)N(CCN(C(c1ccccn1)=O)C(C)C)CCOC 73688,O(NC(=O)CC(C(F)F)NC(=O)C(C(=O)OC)OC)CCCCCC 73689,C1(CNC(C2CC(C)OC2C)=O)CN(C(=O)CCS(C)(=O)=O)CC(C)(C)O1 73690,C1(S(=O)(=O)NC(c2nnnn2CC2CC2)C)(C(C2CC2)OC)CC1 73691,C1(NC(c2n(C(C)C)nnn2)(C)CCN2CCCC2)CC(C)N(C)CC1C 73692,N1(C(c2ccn(CCOC)n2)=O)CCC(C2CC2)C(C)C1.C(C(C)(C)SC)=CC(=O)N 73693,c1(CC(=O)NC(CNC(CC(C=C)C)=O)(C)Cn2cccn2)cccc(C)c1C 73694,c1(C(N2CC3C(CNC(c4c(CC)nccc4)=O)(C3)C2)=O)ccc(Cl)c(OC)c1 73695,C1(OCC)CC2CN(C(=O)NC(c3cccc(Br)c3C)C)CC12.OCC 73696,c1(C(=O)NCC(C)N(C)C(C2OCCCC2(C)C)=O)cccc2sncc12 73697,C1(NC(CNS(NC)(=O)=O)=O)CCCC12CN(C(c1cnc(C3CC3)s1)=O)C2 73698,N1(C(COC(C)C)=O)CC(C(N2CCC(CCCO)C2)=O)C(C2CC2)C1 73699,C(=O)(C1=CC2CCCC12)NCC1C(C)(C)CCN1C(=O)CC1=CCCC1 73700,Cc1cc(F)ccc1NC(C1(C)CCCN1C(=O)COCCN(C)C)=O 73701,C1(C(=O)NCC(CNC(c2ccc(N(C)C)cc2)=O)CO)CN2CCC1CC2 73702,Cc1cc(C(N2CCC(O)(CN(C)C(C3CCCN3C)=O)C2)=O)nc(C)n1 73703,C1(C2CC2)(NC(C2CCC23CC(F)(F)C3)=O)CCN(C(c2cnc[nH]2)=O)C1 73704,c1(Nc2ccc(C(=O)NCC3(O)CC3)cn2)ccc2ccncc2c1 73705,Cc1ccc2nc(C)c(C(=O)Nc3cnc4cccc([N+](=O)[O-])c4n3)n2c1 73706,C1(NC(COCCC#C)=O)CC(C)CN(C(=O)C(c2ccc(C)cc2)F)C1 73707,C(CCC(C(=O)NC1CC(O)C1OC)NC(c1ccc(O)cc1F)=O)OC 73708,C(=O)(C(F)(F)C(C)O)NCCC(C)N(C(C(C)Cc1ccc(N)cc1)=O)C 73709,N#Cc1ccccc1CCCC(=O)NC1CCCCN(C(c2nccs2)=O)C1 73710,N1(C(C(CCC)F)=O)CCN(C(c2cc(CO)on2)=O)C(C2CC2)C1 73711,S(=O)(=O)(CCC(=O)NC(C)(C)CCNC(c1c[nH]nc1-c1ccncc1)=O)NC 73712,C1(CNC(COCCCOC)=O)CN(C)CCN1C(=O)Cn1cccnc1=O 73713,N1(C(C(C)c2cc[nH]n2)=O)CC(NC(c2ccsn2)=O)CCC1C 73714,N1(CCO)CCCC(N2CCC2)C1.c1(C(=O)NC2CC(CC=O)C2)cnn(C(F)F)c1 73715,C1(NC(C2CC(OC)(OC)C2)=O)CC(C(=O)N(C)Cc2nc(C)no2)C12CCC2 73716,c1(N2CCCN(c3c(N)c(Cl)ccn3)CC2)ccc2nncn2n1 73717,c1(C(=O)NCC(C)NC(C2CCCN(CCC)C2)=O)c(Cl)ccc(C)c1O 73718,c1(C(=O)NC2C(NC(c3cnc(CC)s3)=O)CCC2)cc2c(cc1Cl)NCC2 73719,C(CC)(CCC(=O)N(CC)CC1CCCC(C)(C)C1)NC(c1c(CC)ncs1)=O 73720,C1(NC(NCc2nnn(C)n2)=S)C2Cc3ccc(Cl)cc3C12 73721,N1(C(C=C(COC)C)=O)CCOCC1CCNC(c1ocnc1C1CC1)=O 73722,c1(C(N2CC(C(C)NC(C3CCC(OC)C3)=O)C2)=O)cc2sccc2n1C 73723,CCC(O)C(C)(C)C(=O)N1CC(NC(c2c(Cl)n[nH]c2C)=O)C(O)C1 73724,c1(C(=O)NCC2OCCCN(C(C3C(C)CC3)=O)C2)ccc(=O)n2c1CCC2 73725,Cc1nc(-c2ccc(Cl)cc2)oc1COc1cccc(I)c1 73726,C1(C(N2CC(C)N(C(=O)CCc3ccco3)CC2)=O)CC(C2CCOCC2)=NO1 73727,CC(C)C(C)C(=O)NC(C1CN(C(C2CNC2)=O)C1)C 73728,C1(C(N(C2CC2)CC)=O)CCCCC1NC(c1cc(C)nn1-c1ccc(Cl)cc1)=O 73729,C1(C(C)C)(C(=O)NCCCCN(C(=O)C(c2ccc(Cl)cc2)=O)C)CCCCO1 73730,N1(C(C2C(C)OC(=O)N2)=O)CC2(C1)C(NC(=O)CC1(C)CC1)CCS2(=O)=O 73731,C#CC1(N(C)C)CN(C(C2CC=CCN2C(=O)CC2COCC(C)O2)=O)C1 73732,N#CC1(C(=O)NCCC2CC(NC(c3ccc(C(F)(F)F)nc3)=O)C2)CCOC1 73733,c1(C(=O)NC(CNC(C2CC=CCC2)=O)CO)ccc(-c2cnc[nH]2)cc1 73734,CC1Cc2cc(C(N3CCNC(=O)CC3)C(=O)NCC3CC3)ccc2O1 73735,Cc1[nH]nc(C(N2CC(O)CC2C(=O)NC(CO)C2(C)CC2)=O)c1O 73736,C(N=c1[nH]c(C)ncc1[N+](=O)[O-])C1(C)CCN(C(CC(C)SC)=O)C1 73737,CC1(C)CCCCC1CN1CCCC1.C1(=O)C(C(C)(C)C)O1 73738,c1(C(=O)NCCN2CCN(C(C(C(C)C)F)=O)CC2)c(F)ccc2nc[nH]c12 73739,CC1CCN(C(C2CC(CCNC(c3ccc(O)nc3)=O)C2)=O)C(C)C1 73740,C1(O)(CCN(C(CSCC(C)C)=O)C2CC2)CN(C(c2nc(C(F)(F)F)cs2)=O)C1 73741,CCC(C)(C)C(C)CC(=O)NC1CCC(NC(=O)CCOC2CCOCC2)C1 73742,CCC(CC(=O)NC1CN(C(=O)CS(=O)(=O)CC2CCC2)CCC1F)C(C)(C)C 73743,CC1CN(c2nc(C3CC3)ns2)CCC1NC(c1cnn(C)n1)=O 73744,n1(CCSc2ccc(C#C)s2)c(C)cc(CC(=O)N(CC(F)F)C)c1C 73745,c1(SCC(=O)NC2(CO)CN(C(=O)C=CI)C2)ccc(F)c(F)c1 73746,CCC(O)(CN1CCCCC1C(=O)NCCCCCCCSC)C(F)(F)F 73747,CCC(CCC(=O)NCCC1CC(NC(C)=O)C1)NC(=O)CSC 73748,C(=O)(C1=CNC2=NCCC2=C1)N1CCC(CCNC(CSc2n(C)cnn2)=O)C1 73749,c1(C(=O)NCC(CC)NC(c2cnoc2CC2CC2)=O)cnc(-c2cccs2)s1 73750,N1(C(CNC(=O)C=Cc2ccoc2)=O)CCC(OCC2CC2)CC1.C(CO)O 73751,Cc1c(Br)cc(C(=O)NC2C3CN(C(c4ccn(C)n4)=O)CC23)cc1Br 73752,C1(NC(C2(C)C(C)(C)C2)=O)CC12CC(NC(c1csc(Cl)c1Cl)=O)C2 73753,CC(CC(F)(F)F)C(=O)NC12COC(C1)C(NC(c1ccn3ncccc13)=O)C2 73754,N12CCCC3(C1)CN(C3)C2=O.C1CC(C)(O)C1.N1(C(C)C2CC(C)C(CC)C2=O)CCCC1 73755,CCC(C)C(O)C(C)C(=O)NCc1cncc(C(N2CCC(C)(F)C2)=O)c1 73756,c1(C(N2CCN(C(CCc3scc(C)n3)=O)CC2CF)=O)c(C)cc(F)cc1C 73757,Cc1cc(C)c(CN2CCC(C)(C(=O)Nc3cccc(Cl)c3C)C2)cc1C 73758,Cc1nc(C)c(CNC(=O)Nc2ccncc2-c2ccccc2F)s1 73759,C1(C(=O)Nc2c(C)nsc2)N(C(=O)CN(C)C(N)=O)CC12CCCC2 73760,c1(CNC2CCN(C(CC#N)=O)C2)ccc(-n2cncn2)cc1 73761,C1(NC(C2C(C)=CCS2)=O)C=CCC(C(=O)N(CC(C)(C)O)C)C1 73762,CCCCCC(O)C(C)C(=O)N1CCN(C(C2(SC)CC(=O)C2)=O)CC(C)(C)C1 73763,c1(OC)cnc(F)c(C(=O)NCC2(C(C)NC(c3nccs3)=O)CC2)c1 73764,c1(Sc2c(C3(CC(=O)NC(C)=O)CC3)cncn2)cccc2nonc12 73765,C1(C(C(F)(F)F)NC(=O)NCc2c(C3CC3)cn(C)n2)CCCS(=O)(=O)C1 73766,c1(C(=O)NCCCN(C(C2C(C)C2C)=O)C2CC2)cnccc1N(C)C 73767,C1(C(N2CCC(CC)(CC)C2)=O)CC(O)CCN1C(=O)CN1CCCC1C 73768,CCCCCC(C(=O)NCC1=CCN(C(C2CCC(C)O2)=O)CC1)C(C)C 73769,CCC(CC(F)F)C(=O)N1CCN(C(=O)C=Cc2ccc(C(F)F)o2)C(C2CC2)C1 73770,c1(C(=O)NC2CCCN(C(CC3(C=C)CC3)=O)C2)cnc(N)c(CO)c1 73771,N1(CCNC(c2c(C)cccn2)=O)CCCN(C(C2(C)CCOCC2)=O)CC1 73772,Cc1cnn(C)c1CC(=O)NCC1(C)CCCC1NC(c1cc(C2CC2)cs1)=O 73773,C(C(F)(F)CCNC(c1nc(C)oc1C)=O)NC(=O)OC 73774,c1(C(=O)NCCC(=C)CNC(=O)CCC(=O)C2CC2)cc2ccc(Cl)cc2s1 73775,CC1(C)CN(c2nc(N3CCC4(C)C(CC(C)C4)C3)nc3c2SCC3)CCS1(=O)=O 73776,n1(CCC(N2C(C(=O)N(N3CCOCC3)C3CNC3)C=CC2)=O)cc(Cl)cn1.CC 73777,n1(CCOC)cnc(=NC(=O)NC2CCN(C3CCOC3)CC2)[nH]1 73778,N1(C(c2c(C)cc(=N)[nH]c2)=O)Cc2ccccc2C(CNC(c2ccno2)=O)C1 73779,c12ccc(c(C(F)(F)F)c1)C(C)C(=O)N1CC(C1)O2.C1(NC)C2CCCC12.COCC 73780,Cc1cc(C)n2ncc(C(=O)NC3C4CC3N(C(C3(C(C)C)CC3)=O)C4C)c2n1 73781,c1(C(C(=O)NCCSC)N(C2CCNC(C)C2)C)c(Cl)nc2sccn12 73782,CS(=O)C=CC(=O)NCC1CN(C(c2cccc(C(=O)N(C)C)c2)=O)CC1O 73783,C1(NC(CCN(C)CCO)=O)CC(O)CN(C(c2cncc(C(N)=O)c2)=O)C1 73784,c1(C(=O)NCC2N(C(C34CCC(OC)(CC3)C4)=O)CCC2)c(F)ccc(N)c1F 73785,N1(C(Cc2ccc(OC)cc2)=O)CCN(C(c2ccc(F)o2)=O)CC(CO)C1 73786,c1(OC)ccc2c(c1)CCN(C(=O)C(=O)N(C1(C)CCCO1)CCNC(C)=O)C2 73787,C(=O)(CC(C)(C)COC)NCC(CC)NC(=O)C(c1cccc(O)c1)OC 73788,Cc1nnc2n1CCC(C(=O)NC1CC(C)CN(C(=O)CCCS(N)(=O)=O)C1)C2 73789,c1(N2CC(NC(C(C(C)C)O)=O)C(C)C2)ncnc2[nH]ccc12 73790,CC1CC2CC(C(N3CCCN(C(C4CCCC(=O)N4)=O)CC3)=O)(C2)O1 73791,N1(C(C(C)NC(C)=O)=O)CCOC2(C1)CN(C(C1CC1C(=O)OC(C)(C)C)=O)C2 73792,C1(CNC(c2nc(CCC)oc2)=O)CN(C(c2cnsc2)=O)C2CC12 73793,C1(NC(C(C)NC(C)=O)=O)CCC2(CC1)CN(C(c1ccncc1F)=O)C2 73794,CC(C)C(C)C(CNC(=O)CCn1ccnn1)Nc1ncnc(Cl)c1CO 73795,Cc1c(C(N2CC(CNC(=O)C=CS(C)=O)C(C)(C)C2)=O)c[nH]c2nccc1-2 73796,C1(C(=O)NCC=CCNC(c2c(CC)c(C)sc2)=O)COc2ccc(Cl)cc2O1 73797,CN1CCCN(C(=O)CC(C(F)F)NC(C2(C)CCNC2=O)=O)CC1=O 73798,N1(C(c2c(C)cn(C)n2)=O)CCN(C(=O)CCCc2ccc(Cl)cc2)CCC1C 73799,c1(C(=O)NC2CN(C(c3cnccc3Cl)=O)CCC2F)nccc2ccsc12 73800,c1(OCCc2ccccc2)ccc2nc(-n3ccnc3)[nH]c2n1 73801,C(CNC(C1CC(CC2CC2)C1)=O)(C(=O)NCC1(O)CSC1)OC 73802,C1(C(N2C(C=C)CC2)=O)CNC(=O)CN1C(c1nc[nH]n1)=O 73803,C1(C(N(CCCNC(CNC(C)=O)=O)C)=O)CN(C)C2(CCC2)C1 73804,Cc1ccc(F)cc1CC(N1CC=CC(NC(c2occc2CN(C)C)=O)C1)=O 73805,Cc1ccc(C=CC(N2CC(F)CC2CNC(C2(C3CC3)CCCO2)=O)=O)o1 73806,C1(OC)CN(C(=NCCCCl)NCC2CCC(C(F)(F)F)CC2)CC1O 73807,c1(CN2CCC(N3CC(=O)NCC3)CC2)nc2ccc(Br)nc2[nH]1 73808,c1(CC)cc(C(=O)NCC(C2CN(C(=O)C=CC3CC3)C2)F)cn(C)c1=O 73809,n1(CC(=O)NC2CC(N(C(c3cn(CC)nn3)=O)C)C2)cnc2sccc2c1=O 73810,C1(CNC(c2nccc(Cl)c2F)=O)CCN(C(C2(F)CCOC2)=O)C12CC2 73811,CC(=O)C(C)CC(C)C(=O)NC1CC2(C1)CC21CCC1.C12CCCN(C1)C2=O 73812,c1(C(=O)NCC(CC=C)NC(=O)CC2CC(C)C2)ccc(-c2coc(O)n2)cc1 73813,C1(C(=O)NCCC(=O)NC)C2CCC(C2)N1CCC1CCOCC1 73814,c1(C(N(CCNC(CC(CCSC)O)=O)C)=O)c[nH]c2ccc(Cl)cc2c1=O 73815,C1(C(C)NC(=O)CCc2ccnn2C)CCN(C(=O)C(C2CC2)N(C)C)CC1 73816,Cc1nc(CNC(C2(C)CCC2)=O)[nH]c(=NC)c1C 73817,C1(NC(C(C)NC(=O)C(C)CN(C)C)=O)CC2(CCCC2)C1 73818,c1(CC(CN(C(CCC)CO)C)O)cccc(F)c1 73819,C1(CC)CCN(N(C)CCCCc2ccc(Cl)cc2Cl)CC1 73820,N(C)(C(=NCC(O)c1ccccc1)NC1CCCC1)C(C1CCOC1)C 73821,N1(C(C=CSC)=O)C2CCC1CC(N(C)C(c1ccc(C3CCC3)cc1)=O)C2 73822,c1(CC)nc(C(=O)N(C)CC2CCCN2C(=O)C=C(C)C(C)(C)C)cs1 73823,C1(C)(CC)CCC(C(=O)N(CCC(=O)N(CC)Cc2cc(OC)nn2C)C2CC2)O1 73824,C1(C)(C(N2CC(C)C(CNC(=O)CC3=CCCCC3)C2)=O)CCOC12CC2(F)F 73825,N1(C(CC2N(C(C)C)CCC2)=O)CCC(O)(CNC(=O)COC(F)F)CC1 73826,c12cc(ccc1Br)SCC2.c1(C(=O)OC)[nH]nnc1C1CCC1 73827,Cn1ccc2c(C(N3CC4CCC4(NC(=O)CCCN(C)C)C3)=O)ccnc12 73828,NC(=O)CCC(=O)NC1CCCC(CNC(c2coc(-c3cccnc3)n2)=O)C1 73829,N1(C(c2nc(C)n(C)c2)=O)CCC(C)(NC(=O)C(C)C(F)(F)F)CC1 73830,C1(O)(CC(=O)N(CCCNC(c2ncn(C(C)C)n2)=O)C(C)C)CCCCCC1 73831,c1(C(N2CCC(C(C)NC(=O)CN3CCNC3=O)C2)=O)nnc(S)n1C 73832,CC(CC(C)(F)F)C(=O)NC(C)(CNC(C1CN(C(=O)N(C)C)C1)=O)C1CCC1 73833,C#Cc1cnncc1C(=O)NCCC1(C)CCN(C(=O)C(COC)OC)CC1 73834,N1(C(c2n(CC)nc(C)c2)=O)CCN(C(=O)Cc2ccno2)CC2(CC2)C1 73835,C1(NC(c2c(OC)cc(Cl)cc2)=O)CC(C)(C)C12CCC2 73836,C(=O)(C(O)CC(C)(C)C)N(CCN(C(C(=O)NCCCC)C)CCCC)C1CC1 73837,Nc1ccc(C(N2CC3CC3(C(=O)NCC3NC(=O)NC3=O)C2)=O)nc1 73838,S(=O)(=O)(c1ccc(S(N)(=O)=O)c(Cl)c1)NC1C(CC)CCCC1 73839,CC(C(=O)NC1CCN(C(=O)CNC(c2ccc(Cl)cc2)=O)C1)C(C)(F)F 73840,C1(CNC(C=C(CC)CC)=O)(NC(=O)Cc2ccc(Cl)c(Cl)c2)CCCCC1C 73841,CCCC(C)(CC)C(=O)N1CCC(Cn2cc(CCS(=O)(=O)N(C)C)nn2)C1 73842,c1(C(=O)NC(c2ccccc2)C(=O)NC(c2ccn(C)c2)CC)coc(C)c1 73843,c1(OC)cc(C)c(C(=O)NC(C2CCCC2)=O)cn1 73844,c1(C2C(C(=O)NCC3(F)CN(C(CCOC)=O)C3)C2)cccc(OC(F)(F)F)c1 73845,N1(C(C2C(CNC(=O)COc3cccnc3)OCC2)=O)CC2CCC2C1 73846,C(=O)(C1=CCCSC1)NCC(C)NC(=O)CNC(c1c(F)cccc1F)=O 73847,c1(CC(=O)NC2CC(NC(C(CC)OCC)=O)C2)c[nH]c2cccc(Cl)c12 73848,N1(C(C(CC)(C)O)=O)CC2CCC2(C(=O)NCc2ccnnc2)C1 73849,CC1CN(C(C2C=CCC2)=O)CC(C)N1C(c1ccccc1OCC(F)(F)F)=O 73850,C(C)(C)(CC(=O)NCC1CCC(NC(=O)CSc2n[nH]c(=N)s2)C1)SC 73851,C1(CCC(=O)NC)CN(C(c2ccc(C)nc2)=O)CCN1C(=O)C#CC1CCC1 73852,c1(CC(=O)NCCOC2CN(C(C(CCC)O)=O)C2)cccc(C#N)c1 73853,C(C(CC(=O)NCC1(C#N)CC1)C1CCC1)NC(c1c(C)[nH]cc1)=O 73854,c1(NC(CNS(c2ccc(C)c(C)c2)(=O)=O)=O)c(C)cc([N+](=O)[O-])cc1Br 73855,C(=O)(CS(=O)(=O)Nc1ccccc1O)N(C1C(OCC)COC1)C 73856,C1(C(=O)NC(C)CC(=O)NC2CC2)C2CC1N(C(=O)NCc1n[nH]cc1Cl)C2 73857,c1(C(=O)NCC#CCNC(C(C(C)(C)C)N(C)C)=O)cc(N)cc2c1CCC2 73858,C1(C(=O)NCC(O)CNC(N)=O)(NC(C2OCCN(C)C2=O)=O)CCC(C)(C)CC1 73859,N12CC3CC(C1)C3NC(=O)c1ccc(cc1)C2=O.C1(C)(C(N(C)C)=O)CCOC1 73860,C(N=c1[nH]cnc2c1COC2)C1N(C(=O)CC(C(F)F)c2ccccc2)CCC1 73861,c1(C(N2C(COC)(CNC(=O)C3=CCCC3)CCC2)=O)ccc2cccnc2c1 73862,C1(CNC(COc2c(C)cccc2)=O)N(C(=O)C(C)NC(N)=O)CCC1(C)C 73863,N1(C(C2=NOC(C)C2)=O)CC2CCC(CNC(=O)C(F)(F)F)OC2C1 73864,C1(CCC)CCC(C(=O)NC2CCN(C(=O)C(CCC)n3cccn3)CC2)CC1 73865,C(=O)(C)CCN(C(CCC)c1cccs1)CC#C.C(C)(=O)O 73866,C(=O)(C1=NNC(=O)CC1)N(CC(C)(C)NC(c1ccns1)=O)C 73867,C1(C(N2CC3(N(C(=O)CCN4CCCC4=O)CC3)C2)=O)CCCCC(F)(F)C1 73868,N1(C(C2(CCNC(=O)CC3(O)CCCC3)CC2)=O)CC2CC2C2CC12 73869,C(=O)(C(C)(C)C(=O)N(C)C)NCC(C)(CO)NC(c1cn(CC)nn1)=O 73870,C1(NC(C2C(F)(F)C23CC3)=O)CN(C(=O)CCC2CCCC2)CC1CO 73871,c1(C(=O)NC2C(C)CN(C(=O)C#CC3CC3)C2)ccc2ccoc2c1 73872,CCCCC(C(=O)NCC(C)(C)C(=O)N(C)C)NC(c1cc(C)c(C)[nH]1)=O 73873,c1(N(C)C)cc(N2CCC(CSc3conc3C(C)(C)C)C2C2CC2)ncn1 73874,Cc1nc(C(=O)NC(CNC(=O)C=C(C2CC2)C2CC2)C2CCC2)nn1C 73875,C1(C(CC)=O)CC(C)N(CC=CCCCCC)C1.N1(C2CC(CN)C2)CCOCC1 73876,N1(C(CC2(OCC)CCC2)=O)CC(NC(c2cc(O)no2)=O)CC(F)C1 73877,N1(C(C(C)(C)C#N)=O)CC2(CCC(CNC(C3CCC4CC34)=O)O2)C1 73878,C(CC(C)(O)C(=O)NC1CCCC(O)C1O)n1cc(C(C2CCOC2)C)nn1 73879,CC1CCCn2c(COC(C3CCCCC3Oc3ccccc3F)=O)cnc21 73880,C(CCC(C)C)(C(=O)NC(C)C(F)F)NC(C(n1c(C)ccn1)C)=O 73881,c1(-c2c(C(N(CC(CC)NC(=O)CCC(C)=O)C)=O)c[nH]n2)cc(F)cc(F)c1 73882,Cc1nc(N)cc(NCCC(c2ccccc2)O)n1.C1(C)CC(C(C)(C)C)C1 73883,n1(C(CC)C)nc(-c2cccc(N)n2)nc1-c1cnn(CCOC)c1 73884,c1(C(=O)NC(C(C)NC(c2ccoc2C(F)(F)F)=O)C)[nH]nc2ncnc(O)c12 73885,N1(C(=O)CC2CCC2)CCC(C(=O)NCc2ncccn2)C1 73886,C=CC(CCC)CC(=O)N(C)CC1CCN(C(C2CC3C=CC2CC3)=O)C1 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74309,CCC(CN(C)C)CC(=O)NCCC1CCCCN1C(c1cnc(O)c(F)c1)=O 74310,C(C(=O)OC(C)(C)C)(C(=O)N1CC(CC(C)NC(=O)C(F)=C(C)C)C1)OC 74311,C1(NC(C2(CC)CCCCC2)=O)CCCN(C(=O)Cc2ccc(Cl)cc2C)C1C 74312,Cc1cc(C)c([N+](=O)[O-])c(C)c1CCCN1CCN(CC2COC2)CC1 74313,N1(C(c2nc(CC)sc2)=O)CCC(CC(C)NC(=O)CC(=O)OC(C)(C)C)CC1 74314,N1(c2nc(=NC)[nH]c(=NCc3ncnn3C(C)C)[nH]2)CCCC2CCCC(O)C12 74315,C(CC(C)C)(C(=O)N(C(C)CN(C)C(c1ccncc1C)=O)C)OC 74316,CC(C)(C)CS(=O)(=O)NC(C1(O)CC2CCC1C2)=O 74317,C1(CCOC)(NC(c2cn(CCC)nn2)=O)CCN(C(C2CC(=O)CO2)=O)C1 74318,N1(C(c2c(CC)noc2)=O)CCn2ncc(CNC(c3ncsc3C)=O)c2C1 74319,Cc1cccc2c1CCN2C(=O)CC(C)CC(=O)Oc1ccccc1 74320,c1(CC=C)cccc(C(N2CC(NC(=O)CCc3cnn[nH]3)C(C)C2)=O)c1 74321,c1(C(=O)NC(C2(O)CN(C(Cc3nnc(C)s3)=O)C2)C)cnc(F)c(F)c1 74322,C(c1ccccc1Br)=CC(N1C(C)(CNC(=O)NC(=O)C2=CCCS2)CCC1)=O 74323,Cc1ccc(C=CC(=O)NCC2(NC(C3CCN(C)C3)=O)CCC2)nc1 74324,N1(C(C=CCC)=O)CC(C)(C)C(NC(c2cc(CO)[nH]n2)=O)C(C)(C)C1 74325,c1(C(N(CC)CC2CCCCN2C(=O)CCC=CBr)=O)ccc(C)c(F)c1N 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74344,N12CC3CC(CC3C1)SCC2=O.Cc1cc(C2(C=O)CC2)on1.C1CCCO1 74345,Cn1c(C(=O)NC2CCC(CCNC(c3c[nH]c(=N)s3)=O)C2)cc(Cl)c1Cl 74346,N1(C(C2(OC)CC2)=O)CCCC2(C1)CN(C(=O)C(O)CC1CCOCC1)CCO2 74347,c1(C(N2C(C(c3ccc(C)cc3)C)CCC2)=O)ccc(N(C)C)cc1O 74348,CN1CCCCC(C(N2CCOC(CNC(C34CCC(C3)C4)=O)CC2)=O)C1=O 74349,C(=O)(CCN(OC)C(=O)C(CC(C)C)N(C)C)OC.c12cccnc1o[nH]c2=O 74350,c1(CC)cnc(O)c(C(N2CC(NC(=O)CCc3ncco3)CC(C)C2)=O)c1 74351,C1(CNC(c2cc(C(C)C)[nH]n2)=O)CC(C)CCN1C(=O)CCn1cc(Cl)cn1 74352,O=S(=O)(c1cc(F)cc(F)c1)N1CCN(CCc2nc3c(s2)CCCC3)CC1 74353,c1(C(=O)NC(CCNC(C(CC=CC)C)=O)(C)C)ccc(=O)n(CC(=O)NC)c1 74354,c1(OCCCN(C(c2cc3nc(C)sc3[nH]2)=O)CCO)ccc2c(c1)NCCC2 74355,Cc1ccc(C(=O)NC(C)C(C)(C)C(=O)NC(CC2CC2)C2CC2)c(O)c1 74356,N1(CCC#C)CCN(C(=O)C(C(C)C)NC(=O)C(CSC)OC)CC1 74357,C1(CNC(C2OCCN(CC)C2)=O)CN(C(=O)C(C)OC)CCC12CCC2 74358,C=C(Cl)C(C)(C)C(=O)NC(CNC(=O)CSc1ccc(C)cc1)C(C)C(C)C 74359,C12(C(=O)NCCC(C=C)C)CC(CO)(CN1C(=O)CCCN(C)C(C)C)C2 74360,c1(C(N(CCC(C)NC(c2ccoc2Cl)=O)C)=O)ccc2oc(O)nc2c1 74361,C1(C2N(C(CCOC)=O)CC2)CCOCC1.C(C)(C)(C=CC=O)C(N1CCC1C)=O 74362,c1(COC)nc(CC(N2CCCC2C2CCN(C(=O)CC3CC3)C2)=O)cs1 74363,CC1CC(NC(c2cncn2-c2ccccc2)=O)CN1C(=O)C=Cc1nccs1 74364,N1(C(C)=O)CS(=O)(=O)CC1C(=O)NCC(C)(C)CN(C(=O)CCCCC1CC1)C 74365,C(=O)(C1OCCn2ccnc21)NC(C)(C)CCCNC(c1csnn1)=O 74366,c1(C(=O)NCCCOCCCNC(C(CC)(C)C)=O)cn2c(n1)C(C)CCC2 74367,C1(C2CN(C(=O)COC3(C(F)F)CCC3)C2)(NC(=O)CC2(C(F)F)CC2)CC1 74368,C(=O)(CCCC(F)(F)CO)NC1CCCN(c2cn(C)nc2)C1 74369,c1(C(=O)NC(CN(C(C(C2CCCOC2)OCC)=O)CC)C)c(SC)cnn1C 74370,C1(O)(CNC(=O)Cc2csc(S)n2)CCN(C(C2CCC=CO2)=O)C1 74371,N(C1CCCn2nccc21)C(CC1N(C(CCC(CC)C)=O)CC2(CC2)C1)=O 74372,Cc1ccnc(O)c1C(N1CC2C(CNC(=O)CSCC(F)(F)F)C2C1)=O 74373,c1(CNC(=O)NCC#Cc2cn(C)nc2)cc2cc(F)ccc2s1 74374,c1(CCC(=O)NCCOCCCN(C)C(c2cnc(C(N)=O)s2)=O)nc(O)n[nH]1 74375,N(C1CC2CCCc3cccc1c32)C(c1c(S(N)(=O)=O)ccc(Cl)c1)=O 74376,c1(OCC)ccc2cc(C(=O)NC3CCN(C(=O)C(C)(C)CF)CC3(C)C)[nH]c2c1 74377,c1(CNC(CC(COC)NC(c2n[nH]cc2Cl)=O)=O)c(C)cccc1C 74378,CC(=O)CCN=C(NCC(C)CN1CCCCC1C)N1CCC(C)(C)C1 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74414,C1(OCC)CC2(C1)CC2C(=O)NCCn1cc(C2CCN(C(C)C(N)=O)CC2)nn1 74415,C1(Cc2nn(-c3n(C)ccn3)c(C(F)F)n2)CCc2ncsc2C1 74416,C1(CNC(C2(COC)CCC2)=O)CCCCCN1C(c1ccc(O)nn1)=O 74417,N1(Cn2nc(CCC)oc2=O)Cc2ccc(CC(=O)OC)cc2C1 74418,C1(CCOC)(NC(COCCC=C)=O)CCN(C(c2snnc2CC)=O)C1 74419,C1(CC)CN(C(C2(NC(=O)CCCCOC)CCN(C)C2)=O)CCS1 74420,C(=O)(C(CC)CCOC)N1CC(CN2CCN(C(CNC(CC)=O)=O)CC2)C1 74421,C(=O)(CCCN=[N+]=[N-])N(C1CCN(C(c2ccn(CC)c(=O)c2)=O)CC1)CC#C 74422,N1(S(c2ccc(NCC(C)O)nc2)(=O)=O)CC2(CCOCC2)CC1CCO 74423,c1(CC=C)ccccc1C(=O)N(C1CN(C(=O)C2=CCC2)CC1O)C 74424,Cc1cc(C(=O)N(CCNC(=O)Cc2ncoc2C)C(C)C)ccc1OC(F)(F)F 74425,CC1Oc2ccccc2OC1C(=O)NC1COC2(C1)CN(C(C13CC(C1)C3)=O)C2 74426,CC(C)CC(F)C(=O)NCC12CC(NC(C3CCN(C(=O)C4CC4)CC3)=O)(C1)C2 74427,c1(C(N2C3(CCC(NC(CC=C)=O)CC3)CCC2)=O)cc(F)cc2nccnc12 74428,C1(C(=O)NC2(CO)CN(C(C(CC(C)C)=O)=O)C2)CCOC2(CCC2)C1 74429,C(CCC(=O)NC(C)(C)CCNC(=O)CN(C)C(C)C)=CCC=C 74430,c1(C(=O)NC2(CCNC(CC3C(C)C3)=O)CC2)cccc2[nH]ncc12 74431,C1(CCC)(C(N2CC=CC(NC(=O)Cn3ccnn3)C2)=O)CCNC1=O 74432,C1(NC(c2c(C)c(N)ccc2)=O)CC2CC1CN(C(C1CCC(C(N)=O)N1C)=O)C2 74433,c1(C(=O)NCC(CN(C(C2(CC)CCCCO2)=O)C)C)ccc2c(c1)ncn2C 74434,C1(OC)CCN(C(=O)CCC2CCN(C(=O)CCc3cc(C)no3)C2)C1C 74435,C1(C(N2CC(CC(C)NC(c3ccc(C(N)=O)cc3)=O)C2)=O)CC2(C1)CC(F)C2 74436,Cc1ccc(C(C)NC(=O)CSc2nnc3ccccn23)cc1S(C)(=O)=O 74437,C(CCCC(C)NC(=O)CC1(C(F)F)CC1)NC(c1c(C(=O)OCC)con1)=O 74438,c1(OC)c(C(N2CC(O)(C(C)NC(C3(C)CC3(F)F)=O)C2)=O)cc(Cl)cc1Cl 74439,C1(C(=O)NCCOC(C(=O)OC)C)OCCC1C(C)C 74440,C(=O)(CCN(OC)C(=O)C1CN(C(=O)C(C)S(C)(=O)=O)CC(C)O1)OC 74441,c1(OC)ccc(CC(=O)NCCC(C)NC(c2cnc(C(F)(F)F)s2)=O)cc1 74442,C(=O)(CC(CC)CC)NC(CCC)C(N1C2CCC1COC2)=O 74443,C1(C(=O)NCC2N(C(C)=O)CCC2)C=CCN(C(=O)Cc2c(C)n[nH]c2C)C1 74444,C1(NC(CC(COC)C)=O)CN(C(c2conc2C(C)C)=O)Cc2ccnn2C1 74445,C1(NC(CCC)=O)C2CCN(C(c3cccc(CC(C)C)c3)=O)CCC12 74446,C1(C(=O)NCCC(=O)NCC(C2CC2)OC)OCCC1C(C)C 74447,C1(N(CCOC)C(c2ccoc2C2CC2)=O)CCN(C(=O)CC2CCC2)CC1 74448,c1(C(C)C)ncncc1C(=O)NC1CN(C(=O)C(O)CN(C)C)CC1C 74449,N1(C(=O)Cc2ccon2)CCC(C(=O)NC2CC23CCCCC3)C(O)C1 74450,CN1CCn2ncc(C(N3CC4OCC(NC(c5ccoc5)=O)C4C3)=O)c21 74451,C1(CNC(COCC(=O)OC)=O)CC(NC(=O)CCc2cnco2)C1(C)C 74452,N1(C(C(F)=C(C)C)=O)CCC(C)C1CNC(=O)COc1ccccc1F 74453,c1(NC2CC(C)N(C(C3CCc4[nH]nc(O)c4C3)=O)C2)c(Cl)cncc1[N+](=O)[O-] 74454,Cc1ccnc2c(C(=O)NC3CC3NC(=O)CCCCCN(C)C)cccc12 74455,CC1=C(CNC(c2cc(F)cnc2Cl)=O)SCCO1 74456,N1(CCCC2C(F)(F)C2)CCCC1c1ccc(Br)s1 74457,c1(NC(C(n2c(C(F)(F)F)cc(C)n2)C)=O)ccc2ncnn2c1 74458,C1(NC(c2ccc(CO)nc2)=O)CCN(C(C2CCCOCC2)=O)CC1F 74459,N1(C(CC(C)C)=O)CCC2(CCCCN(C(=O)C(O)C(F)F)C2)C1 74460,N1(C(Cn2ccc(C)n2)=O)CCCC(C(=O)NCC2CC23CC3(F)F)(C(C)C)C1 74461,CC(Cc1cnn(C)c1)C(=O)NCCC1CCCN1C(=O)CSc1n[nH]c(=N)s1 74462,C1(CC#C)CN(C(c2ncoc2-c2ccc(OC(F)(F)F)cc2)=O)CCO1 74463,c1(SC)ccccc1C(=O)NCC(CNC(=O)CCC1CC(C)OC1=O)CO 74464,Cc1oc(C)c(C(=O)NC2CCOCC2NC(C2CC2F)=O)c1C 74465,N1(C(c2cn(CC)nc2)=O)CCC(NC(=O)C2=CC(O)CCC2)C(C)(C)C1 74466,CN1CC2CCC(NC(=O)C(=O)NC3CCC4CC34)CC2C1 74467,N1(C(C(C(C)C)O)=O)CCCC(C(N2CCC(CC(N)=O)CC2)=O)CC1 74468,c1(CCn2c(-c3sc(O)nc3C)nc(CCOC)n2)cc(Cl)ccc1Cl 74469,C(CC1(C)CC1)(C(=O)NC1CCC1)N(C(C)C1CC1)CC 74470,C1(NC(c2c(C)ccc(C)n2)=O)CC2CC(C1)N(C(c1ccc(=O)oc1)=O)C2 74471,C1(CNC(c2c(C)cncn2)=O)CN(C(C23CC(C)(CCO2)C3)=O)CCC1C 74472,c1(C(=O)NC23CCCC(NC(c4sccc4F)=O)(C2)C3)cc2n(n1)CCCC2 74473,c1(C(N2CCC(F)(CNC(C(C)C3(O)CCC3)=O)C2)=O)cn2ccnc2cn1 74474,C(=O)(C(C)n1ccnn1)NCC(C)N(C(C1(CCC)CC1)=O)C 74475,CCCC(CNC(=O)CC1CCCOC1)NC(c1ccoc1C(F)(F)F)=O 74476,C1(CNC(C2(C)CC2Br)=O)CN(C(c2nc(Cl)c(Cl)s2)=O)CCO1 74477,CON(C)CCNC(=O)C(C)(C1CC1)N(C)C(C12CC(CO)(C1)C2)=O 74478,C(C(C)C(C)C(=O)N1CC(C)(c2cn(C(c3ccc(Cl)nc3)C)nn2)C1)OC 74479,C12(C(=O)NCC3(OCC)CN(C)C3)CCC(CC1NC(=O)CN1CC=CC1)C2 74480,C(=O)(C(C)(C)C(C)NC(=O)C(F)F)N1CCC(NC(=O)OCC)C1 74481,c1(C(=O)NC2(C(=O)NCCn3c(C)ncc3)CCCC2)cccc(F)c1C 74482,Cn1cc2cc(C(N3CC=CC(NC(c4ccc(O)nc4Cl)=O)C3)=O)ccc2n1 74483,CN1CCOC(C(=O)NC2CCC(CNC(=O)C(F)C3CCOC3)C2)C1=O 74484,C(=O)(C1=CS(=O)CCC1)N(C1CCN(C(C2CCC(F)(F)C2)=O)CC1)CC#C 74485,N1(C(CCC(=C)Cl)=O)CCC2(C1)CN(C(C1CCCC(C)O1)=O)CCO2 74486,c1(OC)cc(-c2cnc(NC(c3cccn3C)=O)c(C)c2)cc(F)c1F 74487,N1(C(C)CN)CCN(CC(C(=O)C=Cc2cccs2)=O)C2(CC2)C1.C(C)(C)(C)O 74488,N1(C(c2nc(C)oc2C)=O)CC(C(=O)NCC(C)(O)C2CCC2)OC(C)C1 74489,C(=O)(C(O)CC(C)(C)C)N1CC(C)N(C(=O)CC2COC(C)(C)CO2)CC1 74490,c1(CC)ccc(F)c(C(N2CCCC(F)(CNC(c3ncc[nH]c3=O)=O)C2)=O)c1 74491,C1(CC(NOCCCCC)=O)CN(C(c2csc(F)c2)=O)C(C)(C)C1 74492,C1(OC)CC2(C1)CC(C(N1CC(NC(=O)C=CC3CC3)C(F)C1)=O)C2 74493,C(=O)(CC1=CCCCC1)NC1(COC)CN(C(C2CC(C)CC(C)C2)=O)C1 74494,Cc1ocnc1C(c1nnnn1C(C)C)NCCC1CC(C)(C)C1 74495,CC(C)(O)C(F)C(=O)NCC(C1CC1)NC(C1CC(CC2CC2)C1)=O 74496,c1(OC)cccc(C(N2CCC(C)C(NC(=O)C(F)C(C)(F)F)C2)=O)c1F 74497,C1(NC(c2n[nH]c(C)c2C)=O)CCCC12CN(C(=O)C#CC(C)(C)O)C2 74498,CN1C2CCC1CC(=CC(N1CCC(NC(=O)C(N)=O)C(CO)CC1)=O)C2 74499,Cc1cc(C(N2CC(CN(C)C(c3cc(CC(C)C)c[nH]3)=O)C2)=O)c(C)o1 74500,CC1CCC(CNC(c2cc(Cl)c(Cl)s2)=O)N(C(c2cnn(C)c2C2CC2)=O)C1 74501,N1(C(C2(CO)CCCC2)=O)CCCC2(CN(CCN3CCOCC3)CCO2)C1 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74819,c1(SC(C(=O)N(C2CCN(C(c3nc(C)nn3C)=O)C2)CC)C)ccccc1C 74820,c1(C(=O)OC(c2ccc(Cc3ccc(Cl)cc3)cc2)C)cc2c(F)cccc2s1 74821,N1(C(C(C=C)CC)=O)CCC(C)(C)C1C(=O)NC1(c2ccncc2)CC1 74822,N1(C(C(CC#C)C2CC2)=O)CCC(C)N(C(c2ccc3nnnn3c2)=O)CC1 74823,c1(OC)n[nH]c(C(N2CC3CC3(NC(c3ccc(NCCO)cc3)=O)C2)=O)c1Cl 74824,C1(CNC(c2cc(C3CCOCC3)no2)=O)CC(NC(C2CCCO2)=O)CC1O 74825,N1(C(CSCC(C)C)=O)CCC2(CC1)CN(C(=O)CC1CCOC(C)(C)C1)C2 74826,C(=O)(C(C)C(C)(C)C)N1CC(CNC(Cc2c(C)ocn2)=O)C(C)C1 74827,c1(C(N2CCN(C(C(N3C(CC)CCC3C)=O)=O)CC2)=O)cc(C)c(=O)n(C)c1 74828,Cc1cc(C(=O)NC2CCC(NC(C3(CC(F)(F)F)CC3)=O)C2)ccn1 74829,C(CN=C(NCc1cc(C(C)(C)C)no1)NC(C)CC(F)(F)F)OCC=C 74830,C(=O)(C(C)(C)c1nccs1)N(CCNC(=O)CCSCC(N)=O)CC 74831,n1(CC(=O)NCCC2CN(C(Cc3ncc(C)[nH]3)=O)C2)cc(C#N)cn1 74832,C1(NC(C(n2ncc(C)c2)C)=O)CCN(C(c2cc(Cl)ccc2N)=O)CC1F 74833,c1(C(=O)NC2CN(C(=O)C(O)C3CCC3)CC2O)ccc2nc(C3CC3)oc2c1 74834,C(CC1=CCCCC1)N(CC(=O)NC1C2CN(C(=O)CCSC3CCC3)CC12)C 74835,C12(NC(C(c3ccc(F)cc3)CC)=O)CCCC(NC(C3CCN(C)C3)=O)(C1)C2 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74888,c1(CC(=O)NC2CCN(CCCC)C2)ccncc1C 74889,Cc1ccc(C#N)cc1C(N1CC(C)(CCC(=O)N(CC(O)CO)CCO)C1)=O 74890,c1(C(N2CCC(O)(CN(C(C3CCC(=C)CC3)=O)C)C2)=O)cc2ccsc2n1C 74891,C1(CNC(C2C(OCC)C2)=O)CN(C(=O)CS(=O)(=O)NC)C2CCCC2O1 74892,C12(C(N(CCCOC)Cc3cccs3)=O)C(NC(=O)COC)C3CC1C2C3 74893,Cc1c(C(=O)NC(C2CCN(C(c3occ4c3CCC4)=O)CC2)C)cncc1Cl 74894,c1(C(=O)NCCC(CNC(c2c(C)n(C)nn2)=O)O)cc(C(F)F)ccc1F 74895,c1(N(CC(C)(F)F)C)nc(N2CC=C(c3cccs3)C2)nc2ccccc12 74896,n1(C(C)C)cnc2c(NCC3(C)CS(=O)(=O)C3)[nH]c(=NC3CCCCC3C)nc12 74897,C1(S(C)=O)(C(=O)OC(c2c(Br)cnn2C(C)C)=O)CCN(CC)CC1 74898,Cn1c(=O)n(CN2CCCC(C(N)=O)C2)c2cc(ON3CCCC3)ccc12 74899,C(CNC(N1CCCC(CCCC(=O)OC(C)(C)C)C1)=O)(CC(C)C)OC 74900,c1(CC(C(=O)N(C2CCN(C(COCC(=C)C)=O)CC2)C)=O)ccc(Cl)cc1 74901,c1(C(=O)OC)nc(Cl)cc(=NC2CC3CN(C(c4ccc5nn[nH]c5n4)=O)CC23)[nH]1 74902,C1(NC(C(CC)=CC)=O)CCCN(C(=O)CCCC(C)N(C)C)C1C 74903,O=C(C1CCc2ccccc21)NCC1CCCC1NC(C1CCCS1(=O)=O)=O 74904,c1(C(N2C(CNC(CC(C(=C)C)O)=O)CC(CC)C2)=O)ccsc1S(N)(=O)=O 74905,N1(C(C23C(CN(C(c4cn5ccccc5n4)=O)C2)C3)=O)CCCC(F)C(F)(F)C1 74906,c1(C(=O)OCCN2CC3CCC2C3)cc(COC)cc(C(=O)OCCOC)c1Cl 74907,C1(C(N2CC(OCCCCC)C2)=O)C=CCN1C(=O)Cn1ccc(C)n1 74908,C1(NC(c2ccc(-c3nc(C)sc3)cc2)=O)CCN(C(=O)C(C)C)C12CCC2 74909,C1(OC)CN(C(C2CCCOCC2)=O)CC1NC(=O)CSc1ccccc1O 74910,CCC(C(=O)N(C1(CC(=O)NCCCSCCO)CC1)C)n1cncn1 74911,N1(C(c2c(CC)ccs2)=O)CCC(C(N2CCCC(C(C)C)C2)=O)C1C(C)C 74912,c1(NC(C2C3(CN(c4nc(SC)c(F)cn4)C3)C2)=O)cc(F)c(C#N)cc1F 74913,C=C(Cl)C(C)(C)C(=O)NCCC1CC(NC(c2cnc(C3CCOC3)s2)=O)C1 74914,c1(C(=O)NC2C(NC(CCSC)=O)CS(=O)(=O)C2)ccc2ncn(C)c2n1 74915,C1(CC)CN(C(=O)CCCN(C)C)CCC1NC(C1(F)CCCC1)=O 74916,C1(CCCNC(COCCC=C)=O)CN(C(c2cnc(NC)s2)=O)CCO1 74917,N1(C(c2ccnc3[nH]nnc23)=O)CCC2CCC(C1)N2C(C1CC=CCC1)=O 74918,N1(C(c2cc(OC)ns2)C(=O)NCCCC2CC2)CCCc2c(C)cccc21 74919,C(C(C)(C)CCC#N)(c1n(CCCC)nnn1)NCc1cc(OC)cc(C)c1 74920,n1(CCCC)ncc(C(=O)NCCCC2(NC(C3CC4(CC4)CO3)=O)CC2)c1C 74921,C1(NC(c2ccc(-n3cccc3)nc2)=O)(CO)CCN(C(c2ccno2)=O)CC1 74922,C(=O)(CC(F)(F)C(F)F)NC1CC(C(C2CC2)(C)NC(c2c(C)nc(CO)s2)=O)C1 74923,C1(CC(=O)N(CC)Cc2nc[nH]n2)(NC(c2nonc2N)=O)CCCCC1 74924,C(=O)(CC(C(F)F)c1ccc(F)cc1)N(C1CN(C(=O)Cc2cnco2)C1)C 74925,n1(CCCC)nc(C)c(C=CC(=O)N(CC(C)(C)NC(=O)CC(C)(C)O)C)c1Cl 74926,C(c1ccc(OCCO)cc1)=CC(=O)NC(n1ccnc1)C 74927,N1(C(C(CC)CC2CCCCC2)=O)CC(C)(CNC(C2(O)CC2)=O)CC1(C)C 74928,C1(C(=O)Nc2cncc(C(=O)OC)c2)CC12CCN(C(=O)C1=CCCCO1)C2 74929,N1(CCCC#C)CC(C)(C)CC(C)(C)C1 74930,C1(F)(C(=O)NCCNC(CC(C)OC)=O)CCS(=O)(=O)C1 74931,C1(C(=O)NCC)CCN(C(c2nc(OC)c(C)s2)=O)C1(C)C 74932,N1(C(C)C)CC(C(=O)NCC2CC(C)N(C(=O)C(C)CSC(F)(F)F)C2)CC1=O 74933,CCCC(C(C)(C)C)NC(=O)CCC1CCN(C(=O)Cc2csnn2)CC1 74934,N1(C(C)C)CC(C(=O)N(C)CC2(NC(C3CC(CCO)C3)=O)CC2)CCC1=O 74935,C1(C(=O)NC2C(NC(C3CC4CCC3C4)=O)CCC2)CCC(F)(F)CC1 74936,c1(OC)ncc(Cl)cc1C(=O)NC1C2CC1N(C(C1CC3CC3C1)=O)C2C 74937,N1(C(C(C=C)OC)=O)CC(O)CC1CNC(C1(SC)CC1)=O 74938,N1(C(c2c(CC)cco2)=O)CCCC1C1CCCN1C(=O)Cc1c[nH]nc1O 74939,c1(C(=O)NC2(C(N(CCSC)C)=O)CCC2)c[nH]c(=S)cn1 74940,C=CCC(CC(=O)NC(C)C(C)(C)OC)NC(=O)COC1CCOCC1 74941,C(=O)(CC(c1ccccc1)N(C)C)N(C)CCOCCN(C)C(C1CCCS1)=O 74942,c1(C(N2CCC(NC(C3N(C(C)=O)CCCC3)=O)(CO)C2)=O)cc(N)ccc1O 74943,C(=O)(C1CCCc2nncn21)N(C)CCOCCNC(c1cn(C2CC2)nn1)=O 74944,Cc1cnc(C)c(NS(=O)(=O)Cc2ccccc2NC2CC(F)C2)n1 74945,c1(C(=O)NC(C2(C(F)F)CC(=C)C2)=O)ccc2c(c1)CN(C(=O)CC1CCCCO1)C2 74946,C(=O)(CC1=NNC(=O)C1)N1CC(NC(c2cnccc2C(F)F)=O)C(O)CC1 74947,C1(C(C(=O)NC(CC)C)N(CCCCO)C)C2CCOCC12 74948,N1(C(C2C(OC)C2)=O)CCCC1C(C)NC(=O)C(C)(C)SC 74949,C(c1ccc(C)cc1)=CC(=O)NC(CC)CNC(=O)C(C#N)=CC1CC1 74950,CC(CCCCNC(=O)CC1CCC(F)(F)C1)NC(C1(C)CC1)=O 74951,N1(C(c2cnn(C(F)F)n2)=O)CCN(C(c2ccc(F)cn2)=O)C(CC(F)(F)F)C1 74952,C1(CC)(CC)CC(NC(=O)C(C(C)(C)C)SC)CN1C(=O)CCC=C(C)C 74953,c1(OC)nscc1CNC(=O)COCCNC(=O)Cc1ncoc1C 74954,C1(F)(C(=O)O)CCCN(C(=O)CN(C(C)(C)C)C2CC2)CC1.CC(C)CC1C(=O)N1 74955,N1(C(c2cn(CC=C)nn2)=O)CCC(F)C(NC(c2cc(C3(C)CC3)n[nH]2)=O)C1 74956,c1(C(N2CCC(C(c3ccccc3)C)C2)=O)[nH]nc2c(=O)n(C)cnc12 74957,c12cccc(c1)CN2CC.c1(SC(c2cc(C)c[nH]2)C)ccncc1 74958,c1(C(N(CCCCN(C)C(c2cc(=O)n(C)cn2)=O)C)=O)ccc(F)c(O)c1 74959,CCCCC(CNC(C1CC1(C)C)=O)NC(=O)CCCN(C)C(=O)OC(C)(C)C 74960,Cn1cc(C(C(=O)N2CCCC2)NCC(=O)NCCC(C)(C)O)nn1 74961,c1(NC)cc(Cl)ccc1C(N1CCCC(O)(CN(C(=O)C(C)N(C)C)C)C1)=O 74962,N1(C(c2c(C)noc2)=O)CCOC2CCN(C(c3ccc4ocnc4n3)=O)CC12 74963,CCC(CC)C(C)NC(c1ccoc1CNC(C1OC2CCC1C2)=O)=O 74964,Cn1ncc([N+](=O)[O-])c1C(=O)NC1CCCC(NC(=O)C=CCF)CC1 74965,c1(C(=O)NCCC(C(C)C)NC(c2c(CC)nc[nH]2)=O)cccc2oc(O)nc12 74966,c1(C(=O)NCCC(C)CCNC(=O)CCc2cnc[nH]2)ccc(F)cc1Cl 74967,CCCC(O)C(=O)N1CCC(C2N(C(=O)C=CC3CC3)CC2(C)C)CC1 74968,C1(NC(C2C(C(=O)OC)C2(C)C)=O)CCC(C)N(C(c2ccc(F)c(F)c2)=O)C1 74969,C1(C)(C(=O)NCC(=O)OC)C=CCCN1C(=O)CCc1cccnc1C 74970,c1(C(N(CCN(C(C=C(C)c2cccs2)=O)C)C(C)C)=O)cnn2c(=O)cc[nH]c12 74971,C(C(C)C(C)C(=O)NCC1(NC(=O)CCCc2nncn2C)CCOCC1)OC 74972,C1(NC(=O)Cc2ccc(Cl)cn2)CC2CC(NC(=O)CC3(C4CC4)CC3)C2C1 74973,c1(C(=O)NCCC(=C)CNC(C2OCC3CCCC2C3)=O)c(C)cc(C)nc1O 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75043,CCCCC(O)CC(=O)NCC1(O)CC(NC(=O)CCCOc2ccc(C)cc2)C1 75044,C1(C)(NC(C(CCC)C)=O)CCN(C(=O)C(C2CCC2)OC)CC1 75045,c1(C(N2CCN(C(C3(CCC=C)CC3)=O)CC2)=O)c(Cl)ccc(OC)c1N 75046,Cc1cc(=NCC(CC2CC2)C(C)C)[nH]c(=NCC(C)Cc2cn[nH]c2)[nH]1 75047,N1(C(C(C(CC)C)O)=O)CCCC2(C1)CN(C(C1CCCN(C(C)=O)C1)=O)C2 75048,C1(C(N(CC(C)NC(=O)CCC(=O)c2ccc(Cl)cc2)C)=O)CCC2CCC1O2 75049,C1(C(=O)OCC2(c3ccccc3)CCCC2)CC(=O)C12CC2 75050,N1(C(C2(F)CCN(C(c3cc(C(C)=O)on3)=O)C2)=O)C2CCC1COC2 75051,Cc1cc(N)nc(CN)n1.c1(C(=O)NC2(O)CCC2)cc(Cl)nc(C(C)(C)C)n1 75052,C1(CNC(C=C(C)C2CC2)=O)(CNC(=O)C(C)OCC2CCCO2)CCCC1 75053,C1(CNC(c2cnc(C)s2)=O)CCN(C(=O)CC2CC(CF)C2)C1(C)C 75054,c1(C(N(CCCOC)CC)=O)ccc(CO)cc1.C(C)(C)(C)N 75055,C12(C(=O)NCCC3CN(C(C4(CC5CC5)CCC4)=O)C3)CCC3CC1C2C3(F)F 75056,N1(C(CCN2CCC(C)CC2)=O)CC(NC(C2CCOC2)=O)C2(CC2)C1 75057,C1(CC(=O)N(CCNC(C(COCC)C)=O)C(C)C)COC2(CCC2)CO1 75058,C1(C(C)=O)CN(C(=O)C(F)=CCCF)CCC1C.c1(C(=O)NC)ccoc1 75059,CC1CC(NC(=O)NCc2ncccc2C2CC2)CN(C(=O)OC(C)(C)C)C1 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75077,Cc1c(CC(CNC(=O)C(=O)N)CO)cccc1Br.c1(C(=O)O)cn(C)c(C)n1 75078,N1(C(c2nc(C(C)C3CC3)oc2)=O)CCC2(CC1)CN(C(=O)C=C1CC1)C2 75079,N#Cc1ccc(C(N2CCCC2C2CCN(C(=O)CCF)C2)=O)cc1Br 75080,C1(C(=O)NCc2cc(C(=O)NCC3(COC)CCCC3)n[nH]2)CCC(O)CN1C 75081,C(=O)(CC(C)C1CCCO1)NC1(C(N(CCF)CC)=O)CCC1 75082,C(=O)(C(=O)N=S(C)(C)=O)NCCC1(CNC(C(C)CC2CC2)=O)CC1 75083,Cn1nc(O)cc1NC(C1(CCNC(c2nnsc2N)=O)CC1)=O 75084,C12(NC(C=CSC)=O)CCCCCC1N(C(c1cc(F)c(N)cc1F)=O)CC2 75085,C1(C(=O)OC)C=CC(C(=O)NCC2CN(C(C)=O)C2)C1.c12c[nH]nc1CNC2=O 75086,c1(CC(=O)N(CC(C)(C)NC(=O)CCC2(C#N)CCC2)C)ccccc1CS(N)(=O)=O 75087,C#CC1CN(C(=O)C(C2CCCO2)NC(=O)CCN2CCOCC2)CCO1 75088,c1(CCC(=O)N(CC(C)NC(C=CCCC=C(C)C)=O)CC)nc2ccccc2[nH]1 75089,N1(C(C(C)OCCOC)=O)CCC2(CCCN(C(=O)CCCN(C)C3CC3)C2)CC1 75090,n1(CC(=O)NCCN(C(=O)CC2(C(F)(F)F)CC2)CC)c(=O)oc2ccccc12 75091,Cc1ccc(C(C)C(C)NC(=O)NCc2ccc[n+]([O-])c2)cc1 75092,C1(C)(CCNC(CCC(C)CN(C)C)=O)CCCN(C(=O)OC(C)(C)C)C1 75093,c1(CNCc2n(CC(C)C)ncc2)cc(F)c(Cl)cc1F 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75147,S(=O)(=O)(c1ccc(=NC2CS(=O)(=O)CC2O)[nH]c1)N1CCCC(C(N)=O)C1 75148,c1(CC)ncncc1C(=O)NC1CCC(CNC(=O)CNC(=O)CCC(C)C)CC1 75149,c1(COC)nc(=NC(=O)Cc2ccc(F)cc2)o[nH]1 75150,N1(C(C23CCC(F)(CC2)C3)=O)CC(NC(C2CC(n3ccnc3)C2)=O)C2(CC2)C1 75151,C1(NC(C2CCC(C)O2)=O)CC2CCC1CN(C(c1nc(CN)cc(O)n1)=O)C2 75152,O=[N+]([O-])c1ccnn1-c1ccc(Cl)c(Cl)c1.c1cnnc(Cl)c1 75153,Cc1ccc(C(N2CCC(C)(C)C2C(N2CC(CO)C(C3CC3)C2)=O)=O)cc1O 75154,c1(C(N(C2CCN(C(C=CC=CC)=O)C2)C)=O)ccc(C#N)n1C 75155,C1(NC(C2=CCSC2)c2n(CCC3(C)CC3)nnn2)CCOC2(CCCC2)C1 75156,CN1CCOCC1C(N1CCC(C)(C(=O)NC2(C3CC3)CC2)C1)=O 75157,C1(N(C)C(C23CC(F)(C2)C3)=O)CCN(C(C2CCC(N(S(C)(=O)=O)C(N)=O)C2)=O)CC1 75158,c1(CC(=O)NC(C2CCN(C(=O)Cc3cnc[nH]3)CC2)(C)C)ccc(=N)[nH]c1 75159,C(C(CC)(CC)C(=O)NC(C)CC1(O)CCC1)N(C(Cc1cn(CC)nn1)=O)CC 75160,N1(C(C(COC)NC(=O)CCc2csnn2)=O)CCS(=O)C(C)C1 75161,c1(CC)ccc(Cl)c(C(=O)NC2CCC(NC(=O)C(CC)SC)CC2)c1 75162,Cc1ccc(C(N)=O)cc1CNC(=O)C(=O)NC(c1cc(Cl)sc1Cl)(C)C 75163,c1(CC(C)C(=O)NCCC(C)N(C(=O)CCc2ccccn2)C)ccc(F)cc1 75164,N1(CCCCCCCCN2CCNC(=O)C2=O)CCS(=O)(=O)N2CCCC12 75165,C(N=c1[nH]c(N(C)CCc2ccccc2Cl)nc2cc[nH]c12)c1c(CC)nco1 75166,N1(C(C(CC)CCOC)=O)CCC2(C1)CN(C(=O)C(C)(O)CCc1ccccc1)C2 75167,C1(NC(c2c(C)cc(C)o2)=O)CC2(C1)CN(C(=O)Cc1cn3ccsc3n1)C2 75168,CCC(CC)(C(=O)NC1CC(C)N(C(C2CCCCC2O)=O)C1)OC 75169,C1(C)(CNC(c2c(CC)n(C)cc2)=O)CCN(C(C2CC(=C3CC3)C2)=O)CC1 75170,c1(C(=O)NCCN(C(=O)CC(=O)N(C)C)CC)c(Cl)c([N+](=O)[O-])nn1C 75171,C(=O)(C(C#N)C(C)C)NC(C(=O)NCC=CCOC)c1ccco1 75172,c1(Cn2cncn2)cccc(F)c1C(N1C(CNC(c2cc(Cl)no2)=O)CC1)=O 75173,CCCC(C(=O)NC12CCCN(C(=O)Cc3cccc(Cl)c3)CC1C2)S(N)(=O)=O 75174,N1(C(C(C)OCC=C)=O)CCC2(CC1)CN(C(c1cc(Cl)cs1)=O)C2C(C)C 75175,C1(O)(CNC(=O)C=C2CCOCC2)CCN(C(=O)CC2CSCCS2)C1 75176,C1(NC(CCCCCOC)=O)CCN(C(=O)C(O)CC(C)(C)C)CC12CCC2 75177,C1(NC(C(CCC)=CCC)=O)CCC2CC1CN2C(c1ncccc1NC)=O 75178,Cc1nc2ccc(F)cn2c1C(N1CCN(Cc2ccc(Cl)nn2)C(CO)C1)=O 75179,C#CC1(O)CCN(C(=O)COCCNC(=O)Cc2nccn2C)C1 75180,Cc1cc(C(=O)NCCCOCCNC(C2CC2(C)C)=O)nnc1O 75181,C#CCC(C)C(=O)NC1CCN(C(C2CCCC2)=O)C1 75182,c1(OC)cc(C(=O)NCCCCC(C)NC(C2CCN(C3CC3)CC2)=O)ccn1 75183,Cc1ncc(F)c(NC(=O)C(N2CCC(CCNC3(CF)CCOCC3)C2)C)n1 75184,C1(C(=O)NC2C(CNC(C(C)(C3CCOCC3)OC)=O)C2)CCC(N(C)C)CC1 75185,Nc1ccc(C(N2CC3CCC2C3NC(C2CCC23CCC3)=O)=O)cc1Cl 75186,c1(C(=O)NC2C(NC(=O)CC3CC3C(F)(F)F)COC2)cc2c(Cl)cccn2n1 75187,C1(NC(Cc2cn(CC)nn2)=O)C=CCN(C(C23CC2C3)=O)C1 75188,C(=O)(C(C)(C)CCOC)N1CC(CCC)C(C(=O)N(CCCCCO)C2CC2)C1 75189,C1(c2nc(COCC)nn2-c2ccnc(C(F)(F)F)c2)CCc2cn(C)nc2C1 75190,c1(CC)n[nH]c(=NC2CCCC(CNC(=O)C(C)CF)C2)s1 75191,c1(C(N(C)C(c2ccc(C(F)F)o2)=O)=O)ccn(C)n1.c12cn(nn1)CCNC2=O 75192,C12(C(N(CCC(C(C)C)NC(=O)C=C3CCCC3)C)=O)CCN(CC1)S(=O)(=O)C2 75193,c1(C(=O)NCCC2CN(C(c3ccccc3)=O)CC(C)O2)cccc2nncn12 75194,CCCC(C(=O)N(CC(O)CN(C)C)C)NC(=O)C(C)NC(=O)C1CC1 75195,Cc1ccc(C2CC2)c(-c2cccc(C(N3CCC(n4cccn4)C3)=O)c2)c1 75196,C1(C)(CNC(C(CCC)C)=O)CC(F)(F)CN1C(=O)C(C(C)C)NS(C)(=O)=O 75197,C(CCCC(C)NC(=O)CC1CNC(=O)C1)NC(c1n(CC#C)cnn1)=O 75198,Cc1ccccc1C(C)N(CC(C)NC(=O)C(F)C1CCC1)C 75199,C(C)(N=c1cc(C)nc(CO)[nH]1)C1CCCN(C(Cc2ccc(OC)c(F)c2)=O)C1 75200,C#Cc1ccc(NC(C2CCN(C(=O)c3ccccc3C)O2)=O)c(C)c1 75201,c1(C(=O)NCC2C(NC(CC(n3c(CC)ncc3)C)=O)C2)cccn2ccnc12 75202,N1(CC(=O)OCCNC(C2CCOC2)C#C)CC(C(F)(F)F)CCC1=O 75203,C1(C#N)(CN(C(=O)CCC(=O)c2cccs2)CC2C(C)C2)CC2(CC2)C1 75204,c1(-c2ccc(C)o2)ccc(S(=O)(=O)N2CCCC2Cc2ccccc2)cc1 75205,N1(C(C2CN(C(C)=O)C2)=O)CCC2(CC(NC(c3ccc(Cl)nc3Cl)=O)C2)C1 75206,c1(SC)ccc(Br)cc1NCc1ccnc(-c2ccoc2)c1 75207,CCC(CN=c1[nH]c(=NCCCc2cc[nH]n2)[nH]c2c1CCC2)C(C)(F)F 75208,n1(CCOC)ccc(C(=O)NCC(C(C)C)N(C(=O)C(C)OCOC)CC2CC2)n1 75209,c1(C(=O)NCC=CCC(=O)N(CCC)Cc2ccnn2C)cccc(F)c1C 75210,N1(C(C(CNC(=O)CC(C)C2CC2)OC)=O)CC(CO)C(C)C1 75211,N1(C(C(CCC)NC(N)=O)=O)CCOC2(CCCN(C(=O)CCF)C2)C1 75212,c1(C(c2ccccc2)C(=O)NCC2CCCN2C(=O)C=CCBr)cccc(F)c1 75213,C1(C(=O)NCC2N(C(C)(C)C)CC2)CN(C(C2COC(=O)N2)=O)CC1C1CC1 75214,N1(C(C(C2CCC2)NC(c2cc(C)nn2C)=O)=O)CC2CC2C2CC12 75215,CC(CC(=O)N1CCCC(N(C(=O)CCCn2ccccc2=O)CCF)C1)C(F)F 75216,c1(-c2cc(CNc3ccc(F)c(F)c3)ncc2)cncc2cnccc12 75217,Cc1nc(O)c(C(=O)NC23CC(C2)N(C(=O)CC(O)C(C)C)C3)nc1C 75218,CC1(C)CCCC1(CO)NC(=O)CNC1CCNC(c2ccccc2)C1 75219,c1(C(=O)NCCCCC(C)NC(C2CCCO2)=O)ccc(N)c(Br)n1 75220,N1(C(c2cccc(CNC(C3(C)CCCNC3=O)=O)n2)=O)CCOC2C(O)CC12 75221,N(C1COCc2ccccc21)C(C#CC(C)(C)C)C(=O)NC1CC1 75222,C1(C(N2CCN(CC3CCC3)CC2)=O)COc2ccc(Br)cc2C1 75223,N#Cc1cnc(NC(C2CCC(NC(=O)C(F)(F)F)C2)=O)nc1 75224,S(=O)(=O)(c1c[nH]c(C(=O)NC2CC(NC(=O)C(C)(C)SC)C23CCC3)c1)NCC 75225,n1(CC(=O)NC2CN(C(CC3(OC)CCC3)=O)C2)nc(C)c2cccnc12 75226,c1(CC(=O)NC(C(C)OC)CO)cc(C)cc(Cl)c1 75227,c1(C(=O)NCC(C)N(C)C(c2cccc(N)c2N)=O)cc2sccc2cn1 75228,c1(C(=O)NC2CC(CNC(c3c(C)nccc3)=O)C2)cn2ncccc2n1 75229,C1(CC#C)CN(C(C2CC(CNC(=O)C(CC)N(C)C)C2)=O)CCO1 75230,c1(CC)cc(C(N2CC(NC(=O)Cc3[nH]cnc3C)C3(CC3)C2)=O)cn(C)c1=O 75231,c1(C(=O)NC(CC=C)CNC(c2nccnc2N)=O)cn(C)c(=O)cc1C 75232,CC1C=C(C(=O)N2CCCCC(NC(c3sccc3CO)=O)C2)CC1 75233,N1(C(=O)COC2CC2)CCC2CC12C(=O)NCC1(CC2CC2)CCC1 75234,C(=O)(C(CO)C(C)(C)C)NC1CCC(NC(C(C)(C)N(C)C)=O)C1 75235,C1(NC(C2C(CCOCCCC(C)C)C2)=O)CCn2cncc2C1.C(=O)N 75236,c1(CC)nccnc1C(=O)NC1CC(CNC(=O)CCn2cnc(=N)[nH]2)C1(C)C 75237,C1(C2CCN(C(c3ccccc3Cl)=O)C2)(NC(=O)Cc2ccno2)CC1 75238,C1(C(N2CCC(CN(C(c3nc(C)sc3)=O)C)C2)=O)CCCS(=O)(=O)C1 75239,Cc1cnn2ccnc(C(=O)CCNc3ccc([N+](=O)[O-])cc3Cl)c12 75240,C1(C(N(CC)CC2CCCN2C(=O)C(C)C)=O)C2CN(c3nnc(C4CC4)s3)CC12 75241,c1(N(C(c2c(COC)noc2)C(=O)NCC2CC2)CCF)cncn(C)c1=O 75242,CC(C)(C(=O)N1CC(OCCNC(C23CC(F)C2C3)=O)C1)n1cccn1 75243,c1(C(N(CCN(C(CC2C(OCC)CC2)=O)C)C)=O)cc(C(C)(F)F)on1 75244,CCN(CCNS(C)(=O)=O)N1CCC2(C=CCO2)C1 75245,CC(C(=O)NC1CCCC(CNC(c2nccnc2-n2ccnc2)=O)C1)C(F)F 75246,CC1CN(C(=O)CCN(C)C)CCC1N(C)C(C1CCCO1)=O 75247,CC1CC(=O)NC1C(=O)NCC(C)(C)NC(=O)CCN1CCOCC1=O 75248,C(=O)(C1CCCc2ncc(C)n21)NCC(C)N(C(c1cc(C(N)=O)c[nH]1)=O)CC 75249,C12(C(=O)OC)CC(CO1)N(C(C1(NC(c3ccncc3F)=O)CC1)=O)C2 75250,CS(=O)(=O)c1cnc(NC2CCC(NC(C3(S(N)(=O)=O)CC3)=O)C2)c(Cl)c1 75251,Cc1cccc(S(=O)(=O)Oc2ccc(C(=O)C(C)C)cc2[N+](=O)[O-])c1Cl 75252,Cc1cc(C(=O)NCCC2CCN(C(=O)C(C)SC(C)C)C2)c(Br)cn1 75253,N1(C(C2CCC(CC)O2)=O)CCC(C(C)NC(C2CSCC(=O)N2)=O)CC1 75254,c1(OC)cc(C(=O)NC23CC(C2)N(C(C2(CC4CC4)CCCO2)=O)C3)ccc1Cl 75255,C(CC(C)C)(C(=O)NC(C)CCN(C)C)NC(CC=CCCCCC)=O 75256,Cc1cccc(C)c1CC(=O)NC(C1CCCN(c2nnc(C(F)F)o2)CC1)C 75257,C1(C(F)F)(NC(C(C2CC2)OC)=O)CC(NC(=O)CC2CCCOC2)C1 75258,CCCC(C#N)C(=O)NCC1C=CCN1C(c1ccc(COC)nc1)=O 75259,CC1(C)CCC(C)(NC(C2CCCN(C(=O)CN3CCC(=O)CC3)CC2)=O)C1 75260,c1(C(=O)NC(CCNC(C(C)SCCCC)=O)(C)C)cccc(OC)c1N 75261,c1(CNC2C=CC(C(=O)Nc3ccc(C=C)cc3)C2)ccc(F)c(C#N)c1 75262,c1(OC)ccc(C(=O)NNC(=O)NCCCN(C(C)C)Cc2ccccc2)cc1O 75263,c1(CC(N2CCC(CCC(=O)NC3CC(C(C)O)C3)C2)=O)coc2ccccc12 75264,C(=O)(C1=CCCCO1)NCCCC(=O)NC(C1CCC1)C 75265,C1(NC(C=C(C)C)=O)CC(C)CN(C(c2cc(C)cc(O)n2)=O)C1 75266,C(CC(C(=O)N1CCC(O)(N(C(=O)CSCCN(C)C)C)C1)N(C)C)SC 75267,c1(OC)c[nH]c(C(=O)N(C)CC2(O)CCN(C(=O)CC3CCC3(C)C)C2)cc1=O 75268,N1(C(CSCCCC)=O)CCC(C(=O)Nc2cn(CC)nc2C#N)CC1(C)C 75269,c1(C(=O)NC(C(C)NC(c2n(CC#C)ccc2)=O)C)nc(=N)[nH]c2ccccc12 75270,C1(C)(C(N(CCCCNC(CCOCCCOC)=O)C)=O)CC(C(F)(F)F)C1 75271,C(=O)(CC(CCCC)NC(c1ccoc1C1CC1)=O)NCC(C=C)O 75272,N1(C(C(C)n2cncn2)=O)CC2CCN(C(C3CCCCC3(C)C)=O)CC2C1 75273,C(=O)(C(F)(F)C(O)C1CC1)N1CCC(O)(CNC(c2c(OC)n[nH]c2)=O)C1 75274,C(=O)(C(C)(CC)C(N)=O)NCCN(C(C1(CC)CCOC1)=O)Cc1ccccc1 75275,CC1(C)CN(C(=O)Cc2csc(Cl)c2)CC1NC(=O)CC1CCOC1=O 75276,C1(NC(C(CCN(C)C)O)=O)CCC2(CC1)CC(NC(=O)CSc1cccs1)C2 75277,C1(NC(CCN(C(C)=O)C)=O)C(C)CN(C(=O)CSC2CC2)CC1C 75278,N1(C(C(n2ccc(C)n2)C)=O)CCC2(CCC2)C(NC(=O)C(C)Cn2cccn2)C1 75279,N1(C(c2oc(C)c(Br)c2)=O)CCC(NC(C2CC23CCC3)=O)C12CCC2 75280,c1(OC)cncc(C(N2CCC(C(N3CCC(F)(CO)C3)=O)(OC)C2)=O)c1 75281,Cc1nc(C(=O)NC2CCN(C(=O)CC3NC(=O)NC3=O)C2)ccc1[N+](=O)[O-] 75282,N1(C(c2c[nH]c(=NC)s2)=O)CCCN(C(=O)C(C)C(F)(F)F)C(CO)C1 75283,Nc1cc(Cl)nc(C(=O)NC2(CNC(c3cccnc3)=O)CCC2)c1Cl 75284,c1(CNC(CCOC(C)C)=O)cc[nH]c1C(=O)NCC1(C)CC1(Cl)Cl 75285,CC1(NC(C2(CO)CCCO2)=O)CN(C(c2cn(C3COCC3F)nn2)=O)C1 75286,Cc1cc2ccc(C(=O)NC3CCC(NC(=O)C#CC4CCCO4)C3)cn2c1 75287,c1(C(=O)NCC2(CN(C(=O)C=C3CCCC3)C)CC2)cnc2ncccc2c1 75288,N1(C(C(C)(CO)NC(C2C(C=C)OCC2)=O)=O)Cc2ncsc2C1 75289,C1(CC)CN(Cc2cc(O)ccc2Cl)c2ccccc2O1 75290,C1(CCC)(NC(=O)C(c2ccccc2Cl)C)CCCN(C(=O)C2=COCCO2)C1 75291,C12(NC(c3cnc(CC)s3)=O)CCCC1(F)CN(C(C1CCC(C)(C)OC1)=O)C2 75292,N1(C(CCn2cc(C(C)=O)nn2)=O)CCCC(n2cc(CN(C)C)nn2)C1 75293,CN1CCN(CCc2nc(-c3ccccc3)n(CCc3ccc(Cl)s3)n2)CC1 75294,Cc1cccc(NNC(=O)C2(n3cc(CN4CCCCC4)nn3)CC2)c1Br 75295,c1(C(=O)NC2(C3N(C(C(C)OCC)=O)CCC3)CC2)ccc(C(F)(F)F)c(O)c1 75296,n1(CCNC(C2C(C(=O)OC)C2)=O)cc(CNC(=O)Cn2cc(C)cn2)nn1 75297,N1(C(CC(C)F)=O)CCC(C)(C(=O)NCC(N2CCCC2)=O)CC1 75298,C1(C(=O)NC(CN(C(c2cc(CC)on2)=O)C)CC)CCc2cnn(C)c2C1 75299,N1(C(=O)COc2ccccc2)CC2CC1CCC2NC(C1(CCOC)CC1)=O 75300,N1(C(C2(COC)CCCCC2)=O)CC(C2CCCN(C(=O)C(C)S(N)(=O)=O)C2)C1 75301,C1(NC(C(c2cnn(C)c2)NC(C(CC)(C)C)=O)=O)(CO)CC2(CCC2)C1 75302,c1(C(=O)NC2(CC(=O)NCCO)CC2)ccn(-c2ccncc2)n1 75303,C(=O)(CCC(C)c1ccccc1)N(CCCN(c1snc(CC)n1)C)C 75304,c1(NC2CCN(CC(F)(F)F)C2)nc2c(c(=NC3CC3)[nH]1)COCC2 75305,N1(C(COCCC)=O)CC(CNC(=O)C2=CC(C)(CC)C2)C2(CCC2)C1 75306,CC1CCC(C)(C)N1C(C1CC(NC(c2csc(Cl)n2)=O)C(O)C1)=O 75307,C(=O)(CC1=NNC(=O)C1)N(C1CCCN(C(=O)CN2CCCS2(=O)=O)C1)CC 75308,N1(C(C(F)=CCC)=O)CCOC(C(=O)NCCc2noc(=O)n2C)C1 75309,CC(C)CC(CNC(=O)C(N1CCN(C)CC1)C)NC(=O)CC1(O)CCC1 75310,CC(C)CCN=C(NCc1ccc(N2CCC2)cc1)NC1CC(=C2CCC2)C1 75311,c1(C(N2CC3(CCN(C(CCOCCOC)=O)C3)C2)=O)nc2nccc(C)n2n1 75312,C(CN=c1cc(CN2C(=O)CCC2=O)nc[nH]1)N(C(c1cnn[nH]1)=O)CC 75313,c1(N(C(=O)COC(F)(F)F)C)cc(C(F)(F)F)nc(N2CCCCC2CCO)n1 75314,Cc1cc(=NCC(CC(C)C)N2CCCC(C)C2)[nH]c(N(CCC(C)C)C)n1 75315,C1(CNC(c2oc(CC)c(C)c2)=O)COC(C)(C)CN1C(=O)CN1CCCC1=O 75316,N1(C(CCC(=O)Nc2ccc(F)cc2)=O)CCC23CCCCC2(C1)C3(F)F 75317,c1(C(COC(C(C(CC)O)C)=O)=O)ccc(S(=O)(=O)CC)cc1.C1C(=O)N1 75318,C1(C(=O)NC(C)CCNC(c2cnsc2)=O)C2CC2CN1C(=O)OC(C)(C)C 75319,C1(NC(c2n(OC)cnc2C)=O)CCC12CCN(C(=O)CNc1cccnc1)CC2 75320,CC(CS(C)(=O)=O)C(=O)N1CCC(Cn2cc(CN3CCOCC3)nn2)C1 75321,C1(CNC(CCC(C)SC)=O)CN(C(=O)Cc2ccnn2C)C2CCCCC12 75322,Nc1cc(C(=O)NCC23CC(NC(=O)C(O)CN4CCCC4)(CO2)C3)ccc1F 75323,C(=O)(CC(C)C(C)(C)C)N1CC(F)(CNC(C(n2cnc(C#N)n2)CC)=O)C1 75324,CC1CN(C(c2ccc(Cl)[nH]2)=O)CCN1C(C1CC(CC(F)F)C1)=O 75325,C1(CC(=O)OC)CC2(C1)CN(C(C1CC1NCc1ccc(Br)c(C)c1)=O)C2 75326,c1(C(=O)NCC2N(C(c3cccc(C)c3C)=O)CC(O)C2)cc2c[nH]cnc-2n1 75327,Cc1cccc(C(CNC(=O)CCCn2ccnc2C)NC(C2CC2F)=O)c1 75328,C(=O)(CC(O)CC(C)C)N1C(CC)C(NC(=O)CCCC(F)F)CC1 75329,c1(CNCc2nc(C(C)(C)C)sc2)cc(I)ccc1F 75330,C12(C(N(CC=C)C3CC3)=O)CC(CCO1)N(C(C1CCCC1O)=O)C2 75331,C1(C(=O)OC(C)=O)C=CCN1Cc1c(C(N(CCOC)CC)=O)cc[nH]1 75332,C(c1cccs1)=C(C)C(=O)N(C(C)CNC(=O)CCn1ccnn1)C 75333,N1(C(C2=CCCCC2C)=O)CCN(C(=O)CCc2cncnc2)C2(CCC2)C1 75334,Nc1nc(C(=O)NCC2CC2CNC(c2cc(Cl)ns2)=O)ccc1[N+](=O)[O-] 75335,N1(C(CC=COC)=O)CC(C)(NCCC(=O)OC)C1.C1(OC)(CO)CCSC1 75336,Cc1nnc2n1CCC(C(=O)N(CC(C)(C)NC(c1nnn3c1CCC3)=O)C)C2 75337,Brc1cccc(C(c2nnnn2CC(F)F)NC(Cc2ccccc2)C2CC2)n1 75338,Cc1ccc(NC(=O)CNC(=O)CSC2CC(=O)N(C)C2=O)cc1C 75339,c1(OC)cc(=O)n(C)cc1C(=O)N(C1CN(C(C2OCC3CCCCC23)=O)C1)C 75340,C1(NC(=O)CC2CC(F)(F)C2)CC2CC1CN(C(c1cccc(CO)c1)=O)C2 75341,N1(C(CC2N(C)CCCC2)=O)CC2CCCC1C2CNC(=O)CCCC1CCC1 75342,N1(C(COCCN(C)C)=O)CCC(CO)C(NC(=O)CCc2ncc(F)cn2)C1 75343,C1(C(=O)NC2CCCC2NC(C2(CO)CCC2)=O)CC2(CO1)CC(F)(F)C2 75344,C1(C(N2CC(CC(C)NC(=O)C(n3ccc(C4CC4)n3)C)C2)=O)CCCC1(F)F 75345,c1(CC(N2CCC(NC(CC3ON=C(CC)C3)=O)CC2)=O)ncnc2sccc12 75346,CCCC(C)(C)CC(=O)NC1CC=C(C(=O)NCc2cc(F)ccc2C)C1 75347,N1(C(c2nn(CC)c(C3CC3)c2)=O)CC(NC(c2ccnnc2)=O)CC2(CC2)C1 75348,N(C1CCc2ccccc21)C(CC(C)CNC(c1nsnc1O)=O)=O 75349,C1(C(=O)NC(CNC(c2cnc(C(C)OC)s2)=O)(C)C)CCc2n[nH]c(C)c2C1 75350,CS(=O)(=O)C1CC(CNC(=O)C(N)C2CSC2)C1 75351,c1(C(C)C)cccc(F)c1C(=O)N(C)CCN(C)C(c1cnc(Cl)s1)=O 75352,C1(CNC(C2C(C)CC2)=O)(NC(C2CCC=CCC2)=O)CCOCC1 75353,c1(C(N2CC(N=[N+]=[N-])C(NC(C3(F)CC3)=O)C2)=O)coc2c1C(O)CCC2 75354,c1(N2CCC(C(N)=O)CC2)nc(N2CCN(c3ccncn3)CC2)c2c(n1)CCS2 75355,C(=O)(C(C)(C)COC(C)(C)C)NC12CC(NC(C=CC(CC)C)=O)(C1)C2 75356,C1(NC(c2cnn(CCOC)c2)=O)CCCN(C(C2(CF)CC2)=O)CC1.CCO 75357,C1(C(N2CC(C)(C(=O)NCC3(O)CCC(C)C3)C2)=O)CCCCCN1C 75358,N1(C(C2CCCN(C)C2)=O)CCC2(C=C(C(=O)NC(c3cscn3)CO)C2)C1 75359,Cc1cn2nc(N3CCC(O)(C(C)NC(=O)CN4CCNC(=O)C4)C3)sc2n1 75360,N1(C(CC2N(CC)CCC2)=O)CCN(C(c2nnsc2C)=O)CC1C(C)C 75361,CC(C(F)F)N(C(=O)CCOCCN(C(=O)CSCCN(C)C)C)C 75362,c1(C(N2C(C(=O)NCC=C)CCC2C)=O)ccc(Cl)c(OC)c1F 75363,c1(CCC(=O)NC(C)(CNC(=O)C=Cc2cn[nH]c2)CO)cccc(O)n1 75364,Cc1ccc(CCCNC(C23CC(CNC(C4COCCN4C)=O)(C2)C3)=O)cc1 75365,C(=O)(CC1=NNC(=O)C1)N(CCCCCCNC(c1c(OC)cc(Cl)cc1)=O)C 75366,c1(C(N2CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C3C2C3)=O)ccnc2ncnn12 75367,Cc1cncc(C=CC(=O)NCC2(CNC(=O)Cc3ccsc3)CC(F)(F)C2)c1 75368,CC(C)C(O)CC(=O)NCc1cn(-c2c(Cl)cccc2Cl)nn1.C12CCCCC1S2 75369,C1(CC=C)(C(=O)NC(CCC)CCC)CCCN1C(C1CN(C(C)=O)C1)=O 75370,c1(NC2N(CC3(S(C)(=O)=O)CCC3)CCC2)ncnc2[nH]cnc12 75371,C(N(Cc1nccs1)N1CCN(CC(C)C)CC1)c1c(C)cccc1 75372,C1(NC(c2cnc(CC(C)C)[nH]2)=O)CCCC12CN(C(c1cc(Cl)ccn1)=O)C2 75373,C12(NC(C(C)Cc3ccncc3)=O)CCCN(C(=O)CC3CCC4CC34)CC1C2 75374,C1(C(N2C3CC(CNC(C4CN(C(C)C)C4)=O)(OC3)C2)=O)CCCCCS1(=O)=O 75375,Cc1ccc(F)c(C(=O)NCC2(CNC(=O)CC3CC=CC3)CCC2)c1 75376,N1(c2cc(CC)ncn2)C2CCC1CC(NC(c1c(C)oc(C)c1Br)=O)C2 75377,c1(C(N(C(C)CNC(=O)CC(C)N2CCCC2=O)CC)=O)nc2cnccc2s1 75378,c1(C(N(C)CC2N(C(C3CN(CC)C(=O)C3)=O)CCC2)=O)ccc(Cl)nc1OC 75379,C1(NC2CC2)CC(=O)C12CCC2.N12CC(C1)C(=O)N(C)CC=CC2=O 75380,C(=O)(C1SCCc2sccc21)NCC(CN(C(C(C)c1ccsc1)=O)C)(C)C 75381,c1(C(=O)NC(C(C)C)CNC(=O)C(C)(F)c2ccon2)ccc2nc(O)n(C)c2c1 75382,C1(C)(CNC(c2c(C)cccc2)=O)CN(C(C2COCCN2C=O)=O)CCO1 75383,C=CCCCCC(=O)N1CC(C(O)C(=O)NCCN2CCC(C)C2)C1 75384,C1(NC(C(N2CCN(C)CC2)C)=O)CCN(C(=O)CCCC2CCC2)C1C1CC1 75385,c1(CN2C(C(N3CCCC3c3ccc(Cl)s3)=O)CCC2)ccc2ncsc2c1 75386,C(=O)(CC(C)C(=O)NC1CN(C(c2cn(CC(F)(F)F)nn2)=O)CC1(C)C)OC 75387,Cc1c(C(=O)NC2CCCC(N(C(=O)C=CCF)C)C2)nnn1C1CCOC1 75388,c1(C(N2CC(NC(C(C)CC(F)F)=O)C3(C2)CC3)=O)cc2ccncc2[nH]1 75389,C1(C)(C(N2C(C3(NC(C4C(C=C)C4)=O)CC3)CCCC2)=O)CCN(C)C1=O 75390,N1(C(CCC=C=C)=O)CCN(C(c2cccc(O)c2F)=O)C(c2ccccc2)C1 75391,c1(CNC(=O)CC2CCN(Cc3ccc(F)c(O)c3)C2)cc2cccnc2[nH]1 75392,C(N=c1[nH]c(N2CCC(O)C2)nc2c1CCCCC2)c1c(OC)nccc1 75393,C(C)(C)(CCN=c1[nH]c(N(C)Cc2nccn2C(F)F)nc2c1SCC2)OC 75394,C1(F)(CNC(=O)CCc2ccncc2)CCC(CNC(C2(F)CCOC2)=O)C1 75395,N1(CC2N(c3nc(CC)nc(C)c3)CCCC2)CCC2CNCCC2C1 75396,C1(Cn2cc(C3CCCN(C(c4c(C)ccs4)=O)C3)nn2)CCCCC1(F)F 75397,N1(C(C=C(C)C2CC2)=O)CCC(C(=O)NCC(O)CCC2CC2)C1 75398,c1(C(N2CC(O)(CNC(C(CSC)O)=O)C2)=O)ccc(Cl)cc1O 75399,C12(C(N3C(C)CN(C(c4cnc(S)[nH]4)=O)CC3)=O)CCN(C1)S(=O)(=O)C2 75400,c1(C(=O)NCCNC(=O)CC2=CSC3=NCCN23)c(F)cccc1[N+](=O)[O-] 75401,c1(-c2nc(C(=O)NCC3C(CC)CCCC3)c(C)s2)ccc(SCC)nc1Br 75402,C(=O)(C(F)CC(C)(C)C)c1nn(C)c(-c2cn(Cc3cscn3)nn2)c1 75403,N1(C(C(COC)NC(C(CC)(CO)OC)=O)=O)CCCC(C2CC2)CC1 75404,C=C(C)CC(=O)N(CCC(C)NC(C1CC(OC)C1)=O)C 75405,C(CC(CNC(c1cnc[nH]1)=O)NC(=O)Cc1ccoc1)OC 75406,C1(C(=O)N)CCCCS1(=O)=O.CC(CCCN)N(C)C.C12CC(C1)C(=O)C2=O 75407,Cn1ncc(CCC(=O)NCC2CC(CNC(c3cnn[nH]3)=O)CO2)n1 75408,N1(C(C2CC(OC)(OC)C2)=O)CC2COCC2(C(=O)NC2CC(F)(F)C2)C1 75409,c1(CC)c(C(=O)NCC=CCNC(=O)C(c2cccc(F)c2)(C)C)ccn1C 75410,C(=O)(C1=CC2CCC(C1)C2)N1CCCN(C(C2C(CC)C(=O)C2)=O)CC1 75411,c1(CNCc2cccc(-c3c(C(=O)OC)ccnc3)c2)ccc(Br)cc1[N+](=O)[O-] 75412,C1(C(=O)NCCCCNC(C)=O)CCN(C(=O)OC(C)(C)C)C1C(C)(C)C 75413,CN1CCN(C(c2ccccc2C2CCC2)=O)C(CNC(c2c[nH]nc2Cl)=O)C1 75414,c1(C(=O)NCC(C)NC(Cc2cnc(C)s2)=O)ccc(C#N)nc1O 75415,S(=O)(=O)(c1nc(N2CCC(COC)C2)ccc1Br)NC1(CC=C)CC1 75416,c1(CC(=O)N(C2CCN(C(c3[nH]c(=NC)sc3)=O)C2)C)ccc2c(c1)CCOC2 75417,c1(C(=O)NC2C3(CN(C(c4c(C)occ4)=O)C3)CCC2)c([N+](=O)[O-])c(C)nn1C 75418,C12(N(C(c3c(CNC(c4ccn(C)c4)=O)occ3)=O)C3CC3)CCC(CC1)C2 75419,CC(C)CC(CNC(C12CC(C(C)(C)C)(C1)C2)=O)NC(=O)Cc1cnn(C)c1 75420,C(CN=c1nc(N2CCN(CC(C)F)CC2)c2nn[nH]c2[nH]1)c1nnc(C)s1 75421,c1(SC(C(=O)NC(C)CNC(=O)CC2CNC(=O)O2)CO)cccnc1 75422,c1(CN(C2CCN(C(CC(=C)C)=O)C2)C(c2ccccc2)=O)ccncc1F 75423,C(=O)(C1=NN(CCO)C(=O)CC1)NC1CCN(C(C(CC#C)O)=O)C1CC 75424,C(=O)(C(C)(C)CF)NC1CCC(N(C(c2c(CC(C)C)onc2)=O)C)C1 75425,CCC(C)(CCC(C)C)C(=O)N1CC(O)CC1C(=O)NCc1cccc(Cl)n1 75426,N1(C(C2(C(CC)=O)CC2)=O)CC(CNC(=O)Cn2cnc(=N)[nH]2)OC(C)(C)C1 75427,C(=O)(CCC(C)C)NCCCN(CCCNC(c1c(CC)nns1)=O)C 75428,c1(C(N2CCN(C(C(CCSC)O)=O)CC2CO)=O)cccc([N+](=O)[O-])c1NC 75429,C1(CC=C)(C(=O)NCC2(CCC)CCC2)CCCN1C(=O)C(C)CC#N 75430,c1(N(CC(C)CO)C)nc2cccnc2c(=NC(C)c2nc3ccccc3o2)[nH]1 75431,Cc1cc(C(=O)NC2C3CC(NC(=O)C(C)Cc4cnn(C)c4)CC23)nc(C)c1 75432,CC1C(NC(C2C3CN(CC(F)(F)F)CC23)=O)CCCN1C(=O)CSC1CC1 75433,C1(OC)CCOC(C(=O)NCCOC2CN(C(=O)CC3CCCC3C)C2)C1 75434,N1(C(c2c(C(=O)OC)scc2)=O)CC(NC(=O)COCCO)CCC1C 75435,C1(N(C(c2cc(C)ns2)=O)C)CN(C(c2cc[nH]c2-c2ccccc2)=O)CC1O 75436,S1(=O)(=O)c2cnc(cc2C)N1.c1(OCC(C)NCCC(=O)NC)cncc(Cl)c1 75437,N1(C(=O)Cn2cncn2)CC2CCN(C(=O)C3=CS(=O)CCC3)C2C1 75438,C(=O)(C(C(C)C)C(C)C)N1CC=CC(C(=O)Nc2ccc(SCC)nc2)C1 75439,c1(C(=O)NCC2CN(C(C(C)CC3CC3)=O)CC2O)ncn2c1COCC2 75440,C(CCCC(=O)N1CC(O)(CC(N2CC(COC(C)=O)C2)=O)C1)OCCC=C 75441,C1(O)(C(C)NC(Cc2cnc(C)s2)=O)CCN(C(c2ccc(Cl)s2)=O)C1 75442,C(=O)(C1=CC2C=CC1C2)NC1COCCN(C(=O)CSc2nncn2C2CC2)C1 75443,N1(C(C23N(C(c4ccc(C)nn4)=O)CCC2CCC3)=O)CC2(CNC(=O)N2C)C1 75444,C1(CNC(C2C(OC)C2)=O)CC2CCC(C1)N2C(c1sccc1-n1ccnn1)=O 75445,Cc1ccc(CC(N2CCCC(C(=O)NC3(CO)CCC3)C2)=O)c(Cl)n1 75446,C(=O)(C(C)(O)CC)N(CC(CNC(C(CC)NC(N)=O)=O)(C)C)C 75447,C(=O)(C(C)(C)CC(C)(C)C)N(CCNC(C1CC1F)=O)CC 75448,c1(C(=O)NC23CN(C(c4cc(C)cc(F)c4)=O)C(C2)C3)ccc2nc[nH]c2c1 75449,c1(CSCCCSC(CNCCO)OC)ccccc1 75450,Cn1cnc2c(C(N3CC(NC(c4cc(Cl)cnn4)=O)CC3CO)=O)ccnc12 75451,N1(C(c2c(CC)oc(C)c2)=O)CCCC(NC(C2CCCN(C)C2)=O)CC1 75452,Cc1cnc(C(=O)NC(CCSC)C(=O)NCC(F)F)c(C)c1 75453,C1(C(=O)NCC2CCCC(OC)C2)N(C(=O)Cc2n[nH]c(C)n2)CCC1(C)C 75454,c1(C(=O)NC(CC)CNC(c2cc(CO)[nH]n2)=O)cnccc1C1OCCO1 75455,Cc1ccn(CC(=O)N(CCCCNC(=O)CSC(C)C)C)n1 75456,N1(C(CCC)=O)CC2CC1CCN2C(=O)C(O)Cc1ccccc1 75457,c1(OC)ncccc1C(=O)Nc1cccc(NC(N)=O)c1.C12CCCN(C1)C2=O 75458,Cc1ccc(C2CN(C(C3CC4CC(=O)C3O4)=O)CCO2)cc1Br 75459,c1(C(=O)NCC(C2CC2)NC(c2cccc(NC(C)=O)c2)=O)c(C)nc(C)n1O 75460,Fc1ccc(F)c(CN2CCC(Nc3ccc(OC)cc3)C2)c1Br 75461,Cc1cccc(C(=O)CCC(=O)N2CCC(NC(C3CC3F)=O)C2C)c1 75462,c1(C(=O)NCC2N(C(C(C)(C)OC)=O)CC2)cccnc1I 75463,C1(OC)CCCC1C(=O)N(CC(F)(F)COC)C 75464,c1(N(c2n(CCCOC)c(-c3scnc3C)nn2)C)ccc(OC(F)F)c(Cl)c1 75465,N1(C(C=CC)=O)CCN(C(=O)C=CC2CCC2)C2CCCCC12 75466,N1(C(COCCOCC#C)=O)CC2CC1C2NC(c1cc(Cl)c(Cl)s1)=O 75467,C1(C(N2CC(NC(=O)C(F)Cl)C(F)CC2)=O)CCc2ccccc2C1O 75468,C1(NC(c2n(CC)cc(Br)c2)=O)COC2(CNC(=O)C3CC3)CC1C2 75469,C1(CC(C)Nc2nnsc2Cl)CCN(C(=O)CCCN2CCCCC2)CC1 75470,C1(C(=O)NCC(C)C(=O)NCc2nccn2C)CCC(=O)CC1C 75471,c1(C(=O)NC(CCCNC(CCCCOC)=O)C)cc(Cl)cc(Cl)c1N 75472,c1(CC(=O)N(CC(C)(C)NC(=O)CC2CC2(Cl)Cl)C)ccccc1OC(F)F 75473,Cc1ccc(CC(N2CCN(C(=O)C(C)Cc3cnc[nH]3)CC2C)=O)cc1F 75474,c1(CCC(=O)NC(C(C)(C)NC(C(=O)NCC)=O)C)ccccc1CC(=O)OC 75475,N1(C(c2ccc(C)cc2O)=O)CC(F)(F)CC1(C)CNC(=O)C(C)C(C)(C)C 75476,Cc1ccccc1CC(=O)NCC(O)CNC(=O)C=Cc1csc(Br)c1 75477,C(=O)(C(O)CCC(C)C)NCC1(F)CN(C(C2(c3c(C)cccc3)CC2)=O)C1 75478,c1(NC(=O)Cc2csnn2)ncnc2c1CCC2.C12CCCCC1CNC2=O 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75496,S(=O)(=O)(c1cccc(F)c1C)N(C1CNCCC1O)C(c1cc(C)cc(C)c1)=O 75497,Cc1cc(Br)c(F)cc1CN1CC2C(C1)N2C(=O)Cc1ccc(Cl)s1 75498,C1(COC)CCC(NC(C2CCN2C(c2ccncc2)=O)=O)C1 75499,c1(C(=O)NCCCC(C)NC(C2CCCO2)=O)ccc(C(=O)NCCO)cc1 75500,Cc1ccc(C(c2nnnn2C)NCCCCSc2ccccc2)cc1Br 75501,c1(C(=O)NCC(C)NC(C=CC(C)(C)SC)=O)cc(C2CC2)n(C)n1 75502,n1(CC(=O)NC(c2ccon2)CC)cc(CNC(=O)COC)nn1 75503,CC1CCCC=C1C(=O)N1CCC(O)(CNC(=O)C(C)NC(C2CCC2)=O)C1 75504,N1(C(c2cnn(C3CCCC3)c2)=O)CC2CCC1CN2C(=O)CCF 75505,N1(C(C(C)=CC2CC2)=O)CC(CNC(c2c(C)ncnc2C)=O)CC(C)(C)C1 75506,Cc1cnc(CNC2CCCC2C(=O)Nc2cc(F)ncc2C)cc1Cl 75507,C=CC(C)(C)C(=O)NCCN(CC(C)O)C(C1CC1C)=O 75508,c1(C(=O)NCC2(CNC(C(C)N(C)C)=O)CCC2)cc(C2CC2)nnc1O 75509,C1(NC(CCC2C(C)(C)C2)=O)CCC(NC(=O)C(O)C2CCCC2)CC1 75510,C1(C(=O)NCC2N(C(C(C)OC3CCCC3)=O)CC2)CCCN1C 75511,c1(C(N2CCC(NC(C(F)=CCC)=O)C(F)C2)=O)c(C)cc(Br)cc1C 75512,c1(C(=O)NC(CC)CNC(C2(C)CCCC2)=O)ccc(C(=O)N(C)C(C)C)cc1 75513,Cc1cccc(C(N2CCN(Cc3ccccc3)CC2)=O)c1C#N 75514,N1(C(C(C(C)C)SCC)=O)CC(C)(CNC(=O)COCCCF)CC1(C)C 75515,C1(C)(C(=O)NC2C(NC(c3ccc(COC)s3)=O)COCC2)CCCNC1=O 75516,N1(C(c2cnn[nH]2)=O)CCN(C(C2CC(O)(c3ccccn3)C2)=O)CC1C(F)F 75517,C(=O)(CCCCCN(C)C(C1CC(C)=NO1)=O)NC(C(C)SC)C 75518,CC1(NC(C2CCO2)=O)CCN(C(c2c[nH]nc2-c2ccco2)=O)CC1 75519,S(=O)(=O)(c1ccc(NCC(C)(C)CCS(C)(=O)=O)nc1)NCC(C)OCCO 75520,C(C(C(C)C(C)C)NC(c1cccnc1C(F)(F)F)=O)NC(COC(C)=O)=O 75521,C1(CNC(C(=O)NCC(C)(C)OC)=O)CCCN1c1ccccc1 75522,Cc1cc(C(=O)NC2CC(C(=O)Nc3ccc(C)s3)C2)c(C)[nH]1 75523,CC(CCCCNC(=O)CSC(F)(F)F)NC(c1ccnc(S)c1)=O 75524,N1(C(C2(CNC(CCC=CC)=O)CCC2)=O)CCCNC(=O)C1 75525,C1(NC(CCSC)=O)CCCCC12CCN(C(=O)CCC1CCCO1)CC2 75526,c1(SC)cc(C(=O)NCC(C)CNC(c2ccc(C(C)C)o2)=O)ccc1F 75527,c1(COC(c2c(C)nn(CC3CC3)c2)=O)ccc(Cl)c(C(F)(F)F)c1 75528,Cc1n[nH]c(=NCC2CCN(C(=O)CCCOc3cccnc3)CC2C)o1 75529,C1(C(=O)NCc2c(C(=O)NCC3CCC=CO3)occ2)CC2(CCC2O)C1 75530,c1(C(=O)NCC(CC)NC(=O)CC2CCn3cncc3C2)cc(Cl)c(O)cc1C 75531,C1(O)(CCNC(CC2C(C)CCC2)=O)CCN(C(c2ccc(N)cn2)=O)CC1 75532,c1(C(N2C(CN(C(CC(=C=C)C)=O)C)CCCC2)=O)ccc2c(c1)CCO2 75533,C=C(Cl)C(C)(C)C(=O)N1CCCCC(NC(=O)C(C(C)C)NC(=O)COC)C1 75534,Cc1csc(C(=O)NCC#CCNC(C2(n3cc(Cl)cn3)CC2)=O)c1 75535,N1(C(c2c(C)nn[nH]2)=O)CC(NC(=O)CCN(C2CCCCC2)C)C2CC2C1 75536,c1(C(=O)NC2(CNC(C3=NNC(=O)CC3)=O)CCOC2)[nH]cc2c1CCS2(=O)=O 75537,c1(C(N2CCC(CC)C2CNC(C2CCN(C)C2=O)=O)=O)cc2cnn(C)c2s1 75538,C1(CCNC(C(CC)N(C(=O)CCNC(N)=O)C)=O)CCC(C)(C)C1 75539,C1(NC(c2c(CC)nc[nH]2)=O)CC2CC1N(C(=O)Cc1cc(C)ns1)C2 75540,c1(C(=O)NC(C(C)NC(c2c(Cl)ccc(C)c2)=O)C)cccc2cnnc(O)c12 75541,c1(C(N2CCC(N(C(C(C)NC(C)=O)=O)C)CC2)=O)c(C)oc(C)c1S(N)(=O)=O 75542,c1(C(=O)NCC(C)(C2CC2)NC(c2cc(CO)[nH]n2)=O)cc2n(n1)CCO2 75543,C(c1c(C)noc1C)=CC(=O)NC(CC)(C)CNC(=O)C(C)(C)N1CCOCC1 75544,c1(C(N2C3C(NC(C=CC(CC)C)=O)C(C3)C2)=O)cc(C)c(F)cc1F 75545,C1(CNC(c2c(C)nc(C)o2)=O)CN(C(C2CC2C(C)(F)F)=O)CCC1(C)C 75546,c1(C(N(C(C)(C)C)CCN)=O)cnn2c1CN(C(C1C=CCN1)=O)CC2 75547,c1(C(N2CC(F)CC(NC(CSCC=C)=O)C2)=O)ccnc(S(N)(=O)=O)c1 75548,C(=O)(C(O)C1=CCCCC1)N(C1CCCN(C(C2(C)CC2)=O)C1)CCCCC 75549,c1(CN2CC(CC(=O)NC(n3ccc4cccnc34)C)C2)c(F)cc(I)cc1F 75550,N1(C(c2noc(CC)c2C)=O)CCC2(CC1)CC2CNC(=O)C(C)NC(=O)CC 75551,N1(C(c2c(C)cc(C3CC3)nc2)=O)C2CCC1CN(C(C1CCCCN1C)=O)C2 75552,c1(NC(C(C(C)C)CNC(=O)C(F)n2ccnc2)=O)ccc2c(c1)COC2 75553,C1(C(=O)NC2CC(CNC(C=C(C)C(F)F)=O)C2)CCCCC1c1nc(S)n[nH]1 75554,C1(C(=O)NCC(C#C)OC)CC(C)N1C(c1coc(C(C)C)n1)=O 75555,C1(CCNC(Cn2c(C)ccn2)=O)CC(F)(F)CN1C(c1c[nH]nc1Br)=O 75556,C(c1cccc(F)c1F)=CC(=O)NCC1(O)CCN(c2nnco2)C1 75557,C(=O)(CCCCC(C)C)NCC(C1CCOC1)NC(c1cccc(CC)c1N)=O 75558,c1(OC)cccc(C2CCN(C(C3CCCSC3)C(=O)NC3COC3)C2)c1 75559,c1(C(c2n(C(CC)C)nnn2)NCc2ncc(Br)s2)cc(C)c(OC)c(C)c1 75560,CC12CCC(C(=O)NC(c3ccnn3C)C(=O)NCC3CCCC34CC4)(CC1)C2 75561,C(CCC(C)C)(C(=O)NC1CC2CC2C(=O)C1)NC(C(C(CC)C)=O)=O 75562,CC1CC(NC(=O)Cc2cnoc2)CCN1C(c1cnns1)=O 75563,CC(CN(C)C(C1C(C)C1C)=O)C(=O)NCC(c1ccsc1)O 75564,CCC(CC(=O)N1CCC1CNC(c1ccc(C(C)=O)s1)=O)C1CC1 75565,N1(C(C(N2CCCC(C)C2C2CC2)=O)=O)CC(=O)N(C)C(=O)C1 75566,c1(C(N2CC3(C)CC2(C(=O)NCCC2CCSC2)C3)=O)ccc2n[nH]cc2c1 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75601,CCCCC(CNC(=O)COCC1CCC1)NC(=O)CN1CCN(C2CC2)C1=O 75602,CC1CCc2[nH]c(=NCCOCC3CC3)nc(N(C)Cc3ccc(F)cn3)c2C1 75603,C(CC)(CCC(=O)OC(C)(C)C)NCc1oc(C)c(Br)c1 75604,N1(C(c2cc(C)[nH]n2)=O)CCC2(CC1)CC2NC(=O)C(C1CC(F)(F)C1)O 75605,Cn1cc(C(=O)NCC2(NC(=O)CC3CCC(C#N)C3)CCC2)c2ccccc12 75606,C1(C(=O)NC2CONC2=O)C2CN(Cc3ccc(CN4CCOCC4)cc3)CC12 75607,N1(C(C(C)=C(C)C)=O)CCC(CCNC(C2CCCCN2C)=O)CC1 75608,c1(C(=O)OC(C)C(N2CCN(C(C3CCOCC3)=O)CC2)=O)c[nH]c2ccccc12 75609,N1(C(C(CCC)OC)=O)CCC2CCC(C1)N2C(C1CC2(CSC2)C1)=O 75610,C#Cc1ccc(C(N2CC(NC(=O)Cc3cncnc3)CC2CO)=O)nc1 75611,c1(COC)ncc(C(=O)NC2(C)CC(NC(=O)C(C)(C)c3ccno3)C2)c(=N)[nH]1 75612,c1(C(=O)NC(CNC(C(CC=C)CC)=O)C)cnc2cc(O)ccc2c1 75613,C(=O)(CCC(C)(C)NC(=O)C(C)Cn1ccnc1)NCC(CCOC)O 75614,C1(NC(c2cnc[nH]2)=O)CC2CN(C(=O)CCc3nccs3)CCN2C1=O 75615,N1(C(CCCC(C)C)=O)CCCC2C(CCCN2C(c2ccnn2C2CC2)=O)C1 75616,C(=O)(CCC(C)SC)NCC(=C)CCNC(=O)CCc1c[nH]c(C(=O)OC)c1 75617,c1(C(=O)NC2(C)CN(C(C3C(C)C3C)=O)C2)cc([N+](=O)[O-])ncc1Br 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75844,Cc1cc(C(=O)NCC(C2CC2)NC(c2ccc(C(F)F)nc2)=O)n(C(C)(C)C)n1 75845,c1(C(C)(C)C)cc(C(=O)NCC2C3CN(C(C4(CO)CCCO4)=O)CC23)nn1C 75846,C(=O)(C1=C(F)CN(C(c2cscn2)=O)CC1)NC(C)CC(F)(F)F 75847,c1(N(CC(CC2CC2)OC)C)ncc(Br)cc1[N+](=O)[O-] 75848,C(c1cn(C)nn1)=CC(=O)NC(C(=O)NC(CC=C)CC)CC1CCC1 75849,c1(C(=O)NCC(C2CC2)NC(C(CC(=C)C)C)=O)cc(Cl)c(Cl)cc1N 75850,N1(C(CCC2N(C)CCCC2)=O)CCCCC(CNC(c2csnn2)=O)CC1 75851,C1(C(N2CCC(NC(C3CN(C)C(=O)C3)=O)C2)=O)Cc2cncn2C(=O)N1 75852,N1(C(c2c(CC=C)cccc2)=O)CC2CC(NC(C3CC3C(F)(F)F)=O)CC1C2 75853,N1(C(=O)Nc2ccc(C)cc2)CCCN(C(c2cc(C)c(C)cn2)=O)CC1 75854,C(=O)(CCCC(=O)NC1CC1)N(C(CCNC(C=CC(C)C)=O)C(C)C)C 75855,N1(C(c2cn(CC=C)nc2)=O)CCC2(CC2C(N2CC(CSC)C2)=O)C1 75856,N1(C(CC=CCC)=O)CC(C)OC2(CCN(c3nc4cc(C)ccc4o3)CC2)C1 75857,C1(NC(Cc2n[nH]c(=NC)s2)=O)CC2CC(C1)N(C(C1(O)CCC1)=O)C2 75858,C=CCC(C)C(=O)N1CCC(C(F)F)(CNC(=O)CN(c2ccnc(Cl)n2)C)C1 75859,c1(C(N2CC(NC(Cc3c(C)noc3)=O)CC2(C)C)=O)cc2cccc(F)c2s1 75860,C(CC(C)(C)C(=O)NCCN(C(=O)C(N1CCCC(O)C1)C)CCOC)OC 75861,C1(NC(c2cc(CCNC(C(CC)C#N)=O)on2)=O)CCOCC1(C)C 75862,c1(NCCNC(N(CC(C)C)Cc2cnccn2)=O)ccc([Si](C)(C)C)cc1 75863,N1(C(c2c(C)scc2)=O)CCOCC(C(=O)NC(c2ccn(C)n2)C)C1 75864,CCC(COC)C(=O)NC(C1CN(C(c2cnn(C3CCC3)c2)=O)C1)C 75865,c1(C(=O)NC(CNC(COCCOCC#C)=O)(C)CO)cccc(F)c1O 75866,N(C(=NCCc1cccs1)N1CC2CC=CCC2C1)C(C)C 75867,c1(Cn2cc(CC(C=C)O)nn2)ccc(CF)cc1.c12ccc(o1)CNC2=O 75868,C1(C(N(CCCCNC(c2cccn2C)=O)C)=O)CCC(C2CC2)C1 75869,O(NC(=O)C(F)C1(O)CN(C(c2ccnn2C2CC2)=O)C1)C(C(C)C)C 75870,C1(CNC(C(CC)CC)=O)CCCCCN1C(c1cc(-c2ccoc2)on1)=O 75871,Cc1cc(-c2ccc(N(C)C)c(F)c2)nc(OC(F)F)n1 75872,c1(C(N2CCC(O)(CNC(c3cn(CC)nc3)=O)CC2)=O)cc([N+](=O)[O-])c(C)s1 75873,c1(C(N2CCC(N(C(C(F)=CC)=O)CC)C2)=O)cnc(OC)c(Cl)c1 75874,c1(CC)ccc(CC(N2CC(NC(=O)CSCC3CC3)C(F)C2)=O)cc1 75875,C1(CNC(C(c2ccccc2)N(C)CC)=O)CC2CC2N1C(C1CC(O)C1)=O 75876,c1(C(=O)NC(C(C)C)C(C)NC(c2ccc(C(N)=O)nc2)=O)cn(C)c(=O)n1C 75877,c1(NCC(CC(C)C)N(C)C)ncccc1S(=O)(=O)NCC12CCN(CC1)CC2 75878,C12(C(=O)NCC(C)(CNC(=O)C(C)(C)OC(C)=O)OC)CCC(F)(CC1)CC2 75879,Cc1c(C(=O)N(CC(C)O)CCNC(=O)C(F)(F)CF)cc(C(C)(C)C)n1C 75880,C1(NC(C2(C)CCOC2)=O)CC2(C1)CN(C(=O)CC1CCNC(=O)C1)C2 75881,c1(OC)noc(C2CC2)c1NC(=O)C(C)(C)C.C12CC(C1)C(=O)NC2 75882,c1(CN(C(CN(C(C2CC2F)=O)CC)=O)CC)cccnc1 75883,N1(C(c2c(C)noc2)=O)CC(O)CCC1OCC(=O)NC1CC1 75884,CCC(C)(C(=O)NC(C)CN(C)CCO)NC(=O)C(COC)OC1CCC1 75885,C1(C(=O)NC2CCC(CNC(C(C=C)(C)O)=O)CC2)CCc2cncn2C1 75886,N1(C(=O)Cc2cnn(C(F)F)c2)CC2CCCC(C1)N2C(C1CCC2CC12)=O 75887,C(CNC(=O)C(O)C1CCC1)(CCNC(=O)CCCN(C)C)OC 75888,c1(C(N(C2CN(C(c3cc(C)c(C)s3)=O)CC2O)C)=O)cc2scnc2[nH]1 75889,Cc1cn(C(=O)NCC2CCN(C(=O)C3=NOCC3)C23CCC3)c2ccccc12 75890,C1(O)(CNC(C2CCN(C)C2)=O)CCCN(C(=O)Cc2ccccc2CO)C1 75891,c1(C(=O)NCC(C)NC(=O)COC(C)(C)C)ccc2c(c1)nc(O)n2C 75892,C(=O)(C1=CCCC1)NC1CCC(NC(c2ccc(COC)s2)=O)C1 75893,c1(C(=O)NCC23C(CN(C(C4(COC)CC=CC4)=O)C2)C3)ccc(C)nc1C 75894,Cc1cc(=NCCN2CCC(O)CC2)[nH]c(N2CC3CC2C2CC32)n1 75895,c1(C(C)=O)ccc(C(N2CCN(C(=O)Cn3cnnn3)CC2)=O)cc1 75896,C1(C(=O)N(C)CC2CCCC2(C)C)(CC)CNC(=O)C1.C12CC1C(=O)NC2 75897,C(=O)(C(CC)C(C)C)N(CCCOC1CCN(C(C2C(CCC)C2)=O)CC1)CC 75898,c1(C(=O)NC2(C)CC(NC(=O)CC3=CCCCC3)C2)n[nH]c2c1CCCC2 75899,C(C)(CC(=O)NCCc1cccs1)NC(COC(C)=O)=O 75900,c1(C(=O)NC2CCC(C(N3CCC4(CC(F)C4)C3)=O)C2)ncc2ccccn12 75901,Cc1cc(=NCCc2cc(C3CC3)n[nH]2)[nH]c(N2CCCC(C#N)C2)n1 75902,C1(NC(c2ccccc2)C)CCOC1c1ccccc1 75903,C(C)(CO)(C(=O)N1CCC(CF)(NC(=O)CC2CC=CCC2)C1)OC 75904,CCCC(C)(CCC)C(=O)NCC1CN(C(=O)C(C)(F)CC2CCCC2)C1 75905,C1(CC(=O)NC2CCN(C(c3scnc3C(F)(F)F)=O)CC2)C=CS(=O)(=O)C1 75906,C1(CC(=O)N(CCCCC)C)CCCC1NC(=O)Cc1nccn1C 75907,C(=O)(CCC(C)(C)O)N1CCCC(C(C)NC(C(CC)OCC)=O)C1 75908,C1(=O)C(CC(C)C)OCNC(=O)CCN1CC=C.C1CCCCC1O.OC 75909,c1(C(N(C2CCC(NC(=O)C(F)F)C2)C)=O)c[nH]nc1S(N)(=O)=O 75910,N1(C(CCC(C)OC)=O)C2CCC1C(CNC(c1cn(C)nc1C(F)(F)F)=O)C2 75911,CC(C)C(C)C(CNC(=O)CCCN1C(=O)CNC1=O)NC(=O)Cc1cscn1 75912,C1(CNC(CC(CC)(F)F)=O)Cc2ccccc2CN1C(=O)CC1CC(C)=NO1 75913,C(CS(=O)(=O)CC(=O)NCc1nnn(C)c1C(F)(F)F)OC 75914,C1(C(N)=O)CCCCC1C(=O)NCC1C2CC1N(C(=O)CSc1ccncc1)C2 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76070,c1(OC)ccc(C(N2CCC(c3ccc(C)cc3)(C(C)C)C2)=O)cc1O 76071,C1(COC)(CNC(=O)CSC(F)F)CCN(C(=O)C(C2CC2)C2CC2)CC1 76072,C1(C(=O)NCC(CN(C(=O)Cn2ncc(Br)n2)C)O)CC2CC2C1 76073,C1(C(=O)NC2CCC(NC(=O)COC(F)F)CC2)CC2CC(O)C(C1)C2 76074,N1(CCCNC(C2CCCSC2)=O)CCN(C(C2CCC(=O)NC2)=O)CC1 76075,S(=O)(=O)(c1cccc(=NC2C=CCC2)[nH]1)NCCc1c(C)nn(C)c1C 76076,c1(C(=O)NCC2CCN(C(c3ccc(C(C)=O)o3)=O)C2)ccc([N+](=O)[O-])n1C 76077,c1(C(C)NC(c2ccc(N3CCC(O)CC3)cc2)=O)ccc(I)cc1F 76078,CC1CN(C(c2cc(C3CC3)ns2)=O)CCN1C(=O)CCCn1cc(CO)nn1 76079,c1(C(c2nnnn2C2CC2)NC(c2cccc(C)c2)CCC)cc(Cl)cc(Cl)c1F 76080,C(C1CCOCC1)=CC(=O)N(C(CC)C(=O)NCC1C=CCCC1)C 76081,Cc1cc(F)ccc1CC(=O)NCC1CCCC1CNC(C1CS(=O)(=O)C1)=O 76082,c1(SC(c2noc(C(C)(C)C)n2)C)cscc1C#N 76083,c1(C(=O)OCC)ccc(C(N2CCC(C)C2c2ccccc2C)=O)cc1 76084,C1(C(=O)NC2CC(CCO)C23CCC3)C2CCC(F)(F)C12 76085,Cc1ccccc1C=CC(=O)NCC12CC(NC(=O)CC3CCC4CC34)(C1)C2 76086,N#Cc1cccc([N+](=O)[O-])c1NCCC(O)(C(F)(F)F)c1ncco1 76087,Cc1csc(C=CC(=O)N(C)CCN(C)C(C2CC2c2nncn2C)=O)n1 76088,CC(CS(C)=O)N=c1ccc(Br)c(S(=O)(=O)NCCCN2CCCCCC2)[nH]1 76089,N1(C(CCCC=C)=O)CCC2C(C1)CN2C(c1cc(-c2ccc(Cl)s2)[nH]n1)=O 76090,C1(C)(C(N2CC(CNC(COCC(=O)NC)=O)C(F)(F)C2)=O)CCC(C)C1(C)C 76091,c1(SCCCOCC)nnc(N2CCOCC2)n1CCCOCC 76092,C(C1(C)CCOCC1)=CC(=O)NC(C1CCCN(C(=O)CCS(C)=O)C1)C 76093,C=C1CCN(C(=O)C(CC)C(C)C)C(C(=O)NC(CO)C(C)(C)C)C1 76094,C(CCC(CC)CC)NC.C1(SCC)C(C=O)CCN1C.N12CCC(C)(C1)C2=O 76095,C(=O)(CC(C)(C)CC(F)F)N1CCC(N(C(C(C)SC)=O)C)C2(C1)CC2 76096,N1(C(CSC(C)(C)C)=O)CCc2cc(N3CCCC(c4ccccc4)C3=O)ccc21 76097,c1(NC(C2CCN(C(c3cccc(C)n3)C(=O)OCC)C2)=O)cccc(OC)c1C 76098,c1(C(N2CCCC(N(C)C(C3CC4CCC3O4)=O)C2)C2CC2)ccccc1F 76099,c1(C(=O)O)cc(Cl)c(S(=O)(=O)N2CCC3CC(O)CCC3C2)c(Br)c1 76100,c1(-c2ccc(CNCc3ccc(OC)nc3OC)cn2)cnn2cccnc12 76101,c1(C(=O)NCCNS(CC)(=O)=O)[nH]ccc1CNC(c1cnco1)=O 76102,C(=O)(C1=C(Cl)CCOC1)N1CCC(CCNC(c2c(C(C)C)nn(C)c2Cl)=O)C1 76103,C(CCCC(=O)NC1CCN(C)C1)NC(CC1C(CC)C1)=O 76104,c1(C(N2CCC(N(CC(=O)NC)C)C2)=O)nccc(Cl)c1C.C(C)(C)(C)OC=O 76105,c1(C(N2CC(OCCNC(c3c(CC)scc3)=O)C2)=O)ccc(C)nc1OC 76106,C1(C(N(C2CC(NC(C3CC3c3ccccc3)=O)C2)C)=O)CCn2nncc2C1 76107,c1(C(=O)OC)ccc(S(C)(=O)=NC(=O)C(C)OC2CCCCC2)cc1 76108,Cc1nn(C)cc1CC(N1CCC(NC(=O)C(=Cc2ccccc2)F)C1C(C)C)=O 76109,N1(S(CCC)(=O)=O)CC2CCC(C1)C2Nc1ncncc1C 76110,C#CCCCCCC(=O)NCCOC1CCN(C(=O)C(C)C2CC2)CC1 76111,c1(CC)ccc(C(=O)NC(C)(CNC(=O)C(C)(C)F)Cn2cccn2)c(C)n1 76112,c1(OCC)cccc(-n2cc(CC(C)O)nn2)c1.N12CC3CC1C3C2=O 76113,C1(NC(c2c(F)ccc(C3(C#N)CC3)c2)=O)C2CC(O)C1N(C(C1CC1C)=O)C2 76114,c1(OCC(N2CC(NC(C3CC(SC)C3)=O)C(C)C2)=O)c(C)occc1=O 76115,c1(CC(=O)NC2CN(C(C(CC=C)C)=O)C(C)CC2)cccc2c1CCC2 76116,Cc1[nH]c(C)c(C(=O)NC2CCC(N(C)C(c3ccc(CO)cc3F)=O)C2)c1C 76117,CCCCCC(F)C(=O)N1CCC(C)C1C(N1CC(C(C)OC)C1)=O 76118,C12(NC(c3occ4c3CCC4)=O)CCCCCC1N(C(C1COC1)=O)CC2 76119,N1(C(C2C(NC(C3C(CCC)C3)=O)C2)=O)CCSCC1 76120,C1(CNC(Cc2c(C)ccs2)=O)CCCC2(CCN(C(c3cnn[nH]3)=O)CC2)O1 76121,N1(C(C2(COC)CC2)=O)CCC(C(C)NC(=O)CCCC2CCCCC2)C1 76122,C(=O)(CCCCCCCCCO)NCC(CN(C(=O)Cn1ccc(O)nc1=O)C)O 76123,C(=O)(CC1=CCN(C)CC1)NCC(CN(C(CSc1ccc(OC)cc1)=O)C)C 76124,N1(S(CCOC)(=O)=O)CCn2c(C(=O)N(CC(F)(F)CO)C(C)C)cnc2C1 76125,c1(C(=O)NCC2CC3CCC2N3C(=O)CCc2ccoc2)cnc2[nH]cncc1-2 76126,N1(C(C=CCN(C)CC)=O)CCN(C(=O)CCCc2ccccc2)C2CC12 76127,c1(NC(c2n(CCSC)nnn2)C2CC2)ccc2oc(C(C)OC)nc2c1 76128,C1(C(C)C)CN(C(=O)C(O)c2cnc[nH]2)CCCN1C(=O)CCCC(N)=O 76129,N1(C(c2cccc(C)c2C)=O)CC2CC(C)N(C(C3CCN(C)C3)=O)C2C1 76130,CCC(CNC(C1C=CCCC1)=O)(CC)NC(c1ccoc1C)=O 76131,C1(NC(c2cn(C)nc2-c2ccco2)=O)CCCC(NC(=O)C2=CSCS2)CC1 76132,CC(N=[N+]=[N-])C(=O)NC(Cc1cc[nH]n1)C(N1CCC(C)(C(=O)N(C)C)C1)=O 76133,c1(CCC)cccc2c1OCCC2NS(=O)(=O)c1cc(COC)ccc1F 76134,c1(OC)ccc(-c2cc(CNC3(c4nnnn4C)CCCC3N(C)C)on2)cc1 76135,O=C(C1COc2ccccc21)NC1(CCCNC(=O)C(F)(F)C2CC2)CC1 76136,CC(C)CC(C)(C)C(=O)N1CCC1CNC(=O)C(=Cc1ccc(F)cc1)C 76137,C(=O)(CC(C)(CN(C)C)C(F)(F)F)N1CCC(N(C(=O)CC(F)F)CC)CC1 76138,CC(C(F)C(=O)N1CCC(CCNC(=O)CCc2nncn2C)CC1)C(F)(F)F 76139,c1(C(=O)NCC2C3N(C(C(CC)C)=O)CC(CC3)C2)nc2nccc(C)n2n1 76140,N1(C(c2cc(CC)nn2C)=O)CCC2(CCC(NC(c3[nH]cnc3C)=O)C2)C1 76141,C1(N=[N+]=[N-])(C(N(C(C)C)CCF)=O)CCN(C(=O)OC(C)(C)C)C1 76142,C1(F)(CNC(c2c(OC)cccc2)=O)CC2CCC(C1)N2C(C1CCC2CC12)=O 76143,C1(CNC(C=CCCC)=O)CN(C(c2ncsc2NC)=O)CC1N(C)C 76144,N1(CC)CCN(CCC(N2CCCC2CN(C)C(=O)Nc2scnc2C)=O)CC1 76145,c1(C(=O)NC(C)CNC(=O)Cn2cc(C3CC3)nn2)cc(Cl)cc(Cl)c1F 76146,C1(C)(NC(C(C2CC(NC(CCCOC)=O)C2)F)=O)CCOC1=O 76147,N#Cc1ccccc1-c1nccc(C(F)(F)F)n1.c12nc(no1)OC2 76148,CC1(CNC(c2ccc(Br)o2)=O)CCCN(C(C2(NC3CC3)CCOC2)=O)C1 76149,C1(C(=O)NCCN(C(C)C)C(C2CC2c2ccccc2)=O)CC(S(C)(=O)=O)C1 76150,c1(C(=O)NC2CCN(C(Cc3cccc(C)c3)=O)C23CC3)ccn2ncccc12 76151,Cn1nc(C(=O)NC2(C)CCN(C(C3CC4(C3)CC(C)(C)C4)=O)C2)c2c1CCC2 76152,C1(C=C(C)C)CCN(c2ncnc(N3CCN(CCCCF)CC3)c2C)CC1C 76153,C1(C(N2CCC(C(CC)CC)C2)=O)C=CCN(C(=O)C(C=C)OCC)C1 76154,c1(CC)onc(C(F)(F)F)c1C(=O)NCC(C(C)(C)C)NC(c1coc(Br)n1)=O 76155,C1(NC(CCc2ccc(OC)cc2)=O)CCC2(CCN(C(c3cnsc3)=O)C2)C1 76156,C1(CNC(C2N(CC)CC2)=O)CN(C(C2OCCO2)=O)CC1C(F)(F)F 76157,N1(C(C=C)C)CCCC(NC(=O)Cc2cccc(OC)c2)C1 76158,C1(C(N2CCCC(NC(C3N(CC)C(=O)CC3)=O)C2)=O)OCCOC1(C)C 76159,CCC(C)(CNC(c1cc(CC)nn1C)=O)C(=O)N1CC(CO)CC1CO 76160,N1(C(C2C(C)(C)OCC2)=O)CCC(C(=O)NCC(O)C2CCC2)=C(F)C1 76161,C1(NC(c2c(C)nsc2)=O)CCC2CC1CN2C(C1C(C(F)(F)F)C1[N+](=O)[O-])=O 76162,N1(CC)CCOC(C(=O)N(C(C)CNC(C2(C3CCCO3)CC2)=O)CC)C1 76163,N1(C(C=CCCC(C)C)=O)CCN(C(c2cc(C3(Cl)CC3)n(C)n2)=O)C2CC12 76164,c1(C(=O)NCC(CN(C(=O)C#CC2(C)CC2)C)(C)C)nccn2ccnc12 76165,C(C)(C)(CCC(=O)N(C)CC1(O)CCN(C(C2CCC(OC)CC2)=O)CC1)OC 76166,CP(C)(=O)CC(=O)NCc1cc(C(=O)NC2CC(CC(N)=O)C2)co1 76167,CC(=O)C1=C(c2ccccc2)CCN1C(c1ccc(C)cc1)=O 76168,C1(NC(=O)CN2CCC2)CCN(C(=O)C2=NOCC2)C(C2CC2)C1 76169,Cc1ccccc1CC(CN1CC(C2CCCO2)C1)CN 76170,c1(C(=O)NC(C(C)C)C(C)NC(c2cc(O)n(C)n2)=O)ccc2ccn(C)c2c1 76171,C1(NC(=O)CCCn2cncn2)CCN(C(C23CCC2CC3)=O)CC1O 76172,C1(CC#N)CN(C(c2csc(O)n2)=O)CCN1C(c1cnoc1)=O 76173,Cc1cc(CC(N2CCCCC2CCCNC(c2nsnc2O)=O)=O)ccn1 76174,Cc1noc2nc(C(=O)N(C3CCN(C(=O)C(F)=C4CCCC4)C3)CCO)ccc12 76175,C(C(CC(=O)N1CCSCC1CCNC(c1cnc(S)n1C)=O)C(F)F)N(C)C 76176,C#CCC(O)C(=O)N1CC(F)(CNC(c2ccc(-c3ccccn3)s2)=O)C1 76177,CC1(NCCS(=O)(=O)c2ccc(F)cn2)CCc2ccccc21 76178,CN1CCCC(C)(NC(C2CCCCC2c2nc[nH]n2)=O)C1 76179,N1(C(C(Cc2ccccc2Br)NC(C2=C(C)CC2)=O)=O)CC2CCC2(C)C1 76180,C1(CC)CCCC1C(N1CCCC1C1(C(=O)N(C)CC2(O)CCC2)CC1)=O 76181,c1(OC)ccc2cc(C(=O)NC3CCN(C(C4CC4C(C)C)=O)C3(C)C)sc2c1 76182,N1(C(c2ccc(Cl)c(F)c2)=O)CC2(CC(NC(c3n[nH]cc3Br)=O)CO2)C1 76183,C1(O)(C(=O)NCCCN(C(CCC(C)SC)=O)CCO)CCCCCC1 76184,c1(CCNC(=O)NC2OCCCO2)cc(C(F)(F)F)ccn1 76185,CCC(C(=O)NC1CC(F)CN(C(c2cc(C(F)F)cs2)=O)C1)C(C)C 76186,S(=O)(=O)(c1cc(Br)c(Br)s1)Nc1nc(C(=O)NC(c2ccncc2)C)n(C)c1 76187,N1(C(C(CC)(O)c2ncco2)=O)CCC(NC(=O)CCN(C)CC2CC2)C(F)C1 76188,n1(CC(N2CC(NC(C3CCN(C(N)=O)CC3)=O)C2)=O)nnc2c1CCCC2 76189,CN1CCCC1C1CCCCN1C(C1CC1C1CC1)C(=O)NCCC1CC1 76190,Cc1ccc(C(C)C(=O)N2CC(CCCCNC(c3ncsc3C)=O)C2)s1 76191,C(=O)(CC(C(F)(F)F)NC(=O)C=CC(=O)OCC)Nc1cn(CC=C)nc1 76192,C1(C(=O)NC2(C)CN(C(C=C(CC)C)=O)C2)C2CCC1(c1cccnc1)C2 76193,c1(C(=O)NCCC2(O)CCN(C(=O)C(O)C(F)F)CC2)cc(Cl)c2n[nH]cc2c1 76194,C(=O)(CC(=O)N(CC(=O)N(C1CCC1O)C)C)NCC#C 76195,c1(-n2c(C(C3CCC3)O)nc(CCCC)n2)ccc(Br)cc1OC 76196,N1(C(c2ccc(C(F)F)cc2)=O)CC2(CCCN2C(c2coc(Cl)n2)=O)C1 76197,CC(C)CC(O)C(=O)N1CC(=O)CC1C(=O)NCC1(C)CCCS1 76198,N1(CC(=O)N(C(C)CC2CC2)C)CCN(C)CC1.C1(CSCC(=O)NC)CCCCO1 76199,c1(C(C)NC(C2C(CNC(C3(SC)CC(=O)C3)=O)CCC2)=O)ccc(C)nc1 76200,N1(C(C(CSC)(C)C)=O)CCC2(CC1)CCN2C(c1cnc2ccc(Cl)nn12)=O 76201,C12(COC)CC(NC(=O)C(C)(C)N3CCOCC3)(CN1C(=O)C(C)CN(C)C)C2 76202,C1(C(=O)NC2ON=C(C)C2)CCCN(c2nccc(-c3ccc(F)cc3)n2)C1C 76203,C12(NC(C(F)=CC)=O)CCC(CC1)N(C(c1cc(C)c(Br)cc1C)=O)C2 76204,c1(C(=O)NCC(CC)(CC)NC(c2ccn(CF)n2)=O)ccc2nc(S)[nH]c2c1 76205,N1(CCC(C)C)CCCC(C)(C(C)C)C1.C1(=O)CCC(=O)NC2CCN1CC2 76206,c12nocc1C(=O)NC2.c1(C(C)C(=O)NC(C2CCC2)C)ccnn1C 76207,c1(OC)ccc(Br)c(C)c1C(N1CC(CNC(c2oncc2C)=O)CC1C)=O 76208,C1=CC(=O)Nc2cc(OC)cc1c2.C1(CC(=O)OCC)CCC2(CC2)CO1 76209,CC(C)C(O)C(C)C(=O)NCCC(C)(C)NC(c1ccncc1Br)=O 76210,C(=O)(CCC(=O)NCCCN(C(C1CCCSC1)=O)Cc1ccccc1)NCC 76211,C(=O)(C1=C(Cl)CCCC1)NC1(CCc2n(C)ccn2)CN(C(=O)COCSC)C1 76212,Cc1ncc(CCC(=O)NCCC2CC(NC(c3ccccc3C)=O)C2)c(O)n1 76213,Cc1cc(CCC(=O)N(CC(C)(C)CNC(=O)CC2CCC(C)O2)C)ccc1Cl 76214,c1(C(C)(C)C)nccn2cnnc12.C1(CNC(CSC)=O)C2CN(C(=O)C=CCO)CC12 76215,c1(C(N(CCCN(C(=O)CC2(C)CC2F)C)C)=O)cnn2c(=N)[nH]cnc12 76216,C1(CCC(=O)NC(CC)CC)CCCCN1C(=O)CCCOC(C)C 76217,C1(O)(CNC(C2CCC2)=O)CCN(C(c2ccc(-c3ncc[nH]3)cc2)=O)C1 76218,N1(C(CC2(C=C)CCC2)=O)CCN(C(=O)C(C2CC2)OC)CC1CCO 76219,N1(C(c2nccc(C)c2O)=O)CCN(C(c2cnccc2Cl)=O)C(C)C1C 76220,c1(CC)cscc1NC(=O)C(N1CCCC1CNC(c1ccncc1)=O)=O 76221,c1(CN(C)C)cccc(C(=O)NCC(c2ccccc2)CNC(=O)C(C)(F)F)n1 76222,c1(C(=O)OCC)cc2cc(C(=O)NC3COCC3c3ccccc3)sc2s1 76223,N1(C(CC(CC)C(C)C)=O)CC2CN(C(=O)C=CCO)CC2(C)C1 76224,C(=O)(CCC(CF)CF)NC1CC2CC(NC(=O)C(O)c3ccsc3)C2C1 76225,c1(CN2CCN(C(c3ccc(CC(F)(F)F)cc3)=O)CC2)c[nH]c2ccccc12 76226,c1(C(C(=O)NCC2(O)CN(C(C(CC)N(C)C)=O)C2)CC)ccc(F)cc1 76227,c1(CO)ccc2cc1NC2=O.N1(CC)CCC(OCCOC)CC1 76228,C(=O)(CCC(N)=O)N1C(C(C)NC(c2cnoc2C2CC2)=O)CCC1 76229,c1(C(=O)NC2(CO)CCCN(C(COCCOC)=O)C2)ccn2cccc2c1 76230,N1(C(c2ccc(O)c(OC)c2F)=O)CCc2sc(-c3ccncc3N(C)C)cc2C1 76231,C1(NC(c2ncn(CC)c2)=O)C(C)CN(C(C2CCOCC23CCC3)=O)CC1C 76232,N1(C(c2nc(C(=O)OC)oc2)=O)CCCCC(NC(=O)Cc2nocc2C)C1 76233,c1(C(N2CCC(O)(C(C)NC(c3cccnc3)=O)C2)=O)cnc(C2CC2)nc1O 76234,CC1CCC(NC(=O)CC2COCC2O)CN1C(=O)C=CC(=O)NCCO 76235,N1(c2nnc(CC)s2)CCC2(CCOC2)C(CNC(c2cnc3n2CCC3)=O)C1 76236,C#CCCCCCC(=O)NCc1nc(C(N2CCOC(CC)C2)=O)c(C)o1 76237,C1(C(N2C(C(C)NC(CCOC)=O)CCC2)=O)CC2(CCOC2)C1 76238,N1(C(C2(C(F)(F)F)CCN(C)C2)=O)CCC(NC(c2cccnc2)=O)C(C)(C)C1 76239,c1(N2CCN(N(C(c3nn(C(CC)CC)c(C)c3)=O)C)CC2)snc(C)c1C#N 76240,c1(CC(=O)NC2CC(C)(CNC(c3csc(C4CC4)n3)=O)C2)ncn2c1CCC2 76241,C(=O)(C(CN=[N+]=[N-])NC(=O)Cn1nccc1C)NCCCc1nc(C)[nH]n1 76242,C=CCCC(C(=O)OC)N(C1CN2CCCC1C2)C 76243,C(=O)(C(F)(CNC(c1cc(C)ccn1)=O)C(C)C)N(C(C)C)CC 76244,CCC(O)(CN(C(=O)C(CO)NC(=O)Cn1c(O)nnc1O)C)CC 76245,CC(C(C)(C)C(=O)NC(c1ccccc1)CO)NC(=O)C(c1cncnc1)C 76246,N1(C(C(C)(C)SC)=O)CCC(NC(C2CCC2)=O)C(CO)CC1 76247,C(=O)(C(C)C(O)C(C)C)N1C2C(OC)CC(C2)C1.N12CCC(C1)n1cc(nn1)C2 76248,C(=O)(C(C)(O)C(F)(F)F)N1CCCC(CN(C(=O)CN2CC(=O)NC2=O)C)C1 76249,C(C)(CCCC(=O)NC(c1nccs1)C)NC(C(C)NC(CC)(C)C)=O 76250,C1(C(=O)NCCN(C(c2c[nH]nc2-c2ccccc2)=O)CC)CC(Br)(Br)C1 76251,CCC(C)C(O)C(=O)N(C1CCN(C(c2cccnc2OC(C)C)=O)C1)C 76252,C1(OC)CN(C(C2C(C)(C)C2(F)F)=O)CC1NC(c1cc(C)c(C)s1)=O 76253,c1(CC(=O)NCCN2CCC(NC(C3CC4CCC34)=O)CC2)ccccc1O 76254,c1(C(=O)NC2CCC(C)N(C(C3CSCCS3)=O)C2)cnc2c(c1)C(=O)CCC2 76255,C=C1CCCN(C(C2CC2C(C)NC(c2coc(CCC)n2)=O)=O)C1 76256,C12(CNC(=O)NC(C)CCCCc3ccccc3)CCOC1CCOC2 76257,C(CCNC(=O)Cc1cccc(NC(C)=O)c1)(C(C)C)NCCCOC=C 76258,c1(C(=O)NCC(CC)(C)NC(c2cncc(N)c2C)=O)nnn2c1COCC2 76259,C(CC)(CC(=O)NCCC(C)OC)NC(C=CC)=O 76260,NC(=O)CCCCC(=O)N1CCCC(CCNC(c2c[nH]nc2C2CC2)=O)CC1 76261,C1(CC(=O)NCCCN(C(=O)CN(C(=O)COC)C)CC)CCC(OC)CC1 76262,CC(C)CC(CN=c1[nH]c(C2CC2)nc2[nH]ccc12)NC(C1CC2(CC2)CO1)=O 76263,N#Cc1c[nH]c2cc(C(N3CC4(CC4)CC3C(N3CCC(Br)C3)=O)=O)ccc12 76264,C1(O)(CC(N2C(CN(C(CCOC)=O)C)CCC2)=O)CCCN(C(C)=O)C1 76265,CC1COC2(CCN(CC(O)Cc3ccc(OC(F)F)cc3)CC2)O1 76266,C12(CC(=O)NCC3CCC3COC)CCC1CN(C(c1cc(O)ncc1F)=O)C2 76267,C(=O)(C(C)(O)CC(C)C)NC(CCC1(NC(c2cn(CCOC)nn2)=O)CC1)(C)C 76268,C1(CC(=O)NCCCC(C)C)CC2(C1)CN(C(=O)C(O)C1CCC1)C2 76269,Cc1noc(Cl)c1CC(=O)NCC12CC1CN(C(c1coc(Cl)c1)=O)C2 76270,c1(CCC(=O)NCC(n2cc(CCN(C)CC)nn2)C)nnc(C)n1C 76271,c1(C(=O)NC2CN(C(c3cc(C)[nH]n3)=O)C3C2C3)c(F)ccc2n[nH]cc12 76272,C#CCC(C)(CC)C(=O)NCCC1CN(C(=O)C=Cc2c(C)coc2C)CCO1 76273,C(=O)(C1=CNS(=O)(=O)N=C1C)NC1C(CNC(C2(COC)CCCCO2)=O)CC1 76274,N1(C(C2N(CC)CC2)=O)CCC(O)(CNC(=O)C(F)=CCCF)CC1 76275,N#Cc1cccc(F)c1C(N1CC2CC(NC(c3cn(C4CC4)cn3)=O)C2C1)=O 76276,c1(C(=O)NC2CN(C(c3ccn(C)c3)=O)CC2F)cc(N=S(C)(C)=O)ccn1 76277,Cc1ccc(CC(=O)NCC2COCCN2C(=O)CCC2CC2C)cc1Br 76278,C12CCN(C1)CC(=O)N(C)C2C1CC1.C(=O)(CCn1cccn1)NC 76279,c1(CC(=O)NCC#CCNC(C2C(C(=O)NCC#C)C2)=O)ccncc1C 76280,C1(C(N2CC(Cn3cc(CCc4[nH]c(=N)sc4)nn3)C2)=O)CCCC2(CCC2)O1 76281,N1(C(c2ccc(CC)s2)=O)CCC(N(C)C(c2ccnc(C)n2)=O)CC1 76282,c1(C(=O)NCC(C)CN(C)C(c2nccn2C)=O)ccc(F)c2c1CCC2 76283,c1(C(c2nnnn2CCCSN(C)C)NC(CC)CC)ccc(SC)s1 76284,Cc1n[nH]c(C)c1CC(=O)N(C)CC1CCN(C(=O)COC2(C)CCCC2)C1 76285,N1(C(c2ccc(COC)[nH]2)=O)CCC2CCC(NC(C3CSC3)=O)C1C2 76286,c1(C(N2CCC3(CC3C(N3CC(O)(CO)C3)=O)C2)=O)cccc2c1CCC2 76287,C#CCC(C(=O)NCCC(=O)NCC#C)NC(C1CCCN1C(C)=O)=O 76288,C(=O)(CC(O)C(C)CC)NC1(CNC(c2ncn(C(C)C)n2)=O)CCCC1 76289,C(=O)(C(CNC(=O)C(C)CCOC(C)=O)C(C)(C)C)N(CC(C)(C)C)CCC 76290,C1(C(=O)NC2(CNC(c3c(C)ncs3)=O)CCCC2)CSC2(C)CCC(=O)N12 76291,c1(C(=O)NCC(CNC(CC(C)C2CCCC2)=O)F)ccncc1Cl 76292,Cc1cc(CCC(C)(c2nnnn2C2CC2)NC(C(C)C)C2CCC2)ccc1Cl 76293,O=S(=O)(c1ccc(Br)cc1N1CCC2(CCSC2)C1)NC(c1cccc(Cl)c1)CO 76294,c1(NC(C(CC)NC(c2cc(C)cc(F)c2)=O)=O)cccc2[nH]ccc12 76295,CC(CONC(C1CCCCC1c1ccccc1F)=O)C(C)C(=O)O 76296,Cc1ccc(COCCC(=O)NCC2CN(C(=O)CCSC(=N)N)CCO2)cc1 76297,C1(C)(C(=O)NC(C)(C)CC2CCOC2)C=CCN1C(=O)CC1CCCC1 76298,S(=O)(=O)(CC(=O)N1CCCC1CCCNC(C1CC2(CSC2)C1)=O)N(CC)CC 76299,O=C(N=c1[nH]nc2ccccn12)NCc1ccc(F)c(F)c1 76300,C1(CNC(CCc2onc(CC)n2)=O)CCCCN(C(c2coc(Cl)c2)=O)C1 76301,C1(CNC(CSCC(=O)OC)=O)C(C)CCCN1C(=O)CNc1ccccn1 76302,C1(C(C)C)CN(C(=O)COC2CCCC2)CCC1NC(=O)CC1C=CS(=O)(=O)C1 76303,C1(C(N(C2CCCN(C(=O)Cn3[nH]cnc3=N)C2)CC)=O)CCNC(=O)C1 76304,c1(OC)ccc(C=CC(=O)NCC(C)CNC(=O)Cn2cc(C3CC3)nn2)cc1Cl 76305,c1(CC)cnccc1C(N1CC(NC(c2ncccc2F)=O)C(O)C1)=O 76306,c1(C(=O)OCC2CCCCC2F)c[nH]cc(Br)c1=O 76307,N#Cc1ccc(F)c(CC(N2CC(NC(c3cnn4c3OCC4)=O)C3CC23)=O)c1 76308,C=CCC(CC(=O)N(C1CC2CC2C1)C)NC(=O)C(O)C1CCC1 76309,C1(NC(C(C)C2CCCC2)=O)C2CC(NC(=O)CP(C)(C)=O)CC12 76310,N1(C(C2CC(C#N)C2)=O)CC2CC(NC(c3sccc3C(F)F)=O)CC2C1 76311,C1(NC(C(CC)CN(C)C)=O)COCCN(C(C2CN(C)CCN2C)=O)C1 76312,c1(C(N2CC=CC(NC(C#CC(C)(C)C)=O)C2)=O)cc2ccc(F)cc2o1 76313,c1(C(=O)NC2CN(C(c3ccc(C)c(I)c3)=O)CC2F)ccc2[nH]nc(O)c2c1 76314,N1(Cc2cc(C)[nH]n2)CCC(O)C(C(=O)Nc2ccc(F)c(C(F)(F)F)c2)C1 76315,C=CC(C)(CCOC)C(=O)N1CCOC(CN(C)C(C2CC(O)(C#N)C2)=O)C1 76316,C1(NC(c2c(OCC)scc2)=O)CC(C)N(C(C2CC3(CCC3)C2)=O)C1 76317,c1(C(N2CC(NC(C(C3CCCOC3)OC)=O)(CO)C2)=O)ccc(N(C)C)cn1 76318,C12(NC(CC(CC=C)(C)C)=O)CC(CO)(C1)OC21CN(C(c2cncn2C)=O)C1 76319,C(CC(C(C)(C)C)NC(c1nsnc1O)=O)N(C(Cc1ncc(C)s1)=O)C 76320,N1(C(C(C)(C)SC)=O)CC2CCOC2(CNC(c2n[nH]c3cccnc23)=O)C1 76321,C1(NC(C(C2CC2)SC)=O)C=CCN(C(c2ccn(C(C)(C)C)n2)=O)C1 76322,C1(O)(C(N2CCC(N(CC#C)C(c3cc(CCC)c[nH]3)=O)C2)=O)CCC(C)CC1 76323,N1(C(c2cccc(C)n2)=O)CCCC12CCN(C(C1CCCSC1)=O)C2 76324,C1(NC(CC(C)(C)C)=O)CC2CCC(C1)N2C(=O)Cc1ccc(Cl)c(N)c1 76325,C(CCCCCNC(=O)C(C)(C)CN(C)C(c1cccc(CC#N)c1)=O)OC 76326,Cn1c(C(N2CC3CC(NC(=O)CC4CCC(=O)N4)CC2C3)=O)cnc1[N+](=O)[O-] 76327,O=C(C#CC1CCOC1)NCCN(CC(O)CF)C(c1ccccc1Br)=O 76328,c1(NC(C2(F)CN(Cc3cc(F)ccc3I)C2)=O)cc(Cl)nc(Cl)c1 76329,c1(OC)cccc(F)c1C(=O)NCC1CCC(NC(c2cnoc2C)=O)CC1 76330,c1(C(N2CCCC(C)(NC(C3C(OC)CCC3)=O)C2)=O)cc(O)cc(F)c1F 76331,CC1CC(C(=O)NCCOCC2CC2)CCN1C(C1CC2CC(=O)C1O2)=O 76332,C1(N(C(=O)Cc2nn(C)cc2Cl)C)CC2CCC(C1)N2C(c1cnccn1)=O 76333,N1(C(Cc2scc(C)c2)=O)CCCC(C2CCN(c3cncc(Cl)n3)CC2)C1 76334,C1(C(N2C(=O)CC(OCC=C)C2)=O)CCCCC12OCCO2 76335,C1(C(N2CC(CC(N)=O)C2)=O)CCC2(CN(C(=O)NC3(Br)CC3)C2)O1 76336,N1(C(c2snc(C)c2N)=O)CC2(CNC(=O)C=CC=C(Cl)Cl)CCC1CC2 76337,c1(CC(N2CC=CC(NC(C3(CC)CC3(F)F)=O)C2)=O)c(C)cccc1C 76338,Cc1nn(C)cc1CCC(N1CC2C(NC(C3(C)CC3(Cl)Cl)=O)C2C1)=O 76339,C1(CNC(C(CCSC)NC(C)=O)=O)C2CN(C(=O)CC3COCCO3)CC12 76340,c1(CNC(c2c(C)ncs2)=O)ccc(-c2ccc(C(F)(F)F)nc2)c2cc[nH]c12 76341,c1(C(N(CCC(C(C)C)NC(=O)CC#N)C)=O)cccc2nc(O)[nH]c12 76342,n1(CC)cc(C(=O)NCC(O)CCNC(c2cnc(C(C)(C)C)[nH]2)=O)c(C)n1 76343,CCCC(CC)C(=O)NC1CCC(NC(c2ccc(Br)cc2N)=O)CC1 76344,c1(CNC(c2cnn(-c3ccccc3)c2Cl)=O)ccc(OCC2CC2)c(F)c1 76345,C#Cc1ccc(C(N2CCCC2CNC(C2CCCC2(F)F)=O)=O)c(F)c1Cl 76346,C1(NC(=O)C(C2CCC2)C2CCC2)CC2CCC1N2C(c1cc2[nH]ccc2s1)=O 76347,CC(CN(C)C)CCC(=O)N1CCCC(N(C)C(c2cccc(F)c2)=O)C1 76348,c1(C(N(CCCN(C(=O)CCC(F)F)C)C)=O)cnc2ccoc2c1 76349,C1(NC(C(C)OCCN(C)C)=O)CC2CN(C(=O)C=Cc3ccc(Cl)s3)CC12 76350,c1(C(C)=O)cc(C)c(C(N2CCCCC2C2CCN(c3nnc(O)s3)C2)=O)o1 76351,c1(NC(C(CC2CCCC2)NC(CC(C)(C)O)=O)=O)ccc(O)c(CO)c1 76352,C1(CCOC)CCN(C(=O)C(=O)NCC(C(C)C)c2ccccc2)CC1 76353,c1(NC(C2C(C(=O)Nc3cc(F)c(OC)c(F)c3)C2)=O)nc2cc(Br)cnc2[nH]1 76354,C1(CC(=O)NCC23CC(NC(C(C=C)O)=O)(C2)C3)CC2(CCOCC2)CO1 76355,ClCCCN=C(NN1CCC(C)C1)NC1CCCCC1.C1(C)CCC1 76356,C(CC(CO)NC(C1CC(NC(C2CC2c2cccs2)=O)C1)=O)SC 76357,N1(C(C2C(=C)C2)=O)CC(C2CC2C(=O)N(C(C)COCC)C)C1 76358,Cc1cc2c(=O)n(CC(=O)NC3CCCCCC3C)cnc2[nH]1 76359,C1(CN(C(C(C)N2C(=O)CN(C)CC2)=O)C)COCC1(C)C.C(C)(=O)OC 76360,Cc1cn2c(C(N3CC4(C3)CN(C(C3(C)CCC3(F)F)=O)C4)=O)c(C)nc2s1 76361,CCCC(C(=O)N(C(C)CC(=O)NCC1(Cl)CC1(C)C)C)NC(N)=O 76362,N1(C(c2cn(CCNC(CC(C)N(C)C)=O)nc2)=O)CCCC12CCNC2=O 76363,C#CCC(O)C(=O)NCC1(CN(C)C(c2cscc2Cl)=O)CC1 76364,c1(C(=O)NC(c2ccccc2)CC)sc(NC(c2occc2Br)=O)nc1C 76365,N1(C(C2CC(OC)C2)=O)CCCC(C)(NC(=O)Cc2nc(C)n(C)n2)C1 76366,Cc1cc(CCC(=O)NCC2CC(NC(=O)C(F)C(F)(F)F)C2)ccc1Cl 76367,c1(OC)cnc(CNC(=O)CCN(C)C(C2CC(=O)CCO2)=O)cn1 76368,CC1CN2CC(O1)C(=O)N1CC(C1)CC2=O.c1(NC(=O)OC(C)(C)C)cn(C)cn1 76369,N1(C(CCCOC)=O)C(C(=O)N(CCS(C)(=O)=O)C)CCC1C 76370,C(=O)(C(C(C)C)NCCC)N(CCCCC=C)C(C)Cc1ccccc1 76371,c1(C(N2C(C(N(C(C(=O)OC)C)C)=O)CC2C)=O)cc(C)ncn1 76372,C1(C#N)(C(=O)NC(c2cccc(C(N3CC[Si](C)(C)CC3)=O)c2)C)CCCCC1 76373,c1(C(=O)NC2CN(C(C3CC(C)(CC)C3)=O)CC2C)cccc2c1C(=O)CCN2 76374,C(Cc1ccco1)(C(=O)Nn1cnnc1)N(C(CS(CC)(=O)=O)=O)CC 76375,C(=O)(CCCN(C)N=O)NCC(C(C(=O)N(CC(=O)OC)CC#C)C)C 76376,N1(C(C)=O)CCCC(O)(CC(=O)NCCOCCNC(c2c[nH]c(=N)cc2C)=O)C1 76377,C1(NC(C(CCCOC)C)=O)CC2CCC(C1)N2C(c1cc2occc2s1)=O 76378,C1(C(=O)NCC2(C)N(C(c3ncc(NC)nc3)=O)CCC2)CS(=O)(=O)CC(=O)N1 76379,Cc1ccnn1CC(N1CCC(C2CCCN2C(c2ccc(Br)o2)=O)C1)=O 76380,N1(C(CCNC(N)=O)=O)CCC(F)(CNC(c2cn(C3CC3)cn2)=O)CC1 76381,c1(COC)cc(C(=O)NC(C)C(C)(C)NC(=O)CSC(C)(C)C)ccc1F 76382,C(=O)(CS(=O)(=O)C(C)C)OC.c1(OCCC)cncc(C(=O)O)c1 76383,CCCCCCC(=O)NC1CCCN(C(c2c(CC=C(C)C)cnn2C)=O)CC1 76384,N1(C(C=CC(C)(C)SC)=O)CCN(C(=O)CNc2n[nH]c(C)c2C)CC1 76385,Cc1cc(NCC2CCC2(F)F)ncc1S(=O)(=O)NC(CC1CC1)C1CC1 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76701,Cc1nc(=N)[nH]cc1C(N1CCC(CNC(c2ccc(F)o2)=O)C1(C)C)=O 76702,C(=O)(C1COc2cc(C)c(C)cc21)N1CCCCC(NC(C(C)(C2CC2)OC)=O)C1 76703,C=CC1(C(=O)NC2C(C)CCC2C)CCN(C(=O)Cn2ncnn2)C1 76704,c1(OCC(C)C)cccc(C(=O)NC2CN(C(=O)C(=O)NCC3CC3)C3CC23)c1 76705,CC1(C)CN(C(c2cccc(Cl)c2)=O)CC1NC(c1c[nH]nc1-n1cnnn1)=O 76706,c1(COCCNC(=O)CC2CCC(Nc3ccccn3)CC2)cccc(F)c1I 76707,c1(CC(=O)NCC2CCCN(C(C(CC)OC)=O)C2)ccc(S(C)(=O)=O)cc1 76708,C1(C)(NC(CCCCC)=O)CCCN(C(=O)C(C)=C(C)CC)C1 76709,C1(C#N)(SC)CN(C(=O)C(CCOCCO)NC(c2ccc(SC)o2)=O)C1 76710,c1(NCC(CC)(C)O)cc(NC2CCN(c3ccccc3)C2)ncn1 76711,CCC(COC1CC1)(c1nnnn1CCCC1CC1)NCCC.C1CC1 76712,c1(CN2CC(NC(=O)CC3CC3)CC(F)(F)C2)ccc(F)c2ccoc12 76713,CCC(C)C(O)CC(=O)N1CC(CCNC(=O)C(=O)Nc2ncc[nH]2)(OC)C1 76714,N1(C(C2CCC(C)CN2C(=O)CCC2CC2(F)F)=O)CCC(C2(C)CC2)C1 76715,C(=O)(C1Cc2ccccc21)NCC1(NC(C=Cc2ccc(OC)cc2)=O)CC1 76716,C1(O)(CNC(CC2N(C)CCOC2)=O)CCN(C(=O)C=Cc2nnn(C)n2)CC1 76717,n1(CC)nc(C(=O)N(C)CCN(C(C2CCCCC2C(C)C)=O)C(C)C)cc1O 76718,c1(C(=O)NCC2C(NC(c3ccc(CC)o3)=O)C2)cccnc1N1CCCC1 76719,N12CCC(C1)C2=O.CC(C(=O)C(=O)Cn1cccn1)N.N1(C2(CN)CC2)CCCC1 76720,C1(NC(c2cnc(SC)s2)=O)CCCCN(C(c2ccn(C3CC3)n2)=O)C1 76721,CCCCCCCCCC(=O)N1CCCC12CN(c1ccncn1)C2 76722,CC1CN(C(=O)Cc2cccc([N+](=O)[O-])c2)c2ncc(Br)cc2O1 76723,C(C(C)(O)CC(=O)N1CCC(N(C)C(C2(c3cccc(SC)c3)CC2)=O)C1)OC 76724,C1(CS(C)(=O)=O)CN(C(c2c(F)cccc2Cl)=O)CCN1C(=O)C(F)C1CCC1 76725,CCCC(O)C(CO)NC(=O)C(C1CCN(C(=O)CN2CCCCC2C)CC1)C 76726,C1(NC(c2nc(C)c(C)s2)=O)(CO)CCCN(C(C2CC3(CCOC3)C2)=O)C1 76727,c1(C(=O)NC23CC(NC(Cn4c(=O)ccc(C)n4)=O)(C2)C3)ccn2ccccc12 76728,C(CN(C)C(C1CN(C)C(=O)N1)=O)(CO)(CO)NC(Cc1n(C(C)C)ncc1)=O 76729,c1(CC)cccc2c(C(=O)NCCCCNC(c3ccc(F)s3)=O)c[nH]c12 76730,Cc1ccc(Cl)c(C(N2CCC(c3nc(-c4ccnn4C)cs3)CC2)=O)c1Cl 76731,C1(OC)CC(CNC(c2cc(NC(C)=O)ccn2)=O)N(C(=O)Cc2ccn(C)c2)C1 76732,c1(N(C)C2CC2)ccc(Cl)cc1F.c1(C2C(=O)N2)ccc(O)cc1.C1(N)CCC1 76733,c1(CC(N2CC(NC(c3c(C(C)C)con3)=O)C2)=O)cc(Br)cnc1F 76734,c1(C(N(C)CCOCCNC(=O)CSCC(N)=O)=O)cc[nH]c1C1CCCC1 76735,N1(C(c2cc(C)oc2)=O)CCC(NC(c2cc(O)no2)=O)C1(C)C 76736,C(CCCCCNC(=O)CNc1cccc(O)c1)NC(=O)COCCc1cccs1 76737,C(=O)(C(C(=O)NC)OC)NCCCCCCNC(C(CC)Cc1ccccc1)=O 76738,c1(OC(c2c(-c3c(C)cccc3)c[nH]n2)=O)cc(Br)ccc1Cl 76739,N1(C(c2cnc(CNC(C(C)c3cc[nH]n3)=O)nc2)=O)Cc2ccc(C#N)cc2C1 76740,N1(C(=O)OC(C)(C)C)CCC2(CCC2)C1C(=O)NC1(C2CCCC2)CC1 76741,C(C)(CNC(c1cc(OC)no1)=O)(C(C)C)NC(Cc1nc(COC)sc1)=O 76742,C1(NC(c2cc(C)sc2)=O)CCCC(CNC(c2cc(C(N)=O)nn2C)=O)C1 76743,c1(C(=O)NCCN2CC(C)N(C(=O)OC(C)(C)C)CC2)cccn2nncc12 76744,c1(C(N2C(CCNC(C(C)n3cncn3)=O)COCC2)=O)ncc2[nH]ncc2n1 76745,N1(C(c2cccc(N(C)C)c2)=O)CCN(C(=O)Cn2ncnn2)CC(O)C1 76746,c1(N2C(CCNC(C3(C(C)(F)F)CCC3)=O)CCC2)ncc2c(n1)COC2 76747,C1(NC(CN2CC(CC)C2)=O)CC2CC1CN(C(=O)C#CC1CCC1)C2 76748,c1(C(N2CC(CNC(C3(C(=O)OC)CCOC3)=O)C2)=O)ccc(N)c(Cl)n1 76749,Cc1cc(N(C)C)ccc1C(N1CCC(C(=O)NCc2nccc(Cl)c2C)C1)=O 76750,CC(Cc1cnc[nH]1)C(=O)NC(CC1CCC1)C(=O)NCC1CC(F)(F)C1 76751,N1(C(c2n(CC)ncc2Cl)=O)CC(NC(=O)CCCCN2CCCC2)C(C)(C)C1 76752,c1(C(N2CC3CN(C(c4cc5c(s4)CCC5)=O)CC32)=O)cc2ccccc2c(O)n1 76753,C(=O)(C1=NNC(=O)CC1)N1CCC(NC(C(C)Sc2ccncc2)=O)C12CC2 76754,c1(C(C)(C)NC(C2(C(C)N(C)C)CC2)=O)c(F)cc(Br)cc1F 76755,CCCC(C(=O)N1CCCC1C1(CNC(=O)Cc2ccsc2Cl)CC1)N(C)C 76756,C(=O)(C(F)(F)C(O)C1CC1)NC1CCC(CNC(=O)CC2(O)CCCC2)C1 76757,C1(NC(=O)C(c2cccn2C)=O)CCCCC1NC(c1n(CC=C)ccc1)=O 76758,C(=O)(C(O)C(F)(F)F)NC(CCCCNC(c1c(C)[nH]nc1Cl)=O)C 76759,N1(C(CCC)=O)CCCC2C1CCCN2Cc1cn(-c2ccccc2C=O)nn1 76760,C12(CC1(C)C)C(=O)N2.c12ccc(o1)C(=O)N(C)C2.C1(SC)(CO)CC1 76761,C#CCC(C(=O)N1CCC(C(C)(C)C)C1)NC(=O)Cc1cccnc1 76762,C(C(=O)NC1CC(CNC(C2CC2(F)F)=O)C1)(C(C)(C)C)NC(C)=O 76763,CCCCCC(=O)NC(C)C(C)NC(=O)C(N1CCN(CCO)CC1)(C)C 76764,C1(C(=O)OC)CN(C)CC1(C)C(F)(F)F.c12c(cccc1Br)NCC2 76765,Cc1cc(CNC(=O)CC2(C(=O)C3CC3)CC2)c(C)s1.c1(N2C(=O)C2)ccccc1 76766,C(=O)(C1=NNC(=O)CC1)N1CC2C(CNC(c3c(C)ncnc3)=O)(C2)C1 76767,N1(C(C2CC(C(F)F)(OC)C2)=O)CCC2(CC1)CC(C)N(C(C1CCCS1)=O)C2 76768,N1(C(CC2(N(C)C)CC2)=O)CCCC2(NC(=O)CCOCC(C)(C)C)CCCC12 76769,C1(CC)C(C(=O)NCC(C)(CNC(=O)CC2CCC(=O)N2C)OC)CCN1C 76770,c1(C(=O)NCC(CCOC)NC(=O)CCNC2CC2)ccc2c(c1)NC(=O)C2=O 76771,CC1CC(NC(=O)CSS(C)(=O)=O)CN1C(=O)Cc1cc(C2CC2)no1 76772,C1(NC(C2(N(C)C)CC2)=O)CCCC1NC(=O)CCOCC(F)F 76773,C#CC(CC)(CC)NC(C1(C(C)C)CCN(C(C2CCSC2)=O)C1)=O 76774,C(=O)(C#CC1CCCCO1)NCC(n1cc(CN(CC)CC)nn1)C 76775,N1(c2nnc(CCC)s2)CCCC2(CC(NC(=O)CC3(O)COC(C)(C)C3)C2)C1 76776,C1(C2(N)CCC2)(NC(=O)CNC(c2c(C)cnn2-c2ccccc2)=O)CCC1 76777,n1(CC)nnc2c(NC(=O)C(C)(C3CCCC3)NC(=O)NC)ncnc12 76778,CCCS(=O)(=O)NC(C)C(=O)NCC(C1CC1)N(C(=O)C(C)Cn1ccnc1)C 76779,c1(C(=O)NCCC2N(Cc3ccc(C)cn3)CCC2)n[nH]c2c(F)cccc12 76780,c1(N2CCN(C(COC)=O)CC2)[nH]c(=NC2CCC2CSC)nc2c1ncn2C 76781,C1(CCC)CN(C(=O)Cc2cncnc2)CCN1C(=O)Cc1scnc1C 76782,c1(N(C2CCCCNC2)C(c2cccc(F)c2Cl)=O)ncnc2c(F)cccc12 76783,CCS(=O)(=NC(=O)C1CCCCCN1C1CCNCC1)c1ccc(Br)cc1 76784,CCCCC(C)C(=O)N1CCN(C(C2CC(C)(C)C2C(F)(F)F)=O)CC1C 76785,O=C(CCCCn1ccnn1)NCC1CCCN1C(=O)C(c1ccc(F)cc1)F 76786,C1(C(=O)NC(C(=O)NC2CC(C=C)C2)CC2CCC2)CC2CCCC2C1 76787,O=CN1CCOCC1C(=O)NC1CCCCN(C(=O)C2=CCCC2)C1 76788,C1(C(=O)NCC(C)S(C)(=O)=O)CC12CCN(C(=O)C=CC1CCCCC1)C2 76789,n1(CC(=O)NC(CC)CN(C(=O)C(F)=C2CCC2)C)ccc2cc(F)ccc12 76790,C(CN(C)C)(C(=O)N(C)C)NC(C=CC(=O)N(C)C)=O.C12(CCC1)CCN2 76791,CC(C)C(C(=O)NC(C)CN(C)C(c1cc(Cl)no1)=O)NC(=O)Nc1ccccc1 76792,c1(CCC(N2CCC(C(C)NC(CC)=O)C2)=O)ccc(F)cc1F 76793,N1(C(C2N(C(C(CCC)NC(C)=O)=O)CC(F)(F)C2)=O)CCCC2(COC2)C1 76794,N1(C(C2C(OC)(OC)CC2)=O)CCC(CC(=O)NC2(C(=O)OC)CC2)C1(C)C 76795,C1(NC(CCn2cnc(=N)[nH]2)=O)CCCCCCC1NC(=O)CC1CCC(=O)N1 76796,N1(C(CCc2n(C)ncc2)=O)CCSCC1C(=O)NC1CC(C)(C)C1 76797,C1(CNC(C2C(C(=O)OC)C2)=O)CC(C(F)F)CN1C(=O)CN(C)C(C)=O 76798,N1(C(c2n[nH]c(CC)c2Cl)=O)CC2CCN(C(=O)Cc3nnc(C)o3)C(C2)C1 76799,Cc1cc(C(=O)N(CCCNC(=O)CS(=O)(=O)C(C)C)C2CC2)c(O)cc1F 76800,c1(C(=O)NC(C)C(N2CCC(O)CC2)=O)cnccc1C#N 76801,c1(OC)cc[n+]([O-])c(C(=O)NCCC2CN(C(c3ccc(Cl)cc3)=O)CC2C)c1 76802,C1(CNC(C(CC)CC)=O)CCC2CN(C(=O)C3=CCCOC3)CCC2C1 76803,N1(C(c2[nH]cc(C)c2)=O)CCn2cnc(-c3ccc4c(c3)OCCO4)c2C1 76804,Cc1cncc(C2C(=O)N2)c1.c1(C(=O)N(C)CCC2CCCN2C)cc(=O)cc[nH]1 76805,C=CCCCC(C)(C)C(=O)NCC1CCC1NC(=O)C(=Cc1cccnc1)C 76806,c1(NC(N2C(C)CCC2C)=O)ccc2cc(Cl)ccc2n1 76807,C12(CNC(C(C)N(CCC)C(c3ccc(C)o3)=O)=O)CCN(CC1)C2 76808,c1(C(N2CCC(OCCNC(C3(C=C)CC3)=O)C2)=O)c(C)nc(O)nc1C 76809,C1(CC(=O)NCC2N(CC)CCC2)CC(C)(C)CN1C(c1cnc(C2CC2)o1)=O 76810,N1(C(C=CCCC)=O)C2CCCC1CC(N=c1ncnc3[nH][nH]c(C)c1-3)C2 76811,c1(CC(C(=O)NCCN(C(C=CCC)=O)C2CC2)O)ccc(C(C)C)cc1 76812,C1(CNC(CCCc2c(C)ccs2)=O)C2CCC(C2)N1C(=O)C1=NNC(=O)C1 76813,N1(C(CC(C)(C)C)=O)CC2CCCC2(NC(c2ccc(N)cc2F)=O)C1 76814,Cc1cnc(N2CCCCC(CNC(C3CCN(S(C)(=O)=O)CC3)=O)C2)nc1O 76815,N1(CC(O)C)CC23CCCC2(C1)C3.c1ccccc1OC(F)F 76816,c1(C(=O)NC2C(C(N3CCC(C#C)CC3)=O)CCCC2)ccc(O)c(O)c1Cl 76817,n1(CC(=O)NCC2(C)N(C(C(C)SC)=O)CC(F)(F)C2)nc2c(n1)CCCC2 76818,CC(C)(C)CC(CO)NC(c1c[nH]nc1CCNC(c1ncccc1F)=O)=O 76819,c1(C(=O)NC23CN(C(Cc4c(C)n[nH]c4C)=O)C(C2)C3)c2c(nn1C)CCC2 76820,C1(C(N2C(C)CN(C(=O)N(C)C)CCC2)=O)COc2ccccc2O1 76821,CCN=c1ccc(C(N2CC(O)(CNC(=O)CCc3nnc(C)n3C)C2)=O)c[nH]1 76822,c1(CC)[nH]c(=N)sc1C(N1CC(O)CC1CNC(C1CC1C(C)C)=O)=O 76823,Cc1cccc(C(=O)NCC2CCC(NC(=O)C(C)(F)F)CC2)c1Cl 76824,C1(NC(CNC(C2CCCCC2)(C)CO)=O)CC2CCCC(C1)N2 76825,C1(CCNC(C(CC2CCCC2)NC(CCOCCOC)=O)=O)CCCN(C)C1 76826,C12(CNC(c3cc(C)cc(C)c3)=O)CC(CCO1)N(C(=O)C(C)CC(C)(C)C)C2 76827,N1(C(CCNC(=O)CO)=O)C(C(=O)NCC2CC23CCCCC3)CC2CCCC12 76828,Cc1cc(NCC2CCCO2)nc(C2CCN(C(=O)C(C)(O)C3CC3)CC2)n1 76829,N1(C(CSCC(N)=O)=O)CCC2CCC(NC(c3ccc(C(N)=O)c(Cl)c3)=O)C12 76830,c1(CO)cccc2ccnn12.Cc1cnc(N2CC(C(N3CCC(O)C3)=O)(CO)C2)nc1 76831,C1(CNC(COC)=O)(CNC(=O)C(C(C)C)NC(c2nccs2)=O)CC12CCC2 76832,C(=O)(C(C)CCC(C)(C)C)NC(C)C(N1CCC2(CCOC2=O)C1)=O 76833,N(C1CCCc2c1cnn2C)C(C(C)n1ccnc1)=O 76834,C(=O)(C(C)CCCOC)NC12CC(CNC(c3ccn(CC)c3C)=O)(OC1)C2 76835,C1(=O)CCCCCCN1.CC1(C)C(CO)CN1C(C1CCCOCC1)=O 76836,N1(CCNC(C(CC)OC)=O)CCCN(C(c2sc(=N)[nH]c2CC)=O)CC1 76837,C#CCCCC(C)C(=O)NCC1CCC12CCN(C(=O)CSC(F)(F)F)CC2 76838,CC1(C)C=C(C(=O)N2CCC(C)(NC(=O)CC3(C#N)CC3)C2)C1 76839,C1(CC=C)(C(=O)NCC2CSC2)CCCN1C(=O)CC1CC2CC2C1 76840,N1(Cc2ccc(SC)s2)CCC(O)C1C(=O)Nc1nc(C#N)cs1 76841,N1(C(Cn2nc(C)oc2=O)=O)CC2(CC2)CC1CNC(C12CCC(CC1F)C2)=O 76842,C1(C(=O)OCC(=O)NC2CC2)CC2CC1CN(C(=O)Cc1cncs1)C2 76843,CC1CC=C(C(=O)N2CC3(CC(NC(c4ccccc4OCCF)=O)C3)C2)CC1 76844,Cc1cc(C(N2CCCC2CC(=O)N(CC(C)(C)N(C)C)C)=O)co1 76845,C#Cc1cncc(C(=O)NC(C)CNC(C2(C)CCCCO2)=O)c1 76846,C=CCCC(F)(F)C(=O)NCC1(CO)CCCN(C(=O)C(CC)C(C)C)C1 76847,c1(C(=O)NC2C(CNC(C34CC(OC)C3C4)=O)CCC2)cc(S(C)(=O)=O)oc1C 76848,c1(OC)ccc(C2CCN(CC(=O)NCC(c3c(C)n[nH]c3C)C)C2)cc1 76849,N1(C(C2C(CC)N(C(=O)C(F)F)CC2)=O)CCCN(C)CC1C 76850,CC(CC(C)(C)C)C(=O)NC1CN(C(C2CCC(=O)N2)=O)CCC1C(F)(F)F 76851,N1(C(CCCCOCCC=C)=O)CCC(C(=O)NC(CC2CC2)C2CC2)CC1C 76852,N1(C(c2cc(C#N)[nH]c2)=O)CCC(CNC(=O)CC2CCCC2O)C(F)(F)C1 76853,C1(C(=O)NS(=O)(=O)CC2(O)CCOCC2)COCC12CCC2 76854,c1(C(N2CC(NC(CCC)=O)C(C)(C)C2)=O)ccnc2[nH]ncc12 76855,N1(C(C=C(CC)C)=O)CCC(C2CCN(C(=O)CCn3nc(C)cc3C)C2)C1 76856,c1(C(COC(C2C(C(=O)OCC)CC2)=O)F)ccc(F)cc1F 76857,N1(C(c2cnc(C(C)(C)C)s2)=O)C2CCC1C(CNC(C1CC1C(N)=O)=O)C2 76858,CC1(C)CCC(C)(C(=O)NC2CN(C(c3cncc4c3CCC4)=O)C3CC23)CC1 76859,c1(OCCC(=O)NCC2CCN2C)ccc(Cl)c(F)c1.C(=O)(CSCCCF)NC 76860,C1(NC(CNC(C)=O)=O)CC2C1CCN2C(c1cnn(C)c1Cl)=O 76861,N1(C(Cc2cccc(CC)c2)=O)CC(C)CN(C(=O)C(C)(C)CO)C(C)C1 76862,c1(CCC(=O)NCC2C(NC(C3CC(OC(F)F)C3)=O)COC2)nnc(S)nc1O 76863,N1(C(C(CC)C)=O)CCN(C(c2cc(C(=O)OC)on2)=O)CC1CC(F)F 76864,c1(C(=O)NCC2N(C(C(COCC)C)=O)CC2)cnn2ccsc12 76865,N1(C(CCn2c(C)csc2=O)=O)CCCN(C(=O)CCCCC#N)CC1C(C)C 76866,c1(C(=O)NCC(C(C)C)NC(c2cccc3nn[nH]c23)=O)ccnc2[nH]cnc12 76867,C1(C(=O)NCCC(C)(C)O)(CC)CCCN1C(c1ncccc1O)=O 76868,C(=O)(C(C)(C)CC=O)NCC.C(CCCNC(=O)CSCC)OCC 76869,C12(CCOC)CCN(C1)C(=O)c1csc(n1)C(C)O2.c1(C(=O)NC)ccns1 76870,Cc1c(F)ccc(C(=O)NC2(CNC(C3CCCCO3)=O)CCOC2)c1O 76871,CCC(C)CCCC(=O)NCC(N1CC(N(C)C)C2(CC2)C1)=O 76872,N1(C(CCCCCOCC)=O)CCC(N=c2cc[nH]cc2C#N)CC1 76873,N1(C(C2(C(=O)NC)CC2)=O)CC2CN(C(c3csnn3)=O)CC2C1C(C)C 76874,c1(OCC(=O)NCC2CN(C(C=C(C)C(C)C)=O)C2)cccc(C#N)c1 76875,C1(CC(=O)N(C(CNC(C2COC(=O)N2C)=O)C2CC2)C)CCCCC1(C)C 76876,C1(CC=C)(C(=O)NCCN(CCCC)CC)CCN(C(=O)CN2CC=CC2)C1 76877,C=CC(C)C(C)C(=O)N1CC(OCCNC(c2ccc(NCC)nc2)=O)C1 76878,C1(NC(CCSCCC)=O)CN(C(=O)C(C)(O)COC)CCC1C(F)(F)F 76879,C1(C)(CNC(C23OCC(COC)(C2)C3)=O)COCCN(C(c2cc(C)no2)=O)C1 76880,CCC(CC)CC(F)C(=O)NC1CC=C(C(=O)N(C2CCNC2=O)C)C1 76881,C1(CNC(COCCC)=O)CN(C(=O)C=Cc2cccc(O)c2)CC(C)(C)O1 76882,C(=O)(CCC(=O)C(C)(C)C)N1C(C(=O)NCCN(CCC)CCC)CNC(=O)C1 76883,c1(-c2onc(C(=O)Nc3ccc(C4CC4)cc3)n2)cc(Br)c2ccccc2c1 76884,C(=O)(C(C(=O)NC1CCCN(C(=O)C(N2CCSCC2)C)CC1)C(C)C)OCC 76885,C1(O)(CNC(C2(COC)CCC2)=O)CCCN(C(=O)C(=O)NCC(F)(F)F)CC1 76886,N1(CCCCC(c2nn[nH]n2)N(CC)CC)CCCC(C)C1C 76887,C1(N(CCOC)CCN2CCOCC2)CCN(C(=O)NC2CCCC2(C)C)CC1 76888,CC(C)C(F)(F)CC(=O)NC1CN(C(=O)CCCC2CCCC(=O)N2)C(C)(C)C1 76889,CC(C(C)C(=O)N1CCCC(N(C)C2CC2)C1)NC(=O)CCCNC(N)=O 76890,C(=O)(C(C#N)C(C)C)NC1CN(C(CC2(COCC)CC2)=O)CC1C(F)(F)F 76891,Cn1[nH]c(C(=O)NCCC2CCN(C(=O)CC34CCCC3C4)C2)nc1=O 76892,C1(C(=O)NCC2(CC(=O)Nc3cn(CC#C)nc3)CC2)CC(=O)OC1(C)C 76893,c1(C(=O)NCC(C)N(C(=O)CC(O)C(C)C)CC)c[nH]c2c(C)cccc12 76894,c1(NC(=O)NCC2C(N)CC2)nc(O)cc(O)n1 76895,c1(OC)cccc(C2CC2C(N2CCC(N(C)C(c3[nH]c(C)nc3C)=O)CC2)=O)c1 76896,c1(OC)ccc(C(c2c(C)ncn2C)NC(=O)CNc2ncc(F)cn2)cc1 76897,c1(C(N2CCN(C(c3cc(CCO)on3)=O)C3CC23)=O)cc2c(cn1)OCCO2 76898,C1(NC(=O)CCCF)CN(C(C23CCCC2CCC3)=O)CC2(CCC2)C1 76899,N1(C(C(C(CC)CC)F)=O)CC2(CCCN(C(=O)C(F)CCC(C)(C)C)C2)C1 76900,C1(C(=O)NCc2ccccc2CO)CCC(CN(C(=O)CC2CC2(Cl)Cl)C)CC1 76901,C1(F)(C(=O)NC(CNC(c2cc(C)[nH]c2)=O)CC(C)C)CCN(C)CC1 76902,c1(C(=O)N(C2CC3CC3C2)C2CC3CC2CN3)[nH]nc([N+](=O)[O-])c1Cl 76903,c1(C(=O)NCC(C)NC(C(C)C2CCC2)=O)cnc2ccccc2c1C(F)(F)F 76904,c1(C(N(CC(C)NC(=O)C2=COCC2)C)=O)nc[nH]c2ncc(Br)c1-2 76905,N1(C(C(C)=CC2CC2)=O)CCC2CN(C(=O)Cc3cnccc3C)CC2C1 76906,c1(CC)ccc(C(=O)NCC2CCN(C(C3CCC4(CC4)C3)=O)C2(C)C)c(C)c1 76907,c1(NC2CCCC2)ncc([N+](=O)[O-])cc1F.c12ccc(o1)C(=O)NCCN(CC)C2 76908,CC1CN(c2ncc(C#N)cn2)CC(C)CN1C(=O)OC(C)(C)C 76909,Cc1cccc2cc(C(N3CCCC(CO)(NC(=O)C4=CSCS4)C3)=O)sc12 76910,n1(CC=C)nc(-c2ccc(C)cc2)nc1C(F)C1CC1 76911,N1(C(C(C)NC(=O)C(N)=O)=O)CCN(C)C(CO)C1 76912,N1(C(=O)CC2CCOC2)CCC2(CCN(C(=O)CNc3ccccn3)C2)C1 76913,c1(N(C)C)ccc2c(N3CCN(c4cccc(Cl)n4)CC3)nc(Cl)nc2c1 76914,c1(C(N2CC(Cc3ncc(C)s3)C(F)C2)C(=O)NCCCF)cc(C)nnc1C 76915,C1(C(=O)NCC(N2CCCCC2)C)(NC(=O)CN(C)C)CCN(C)C1 76916,c1(NCC(CNC(C(C(CC)C)NC(C)=O)=O)CO)cc(C)c(OC)c(C)c1 76917,CCCC(C)(C)C(=O)NC(c1ccccc1)CNC(=O)C(C)S(C)(=O)=O 76918,Cc1ncnc(C)c1CC(=O)NCC(C)(C)CN(C(=O)CC1CCOC1(C)C)C 76919,N1(C(COCCC#C)=O)CC(C(=O)NCC(C)C(C)O)C(CC)C1 76920,c1(CN2C(C(N3CCSCC3)=O)C=CC2)cc2cc(Br)ccc2o1 76921,C1(C(=O)NCC2N(C(C)=O)CCC2)CCN(C(=O)Cc2ccccc2)C1(C)C 76922,N1(C(=O)COC2CCCCC2)CC2(CC(CC(N3CC4(CC=CC4)C3)=O)C2)C1 76923,O(C=CC(=O)N1CC(NC(=O)CSCC(=O)OC(C)(C)C)C1)CC 76924,N1(C(C2NC(=O)OC2)=O)CC2CCCC(NC(c3cc4ncccc4s3)=O)C2C1 76925,c1(N2CC(O)(C(C)NC(=O)C(N)=O)C2)ccc(C(N)=O)cc1[N+](=O)[O-] 76926,c1(C(=O)OCC(c2cccc(OC)c2)C)c[nH]c2ncc(F)cc12 76927,c1(C(=O)NC(CC)CN(C(=O)CNC(N)=O)CC)ccn(C)c(=O)c1 76928,c1(OC)ccccc1C(=O)N(C1CCC(NC(c2cnns2)=O)CC1)CC1CC1 76929,N1(C(C=CCC)=O)CC(NC(=O)CC2(C#N)CCC2)CC1CO 76930,N1(C(CCC(C)OC)=O)CC(C2CCN(C(c3cc(C)c(C#N)cn3)=O)CC2)C1 76931,Cc1c(C)n(C)c2ccc(C(=O)NC3CCOCC3NC(C3CC(O)C3)=O)cc12 76932,C=CC1OCCCC1C(N1CCC(OCCNC(c2nn(C)c(C)c2Cl)=O)C1)=O 76933,c1(OCC(=O)NC(C)C(C)NC(=O)CN2CCNC2=O)ccccc1Cl 76934,N1(C(C2C(CC)CCC2)=O)CCc2sc(C(=O)NC(C)C3CC3)cc2C1 76935,C1(N(C(C(C)OCC#C)=O)CCO)CCCN(C(=O)C(=Cc2ccccc2)C)C1 76936,C1(NC(c2ccc(C)o2)=O)(CNC(C2CCOCC2)=O)CC(F)(F)C1 76937,C1(CC)CN(C(c2ccc(Cl)nc2)=O)CCN1C(=O)CCc1cccc(OC)n1 76938,c1(CCCC)ccc(CC(=O)NC2CC2NC(=O)C(C)OCC2CCC2)cc1 76939,C1(C)(CC)CCC(C(=O)NCC(C)CC(=O)N(CC(N2CCCC2)C)C)O1 76940,c1(-c2ccc(C3(C(N4CC(OC)C(C)C4)=O)CC3)cc2)cc(F)cc(F)c1C 76941,C=CCC(C)C1(C)c2nnnn2CCN1.C1(SC)CCC(F)(F)C1 76942,CC(C)(C)C(CNC(=O)Cn1ncnn1)C(=O)NC(CCO)C(C)(C)C 76943,N1(C(Cc2c(C)cccc2F)=O)CCN(C(=O)COc2ccsc2)CC12CCC2 76944,C(=O)(CC(CNC(=O)C(COC)CC)OCC)NC1CC(C=C)C1 76945,C1(F)(C(N2CC(OCCOC)C2)=O)CCCN(C(=O)CC2CCCSC2)C1 76946,Cc1cc2c(C(=O)NCC3(C)CCCN3C(=O)Cc3cnc[nH]3)nccn2n1 76947,N1(C(CC(C=C)CCC)=O)CCN(C(=O)C(CC2CCCC2)CC)CC(C)(C)C1 76948,S(=O)(=O)(c1cccc(N2CCOC3(CCC3)CC2)n1)NC1C(C)N(C)CCC1 76949,N1(CCCn2cc(C)nc2)CCc2cnn(-c3ccc(C#N)cc3)c2C1 76950,N1(C(C(CCC)C)C(=O)NC2CCC2)CCc2c(CCC)cccc2C1 76951,c1(C(=O)CC=O)cnnn1-c1ccccc1.CC(CO)C1CCC1 76952,C1(NC(C2CN(S(CC)(=O)=O)C2)=O)CCCC(NC(=O)CSC2CC2)C1 76953,C(=O)(CCC(=O)NC=O)NC(C(=O)NCC(=O)N(C(C)=O)CC)COCC 76954,C123COC(C1)(C2)C(=O)NCC(CO)NC3=O.C1(CC)CCCN(C(=O)C(C)C)C1 76955,N1(C(COCCCCOC)=O)CCC(C(C)NC(C2(C)CC3CC3C2)=O)CC1 76956,C#CCC(CC(=O)NC1(C(F)(F)F)CC1)NC(C1(COC)CCOC1)=O 76957,c1(C(N)=O)nc(C(=O)NC2CC(CNC(c3cnn(CC(F)(F)F)n3)=O)C2)cs1 76958,c1(C(=O)NCC(C)CNC(c2ccc(-c3cc[nH]n3)s2)=O)ccc(C#N)c(Cl)c1 76959,N1(C(c2cnc(N(C)C)c(Cl)c2)=O)CCC(NC(C2(C)CCN2C)=O)C(C)(C)C1 76960,CC#CCCC(=O)NCC1CC(F)(CNC(c2c(SC3CC3)noc2C)=O)C1 76961,c1(OC)cc(C(=O)NCC2CCC2NC(=O)CCSC)cnc1OC 76962,C12(NC(c3ccc(CC)[nH]3)=O)CC1CN(C(=O)C(F)=C1CCCC1)C2 76963,C1(C(c2nnnn2C(C)(C)C)NCCc2c(OC)cccc2)CC2CCC(C1)O2 76964,c1(C(=O)NCC(CC)N(C(=O)CC2(C)CC2)C)cn(C)c(=O)c2cccnc12 76965,c1(OC)ncc(C)cc1C(=O)NCC1(C)CCCN1C(c1cnc(SC)nc1)=O 76966,C1(CCNC(CC2(OC)CCC2)=O)CCN(C(=O)CCn2cnnn2)C(C)C1 76967,c1(CC(=O)Nc2nnc(NC(c3onc(OC)n3)C)s2)ccc2c(c1)CCC2 76968,N1(C(COCC)=O)CC2COCC(C1)C2NC(=O)CCC1CCC(=O)N1 76969,c1(OCC)ccc(CC(=O)NC2(C)CCCN2C(c2cnc(C)[nH]2)=O)nc1 76970,C1(CC(=O)NCC(=O)NCCC2CC(NC(C(C)C)=O)C2)CC=CCC1 76971,N1(C(c2c(Br)cn(CC)n2)=O)C2CCC1(CNC(=O)CCCC(N)=O)CC2 76972,C=Cc1ccc(C(N2CC(O)CC2C(=O)Nc2cnc(C)c(C(N)=O)c2)=O)cc1 76973,c1(CC)ccc(C)cc1C(=O)NCC(CNC(c1ccc(C)o1)=O)S(C)(=O)=O 76974,c1(C(N(C2CCC(C#N)C2)CC(=O)NC(=O)C2CC2)=O)coc2c1COC2 76975,c1(NC(C(C)N(C(=O)COCCCN=[N+]=[N-])C)=O)cncc(Cl)c1 76976,C(=O)(C(F)CC(C)(C)NC(c1ccc(F)cc1O)=O)N(C1CCC(C)(C)C1)C 76977,c1(NC(C2CCN(C(c3c(Br)ccnc3Cl)=O)C2)=O)cccc2nsnc12 76978,N1(C(C(C)CCN(C)C)=O)CCC2(CCC(NC(=O)Cc3nccn3C)CC2)C1 76979,c1(C(C)Nc2nccc(=NCC3CC(=C)C3)[nH]2)cc2c(cc1OC(F)F)OCO2 76980,C1(NC(c2n(C)ccc2)=O)CCN(C(=O)CCC2CC2)CC12CCC2 76981,N1(C(C(COC(C)C)NC(C(CCC)OC)=O)=O)CCN2C(=O)CCC2C1 76982,c1(NC(C(=O)NC(CC)C2CC2)=O)cc(S(C)(=O)=O)ccc1OC.N1(CC)CCCCC1 76983,C1(N(C)C(C2CCCC2F)=O)(C(=O)NCC2(C)CCCCCC2)CCC(C)(C)C1 76984,N#Cc1c[nH]cnc1=NC1COc2cc(C(=O)N=c3ccnc(Cl)[nH]3)ccc2C1 76985,C1(c2nnnn2C(C)(C)C)(NCc2ccc(C(C)(C)C)nc2)CC2COCC2C1 76986,c1(C(N2CCC2c2ccccc2)=O)cnc2c(c1)CN(Cc1c(C)nc(C)s1)CC2 76987,CC1(C)C(CNC(=O)CCNC(=O)CO)CCN1C(=O)C(O)C1CC1 76988,C12(NC(c3c(OC)c(=O)cco3)=O)CCCC1CN(C(c1cc(=O)cc[nH]1)=O)C2 76989,CCC(C)C(=O)C(=O)N1CCC(F)(C(=O)Nc2cnc(F)nc2)CC1 76990,N1(C(Cc2nc(C)oc2)=O)CCOC(CCNC(c2cc(C(F)F)ccn2)=O)C1 76991,C12(NC(c3c(C(C)=O)scc3)=O)CCCC1N(c1ncnc(Cl)c1C#N)CC2 76992,C1(C(=O)NC2(CF)CCN(C(CSCC(N)=O)=O)C2)CC(=O)NC(=O)C1 76993,C1(C)(C(=O)OC)CN(C(=O)CC2CC(F)(F)C2)C1.c12cc([nH]n1)CNC2=O 76994,CC(C)C(C)CC(=O)N(C1CC(C(=O)NC(C)CS(C)(=O)=O)C1)C 76995,O=S1(=O)CC2CN(c3ncnc(-c4cnn5ccccc45)n3)CC2(C(F)(F)F)C1 76996,c1(C(=O)NCC2C(C)CN(C(=O)Cn3nnc(=N)[nH]3)C2)csc2cc(Cl)cnc12 76997,CCCC(C(=O)NCC(C)(C)NC(=O)CC1CC(OC)C1)OC 76998,c1(C(N)=O)ccc(Br)c(S(=O)(=O)N2CCN(CC3CCOCC3)CC2)c1 76999,N1(C(CC)=O)CCC(C(=O)NC2CC(F)(C(=O)OCC)C2)CC1 77000,c1(NC(=O)CNC(c2ccns2)=O)cccc(Cl)c1Cl.N12CC3CC1C3NCC2=O 77001,c1(CN2CCC(CNC(c3cccc(C)c3)C(C)C)CC2)c(F)cccc1Cl 77002,N1(C(CCC=CCC=C)=O)CCCC(CNC(c2csnc2C)=O)C1C 77003,CS(=O)(=O)c1cnc(CCNC(=O)NC2COCC2C2CC2)nc1 77004,CC1CCC(C)C1NC(=NCCCCCCCCOC(F)F)N.c1(OC)ccc(Cl)cc1 77005,c1(C(=O)NC2CC(CNC(C3C(C)CCC3)=O)C2)cc2sc(Br)cc2s1 77006,c1(N(C)CCc2ccco2)cc(Br)ccc1S(=O)(=O)N1CCC(C2CC2(F)F)C1 77007,C(=O)(CC(C)(C)C(=O)OC)N1CCC(OCC2(C#C)CCCC2)C1 77008,C(=O)(CC(COC)NC(C1(C)CNC(=O)C1)=O)NCC(C(=O)NC)O 77009,C(=O)(C(C)CC(C)(C)C)N.C1(COCC)CCN(C(C2(CC)CCOC2)=O)CC1 77010,C=CC(CCC)CC(=O)N(C(C)CNC(c1ccc(CN(C)C)[nH]1)=O)C 77011,C1(C(=O)NC2CCCC2CNC(=O)CCc2ccncc2)(COC)CCCC1 77012,Cc1onc(C(=O)NCc2ccc(CF)cc2)c1CS(N)(=O)=O 77013,c1(C(=O)NCCCC2N(C(C#CC(C)C)=O)CCC2)nccc2c(Cl)cccc12 77014,c1(C(=O)NC(C(C)NC(c2cccc(CO)c2)=O)C)ccc(O)c(N)n1 77015,C(=O)(CCCCCC(C)O)NCC1CC(NC(c2cc(C)c(C)[nH]2)=O)C12CCC2 77016,N1(C(C(c2n(C)ncc2)NC(C2CC3(CCC3)C2)=O)=O)CC(O)C(O)C1 77017,c1(C(N(C(CSC)C)C)=O)cc(CNC(c2csnn2)=O)ccn1 77018,C(=O)(C(C1CC1)N(C)CC1SCCS1)NCC(=C)C 77019,C1(NC(C(C=CC)O)=O)CCCC(CC(=O)NCCc2cc(CC)no2)C1 77020,C(CNC(=O)C(C)Cc1ccccn1)(CC(F)(F)F)NC(C=C(C)C(F)F)=O 77021,Cc1ccc(Br)c(C(=O)NC2(C)CCN(C(c3c(C)cccc3O)=O)C2)c1 77022,c1(NC(c2c(CNC(c3cnsc3)=O)ccs2)=O)cnc2ccnn2c1 77023,C(=O)(C(C1CCOc2ccccc21)N1CCc2cc(Cl)cc(C)c2C1)NCC=C 77024,C1(CNC(C2N(CC)CC2)=O)CN(C(C2CCCSC2)=O)CCC1(C)C 77025,c1(NC(CNCC(=O)OC)=O)ccc2ccccc2n1.C(C(F)(F)F)O 77026,C(=O)(C(F)CCC(C)(C)C)NC(CN(C)C)C(N1CCC(CO)C(C)(C)C1)=O 77027,C(=O)(C1(C)CCc2ccccc21)NCCCNC(C1CCC(CC)CC1)=O 77028,CC(CC(C)(C)O)c1nc(Cc2nnc(-c3ccccc3Br)o2)no1 77029,C(CCCCC(=O)NC1CCCCCC1C(=O)NCCC(COC)OC)OC 77030,C(=O)(C1=CC2CC=CCC12)NCC1CCN(C(c2c[nH]c(=NCC)s2)=O)CC1 77031,Cc1c(C(=O)N(CCCNC(C2CC(C(C)(C)C)C2)=O)C(C)C)nnn1C(C)C 77032,CCC(CC(F)F)C(=O)NCC1(F)CN(C(C2(C3CCCCC3)CC2)=O)C1 77033,N1(C(C2C(C)(CC)C2)=O)Cc2nccn2CC(NC(=O)C(c2cnn(C)c2)C)C1 77034,Cc1cc(C(=O)NCCN(C(=O)C(F)F)C(C)C)n2ncnc2n1 77035,C#Cc1ccc(C(N2CC(C(N3CCC(N(C)C)C3)=O)C(C3CC3)C2)=O)c(C)c1 77036,CN1CCC2(C1)C(=O)N2.C(=O)(C#CC1CC1)N1CC(c2ccccc2)C1 77037,N1(C(c2c(C)nccn2)=O)CCCC(C2CCCN(C(=O)Cc3cocn3)C2)C1 77038,c1(NC(C2C(C(=O)OC)C2)=O)cccc2c1NC(=O)CO2.C1(=O)C(N(C)C)CN1 77039,C(=O)(C(C)(O)C(F)(F)F)C(C)=O.c1(COCC)cnc(OC)c(C(N2CC(N)C2)=O)c1 77040,C1(NC(C2(C)CC=CC2)=O)CN(C(=O)C(F)=C2CCC2)CC1O 77041,CCCC(CC(=O)NCCC(C(C)C)OC)NC(=O)CC1COCCO1 77042,C1(CNC(C(C(C)C)N2CCCC2)=O)CCN(C(=O)CCC(F)F)C1(C)C 77043,Cc1cc(C)c(C(N2CCOCC(NC(=O)Cn3cccn3)C2)=O)c(Cl)n1 77044,N1(C(c2c(CC)nco2)=O)CC2CCCN(C(c3ccc(C)c(C)c3O)=O)C2C1 77045,c1(NCC(=O)NC(CC2CN(C(C(CC)C)=O)C2)C)cccc(Cl)c1 77046,c1(OCC)ccccc1C=CC(N1CCCC(CNC(C2(COC)CC2)=O)C1)=O 77047,n1(CC(C)C)cc(C(F)F)c(NC(c2cc(CCN(C)C)on2)=O)n1 77048,C1(CC(=O)NC(c2cc(F)cnc2Cl)C)CCCCC1(F)F 77049,N1(C(CCc2c(C)n[nH]c2C)=O)CCC2(CCCN2C(=O)CC2CSCCS2)C1 77050,CCCCCCC(C)C(=O)NC(CNC(=O)C(CC)n1ccnc1)CC 77051,N1(C(C(CCC#C)O)=O)C2CCC1CC(CNC(c1cc(Br)no1)=O)C2 77052,C1(CC)CCN(C(=O)C(C)Cc2ccccn2)C1CNC(=O)C(F)CC 77053,CCC(CC(F)(F)F)C(=O)NC1CC(NC(=O)CC(CN(C)C)C(F)(F)F)C1 77054,C1(CNc2[nH]c3ccccc3c2C2OCCO2)CCc2cc(Br)ccc2NC1=O 77055,CC(C)(C)C(CNC(c1nsnc1O)=O)NC(C1C=CCCC1)=O 77056,C1(COC)CC(CNC(c2nc(Cl)sc2C)=O)N(C(C2CCC(=O)NC2)=O)C1 77057,N1(CCCOC)CCC(NC(N2CCN(c3ccnc(C)n3)CC2)=O)CC1 77058,c1(OC)nc(=NCCc2ccc(OC3CCN(CCF)C3)cc2)[nH]c2c1CSC2 77059,N1(Cc2n(CCC)ncc2)CCCC(CNC(c2ncccc2Cl)=O)C1 77060,CCS(=O)CC(=O)N1CCCC1C1CCN(C(C2COCCN2C)=O)C1 77061,C1(CNC(C2CCC(NC(C3(CC)CC3)=O)CC2)=O)CC2(C1)CC(O)C2 77062,C1(COC)(NC(=O)C(C)Cc2ccncc2)CCN(C(C2(C)CC(C)=NO2)=O)C1 77063,n1(CC)cc(C#N)c(=NC(=O)C2C3CN(C(C4CCCC4C)=O)CC23)[nH]1 77064,N#CC1CN(C(c2cccc3c2OCO3)=O)CCN1C(c1ccccc1)=O 77065,C(C(C)(COC)C(=O)N1CCCCC1CNC(c1cnn(C)c1)=O)OC 77066,CCCC(C)(O)CC(=O)NCC1CC2CCC1N2C(c1cc(C#N)ccc1C)=O 77067,N1(C(=O)CSCc2cccc(Cl)c2)CC2CC(NC(C3(Cl)CC3)=O)C(C2)C1 77068,c1(C(N(C(CNC(CC(C)c2ccco2)=O)C)C)=O)ccnc(-c2ccco2)c1 77069,N1(C(c2c(SC)cccc2)=O)CCN(C(=O)C(C#N)C(C)C)C(CCO)C1 77070,c1(C(N(C(C)CNC(c2nnsc2C(F)(F)F)=O)C)=O)nc2ncccn2n1 77071,C(=O)(C(C)(O)c1ccccc1)N(CC(CC)NC(=O)Cc1cncs1)C 77072,c1(NC(C2N(C(=O)Nc3c(C)cc(F)cc3)CC2)=O)ccc(C)c(C)c1F 77073,C1(CNC(c2c(C)[nH]nc2C(C)C)=O)COC(C)(C)CN1C(C1CC12CC2)=O 77074,CN1C(=O)NCC1C(=O)NCC1CC(NC(c2cnc(C(F)(F)F)nc2)=O)C1 77075,C(=O)(CC(C)CCCCC)N(S(c1c(CCC)c(C)[nH]c1C)(=O)=O)CC(=O)OC 77076,N1(C(C2CC(=C)C2)=O)CC(C)CCC1CNC(c1ccc(C(C)C)c(F)c1)=O 77077,C(=O)(C(O)C(C)(C)CC)NC1CC(C(=O)NC(C#C)C2CC2)CC1O 77078,CN1CCCCC1C(N1CC2CC2(CNC(=O)C=Cc2ccncn2)C1)=O 77079,C1(CC(=O)N(CCOC)CCNC(=O)C=C(C)C(F)F)CNC(=O)C1 77080,O(P(C)(=O)CNC(C1CCN(C(c2cc(C)c(N)o2)=O)C1CC)=O)CC 77081,c1(C(=O)NC2CCC(CCNC(C3N(CCC)CCC3)=O)C2)ccc(F)c(O)c1 77082,c1(NC(=O)CNC(C23C(CN(C(C4C(COC)C4)=O)C2)C3)=O)cccc([N+](=O)[O-])c1 77083,CC(CNC(=O)C(Cc1ccoc1)NC(=O)CSc1cn[nH]c1)C(C)(C)C 77084,C1(CC)CCCCN1CC(=O)NC12CC(C(=O)OCCN(C)C)(C1)C2 77085,c1(OC)ccc(-n2nc(C(C)OC)nc2-c2nnc(C3CCC3)o2)cc1 77086,c1(NC(C2CC2C(N2CCCC(C#C)C2)=O)=O)cccc([N+](=O)[O-])c1C 77087,c1(C(=O)NC2C(NC(C(COC)N(C)C)=O)CCC2)ccn(C)c1C 77088,c1(C(N2C3C(C(=O)NC4(C(C)C)CCC4)C(C3)C2)=O)nnc(O)nc1O 77089,c1(CC)[nH]nc(C(N2CCC(CCNC(=O)CC3(C4CC4)CC3)C2)=O)c1Br 77090,C1(=O)C(C)(C)C(=O)N(C)CC(C)N1.C#CCCCOCC(=O)OC 77091,c1(CC)c(C(N2CCCC(NC(C3CC(C)(F)C3)=O)C2)=O)cnn1C(C)(C)C 77092,C1(CC=C)(C(=O)NC(C)CCF)CN(C(C2CCC(=O)C2)=O)C1 77093,C1(N(C(=O)CCCF)CC)CCCN(C(c2cn(C(C)(C)C)nc2Br)=O)C1 77094,C1(N(CC)CC)CCN(C(=O)CC(CCC)NC(=O)CN2CCCC2C)C1.OC 77095,C12(NC(c3cn(CC)nn3)=O)CCCC1N(C(c1c(C)cc(O)nc1C)=O)CC2 77096,N1(C(COCC)=O)CCCCCC(NC(c2cnn(CC(C)(C)O)c2C)=O)C1 77097,C1(NC(c2n(CCC)nnn2)C2CCCOC2)CCC(=O)N(CC)C1 77098,c1(C(=O)NCCOCCN(C(C2C(CC)OCC2)=O)C)ccn2cc(C)nc2c1 77099,c1(OCC(=O)NC2(CNC(CSCC)=O)CCOC2)ccccc1Br 77100,CC(N=c1nc2scnc2c(NCCS(=O)(=O)C(F)F)[nH]1)c1cn[nH]c1 77101,c1(NC(C2C(C)(C)COCC2)c2nnnn2C2CC2)cccc(P(C)(C)=O)c1.C1CC1 77102,C(=O)(CCCC(C)(C)C)N1CCCC(CCNC(c2cn(CCOC)nn2)=O)C1 77103,C(C1(C)OCCc2ccccc21)NC(C1CN(C)CCO1)C 77104,N1(C(c2cc(C)on2)=O)CCCC(N(C(=O)CCCOc2ccccc2F)C)C1 77105,c1(CC(=O)OC)ccc(Cl)c(CN2CCCC(OCC(C)C)C2)c1 77106,N1(C(C(CC)CC2CCCC2)=O)CCN(C(c2cccc(Cl)c2N)=O)CC1CF 77107,CC(C)CCC(C(=O)NCC1(F)CC(CO)C1)NC(=O)CC=CC(C)(C)C 77108,C(=O)(C1=CC2C=CC(C1)C2)N1CC(NC(C(COC)(C)C)=O)C(C2CC2)C1 77109,c1(C(=O)NCCC(C)=O)ccc(-c2cn(CCCCCO)nn2)o1 77110,c1(C(=O)OC)cc(C(N2CC(NC(=O)CN=S(C)(C)=O)CC(F)C2)=O)cc(C)c1 77111,S(=O)(=O)(c1ccc2nc(N3CC4CC=CC3O4)sc2c1)N1CC2C(C)(CC2)C1 77112,N1(C(c2csc(C#N)c2)C(=O)NCCCCCC)CC2CC(O)C(O)CC2C1 77113,Cc1c(N)ccc(C(N2CCC(=CCNC(C3CCCC3(F)F)=O)CC2)=O)c1F 77114,Cc1nc(C(=O)N(C2CC(NC(C3(Cl)CC3(C)C)=O)C2)C)c(=O)[nH]c1C 77115,C1(CCC(N2CCC(CN(C)C(C3(F)CC3)=O)C2)=O)CC(C)(C)CO1 77116,N1(C(CCCn2c(C)nc(C)n2)=O)CCCCC(CNC(c2ncccc2C)=O)C1 77117,CC1(C)CC(NC(=O)CNC2(C)CCC2)c2cc(F)ccc2O1 77118,c1(C(=O)NCC2CC(CNC(c3nc(CCC)oc3)=O)OC2)cc(C)n(C)n1 77119,CCCC(CC(=O)NCc1c[nH]nc1C1CCC1)NC(=O)OC(C)(C)C 77120,c1(C(=O)NC2(CN(C(C(CC(C)C)(C)O)=O)C)CC2)ccc2c(c1)C=CS2(=O)=O 77121,N1(C(c2c(OC)ccs2)=O)CCC(CC(C)NC(=O)C(C)(C)CC)CC1 77122,c1(C(=O)NC(C(C)C)CNC(c2ccc(C3(C)CC3)cc2)=O)ccc([N+](=O)[O-])[nH]1 77123,c1(OC)ccccc1C(N1CCC=C(F)C1)C(=O)NCCCOCC1CC1 77124,C12(NC(CCN(C(C=C(COC)C)=O)C)=O)CCC(C1)OC2C 77125,C1(NC(CC(CC)COC)=O)C2CCCN(CCCS(C)(=O)=O)C2C1(C)C 77126,CC(O)C(C)(C)C(=O)N1CC2CC1(C(=O)NC(C)Cn1cnnc1)C2 77127,c1(COC)ccc(C(=O)NC2CC(CNC(C3CCC(=O)C3)=O)C2)cc1F 77128,C1(CNC(c2c(C)nc(CO)o2)=O)CCC(C)CN1C(=O)CC1(C2CC2)CC1 77129,C=CC(C)(O)CC(=O)N(CCC(=O)N1CCC(CSC)C1)OC 77130,c1(C(=O)NCC2CCC(NC(C3C=CCC3)=O)CC2)c[nH]c2nc(Br)ccc12 77131,c1(C(N(CCCNC(C2CCC(C)CC2)=O)C2CC2)=O)cc([N+](=O)[O-])ccn1 77132,c1(C(N2C(C(C)NC(=O)CCF)CCCC2)=O)cnc2[nH]cnc2c1 77133,C(=O)(C(C(CC)CC)OC)NC(CCCC)CNC(=O)C(C)(C)CC1CC1 77134,C1(NC(C=Cc2ccc(C)o2)=O)CCC12CN(C(c1cc(Br)cn1C)=O)C2 77135,c12coc(c1)CNC(=O)CN2C.c1(CNC(=O)CCn2cccn2)nnc(S)s1 77136,CCCS(=O)(=O)N1CCCC1C(N1CC(NC(C23CC(C)(C2)C3)=O)C1)=O 77137,c1(CNC(C2(CC#C)CCC2)=O)nc(CNC(C2CCC2C(F)F)=O)cc(O)n1 77138,CCS(=O)(=O)c1ccccc1CC(=O)NCC1CC(NC(C2(CF)CCC2)=O)C1 77139,C1(C(N(CCCCNC(CSCC=C)=O)C)=O)CCC(=O)CC1C 77140,N1(C(C(CO)N(C)C)=O)CC2CC(C1)CN(C(c1n[nH]c3c1CCOC3)=O)C2 77141,C1(CC(=O)NCC=CCNC(c2ccn(CCF)n2)=O)CCC(=O)NC1=O 77142,n1(CC(=O)NC2C(NC(C(C)c3ccco3)=O)CC2)nccc1C1CC1 77143,c1(CNC(=O)Nc2c(CS(C)(=O)=O)cccc2)nc2ccc(F)cc2[nH]1 77144,N1(C(c2cc(C(C)C)oc2C)=O)CC2(CC2)CC1CNC(C1(C)CC(OC)(OC)C1)=O 77145,N1(C(C(C=C)O)=O)CCC2CCCN(C(=O)COc3ccc(F)cc3)C2C1 77146,CC1CC(=O)NC(C(=O)NCC(O)CNC(=O)C(=O)NCCC(N)=O)C1 77147,c1(CNC(=O)CC2CCCO2)cccnc1CNC(C1CCC(F)(F)C1)=O 77148,CCCC(CNC(c1cc(C(=O)NC)co1)=O)C(=O)N1CCC1CF 77149,CCC(C)(C)C(O)C(=O)NCC1CN(C(=O)COC2(C)CCCC2)CC1(C)C 77150,CN1CCn2nc(C(NC3CCc4ccc(C(=O)O)cc43)=O)cc2S1(=O)=O 77151,c1(C(=O)NCC2=CCCN(C(CCC(CC)C)=O)C2)nccn2cnnc12 77152,CC1CC(CC(=O)NCCCn2cnnc2)CN1C(c1ccnc(CO)c1)=O 77153,c1(C(=O)NCCN(CC(C)O)C(=O)CC2C=CS(=O)(=O)C2)cc2c(nc1N)CCC2 77154,c1(C(N(CCC)CCNC(C2CC2Cl)=O)=O)ccc(-n2ccnc2)c(C)c1 77155,Cc1n[nH]c(=NCO)o1.c1(COC)ccco1.C(=O)(C1CC1)NCCOCCOCC 77156,C(=O)(C1OCCn2ccnc21)NC(C)CNC(c1ccc2c(c1)NC(=O)CO2)=O 77157,CCCCC(CNC(=O)CCC(C)=O)NC(=O)Cc1csc(C)c1 77158,c1(-n2c(-c3cnns3)nc(-c3ccc(O)cc3)n2)nc2ccccn2n1 77159,N=c1ccc(C(N2CCC(CNC(c3csc(O)n3)=O)C2)=O)n[nH]1 77160,C1(C)(C(=O)NCC2C(C(N3C(C(=O)OC)CC3)=O)CC2)CCC2CC2C1 77161,C1(C(=O)NCCCn2cc(CNC(C(C(C)C)C)=O)nn2)CCCCNC1=O 77162,Cc1cc(Cl)cc(Cl)c1OCC(N1CCC(CCNC(C2CC(C)CO2)=O)C1)=O 77163,C1(C)(CNC(=O)OC(C)(C)C)CCN(C(c2cc(N)c(O)nn2)=O)CC1 77164,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CCN(C(CCCNC(=O)OC)=O)CC1CO 77165,c1(C(N(CC(C)NC(c2ccc(C(C)(F)F)cc2)=O)C)=O)ccc(N)c(O)c1 77166,c1(N(C)C)ccc(CN2CCOC(C(=O)Nc3nncn3C)C2)c(F)c1 77167,CCC(CC)C(c1nnnn1CCCF)Nc1cncc(C)c1 77168,N1(C(C(=O)NC2C(C(=O)OC)CN(C(C)C)C2)=O)CCCCC(C)C1 77169,Cc1cc(C(N2CC(NC(=O)Cc3cc(Cl)ccc3Br)CC(F)C2)=O)c(Cl)cc1F 77170,CCCC(C(=O)N1CCC(NC(=O)COC2CN(C(C)=O)C2)C1)NC(C)=O 77171,C1(C(=O)Nc2cccc(CNC(=O)C(O)c3ccco3)c2)(OC)CCCCCC1 77172,C(=O)(C(CNCC)N(C)C)N(CCC)C.C1(CC=O)OCCCOC1 77173,C1(C(N(CCNC(=O)CSC)CC)=O)CC(NC(=O)C(C)O)C1.C1(C)CC1 77174,c1(CN(C(=O)C(C2CCC2)NC(=O)CCc2cnn(C)c2)C)cccnc1 77175,C1(C(=O)NC(CCO)C2CCC2)(CC)CN(C(C2CC2Cl)=O)C1 77176,c1(OCC)cc(C(=O)NC2(CNC(C3CCC3(C)C)=O)CC2)on1 77177,c1(NC(C(=O)OC)Cc2cnc[nH]2)ccccc1NC(C1CC1N(C)C)=O 77178,N1(C(Cn2cc(C(C)O)nn2)=O)CCC2CN(C(=O)Cn3cccn3)CC2CC1 77179,CC(C(F)F)=CC(=O)NC(CNC(=O)CSc1cn[nH]c1)C1CC1 77180,c1(C(N2CC3C(NC(C(C=C)O)=O)CC(CC3)C2)=O)cc(F)c2ncccc2c1 77181,C(=O)(C(C)(C)CC(F)F)NCC(CCC)C(=O)NC1CCC(C#N)CC1 77182,c1(OC)ccc(CNC(=O)CC2CCCN2S(=O)(=O)Cc2ccccc2)cc1O 77183,CN1CCCN(C(CC2CC(F)(F)C2)C(=O)NCCC2(C)CC2)CC1 77184,c1(OCC(N2C(CN(C)C(c3cc(C(F)F)on3)=O)CCC2)=O)ccccc1F 77185,N1(C(C(C)CC2CCC2)=O)CCC(C(C)NC(=O)CC(C2CCCC2)C2CC2)CC1 77186,N1(C(CCCC2C(C)C2)=O)CC(N(C(=O)COCCN(C)C)C)C2(CC2)C1.CNC 77187,C1(=O)CCC(=O)NC(CC)CN1C.C1(CCNC(=O)C2CC2)(SC)CCCC1 77188,C1(CC#C)(C(=O)NC(C)CCN(C(=O)Cn2cc(Cl)c(C)n2)C)CC=CCC1 77189,c1(C(=O)NCC2(CCNC(c3cc(C(C)C)no3)=O)CC2)cc(C#N)ccc1O 77190,c1(C(=O)NC(CNC(c2ccc(C)o2)=O)C2CCC2)cc(N)ccc1[N+](=O)[O-] 77191,C(=O)(CC(C)(C)CNC(=O)C(CC(C)C)OC)N1C(C(=O)NC)C=CC1 77192,c1(C(C(=O)NCCCOCCO)N(C(C)C)C)cccc(Cl)c1 77193,CC1C(C(N2CC=CCC2)=O)CCN1C(=O)CC1CCCCCC1 77194,N1(C(C2(SC)CCOCC2)=O)CCC2(CC1)CCN(C(=O)Cc1n[nH]c(C)n1)C2 77195,N1(C(C(C)NC(C)=O)=O)CCC(CNC(C(F)(F)F)c2cnn(C)c2)C1 77196,CC(C)CC(C)C(=O)N1CCCC(F)(C(=O)NCCCc2cc[nH]n2)C1 77197,N1(C(COc2ccn(C)n2)=O)CC2CC1(C(N1CCOCC1CC1CC1)=O)C2 77198,c1(CCC(=O)NCC23CCC(C2)C3)cc(Br)sc1Br 77199,c1(C(=O)NCCOCCNC(C2C(SC)CCC2)=O)c(C)nc(C)n1O 77200,C1(CNC(C(C)OCCC#C)=O)N(C(=O)C(C)C2CCCC2)CCC1(C)C 77201,c1(SCCCNC(CN(C(=O)CCC(N)=O)CC)=O)ccc(OC)c(O)c1 77202,c1(C(N(CC(C)(C)CNC(C2CC2F)=O)CC)=O)ncccc1Br 77203,C1(C(=O)NCC2(C)CC2)(NC(C2CC23CCOC3)=O)CC(F)(F)C1 77204,c1(NCc2ccc(-c3c(C)ccc(O)c3)o2)cc(F)c(Br)c(F)c1 77205,C1(CNC(COCCCOC)=O)CC2CCC(C1)N2C(=O)C(C)(C)C(C)C 77206,Cc1ccc(O)c(C(=O)NC(C)(CO)C(=O)NCCN2CC3CC3C2)c1 77207,c1(CC)nnsc1C(N1CC(N(C(=O)COCC2CC2)C)C1)=O 77208,N1(C(c2c(C)n(C)nn2)=O)CC(CNC(c2nccs2)=O)CC(C)(C)C1 77209,C1(NC(c2cccc(C)c2)=O)CCN(C(c2ccc(C(N)=O)[nH]2)=O)C(C)C1 77210,c1(C(N2CCN(C(C3CCc4cnnn4C3)=O)C(CO)C2)=O)cc2n(n1)CCCO2 77211,NS(=O)(=O)CCCCC(=O)N1CCC(NC(=O)CCc2ccccn2)CC(O)C1 77212,Cc1nn(CCO)cc1C(N1CCOC(C2CN(C(=O)CCC3CCC3)C2)C1)=O 77213,c1(C(N2C(C)CCC(CNC(=O)CC3CC3(C)C)C2)=O)ccc(Cl)c(Cl)c1N 77214,n1(CC(=O)N(C2CCN(C(C(C)SCC)=O)CC2)CC2CC2)ccc(C)cc1=O 77215,C1(CN(C(=O)Cc2cn(C)nc2Cl)C)CCN(C(=O)CCN2CCCCC2)CC1 77216,c1(N2CC(C)CS(=O)CC2)nc(=NCc2nc(C(C)(C)C)n[nH]2)[nH]c2c1COC2 77217,C(=O)(CCC(=O)N(C)CCN(C)C(C1OCCOC1C(F)(F)F)=O)OCC 77218,C1(CNC(CSCC#C)=O)CN(C(c2cccc(F)c2CC)=O)CCC1(C)C 77219,c1(OC)ncnc(C)c1NC(=O)C(N1CCN(C2CCOCC2OC)CC1)=O 77220,N1(C(C2C(C(=O)OC)C=C2)=O)CC=C(CNC(C2CCCN(C)C2)=O)CC1 77221,CCC(CNC(c1ncccc1F)=O)(CC)C(=O)NC1CC1CF 77222,C(CCS(C)(=O)=O)NC(C1N(C(C(c2ccnn2C)NC(C)=O)=O)CCC1)=O 77223,CC1CN(C(CCn2cc(-c3cccn(C4CCC4)c3=O)nn2)=O)CC(C(=O)O)O1 77224,C1(CC)CN(C(c2cn(CC)nn2)=O)CCC1NC(C1(C)CCN(C)CC1)=O 77225,N(C(=NCCF)NCC12CC(C1)C(C(F)(F)F)O2)C(C)C1CC1 77226,c1(C(N(C)C)=O)cccc(C(N2CC3CC3(CNS(=O)(=O)CCCl)C2)=O)c1 77227,c1(N2CCC(CC=C)(NC(=O)CN3CCOCC3)C2)ncnc2c1CCC2 77228,N1(C(C2CCC(C(=O)OC)C2)=O)CC(C(=O)NC(C)CC(C)C(F)F)CC1(C)C 77229,C1(C(=O)NCC(C)(C)OCCCNC(C=CCCC)=O)CC(=O)NC(C)C1 77230,c1(C(=O)NCc2cnc(=N)[nH]c2)ccc(C(=O)O)c(F)c1 77231,C(=O)(C1=NN2CC(C)CN=C2N1)N1CC(O)(C(C)NC(c2cc(C)sc2)=O)C1 77232,Cc1cc(N2CCN(C(C3CCCC4(CC4)C3)=O)CCC2C)n2ncc(C)c2n1 77233,C1(O)(COC(C)=O)CCN(C(=O)C(c2cccs2)NC(=O)C(C)(F)c2ccon2)C1 77234,N1(C(C2(CN(C)C)CC2)=O)C2CCC1CC(NC(=O)CCC(=O)OC(C)(C)C)C2 77235,C1(OC)CC(NC(=O)C2=CSCS2)C12CCN(C(=O)C(C)(C)C(F)F)CC2 77236,c1(CC(=O)N(CCCNC(c2nc(C)sc2C)=O)C(C)C)cc(F)ccc1Cl 77237,C(=O)(C(C)(O)C(C)C)NCCSCC(=O)NC(c1nn[nH]n1)CC 77238,c1(OCC)ccccc1C(C(=O)NC1CCC1)N(C)CCNC(C1CCCS1)=O 77239,O=C(CCCCCCNC(c1cc2cc[nH]c2cn1)=O)NCc1cnn[nH]1 77240,C1(N(C(C2C(C)OC(=O)N2)=O)C)CCCN(C(=O)CC2CCCCC2(C)C)CC1 77241,C1(OC)CCCN(C(C2CC(O)CN2C(c2cc(C)ns2)=O)=O)CC1 77242,c1(SC)nc(O)nc(C)c1C(=O)N(CC(CO)(CO)NC(=O)C(C)C#N)C 77243,C1(C(N(CCNC(C(C(C)c2ccccc2)O)=O)C2CC2)=O)CC2C=CC1CC2 77244,Cc1c(CCNC(C2(F)CCN(C(C3CC(CO)(CO)C3)=O)C2)=O)cnn1C 77245,n1(CC)cnc2nc(=NCC3CCCCCC3)[nH]c(NCC3CCCC3(F)F)c12 77246,N1(C(C2CCC(C3CC3)O2)=O)CCOC(c2n[nH]c(-c3ccccc3)n2)C1 77247,C1(NC(c2ccc(C(C)C)cn2)=O)CCC(C)N(C(C2CCOC2C)=O)C1 77248,C1(C(=O)NCCn2ncc(C)c2)CCCN(C(c2scnc2C(C)C)=O)C1 77249,N1(C(C2(NC(C3CC(CC)C3)=O)CC2)=O)CC2CCCN2CC1CN(C)C 77250,C1(C(N2CCC(CF)(NC(c3cnco3)=O)C2)=O)(CC)CCNC1=O 77251,c1(-n2cc(CCc3nc(C)sc3)nn2)cccc(C(=O)NCCCNC(N)=O)c1 77252,c1(NC(C)CCC(=O)OC(C(C)NS(CC)(=O)=O)=O)cccc([N+](=O)[O-])c1 77253,c1(OC(C2C(c3onc(C)n3)C2)=O)cc(Cl)cc(Cl)c1 77254,N1(C(COCCCCC)=O)CCN(C(C2CNC(=O)N2)=O)C(C2CCC2)C1 77255,c1(C(=O)NC2(CCNC(=O)CC3CCC(=O)N3)CCC2)cc(C2CC2)ccc1F 77256,CCCC(C(O)C(=O)N1CCC(OC(=O)CC(C)(C)CC)CC1)NC(=O)C(C)C 77257,C#CCC(C(=O)NOCC1CC1)NC(C1CC12CCC2)=O 77258,c1(CNC2C(C(=O)NCCC#N)CCCC2)cc(O)c(O)c(O)c1 77259,C1(NC(c2cnc(CCCC)s2)=O)C2CCN(C(=O)CCN3CCCC3)CCC12 77260,C12(C(N(CCC(=O)OC)C)=O)CCC(CC1)N(C(C1C=CCS1)=O)C2 77261,c1(C(=O)NCC2C=CCN2C(=O)CC2CC2)c[nH]c2ccc([N+](=O)[O-])cc12 77262,N1(CC(=O)O)CCCC2(CCCN2Cc2nc3sccn3c2[N+](=O)[O-])C1 77263,C1(NC(CCCCOC)=O)CC2CCC1N2C(=O)C(C)Cc1cccc(Cl)c1 77264,C#CC1(C(=O)NCC(CC)C(C)C)CN(C(=O)C(F)CC2CCOC2)C1 77265,C(N=c1cccc(S(=O)(=O)NC2CCC=CCC2)[nH]1)C1CC(C)(C)OC1 77266,C=CC1(C(=O)NC(c2nccs2)CC)CCN(C(=O)CC=CCC)C1 77267,c1(CC(=O)NCC2CCN2C(c2cc(C(F)F)no2)=O)ccccc1Br 77268,c1(C(=O)OC)cc(S(N)(=O)=O)c(F)cc1NC(=O)NCC(c1ccc(C)cc1)O 77269,C(=O)(C1=CS(=O)(=O)CCC1)N1CC(NC(c2c(O)cccc2F)=O)(CO)C1 77270,c1(CNCC(C)N(CC)CC)c[nH]c(C)c(Br)c1=O 77271,C1(C(N2C(C(N(C(CC3CC3)CO)C)=O)CCCC2)=O)CCCC12CCC2 77272,c1(C(=O)Nc2c(COC)n(C(CC)CC)nc2)ccc(F)cc1F.C1(CO)CC(C)C1 77273,N1(C(C2C(NC(c3ncn(C)c(=O)c3)=O)CCO2)=O)CCCC(N=[N+]=[N-])CC1 77274,CC1CN(C(C2C3CCC(C3)C2NC(=O)Cc2cccn2C)=O)C(C)(C)C1 77275,C1(C(N(C(C)C)CCNC(c2ccoc2Cl)=O)=O)CCn2c(O)nnc2C1 77276,C1(NC(C2(N(C)C)CC2)=O)C=CC(CC(=O)NCC2CC(F)C2)C1 77277,C1(CNC(c2n(CC)ncc2)=O)CCCCN1C(C1OCCOC1C(F)(F)F)=O 77278,c1(CN(C)C(C2CC(C)(NC(=O)OC(C)(C)C)C2)=O)ccc(OC)nc1 77279,C(=O)(C(C)N=c1cncc[nH]1)N1C(C(=O)Nc2cccc(OC)c2Br)CC(F)C1 77280,CC(C)(C)C(CNC(=O)Cn1cc(C#N)cn1)NC(C1COCCN1C1CCC1)=O 77281,Cc1cc(C(N2CC(CCNC(C3CCOC3(C)C)=O)C(C)C2)=O)ccc1F 77282,CN1CC(C(N2CC(F)(CNC(c3csc(C(N)=O)n3)=O)C2)=O)CC1=O 77283,C1(CC(N2CCC(CCOC(C)=O)CC2)C(=O)NCC)Cc2ccccc2O1 77284,N(C(=NCc1nc(C(C)O)n[nH]1)N1CCC(C)C1)C(COC)C 77285,C1(CNC(COCCC=C)=O)CCC2CN(C(=O)CC3CCSC3)CC12 77286,c1(C(=O)NCCCN(C(CC2(OC)CC2)=O)CCO)cc2cc(Cl)ccc2s1 77287,C1(C(N2CCC(CN(C(=O)C(CC3CC3)NC=O)C3CC3)C2)=O)CC(F)(F)C1 77288,Cc1ccc(C(=O)C(=O)NCC2(COC)CN(C(C)C(c3ncc[nH]3)=O)C2)cc1 77289,C(N=c1[nH]c(=NC(C)C)c2ncccc2[nH]1)C1CCOC1c1c(C)ccc(F)c1 77290,c1(C(N(CC(=O)N(C)Cc2c(CC)n[nH]c2)CC)=O)ncncc1Cl 77291,C1(NC(C2(CF)CCN(C(c3cc(OC)ns3)=O)C2)=O)CCCCC1(C)C 77292,Cc1cc2ccc(C(N3CC(NC(C4SCCCS4)=O)C4(CCC4)C3)=O)cn2c1 77293,N1(C(CCS(C)(=O)=O)=O)CC(C)(CNC(=O)Cc2csc(C3CC3)n2)CC1(C)C 77294,N1(C(C2COCCO2)=O)CC2CC(C(N3CCC(c4cnn[nH]4)C3)=O)(C2)C1 77295,C(=O)(C#CC1(C)CC1)NC(CC)CNC(=O)CCC1CC1(Cl)Cl 77296,CCCC(O)CC(=O)NCC(CC)NC(C1CC2CCC(C1)S2)=O 77297,C12(C(=O)NCc3c(CC)noc3)CCN(C(=O)Cc3ccccc3)CC1C2 77298,CC1CN(c2cccc(C=O)c2CCN)CC(C)CN1C(=O)CC1CC1C(F)(F)F 77299,c1(C(=O)NC23CC(CNC(C#CC(=O)N(C)C(N)=O)=O)(C2)C3)nnc2ccccn12 77300,Cn1nc2c(c1C(N1CC(NC(c3ocnc3C(F)(F)F)=O)C(O)C1)=O)CCC2 77301,C1(N(C(Cn2c(C)ncc2)=O)C)CN(C(C2CC=CCC2)=O)CC1O 77302,c1(CC)cc(Cl)ccc1C(=O)NC1CCC1CNC(c1ccccc1C)=O 77303,C1(C(N(CC#CC)C)=O)(CNC(=O)Cc2ccn(C)c2)CC12CCC2 77304,C1(NC(C(c2cnn(C)c2)OC)=O)CCC(N(C)C(C2CC(C)(F)C2)=O)CC1 77305,c1(NC(C=Cc2nnc(C(C)C)o2)=O)cc2c(I)cnn2cn1 77306,C(=O)(C(F)(F)CC(C)C)NCC(CN(C(c1cnc2ccnn2c1)=O)CC)(C)C 77307,O=C(CCC(F)(F)F)NCC1COCCN1C(=O)C(O)CN1CCCCC1 77308,N1(C(c2cccc(C)n2)=O)CCC(C)C(N(C)C(C2CCCNS2(=O)=O)=O)C1 77309,N#CC1(C(N2CC3CC3C2C(N2CCC(C(F)(F)F)C2)=O)=O)CC12CCC2 77310,c1(C(=O)OCC)cc(C(=O)NC(CNC(c2nccn2C)=O)CO)ns1 77311,c1(NC(C)=O)ccc(F)c(C(N2CCC(N(C(=O)CC3CC3(C)C)C)C2)=O)c1 77312,CC1=C(CNC(=O)CC2(NC(C3CC3(C)C(F)F)=O)CCC2)CCC1 77313,c1(C(=O)NC(C(=O)NCc2onc(CC)n2)C2CCOC2)cc(C)ccc1O 77314,c1(C(=O)OC)cc(COC(c2cn(Cc3csc(Br)n3)nn2)=O)c(C)s1 77315,C=CC(CC)CC(=O)N1CCOCC1CN(C)C(c1cn(C(F)F)cn1)=O 77316,CC1(C(N2CC(OCC(=O)NC34CC=CC(C3)OC4)C2)=O)CCCCCC1 77317,C1(NC(c2cn(CC(CC)O)nn2)=O)CN(C(C2CC23CC3)=O)CC12CC2 77318,c1(C(=O)NC2(C)CN(C(c3nccc(CC)c3)=O)C2)cccc(F)c1C 77319,CC(C)C(O)CCNC(=O)C(CCF)NC(=O)COC1CCC1 77320,c1(C(N(CCCNC(CCSC)=O)C(C)C)=O)c(C)cc(C)nc1N1CCOCC1 77321,C1(C(N(C)CC2CCN(C(=O)CS(N)(=O)=O)C2)=O)CCC2(CCC2)O1 77322,CC1CC(NC(c2ccco2)=O)CN1C(C1CCCC(O)C1)=O 77323,c1(OC)ccc(CC(=O)NC2CN(C(c3c(N)cccc3Cl)=O)CC2C)cc1F 77324,C1(N(C(c2cc(CC)no2)=O)C)CCN(C(=O)CC2(CC(=O)OC)CC2)CC1 77325,c1(C(=O)NC2CC(CCC(=O)NC3C(CCC)CC3)C2)csc(CO)n1 77326,Cc1cc(C)c(C)c(C(=O)NCC2CCN(C(c3cn[nH]c3)=O)C23CC3)c1C.C1=CC1 77327,c1(OCC(=O)NCCCC(C)NC(CC2(C=C)CCC2)=O)cccc(C)c1C 77328,C1(C(=O)NC(CNC(COCC#C)=O)C)CC12C(O)C(O)Cc1ccccc12 77329,C(=O)(CN=c1cc[nH]cc1)N1CC(CNC(c2c(C)scc2)=O)C(C)(C)C1 77330,c1(OC)cc(Br)c(C(N2CC(NC(C3CCCCO3)=O)CC(F)C2)=O)cc1O 77331,N1(C(C(C)Cc2ccc(F)cc2)=O)CC2CC(NC(=O)CCC3CC3)CC1C2 77332,N1(C(C(C)=O)=O)Cc2ccccc2C1CNC(c1cnc(C(C)C)o1)=O 77333,c1(CCC)cc(C(=O)NC2CCN(C(=O)C(CC)CC)C2C2CC2)c(C)o1 77334,C1(CC(=O)NCCC2(OC)CN(C(=O)CCNC(C)=O)C2)CCCC(C#N)C1 77335,C(=O)(C1=CCC2CCC1N2C(C1(C)CSC1)=O)N(C)CC1CCCCO1 77336,CC(=O)CCC(=O)NCC1CCCCN1C(c1cnc(C2CCOCC2)s1)=O 77337,C(CC(C(=O)NC(C)C(C)N1CCC1)NC(=O)CSC(F)F)SC 77338,C1(C)(CNC(c2cnn(CC)c2C)=O)CCCN(C(c2c(C#N)cnn2C)=O)C1 77339,Cn1nnc(CNC(=O)C(C)(C)C#N)c1C(N1CC(CO)C1(C)C)=O 77340,N1(C(CCc2n(C)cnn2)=O)CCOC2(CCN(C(=O)C=CCO)C2)C1 77341,C1(CNC(c2[nH]cc(C(=O)OC)c2)=O)CCN(C(=O)C(C)SC)CC1C 77342,c1(CNC(=O)C(O)c2ccsc2)csc(CC2CNC2)n1 77343,N1(CCC)CCC(C(=O)NC2CCCC(CNC(=O)C(C)(CC)OC)C2)CC1 77344,CCC(C(=O)NCc1ccco1)N(C(=O)CC1CCCN1C)C 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77413,c1(C(=O)NC(CCNC(C2(C(=O)OCC)CC2C)=O)C)cc(C)nc(O)c1 77414,N1(C(C(C)(C)C2CCCO2)=O)CCC(C)(CNC(=O)C=C2CCCC2)C1 77415,c1(C(=O)NC2CN(C(CC(C)F)=O)CC2(C)C)c2ccccc2nn1C 77416,c1(C(=O)NCCN(C(=O)CC2CCC(=O)N2)CCC)c[nH]c(=N)o1 77417,N1(C(C(C(C)SC)O)=O)CCC(C)(CNC(=O)CN(C2CCCCC2)C)CC1 77418,c1(CC(=O)NC2C3CN(C(=O)CC4CCCOC4)CC23)c[nH]c2cnccc12 77419,Cc1cc(C)n(CCNC(C2C=CCN(C(=O)CC3CC(F)(F)C3)C2)=O)n1 77420,Cn1nc([N+](=O)[O-])cc1C(=O)NCC1CN(C(C2CCS(=O)(=O)CC2)=O)C2CC12 77421,C1(OC)C(NC(=O)C(C)(C)Cc2ccc(C)c(Cl)c2)CC12CCC2 77422,S(=O)(=O)(c1ccc(F)c(C(=O)NC2CCC(C(N)=O)C2)c1)NC(N)=O 77423,c1(CCC)cccc(C(=O)NC2(CNC(=O)C(c3ccc(Cl)s3)C)CC2)c1 77424,C(=O)(CC(CC(C)C)NC(=O)C(F)CCC)NCC(CCC)O 77425,Cc1cc(C)n(CC(=O)NCC2CC2C(=O)NCc2cc(C3CC3)no2)n1 77426,c1(NC(CC2CCN(C(C(CC)C)=O)CC2)=O)cc(OC)c(OC)cc1F 77427,Cc1cnc(C(=O)NCC(CO)NC(c2nocc2-c2ccccc2)=O)c(F)c1 77428,N1(Cc2cn(CCC)nc2)CC2CN(C(C)C(=O)NC3CC3)CCC12 77429,N1(C(C(C)OCC#C)=O)CCCC(C2CC2NC(c2cc(OC)cc(F)c2)=O)C1 77430,c1(CNCC(=O)NCCCOCCCC)conc1SCC 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77448,N(C(=NCCCCC)N1CCc2c(cc(F)c(F)c2F)C1)C(C#C)(C)C.C1C(=O)N1 77449,CCCCC(C(=O)NC)NC(=O)C=CC(C)(C)NC(c1cn(C)cc1C)=O 77450,N1(C(COCC)=O)CCCC12CCN(C(=O)CC(F)(F)Br)CC2 77451,n1(CC)nc(C)c(C(=O)NC2CC(n3cc(-c4cccnc4)nn3)C2)c1C 77452,c1(SC)cn(C)nc1C(N1CC(NC(C2(C(N3CCCC3)=O)CC2)=O)C(F)C1)=O 77453,CCC(C)(C)CC(=O)NCC1CN(C(c2ccc(F)c(CC=C(C)C)c2)=O)CC1O 77454,c1(CC(=O)NCC=CCNC(=O)CCC2CCCO2)ccc(Cl)nc1F 77455,c1(C(=O)NCC(C)N(C(=O)C(C)CC(F)F)CC)ccnc2[nH]c(C)nc12 77456,Cc1cc(C(=O)NCC(CNC(=O)CC#N)CO)n(C(C)(C)C)n1 77457,n1(CCC)ccnc1C1CC1.C1(C(=O)CCC(=O)N)CSCN1C(=O)CN(C(C)C)C 77458,c1(CC(=O)NCCC2(CNC(CN(C(C)=O)C)=O)CC2)csc(C)n1 77459,c1(OCCNCCOCCOC(C(=O)OC)C)ccccc1 77460,n1(CCC)ccnc1C(F)(F)C(=O)N(C)CCN(C(=O)CC(C)C1CC1)C 77461,CCC(C)CC(C)NC(C(C)(C)CC1CC1)c1nnnn1C 77462,C1(NC(C(=O)OC(C)C)=O)CCN(C2CCCCC2NC(=O)OC(C)(C)C)CC1 77463,CCCCC(O)C(=O)NCCC1CCCN(C(c2ccc(C)c(OC)c2)=O)CC1 77464,N1(C(C2C(=C)C2)=O)C(C(=O)NC2(CC3CCC3)CC2)CCC12CC2 77465,CCS(=O)(=O)CC(=O)N1CC2CC2C1C(=O)NC(c1nn[nH]n1)C1CC1 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77519,C1(C(=O)NC(C(C)C)(C)CNC(=O)Cc2cnnn2C)OCCN(C)C1=O 77520,C1(CNC(c2csc(C)c2C)=O)CN(C(C2CCOC2)=O)CC(C)(C)C1 77521,C1(NC(C2(C=C)CCC2)=O)CC(O)CN(C(c2ccc(OC)c(C)c2)=O)C1 77522,c1(-c2ncc(C(N(C)CC3CCN(C(COCC=C)=O)C3)=O)s2)ccc(C)cc1 77523,c1(C(=O)NC(CC2CN(C(c3cnc(C(C)=O)s3)=O)C2)C)c(Cl)c(C)nn1C 77524,c1(C(N(C2CCN(C(CCCOC(C)C)=O)C2)C)=O)nccc(Br)c1O 77525,c1(OC)cc(C(N2CCCC(O)(CCNC(=O)C(C)CO)C2)=O)c(N)c(C)c1 77526,c1(NC(c2c(NC(Cc3n(C)cnn3)=O)c[nH]n2)=O)cccnc1O 77527,N1(C(c2n[nH]c(C)c2C)=O)CCC(C)(CNC(C2CC2C(=O)NCCO)=O)CC1 77528,N1(C(Cn2ncc(CC)c2)=O)CC=C(CNC(C2CCN(C(C)=O)CC2)=O)CC1 77529,C1(NC(c2nn(CC)c(=O)cc2)=O)C2CCCC1CC(NC(C1CCCC1)=O)C2 77530,c1(COC)cc(C(N2CC=CC(NC(C3(c4cccnc4)CC3)=O)C2)=O)n(C)n1 77531,C1(CCCNC(=O)C(c2cnn(C)c2)C)(CNC(CC=C)=O)CCCC1 77532,Cc1[nH]c2ccccc2c1CNC(=O)C(=O)N(C(CN)C1CC1)C 77533,c1(CNC(c2cnco2)=O)cccc2c1CN(C(C1CC(O)C(F)C1)=O)C2 77534,c1(C(=O)NC(C2COC(C)(C)C2)C)ccc(Cl)cc1N=[N+]=[N-] 77535,C1(C#N)(CNC(C(=O)N(CC(C)(C)Cc2ccccc2)C2CC2)=O)CCCO1 77536,C=CCCCCC(=O)NC(C)CCCCNC(C1CCCN1c1cnccn1)=O 77537,NC1CC2(CC(NC(=O)C(=O)NCCCOc3ccccc3)C2)C1 77538,C1(C)(c2cn(C(C3C=C(C)CCC3)C)nn2)CN(CC2C3CC4C(C3)C24)C(C)(C)C1 77539,C(=O)(C1=C(Cl)CCC1)N1CCC(CNC(=O)CCC(=O)c2ccc(O)cc2)C1 77540,Cc1cc(C(N2CC(CNC(C3COC3)=O)CC2C)=O)c2nc(C)n(C)c2n1 77541,CCC(C)(O)C(=O)N1CCCC1CNC(c1cc(SC)oc1C)=O 77542,c1(COC)ccsc1C(=O)NC(C)C(C)NC(=O)C(C)Oc1ccccn1 77543,c1(C(N(CC(CC)NC(=O)C#CC2(C)CC2)C)=O)c(SC)cccc1F 77544,c1(NC(C2C(C)(C(=O)OCC)C2)=O)ccc(Br)cc1Br 77545,C(=O)(CC(C)CC(C)(C)C)NC1CCC(NC(c2n(C=C)ncc2)=O)CC1.C1CO1 77546,c1(C(N2CC(OC3CCN(C(CC(C(C)C)O)=O)CC3)C2)=O)cc(Cl)c(F)cc1F 77547,CC1CC(C)(C)CN1C(=O)CC1CCN(C(=O)C(O)CN2CCCC2)CC1 77548,c1(CC(N2CC(O)(C(C)NC(CC(C=C)C)=O)C2)=O)cn2cccc(C)c2n1 77549,Cc1noc(C(N2CC(CC(C)NC(=O)COc3cnn(C)c3)C2)=O)c1C 77550,C(=O)(CCC(F)(F)C(F)(F)F)NCC1CN(C(c2c(C)cc(O)nn2)=O)C1 77551,N1(C(c2cc(SC)oc2)=O)CC(C2CCN(C(C3CCOC(C)(C)C3)=O)CC2)C1 77552,C(CC(=O)NC(C)COCCOC)N(CC(=O)NC1CC1)CCC 77553,C1(N)CC1C1CN(C(C2CCCCCC2)=O)C1.CC(CO)(C1CCCC1)N 77554,CC(CC(=O)NCCCC1CCCN1C(=O)CCN1CCCC1)P(C)(C)=O 77555,C(CC(C)(C)CC(=O)NCC(c1cc(Br)cc(Br)c1)(C)C)OC 77556,c1(C(=O)NC2CCC(C(N3C(C#C)CC3)=O)C2)ccc(F)cc1F 77557,N1(C(c2ncc(OC(C)C)nc2)=O)CCC2(NC(c3c[nH]c(=N)o3)=O)CC2C1 77558,C(C(N=[N+]=[N-])C(=O)NCc1nc(C(=O)NOCC(C)C)co1)OC 77559,C#CCC(CC(=O)N(C)CC1(CC=C)CCC1)NC(=O)CC(C)C(F)F 77560,C#CC1(C(=O)NC2CN(C(C3CC4(CCO3)CC4)=O)CC2OC)CCOCC1 77561,c1(N(CCOCCN(C(C(C)n2cccn2)=O)C)C)cc(N)c(O)cc1F 77562,C1(NC(C2CCCC2)=O)CC2CCC1CN2C(c1cc(O)ncc1F)=O 77563,N1(C(CCN(C)CCO)=O)CCC(CF)(NC(=O)CCSc2ccccn2)C1 77564,C1(C(=O)NC2CC(=O)N(C(C)C)C2)CCC2(CCC2)C1.C=C1CC2(C1)C(=O)N(C)C2 77565,Cn1nc(CC(=O)NC2CC(F)(CNC(c3cc[nH]n3)=O)C2)cc1C(F)(F)F 77566,C(=O)(C(C)(C)C(C)(F)F)N1CCC(F)(CNC(C2(C)CCCCCC2)=O)C1 77567,C1(C)(NC(=O)CO)CCCC1NC(=O)C(N1CCC(OC2CC2)C1)=O 77568,C1(CNC(=O)C(C2CCC2)C2CCC2)CCN(C(C2CSCCS2)=O)C12CC2 77569,c1(C(=O)OCC)nnc(C(C)NC(=O)N(c2nc(C)no2)C2CC2)s1 77570,C1(C(N2CCN(C(CSCCCC)=O)CC2CF)=O)COC2CCCCC12 77571,c1(C(N(CCOCC#C)C)=O)coc(CNC(C2CCC(=O)C2)=O)n1 77572,c1(NCCC(=O)NC(C2(C)CNC2)CC)ncnc2sccc12 77573,c1(C(N2CCC(NC(C3C(OCC)C3)=O)C(CO)C2)=O)cc2cc(Cl)cnc2o1 77574,CN1CCC2(CCN(C(C3CC(CC(=O)O)C3(C)C)=O)C2)C1=O 77575,C1(NC(C(C)c2ccco2)=O)CC(CNC(C2(C3CC3)CC2)=O)C1(C)C 77576,N1(C(=O)NCCOCc2ccccc2)CCC(Nc2cc(Br)co2)CC1 77577,c1(C(N(C2CCN(C(=O)CC(c3ccc(C)s3)C)C2)CC)=O)nc(C(C)C)oc1C 77578,Cc1ccnc(C)c1C(N1CCC(O)C(NC(c2csc(C(N)=O)n2)=O)C1)=O 77579,C(=O)(CC(CC)CCCC)NC(CN(C(C1C(=C)C1c1cccnc1)=O)C)CC 77580,C(=O)(C(C)(C)C(=O)N(CC(O)CNC(C1CCNC1=O)=O)C)N(C)C 77581,N1(C(c2c(NC)nccc2)=O)CC(C(N2CCC(CO)CC2)=O)CC12CCC2 77582,C(C)(CN=c1[nH]c(N(C)Cc2cnn(-c3cccc(Cl)c3C)c2)nc(=N)[nH]1)SC 77583,c1(CC)nc(C)cc(=NC(=O)C2CC(O)CCN2Cc2ncccc2Br)[nH]1 77584,C1(CCNC(C(n2ccc(C)n2)(C)C)=O)CCCCN1C(=O)Cc1cnccn1 77585,Cc1cc(F)cnc1-c1cn(CCC(=O)N(CC)Cc2nc(C(F)(F)F)cs2)nn1 77586,C1(c2n(C(C)C)nnn2)(NCc2cnc(C(C)C)o2)CCC(F)(F)CC1 77587,c1(NS(C)(=O)=O)cccc(CNC(=O)CC2CC(=O)N2)c1.N12CCCCC1C2 77588,C1(F)(CNC(C(CC)F)=O)CCN(C(=O)C(C)(C)N2CCOCC2)C1 77589,N1(C(C(C)ON)=O)CCCCC(SC(C)(C)C)C1 77590,c1(N2CC(=O)N(c3ccc(Br)cc3)CC2)ncccc1S(=O)(=O)NCC(F)CO 77591,C(CCCC(C)(C)NC(=O)CC1CCN(C)C1=O)NC(CC1CN(C(C)=O)C1)=O 77592,c1(C(N)=O)ccc(NC(C2CC(F)CN(Cc3ccc(Br)s3)C2)=O)c([N+](=O)[O-])c1 77593,c1(C(=O)NCCNC(C(C)C2CCCC2)=O)c[nH]c(=NC2CCOCC2)cn1 77594,CC1(C)CNCCC1N1CCN(Cc2cc(Cl)ncc2Cl)CC1 77595,c1(C(N2CC(CNC(c3nocc3C3CC3)=O)OCC2)=O)cc(Cl)c(O)c(Cl)c1 77596,C1(O)(CNC(CCCC#C)=O)CCCN(C(c2ccc(C(F)F)cc2F)=O)CC1 77597,c1(C(=O)NCC2OCCN(C(CN(C3CC3)CC)=O)C2)cc(C)cc2c1CCC2 77598,CC(CC(=O)N1CC(O)(C2CCCN2C(c2cnc3n2CCC3)=O)C1)C(F)F 77599,c1(C(N2C3C(NC(=O)C=CC4CCC4)CC(C3)C2)=O)ccc2ccncc2n1 77600,c1(N2CCN(C(=O)Nc3cc(C)ncc3Cl)CC2)cccc2nsnc12 77601,C=Cc1cncc(NC(C2(NC(=O)CN(C)C)CCN(C)C2)=O)c1 77602,N1(C(C=CC=CCCCCC)=O)CC2C(CNC(C3CCC(=O)N3C)=O)C2C1 77603,N1(C(C2N(CC)CC2)=O)CCOC(CCCNC(C2CC(n3cnnc3)C2)=O)C1 77604,N1(C(CCc2c(C)noc2Cl)=O)CCC2(CCN(C(=O)CCc3cncs3)C2)C1 77605,N1(C(C(C)S(N)(=O)=O)=O)CC2CCC(C1)C2NC(C1CCC2(CCCC2)C1)=O 77606,c1(NCc2ccn(CC)n2)ccc2c(c1)OC(F)(F)O2 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77678,C(=O)(C1=NNC(=O)CC1)N(C1CCN(C(C2(C3CC3)CC2)=O)C1)CC 77679,C1(NC(c2ccc(F)c(CO)c2)=O)CCS(=O)(=O)C12CN(C(C1C=CCC1)=O)C2 77680,N1(C(C2(NC(c3ccc(OC)cn3)=O)CC2)=O)CCC(O)C(C)(CO)C1 77681,CC1=CCC(C(N2CCN(c3ccccc3CNC(=O)C(F)F)CC2)=O)CC1 77682,c1(OC)ccc(CC(=O)NC(C)C(C)NC(c2csnn2)=O)c(Cl)c1 77683,N1(C(C(C)n2cccc2)=O)CCc2sc(CNC(=O)CCS(C)=O)nc2C1 77684,C(C1=CCCOC1)N(C)C(C1CCC(NC(c2cnc(C3CC3)o2)=O)CC1)=O 77685,N1(C(C2N(CC)CCC2)=O)CCC2CCCC12C(=O)NC(C)C(C)SC 77686,C(CCNC(=O)Cn1nnnc1C(C)C)(C(C)C)NC(CNS(CC)(=O)=O)=O 77687,C(C)(C)(CC(F)C(=O)N1CCC(OCCOC)C1)NC(c1c(CC)occ1)=O 77688,N1(C(C2(SC)CC2)=O)CC2CCC1CN2C(C1(CO)CC1)=O 77689,c1(C(N2CC(CNC(C3(CC#C)CCC3)=O)C2)=O)nccc(C)c1Br 77690,c1(OC(C)C(=O)N(CCCCNC(=O)CC2COC(=O)C2)C)cc(Cl)cc(Cl)c1 77691,n1(CC(=O)N(CCC)CCN2CCC2C)cc(-c2ccnn2CC)nn1 77692,CC(C)(F)CCC(=O)NCC1CCCC1C(N1CCC(CC(N)=O)CC1)=O 77693,c1(C(=O)NCC2C(NC(C=NOC)=O)CCC2)cnc2c(c1)CCCC2 77694,c1(C(=O)NC2C(C)CN(C(=O)CC3SC(=N)NC3=O)C2)nc2ccccc2[nH]1 77695,N1(C(CN(C)C(C2CC2)=O)=O)CCC2(CC1)CN(C(c1ccnnc1N(C)C)=O)C2 77696,c1(C(=O)NCC(C)(C(C)C)NC(c2ccc(C)s2)=O)ccc2ncnn2c1 77697,C1(NC(C(c2cccnc2)OC)=O)CC=CCC1C(=O)NCCF 77698,c1(C(C(=O)NCC(C2CC2)NC(C(C)OCCN(C)C)=O)=O)cccn1C 77699,C1(CC(N2CCC(COC)(NC(=O)C=C3CCSCC3)C2)=O)CCCNC(=O)C1 77700,n1(CCC)cc(C(=O)N(CCC(=O)NC2(C(O)COC)CC2)CC)cn1 77701,C#CCC(C)(C)C(=O)NCc1ncccc1C(=O)Nc1ccc(C(C)C)cc1 77702,O=C(C1=Cc2ccc(Cl)cc2OC1)NCC(C1CC1)NC(c1cscn1)=O 77703,n1(CC(N2CCC(CCCC)C2)=O)ccc2ccc(F)cc12 77704,c1(CNc2ccc(CO)cn2)cc2c(o1)=CCC(c1sccc1C1OCCO1)=CC=2 77705,C(=O)(CCC(C)CC)N1CC(CCNC(C2CC(=C)C2)=O)OCC1 77706,N1(C(CN2CC(C)(OC)C2)=O)CCN(C(C2CCCC2C2CC2)=O)CC1C 77707,c1(C(N(CC(O)CNC(=O)C(C)(C)O)C)=O)cnn(C)c1C(F)(F)F 77708,C(Cn1cccn1)(CCNC(C1CC1c1cnn(C)c1)=O)NC(C)=O 77709,CCC(CCCC(=O)N1CC2(CSC2)C1)NC(=O)C(c1ccnn1C)O 77710,N1(C(C=CCN(CC#C)C)=O)CCC2CN(C(c3c(Cl)cccc3Cl)=O)CCC2C1 77711,CC(C)(CC(=O)NC1(C2CCN(C(=O)C(F)CC3CCOC3)C2)CC1)C(F)F 77712,C1(O)(CN(C(c2ccc(-n3cc(C=CC)nn3)cc2)=O)C)CCC(F)(F)CC1 77713,C1(CC)CCCC1(C)C(=O)NCCCNC(c1ccccc1OCC(N)=O)=O 77714,c1(NCCSCC(C2CCCC2)C)nc(=N)[nH]c(=NCCN2CCCC(C)C2)[nH]1 77715,C1(C(=O)NC(C(C)C)c2nn[nH]n2)CC12CCN(C(c1ccc(Br)cc1F)=O)C2 77716,C(C(C(=O)N1CC(OC(C)=O)C1)NC(C1C=C(C)CS1)=O)OC 77717,N#Cc1cncc(C(N2CC(NC(=O)Cc3cncnc3O)C(F)(F)C2)=O)c1 77718,Cc1ncnc(C)c1C(=O)NCC1(C(N)=O)CN(C(=O)Cc2cccc(F)c2)C1 77719,C1(C(=O)NCC2(C(=O)OCC)CCC2)CC2(CCCN1C(=O)CCCCNC)CC2 77720,c1(CCC(N2CCCC(C(C)NC(c3c(C)nns3)=O)C2)=O)cc(Cl)cc(Cl)c1 77721,c1(C(=O)NCC(C2CC2)NC(=O)CN2CCCCCC2)cc2c(Cl)cncc2o1 77722,C(=O)(C1=CC2C=CC1C2)N1CC2C(CC(=O)N(CCCO)C)(CC2)C1 77723,N1(CC(=O)NC2CCC(NC(c3c(C)nc[nH]3)=O)C2)CCN(S(C)(=O)=O)CC1 77724,Cc1cccc2c(C(=O)NC3CC4CCC(C3)N4C(=O)Cc3nc[nH]n3)csc12 77725,c1(OC)cc(=O)n(C)cc1C(=O)NCCN(C(=O)C1=CCS(=O)(=O)C1)CC1CC1 77726,N1(C(CCc2cc(C)on2)=O)CCC(NC(=O)Cc2coc(C)c2)C(O)C1 77727,C1(C(=O)NC(C(C)NC(c2c(C)n(C)nn2)=O)(C)C)CC2C=CCC(C1)C2 77728,N1(C(C=C(CCC)C)=O)CC=CC(C(N2CCC(OCC)C2)=O)C1 77729,c1(C(=O)NCCC2(NC(CC3CC(=C)C3)=O)CC2)sc2ccccc2c1Cl 77730,n1(CC#C)ccnc1C(C(=O)NC)N(CCC(N)=O)CCOC 77731,c1(CNCc2c(NC(CC(c3ccccc3F)C)=O)c[nH]n2)ccccc1CO 77732,c1(C(=O)NCC(CNC(=O)C=CBr)OC)c[nH]nc1-c1cnn(C)c1 77733,n1(CC(C)C)c(N2CC=CC2)nnc1C(c1cccs1)O 77734,c1(-n2ncc(C)c2)ccc(CNC(N2CCOC(C)(C3CC3)C2)=O)cc1F 77735,N#Cc1c[nH]c2ncnc(N3CC(F)CC3C(N3CCC(Br)C3)=O)c12 77736,N1(C(C2(COCC)CCC2)=O)CCSCC1C(N1CCCOCC1)=O 77737,CC(C)CC(C)CNC(=O)CC1CCCCN1C(C1CN(C(C)C)C1)=O 77738,C1(NC(C=C(C)C(F)F)=O)CN(C(=O)C(CCN(C)C)N(C)C)CCC1O 77739,CCC(=O)CCC(=O)NC(C)CCCC(=O)N1CC(CO)CC(C)C1 77740,C1(CNC(C2CC=CCO2)=O)CC(F)(F)CN1C(c1cc(F)cc(Cl)c1)=O 77741,c1(C(N2C(CNC(C(C)Cc3ccccc3)=O)CCC2)=O)nc[nH]c2ncnc1-2 77742,O=C(CC1=CCOCC1)NC1(CCNC(c2ccc(C(N)=O)cn2)=O)CCC1 77743,c1(C(CC)=O)ccc(NC2CCC(CCCNC(=O)OC(C)(C)C)C2)c([N+](=O)[O-])c1 77744,C1(CNC(C2(SC)CCC2)=O)CN(C(c2cc(C)c(C)o2)=O)CC1C 77745,Cc1noc(COC(=O)CCNC(=O)CNC(c2ccco2)=O)n1 77746,c1(C(N2C(CNC(C3C(CC)CCC3)=O)CC(O)C2)=O)cc(Cl)c(Cl)cc1O 77747,C1(C)(C(=O)NC(CCNC(C(=O)NCCOC)=O)C)CCNCC1 77748,Cc1ccc(C(N2CCOC(CCNC(C3(C(F)F)CCCO3)=O)C2)=O)c(N)c1 77749,c1(NCC2CCN(C)CC2)ccc2c(c1)CCN2C.N12CC3(CCC(O3)C1=O)C2 77750,c1(C(=O)NCC2(C(N)=O)CN(C(=O)CC#N)C2)ccc(O)cc1O 77751,N1(C(C)=O)CCC2(CC1)CC(NC(=O)C(C)CS(C)(=O)=O)C2 77752,c1(CC)noc(CCCC(=O)NCC(C)N(C)C(c2nccn2C)=O)n1 77753,C(=O)(C1=Cc2ccccc2C1)N1CCC(CNC(C(CO)N(C)C)=O)C1 77754,C1(CC)CN(C(=O)C(N2CCCC2)C2CC2)CCC1NC(c1ccncc1)=O 77755,N1(C(CCC(=O)NCCCOC)=O)CCC(NC(=O)C(C)(C)CO)C(C)(C)C1 77756,C1(C(N)=O)CN(C(C2CCCN(C(=O)CC3(O)CCCC3)C2)=O)CCO1 77757,C(CC1c2ccccc2CCN1C(c1c[nH]nc1C)=O)NC(C(F)=CC)=O 77758,O=C(C1CCc2snnc21)N1CCCCC(CNC(C2(Cl)CC2)=O)C1 77759,C(C)(C)(CCCNC(=O)C(F)OC(F)(F)F)NC(C1CCC(CC(=O)OC)O1)=O 77760,CC1CCCCC1(CNC(c1cc(CO)on1)=O)NC(=O)CCN1CCOCC1 77761,c1(C(=O)NC(CC)CN(C(=O)C#CC(C)C)C)ncc(OC)cc1F 77762,N1(C(CSCCCC)=O)C2CCC1C1CC1(NC(=O)Cc1ccsc1C)C2 77763,C#CCC(C)(C)C(=O)N(C1C2CN(C(c3ccc(CC)nc3)=O)CC12)C 77764,Cc1ccncc1C(=O)NC1(CCNC(c2occc2Cl)=O)CC1 77765,C1(CNC(=O)CC2COCCO2)CCCCCN1C(c1cn[nH]c1)=O 77766,C1(NC(c2ncc(OC)nc2)=O)CC(NC2CCS2(=O)=O)C12CCOCC2 77767,C(=O)(C(C)(C)CN(C)C)N(CCOC(C)=O)C.c12occc1CNC2=O 77768,C(=O)(CCC(C)NC(N)=O)NC(C1CCN(C(C2(C=C)CCC2)=O)C1)(C)C 77769,N1(C(c2cnc(S)[nH]2)=O)CCC2CN(C(c3cccc4sccc34)=O)CC2C1 77770,c1(C(=O)NCCCN(C(=O)CCC2CCCCO2)C)cccc2c1C(C#N)C2 77771,N1(C(=O)C(Cl)=CCl)CC(NC(C2(c3ccco3)CC2)=O)C(F)C1 77772,N1(C(c2cc(C)c(C)nc2)=O)CCCC(NC(=O)C(O)CCC(C)C)CCC1 77773,N1(C(C=CC=CC)=O)CCCC1CN(C(c1cc[nH]c1CCC)=O)C1CC1 77774,N1(C(Cc2c(C)cc(C)s2)=O)CC2CCN(C(=O)CCNS(C)(=O)=O)C2C1 77775,C1(COC)CN(C(=O)NCC2CCCN(c3cccnn3)C2)CCO1 77776,n1(CC)nc(C)cc1C(=O)NCC12CC1CN(C(c1n[nH]c(C)c1C)=O)C2 77777,C1(C(=O)NCC(C)(C2CC2)OC)C2CC3C(C2NC(c2ccc(=N)[nH]n2)=O)C13 77778,Cn1ncc2c(NCC3CC=CC3)nc(N3CCOC(C4CCOC4)C3)nc12 77779,C1(C(=O)NCCP(C)(C)=O)C2CN(C(=O)C(=O)NCC(F)F)CC12 77780,N1(C(CCCCC)=O)CCN(C(c2ccn(C(C)C)n2)=O)C(C)C1C 77781,C#Cc1ccc(C(N2CCC=CC2C(=O)NCC(O)CO)=O)cc1C 77782,c1(NC(CNC(=O)CNC(C2CCCC(O)C2)=O)=O)cc2ccccn2n1.C(=O)CC 77783,CCN=C(NCc1noc(-c2ccco2)n1)NC(c1cccs1)C 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78031,C(CC(CC)C(=O)NCCOCCNC(=O)C(C)NC(=O)NC)=CC 78032,N1(C(CCc2ccc(C(=O)OC)nc2)=O)CCCC(NC(=O)C(F)C(C)(C)O)C1C 78033,C(=O)(C(CC(C)C)C(N)=O)NCc1occ(C(N2CCCC(C#C)C2)=O)c1 78034,C1(C(=O)NCC2(CC)CCCC2)CC(F)CN1C(=O)N(C(F)(F)C(F)(F)F)CC 78035,C1(C(N(C)CC2CN(C(=O)CCNS(C)(=O)=O)C2)=O)CCC2CCCCN12 78036,Cc1ccc(C(N2CC=CC2(C)C(=O)NC(C)CF)=O)nc1C 78037,c1(CC(N2CC(CN(C(c3cc(C)n(C)n3)=O)C)C2)=O)ccc(F)c(Cl)c1 78038,C12(C(N)=O)CCCC1(C(=O)NC1CCCC1NC(c1nncs1)=O)C2 78039,C1(C(N)=O)COCCC12CN(C(=O)OC(c1ccnc(O)c1)=O)C2.C1CCOCC1 78040,N1(C(c2cc(CC)ncn2)=O)CCCC(O)(CCNC(c2ccc(Cl)nn2)=O)C1 78041,c1(C(=O)NC(CNC(C2N(CCC)C(=O)CC2)=O)CO)ccn2c1CCCC2 78042,N1(C(CC(C)n2ccnc2)=O)CCC(CO)(NC(C2CCCCS2)=O)CC1 78043,C(=O)(C1CCCc2sccc21)N1CC(CC(=O)NC)N(C(=O)C2CC2)CC1 78044,C1(OC)CCC(C(N2CC(F)CC2CC(=O)NC(c2nc(C)oc2C)C)=O)CC1 78045,c1(CNC(=O)C=CCF)cn(C2CCOC2)nn1 78046,C(CC(=O)N(CC(C)N(C(=O)C(C)n1ccnn1)C)C)OCC(C)C 78047,c1(OC)ccc(C(=O)CCC(=O)N(CCNC(=O)C(O)C(C)C)CC2CC2)cc1 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78083,C(=O)(C#CC1CCCOC1)N(CC(C)(C)CNC(c1ccc(CC2CC2)s1)=O)C 78084,c1(OC)ccc(NC2CN(c3nccc(OCCCO)n3)CCN2C)cc1O 78085,C(=O)(CC(C)CC(=O)N(C(CC(F)F)C(=O)NCC1=C(C)CCC1)C)OC 78086,N1(C(c2c(C)n3c(n2)scc3)=O)CCC2C1CCCN2C(=O)CC(C)F 78087,C12(C(=O)NC(CC(C)(C)OC)C)CCNC1CNC2 78088,CC1CC(=O)NCCN1C(c1c[nH]nc1-c1ccc(Cl)s1)=O 78089,N1(C(C23CC(CC(C)O2)C3)=O)CC2CCCC(C1)N2C(=O)C(N)=O 78090,c1(C(=O)NC(CCSC)C)cc(CNC(=O)CCc2nncs2)[nH]n1 78091,C1(N(C(C2C(C=C)C2)=O)C)CC2CCC(C1)N2C(c1cnnn1C=C)=O 78092,C1(C(=O)NCCC2CCCN(C(CCCCC#N)=O)C2)CC12CCC1(CC1)CC2 78093,S(=O)(=O)(CCC(=O)NC1CC(NC(c2ccc(Cl)c(Br)c2)=O)C1)NC 78094,C1(C(N(CCNC(C(F)=CCC)=O)C)=O)CC(CC)=NO1 78095,CCC(C)CC(C(=O)NCC1=CCCOC1)NC(C1CN(C(=O)NC)C1)=O 78096,C1(C(N2CC(CC)(OC)C2)=O)CCCN(C(c2cc(C)ncn2)=O)C1C 78097,c1(C(=O)NC(C(C)C)C(N2CCCC(C#N)C2)=O)ccc2nncn2c1 78098,C(=O)(CC(C)CC(C)(C)C)NCC(CC)(CC)NC(C1CC(O)CN1C)=O 78099,N1(C(C(CC)c2ccccc2)=O)CCC(N(C(=O)CCCc2ccsc2)C)CC1 78100,C12(NC(=O)C(C3CCOCC3)O)CCCC1N(C(=O)Cn1ccnn1)CCC2 78101,N1(C(CCc2ncc(C)[nH]2)=O)CCC2CN(C(=O)C#CC3(C)CCCO3)CC2C1 78102,c1(C(C(N2CCC(O)(CNC(CC(C=C)C)=O)C2)=O)(F)F)ccc(C)c(OC)c1 78103,c1(C(=O)OC)cc(NC(=O)NCC2CCCC2SC)c2c(c1)CCC2 78104,CC1CCC(NC(=O)C=C2CCCC2)CN1C(c1cc(Br)n(C)c1)=O 78105,c1(CC(CN(C(=O)NC(CC)C(F)F)C)=O)ccc(F)c(F)c1 78106,N1(C(c2cc(SC)ncc2)=O)CC2CN(Cc3cccc(C(F)(F)F)c3)C2C1 78107,N1(C(C2(COC)CC2)=O)CC(OC)C(NC(c2cc(OC)ns2)=O)C1 78108,c1(C(=O)NC2CC3(CC(CNC(COC(C)C)=O)C3)C2)cn2c(n1)CC(C)CC2 78109,c1(OC)cc(C(N2CCCC(SC)CC2)C(=O)NC2CCC2)ccc1S(C)(=O)=O 78110,C1(OC(C)(C)C)CCCN(C(=O)CCC2(CN)CCCCC2)C1 78111,C1(CC=C)(NC(=O)CCN2CCCC2)CCN(C(C2(CN(C)C)CCC2)=O)C1 78112,C1(CNC(=O)C=CCN2CCCC2)(NC(C2COC(=O)N2)=O)CCOC1 78113,c1(CC)cccc(C(=O)NC2(CF)CCN(C(C3CC(n4ccnn4)C3)=O)C2)c1O 78114,CC1CCN(C(c2coc(Oc3ccccc3)n2)=O)CC1CNC(=O)CC(F)F 78115,CC(C)CCCC(C)C(=O)NCC1(C(N2CCCC2CC(N)=O)=O)CC12CCC2 78116,CCC(C)(C(=O)NC1CC(NC(c2cncc(SCn3cccn3)c2)=O)C1)OC 78117,c1(N2C(C(=O)NC(C(C)C)CN3CCCC3)CC(F)C2)cc(C(C)(C)C)ncn1 78118,c1(C(N2C(CNC(=O)CN3CC(CF)C3)CC(OC)C2)=O)cc2cnccc2o1 78119,c1(C(=O)NCC2CCCN(Cc3cnc(Br)s3)C2)cc(C(=O)NC)ccn1 78120,C(=O)(C1=CCCC1C)N(CCN(C(c1ccc(C(C)=O)o1)=O)C)C(C)C 78121,Cc1cc(C)c(CN2C(C(NOC(c3ccc(CO)cc3)=O)=O)CC2)s1 78122,CC1CN(C(c2cnc(Cl)cn2)=O)CC(C)N(C(C2CC(=O)CO2)=O)C1 78123,c1(CC)cc(C(N2CC3C(CC(=O)NCc4ncon4)C3C2)=O)n(C)n1 78124,n1(CC(N2CCC(c3onc(NC)n3)CC2)=O)cc(C)c(=O)cc1C 78125,Cc1ccc(=N)[nH]c1C(N1CC(NC(=O)C(C)(C)c2cnsc2)CC1C)=O 78126,N1(C(c2cnc(C)s2)=O)CCCN(C(c2coc(Cl)c2)=O)CC1c1ccccc1 78127,Cc1nn(Cc2ccc(F)cc2)cc1C(=O)NCC1CC1NC(=O)C#CC(C)C 78128,C1(NC(C(C)(C)N(C)C)=O)CCCC(NC(c2cncc(C(=O)N(C)C)c2)=O)C1 78129,C(CC(=O)N1CC2CN(C(c3ncccc3Br)=O)CCC12)(C(F)(F)F)OC 78130,CCC(O)C(C)C(=O)NCC1CN(C(=O)Cc2cn[nH]c2)CC1C(F)(F)F 78131,C1(C(=O)NCC(C)CN(C(=O)COCc2ccncc2)C)CCC(F)(F)C1 78132,N1(C(CC(CNC(C2C(C(C)(C)C)CC2)=O)(C)C)=O)CCc2ccncc21 78133,N1(C(c2c(CC)noc2)=O)CC2(CCOCC2)CC1CNC(=O)CC(F)F 78134,C(CCC(C)CC(=O)NCCNC(c1cccc(O)c1F)=O)=C(C)C 78135,C(=O)(C1CCCS1(=O)=O)NCCCCC(C)NC(C=NOC)=O 78136,C1(F)(CNC(c2n(CC(C)C)ncc2)=O)CCN(C(c2nc(=O)n(C)[nH]2)=O)CC1 78137,N1(C(CCCCC)SC)CCC(S(=O)(=O)N2CCOCC2)C1 78138,c1(CNC(C2C(C(=O)Nc3ccccc3CO)C2)=O)c(Cl)cccc1[N+](=O)[O-] 78139,C1(O)(C(C)NC(=O)C=C2CCCC2)CCN(C(=O)CC(c2ccc(Cl)cc2)O)C1 78140,N(C(=NCCOc1nccc(C)n1)NCC(C)C)C(C=C)C 78141,N1(C(c2cc(C(CC)CC)no2)C(=O)NC(C)(C)C)CCC(O)C(O)C1C(=O)OC 78142,C1(C(=O)NCC(=O)NCCC)CN(C(=O)C(C2CC2)OC)C2(CCC2)C1 78143,N#Cc1ccccc1C=CC(N1CC2(CC(NC(C3(CO)CC3)=O)CO2)C1)=O 78144,C(=O)(CCCC(N)=O)NC(CCCCNC(C(C)OCC(C)C)=O)C 78145,N1(C(c2ccc(CC#C)cc2)C(=O)NCC(F)F)CCOCC1C=C 78146,c1(CC2(CNC(C3(C(C)(C)C)CCC3)=O)CC2)cccc(F)c1.C12CN(C1)C2=O 78147,c1(-n2cc(CCCC(=O)NCCCC(=O)O)nn2)ccc(C(=O)O)c(Cl)c1.CCOC 78148,c1(C(C)C)noc(CCCC(=O)N(CC(C)NC(c2ncc(Cl)s2)=O)C)n1 78149,C12(C(=O)NC3CCN(C(N)=O)C3)CC1CN(C(=O)COC1CCC1)C2 78150,c1(C(C)C)ncc(CN(C)Cc2cnc[nH]2)s1 78151,N1(C(c2ccc(COC)s2)=O)CCC(NC(C2CC3(C2)CCCC3)=O)C(O)C1 78152,CC1(C)OC2CC(C(N3CC(CCCCNC(=O)CCCS(C)(=O)=O)C3)=O)CC2O1 78153,c1(C(N(C2CCN(C(C(CCC)CC)=O)C2)C)=O)ccc2occ(C)c2c1 78154,N1(C(=O)C=CCN2CCOCC2)CC2CCN(C(c3cn[nH]c3)=O)CC(C2)C1 78155,C(=O)(C(C1(C)CC1)NC(=O)C(F)OC(F)(F)F)NCC(C1CCC1)OCC 78156,N1(C(c2ccc(C#N)s2)C(=O)Nc2c(C)cc(F)cc2)C2CCC1CC(CO)C2 78157,N1(C(c2cc(OC)ns2)C(=O)NCCc2cccs2)CCOC(C)(CC(=O)OC)C1 78158,CC(C(=O)Nc1cn[nH]c1)CCCSC(F)(F)F 78159,Cc1ncncc1C(=O)NC1CN(C(=O)CCOCC2CCCO2)CC1C 78160,c1(OC)cc(C(=O)NC2(C3CN(C(=O)C4=COCC4)C3)CC2)cc(OC)c1C 78161,N1(C(C=C(CC)CC)=O)CCC2(CCCC2NC(C2CCS2(=O)=O)=O)CC1 78162,C1(CC=C)(NC(=O)C(C)OCC(F)(F)F)CCCN(C(c2n[nH]c(C)c2O)=O)C1 78163,c1(C(=O)NCCCCN(C(=O)C(c2ccnn2C)O)C)ccc(C#N)cn1 78164,CN1CC(C(N2CCCCC2C2CCN(C(=O)Cn3[nH]cnc3=N)C2)=O)NC1=O 78165,C1(C(=O)NC(c2nocc2C(=O)N(CCF)C2CC2)C)CC=CCC1 78166,C12(C(=O)OC(C(=O)CCCO)CO)CCCN1S(=O)(=O)CC2 78167,c1(CC(N2CC3C(CNC(C(CC4CC4)OC)=O)C3C2)=O)c(C)cccc1Cl 78168,Cc1nn(C)c(C(=O)NC(c2ccc(Cl)cc2Cl)C2CC2)c1CC1(F)CCOCC1 78169,N(C1c2ccccc2OCC1F)S(=O)(=O)c1c[nH]ccc1=NC1C=CCCCC1 78170,c1(C(=O)NCC2(O)CC(CNC(CCC=C)=O)C2)cc(C(=O)NC)ccc1F 78171,c1(OC)cc(C)cc(C(=O)NC(C2(O)CN(C(=O)C3=COCCC3)C2)C)c1O 78172,c1(C(C(=O)NC(C)CC)N(CCCN(C)C)CCC)ncc(C)c(OC)c1C 78173,c1(C(=O)NC2(N)CCOC2)cc(Cl)c2cccc(Br)c2n1 78174,C1(C)(NC(c2n(CC)ccc2)=O)CCCN(C(c2cc(N(C)C)cnc2O)=O)C1 78175,C1(CNC(c2ccn(CC)n2)=O)CC2(CCC2)CN1C(=O)Cc1ccsc1 78176,C(c1csc(C(F)(F)F)c1)=CC(N1CC(N(C(C(CC#C)C2CC2)=O)C)C1)=O 78177,C1(CNC(c2c(C)snn2)=O)CC(NC(c2cnc(C3CCCO3)s2)=O)C(O)C1 78178,N1(CC2(C)CC2(F)F)C(=O)COCC1=O.c1nc(-c2ncccn2)no1 78179,C1(C(=O)NC2CCN(CCNC(c3c(C)n[nH]c3)=O)CC2)CC(C)CC(C)C1 78180,C1(CC(=O)Nc2ccc(CNC(C(C)NC(CC)=O)=O)s2)Cc2ccccc2O1 78181,N1(C(c2cnc(-c3cccc(C#N)c3)s2)=O)CCC2(CC(=O)NC2=O)C1 78182,CC1(C)CCN(C(=O)COCc2nccs2)CC1C(=O)NCCCc1nccs1 78183,C(N=c1[nH]c(C)c([N+](=O)[O-])cc1Cl)C1CC(NC(Cc2c(SC)cccc2)=O)C1 78184,c1(CC)c[nH]c(=NC)nc1CN(C(N1CCCCC(CN=[N+]=[N-])C1)=O)C1CC1 78185,N1(C(C(C)NC(C2CCCC2)=O)=O)CCCC(CNC(c2ccc(F)cc2)=O)C1 78186,C1(N(CC(=O)OC(C)(C)C)C(c2cccc(Cl)c2)CO)CCC2C(CC1)C2(F)F 78187,C(=O)(CCS(=O)(=O)N(C)C)NC1(C)CC(NC(c2cc(CC)nn2C)=O)C1 78188,C1(CNC(Cn2ncc(C)c2)=O)CC2(CO1)CN(C(=O)C(N1CCCCC1)C)C2 78189,CC1CN(C(c2ccc(CO)cc2)=O)CC(C)N(C(c2cccnc2)=O)C1 78190,C(CC(C)C(=O)NCC1(NC(=O)CCCc2n[nH]c(=N)s2)CCCC1)OC 78191,N1(C(CC(=C)C)=O)CC(NC(=O)C=Cc2cc[nH]n2)CC12CCC2 78192,CC(=Cn1ccnn1)C(=O)NCCCCC1(NC(C2CCCN2N=O)=O)CC1 78193,Cc1nc2[nH][nH]cc-2c(=NCC=CCNC(c2cc3n(n2)CCNS3(=O)=O)=O)n1 78194,C1(CNC(C2(C3CC3)CC2)=O)CC2(CCOCC2)CN1c1ncc2ncnc-2[nH]1 78195,C1(N(C(c2cccs2)=O)CC)CCCN(C(=O)CSc2ccccc2)C1 78196,C(=O)(C(C)(C)CCCNC(=O)C(N1CCCCC1)C)N(C)CCOCCO 78197,c1(C(=O)NCC(C2CCCCC2)NC(C(C=C)O)=O)ccnnc1Cl 78198,N1(C(C2N(C(C(C)OC)=O)C3C(O)CC2C3)=O)C2CCCC1CN(C)C2 78199,C(CCCCC(=O)NC1CCC1CNC(=O)CC12COC(C)(C1)C2)SC 78200,c1(SC)n[nH]c(CN2CCN(CC(=O)NC(=O)NC(C)(C)C)C(=O)C2)c1C#N 78201,c1(NC(C(c2ccccc2)C)=O)cccc(C(=O)NOCC(F)(F)F)c1 78202,c1(C(=O)NCC2(F)CC(NC(CCCCOC)=O)C2)cc2ccccn2c1 78203,C(=O)(C(O)CCCC)N1CCC(CC=C)(C(N2CC(O)(c3cnn[nH]3)C2)=O)C1 78204,c1(C(N2CCOCC(NC(C3(CCC)CCOC3)=O)C2)=O)ccc(C#N)cc1O 78205,N1(C(=O)Nc2ccc(SCC(=O)NC)cc2)CCCCCC2(CCCCC2)C1 78206,N1(C(CSSC)=O)CC(CNC(c2cc(C(F)(F)F)ncn2)=O)C(O)C1 78207,c1(C(=O)NCC2(F)CC(NC(=O)CC3CSCCS3)C2)ccc(F)c2ccoc12 78208,C1(C)(C(=O)NCCN(C(C2(c3ccc(C)nc3)CC2)=O)C2CC2)CCC(=O)NC1 78209,c1(NC(C2CC3(CC3)CN2Cc2n[nH]cc2Cl)=O)cccc(I)n1 78210,CCC(C(=O)N1CCC(CC(=O)NC(C)C(C)C)C1)C(C)C 78211,N1(C(C(C(C)C)N2CCCCC2)=O)CC2CCC1CN2Cc1ccc(CF)cc1 78212,Cc1ccc2c(C(=O)N(C(=O)CC(C)CC(C)(C)C)CC3CCN3)cccc2c1 78213,S(=O)(=O)(c1ccc([N+](=O)[O-])cc1F)N(c1cccc2c1CN(c1ccccc1)CC2)C 78214,C1(NC(c2c(C)sc(O)n2)=O)CC(O)CN(C(c2cc(C(C)C)on2)=O)C1 78215,c1(C(=O)NC2C(F)(F)CCN(C(C(=O)NC(C)C)=O)C2)cc(Br)cc2[nH]ccc12 78216,C1(F)(CNC(C2SCCS2)=O)CCN(C(=O)CSc2ccccn2)C1 78217,c1(C(=O)NC2CC(NC(C(c3ccn(C)n3)C)=O)C2)cc([N+](=O)[O-])n(C)n1 78218,C1(C(=O)NCCNC(C2CC(C)(C)C2)=O)(N(C)C)CCCCC1 78219,Cc1cc(C(=O)NC(CO)CCCCNC(=O)C(C)C(C)(C)C)cc(=O)n1C 78220,Cn1nnc2ccc(C(=O)NC(CNC(=O)C=Cc3cccnc3)CO)cc12 78221,Cc1nc(CNC2CC(C(=O)NC(c3cccc(C#N)c3)CO)C2)ccc1F 78222,N1(C(c2cc(C(CC)CC)no2)=O)CC(C2CN(C(C3(CN(C)C)CC3)=O)C2)C1 78223,C1(C(N(C)CC2(NC(C3OC4CCC3C4)=O)CC2)=O)CC2CCC1CC2 78224,CC1(CO)CCCC1NC(C1CCC1NC(C1CC1(F)Cl)=O)=O 78225,N1(C(C(c2cccnc2)C)=O)CC2CCCN(C(C3COC4COCC34)=O)C2C1 78226,c1(SC)nc(N2CCC(CNC(=O)C(O)CC(C)(C)C)C2(C)C)c2ccsc2n1 78227,C1(F)(C(=O)NCC(C)CC2CCC2)CCN(C(=O)C=Cc2cn(C)nn2)C1 78228,C(=O)(CCCCC(C)(C)C)N1C(C(=O)NCC2CCCC(C)(C)O2)CC(OC)C1 78229,C(=O)(C1CCc2snnc21)N(C)CC1CCN(C(C(n2ccc(C)n2)(C)C)=O)C1 78230,c1(C(=O)NCC(C)N(C)C(C2OCCO2)=O)ccnc2ncsc12 78231,c1(CNC(=NCC)NC2CCCC(N(C)C)C2)nnc2n1CCCC2 78232,C1(C(=O)NCC(C)(C2CC2)NC(C=CSC)=O)CCCCN1C(=O)OC(C)(C)C 78233,c1(C(N2CC3C(CNC(C)=O)(C3)C2)=O)cccc2c1OC(C)C(=O)N2 78234,Cc1ccc(C(N2CC(NC(c3cncc(N)n3)=O)C(C(F)F)C2)=O)nc1C 78235,N1(C(c2ccc(C(C)C)nc2O)=O)CCN(C(C2CCCCN2C)=O)C(C)C1C 78236,C1(n2cc(C(CC)OC)nn2)CCCN(C(=O)C(F)(F)c2ccsc2C(F)F)C1 78237,N1(C(c2c(C)nsc2)=O)CCCC2(C1)C(NC(c1cn(C)nc1Cl)=O)CCN2C 78238,N#Cc1ccc(CF)cc1.CN=c1[nH]nc(C2CC2)s1 78239,N1(C(C(C(C)C)NC(C)=O)=O)CCN(C(=O)CNC(=O)C2CC2)CCC1C 78240,Cc1cc(C(=O)NC2COCC2NC(c2sccc2C#N)=O)ccc1S(N)(=O)=O 78241,c1(C(=O)NC2CN(C(C3CN(C(C)C)C3)=O)C(CO)C2)ccc2ccc(F)cc2n1 78242,C1(CNC(CNC(CNC(C)=O)=O)=O)CN(C(c2cnncc2O)=O)CCO1 78243,C1(C(=O)NC2C(NC(c3cc(CN(C)C)on3)=O)CCC2)CC2(C1)CC(C)(C)C2 78244,c1(CC(=O)N(C2CCN(C(C=C(COC)C)=O)CC2)C)ccc(C)c(OC)c1 78245,C1(C)(CCNC(C(C2CN(C(=O)CC3(C)CCOC3)C2)OC)=O)CCCC1 78246,c1(C(=O)NCCCC(C)NC(C2CC3(CC(=C)C3)C2)=O)ccc2sc(=N)[nH]c2c1 78247,C1(N(C(C(C)SCC)=O)CC)CCC(NC(=O)CC2COCCN2C)CC1 78248,C(CCCC(C)NC(c1ccnc(C2CCC2)c1)=O)NC(C1C(CC)OCC1)=O 78249,c1(C(N(C2CCCC(NC(c3occc3F)=O)C2)C)=O)ccc(F)cn1 78250,Cc1nc(CNC(=O)C(C2(O)CCC2)NC(C2CC(C3CC3)C2)=O)sc1C 78251,C12C(C1(C)C)NC2=O.C(=O)(C(C)CO)NCCOCCC(=O)NC 78252,Cc1cc2nccnc2cc1C(N1CC(C)N(C(c2ccc(Cl)s2)=O)CC1C)=O 78253,CC(CC(=O)N1CC(NC(=O)Cc2cc(F)cc(Br)c2)C(O)C1)C(F)F 78254,N1(c2snc(CCC)n2)CC(CNC(=O)C(N2CCSCC2)C)OC(C)(C)C1 78255,N1(C(c2nc(OC)c(C)s2)=O)C2CCC1CN(C(C1(CSC)CCCO1)=O)CC2 78256,C1(C(N2C(C)C(NC(C3(C)CC(C)=NO3)=O)CC2)=O)CC2C(C1)C2(F)F 78257,CCC(C)(COC)C(=O)N1CCC(CNC(c2cnn(C3CCC3)c2)=O)C1 78258,CCC(CC(C)C)C(=O)N1CC(O)(CNC(c2nc(Cl)sc2Cl)=O)C1 78259,c1(OCC(N2CCCC(C(O)C(F)F)C2)=O)cccc(-c2ccc[nH]2)c1 78260,c1(CC)cc(C(=O)NC2CN(C(C3CC3OCc3ccncc3)=O)C2)oc1CC 78261,C(=O)(CCC1=CCCCC1)NC1CN(C(c2c(N)nc(C(F)(F)F)cc2)=O)C2C1C2 78262,CC1=NOC(CNC(=O)C(C)(C2CC2)N(C(=O)CN=[N+]=[N-])C)C1 78263,c1(C(N2CCC(NC(C(C=C)(C)O)=O)C2)=O)ccc([N+](=O)[O-])c(C(C)=O)c1 78264,C1(C)(NC(=O)Nc2cccc(SCc3cnc(C)[nH]c3=N)c2)Cc2ccccc2C1 78265,CCCC(CC)CCC(=O)NC1CC2(C(=O)NC(C)(CO)CO)COC1C2 78266,C12(C(=O)NCCc3nc(C)[nH]n3)CCCC1CCN2C(c1ccc(F)c(N)c1)=O 78267,C(CNC(=O)CCC(C)N(C)C)(CC(F)(F)F)NC(Cn1c(C)nnn1)=O 78268,C1(C(=O)OCC)CC(C(N2CCC2(C)NC(CCC)=O)=O)C1(C)C 78269,C(C(CN=c1[nH]cnc(Cl)c1[N+](=O)[O-])C(C)(C)C)NCCC(=O)ON(CC)CC 78270,C(C(O)C(=O)NCC(c1ccccc1)NC(=O)CC1CC12CC2)SC 78271,C(CCC(=O)N(C)C)(C(C)C)NC(C1(CC(=O)OC)CC1)=O.C1(C)C(=O)N1 78272,C1(NC(CCNC(=O)NC)=O)CN(C(c2cscc2Br)=O)C2CCCCC12 78273,c1(C(=O)OCC)cccc2c1ccn2CC(=O)OCc1ccnnc1O 78274,C1(C(=O)NC(CC)C(F)(F)F)CN(C(c2ccncc2F)=O)CC12CCC2 78275,CC1C(NS(=O)(=O)c2ccc(C(=O)O)cc2)C(NS(=O)(=O)C(F)F)CCS1(=O)=O 78276,c1(CC(=O)NC2CC(C(=O)NCc3c(C)nns3)OCC2)c(F)cccc1F 78277,C1(O)(CN(C(C(C=C)O)=O)C)CCN(C(=O)C(C2CC2)C2CC2)C1 78278,c1(OCC(N2C(Cn3cc(CCS(C)(=O)=O)nn3)CCC2)=O)ccc(F)c(F)c1 78279,C1(C(=O)OC)CC(NC(=O)CC=CCNc2ccsn2)C1 78280,C1(OC)C(OC)CN(C(c2cc[nH]n2)=O)C1CNC(=O)C(C)N1CCC1 78281,Cc1cc(C(N2CC(CNC(C3COC(=O)C3)=O)CC(C)C2)=O)ncc1F 78282,N1(C(c2c(C)noc2C(F)(F)Cl)=O)CC2CC1CN2C(c1sccc1CC#N)=O 78283,C(C)(C(C)NC(n1cc(C(c2ccccc2)C2CC2)nn1)=O)(C1CC(F)(F)C1)OC 78284,N1(C(c2c(C)cccc2N)=O)CC2(CCCC2NC(C2CC(C3CC3)=NO2)=O)C1 78285,c1(COC)ccc(C(N2CC(O)(C(C)NC(=O)C(C)c3ncco3)C2)=O)s1 78286,CCC(COC(C1(C)CCCC1)=O)CO 78287,CC1(C)CC(C(=O)NCC2CC2(F)F)CN1C(=O)CCc1cccc(O)n1 78288,N1(C(C2C(C(C)N)OCC2)=O)CC(S(N)(=O)=O)C1.C1CCC(C)(C)OC1 78289,c1(C(=O)NC(CC)CC(=O)NCC(F)Cl)ccnc(C)c1C 78290,c1(CC)ccc(C(=O)NC2CCC2NC(C2CNC2)=O)cn1 78291,Cc1ccc(C(c2ccccc2)NC(N2CCCC2CCC(=O)O)=O)c(Cl)c1 78292,c1(C(=O)NC(c2c(F)ccc(N(S(CC)(=O)=O)C)c2)C)nc2c(s1)CN(C)CC2 78293,C1(NC(COCCCOC)=O)CCN(C(c2cnn(C)c2C)C)CC12CCC2 78294,c1(C(=O)NC2CC3CN(C(C4(C)CCCC4)=O)C(C2)C3)cccc2cccnc12 78295,C1(CC(=O)N(C2CCN(C(=O)C(C)CSCC)C2)CCC)CCCOC1 78296,C=CCCCCC(=O)N(C)CC1(C)CCCC1NC(c1ccc(C)s1)=O 78297,C1(CC(=O)N(C)C2CC2)CCCCC1.C1C(=O)N(C)CC2(CC2)CC(=O)CN1.CC(=O)N 78298,N1(C(C(C)C)=O)CCCN(C(=O)C(n2nnnc2C(C)(C)C)C)C(C)C1 78299,c1(OC)ccn2c(C(=O)NCCN(C(c3c(C)nsc3C)=O)C(C)C)cnc2c1 78300,CN=C(NCCc1cc(-c2ccccc2)n[nH]1)NCC(C)(C)n1ccnn1 78301,N12CC3C(C3C1)C2=O.C1(C(=O)O)CC(C(=O)NC(c2cnc[nH]2)C2CC2)C1 78302,C1(C(=O)NCCC2C(C)CN(C(c3c[nH]c(C#N)c3)=O)C2)CN2CCCN1CC2 78303,C(=O)(C(COC)CC(C)C)NC1CCC(CNC(C(COC(C)=O)N(C)C)=O)CC1 78304,C=CC1(CO)CCN(C(=O)C(CCC)NC(=O)CSCC(F)F)C1 78305,C1(NC(C=CC(N)=O)=O)CC2(CCCCN2C(c2cc(CC3CCC3)c[nH]2)=O)C1 78306,C(=O)(CC(O)C(=O)NCC1CCC(NC(=O)C2CC2)CC1)NC(C)C 78307,S(=O)(=O)(c1cccc(=NCc2cn(C3CCCC3)nn2)[nH]1)NCCc1ccn(C)n1 78308,N1(C(C)=O)CC(O)CC1C(=O)NCC1CCN(C(C2(C)CSC2)=O)C1 78309,C(=O)(CCCCCCCCCO)N1CCC(CN(C(=O)COC(F)(F)F)C)CC1 78310,Cc1ccccc1C=CC(=O)NCC12CC1CN(C(=O)C(C)O)C2 78311,c1(SC)cccc(C(N2CC(O)CC2C(=O)NC2CN(c3cncs3)C2)=O)c1 78312,c1(C(C)=O)cc(C(N2CC(n3cc(CNC(=O)C(C)CO)nn3)C2)=O)oc1C 78313,N1(C(C2ON=C(CC)C2)=O)CCCC2CN(C(=O)C(C)NC(C)(C)CC)CC12 78314,n1(CC)cnc2c(NCc3nc(=N)[nH][nH]3)nc(N(C)CCC3CCOC3)nc12 78315,C1(N(C(=O)CNS(C)(=O)=O)C)CCCN(C(=O)Cc2nc(C3CC3)no2)CC1 78316,c1(C(=O)NCC(C)CN(C)C(C2CNC(=O)N2C)=O)coc2c(F)cc(F)cc12 78317,O=C(CCCC1CCC1)N1CCC(CC(=O)NC2(C(N3CCCC3)=O)CCCC2)C1 78318,C1(C(=O)NCC2(OCC)CN(C(C3CC3[N+](=O)[O-])=O)C2)CCNC(=O)C1 78319,c1(OC)ccc(=NC(=O)C23CC2CN(C(c2cc(Br)ncc2F)=O)C3)[nH]n1 78320,n1(CC(N2CC(N(C)C(c3ncccn3)=O)C(F)C2)=O)nc(Cl)ccc1=O 78321,N1(C(C(C=C)O)=O)CCC(C(F)F)(CNC(c2cnn(CC)n2)=O)C1 78322,N1(CC)CC2=C(C1=O)C(c1ccc(F)c(F)c1)NC(=O)N2CCC1CCCO1 78323,c1(C(N2CCC(NC(C(C)CF)=O)(CO)CC2)=O)c(O)cnc2ccccc12 78324,C1(c2n(CCCOC)nnn2)(NC2CC(NC3CCCC3)C2)CCC(C)C(C)C1 78325,N1(C(c2c(CC)noc2)=O)CCC(CO)(NC(=O)Cc2cnn(C3CCC3)c2)C1 78326,C1(CNC(=O)COC2CCC2)CCC2CN(C(c3ccc(O)cc3)=O)CCC2C1 78327,C1(NC(C(C)(C)SC)=O)CC12CCN(C(=O)Cc1ccoc1C)CC2 78328,C(c1cn(C)c2ccccc12)=CC(=O)NC1CN(C(CN(C(C)C)C)=O)CC1C 78329,C(=O)(C(C)N(N(CC(=O)NC)CCOC)C)OC.C1(C=O)CCC1OC 78330,c1(C(N(CC(CNC(c2n(C(C)C)ccc2)=O)C)C)=O)[nH]ncc1C#N 78331,CCCCS(=O)(=O)NC(=O)COc1ccccc1OCC1CCCCN1C(C)=O 78332,c1(NC(=O)NC2CN(C(C3(OC)CCOC3)=O)C2)ccccc1N=[N+]=[N-] 78333,c1(C(=O)NC(CCCNC(c2nnc(C)s2)=O)C)cccc(CO)c1C 78334,CC(C)(CCC#N)C(=O)NC(CNC(=O)Cc1ccc(Cl)cc1Cl)CC(F)(F)F 78335,c1(C(C)NC(CCC2(NC(C=CCOC)=O)CCCC2)=O)c(F)cccc1F 78336,N1(C(Cc2ccc(OC)nc2)=O)CCC2C(C1)NC(=O)CN2C(C1CC1F)=O 78337,N1(C(C(CC)(F)F)=O)Cc2occ(C(N3CCC(CCCO)C3)=O)c2C1 78338,Cc1cc(C)n(CCCC(=O)N(C(=O)CCCCCl)C(C)C)n1 78339,Cc1ccc(-c2cn(-c3ccccc3Oc3ccccc3)nn2)cc1C(=O)N(C)C 78340,c1(CC(=O)NC2C(OC)CN(C(C3C(C)(C)C3(F)F)=O)C2)ccc(Cl)cc1Cl 78341,Cc1cc(C)c2c(=NC=C3CCCC3)[nH]c(=NCCOCC(C)(F)F)[nH]c2c1 78342,Cc1nc2ccc(S(=O)(=O)NC3CCC4CCCC34)cc2o1 78343,Nc1ccc(Br)c(F)c1C(N1CC(NC(c2csc(Cl)n2)=O)C1)=O 78344,N1(C(c2cn(CC)nn2)=O)CC2CCC2(CNC(c2occc2C)=O)C1 78345,c1(CC(=O)NCC2N(C(C(CC)C(C)C)=O)CC2)ccccc1[N+](=O)[O-] 78346,C1(NC(C(C)NC(C)(C)C)=O)C2CC1CN(C(=O)C=Cc1cn(C)cn1)C2 78347,C1(=CC(N2C(CCNC(CSCC#C)=O)COCC2)=O)C2CC3CC(C2)CC1C3 78348,N1(C(c2nc(CC)oc2)=O)CC(NC(c2sc3cncn3c2C)=O)C(C2CC2)C1 78349,C(CCCCCC(=O)N1CC2CCC2(CNC(=O)C(O)CF)C1)SC 78350,C(=O)(CC(C)(C)C(F)F)NC1(CC(=O)NC(CCC)C(=O)N(C)C)CCC1 78351,c1(C(=O)NCC(C)CNC(=O)CCCC(C)(C)C)n[nH]c2c1CCCCC2 78352,Cc1cc(C(=O)NCC#CC(N2CCOC(C(N)=O)C2)=O)sc1C 78353,C(N=c1[nH]c(=NC(CCO)C2CC2)[nH]c2ccsc12)c1n(CC)cnn1 78354,c1(OC)ccc(C(N2CC(NC(=O)CC3(O)CCCCCC3)CC2C)=O)cc1C 78355,C1(N=[N+]=[N-])(C(N2CC(NC(COC)=O)C2)=O)CCN(C(c2cc(Cl)n(C)n2)=O)C1 78356,C(=O)(N=c1cc(Cl)c(C#N)c[nH]1)C1C2(CN(Cc3c(C)cc(OC)c(OC)c3)C2)C1 78357,N1(C(CC2(OCC)CC2)=O)CCCC1C(C)(C)C(=O)NC1CC(F)C1 78358,c1(OCCOC)ccc(C(=O)NC2CCC(NC(=O)C(C)C(C)C)CC2)cc1 78359,C1(C(=O)NCC2CN(C(CSCCOC)=O)C2)CCc2cncn2C1 78360,N1(C(COCC(C)C)=O)CC2C3CCC(C2C1)N(C(c1ncccc1CO)=O)C3 78361,Cc1cccc(C(=O)NCC(CNC(c2nn(C)cc2Cl)=O)=O)c1.C1(CN)CC1N 78362,C1(C(=O)Nc2snc3nccnc23)CCc2nnc(O)cc2C1 78363,c1(CC)ccc(CNC(=O)C(CCCC(N)=O)NC(=O)C(C)C(=O)OC)cc1 78364,Cc1nsc(N)c1C(N1CSCC1C(=O)NCCSCCO)=O 78365,CCCC(C)C(=O)N1CC=CC1CNC(C1CC(O)C1)=O 78366,C(=O)(C1=NOC2(CCOC2)C1)N(CCN(C(c1cn(CC=C)nn1)=O)C)C 78367,Cc1nn(C)c(C)c1CC(N1CC(C)(C)CC1CNC(C1C2(CC2)C12CC2)=O)=O 78368,C(N=c1ccc2c([nH]1)CCC2=O)C1CC(NC(C(C(C)C(F)(F)F)F)=O)C1 78369,c1(OC)c(C(=O)NCCCN(C(=O)CCc2nncs2)C2CC2)cccc1F 78370,CC1CC=C(C(=O)NC2CN(C(c3cccc4nccn34)=O)CC23CC3)CC1 78371,C1(C)(C(N(CC(C)C)Cc2ncccn2)=O)CCCN(c2cc(=O)cco2)C1 78372,CC1(C)CC=C(C(=O)N2CCCC2CCCNC(=O)CC2CCC(=O)N2)CC1 78373,c1(OCCOC)cc(C)c(Cl)cc1N.N1(CCCCCN)C(C)CCCC1C 78374,CC1=C(C(=O)N2CC(C)CN(C(=O)C=Cc3ccsc3)CC2C)C(C)(C)CCC1 78375,Cc1ccc2c(c1)C(=O)OC(C)(C(=O)NC(C)CNC(c1sc(C)nc1C)=O)C2 78376,c1(CCC(=O)OC)cccc(CN2CCCC(CN3CCSCC3)C2)c1 78377,N1(S(CCC)(=O)=O)CC2CC1CN2C(c1ccc(N2CCOCC2)cc1)=O 78378,C=CC1(C(=O)NC(C)C(C)C(=O)NCc2cncc(Cl)c2)CCCCC1 78379,C1(NC(C(CCOC)OC)=O)CCN(C(=O)Cn2ccsc2=N)C(C)C1 78380,N1(C(COc2cc(C)on2)=O)CCC2CN(C(C3CCC=CCOC3)=O)CC2CC1 78381,N1(C(COCC)=O)CCC(C)(C)C(NC(=O)COCC(=O)OC)C1 78382,C1(C(=O)N(CCCN(C)C(c2cnn(CCOC)c2C)=O)C)(CC)CCNC1=O 78383,c1(C(=O)NC(CC)CNC(C2(F)CCOC2C)=O)c(C)nn(C)c1N 78384,Cn1cnc(CNC(=O)CC2CC2CNC(=O)CSCC2CC2)n1 78385,CCC(C(=O)N1CC(OCC(=O)NC2CCOC2)C1)OC 78386,N1(C(C#CC2(CC)CC2)=O)CC=C(C(=O)N2CC3CCC(C2)O3)CC1 78387,CC1(C)COCCC1CNC(=O)COc1ccccc1-c1nc[nH]n1 78388,C(CCC(F)(F)F)N(C(=O)CC1(O)CCOC1)C.c12cn(nn1)CCOCCOC2 78389,C(=O)(CC(CC)C(C)(C)C)NCC(CC=C)NC(=O)CN(S(=O)(=O)CC)C 78390,c1(C(=O)NC(CC(C)C)CNC(c2cc3sccc3[nH]2)=O)c(F)ccc(N)c1F 78391,c1(-n2c(CC3CC(C(CC=C)O)C3)nc(-c3ccncc3)n2)cccc2nc[nH]c12 78392,C(=O)(CC(C)(C)CNC(c1ccnc(C)c1)=O)N(C(CC)CO)CC 78393,C1(C(N2C(CCC(=O)N(C)Cc3cc(=O)cc[nH]3)CCC2)=O)CC2(CCC2O)C1 78394,CC(CCCC(=O)N(C)CCn1cccn1)NC(=O)C=Cc1ccccc1 78395,c1(C(C(=O)NCCCC)N(C)C(c2ccncc2)C)ccc(OCOC)cc1Br 78396,c1(C(=O)NC2CCN(C(COC(C)C)=O)C(C3CC3)C2)ccc2n[nH]cc2n1 78397,c1(C(=O)NC2CC3(C(C(CC)(C)OC)=O)CC(C3)N2)ccc(P(C)(C)=O)cc1 78398,C#CC1(O)CCN(C(C)C(=O)NC(C)(C)CCNC(C2CCC(F)C2)=O)CC1 78399,CCCCCCCCCC(=O)N1CC(NC(=O)COCP(C)(C)=O)CC(C)C1 78400,C1(C(=O)NCCCCCN(C)C(C2CC(NS(C)(=O)=O)C2)=O)CCCS1(=O)=O 78401,c1(C(=O)NC(C2CCCC2)CC)ccn(CCNC(=O)CCCc2ncco2)c1 78402,C1(CN)CCC2(CCC2)O1.C1(CCCOC(C)C)CCCN1C=O 78403,N1(C(CCCc2cc(C)no2)=O)CC(NC(=O)CC2CC2(C)C)C(F)C1 78404,C(=O)(CCS(N)(=O)=O)N(C(CC)C(=O)N1CCC(N2CC(O)C2)C1)C 78405,c1(C(c2cccc(OCC)c2)NCC2CCC3CC3C2)cc([N+](=O)[O-])ccc1Cl 78406,C1(NC(=O)CC2COCC2O)C2CN(C(=O)CCCc3ccccn3)CC12 78407,C1(NC(=O)COCC2CC2)CC2CCC1(C(=O)N(C)CC1(F)CCC1)C2 78408,C1(N2C(=O)C2)CCN(C(C2CCOC2C(F)(F)F)=O)C1.C(C(C)C)SC 78409,C1(C(=O)NCCSCCC(=O)NCc2c(C)nc[nH]2)CCCN1C=O 78410,C1(OC)CC(C(=O)NC(Cn2cncn2)C(F)F)N(C(=O)OC(C)(C)C)C1 78411,N1(CC)CCOC(CNCCCC2CCCC2)C1 78412,Cc1ccc(F)c(C(=O)NCCC2(O)CCN(C(=O)CCC3(O)CCC3)C2)c1F 78413,C1(C)(C(N(CCCO)C)=O)CCN(C(c2cc(C(F)F)[nH]n2)=O)CC1 78414,C12(NC(CCC)=O)CCCC1CN(C(c1sc(C(C)C)nc1C)=O)C2 78415,C1(C(N2CCC(C(C(=O)NCCc3ccc(O)cc3)F)C2)=O)CCC2(CCC2)C1 78416,c1(C(=O)NC(C2CN(C(=O)CCn3cncn3)CCO2)C)ccc2[nH]ccc2n1 78417,C1(CNC(c2c(C)sc(C)c2Br)c2n(CCC)nnn2)CSc2ccccc2O1 78418,N1(C(c2cc(COC)sc2)=O)CC2C(NC(C3CCCC(COC)C3)=O)C2C1 78419,CCC(CC)(C(C)C)NC(=O)C(CNC(c1ocnc1C)=O)N(C)C 78420,c1(CC(C(=O)N(CCCCNC(C2(C)CCCCC2)=O)C)O)ccc(F)cc1 78421,N1(C(c2c(C)[nH]cc2)=O)CC2C3CCC(C2C1)N(C(=O)Cc1cnoc1)C3 78422,C1(NC(Cc2c(C)nc(O)nc2O)=O)CC(N=c2[nH]c3cccc(Cl)c3o2)C1 78423,N(C1CCc2ccccc21)C(=O)C(O)CNC(C1CCOCC12CCC2)=O 78424,C1(C(=O)NC(C(C)NC(COCCOC)=O)CO)CC2(CCCCC2)S1(=O)=O 78425,c1(C(=O)NC(C)CCNC(C2(C)CCCOC2)=O)cc2c(nn1)CCCC2 78426,N1(C(c2ccc(F)cc2I)=O)CCC(O)C(N=c2ncnc(C(F)(F)F)[nH]2)C1 78427,c1(C(=O)NCC(CNC(C(C)Sc2nncn2C)=O)F)nnc(O)cc1O 78428,C(C)(C(C(=O)NCCN(C(C)C)C1CC1)C(C)C)NC(C=CC(=O)OC)=O 78429,c1(NC2C(OCC)CC2)cc([N+](=O)[O-])cc(-c2cccc(OC)c2)c1O 78430,C1(NC(C2(CCOC)CC2)=O)CCN(C(=O)COCCSC)CC12CCC2 78431,c1(C(N2CC(CNC(C3CCC=CCCC3)=O)OCC2)=O)cc2n(n1)CCCO2 78432,N#CC1NC(=O)CC1C(=O)N(C1CCN(C(=O)Cn2ccccc2=O)CC1)CCO 78433,Cc1onc(C2CCCCC2)c1C(=O)N(C(CNC(=O)CC(F)(F)F)C1CC1)C 78434,Cc1ccc(F)c(C(=O)NCC2(C)CC(NC(c3cnc4n3CCS4)=O)C2)c1F 78435,N1(C(C2(CC(C)C)CC2)=O)CC(C(=O)NCC2C3COCC23)C(C)(C)C1 78436,CC(C)(CC=CC(=O)NC1CCCC1C)NC(=O)CC1CCSC1 78437,c1(C(N2C(CC)CN(C(=O)C(F)=CC3CC3)CC2)=O)cccc2cc(Cl)ccc12 78438,C1(C(=O)NCC(CN(C)C)(C)C)CNC(=O)CN1C(=O)CC(=O)NC1CC1 78439,C1(N(C)C)CN(C(=O)Cc2csnn2)CC1CNC(C1COCCN1C)=O 78440,C1(C(=O)NC2CCC(CNC(c3coc(C4CC4)c3)=O)C2)CCc2n[nH]cc2C1 78441,c1(C(N2CC(CC)C(NC(=O)C(C)C)CC2)=O)cnc(S(C)(=O)=O)s1 78442,N#CC12CCCCC1CN(C(c1cscc1Cl)C(=O)NC1COC1)C2 78443,CCCC(O)C(=O)NCCCN(C(C1C2CC2C2CC12)=O)Cc1ccccc1 78444,N(C(=NCC1CCOC1)NCC1(C(=O)OC)CCC1)C(CC)C 78445,c1(C(=O)NCCCCNC(C2(C#C)CC2)=O)ccsc1S(N)(=O)=O 78446,CC(CNC(C1(C(C)(C)O)CC1)=O)CC(=O)Nc1cccc(O)c1 78447,CN=c1[nH]c(=NCC23CC(CN2C)C3)[nH]c(=NC(C)c2cc(C)on2)[nH]1 78448,Cc1cnc(C(=O)NCC2(CNC(=O)C(c3ccn(C)c3)C)CC2)cn1 78449,C(C(F)(F)C(=O)Oc1ccc(F)nc1)NC(C1N(C(C)(C)C)CC1)=O 78450,N1(C(c2ccccc2[N+](=O)[O-])=O)CC2CCN(C(C3CC3(Cl)Cl)=O)CC2C1 78451,C1(CNC(CCC#C)=O)CCC(C)(C)CN1C(c1sc(C)nc1C)=O 78452,C1(NC(C(C=CC)O)=O)CCCN(C(CO)C(C)C)C1 78453,C1(NC(CS(=O)(=O)NCC)=O)(CNC(c2ccoc2C)=O)Cc2ccccc2C1 78454,C12(C(N3CCC(OCCNC(CCCOCC)=O)C3)=O)CCCC1CC(=O)CC2 78455,c1(CNC(c2scc(C(=O)NC3CC(Cl)(Cl)C3)n2)=O)cc(F)c(F)cc1O 78456,c1(NC(N(C)CC2CC(C)(C)C2)=O)ccc(S(N)(=O)=O)cc1F 78457,c1(CC)ccc(NN2CC(=O)N2C2CC2)c(OC)c1.S(C)(=O)(=O)N(CC)C 78458,CC1CCNCC1CC(=O)N(Cc1ccccn1)Cc1cccc(F)c1 78459,N1(C(C(C=C)C)=O)CCC2(C=C(C(=O)N3CCOCC3C3CC3)C2)C1 78460,c1(C2N(CC)CCC2)ccc(F)c(Cl)c1.c1(NC(C2CCOC2)=O)nccnc1OC 78461,C(CC(C)(C)CNC(=O)C(=O)NCc1ncc(C)o1)OC 78462,C(=O)(CC(C)(C)COC)NCC(CCC)NC(=O)C(c1cccs1)SC 78463,CC1CC2(CCCC2)CN1C(C1CCC(C2CC2)N1C(C1CCCN1C1CC1)=O)=O 78464,CC1CC(NC(=O)CCc2ccsc2Br)CCS1(=O)=O 78465,N1(C(C(C)(C)C2CCCO2)=O)CCN(C(=O)C(C)(C)C2CCCCO2)CC1 78466,C(CS(=O)(=O)c1ccc(C(=O)NC2CN(C(=O)C3=CCCS3)C2)cc1)OC 78467,C(C(C)C(F)C(=O)N(C)Cc1cccs1)NC(CCn1ncc(C)c1)=O 78468,C(=O)(C(C)(C)NC(=O)C=CC(C)(C)NC(c1cc[nH]c1)=O)NC 78469,C(=O)(CCCCC(C)=O)N1C(CC(N2CCC(CC#CC)CC2)=O)CCCC1 78470,N1(C(Cc2c(C)n[nH]c2)=O)CCCC(NC(=O)CC2CCC(C)(O)CC2)C1C 78471,c1(NCC(=O)NCC(CNC(CSCC=C)=O)F)c(C)cc(Cl)cc1C 78472,C(CCC(=O)NCCC1CCCO1)NC(CC1CC(=C)C1)=O 78473,CC1CN(C(c2ocnc2C(F)F)=O)CC(C)C1NC(=O)Cn1nnnc1C1CC1 78474,Cc1nn(C)cc1C(=O)NCCCOCCN(C(=O)Cc1ccc(C#N)o1)C 78475,Cc1ncc(C(C)NC(c2cn(CCNC(=O)CC34CCCC3C4)cn2)=O)s1 78476,c12cc(ccn1)OCCNC2=O.c1(C(NOCCC)=O)c[nH]c(=NC)cc1 78477,CCC(C)C(=O)NCC(=O)NCC(C1CCCC1)CNC(=O)Cc1cc(C)no1 78478,N1(C(c2c(CC)c[nH]c2)=O)CC(N=[N+]=[N-])CC1C(=O)N(C)CC1CCCCO1 78479,Cc1cc(C(N2CCCC2CCCNC(c2cc3sccc3s2)=O)=O)ccc1Cl 78480,N1(CCC#C)CCN(C(=O)C(C)(CO)NC(=O)CC2CCCCC2O)CC1 78481,N1(CC(=O)NC(C2(O)CCN(C(c3cn(CCO)nn3)=O)C2)C)CCNC(=O)C1 78482,c1(N(C)Cc2ccnc(C)n2)nc(N2CCn3nncc3C2)c2c(n1)CSC2 78483,C1(C(=O)NCC2CCCN2C(=O)C2=CS(=O)CCC2)CCN(CP(C)(C)=O)CC1 78484,N1(C(CNC(CCC(C)C)=O)=O)CC2CCCC1(CNC(=O)Cc1cncs1)C2 78485,C1(F)(C(=O)NC(CC)CC(=O)OC)CCN(C(C2CCN(C)C2=O)=O)CC1 78486,CC1(C)CC(NC(=O)C=Cc2cncs2)CN(C(=O)COC(F)(F)F)C1 78487,Cc1cnc(C(=O)NCC(=O)N(C2(NC(=O)CN3CCC3C)CC2)C)[nH]1 78488,Cc1cc(C(=O)NC2C3CN(C(c4cc(F)cc(Br)c4C)=O)CC23)c(Br)cc1F 78489,c1(C(=O)NC2CC3CN(C(CCOCCC)=O)C2C3)nc2cc(O)ccc2[nH]1 78490,C1(CC(=O)NC(C)COC(F)(F)F)COCCN1C(C1OCCC1(C)C)=O 78491,N1(C(C(CC=C)OC)=O)CC2OCCN(C(c3ccc(O)nn3)=O)C2C1 78492,Cc1csc2cc(C(=O)NC(C)CNC(c3cnn(CC4CC4)c3)=O)[nH]c12 78493,CC1(C)C(NC(=O)C=Cc2cncs2)CCN1C(C1CC2CC2C1)=O 78494,c1(CN(N=CCC)C(=O)Oc2ccc(COCC)cc2)ccc2c(c1)CC(C)O2 78495,C#Cc1cccc(OCC(N2CC3(CCN3C(c3ccccc3SC)=O)C2)=O)c1 78496,c1(C(=O)NC23CC(NC(C4C(C)(CC)C4)=O)(C2)C3)cnc2ncc(Cl)cn12 78497,C12CC(F)CN(C1)C2=O.N1(C(=O)CSc2ccccc2)CCC(CO)C(O)C1 78498,c1(C(=O)NCC(C(C)C)NC(c2c(OC)cco2)=O)ncc(N)cc1C 78499,c1(OC)cc(CN(CCS(N)(=O)=O)C)ccc1OCCO.C1(C)CC1(F)F 78500,C1(O)(CN(C(c2[nH]cc(CC)n2)=O)C)CCCN(C(C23CCC(C)(C2)OC3)=O)C1 78501,C(=O)(CCCC(F)(F)F)N1CCC=C(COCCOCCOc2cn(C)nc2)C1 78502,N1(C(CC2CCC(C)O2)=O)CC(NC(=O)Cn2cnnn2)CC(F)C1 78503,CCC(O)C(C)C(=O)N1CCC(O)(C(F)(F)C(N)=O)CC1.C1(O)CCCCC1 78504,c1(C(N2C(C)CCC2C(=O)Nc2ccc(Cl)nc2F)=O)cc(F)ccc1[N+](=O)[O-] 78505,c1(CC)cc(=NC(=O)C(C)C(C)NC(C2C3CC(=O)CC23)=O)[nH]n1C 78506,CC1(C)C2CCC(C(=O)NC3C4CN(C(c5ccc(C(F)F)nc5)=O)CC34)C1C2 78507,C1(NC(=O)OCC)CN(N2CCCOC(C(C)C)C2)CC1OC 78508,Cc1ncc2n1CCC(C(=O)NC1(CNC(=O)Cc3sc(O)nc3O)CCC1)C2 78509,C(=O)(CCCCC(F)(F)F)NCCCN(C)C(c1nnc2n1CCCC2)=O 78510,CC1CCCCC1(CNC(c1ccsn1)=O)NC(C12CCCC1CCC2)=O 78511,C1(C(=O)NCCC2CC(O)C2)COCCN(C(c2n[nH]cc2[N+](=O)[O-])=O)C1 78512,c1(C(N2CC3CCN(C(CCN(CCC)C)=O)C3C2)=O)ccc2nc(C)cn2c1 78513,CC1=CC2CC(C1)CC(c1nnnn1CCC1(C)CC1)(NCC1CC1)C2 78514,N1(C(C2C(CCNC(CCn3c(C)ncc3)=O)C2)=O)Cc2ccc(Cl)nc2C1 78515,N1(C(C2(C(F)F)CC(=C)C2)=O)CC2CN(C(c3cnn4ccsc34)=O)CC(C1)O2 78516,C1(NC(=O)OC(C)(C)C)(CC)CCN(C)CC1.CCC1CN(CC(C)C)C(=O)N1 78517,c1(CCC(=O)CC(n2cc(C(C)(C)OC)nn2)C)cccc(Cl)c1Cl 78518,C(=O)(C(CNC(c1cccnc1Oc1ccc(Cl)cc1)=O)C(C)C)NCC 78519,Cc1c(N)cc(C(N2CCC(CO)(NC(=O)C(C)C(C)O)CC2)=O)cc1N 78520,Cc1cc(C(N)=O)sc1C(=O)N(CCC(C)NC(c1cnc(N)cn1)=O)C 78521,C1(NC(C(CC)N2CCCC2=O)=O)CN(C(=O)CN(C(=O)COC)C)CCC1F 78522,C(=O)(C(C)CSC)N(CC=CC(=O)N(C1CCCCC1)CC)C.O(C(F)(F)F)CC 78523,C1(CCCC)CN(C(=O)Cc2ccccc2)CCN1C(=O)C(O)CN(C)C 78524,C(c1ccc(Br)cc1)=CCC(=O)NCC(CNC(C(C)C1CC1)=O)CO 78525,N1(C(C(CCCC)O)=O)CC2CCCC2(CNC(c2ncc(Br)cc2OC)=O)C1 78526,C1(NC(c2c(CC)n(C)nn2)=O)CCCCCC1NC(=O)CCCn1ccnn1 78527,N1(C(C2N(CC)CCOC2)=O)CCCC(NC(=O)C=Cc2cccc(F)c2)CC1 78528,c1(C(=O)NCC(C2CC2)NC(CC2(N(C)C)CCC2)=O)c[nH]c2nccc(Cl)c12 78529,C(C)(CCC(C)(C)C)(c1nnnn1C1COC1)NCC(=C)Br.C12(CC1)C(=O)O2 78530,C1(C)(COC)CC(NC(C2CC23CCCC3)=O)CN1C(c1cnccn1)=O 78531,CC(C)C(N=[N+]=[N-])C(=O)NC1CC(C(=O)NC(C)(C)CC2CCC2)C12CCC2 78532,C1(NC(=O)Cc2ccncc2)CC2(C1)CN(C(=O)CCCN1C(=O)CCC1=O)C2 78533,C1(C(=O)NC2C3CN(C(C=CC(C)C)=O)C(C3)CC2)CC2CCC(C1)S2(=O)=O 78534,Cc1ncc(NC(C2CCN2C(c2cc(Br)cnc2F)=O)=O)c(C)n1 78535,C1(O)(CN(C(c2ccc(COC)o2)=O)C)CCN(C(=O)C2=COCCC2)CC1 78536,C1(C(N2CCC(CCNC(c3cscn3)=O)CC2)=O)CC1C1CC(F)(F)C1 78537,C(=O)(C(F)C(C)CNC(=O)C(C)OCC=C)NCCSCC#C 78538,c1(CC)ccc(C(N2CC(NC(=O)CC(C)c3ccncc3)C(O)C2)=O)nc1 78539,N1(C(c2c(C)snn2)=O)CC2ON=C(CNC(=O)COCC3CC3)C2C1 78540,c1(NC(c2[nH]nc(C3N(C(C(CCC)C)=O)CCOC3)n2)=O)cc(C)cnc1O 78541,C1(C(=O)N(c2cnoc2)C2CC2)CCN(C(=O)CCc2ccccc2)CC1O 78542,C1(C(=O)NC(c2nc(=O)o[nH]2)C)CC2(CCN1C(C1CC(=O)C1(C)C)=O)CC2 78543,Cc1nn(C)c(C(=O)NC(CN=c2[nH]nc(CO)s2)C2CC2)c1I 78544,C1(C(C)C)CN(C(=O)Cc2cn[nH]c2)CCN1C(c1cc(Cl)n(C)n1)=O 78545,c1(C(=O)NC2CC2C(=O)NCC2(C)CC2)cc(Cl)c(Cl)c(Cl)c1 78546,N1(C(C(CC)C2CCOCC2)=O)CCN(C(C2(C)COC2)=O)C(C)C1 78547,c1(C(=O)NCCC23C(CN(C(CCC)=O)C2)CC3)n[nH]c2cccc(OCC)c12 78548,CCC1=NOC(CC(N2CCC(CC(=O)NCCCC(=O)NO)C2)=O)C1 78549,Cc1cc(C(=O)NC(c2ccc(N(C)C)cc2)CNC(=O)C(C)O)ncn1 78550,N1(CC(C(C)C)(C)O)CCN(N2CCCC(c3cnc4ccccn34)C2)CC1 78551,CC(C)CCC(C(C)C)NCc1cn(-c2cc(Cl)ccc2Br)nn1 78552,O=C(O)CC(C(=O)NC1CCC(n2ccnn2)CC1)c1ccc(Cl)s1 78553,c1(C(=O)NCC2(CCO)CCC2)cc(CN)cs1.C1(C(=O)C2CC2)(CO)CCCO1 78554,C(=O)(CC(C(F)F)NC(=O)C(C)=CC1CC1)NC(C#C)(CC)CC 78555,O=C1CCC2(CC1)CC2C(=O)Nc1cccc(Oc2nccs2)c1 78556,c1(C2(C(N(CCOCCCNC(CC=C=C)=O)C)=O)CCC2)cccc(Cl)c1 78557,C1(CC(N2CC(CCCCNC(=O)CCc3ncc[nH]3)C2)=O)Cc2ccccc2O1 78558,CC1CN(C(=O)CCCc2ccccc2)CC(C)C1NC(=O)C(C)(C)C(=O)N(C)C 78559,C1(C(=O)NC(CCOC)COC)CN(C(=O)CCn2cccn2)CCC1C 78560,C12(CC(=O)NCc3ccccc3N3CCN(C(=O)C(F)F)CC3)CCC(CC1)C2 78561,C(C(N=[N+]=[N-])C(=O)NCC1CCCN(C(=O)CCN2CCN(C)CC2)C1)OCC 78562,c1(C(C(=O)N(CCNC(C2CC3(CC3)C2)=O)C2CC2)(F)F)cccc(F)c1F 78563,Cc1cc(C)c(NC(=O)C(C(C)(C)C)n2cc(CCCCCO)nn2)cc1O 78564,C1(OC)(OC)CC(C2CCN(c3nnc(-c4ncccc4F)n3CCCO)C2)C1 78565,c1(C(CC)NC(N2CCCC2)=O)ccc(-c2nc(C(F)(F)F)no2)cc1 78566,Cn1[nH]c(=NC(=O)NC2CCN(Cc3ccc(F)cc3)CC2)c2ccc(Br)cc12 78567,C1(CNC(CCCCC=CC)=O)CN(C(=O)C=C(Cl)Cl)CCC12CCC2 78568,N1(C(c2c(C)c(N)cnc2)=O)CCC(C2CCN(C(c3ns[nH]c3=O)=O)C2)C1 78569,O=C(CC1=CCOCC1)N1CC(N2CCN(C(C3CCCC4(CCC4)C3)=O)CC2)C1 78570,C12(C(=O)Nc3c(CC)ccnc3)COCC1CN(C(c1cn(C)cn1)=O)C2 78571,C1(C(C(=O)NCCC2CC2)N(CCF)CC)CC2CC1C1CC21 78572,N1(C(C=CC(C)C)=O)CCN(C(=O)CC2CCCC2(F)F)CC(C)(C)C1 78573,N1(C(c2scc(OC)c2)=O)CC(NC(=O)CCCc2cnn[nH]2)CC12CCOC2 78574,c1(CC)cccc(C(=O)NCC(C)(C)NC(c2cc(C3CC3C)on2)=O)c1 78575,CC1CC(C)CN(C(=O)C(C)CC(N2CCCC2C(C)(C)C(N)=O)=O)C1 78576,CN(C)NC(=O)CCC(=O)NC1C=CC(CNC(C2CC3CCCCC23)=O)C1 78577,N1(C(C=Cc2ccc(C)o2)=O)CCN(C(=O)Cn2cccn2)C2CC12 78578,N1(CC(=O)N(CC(F)(F)Br)C)CCn2c(C(F)(F)F)nnc2C1 78579,C1(CN(C(CN2C(C)CCC2)=O)C)C2CN(C(c3csc(C(C)(C)C)c3)=O)CC12 78580,C1(C(N(CCNC(c2sc(Cl)c(Cl)c2OC)=O)CC)=O)CC2COCCN2C1 78581,c1(C(=O)NC2CN(C(C(CC)COC)=O)CC2C2CC2)cc2cc(F)ccc2[nH]1 78582,N1(CC(C)(C)C(=O)NC2CCOC2)CCC2(CCN(c3ccc(C#N)nc3)C2)C1 78583,c1(C(=O)NCC2N(C(COCC=C)=O)CCOC2)cc(S(=O)(=O)N(C)CCC)c[nH]1 78584,N1(C(CN(C(C2(COC)C=CCC2)=O)C)=O)CCN(C(c2nnc(C)s2)=O)CC1 78585,N1(C(c2c(C)cco2)=O)CC2CC2(CNC(c2sccc2-n2ccnn2)=O)C1 78586,c1(NCC(=O)N(CC)CC)nccc(N2CCCC(c3nc(=N)[nH]s3)C2)n1 78587,C1(NC(c2c(CC)c[nH]c2)=O)C2CC3CN(C(c4cnsc4C)=O)C1C3C2 78588,n1(CC)c(O)nc2ccc(NC(C3CCN(CC(O)COC)CC3)C(C)C)cc12 78589,CCCCC(F)C(=O)N1CCC(CC(C)NC(=O)C(C)N2CC(C)C2)CC1 78590,C(CCF)(C(=O)NCC(C)N1CCC1)NC(C1(COCC)CCC1)=O 78591,CC1(CNC(C2CC(C(F)F)C2)=O)CCN(C(=O)C(F)(F)c2csc(=N)[nH]2)C1 78592,c1(CC)cc(CC(=O)N(CCCCCNC(=O)CN2CC(C)C2)C)on1 78593,C1(NC(C(CCC)C)=O)(CNC(c2cc(C)nc(OC)n2)=O)CCCCC1C 78594,C(=O)(CC(C)CC(F)(F)F)NC1CCC(C)N(C(C2(O)CCCC(C)(C)C2)=O)C1 78595,C(CC(C)C(=O)NCCC(O)CNC(C1CN(c2nnnn2C)C1)=O)=CC 78596,S(=O)(=O)(c1ccccc1F)NCCC(=O)N(C(CCCC=C)c1ccccc1)C 78597,C1(CC)CC(C(=O)NC(c2nccs2)CC2CC2)CCO1 78598,c1(C(=O)NCC(CNC(C(N)=O)=O)CO)ccc(OCC2CC2)nc1 78599,C1(C(=O)NCCCOCCN(C)C(c2n[nH]c(C)c2C)=O)CCCC(N)C1.COC 78600,c1(OCC)ccc(Br)cc1CN1CCC(NC(c2ccc(CC)o2)=O)C(F)C1 78601,N1(C(C2(CNC(C3C(CC(C)(C)C)C3)=O)CC=CC2)=O)CC2(CCCC2)C1 78602,C1(NC(C=CC(C)(C)C)=O)CN(C(=O)CNC(c2ccc(Cl)cc2)=O)CC2(CC2)C1 78603,C12(NC(C(C)CC(N)=O)=O)CCC(CNC(c3cccnc3O)=O)(CC1)OC2 78604,c1(C(=O)NC(C)CNC(c2ccccc2F)=O)cc(=NS(C)(=O)=O)cc[nH]1 78605,c1(CC)c[nH]nc1C(=O)NC(Cn1cccn1)C(=O)NC(CC1CCCC1)CO 78606,Cc1ncccc1C(N1CC(NC(=O)COC2CCN(C)CC2)C(C(F)F)C1)=O 78607,c1(C(=O)NC(C2CN(C(c3ccccc3C(F)F)=O)C2)C)nc(=O)n(C)[nH]1 78608,C(CCC(C)C(=O)N1CCOC(c2cn(CC(C)C)nn2)C1)OC 78609,c1(OCC(C)C)ncc(C(N2CCC(NC(C3CC(O)CN3C)=O)C2)=O)cc1Cl 78610,N1(C(COC)=O)CC2CC(C(=O)Nc3c([N+](=O)[O-])cnn3C(C)(C)C)CC1C2 78611,C(C(C)(C)C1=CCCC1)NCCNC(NOCCOCC)=O 78612,N1(C(CC2(CC=C)CCCC2)=O)CC2CCC(NC(=O)CCS(C)=O)CC1C2 78613,c1(C(=O)OC)ccc2[nH]c(=NCC3CC(C)N(C(C4CCS4(=O)=O)=O)C3)sc2c1 78614,C1(CC)(CC)CC(NC(=O)C(C)CC2CC2)CN1C(c1ncn2c1CCC2)=O 78615,c1(OC)cncc(C(=O)NCC2CC2NC(C2CC(n3cnnc3)C2)=O)c1 78616,n1(CCONC(C2N(C(C(CO)N(C)C)=O)CSC2)=O)nnc2ccccc12 78617,C(=O)(C1=CCCOC1)N(C1CCCCC1NC(c1ccc(C(=O)C2CC2)nc1)=O)C 78618,CC(=O)CCCC(C)C(=O)NC1(C(N2CC([N+](=O)[O-])C2)=O)CC(O)C1 78619,c1(CC)cccc(C(N2CC3CCC3(CNC(c3cscc3CC)=O)C2)=O)c1O 78620,N1(C(CSc2n(C)cnn2)=O)CC(NC(=O)CCNC2CCC2)CC1CO 78621,c1(CN(C(C(C2CCCC2)NC(C2CC(=C)C2)=O)=O)C)cccnn1 78622,C1(C(C(=O)NCC2C(OCC)CC2)(C)C)CCCN(C(=O)CC(C)C2CC2)C1 78623,C1(CNC(c2cn(C)nc2)=O)CCC2(CO1)CC(NC(=O)C=Cc1ccc[nH]1)C2 78624,CC1CCc2ncc(C(=O)NC3CCN(C(C4CCCSC4)=O)CC3C)n2C1 78625,N1(C(C(C(C)C)OCC)=O)Cc2occ(C(=O)NC(C)C(O)C(F)F)c2C1 78626,C=CCC(CNC(=O)C(CC)C(=O)OC)C(=O)NC(C)C(C)(C)SC 78627,C1(NC(c2c(CNC(CCC(C)N(C)C)=O)n[nH]c2)=O)CCC(O)C(O)C1 78628,C1(C(=O)NC(C(=O)OC)Cc2cn(CC(C)(C)C)nn2)CCn2cncc2C1 78629,Cc1cnccc1CC(N1CC(NC(c2cnn(C)c2N)=O)C1)=O 78630,C1(NC(CS(CC)(=O)=O)=O)CN(C(c2coc(C(C)C)n2)=O)Cc2ccnn2C1 78631,c1(OC)ccc2c(N(C3CCN(C(C4CCNC(=O)C4)=O)C3)C)ncnc2c1 78632,CC1(C(=O)NC2CC2NC(=O)CC2(CN(C)C)CCOCC2)CCCCO1 78633,c1(C(N2C(C)(C(=O)NCCCc3cn[nH]c3)CCC2)=O)cc(F)cc(F)c1 78634,CC1(C)Oc2ccsc2C(N=c2[nH]c(=N)[nH]c(=NCc3nc(O)n[nH]3)[nH]2)C1 78635,c1(C(N2CC(C(=O)NCCCCCCO)OCC2)=O)c(I)ccnc1F 78636,n1(CCC)cccc1C(=O)NCC(C)(F)CNC(=O)C(C)=C1CCC1 78637,C(=O)(C#CC1CCC1)NC(c1ccccc1)C(=O)Nc1c(CC)nn(C)c1 78638,N1(CC(C)(C)N(C)C)CCN(C(=O)C(C)(F)NC(=O)NC(C)(C)C)CC1 78639,C1(CCCNC(C2CC(OC)C2)=O)CCN(C(=O)Cc2nnc(C)o2)CC1 78640,Cc1cnc(C(=O)NCC2(F)CC(NC(C3CC3C(F)F)=O)C2)nc1 78641,C(=O)(CC(C)(C)CN(C)C)NCC1(OC)CN(C(=O)CC2CCOC2=O)C1 78642,C=CCCCC(=O)NC(C1CCCCC1)C(C)NC(=O)CCc1ccoc1 78643,N1(C(c2cc(C)no2)=O)CC2(CC2)CC1CC(=O)NCC1CC(CF)C1 78644,C1(N(C(c2c(CC)c[nH]n2)=O)C)CCN(C(=O)CCc2cn(C)nn2)CC12CC2 78645,CS(=O)(=O)c1ccc(F)c(C(N2CCCN3CCCCC23)=O)c1 78646,C1(C)(C(N(CCCCN(C(C(CC)(C)C#N)=O)C)C)=O)CCCNS1(=O)=O 78647,c1(C(=O)NC(C)CNC(=O)Cc2ccnc(C(N)=O)c2)c(F)ccc2[nH]ccc12 78648,CN1CCOC(C(=O)NCC2CN(C(=O)CCc3ncc[nH]3)CC2(F)F)C1=O 78649,c1(CC(N2CC(N(C)C(C3CCCCC3O)=O)C2)=O)ccc(O)cc1Cl 78650,C1(C)(CNC(CSCCC)=O)CCCN(C(C2C3C4CCC(C4)C23)=O)C1 78651,c1(CNCC2N(C(c3ccc(C(F)F)cc3)=O)CCC2)c(Br)cccc1[N+](=O)[O-] 78652,CC1(C(=O)NC2C3CC2CN(C(=O)CC2CC4CCC2CC4)C3)CCCCCC1 78653,c1(CC)ncc(C(=O)N(C2CCCC2)CCNC(C2CNC(=O)C2)=O)c(O)n1 78654,N1(C(c2nnn(C)c2N)=O)CCCC(NC(=O)Cn2cnc([N+](=O)[O-])c2)C(F)C1 78655,C(CCC)(C(=O)NCC(CC(C)C)NC(c1cc(CN(C)C)on1)=O)=CC 78656,Nc1cc(Cl)ncc1C(=O)NC1CC2CCC1(CNC(=O)Cn1ncnn1)C2 78657,C1(CN(C)C(c2ccncc2)=O)COCCN1C(c1c[nH]nc1C(F)(F)F)=O 78658,CC(CS(C)(=O)=O)C(=O)NC1CC(CNC(c2ccc(-c3cc[nH]n3)s2)=O)C1 78659,Cc1ccccc1S(=O)(=O)N(C1CCC2(CC1)CNC2)CC(=O)O 78660,c1(CC)ccnc(CNC(=O)CC(C2CC2)NC(C2NC(=O)OC2C)=O)n1 78661,O=C(C1=CS(=O)CCC1)NC1CC2CC1N(C(c1cncc3[nH]ccc13)=O)C2 78662,N1(CCCNC(C2C(=C)CC2)=O)CCN(C(c2nc(C)[nH]c2C(=O)OC)=O)CC1 78663,CC1(O)CCN(C(=O)CCC2CCCCN2C(=O)CCOCC2CC2)CC1O 78664,C1(CNC(C(CC)C#N)=O)CC2CCCC2N1C(c1ccccc1F)=O 78665,C1(C#N)(C(=O)OCC)CCN(CC(CO)C(F)(F)F)CC1 78666,c1(OC)cc(N)c([N+](=O)[O-])cc1C(=O)NCC1CC1NC(c1nn(C)cc1N)=O 78667,N1(C(C2N(CC)CCC2)=O)CCC(O)CC1C(=O)NC1C2C=CC(C2)C1CO 78668,c1(C(=O)NC(C(=O)NCCOCCOC)CC2CC2)ccc(=O)n(C)c1 78669,C(=O)(C1=CCCCCC1)N1C(C)(C(=O)NC(C)CN2CCCCC2)CC(O)C1 78670,C1(C)(C(N2C(CNC(c3ccc(CC)[nH]3)=O)CC2)=O)CCCCCC1 78671,C(c1ccco1)=C(C(=O)N)C.c1(COCCN(CC(C)O)C(=O)C)cc(Cl)ns1 78672,Cc1cc(C(N2CCC(N(C(=O)CC3(CO)CCC3)CCO)C2)=O)cc(O)c1 78673,c1(C(=O)NC2C=CC(CC(=O)NCCCCN(C)C)C2)cc(O)cc(F)c1 78674,C1(C=C)(NC(CCN(C(=O)C(N2CCOC2=O)C)CC=C)=O)CCCCC1 78675,N1(C(C(C)C)=O)CC(NC(C2CN(C(=O)OC(C)(C)C)C2)=O)C1(C)C 78676,C1(NC(=O)CCc2cn[nH]c2)C=CCC(C(=O)NCC2CCC(F)C2)C1 78677,Cn1cc(C(=O)NC2CN(C(c3cc(C(N)=O)[nH]n3)=O)CC2O)nc1O 78678,n1(CC)ncc2c(NCCCCCO)[nH]c(=NCC(C)=C(C)COC)nc12 78679,C#CC12CCN(C1)C(=O)OC1CCN(C1)C2=O.C1(C(=O)NC)CN(C2CCC2)C1 78680,Cc1onc(Br)c1C(N1CCC(NC(c2cccnc2O)=O)C1)=O 78681,CC(C)C(F)(F)CC(=O)NCCCOCCNC(C1CCC(C)CN1C(N)=O)=O 78682,c1(OC)ccc(C(N2CC(CN(C)C(c3conc3C(C)(C)C)=O)C2)=O)c(F)c1 78683,C(CC(O)CC(=O)NC1CC(NC(=O)CC(C)O)C1)SC 78684,c1(N2CCC(CC=C)(NC(C3CC4CCCC34)=O)C2)ncnc(Cl)c1C#N 78685,C1(NC(C2C3CN(C(c4cn(CC)nc4C)=O)CC32)=O)CC2(CCC2)C1OC 78686,C(C)(C(=O)N(CCC(=O)NCC1CNC(=O)CO1)OC)OCCCC 78687,CCCN=C(NCC1CS(=O)(=O)c2ccccc2O1)N1CCN(C2CC2)C(=O)C1 78688,CC(C)(C(C#N)OC(c1cc(C2CCC2)no1)=O)c1ccc(Cl)cc1 78689,c1(C(=O)OC)ccc(NC(C)C(CO)NC(=O)CSC)c([N+](=O)[O-])c1 78690,c1(OC)cccc(C(=O)NC(CO)C(C)NC(C2CCNC(=O)C2)=O)c1O 78691,n1(CC(=O)NC2CC3CC(NC(CC4CC(SC)C4)=O)C3C2)nc(C)ccc1=O 78692,C(=O)(C1=CCCCC1)N(CC(O)CNC(C1CC12CC2)=O)C 78693,C1(CNC(c2cncc(NC)c2)=O)CN(C(=O)C(C)OCC(C)C)CC(C)(C)O1 78694,N1(C(C(C(CC)O)C)=O)CC2CCC(C1)N2C(=O)CNS(=O)(=O)N(C)C.C(COC)S 78695,C1(C(=O)NC(C)Cc2ccco2)CN(C(=O)C(F)CC(C)(C)C)CC1C1CC1 78696,CC(Cn1ccnc1)C(=O)NCC1CCCN1C(=O)COCP(C)(C)=O 78697,CCC(C)(O)C(=O)NN1CCCC1NC(=O)NC1CC(=C2CCC2)C1 78698,N1(C(CCNC(C)=O)=O)CC(N(C)C(c2ccc(Cl)cc2Cl)=O)C(C)(C)C1 78699,C(=O)(CC(C)n1cccn1)NCC(C)N(C(COCCSC)=O)C 78700,c1(C(N2CCC(NC(C(P(C)(C)=O)O)=O)C2)=O)cc2ccccn2n1 78701,c1(N2CCCN(CCC(C)C)CC2)nccc(=NCCC2CCC3(CCC3)O2)[nH]1 78702,CC(CNC(C12CC1CCN2C(=O)CC1(C)OCCO1)=O)C(F)(F)F 78703,N1(C(c2c(C)onc2)=O)CCC2(CCC2)C(NC(C2CC3CC3C2)=O)C1 78704,C1(N(C(C(c2cnn(C)c2)OC)=O)C)CC2CC1N(C(c1ccc(F)cc1)=O)C2 78705,CC1(C)CCC2(CC1)CC2C(=O)NCC1CCN1C(=O)CCc1nccs1 78706,c1(C(=O)NCCN(C)C(c2cc(C(F)(F)F)nn2C)=O)cc2cn[nH]c2cn1 78707,C1CCC(O)C(=O)O1.c1(-n2cc(C3C(C(=O)NC)C3)nn2)cncc(Br)c1C 78708,C1(C#N)(C(=O)NCC2(O)CN(C(c3ccc(SC)o3)=O)C2)C(C#N)C1(C)C 78709,C(C(C(=O)N1CCOC(C(=O)NC)C1)C(C)(C)C)NC(C(C=C=C)C)=O 78710,CC(O)CCCCCC(=O)N1CC2(CC(NC(=O)CP(C)(C)=O)CO2)C1 78711,C1(C)(C(N2CCC(OC)(CNC(=O)CN(C)C(=O)C3CC3)C2)=O)CC2C=CC1C2 78712,N1(C(c2n(CC)ncc2)=O)CC(CNC(=O)C(F)(F)C(O)C2CC2)CC1(C)C 78713,N1(C(c2nc(C)sc2)=O)CC2CCCC2(NC(=O)CN2CCC(=O)NC2=O)C1 78714,N1(C(Cc2c(C)ncs2)=O)CCC(C(N2CCN(C)CC2C)=O)C12CCC2 78715,N1(C(c2cc(C)[nH]n2)=O)Cc2ccc(O)cc2CC1C(=O)NCc1cc(C)on1 78716,CCCC(CC(=O)NC(C)(CO)CCC)NC(C1OCCCC1(C)C)=O 78717,Cc1c(C(N2CCC(NC(c3cnn(C)c3N)=O)C2C)=O)cnn1C(C)C 78718,C1(CC(=O)NC2CN(C(c3c(C)oc(C(C)C)c3)=O)C(C)C2)CCCC(C#N)C1 78719,C(CC(C(=O)NCCC1CCCN1C(c1oc(CC2CC2)nc1C)=O)OC)OC 78720,Cc1cc(C(=O)NC2CCN(C(c3cccnc3Br)=O)CC2)c(C(F)(F)F)o1 78721,C(=O)(CC1OC(=O)c2ccccc21)Nc1c(C)ccc(F)c1.C12(CC1)CN2 78722,CC(C)C(O)C(C)C(=O)N1C(CC(=O)N(C)CC2CN(C)C2)C2CCCC12 78723,C(=O)(CC(CNC(=O)C1=CCCC1)C1CCC1)NC(C)Cn1ccnc1 78724,c1(CC(=O)NC(CNC(C2CCCC(N(C)C)C2)=O)C)cccc(Cl)c1F 78725,C1(NC(CCCCCC)=O)CCC(O)CN(C(=O)C(C)(O)C(C)C)C1 78726,C1(OCC=C)CN(C(=O)C2CC2)C(C)(C(=O)OC)C1.C(=O)(COC(C)(C)C)NC 78727,C1(C(=O)NC(CNC(c2cnc(NC(C)=O)o2)=O)CC(C)C)CC12CCCCC2 78728,CON(C(=O)C(C)C1CCCN(C(=O)CC(C)(C)C2CC2)C1)C(C)C 78729,N1(C(c2c(C)nco2)=O)CCOCCC1C(=O)NC1CCCCC1(C)C 78730,C(C(CNC(c1ncnc(C)c1C)=O)C(F)(F)F)NC(C=C(CC)C)=O 78731,N1(C(Cc2cccc(OC)c2)=O)CCN(C(=O)C(C)CF)CC(C)(C)C1 78732,c1(OC)ccc(NC(C2CC(NC(c3cnc(N(C)C)nc3)=O)C2)=O)cc1Cl.NC 78733,Cc1cc(Br)ccc1C(N1CCC(CN(C)C(c2cccc(Cl)c2F)=O)CC1)=O 78734,c1(C(=O)NC2C(NC(=O)CC3C=CCCC3)CC2)cnc2ccccc2n1 78735,C1(C(=O)NC2CCCC(C(N(CCCC)CC)=O)C2)CC2(C1)CC(C)C2 78736,C1(C(=O)NCC(=C)CCNC(=O)C(C)Sc2cccs2)(CO)CCCCC1 78737,C1(C(N2CCC(N(C(=O)Cc3nocc3C)CC#C)CC2)=O)CCCCCN1C 78738,c1(C(N2CCC(CCNC(CN(C(C)=O)C)=O)CC2)=O)cc(N)c(Cl)c(O)c1 78739,c1(C(=O)NCCN2CCC(NC(CC(CC)C)=O)CC2)cc(N)ccc1Cl 78740,CC(=O)CCCCC(=O)N1CCC(C(=O)NCc2ncccc2F)(CF)C1 78741,N1(C(c2c(N)snn2)=O)CCCC2(CCCN2C(C2C3CCCOC23)=O)C1 78742,C(CNC(c1ccc(F)s1)=O)(CC(F)(F)F)NC(C1(C#N)CCOC1)=O 78743,c1(CC(=O)NCC23CN(C(C(C)CO)=O)C(CC2)C3)cn2cc(Cl)cc(Cl)c2n1 78744,c1(C(=O)NCC(C)(CO)NC(=O)C=CC=C(Cl)Cl)ccc(C2=CCOCC2)cc1 78745,CCCCCCCCC(=O)NC1CCN(C(c2ccc(N)c(O)c2)=O)C1 78746,CCC(C)(CC)C(=O)N(CCNC(C1CCCC(N(C)C)C1)=O)CC1CC1 78747,CC1(C)COCC1CC(=O)NCC1(NC(c2ccc(C(=O)N(C)C)cc2)=O)CCC1 78748,C=CCC(CC=C)C(=O)NC(C1(O)CCN(C(c2ccn(C)c2)=O)C1)C 78749,CC(C)(CC(=O)NCC12CN(C(=O)COC(F)F)C(C)(CO1)C2)CC(F)F 78750,C#CCC(CC(F)F)C(=O)N1CCC(CC)C1C(=O)NOCCC(C)O 78751,c1(C(=O)NC2CC(NC(=O)C(F)n3ccnc3)C2)ccc(F)c(OC(F)(F)F)c1 78752,CN1CCN(C(=O)Cc2csnn2)C(CNC(c2cc3[nH]ccc3s2)=O)C1 78753,c1(OC)cccc(Cl)c1CN1CC(CO)(NC(c2cccnc2C(F)(F)F)=O)C1 78754,CC1=C(C(=O)NC2CC(C)N(C(=O)CCCn3ccnc3)C2)CCC(C)(C)C1 78755,C1(NC(=O)Cc2sc(O)nc2O)CCCC12CN(C(C1CCC(C(N)=O)O1)=O)C2 78756,C(CC)(CCCC(=O)NCC1CCC(=O)N1)NC(c1c(CC)[nH]cc1)=O 78757,Cc1cc(Br)c(C(=O)NC(c2cccc(Br)c2)CC(N)=O)c(Br)c1 78758,C1(NC(C=CSC)=O)CCS(=O)(=O)C2(C1)CC(CNC(=O)C(C)C(F)F)C2 78759,c1(C(=O)NCC2C(O)C(O)CN2C(=O)C=CCF)cc2c(nc1O)CCSC2 78760,CC(CC(F)(F)F)C(=O)N1CC(N(C)C(c2occc2Br)=O)C(O)C1 78761,C(CC(C)(C)C)(C(=O)N(CC(C)(C)CNC(C1(CO)CCCO1)=O)C)OC 78762,c1(NCC(=O)NCCCNC(C(C)=CC)=O)ncnc2sc(C)c(C)c12 78763,N1(C(COC(C)=O)=O)CC2CCC(CNC(c3ccc(C(F)F)s3)=O)(C2)C1 78764,c1(N2CCC(NC(C3N(C(C)=O)CCC3)=O)(CO)CC2)nccc(S(C)(=O)=O)n1 78765,n1(CC#C)c(C)cc(C(N2CCC2CNC(c2c(C)csc2Cl)=O)=O)c1C 78766,CON=Cc1ccc(NC(C2CCN(C(=O)C(N)=O)CC2)=O)cc1 78767,N1(C(c2cnn(C)c2)C(=O)Nc2c(C)cccc2)CCc2ccc(C#N)cc2C1 78768,N1(C(C(=O)NCCCC)c2csnn2)CCCC(c2nn(C)cc2C(N)=O)C1 78769,C1(C2(NC(CNC(c3ccoc3)=O)=O)CC2)CCCN1C(=O)CCC1CC1 78770,C(C(C(=O)N(C1CC1)CC1CCCN1C(=O)CCNC=O)N(C)C)N(C)C 78771,c1(C(=O)NC(CC)CNC(=O)CC(C)SC)ccc(N)c(Cl)n1 78772,C1(CC)CN(C(c2c(C(F)(F)F)cnn2C)=O)CCC1NC(c1cc(C)cs1)=O 78773,N1(C(C23CN(C(C4C(CC)C4)=O)C(C2)CO3)=O)CCN2C(=O)NCC2C1 78774,c1(C(CC)NC(c2coc(Cl)c2)=O)nc2ccc(C)cc2[nH]1 78775,C1(N)CCCCC1OCC(=O)N(CC(CNC(C=CC)=O)(C)C)C 78776,N1(C(CN2C(=O)CNC2=O)=O)C2CCC1CC(NC(=O)CCCC1CC1)C2 78777,C(C)(CC(=O)NC12CC(NC(=O)C(C)CC3CC3)(C1)C2)SC 78778,C(=O)(CCCCCCCCCO)N(CCNC(c1cccc(C(F)F)c1)=O)CC 78779,CC1CN(C(=O)CCc2cncn2C)CCN1C(=O)CC(c1cccc(F)c1)O 78780,Cc1nc(O)c(C(=O)NCC(N2CCCCC2)Cc2cccnc2)c(C)c1[N+](=O)[O-] 78781,C(=O)(C(O)C(F)(F)F)NCCOCCCN(C(=O)CCc1ccccc1Cl)C 78782,C(CCC)(C(=O)NCc1ncc(C)s1)NC(C(C=C)C)=O 78783,N1(C(C(C2CCOCC2)C)=O)CC=C(C(=O)Nc2c(O)cccc2Cl)CC1 78784,CC(C)(C)C(CNC(c1cccc2nccn12)=O)C(=O)N1CC=CCC1 78785,N1(S(CCCOCC)(=O)=O)CC(C(=O)OC)CCC1C 78786,c1(N2CCC(C)C(NC(c3cc4c(s3)CCC4)=O)C2)ncnc2cc(F)c(F)cc12 78787,C1(C)(C(N2CC(COC)(CNC(C3CCCOC3)=O)C2)=O)CC2CC2C1 78788,N1(CCC)CCCC(C(N2CCCC2C(C)(C)NC(=O)CC(C)(F)F)=O)C1 78789,CCC(CCCC(=O)N1CCCC1SC)NC(c1csc(C(N)=O)n1)=O 78790,c1(C(=O)NCCCN(C(=O)CCc2cn[nH]c2)CC)ccc2ccnc(Cl)c2n1 78791,N1(C(COCCCC#C)=O)CCC2CN(C(C3CC4C=CC3CC4)=O)CCC2C1 78792,N1(C(c2c(C)cc(F)cc2)=O)CC(C2CN(C(C3CC3(C)C(F)F)=O)C2)C1 78793,Cc1cc(C(=O)NC23CCOC(CNC(C4CCCCC4C)=O)(C2)C3)ccc1Cl 78794,c1(C(N2CCN(C(c3ns[nH]c3=O)=O)C(CO)C2)=O)ccccc1[N+](=O)[O-] 78795,c1(CC)ccc(NC(C2CCCN2C(C2CCCN2C2CC2)=O)=O)cn1 78796,CC(C)C(CNC(c1ccc(O)cc1)=O)C(=O)NCC1CCC(CO)O1 78797,O=S(=O)(c1cccc(Br)n1)N.c1(CN2CCOCC2)ccc(Cl)c(Cl)c1Cl 78798,Cc1ocnc1CC(=O)NC(CNC(=O)C=CC1CCCO1)C1CCC1 78799,C1(CNC(CCCCSC)=O)CC2CCC1N(C(c1cnnc(C)c1)=O)C2 78800,CCC(CC(=O)NCC1(C)CCC(NC(c2ccc(C(N)=O)o2)=O)C1)CC(F)(F)F 78801,c1(C(=O)NC2C(C)CCN(C(=O)C=CBr)C2)nccc2ncccc12 78802,N1(C(C(Cc2cn[nH]c2)NC(=O)CC2CCCCC2)=O)CCC(O)(C(F)F)C1 78803,C(=O)(C1SCCc2sccc21)N(C)CCNC(c1cc2c([nH]1)CCOC2)=O 78804,c1(OC(C(=O)NC2(C)CCN(C(c3c(CC)nns3)=O)C2)F)ccc(Cl)c(F)c1 78805,C(C)(CCCNC(=O)Cn1cc(C2CC2)cn1)NC(C1C(CC)C1)=O 78806,c1(C(N(CC(CNC(CCC(C=C)(C)C)=O)O)C)=O)ccc2c(c1)nnn2CC 78807,Cc1occc1S(C)(=O)=NC(=O)C12CCC(CO)(C1)OC2 78808,c1(CC(C(=O)O)NC(C2CCC(C(C)(C)C)C2)=O)c(F)cccc1Cl 78809,C(=O)(CC1=CCCCC1)N1CC2(CN(C(C(CC)SC)=O)C2)C1 78810,N1(C(CC(C)SC)=O)CCOCC(CNC(=O)COc2cccc(Cl)c2)C1 78811,c1(CCC)cc(C(=O)NC2CC(CNC(C3CC34CCC4)=O)CC2O)nn1C 78812,c1(C(=O)NCC2(CN(C(C(CC)SC)=O)C)CC2)cnn(C(C)C)c1C 78813,Cc1ncc([N+](=O)[O-])n1CC(=O)NCCCCC(CO)NC(c1n[nH]cc1Cl)=O 78814,c1(OC)cccc2c1C(N=c1ccc(Br)c(S(=O)(=O)NCc3ccns3)[nH]1)CC2 78815,Cc1ccc(S(=O)(=O)NC2CCCN3CCCCC23)cc1[N+](=O)[O-] 78816,C(C(=O)NN1CCCN(C)CC1)C1CC2N(C(=O)OC(C)(C)C)C(CCC2)C1 78817,N1(C(C2CC(C)(F)C2)=O)CCN(C(=O)C(C)(C)c2cc[nH]n2)CC2CCCCC12 78818,C1(NC(c2cn[nH]c2)=O)CCN(C(=O)CCN2CCC2)CCC1(F)F 78819,C1(CNC(=O)NC(c2noc(C3CCC3)n2)C)CCC(N2C(=O)CCC2=O)CC1 78820,N1(C(c2c(OC(C)C)cncc2)=O)CC2CC(NC(=O)C=C3CCC3)CC1C2 78821,CC(C)CCCC(=O)N1CC2(CNC(=O)C(O)CN3CCCC3)CC1CO2 78822,N1(C(C(C2CC2)OC)=O)CC=CCC1C(=O)NCCOCCC(C)C 78823,c1(C(=O)NC2C(CCC)CN(C(=O)C(c3ccccc3)F)C2)cc(C)cc(O)c1 78824,N1(C(C2C(=C)C2)=O)CCC2(COC(CNC(c3sc4cncn4c3C)=O)C2)C1 78825,c1(NCCCCCOC)ccc(S(=O)(=O)NCC2CCOCO2)c(Br)c1 78826,C1(C(C)NC(=O)NC2CCN(C(C)=O)C2C)CCC2CC1CO2 78827,N1(C(CCCC)=O)CCN(C(C2C(C)C2C)=O)CC1c1cc(F)cc(F)c1 78828,C1(C(=O)NCC(C(C)(C)C)(C)O)CC2(CCN(C(=O)CCc3cnco3)C2)C1 78829,Cc1oc(CNC(C2CCCC(F)C2)=O)nc1C(=O)NC1CSC1 78830,c1(C(=O)NCC2CC(NC(C3C(C)(CC)C3)=O)C2)cnc(C)n1C(F)F 78831,C1(CC=C)(C(N(CCN(C)C)CC)=O)CCN(C(c2cccn2C(C)C)=O)C1 78832,C1(NOCC)CN2CCC1(C)CC2.C1(C)C(=O)NCC=CC(=O)N1C.C.N 78833,c1(CCC)cccc(C(=O)N(C)CC2CCN(C(C34CC(C)C3C4)=O)C2)c1 78834,N1(C(CCC(=O)NC)=O)CCn2nc(CNC(=O)CCC3CCOC3)cc2C1 78835,c1(C(=O)NCCNC(C(C=C=C)C)=O)cc(Br)ccc1N1CCCC1 78836,c1(-c2nc(CC(C)(C)Oc3ccc(Cl)cn3)on2)ccccc1Cl 78837,N1(C(c2c(C)nccn2)=O)CCCCCCC1C(=O)NCC1CCCCCC1 78838,N1(C(C2(OCC)CCCC2)=O)CCC(C)(C(=O)NCCF)CC1 78839,c1(OCC)cnc(C(N2CCC(CC)(NC(=O)C(OC)OC)CC2)=O)c(Cl)c1 78840,C1(NC(C(C2CCC2)NC(C=CCC)=O)=O)CC(F)(F)C1(C)C 78841,C1(Nc2cc(O)cc(C(N)=O)c2Br)CNC(=O)CC12CCC2 78842,C1(C(=O)NC2CC(CC(=O)NCCC(=C)C)C2(C)C)CCCCC(=O)C1 78843,C(C(=O)NCCOCCCN(C)C(c1cnns1)=O)(C(C)C)OC 78844,N1(C(c2c(C)c[nH]n2)=O)CCN(C(c2ccnc(C3CC3)n2)=O)C2CCCCC12 78845,C(=O)(CC(C(F)(F)F)NC(=O)C(F)=CC1CC1)NC(CC)COC 78846,C12(CC(=O)NC(C3CCCN3C(=O)CC3CCNC3=O)C)COC(C)(C1)C2 78847,C(C1=CCN(C(c2ccc(C)nc2)=O)CC1)NC(c1c(CC)n(C)nc1)=O 78848,CC1CCCN(C(=O)CCCCCNC(N)=O)C1CNC(=O)Cc1cc[nH]c1 78849,n1(CC(CC)O)cc(C(=O)NCC#CCNC(=O)C(C2CCCC2)OC)nn1 78850,c1(C(=O)NCCCCNC(C2C3CCC2(c2cncs2)C3)=O)cccc(Cl)c1F 78851,CC(C)CCCCCC(=O)NCC(O)CNC(=O)C=CC1CCOC1 78852,CCC(C)(C)C(O)C(=O)NCC1(O)CCCN(C(=O)CN2CSCC2=O)CC1 78853,CCCCC(CC)CC(=O)NC1CN(C(c2c[nH]nc2CCC)=O)CC1N=[N+]=[N-] 78854,C=CCCC(CC(C)C)C(=O)N(CCCCCNC(C1CC12CC(C)(C)C2)=O)C 78855,N1(C(COCCCC#C)=O)CCC2(CCCCN(C(=O)C#CC(=O)N(C)C)C2)C1 78856,CC1CCN(C(=O)COC2CC=CC2)CC1NC(C1CCOCC1(C)C)=O 78857,C1(NC(CCc2c(C)ncs2)=O)(CO)CCN(C(C2CCC(=O)O2)=O)CC1 78858,C(c1ccccn1)=C(C)C(=O)NC1CC(CNC(C2(C#N)CC(=O)C2)=O)C1 78859,C(CO)(CCCCNC(=O)C(F)CC1CC1)NC(CCC)=O 78860,C1(CN(C(CC2(C=C)CC2)=O)C)CCN(C(=O)CC(=O)NC2CC2)C1 78861,CC1COC(C)CN1C(=O)CCN(C)C1CC1 78862,C1(C)(NCC)CCCN(C(=O)Cc2cccnc2Cl)C1.c1(CC)ccoc1C(=O)OC 78863,Cc1ccc(NC(=O)COCCCCCCNC(=O)C=CC(C)C)cc1O 78864,c1(NC(C(N2C(C(C)(C)O)CCCC2)=O)=O)coc(S(C)(=O)=O)c1 78865,C1(OC)CN(C(C2(Cn3ccc(C(=O)CC4CC4)n3)CCC2)=O)C(C)(COC)C1 78866,c1(CNC(C(C)CNC(C2CCN(C)C2)=O)=O)cnn(C)c1Cl 78867,c1(C(N(C(C(=O)Nc2cnnn2C2CC2)C2CC2)C)=O)cnn(CCF)c1 78868,n1(CC(=O)N(C(C2CCN(C(=O)CCc3nncs3)C2)C)C2CC2)cc(Br)c(=N)[nH]1 78869,c1(NC(=O)NCCCCCNC(CNC(=O)CN2CCCC2)=O)ccc(O)nn1 78870,c1(OC(C)(C)C)ccc(-c2ncn(CCCOC(=O)C(F)(F)F)n2)cc1 78871,Cc1nc[nH]c1C(=O)OC(C)(C)C.C12(CC(CO)C1)N1CC(CS(=O)(=O)NC2)C1 78872,c1(CCC(N2CC(NC(C(C(CC)O)(F)F)=O)C2)=O)ccc2cccnc2c1 78873,c1(C(=O)NCCC2CC(NC(C(C)NC(CC)=O)=O)C2)nnn2c1CCCC2 78874,C(=O)(C1=COCCC1)N1C(C2(NC(C3(C#C)CCC3)=O)CC2)CCCC1 78875,C1(C(=O)NCC2(CNC(c3c(C)cncc3)=O)CCCC2)CC2(C1)CC(C)(C)C2 78876,N1(C(=O)OC(C)(C)C)CC2(CCC2)CC1C(=O)N(C1COCCNC1=O)C1CC1 78877,C(=O)(CCCCCC#N)NC(C)C(C)(C)NC(c1cccc(SCC#N)c1)=O 78878,N1(C(c2ccc(C)nn2)=O)CC2CCCC1(CNC(=O)C(O)C1CCCC1)C2 78879,N1(C(C(C)(C)SC)=O)CCC2CN(C(=O)CCCc3ccc(Cl)cc3)CCC2C1 78880,c1(C(N2CC(CCCCNC(C(CCOC)OC)=O)C2)=O)ccc(Cl)c(F)c1 78881,C(CC(=O)NC(c1ccc(C)nc1)C)(C(F)(F)F)NC(C=CC(CC)C)=O 78882,CC(C)(CNC(=O)C(F)CC1CN(C(=O)CC(C2CC2)C2CC2)C1)C(F)(F)F 78883,CC(CCC(=O)NC1(CC(=O)N(C(C2(CCO)CC2)=O)C2CC2)CCC1)N(C)C 78884,C(N=c1[nH]c(=NCc2c[nH]nc2C2CC2)[nH]c2c1CCC2)C1CC(=O)N(C2CC2)C1 78885,N1(Cc2c(NC(C(CC)N(C)C)=O)cccc2Cl)C(=O)c2ccccc2C1=O 78886,C1(N(C(CCSCCC)=O)C)CCCCN(C(=O)CCC2CCCCO2)C1 78887,N1(CC(c2ccco2)C(=O)OC(=O)NC(C)(C)C)CC2CCCCC2C1 78888,C12(NC(C=NOC)=O)CCCC1N(C(c1cc(F)cc3c1CCC3)=O)CCC2 78889,C1(NC(C2CN(C(C)C)C2)=O)(CF)CCN(C(=O)COCCF)C1 78890,N1(C(c2csc(CO)n2)=O)CC2=C(C1)CN(C(C1(C(F)(F)F)CC3CC3C1)=O)C2 78891,CCCC(C)CC(=O)NC(C1CCN(C(c2c[nH]c(C(=O)OC)c2)=O)CC1)C 78892,c1(C(N2CCN(C(C3CCS3(=O)=O)=O)C3C2C3)=O)cc2nc(=O)ccn2[nH]1 78893,N1(C(C2CN(CC)C(=O)C2)=O)C2CCCC1CC(NC(c1csnc1C)=O)C2 78894,Cn1c(C(=O)NC2CCCC(CNC(C3CC4(CC4)C3)=O)C2)cnc1S 78895,c1(C(C)=O)ccc(C(N2CC(NC(=O)C(C)NC(C)(C)C)CC2C)=O)cc1C 78896,C(C(F)(F)C(=O)NCC1(C)CCCC1NC(=O)CC1COCCN1C)N(C)C 78897,C1(NC(c2cccc(CSC)c2)=O)CN(C(c2n[nH]c(C)n2)=O)CCC12CCC2 78898,c1(C(=O)NCC(C)N(C(=O)C(C)Cc2cnn(C)c2)C)cn2c(n1)COCC2 78899,c1(C(=O)NC(CNC(c2c(COC)nc(C)[nH]2)=O)CC)cc(N(C)C)nc(Cl)c1 78900,C=C(Cl)CC(C(=O)NC(c1ncccc1F)C)NC(c1nc(Cl)cs1)=O 78901,c1(C(=O)NC(C2CCOC2)CNC(c2c(CC)ncs2)=O)c(C)nnn1CC 78902,N1(C(CCOCCOC)=O)CCC2(NC(c3ccc(C(C)C)cc3C)=O)CC2C1 78903,CC(C)(CC(=O)NCC(CO)NC(=O)C(c1c(F)cccc1F)(F)F)C(F)F 78904,CC(C)(O)CC(=O)NCC(O)CCNC(C1CCCC(O)C1)=O 78905,N1(C(C2CCC(CNC(C3(COC)COC3)=O)O2)=O)CC(C#N)C1 78906,C1(NC(C(c2cccc(F)c2)C)=O)CC(NC(c2cc(C(N)=O)c[nH]2)=O)C(O)C1 78907,C1(NC(C2C(OCC)C2C)=O)CC(F)CN(C(=O)CCn2cc(C)cn2)C1 78908,N1(C(CCC(C)SC)=O)CCCC(NC(=O)C=Cc2cnn(C(C)(C)C)c2)CC1 78909,C1(CC)(CC)CC(NC(c2ccnc(OC(F)F)c2)=O)CN1C(=O)C(=O)N(C)C 78910,c1(OCc2cccc(OCC=C)c2)cccc2c1NC(C)CC(=O)N2 78911,c1(C(=O)NC2C(NC(c3c(N)c(Br)ccc3)=O)CCCC2)ccc2ncnn2c1 78912,C1(NC(C=CC(C)C)=O)CN(C(C2CC2C2CC2)=O)CC1c1cccc(F)c1 78913,Cn1cc(S(=O)(=O)NC2CC(CO)(CO)C3CC23)nn1 78914,c1(C(=O)NC(CC)CNC(=O)COCCC(C)C)ccc(O)nc1Cl 78915,C(CNC(=O)CSCCNC(=O)CC(C)Cn1cccn1)(C(C)(C)C)OC 78916,N1(C(C(C(=O)OC)(C)C)=O)CC2CC(NC(c3cn(C)c(C)cc3=O)=O)CC2C1 78917,N1(C(Cc2c(C)n(C)nc2)=O)CC(NC(=O)C=CC(C)C)CC(F)C1 78918,CON1CCC(C(=O)NCC2CCCCC2NC(c2cc(C(F)F)no2)=O)CC1 78919,CC1CC(=O)CCC1C(=O)NC1CC(C(=O)NC(C[N+](=O)[O-])C2CC2)C1 78920,N1(C(C2C(C)(C)COC2)=O)CC2(C1)CN(C(=O)CNC=O)Cc1ccccc1O2 78921,N1(C(C(CCC)Cl)=O)C2CCC(C2)C1C(N1CCC(C)(CO)C1)=O 78922,C(=O)(C(C(C)C)OC)NCC(CC)(C)NC(=O)CSCCN(C)C 78923,C1(NC(CC(C)C(F)F)=O)CC2CC(C1)N(C(c1ccc(N)cc1)=O)C2 78924,C(=O)(C#CC(=O)NCC1(CNC(c2c(Br)noc2C)=O)CC1)OC 78925,Cc1nccc(C(N2CCC(O)(C(C)NC(c3cc(Cl)n(C)n3)=O)CC2)=O)c1C 78926,c1(CNC(C)=O)cn(C2CC(C(=O)N(c3cscn3)C)C2)nn1 78927,CC1(CC(N2CC3CC3C2C(=O)NCC2C3COCC23)=O)CCCCC1 78928,Cc1nc(C)n(O)c1C(=O)NCC(CNC(=O)Cn1ccc([N+](=O)[O-])n1)CO 78929,N1(C(C(N2CCOC2=O)C)=O)C2CCC1CN(C(=O)C(c1cncn1C)=O)CC2 78930,C1(C(=O)NCC2(F)CCN(C(C(C=C)O)=O)C2)(OC)CCCCCC1 78931,C(=O)(CCC(F)(F)F)N1C(C)(CC(=O)NC(C(=O)OCCCC)C)CC1 78932,N1(C(C2CCN(C(CCC)=O)CC2)=O)CCCC2(NC(C3CCC3)=O)CC2C1 78933,C1(NC(c2ccc(Cl)c(F)c2)=O)CC2CC(C1)N(C(c1ccsn1)=O)C2 78934,CC1(C(=O)NCC2CCC(CNC(=O)COc3ccsc3)CC2)CC2C=CC1C2 78935,c1(C(=O)NCC2C(NC(COCCC)=O)CCC2)ccn2c1CCCC2 78936,C123CN(CC1CCO2)C3=O.c1(N(C(=O)CC2CC=CC2)C)cnc2nccn2c1 78937,c1(OCCCC)ccc(C(=O)NCCNC(=O)CC2CC(C)(C)C2)c(Cl)c1 78938,c1(SCC(=O)NCCCc2nc[nH]n2)ccccn1.C12CC1C(=O)NC2 78939,C1(C(=O)NC(c2ccc(F)cc2)CO)CC(O)CN1C(C1CC=CCO1)=O 78940,c1(C(C(=O)NCC(C)NC(C2(CC#C)CCCOC2)=O)OC)c(F)cccc1F 78941,CCC(C)CCC(=O)N(C)CC1(O)CCCN(C(=O)CSc2nncn2C)C1 78942,c1(C(N2C(C(C)(C)NC(=O)Cc3ccns3)CCC2)=O)cc(C(F)F)cc(Cl)c1 78943,Cc1cc(C(=O)NC2CCC(CNC(=O)Cn3cccc(O)c3=O)C2)cc(O)c1 78944,CC#CCCCC(=O)NCC(CNC(=O)CC(COC)COC)CO 78945,Cc1nn(C)c(N2CCN(C)CC2)c1CNC(=O)CC1CC12CC2 78946,C(=O)(C(O)CC(F)(F)F)NC(CC#C)C(=O)Nc1ccc(CC)cc1O 78947,c1(CNC(=O)C(O)C(C)(C)C)nc(CNC(C2CCC(C(N)=O)C2)=O)cc(O)n1 78948,C1(NC(c2ccnc(C3CC3)n2)=O)C2CC1N(C(C1CC3CCC1O3)=O)C2 78949,C1(C(N(CCCNC(=O)C2=CCCCC2)C2CC2)=O)CCCC2CCCN12 78950,c1(CCCC)cc(C(=O)NC2CCCCC2NC(c2n[nH]c(C)n2)=O)c(C)o1 78951,C1(COC)CN(C(=O)CCc2ccsc2)CCN1C(C1COC(=O)N1)=O 78952,N1(C(c2n(CC)nnc2)=O)CC(NC(=O)C2=CCCC(C)(C)C2)CC12CCOC2 78953,N1(C(c2c(O)ccc(C)c2)=O)CCCC(C)(C)C1CNC(c1ccoc1Cl)=O 78954,c1(C(=O)NCC2(C(C)NC(C3CCCC3)=O)CC2)ccc2c(=N)[nH]cnc2c1 78955,c1(C(C(N2CCC(N(C(=O)CC3CC3)CCO)C2)=O)O)ccc(Cl)c(Cl)c1 78956,c1(C(C)C(=O)NC2C3CCC2N(C(C2CCCO2)=O)C3)n[nH]c2c1CCCC2 78957,C12(C(=O)NCC3N(C(=O)CCCc4ncco4)CC(F)C3)CC1COC21CCC1 78958,c1(C(=O)NCc2c(C(=O)NC3CC(CSC)C3)ocn2)cccc(C(C)=O)c1 78959,Cc1c(C(=O)NC2CCCC2NC(c2ccn(C(F)F)n2)=O)ccn1C(C)C 78960,c1(C2(C(CCCCCn3cc(C4CCCC4)nn3)=O)CC2)ccc2c(c1)OCCO2 78961,c1(CC)cc(C(=O)NCc2cc(C(=O)NCC3CNC(=O)CO3)n(C)n2)nn1C 78962,c1(CC)c(C(=O)NCCCCN(C)C(C2C3CC3C3CC23)=O)oc2ccccc12 78963,C12(CCCC1C)C(=O)N2.Cc1cc(OCCCN(C)C(=O)C2CC2)no1 78964,C1(NC(c2cc(Cl)cc(F)c2F)=O)CN(C(C2(O)CCOC2)=O)CC2(CC2)C1 78965,c1(C(=O)NCC2CC(NC(C3N(CC)CCCC3)=O)C2)ccnc2c1nnn2C 78966,N1(C(CC(C)(C)N(C)C(C2CC(=O)CC(=O)C2)=O)=O)CC2(CCC(=O)N2)C1 78967,N1(C(C(CC)COC)=O)Cc2ccc(CNC(C3CCCC3)=O)cc2C1 78968,c1(C(=O)NCC2C3CN(C(C(CC(N)=O)O)=O)CC32)cccc2nc(O)[nH]c12 78969,Cc1ccc(O)cc1CN1CCCC(C)C1C.C12CCC(CC1)C(=O)NC2 78970,N1(C(CCSCC(N)=O)=O)C2CCCC1CC(CNC(C1CCC=CCC1)=O)C2 78971,C1(O)(C(=O)Nc2cnc(C(N)=O)cn2)CCCN(Cc2oc(C)c(C(=O)O)c2)C1 78972,C(C)(C)(CC(=O)NC1COCC1c1ccc(F)cc1)OC.C12CCCN(C1)C2=O 78973,N1(C(C(COCC)n2cc(COC)nn2)=O)CCCC(OC2CC2)C1 78974,C(=O)(C1=CCCOC1)N(C)CC1N(C(C2OCCN(C)C2)=O)CCOC1 78975,c1(OC(C)C(=O)NCCC(F)Cn2cc(C(C)(O)CCO)nn2)cccnc1 78976,c1(CCC)ncc(C(=O)NC)cn1.C1(C(C)C)CCNC(=O)C(=O)N1 78977,C12(C(=O)NC(C#C)C(C)OC)CCCC1CCN2C(c1cc(CCC)on1)=O 78978,c1(C(=O)NC2CN(C(CCC(=O)NC)=O)CC(O)C2)cccn2cnnc12 78979,C#CC1(C(N2CCC(CO)C(NC(=O)CCC3CC3(C)C)C2)=O)C=CCCC1 78980,O=[N+]([O-])c1cc(Cl)c(F)c(S(=O)(=O)NC(C(F)F)c2cccs2)c1 78981,CN1Cc2ccc(C(N3CCC(N(C(=O)CCCn4cccc4)C)C3)=O)cc2C1 78982,N1(C(C2N(C)CC2)=O)CCC(C(=O)NCC(c2ccco2)O)C1(C)C 78983,c1(COCC)cnoc1CNC(C1CCN1CC)=O 78984,N1(C(C(C=C)C)=O)CC2(C=C(C(=O)Nc3cccc(SC)c3)CO2)C1 78985,C12(CC3CN(CC(CC)C4CCC4)C3)C=CCN1C2=O.C1(C(=O)NC)CC(C)=NO1 78986,CC(C)(C(=O)NCC1(O)CCN(C(c2ccccc2O)=O)CC1)C(N)=O 78987,c1(CC(=O)NCC(C)N(C(C(C)SC)=O)C)c(C)nc(-c2ccccc2)nc1O 78988,N(C)(S(N)(=O)=O)CC(=O)NCC1N(C(CSCC#C)=O)CC1 78989,C(CC(C)C)(C(=O)NC1CC(C)CCC1O)NC(C(CC)COC)=O 78990,C(=O)(CCC(C)NC(=O)CCc1cnn(C)c1)N(CC(C1CC1)OC)C 78991,CC1OCCC1CC(=O)NC1CCC1C(=O)N(C)CCc1ccccc1 78992,C(=O)(CCCC(=O)NCC1CCCN1C(c1c[nH]c(C#N)c1)=O)N(C)C 78993,C1(CC)C(NC(=O)Cc2ccccc2O)CCCN1C(=O)Cc1cccs1 78994,c1(SCC(N2CCCC2Cn2cc(C(=O)O)cn2)=O)ccccc1Cl 78995,c1(CCC(N2CCC(O)(CCNC(C(CC)(C)O)=O)C2)=O)c(Cl)cncc1Cl 78996,C1(C(N2CCC(C(C)(C)NC(c3ccc(CN4CCCC4)o3)=O)C2)=O)CCOCC1 78997,C1(C(N2CC(CN(C(C(C)Oc3cccnc3)=O)C)C2)=O)CC2C(C1)C2(C)C 78998,c1(SC)nc(=N)[nH]c(=NC2CC3CC(C2)N(C(C2CCCC2CF)=O)C3)[nH]1 78999,C1(CNC(=O)Nc2cc(C)c(CN(C)C)cc2)CC2(C1)CC2S(C)(=O)=O 79000,C12(CC)CC(NC(C3(CCF)CC3)=O)(CN1C(=O)CNC(=O)C(F)(F)F)C2 79001,CC1=C(C(=O)NCCc2nn(C)cc2Cl)C(C)(C)CCC1 79002,c1(OCCC(=O)NCC(C(C)C)NC(c2cn(CCC)nc2)=O)cccc(F)c1 79003,N1(C(CCNC(=O)C=CCl)=O)CCC2(CC(NC(C3CCCCC3(F)F)=O)C2)C1 79004,C(=O)(CCC(C)(C)F)NC(C1CCN(C(=O)CCc2ccn(C)n2)C1)C 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79109,c1(C(N2CCN(C(C3C(CC)CCO3)=O)CC23CC3)=O)cc2c(O)ccc(F)c2[nH]1 79110,c1(CC=O)n[nH]c(=NC2CCC2)s1.C(c1ccco1)=C 79111,C1(C(=O)NCC2(F)CCN(C(C=C(C)Cl)=O)CC2)CC(C)(C)OC(C)(C)C1 79112,C1(C(N2CCC(NC(=O)Cn3nnc(C4CC4)n3)CC2)=O)OC2CCC1CC2 79113,c1(C(=O)OC)ccn(CC(=O)NCCN(CC(C)O)C(c2cnccn2)=O)n1 79114,N(C(=NCc1ccc(OC)cc1)NCC1(OC)CCCOC1)Cc1n(CC)cnc1 79115,c1(C(=O)NCC(CCOC)OC(C(C)NC(C)=O)=O)ccnc(C)c1N 79116,c1(C(N2C(CNCC)CCCC2)C(=O)NCCCSC)cc2c(cn1)OCCO2 79117,C=CCCCC(C(=O)NC(CF)C(F)(F)F)NC(=O)C(C)c1cc[nH]n1 79118,N1(C(C2N(CC)CCOC2)=O)CC(C)(C)CC1CNC(=O)CCP(C)(C)=O 79119,Cc1cc(C(=O)N(CCC(=O)NC(C2CCC(C)(C)O2)C)C(C)C)cn1C 79120,C1(C(=O)Nc2cc(O)n[nH]2)CCCC12CCN(Cc1cscn1)C2 79121,Cc1cc(=NC(CCO)C2CCSC2)[nH]c(=NCc2cccc(CO)c2)[nH]1 79122,C1(NC(C(CC)OC)=O)(CF)CCN(C(C2(n3cc(Br)cn3)CC2)=O)C1 79123,c1(C(=O)NC(CNC(c2c(SC)ccs2)=O)C2CCC2)ccc(F)c(C)c1F 79124,C=CC(C)(CC)C(=O)NC(C)CCC(=O)Nc1cnc(OC)c(C)c1 79125,n1(CC)ncc(Cl)c1C(=O)NCC1(COC)CN(C(C2CC(=O)N2)=O)C1 79126,C1(NC(CCSCC)=O)CCCCC1NC(c1ccc(C)nn1)=O 79127,Cc1c(CNC(=O)N(C)CC2CCN(S(C)(=O)=O)C2)cccc1O 79128,c1(C(=O)NCCCNC(C(CC2CCCCC2)OC)=O)c([N+](=O)[O-])c(C)nn1C 79129,n1(CC(=O)NCC(N(C(C(CSC)C)=O)C)C2CC2)nc(C(F)F)cc1C(F)F 79130,c1(C(=O)NC2C(C)CN(C(c3ccc(C(N)=O)s3)=O)C2)cccc(S(N)(=O)=O)c1 79131,c1(C(N2CCCC(NC(C3C=CCCC3)=O)C2)=O)c(F)cncc1Cl 79132,c1(C(N2C(C)C(NC(c3ccccc3C3(C)CC3)=O)CC2)=O)cc(=O)cc(Cl)[nH]1 79133,C=C(C)CCCC(=O)N(C1CCCN1C(=O)C(N1CCOCC1)C)CCO 79134,N1(C(C(C)OCCOC)=O)CC(CO)C2(C1)CN(C(=O)C(C)C(C)(F)F)C2 79135,N1(c2cc(NCc3cnc(N(C)C)cc3C)nc(C)n2)CC2CCCCC2(CO)C1 79136,c1(C(=O)N(CCOCCNC(=O)CC2CC3COCC23)C2CC2)cnn2ccsc12 79137,Cc1cc(C(N2CCC(CNC(=O)CN3CCCC3=O)C(C)C2)=O)c(N)c(Cl)c1 79138,c1(OC)cccc(NC(=O)COC(C)(C)CNC(c2nc(C)oc2C)=O)c1 79139,C(CC(O)C(=O)N(CC(C)(C)CNC(=O)CCC(C)OC)C)SC 79140,Cc1c(COCCOC(C)(C)C)ccoc1=NCS(=O)(=O)c1ccc(F)cc1Br 79141,C(=O)(CS(=O)C(F)(F)F)NCCCCN(C)C(c1cnc2[nH]cncc1-2)=O 79142,c1(C(N2CC(F)(CO)CC2)C)ccc(Br)cc1.c1(C2C(=O)N2)cccnc1 79143,N1(C(c2cccc(N(C)C)c2)=O)CCN(C(C2CC(C)(F)C2)=O)C2COCC12 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79248,c1(-c2nc(C(C)O)nn2Cc2cccs2)oc2ccccc2c1Cl 79249,C1(CNC(C(C)=O)=O)CCN(C(C2CC(n3ccnc3)C2)=O)C1 79250,c1(C(N2C(C(=O)Nc3cc(C)c(O)cn3)CCCC2)=O)cc(F)c(Cl)c(F)c1 79251,C1(NC(C(C)NC(C)=O)=O)CC2CCC1CN(C(=O)C(c1c(C)n[nH]c1C)C)C2 79252,C12(C(N3CC(O)(CCNC(c4ccc(C)c(C)n4)=O)C3)=O)CC3CC1C2C3(F)F 79253,c1(C2C(C(N3CCC(NC(c4cc(C)ns4)=O)C3)=O)C2)ccc(F)c(F)c1 79254,C1(F)(CNC(C(COC)O)=O)CCC(NC(C2(C)CC(F)(F)C2)=O)C1 79255,CCCC(CCCNC(c1cc[n+]([O-])cc1)=O)NC(C1CCCCO1)=O 79256,C(=O)(C(F)(F)C(F)(F)C(=O)O)N1C2(CCCN(C(=O)OC(C)(C)C)C2)CC1 79257,Cc1nc2ncnn2c(N2CCC(Oc3ccc(F)c(Cl)c3)C2)c1C#N 79258,C1(Cl)(C(=O)NCC#CCNC(c2c[nH]nc2C(F)F)=O)CC1(F)F 79259,CC(O)C(C)C(=O)N1CCCC(NCc2ccc(Cn3ccnc3)cc2)C1 79260,C1(CCNC(c2coc(C(F)F)c2)=O)COCCN1C(c1ccsn1)=O 79261,C=CC(C)(CC)C(=O)NC1CC(C)(C(N2CCC(C)(C(=O)NC)C2)=O)C1 79262,CCCC(C)(C(=O)OC)NC(=O)OC(C)(C)C.c12ccn(n1)CCN(C)C(=O)C2 79263,N1(C(c2cnc(O)[nH]2)=O)CC2CN(Cc3ccc(F)cc3-c3ccccc3)C2C1 79264,C1(C(N(CC(C2CC2)OC)C)=O)C=CCCN1C(c1nonc1N)=O 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79282,Cc1cc(Cl)ccc1OC(C)C(=O)NCC(F)CNC(C1(CC(F)(F)F)CC1)=O 79283,c1(C(N2CCC(N(c3ccn4nccc4n3)C)C2)=O)ccc2cccc(F)c2n1 79284,c1(SCC(=O)NC(c2ccccc2)CNC(C=C(COC)C)=O)ccc(C)cc1 79285,C1(C(C)C)NCC12CCN(C(c1ncccc1N)=O)CC2 79286,C(=O)(C1=CCC(NC(C2(C3CC4(CCC4)C3)CC2)=O)C1)NC1C(C)C1(C)C 79287,c1(CNC(C(CN(C(C2C(CC)CCC2)=O)C)C)=O)cc(C)cc(O)c1 79288,CCC(CC(=O)NCC(CN1CCN(C(=O)C(N)=O)CC1)OC)SC 79289,Cc1noc(C)c1CC(C)C(=O)NCC1CC(NC(c2[nH]nnc2C(F)F)=O)C1 79290,c1(C(=O)NC2(C)CN(C(C(C)NC(C)=O)=O)C2)cc2ccc(C)cn2c1 79291,Cc1cc(O)c(C(=O)NCCOCCCN(C(=O)C(CO)NC(N)=O)C)cc1F 79292,C1(CC)CCC(C(=O)NCC(C(=O)NCCC(=O)NC)N(C)C)O1 79293,S(=O)(=O)(c1ccc(Br)cc1[N+](=O)[O-])Nc1c(SCCC)ccc(Cl)c1 79294,C1(CNC(c2c(CCC)cccc2)=O)CC2(CC2)CN1C(C1CCC(C)O1)=O 79295,c1(C(=O)NC(CCCCNC(c2c(OC)cccn2)=O)C)cc2sc(C)cc2[nH]1 79296,C(=O)(C1=CCS(=O)(=O)C1)N1CC(NC(c2ccncn2)=O)C(CO)CC1 79297,c1(C(=O)NCC(C2(O)CCN(C(CSCC#C)=O)C2)C)c(F)cc(F)c(F)c1F 79298,C1(C(=O)NCc2cc(C(NOCCCOC)=O)ncc2)CN(C)CCN1C 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79349,c1(OC)ccc(C(N2CCCC2C2CCN(C(C3(N(C)C)CC3)=O)C2)=O)c(Cl)c1 79350,c1(C(=O)NC2C(NC(C(CC)F)=O)C2)cncc(-n2cccn2)n1 79351,C1(C(N2CCC(C(CNC(CN(C)CC)=O)(C)O)CC2)=O)CCn2ccnc2C1 79352,CCC(CC(=O)NC(C)CCCN)OC.c12cn(nn1)CCOC2 79353,C1(NC(c2c(CC)c[nH]n2)=O)CN(C(c2noc(C3CC3)c2C)=O)CCC12CCC2 79354,C1(O)(CNC(C(C)OC)=O)CCN(C(c2cnn(C(C)(C)C)c2)=O)C1 79355,N1(C(c2onc(CC)n2)=O)CCC2CCC(C1)N2C(c1cnoc1)=O 79356,CCCCC(O)C(=O)NCC(CC(=O)N1CCC(C(C)C#N)CC1)C1CCC1 79357,N1(CC)C(C)CN(C(=O)C(n2cc(CCOCP(C)(C)=O)nn2)C)CC1C 79358,N1(C(C2C(C(C)(C)C)C2)=O)CC2CCC(C1)N2C(c1nccn1C(=O)C1CC1)=O 79359,Cc1ccc(C(=O)NCCC(C)N(C)C(C2CCS(=O)(=O)N2)=O)c(Cl)c1 79360,c1(NCCCC2CCC3(C(CO)C3)CC2)nc(=NCc2nncs2)[nH]c2c1COC2 79361,CCCCCC(O)C(=O)N1C(CNC(=O)CCc2csc(C)n2)CC2CC12 79362,c1(N2CC2)cccc(S(C)(=O)=O)c1.C1(C)(CS(=O)(=O)N(C)C)CCOC1 79363,S(=O)(=O)(c1cc(F)cc(Br)c1)N1C(C(=O)Nc2cnsc2)CCC1 79364,O(C1CCCc2ccccc21)CC(=O)NC1CN(C(C2CCC2)=O)CC1CO 79365,c1(C(=O)NCC2(O)CN(C(COC3C(CC)CCCC3)=O)C2)ccc(O)cc1F 79366,C1(CNC(c2n(C)ccc2)=O)C(C2CC2)CCN1C(C1C(C)(C)C1(C)C)=O 79367,C(=O)(CC(O)CC(C)C)N1CC(CCC)N(C(=O)CSC2CCOC2=O)CC1 79368,c1(NC(C(c2cn(-c3ccc(OC)cc3)nn2)N2CCCC2)=O)ccc(Br)cc1Br 79369,C1(NC(CNC(C)=O)=O)CN(C(C2CC3(CCOCC3)CO2)=O)C2CCCCC12 79370,C1(CCNC(c2ccc(SC)s2)=O)CSCCN1C(c1coc(C(F)(F)F)n1)=O 79371,C(N=c1[nH]c2c(c(=NCc3cccc(C(F)F)c3)[nH]1)CCC2)c1c(CC)nns1 79372,C(CCN=c1[nH]c2c(c(=NCCOCCCF)[nH]1)CSC2)c1n[nH]c(=N)o1 79373,C#CC1(C(N2CCN(C)C(C)C2)=O)CCN(C(=O)OC(C)(C)C)C1 79374,C1(NC(CN(c2ccncc2)C)=O)CN(C(C2CCOC2C2CC2)=O)CC12CC2 79375,CCC(CC)C(F)C(=O)NCC(CNC(c1cccc2ccoc12)=O)C(F)(F)F 79376,C1(N(C(COCC(C)C)=O)C(C)(C)C2CCC2)CN(C(=O)CC2CC2)C1 79377,CCC(CNC(=O)C(O)CCCNC(C1CCC(=O)CC1)=O)(CC)C(N)=O 79378,CCCCC(CC(=O)N1CCC(F)C(O)C1)NC(C1CC2(CCC2O)C1)=O 79379,c1(C(=O)NCC2(F)CN(C(C3(C)CCOC3)=O)C2)cc2scnc2[nH]1 79380,c1(C(N(C(C)C)CCNC(c2cnn(C3CC3)c2Cl)=O)=O)cc(F)c(F)cc1Cl 79381,C1(C(C)NC(c2c(CC)ocn2)=O)CCCCN1C(c1ccn(C(F)F)n1)=O 79382,C1(NC(c2nc(C)oc2)=O)COC2(C1)CN(C(=O)CC1CCOC1=O)C2 79383,N1(CC(=O)NCC(CNC(C2C(CC)OCC2)=O)F)CCC(C)(C)CC1 79384,C(=O)(CC(F)(F)F)NC(C)C(=O)N(CC(O)CN(C(=O)CCc1ncco1)C)C 79385,CN1CCC(CC(=O)N2CCN(C(=O)C(N)=O)CC23CC3)c2ccccc21 79386,c1(C23CC(C(N(C)CCNC(C4CCN4C4CCCC4)=O)=O)(C2)C3)ccc(F)cc1 79387,C1(F)(CNC(c2cnc(S)[nH]2)=O)CCC(CNC(=O)C(O)C2CCC2)CC1 79388,C(CCF)(C(=O)N1CC(F)(CF)C1)NC(CN1C(C)CCC1)=O 79389,c1(OC)cc(N)c(C(N2CCCC(O)(CNC(c3ccc(Cl)s3)=O)C2)=O)c(F)c1 79390,c1(NC(C)C)ccc(C2(CNC(=O)NC3C(C)CC3C)CCC2)cc1 79391,c1(C(=O)NC(C2CCCC2)CNC(CCSCC(N)=O)=O)cc2cccnc2[nH]1 79392,C1(C(=O)NCCC2CCN(C(C=CC(=O)OCC)=O)C2)CC(=O)N(CCC(C)C)C1 79393,C(c1ccc(C(F)F)o1)=CC(=O)NCCC(C)NC(c1cc(Cl)c[nH]1)=O 79394,C1(NC(c2c(C)ncn2O)=O)CCOC2(CCN(C(c3cnc(O)s3)=O)CC2)C1 79395,C=CCCC(C(=O)N1CCCC(CCOC)C1)NC(C1(O)CCCC1)=O 79396,c1(CNC(C2CCSC2)=O)ccc2c(c1)CN(C(C1CCCC(CF)C1)=O)C2 79397,C=CCC(C)(C(=O)N1CC2(C1)CN(C(C1(OC)CCCC1)=O)C2)N(C)C 79398,C(=O)(CC(C)(C(F)(F)F)N(C)C)N(C)Cc1cc(N)cc(S(C)(=O)=O)c1 79399,c1(CC(C(=O)NC(c2ccc(F)cc2)CC)N)c[nH]c2cc(Cl)ccc12 79400,O=S(=O)(c1cccnc1NC1(CN2CCN(C3CCOC3)CC2)CC1)NCCO 79401,c1(C(c2n(C)nnn2)NCC2CC(F)C2)cncc(C(F)(F)F)c1 79402,c1(CC(=O)NCC2CC(O)(CNC(CC=C=C)=O)C2)c(OC)cccc1Cl 79403,N1(C(C)=O)CC(C(N2CC(C(F)CNC(=O)CC3(C(=O)N(C)C)COC3)C2)=O)C1 79404,C(C(CC(=O)N(C1CC(F)(F)C1)C)NC(C1CCC(=O)CC1)=O)OC 79405,N(C1CN(C(=O)CC2CC3CC3C2)CCc2ccccc21)C(C=CC)=O 79406,c1(OCC)ccc(COC)cc1-c1c(CN2CC(C)OC(C)C2)ccnc1F 79407,c1(C(=O)NC2(CN(C(C(CC)N3CCOCC3)=O)C)CC2)cccc2ncoc12 79408,C12(NC(CCOCC#C)=O)CCCC1N(C(c1cc(SC)ccc1C)=O)CCC2 79409,C1(CCN2CCC(NC(CNC(CN(C)C(N)=O)=O)=O)C2)COCC1C1CC1 79410,c1cn(C)c(=O)c2ccccc12.CN1C(=O)CCCN(N2CCC3(C)OCC23)C(N)C1=O 79411,c1(CC2(C(=O)NC3(CC(N4CC(CCCCC)C4)=O)CCC3)CC2)nccn1C 79412,C1(CC)(C(=O)NC(C2CC2C(N)=O)C)CCN(C(=O)C(C)n2cnnn2)C1 79413,C1(OC)CC(C(=O)N(CCCNC(C2CCC2(F)F)=O)CCO)CC1NC(C)C 79414,C1(CCNC(=O)Cc2cccc(O)c2)(NC(=O)CC2CCC3CC23)CCOCC1 79415,CCC(C)C(C(=O)N1CCCCC1c1nccs1)n1ccc(-c2cn(CC)nn2)n1 79416,c1(C(N(C2(CC(=O)N(CCC(N)=O)CC)CC2)C)=O)cnc(C2CC2)o1 79417,C1(NC(C2CNC(=O)N2)=O)C2CC1N(C(C13CCCCC1C3)=O)C2 79418,C(=O)(C(C)CC(C)(C)C)NC(CC)CN(C)C(C1CC(N2CCCC2)C1)=O 79419,c1(C(C)NC(C2C(c3ccc(C(=O)OC)cc3)C2)=O)ccc(F)cc1Cl 79420,N1(C(C(CCC)NC(c2ccc(C#C)cc2)=O)=O)CC(C)(C)CCC1C 79421,C1(C(N(C(C)CNC(=O)Cc2cn(C3CCC3)nn2)CC)=O)CCC2(CCC2)O1 79422,C12(C(=O)NCC3N(C(CC4C(CC)C4)=O)CC(F)C3)CCCN(CCC1)C2 79423,C1(NC(C2CC(=O)NC2)=O)CCCCN(C(c2cccnc2C2CC2)=O)C1 79424,Cc1ccncc1C(C)NC(c1nc(CNC(c2cc(C)c(C)[nH]2)=O)oc1C)=O 79425,N12CCC(C(F)(F)CC1)C2.CCCCNC(=O)CNS(C)(=O)=O 79426,C(=O)(C1CCCc2sccc21)N1C2C(NC(C3C(CCC)CCC3)=O)C(C2)C1 79427,C(=O)(C1=Cc2ccccc2C1)N(CCOCCCN(C(CCC(C)SC)=O)C)C 79428,c1(OC)ccc(Cl)c2[nH]c(C(=O)NC3(CNC(=O)C(C)N4CCC4)CCC3)cc12 79429,Cc1n[nH]cc1C(=O)NCCCCC1CN(C(=O)C(c2cc(C(N)=O)c[nH]2)=O)C1 79430,C1(C(=O)NC2CCN(C(C(CN(C)C)(C)C)=O)C2)CC2CCC(C1)N2C 79431,c1(CN2CCC(NC(c3n(C(C)C)ncc3)=O)C(F)C2)cc(F)ccc1[N+](=O)[O-] 79432,c1(CC(=O)N(CCCCN(C(c2ccc(CC)[nH]2)=O)C)C)cccc2nsnc12 79433,c1(C(=O)NC(CC)CN(C(c2cnco2)=O)CC)ccc(Br)c(C)n1 79434,C1(NC(C(C)(C)n2cc(Cl)cn2)=O)CCC(O)CN(C(c2ccc(Cl)o2)=O)C1 79435,C1(S(N)(=O)=O)(C(c2nnnn2C(C)(C)CC)NCc2c(CC)cnn2C)CCC1 79436,C(=O)(C(C(=O)NCC1CCN1C(=O)Cc1cc(Cl)cnc1C)C(C)(C)C)OCC 79437,Cc1cccc2[nH]cc(C(=O)NCC(CC(C)C)NC(C3CCC(=O)N3C)=O)c12 79438,c1(C(=O)NCC(=C)CCNC(c2cc(-c3cccs3)on2)=O)c(C)ncn1O 79439,c1(CC)nc(C(=O)N(CC(CC)NC(=O)CCc2cc(OC)no2)C)c(C)o1 79440,N1(C(c2c(CC)nc[nH]2)=O)CCN(C(c2cc(C)on2)=O)C2(CC2)C1 79441,C1(NC(=O)Nc2cc(C(C)C)sn2)CS(=O)(=O)CC1C(=O)OC(C)(C)C 79442,C(=O)(CCC(C)(C)F)NC(c1ccc(OC)cc1)CNC(C1CC(COC)C1)=O 79443,N1(C(C(C)(C)OCC)=O)CC2(CC(NC(c3ccc(CO)nc3)=O)CO2)C1 79444,c1(C(=O)NC2(C)CN(C(c3ccnc(C)n3)=O)C2)ccc2ncn(C(C)C)c2c1 79445,C1(CN(C)C(C2(C)CC3CC3C2)=O)CCCN(C(=O)C2=COCC2)C1 79446,Cc1cc(CNc2ccc(NC(C3CC3C)=O)c(F)c2)cc(O)c1 79447,c1(C(=O)Nc2ncc(C)cc2Cl)n[nH]c2c1CN(C(=O)CCCCBr)C2 79448,CCC(CC(=O)N1CC2(CC(NC(C3CCCCCC(=O)C3)=O)C2)C1)C(F)F 79449,N1(C(C(CC)(C)O)=O)CCC(C2CCN(C(c3cc(C)cc(C)c3N)=O)C2)CC1 79450,N1(CCC)CC(C(=O)N(CCCCN(C(=O)CC2CC2(Cl)Cl)C)C)CC1=O 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79521,C1(C(=O)NCC(N2CCC(CNC(=O)OC)C2)=O)CCC=CCCC1 79522,C1(NC(C(C)NC(c2ccc(C3CC3)nn2)=O)=O)C2CCCOC12 79523,C1(N)CCCC(SC)C1.CCC(C)(C)OC.C1C(=O)NC2(CC2)C(=O)NO1 79524,Nc1ccnc(C(=O)NC(CNC(c2cc(C(F)(F)F)on2)=O)C2CC2)c1 79525,C=C(C)CCCN=c1c(Br)ccc(S(=O)(=O)N2CCC3CCCCC3C2)[nH]1 79526,C1(C(N(C2CCCCN(C(=O)CC(C)(C)O)C2)C)=O)CCC(=C(F)F)CC1 79527,C1(NC(C2C(CNC(c3c(CC)oc(C)c3)=O)CCC2)=O)CC2CC1C(O)C2O 79528,C1(CNC(C(CCCC)O)=O)CCC12CCN(C(c1cnc(C)[nH]1)=O)CC2 79529,N1(C(C=CC2N(C)CCC2)=O)CCN(C(c2cc[nH]c(=N)c2)=O)CC1CC(F)F 79530,C1(C(=O)NCC(CN(c2ccccc2)C(C=C(COC)C)=O)C)CC1C1CC1 79531,C1(NC(CC(C)N2CCCC2=O)=O)CN(C(c2cn(C)nc2O)=O)CCC12CCC2 79532,CC1CN(C(C2(C(C)(C)C)CCCC2)=O)CCC1NC(c1cn(C)c(=O)n1C)=O 79533,C1(CC=C)(C(=O)NCCC2CN(C(C3CC3c3ccoc3)=O)C2)CCC1 79534,CCC(O)C(C)C(=O)N(CC)CC1CCN(C(=O)CC2C(COC)C2(F)F)CC1 79535,C1(NC(c2ccc(F)c(Br)c2)=O)CC2CC1N(C(c1ccc(C3CC3)o1)=O)C2 79536,CC(O)C(C(=O)NCCC1CCCN(C(c2csc(Cl)n2)=O)C1)N(C)C 79537,Cc1ccc2c(=NC3CCOCC3)[nH]c(=NCc3nnc4ccccn34)[nH]c2c1 79538,c1(CC)ncc(C(=O)NC2CCC(NC(=O)CSc3nncn3C(C)(C)C)C2)s1 79539,C(=O)(C#CC1CCOC1)N1CC(NC(c2c(C)nc(-c3cnn(C)c3)s2)=O)C1 79540,C12(CNC(=O)CC3CCC(=O)N3)CC1CN(C(c1cccnc1-n1nccn1)=O)C2 79541,c1(OC)ccc(F)c(CNC2CCC(NC(=O)CCc3nc(Br)ccc3Br)C2)c1F 79542,c1(C(=O)NCCN(C(c2ccc(N)cn2)=O)CC)ccc2c(C)[nH]nc2c1 79543,C1(C(N(C)CC2(O)CCN(C(Cn3c(C)csc3=O)=O)C2)=O)C2CCC(F)(F)C12 79544,c1(C(=O)NC2CC(C(N3CC(O)(C(N)=O)C3)=O)OCC2)cc(O)cc(Br)c1 79545,CC1COc2ccc(C(=O)NC3CCC3NC(=O)CCCc3ccsc3)cc21 79546,c1(C(CNC(C2(NC(C)=O)CC2)=O)NC(C2(C(=O)OC)CCC2)=O)cc([N+](=O)[O-])c[nH]1 79547,C1(CNC(C2C(=C)C2)=O)(CC)CN(C(=O)C(C)C2CCCC2)C1 79548,C1(CC(N2CC(NC(CC=C=C)=O)C(F)C2)=O)OC(C)(C)OC1=O 79549,C(=O)(C(C)C(O)CC(C)C)NCC1(CC(C)C)CC1.C12CC(C1)NC2=O 79550,C(=O)(C(CC)(CC)CC)NCC1COCCN(C(c2cn(CCOC)nn2)=O)C1 79551,C1(C(=O)NC(CNC(CNS(CCCOC)(=O)=O)=O)CC)CC2(C1)CC21CCC1 79552,C1(CC=C)(NC(=O)CC2CCCC2C)CCCN(C(c2cc(O)ccc2O)=O)C1 79553,n1(CCNC(C2CC(CNC(=O)C(C3CC3)C3CC3)C2)=O)cc(CO)nn1.C1CC1 79554,C1(CCC)COCCN1C(=O)C(=O)NCC1(SC)CCC1 79555,C1(NC(c2nccs2)=O)CN(C(C2CN3CCC2CC3)=O)CC12CCCC2 79556,C1(CC(=O)OC)CN(C(=O)NC2CCNC(=O)CC2)CC(C(F)(F)F)O1 79557,C1(C(C(=O)C(F)(F)F)=O)COC(=O)N1C.C(=O)(C(CO)N)N(C1CCN(CC)C1)C 79558,C1(N2CCC(NC(=O)C3=NOCC3)C2)CC12CCOCC2 79559,N1(C(C(C)OC2CCOC2)=O)CCCC12CCN(C(=O)CCc1cnoc1)C2 79560,C1(NC(Cc2ccc(C)nc2)=O)CC2CC(C1)N(C(=O)CCc1cccs1)C2 79561,c1(CCNC(=O)NC(CC=C)CC=C)noc2c1CCC2 79562,C1(NC(C(CN(C)C)(F)F)=O)CCC2(CCCN(C(=O)CSS(C)(=O)=O)C2)C1 79563,N1(C(CCC)=O)CCN(C(=O)C=CC2CCC2)C(C)CC1C 79564,Cc1snnc1C(N1CC(C(C(=O)NCCN2CCC(OC)C2)OC)C1)=O 79565,C1(CNC(c2cccc(C3CC3)c2)=O)COCCN1C(C1CC1C1CCCO1)=O 79566,c1(C(=O)NCC(CCCC)O)cc2[nH]nnc2cc1OC 79567,C1(C(N(C(CCSC)C)C)=O)CC(=O)CN1C(c1cc(C)[nH]c1C)=O 79568,N1(C(CN2CC(C)C2)=O)CCCC(n2cc(CNC(C3CC3(Cl)Cl)=O)nn2)C1 79569,CCCCCCC(O)CCC(=O)NC1(C)CCCN(C(C2OCCC2C)=O)C1 79570,N1(C(C2NC(=O)OC2)=O)CC2CN(C(c3cc4n(n3)CCCN4)=O)CC2C1 79571,C(=O)(C1SCc2cccnc21)N1CCCC(N(C(c2cncc(C)n2)=O)C)C1 79572,C1(CN(C(=O)C(C)C2CCC2)CC)CCN(CC(c2ccccc2Cl)OC)CC1 79573,CN=c1ccc(C(=O)NCCCN(CCO)C(c2csc(CO)n2)=O)c[nH]1 79574,C(=O)(C(C)S(=O)(=O)N1CCOCC1C1CC(F)(F)C1)OC 79575,N1(C(C(CCO)N(C)C)=O)CC(C2CCN(C(C3CC3(C)C)=O)CC2)C1 79576,N(C(=NCc1ccc(OCC(F)(F)F)cn1)N(C)Cc1nc(Cl)ccc1Br)CC 79577,CC1(NC(c2cc(-c3ccoc3)[nH]n2)=O)CCCN(C(=O)CC2CCC(=O)N2)C1 79578,CCS(=O)(=O)CC(=O)NCC1C(C(=O)Nc2ccc(O)c(C(N)=O)c2)C1(C)C 79579,Cc1cnc(N2CC=CC(NC(C3CCCC3(C)C)=O)C2)nc1O 79580,c1(C(=O)NC2CN(Cc3ccc(Br)nc3)CC2F)ccnc(Cl)c1Cl 79581,c1(CC(=O)NCC(CC=C)NC(=O)Cc2cc(C)cc(C)c2)cc(OC)ccc1Cl 79582,C(=O)(C1=CCCS1)N1CCC(CNC(C(C)NC(=O)C2CC2)=O)C1 79583,c1(C(=O)NCCCNC(C(c2c(C)cccc2)(C)C)=O)c(C)cc(O)nc1C 79584,Cc1cc(F)ccc1CN(C(c1csc(C#N)c1)C(=O)NCCCF)C 79585,N1(C(CNC(=O)OCC=C)=O)CCC(NC(=O)CC(C)(C)CC)C(C)C1 79586,C1(NC(COCCOC)=O)CCCC1SCCCCNC(C1CS(=O)(=O)C1)=O 79587,C1(C(N(C)CC2CN(C(c3cc(Cl)ccc3F)=O)C2)=O)Cc2ccccc2N1 79588,c1(C(N2C(C(=O)NC3C(CC=C)COC3)C3CC3C2)=O)ccc(C#N)cn1 79589,C12(CNC(Cc3cccc(C)c3F)=O)CCCC(CN1C(=O)C(F)F)C2 79590,C(=O)(C(F)CCC(C)C)N1CCN(C(CCCC#C)=O)C(CCO)C1 79591,C=CC1(CC(N2CC(C)(CCC(=O)NC3CCC4CC34)C2)=O)CCCC1 79592,C1(CNC(=O)Nc2cc(C)nn2C2CC2)CCCN(C(=O)OC(C)(C)C)CC1 79593,c1(C(N2C(=O)C(C)C(=O)NCC2C)=O)ccc2nccn2n1.c1(CC)nccs1 79594,c1(C(=O)NCCOC2CN(C(C3C(C)(C)CO3)=O)C2)c[nH]c2c(C#N)cccc12 79595,C(=O)(C(C(C)C)NC(=O)CC(C)C)NC1CC(F)(CNC(CC(OC)OCC)=O)C1 79596,NC(=NCCF)NCC(c1cccs1)O.C1(C2(C)CC2)CCOC1 79597,c1(C(=O)NC2C(C)CN(C(C3CCC(C)O3)=O)C2)cc2cccc(Br)c2[nH]1 79598,C1(C)(CC)C=C(C(=O)N2CCN(C3CCCN(C(=O)C(O)C(C)(C)C)C3)CC2)C1 79599,C1(OCCOC)CC(CF)N(C(c2cnc(C)s2)C(=O)NC2CCCC2)C1 79600,Cc1ncncc1C(=O)NC1CN(C(c2occc2CN(C)C)=O)CC1F 79601,C(CC1=CCN(C(C2CC23CC(C)(C)C3)=O)CC1)NC(CCCC(=C)C)=O 79602,N1(C(C=C)=O)C2CCC1C(C)C(NC(=O)C(COC)N=[N+]=[N-])C2 79603,c1(-c2cccc(C(C)O)c2)ccc2cc(NC(C3COC(C)(C)OC3)=O)[nH]c2c1 79604,c1(C(=O)NC2CCC(C(=O)NC(c3ccnn3C)C)CC2)cccn(C)c1=O 79605,CCC(CC)C(C(=O)N1CCCC1C(C)NC(c1ccoc1)=O)OC 79606,C1(N(C(C(F)=CCC)=O)CC)CCCC(NC(c2ccn(C(C)(C)C)c2)=O)C1 79607,n1(CC)cc(NC(c2ccn(C)c2)c2nnnn2C)cn1 79608,c1(N(CC(=O)NC2CCCC2CNC(=O)Cc2cc[nH]n2)C)cccc(F)c1F 79609,c1(OC)ccncc1CNC(=O)CC(C)(C)OC.C12CC(C3CC3)N1C2=O 79610,C1(C(C(C)NC(=O)CSc2nc[nH]n2)NC(=O)COC2CC2)CCCCC1 79611,CC1(C)CN(C(C2(Cl)CC23CCC3)=O)C(CNC(c2csc(C3CC3)n2)=O)CO1 79612,C(C(CO)(CO)NC(c1cc(C(C)(C)C)c[nH]1)=O)N(C(c1nc(SC)sc1)=O)C 79613,C12(C(=O)NCC3C4CN(C(c5nncs5)=O)CC43)CC3CC(C1)CC(F)(C3)C2 79614,N1(C(C=CC(C)(C)C2CC2)=O)CCC(C(=O)N2CC(CS(C)=O)C2)=C(F)C1 79615,N12CC3CCC3(C1)CC=CC2=O.C(=O)(C(C)(C)SC)NC(c1noc(C)n1)CC 79616,N1(C(=O)C=Cc2ccncn2)CCN(C(C2(O)CC2)=O)CC(O)C1 79617,C(=O)(CCCCCCCCC1CC1)NC1CC(Cn2cc(C(C)OCC)nn2)C1 79618,C1(C(NOCCCCC)=O)CC(C)CN1C(=O)C(=O)NOC 79619,C(C(O)CC(=O)NCCC1(C)CCN(C(C2(CCCC#N)CCC2)=O)C1)SC 79620,C(=O)(C(C)(C)C(F)(F)F)N1CCCCC(CNC(C=CC=CCCCCC)=O)C1 79621,C1(NC(CSCC)=O)CN(C(c2ccn(C3CC3)n2)=O)CCC12CCOCC2 79622,C(=O)(C1=CS(=O)CCC1)N1CCC(NC(c2cn(C(F)(F)CO)nn2)=O)C1 79623,N1(C(c2c(CC)con2)=O)CC(CCNC(c2cc(C(=O)OC)c[nH]2)=O)OC(C)C1 79624,C12(NC(C3CCC(=O)N3)=O)CCCC1N(C(C1CC(F)(CO)C1)=O)CCC2 79625,C(=O)(C1CCc2cc(Br)ccc21)c1ccc(C2CCCN(C)C2)cc1 79626,C1(CNC(c2ccc(CSCCC)o2)=O)CCCN(C(=O)CN2CCCC2)C1 79627,c1(C(N2C(n3cc(C(CCC)CC)nn3)CCC2)=O)ccc(=N)[nH]n1 79628,c1(CNC(c2csc(C)c2C)c2n(CC)nnn2)cccc(F)c1 79629,Cc1cc(C(N2CCC3(CC3C(=O)Nc3cc(Cl)cc(I)c3)C2)=O)ccc1O 79630,C(C(=O)NN1CCCC1C(N1CCCC1)=O)N.N1(C(C)=O)C(C)CCC1C 79631,C(=O)(C1CCCc2ccccc21)NC(C1N(C(Cc2cnc(C)[nH]2)=O)CCC1)C 79632,c1(C(N2CC(O)(C(C)NC(C3CCCN3C)=O)C2)=O)ccccc1Br 79633,C1(NC(c2cc(C3CC3)ncn2)=O)CCN(c2ncnc(O)c2Br)CCC1CO 79634,c1(OCC(=O)NC2C(NC(c3c(CC)non3)=O)C2)ccc(Cl)cc1[N+](=O)[O-] 79635,Cc1cc(C(=O)N(CCC(C)NC(c2ccc[n+]([O-])c2)=O)C)ccc1F 79636,N1(C(c2cncc(CNC(C(CC=CC)C)=O)c2)=O)CCCC(C)(N(C)C)C1 79637,c1(OC)cc(Br)c(C(=O)NC2CC2CNC(=O)CC(F)F)cc1F 79638,N1(C(c2ccn3cncc3c2)=O)CCCC2(CCCN2C(=O)C2=NOCC2)C1 79639,C1(NC(c2c(C)[nH]cc2)=O)CCN(C(C2CC3CCC2C3)=O)C(C)C1 79640,c1(C(=O)NCCCC(C)NC(C2(OC)CCOC2)=O)cccc2cc(F)ccc12 79641,N1(C(C(CC)Oc2cccc(C)c2)=O)CC(F)CC1CNC(c1nc(Cl)cs1)=O 79642,CC(C)C(C)(C)C(=O)NCC(C)(C)NC(C1CCC(O)CN1C)=O 79643,c1(CC(=O)NC2(CNC(=O)C(O)Cn3cncn3)CC2)ccccc1F 79644,CC1CC(C)(C(N2CC(Cn3cc(CC4CCNC4=O)nn3)C2)=O)C1 79645,c1(SCC(N2CCCC(NC(=O)Cc3nc(O)n[nH]3)C2)=O)nc2ccccc2[nH]1 79646,c1(CC(N2CCC(C(C)(C)NC(=O)CSc3cccs3)C2)=O)cnncc1O 79647,C1(C(=O)NCC(CNC(c2ccn(CCN(C)C)n2)=O)O)CC2C=CCC(C1)C2 79648,Cn1nc(Br)c2c(NC3CC(=C4CC4)C3)ncnc12 79649,c1(C(=O)NC)ncccc1NC(=O)NC1CCN(CCF)C1=O 79650,N1(C(=O)NCC(C2CC(F)(F)C2)OC)CCC2(CC1)OCCO2 79651,N1(C(Cc2onc(CC)n2)=O)CC2(C1)C(NC(=O)CC(C)C(F)F)CCS2(=O)=O 79652,c1(NC(C(=O)NC(CC=C)C)=O)ccc(OC)c(CC)c1 79653,n1(CCC)c(N)c(C(=O)CN(C(=O)Cc2c(C)noc2C)C2CC2)c(O)nc1=O 79654,c1(C(N2C(C)(CC(=O)NCCCc3cc(C)no3)CC2)=O)cc2ccncc2[nH]1 79655,O=C(C1=CC2CCC(C1)C2)N1CCC2(CC1)CC2C(=O)NCc1ncccc1F 79656,c1(C(=O)NCC2(C)N(C(CC(C=C)(C)O)=O)CCC2)cccc([N+](=O)[O-])c1 79657,CC(O)C(C(=O)N1CCC(O)CC1)N(C)C1CC1.C(CCN)NC(=O)OC(C)(C)C 79658,C1(NC(c2cc(CNC(=O)COC3CCC3)ncc2)=O)CC2C(C1)C2(F)F 79659,C1(C(N2CC(CC)C(NC(=O)COCCOC)C2)=O)CC2C(C1)C2(C)C 79660,O=S(=O)(c1cccnc1NC(Cc1ccco1)CO)NCCN1CCCS1(=O)=O 79661,c1(SCC(=O)NC(CCNC(C(CC)F)=O)C)ccc(F)c(F)c1 79662,Cc1ccc2c(C(N3CCC(N(C)C(c4c[nH]nc4[N+](=O)[O-])=O)C3)=O)n[nH]c2c1 79663,N1(C(C2N(C)C(=O)C(F)C2)=O)CCS(=O)(=O)CC1C1CC1 79664,c1(OC)ccccc1C1(Cc2ncc(Br)cn2)CC1.c12n[nH]cc1NC2=O 79665,C1(NC(C(C=C)(C)O)=O)CCCCC12CCN(C(=O)C1=CCSC1)CC2 79666,Cc1nc2ncnn2c(C)c1CC(=O)NC1CC2CC1N(C(=O)C(C#N)C1CC1)C2 79667,C(c1cccc(Cl)c1)=CC(N1CCC(N(C(=O)C(C)O)CCC)C1)=O 79668,N1(c2nc(C(=O)OC)c(C)s2)CCC(C)(NC(=O)CCN2CCC(F)C2)CC1 79669,c1(N2C3CC(CNC(C4CCSC4)=O)CC2CC3)nc2ccc(Br)cc2s1 79670,CCN=C(NCc1ccc(C#N)cc1Br)N1CCCC1 79671,C(C(=O)N(C1CCCCC1C)C1CC1)(C(C)(C)O)NC(c1ccc(OC)s1)=O 79672,C1(C(N2CCN(C(C(C)NC=O)=O)C(CC(F)F)C2)=O)CCCC2(CCC2)C1 79673,N1(C(c2n(C)ncc2Cl)=O)CCCCC2C1CCCN2C(=O)CC1CNC(=O)C1 79674,O=NN1CCCCC1C(N1C2CCC1(CNC(=O)CC1CC1)CC2)=O 79675,n1(CC)nc(C)c(C(N2CCCC(NC(=O)CC3(C#N)CCC3)C2)=O)c1Cl 79676,c1(NC(c2nc(COC)sc2)C)nccc(=NCc2c(C)coc2C)[nH]1 79677,c1(C(=O)NCC(CO)NC(C(CC)OC)=O)ccc(N2CCOCC2)cc1 79678,Cc1c(NC(C)C(=O)OCCSC(C)C)c(-c2ccccc2)nn1CC(=O)O 79679,C#Cc1ccc(C(=O)NC(CC(C)C)C(=O)NCC2CC2C(=O)OC)nc1 79680,N1(C(CC2CC(=O)C2)=O)CCCC(C2(NC(c3nccc(C(F)F)n3)=O)CC2)C1 79681,CC1CC(NC(C2CSCN2C(=O)CC2OCCO2)=O)C(=O)O1 79682,n1(CC)cnnc1NC(C1CN(C(C)=O)C1)=O.N1(CC(C)N)CCCC1 79683,c1(CC(N2C3CC(NC(c4cc(Br)co4)=O)(C3)C2)=O)ccc2c(c1)OCO2 79684,c1(-c2nc(C(=O)NC(c3cccc(Br)c3)C(C)C)on2)cccc(OC(C)C)c1 79685,CC(C)S(=O)(=O)CC(=O)N(CC(O)CNC(=O)CNC(c1cccc(O)c1)=O)C 79686,Cc1ccc(C(=O)NCC2CN(C(=O)Cc3ccon3)CC2C)c(C2CC2)n1 79687,CCC(C)C(O)C(=O)NCCC1(O)CN(C(=O)Cc2cc(Cl)ccc2OC)C1 79688,CCC(C)(C(=O)N1CC2CC(C1)N(C(=O)CCNC(c1cnccn1)=O)C2)C(N)=O 79689,c1(-c2ccc(CNC(c3cc(Cl)cnc3O)=O)cn2)cccn2ccnc12 79690,Cc1cnc(C(N2CCC(CNC(=O)CC3CCCCCC3)C(C)C2)=O)c(F)c1 79691,N1(C(c2cnc(CC)s2)=O)CCC(F)(C(=O)Nc2ccc(F)c(C)c2)CC1 79692,CCC(CC(F)F)C(=O)NCCNC(C1NC(=O)C2CC12)=O 79693,c1(C(=O)NCC23CC(NC(CC4CC(C)OC4)=O)(C2)C3)cccc2ccn(C)c12 79694,CC(CC(C)NC(=O)C(C)OCC1CC(c2ccccc2)C1)NC(C1CC1)=O 79695,N1(C(C2(c3ccc(C)cc3)CC2)=O)CCC(C(N2CCC(C)(N(C)C)C2)=O)CC1C 79696,c1(C(=O)NC2CCC(NC(C3C(COC)CC3)=O)C2)nc(C(F)(F)F)cn1C 79697,c1(CNC(C2CCCO2)C)cnn(CC2CC2)c1C(F)(F)F 79698,c1(C(N2CC(OC(C3(C=C)CCC3)=O)C2)=O)ccnc2c(OCC)cccc12 79699,c1(C(C)NC(CC2(NC(Cn3c(C)nnn3)=O)CCC2)=O)cc(Cl)ccc1F 79700,C(CN1C(=O)Cc2ccccc21)NC1(c2n(C3(C)CC3)nnn2)CCNC(=O)C1 79701,C#Cc1cncc(C(=O)NC2(C(N3CC4(C3)CN(COC)C4)=O)CCCC2)c1 79702,N1(C(CC(=C)Br)=O)CC(NC(=O)CCCN(C)C(C)=O)CC1C 79703,C(=O)(C(O)C(C)(C)CC)N1CC(C(=O)NCC(CC)NCCN2CCC(C)CC2)C1 79704,C(=O)(N=c1cc(-c2ccco2)o[nH]1)N(C(c1cnc(C)s1)=O)C 79705,c1(C(N2C(CN(C(=O)C=CC3CCOC3)C)CC(F)C2)=O)cc2n(n1)CCC2 79706,C1(C(=O)NC)CCN(C(=NCCCC2CC2)NCC(C2CC2)C2CC2)C1 79707,c1(C2C(C(=O)NC3C(CNC(=O)C(c4ccc(Cl)cc4)=O)C3)C2)ccccc1C#N 79708,C1(NC(C=NOC)=O)CCN(C2CCN(C(C34CC(O)C3C4)=O)CC2)CC1 79709,C(CCCC(=O)N1CC(C(C)(C)O)(CNC(c2cccn2C(C)C)=O)C1)OCC 79710,O=C(C#CC1CCCOC1)NC1(CNC(c2ccnc(S)c2)=O)CCOC1 79711,c1(NCc2cc[nH]n2)cc(N2CC3C(C2)C3(F)F)ncn1 79712,CN1CCN(c2nc(Cl)ncc2Cl)C(CNC(C2CC3CCC(C2)S3)=O)C1 79713,C1(F)(CNC(c2ncc(C)s2)=O)CCCN(C(C2(C)CC2C)=O)C1 79714,S(=O)(=O)(c1ccc(NCCS(N)(=O)=O)nc1)NC1C(C)CCc2ccccc21 79715,c1(C(=O)NCc2ncoc2CNC(C(CCC)C#N)=O)cnn2c(Br)cccc12 79716,C1(NC(CC(c2ccc(F)cc2)C)=O)CCCCC1NC(=O)C(N)=O 79717,C1(C(=O)NCC(COC)(C)C)CCN(C(=O)C(C)N(C)C(C)=O)C12CC2 79718,c1(-c2cn(C(C)C(N3CCN(C)C(C)C3C)=O)nn2)ccc([N+](=O)[O-])cc1 79719,c1(C(=O)NCC23C(CN(C(C(C(=C)Cl)(C)C)=O)C2)C3)cccc2c1ncn2C 79720,C1(C(=O)O)(NC(C2CN(C(C(C)NS(CC)(=O)=O)=O)C2)=O)CC(CO)C1 79721,c1(NCC2CCCCN(C(Cc3ccc(C)s3)=O)C2)nc(Cl)nc2sccc12 79722,Cc1c(NCCCOCCC(C)C)ncnc1N1CCC(C)(F)C1 79723,c1(CN(C(=O)C=CC2(C)CCOCC2)C)cc2ccccc2[nH]1 79724,c1(C(=O)NC(CC=C)CNC(C2CC(F)(CO)C2)=O)cc2ccccc2nc1C 79725,c1(C(=O)NC(c2nc(C)c(C(C)C)s2)C)cc2ccc(OC)cc2[nH]1 79726,O=C(CCCCc1ccc(F)cc1)NCCC1CN(C(C2C3CC3C3CC23)=O)C1 79727,C1(NC(C2C(C(C)O)C2)=O)CCCN(C(c2cncn(C)c2=O)=O)CC1 79728,C1(NC(=O)CCc2ccccn2)CCN(C(c2cc(O)nc(Cl)c2)=O)CC1CO 79729,c1(C(=O)NC(CNC(C2C(C)C2)=O)C)nc(C2CC2)ncc1Br 79730,c1(CC)ncc(C(=O)N(CCCNC(C2CC2C2CC2)=O)C(C)C)s1 79731,c1(C(N2CCCC2c2c(F)cccc2Cl)=O)cc(Cl)cc2nc[nH]c12 79732,C1(C(C)C)C2CCN1C(CCC1CC1)C(=O)N2.C1(CC2CC2)CCOC1 79733,c1(C(N2CCN(C(C(CC)C)=O)C(C)C2)=O)oc2ccccc2c1CS(C)(=O)=O 79734,n1(CC)cc(Br)c(C(=O)NC(C)CC(C)NC(C2CS(=O)(=O)C2)=O)n1 79735,N1(C(C(C)NS(C)(=O)=O)=O)CC(NC(c2ncn3c2CCC3)=O)C(C2CC2)C1 79736,C1(C(N(CC(CN(C)C(c2ccn(C)c(=O)c2)=O)O)C)=O)CCC2CCC1O2 79737,N1(C(C2C(CCOC)C2)=O)CCCCC(NC(C2NC(=O)OC2C)=O)C1 79738,C1(C(=O)NC2CC(n3cc(C(C)C4CC4)nn3)C2)CCC(C2CC2)C1 79739,C(C)(C)(CNC(=O)C(C1(C)CC1)NC(=O)CC1(C)CC1)OC(C)C 79740,c1(OCCOC)cncc(C(=O)NC2CCC(NC(C3CC=CC3)=O)C2)c1 79741,N1(C(CC2(COC)CC2)=O)CCOC2CN(C(C3CCSCC3)=O)CC12 79742,N1(C(c2cnc(OC)nc2)=O)C(CNC(c2cc(Br)c[nH]2)=O)CC2COCC12 79743,c1(C(N2C(CCNC(CCOCCOC)=O)CSCC2)=O)cnc2ccoc2c1 79744,c1(C(=O)OC)sc(NC(C2C(O)CCN2Cc2nccn2C)=O)c(C#N)c1C 79745,CC(C)CCC(=O)C(=O)NCC#CC(=O)NCC1CCOCC1(C)C 79746,C1(C(N2C(CC#C)CCCC2)=O)CC(C)CN(C(c2cc(C)cc(Cl)c2)=O)C1 79747,C=CC(C)(CC)C(=O)NC1(O)CC(CNC(=O)C(c2c(C)cccc2C)O)C1 79748,C12(CNC(C(CSC)(C)C)=O)CCC(CNC(=O)C3=CSCS3)(CC1)CO2 79749,N1(C(CCCNC(=O)OC)=O)CCN(C(C)CNC(=O)Cn2ccnc2C)CC1 79750,C#CCCC(O)C(=O)N1CC(CNC(c2ccc(-c3cc[nH]n3)cc2)=O)C(O)C1 79751,Cc1c[nH]c(N2C3CCCC2CC3)nc1=Nc1ccc(Cl)cc1 79752,C(=O)(CC(CC(C)C)NC(c1cnc(OC)s1)=O)NC(C#C)(C)C1CC1 79753,CCCCCCC(C)CC(=O)OC(C)C(=O)NCC1(O)CCCC(C)C1 79754,N1(C(C2(OC)CC(CF)C2)=O)CCC(C)(NC(C2(C#N)CCCO2)=O)C1 79755,CC(C(C)(C)C(=O)Nc1cc(CO)cc(F)c1)NC(c1ccc(CO)nc1)=O 79756,Cc1ccc(CC(=O)NNC(=O)c2ccccc2C(F)(F)F)c2c1CCC2 79757,C(CCOCCO)(C(=O)N(CC(F)F)C)NC(Cc1c(C)scc1)=O 79758,CCCN=C(NCc1nn(C)cc1Br)NCCCC(C)(C)OC 79759,C1(C(=O)NCC2(C(=O)NC)CC(=C)C2)CCCCC1NC(=O)CC1(CCO)CC1 79760,c1(C(=O)NC(CCNC(C(C(C)C)NC=O)=O)C)ccc(F)cc1Cl 79761,N1(C(C2COC3(CCC3)C2)=O)CCC2(CCCN2C(=O)COC(F)(F)F)C1 79762,n1(C(C)C#N)cccc(NC(=O)C(C)Cc2cnn(C)c2)c1=O 79763,C=Cn1ncc(C(=O)NCC2CCCN2C(=O)CCc2ccc(C)o2)c1N 79764,CC1(C(=O)NCCCOCCNC(C2CCCCS2)=O)CC1(F)F 79765,N1(C(c2nc(NC(C3C(C)C3)=O)sc2)=O)CCCOC(CNC(=O)CCCC#N)C1 79766,N1(C(CCC(=O)OCC)=O)Cc2ccnn2CC(NC(=O)CC23CCCC2C3)C1 79767,c1(C(=O)NCC(CNC(C2CC(C(C)=O)C2(C)C)=O)F)ccc(F)cc1F 79768,N1(C(c2cc(C)c(Br)cc2)=O)CC(CNC(c2cncnc2)=O)C2(CCC2)C1 79769,C1(C)(N(C(C2(OCC)CCC2)=O)C2CC2)CCN(C(c2sncc2C)=O)C1 79770,C1(=O)CC(C)N1.C1(OCC)CC(NC(=O)CCC2CC(N(C)C(N)=O)C2)C1 79771,C1(C(=O)NCC(C)(C)CCNC(C2(CO)CC2)=O)(CC)CCC(C(C)(C)C)CC1 79772,Cn1nc(C(N2CCCC2CNC(=O)C2=NOCC2)=O)cc1OC(F)F 79773,C(=O)(C(C)(C)CCNC(c1csc(C)c1)=O)NC(CSC)(C)CO 79774,C(=O)(C1=CCCN(C(c2ccoc2Cl)=O)C1)N1C(C)CC(C)C1 79775,c1(NC(C=C2CCN(Cc3ccc(OC)cc3O)CC2)=O)nc(Cl)c(C)c(Cl)n1 79776,C1(C(=O)NC2CC3(C(NC(C4CCN(C)C4)=O)C3)C2)Cc2ccccc2NC1=O 79777,Cc1ncnc(C)c1C(=O)N(CC(C)N(C(=O)C(CC(C)C)n1ccnc1)C)C 79778,Cc1cc(C(=O)N(C2CCC(NC(C3(C)C=CCCC3)=O)CC2)C)ncc1CO 79779,CC1CCCCC1(C)C(N1CCC2(CC2C(=O)N(CCS(N)(=O)=O)C)C1)=O 79780,N1(C(C2C(C)C2)=O)CC2CC2(NC(c2coc(Cc3ccccc3)n2)=O)C1 79781,C1(OC)CCN(C(=NCCNc2ccc(F)cc2)NCCF)CC1(C)OC 79782,n1(C(C(=O)NCC2CCN(C(C(C=C)O)=O)CC2)C)nc([N+](=O)[O-])cc1C 79783,N1(C(c2cn(C)nc2)=O)CCCC2CCN(C(c3cc(C(N)=O)cs3)=O)CC12 79784,C1(NC(COCCCCC)=O)CCCC(NC(C2CC(N(C)C)C2)=O)C1 79785,N#Cc1cc(NC(C2CN(C(=O)CC3CCCCO3)CCS2)=O)cnc1Cl 79786,C1(NC(CNC(CC(C)C)=O)=O)CC2CC1CC2C(N1CC(C)C(O)C1)=O 79787,Cc1cc(-n2nc(Cc3cnn(C)c3)nc2CCc2cc[nH]n2)ccc1Cl 79788,C1(C(=O)Nc2ccc(C3CCN(C(C(C)OC)=O)CC3)cc2)CCCC(C#N)C1 79789,C(=O)(C(CC1CC1)NC(c1ccncn1)=O)NC(C(=O)OCC)C 79790,C1(O)(CNC(CCC(C)SC)=O)CCCN(C(=O)C(F)=CC2CC2)C1 79791,N1(C(CC2CC(C(=O)OC)C2)=O)CCCC1C1CCCN1C(C1CC(O)C1)=O 79792,N1(C(c2cccnc2)=O)CCN(C(C2CC2(Cl)Cl)=O)C(CF)C1 79793,N1(CC(=O)N(C(C)CC2CCOCC2)CC=C)CCC(OCC)C1 79794,c1(NC(=O)NCCc2ncn(C(C)C)c2)cc([N+](=O)[O-])ccc1-n1cnnn1 79795,N1(C(c2nnn(CC)c2C)=O)CC2(CNC(c3cnnn3C(C)C)=O)CC1CO2 79796,C(CCC(C)C)(C(=O)NC1CCCC1(C)CN(C)C)NC(c1ccc(C)n1C)=O 79797,c1(C(=O)NC(C2CCCO2)CC)ccc(CNC(C2CC(C)(O)C2)=O)o1 79798,CC(CNC(=O)CNC(=O)NC1CC1)N=c1ccnc(C2CCCC2)[nH]1 79799,N1(C(CC(C=C)CC)=O)CCC(CNC(=O)C2=CCCC2(C)C)C(F)(F)CC1 79800,N(C1CC2(CN(C(=O)CCn3cc(C)cn3)C2)n2ccnc21)C(C(CC)SC)=O 79801,C1(C(N(CCN(C(C2CC2(C)CC)=O)CC)CC)=O)CNC(=O)C1 79802,c1(C(N2C(C)CCC(NC(=O)Cc3cnco3)C2)=O)cccc2oncc12 79803,c1(NC(C(=O)NCCc2cn(C3COCC3F)nn2)=O)cc(Cl)ncc1Br 79804,C(=O)(NN=c1ccc2nccn2[nH]1)c1c(C)ccc(CCC(=O)OC)c1 79805,c12cccc(c1)S2.N1(C(CC)=O)CCCC1C(c1cnn(C)c1)O 79806,C1(C(=O)NCC(c2ccccc2)O)(CC)CCCN1C(C1CC(C)(C)CN1)=O 79807,CN(C)NC(=O)CCC(=O)N1CC2(n3cc(-c4cc(F)ccc4Cl)nn3)CC1C2 79808,C1(C(C)C)CCCCC1C(=O)N(C)CCOCCNC(C1(C)SCCCS1)=O 79809,C1(C)(CCNC(C2(N(C)C(c3nc(Cl)cs3)=O)CC2)=O)CCOCC1 79810,c1(C(=O)NC(C2CC2)=O)nnn2ccccc12.N12CC3C(C3C1)CN(C)C(C)C2=O 79811,C1(C(N(C)Cc2n(CC)ncn2)=O)CCOCC1NC(=O)C(C)=NOCC#N 79812,N1(C(CC=CC)=O)CCC(CNC(=O)C=Cc2cscn2)CC1C 79813,Cc1ccc(C)c(C(=O)N(CC(=O)NCC23CC(CN2C)C3)CCO)c1 79814,CCCC(F)C(=O)N(C1CCN(C(=O)CCOc2ccc(C)cc2)CC1)C 79815,n1(C(CC)C)nnnc1C(c1sccc1Cl)NCC1CC2(CC2)C1 79816,S(=O)(=O)(c1ccc(C(=O)NCC(C)CNC(=O)CC2CCC(OC)CC2)o1)NC 79817,Cc1ccc2c(c1)CC(C(=O)NCC(O)CN(C(=O)CN1CSCC1=O)C)O2 79818,N1(C(c2cncc(OC(C)C)c2)=O)CC(C)(C)CCC1CNC(C1CCSC1)=O 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79837,C(CCCCCNC(C1(C)CC=CCC1)=O)N(C)C(c1cccc(CS(C)=O)c1)=O 79838,c1(CC)ccc(F)c(C(=O)NCC2(O)CC(NC(=O)C(C)SC(F)(F)F)C2)c1 79839,C(=O)(C1=CC2(CCN(C(=O)C(C)N(C)C(C)=O)C2)C1)NC1CCN(CC)C1 79840,C(=O)(CCP(C)(C)=O)N1C(CN(C)C(c2ccon2)=O)CCC1 79841,C1(C2CCCO2)C(=O)N1.C1(COCC)(NC(=O)CCc2nccs2)CCC1 79842,C=CC(C)(C)CC(=O)NC(C1CCCCN1C(c1ncccc1NC(C)=O)=O)C 79843,c1(C(N2CC(NC(C34CC(C(=O)OC)(C3)C4)=O)C2)=O)cncc2c[nH]nc12 79844,C1(NC(C(C(C)C)O)=O)C2CC1CN(C(c1cc(C#N)c[nH]1)=O)C2 79845,N1(C(C2N(C(C3CC(C)=C(C)CC3)=O)CCC2C)=O)CC2CCCC(C2)C1 79846,N1(C(C(C(C)C)OC)=O)CCCC2(C1)CN(C(c1cccc(O)c1Cl)=O)CCO2 79847,C12(C(N(C3CCN(C(c4n[nH]c(C)c4Cl)=O)C3)C)=O)CCCN(CC1)C2 79848,CC1(CNC(=O)C=CCO)CCCN(C(c2cc(N)ccc2O)=O)C1 79849,CC1(C)CN(C(c2cc(C3CC3)no2)=O)C(CNC(C2CCCOC2)=O)CO1 79850,c1(C(N(C2CCN(C(=O)CCCC(C)C)CC2)CC)=O)cc2cncn2c(O)n1 79851,c1(C(N(C2CCN(C(CC(C=C)C)=O)C2)CC)=O)cc2nc(Cl)ccc2s1 79852,c1(NC(c2ccc(Cl)s2)CC)nccc(N2CCC(c3nc(=N)n(C)[nH]3)CC2)n1 79853,C1(NC(CC(C)SC)=O)CCOCC1C(=O)NC(C)(C)C#N 79854,C1(C(=O)NC(C2(O)CN(C(=O)CN(S(C)(=O)=O)C)C2)C)CC1[N+](=O)[O-] 79855,c1(C(CO)NC(NNC(c2cccc(OC)c2)=O)=O)ccc(S(C)(=O)=O)cc1 79856,c1(C(=O)NC2CC(NC(C34C=CC(CC3)C4)=O)C2)c[nH]c2ccc([N+](=O)[O-])cc12 79857,C1(C(=O)NCCCN(C(c2cncc(N(C)C)n2)=O)CC)CCCCC1C1CC1 79858,N1(C(CC(CC)NC(c2c(C)nsc2C)=O)=O)CCC(O)C(CO)C1 79859,Cc1nc(NC(C2CN(C(=O)CC(C)C)CCN2)=O)ccc1CO 79860,C(=O)(C(C)(C)C(=O)N(C)C)NCCN(C(=O)C=C(C)c1ccsc1)CCOC 79861,Cc1ccc(O)c(C(N2CCC(CNC(=O)C=Cc3cccnc3)C2)=O)c1 79862,c1(OCCOC)ccc(CN2CC(C(=O)NC3CC(C(=O)O)CC3O)C2)cc1 79863,C1(CNC(=O)Cc2csc(-c3ccco3)n2)COCCN(C(=O)C=C2CCC2)C1 79864,C(=O)(C1CCc2cc(C)ccc21)N1CC(C(=O)NCCOCC)(CNC(C)=O)C1 79865,C12(C(=O)NCCCNC(c3cccc(C(N)=O)n3)=O)CCCCC1CS(=O)(=O)C2 79866,c1(C(=O)NCC(N(C(C2CCN(CC)C2)=O)C)C2CC2)c[nH]c(=N)c(C)c1 79867,O(NC(=O)C(CCF)NC(c1cccc(O)c1F)=O)C(C=C)C 79868,c1(C(=O)NC2CCCN(C(CC3(C=C)CCC3)=O)CC2)cc(C)cc(OC)c1C 79869,N1(C(c2[nH]cc(C)c2)=O)CCC2(C1)CN(C(=O)CCCNS(C)(=O)=O)C2 79870,c1(OC)ccc(C(=O)NCC(C2(O)CN(C(C3CCCSC3)=O)C2)(C)C)cn1 79871,c1(C(N2C3C(N(C(C(CC)SC)=O)C)CC(C3)C2)=O)ccn2ncccc12 79872,Cc1nc(N2CCCCC(CNC(=O)CC(C)C)C2)c2c[nH]nc2n1 79873,CC(N=c1cc[nH]cc1S(=O)(=O)N1CCC1C1CCCCC1)C1CC2(CCC2)C1 79874,c1(C(N(CCN(C(C2(C(=O)NC)CC2)=O)C)C(C)C)=O)c(C)cc(Br)cc1F 79875,CCCC(C(=O)OC)NC(=O)C(C1CCC1)NC(c1cnccn1)=O 79876,C(C(=O)NCCC1CC(NC(=O)C=CBr)C1)(C(C)C)SCC 79877,N1(C(c2cc(CC)nn2C)=O)CC(NC(C2CCC(CC)CC2)=O)CC12CCC2 79878,N1(C(C2C=CCCC2)=O)CCC(O)(c2ccccc2)C(O)C1.C1(N)CCS(=O)(=O)C1 79879,CC(C)C(C)CC(=O)NCC1(O)CC(C(N2CCOCC2)=O)C1.C1C(=O)N1 79880,N1(C(C2(C)CCNC2=O)=O)CC2(CCCN(C(=O)Cc3ccc(F)cc3F)C2)C1 79881,c1(CCC(N2CCC(N(C(=O)CC(C)OC)CCC)C2)=O)ccc2c(c1)CCO2 79882,C1(NC(C(C)NC(N)=O)=O)CCSC12CN(C(c1cccc(C(F)F)n1)=O)C2 79883,C(c1ccc(=N)[nH]c1)=CC(N1CC(NC(C#CC(=O)N(C)C)=O)(CO)C1)=O 79884,N1(C(c2cccc(N3CCCC3=O)c2)=O)CC2CCC(C1)N2C(C1CCC1F)=O 79885,CC1CCN(C(c2cnn(C)c2Cl)=O)CC1C(N1CC(O)(C(F)(F)F)C1)=O 79886,C1(COC(=O)Cc2cccnc2O)CC2CC1CC2O 79887,n1(CC)ncc([N+](=O)[O-])c1C(=O)NCC(C)CNC(c1ncn(C(C)(C)C)n1)=O 79888,c12n[nH]c(n1)CNC2=O.c1(N(C)C)cc(CNC(C2CC2(Cl)Cl)=O)on1 79889,N1(C(C(c2scc(C)n2)C)=O)CCC(=CCNC(c2[nH]nnc2C)=O)CC1 79890,c1(C(=O)NC2CCCCN(C(CCCCC)=O)C2)cc2cc(OC)ccc2o1 79891,n1(C(CC)CCCO)cnc2c(N3CCC4CCC(C4)C3)ncnc12 79892,c1(NC(c2c(OC)ccs2)=O)ccc2c(C(N3CCOCC3(C)C)=O)ncn2c1 79893,C1(C(=O)NC2C=CC(Cn3cc(CNC)nn3)C2)CC12CC(F)(F)C2 79894,c1(N2CCC(C)C(NC(C3CCS(=O)(=O)C3)=O)C2)ncnc2[nH]cnc12 79895,N1(C(C2C(C)CCOC2)=O)CC2(CCN2C(C2CCC(=O)O2)=O)C1 79896,c1(CC(C)OC)nc(C2CCN2C)n(-c2ccnn2C)n1 79897,C#CC1(NC(=O)CCCCC(N)=O)CCN(C(C2(COC)CC2)=O)CC1 79898,C1(CCOC)(NC(C(CC)F)=O)CCCN(C(=O)CC(C)OC)C1 79899,N1(C(Cc2cnc(C)s2)=O)CCC(CNC(c2c[nH]nc2C)=O)C(C)C1 79900,C1(NC(C2CCn3nncc3C2)=O)CCC2(CCNC2)C1 79901,c1(C(c2nnnn2C2CCC2)NC(c2cncc(C)c2)C)nc2c(s1)CCCC2 79902,c1(C(N(C(C)C)CCNC(=O)CC2CC(C(F)F)C2)=O)coc2c1CCCC2 79903,C(=O)(C1Cc2ccccc21)NCCOCCC(=O)NCC1N(C)CCOC1 79904,N1(CC(N2CC(OCCNC(C3(COC)CCC(=O)N3)=O)C2)=O)CC2CCC1C2 79905,c1(NC(C2CCCN(Cc3cccc(Cl)n3)C2)=O)ccc(O)cc1O 79906,C1(COC)(NC(=O)CC(C)(C)C2CC2)CCN(C(=O)C2=NOC(C)C2)CC1 79907,CCCCCC(O)CC(=O)NCC12CC(CN1C(=O)C(N1CCCC1)C1CC1)C2 79908,C12(C(=O)NC3CCCN(C(c4cc(OC)ncc4)=O)C3C)CCC(O)(CC1)CC2 79909,c1(C(N2CC3CC2C3CNC(C2(C(F)F)CCCC2)=O)=O)cc2occc2[nH]1 79910,CC(C)(C)C=CC(=O)NCCNC(=O)C(=O)NCC(C1CCCO1)SC1CC1 79911,c1(CC)cnc(O)c(C(=O)NC(C)(CNC(C2CC2(Cl)Cl)=O)C2CCC2)c1 79912,S(=O)(=O)(c1ccc(Cl)s1)N1CCN(C(C2CC(NC3CCC(=O)C3)C2)=O)CC1 79913,C1(NC(C(CSC)O)=O)CCN(C(=O)Cc2c(F)cncc2Cl)CC(O)C1 79914,C=CCC(CC=C)C(=O)N1CCC(F)(F)C(CNC(c2cncn2C2CC2)=O)C1 79915,c1(C(N2C(CC(C)O)CCCC2)=O)cccc2c1COC2 79916,c1(C2(Oc3ccc(Cl)cc3)CC2)cc(F)c(N)cc1F.C1(=O)C(=O)NC(C)CN1 79917,C1(CC)CCCC1(C)C(=O)N(C1CN(C(c2cccc(OC3CCC3)c2)=O)C1)C 79918,CCCCS(=O)(=O)CC(=O)NC1(CO)CCN(C(c2ccc[nH]2)=O)C1 79919,c1(NCc2ccc(C(C)(C)C)cc2)ncccc1S(=O)(=O)NC1CCC12CCC2 79920,c1(C(N2CC(C)(CNC(CC(C)OC)=O)C(C)C2)=O)cnc(O)c(C(C)=NO)c1 79921,c1(CC(=O)NCC2N(CC(=O)NS(CC)(=O)=O)CCC2)nccc(N(C)C)c1F 79922,N1(C(CC(CC)(F)F)=O)CCC2CCN(C(C3C(C=C(C)C)C3(C)C)=O)C2C1 79923,C1(CNC(CC(CNC(c2ncccc2O)=O)C2CC2)=O)CC2CCCC2C1 79924,CCCC(CCCNC(c1cc(C)nn1CCN(C)C)=O)NC(=O)Cn1cnnn1 79925,C(=O)(CCN(OC)C(=O)CC(C)n1ccnc1)N(C(CC(=O)OCC)C)C 79926,C1(OC)(CNC(c2cccc(CSC)c2)=O)CCN(C(=O)Cc2cnc(C)[nH]2)C1 79927,C1(C(=O)NCCOC)CCN(N2CCC(c3ncc(C)o3)CC2)C1 79928,C1(F)(CNC(C(C)c2ccsc2)=O)CC(NC(C2(c3ccccc3)CC2(Cl)Cl)=O)C1 79929,C=CCC(CC)C(=O)NCC(C)NC(C1(C)COC1)=O 79930,N1(C(c2cn(C3CC3)nn2)C(=O)NCCSC)CCc2ccc(Br)cc2C1C 79931,N1(C(c2c(CC)nc(C)o2)=O)CC(C(=O)N(CCCO)C2CC2)C(C)(C)C1 79932,c1(CNC(=NCc2cc(C)oc2C)NC(C)CN(C)C)ccc(S(C)(=O)=O)cc1 79933,C1(CNC(=O)CCc2ccc(Cl)s2)CCCC(CNC(=O)C2=CCSC2)C1 79934,c1(C(=O)OC)ccc(C(N2CCCC2CNC(c2cc(O)n(C)n2)=O)=O)cn1 79935,C1(C(N2CCCC(NC(C(F)=C(C)C)=O)C2)=O)OCCOC1(C)C 79936,C1(NC(=O)OC(C)(C)C)CCCC12CCN(C(c1cc[nH]c(=NCCF)c1)=O)C2 79937,C1(CC(N)=O)(NC(C2CCCN2C=O)=O)CCN(C(c2ccccn2)=O)CC1 79938,N#Cc1ccc(C(=O)NCCN(C(C2CCC3(CC3)CO2)=O)CC2CC2)cc1 79939,C(=O)(C(F)(CC)C(=O)OC)NCC1N(C(C(CC)CC)=O)CCCC1 79940,C(=O)(C(O)CC(C)C)NC1CCN(C(C2CN(CC)C(=O)N2)=O)C1 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79976,c1(OC)cc(C(N2CC3C(C2)N3C(C2CCCC(C)C2)=O)=O)cc(C(F)(F)F)n1 79977,Cc1cc(Cl)ncc1NC(C1CCC(C)N1C(=O)Cc1cccs1)=O 79978,CC(C)CC(C)(O)C(=O)N1CCN(CC(CNC(=O)COCCF)C(F)(F)F)CC1 79979,C1(C(=O)NCC(CNC(C(C)(CO)OC)=O)(C)O)CC2(C1)CC(C(N)=O)C2 79980,C(C1c2ccccc2CCN1C(c1cnsn1)=O)NC(c1cccc(OC)n1)=O 79981,Cc1noc(C(=O)NCC2C3CN(c4nnco4)CC23)c1C 79982,C1(C(C)NC(CCNC(=O)NC)=O)CCCCC1.C1(=O)C(C)C2(CC2)CN1 79983,C1(C(=O)NC2(C)CCN(C(CCc3n(C)cnn3)=O)C2)COc2ccccc2O1 79984,N1(C(c2cccs2)=O)CCC2CN(C(C)C(=O)O)CC12.c1(OC)cc(OC)ccc1O 79985,N1(CCN(C(CN(C2CCC2)CC)=O)C)CCN(C(c2c(C)n[nH]c2C)=O)CC1 79986,C(=O)(C1=NN(C)C(=O)CC1)N1CCCCCC(NC(Cc2cn(CC)nc2)=O)C1 79987,N1(C(c2c(C)n(C)cc2)=O)CC(CC(=O)NCc2cnc[nH]2)CC1(C)C 79988,C1(NC(C(C(CC)O)(C)C)=O)CN(C(=O)CC2=CCCCC2)CC2CCCC12 79989,N1(C(CCS(=O)(=O)NC)=O)Cc2ccccc2CC1C(=O)NC1(CC(C)(C)C)CC1 79990,N1(C(C(C)NC=O)=O)CCC(C)C(CNC(c2cc(O)nn2C)=O)C1 79991,Cc1nc(Cl)ccc1C(N1CCN(C(c2c[nH]nc2C(N)=O)=O)CC1C1CCC1)=O 79992,CC1CCCCC1C(=O)NCC(C)(C)CCNC(=O)Cn1cccc1 79993,CS(=O)CCC(=O)N1CCCC(CCNC(C2(c3ccc(Cl)nc3)CC2)=O)C1 79994,CN1CC(O)(CNC(=O)C(Cn2cncn2)NC(=O)Cc2cn[nH]c2)C1 79995,N1(C(C2C(C)(C)C2)=O)CCCC2(CC(NC(=O)Cn3ncc4ncccc34)C2)C1 79996,C1(C(=O)OC)(C(=O)NC2CCCC2NC(=O)CC(C)(C)O)CC2(CCC2)C1 79997,c1(NC2CN(C(Cc3scc(C)c3)=O)C(C)C2)ncnc(Cl)c1Br 79998,C1(=O)C(Cc2ccccc2)N1.c1(CN(C)CCOCCO)coc(Br)n1 79999,CN=c1[nH]cc(C(=O)NCC2CCC(C(=O)NCCC3(O)CCOC3)C2)o1 80000,c1(C(=O)NCC2(NC(C3CCCCS3)=O)CCC2)ccnc2nccnc12 80001,Cc1nc(C=CC(N2CC(NC(c3ccc(O)cn3)=O)C(n3ccnn3)C2)=O)cs1 80002,N1(C(CC2C(NC(=O)Cn3ccnn3)COCC2)=O)CCCOC(CO)C1 80003,C1(NC(CC(C)OC)=O)CC2CC(C1)N(Cc1cc(F)cc(F)c1)C2 80004,CC(C)C(C(C)NC(c1cncc(C2CC2)c1)=O)NC(=O)C(F)(F)CO 80005,C=CCCCC(C(=O)N1CCSC(C)(C)C1)NC(=O)CC1CCC(=O)CC1 80006,c1(NCc2n(C)nnc2Br)[nH]c(=NC2CCC3CCC23)nc2scnc12 80007,c1(CCS(N2CC(CC)(CO)C2)(=O)=O)ccc2ccccc2c1 80008,Cc1csc2c(NCC(C3CCCCCC3)NC(=O)CCC(C)(C)C)ncnc12 80009,c1(-n2cc(C3C(NC(N4CCCCC4CCF)=O)C3)nn2)ccnc(Cl)c1 80010,c1(C(=O)NCCN(C(=O)CN2CCCCC2)C(C)C)ccc(C2CCC2)cc1F 80011,c1(C(N2CC(CC)C(NC(C)=O)C2)=O)ccc(OC)cc1OC(F)F 80012,C1(CC)C(NC(c2cncs2)=O)CCN1C(C1C2CC3C(C2)C13)=O 80013,N1(C(c2[nH]cc(C)c2C)=O)CCC2CN(C(C3CN(C)CC(C)O3)=O)CC2C1 80014,N1(C(C2(COC)CCOC2)=O)C2CCC1CN(C(=O)C(C1CCC1)N(C)C)CC2 80015,N=c1cc[nH]c(C(=O)N(C2CCN(C(=O)CC3CCOC3CO)CC2)CCO)n1 80016,C1(C(=O)NCCNC(C2CN(S(CC)(=O)=O)C2)=O)C2CCCCCC12.C12CC1N2 80017,c1(C(N(CCCCN(C(c2n(C(C)C)nnc2)=O)C)C)=O)cc2c(ccn2C)[nH]1 80018,c1(C(=O)NC2CC(C)(CNC(C3C(C(C)C)CCC3)=O)C2)ccc(CC)cc1 80019,c1(C(=O)NCCOCCNC(C(C)OCCC#C)=O)cc(F)c(F)c(C#N)c1F 80020,c1(-n2nnc(C(=O)OC)n2)cccc(NC(C2(CO)CNC(=O)C2)=O)c1C 80021,c1(C(CNC(=O)CC2CCCCC2C(F)(F)F)O)cccc(O)c1 80022,O=C(C#CC1CCCO1)NC1CN(C(C2CCc3nn[nH]c3C2)=O)C1 80023,CC(CCC(F)(F)F)NC(=O)CC(C)NC(=O)CC1OCCCO1 80024,c12ccc(cc1O)NC2.N1(C(CC)C)CCC(C(=O)OC)CC1 80025,c1(OC)ccc(C2CC2C(=O)NCC(C)CNC(=O)CCC2CCOC2)cc1F 80026,c1(NC(=O)OCC)cccc(C(C(=O)C(CC)OC)=O)c1.C12(CC1)C(C)N2 80027,Cc1csc(CCNC(C2C(CNC(c3csc(=N)[nH]3)=O)C2(C)C)=O)n1 80028,c1(C(=O)NC2CN(C(C3CCOC3)=O)CC2CO)ccc(C(F)(F)F)cn1 80029,N1(C(c2ccc(O)nn2)=O)CC2(C1)CN(C(c1ncoc1C(F)(F)F)=O)C2 80030,C#CCCCC(=O)N1CC(N(C(=O)CC2CCC(C3CC3)O2)CC)C1 80031,c1(OC)ccc(NC(=O)C(N2C(C)CCC2(C)C)=O)cc1C 80032,c1(C(N2CC3CN(C(C4(Br)CC4)=O)CCC23)=O)n[nH]c2c1CCSC2 80033,Nc1cccc(C(N2C(CNC(c3ccc(-c4cc[nH]n4)s3)=O)CC3CC23)=O)n1 80034,C1(CC)CC(C(=O)NC(C)CC(C)(C)OC)CCN1C(c1ccnc(C)c1C)=O 80035,CCS(=O)(=O)c1ccc(CNC(=O)Nc2c(Br)cnn2-c2ncccn2)cc1 80036,N(C)(C(=NCC(C)C)NC(c1ccccc1C)C)CCc1c(C#C)cccc1 80037,c1(C(=O)NCCN2CCN(C(C3(C(F)(F)F)CC3)=O)CC2)ccc(CCO)cc1 80038,C1(c2nccn2C)(NC(C)=O)CN(CS(=O)(=O)NC2CCOC2)C1 80039,C(CCCC(=O)N1CC(CC(C)(C)CNC(C2(Cl)CC2(C)C)=O)C1)N(C(C)=O)C 80040,c1(C(N(C2CCC23CCNCC3)c2cccc(N)c2)=O)nc2n(c1Cl)CCCC2 80041,CCCCC(C(=O)NC1(CC(=O)NCCOC2(C)CCC2)CCC1)C(C)C 80042,Cc1nscc1CC(N1CC(F)(CNC(C23CC(CO)(C2)C3)=O)C1)=O 80043,C(=O)(C1=CC2CCCC12)N1CCN(C(c2c(OC)ccc(OC)n2)=O)CC1C 80044,C1(C)(NC(C(c2cccc(C)c2)(F)F)=O)CCCN(C(=O)C(C)n2cccn2)C1 80045,CC(C)CC(O)CC(=O)N1CC(C2(NC(c3ccncc3F)=O)CC2)C1 80046,C1(C(=O)NCC2CC(F)C2)CC2CC1CN(C(=O)CCCC1CCC1)C2 80047,N1(C(C#CC2(CC)CC2)=O)CCC2CN(C(c3cccn(C)c3=O)=O)CC2CC1 80048,C1(F)(C(=O)NC(C)C)CN(C(=O)CCc2cn(C)nn2)C1 80049,c1(C(N(C2CCN(C(Cn3c(C)nnn3)=O)C2)C)=O)cnc2ncnn2c1O 80050,C1(F)(C(=O)NCC2C(C)OCC2)CCN(C(=O)CN(C)C(=O)C2CC2)CC1 80051,c1(C(=O)NCCOC2CCN(C(C(C=C)O)=O)C2)ccc(C2CCOCC2)cc1 80052,c1(OC)cccc(C(N2CC(CNC(c3cnoc3C3CC3)=O)CC2C)=O)c1 80053,C(=O)(C1CCCc2ccccc21)NC1CCN(C(CC=CCC)=O)CC1(C)C 80054,CC1COC2(C1)CN(C(C13CC1CCN3C(C13CCC(C1)C3)=O)=O)C2 80055,c1(CCC(=O)NCC(C2(O)CCN(C(CSCC#C)=O)C2)C)cccc(F)c1Cl 80056,C12(NC(C3OCCN(C(C)C)C3)=O)CCCC1N(C(C1(F)CCCC1)=O)CC2 80057,c1(CN(C(C(c2onc(CCC)n2)NCCCC2CC2)=O)CC)cccc(CC)c1 80058,c1(OC)cc(C(=O)NCCOC(c2cccc(F)c2)=O)c([N+](=O)[O-])c(F)c1 80059,C1(C(N2C(CC)CC(O)C2)=O)CCC(C)(C)N(C(=O)C=CC(F)F)C1 80060,C(=O)(C1=NOC2COCC12)NCCCCCCNC(C(C)Sc1cccc(Cl)c1)=O 80061,c1(OC)ncccc1C(=O)NC1(C2CCCN2C(C23CC(F)(C2)C3)=O)CC1 80062,C12(C(N3CC(CNC(C4CC5(CCC5)CO4)=O)C3)=O)CCC(C(F)(F)F)(C1)OC2 80063,N1(C(C(CC)=CCCC)=O)CCN(C(=O)C(C)ON2CCOCC2)CC1C 80064,c1(C(=O)NC2CC(CNC(C(=Cc3cccs3)C)=O)CC2O)csc2nccn12 80065,CC1Cc2ccccc2C(Nc2nnnn2Cc2cc(Br)cs2)C1 80066,C(=O)(C1=C(C)OCCC1)N(CCNC(c1nc(C(F)(F)F)ccc1F)=O)CC 80067,C(=O)(CCCCN(C)C)N(C1(CC(=O)NC(C(=O)OC)C2CC2)CC1)C 80068,c12ccc3ncc-1n3c2.c1(C(=O)NCCN(C)C)c[nH]nc1Cl 80069,CCC(CC)(CO)C(=O)N1CC(NC(=O)C(c2ccc(F)cc2)(C)C)CC(C)C1 80070,C1(C(=O)NCCN(C(C(C2CCCC2)NC(C)=O)=O)C)(NC(C)C)CCCOC1 80071,C(=O)(CC(CC)C(C)(C)C)N(C1CCN(C(c2cncc(C#C)c2)=O)CC1C)C 80072,C1(CNC(c2c(CNC(c3cnc(C(C)C)o3)=O)occ2)=O)CCC(=O)NC1 80073,CON(C(=O)C1CC(C)(C)C1)C1CCCOc2ccccc21 80074,C=C=CC(C)C(=O)N1CC(N(C)C(c2cc(C(F)(F)F)ns2)=O)C1 80075,c1(SC)cccc(F)c1C(=O)NC1CCCC(NC(c2sccc2C2CC2)=O)C1 80076,C(C(C)(C)CC(C)C)NC(C1(CNC(C2C(CC)CC2)=O)CCCO1)=O 80077,C1(C(N(C)CC2(CNC(C3CC4C=CC3C4)=O)CC2)=O)CC2CC1C1CC21 80078,C(=O)C(O)CC(F)(F)F.CCC1C(=O)N1.C1(C(=O)OCC)CCCN1C(=O)C(C)C 80079,n1(CC(=O)NC2CCC(NC(c3csc(C(F)(F)F)n3)=O)CC2)ccccc1=O 80080,c1(C(=O)NCC(N(C)C(c2cc(C3CC3)cs2)=O)C2CC2)ncn2c1CCCCC2 80081,CCCCCS(=O)(=O)CC(=O)N1CCCC2(C1)CN(C(C1(CF)COC1)=O)C2 80082,CCC(C(O)C(=O)OC)NCc1cc(C#N)c(Br)s1 80083,c1(CNC(C2C(CNC(CCC=C=C)=O)CCCC2)=O)cc(C)nc(C)c1 80084,CC1(C)CC(NC(c2ccncn2)=O)CN1C(c1cn(C2CC2)nn1)=O 80085,C1(NC(CNC=O)=O)CCN(C(=O)C2=CCOC2)CC1O 80086,c1(CN2CCCC(C)(C(=O)Nc3cc(F)ccc3O)C2)cccc2nonc12 80087,c1(C(N2CC(C(C)NC(CC(CC)C)=O)C2)=O)cc2c(C)c(F)ccc2[nH]1 80088,C1(C(C)NC(=O)C(C2CCCC2)NC(c2ccc(CO)o2)=O)CC2(CCC2)C1 80089,CC(C)(C(=O)N1CCC(NC(c2csc(C(F)F)c2)=O)C1)S(=O)(=O)C1CC1 80090,Cc1cc(C(=O)NCCC2CCN(C(c3cc(Cl)no3)=O)CC2)cc2nn[nH]c12 80091,c1(C(N2CCC(NC(CCC(C)O)=O)C2C2CC2)=O)cc2c(cn1)CCCC2 80092,Cc1ncnc(C(=O)NC2CCC2NC(=O)Cc2ccc(F)cc2F)c1C 80093,c1(CC)ccn(CC(F)(F)F)n1.C1(=O)CN(CCOC)N(CCC)CCN1 80094,c1(C(=O)O)ccc(C(N2CC(O)CC2C2CCOCC2)CC2CCCC2)n2nccc12 80095,CC1C(NC(=O)C=Cc2ccc(=N)[nH]c2)CCCN1C(c1cc(CCO)on1)=O 80096,c1(C(N(CCCOCCNC(C(C)SCCCC)=O)C)=O)cc(=O)cc(Cl)[nH]1 80097,c1(C(=O)NC(C2(O)CN(C(c3cc(C)sn3)=O)C2)C)cc2c(nn1)CCC2 80098,c1(OCC)ccc2c(C(=O)NCc3cccc(C(F)(F)F)c3F)coc2c1 80099,C1(NC(c2cc(C)nc(O)c2)=O)CC2CC1CN(C(=O)C=Cc1ccn(C)c1)C2 80100,Cc1nc(CS(=O)(=O)NC(=O)C(C)(c2ccccc2)NC(N)=O)co1 80101,c1(-c2cc(C)c(C)nc2)cccc2sc(C(=O)NC(C)C(F)(F)F)cc12 80102,C(CS(=O)(=O)c1ccc(F)cc1)NC(c1cnn(C)c1C)c1n(CC)nnn1 80103,c1(N2CCC(C(C)C)(COCC)CC2)cc2c(cc1[N+](=O)[O-])CCC(=O)N2 80104,C1(NC(c2c(OCCC)cccc2)=O)CCN(S(=O)(=O)CC(C)C)CC(C)(C)C1 80105,c1(N2CCC(C3C(C)(C)CCC3)C2)ccc(S(=O)(=O)NCC2C=CCC2)c(Cl)c1 80106,c1(CC)cc(CNC(c2[nH]ccc2CNC(=O)C(C)CC2CCC2)=O)on1 80107,Cn1cc(C(C)(C)C(=O)N2CCC2CNC(C2C=CCC2)=O)cn1 80108,C1(NC(=O)OC(C)(C)C)CCC(O)(Nc2cc(-c3cccnc3)cc(F)c2)CC1 80109,C(=O)(C(C)(C)CSC)N1CCC(CCNC(Cc2c(C(=O)OC)csc2)=O)C1 80110,C1(C(=O)NC(CN(C(c2ncccc2Cl)=O)CC)C)CC(=O)NC1(C)C 80111,N1(C(c2cc(C#N)sc2)=O)CCN(C(=O)CC2C=CCCC2)CC1C(F)F 80112,C(c1ccncc1)=C(C)C(=O)NCCC1CSCCN1C(=O)CC(C)F 80113,c1(C(=O)OC)c[nH]nc1C(=O)NCCCC(C)NC(C1COC(=O)N1)=O 80114,Cc1ccc(C(=O)NC2CC2NC(c2n[nH]cc2C)=O)c(C(C)C)n1 80115,C1(C(=O)NCC2(C(=O)NC3CCCCC3)CCCCC2)CC(=O)C12CCCC2 80116,N1(C(CCNC(C)=O)=O)CCOc2ncc(-c3csc(C(F)(F)F)n3)c(C)c21 80117,Cc1cc(C)c(C(C)NC2COCC2C(=O)Nc2ncccn2)c(C)c1 80118,N1(C(CCCC#CC)=O)CC2(CCCC2NC(C2CN(C(C)C)CCO2)=O)C1 80119,c1(C(N2CC(NC(C=C(CC)C)=O)C(O)CC2)=O)oc2cc(Cl)ccc2c1C 80120,CCC(CCCC(=O)N(C)CCC1CCOCC1)NC(=O)CCC(CF)CF 80121,c1(NCC2(CCOC)CCCC2)ccc(S(=O)(=O)N2C3CCC2COC3)cc1Cl 80122,C1(CCNC(c2onc(CC)c2C)=O)CN(C(c2c(Cl)cnn2C)=O)CC(C)O1 80123,C1(NC(CCCCCC)=O)CC2CCC(C1)N2C(=O)CS(=O)(=O)NC(C)(C)C 80124,c1(C(N2C(C(N(C(C)COC)CC=C)=O)CCC2)=O)ncccc1N 80125,N1(CC)CC(C(=O)NCC2CCCN(C(c3ccccc3F)=O)C2)CC1=O 80126,c1(C(=O)NCC(Cc2ccccc2)N(C(CC=CC)=O)C)ccncc1N(C)C 80127,c1(NC(=O)Nc2cccc(-c3nc(C)[nH]n3)c2)c[nH]c2nccc-2c1 80128,CC1CCC(O)(C(=O)N(CCCNC(=O)CCCc2cc[nH]n2)C)CC1 80129,c1(OC)ncc(C=CC(=O)NCCC2(NC(c3ocnc3C(F)F)=O)CC2)cn1 80130,C1(NC(c2c(NCC)cccc2)=O)CCC(C)N(C2CCCC2OCC)C1 80131,C(=O)(C(CN(C)C)NC(=O)Cc1cc[nH]c1)N(CC(C)OC)C 80132,C(N=c1[nH]c(C#N)c(Cl)s1)C1CCN(C(CSCC(C)C)=O)CC1C 80133,c1(CC)nc(C(=O)N(CC(=O)NC(C2CCCC2)CO)CC2CC2)c(C)o1 80134,Cc1cn2c(n1)C(C(=O)NC(C)(CNC(=O)Cn1nccn1)C(C)C)CCC2 80135,CC1CN(CCNC(C2CC2C2CCCC2)=O)CC(C)(C)O1 80136,Cc1nc(C(=O)NCC2CCC(NC(=O)CN3CCNC(=O)C3)C2)ccc1C#N 80137,C=CCCCC(=O)NC1C2CN(C(C3(c4ccccc4)CC(C)(C)C3)=O)CC12 80138,C1(CCC(=O)OC)(Nc2cnn(SC(F)F)c2)CCNCC1 80139,c1(CC(=O)NC2COCCN(C(CCCC)=O)C2)ccc2ncsc2c1 80140,c1(C(N2C(C)(CNC(C3C(=C)C3)=O)CCC2)=O)cccc2c1OCC2 80141,c1(C(N(C(C=C)C)C)=O)cc(CNC(=O)CSC)nn1C 80142,C1(C(N(C2CCCN(C(=O)CSc3csc(=N)[nH]3)C2)CC)=O)CCCN(C)C1 80143,c1(C(N2C(C(C)C)C(NC(=O)C3CC3)CC2)=O)ccc2c(c1)N(C)C(=O)CO2 80144,c1(Cc2cccc(C(N(CCC)Cn3cncn3)=O)c2)nccc2ccccc12 80145,c1(CC(=O)NC2CCCN(C(Cc3c(C)nsc3)=O)CC2)cc2ccccc2s1 80146,c1(CCC(=O)NC2C(NC(C=CSC)=O)CCC2)ccccc1Cl 80147,n1(CC)cc(C(=O)NCC(C(N2CCC3(CC3)C2)=O)OC)cn1 80148,c1(C(C(=O)NCCOC(=N)O)NC(C(CC)C#N)=O)c(C)cccc1Br 80149,N1(C(C=CCCC)=O)C2CCCC1CC(NC(c1cc3cc(Cl)ccn3n1)=O)C2 80150,C1(CC)CCCCC1NC(C1(CCNC(=O)C(C2CCCC2C)=O)CCCC1)=O 80151,C1(NC(Cc2c(COC)cccc2)=O)COC2CN(C(=O)CC3CCC3)CC12 80152,Cc1ccc(-n2ncc(C(=O)NC3CCN(C)C3C)c2C2CC2)cc1 80153,CC(C)CCCC(=O)N(C(C)C(=O)NC1CCCC(F)(F)C1)C1CC1 80154,c1(NC(CN(C(C2(COC)CCCO2)=O)C)C)ncnc2c1c(Br)nn2C 80155,CCC(CCCC(=O)NCCCC(C)O)NC(=O)C(C)(C)C1CCCO1 80156,C1(C(=O)NC2CC(N(C(C(C)COc3ccccc3)=O)C)C2)CCOCC1(C)C 80157,C1(N(C(C(C)N(C(=O)C(C)C2(O)CCC2)CCC)=O)C)COC(C)(C)C1 80158,C(CNC(C1CCC(C(C)C)N1C(C1CCN1C(C)(C)C)=O)=O)(C(F)(F)F)OC 80159,CC1(C)CCC(C(=O)NCCNC(c2ccccc2OC(F)(F)F)=O)C1 80160,N1(C(C(C)C)CN2CCOCC2)CCCCCC1 80161,CC(C)(C)CC(=O)NC1CCCC1CNC(C1(C)CS(=O)(=O)C1)=O 80162,N1(C(CC2(C)CCOCC2)=O)CCC(NC(C2COC3(CCC3)C2)=O)C(F)C1 80163,N(C1CCCn2ccnc21)C(C1(NC(CC2CCC(C)(C)C2)=O)CSC1)=O 80164,C(C(=O)NCCC(C)C(C)C)(C(C)(C)C)NC(c1cc(C)n(C)c1)=O 80165,C(=O)(CCCC(=O)N1CCCC(NC(c2nncn2CC)=O)C1)OCC 80166,N12CCC3C(CCCN3CCC1)C2.c1(CN)nc(C2CC2)cs1 80167,N1(C(c2c(N)ccc(-c3nn[nH]n3)c2F)=O)CCC2CC(F)(F)CCC2C1 80168,c1(CC(N2C(CNC(C(C=C)(C)C)=O)COCC2)=O)ccc2sccc2c1 80169,c1(C(=O)NCCCCC(CO)NC(c2nnn(C)c2C(F)F)=O)cnc2sccn12 80170,C(=O)(CC(=O)N(C)C)NC(C1CC(NC(=O)CC2CSC2)C1)C 80171,c1(CC)ccc(C(N2CC(F)CC2CNC(=O)Cc2cc(C3CC3)on2)=O)cn1 80172,N1(C(CN(C)CC)=O)C2CCCC1CN(C(C13COCC1C3)=O)CC2 80173,C1(C)(CNC(c2ccn(CCCC)n2)=O)CCCN(C(C2(C)COC(=O)N2)=O)C1 80174,N1(C(c2n(CCC)ncc2)=O)CC2CN(C(=O)CCn3c(C)ccc3C)CC2C1 80175,CC(CC(=O)N1CCCC(F)(CNC(c2noc(C3CC3)n2)=O)C1)P(C)(C)=O 80176,c1(NC(CCCOC)c2nnnn2C2CCC2)cc(S(N)(=O)=O)cc(Br)c1F 80177,C1(CC2(C)N(C(=O)NC3C(c4onc(C)n4)OCC3)CCC2)CCC(CO)CC1 80178,CC(C)C(C(=O)N1CC(NC(c2cc3ccccn3c2)=O)CC(F)C1)C(C)C 80179,C(=O)(CCCCC(F)F)N1CC(CNC(C(C)CC(F)F)=O)N(C)CC1 80180,N1(C(C2C(C(C)C)C2)=O)CC(CNC(c2ccnn2CCF)=O)CC1(C)C 80181,C(=O)(CCNC(=O)COCC1(F)CC1)N(CC(C)OC(F)F)C 80182,N1(C(C(CC)F)=O)CC(NC(c2ccc(-c3ccccc3)c(Cl)c2)=O)C2(CC2)C1 80183,C1(NC(C2C(CC)OCC2)=O)CCCCC12CCCN(C(=O)C(=O)NC1CC1)C2 80184,c1(C(N2C(CNC(CSC(C)C)=O)CC(O)C2)=O)ccn2nccc2n1 80185,C1(NC(C(C)OCC#C)=O)CC2CC(NC(=O)CSc3ccccn3)CC12 80186,C1(NC(CNc2cccc(C)c2)=O)CCCC12CN(C(=O)C(F)C1CCOC1)C2 80187,CC(C)CCCCC(=O)NCC1CC(n2cc(-c3cccc(N)c3)nn2)C1 80188,n1(CC)cc(C(N2CC(NC(c3cnc[nH]c3=N)=O)C3CC23)=O)c2ccccc12 80189,N1(C(C2(OC)CCCC2)=O)CC(NC(C2CC23CC(O)C3)=O)CC(F)C1 80190,N1(C(C2(C(=O)NC)CC2)=O)CC(=O)NCC1C(=O)NCC1CC2CCC2C1 80191,C1(C)(COCCC=C)CCCN(c2ccc(Cl)cc2C(=O)OC)C1 80192,C1(NC(CC2(C=C)CC2)=O)CCC(C)N(C(c2sccc2CO)=O)C1 80193,C1(C2(O)CN(C(=O)C#CC3CCCC3)C2)(CNC(C2(F)C(C)OCC2)=O)CC1 80194,c1(CC(N2CC(=C(CN(C(C(C)NC3CCCCC3)=O)C)F)C2)=O)nncn1C 80195,C1(C(C(=O)NC(CC)C)NCC2CCCO2)CCOCC1 80196,C1(CC)CC(CC(=O)N(C2CC2)CC2CCCN2C(C2CC3CC3C2)=O)CCO1 80197,Cc1cc(C(=O)N(C2(C(N3CC(c4c[nH]nc4C)C3)=O)CC2)C)c(C)cn1 80198,Cc1cccc(-c2nc(OC(=N)O)n(CC3CC4CCC3C4)n2)c1 80199,C1(NC(C(C)OCC#C)=O)C2CCC(C2)C1C(=O)NCc1[nH]nnc1CC 80200,CN1CC(=O)N(CC(=O)NC2CCN(Cc3cnon3)CC2C)C1=O 80201,Cc1nn(C)c(Cl)c1C=CC(=O)NCCCNC(c1cnc(C2CC2)[nH]1)=O 80202,CC1CCC=C1C(=O)N1CC(C)CCC1C(=O)Nc1ccc(O)c(F)c1 80203,c1(C(N2CCCC(N(C(=O)C(C3CC3)OC)CC)C2)=O)ccc2cnccc2c1 80204,n1(CC)nc(C(C)NC(c2ccc(Cl)cc2)Cc2ccccc2)ccc1=O 80205,Cc1cc(C)c(C(=O)NC2CC3CN(C(c4n[nH]c(=N)[nH]4)=O)CC23)c(C)n1 80206,N1(CC(=O)N(C(C2CN(C(=O)C(C)CC(F)(F)F)C2)C)CC)C(=O)C(=O)N(C)C1=O 80207,C(=O)(C(Cc1ncoc1C1(C2CCCCC2)CC1)CCS(C)(=O)=O)OC 80208,c1(CC(C)C)n[nH]c(=NC(CNC(C2CCn3nncc3C2)=O)C(C)C(C)C)s1 80209,C1(NC(C2C(C)C2)=O)CCC2(CCN(C(c3n[nH]cc3[N+](=O)[O-])=O)C2)C1 80210,C1(C)(C(N(CC=C)C2CC2)=O)CC12CCN(c1cnc(=N)[nH]c1)CC2 80211,C(=O)(CC(C)(C)CC(F)F)NCC1CN(C(C(C(C)O)(F)F)=O)CC12CCC2 80212,C1(CC)(CC)CNC(=O)C1Nc1nnn(CCc2ccccc2)n1 80213,c1(C(=O)NCCC(C)N(C(=O)CNC(c2nccs2)=O)C)coc(S(C)(=O)=O)c1 80214,c1(C(N2CCCC(NC(C(CSC)OC)=O)(CO)C2)=O)cccc2oc(C)cc12 80215,c1(CC(N2CC3C(CNC(C(CC)SC)=O)(C3)C2)=O)coc2c(F)c(F)ccc12 80216,C1(N(C)C)CCC(C(=O)NC(C)(C)CNC(=O)CCC2CCCC2)C1 80217,C12(C(=O)NCC3(F)CC(NC(c4c(N(C)C)nccc4)=O)C3)CCCC1OCC2 80218,c1(C(=O)NC(C)CNC(=O)COC2CCC2)csc(S)n1 80219,c1(C(N(C2(c3ccc(F)cc3)COC2)C)=O)ccc(F)c(C(F)F)n1 80220,N(C1c2ccccc2CC1NC(c1conc1C)=O)C(c1nc(OC)c(C)s1)=O 80221,CCC(CCCC(=O)NC1CC1CN(C)C)NC(c1ccc2[nH]ccc2c1)=O 80222,N1(C(C2CC(=C)C2)=O)CCC(NC(=O)C(CC)N2CCCC2=O)C1 80223,c1(CCN2CC(CNC(C(=Cc3ccccn3)C)=O)C(C)C2)ccc(C)c(C)c1 80224,C1(C(N2C3CCC(NC(COCCCCC)=O)(C3)C2)=O)CCCCN(C)C1=O 80225,C(CC1=CCCCC1)N(C(C=CC(C)(C)NC(C(CC)O)=O)=O)C 80226,C1(n2cc(CN=S(C)(C)=O)nn2)(CCNC(=O)CC2(O)CCC2)CCOCC1 80227,C1(NC(=O)CCOC2CN(C(C3(CO)CCCC3)=O)C2)CCN2CCCC2C1 80228,c1(C(N2C(CC)CN(C(C3COC(=O)N3)=O)CC2)=O)n[nH]c2c1CCSC2 80229,C1(N(C)C=O)CCCN(C(=O)CCC2CC2)CC1.n1(CC=O)ccc(=N)[nH]1 80230,CS(=O)(=O)c1nc(Cl)cc(=NCC2CN(C(=O)C(F)CC3CC3)CCO2)[nH]1 80231,CP1(=O)CCN(CC(=O)NC2CCCC(CNC(c3ccoc3)=O)C2)CC1 80232,N1(C(C(C(C)C)F)=O)CCC(C(=O)NC2CCN(C3CC3)C2=O)C(C)(C)C1 80233,c1(C(=O)NC(CC)CN(C)C(C2(C)CNC(=O)C2)=O)cc(F)cc(F)c1 80234,Cc1ccc2nc(C(N3CCC4CN(C(c5cnsn5)=O)CCC4C3)=O)cn2c1 80235,c1(C(=O)NC(C(C)NC(c2cc(C)on2)=O)C(C)C)cc2ccc(Cl)cc2o1 80236,N1(C(C2(OCC#C)CC2)=O)CC(C)N(C(=O)Cn2nc(C)cc2OC)CC1C 80237,c1(CC)oc(C)cc1C(=O)NCC1(CCNC(c2cn(C)cn2)=O)CC1 80238,C(=O)(C1CCc2nccn21)N1CC(C(=O)NC(CC#C)C(=O)OC)N(C)CC1 80239,CN1CCN(C(=O)CCCCC2CC2)CC1CNC(c1cc(C(F)F)nn1C)=O 80240,N1(C(c2cnc(C)[nH]2)=O)CC(C)N(C(c2cn(CCO)nc2C)=O)CC1C 80241,CCCC(C)C(=O)N1CCN(CCNC(=O)CC(=O)NC2CCCC2)CC1 80242,C(=O)(CC1=CCOCC1)N1CCCC(CN(C(=O)CC2(CO)CCCCC2)C)C1 80243,CCC(CC(=O)NC1CC(C(=O)NCc2noc(C(C)C)n2)CC1O)SC 80244,c1(N2CC(NC(=O)CC3NC(=O)NC3=O)(CO)C2)ncc([N+](=O)[O-])cn1 80245,c1(C(=O)NCC2CN(C(c3c(C)ccc(N)c3)=O)C2)[nH]c2ccc(F)cc2c1C 80246,c1(CC)cc(C(=O)NC(C)(C)CN(C)C(c2cn(C(C)(C)C)nn2)=O)cc(C)c1 80247,CCCCCC(O)C(=O)N1CC(CN2CCN(C(=O)C(C(C)C)SCC)CC2)C1 80248,C1(c2nn[nH]n2)(CC)CCN(C(=O)OC(C)(C)C)CC1.C12CCN(C1C)C2 80249,c1(C(N(CCCCN(C)CC)C)=O)ccnc(C2CC2)n1.c12nc(co1)NC2=O 80250,N1(C(C2(CC=C)COC2)=O)CCC(C)N(C(=O)CC2CC3CCC2CC3)CC1 80251,c1(C(=O)NC(CNC(c2ccc(OC)s2)=O)CO)cn(C)c(=O)cn1 80252,c1(C(N2CC(C=C)(CC(N3CCC4(CC3)CC4CO)=O)C2)=O)ccn2cncc2c1 80253,c1(NC2CCN(C(C)C)CC2)ccc(S(=O)(=O)NC(C2CSC2)C)cc1Br 80254,C1(SCC(=O)O)CSCCO1.C1(C(n2cc(C)nn2)CC)CCN(C(=O)C)C1 80255,CCCCC(C(=O)N1CCN(C2CCC2)CC1)NC(=O)CN(C)C(C)C 80256,N1(C(c2scc(C)c2)=O)CCC(C(F)CNC(=O)C(F)(F)C2(O)CCCC2)CC1 80257,C12(NC(C(C)NS(C)(=O)=O)=O)CCC(CC1)N(C(=O)CCc1nc(O)n[nH]1)C2 80258,C1(C(=O)NCCC(=O)N(C)CC)CC12CCS(=O)(=O)CC2 80259,c1(C(=O)NCC(C)CN(C)C(C2CC(C)(C)O2)=O)cc(Cl)c(F)c(Cl)c1 80260,Cc1nc(C2CC2)ncc1C(=O)NCC1(C)CN(C(=O)CC2CCSCC2)CC1C 80261,CC(CNC(=O)OC(C)(C)C)CC(=O)NCC(C)N(C)C(C12CC(F)(C1)C2)=O 80262,Cn1nnc2cc(C(=O)NCCN(C3CCCCCC3)C(C3CCC3F)=O)sc12 80263,N1(C(C(CC)O)=O)CCC(CO)C(NC(=O)Cc2c(Cl)cnn2C)C1 80264,c1(C(=O)NCC2CCC(NC(C3(N(C)C)CC3)=O)C2)nnn(C)c1N 80265,Cc1ncc(CCC(=O)NC(C(=O)NC2CCNC2=O)C2(C)CC2)o1 80266,Cc1cc(F)cc(F)c1S(=O)(=O)NC(C1CCc2nnnn2CC1)=O 80267,N1C(=NCCCN2CCCCCC2)NCC(C)C1C.C1(C(N)=O)(NC2CC2)CCCCC1 80268,N1(C(C2CC(C)CC(C)C2)=O)CCCN(C(=O)CCSc2ccccn2)CC1C 80269,c1(CC(C)C)cc(C(=O)NC2(c3ccc(NC(=O)C(=O)NC)cc3)CC2)ncn1 80270,C(=O)(C(C)(C)CCNC(C1CC(F)C(=O)N1)=O)NCC1CCN(C(C)=O)C1 80271,C(C)(C)(CCCCC(=O)NC1CN(C(C2CCOC3(CCC3)C2)=O)C1)OC 80272,C1(C(N2CCC(N(C(CSC)=O)C)C2)=O)CC12CCCCC2 80273,CC1CCN(C(C2CCCCCN2Cc2ccccc2F)=O)C(NC2CCC2)C1 80274,C1(NC(c2ccc(CC)nc2)=O)Cc2ccccc2C1NC(=O)C(C)NC=O 80275,C12(CNC(c3nc(C(C)C)sc3)=O)CCC1CN(C(c1ccc(O)c(N)n1)=O)C2 80276,N1(C(C#CC(C)(C)C)=O)CCCCC12CN(C(=O)C=C1CCCCC1)C2 80277,c1(C(C)C(=O)NC2COCC2NC(C2(CC#N)COC2)=O)c(F)cccc1F 80278,N1(C(Cc2c(C)noc2)=O)CCN(C(=O)C2=NOCC2)CC1CF 80279,C1(OC)CN(C(=O)C(O)C2CCCC2)CC1C(=O)Nc1ccc(F)nc1 80280,c1(C(=O)NCCC(=O)Nc2cnn(CC(F)F)c2)ccc2c(c1)OCCO2 80281,CCC(C#N)C(=O)NCCC(O)C(N1CCCN(C(C)=O)CC1)=O 80282,c1(C(=O)NCC#CCNC(C(CSC)OC)=O)cccc2c1OCCO2 80283,c1(C(N2CCC(OCCNC(c3ccns3)=O)C2)=O)ccc2n[nH]cc2c1F 80284,C1(C(=O)NCC2CN(C(c3ccnc(CC(C)C)n3)=O)C2)CC2CCC1C21CC1 80285,C(=O)(CC(C1CC1)OC(C1CCN1C(=O)CC1CN(n2cnnn2)C1)=O)NC 80286,c1(Cn2cc(CNC(CC)CC(C)C)nn2)c(OC)cccc1Cl 80287,N1(C(c2cc(CC)nc(O)c2)=O)CC(NC(=O)Cc2cnco2)C2(CCCC2)C1 80288,C(c1nnc(CC(=O)N(CCN(C)CC)C)o1)=CC(=O)NC1(C(C)C)CC1 80289,C12(CNC(c3ccc(CC)o3)=O)CN(C(C3(C)CCOC3)=O)CC1CCO2 80290,C1(C(N(C)Cc2c(C)nsc2)=O)CC12CCN(C(c1ncccc1Cl)=O)CC2 80291,CC#CCCC(=O)N1CCC(NC(c2cc(C(C)=O)cs2)=O)C1C1CC1 80292,C(C(N=[N+]=[N-])C(=O)NCC(C(C)C)NC(c1ccncc1O)=O)OCC 80293,c1(NC(=O)NC2OCC(C)C2)cc(Cl)ccc1F 80294,N1(C(C(P(C)(C)=O)O)=O)CCC2(CCN(C(=O)CSc3nc4ccccc4o3)C2)C1 80295,C(C)(C)(C(C)(C)C)NC(CC1CCN(C(C(C(C)C)=O)=O)C1)=O 80296,c1(CNC(CCCC)(C)c2nnnn2C2CC(F)(F)C2)ccc(O)c(Br)c1 80297,c1(CCNC(=O)Nc2ccnc(N3CCOCC3)c2)ccc(F)c(F)c1 80298,Cn1cnc(C(=O)NC(C)(C)CCCNC(C2CC23CC3)=O)cc1=O 80299,C1(CNC(C2(NC(C)=O)CCC2)=O)CCN(C(c2cnc(CC(C)(C)C)o2)=O)C1 80300,c1(COCC(=O)NCCNC(=O)CN2CCCC2)ccccc1.C12CC(C1)NC2 80301,c1(C2(C(=O)NCC(CN(C)C(c3sccc3F)=O)(C)C)CC2)ccnc(Cl)c1 80302,C1(N(C(=O)C(O)CC(N)=O)C)CC2CCC(C1)N2C(c1ncc[nH]c1=O)=O 80303,C(=O)(C1=CCC(NC(=O)C(=O)NC(C)C)C1)NC(C(=O)OC)C 80304,C1(C#N)(C(N(CCCCCC)CCNC(C2CCOCC2)=O)=O)CCOC1 80305,C1(CNC(C(c2cn(C)nc2)(F)F)=O)CCN(C(C2CC2[N+](=O)[O-])=O)C1(C)C 80306,c1(C(N2CC(O)(C(C)NC(COC(C)=O)=O)C2)=O)c(Cl)cc(Cl)c2cccnc12 80307,N1(C(C(C)CNC(=O)OC(C)(C)C)=O)CCC2CN(C(=O)NC3CC34CC4)CC12 80308,CC1CC(C2CN(C(C3CN(C(C4CC4Cl)=O)CCO3)=O)C2)=NO1 80309,C1(C(=O)NC2(CC)CN(C(C34CCC(OC)C3C4)=O)C2)COCCN1C 80310,CC(C)CC(C(=O)NCC1CCCCC1(F)F)ONC(c1ccsn1)=O 80311,c1(NC(CN(C2CCN(C(C(CC)(C)C)=O)C2)C)=O)cc(OC)ncc1Cl 80312,c1(C(=O)NC(C2CN(C(c3c(C(C)C)ncs3)=O)C2)C)cccc(Br)c1O 80313,c1(N2CC(C)=C(C)C2)nc(N2CCC(C)(CCO)CC2)nc2c1CC(C)CC2 80314,c1(C(N(C2CCN(C(c3c(C)n[nH]c3)=O)CC2)CCO)=O)cc2ccsc2n1C 80315,c1(C(=O)NCC(C)(CC)NC(CCOCC)=O)ccnc(C(F)(F)F)n1 80316,c12ccc(cc1)S(=O)(=O)N(C)C(=O)NCC2C.c1(SC2CC2)c(F)cccc1F 80317,C(CC(F)F)(C(=O)NOCC1CCCO1)N(C(c1c(OC)n(C)nc1)=O)C 80318,c1(NC(C(C)NCC2CC2)=O)ncc(C(=O)NCc2n[nH]cc2CC2CC2)cn1 80319,C1(OCCC)CCCCC1C(=O)NC(C)CNC(c1c(C)noc1C1CC1)=O 80320,c1(C(=O)NC2CCC(NC(C=CC(=O)N(C)C)=O)C2)cn(C)c(=O)nc1O 80321,C12(C(N3C(C)CN(C(c4ncc(F)cn4)=O)CC3)=O)CCC(C)(CC1)CO2 80322,c1(CC)ccc(F)c(C(N2CCN(C(c3snc(C)c3N)=O)C(CF)C2)=O)c1 80323,C1(NC(c2cnc(Cl)s2)=O)CCCCCC1C(N1CC(Cc2ccoc2)C1)=O 80324,C#CCC(CC(F)F)C(=O)N1CC(NC(=O)CC2CC(C3CC3)C2)C2CCCC12 80325,C1(CNC(C2CCN(C(CC)=O)CC2)=O)CC(C)CN(C(=O)C=C2CCCC2)C1 80326,n1(C(C)C)ncc2c(N3CC(F)C(F)C3)[nH]c(=NCC3C=CCCC3)nc12 80327,c1(C(=O)NCCC2CCN(C(C(C)N(C(C)=O)C)=O)C2)onc2c1CCCC2 80328,C1(C(N2CC(NC(COC)=O)CC2(C)C)=O)Cc2ccccc2NC1=O 80329,N1(C(CN(C(CCSCC(C)C)=O)CC2CC2)=O)CC(C2CCCC2)C1 80330,C1(C=O)CCc2nnnn2C1.c1(C(=O)NCC(C)OC(F)F)ncsc1C(F)(F)F 80331,Cc1ccc(CC(=O)NC(CNC(c2scnc2C(F)F)=O)CC(C)C)cc1O 80332,CC1CC(=O)NCC1C(=O)NCCC1CCCN(C(=O)C(C)C2CCC2)CC1 80333,c1(C(N2C(CC(=O)NCCCOC(C)C)CCC2)=O)ccc(-n2ccnc2)cc1 80334,c1(OC)c(F)cc(Nc2ncc(CC(=O)NCc3ccncc3)s2)cc1F 80335,C#CC(CNC(C1CN(C(=O)CC(F)(F)F)CCC1O)=O)CC(C)(C)C 80336,Cc1nc(NCC(C(C)(C)C)NC(=O)C=CSc2ccccc2)cc(C#N)n1 80337,c1(CCC(N2CC(O)(CC(=O)NCCCC)C2)=O)ccc2c(c1)OCO2 80338,C(CCC(N)=O)(C(=O)N)n1cc(C(C)NC)nn1.c1(CC2CCCC2)ccc(Cl)s1 80339,c1(C(=O)OC(c2ccccc2)C(=O)OCC)ccnc2[nH]cnc12 80340,CC1OCCCC1C(=O)NC12CC(C(=O)NCCC3CC(O)C3)(C1)C2 80341,N1(C(C(CCSC)NC(=O)CSCCN2CCC2)=O)CCCCCCC1 80342,C(=O)(CC(C(C)C)NC1CCC(=O)NC1)OCC 80343,c1(C(=O)NC)cccc(CNC(C2CC23CN(C=O)C3)=O)c1.C1C(=O)N1.C(C)C 80344,C(C(=O)N=c1ccn(CCCO)[nH]1)=CC(=O)NC(c1ccccc1)COC 80345,C1(C(N(CCOC)CCNC(=O)C(C)(C)CC2CC2)=O)CCC(=O)CC1(C)C 80346,c1(C(=O)NCCCCCCC=C)ccc(O)c([N+](=O)[O-])c1 80347,Cc1cc(C)cc(C=CC(N2CC3(CCCC3NC(=O)C(F)C3CCC3)C2)=O)c1 80348,C1(C(N2C(C(=O)NCC(C)C(F)(F)F)CCC2C2CC2)=O)CC2(CC(=O)C2)C1 80349,C1(CC(=O)NCC(C)(C)COC)CN(C(=O)CCCOC)CCC1C.C(=O)OCC 80350,Cc1cc(C#N)ccc1C(=O)NCCOCCNC(c1cnc2ccnn2c1)=O 80351,N1(C(C(C(C)C)C#N)=O)C(C)CC2CN(C(c3sccc3CN(C)C)=O)CC12 80352,N1(C(CN(CCC)C)=O)CC2CC1CN(C(C1CC(C)OC1C)=O)C2 80353,n1(C(C)C)cc(C(=O)N(C2CCN(C(=O)C=CC(F)(F)F)C2)CCO)c(O)nc1=O 80354,Cc1ccc(OCC(N2CCC(NC(C3CC3(F)Cl)=O)CC2)=O)cc1C 80355,c1(C(=O)NCC(C2CCC2)NC(C(C)N(C(C)=O)C)=O)ccc(C(C)C)s1 80356,C1(CC(N2C(C)(C(=O)NC)CC2)=O)CCCN(C(C2C3CN(C)CC23)=O)CC1 80357,N1(C(CNC(CC)=O)=O)CC=CC1(C(=O)N(C)Cc1cnn(CC)c1C)COC 80358,c1(OC)cccc2c1C(C(=O)N1CCCC1CN(C)C(C1(CCO)CC1)=O)CC2 80359,Cc1nn(C)c(C)c1C1OCCO1.C12(CCOC1)CC(=O)N2 80360,CC1(C)C2CCC(C(N3CCCC(N(C(=O)CP(C)(C)=O)CCO)C3)=O)C1C2 80361,CC(C(C)(C)C(=O)N1CCOC(C)(C)C1)NC(c1ccc(F)cc1)=O 80362,c1(C(N2CC(CCNC(CNC(C)=O)=O)C2)=O)ccc2c(c1)C(=O)NC2 80363,CCCCC(CNC(c1n[nH]cc1C(C)C)=O)NC(c1cnccc1Br)=O 80364,CC1CCCCC1(C)C(N1CC=CC(NC(c2cc(Cl)ncc2Cl)=O)C1)=O 80365,N1(C(CCC)=O)CC2CS(=O)(=O)CC2(NC(c2cnn(CC(F)(F)F)c2)=O)C1 80366,C12(CNC(C(c3ccccc3)OC)=O)CC(NC(=O)C=CS(C)=O)(C1)C(C)(C)O2 80367,C1(C(=O)NC(C)Cc2cccnc2)CC(NC(c2cccc(F)c2)=O)C1(C)C 80368,N1(CCCC)CSCC1C(=O)N(CCC(C)NC(=O)C=CC(=O)OCC)C 80369,C=CCCCCC(=O)N1CCC(CNC(c2nc(C)n(-c3ccccn3)n2)=O)C1 80370,C(=O)(CCCCCCCC1CC1)N(C1CCCN(C(C(CC)=CC)=O)C1)CCO 80371,C1(CC=C)(NC(=O)Cc2ccnn2C)CCN(C(=O)CCc2ccoc2)C1 80372,C(C)(CCC)=CC(=O)N(CC(=O)N(CC(=C)C)CC)C(C)C 80373,S(=O)(=O)(c1cc2ccccc2s1)N1CCCC(C(=O)NCC2CCOCC2)C1 80374,c1(CNC(C2CC2CNC(C2C3CCCCCC23)=O)=O)ccc(F)c(O)c1 80375,Cc1c(C(C(N2CCN(C)C3CC23)=O)N(CCCF)C)cccc1F 80376,N1(C(=O)C=Cc2cscn2)CCOC2C(O)CC12.O=C1C(O)C2CN1C2 80377,N1(C(C2C(NC(=O)NC(C)(C)CO)C2)=O)CCCOCC1 80378,Cc1cccc(C(N2CCCC(NC(C3CCC(C(C)(C)C)CC3)=O)C2)=O)c1Br 80379,C1(C(N(CC(C)C)CCOC)=O)CC(CCNC(=O)C(F)n2cccn2)C1 80380,S(=O)(=O)(c1ccc(OC(C23CC(CO)(C2)C3)=O)cc1C)NC(CCC)CCO 80381,C1(CNC(CN(C(C)=O)C)=O)(CNC(C2C(C)(C)C2(C)C)=O)CCOCC1 80382,c1(COCCOC)ccc(-c2cn(-c3ccc(OC)cc3)nn2)cc1 80383,C1(C(=O)NC2CN(C(c3ccc(C)nc3)=O)CC2C(F)(F)F)C2C3CCC(C3)C12 80384,C1(NC(CC(=O)NCC#C)=O)CCN(C(=O)C=Cc2cncn2C)C1C 80385,Cc1ccc(C(=O)NC2CCCC(NC(=O)CCC3CCOC3)C2)nc1O 80386,N1(C(C23CC(COC)(OC2)C3)=O)CC(NC(C2(C)CCC(C)C2)=O)C(C(F)F)C1 80387,C(=O)(C(CC(F)F)C1CC1)NCC(N(OC(C(=O)OC)CC1CC1)C)=O 80388,N1(C(C(C(C)C)OC)=O)CCC(C2CN(C(c3cc(OC)ns3)=O)C2)CC1 80389,CCCC(C)(CC)C(=O)NC1CC(N(C)C(c2cc3occc3s2)=O)C1 80390,c1(OC)cccc(C(C(=O)NCCC#N)N(C)Cc2cncs2)c1Br 80391,C#CC1CN(C(=O)CC=C(Cl)Cl)CCN1C(=O)COCC(c1ccccc1)C 80392,c1(C(=O)NCCCCNC(C2CN(C(N(C)C)=O)C2)=O)csc([N+](=O)[O-])c1 80393,C(=O)(C(F)CC1CN(C(=O)COCCF)C1)N(C1CCCCO1)C 80394,C1(C)(C(N(c2c(C(=O)NCC(C)C)cccc2)C)=O)CC(C(C)(C)C)=NO1 80395,c1(Cc2cn(CC(CC)(CC)CCO)nn2)ccc2c(c1)CNC2 80396,c1(CCC(=O)NC(C2CCN(C(Cc3nnc(C)o3)=O)C2)C)ccc(C#N)cc1 80397,Cc1cc(CC(=O)NC2CCC2NC(=O)C(N2CCCC2)C2CC2)cc(F)c1 80398,CN=O.C(C)(C)(C)N(C1(N(C)C=O)CC1)C(=O)OC(C)(C)C 80399,C1(C(N(CC(C)NC(c2c(CCC)nco2)=O)CC)=O)CCCCC1O 80400,C12(NC(Cc3scc(C)c3)=O)CCCC(NC(=O)CC(C)(C)O)(C1)C2 80401,c12cnc(c(Br)c1)[nH]c2=O.c1(C2(NC(C3CC3)=O)CC2)ccccc1Br 80402,C1(NC(=O)CO)CCCCC1C(=O)N1CCCCCC1.c1(O)cccc(Cl)c1 80403,c1(C(=O)NCC(COC)(C)OC)cc2c(s1)CC(C)(C)C2 80404,C=C(C)CCCC(=O)N1CC(c2ccccc2)(CNC(=O)CC2CNC(=O)O2)C1 80405,N1(C(Cc2nnc(C)s2)=O)CCSCC1CCNC(=O)C=CC1CCOC1 80406,Cc1csc2ncnc(NC3CC(C)CN(C(c4ccc(F)s4)=O)C3)c12 80407,C(CN=c1[nH]c(=NCc2cccnc2C)[nH]c2c1COCC2)OCC 80408,c1(C(=O)OC)cnc(NC(C2CC2C(=O)Nc2ccc(C(C)O)cc2)=O)cn1 80409,c1(C(=O)NCC(C)NC(C2CC2c2cccc(F)c2)=O)ccc(F)c2c1CCC2 80410,C1(CNC(c2cc(C)[nH]n2)=O)CCC(C)CN1C(c1cncc(NC(C)C)c1)=O 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80428,C1(C#N)(C(=O)NCC2C(CC(=O)N(C)CC3CCCCC3)C2)CC12CCC2 80429,N1(C(CC(=C)Br)=O)CC(NC(=O)COc2ccc(Cl)nc2)CC(C)C1 80430,CC1(NC(c2ncccc2CO)=O)CCN(C(=O)CC2COCC(C)(C)O2)CC1 80431,C(=O)(C1=CCC(C)(C)CC1)N1CCC(NC(Cc2ccc(CC)cc2)=O)C1C 80432,Cc1cncc2cc(C(N3CC(N(C(=O)C(O)C4CC4)C)C4(CC4)C3)=O)sc12 80433,Cc1ccccc1C(CNC(c1cc(-c2ccco2)no1)=O)NC(C1(SC)CC1)=O 80434,C1(C(C)=O)(NS(C)(=O)=O)CCCCO1.N12CCCCC1Cc1cn(nn1)CC2=O 80435,c1(C(C(=O)NCC2(CNC(CSCC=C)=O)CC2(F)F)(C)C)cccc(O)c1 80436,N1(C(C2N(C(C(C)Oc3ccc(F)cc3)=O)CC(O)C2)=O)CCC2(CCCO2)C1 80437,C1(C(=O)OC)N(C(=O)C(CN(C)C)NC(C2(C(C)(F)F)CC2)=O)CC1(C)C 80438,C(CC(C)C(=O)NCC1(NC(=O)CN2CCCCC2=O)CC(F)(F)C1)OC 80439,C(=O)(CC1=CCCC1)NCCN(CC(C)O)C(c1ccc(Br)nc1O)=O 80440,C1(C(N2C(C=C)CCC2)=O)CC2CCC1N2C(=O)C(C)=NOCC#N 80441,N1(C(C(C)(C)N(C)C)=O)CC(CNC(=O)CC2=CCCC2)C(C)(C)C1 80442,C1(NC(C(C)(C)c2cc[nH]n2)=O)CCN(C(C2CCCO2)=O)CC1 80443,N1(C(CCn2c(C)nc(C)n2)=O)CCCC(C)(CNC(C2CC3(C2)CC3F)=O)C1 80444,C1(C(=O)NCCC(C)NC(=O)C(C)(C)C#N)COc2ccc(Cl)cc2C1 80445,C1(C(=O)NCC(C(=O)N2CC(N(CCC)C)C2)SCC)CCCCC1OC 80446,Cc1nc(SCC(N2CC(CO)(NC(=O)Cn3nnc(=N)[nH]3)C2)=O)n[nH]1 80447,C(CCC(C)(C)NC(=O)C(c1ccccc1)F)NC(c1c(CC)c[nH]n1)=O 80448,N1(C(CN)=O)CCCC2CN(CCO)CCC12.CCS(=O)(=O)N(CCCOCCOC)C 80449,Cc1cc(C(N2CC3(CCC3)CC2CNC(c2cc(O)no2)=O)=O)ncc1C#N 80450,CC(C)(C)C(O)C(=O)N1C2CCC1C(NC(c1cnc(S)nc1)=O)C2 80451,C12(NC(c3c(CC)nco3)=O)COC(C1)C(NC(c1ccnc(Cl)c1OC)=O)C2 80452,C1(NC(C2C(C(C)C)C2)=O)CC2(C1)CN(C(c1cnn(CC3CCOC3)c1)=O)C2 80453,n1(CC)cnc(CCNC(C2CCCC2CN(C(=O)CCn2cnc(=N)[nH]2)CC)=O)c1 80454,C(=O)(C(O)CC(F)(F)F)NC1(CO)CCN(C(CCCc2ccc(C)s2)=O)C1 80455,C#Cc1cccc(CCCC(=O)NCc2ccc(Cl)cc2C2(S(C)(=O)=O)CCC2)c1 80456,c1(C(C)C)cccc(C(=O)NCC2C3CN(C(=O)CN(C)C(N)=O)CC23)c1 80457,c1(NC(c2nccc(-c3ccc(C)nc3)c2)=O)cc(S(C)(=O)=O)ccc1C 80458,C1(C(=O)OCC)COCCN1C(C1(C)CCN1C(C1CC=CCC1C(F)(F)F)=O)=O 80459,C1(NC(C2CC(=C)C2)=O)CC=C(C(=O)NCc2ccnc(CO)c2)C1 80460,C1(N(C)C(C2(C(=O)N(C3CCCC3(F)F)C3CC3)CC=CC2)=O)CN2CCC1CC2 80461,N1(C(CC(C2CC2)NC(C(COC)NC(C)=O)=O)=O)CC(C)CC(O)C1 80462,N1(C(C2(SCC)CC2)=O)CC2(CC(NC(c3c(C)ncn3OC)=O)CO2)C1 80463,c1(C(N2CCCC(C(=O)NCC3(C#C)CCCC3)C2)=O)cnc(O)c(Cl)c1 80464,C1(C(=O)NC(COCC)C(=O)NCc2oc(CC)nc2C)CCCC(=O)N1C 80465,C(=O)(CC(C)CC(=O)N1CC(CNC(=O)CC23CCC(CC2)OC3)C(F)C1)OC 80466,C1(OC)CC(C(=O)NC2CC2(C)C)N(C(=O)Cn2c(O)nnc2O)C1 80467,C1(NC(C(C)=C(C)C)=O)CN(C(c2ccc(SC(F)(F)F)cc2)=O)C(C)(C)C1 80468,c1(C(=O)NC(C)CNC(=O)CCCC2CC2C)cc2ccccc2oc1=O 80469,N(C1CCc2ccc(-c3ccccc3)cc21)Cc1ccc(C(F)(F)F)s1 80470,CC1(C)CN(C(=O)CC2CCCO2)CCC1NC(=O)CCc1ccc(Cl)cc1 80471,c1(C(N(C)CC2N(C(C3CCN(C)CC3)=O)CC(F)C2)=O)nnn2c1CCC2 80472,C1(O)(CC(=O)NCCC2CCCN(C(c3scc(C)c3)=O)C2)CCCN(C)C1 80473,C=C(Cl)CC(C(=O)N1CC(F)(F)CC1C)NC(C1CCC(C(N)=O)C1)=O 80474,C1(NC(COC2(C)CN(C(=O)Cc3ccoc3)C2)=O)CC2CCC1C2 80475,C1(NC(c2cn(CCC)nn2)=O)CC2CC1N(C(=O)CCN(C)CC)C2 80476,C1(C(=O)NC2CCCC(C(=O)NCCC3CC(C)OCC3)C2)CC2CCC(C1)O2 80477,O(N1CCC(CC(=O)NCC(O)CN(C(=O)Cc2cn[nH]c2)C)CC1)CC 80478,C1(C(=O)NCC(C)CNC(=O)C=CC2CCOC2)CCc2c[nH]nc2C1 80479,c1(C(=O)NCC(CC)NC(c2cc(C(F)F)[nH]n2)=O)cc(F)cc(Br)c1 80480,O=C(CC(F)(F)C(F)(F)F)NC1CC2CC1CN2C(C1(CF)CCOCC1)=O 80481,C1(CNC(C(C)=C(CC)C)=O)COC(C)(C)CN1C(C1CCCCC1)=O 80482,C1(CNC(C(c2ccc(OC)cc2)=O)=O)CCN(C(=O)C2=NNC(=O)C2)C(C)C1 80483,N(C(=NCCC1COC(C)(C)C1)NCC(=O)NCCOC)CC=C 80484,Cc1nc(O)ccc1-c1nc(C2CCCN(C(=O)CSC(=N)N)CC2)no1 80485,Cc1ccc(CO)cc1NC(=O)CCC1CC(NC(c2cccn2C(C)C)=O)C1 80486,C(=O)(C1Cc2ccccc21)NC(CC(C)NC(c1cc(OC(C)C)ncc1)=O)C 80487,C(N=C(NC1CC1)N1CCC2NC(=O)OCC2C1)c1nn(C)c2c1cccc2 80488,CC(CCC(=O)NC1CN(C(C2CC2Br)=O)C1)N(C)C 80489,CC1(CNC(=O)CCCC#N)CCN(C(=O)COCC2CCCO2)CC1 80490,C1(C(=O)N(C2CCCCC2)CCO)CCCC(NC(c2cn[nH]c2)=O)C1 80491,CC(O)(CC(=O)NC1CC1C(N1Cc2ccc(Cl)cc2C1)=O)CC(=O)O 80492,C1(NC(C2CC(OCC)C2)=O)CN(C(c2csc(-c3ccco3)n2)=O)CC1C 80493,c1(CNC(=O)NC(CC(=O)OC)CC(C)C)cccc2nc(CO)[nH]c12 80494,C12(C(N(CC(C)CNC(c3cc([N+](=O)[O-])nn3C)=O)C)=O)CCCN(CCC1)C2 80495,c1(C(=O)NCC(C)NC(c2cccc(SCCC)c2)=O)cnn2c1CCCC2 80496,N1(CCCNCc2ccc(C)o2)C(C)CCCC1C 80497,S(=O)(=O)(c1cccc(C(C(=O)OC)NC2CCCCCC2O)c1)NC 80498,C1(CCNC(c2nn(CC)c(C3CC3)c2)=O)CCCN(C(=O)C(N)=O)CC1 80499,c1(N(C)CC2CCN(C(C3C(C#C)C3)=O)C2)ccc2c(n1)CCC2=O 80500,C1(CC=C)(NC(c2cnc(C)o2)=O)CCCN(c2cc(C)nc(SC)n2)C1 80501,N1(C(C(C)(C)C2CCCO2)=O)CC(CO)C2(C1)CN(C(=O)C(C1CCCCC1)F)C2 80502,CCC(CCCC(=O)NCCN1C(=O)CNC1=O)NC(C1CC(O)C(F)C1)=O 80503,Cc1oc(CO)cc1C(N1CCC(F)(C(N2C3COCC2C3)=O)C1)=O 80504,C1(CN(C(C(C)OCc2cccc(Cl)c2)=O)C)COCCN1C(=O)C(F)(F)CO 80505,C(=O)(C(CC)C(=O)N1CC=C(CNC(=O)CN2CCCC2CO)CC1)OC 80506,N1(C(c2nnn(C(C)(C)C)n2)=O)CCC(C(F)(F)F)C(NC(=O)C(C#N)C2CC2)C1 80507,C1(C(N2CC(CN(C(=O)COCC3(F)CC3)C)OCC2)=O)Cc2cscc2C1 80508,c1(CCC)cc(C(=O)NCc2ncoc2CCNC(=O)CC2CC2C)ccn1 80509,N12CCC(OCCC(=O)N(CCCO)C)(C1)OCC2=O.C(COCCOC)OCC 80510,C(CC(F)(F)Cn1cc(-c2conc2C(F)(F)F)nn1)NC(C1CCCCO1)=O 80511,N1(C(c2c(C)nn(C)c2)=O)CCN(C(c2cc(C(C)C)ccc2F)=O)C(CF)C1 80512,c1(C(N2C(CC#N)CCCC2)=O)ccc(Br)c(C(N)=O)c1 80513,C1(CC(=O)NC2C(c3c(C)n(C)nc3)N(C)C(=O)C2)CCCCCC1(F)F 80514,Cc1nn(C2CCC2)cc1C(N1CC2CC2(NC(=O)CC2OCCC2C)C1)=O 80515,Cc1cccc(C)c1CC(N1CC(NC(c2ccn(C3CC3)n2)=O)C2(CC2)C1)=O 80516,C1(NC(C2(CSC)CCC2)=O)CC(C)CN(C(=O)CC2CCOC2)C1 80517,C1(C(=O)NCC(COC)C)C=CCN1C(=O)C=C1CCCCC1 80518,C1(NC(c2cc(C)c(C(C)C)cc2)=O)CCSC12CN(C(C1CC13CC3)=O)C2 80519,C1(C(=O)NCCCN(C(CN(CCOC)C)=O)C2CSC2)CCCO1 80520,C1(C(=O)NCc2ncc(C)s2)CC2(CCN1C(C1CC(C)CCO1)=O)CC2 80521,c1(C(=O)NC(CCC)C(=O)O)cnc2c(c1)C(N)CCC2 80522,C(C1=CN(Cc2ccccc2)CCC1)(c1nnnn1C)NCC(C)(C)CCCl 80523,CC#CCCCC(=O)NCC12CC1CN(C(c1ccccc1OC)=O)C2 80524,c1(NC(CN2CCCC(C(=O)Nc3cccc(F)c3)C2)=O)c[nH]c2cccnc12 80525,C1(NC(c2c(CC)nns2)=O)CCC(C)N(C(C2(COC)COC2)=O)C1 80526,CCC(COC)C(=O)N1CCC=CC1C(=O)NCC(O)C(C)(C)O 80527,C1(CNC(C(C)C2CCCC2)=O)C2CN(CCCOc3cccc(Cl)c3)CC12 80528,c1(C(=O)NC(C2(O)CN(C(C3(CC)CC3(F)F)=O)C2)C)cnc2ccccn12 80529,C1(CNC(c2cc(C)c(Cl)cn2)=O)C(C2CC2)CCN1C(=O)CCc1cnco1 80530,C1(CC(=O)NC2(C)CC(C(=O)NC(C(=O)OC)C3CCC3)C2)CCCN(C)C1 80531,C1(C(N2CC(COC)(NC(=O)CC3CCC(=O)O3)C2)=O)CC2C=CC1O2 80532,C1(NC(CC)=O)CCC(CNC(C)=O)CC1.c1(N2C(C)C2=O)ccncc1 80533,N1(C(=O)C(Cl)=CCl)CCC2CN(C(=O)C(F)(F)c3ccsc3Cl)CC2C1 80534,N1(C(c2c(C)sc(O)n2)C(=O)NCSc2ccccc2)CCC2(CC1)CNC(=O)O2 80535,C1(CC(=O)NCCOCCCNC(C2CC(CC)C2)=O)CCCC2CCCCC12 80536,C12C=CC(C1)CC(=O)N2.C(CCCO)N(C(CC1(CC(=O)OC)CC1)=O)C 80537,C1(C(=O)NC(C2(O)CN(C(c3cc(N(C)C)ccn3)=O)C2)C)CC(C2CC2)=NO1 80538,C(=O)(CCCC(C)C)NC(C(=O)N(CC(=O)OC)CCC)CCOCCO 80539,C(=O)(C(C)C(F)(F)F)N(C(=O)Cc1cn(Cc2nnn(C(C)(C)C)n2)nn1)CC 80540,C(=O)(C1=CC(C)(CC)C1)NC(C1(O)CN(C(c2c(CCC)[nH]cc2)=O)C1)C 80541,N1(C(=O)C=Cc2cc(Cl)cc(Cl)c2)CCOC2(C1)CN(C(=O)COCC(F)F)C2.C 80542,CC(CC(=O)N1CC2(CNC(c3ccc4nnnn4c3)=O)CC1CO2)C(C)(C)C 80543,c1(C(N(C(CNC(C2C3CCCC23)=O)C(C)C)CCOC)=O)cccc(OC)c1 80544,C(=O)(C1CCc2ccccc21)N1C(CNC(c2cncs2)=O)CCCC1 80545,c1(C(C)C)cc(N2CCC(CF)(NC(=O)Cc3ccc(F)cn3)C2)nc(Cl)n1 80546,C1(NC(=O)NCCc2ncc(-c3cccnc3)[nH]2)CCCCCCC1CO 80547,Cc1c(Br)ccnc1C(N1CCOCC(CNC(=O)C#CC(C)C)C1)=O 80548,c1(C(N(C2(CC(=O)NCC(O)CC(F)(F)F)CC2)C)=O)cccn2nccc12 80549,N1(C(=O)OC(C)(C)C)CCC(NCC2=NC=c3[nH]ncc3=NC(=N)N2)C2(CCC2)C1 80550,CC(C)(CC(F)C(=O)N1CCC(N2CCCC2)C1)NC(c1cccc(CO)n1)=O 80551,Cc1nn(C)c(C(=O)NCCCN(C)C(C2CCCCN2C)=O)c1Br 80552,N1(C(C(C)OCCC(C)C)=O)CCC(C(C)CNC(C2(C)CCCO2)=O)CC1 80553,C12(C(=O)NCCN(OC)C)CCCC1CCN2C(C1CCOCC1)=O 80554,N1(C(c2n(COC)ncc2)=O)CCC(NC(=O)C(N2CCN(C)CC2)C)C12CC2 80555,CC1(C)CC(C(=O)NCCC2(C)CCCC2)CN1C(c1ccc(C#N)cn1)=O 80556,N1(C(C(CC2CC2)SC)=O)CCC(c2ccccc2)(NC(=O)C(C)C(F)F)C1 80557,c1(OCC(=O)NC(CNC(c2c(CC)c[nH]n2)=O)C2CC2)nn(C)cc1[N+](=O)[O-] 80558,C1(CC(=O)NCC2CC2CNC(=O)C(c2ccc(C)s2)C)(CC)CCOCC1 80559,C#CCC(CC(F)F)C(=O)N1CC(CC(N2CC(CC(C)(C)C)C2)=O)CC1C 80560,C(=O)(C1=NNC(=O)C1)NC1C(C(C)C)N(C(=O)CC(C)(C)O)CC1 80561,Cn1ccnc1C(F)(F)C(=O)NC(C1CCN(C(=O)Cc2cn[nH]c2)C1)(C)C 80562,c12cnc(nc1C)N1CC3C(C3C1)CNC2=O.N1(CC)CCC1C1CCCC1 80563,C(c1cccnc1)=CC(=O)N(C(C(=O)NCC(C)(C)O)C1CC1)C 80564,Cc1ccc(SCCNC(c2ccccc2Cl)c2nnnn2C2CCOC2)c(C)c1 80565,C(=O)(C(C)(C)C(C)NC(c1cn(C(C)C)cn1)=O)NCC1CN(C(C)C)C1 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80600,c1(C(N2C(C(=O)OC(C)(C)C)CC(O)C2)=O)c[nH]c2c(F)cc(Cl)cc12 80601,C12(CNC(CSCC#C)=O)CN(C(c3sccc3C#N)=O)CC1CCO2 80602,C(=O)(C(C)(C)C(=O)NN1CCCC1C(N1CC2(CCCO2)C1C)=O)OC 80603,C1(NC(Cc2cnc(C)s2)=O)CC(C)N(C(=O)Cn2cc(CO)nn2)C1 80604,CCCC(C)(C)C(=O)NCC1(F)CCN(C(c2noc(C3CC3)c2C)=O)C1 80605,C12(CNC(C3C(C)(C)CO3)=O)CC1CN(C(C1CN(c3nncs3)C1)=O)C2 80606,C1(NC(Cc2scc(C)c2)=O)CCC(CNC(c2cn(C)cc2C(F)F)=O)CC1 80607,CC1(C(N2CCOC(CNC(C3(n4ccnn4)CC3)=O)C2)=O)CC2CCC1C2 80608,CCCC(CNC(c1ncc[nH]1)=O)C(=O)N(CC)OC 80609,Cc1ccc(-c2cc(F)ccc2CNC(C)Cc2ccc[nH]2)c2nc(C(=O)O)cn12 80610,N1(C(CNC(C2C(C)=CCS2)=O)=O)CC2CCCCCC2C1 80611,Cc1ccc(C2CC2C(N2CCCC2(C)CNC(c2cn[nH]c2)=O)=O)cc1Cl 80612,c1(COC)nn(C)c(Cl)c1C(N1CCCCC(NC(=O)C(C)=CC(C)(C)C)C1)=O 80613,c1(C=O)cnc(S(C)(=O)=O)s1.C1(N(C)C)CCCN(N2CC(C)(C=O)C2)C1 80614,c1(C(=O)NCC2CN(C(CNC(C(CC)C)=O)=O)CC2C)cc(C)c(F)c(C)c1 80615,CC1CN(C(C2CCC(C)C2)=O)CC1C(=O)NCc1ncc(C2CC2)o1 80616,c1(NC(C(CC=CC)NC(C2CCCN2C)=O)=O)cnc(C)nc1C 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80635,CCC(CC)(C(=O)NC1CCCC(CC(=O)NC(CN(C)C)C(C)C)C1)OC 80636,C=C1CC(C)(C(=O)NCC2C=CCN2C(=O)CC#N)C1 80637,C1(CC)CN(C(C2(Cl)CC2(F)F)=O)CC2(CCCOC2)O1 80638,CCC(F)(F)CC(=O)N1CCCC1CCCNC(=O)CCn1cc([N+](=O)[O-])cn1 80639,C(=O)(CCC(F)(F)C(=O)N1CC(C)N(C(=O)CC(C)(C)CC)CC1C)OCC 80640,C12(C(=O)CC3CC(C(=O)NCCC(=O)OC(C)(C)C)C3)CCC(C(F)F)(CC1)C2 80641,c1(C(N2CC(C(N)=O)(CNC(C3C(CC)CC3)=O)C2)=O)ccc(=N)[nH]c1Cl 80642,c1(C(=O)NCC(C)NC(C(c2c(C)cccc2)C)=O)ccn(CC(F)F)c(=O)c1 80643,C12(CC(=O)N(C3CCC3O)CC)CCC1CN(C(C1(C)CCCN1C)=O)C2 80644,C(=O)(C(Cc1ccco1)NC(C1CC1Cl)=O)NC(C(C)C)C1CCC1 80645,C(c1cc2ccccc2o1)=CC(N1C(C(=O)Nc2c(CC)cc(Cl)cc2)CC1)=O 80646,c1(CCC(=O)NC2CCC2NC(=O)C=CCOc2ccccc2)ccccc1F 80647,C1(NC(c2cn(CCC(C)C)nn2)=O)CCN(C(C2CCN(C)C2=O)=O)C1(C)C 80648,C(=O)(C(O)C(C)C)NCC(C1CCC1)NC(c1cnc(COC)s1)=O 80649,C1(NC(C2CCN(C(C=CCOC)=O)C2)=O)CN2CCC1(C)CC2 80650,C(CO)(CCCNC(c1coc(C)c1)=O)NC(C(CSC)OC)=O 80651,CC#CCC(C(=O)N1CC=CC1CF)NC(c1ccc(CO)nc1)=O 80652,c1(NC(=O)COCP(C)(C)=O)ccc(N)cc1[N+](=O)[O-].C12CCN(CC1)C(=O)C2C 80653,C1(C(N(C(C)CCNC(C2(C(F)(F)F)CCC2)=O)C)=O)CCOC2(CCCC2)C1 80654,C1(CC)C(C(N2CC(O)(CC(C)C)C2)=O)CCN1C(c1cc(CO)oc1C)=O 80655,c1(C(C(=O)NCC(CNC(c2ccc(CC)o2)=O)(C)O)(C)C)ccc(F)c(Cl)c1 80656,C1(CC#C)(C(=O)NC(CO)C(C)NC(c2cc(Cl)cs2)=O)CCCC1 80657,Cc1cncc(NC(=O)C(C)(C)C2CCCN2C(C2CCCCN2C)=O)c1 80658,c1(OCCOC)ccc(C(=O)N(CCC(C)NC(C2CCO2)=O)C)cn1 80659,CC1(CNC(C2CCC(=O)NC2)=O)CCN(C(=O)Cn2cc(C3CC3)nn2)C1 80660,c1(OCCC)ccc(C)cc1C(=O)NC1CCN(C(C2(C)COC2)=O)CC1F 80661,N1(C(C(CC)F)=O)CCC2C(CCN2C(=O)Nc2cccc(NS(C)(=O)=O)c2)C1 80662,c1(NC(=O)NCC(CNC(=O)OC(C)(C)C)OC)c(Cl)cccc1Cl 80663,N1(C(C(c2cccc(OC)c2)OC)=O)CCC(C)(C)C(C(=O)NC2CC=CC2)C1 80664,C1(C(N2CC(NC(=O)C(Cc3ccccc3)OC)C(F)C2)=O)(CC)CCOCC1 80665,c1(C(N2CC(n3ncc(Nc4ccnc(C(C)C)n4)c3)C2)=O)cnc(Br)c(F)c1 80666,c1(C(N2CCC(C)(CNC(=O)CC3CC3C3CC3)CC2)=O)cc2c([nH]1)CCCC2 80667,C#Cc1cc(C(=O)NCc2cn(-c3ncc(Cl)cn3)nn2)ccc1Cl 80668,C(CO)(CN=c1[nH]c(=NC)[nH]c(=NCCc2ccc(C)c(Cl)c2)[nH]1)OC 80669,c1(C(=O)NC(COC)CNC(c2ccn(C)c2C)=O)c(Cl)cccc1[N+](=O)[O-] 80670,CCCCC(CCCC)C(=O)NCCCc1nnc(Cl)s1 80671,C1(NC(C2(SC)CC2)=O)CCN(C(c2ccc(-c3sccc3C)s2)=O)CC1F 80672,C(N=c1ccc(NC(=O)C(OC)OC)n[nH]1)C1(OC)CCOCC1 80673,N1(C(CCC2CCC(NC(CC3CC(C)(C)C3)=O)C2)=O)CCC(C#N)C1 80674,CN1N=C(CC(=O)NCCC2CCCN(C(c3c[nH]c(=N)s3)=O)C2)CC1=O 80675,Cn1ncc2c(N3CCC(C)(CNC(c4cc(Br)nc(Br)c4)=O)CC3)ncnc12 80676,c1(C(=O)NC(CCNC(c2c(NC)cccc2)=O)C)ccc(F)c(F)c1 80677,c1(C(N(CCC)CCN(C(c2sccc2F)=O)C2CC2)=O)cnc(OC)nc1.C(C)(=O)O 80678,c1(CC(=O)NC(C)C(c2ccccc2)N(C(=O)C(C)(C)C)C2CC2)cnnn1C 80679,Fc1cncc(-c2nc(-c3ccc(-n4ccnn4)o3)n(C3CCSC3)n2)c1 80680,C12(NC(c3n[nH]c(C)c3C)=O)CCOCC1CN(C(C1C3(CC3)C13CC3)=O)C2 80681,c1(C(=O)NCC2CCN(C(C(N3CCN(C)CC3)C)=O)CC2)cc(Br)cc(Br)c1C 80682,CCC(CNC(=O)CCC(=O)c1ccc(C2CC2)cc1)CC(F)(F)F 80683,c1(-c2cn(CC3N(C(C4(CC(C)C)CC4)=O)CCC3)nn2)ccc2[nH]ccc2c1 80684,C1(C(=O)NCC(CC)(C)CC)CCCCCN1C(C1OCCC1C)=O 80685,C1(C(N2CCC(CC)C2CNC(=O)CCC2CCCC2)=O)CC12CCC(=O)CC2 80686,N1(C(CCN(c2nnnn2C)C(C)C)=O)CCN(C(c2ccc(Cl)s2)=O)CC1 80687,C(C)(C)(C(=O)N1CCC(N(C)C(c2cnc(Nc3ccccc3)s2)=O)C1)SC 80688,N1(C(C(CNC(C2(CCCC)CC2)=O)O)=O)CC2CCCC1C2 80689,c1(C(=O)NC(C)C(=O)NC2(CF)CC2)cn2ccccc2n1 80690,N1(C(c2nc(C(C)C)oc2)=O)CCN(CCN(C(=O)C(C)(C)CF)C(C)C)CC1 80691,CC(C(=O)NCCc1ccc(I)s1)S(=O)(=O)CCCCCCCC#N 80692,c1(-c2ccc(OC)cc2OC)c[nH][nH]c1=NCCc1cc(Br)n(C)n1 80693,C1(C#CC(=O)N(CC(=O)NCCCc2cncnc2)C(C)C)(CC)COC1 80694,c1(C(=O)NCC2(O)CN(Cc3ccsc3)C2)cccc2nsnc12 80695,CC1CN(C(C23CCCC2N(C(=O)OC(C)(C)C)CC3)=O)CCN(C)C1 80696,Cc1ccc(C(N2CCCC(C)(NC(=O)Cc3ccn(C(C)C)n3)C2)=O)nc1F 80697,CC1C(C(=O)NCCCOCCN(C(=O)CC2NC(=O)NC2=O)C)CC(C)(C)C1 80698,CC(C(=O)NCC1CN(C)CCN1C(C1CCn2ccnc2C1)=O)P(C)(C)=O 80699,N1(CC(=O)NCCN(C(=O)C(O)C2CCC2)C)CCCCCC1=O 80700,c1(CCC)ccc(C(=O)NCCCCCCNC(=O)CC2CC2CC)cc1 80701,C1(C(=O)NCC(CNC(C(CC)NC(N)=O)=O)CO)COCCN1C=O 80702,N1(C(c2cc(C(C)=O)on2)=O)CC2CCN(C(=O)C(O)c3cnc[nH]3)CCC2C1 80703,C1(NC(C2CCN(C(C3CCCCO3)=O)CC2)=O)CC2CCCC2C1 80704,C#CCCCCN=C(NCC1CC1)NC1CCN(S(C)(=O)=O)C1 80705,Cc1nn(CCC(N2CCOCC2C(C)(C)OC(F)F)=O)c(C)c1[N+](=O)[O-] 80706,CC1CN(c2ncncc2Cl)CC1NC(=O)CC1CC=CCC1 80707,Cc1cccc(C)c1C(N1CCC1CNC(C1(F)CCOC1C)=O)=O 80708,c1(C(=O)NC2C(CC)N(C(c3ncccc3F)=O)CCC2)ccc(Cl)c(Cl)c1N 80709,C1(C(N2CCC(CNC(CC3CC(=C)C3)=O)(COC)C2)=O)CC(C)CC(=O)N1 80710,c1(C(N2CC3CC3(C(=O)Nc3cnc(Br)cn3)C2)=O)ccc2c(c1)CCCO2 80711,c1(OCC)cccc(CC(=O)NC(C2CCN(C(C34CCC(C3)C4)=O)C2)(C)C)c1 80712,C(C(C)CC(=O)N1CCC(C(C)(C)NC(c2cn(C)cc2C)=O)C1)OC 80713,c1(CNC(=O)C(C)C)ccccc1.CCCCCCOCC(=O)NOCC(F)F 80714,C(=O)(C1CCOc2ccccc21)N(CC(C)C#N)NCC(N)=O.Cc1nc(C)cs1 80715,N1(C(c2nc(N(C)C)oc2)=O)CCC2(CCC(NC(=O)Cn3cnnn3)C2)C1 80716,C12(C(=O)NC(C)(C)CCNC(=O)C3=NNC(=O)CC3)CC(C)(C1)OC21CCC1 80717,N1(c2c(C#N)cnc(SC)n2)CCC2(CCC2NC(C2CC=CCC2)=O)CC1 80718,CC1CN(C(C2CCN(C(C3CC(O)CN3)=O)CC2)c2ccccc2)CC(C)O1 80719,N1(C(c2c(C)cno2)=O)CCCC(N(C)C(c2ccc(-c3ncc[nH]3)nc2)=O)C1 80720,c1(C(=O)NCC2CC(CNC(CC=C)=O)OC2)cc(C)nc2[nH]nc(C)c12 80721,c1(OC)ccc(C(=O)NCCN(C2CCCC2)C(=O)Cc2ccccn2)nc1Cl 80722,Cn1nccc(C(=O)NC2(CO)CN(C(=O)C(c3ccc(F)cc3)O)C2)c1=O 80723,c1(OCC)nc(Cl)ccc1C(=O)NCCC(C)(C)NC(c1cnc(C2CC2)[nH]1)=O 80724,c1(N(CC(C(C)C)NC(CCOCCOC)=O)C)cc2c(cn1)C(=O)CCC2 80725,N1(C(C=CCC)=O)CCC2(C1)CN(C(=O)CCCc1n[nH]c(=N)s1)CCO2 80726,c1(CC)cncc(C(=O)NC2CCCCC2NC(=O)CCC2CCCO2)c1 80727,Cn1nnc2cc(C(=O)NC3CCC34CN(C(c3cc(Cl)cs3)=O)C4)cnc12 80728,C1(C(=O)NCC(O)CNC(=O)CCn2cnnn2)(OC)CCCOC1 80729,C1(C(=O)OC)N(C(=O)C(=O)NC(CCO)C(C)(C)C)CC12CCCC2 80730,N1(C(C2CCN(C(C(C)OCCOC)=O)C23CCC3)=O)CCC2(CNC(=O)C2)C1 80731,C1(CNC(C2CCC(C)C2)=O)CC2CCC(C1)N2C(c1ccc2cccnn12)=O 80732,c1(C(N2CCC(C(C)NC(=O)C(C)=CC3CC3)C2)=O)ccccc1S(C)(=O)=O 80733,C1(CC(=O)NCC(O)CNCCc2nnnn2C2CCC2)CCC(=O)N1 80734,c1(CC)cc(=NC(=O)NCCCc2ccc(Br)c(F)c2OC)[nH]n1C 80735,CCC(C)(CCC(C)C)C(=O)NC1CC(C)(NC(=O)C(C)S(=O)(=O)C(C)C)C1 80736,c1(C(CN(C(C(=O)NCC)CC2CCCCC2)CC(C)C)O)ccc(F)cc1Cl 80737,C1(COC)CCN(C(=NCC(F)(F)c2ccc(OC)cc2)NC2CC2CF)CC1 80738,C(N=c1[nH]ncs1)C1CCN(C(Cc2cc(C)[nH]n2)=O)C1 80739,C=CC1CN(CC(C)(C)O)CCC1C(F)(F)F.S(=O)(=O)(CI)N 80740,C1(CC(=O)N(CCC(=O)NC(C(=O)OC)C2CC2)CC)CCCCO1 80741,c1(C(N(CC(C)NC(c2ccnn2CC(F)F)=O)CC)=O)nccn2nccc12 80742,C1(C(=O)NC2CC(C)C2)C=CCN(C(=O)CC2C(C)(C)C2(C)C)C1 80743,c1(CC(N2CC(F)(C(N3C(CO)CC3CO)=O)C2)=O)ccn2ccnc2c1 80744,c1(C(C(=O)Nc2ccc(F)cc2)N(CCOC)CCF)cc(Br)c(C)nc1OC 80745,Cc1nc(C(N2CC=CC2(C)C(=O)NCC2(CO)CC3CC3C2)=O)cc(O)n1 80746,N1(C(c2c(C)nn[nH]2)=O)CC(NC(C2CC(=O)N(C(C)C)C2)=O)C(CC(C)(C)C)C1 80747,c1(SCC(=O)NCCCc2cn[nH]c2)cn(CC(N2CC3CC3C2)=O)cn1 80748,Cc1cc(C#N)cc(C(N2CC=CC2CNC(=O)CCc2ccccc2C)=O)n1 80749,C(=O)(C(C#N)C(C)C)NC(CCC)C(=O)NCCc1cc[nH]n1 80750,C(=O)(C(F)(F)C(F)F)NC1CCC(CNC(CC(C)(C)C2C(C)C2)=O)C1 80751,c1(C(=O)OCc2cnc(C)s2)ccc2c(c1)S(=O)(=O)N(C)C2=O 80752,Cc1cc(Cl)cc(C)c1OCC(=O)NCC(O)CN(C(=O)CC1(O)CCOC1)C 80753,Cc1cc(C(=O)NC(C2CCN(C(c3ccnnc3C)=O)CC2)C(C)C)ccn1 80754,C=C(C)CC(C)C(=O)NCC(C)(CO)NC(=O)COc1ccc(Cl)c(Cl)c1 80755,C1(CNC(Cc2cn(CC)nn2)=O)CC(C)(C)CN1C(=O)Cc1ccnc(F)c1 80756,N1(C(c2c(C)nsc2)=O)CCC12CN(C(=O)C(O)C(C)(C)C)C2 80757,n1(CC)cc(C(=O)NCCN(CC(C)O)C(C2CN(c3nncs3)C2)=O)cn1 80758,N1(c2cc(N3CCCC(c4n(C)cnc4)C3)ncn2)CC2C3CCC(CC3)C2C1 80759,C12CN(CC1C)C2.c1(NC(CNS(CC)(=O)=O)=O)cn(-c2ccccc2)nn1 80760,C(=O)(C1=CCC(C(F)(F)F)OC1)NC(C)CCCNC(c1cnc(S)nc1)=O 80761,C1(C(=O)NC2C3CN(C(=O)Cn4cc(Cl)cn4)CC23)CCC=CCCC1 80762,c1(C(N2CCN(C(C)C)C(=O)C2)=O)cnn2cc(F)cc(F)c12 80763,C1(C(=O)NC(CCCCNC(c2c(C)n[nH]c2C)=O)C)CCCCC(=O)C1 80764,c1(C2C(C(N(C)CC3(O)CN(C(C(CC)F)=O)C3)=O)C2)ccc(Cl)cc1F 80765,C(CCCCC(=O)NC1(C)CCN(C(=O)C(C)Cc2cnn(C)c2)C1)OC 80766,N1(C(CN(C)C)=O)CCN(Cc2ccc(OCF)c(I)c2)C2CC12 80767,C12(NC(C3CCC(F)(F)C3)=O)CCN(C(c3ccccn3)=O)CCC1C2 80768,C1(NC(C=CCC)=O)CCCC12CN(C(c1ccc(CCNS(C)(=O)=O)s1)=O)C2 80769,c1(C(=O)NC(CNC(CC(CCC)O)=O)C2CCC2)c(F)cc(F)c(O)c1F 80770,C1(NC(C(C)CF)=O)CN(C(c2cc[nH]n2)=O)C2(CCOCC2)C1 80771,c1(C(=O)NCC(C2CCOC2)NC(=O)COCCCF)c[nH]nc1C(F)F 80772,Cc1cccc(Cn2nc(-c3ccc(C(C)C)nn3)nc2C2CCCC2C(C)C)c1 80773,O(NC(=O)C(CCOCCO)NC(c1ccn2cncc2c1)=O)CCCC=C 80774,c1(C(=O)NC(CCCNC(C2(C)CCC(OC)CC2)=O)C)ccc(C#N)c(C)c1 80775,CCCCCCCCC(=O)N1CC2(CC(NC(C3(C)C=CCCC3)=O)CO2)C1 80776,C1(C(=O)NC2(C)CC(C(N(CCOCC)C)=O)C2)CC(C)(C)CO1 80777,C=CCC(C)(C)C(=O)NC(C)CC(C)NC(c1cc[nH]n1)=O 80778,CC1(C)CC(CC(=O)NCCCCC(CO)NC(=O)CSc2nc[nH]n2)CCO1 80779,Nc1cc(C(=O)NCC2CN(C(c3cc[nH]n3)=O)CC2(F)CO)ncc1Cl 80780,C=CC(C)(C)CC(=O)NCC1CN(C(=O)C(C)=C(C)CC)CCC1C 80781,C(=O)(C1=CCCC1(C)C)N1CCC(C(CNC(c2ccc(C#C)cn2)=O)O)CC1 80782,c1(N(C(C=C(C)C)=O)Cc2cc[nH]c(=N)c2)ccccc1CC(N)=O 80783,N1(CCCNC(c2nnnn2C2CCCC2)(CC2(C)CC2)C)CCNC1=O 80784,N1(CCNC(c2c(SCC)nc(-c3nc[nH]n3)s2)=O)CCc2ccccc21.C1(C)CC1 80785,c1(C(=O)NCCC2(CNC(C3(C)CCC3)=O)CC2)cccc2sncc12 80786,C(=O)(CC(C)(O)C=C)NCCCCC(CO)NC(CCNC(COC)=O)=O 80787,N1(C(CC2ON=C(CC)C2)=O)CCN(C(c2cnc(C(C)(C)C)o2)=O)C(CO)C1 80788,C1(C#N)(C(=O)NCC2(F)CC(NC(C3CC(C(C)=O)C3(C)C)=O)C2)CC12CCC2 80789,C1(C(=O)Nc2c(C(=O)OC)n[nH]c2)C2CN(CCn3cc(Br)cn3)CC12 80790,N(C(=NCC1(N2CCCC2)CCC1)N1CCC(CC(N)=O)C1)Cc1c(Br)c[nH]n1 80791,C(=O)(C1=NN(CC)C(=O)CC1)N1CCC(N(CC#C)C(C2C=CCC2)=O)CC1 80792,Cc1cc(CN2CCC(C(N3CCCCC3CO)=O)C2)c(Br)cc1F 80793,c1(C(N(c2ncc(SC)cn2)C2CCNCC2F)=O)cc([N+](=O)[O-])c(F)cc1F 80794,C#Cc1c[nH]nc1C(N1CC2CC2(CNC(C2(COC)CCCC2)=O)C1)=O 80795,N1(C(c2c(C)n(CC(F)F)nc2)=O)CC2CCCC2(NC(C2OCCCO2)=O)C1 80796,c1(C(N2CC(C3CC3)(C(=O)NOCC3CCCC3)C2)=O)cccc2ccoc12 80797,CC(CC(=O)NCCCCCNC(C1(O)COC1)=O)c1cccnc1 80798,C#CC1(O)CN(C(=O)C(C)(C)CNC(=O)CC2NC(=O)NC2=O)C1 80799,n1(CC(N2CC(O)(CNC(CSCCC)=O)C2)=O)c(C)cc2ccccc12 80800,C1(CNC(CN(CCC)C)=O)CN(C(=O)CCNC(=O)NC2CC2)CCC1F 80801,C1(N(C(=O)C(=O)NC2C=CC(NC(=O)OC(C)(C)C)C2)C)CCCOC1 80802,N1(C(Cc2c(C)cc(C)s2)=O)CC2=C(C1)CN(C(C1(CCF)CC1)=O)C2 80803,C1(C(=O)Nc2ccccn2)CC12CCN(Cc1cncnc1)CC2 80804,N1(C(C2CN(C)C(=O)N2)=O)CC(NC(=O)C(F)=C2CCCC2)C2(CCOCC2)C1 80805,CC(C)C(C)(O)C(=O)NCC1CC(NC(C2CCC(=O)NC2=O)=O)C1 80806,C(=O)(C(C)CCCC(C)=O)NC(CC#C)(C)C(=O)NCC1(O)CC=CC1 80807,N1(CC(=O)NCC2(F)CN(C(c3cc(CCO)on3)=O)C2)CCNC(=O)C1 80808,C12(C(=O)OCCCNC(C=CCC)=O)C(NCCO)C3CC1C2C3.C(CCO)O 80809,c1(CC)nc(=N)[nH]cc1C(=O)NC1CCC1NC(=O)CSCc1ccccc1Cl 80810,c1(C(C)C)nc(NC2(C(=O)OCC(C)(C)C)CCC2)cc(=NC2CCC(=O)NC2)[nH]1 80811,N1(C(c2cc(-c3cc(C)c(C(F)(F)F)cc3)ncc2)=O)CC(F)(F)C(F)(F)C1 80812,C1(CNC(c2scnc2C(F)F)=O)CCCCN(C(=O)CC2CCOCC2)C1 80813,C1(NC(C(C)C2CC2)=O)C2CCC1N(C(c1cccc(-c3nnco3)c1)=O)C2 80814,CC12CN(C(=O)C3=CCC3)CC1(C)CN(C(=O)CCOCC1CCCO1)C2 80815,c1(CN2CCCCC(NC(=O)C(CO)c3ccccc3)C2)cc(I)ccc1[N+](=O)[O-] 80816,C(=O)(CS(=O)(=O)C1CC1)N1C(CNC(c2cccc3c2CCC3)=O)CCCC1 80817,Cc1nn(CC(=O)NCCOC(C)(C)CNC(C2(CO)CCCCC2)=O)c(=O)o1 80818,C(CC1=CCN(C(=O)CC23CCCN2CCC3)CC1)NC(C1CC1(Cl)Cl)=O 80819,C12(NC(C(=O)Nc3cn(CCC(=O)O)nc3)=O)CCOCC1C2(F)F 80820,N1(C(C(C)CO)=O)CC2(C1)CN(C(c1c[nH]ccc1=O)=O)CC2CO 80821,N1(C(C2C(C)C2)=O)CCCC2(CCN(C(=O)C=CCN(CC(F)(F)F)C)CC2)C1 80822,C1(CC)CCCC(C(N2CCC(CN(C)C)C2)C(=O)NC2COC2)C1 80823,CCCC(CCO)N=c1[nH]c(NC2CC2C2CC2C)nc2ccc(Cl)cc12 80824,C1(NC(c2ccsc2)=O)CC(NC(c2cc(C3CCC3)[nH]n2)=O)C12CCC2 80825,C(CC(O)C(C)(C)C)N(C(c1cc(C(=O)N(C)C)n(C)n1)C)C 80826,C1(NC(CC2(C)CCN(C(=O)C(F)C3CCCC3)C2)=O)C(O)C2CCOC12 80827,C1(C#N)(CC)CCN(C(=NCCOC(C)C)NC(C)C2CC2)CC1 80828,C1(C#N)(C(=O)NCC2(CC)CCN(C)CC2)CC2CCC1C2 80829,c1(C(N2CC=C(CNC(C3C(OCC)C3)=O)CC2)=O)ccc2scc(C)c2c1 80830,c1(C(=O)NC(CNC(CC(=C)C)=O)CC(F)(F)F)cc(Br)c2[nH]nnc2c1 80831,N1(C(C2CCC(C)C2)=O)CCC2(CC(NC(=O)CSc3ccccn3)C2)C1 80832,c1(C(=O)NCC2C(OCC)CN(C(=O)C(C)(C)C)C2)cc(C)c(C)cc1N 80833,C1(NC(C2CCC(C(F)(F)F)O2)=O)CCCN(C(C2(O)CCSC2)=O)C1 80834,N(C1CC2(CCC2)Oc2ccccc21)C(=O)NCc1cccc(C)c1 80835,N(C1CC2(CCN(C(=O)C(N)=O)CC2)Oc2ccccc21)C(c1c(C)scn1)=O 80836,N1(C(=O)CC2CC2c2ccccc2)CCCC1C1CCCN1C(C1CCC1)=O 80837,N1(C(C2CCCC(=O)O2)=O)CC(NC(C2C3COCC23)=O)C2(CCC2)C1 80838,C(=O)(CC(C)(O)CCC)NCCC(C(=O)NCC(C)OCC#C)(C)C 80839,N(C1CCc2ccc(C)cc21)c1nc(N2CCCC(C=C)C2)c2c(n1)CSC2 80840,Fc1cc(-n2cc(CN3CCCC(CCC4CCCC4)C3)nn2)cc(Br)c1 80841,N1(C(COCCC=C)=O)CCCN(C(=O)COc2cc(F)cc(Cl)c2N)C(C)C1 80842,c1(C(=O)NC2CCN(Cc3c(C)ccc(C)c3)CC2O)cc(F)c(Cl)cc1F 80843,C1(CNC(COCCCC#C)=O)CN(C(C2CC(Cl)(Cl)C2)=O)CCC12CCC2 80844,C1(CC=C)(NC(C2CC2C(C)C)=O)CCN(C(=O)C(C)(C)n2cnc(C)c2)CC1 80845,c1(OC2CCN(CC(=O)NCCC)C2)cc(C)c(Cl)cc1CC.C1(=O)CN1C 80846,N1(C(c2cnc(C)[nH]c2=N)=O)CC2(CCN(C(c3cn(C)c(C)n3)=O)CC2)C1 80847,c1(CC2(OC)CCC(C(N)=O)CC2)nc(C)cc(=NCc2cc(Cl)cs2)[nH]1 80848,N1(C(=O)NCCc2nc(CC(=O)OC)sc2)CCc2cc(OC)ccc2C1C 80849,C1(C2CCC(=O)NC2)(C(=O)NC2C(NC(C(C)(C)C#N)=O)CCC2)CCC1 80850,c1(C(=O)NC2CN(C(c3c(C)scc3)=O)C(C)(C)C2)c[nH]c2ccccc2c1=N 80851,C(C(=O)NC(C1CCCC1)CO)(C(C)(C)O)NC(c1c(C)nc(C)s1)=O 80852,c1(Cc2c(C(=O)NCC3C(NC(CSCC#C)=O)C3)non2)ccccc1Cl 80853,c1(C(N(CC(=O)NC(c2nc(-c3ccccn3)no2)C)C)=O)ccncc1I 80854,n1(C)cc(C(C)(C)C)cn1.C1(NC=O)CCC(CNC(C2(C3CC3)CCC2)=O)C1 80855,CCCCCC(C(=O)NC1CC2C(NC(C3CC(OC)C3)=O)C2C1)C(C)C 80856,S(=O)(=O)(c1ccccc1Cl)NC(=O)CCN(C1CC1)CC1CCCNCC1 80857,N(C(=NCCCOc1ccccc1)NCCNCC)CC(C)SCCC#N 80858,CCCCCCC(CC)(CC)C(=O)NCC(C)(O)CNC(C1CC(C)(C(=O)OC)C1)=O 80859,C1(NC(N2CCC(c3ccccc3)C(F)(F)C2)=O)COc2ccccc2C1 80860,Cc1oc(C(=O)NC2CC2NC(=O)CCc2ccc(C(F)(F)F)cc2)cc1Br 80861,C(=O)(C1=C(Cl)CCOC1)NCC(CN(C(C(C(C)C)n1ncc(C)c1)=O)C)O 80862,N1(C(C#CC(C)(C)C)=O)CCCC12CCN(C(C1(CCF)CC1)=O)CC2 80863,c1(N2CCC(C(=O)NC3CC=CC3)C2)ncc2scc(Br)c2n1 80864,N1(C(CC(C)C)=O)CCC(F)(CNC(C2(c3cccs3)CCCCC2)=O)CC1 80865,CC1CC(C)CN(C(=O)CN2CCCC(N(C(=O)CCc3cocn3)CCF)C2)C1 80866,c1(C(=O)OC)ccc(C(=O)NCC(CO)NC(c2cc(C)n(C)c2)=O)cc1C 80867,c1(C(=O)NC2C3CN(C(C(C)OCC)=O)C2C3)ccc2nc(C)n(C)c(=O)c2c1 80868,Cc1c(Cl)cccc1S(=O)(=O)NCC1CCN(C(=O)CCn2ccc(C)n2)CC1 80869,c12cc(Cl)ccc1OCC1N(CC1)C(=O)N2.c1(SCC=C)ccncc1 80870,C1(NC(=O)C(c2ccc(F)cc2)CO)CN(C(c2coc(Cl)c2)=O)CC1C(F)F 80871,CC1(C)CCC(CNC(=O)CC2CCCNC2=O)N(C(=O)C=Cc2cnc[nH]2)C1 80872,c1(C(=O)NCC2CN(C(=O)C(F)Cc3ccccc3)CC2O)cc(O)ncc1F 80873,c1(C(C)C)nnc2n1CC(C(=O)Nc1cc(C(F)(F)F)cc(O)n1)CC2 80874,N1(C(C(C)OCC=C)=O)CC(CO)C2(C1)CN(C(=O)CCCC1CCOCC1)C2 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81116,Cn1cc(S(N)(=O)=O)cc1C(=O)NC1CCCC1NC(C1CCCN1C1CC1)=O 81117,CC1CCN(CC(N2CCC(NC(=O)CCc3nccs3)C2C)=O)CC1.C1CC1 81118,CC1CN(C(=O)Cc2csc(Br)c2)CCN1C(=O)C(=O)CC(N)=O 81119,C(C(=O)NCCC(C)CCNC(c1cc(C(F)F)nn1C)=O)(C(C)C)SC 81120,C(C)(c1ccccc1OC)=CC(=O)NCC1(C)CC(NC(CC2CC(CC)C2)=O)C1 81121,N1(C(c2cn(CCNC(C(C)OCC(C)C)=O)nn2)=O)CC2(CCCN2C)C1 81122,CC1(C)CN(C(=O)Cc2cc(Cl)ccc2Cl)CC1NC(C1(O)CCOCC1)=O 81123,N1(C(CNC=O)=O)CCSCC1C(=O)NCc1cncs1 81124,CC1CN(C(C2C(C)(C)C2(F)F)=O)CC2(CCN(Cc3cc(F)cc(F)c3)C2)O1 81125,C(=O)(C1=CS(=O)CCC1)NCC(C(C)(C)C)NC(COCC(C)(C)C)=O 81126,c1(C(=O)OC)cc(C)ccc1S(=O)(=O)N1CCC12CN(Cc1nccs1)C2 81127,CC1(C)C(NC(=O)CCc2csc(=N)[nH]2)CCN1C(=O)CCC1OCCO1 81128,C12(NC(CCOC)=O)COCCC1CN(C(=O)CNS(=O)(=O)CCCC(F)(F)F)C2 81129,C1(NC(C=C(C)C)=O)CC2(C1)CC1(CC(NC(=O)CS(=O)(=O)C(C)(C)C)C1)C2 81130,C(C(=O)NNC(=O)CNc1nnc2cnccn12)OC(CC)(C)C 81131,CCC1=NOC(C(N2CCC(N(C(=O)CC3C(=O)NN=C3C)CCO)CC2)=O)C1 81132,N1(C(Cc2n[nH]c(=N)s2)=O)CCC(Nc2cc(-c3ccccc3)ncn2)CC1C 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81622,c1(OCC)cccc(C=CC(=O)NCC=CC(F)(F)F)c1OCC 81623,c1(C(N(C2CN(C(C3(CN4CCCC4)CC3)=O)CC23CC3)C)=O)cccn(C)c1=O 81624,C(=O)(C(C)(C)CCSC)NCC1(OC)CN(C(C2(F)CCCN(C)C2)=O)C1 81625,C1(NC(C(C)OC(C)(C)C)=O)CC(C)CN(C(c2cc(Cl)c[nH]2)=O)C1 81626,c1(C(=O)NC2C(NC(CCc3n(C)ccn3)=O)CC2)cnc2n1CCCCC2 81627,C1(C(=O)NCC2OCCN(C)C2)COC2(C1)CN(C(C1CN(C3CCC3)C1)=O)C2 81628,c1(OC)ccc(C(N2CCC(NC(=O)C=Cc3ccn(C)c3)CC2C)=O)cc1F 81629,C1(CNC(C2(OC(C)=O)CC2)=O)COCCN(C(=O)COC(F)(F)C(F)(F)F)C1 81630,c1(COC)cccc(C(=O)NCC#CCNC(=O)CSc2ccccn2)c1 81631,c1(-c2n(-c3cnc(C)s3)nc(C3CCOC3)n2)cnn2c1CN(C)CC2 81632,c1(C(N2CCCC(C)(NC(=O)C=CC3CCOCC3)C2)=O)cnc2scnc2c1 81633,C1(NC(C2(c3cc(C)no3)CC2)=O)CCC(C)N(C(=O)C(C(C)C)C2CCC2)C1 81634,CC(C(C)C(=O)N1CC(C)(C#N)C1)NC(c1csc(Cl)c1)=O 81635,C(c1cncnc1O)=CC(=O)NCC1CC(NC(c2c(C)oc(C3CC3)n2)=O)C1 81636,c1(C(=O)NCCCC(C)NC(C2CC2F)=O)cc(F)c(Br)cc1F 81637,N#CCCCCCC(=O)N1CCN(C(=O)C(F)OC(F)(F)F)C(C(F)F)C1 81638,CC(C)(C(=O)N1CCC(O)(CCNC(C23CC(CCO2)C3)=O)CC1)C(N)=O 81639,CCC(C)(CCC(C)C)C(=O)N1CCCC(CCOCC(C(=O)NCC)(C)C)CC1 81640,N1(C(c2ccc(C(C)(C)C)[nH]2)=O)CCOC2(CCC(NC(c3ccsn3)=O)CC2)C1 81641,C1(NC(c2c(C)sc(O)n2)=O)CN(C(c2cc(F)cnc2O)=O)CCC1C 81642,C#Cc1cccc(CC(=O)NCCC(C)(C)NC(=O)COC2CCC2)c1 81643,c1(C(C)C(C2C(C(=O)NCCSC)C2)=O)cncn1C.C1(=O)CC=CCN1 81644,N1(CC(C)(C)NC(C2N(CC)CCC2)=O)CCN(C(=O)Cc2scnc2C)CC1 81645,c1(SCC(C(=O)NCCCc2c(C)noc2C)C)ccc(Cl)cc1F 81646,CC(F)(C(=O)N(CCNC(C1CCCOC1)=O)CC1CC1)c1ccon1 81647,C(=O)(C(Cn1cccn1)NC(C1C2CCCC12)=O)N(C1CC(C)C1)C 81648,Cc1nnc2n1CCN(C(C1CC(F)CCN1C(=O)C(C)C#N)=O)C2 81649,S(=O)(=O)(c1cccs1)NCCC(=O)NCC1(O)CCN(CC)C1.C1CC(=O)N1 81650,C1(CC)CN(C(C2CCS(=O)(=O)C2)=O)CCN1C(c1cc(C)oc1C)=O 81651,N1(C(C2(COC)CC=CCC2)=O)CCC2(CCCCN(C(=O)CC(F)(F)Cl)C2)C1 81652,Cn1cc(CNC(N2CCN(CCC3CCCN3)CC2)=O)c(C(F)(F)F)c1 81653,Cc1noc(CCC(=O)NCC(CNC(=O)CC(C)c2ccco2)CO)n1 81654,c1(CC)nn(C)c(C(=O)NCCN(C(=O)C(CC)C(C)O)C2CC2)c1Cl 81655,C=CC(C)(C)C(=O)NCC12CC(CN1C(=O)C(C)NS(=O)(=O)CCCC)C2 81656,c1(C(=O)NCC2CN(C(C=C3CCN(C)C3)=O)C(C)(C)C2)csc(S(C)(=O)=O)c1 81657,C(=O)(CC1=CCCCC1)N(C)CC1CN(C(C2CCCN2N=O)=O)CCO1 81658,C1(NC(C2CC2Cl)=O)CC2CCC1CC2NC(C1CCC(c2ccccc2)CC1)=O 81659,S(=O)(=O)(c1ccsc1C(=O)NC12CCN(C(c3cn(C4CC4)nn3)=O)CC1C2)NC 81660,C1(C)(CC(=O)N(C2CN(C(C=C(COC)C)=O)C2)C)CC1(Cl)Cl 81661,N1(C(c2cncn(C)c2=O)=O)CCOCC(CNC(C2(O)CCSCC2)=O)C1 81662,Cc1noc(Cl)c1CCC(=O)NCC(O)CN(C)C(c1c(C)nnn1C(F)F)=O 81663,c1(N2CC(CC)C(NC3(C(C)C)CC3)C2)ncc(C)cc1S(=O)(=O)NC 81664,Cc1oc(-c2ccco2)nc1CC(=O)NCC(C)(C)N(C(=O)C=CCF)C 81665,c1(CNC(C(c2ccccc2)NC(C(C)OCCCC)=O)=O)ccc(F)cc1 81666,c1(CCC(=O)NC2CC2C(=O)NCCC#N)cccc(O)n1.c12ccnc(c1)S2 81667,c1(C(=O)NC2C(C)CN(C(=O)CCc3nc[nH]n3)C2)cccc(Cl)c1N 81668,C1(CC)CN(C(=O)CCc2ccc(O)nc2)CCC1N=c1nc[nH]s1 81669,c1(C(N(CC(CC)NC(=O)C(O)CC[S+](C)C)C)=O)cccc2cc[nH]c12 81670,N1(CC)OCC(OC(c2cc(C)c(C)s2)=O)C1=O 81671,CCCC(C(=O)NC(C(=O)NC1CCCCC1N(C)C)C1CCCO1)OC 81672,C1(C(=O)NCC2CN(C(c3scc(C)c3Cl)=O)C(C)C2)CCC(=O)C(C)C1 81673,N1(C(C(=Cc2cccs2)C)=O)CC(NC(=O)CC2CCCCC2O)C(C(F)(F)F)C1 81674,c1(NC(=O)CC)ccc(Cl)c(I)c1Cl.N1(CC(COC)O)CCN(C(=O)N)CC1 81675,C1(N(CCOC)C(c2ccc(SC)s2)=O)CCN(C(C2CCS2(=O)=O)=O)CC1 81676,c1(C(N2CCC(NC(C3CC=CCC3)=O)C(O)C2)=O)cccc2nc(CO)[nH]c12 81677,C1(OC)(CNC(C2CC(=O)N(C(C)(C)C)C2)=O)CCN(C(C2CCSC2)=O)C1 81678,C1(N(C(=O)CCn2cncn2)C)CCN(C(c2ncncc2Cl)=O)CC1 81679,C=CCC(CC=C)(C(=O)N1CCCC(CSC)(COC)C1)NC(=O)OC(C)(C)C 81680,c1(OC2(C(=O)NCCCCN(C)C(C3CCCC3)=O)CC2)cnn(C)c1 81681,Cc1cccc(CC(=O)N(C(C)CCNC(=O)C(c2cccc(C)n2)(C)C)C)c1 81682,C(C(C)(C)CC(=O)N1CCCC1CN(C)C(c1c(C(F)(F)F)n[nH]c1C)=O)OC 81683,N1(C(c2c(C)scc2)=O)CCCC(O)(CNC(=O)C(C)OCC2CC2)C1 81684,Fc1ccc(C(F)(F)F)cc1OCc1cc(I)cs1.C12(CC1)NC2 81685,Cc1ccc(=NCCC(=O)NCCNC(c2cc3n(n2)CCN(C)C3=O)=O)[nH]c1 81686,n1(C(C)C)ccc(C(=O)NCC2COCC2NC(c2cnoc2C2CC2)=O)n1 81687,c1(SCC(=O)NCC(CNC(c2ccc(C)o2)=O)O)ccccc1C 81688,C(C(=O)NCCCCN(C(=O)C(F)CC)C)(C(C)C)N(CC)CC 81689,C(=O)(CCCC(C)CC)NCC1CN(C(C(C)(C)NC(=O)NCC)=O)CC1O 81690,C(CC(C)C(=O)N1CC(F)(CNC(C2(CC)CC(C)(C)C2)=O)C1)=CC 81691,Nc1c(F)cc(-c2ccc(-c3ccc(C=CC(=O)NC)cc3)c(F)c2)cc1F 81692,c1(OCC)cnc(C(N2CCC(C)C2CNC(C2CN(C(C)C)C2)=O)=O)cn1 81693,C1(CNC(CCOCC#C)=O)CCN(C(=O)CCc2ccccc2Cl)CC1C 81694,C1(NC(C(CC)OC)=O)CCCCN(C(=O)C(=O)Nc2ncc[nH]2)C1 81695,O(NC(=O)C(c1ccoc1)NC(=O)CC1CCCC(=O)C1)CC(C)C 81696,c1(OC)ccc(F)c(C(=O)NCCC2CCCCN2C(c2csnn2)=O)c1Cl 81697,C1(CC(=O)NCCOCCNC(C(C)=CCC)=O)CCCNC(=O)C1 81698,c1(CNC(=O)NC2C(c3ccc(C)o3)C2)cccnc1N1CCCC1 81699,n1(COCC)c(C)cc(C(N2CCCC(CO)(CO)C2)=O)c1C 81700,c1(C(=O)NCC(CNC(C(CCC)F)=O)(C)C)cccc(C(N)=O)c1F 81701,C12(CCNC(COCCN(C)C)=O)CCC(C1)N(C(c1ccc(Cl)cc1)=O)C2 81702,C1(CC(N2CC(C(N)=O)(CNC(=O)C=CCO)C2)=O)CCOCC1(C)C 81703,N1(C(c2cncc(CC)c2)=O)CCN(C(c2cc(C(N)=O)co2)=O)C(CCO)C1 81704,Cc1cccc2c1ccn2CC(=O)N(C1CN(C(=O)C(F)C(F)(F)F)CC1O)C 81705,N1(C(=O)Cc2cnsc2)CCN(C(C2C3CNC(=O)C23)=O)C(c2ccccn2)C1 81706,Cc1c(CNC(C2C=CCN(C(=O)CCS(C)(=O)=O)C2)=O)sc2cncn12 81707,c1(OC)ccnc(C(N2CCC(C)(CC(=O)OC)C2)C(=O)NCCCF)c1 81708,CCC(CCC(=O)N1CC(C(=O)OC)C1)NC(C1CCN(CC)C1)=O 81709,c1cc(O)n(C)n1.n1(CCC(=O)NCCCN(CC)CC)cc(C)cn1 81710,N1(C(c2c(OC)cccc2)=O)CCN(Cc2cc(C)sc2C)C2CC12 81711,N1(C(c2cncnc2)C(=O)NC)CC(F)(F)CC1C(=O)Nc1cccc(OC)c1 81712,CC1CCC(C)(C=CC(=O)NCC2CN(C(C3(F)CCOC3)=O)CCO2)C1(C)C 81713,c1(NC(=O)NC(c2ccc(C(F)F)cc2)C)cc(Cl)ccc1NCCC(N)=O 81714,c1(CC)cccc(C(=O)NCC2(C)CCCN2C(=O)CCC(C)C#N)c1N 81715,c1(C(C)NC2CCCN(C(=O)Nc3ccco3)C2)ccc(F)c(Cl)c1F 81716,c1(CC(=O)NC23CCN(C(C4CC(O)C4)=O)CCC2C3)cnc2ncccn12 81717,C1(CNC(C#CC(=O)N(C)C)=O)CN(C(C2CCC3(CC2)N=N3)=O)CCC1(F)F 81718,C(=O)(CC1OCCc2ccsc21)NCC1CC(C)N(C(C2CCCOC2C)=O)C1 81719,c1(CNC(C(C2CCOC2)NC(C(F)=CCC)=O)=O)ncnn1C 81720,C12(NC(C(C)c3ccsc3)=O)CCC(NCc3ccc(C(=O)O)cn3)(CC1)C2 81721,C(=O)(CC(O)C1CCCC1)NC(C1CN(C(=O)Cc2csc(Br)n2)C1)C 81722,c1(N2CC(CCC)(C(=O)N(c3ccc(C)cc3)C(C)CO)C2)nc[nH]c2ncnc1-2 81723,N1(CCC(=O)Nc2ccccc2)CCN(c2nnc(-c3occc3Cl)s2)C2CC12 81724,C1(CC(=O)NCC2CC2)(N(C)C)CCCCC1.C(=O)(C(C)(C)c1ncco1)N1CCC1 81725,C(=O)(C(C)CC(N)=O)N1C(CC(=O)NCc2n[nH]c(C)c2C)CCCC1 81726,N1(Cc2nc(C)sc2)CCCC(CNC(=O)COC2CCCOC2)C1 81727,CC(C)(C)CCCC(=O)NC1(C)CCN(C(C2(C)CCCO2)=O)C1 81728,N1(C(C(OC)OC)=O)CC(=O)NCC1C(=O)NCCOCCCF 81729,c1(C(N2CC3CN(C(C(n4cc(Br)cn4)C)=O)CC32)=O)ccc2cnn(C)c2c1 81730,c1(C(N2CCN(C(CSC(C)C)=O)C3C2C3)=O)ccc2oc(O)nc2c1 81731,C1(C(=O)NCC(CSC)(C)C)CC=CCN1C(c1cc(F)n(C)n1)=O 81732,C(=O)(C1CCCc2nn[nH]c21)N1CC(CCNC(C23CC(C#N)(C2)C3)=O)OCC1 81733,N1(C(CCSC)=O)CC2C(CC(=O)NCCc3scnc3C)C2C1 81734,Cc1c(F)ccc(C(N2CCOC(CNC(C3(C)C=CCC3)=O)C2)=O)c1Cl 81735,CCC(CC)CCC(=O)NC1CCOC(CNC(=O)C(N2CCCCC2=O)C)C1 81736,N1(C(CCCCC)=O)CCN(C(C2CC(=O)N(C)C2)=O)C2(CCC2)C1 81737,c1(N(C)C)ccc(C(=O)NC2CCC2NC(c2ccncc2F)=O)cc1[N+](=O)[O-] 81738,O=C(NNc1ncccc1Cl)c1ccc2n[nH]cc2n1 81739,C1(NC(c2cnc(CC(C)C)[nH]2)=O)CCSC12CN(C(=O)CCc1nc[nH]n1)C2 81740,C1(CC(N)=O)COCCN1C(=O)NC1CCN(N2CCCC2)C1 81741,c1(SCC)ccc(NC(C23CC2CN(C(=O)OC(C)(C)C)C3)=O)c(C(=O)O)c1 81742,c1(-c2nnc(C(C(CC)CC)Oc3ccc(F)cc3)o2)c(Br)cccc1[N+](=O)[O-] 81743,C1(CC)CCC(O)(C(=O)NCCN(C(=O)CS(C)(=O)=O)C2CC2)C1 81744,n1(CC(N2C(C)C(NC(=O)Cc3cnc[nH]3)CC2)=O)nc(O)ccc1=O 81745,C(N=c1[nH]c(C)ncc1F)C1C(NC(Cc2c(C)cccn2)=O)C2(CC1)CCC2 81746,N1(C(CCc2cnc(C)o2)=O)CCCC2(CCC(NC(C3(C)CC(F)(F)C3)=O)C2)C1 81747,C1(CC(=O)NC(C(C)C)CNC(C2(O)CCOC2)=O)(CSC)CCOCC1 81748,Cc1cc(N)ccc1C(N1CCC(O)(CCNC(c2ccnc(CO)c2)=O)C1)=O 81749,c1(C(N2CCCC(Nc3cc(C)nc(C)n3)C2)=O)cc(C)c(F)cc1F 81750,C1(CNC(=O)NC(c2nc(=O)o[nH]2)C)CC(O)CN1c1ccncn1 81751,N1(C(C2CCC(CNC(CC(C)F)=O)C2)=O)CCOC2(CCCC2)C1 81752,C1(C(=O)NCC2CC(O)CN2C(=O)CCc2ccc(F)nc2)CCC2CC2CC1 81753,C(=O)(CC(C)(C)CCOC)NCC(CCC)C(=O)NC(C1CCCC1O)C 81754,c1(CC)nc(C)ncc1C(=O)NC1CC(NC(c2cc(OC)no2)=O)CC1O 81755,N1(C(c2c(OCC)ccc(C)n2)=O)C(CNC(=O)C(N)=O)CC2COCC12 81756,N1(C(c2cc(CC)on2)C(=O)NCC2CCCO2)CCCCC1c1cncnc1 81757,N1(C(c2c(CC)c[nH]c2)=O)CCOC2CCN(C(c3ccc(N)cc3)=O)CC12 81758,CC(CC(F)F)C(=O)NCC1CCCCN1C(=O)CCCNC(N)=O 81759,N1(C(c2scc(C)c2)C(=O)NCCCF)CCN(Cc2ccccc2)C(=O)C1 81760,c1(OC)cc(F)c(S(N)(=O)=O)cc1C(N1CCC(C(c2ccccc2)C)C1)=O 81761,n1(CCOC)cccc(C(N2CCOC(C3CCCCC3)C2)=O)c1=O 81762,C1(CC#C)CCN(C(C2CCC(NC(=O)CCC3CC3C)CC2)=O)CC1 81763,C1(C(=O)NC2(CF)CN(C(C3C(C)CCC3)=O)C2)COCCN1C=O 81764,N1(C(COC2N(C(c3ccc(C#N)s3)=O)CCC2)=O)CC2CCC(C1)O2 81765,c1(C(N2C(C(=O)NC(CCC)CCC)CSCC2)=O)ncc(F)cc1C 81766,C12(C(=O)NC3(C)CC(NC(C(C)Cc4ccncc4)=O)C3)CCC(C1)OC2 81767,N1(C(c2c(C(C)NC(C3C4C5CCC(C5)C34)=O)noc2)=O)CC(O)C(C)(C)C1 81768,C(=O)(C(C(C)C)NC(=O)CCN(C)CC)NC(C(=O)NCCC)C 81769,c1(C(=O)NCC(CN(C(C(CC#C)C2CC2)=O)C)O)cnn2c1N(C)CC2 81770,C1(C(=O)NCC(CNC(=O)CCc2ccc(Cl)cc2)O)NC(=O)C2CCC12 81771,N12CC3CC(C3C1)Nc1nc(cs1)C2=O.c1(N)nccnc1F.CC(C)(C)OC(C)=O 81772,c1(CCCCC(=O)NCC2(C)CCN(C(C3COC3)=O)C2)ccc(F)c(F)c1 81773,C(=O)(C1=NNC(=O)CC1)N(C)CC1CCCC(NC(=O)CCc2nncn2C)C1 81774,C1(C(=O)NCCC(CCC)O)C2CCC(C2)N1C(c1coc(N(C)C)n1)=O 81775,C(=O)(CC(C)(C)C(F)F)NC(CCC)C(=O)NC(CO)CCC(C)C 81776,N1(C(COC(C)C)=O)CCC(O)(CNC(=O)CCc2cnn(C)n2)C1 81777,Cn1cc(C(=O)NCCCC2CCN(C(c3cccc(CF)c3)=O)CC2)nc1O 81778,C1(C(=O)OCc2cncc(CN)c2)CCC=CCCC1 81779,C(c1cccc(Cl)c1)=CC(N1CC(NC(c2ccc(OCC)nc2)=O)C(O)C1)=O 81780,C1(NC(c2c(C)noc2N)=O)CN(C(C2CCCN2C)=O)C2(CCOCC2)C1 81781,N1(C(c2ccc(OC)cc2O)=O)CC(NC(c2ccsn2)=O)CC12CCOC2 81782,c1(CC(=O)NC2CCCC(CNC(C=CC=CC)=O)C2)ccc(C#N)nc1 81783,CC1CCOCC1C(=O)NC(C)(C)CNC(C1(n2cnnn2)CCCCC1)=O 81784,c1(CC(N2CC(CCCC)N(C(=O)C(C)CCC)CC2)=O)cnn2c1CCCC2 81785,Cn1cc(C(=O)NC(c2ccc(Cl)cc2)Cc2cccnc2)c(=O)c(Br)c1 81786,c1(NC(=O)NC2C(CC)COC2)ccc2c(c1)C(O)CCC2 81787,C12CCCN(C1)C2.C1=CCC(Cn2cc(CC3C=CCC3)nn2)CC1 81788,C1(C(=O)NC2CC(NC(c3ccc(C(C)(F)F)cn3)=O)C2)C(F)(F)C12CCC2 81789,c1(N(CC(CN(C(C(COC)(C)OC)=O)C)O)C)nnc(O)c2ccccc12 81790,C1(C(=O)NCC2(COC)CN(C(c3coc(C)n3)=O)C2)CC2(CSC2)C1 81791,c1(CC=C)cccc(C(=O)OCc2ccns2)c1.C1(C(C)C)C(=O)O1 81792,c1(C(=O)NCc2ccc(C(C)NC(CC(C)SC)=O)cc2)ccc2nn[nH]c2n1 81793,N1(C(c2c(C)cc(C(C)C)o2)=O)CC(C)N(C(C2CCNC(=O)C2)=O)C(C)C1 81794,C(N=c1[nH]c(=NCc2ncco2)[nH]c2ccsc12)C1(C)CC1 81795,c1(-c2ccn(C)n2)cc(C(=O)Nc2cc(Cl)nc(Cl)c2)cc2cc[nH]c12 81796,Cc1cc(C(=O)NCc2cnn(C)c2C(=O)NC(C2CCCO2)CO)c(C)nn1 81797,N1(C(c2ccc3nc(Br)nn3c2)=O)CCC2(CCCC2C(N2CCCOCC2)=O)C1 81798,N1(C(C(C(C)C)N(CC)CC)=O)CC2CC3CC2C1C3NC(=O)C1=CCC1 81799,c1(NC(=O)NC2C(C(C)C)CNCC2)ccc(-n2cncn2)c(Cl)c1 81800,c1(OC)nc(C)c(C(C)OC(C2CC(C)(C)C2)=O)s1 81801,C(=O)(CCC(=O)NCC1CCCC1)NC(C1(NC(=O)Cc2ccn(C)n2)CC1)C 81802,c1(C(N2CC(O)CC2C)C(=O)NC(CC)C)cc(C)c(Br)s1 81803,C1(CNC(C=C(C)C)=O)COC(c2ccccc2)CN1C(c1coc(Cl)n1)=O 81804,c1(C(=O)NC2C=CC(CC(=O)N(C)Cc3c(C)occ3)C2)cc(C#N)cs1 81805,CC(CNC(=O)C(C1CC1)NC(=O)CN1CCOC1=O)(CO)CO 81806,c1(C(=O)NCC2C(CNC(C34CCCCC3C4)=O)C2(F)F)ccc(F)cc1F 81807,C1(NC(c2ccnc(C)n2)=O)CCCN(C(c2cc(C(C)(C)C)on2)=O)C1C 81808,C1(NC(c2cn(CCOC)nn2)=O)CCN(C(c2cc3n(c2)CCC3)=O)C(C)C1 81809,Cc1ccc2nc(C(N3CCN(C(=O)CC4(CO)CC4)C(CO)C3)=O)cn2c1 81810,C1(CNC(C2C3CNC(=O)C32)=O)CCCCN(C(c2occ3c2CCC3)=O)C1 81811,CC1(C)C=C(C(=O)NCC(O)CCNC(c2cncc(Cl)c2Br)=O)C1 81812,C1(CNC(c2c(C)cnn2C(C)C)=O)CN(C(=O)CCCC2CC2C)CC1(F)F 81813,C(=O)(C1=C(C)CCCC1(C)C)N(CCOC)CCNC(=O)C(C(C)O)NC(N)=O 81814,C1(=CC(=O)NCC(CN(C)C(c2cncc(Cl)c2Cl)=O)O)CN2CCC1CC2 81815,C1(C)(N(CC(=O)NC)C)CCC(NC(=O)CCC2CC(C)(C)CO2)CC1 81816,CON=CC(=O)N(CC(C)CNC(c1cc(CN(C)C)on1)=O)C 81817,CC1(NC(=O)Cc2csc(S)n2)CCCN(C(C2CCCC2(F)F)=O)C1 81818,N1(C(COCC=C)=O)CC(CNC(c2cc(OCC)n[nH]2)=O)CC1C 81819,CN1CC(C)(C(=O)NCC2CC3CCC2N3C(=O)CCc2ccncn2)CC1=O 81820,C(CNC(=O)Cc1cccs1)(CC(=O)NCCC1CC(F)C1)OC 81821,n1(C(C(=O)NC(C)CSC(F)F)C)cc(C2(N3CCC3)CCC2)nn1 81822,C1(OC)CC2CCC1CC2C(=O)N(c1ccc(F)cc1)C1CN(C(=O)C=C(Cl)Cl)C1 81823,c1(C(CF)NC(=O)NCC2(C(=O)OC)CC2)cccc(OC)c1 81824,c1(C(N2CC3CCN(C(C4CC(C)(O)C4)=O)CC32)=O)cnc2ccc(F)cc2c1 81825,C1(C(N2CC(C(C(N3CCC(NC(=O)NCC)C3)=O)O)C2)=O)CC2C=CC1C2 81826,c1(CN(C(C(COC)O)=O)CCNC(=O)Cn2ccnc2C)ccc(F)cc1 81827,C12(C(=O)Nc3c(C(=O)OCC)c[nH]n3)CCC(CC1)N2C(c1scnc1C)=O 81828,c1(NC(C23CCC(OC)C2C3)=O)cc(Cl)c(N=[N+]=[N-])cc1Br 81829,C(=O)(C(CO)C(F)(F)F)NCC(C1(O)CCCCC1)(C)C 81830,c1(C(N2C(CN(C(=O)Cc3cc[nH]n3)C)COCC2)=O)occ2c1CCC2 81831,C1(CNC(CN(C)C2CC2)=O)CN(C(=O)CC2NC(=O)NC2=O)CCC1(C)C 81832,C1(NC(c2c(C)n(C)nn2)=O)C2CC3C(C2)C13C(=O)N(C1CCCC(C)(C)C1)C 81833,Cn1cc(C(N2CCN(C(=O)COC3(C)CCCC3)C(CCO)C2)=O)ccc1=O 81834,C1(C(N(C2CC(=C)C2)C)=O)C=CCCN1C(=O)C(C)OCOC 81835,C1(CC(=O)N(C)CC2CCCCN2C(C2CCCSC2)=O)CCC2(CC1)CC2 81836,c1(SC)nc(N2CCC(NC(=O)CSCCN(C)C)C(F)C2)c(C)c(Cl)n1 81837,Cc1sncc1C(=O)NCC(C)C(=O)NCCCN1CCCCC1 81838,c1(C(C(=O)OCC2CCOCC2)N(C(C(C)SC)C)C)noc2c(Br)cccc12 81839,C1(C)(C(N2CCCC(N(C(=O)Cc3cc(C(F)(F)F)co3)C)C2)=O)CCC(=O)NC1 81840,c1(C(=O)NCC2CCC(NC(C3C(C)(C)CC3)=O)C2)ccn2nccc2c1 81841,c1(C(N2CCCC(CNC(C(C)(C)SC)=O)C2)=O)nn(C)c(Cl)c1Cl 81842,C(C1c2ccccc2CN1C)=CC(=O)NCC(C)N(C(=O)C=C(Cl)Cl)C 81843,CN=c1[nH]cc(C(N2CCC(OCCNC(c3cc(C(N)=O)co3)=O)C2)=O)s1 81844,C1(C(=O)NC(CN(C(CCOCC#C)=O)C)CC)CCOC1(C)C 81845,C(CC(=O)N1CC(NC(C2CC3(C2)CS(=O)(=O)C3)=O)C1)(C1=CCCC1)OCC 81846,C(C(C(=O)NCCC#CCO)NC(=O)C(n1ccc(C)n1)C)OC 81847,C12(C(=O)OC)CCC(CC1NC(=O)C(C)CCNC(=O)CN1CCC(OC)C1)C2 81848,C1(N(C(=O)C=CC(=O)NCC2(NC(=O)CSCC(N)=O)CC2)C)CC1 81849,C1(C(N(CC(=O)Nc2ccc(Cl)cc2Cl)C)=O)CC(=O)N(C)C1c1ccccc1 81850,C(N=c1nc2c(cnn2C)c(NC(C2CCCO2)C)[nH]1)C1(OC)CCC1 81851,C1(CC(=O)NC)CN(C(=O)CC2(SC)CC2)CCN1C(c1ccc(C)nc1OC)=O 81852,N1(C(CCCN(C(=O)OCC)C)=O)CC=CC(NC(C2C=CCC2)=O)C1 81853,C1(CC)CN(C(C2(CC)CCOCC2)=O)CC1C(=O)N(C)CC1CC1(F)F 81854,C1(C(N(CCC=C)CC)=O)CCN(C(=O)C(C)CC=CC=C)C1C(C)C 81855,C12(CC)CN(C(c3ccnn3CC(F)F)=O)C(CNC(C3CC(C)=NO3)=O)(C1)C2 81856,N1(C(Cc2n(C)ccc2)=O)CC(CNC(C2CCSC2)=O)C(C)(C)C1 81857,N1(C(C(c2cnn(C)c2)OC)=O)CC2(CCN2C(c2ccc(Cl)c(C)c2)=O)C1 81858,c1(CN(CCCNC(COCC(=O)OC)=O)C(C2CC2Cl)=O)ccccc1 81859,C(=O)(CCCCCNC(=O)CC1C=NNC1=O)NCCCS(C)(=O)=O 81860,CC1C(C(N2CCC(C(CO)NC(C3CCS3(=O)=O)=O)CC2)=O)CCN1C 81861,c1(CC)conc1C(=O)NCC1(CNC(c2nnn(C(C)(C)C)n2)=O)CCC1 81862,S(=O)(=O)(c1ccc(Br)c(C)c1C)N(c1c(C)n(C)nc1C(F)(F)F)C1CC1 81863,c1(C(N2CCC(N(C(C3C(OC)CC3)=O)C)C2)=O)cn(C)nc1O 81864,C1(CCOC)(NC(c2ccc(CC(C)C)s2)=O)CCN(C(=O)C=C(C)Cl)C1 81865,CC1C(C)N(C(C2CCn3nccc3C2)=O)CCN1C(C1CC(=O)NC(=O)C1)=O 81866,c1(OC)cccc(C(=O)NC2CCN(C(c3csc(Cl)c3)=O)C2C(C)C)n1 81867,N1(C(C2N(C(c3c(OC)scc3)=O)CC(C)C2)=O)CC(N(C)OC)C1 81868,c1(C(=O)OC)cnc(NC(C(C)NC(c2ncc(F)cn2)=O)C(C)C)cc1C 81869,c1(C(=O)NC2(CO)CN(C(c3c(N)cnc(SC)n3)=O)C2)cc2cnccc2o1 81870,CC1(C(=O)NCC2CCCN(C(=O)CCSCc3ccccn3)C2)CC=CCO1 81871,C1(O)(C(=O)NC(C2C(C(=O)NCC3C(OCC)CC3)C2)C)CCSCC1 81872,c1(C(=O)NC(c2nnc(C)s2)C)cc2cc(F)ccc2o1.N12CCCC(C1)C2 81873,c1(C(N(C(CNC(C(F)OC)=O)C)C)=O)cnc2c(cnn2C)c1O 81874,c1(C(=O)NCC2(COC)CCCN2C(C2CCNC(=O)C2)=O)cnc(C)c(C)c1 81875,N1(C(c2ccc(F)cc2F)CC)CC2CN(C(=O)C(C)(C)CC(F)F)CC2C1 81876,C1(CNC(CCNC(C)=O)=O)C2CCCC1N(C(c1ccc(C)s1)=O)C2 81877,Cc1c(C(=O)NCC(C(C)(C)C)NC(c2cccnc2)=O)ccc([N+](=O)[O-])c1O 81878,C(=O)(C1=CC2(CCOC2)C1)NCC1(CNC(=O)CCCCc2cnn[nH]2)CCC1 81879,CC1(C(N2CCCC(Nc3nccc(C(F)(F)F)n3)C2)=O)CCOC12CC2(F)F 81880,n1(N(CCNC(=NC)NCCCCN(C)C)C)ccc2ccccc12 81881,N1(C(C(C)NC(C)=O)=O)CCC2(CC1)OCCC2NC(c1ccc(N(C)C)cn1)=O 81882,c1(C(=O)NCC(C)NC(=O)C(C(C)O)NC(=O)C(C)(C)C)cc(F)c(F)cc1O 81883,N1(C(c2c(C(C)C)n(C)nc2)=O)CCCC(N(C(=O)C=CC2CCCO2)C)CC1 81884,C1(NC(C2C(=C)CC2)=O)CN(C(c2[nH]c(C)nc2CC)=O)CC1C(F)F 81885,C1(C(=O)NCC2CCCOC2)(CNC(=O)CCc2cnoc2)CCCCC1 81886,c1(-c2c(C)n[nH]c2C)ccc(=NCc2cc(Cl)cc(Cl)c2)[nH]n1 81887,c1(C(=O)NC(C(C)NC(c2ccc(COC)o2)=O)C(C)C)cc(=N)[nH]c(Cl)n1 81888,C1(CNC(CS(CC)=O)=O)CCC2CN(C(c3cn4ccsc4n3)=O)CC12 81889,c1(C(N2CCCC(CN(C(C(C)C3CC3)=O)C)C2)=O)coc2c1CSC2 81890,n1(C2(OC)CC2)cc(CN(C)C)nn1.n12cc(nn1)CCC(=O)NC(=O)C2C.C(F)(F)F 81891,C(C1CCN(C(=O)CSC(F)F)CC1)=CC(=O)NC1CN(C2CCC2)C1 81892,c1(NC(=O)CC2CC(C(=O)NCC3NC(=O)NC3=O)C2)ccc(O)nc1 81893,O=C(N=c1[nH]nc(C2CNC2)s1)C1CC(O)(C(F)(F)F)C1 81894,C(=O)(CCC(=O)N(C)C)N(C1(C(=O)NC(CCOC)C)CC1)C 81895,N1(C(C(=O)NCCOCCOC)=O)CC(CNC(c2scnc2Cl)=O)C2CC12 81896,C(CCC(O)C(=O)NCc1ncn(C2CC2)n1)NC(c1ccc(C)[nH]1)=O 81897,c1(C(N2C(C(=O)NCc3ccsc3)CC(OC)C2)=O)ccc(C)cc1O 81898,C1(OC)(CNC(=O)CSC2CCOC2=O)CCN(C(c2nccn2C)=O)C1 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81917,N#Cc1ccc(=NC(=O)NCCN2Cc3ccccc3C2)[nH]c1 81918,c1(C(=O)NC(CCCC)CNC(c2cn[nH]c2)=O)ccc(C(F)(F)F)nc1OC 81919,C1(C(=O)OC(C)CF)COCCN(c2ccc(Cl)c(OC(C)(C)C)n2)C1 81920,C1(CC(=O)N(C)Cc2cn(CC)nc2)CCCN(C(c2cccnc2C)=O)C1 81921,Cc1cc2ncc(C(N3CCC(O)(CN(C(=O)C(C)CO)C)C3)=O)cn2n1 81922,N1(C(c2nc(CC(C)(C)O)sc2)=O)CC2CCC(C1)NC2 81923,C(=O)(CCCCNC(N)=O)NC1CCC(CNC(CC2(C=C)CCC2)=O)C1 81924,C(=O)(C(CC(C)C)ONC(C1CN(C)C1)=O)NC(c1nn(C)cc1O)C 81925,c1(C(N2C(C)(NC(=O)CCc3nccs3)CCC2)=O)cc(Cl)ccc1OCC#N 81926,c1(C(=O)C(C)C)cccc2c1OC(F)(F)O2.n1(CC)cc2c(n1)C(=O)O2.N 81927,CC(C)CC(CNC(c1cn(C)cn1)=O)C(=O)N1OC2CCC1C2 81928,C12(NC(C(C)CC3CCCCC3)=O)CCC(CNC(=O)C(=O)N(C)C)(C1)OC2 81929,O=C(CC(C(F)(F)F)NC(=O)CCC1CCC(=O)C1)NCC1CC1(F)F 81930,C12(NC(CSC(C)C)=O)CCCC1CCN2C(c1csc(Nc2ccc[nH]2)n1)=O 81931,O=C(CCS(=O)(=O)NC1CC(NC(=O)CCn2ccccc2=O)C1)NC1CC1 81932,c1(C(=O)NC(C)CCNC(=O)Cc2ccno2)cncn1C1CC1 81933,c1(CC)ccc(C(=O)NCC(C)(C)CN(C)C(C2CCCCNC2=O)=O)c(C)n1 81934,N1(C(C2(F)CCC2)=O)CCOC2(C1)CN(C(=O)CC(C(F)F)n1cccn1)C2 81935,c1(C(=O)NCCCC2OCCN(C(c3n(CC)nnc3)=O)C2)nc(C)ccc1C 81936,c1(NC(C(=O)NCC2C(NC(CCC#C)=O)C2)(C)C)ccc2c(c1)OCCO2 81937,N1(C(=O)Nc2c(C)cccc2I)CC(C)C(NC(=O)OC)CC1C 81938,c1(C(=O)Nc2scnc2C(=O)N(C2CCN(C(=O)NC)C2)C)nnccc1C 81939,CC1(C)COCC(NC(=O)CC2CCC(C)(F)CC2)CN1 81940,C=CC(C)(O)C(=O)N1CCCC(CCNC(c2cnn(CC)c2C)=O)C1 81941,c1(C(C)(C)C)ncc(C(=O)NC2CCN(C(=O)CCN3CCCC3=O)C2)s1 81942,Cc1cc(Br)cc(C)c1CC(=O)NCC1C2CN(C3CCS(=O)(=O)C3)CC12 81943,CC(C)(C#N)CC(=O)N1CC(n2cc(CCCO)nn2)C1.c12ocnc1CNC2=O 81944,C1(N2CCC(OC)C2)CCN(C(=O)C(=O)Nc2ccncc2)CC1 81945,N1(C(C(C)N(C(C)=O)C)=O)CCCCC1CCNC(c1occc1C)=O 81946,C(=O)(C(C(C)C)n1cc(C)cn1)NCC(CNC(CC(=O)NCC#C)=O)O 81947,C1(CN(C(C(=O)OC)C)C(=O)C=Cc2ccoc2)CC(=O)NC1=O 81948,c1(C(N2CC(CCC)C(C(=O)NC(c3nc(C)cs3)C)C2)=O)ccc(F)c(C)c1 81949,c1(NC(=O)NCC2(C(=O)NC3CCOC3)CCC2)ccc(Cl)c(Cl)c1 81950,C(C(F)(F)F)(C1CC1)OC1CC(CC(=O)NC2CCCO2)C1 81951,C1(C(=O)NC2CCCCC2)CCCCC1CNC(c1sccc1CO)=O 81952,n1(CCOC)nc(C)c([N+](=O)[O-])c1NC1CC(OC)CN(C(=O)C=CC(C)(C)C)C1 81953,CC(C(C)(C)C)NC(=O)C(c1cn(C)nn1)NC(=O)C(C)OCC1CC1 81954,C(=O)(CC(C)C(=O)NCCC)N(CC(=O)NC1CCC1CO)CCC 81955,c1(C(N2CCC(F)(C(=O)NC(C3CCOCC3)C#C)C2)=O)ccc(C#N)cc1 81956,C(C(F)(F)C(=O)N1CCCC1(C)C(=O)NC1CCC(c2ccccc2)C1)OC 81957,c1(C(=O)NCCN(C(=O)C2=CCCC2C)CCC)cc(C)ccc1[N+](=O)[O-] 81958,CC1=CCC(C)(C(N2CCC(CN(C(=O)CC3CC(=O)NC(=O)C3)C)C2)=O)CC1 81959,N1(C(c2cc(C)c(C)nc2)=O)CC(NC(=O)CNC(N)=O)C(S(C)(=O)=O)C1 81960,CC(F)(F)C(C)(C)C(=O)NCCC(N1CCC(c2nc[nH]n2)C1)=O 81961,CS(=O)(=O)C1(CNC(c2ccnn2C2CCCC2)c2nnnn2C2CCC2)CC1 81962,Cc1ccc(F)c(C(=O)N(C)CC2CCCN(C(C3CCC(C)O3)=O)C2)c1F 81963,Cc1cc(NC(c2ccccc2F)=O)ccc1OCc1nnc(O)o1 81964,c1(C(=O)NCC2CN(C(CS(CC)(=O)=O)=O)CC23CC3)cc2c(s1)CCCC2 81965,Cc1c(C(N2CCC(O)(CNC(c3cnsc3)=O)C2)=O)cnn1C1CCC1 81966,C1(NC(CC(c2ccc(Cl)cc2)C)=O)CCCN(C(=O)C=Cc2cncs2)C1 81967,C1(CNC(=O)Nc2nc3ccccc3[nH]2)COC2(CCCCC2)O1 81968,C1(COC)COCCN1N(C)C1CCCC1c1ccc(C)cc1C 81969,C1(NC(C(=O)NC(C)C)=O)CCOCC1NC(=O)NC(=O)N(C)C 81970,n1(CC(=O)NCC(CC)NC(c2ccc(N)cc2F)=O)cc(C)c2ccccc12 81971,C1(CC#C)(C(=O)NCC2CCN(C(c3c[nH]nc3C(C)(C)C)=O)C2)CCOCC1 81972,C(=O)(C(F)(F)C(F)F)N1CCC(C(C)NC(=O)CC2CCCOC2)CC1 81973,C(c1cnc[nH]1)=CC(=O)NCC(C)N(C(=O)C(O)C1CCCC1)CC 81974,N1(C(CCCC)=O)CCCC2(NC(c3ncn(C)n3)=O)CC2C1 81975,c1(C(N(C(CNC(C(C)=C(CC)C)=O)C)C)=O)cc(OC)nc2ccccc12 81976,c1(CN(c2nnc(C3CCC(=O)N3)n2CC2CCCCC2)C)cccc(F)c1C 81977,c1(NC(C)CN(C)C(c2c(O)cc(F)cc2F)=O)ncc2ncn(C)c2n1 81978,N1(C(c2c(C)cn(C)c2)=O)CCC(CO)(CNC(c2cnc(S)[nH]2)=O)CC1 81979,CCCCCC(O)C(C)C(=O)NCCC1(CNC(c2ccnn2CCC)=O)CC1 81980,Cc1cc(C(=O)C(=O)NC2CC2NC(=O)C=CC2CC2)ccc1F 81981,C1(NC(CNC(C)(C)C)=O)CC(F)(CNC(c2csc(-c3cn[nH]c3)n2)=O)C1 81982,C1(CNC(=O)CCC2OCCO2)CC(NC(c2ccn(CC(F)F)n2)=O)C(O)C1 81983,c1(C(N2C(CNC(C(C)(C)O)=O)CCCC2)=O)cccc2nc[nH]c12 81984,c1(C(=O)NC2(CF)CCN(C(c3ncc(CC)nc3)=O)C2)cc2ccncc2s1 81985,N1(C(CN(C)C2CC2)=O)CCOC2(C1)CN(C(C1(C)CCC1)=O)C2 81986,C1(OC)(CNC(=O)Cn2ccccc2=O)CCN(C(c2cccnn2)=O)C1 81987,C(CN=c1[nH]c(=NCc2ccc(C3CC3)o2)[nH]c2c1COCC2)(NC)C1CC1.CS 81988,CON(CCO)C(=O)C1CC(=O)CN1C(C1COCC1(C)C)=O 81989,C1(CNC(C(C)CF)=O)CN(C(c2cc(C(F)F)on2)=O)CCC12CCC2 81990,C1(C)(c2nc(C3CCC(C)(O)CC3)on2)CN(C(C)(C)C)CC1(F)F 81991,CC(C)C(C(=O)NC1CCN(C(c2cc(C(N)=O)co2)=O)C1C)n1cncn1 81992,C(c1cn[nH]c1)=CC(=O)NC(C1CCCN1C(=O)C(=O)NCCn1cccn1)C 81993,c1(OC)ccc(C(C)CC(=O)NCC(O)CN(C(=O)C(C)O)C)cc1 81994,C(c1cc[nH]c1)=CC(=O)NC1C(CNC(=O)C=CI)C1 81995,C1(NC(C(CSC)OC)=O)COCCC1NC(=O)CC1CC(C)(C)C1 81996,C#Cc1ccc(Br)c(C(=O)OCC)c1.C12CCC(C)CN1C2=O 81997,C1(C(=O)NC(C)CC(C)NC(C2COC(=O)O2)=O)CN2CCN1CC2 81998,c1(N(C2CCN(C(c3ccc(C)c(F)n3)=O)C2)C)ccc2c(n1)CCC2=O 81999,C1(C)(CC)CCCN(C(=O)C(c2cn(C)nn2)NC(=O)CCC(C)=O)CC1 82000,C(C)(N=c1[nH]c(Cl)ncc1Br)C1OCCN(C(CC2C(C)=NN(C)C2=O)=O)C1 82001,Cc1cc2cc(NC(c3cccc(Br)c3F)=O)ccc2nc1Cl 82002,C1(N(C)C(c2cc(S(N)(=O)=O)co2)=O)COC2(CCN(C(=O)C(C)(C)O)C2)C1 82003,C1(N(C)C(C2(C)CC2C(F)(F)F)=O)CCCCN(C(c2ccnnc2)=O)C1 82004,c1(NCCCCOCC)cc(C)c(S(=O)(=O)N2CCCCC(C)(C)C2)cn1 82005,C1(CNC(CCCSC)=O)CN(C(C2CCCC(C#N)C2)=O)C2CCCC2O1 82006,C12(CNC(C(CCC)F)=O)CC(CO1)N(C(=O)CC(C)n1ccnc1)C2 82007,O(C=CC(=O)NCC(C)N(C)C(c1ccn(CC)n1)=O)CC 82008,C1(NC(Cc2nnc(C)s2)=O)CC2CC(NC(=O)CCc3ccccn3)CC12 82009,Cc1ccc(F)cc1C(=O)N1CCC(=O)NC(CN(C)C)C1.C(CCO)O.C1CC1 82010,C1(F)(C(=O)NCC(C)(CO)NC(C(CSC)OC)=O)CCCCCC1 82011,C1(C(=O)NCCCCOCC)CCC(CF)CC1.c12cccc(c1)S2 82012,C(CCCC(=O)NC1C2CC1N(C(C1(C)CCN(C(C)=O)C1)=O)C2)SC 82013,CC(O)C(C(F)(F)F)NC(=O)Nc1ccn(CCNc2ccc(C#N)cc2)n1 82014,C1(C(=O)NCC2CCC2NC(C2(CC3CC3)CCC2)=O)CCC2(CC1)OCCO2 82015,CC(C)CC(C(=O)NCC(C)N(C)C)NC(=O)CN(C)C(C1CCC1)=O 82016,N1(C(C(F)OC)=O)CC(O)(CNC(=O)CCCC2CC2)C1 82017,c1(C(N(C2CCCN(CCNS(C)(=O)=O)CC2)C)=O)cccc(N=[N+]=[N-])c1 82018,C12(NC(c3ccc(C#N)o3)=O)CCN(C(c3nocc3Cl)=O)CC1C2 82019,Cc1c(C(N2CCN(C)CC2CNC(=O)C(O)CF)=O)cccc1CO 82020,C(=O)(CC(C)C(F)(F)F)NCCC(C)NC(C1CCN1C1CCCC1)=O 82021,C1(CNC(c2cn(C)nc2)=O)CCCC(NC(C2CN(C3CCOCC3)C2)=O)C1 82022,C1(C(=O)NCc2cn(CC(C)C)nn2)CN(C(=O)OC(C)(C)C)CC1(C)C 82023,N1(C(C(C2CC2)OCC)=O)CC(N(C)C(C2CC(CN(C)C)C2)=O)C(O)C1 82024,c1(C(=O)NCC2C(CNC(C(C)OCC)=O)CC2)cc(Cl)ccc1-n1cccn1 82025,n1(CCCNC(CN(C)CC)=O)cc(CCNC(C2COCC2C(N)=O)=O)nn1 82026,CCC(C)CCC(=O)NC(CCN(C(=O)CC1(O)CCCC1)C)C(C)C 82027,N1(C(CC(C=C)C)=O)CC2(C(=O)NCCCCN=[N+]=[N-])CC1CCO2 82028,C(=O)(C1=C(NCC)CCCC1)OCc1cnccc1-c1ccc(CC(=O)O)cc1 82029,N1(C(Cc2ncc(C)[nH]2)=O)CCCC(NC(C2CC2(Cl)Cl)=O)C1C 82030,Cc1cc(C#N)ccc1C(N1CCOC(CNC(=O)Cc2ncc(Cl)s2)C1)=O 82031,CC(C)(CCCF)C(=O)NC1CCCCC1CC(=O)NCC1(C)CC2(CCC2)C1 82032,N1(C(CS(=O)(=O)NC(C)(C)C)=O)CCC2C(C1)NC(=O)CN2C(=O)OC(C)(C)C 82033,c1(CN(C)C(=O)NC2COC3(CCOC3)C2)nc2ccccc2[nH]1 82034,C(C(C(=O)NC1(C(F)(F)F)CCC1)C(C)(C)C)NC(CCC(C)(C)OC)=O 82035,c1(OC)cc(CNC(=O)Nc2ccccc2-n2ccnn2)ccc1C 82036,C1(N=[N+]=[N-])(C(=O)Nc2c(C)cccc2F)CCN(C(c2csc(C)c2C)=O)C1 82037,C(=O)(C1CCCc2nncn21)c1ccc(NC(C)=O)c(F)c1 82038,C12(CC(=O)N(C3CC(CF)C3)C)CCCCC1C2(F)F.C12CCCC1CNC2=O 82039,N1(C(c2c(C)nc(C)[nH]2)=O)CC(N(C)C(C2CCCSC2)=O)C(C)(C)C1 82040,CCC1=C(C(=O)N2CCC(n3cc(-c4cc(F)ccc4OC)nn3)C2)CCCO1 82041,N1(C(C(CCCC)F)=O)CCC2(C1)CN(C(c1ccc(CCC(N)=O)cc1)=O)C2 82042,c1(COC)ccnc(C(=O)NC(C)(CNC(c2cc(C)c(C)s2)=O)C2CCC2)c1 82043,C=CCC(C)C(=O)N(CCCNC(c1ccc(OC)cn1)=O)C(C)C 82044,C(=O)(C(C)CCC)NCC1N(C(C=C(CCC)C)=O)CCC1 82045,CC1(C)CN(C2CCN(C3CC3)C2=O)CCC1C(=O)OCC(F)(F)F 82046,C1(CC)CCN(C(C2OCCC2C(C)C)=O)C1C(=O)NCCNS(C)(=O)=O 82047,CCC(CNC(c1nc(O)c(C)s1)=O)(CC)NC(=O)CN1CCCC1=O 82048,CC#CCC(C(=O)N1CC(c2ccccc2)C1)NC(C1CC2CCC2C1)=O 82049,C1(C(C(=O)NCC(C)(C2CC2)OC)C)CCN(C(=O)Cc2nc[nH]n2)CC1 82050,C1(NC(=O)C(O)C2CN(C(C3CC(C)C3)=O)C2)CCC(C)(C)CC1 82051,CCC(Cc1ccccc1)N=c1[nH]c(N2CCN(C(C)=O)C(C)(C)C2)nc(=N)[nH]1 82052,N1(C(C(C)NC(CC)=O)=O)CCN(C(=O)C=CCN(C)C)C(C(C)C)C1 82053,C(=O)(CC(F)(F)CC(=O)N1CCCC1Cc1cn(CC(F)(F)F)nn1)OC 82054,C1(CCNC(c2nn(C)c(C(N)=O)c2)=O)CN(C(=O)C(C)(C)C)CCS1(=O)=O 82055,c1(C(C2CCOCC2)CC=C)nnnn1CC=C.C(=O)(CNC(C)COC(F)F)N 82056,Cc1cccc(C(=O)NCC2(F)CCC(NC(=O)C(c3ccccc3Cl)C)C2)n1 82057,C12(C(=O)NC(C3CCC(=O)N(C)C3)=O)COCC1CN(Cc1c(C)cco1)C2 82058,Cc1nccc(C(=O)NC(C)CC(C)NC(=O)CCSc2ccccn2)c1C 82059,C1(CNC(c2c(C)cncc2)=O)CN(C(=O)CN2CCOCC2=O)CCCO1 82060,N1(C(c2cnc(CC)[nH]2)=O)CCC(C)(NC(c2cccc(OC)c2N)=O)CC1 82061,N#CC1(C(N2CCC=C(Cc3ccccc3OC(F)F)C2)=O)CC12CCCC2 82062,N1(C(=O)C2=CCCSC2)CCC2CCN(C(c3ccccc3C(F)F)=O)C2C1 82063,n1(-c2cc(CC)c(C)cc2)ncc2ccc(C(N3CCOCC3COC)=O)cc12 82064,C1(C(=O)NCCCc2cscc2Br)C2CC1N(Cc1ccncc1)C2 82065,Cc1cc(Br)c(S(=O)(=O)NCC2(CO)CC23CCOCC3)cc1Br 82066,c1(NC(CC(C)(C)N(C(C(C)=C2CCC2)=O)C)=O)cnc(F)cc1C 82067,CCCC(C(=O)NCC1(F)CCN(C(c2ccc(OC)c(C)c2)=O)C1)S(N)(=O)=O 82068,CC(CC(=O)NC(c1ncnn1C)C)C(C)(C)NC(=O)C=CC(F)F 82069,N1(C(c2n(CC)cc(Cl)c2)=O)CCC(C[N+](C(=O)CC2CCCOC2)([O-])NC)C1(C)C 82070,C(C(C)(C)CNC(=O)C(C1CC1)NC(c1ccc(Cl)s1)=O)SC 82071,C1(C(=O)NC2CC(N(C(=O)C=CBr)C)C2)CN(C)CCN(C)C1 82072,Cc1c(C(=O)NCC(C)(C)NC(C2CCCS2)=O)ccc(F)c1F 82073,C12(C(N3CC(N(OC)C)C3)=O)CCC(CC1)N(C(=O)CC(C)C(F)F)C2 82074,C1(CC)CCC(O)(C(=O)NCCOC2CCN(C(=O)CCC3CCC3)CC2)C1 82075,c1(N(C)Cc2n[nH]c(=N)s2)nc2c(c(=NC3COC4(CCC4)C3)[nH]1)CCCC2 82076,C(N=c1[nH]c(O)nc(N)c1[N+](=O)[O-])C1CN(C2CC3(ON=C(C)C3)C2)C1 82077,Cc1cnc(C(=O)NCC2CCN(C(=O)C=CC3CCCC3)CC2)cc1C#N 82078,c1(N(C)C)cc(C(N)=O)cc(F)c1.CCC1C(=O)N2CCC2C(=O)OC(=O)N1 82079,c1(C(=O)NCC2(CN(C(CNC(=O)NC)=O)C)CC2)cnc2[nH]cncc1-2 82080,C#Cc1nc(C(=O)NCC(C)N(C)C(C2CC2C#N)=O)cs1 82081,C1(CN(C(CCC#C)=O)C2CC2)CCCCN1C(c1c[nH]nc1Br)=O 82082,C1(C(=O)NC(CCNC(c2cc(CCC)[nH]n2)=O)(C)C)COCC(C)O1 82083,C1(CNC(c2cccc(OCC(F)(F)F)c2)(C)C)CCN(CCCCO)CC1 82084,Cc1ccc(F)cc1CNC(C1(C#N)CC1(C)C)=O 82085,C1(CCC)CN(C(=O)CNC(c2ccccn2)=O)CCN1C(=O)C(C)CC(N)=O 82086,c1(OC)ccc(C)c(C(=O)NCC2CCC(NC(C3CC3CF)=O)CC2)c1 82087,Cc1noc(-c2ccccc2)c1C(=O)NCCCN(C(=O)CC1(O)CCOC1)C 82088,c1(C(=O)NC(CNC(Cc2c(C)scc2)=O)C)cccc(-c2ccccc2)c1 82089,Cc1cc(C(=O)NCC2(O)CCN(C(c3c[nH]cc(C)c3=O)=O)CC2)ccc1Cl 82090,N(C1CCCn2nccc21)C(c1nc(C)c(C)s1)c1nnnn1CCOCC1CC1 82091,CC1(C)CN(C(=O)C(C)(C)CC2CC2)CCN(C(=O)CC(O)c2ccccc2)C1 82092,c1(CN2CCC(N(C(c3c(C)nc(F)cc3)=O)C)C2)ncccc1[N+](=O)[O-] 82093,c1(C(N2CCC(C(C)(C)NC(COCCCC)=O)C2)=O)cc(C#N)c(N)cc1O 82094,S(=O)(=O)(c1ccccc1[N+](=O)[O-])C(CCC(=O)NC(C(CC)C)C(=O)O)=O 82095,c1(C(=O)NCC23C(CN(C(CC4(C)OCCO4)=O)C2)C3)cc2cc(Cl)ccn2n1 82096,C(=O)(CC(C)N(C)C(C1CC(C)(C)C1)=O)NC(CNC(=O)OC)C 82097,c1(SC(C(=O)N(C(C)CCNC(C2CCCO2)=O)C)(C)C)nc2ccccc2[nH]1 82098,c1(C(N(CCCNC(=O)CC2(CO)CC2)C2CC2)=O)coc(-c2ccccc2)n1 82099,C(=O)(CCCCCN(C)C)N1C(C(C)NC(=O)Cc2cscn2)CCC1 82100,N1(C(c2cnsc2)=O)CCC2(CCCN(C(C3CC34CC(O)C4)=O)C2)C1 82101,c1(C(=O)NC(C(C)NC(c2ccccn2)=O)C)occ2c1CCC2 82102,CC(C(C)(C)C(=O)NC1C=CCCC1)NC(=O)C=CC(F)(F)F 82103,C1(NC(CNS(CCCC)(=O)=O)=O)CCN(C(c2cc(Cl)cs2)=O)CC1C(C)C 82104,N1(C(C(C2CC2)OC)=O)CCC2CCC(C1)N2CC1CCCO1 82105,C(=O)(C1=CCC(C)(C)CC1)NC(C1CN(C(c2cnncc2O)=O)CCO1)C 82106,c1(CNC(C2CN(C(C3C(c4n(C)cnc4)C3)=O)C2)=O)cccc2c1OCCN2 82107,N1(C(CCc2n(C)ncc2)=O)CCCC1(C(=O)NC12CC(C1)C2)C(C)C 82108,c1(N(CC(=O)NCCN(C(c2csc(C3CCCN3C)n2)=O)CC)C)ccccc1 82109,CCCCCCCCC(C)C(=O)N1CCN(C(c2ccc(C)cc2)=O)CC(O)C1 82110,C(CC(F)F)(C(=O)N1CC=CCO1)N(C(c1ccc(CC)cn1)=O)C 82111,c1(CCCNC(C(CNC)O)=O)nc(O)c2c3c(sc2n1)CC(C)CC3 82112,N1(C(C2(OCC)CCOC2)=O)CCOC(C(=O)NC2CCCC2(F)F)CC1 82113,C1(C(=O)NC2(CCO)CC2)CCN(C(=O)C=C(C2CC2)C2CC2)CCO1 82114,CC1(C)CC(C)(C(N2CCN(C(N)=O)CC2)=O)CN1C(c1cscc1Cl)=O 82115,C(=O)(C1SCCc2ccccc21)N1CCN(C(C=C=C(C)C)=O)C(CCO)C1 82116,C(C)(CC(C)C(F)F)C(C1CCC2(CCC2)C1)=O.CC1=CC(=O)NC1 82117,c1(C(=O)NCc2nc(N3CCCCC3C(F)(F)F)sc2)c(F)c(F)nc(F)c1F 82118,Cc1ccc2[nH]c(C(N3CCCC(NC(=O)CSC4CC4)C3C)=O)cc2c1C 82119,CCCC(CC(=O)NCCCCCCO)NC(=O)C=Cc1cncs1 82120,N1(C(c2c(C)ccnc2O)=O)CCC(C)N(C(=O)C2=COCCO2)CC1 82121,N1(C(COC2(C)CCCC2)=O)C(CNC(C2CCC2(C)C)=O)CC2CC12 82122,C1(C(=O)NCC2(CNC(=O)CCc3cnco3)CC2)COC2(CCC2)CO1 82123,N1(C(CCC(=O)NC)=O)CCN(C(C2CCC2)=O)CC(O)C1 82124,Cc1ccc(N2CCC(NC(C3(F)CCCCC3)=O)C(O)C2)c([N+](=O)[O-])c1 82125,Cc1ccc(C=CC(=O)NCC2CN(C(=O)CCC3COC(C)(C)O3)C2)c(C)c1 82126,C(C(=O)NCCC1(O)CN(C(C2CCCC2SC)=O)C1)(C(C)(C)C)OC 82127,c1(OC)nccc(C(=O)N(c2nc(C)cc(C)n2)CC2CNCCO2)c1F 82128,C1(C(N2C(CC(=O)NC)CC2)=O)CCCN1C(=O)Cc1cncs1 82129,Nc1cncc(C(N2CCCCC2CCNC(=O)CCCCc2cnc[nH]2)=O)c1 82130,c1(-c2cc(NC(c3ccc(F)nc3)=O)sc2)ccccc1C(F)(F)F 82131,c1(C(=O)NC2CC(NC(C(CC(N)=O)O)=O)C2)n[nH]c2c1CCSC2 82132,O=C(NNC(=O)N1CC(c2nc[nH]n2)C1)c1cccc(-c2cccc(O)c2)c1 82133,N1(C(C2(CNC(C(CC=CC)C)=O)CCCC2)=O)CCC(C2=NOCC2)C1 82134,C1(NC(CCC#C)=O)CN(C(=O)CSc2nncs2)CC1C 82135,c1(CC)ccc(C(=O)N(C2CCN(C(C3CCCC(O)C3)=O)C2)C)cn1 82136,n1(C(CC)C)ncc(C(=O)NCC(O)CCNC(=O)C=Cc2cnc[nH]2)c1C 82137,C(CO)(CCC(C)C)NC(CC1(C)N(C(C(C)SC)=O)CC1)=O 82138,C(CN=c1ccnc(N2CCC=C(F)C2)[nH]1)c1n(C)nc(C(F)(F)F)c1 82139,C(c1cn(C)cn1)=CC(=O)NC1CCN(C(c2nc(CC)oc2)=O)C1 82140,CC1(c2cn(C3CCC(C(=O)NCCC4CCCCO4)C3)nn2)CCOC1 82141,Cc1cc(Cl)cnc1C(N1CC(F)CC1C(N1CC2CCC(C1)O2)=O)=O 82142,C1(=CCC)CCN(C(c2nocc2C)C(=O)NCc2ccco2)C1 82143,C1(NC(C=CCC)=O)CC2CN(C(=O)CS(=O)(=O)N(CC)CC)CCN2C1=O 82144,c1(C(=O)OCC(c2ccc(Br)s2)C)ccc(C2CCCC2)c(F)c1 82145,n1(CCC(=O)OC)cc(S(=O)(=O)N2CC3CCN(C(C)=O)C3C2)cn1 82146,N1(C(C)C)CCCC1C(=O)N(CCNC(=O)COCc1ncnn1C)C1CC1 82147,N1(C(C(c2c(C)cccc2Br)NC(C(COCC)C)=O)=O)CCCCCC1CC 82148,C1(C(=O)NCCOC)C2CN(C=O)CC12.c1(-c2ccnn2C)cc(C)[nH]n1 82149,C12(CNC(Cn3ncc(C)c3)=O)CN(C(=O)Cn3ncn(C)c3=O)CC1CCO2 82150,c1(C(N2CC3(CC(NC(=O)Cc4c[nH]nc4O)C3)C2)=O)cnn2c1OCC(O)C2 82151,Cc1cccn2cc(C(N3CC4CN(c5nccc(CC#N)n5)CC4C3)=O)cc12 82152,O=C1CC2(CCN(C(C3CC4C(C3)C4(F)F)=O)C2)CN1.c12cn(nn1)CCOC2 82153,C1(CNC(C2(NC(C3C(CC(C)(C)C)C3)=O)CC3(CC3)C2)=O)CCC=CCCC1 82154,N12CC3(CC1CO3)C2=O.N1(CC)CCOC(CCNC(=O)C=CC(C)(C)SC)C1 82155,C1(N(C(CCc2cccc(OC)n2)=O)C)CCN(C(=O)CCSC)CC12CC2 82156,C12COC3(C1)CN(C3)C(=O)C1(CC1)NC2=O.CC1(CCO)CC1 82157,C(C(C)(O)C(F)(F)F)C(=O)NC1CCN(C(COC(C)C)=O)C1C 82158,CC1COCC(CNC(=O)C(C)N(C(c2cnc(Cl)s2)=O)C2CC2)O1 82159,C(=O)(C(C)(C)COC(=O)Nc1ccccc1)N1C(C(C)OC(=O)C(C)(C)C)CCC1 82160,C12(NC(COC)=O)CN(C(=O)C(Cl)=CCl)CC1CS(=O)(=O)C2 82161,C1(C(=O)NCC(=O)Nc2ccc(Cl)cc2)C2CCC(C2)N1C(=O)CSCC(F)F 82162,c1(COC)cc(C(=O)NC2CCCN(C(c3cnn(C(F)F)c3)=O)C2)c(C)o1 82163,c1(C(c2nnnn2C(C)(C)CC)NCCCCCS)cnnn1C.CCC(C)CO 82164,C=CCC(CC(=O)NCC(O)(COC)CO)NC(c1nc[nH]n1)=O 82165,Cc1[nH]c(C)c(C(=O)NCC2CCCC2NC(c2c(C)n[nH]c2C)=O)c1C 82166,C1(NC(CNC(C)=O)=O)CN(C(c2cnn(C)c2Cl)=O)CC1C#N 82167,c1(CNC(C(c2ccccc2F)C)=O)cnn2c1CN(C(=O)CCS(C)=O)CC2 82168,C(=O)(C1=C(C)OCCS1)N1C(C(=O)NCC2COCC2(C)C)(COC)C=CC1 82169,CC(=Cn1ccnn1)C(=O)N1CCCC(n2cc(C3(CCO)CC3)nn2)C1 82170,c1(C(=O)NC2C(NC(c3c(C)nncc3)=O)COC2)cc2ccccc2[nH]1 82171,N1(S(C)(=O)=O)CCCC(C(=O)NCC(C)(C)NC(C2CCC(C(N)=O)CC2)=O)C1 82172,C(C1CN(C(=O)CC(C)COC)CC1C(N1CCOC(CO)C1)=O)=CC 82173,C1(N2CC3=CCN(CC3)C2=O)CCCN(S(N)(=O)=O)C1.NC(=O)C.C(C)(C)(C)C=O 82174,CCCC(O)CC(=O)NCC1CCC1NC(C1(C2CCC2)CC1)=O 82175,C1(CC(=O)NC2C(OC)CC2O)COCCN1C(=O)CC1CCCC(=O)C1 82176,c1(CNC(C(=O)OCC=C)CC2CCOC2)cc(OC)ncc1Br 82177,N1(C(C2C(COC)C2)=O)CC(NC(c2cc(N)cnc2C)=O)C(C)(C)C1 82178,c1(C(=O)NC(CCCNC(CC(CC)CC)=O)(C)C)ccn2ncccc12 82179,C1(CNC(=O)C(O)c2cnc[nH]2)CCCN1CC(F)F 82180,N1(C(C2CCC(C)(CC)O2)=O)CC(C2CCCN(C(c3coc(Cl)n3)=O)C2)C1 82181,C1(CC)CN(C(=O)C=NOC)CC1NC(c1cn(CC2CCCO2)nn1)=O 82182,C1(N(C(C(c2scc(C)n2)C)=O)C)CCCCC1N(C)C(c1ccc(O)cn1)=O 82183,C(=O)(C1Cc2ccccc21)NCC1(C(N)=O)CN(C(C2CCN(C)CC2)=O)C1 82184,C1(=CCNC(C2CC(=C)C2)=O)CCN(C(=O)Cc2cc[nH]n2)CC1 82185,C(=O)(C1=CCCCO1)NCCCC1(NC(c2snc(C)c2Br)=O)CC1 82186,C1(NC(CCCC=C)=O)CN(C(=O)Cc2cccnc2C)CC1C=C 82187,C1(NC(C#CC)=O)CCC(C(=O)Nc2cccc(CS(C)(=O)=O)c2)OC1 82188,c1(OC)cc([N+](=O)[O-])ccc1C(=O)NC1CC(NC(=O)Cc2ccccc2O)C1 82189,C1(CCC(=O)N(C2CCCCC2)Cc2ccc(F)cc2)CCC(C(F)(F)F)CC1 82190,C(=O)(CCC(=O)N1CCCCC1CCNC(c1c(C)nsc1C)=O)NC 82191,c1(C(=O)NC2C(CNC(C3C(OC)CC3)=O)CC2)cc([N+](=O)[O-])c(C)s1 82192,N1(C(CCN(C(=O)CCNC(C)=O)CC#C)=O)CCCC(C2CC2)CC1 82193,C1(NC(c2cn(C(C)(C)C)nc2)=O)CCC(O)CN(C(C2CCCN2N=O)=O)C1 82194,Cc1cc(Br)c(S(=O)(=O)N2CCOCC2CCC(F)(F)F)s1 82195,c1(C(C)C(N2CCC(n3cc(CN4CCOCC4C)nn3)C2)=O)ccc(F)cn1 82196,C1(C(=O)NCC(n2cccn2)C)(NC(=O)CCN2CCCC2=O)CC(F)C1 82197,C(C(C)(C)C(=O)NC(C)CCNC(=O)CN1C(=O)CNC1=O)SC 82198,C1(C(=O)NCC(CNC(C2(OCC)CCC2)=O)(C)F)CCCC2(CCC2)C1 82199,c1(NC)cccc(C(N2CC(C(O)C(N3CCC(CC(C)(C)C)C3)=O)C2)=O)n1 82200,c1(C(=O)NC2CN(C(C(N(C)C)N(CC(F)(F)F)C)=O)C2)ccn(C)c(=O)c1O 82201,Cn1c(C(=O)NCCC2CN(C(C3CCCCC3C(F)(F)F)=O)C2)cccc1=O 82202,C1(C(=O)NCC(C)N(C(CCN(C)CC)=O)C)CCCN1Cc1ccsc1 82203,c1(CC(=O)NCC2(O)CN(C(c3c(C)nc(C4CC4)o3)=O)C2)nc([N+](=O)[O-])n[nH]1 82204,C(c1cncs1)=CC(=O)NC(CNC(CCN(C)CCO)=O)(C)C1CC1 82205,CC1CN(C(=O)CC2CC2)CC1NC(C1CC1c1cccs1)=O 82206,N1(C(c2n(C)nc3c2CCC3)=O)CCOC2(CCN(c3nnc(C4CC4)o3)CC2)C1 82207,C(=O)(C#CC1(C)CC1)N(C1CCN(C(C(CC)COC)=O)C1)CCO 82208,c1(C(N2C(C(=O)Nc3ccccc3)CC(F)C2)=O)cncc2ccccc12 82209,Cc1csc(CCCC(=O)NCC(C)(C)CNC(=O)C(C)Cc2cccnc2)c1 82210,C1(NC(C(=O)N(CC)CC2CCCCO2)=O)CCCN(CC)C1 82211,C1(C)(NC(CC2CC(=C)C2)=O)CCCC1C(=O)NC(C)COCC1CC1 82212,CC1CN(C(=O)CCC2CC2)CC1NC(=O)CC1CC(=O)NC1=O 82213,n1(CC(N2CC(NC(C(COC)(C)OC)=O)C(O)C2)=O)cc(P(C)(C)=O)cn1 82214,C(C(C)(C)C1=CCCC1)NC(C1(OC(C)=O)CCCCC1)=O.C1C(=O)N1 82215,C(=O)(CP(=O)(C(C)C)C(C)C)N1C2CC(NC(C(F)=CC)=O)CC1CC2 82216,Cc1cc(C(=O)NC(C)CC(C)NC(=O)CC2CCC(C)(C)CO2)n2nccc2n1 82217,C12(NC(c3nc(C)sc3)=O)CC1CN(C(c1cccnc1SCCC(C)C)=O)C2 82218,n1(CC(=O)NCC(CO)NC(CCCOC(C)C)=O)ncc2ccccc2c1=O 82219,c1(CCC)cc(C(=O)NCC2CCCC2NC(c2cc(CO)oc2C)=O)c(C)o1 82220,N1(C(C(CO)NC(CCCCC=CC)=O)=O)CCOC(C)(C)CC1 82221,CC(CC(N)=O)N=c1[nH]c(C(F)(F)F)c(C2OCCO2)s1 82222,N1(C(CC2(C)CC2)=O)CCOC2(CCN(C(c3cccn(O)c3=O)=O)CC2)C1 82223,N1(Cc2c(C)ccnc2)CCC(NC(c2ccc(C(C)(C)C)o2)=O)CC(C)(C)C1 82224,N1(C(Cc2n(C)ccc2)=O)CCCC(O)(CCNC(C2CNC(=O)N2)=O)C1 82225,C1(NC(=O)CCSCc2ccccc2)CCC12CN(C(=O)C1=COCC1)C2 82226,N1(C(C=C(C)C(C)C)=O)CCC2CN(C(=O)CCN3CCC3)CCC2C1 82227,N1(C(C(=O)N(C)C)=O)CCN(C(C2CCC3(CC2)CC3)=O)C2(CC2)C1 82228,n1(COC)nccc1C(N1CCC1C(=O)N(C)CCN1CCOCC1)=O 82229,N1(C(CNC(N)=O)=O)CCOC2(CCN(C(C3CCC(F)C3)=O)CC2)C1 82230,c12cccc(c1)C(=O)N2.C(CCCCCO)NCc1cnc(Br)s1 82231,Cc1ccc(C(N2CCN(C(=O)CC3CCOCC3)CC2)=O)cc1Br 82232,n1(C(C)CC(=O)N(C)CCN(C)C(=O)SC2CCCCO2)cnc2ccccc12 82233,c1(C(=O)NC2CC(F)(CNC(C3CC(OC)(OC)C3)=O)C2)nc[nH]c2nccc1-2 82234,C1(O)(CC(=O)NC(COC)(C)COC)CCN(C(c2ccc(OC)nc2)=O)CC1 82235,N1(C(C2(OC)CC(C(F)F)C2)=O)CCCOC(CNC(=O)CSC)C1 82236,C(C(C)(O)CC(=O)N(CC(=O)NCC#CC(F)(F)F)C(C)C)OC 82237,N1(C(C(CCC)C(C)C)=O)CC2CCCC(C1)N2C(=O)Cc1cnnn1C 82238,CC(O)C(=O)NC1(CCNC(=O)CCC2CC2CC2CC2)CCC1 82239,C(=O)(C(O)CC[S+](C)C)NC(C)CNC(=O)C=CC(=O)N(c1ccccc1)C 82240,C(=O)(C(C)(C)C)N(C1CN(C(=O)C(C)OCCOC)C1)CC 82241,C(=O)(C(Cc1ccco1)C(=O)NC1CC(CNC(=O)Cc2cc(C)ns2)C1)OC 82242,N1(C(C(C)=CC2CC2)=O)CCC(C)(C)C(NC(=O)CCC2CCCN2C)C1 82243,CC(Cc1ccco1)C(=O)NC(CNC(c1nocc1C(C)(C)C)=O)C1CCC1 82244,c1(C(N2CCC(N(C(CC=CCC)=O)CC)C2)=O)cccc2c1C1CCC2OC1 82245,C1(NC(C(c2cncnc2)C)=O)COCCC1NC(c1cc[nH]c1C1CCC1)=O 82246,c1(OC)cn(CC(=O)NC2(CNC(=O)CCCC(N)=O)CCOC2)c(C)cc1=O 82247,C1(OC)CC(C(=O)N(C)Cc2cnc(C)s2)N(C(=O)CCn2ccnn2)C1 82248,C(=O)(C1=CCC(F)(F)CC1)N1CC(C)N(C(=O)Cc2cccc(O)c2)CC1 82249,N1(C(c2c(C)cccc2O)=O)CC2CCN(C(c3snnc3C)=O)C2C1 82250,N1(C(=O)CC2CC(F)(F)C2)CCOCC(CNC(C2(CCO)CC2)=O)C1 82251,N1(C(C=C(C)C)=O)CC2CCCC(NC(=O)CN3CCn4nccc43)C2C1 82252,N(S(=O)(=O)N1CCCCC(C)(F)C1)(C(C)C)Cc1ccc(F)cc1 82253,c1(C(=O)NCC(CC)NC(c2cnc(O)nc2O)=O)ncc(Cl)cc1Cl 82254,C1(NC(CSCCC)=O)CCCC1NC(=O)C(C)(C)n1cnnn1 82255,C(=O)(CS(=O)(=O)NCC1CC1)N1CC(O)(CN(C(=O)CCC2(C)CC2)C)C1 82256,N1(C(c2nc(C)sc2)C(=O)NCCC2=CCCCC2)CCn2ncc(C)c2C1 82257,CC(C(C)(O)C(=O)N(CCCN(C(=O)CSC(C)(C)C)C)C)c1ccccc1 82258,CCC(C)C(CC(=O)N1CCC1C)NC(=O)C(C)CC#N 82259,Cc1cc(C)n(CC(=O)NCCCN(C(=O)CCc2ccc(Cl)s2)C2CC2)n1 82260,C1(C)(C(=O)NCC(C)(O)C2(C)CC2)CC(O)CN1C(C1C2CCC(F)(F)C12)=O 82261,Cc1cccc2cccc(NC(C3(O)CCN(C(C4(C)CC4)=O)C3)=O)c12 82262,CC(C)C(C)C(=O)N1CCN(CCc2cn(CCOCCO)nn2)CC1 82263,C1(N(C(c2coc(C(N)=O)c2)=O)CC)CCCN(C(C2CCCN2S(C)(=O)=O)=O)C1 82264,C1(CC(=O)NC(C)C(O)Cc2ccccc2)CN(C(=O)OC(C)(C)C)CCC1(F)F 82265,S(=O)(=O)(c1c[nH]c(=NCC(C)(C)C)cc1C)N(C)Cc1c(OC)cccc1F 82266,C12(NC(C(Br)=C(C)C)=O)CCCC1CN(C(c1[nH]c(C)nc1C)=O)C2 82267,c1(OC)ccc(Cc2noc(-c3c[nH]nc3-c3cnn(C)c3)n2)cc1 82268,Cc1n[nH]c2nccc(N3CCN(C(C4=CCSC4)c4nnnn4C)CC3)c12 82269,CN1CCCC(CC(=O)NCC23CC2CN(C(=O)CN(c2ccccc2)C)C3)C1 82270,C(CC(=O)NC=CC(C)(C)SC)NC(COC)=O 82271,C1(C(=O)NC(CN(C(C2CCCN(C)C2)=O)C)(C)C)CN=C2N=CNN2C1 82272,C1(CCC)(C(=O)N(C(C)COC(C)=O)CC=CC(=O)NCC(C)C)CCC1 82273,C(=O)(C1CCCc2sccc21)NC1(CO)CCN(C(c2c(C(N)=O)ccs2)=O)C1 82274,N1(C(C(C)=C2CCC2)=O)CCN(C(=O)CCC(C)C)C(C2CCC2)C1 82275,c1(C(N2CCC(CNC(=O)Cc3cc[nH]c3)CC2)=O)nccc2cc[nH]c12 82276,C=CCC(CC)C(=O)N1CC2CC(C(=O)N(c3ccc(F)cc3)C)(C2)C1 82277,C1(C(=O)NCCN(C(c2cn(CC(F)F)cn2)=O)CC)CC1C1CC(F)(F)C1 82278,c1(OC)cc(C(=O)NCC2CN(C(=O)CCc3nccn3C)C3CC23)n(C)n1 82279,c1(CN(C2CCCN(CCF)C2)C(=O)CC2COC3CC2C3)occ2c1CCC2 82280,c1(OC)nc(C)ccc1C(=O)NCC1(OC)CN(C(C2(C)CC(OC)C2)=O)C1 82281,C(c1cccc(Cl)c1)=CC(=O)NC1CCCC1NC(C1CCCC12CC2)=O 82282,N1(C(C(n2cc(C)nc2)(C)C)=O)CC(C(=O)NCC2CCC=CCC2)CCC1C 82283,Cc1nscc1C(=O)NCC(C)N(C)C(C1CC2CC2C1)=O 82284,C1(CNC(C2C(C(C)O)C2)=O)C2CCCC1N(C(=O)C=Cc1ccc(=N)[nH]c1)C2 82285,Cc1cc(C(=O)NC(C)CNC(=O)C(C)(C)Cc2ccc(Cl)cc2)ccc1F 82286,C1(C(=O)NCc2nccc(CC)c2)CCCCCN1C(c1csc(C)c1C)=O 82287,N1(C(CSc2cn(C)nc2)=O)CC2CN(C(=O)CNS(N)(=O)=O)CC2C1CO 82288,C1(OC)CN(C(c2cnc(Cl)[nH]2)=O)CC1NC(=O)C(F)(F)c1ccncc1 82289,c1(C2CC2)c(C(=O)N(C(C2CCCCN2C)=O)CC)[nH]c2ccccc12 82290,O=C(C1=CCCN1Cc1ccccc1F)N=c1cc2n([nH]1)CCOC2 82291,CC#CCCCC(=O)NC(CCCC)C(=O)NCCCC(C)CO 82292,C1(O)(CN(C)C(C2CCCCN2C)=O)CCN(C(C2CCC(=O)O2)=O)C1 82293,n1(CCC(=O)NCCN(C(=O)CC2CCCCO2)CC)c(C)ccc1C 82294,c1(C(=O)NCC2C(NC(C3C(CCOCC)C3)=O)C2)nc[nH]c1C(C)(C)C 82295,c1(CCN2CCC(=O)N(Cc3cccnc3)C2=O)cc(Cl)c(Cl)c(Cl)c1 82296,c12cnc(nc1)c(=O)[nH]2.C1(CNC(C(C)N2CCCC2)=O)CCC2(CC2)C1 82297,CN1CCN(C(=O)C#CC2CCC2)C(C(=O)NCC(O)CCC2CC2)C1 82298,n1(CC)ncc(C(=O)N(C)CC=CC(=O)NCC2CNC(=O)O2)n1 82299,C(C(=O)NCC1CCCO1)(C(C)CC)N(C(C(C=C)CC)=O)C 82300,c1(NC(CCCC)=O)ccc(-c2ccc(-c3ccccc3)cc2)nn1 82301,N1(C(c2c(=O)ccn(C)c2)=O)CCC2(CCN(C(c3cn(C)c(O)n3)=O)C2)C1 82302,CC(C)C(O)CC(=O)N1CC=C(CNC(c2cc(C3CC3)ccn2)=O)CC1 82303,c1(NC(c2cn(C)nc2)O)nc(C(F)F)nn1-c1cnccn1 82304,CC1(C)CN(C(=O)CC2COC(C)(C)CO2)CCN(C(C2(O)CCCCCC2)=O)C1 82305,C1(NC(CC(=O)NC)=O)C2CC3CN(C(c4cc(C)nc(C)c4)=O)C1C3C2 82306,N1(C(c2ccc(CSC)o2)=O)CC(NC(c2sccc2OC(F)F)=O)C(C)C1 82307,C#Cc1ccc(C(=O)NC2(CNC(=O)C3=NOC(CC4COC4)C3)CC2)cc1F 82308,c1(C(c2n(CC)nnn2)NCC2C=CCCC2)c(I)cnn1C 82309,C(=O)(C(CCOC)NC(=O)CCCn1cccc1)NCC1(CC)CCCO1 82310,N1(C(C(c2cccnc2)NC(C(CC#C)C2CC2)=O)=O)Cc2ccccc2C1 82311,CC(CCC(=O)N(C)CC1C2CN(C(=O)C=C3CCC3)CC12)N(C)C 82312,C1(N(c2ccc(-c3cnccn3)cc2)C(c2cc(C)oc2)=O)CCNCCC1C 82313,c1(CC)cccc(C(=O)NCCCOCCN(C)C(C2(C)COCCO2)=O)c1C 82314,C=CC(C)CC(=O)N1CC(NC(=O)CCCOc2ccccc2)CC1C 82315,C(CC(C)(C)C)(C(=O)N1CCC(NC(c2csc3cncn23)=O)C(CO)C1)OC 82316,c1(COC)cccc(C(=O)NC(CC2CCC2)C(=O)NCC2(C)CC(C)=NO2)c1 82317,N1(C(C2CC(CNC(C(C(C)(C)C)C#N)=O)OC2)=O)CCC2(CCCOC2)C1 82318,C1(O)(CN(C)C(C2(F)CCCCC2)=O)CCCN(C(C2(C)CCOC2=O)=O)C1 82319,C1(CN(C)C(c2ccc(C#N)[nH]2)=O)CC(F)CN1C(c1cc(Br)c[nH]1)=O 82320,C1(CN2C(=O)CN(CCC(COC)C)C2=O)COc2ccccc2C1 82321,N1(C(c2c(C(C)=O)cn(C)n2)=O)CCN(c2nnc(C(F)F)s2)CC(O)C1 82322,Cc1nn(C)c(C)c1CCNC(=O)NC1(C)CC1(F)F 82323,C12C3CC4C(C3NC1=O)C24.C1(C(N(C(CC#C)C(=O)OC)C)=O)CCCC(=O)CC1 82324,N(C1CCCn2nccc21)c1c(C)c(NCc2nnc3n2CCC3)ncn1 82325,c1(NCc2c(C)cncc2)nccc(=NCc2cccc(Br)c2C)[nH]1 82326,c1(OC)c(C(N2CC(C)(NC(C3CC(C(C)C)=NO3)=O)C2)=O)[nH]c2ccccc12 82327,CN1CC(C)(C(=O)NC2CCCCC2CNC(c2cc3[nH]ccc3s2)=O)CCC1=O 82328,CC1(C(=O)NCCCCC2CN(C(c3ccnn3C3CC3(F)F)=O)C2)CC2(CC2)C1 82329,C1(NC(c2ccc(OC)nn2)=O)CCC(C)N(C(c2cnc(C)nc2CO)=O)C1 82330,C#CC1CCCN(C(c2cccc(-c3nnc(S)o3)c2)=O)CC1 82331,C1(NC(C(C)(C)C)=O)CCCN(C(=O)Cn2ccc(Br)cc2=O)CC1F 82332,c1(CNC(C2(NC(C3(c4c(C)cccc4)CC3)=O)CC2)=O)ccc[n+]([O-])c1 82333,c1(C(C)NC(C2COCC2NC(=O)Cc2cscn2)=O)ccc(C)nc1 82334,C(C(=O)N1CCSCC1C1CC1)(C(C)C)NC(C(n1ncc(C)c1)C)=O 82335,C1(NC(C2C3CC4C(C3)C24)=O)CN(C(C2CC(C)(CC)C2)=O)CC1OC 82336,C#CCCCC(C)C(=O)N1CCCC1CCc1cn(CC(C)(C)C)nn1 82337,c1(C(=O)N(CC(N2CC(n3ccnc3)C2)=O)C2CC2)c[nH]c(C(N)=O)c1 82338,c1(C(=O)NCC23CC(NC(C4C(CCC)C4)=O)(C2)C3)cccc(O)c1F 82339,C1(CNC(c2ccc(CCC)cc2)=O)CC2CN(C(=O)COc3ccsc3)CC12 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82533,c1(N2CC(C)C(NC(=O)CC3CC(F)C3)CC2)ccc(Br)cc1[N+](=O)[O-] 82534,N1(Cc2cn(-c3c(CC)ccnc3)nn2)CC2CC(OC)C(C2)C1 82535,N1(C(CSCC)=O)C2CCC(C2)C1CC(N1CC(C(=O)OC)C1)=O 82536,N1(C(CC2CCCC(OC)C2)=O)CCCC(CNC(=O)COCC2CCC2)CC1 82537,c1(CC(=O)NCC(CNC(CC2(OC)CCCC2)=O)OC)ccncc1F 82538,CC1CN(C(=O)Cc2ccon2)CC2(CCN(C(C3CC(C)(F)C3)=O)C2)O1 82539,c1(C(=O)OCC)ccc(C(=O)NC2C=CC(C)(C)OC2)nc1C 82540,C1(C(=O)NCc2n(CC(C)C)ccn2)C2CC(C)(C)C1NC2 82541,Cc1cc(=NCC2CCCC(C)CC2)[nH]c(=NCCc2cccc(N)c2)[nH]1 82542,CCCC(CC)CCC(=O)NC1CCC(NC(c2sccc2OC)=O)CC1 82543,N1(C(C(C)OCCN(C)C)=O)CCC(NC(C2CCOCC2)=O)C(CO)C1 82544,CC1(C)CC(CNC(C2CC23CC(F)(F)C3)=O)CN1C(=O)CCC1CCC1 82545,c1(C(=O)NC(CNC(CNC(C)=O)=O)C)cnc[nH]1 82546,Cc1cc(C)c(CC(N2CCOC(CCNC(C3CCC3)=O)C2)=O)c(C)c1 82547,C1(CC=C)(NC(c2[nH]nnc2C)=O)CN(C(=O)CNc2cnn(C)c2)C1 82548,CC1CCCC(NC(C2(C(C)NC(=O)COCCC(C)C)CC2)=O)C1 82549,c1(C(=O)NC(C(=O)N(CCNC(c2c(C)occ2)=O)C2CC2)C)cccc(Cl)c1 82550,C1(C(=O)NCc2cncc(C)c2)CCN(C(=O)COCCN(C)C)CC1(C)C 82551,C1(C(=O)N(CCC(C)(C)C)C)(NC(C(CC)SC)=O)CCN(C)C1 82552,C(=O)(C(C=CC)NC(=O)C(C)OCCOC)NCC1CC(=C)C1 82553,C1(CNC(CN(C(C(C)OCC)=O)C2CC2)=O)CCCC12CCC2 82554,c1(C(C)(C)C)ccccc1C(=O)NCC1C2CC2CN1C(C1C2CC3C(C2)C13)=O 82555,c1(OC(CN(CCOC)C(C)N)=O)ccc(OC)cc1.c1(C)cccc(OC)n1 82556,N(C(=NCCN(CC(F)(F)F)C(C)(C)C)NCCN1CCCC1)C1C(C)OCC1 82557,C1(C(=O)NCCCCCN(C(=O)CC2COC(=O)N2)C)(COC)CCCO1 82558,C1(CNC(=O)CSC2CC2)CCCC1NC(C1CCC1)=O.c12c[nH]nc1N2 82559,C1(C)(C(N(CC2CCCSC2)CC2CN(C)C2)=O)CCC2CC2C1 82560,N1(C2CCN(CC=C)C2=O)CC(NC(=O)OC(C)(C)C)C(C)(C)C1 82561,c1(C(=O)NC)ccc(CNC(=O)N(CC(c2cccc(OC)c2)O)C)cn1 82562,C12(CN)CC(C1)C(NC(c1cncc(-c3ccoc3)n1)=O)CO2 82563,C=CC(O)C(=O)OC.N12CCC(C1)OCCCCNC(=O)C2 82564,c1(N2CCN(C(CC)=O)CC2)nc(NCc2cn(C)nn2)c2ncn(CC)c2n1 82565,c1(C(=O)NCC2(C)CCCN2C(c2ncccc2Br)=O)n[nH]c2c1COC2 82566,C1(NCC=Cc2ccccc2)COCCC1c1nnnn1C1CCCCC1.CC=C 82567,C1(NC(c2c(CC)nco2)=O)CCC2CCN(C(C3(C(F)(F)F)CC(C)C3)=O)C1C2 82568,c1(C(N2CC3C(N(C)C)C3C2)=O)nccc(=NCCOC2CCOC2)[nH]1 82569,c1(C(C)C(N2CCC(CNC(C3(O)CCSCC3)=O)C2)=O)c(F)cccc1F 82570,C(=O)(C1=Cc2ccccc2C1)N1CC(NC(C2C3CC3C3CC23)=O)(CF)C1 82571,N1(C(C(C2CCCO2)OCC)=O)CC2(CCCCN2C(c2ccnc(S)c2)=O)C1 82572,CC(C)(C)CC(F)C(=O)N1CCC(NC(c2cc3cnccc3[nH]2)=O)C(O)C1 82573,CCCC(C(=O)N1CCC(C)N(C(c2cc(C)c(F)c(C)c2)=O)CC1)S(N)(=O)=O 82574,N1(C(C(CC)OC)=O)CCN(CCF)CC1.N12CCC(C1)CC2=O 82575,Cc1coc(C2CC2)c1C(=O)NCC(CC(C)C)NC(c1cnco1)=O 82576,Cc1cc(=NC(=O)NC(CO)CC(O)C(C)(C)C)[nH]n1-c1ccc(Cl)c(F)c1 82577,Nc1sc2ccccc2c1C(N1CCOCC(NC(c2nccnc2N)=O)C1)=O 82578,CCC(CC(C)C)C(=O)NC1CC(F)(CNC(c2cc3ccccc3o2)=O)C1 82579,CCC(CC)(C(=O)N1CCC(NC(=O)CCC(C)(C)F)C(C)C1)OC 82580,c1(OC)cc(C)cnc1C(=O)N(C)CC1C2CN(C(C3CC3C)=O)CC12 82581,c1(C(=O)NCCN(C(c2ncoc2C(C)C)=O)CC)cnc(CC(C)C)cn1 82582,CCCC(O)CCCNC(c1nnnn1C1CCCC=C1Br)C1(C2CCC2)CC1 82583,C1(C(=O)NC(C(=O)NC2CN(C(C)C)C(=O)C2)C2CC2)CN(C)CCN1C 82584,CC1CN(C(=O)C2=CCC(NC(=O)CSC(F)(F)F)C2)C(C)C1C 82585,Cc1cccc(C(=O)NCC(N2CCCCC2CCCC(=O)NC(N)=O)=O)n1 82586,Cc1nc(CO)ncc1C(N1CC(NC(C2OCC2(C)C)=O)CCC1C)=O 82587,c1(C(=O)NC2(C(N3CC4CCC4C3)=O)CCCCC2)ccc2[nH]ccc2n1 82588,C(=O)(C(F)C(=O)NCCN(C(=O)CCCSC)C1CCCCC1)OCC 82589,CCC(C(=O)NC1CC(F)(CNC(=O)C(C)CC2CC2)C1)OC 82590,C(CCCc1ccccc1)(c1ccccc1)NC(=O)NC(C)Cc1nc(O)n[nH]1 82591,CCS(=O)(=O)C=CC(=O)NCC(C)CNC(=O)CN1C(=O)CNC1=O 82592,C12(C(N3CC(CNC(C(CC)O)=O)C(C(F)(F)F)C3)=O)CCC(CC1)CC2 82593,c1(C(=O)NCC(COC)NC(=O)C(C)(C)n2ccc(C(=O)O)n2)ccc(C)n1C 82594,C1(CNC(c2[nH]cc(CC)c2)=O)CCCCN1C(C1(n2nccn2)CC1)=O 82595,C1(NC(Cc2c(C)nc(S)s2)=O)CS(=O)(=O)CC1NC(c1cc(O)nn1C)=O 82596,C1(CCNC(C2C(C)CCC2)=O)CSCCN1C(=O)COc1ccsn1 82597,C1(C#CC(=O)NCCC2CN(C(C3CCCS3)=O)CC2C)(CC)CC1 82598,Cn1cnc2nc(=NCc3cncs3)[nH]c(NCC3C(F)(F)C34CCC4)c12 82599,C=C(Cl)C(C)(C)C(=O)N1CC(N(C(=O)CCc2cc(OC)c(C)o2)C)C2(CC2)C1 82600,CC(C)CC(C(=O)NC12CC1CN(C(c1cn3cc[nH]c(=O)c3n1)=O)C2)C(C)C 82601,C12(C(=O)Nc3cccc(Cn4ccnc4)c3)CCCC1C2(F)F 82602,C(=O)(N=c1[nH]onc1C1CC1)OC.c12cn(nn1)C(COC)C(=O)N(CC)CC2 82603,C(CCCCCNC(c1ccc[n+]([O-])c1)=O)NC(c1ccsc1)=O 82604,C1(C(N2C(CCCCNC(=O)OC)CC2)=O)CC(OC2CC2)CN1C(=O)CC#N 82605,C1(N(C(C(C)Cc2ccccn2)=O)C)CCCN(C(c2cncnc2)=O)CC1 82606,C12(NC(c3cn(C)nc3)=O)COCCC1CN(C(=O)C=Cc1cnc[nH]1)C2 82607,Cn1cc(C(=O)NC2CCCCC2NC(c2nc(C3CC3)cs2)=O)nc1O 82608,C1(C(=O)NC2(CC=C)CCCCC2)CN(C)CCN1C(c1ccc(F)c(O)c1)=O 82609,C1(OC)CC(NC(C2(C)CCCN(C)C2)=O)CN(C(c2ccc(C)cc2Cl)=O)C1 82610,c1(OCC)cc(OC)ccc1C(=O)NCCC1(NC(=O)CC(C)C)CC1 82611,C(CC1CC1)(C(=O)N(C(CC1CC1)C(=O)N1CCC(c2ccon2)C1)C1CCCC1)OC 82612,Cc1cc(C(N2CC3CCC3(CCNC(c3cnc(N)cn3)=O)C2)=O)cc(C)c1 82613,C1(C(=O)NC(CC(=O)OC)C)CN(C(=O)Cn2cc(C)cn2)CC1C1CC1 82614,CC(CC(=O)c1ccc(F)cc1)C(=O)NCCCCCNC(=O)C(C)(F)F 82615,C(=O)(C(O)C(F)(F)F)N.C12CCC(C1)CCC(=O)N2.C(C(C)(C)C)N(CC(=O)OC)C 82616,c1(NC(C2CC(C)CN2C(c2cc3sccc3[nH]2)=O)=O)nc2ccccc2s1 82617,C1(NC(C(=O)N(C)C)=O)CC(C(=O)NC2C(O)CC2O)C12CCC2 82618,c1(OC)cc(C(=O)NCC(CNC(=O)CCSC2CCCC2)OC)cc(F)c1 82619,c1(OCC)c(Br)cccc1S(=O)(=O)N1CCC(SC(F)F)C1 82620,C12(C(N3CC(CC=C)(NC(C4CCC(C)(C)CO4)=O)C3)=O)CCCC1CC(=O)C2 82621,C1(C)(CC)CC(C(N2CCC(F)(Cn3cc(C(O)CC(C)C)nn3)C2)=O)CCO1 82622,n1(CC)ncc(Cl)c1C(N1CCCCC1c1ccc(Br)cc1)C(=O)NC(C)(C)C 82623,Cc1ccc(C(=O)NC2CCC(C)N(C(C3CC4(C3)CC(O)C4)=O)C2)cc1C#N 82624,C1(C(N2CCC(CCNC(C3C(C)(C)CC3)=O)CC2)=O)OCCOC12CCC2 82625,c1(CN(C(=O)CNC(C2CCCO2)=O)C)ncc(Br)s1 82626,c1(C(=O)NCC2(C)CCC(NC(c3ccc(Br)o3)=O)C2)cnc2n1CCC2 82627,c1(CCCC)nc(C)c(C(=O)NCCNC(C2C3CN(CC(=C)C)CC23)=O)s1 82628,CC1C(=O)N(C)CCN1C(=O)C(C)(c1ccccc1)NC(=O)CCCC1CC1 82629,Cc1cc(N2CC(NC(=O)C3=C(Cl)CCC3)CC(C)(C)C2)cc(C#N)c1[N+](=O)[O-] 82630,CCCC(C(=O)NCc1ccccc1)N1CCCC1CC 82631,c1(CC)cc(C(N2CC(CNC(c3cc(Br)n[nH]3)=O)CC2C)=O)cc(Cl)n1 82632,c1(OS(CC2CCCC(C)C2)(=O)=O)ccc2cccnc2c1 82633,C1(NC(C2C(NC(C(CO)OC)=O)CCO2)=O)C=C(C)CCC1 82634,N1(C(CCC=C(C)C)=O)CCN(C(c2cccnc2C(N)=O)=O)CC1C(F)F 82635,c1(C(N(CCC(=O)NC(C2CCCC2)C)CCO)=O)cccnn1 82636,CC#CC1CCN(C(c2cc(CNCC3CC3CC)nn2C)=O)C1 82637,Cc1cc(O)ncc1NC(C1(C)CC(O)CN1C(=O)C(C)C(F)(F)F)=O 82638,c1(OC)ccc(C(=O)C(=O)NCC2CCCN2CC2CC2)cc1 82639,C1(CNC(=O)CCc2nc[nH]n2)CCCCC1C(N1CC=CC1)=O 82640,N1(S(CCC)(=O)=O)CCCCC1C(=O)NCC(C)CCNC(=O)CS(N)(=O)=O 82641,N1(C(=O)CC2CC2)CCCCC1C1CCCN1C(=O)Cc1ccccc1 82642,C1(CCNC(C(C(C)C)OC)=O)CCCN(C(c2nscc2N)=O)CC1 82643,CN1C2CCCC1CC(n1cc(C3CCN3C(c3ccc(Cl)c(F)c3)=O)nn1)C2 82644,Nc1cc(C(=O)NC2CCCCC2O)ccc1OCC1CCCCCO1 82645,C1(F)(C(=O)NCC(=O)NCC#C)CCN(C(=O)C(CC2CC2)OC)CC1 82646,C(=O)(CC(C)(C)COC)NCC1N(C(c2cc(C(C)=O)[nH]c2)=O)CC(OC)C1 82647,C(=O)(C(C)CC(F)F)NC1CN(C(c2c(C(C)C)ccs2)=O)CC1O 82648,Cc1ccc(C(N2CC3CCC2C3NC(C2(C)CC2(F)F)=O)=O)cc1OC(F)F 82649,N#Cc1ccc(S(=O)(=O)N2CCCC3CC2C3)cc1NCc1c[nH]c(=N)s1 82650,c1(C(N(CCN(C(C2CC(C)(C)O2)=O)CC)CC)=O)cc2cccnc2s1 82651,N1(C(CC2CN(C(C)=O)C2)=O)CC(NC(=O)C2CC2)CC1CSc1ccc(C)cc1 82652,C1(C(N2CCCC2)=O)COC2(C1)CN(C(C1(c3ccon3)COC1)=O)C2 82653,N1(C(CC2C(C)CCO2)=O)CCCCC2(CCN(C(C3CS(=O)(=O)C3)=O)C2)C1 82654,N1(C(c2c(CC)nn[nH]2)=O)CCOC(C(=O)NCc2nc(C)cs2)CC1 82655,C(CC(CC)C(=O)NCCCCCCN(C(=O)CN(C)CCC)C(C)C)=CC 82656,C1(NC(C2C(OC)CC2)=O)CC2CCC(C1C)N2C(c1cc(C)ncn1)=O 82657,C1(NC(C(N2CCOC2=O)C)=O)CC2(C1)CC2NC(c1ccc(Cl)s1)=O 82658,C1(C(=O)NCCCCC2C(C)C2)CN(C(=O)CC2CCCC(=O)C2)CC(C)(C)C1 82659,N1(C(c2cn(C)nc2)=O)CCN(C(c2cc(S(N)(=O)=O)ccn2)=O)C2(CCC2)C1 82660,N#Cc1cccc(I)c1NC(C1CCCCC1NC(c1ccc(CO)cc1)=O)=O 82661,c1(NC2(CC(=O)NC(CC)C(C)O)CCC2)ncnc2ccc(OC)nc12 82662,c1(CNc2c(OC)cn(-c3ccccc3)n2)ccc(I)cc1OC 82663,c1(C(=O)NCC(C)CN(C(=O)CN2CCSCC2)C)conc1C1CCCO1 82664,c1(NC)c(C(=O)OC(c2noc(C)n2)C)ccn1C 82665,Cc1c(F)ccc(C(=O)NCC(CO)NC(=O)CC2OCCC2(C)C)c1C#N 82666,Nc1ccc(C(=O)N(CCC(=O)NCCC2CCSC2)CC2CC2)nc1 82667,C1(NC(C2N(CC)CCOC2)=O)CC(N=c2[nH]c(C#N)c(Cl)s2)C1 82668,Cc1ccnc(-n2nc(C)cc2NC(=O)NC(c2noc(C)n2)C)c1 82669,C1(CCNC(C(C)SC(C)C)=O)CCN(C(C23CCCC2C3)=O)CC1 82670,N1(C(c2cnn(CC(F)F)c2)C(=O)NC)CCOCC2(CSC2)C1 82671,C(=O)(C(C)(C1CCCOC1)Sc1conc1C(C)C)OCC 82672,CC1C(C)N(C(c2coc(C#N)c2)=O)CCN1C(=O)Cc1cc(F)ccc1O 82673,c1(NC(c2nc(NC(c3c(=N)[nH][nH]c3)=O)sc2)=O)cc(O)nc2ncccc12 82674,c1(C(C)(C)C)ccc(CN2CCNC(=O)CC2)c(O)c1.C123CC(C1)(C2)C(=O)N3 82675,C1(C(N2CCC(C3CCCN3C(c3ccc(=O)oc3)=O)C2)=O)COCCC1CO 82676,c1(OC)cc(O)c(C(N2CCC3CN(C(c4ccsc4Cl)=O)CC23)=O)cc1OC 82677,C(=O)(C(F)(F)C(O)CC)N(CC(CC)NC(=O)Cc1sc(C)nc1C)C 82678,C12(CNC(Cc3c(OC)cccc3Cl)=O)CCCC1CN(C(=O)Cc1nc[nH]n1)C2 82679,N1(C(=O)COCC2CCCCO2)CC2CC(C1)CN(C(c1cocn1)=O)C2 82680,Cc1cc(N)c(C(=O)NCC2CC(NC(C3C4CCN3CC4)=O)C2)c(F)c1 82681,C(=O)(C1CCCc2cncn21)NC(C)CCNC(c1c(O)ccc(Br)c1Cl)=O 82682,c1(N(CC(C#C)C)C)sc(C(C)(C)C)cc1C#N 82683,c1(C(=O)NCC(CC=C)NC(C2CS(=O)(=O)C2)=O)cnc2c(F)cc(C)cc2c1 82684,CCCCCCCN=c1nc(N(C)Cc2ncccc2C)c2ccc(C)cc2[nH]1 82685,C1(CCC(=O)NC2C(NC(CN(C(=O)OCC)C)=O)CCC2)NC(=O)NC1=O 82686,C1(F)(CNC(C(C)(C)OC(C)C)c2nnnn2CC2CC2)COCCOC1 82687,C#Cc1cc(C(N2CCC(O)(CNC(c3ccc(Cl)nc3O)=O)C2)=O)ccc1C 82688,CC(=O)CCCC(C)C(=O)N1CCC(C)(C(=O)NC(C)(C)C(F)F)C1 82689,C1(C(=O)NC(C(C)NC(CNS(CCCOC)(=O)=O)=O)CO)CC12CC(F)(F)C2 82690,C1(N(C)C(C2CCCOC2)=O)CCCN(C(=O)C(C)(C)c2ccno2)CC1 82691,c1(C(N2CC(CC(C)NC(=O)C(=CC3CCCCC3)F)C2)=O)cccc(N)c1 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82745,c1(CN(C2CN(C(c3ccccc3C#N)=O)C2)C)cnc2ccc(F)cn12 82746,N1(C(Cc2c(SC)cccc2)=O)CCCC(O)C1C.CCC1CC1 82747,C1(NC(c2c(CC)scc2)=O)CCC2(CC1)CC2NC(=O)CCC1CC1C 82748,C1(NC(c2cc(C)n(C)c2)=O)C2CC1CN(C(C1(COC(C)C)CC1)=O)C2 82749,C(c1ccc(F)cc1)=C(C(=O)NCC1(C)N(C(C2C(=C)C2)=O)CCC1)C 82750,c1(C(C(=O)NC2COC2)N(CC(CCC)C)C)cc2ccccc2oc1=O 82751,C1(C(=O)Nc2c(C)ncnc2)CC(F)CN(S(=O)(=O)C(F)(F)F)C1 82752,c1(CC)ccc(C(=O)NC2CC2CNC(=O)C(C)OCC2CCCO2)s1 82753,c1(C(=O)NC2CC3CC(NC(c4scnc4Cl)=O)C2C3)cccc2c1OCC2 82754,c1(C(CO)NC(c2ccn(C(F)(F)F)c2)=O)ccccc1F 82755,C=C(C)CC1C(=O)N(C)CCCCOCCC(=O)N1.C(C)(=O)OCC 82756,Cc1ccc(CCC(=O)NCCCCC(C)NC(=O)C(C)C2CC2)cc1 82757,C(=O)(C(C)CCCCCCC)N1CCN(C(C2(CC=C)CC2)=O)C(CCOC)C1 82758,N1(C(CCc2cccc(C)c2)=O)CCN(C(C2CC2F)=O)CC1C 82759,N1(C(C2(CC)CCCO2)=O)CCC2(COC(CNC(=O)C(O)CC(C)(C)C)C2)C1 82760,N1(C(=O)CNC(C)C)CCCC(O)(CNC(=O)CC2CN(C(C)=O)C2)C1.C(C)(C)(C)O 82761,N1(C(C2(CC)CCC2)=O)CC=CC1(C)C(=O)NCCc1nccc(O)n1 82762,c1(OC)cc(C(N2CCCC(C)(C(=O)NC3CSCS(=O)(=O)C3)C2)=O)cc(OC)n1 82763,CS(=O)c1cccc(C(=O)NC(CNC(c2ccnnc2)=O)CO)c1 82764,N1(C2C(C(C)(C)C)P=N2)CCCCC1C(N1CC2(CSC2)C1)=O 82765,c1(OC)cccc2[nH]nc(C(=O)NCCNC(C3CCC(F)(F)C3)=O)c12 82766,C#Cc1cn(C)nc1C(N1CCC(CO)(CNC(c2cccnc2N)=O)CC1)=O 82767,N1(C(CC(C=C)CCC)=O)CC=C(CC(=O)N2CC(C)CCC2CC)CC1 82768,N1(C(c2ccc(CNC(Cc3cn(C)nn3)=O)o2)=O)CCCC1(C)C1CCC1 82769,c1(C(=O)NCCCN(C(CC(C(=C)C)OCC)=O)C(C)C)cnc2ccsc2c1 82770,N1(C(CCOC)=O)CCC2(CC1)CCN(C(=O)C(N1CCOC1=O)C)CC2C 82771,N1(C(C2(C)CC(C)C2)=O)CCOCC(F)(CNC(c2nccc3cc[nH]c23)=O)C1 82772,C1(SCC(=O)NC2(C)CC(NC(C(C)N(C(C)=O)C)=O)C2)Cc2ccccc2C1 82773,Cc1nc2c(F)cccc2cc1C(N1CC2CC1C2NC(c1cnsn1)=O)=O 82774,Cc1nc(C(N2CCC(C(C)NC(=O)CN3CCC(CO)CC3)C2)=O)cc(O)n1 82775,CN1CC(NC(=O)Cc2ncc[nH]2)C(c2ccccc2Br)C1 82776,C1(NC(C(C2CCN(C(CCCC#C)=O)C2)(C)C)=O)CCn2ccnc2C1 82777,n1(CC(=O)NCCCC(CO)NC(CCNC(N)=O)=O)cnc2c1CCCC2 82778,c1(CCCC(=O)NC(c2cn(C3CCCC3)nn2)C)ccc(Cl)cc1Cl 82779,N1(C(C(CNC(c2cc(O)cc(OC)c2O)=O)O)=O)CCn2c(C)nnc2C1 82780,C1(C)(CNC(c2c(CC)nn[nH]2)=O)CCCC1NC(=O)C(F)n1ccnc1 82781,C1(C#N)(SC)CN(C(C2CCN(C(=O)Nc3ccccc3)C2)=O)C1 82782,CCC(O)CC(=O)N1CCCC1C(=O)NCCN=[N+]=[N-] 82783,N(C1CCc2c(Br)cccc21)C(C1CCCC(N)CC1)=O 82784,C1(C(=O)NC2(CC=C)CCN(C(=O)Cc3cnns3)C2)CCC=CCCC1 82785,C1(C(=O)NCC(=O)NC(C=C)(C)CC)CC2(CCC2)CO1 82786,c1(NC(C(=O)NCC2(C(=O)OC)CC2(F)F)=O)ccc(C#N)c(F)c1Br 82787,C1(C(=O)NC2C(NC(=O)Cc3cccnc3)CCC2)CCC2CCC1O2 82788,C1(C(N2C(CN(C(C3CCC(C)O3)=O)C)CC(F)C2)=O)NC(=O)OC1(C)C 82789,c1(C(=O)NC2C(C)CN(C(=O)C(C)(C)C3CCOC3)C2)cn2ccsc2n1 82790,C1(C(N2C(CNC(C3CC(SC)C3)=O)CC(C)CC2)=O)CC2CCC(C1)C2=O 82791,N1(CCNC(C(C2N(C(Cn3c(C)nnn3)=O)CCC2)(C)C)=O)CCOC(C)C1 82792,O=C(N=S1(=O)c2ccccc2CCC1F)C1CC2CCC1C(C(=O)O)C2 82793,C1(NC(c2cccc(O)n2)=O)COCCC1C(N1CC(c2nncs2)C1)=O 82794,C(=O)(C1=CCC(C(F)(F)F)OC1)C(C1CC2CN(C(=O)C3=CCCOCC3)CC12)=O 82795,C(=O)(C1=C(c2csc(Cl)c2)N(CCOC)C(=O)NC1c1ccc(CC)o1)OCC 82796,N1(C(CC(COC)C)=O)CC(C)(C)C(NC(=O)C(C(C)C)N(C)C)C(C)(C)C1 82797,CC(CC(=O)N(CC(C)NC(=O)Cc1nnc(O)s1)C)P(C)(C)=O 82798,c1(CNC23CC(C(=O)NC(c4ccc(C)o4)CC)(C2)C3)c(F)ccc(Cl)c1F 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83047,CCCCC(C(=O)N(CCCCC(=O)NC(c1cncn1C)CO)C)N(C)C 83048,n1(CC(=O)NC(CNC(C(CC)O)=O)(CC)CC)ccc2ccc(Br)cc12 83049,CN1C(C(=O)NCC2(NC(=O)Cc3ccc(O)cc3F)CC2)CCS1(=O)=O 83050,N1(C(Cc2c(CC)con2)=O)CC(NC(=O)C(O)CSC)C(S(C)(=O)=O)C1 83051,c1(C(=O)NC2C(F)CCN(C(C(C(C)C)O)=O)C2)cn2ncccc2n1 83052,c1(OC)ccc(CC(=O)NCC2CC2NC(C2CCCOC2C)=O)nc1 83053,N1(C(c2cncn(C)c2=O)=O)CC2CN(C(=O)C(CN(C)C)N(C)C)CCC12 83054,c1(C(=O)NCC(c2ccc(C)cc2)NC(=O)NC2CCC3CC23)ccc(C)c(C)n1 83055,Cc1ccc2nc(C(=O)NC3CCN(C(=O)C(C)c4cccs4)CC3C)cn2c1 83056,N1(C(CNC(=O)OCC=C)=O)CC(N(C)C(c2scnc2C(F)(F)F)=O)C(O)C1 83057,C12(CNC(=O)NCC(C(C)C)O)CCC(CC1)O2 83058,C(=O)(C1=C2CCN=C2NC=C1)N1CC2C(NC(C3COC4(CCC4)CO3)=O)C2C1 83059,N1(C(C(C)OCC)=O)CC(F)(F)CC1C(=O)NCC1CCCC(O)C1 83060,c1(NC(=O)CCCOC)ccccc1-c1ccc(SC)cc1.CCO 83061,Cc1oc(Cl)nc1C(=O)N(C)CC1CCN(C(c2cncn2C)=O)C1 83062,C#Cc1ccnc(C(=O)NC2CN(C(=O)C(O)CN3CCCC3)C(C)(CC)C2)c1 83063,C=CCC(CNC(=O)CC1CC1CNC(=O)CCOCC(C)C)CC(C)C 83064,C1(C(=O)NC(c2occ(C(N(CC(=C)C)CC)=O)n2)C)C2CC3C(C2)C13 83065,N1(C(C2CCOC(F)(F)C2)=O)CC2(CCN(C(C3CCCC4(CC4)C3)=O)CC2)C1 83066,c1(C(=O)NC2CN(C(c3c(C)sc(Cl)n3)=O)C(C)CC2)cc[nH]c(=N)c1[N+](=O)[O-] 83067,C1(NC(Cc2ncn(C)c2)=O)CCCC12CN(C(=O)C(C1CCOCC1)O)C2 83068,C#Cc1ccc(C(N2CCC3CCC23CNC(c2ccc(Cl)c(F)c2)=O)=O)cn1 83069,c1(NCC(=O)NCC(C)(CO)NC(=O)CC2NC(=O)NC2=O)ccc(F)cc1F 83070,C1(C(=O)NC(C(=O)NC(c2ccncc2F)C)(C)C)CCCC(O)C1 83071,N1(C(c2sccc2Cl)=O)CCC2CN(C(=O)C3CCCc4ccnn43)CC2CC1 83072,N1(C(C(C2CC2)OCCC)=O)CC=CC1C(=O)NCc1cc(C(=O)OC)on1 83073,c1(C(N2CCCC(N(C)C(C)=O)C2)C(=O)NC)cnc(C)n1C 83074,Cn1nc(C(N2CCCCC2Cn2cc(CNC=O)nn2)=O)c2c1CCSC2 83075,C1(CNC(CCOC(C)C)=O)CC(NC(C2(C(F)F)CCC2)=O)CCO1 83076,N1(C(CS(=O)(=O)N(C)C)=O)CC2(CCCC2NC(C2CC3CC3C2)=O)C1 83077,c1(N(C(C(C2N(C(C)=O)CCC2)(C)C)=O)C)ccc2c(c1)OCCO2 83078,c1(C(=O)NCCC(C)N(C)C(C2CC2c2ccc(Cl)cc2)=O)nc(Cl)ccc1N 83079,C(=O)(CS(=O)(=O)CC)NCC1N(C(C2CN(S(CC)(=O)=O)C2)=O)CC1 83080,N1(C(COC2(C)CCC2)=O)CCOC(CCNC(c2cc(F)c[nH]2)=O)C1 83081,c1(OC)cnc(Cl)nc1N1CCC(Cc2ccccc2)C1.C12CCCN(C1)C2=O 83082,c1(C(N2CC3CCCC23)C(=O)NCc2cccs2)nc2c(s1)CCCC2 83083,C12(C(N3CC(OCCNC(=O)CC4CCCO4)C3)=O)C3CCC(CC13)C2(F)F 83084,N1(C(C(C)SC)=O)CCC(NC(c2ccn(-c3ccncc3)n2)=O)C(O)C1 83085,c1(C(N2CC(CNC(C(C)(CO)OC)=O)C(C)C2)=O)ccn2c1CCCC2 83086,C(CS(=O)(=O)NCC1CC1C#N)(C1CC1)OC 83087,c1(C(N(CC(C)NC(=O)Cc2nc[nH]n2)C)=O)ccc2nnn(C)c2c1 83088,N#CC1CN(C(C2CC3CCC2N3C(c2ccccc2F)=O)=O)CCO1 83089,N1(C(c2scc(CC)c2)=O)CCN(C(=O)C(C)(C)N2CCCC2)CC1C1CC1 83090,c1(C(CNC(C2CC2C2CC2)=O)NC(COCC)=O)cccc(Cl)c1 83091,c1(OC)nccc(C(N2CCC(NC(=O)C(C)=C(C)C)C(CO)C2)=O)c1F 83092,C(C(CNC(=O)CC1CCC(C)O1)S(C)(=O)=O)NC(C(COC)(F)F)=O 83093,c1(NC(c2ccc(Cn3cc(CSC)nn3)o2)=O)ccnc(CC2(F)C(C)C2)c1 83094,C1(C(=O)OC)CCCC1Cn1cc(-c2ccn(C3CCOCC3)n2)nn1 83095,C(CNC(=O)C(O)Cn1cncn1)(CC(=O)NCC(O)CC(C)C)OC 83096,c1(C(N(CCN(C(C2C(CC)CCC2)=O)C)C(C)C)=O)cc(=O)n2nccc2[nH]1 83097,CC(C)(C)CCNC(=O)CCC1CCC(=O)C1.C(=O)(CCc1cn[nH]c1)NC1CC1 83098,CC1(C(=O)NOCC2CCOC2)CCN(C(C2CC23CC3)=O)CC1 83099,C(=O)(CC(C)c1cnn(C)c1)NCCC1CC(NC(COC(CC)(C)C)=O)C1 83100,C(C1=NOC2CN(C(c3cc(Cl)c(Cl)s3)=O)CC12)NC(c1cn(C)nc1)=O 83101,CC(C)CS(=O)(=O)CC(=O)NCC1CCN1C(C1CC2(C1)CC21CC1)=O 83102,N1(C(CCSCC)=O)CCN(C(=O)CCc2ccc(OC)cc2)C(CC)C1 83103,C1(NC(C2(C(N(C(C)C)C)=O)CC2)=O)CCCC1NC(=O)C1=CCC1 83104,c1(C(=O)NC)cccc(OC(C)C(=O)NC2CC2NC(c2c(C)coc2C)=O)c1 83105,CC1(C)C(C)(C)C1(F)C(=O)NC1CN(C(=O)C(CO)c2ccccc2)CC1CO 83106,C1(CCNC(C(C)SCC)=O)CN(C(=O)C=CCn2cncn2)CCC1(F)F 83107,C1(O)(C(N2C(C)(CNC(C3CN(C4CCC4)C3)=O)CCC2)=O)CN2CCC1CC2 83108,C1(C(N(C)Cc2cc(OC)no2)=O)C=CCCN1C(=O)Cn1cnnc1O 83109,C=C1CC2(C1)CC(C(=O)N(C1CC3CC1N(C(=O)C(C1CCCCC1)F)C3)C)C2 83110,C1(N(C(Cc2c(C)con2)=O)CCF)CCCN(C(C2OCCC2C(C)C)=O)C1 83111,c1(CC(=O)NCC(C(C)C)NC(=O)C(C)CO)cnc2n1CCCC2C 83112,C1(NC(CNC=O)=O)CN(C(=O)Cc2cccc(Cl)c2)CC1n1cccn1 83113,C1(CCNC(C2(NC(SCC(C)(C)C)=N)CC2)=O)CCOC1=O 83114,c1(NC(=O)C(N2CC(F)CC2CO)=O)cnncc1Br 83115,C1(NC(c2ccc(C(C)C)o2)=O)CCCCN(C(C2CC3(CCO3)C2)=O)C1 83116,C1(NC(CC2C(C)CCO2)=O)CC(F)CN(C(=O)CN(S(C)(=O)=O)C)C1 83117,c1(NC(C23C(CN(C(C(C)OCC=C)=O)C2)C3)=O)cccc(I)c1Cl 83118,C1(CC)CNCCN(N2CCCC3(CC2)NC(=O)NC3=O)C1 83119,c1(CC(=O)NC(CNC(=O)COCCF)C2CCC2)ccsc1Br 83120,C(=O)(C(C)(F)C(C)(C)F)N(C)CCN(C)C(C1(F)CCCOC1)=O 83121,CC(C)CC(C(=O)NC(C)C(C)C(=O)N1CCCC(CF)C1)N(C)C 83122,C(=O)(CS(=O)(=O)Nc1ccco1)NCC1CN(C(C2C(=C)CC2)=O)C1 83123,C1(CNC(CC2N(C)CCCC2)=O)CC(F)(F)CN1C(=O)CCCCO 83124,c1(CC)ccc(Br)c(C(=O)N(CC(C)CNC(=O)C#CC2CC2)C)c1 83125,c1(CCC(N2CCC(Cn3cc(CC(C(C)C)O)nn3)C2)=O)ccc(F)cc1F 83126,C(=O)(C(F)C(C)CNC(=O)CN1CCCC1)N(CC(CC)CC)CC 83127,C1(CCC#C)CCCN1C(C1CCC(CNC(=O)Cc2cc(C)[nH]n2)C1)=O 83128,c1(OC)cccc2c(C(C)NC(=O)Nc3n[nH]cc3OC(C)(C)C)c(C)[nH]c12 83129,CC1CC(CNC(c2cn(C)cn2)=O)CN1C(c1cc(C2CCC2)nn1C)=O 83130,c1(C(=O)NC2CCC(NC(CC(CCC)(C)C)=O)C2)ncc(F)c2ccccc12 83131,CC1(NC(C2(c3cn[nH]c3)CC2)=O)CN(C(c2cnsn2)=O)C1 83132,Cc1cc(Br)cc(C)c1CN1CCN(C(c2cc(O)n(C)n2)=O)C(C(F)(F)F)C1 83133,N1(C(c2nc(CNC(=O)C(C3CC3)C3CC3)oc2)=O)CCCC(C2CC2)CC1 83134,N1(C(C(CNC(c2c(CC)ncnc2)=O)O)=O)CCN2CCCCC1C2 83135,c1(C(N(C2CC(NC(C3(CC=C)CCCC3)=O)C2)C)=O)ccccc1C1CCC1 83136,C1(NC(C(C)OCCC#C)=O)CN(C(c2cnn(C)c2)=O)CC12CCC2 83137,c1(OCC)ccc(C(C)NCC(C)C(C)(C)C)c(Cl)c1OC 83138,C1(C(=O)NC(C)CNC(=O)Cc2csc(CC(F)(F)F)n2)CC(C)(C)CCO1 83139,C#CCCCC(C)C(=O)NC1(CNC(=O)Cc2nocc2CC)CCCCCC1 83140,N1(C(C(C(=O)OC)OC)=O)CCOC2(C1)CN(C(=O)COC1CCCCCC1)C2 83141,C#CC1CCC(CN2CC(C)CC(C(=O)NCc3c(C)cccc3F)C2)CC1 83142,C1(NS(=O)(=O)CCc2c[nH]nc2O)CCC12CCCCC2 83143,CC(CC(=O)NC1CN(C(=O)COC(F)(F)F)CC1O)C(=O)c1ccccc1F 83144,CC1(CNC(=O)CC2CCCN(C(C3(F)C(C)(C)C3(C)C)=O)C2)NC(=O)NC1=O 83145,c1(C(=O)NCCSCC(=O)NC(c2nncs2)C)cccnc1S 83146,N1(C(CCCNC(C)=O)=O)CCC(CO)(CNC(=O)CN2CCNC(=O)C2)C1 83147,CCC(CC(c1nnnn1C1(C)CC1)NCCc1ncc(F)cn1)OCOC.C1CC1 83148,C#Cc1cccc(CC(=O)N(c2nc(NC(C)(C)CCO)ns2)C)c1 83149,C1(CN(C(C(C)SCC)=O)C)CCN(C(=O)C(O)CC2CCOCC2)CC1 83150,C#CCC(CC(F)F)C(=O)N(C1CCC(NC(=O)C2=C(Cl)CCC2)CC1)C 83151,c1(SC)cc(C(=O)NCC2CC(=O)N(c3ccc(OC(C)C)cc3)C2)nn1C 83152,Cc1c(CCC(N2CC(O)(CCNC(=O)C(CCO)N(C)C)C2)=O)cnn1C 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83188,N1(CC(=O)NCCCCN(C)C)CCC12CC(CO)C2 83189,C=C1CC(COC)N(Cc2cn(-c3cccc(Oc4cccc(C)n4)c3)nn2)C1 83190,CC(C)S(=O)(=O)C(C)C(=O)NCC(C)(C)NC(=O)Cn1cc([N+](=O)[O-])ccc1=O 83191,c1(OCC)oc(C)nc1C(=O)NC1CC(C)N(C(c2cscc2F)=O)C1 83192,C1(OC)CN(C(=O)CN2CCC(C)C2)CC1NC(C1(C)SCCCS1)=O 83193,C1(C)(c2n(C)cnn2)CCCN1C(C1(C(F)(F)F)CC1)=O 83194,C1(CC(=O)NC2CCN(C(=O)CC3CC4(CC4)C3)C2)CC2(CCC2)C1 83195,c1(NC(c2c(C)cncc2F)=O)ccc2c(n1)CCC2=O.C12CC(C1)CNC2=O 83196,C1(CNC(C(CCC)F)=O)N(C(=O)CN2CC(C)(OC)C2)CCCC1(C)C 83197,N1(C(C(c2n(C)ncc2)O)=O)CC2(C1)CN(C(=O)C(F)C(C)(F)F)C2 83198,C1(C(=O)NCC2N(C(c3c(C)ccc(N)c3)=O)CCC2)CCCN1S(=N)(=O)N(C)C 83199,N1(C(C(CCC)N(C)C)=O)CCC(NC(C2CN(C)CCN(C)C2)=O)C12CCC2 83200,CC(C)C(F)C(=O)N1CC(=C(F)CNC(=O)Cc2csc(=N)[nH]2)C1 83201,C(c1ccc(S(N)(=O)=O)cc1)=CC(=O)NC1C(CNC(CCC(N)=O)=O)CC1 83202,CC1C(=O)NC(=O)CN1C(=O)C(CN=[N+]=[N-])NC(c1ccc(C(F)F)o1)=O 83203,N1(C(C2CC(C)N2C(c2cc[nH]c2)=O)=O)CCCC12CCNC2=O 83204,c1(C(=O)NC(C)CNC(c2cc(-c3cccnc3)on2)=O)cc(Cl)ncc1F 83205,Cc1nnc(O)c(C(=O)NCC2CC3CN(C(c4ccccc4F)=O)CC23)c1C 83206,C(=O)(C1=CCCOCC1)N1CCC(NC(c2ccsc2-n2cnnn2)=O)(CF)C1 83207,Cc1ccc(O)c(C(N2CC(CC(=O)NC3CC(C(C)O)C3)C3(CC3)C2)=O)c1 83208,c1(OC)ccc(CC(=O)NC2CCC2NC(c2sc(N)nc2C)=O)cc1F 83209,C1(C)(C(N2CC(CNC(c3n(CCC)nc(C)c3)=O)(OC)C2)=O)COCC1(F)F 83210,C=CCC(C)C(=O)NCCOC1CN(C(=O)CC2COC(C)(C)C2)C1 83211,CCCC(CCC)C(=O)N1CCCCCC1C(=O)N(C)CC1CCCOC1 83212,Cc1cnc(C(C(=O)NCCC#N)N(CCCNC(C)(C)C)C)s1 83213,N1(C(=O)Cc2ccncn2)CC(NC(COCCC(C)C)=O)C(n2ccnn2)C1 83214,CC(C)CCCCN(C(=O)C(n1cc(-c2cnc(C3CC3)s2)nn1)C)C 83215,C1(C(=O)NCC(CC)(CC)NC(=O)Cc2ccc(C)c(O)c2)CC12CCSCC2 83216,C(=O)(C(C)(CCC)CCCCCC)NCC(CC=C)NC(c1ccoc1CC)=O 83217,c1(C(N2CC(C=O)NCC2)=O)cc(Cl)c(Br)cc1Cl.CCCCCCOCCC=C 83218,Nc1ccc(F)c(CNC(=O)NCCn2nccn2)c1 83219,C1(NC(=O)NCCNC(C2CC(N(C)C)C2)=O)CCc2ccccc2N1 83220,c1(C(=O)NCC(=O)NCc2cncn2C2CC2)cc2ccccn2n1 83221,N1(C(C=Cc2ccc(C)o2)=O)CC(NC(=O)CN2CC3CC3C2)CC(C)C1 83222,Cc1cccc(O)c1C(=O)NC1CC(C)CN(C(=O)Cc2c(F)cccc2F)C1 83223,C1(C)(CNC(COC(CC)C)=O)CCCN(C(c2cc(C(C)(C)C)n[nH]2)=O)C1 83224,N1(C(C(C(C)(C)C)C2CCC2)=O)CCCC(C2(NC(=O)CC3(CO)CC3)CC2)C1 83225,O=C(CCCCC1CC1)NC1CN(C(C2(c3ccc(F)cc3)CCCCC2)=O)C1 83226,N1(C(c2n(C=C)ncc2)=O)CCCC(N=c2cc[nH]c(-c3nccs3)n2)C1 83227,C(=O)(C(=O)N=S(C)(C)=O)N1CCC(C)(NC(C2C(=C)CC2)=O)C1 83228,C1(CCNC(CC2CC(C)C2)=O)CN(C(C2C=CCCC2)=O)CC1C 83229,C(=O)(C(CCO)N(C)C)N(C)CC1CCN(C(C(C)NC(COC)=O)=O)C1 83230,CC#CCCCC(=O)N1CCCC(CCNC(=O)CS(=O)(=O)NCC)CC1 83231,N1(C(c2c(C)oc(CO)c2)=O)CC2(CNC(=O)CN(C)CCO)CC(F)(C1)C2 83232,CCC(C)C(C(=O)NC1CCN(C(=O)C#CC(C)(C)O)C(C)C1)OC 83233,c1(CCCC)nnc(C(N2CC(CCNC(c3cn[nH]c3)=O)C2)=O)s1 83234,c1(C(C)NC(C2CCN(C(=O)CCCC3CC3C)C2)=O)nn(C)cc1O 83235,C1(NC(c2cnccc2Cl)=O)CN(C(=O)CCC2CCCC2)CCC1CO 83236,C1(OC)CN(C(C23CCN(CC2)CC3)=O)C(C)(CNC(=O)CCc2cnco2)C1 83237,c1(C(=O)NCc2c(CCC)n[nH]c2)cc(CC)c(C)s1.N12CCC(C1)C2=O 83238,C1(CC(=O)NCC2CN(C(=O)Nc3ccc(Cl)cc3)C3CC23)CN2CCC1CC2 83239,C12(C(=O)NCCOCCO)CCC(C(=O)NCC3(Br)CC3(F)F)(CC1)CC2 83240,C1(N(C(C2CC(SC)C2)=O)C)CCCC(NC(c2ccccc2CO)=O)C1 83241,c1(C(=O)NC2CC(N(C(=O)Cc3ccon3)C)C2)cnnn1C 83242,c1(C2C(C(=O)NCC3(CF)CCOCC3)C2)ccc(F)nc1 83243,C1(C(N2CCC(C)(CO)C2)=O)(COC)C=CCN1C(=O)CCC=CC(C)C 83244,CCCCCC(C)CC(=O)NCCCCCNC(=O)CCS(C)=O 83245,C1(CNC(CCC(N)=O)=O)(NC(C2CC(=O)N(CCF)C2)=O)CC2CCC1CC2 83246,c1(CCC)nc(CN(CC(F)F)CC)no1.C(C)O 83247,CC1CN(C(C2C3CCC2(c2cncs2)C3)=O)CC1CNC(=O)CN(C)C 83248,C1(C2CN(C(=O)COc3cccc(Cl)c3Cl)C2)(NC(c2nc(C)nn2C)=O)CC1 83249,C1(CC=C)(C(=O)N(C(C(N)=O)C2CC2)C)CCCN1C(c1ccncn1)=O 83250,c1(C(=O)NCC(C)(C2CCC2)NC(CC2C(C)C2)=O)cnn(CC(F)(F)F)n1 83251,CC1CC(C(=O)NCCN(C(=O)CCCOc2ccc(C(N)=O)cc2)C)C(=O)O1 83252,C#CC(CNC(=O)CCCC(C)NC(c1cnn(CC)c1C)=O)CC(C)(C)C 83253,c1(C2(C(N(CCCCC)C(C3CCCSC3)=O)=O)CCC2)ccc(F)cc1C 83254,C(=O)(C#CC1CCC1)N1CCC(CNC(CSc2n(C(C)(C)C)cnn2)=O)C1 83255,C(=O)(C1=NNC(C(F)(F)F)C1)N1CC(O)(CCNC(C(C(C)C)SCC)=O)C1 83256,N1(C(CCC(C)OC)=O)C2CCC1CC(N(C(=O)CCc1cc(C)no1)C)C2 83257,Cc1noc(N)c1C(=O)NCc1cc(C(=O)NCCc2ccccc2Cl)n(C)n1 83258,C1(NC(C(CC2CCC2)NC(C)=O)=O)CCSC12CN(c1nc(C)ns1)C2 83259,c1(NC(CC2(C(=C)F)CCC2)=O)cc(=O)c2cc(O)ccc2o1.C1(=O)CN1C 83260,C1(OC)CN(C(c2ccc(CO)cc2)=O)CC1NC(c1scnc1C)=O 83261,c1(C(=O)OC)ccc(C)nc1N(C)CC1CCCCN1C(=O)C1=CCCOC1 83262,N#CC1CN(C(=O)CC2CCN2C(=O)C2=CCOCC2)CCO1 83263,C(=O)(C1=NNC(=O)C1)N(CC(C)C)CC(=O)NCCC1CCCN(C)C1 83264,N1(C(C#CC(C)(C)O)=O)C2CCC1C(F)C(NC(c1cc(Cl)c([N+](=O)[O-])[nH]1)=O)C2 83265,C(C(=O)C(C)(C)C)OC1CCN(C(C)=O)C1 83266,N1(C(CC(CSC)OC)=O)CCC(C=CC(N2CC(SC)C2)=O)CC1 83267,c1(CC)cc(F)c(F)cc1NCc1cc(-c2c(F)cccc2Br)n[nH]1 83268,c1(-n2cc(CNC(c3n(C)cnc3Br)=O)nn2)cccn2ccnc12 83269,c1(C(=O)NC(C2CCN(C(C3(CC#C)CCOC3)=O)C2)C)cccc(C)c1Cl 83270,Cc1occc1C1CC1C(=O)NCC1C=CCN1C(c1c[nH]c(=N)s1)=O 83271,Cc1nc(C)c(C(N2CC3(COC(CNC(C4CN(C)C4)=O)C3)C2)=O)c(C)n1 83272,CC1CN(C(=O)CS(=O)CCNC(c2sccc2F)=O)CC1(C)CO 83273,C=CC1OCCC1C(N1CCCC(CNC(C2CCC(C(=O)OC)CC2)=O)C1)=O 83274,N1(C(C=CS(C)=O)=O)C2CCC1CN(C(c1ncn3c1CCC3)=O)C2 83275,C1(C(=O)NC2C(CCOC)CCC2)(NC(=O)Cc2n[nH]c(C)n2)CCN(C)C1 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83451,C(CCC(O)C(=O)NC1CCN(CCC)C1)NC(CC(C=C)C)=O 83452,C=CC1(CC(=O)NCCCN=[N+]=[N-])CN(C(=O)C(C)n2ccnn2)C1 83453,Cc1ccsc1C1CC1NC(C1CC(NC(=O)COc2cccnc2)C1)=O 83454,N1(C(c2ccc(C3C(C)C3)o2)=O)CCC2(C1)CN(Cc1ccc(C#N)cc1F)C2 83455,C1(CC)(NC(=O)CC2CN3CCC2CC3)CCCN(C(C2(C(=O)NC)CC2)=O)C1 83456,Cc1nc(C)n(CC(N2CC(NCC3CCC3(F)F)C(c3ccccc3)C2)=O)n1 83457,c1(OC)ncc(C(N2CCOCC2)=O)cc1-c1c[nH]nc1C(=O)NC1CC1 83458,N1(C(C(C)(C)OC)=O)CC2CCC(NC(=O)CSC)(C2)C1.c1(C)ccc(Cl)cc1 83459,Cc1cc2cc(C(=O)NC3CC(NC(=O)C=CC4C(C)C4(Cl)Cl)C3)oc2cc1C 83460,N1(C(C(CC)CC)=O)CC2CC(NC(=O)CCC3CCOCC3)C(C2)C1 83461,C(C)(CCC(=O)Nc1cnccc1CO)NC(C(C1CC1)SC)=O 83462,C#CC1CN(C(=O)CC2CCC3CC23)CCN1C(c1ccc(C)nc1O)=O 83463,c1(CC)ccc(C(C)Nc2ccnn2C(C)C)cc1 83464,Cc1nn(CC(=O)NCC(Cc2ccccc2)NC(=O)C(O)C2CC2)c(C)c1C 83465,C(CCC(=O)NCC(C)(F)CNC(=O)C(C)c1cccs1)C1C(C)C1 83466,CCCCC(O)CC(=O)NC(CC(F)F)C(=O)N(C1CCCCC1O)C 83467,C1(CC(=O)NC(C)Cc2cnc[nH]2)CCCN(C(=O)CC2CSC2)CC1 83468,CC1(C)CC(CC(=O)NCCCC(N)=O)CN1C(c1ccc[n+]([O-])c1)=O 83469,c1(C(=O)NCC2(O)CC(NC(CCc3onc(CSC)n3)=O)C2)ncccc1N 83470,C12(NCC3C(NC(=O)OC(C)(C)C)COC3)CCC(n3cc(CO)nn3)(CC1)C2 83471,CN1CCN(C(c2ncccc2Br)=O)CC1CNC(=O)CC1COC(C)(C)C1 83472,N1(C(C(C)=C2CC2)=O)CCC2CCN(C(C3(C#N)CCC3)=O)CC2C1 83473,C1(CCC(=O)OC)CCN(C(c2c[nH]cc2-c2ccccc2F)=O)CC1 83474,c1(C)cc(C(=O)NC2CC(C)(NC(C3N(CC)CCC3)=O)C2)ccc1C.C(=O)OC 83475,c1(OC)ccc(F)cc1CCC(=O)NC1(CCNC(=O)CCSC)CC1 83476,N1(C(c2c(C)sc(Cl)n2)=O)CCC2(CCCN2c2ncnn3cccc23)CC1 83477,C12(CNC(C=CCCC)=O)CCCC1CCN2C(=O)CCOc1ccccc1 83478,C1(NC(C2C(NC(Cc3n(C)cnc3)=O)COCC2)=O)CCN(C)C(=O)C1 83479,c1(C(=O)NCC2(O)CC(NC(C3C(CCC)C3)=O)C2)coc2ccc(C)cc12 83480,CCCCCC(C)(CC)C(=O)NCC1(F)CCN(C(c2ccc(C)cc2)=O)C1 83481,c1(SC)ccc(C(N2CCC(c3cn(-c4cccnc4)nn3)C2)=O)cc1C#N 83482,c1(CN(C(c2ccc(F)c(Cl)c2)C(=O)NC2(C)CC2)C)cc(F)ccc1F 83483,CCCC(C(=O)NCC1CC2CCC1N(C(=O)CCC1CCCC1)C2)S(N)(=O)=O 83484,CCC(C)C(C(C(=O)Nc1ccccc1Cl)N(C1CCC(F)CC1)C)OC 83485,C=CC(C)(CCOC)C(=O)NCC(c1ccc(C)cc1)NC(=O)C=CC1CCCC1 83486,C1(C(N2C(CNC(Cc3n(C)nc(C4CC4)n3)=O)CC2)=O)CC2CC(=O)C1O2 83487,c1(-n2c(CCC(=C=C)C)nc(C3CSC3)n2)nc2ccccc2n1C 83488,C1(CNC(C(=O)N(C)C)=O)CCN(C(=O)CC(C)(C)Cc2ccccc2)C12CC2 83489,N1(C(CN(C)C)=O)CC(NC(C2CCCN(S(=O)(=O)C(F)F)C2)=O)CC(F)C1 83490,C1(NC(c2ccc(C(F)(F)F)nc2)=O)CN(c2cc(O)ncn2)CC2(CC2)C1 83491,c1(C2(CN(C)C(=O)NCC34CCCC(CO3)C4)CCOCC2)ccc(F)cc1F 83492,N1(C(CC(C#CC)c2ccc(O)cc2)=O)CCCC2(CCCN2C(C2CC2F)=O)C1 83493,C1(O)(C(=O)NC(CNC(C(C(C)C)OCC)=O)C2CCC2)CCCCCC1 83494,Cc1cc(Cl)ccc1OCC(N1CCCOC(CNC(=O)C(C)(C)C(C)O)C1)=O 83495,C#CC(C1CCc2ccccc21)NC(=O)Nc1ccnc(CS(C)(=O)=O)n1 83496,c1(CN(C(CN(C(=O)C2=CCCC2)CC#C)=O)C)ccc(C)nc1 83497,C1(NC(CCNC(C)=O)=O)CN(C(=O)CCSC(C)C)CCC1C 83498,N1(C(C2(CC)CC2)=O)CC(NC2CC2)C2(CC2)C1.C12COC(C(=O)N)(C1)C2 83499,c1(N2CC3C(C)(C)C(C3)C2)nc2ccccc2nc1NC1CCCN(S(C)(=O)=O)C1 83500,Cn1ncc(NC2CCC3CC23)c1Br 83501,N1(C(CC(C)(C)C2CC2)=O)C2CCC(C2)C1CC(N1CCN(C2CCC2)CC1)=O 83502,C1(NC(CCSC)=O)CC(NC(c2cc(N)ccc2C(F)(F)F)=O)C12CCC2 83503,C(CC(F)F)(C(=O)NC1CCC(O)CC1)NC(=O)CC1(O)CCC1 83504,c1(COC)nn(C)c(Cl)c1C(N1CCN(C(=O)CC2CC(C)=NO2)C(C2CC2)C1)=O 83505,C1(C(F)(F)F)CN(C(c2c(CN)csn2)=O)CCN1CC1CC1 83506,C1(C(N(C(C)C)CCN(C)C(C2CCNC2=O)=O)=O)CCCC1(F)F 83507,C1(C)(NC(C(C)N(CCC)C(c2coc(C)c2)=O)=O)CC2CCC1C2 83508,c1(C(=O)NC2CCCN(C(c3nccc(CC)c3)=O)C2)coc2ccc(C)cc12 83509,c1(CCC(=O)NCCC(C)N(C)C(c2cccn2C2CC2)=O)cc(C2CC2)on1 83510,C(=O)(C(C)C(C)NC(=O)Cc1nc[nH]n1)N(CCCOC)CCO 83511,C1(C(=O)NCCCSCC)CC(NC(c2cnn[nH]2)=O)C12CCC2 83512,Cc1cc(C(N2CCCC2C(N2CCN(C)C(Cc3cnsc3)C2)=O)=O)ccc1F 83513,C1(CNC(CNC(=O)OC)=O)CC2CCC1N(C(=O)C(C)Cc1cccnc1)C2 83514,n1(C(N2CC(CCNC(C3(C(C)C)CC3)=O)(OC)C2)=O)cc([N+](=O)[O-])nc1C 83515,C1(C(=O)NC23CC2CN(C(C2CC4(C2)CC(F)C4)=O)C3)CCc2ncccc2C1 83516,C12(C(=O)NCC#CCNC(c3n(C)ncc3C(F)F)=O)CCCCC1NC(=O)C2 83517,CCC(O)C(C)(C)C(=O)N(CCCN(C)C)CCNC(=O)C(C1(CC)CCCC1)C 83518,C(=O)(CC(C(F)(F)F)C1CCOCC1)N1CC(CC(CC)O)C1 83519,n1(CC(=O)NCCOCCN(C(CCC=C(C)C)=O)C)ncn(C)c1=O 83520,CCC(CC(F)(F)F)C(=O)N(C)Cc1nc[nH]n1.C12(CC1)NC(=O)COC2 83521,c1(C(=O)NC2C(F)CCN(C(C3ON=C(C)C3)=O)C2)c(C)ccc2c1CCCN2 83522,c1(C(=O)NCc2ccc(C(F)F)c(F)c2)cc2cccc(C(F)F)c2nc1O 83523,N1(C(c2on(C)c(=O)c2)=O)CCC2CCC(C1)N2C(=O)COC1(C)CCCCC1 83524,N=c1nc(Cl)cc(C(c2nnnn2C2CCCCC2)NCCOC2CCOC2)[nH]1 83525,C1(NC(CCCNC(CC(CC)(F)F)=O)=O)CCCCC12CCC2 83526,N(C(=NCCOCC1CCCCO1)NCC1CCCCC1)Cc1ncn(C)c1 83527,c1(N(C(C2N(C(C)=O)CC2)=O)CC2CCCC2)ccc(N)cn1 83528,C(=O)(C(O)CC1CC1)NC(C)C(=O)N(C1CCCCC1)C 83529,c1(COC)cc(F)c(C(c2nnnn2C2(C)CC2)NCc2cc(C)c(C)s2)cc1Br 83530,c1(SC)cccc(C(N2CCC(CCNC(=O)CCc3cccc(O)n3)C2)=O)n1 83531,C(=O)(C#CC1CCOC1)N(C(C(=O)NC(CC#C)CC(F)F)C1CC1)C 83532,C1(CNC2(F)CC2)CCCCC1.C1C(O)CNC(=O)COCC(=O)N1 83533,CC1C(C(=O)N(C)CC2CC2)CCN1C(=O)Cc1ccccn1 83534,Cc1cc(=NCC2(NCCC(=O)Cc3ncccc3C)CCCC2)c(C#N)c[nH]1 83535,N1(C(CC(C(=C)C)O)=O)CCCc2nc(O)ccc2C1 83536,C1(C(=O)NCC=CCNC(C2CC3CCCCN3C2)=O)CCC2(CCCC2)CC1 83537,C(=O)(C1=CC=CN2CCS(=O)(=O)N=C12)NC(CNC(C1C(C(=O)OCC)C1)=O)C 83538,N1(C(c2nn(C)cc2Br)C(=O)NCC(=C)C)CC(S(C)(=O)=O)CCC1C 83539,c1(C(=O)NCC2(NC(CCc3cc(C)sc3C)=O)CCOC2)ccnc(C)c1N 83540,[N-]=[N+]=Nc1cnn(CCCC(=O)NCC2(c3cccc(Cl)n3)CCC2)c1 83541,c1(C(=O)NCC2N(C(=O)COCC3CCCO3)CC(O)C2)cc2ccccc2s1 83542,c1(C(=O)NCc2cc(C(=O)NCC(C)SC)sc2)cc2n(n1)CCC2 83543,CC(C)CC(C)CC(=O)NCC1(F)CCN(C(=O)COc2ccc(Cl)c(F)c2)C1 83544,C1(C(N2C(CCNC(C(CCCOC)C)=O)CCCC2)=O)CC1C1CCCCC1 83545,C(N=c1cc(Cl)nc(C(F)(F)F)[nH]1)C1OCCCN(C(c2cn(CC)nn2)=O)C1 83546,N1(C(c2c(COC)ncs2)=O)CCC(CNC(c2ncc(Cl)n2C)=O)C(C)C1 83547,C1(CCC)CN(C(c2ccncc2Cl)=O)CC1C(=O)NOCC(O)C(C)(C)C 83548,C1(NC(c2nn(-c3ccc(Cl)c(Cl)c3)cc2O)=O)CC2=CC3=C1CCC2(N)C3 83549,Cc1ccccc1C=CC(N1CCC(C)(CNC(C2C3CCC(=O)C23)=O)C1)=O 83550,c1(C(N(CCCOCCNC(C(C)SC)=O)C)=O)cnc2[nH]c(C)nc2c1 83551,c1(OC)cccc(C(=O)NCC(C)(C)NC(C2CCN(C)C(=O)C2)=O)c1N 83552,C(CCCN=c1[nH]c(Cl)nc2c1SCC2)NC(C(CCCC)O)=O 83553,Cn1nc(C(N2CC(c3nc(Oc4ccccc4)no3)C2)=O)ccc1=O 83554,Cc1cc(C)c(C(N2CC(NC(=O)CCCc3ccncc3)C(O)C2)=O)c(N)c1 83555,Cn1c(C(N2CCC(CCC(N3CCC(F)(CF)C3)=O)C2)=O)nnc1S 83556,c1(CNC(C(CNC(CCC=C(C)C)=O)O)=O)cccc(C#N)c1 83557,n1(CC(OC(F)(F)F)=O)cnc2c(N)ncnc12.CC(C)(CCO)n1cnnn1 83558,c1(NC(C2CC(NC(C3CC(CSC4CC4)C3)=O)C2)=O)ccccc1Br 83559,N1(C(c2cnc(SC)s2)=O)CC2CC(C1)N(C(C1CCC(C)(C)O1)=O)C2 83560,CCCCCC(O)CC(=O)NC(C)(CC)CCNC(C1CCCC(O)C1)=O 83561,N1(C(C2OCCC(C)(C)C2)=O)CC(CNC(C2CCCC2)=O)CC12CCC2 83562,C#CCC(C)(C(=O)NC(C(O)CO)C1CC1)NC(=O)C(C)C1(O)CCC1 83563,N1(C(Cc2ccc(C)o2)=O)CC(NC(c2sccc2C)=O)CCC1C 83564,c1(COC)nc(OC)c(C(=O)N(C)Cc2cn(C(CC)CC)nn2)c(Cl)n1 83565,Cc1cc(NCC2CN(C(C3(C)CCCOC3)=O)C2)ccc1[N+](=O)[O-] 83566,c1(C(N2CCC(CC(F)F)CC2)C(=O)NCCCCCC)cc(C)nnc1C 83567,Cc1ccc(C2CC2NC(C2CCC2CNC(=O)CC(C)C(C)C)=O)c(Cl)n1 83568,Cc1c(C(=O)N(CC(=O)NC(C2CCCO2)CO)C)cccc1C#N 83569,N1(C(c2c(F)ccc(C)c2)=O)CCCN(C(c2cc(Cl)cs2)=O)CC1C 83570,Cc1cnc2c(C(N3CC(CNC(=O)CC4=CCOCC4)C3)=O)cccn12 83571,C1(C(=O)NC2CCC(CN(C(C(COC)(C)O)=O)C)CC2)CC(C(N)=O)=NO1 83572,N1(C(CN2CC(C)(OC)C2)=O)C2CCC(C2)C1C(N1CC(C)C(O)C1)=O 83573,c1(C(N2CCC(NC(c3cc(Cl)c(Cl)c(Cl)c3)=O)C2)=O)cnc2cc(Cl)ccn12 83574,C12(C(N3CCCC(CC)(NC(=O)C=CCO)C3)=O)CCC(C#N)(CC1)CC2 83575,CC(CC(=O)NC1CSC1)N(C(=O)Cc1ccn(C)n1)C 83576,c1(CC)ccc(Br)cc1C(N1CCCCC1C1CCN(CCN(C)C)C1)=O 83577,C(CCCCC(=O)N1CCCC(CCCCNC(=O)C=C2CCCCC2)C1)SC 83578,O=C(N1CC(Cc2ccccc2)CO1)C1CCCCN1C(=O)CN1CC=CC1 83579,C(=O)(C(CCC)C(C)C)NCCC1CCCN(C(C(CCC)F)=O)CC1 83580,C(=O)(CC(C)(C)OCCCOC)NCCNC(CC1CCN(C(CC)CC)C1)=O 83581,C1(NC(CN(CCC)C)=O)(CC)CCCN(C(=O)C(c2cnn(C)c2)=O)C1 83582,C(=O)(C(C)(C)C(C)(F)F)N(C(C(=O)NCCCOCC=C)CC(F)F)C 83583,C(=O)(CCCCC(F)F)NC1(CNC(c2cnn(C)c(=O)c2)=O)CCCC1 83584,c1(C(=O)NC2C(NC(c3[nH]cc(C(N)=O)c3)=O)C2)ccc(Br)nc1N 83585,C1(C(=O)NCC(C)(C)NC(c2cn(C)nc2O)=O)CC(Cc2ccccc2)=NO1 83586,c1(CC(=O)NCC(CC=C)NC(=O)C(O)C=CCCC)ccc(Cl)cc1C 83587,c1(C(=O)NCC(C)NC(C2CC3CC2C3)=O)ccc(OC(F)F)cc1 83588,CC1(C)CN(C(c2ccc(O)c(O)c2)=O)CCC1NCc1ccc2ncoc2c1 83589,CC(C(=O)NC1C2CC1CN(C(c1ccnn1C1CCOCC1)=O)C2)C(C)(C)C 83590,CC1(C)CCCC(CC(N2CC(CCO)(NC(C3CCCOC3)=O)C2)=O)C1 83591,C=CCC(C)(C)CC(=O)N1C(C)C2CC1C2NC(c1cnc(O)c(Cl)c1)=O 83592,C1(CC(C)Sc2nncn2C)CCN(C(=O)CNC(=O)C=CC(C)(C)C)CC1 83593,CN1CCN(N2CCC(CN3CCN(C(C4CCCC(=O)O4)=O)CC3)C2)CC1 83594,c1(C(N(C2CCN(C(=O)Cc3c[nH]nc3O)C2)C)=O)cc2cnn(C)c2s1 83595,CC(CC(=O)NCCC1(CNC(c2ccn(C)c(=O)c2)=O)CC1)CC(F)(F)F 83596,N1(C(CC(C(C)C)O)=O)CCC2(CCCCN(C(c3cn(C)c(=O)cn3)=O)C2)C1 83597,C(C)(CNC(=O)C(C)C(C)(F)F)(CC(C)C)NC(CCOC(C(C)C)=O)=O 83598,c1(C(N2C(CNC(CC)=O)CCCC2)=O)n[nH]cc1[N+](=O)[O-] 83599,c1(CN2CC(C(=O)Nc3ccc(CC)nc3)OCC2)ccc(I)c(O)c1 83600,C=Cc1cc(C(=O)NC(C)C(C)NC(=O)CNC(c2ccccc2)=O)cc(F)c1 83601,c1(C(=O)NC(CCOC)CNC(=O)C(F)(F)CNC(C)=O)sc(C)c(C)c1C 83602,C(=O)(C1CCCc2nncn21)NCC(C)(C1CC1)NC(c1cc(C)c(Cl)s1)=O 83603,C1(NC(C(F)=CC)=O)CN(C(c2ccc(-c3cnn(C)c3)o2)=O)CC1(C)C 83604,C1(C(N2CC(CC(C)NC(c3[nH]c(C)c(C)c3C)=O)C2)=O)CC1C1CCCCC1 83605,c1(CC(=O)N(C2CCCN(C(c3c(C)ncnc3)=O)C2)C)ccc2nn[nH]c2c1 83606,CC1(C)CC(=O)N(CC(=O)NCC2CC2CNC(=O)CCC2CCC(=O)N2)C1=O 83607,N1(C(C)C)CC(C(N2CC(CN(c3ncc(C(C)(C)O)cn3)C)C2)=O)CC1=O 83608,C1(O)(C(=O)NC2C(NC(c3cc(OCC)n[nH]3)=O)CCC2)CC2(CCOCC2)C1 83609,C1(NC(Cn2c(C)ccn2)=O)CCN(C(=O)C(=O)NCC2CC2)CC(O)C1 83610,Cc1noc(C2CC2)c1C(=O)NC1CCN(C(=O)C(n2nccc2C)C)C1C1CC1 83611,CCCC(CC(C)C)C(=O)N1CCOCC(NC(c2occc2COCC)=O)C1 83612,c1(C(=O)NCCCN(C(CCCOC)=O)C2CC2)c(C)cc(C)oc1=O 83613,CC1CCN(C(c2cnc(Cl)cn2)=O)CCN1C(=O)CC1CCC=CCC1 83614,N1(C(C2N(CC)C(=O)CC2)=O)CCCC2(CCN(C(=O)CN3CCC(C)C3)C2)C1 83615,C(CC(C(C)C)NC(c1nccnc1C(N)=O)=O)NC(C(C)=C(C)C)=O 83616,CC(C)CC(CNC(=O)CC1(C)CC1)NC(c1ccc(C2CC2)o1)=O 83617,c1(OCC)ccc(-c2nc(COC)nn2-c2ccnn2C)cc1OC 83618,C(C)(N=c1ccnc(Cn2cc(C)cn2)[nH]1)C1CCCN(C(C2C(=C)C2)=O)C1 83619,CC(C)(C)CCCCNC(C1(NC(c2ccon2)=O)CCSC1)=O 83620,N1(CC(=O)N(C)CC2(O)CCN(C(c3cn(C)nc3Cl)=O)C2)CCCCCC1=O 83621,c1(NC2CCN(C(CC)C)CC2)[nH]c(=NCC(CC)C(C)(F)F)nc2sccc12 83622,c1(C(N(C2CCCC2)CC#C)=O)cc(CNC(=O)C(C)C2CCC2)no1 83623,C(=O)(C(C)C(C)(C)C)N1C(C(=O)NC(c2ccccc2O)C)CCC1C(C)C 83624,N1(C(C(C)N(C)C)=O)CC2CCC(C1)C2C(N1CCCC1c1ccccc1)=O 83625,c1(C(N(CC(CNC(C(c2cccc(C)c2)=O)=O)O)C)=O)cc2sccc2n1C 83626,Cc1cc(C(=O)NCC2C3CN(C(=O)C(F)C(C)C)CC23)c(C)cn1 83627,C(=O)(C(C)(C)CC(F)F)NC1(CF)CCN(C(c2cnn(C)c2C(C)(F)F)=O)C1 83628,C(C(N=c1nc(C2CC2)[nH]s1)C1CCC1)NC(C(C)Nc1ccccc1)=O 83629,C#CCCN=C(NCC(=O)NC1(OC)CCS(=O)(=O)C1)NC(c1cccc(F)c1)C 83630,C1(CNC(CNC(C(CC)C)=O)=O)CC2CN(C(=O)Cc3ccc(F)c(C)c3)CC12 83631,N1(C(COCC=C)=O)Cc2n[nH]cc2C1C(=O)N(C1CCCCCC1)C 83632,C(c1c(OC)cnn1-c1ccccc1)=CC(=O)NCC(CCC)OC 83633,c1(C(C(N2CCC(n3cc(COCC=C)nn3)C2)=O)(C)C)cccc(C(=O)O)c1 83634,c1(CN2CCC(O)(CCc3ccccc3)C2)noc2c1COCC2 83635,CCC(C)CC(=O)NCC(C1CC1)NC(=O)Cc1n[nH]cc1C 83636,N1(C(C2C(=C)C2C(=O)OC)=O)CCN(C(C23CCOC(C)(C2)C3)=O)C(C)C1 83637,c1(C(=O)NC(C(C)NC(c2cc(C)nc(O)c2)=O)C)ccc(N)c(C)c1C 83638,O=C(C1=CCCOC1)N1CCN(C(=O)CC2CSC2)C(C2CC2)C1 83639,c1(C(=O)OC2(C=C)CCC2)ccc(F)c(SC2CC2)c1 83640,N1(C(C(CC(=O)OC)c2ccc(Cl)cc2)=O)CCc2ccc(N=[N+]=[N-])cc2C1 83641,N1(C(c2c(CC)nn[nH]2)=O)CCC(CF)(NC(=O)CCCN(C)C)C1 83642,CC1CN(C(C2(C#N)CCCC2)=O)CCC1N(C(=O)C1=NOCC1)C 83643,N1(C(C=CCCC(C)C)=O)CCN(C(=O)Cc2ccc(Cl)c(F)c2)CC1CCO 83644,c1(NC(C23CCC(C(N4CC(O)C4)=O)(CC2)CC3)=O)cc(Cl)cc2cccnc12 83645,C(C)(c1ccc(F)cc1)=CC(=O)NCC1N(C)CCN(C(C(C(CC)O)C)=O)C1 83646,c1(C(=O)NCC2C(NC(C(c3ccccc3F)OC)=O)C2)cc(C#N)[nH]c1C 83647,N1(C(CCOCC)=O)CC(NC(c2cc(F)c(Br)c(F)c2)=O)CC2(CC2)C1 83648,C1(CCNC(C(CC)F)=O)CN(C(c2cc(Br)cn2C(C)C)=O)CCO1 83649,CC(O)C(C(=O)N1CCC(CCNC(=O)C(c2ccccc2F)O)CC1)N(C)C 83650,C1(C(N2C(COC)(CNC(C3CC4(CC4)C3)=O)CCC2)=O)CCC2(CCCC2)C1 83651,N1(C(c2c(C)c(Br)sc2)=O)CC(C)(C)CCC1(C)C 83652,CC(CC(=O)NCC=CBr)C(C)(C)NC(=O)C(C)CC#N 83653,c1(OC)cc(C(N2CC(NC(c3cc(C)no3)=O)CC2(C)C)=O)c(F)cn1 83654,C(CNC(=O)CCc1ccccc1Br)(C(C)C(C)C)NC(COC)=O 83655,N1(Cc2ccc(OC)cn2)CCOCC(CNC(=O)Nc2cnccc2C)C1 83656,N1(C(CC(=C=C)C)=O)CCC(C2CCOCC2)(CNC(=O)Cc2cn[nH]c2)C1 83657,C1(NC(c2cc(C)c(C3CC3)cc2)=O)CCCC12CN(C(=O)C(O)CF)C2 83658,Cc1nn2ccccc2c1C(=O)NCC1(C(C)NC(C2(C)CC=CCC2)=O)CC1 83659,N1(C(COCC)=O)CCC2(CCC2NC(=O)C=Cc2ccc(F)c(F)c2)CC1 83660,N1(C(CC(C=C)C)=O)CCC2(CC1)CCN(C(c1ccc(O)c(Br)c1)=O)C2 83661,c1(C(=O)NCC(CC)N(C)C(c2ccn(C)n2)=O)cccc(I)c1 83662,CC1CC(C(=O)NCCn2cccnc2=O)CN(C(=O)CCc2cccc(F)c2)C1 83663,C1(NC(c2c(C)coc2)=O)C2CCCN(C(C3CC4C=CC3C4)=O)C2C1(C)C 83664,C1(NCc2ccc(OC)c(SC)c2)C2CCCC(F)(F)C12 83665,n1(CCCC(=O)NCC2(C)CC(NC(=O)Cc3n[nH]c(=N)s3)C2)ccccc1=O 83666,c1(C(=O)NCC2(NC(c3c(C)ncnc3)=O)CCCCC2)cc([N+](=O)[O-])c[nH]1 83667,C1(C(=O)Nc2ccc(C(C)(O)CF)cc2)CC2C(C1)C2(F)F 83668,c1(N(CCC)C(C)=O)cccc(NC(=O)CC(C)CNCc2nc[nH]n2)c1 83669,c12ccc3c(c1)N(CC3)C2=O.C1(NC(C2(CC=C)CC2)=O)CCCC(SC)CC1 83670,N1(C(Cn2nnc(C)n2)=O)CCC2(CCN(C(c3cc4cnccc4[nH]3)=O)C2)C1 83671,c1(CC)cnc(CNC(=O)CN(C2CCC2)C(C2(Cl)CCC2)=O)o1 83672,Cc1cc(O)ccc1NC(C1CC1NC(=O)Nc1ccsc1)=O 83673,C1(NC(C2(C)ON=C(C)C2)=O)CC2(CCN(C(c3sc(C)nc3C)=O)C2)C1 83674,N1(C(c2c(C)ccc(OC)c2)=O)CCCCC(CNC(=O)C(F)=CC2CC2)CC1 83675,C1(C(N(C)C)=O)CCCC(NC(=O)CC(=O)NCc2ccnc(O)c2)CC1 83676,C12(CCCCC1)C(=O)N2.C1(O)(CC#C)CC(C(=O)N(C2CC2)CC2(C)CC2(C)C)C1 83677,CCC(CC)C(C)C(=O)NCCC(O)CNC(=O)CCCc1ccccc1 83678,C1(C(=O)NC(COC)C2CC2)CCCN(C(=O)C(c2ccccc2)=O)C1 83679,C12(CC(=O)NCCC#N)CCCC1(F)CN(Cc1coc(-c3ccccn3)n1)C2 83680,Cc1cc(C(N2CCC(CNC(=O)CN(C3CCCC3)C)CC2C)=O)nnc1O 83681,C1(C(N2CCC(n3ccnn3)C2)=O)CCCN(CC2CC23CC3(F)F)C1 83682,C=CC1(CC(=O)NCC2(C3CC3)CCCO2)CN(C(C2CCC(C)(C)C2)=O)C1 83683,N1(C(C=CSC)=O)CCn2nc(C)c(CNC(=O)C(C)C(C)CC)c2C1 83684,c1(-c2c(C(N3CC(CNC(=O)CC4COC(=O)C4)C3)=O)cno2)ccccc1F 83685,c1(NCC(C)NC(C(C)OCC(C)C)=O)nc(Cl)nc2[nH]c(O)nc12 83686,C12(C(N(CCCCCC)CC(F)F)=O)CC1CN(C(=O)C(n1ccc(C)n1)C)C2 83687,Cn1cc(C(=O)NC2CCCC(CC(N3CCCC(CF)C3)=O)C2)ncc1=O 83688,c1(C(=O)NCC=CC=CC(=O)NC2(CCCC)CCC2)cccc(F)c1O 83689,C1(CC=C)(NC(c2cccnc2CO)=O)CCCN(C(=O)CC(C)C=C)C1 83690,N1(C(CCc2cnc(C)s2)=O)CC(NC(=O)C(C)(C)C(C)(C)C)CC2(CC2)C1 83691,c1(C(C(=O)N(CCNC(CCOC)=O)CC2CC2)O)cnn(C)c1 83692,C1(C2(NC(C3CCN(C(C)=O)C3)=O)CC2)CCCCN1C(c1ccsc1C)=O 83693,C1(NC(C2CC(O)(CNC(c3c(CC)nccn3)=O)C2)=O)CC(C)(C)C12CC2 83694,c1(CNC(C2CCCC(F)C2)=O)ccc(C(=O)NCC2CC(F)C2)nc1 83695,N1(C(CCC2CCN(C)C2)=O)CCC2(CCN(C(C3CC4CC4C3)=O)CC2)C1 83696,c1(-n2ncc(NC(C3(CCl)CN(C(=O)C#CC4CC4)C3)=O)n2)ccc(Br)cc1 83697,n1(CC(N2CCC(NC(C3(OC)CCOC3)=O)C2)=O)nc(C)n(C)c1=O 83698,N1(C(c2c(C)cc(F)cn2)=O)CCC2(C1)CN(C(=O)C(C(C)O)N(C)C)C2 83699,C1(C(=O)NCCN(C(CC=CC)=O)CCC)COC2(CCC2)CO1 83700,C(N=c1[nH]c(NCc2cc(Br)cc(Br)c2O)nc(=N)[nH]1)c1c(C)[nH]nc1O 83701,N1(CC(=O)NC(CN(C)C(N)=O)(C)C)CCC(F)CC1.C12CCCN(C1)C2=O 83702,C1(CC)CCN2C1C2=O.c1(NC(=O)CCCSC)cnn(CCF)c1OC 83703,N1(C(C2(CC=C)CN(C(=O)C(C)CC3CCC3)C2)=O)CC2CC=CCC2C1 83704,N1(C(c2ccc(C)o2)=O)CCC2(CC1)CC2(C)C(=O)Nc1cccnc1 83705,Cc1nc2ccc(C(N3CC4CN(Cc5nccnc5Cl)C4C3)=O)cc2o1 83706,c1(OC)ccc(OC)c(CC(=O)NC(C2CCN(C(c3cnc[nH]3)=O)CC2)C)c1 83707,c1(C(N2CC3CCC(C2)N3C(=O)Cc2ccnc(O)c2)=O)cccc2nsnc12 83708,c1(C(N2CCCC(COC)C2)=O)ccc(Cl)cc1N.c12cn(cn1)CCNC2=O 83709,CCCC(C(=O)OC)C(=O)NCC(=O)Oc1ccc(NC(=O)CCC(C)=O)cc1 83710,CCCCC(O)CCC(=O)N1CCC(CCNC(=O)CC2CC(CC)C2)C1 83711,C1(C(=O)NCC(c2cccc(C)c2)NC(=O)C(Cl)=CCl)CCn2cncc2C1 83712,C1(C(=O)NC(C#CC#C)(C)C)CC(C)CCN1C(C1OCCC1C)=O 83713,Cc1nc(C)c(C(=O)NC(C)CCCNC(c2ccc(SC(F)(F)F)s2)=O)[nH]1 83714,c12ccc(cc1)C(C)NC(=O)CC2.C1(N(C(=O)C(F)F)CC)CCC(CO)CC1 83715,C(=O)(C(C)CC(N)=O)NCC(C)CN(C(=O)CC1CC(=O)C1)C 83716,c1(C(N(CCCNC(CC(=C=C)C)=O)C2CC2)=O)c(OCC)cnnc1OC 83717,CC(CC(=O)NC(C1CCN(C(=O)CCCC(=O)N(C)C)CC1)CO)C(F)F 83718,N1(C(CC=C)=O)CCC2(CCCN2C(=O)C(CCOC)N(S(C)(=O)=O)C)C1 83719,CC1C(NC(c2nnc(O)nc2O)=O)C(C)CCN1C(=O)C=CC1CCCC1 83720,c1(OCC)ccc(NC(c2sc(Br)cc2Cl)c2nnnn2C(C)(C)C)cc1Br 83721,c1(C(N2C(C)(COC)CC(NC(=O)COC(C)C)C2)=O)n[nH]c2cc(Cl)ccc12 83722,CC1CC(CO)CN(C(=O)CCCCCNC(c2coc(C(N)=O)c2)=O)C1 83723,Cn1cc2c(n1)CCC(CNC(=O)NC(c1cc3ccc(Br)cc3o1)C1CC1)C2 83724,C=C(CCNC(=NCc1nccc(C(F)F)n1)NC1CC1C)C(=O)OC 83725,C1(C(N2CCCC2C(C)NC(=O)CCCNS(C)(=O)=O)=O)(OCC)CCCC1 83726,N1(C(C(CC=C)C)=O)CCC(CO)(NC(C2CC3(CCC3)C2)=O)CC1 83727,C(=O)(CCCCC(=O)NC1CC(CNC(=O)C=C(CCC)CCC)C1)NC 83728,N1(C(C(N2C(=O)CCC2=O)CC)=O)CCOC(CNC(C2(O)CCC2)=O)C1 83729,C1(C(N2CC3CC3(CO)C2)=O)(NC(CN(CCOC)C)=O)CCN(C)C1 83730,c1(C(N(CCC(C)NC(C2C3COCC23)=O)C)=O)sccc1F 83731,c1(C(=O)NC2(C)CCCN(C(COCC(=O)OC)=O)C2)c(F)ccc(F)c1OC 83732,c1(C2(C(N(CCC(C)NC(=O)CC3(CO)CC3)C)=O)CC2)ccc(F)c(F)c1 83733,Cc1cccc(CN(C(=O)C(F)(F)c2ccncc2)C)c1 83734,c1(C(C)=O)c(CCC(=O)NCCCCN(C(=O)CCN2CCC2)C)c[nH]c1C 83735,C(=O)(C(C)(C)CCC)N1CC(C#C)(C(=O)NC2CCCC2C#N)C1 83736,CN1CCCC(CCC(=O)N2CC(CNC(C3(CO)CCCC3)=O)C2)C1 83737,C1(C(=O)NC2CC(C)(C(=O)OC)C2)(NC(C2CC(=O)N(C)C2)=O)CCN(C)C1 83738,N1(CC(=O)NCCC)CCCC(C2CCN(C(=O)CC3=CCN(C)CC3)CC2)C1 83739,CCC(C)(C#N)C(=O)N(C)CCOCCNC(=O)CC(c1ccc(SC)cc1)C 83740,c1(-c2nc(CC(CC)C)nn2-c2c(C)ncnc2C)cc2c[nH]cnc-2n1 83741,C(=O)(CC1CCCc2oc(C)nc21)NCC1(OC)CN(C(COCC#C)=O)C1 83742,C1(CNC(CCOCC#C)=O)(COC)CN(C(C2CCCOC2)=O)C1 83743,C1(NC(C2CCCC(OC)C2)=O)CCN(C(=O)CC2=CCCCC2)CC12CCC2 83744,c1(C(N2CCC(CNC(C34CC(c5ccccc5)C3C4)=O)C2)=O)cccc(O)n1 83745,c1(NC23C(CN(C(c4cnc(CC)s4)=O)C2)CCC3)nc(Cl)nc2cnn(C)c12 83746,C1(C(=O)NC2(C)CCN(C(CNC(C)=O)=O)C2)CC(c2cn(C)nc2C)=NO1 83747,C(=O)(CCCS(C)(=O)=O)N(CC(CNC(c1c(C)c(C(N)=O)ccc1)=O)O)C 83748,C1(NC(C(C(C)C)SCCCC)=O)CCCCCN(C(c2nnc(C)s2)=O)C1 83749,c1(C(=O)NCC2CC2OC(C)(C)C)cn(C)nc1C(N1CC(OC)(CO)C1)=O 83750,Cc1ccc(C(=O)NC(CCN(C(=O)CC2(CO)CC2)C)C(C)(C)C)c(C)n1 83751,c1(-c2c(C)noc2)ccc2c(C(N3CCCC(C)CC3)=O)cnn2c1 83752,C1(CCSC)COCCN1C(c1nscc1Br)C(=O)NC1CCOC1=O 83753,N1(C(C=NOC)=O)CCC(O)(CCNC(c2ccc(CO)cn2)=O)CC1 83754,C1(C)(CNC(CC(C=C)C)=O)CN(C(C2CC(S(C)(=O)=O)C2)=O)CCO1 83755,c1(C(=O)NCC(C)N(C(C2C(C(F)F)C2(C)C)=O)CC)cccc2[nH]nc(O)c12 83756,C1(OC)CN(C)C(C)(C(N2CC(CO)(NC(=O)CC(C)(F)F)C2)=O)C1 83757,C1(CC(=O)NC(C=CC(=O)N(C(CC)C(N)=O)CC)(C)C)CCCOCC1 83758,Cc1cc(O)c(C(=O)NC2(CO)CCCN(C(c3c[nH]c(Br)c3)=O)C2)nn1 83759,c1(OC)ccc(C(O)CNC(c2ccnc(-n3ccnc3)c2)=O)cc1OC 83760,C#Cc1cccc(NC(C2CCN(C(=O)CCC(=O)OC(C)(C)C)C2)=O)c1 83761,N1(C(CSC(C)(C)C)=O)CCC2(CNC(c3ccnc(F)c3N)=O)CCCCC12 83762,C(CCN=c1ccn2c(Br)cnc2[nH]1)N(C)CCN(C(=O)C=CC1CCCC1)C 83763,C1(NC(c2ccc(CCC)s2)=O)CCC(F)(CNC(c2ccc[n+]([O-])c2)=O)C1 83764,C12(NC(C#CC3(CC)CC3)=O)CCC(CN(C(C3CCCN(C(N)=O)C3)=O)C1)C2 83765,CC(O)(CC(=O)NCC1CC2CN(C(=O)CCc3nc(O)n[nH]3)CC12)C(F)(F)F 83766,c1(C(N(C2CCCN(C(c3cc(CO)[nH]n3)=O)C2)CC)=O)nccc2[nH]ccc12 83767,C1(NC(C(C)=C2CCCC2)=O)CCCCC1CNC(c1cnc(S)[nH]1)=O 83768,c1(OC)ccc2c(CC(=O)OCC3CC34CCSCC4)c[nH]c2c1 83769,C1(C(=O)NCC(C(C)C)NC(=O)C(O)C(C)(C)C)CCC(F)(F)CC1 83770,c1(C(N2CC(C)C(NC(=O)CC3CCCCC3O)C2)=O)cc(F)cc2cnccc12 83771,c1(CC(N2CC3CC2CN3Cc2c[nH]c3ncccc23)=O)cccc2c1OCC2 83772,C1(CNC(Cc2ccc(OC)nc2)=O)CC(C)CCN1C(c1c(Cl)cnn1C)=O 83773,N1(C(COCC)=O)CC(NC(=O)Cn2cc(CCN(C)C)nn2)CC(F)(F)C1 83774,C12(NC(=O)Cc3ccon3)CCCCC1CN(C(=O)Cc1ccc(F)c(F)c1)C2 83775,C=CCCC(C(=O)NCC1CN(C2CC2)C1)NC(C1CC12CCOCC2)=O 83776,CCCCC(C)(F)C(=O)N1CCC2CN(S(=O)(=O)CC3(COC)CC3)CC12 83777,N1(C(C(C)N)=O)CCC(C(=O)N)C(C)(C)C1.C(C)(C)(C)C(=O)C(=O)C1CC1 83778,C1(CC)(OC)CCCN(C(C2(C3(c4ccccc4)NC(=O)NC3=O)CC2)=O)C1 83779,c1(C(=O)NCC23C(CN(C(COCC(=O)NC)=O)C2)C3)n[nH]c(CC)c1[N+](=O)[O-] 83780,c1(C(N(CC(=O)OC)CC#C)=O)n[nH]cc1CNC(=O)C(F)C1CCOC1 83781,N1(C(c2cc3ccccc3cn2)C(=O)NC(CC)C)CCN2CCN(C)CC2C1 83782,C12CC3CC(C1)N(C3)C(=O)c1cncc(c1)C(=O)NC2.C12CC(F)(C1)C2.CCN 83783,N1(C(C2C(NC(C3C(C(=O)OC)C=C3)=O)CCO2)=O)CCN(C)CC1C 83784,N(C(=NCCCC(=O)N1CC=CC1)NCC12CCCC(C)(CO1)C2)CC(C)(C)C 83785,c1(C(=O)NC(CNC(c2ccc(=N)[nH]c2)=O)C2CC2)ccc2cnnn2c1 83786,C(=O)(CC(C)NC(C1CC=CCC1)=O)NCC(CNC(=O)C(=O)N(C)C)OC 83787,Cc1nn(Cc2nc(C3CC3)n(-c3ccccc3OC(C)C)n2)c2ncccc12 83788,N1(CC(=O)NCc2c(Cn3cc(C(CCC)N(C)C)nn3)nco2)CCCCCC1 83789,c1(C(CNC(c2n(C(CC)(C)C)nnn2)c2cc(C)co2)(C)C)cc(C)cc(C)c1 83790,Cc1cc(NC(C2(NC(=O)CSC(C)C)CCCCC2)=O)ccc1O 83791,C1(CC)(CC)CN(C(C23CC(C(F)(F)F)(C2)C3)=O)CC(C)O1 83792,C(C(=O)N1CC(NC(c2cc(O)n(C)n2)=O)CC1(C)C)(C(C)(C)C)NC(C)=O 83793,C(C)(C)(CCCC(=O)N1CCOC(C(N)=O)C1)NC(C1(C)CCN(C)C1)=O 83794,N1(C(CC2C(C)CCC2)=O)CCC(C(C)(C)NC(C2(n3cc(Cl)cn3)CC2)=O)CC1 83795,CCC(CC)CCC(=O)N(CN(C(C)C(=O)Nc1ccc(F)cc1OC)C)CC 83796,Cc1ccc(C(=O)NCC2CCCC2NC(=O)CSc2cccc(F)c2)cc1Cl 83797,N1(C(C(CSC)OC)=O)CCC2(CC1)CC(CNC(C1CC3CC3C1)=O)C2 83798,N1(C(c2c(C)c[nH]c2)=O)CCc2cc(C(=O)NCC(N)=O)cnc2C1 83799,C1(CC)(CC)CCCC1O.N12CC(CO)(C1)CC2=O.C(=O)(CC(=O)O)NC1CCC1 83800,N1(C(C#CC2(C)COC2)=O)CCC2CCN(C(=O)CCc3ncc(F)cn3)C2C1 83801,N1(C(C)C)CCCC(CCNC(C2CCCCN2C(=O)COC(C)(C)C)=O)C1 83802,c1(SC)nc(CCCCO)c(-c2nc(C)no2)s1 83803,CC(C(=O)N1CCCN(CCC2CN(C(=O)Cn3nccn3)C2)CC1)C(C)(C)C 83804,C=CC(C)(C)CC(=O)NCCCN(C(C1CC(O)CN1c1ccncn1)=O)CC 83805,C(=O)(CCCN(C)N=O)NCCCCNC(C1CC(C)SC1)=O 83806,c1(C(N2C3CN(C(C(COC)OC)=O)C(C3)C2)=O)oc2ccccc2c1C 83807,C1(C(N(C2(C(=O)NCc3nccc(C)c3)CC2)C)=O)C2CCC(C2)C1C 83808,C(C)(CNC(C1(c2ccno2)CC1)=O)(C(C)C)NC(c1c(SC)ccs1)=O 83809,N1(C(COc2ccc(CC)cc2)=O)CCC2CC2(NC(=O)CC(C)C(C)C)CC1 83810,CC1=CCC=CC1C(N1CC2C(NC(=O)CC(C)O)C2C1)=O 83811,S(=O)(=O)(C1(C(c2cccc(OCc3ccc(F)cc3)c2)Nc2ncoc2Cl)CC1)NC 83812,N1(C(C(C)CC2CCCO2)=O)CCC(CN(C)C(C2(n3cccn3)CC2)=O)CC1 83813,C12CC3CCC(C1)N3C2.C1(C(=O)NCC(=C)C)CCN(CCc2ccccc2)CC1 83814,N1(c2nc(OC)c(F)c(C)n2)CCCC2(CCN(C(=O)C(C)(C)SC)C2)C1 83815,C1(C(NOCCCCCC)=O)CCCN(C(=O)Cc2cnccc2C)C1 83816,N1(C(c2cccc(C#C)c2)=O)CCCCCCC1C(=O)NCC1CCC(C)C1 83817,C(=O)(C(C)(C)C(N)=O)N(CCC(C)NC(c1cnn(C(C)C)n1)=O)C 83818,N1(C(=O)OC(C)(C)C)CCC2(C1)C1CN(C1)C(=O)N2.N1(CC(=O)O)CCNC1=O 83819,n1(C(C)C)cnc(C(=O)N(C2CCC(NC(=O)CC3(N(C)C)CCCC3)C2)C)c1 83820,C=CCC(CC(C)C)C(=O)N1CC(C2CC2)C1Cn1cc(CNS(N)(=O)=O)nn1 83821,c1(OC)ccc(C(N2CCCC(NC(c3cccnc3OC)=O)C2)=O)cc1F 83822,C1(CNC(=O)OCC)CCN(N2CCOC(Cc3ccc(F)cc3)C2)CC1 83823,CN1CC(C(=O)NCCCN(C(C2CCCS2)=O)CC2CCCC2)CC1=O 83824,c1(C(=O)NC2CC(CNC(CN(C)C)=O)C2)cc(F)cc2nc(S)[nH]c12 83825,c1(C(N2C(CNC(CCC=CCC=C)=O)COCC2)=O)cc(F)cc(C)c1N 83826,C(C)(C)(C#Cc1cn(-c2ccncc2)nn1)NC(c1c(C)ccc([N+](=O)[O-])c1)=O 83827,CCCC(CNC(=O)CC1(C)CCOC1)C(=O)N1CCCC(OCC)C1C 83828,C(=O)(CCC(C)(C)[N+](=O)[O-])NCCN(C(C(C)N1CCCC1)=O)C1CC1 83829,C(=O)(CCCCC(=O)NCC(O)CN(C(=O)C(O)C1=CCCCC1)C)OC 83830,CN1CCC(=CC(N2CC3C(CC(=O)NCCc4ccsc4)C3C2)=O)CC1 83831,Cc1csc2ncc(C(=O)NC3CN(C(=O)CSCCC(F)(F)F)CCC3F)n12 83832,c1(C(=O)NC2(C(=O)NC(C(C)OC)C)CC2)ccc(CC(=O)C2CC2)nc1 83833,C(CC(O)C(=O)N)NC(CCN(C(C=CC)=O)CCO)=O 83834,c1(CCC(=O)N(C)CC2(O)CN(C(CNC(C3C(C)C3)=O)=O)C2)ccc(Cl)cc1 83835,C(=O)(CC(C)COC)NCC(CC)NC(c1cccc(CN2CCCCC2)c1)=O 83836,C(CN=c1[nH]c(N2CCCC(C(C)C)CC2)nc2cccnc12)=CC 83837,N1(C(C2CC2C(F)F)=O)CC2CCC(C1)N2C(c1cc(-c2ccns2)on1)=O 83838,c1(C(N2CCCC2c2cccc(Cl)c2)=O)cc(Cl)c(F)cc1[N+](=O)[O-] 83839,c1(CC(=O)NC2CCN(C(c3c(C)ncnc3)=O)C2)cnn2c1OCCC2 83840,N1(C(C2CCCC(CC)C2)=O)CC2=C(C1)CN(C(c1cc(F)cc(Cl)c1)=O)C2 83841,c1(OC(C(=O)NCCN(C(=O)C(O)C(C)C)CC)C)cccc(C(N)=O)c1 83842,CC(C(F)(F)C(F)(F)Br)Oc1ccc(OC(=O)CCCc2ccccc2)cc1 83843,C(=O)(C(CN(C)C)NC(=O)Cc1cnoc1)NCC(C)CN(C)C 83844,N1(C(CN(C(COC)=O)C)=O)CCN(C(=O)CCCCCSC)CC1CC(F)F 83845,c1(CCC)cc(C(=O)NC2CCN(C(=O)C(O)CC3CC3)C2C2CC2)c(C)o1 83846,c1(CNC(=O)CC2CC(NCc3ccnc(O)c3)C2)cccc2c1CCC2 83847,C(CC(CNC(C1(C)CC(F)C1)=O)NC(=O)C(C)OCC1CC1)OC 83848,c1(C(N2CC3CC(NC(COC4(C)CCC4)=O)C3C2)=O)ccc2ncsc2c1 83849,N1(C(C2N(CC)CCOC2)=O)CCC2OCCN(C(=O)CC(C)(C)OC)C2C1 83850,C1(C(N(CCN(C)C)CCO)=O)CSCCN1C(c1ccc(CO)s1)=O 83851,C12(CC)CCCC(CN1CC=Cc1cn(C3CC3)nn1)C2.C1(F)(C=O)CC1 83852,C1(C(=O)NC2CN(C(c3cc(SC)oc3C)=O)CC2C)(OC)CCOCC1 83853,S(=O)(=O)(c1cccc(C(=O)O)c1)N1C(C2CCN(C(C(=C)F)=O)CC2)CCC1 83854,c1(C(=O)NC2CCN(C(c3[nH]cc(CC)c3)=O)C2C)ccc(OC)c(C(F)F)c1 83855,c1(CC(=O)NC)cc(F)ccc1C(=O)NOCC(CNC(C(C1CC1)OCC)=O)CO 83856,C1(C(=O)NCCNC(CC2CCCN(C)C2)=O)CCCN2CCCCC12 83857,CC(C)CCCCC(=O)NC1(C)CC(NC(c2cnn(CC3CC3)c2)=O)C1 83858,c12c(nnn1C)NC(=O)C(C)N(CC)C2=O.C(CC(C(=O)OC)OC)N 83859,C(=O)(CC(CC(C)C)NC(=O)Cn1cc(C2CC2)nn1)Nc1onc(C)n1 83860,C1(N(C)CC)CCCCC1NC(=O)NC1CCCN(C(=O)N(C)C)C1 83861,N1(C(CN2CCN(C(C=CC(CC)C)=O)CC2)=O)CC2CCCCC2C1C 83862,C(C)(CNC(c1c[nH]nc1C(F)F)=O)(C(C)C)NC(C(CO)OC)=O 83863,C1(OC)CCC(C(=O)NC2C3CC2N(C(C2(C)CC=CCC2)=O)C3)CC1 83864,c1(NCc2c(OC)ncc(F)c2)cnc2ccc(F)cc2c1 83865,N(C(=NCCF)N(C)Cc1noc(-c2cccc(Cl)c2)n1)C1C(C)CCC1 83866,C1(C(=O)NCC(C(C)C)NC(c2cccc(C(N)=O)n2)=O)CCCCC1(F)F 83867,c1(OC)c(C(=O)NC2CCC(CNC(C3(C)CCOC(C)C3)=O)C2)c(C)nn1C 83868,C1(O)(CC)CCCN(C(C2CC3C=CC2C3)=O)C1 83869,CCC(COC1CCOC1)(CC)C(=O)N1CCC(C(=O)NC2CC2)O1 83870,N1(C(c2c[nH]c(=NC)s2)=O)CCC2(CC1)CC2C(N1CCOC(C(C)(C)C)C1)=O 83871,c1(C(=O)NC2(CNC(=O)C(O)C3CCC3)CCOC2)cc2ccccc2cn1 83872,Cc1c(C(N2CCC(C(C)NC(c3cnc(N(C)C)nc3)=O)CC2)=O)nnn1C 83873,C1(COC)(NC(C2(n3cccn3)CC2)=O)CCN(C(=O)CCn2cncn2)C1 83874,C1(C(=O)NCC(CNC(c2cc(C)ns2)=O)CO)CCC(=O)NC1 83875,C(=O)(C(C)(C)C(N)=O)N1CCN(CCCN(c2cnc(O)c(F)c2)C(C)=O)CC1 83876,N1(C(C(=O)NCC2(OC)CN(C(C3CC3[N+](=O)[O-])=O)C2)C)CCCC(O)C1 83877,CC(=O)CC(C)(C)C(=O)NC1C=CC(C(N2CCC23CCCCC3)=O)C1 83878,C1(C(N(CCCC=C)CC)=O)CCC(C2CC2)N1C(=O)C=Cc1cc[nH]n1 83879,c1(C(=O)NCC2CCCC2C(N2CC(c3nncs3)C2)=O)ccncc1F 83880,c1(C(=O)NC2(COC)CCN(C(=O)CC3CCOCC3)C2)cnc2n1CCCC2 83881,C(CO)(CCCCNC(=O)CCc1cscn1)NC(c1nc(CC(C)C)sc1)=O 83882,c1(C(=O)NCCCNC(CC2COCC(C)O2)=O)cccc(F)c1F 83883,C(CCCCNC(=O)CCCF)NC(C(C)c1cccs1)=O 83884,C1(N(C(=O)COC2CC2)C)CCCCN(C(=O)C(C)(C)n2cccn2)C1 83885,C(=O)(C1=CCOCC1)NC(C1(O)CCN(C(C2SCCS2)=O)C1)C 83886,n1(Cc2ccc(NC(=O)NCC(n3ccc(C(F)(F)F)n3)C)o2)ccccc1=O 83887,c1(CNC(CCOCCC)=O)ocnc1C(=O)NCC1CCN(CCF)C1 83888,Cc1ccc(C(N2CCCOC(CNC(=O)C(CO)N(C)C)C2)=O)c2c1CCC2 83889,N1(C(C(C2CCN(C(C(=O)NCC(CC)C)=O)CC2)C)=O)CCN(C)CC1 83890,c1(NC(C(C(C)C)SC)=O)ccc(NC(=O)C(C2CCCC2)OC)cc1C 83891,C(=O)(C(C(C)(C)C)c1ccccc1)NCCCNC(C(c1ccc(F)cc1)C)=O 83892,CC1CN(C(c2ccc(-c3ccc(O)cc3)cc2)=O)CCN1C(C1CC1F)=O 83893,CCCC(C)C(=O)NC1CCCN(C(C2(C#N)CCC2)=O)C1 83894,Cc1cc(F)c(C(=O)NCC(C)CNC(c2csc(C(N)=O)n2)=O)cc1Br 83895,CCC(CNC(=O)C(c1cncnc1)C)(CC)C(=O)NCC(O)C1CC1 83896,Cc1scc(C(N2CCC(C)(CC(=O)NCc3cnns3)C2)=O)c1C 83897,CC1(C)COC(CCC(=O)NCCCOCCCNC(=O)CCn2cncn2)C1 83898,c1(OC)cc(F)cc2[nH]c(C(=O)NC(C)(C)CCNC(=O)C3=CCCC3C)cc12 83899,Cc1cc2[nH]c(C(=O)NC(CNC(C34CCN(C3)S(=O)(=O)C4)=O)C(C)C)cc2o1 83900,C(CC(C(=O)N(C)Cc1nnnn1C)NC(C1CC(OC)C1)=O)OC 83901,C12(NC(=O)Cc3ccc(F)cc3Cl)CCCC1N(Cc1cccc(Cl)c1Cl)CC2 83902,N#Cc1ccc(CC(=O)NC2CCC(NC(c3cc(C#N)c[nH]3)=O)C2)cc1 83903,CC(O)C(CC(=O)NC1CCN(c2ccncc2)C1)c1ccccc1 83904,Cc1cc(C(=O)NCC2(F)CN(C(=O)CCCCC(C)(C)C)C2)cc2c1CCC2 83905,C1(CC(=O)NCC(C)N(C)C)CCCCN1C(C1CCCCO1)=O 83906,C1(NC(C=C(CC)C)=O)C2CC3CN(C(c4ccc(F)c(Br)c4)=O)C1C3C2 83907,c1(C(=O)NCC#CCNC(=O)CC2CCC(O)C2)cn2ccc(F)cc2n1 83908,C(CSC1CC1)(CC1CC1)OCC 83909,C12(C)CN(CCO1)CC(=O)N2.c1(C(C)C(F)(F)F)cccc(-c2nn[nH]n2)c1 83910,c1(C(CC)C(=O)N(C)CCN(C)C(C2CNC(=O)C2)=O)cccc(Cl)c1 83911,c1(C(=O)NCCN(CCC)C(C2C3COCC23)=O)cc(C2CCCCC2)nn1C 83912,C=C(CNC(C)=O)CCNC(=O)CC1(C(=O)OC)CC1.c1(CC(=O)N)ccon1 83913,C(=O)(C1=CC(C)(C)C1)NCC(CNC(c1ccc(N(C)C)cc1)=O)(C)F 83914,c1(C(N2CC(CNC(C(C)N(CC)CC)=O)C(O)C2)=O)cccc2ccoc12 83915,C1(C(=O)NCc2ncccc2C)(CC)CCCN(C(c2cnn(C3CC3)c2)=O)C1 83916,N1(C(c2csc(C)c2C)C(=O)NC2CC(SC)C2)CCC(F)(F)C(C)C1.C(C)(C)C 83917,c1(N(CCNC(c2ccc3ocnc3c2)=O)CC)nc(O)c2ccc(Cl)cc2n1 83918,c1(NC(C)=O)cnccc1C(=O)NC(C)CNC(c1csc(C(C)C)n1)=O 83919,CN1CCC(C(=O)OCC2(CF)CC3(CCC3)C2)CC1=O 83920,C1(CNC(=O)CCOc2ccccc2)CC2(CC(NC(c3c[nH]c(Br)c3)=O)C2)C1 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83973,c1(C(=O)NCCC2CCCN(C(C3C(CC)OCCC3)=O)C2)cc2occc2s1 83974,Cc1cc(C(=O)N(C2CN(C(=O)C(C(C)C)N(C)C)CCC2C)C)nc(C)c1 83975,CCCCCS(=O)(=O)CC(=O)N1CC2CCN(C(=O)Cc3ccccc3)CC2C1 83976,Cc1cc(=NCCCCNC(c2cc([N+](=O)[O-])c[nH]2)=O)[nH]c(Cl)n1 83977,c1(CN2CC(CN(c3nc(C)cc(C)n3)C)C2)ccc2c(cnn2C)c1 83978,N1(C(CC(CCC)C)=O)CCOC2(CCS(=O)(=NC(=O)CCCC(C)C)CC2)C1 83979,c1(C(=O)OC)cccc(NC(=O)Cc2coc(C)n2)c1O.C12CC1NC2=O 83980,C1(NC(Cc2cc(C)on2)=O)C2CCC1N(C(=O)COCc1nccn1C)C2 83981,c1(C(=O)NCC2(CNC(C(C)Cn3cccn3)=O)CC2)cccc2oc(O)nc12 83982,C(=O)(C(C(C)(C)C)OC)N1CC(NC(CC(CC)SC)=O)(CO)C1 83983,C(=O)(C#CC1(C)COC1)N1C(C)CCC(C(=O)NCC2CN(C)C2)C1 83984,CC(CC(=O)NCC1CC1C(=O)NC(C)(C)C(C)(C)C)CC(C)(C)C 83985,c1(C(C)C)cccc(CC(N2CC(C)(NC(=O)CSCC3CC(F)(F)C3)C2)=O)c1 83986,N1(C(CN(C(c2cccc(C)c2N)=O)C2CC2)=O)CC(C)C(O)C(C)C1 83987,Cn1cnc(C=CC(=O)NC2CCCC2NC(C2(N(C)C)CCC2)=O)c1 83988,C(=O)(CCC(=O)NN(C)C)NC(CSCC)C(=O)N(C)CCn1ccnc1C 83989,Cn1c(N)c(CN2CCC(C3CCCC4(CCC4)O3)CC2)c(O)nc1=O 83990,C1(n2cc(CCOC)nn2)CC2CCC1(NC(=O)C(F)C(C)(C)O)C2 83991,c1(CC(N2CC(CNC(CCCOC(C)=O)=O)C2)=O)ccc2c[nH]nc2c1 83992,C(C)(CO)(C(=O)N1CC2C(CNC(C3(c4cccc(F)c4)CC3)=O)C2C1)OC 83993,C(=O)(C(C)(C)C(C)C)NC(CC)CN(C)C(C1CCN1C1CCCC1)=O 83994,CCC(F)(F)CC(=O)NCC1CC(C)CCN1C(=O)CC(c1ccc(F)cc1)C 83995,N1(C(c2c(F)cccc2Cl)=O)CCCC12CCC(NC(C1(C(F)F)CC1)=O)CC2 83996,c1(CC)ccc(C(=O)NC2CCC(CNC(c3cc(C(N)=O)cs3)=O)C2)s1 83997,c1(C(=O)NC2(C)CC(C(N(CC(COC)(F)F)C)=O)C2)ncccc1O 83998,N1(CC(=O)NC(COCC)C(=O)N(C)CCC2CCCN2C)CCC(=O)CC1 83999,c1(C(=O)NCC2C(CNC(c3c(OC)cccc3F)=O)C2)nc(C)c(C)nc1O 84000,CC1CCC(CC(=O)NC2(CNC(C3CCCC3C)=O)CCCC2)CC1 84001,CCC(CC)(CN=c1[nH]nc(C(C)(C)C)o1)NC(c1nocc1C)=O 84002,CCC(CNC(C1C2CN(C(=O)C#CC(C)C)CC12)=O)CC(C)C 84003,N1(C(c2c(CC)cco2)=O)Cc2[nH]nc(C(=O)Nc3cccc(C)c3)c2C1 84004,Cc1ccc2c(c1)CC(C(=O)NC(CNC(c1ccc(C(F)F)cc1)=O)CO)S2 84005,CCCCC(F)C(=O)NC1(C(=O)N(C)CC2(O)CCC2)CCN(C)C1 84006,N1(C(C(COC(C)=O)O)=O)CCC2(C(N3CC(CO)C(O)C3)=O)CC2C1 84007,N1(C(C2C(OC)(OC)CC2)=O)CCC2CCC(NC(=O)CC3CC3(C)C)C1C2 84008,N1(C(c2c(Cl)cn(CCC)n2)=O)CCN(C(c2ccccc2)=O)CC(CO)C1 84009,CC1CN(C(=O)C(=O)NCCC(N)=O)CCCN1C(c1ccc2sccc2c1)=O 84010,c1(C(N2CCCC(N(C(=O)CCP(C)(C)=O)C)C2)=O)ccc2c(c1)[nH]c(=N)n2C 84011,Cc1ncn(C)c1NC(=O)NCC(Cc1ccccc1)C(C)C 84012,N1(C(Cc2c(C)cnn2C)=O)CCC2CCC(C1)N2C(=O)CC1CC(F)(F)C1 84013,Cc1cc(C(=O)Nc2ccc(-c3nnc(S)n3C(C)C(=O)O)cc2)c(C)o1 84014,C(=O)(C(CCOC)NC(C1CCC2CC12)=O)NCC#CC 84015,c1(OCC(=O)NC(C)CNC(c2cnc(N)cn2)=O)ccccc1C(N)=O 84016,C1(O)(C(N2C(C)CC(NC(=O)Cn3cc[n+](C)c3)CC2)=O)CCCC(C)(C)C1 84017,C(=O)(CC(C(C)C)NC(c1cnc(Cl)s1)=O)NCC(C(=O)OC)(F)F 84018,CC1(C)OCCC1CC(N1CCC(C)(NC(c2cnc(N)cn2)=O)C1)=O 84019,N1(C(CC(C=C)(C)O)=O)CCN(C(=O)C=CCN(CC(F)(F)F)C)C2COCC12 84020,c1(CC(=O)NC2CCC(N(C(C3(C(COC)OC)CC3)=O)C)C2)ccccc1C 84021,C1(C(=O)NC(c2ccc(C)cc2)C)CC12CCN(C(=O)C(C)CC1CCC1)CC2 84022,C(c1c(F)cccc1F)=CC(=O)NCC1(O)CCN(C(COCC#C)=O)C1 84023,C(=O)(C(C)(C(F)F)C1CCC1)NC(CC(=O)OCC)COC(C)(C)C 84024,C1(NC(C(c2ccc(F)cc2)C)=O)CC(CO)N(C(=O)Cc2cncs2)C1 84025,C(=O)(C#CC1CCOC1)NCC(CNC(c1c(F)ccc(C(C)C)c1)=O)O 84026,c1(C(N2CC3C(C(=O)NC(c4cccs4)C)C3C2)=O)cnc2n1CCC2 84027,CCC(C)(CO)C(=O)NCCN(C(=O)CNc1ccccc1SC1CCCC1)C 84028,Cc1cc(N2CCCC2)ccc1C(=O)O.C12CCCC(C1)NC2C 84029,c1(C(=O)NC2CC(CCNC(C(n3cc(Br)cn3)C)=O)C2)cc(C(N)=O)on1 84030,C12(CNC(C(C=C)(C)C)=O)CCCC1CCN2C(=O)CC1(O)CCC1 84031,c1(CNC(C(CCC)C)C)cc(C#N)ccn1 84032,C1(NC(CC=C)=O)CCN(C(c2ccc(-c3cc[nH]n3)cc2)=O)CCC1(F)F 84033,C(=O)(C(F)(CNC(C1CCCCO1)=O)C(C)C)NCc1n(CCC)ccn1 84034,N1(C(CC2N(C(C(C)OCCCC)=O)CCCC2)=O)CCCC(C#N)C1 84035,N1(C(c2c(C)cns2)=O)CC(NC(=O)CCc2cccc(O)c2)CC1C 84036,c1(C2C3CCCN(C3)c3nnc2n3C)ccc(F)cc1.C1(COC)CCCC=C1Br 84037,CCCC(F)C(=O)N1CCC(COC)(NC(c2csc(NC(C)=O)n2)=O)C1 84038,N1(C(c2cc(F)c(C)c(N)c2F)=O)CC(=O)NC2CCCCC12 84039,N1(CC(N2CC(C)(NC(c3c(C)n(C4CC4)nc3)=O)C2)=O)CCC(=O)NC1=O 84040,C1(C(=O)NCc2c(CC)c[nH]n2)CCCN1NC(=O)C=CC(=O)NC 84041,c1(N(C)C)ccc(N(C)C(c2ccccc2NOC2CCCCC2)=O)cc1 84042,C(=O)(C(F)(F)C(F)F)NCCCCC1CCCN(C(C(CSC)C)=O)C1 84043,C=CC(F)(F)C(=O)NC(CNC(c1cnn(CC2CC2)c1)=O)CC1CCCCC1 84044,C12(C(=O)NC3CC(NC(C(C)OCCCC)=O)C3)CCCN(CCC1)C2 84045,c1(C(N2CCC(NC(C=C(CC)CC)=O)C2)=O)nc(Br)sc1C1CC1 84046,C1(NC(CN(CCC)C)=O)CC(C(=O)Nc2cc(C)ccc2CO)C12CCC2 84047,C(=O)(C1=NOC2COCC12)NCC(=O)NC1CC(n2cc(C(N)=O)nn2)C1 84048,c1(C(=O)NCCC(=O)NC2C(CN(CC)CC)C2)sc(-c2ccc(C)o2)nc1C 84049,N1(C(C2C(C)CCCC2)=O)CC2(C=C(C(=O)N(C3CN4CCC3CC4)C)CO2)C1 84050,Cc1ncc(OCCC(N2CCOCC2)C)cc1NC(c1ccccc1)=O 84051,C1(CC(N2CC(O)(CCNC(C(C)CCN(C)C)=O)C2)=O)CC(O)C12CCC2 84052,C12(C(=O)Cc3c(C(=O)OC)n(C)nn3)CCCCC1OCC2 84053,n1(CC)nnnc1C1(C(=O)NC2(CC(C3CN(C(=O)NC)C3)C)CCC2)CC1 84054,Cc1nnc2cc(NC3CCCC34CN(C(C3C5C6CCC(C6)C35)=O)C4)ncn12 84055,CC1(O)CCN(CC(=O)NCCCNC(C2CCCCC2C(F)(F)F)=O)C1 84056,Cc1cccc(C(N2CC(C(=O)NC(C)(C)CCO)CCC2C)=O)c1C 84057,c1(OC)c(C(=O)NCC(F)CNC(c2c[nH]nc2[N+](=O)[O-])=O)cccc1F 84058,N1(C(COCCC#C)=O)CC(NC(c2nnc(O)cc2C)=O)C(C)(C)C1 84059,C1(C(=O)N)C2CC3C(C2=O)C13.C1(NC)CCN(c2nc(CC3CC3)ns2)C1 84060,C1(C(=O)NC(c2ncnn2C)CC)CC12CCN(C(C1(C)CC1)=O)C2 84061,CC1CN(C(c2ccccc2O)=O)CC1CNC(c1nnn(C)c1N)=O 84062,C(CC(C)C(=O)N1CCOCC1CNC(=O)Cc1ccc(C(N)=O)cc1)OC 84063,C=C(Cl)CC(C(=O)NCC(C)C(C)O)NC(c1ccc(=O)n(C)c1)=O 84064,C(=O)(C(O)CC(F)(F)F)NCCN(C(c1cc(S(C)(=O)=O)co1)=O)CC 84065,c1(C(N(C2CCCN(C(C3CC34CCC4)=O)C2)CCO)=O)cc2n(c1)CCSC2 84066,Cc1nnc2n1CCC(NC(=O)CNC(=O)C(=O)NC1CCCN(C)CC1)C2 84067,C1(NC(C(CCC2CC2)OC)=O)CN(C(=O)CN2C(=O)CN(C)C2=O)CC12CCC2 84068,C1(CC(=O)NC(C2N(C(C=CC(C)C)=O)CCC2)(C)C)CCC(=O)NC1 84069,C1(C#N)(C(=O)NCC(CN(C(C2(CC#C)CC2)=O)C)O)CC12CCCC2 84070,C1(OC)CCCN(C(C2C(NC(c3cnc(O)c(C)c3)=O)CCCCC2)=O)C1C 84071,c1(C(=O)NC2CCC(N(C(C(COCC)C)=O)C)CC2)csc(S(C)(=O)=O)c1 84072,C1(OCC)CCCCC1N=c1nc(N(C)CCc2nccs2)c2c([nH]1)CCC2 84073,c1(CC)cncc(C(=O)NC2CC2CNC(=O)C(C(=O)OC)OC)n1 84074,N(C1CCCc2nn(C)cc21)C(c1ccc2c(c1)CCCN2CC(=O)NCC)=O 84075,c1(C(=O)NC2C(NC(=O)Cc3ccc(CO)cc3)CCC2)cccc2[nH]ncc12 84076,c1(C(C)C(=O)NC2CCCN(C(c3csc(Cl)n3)=O)C2)ccc([N+](=O)[O-])cc1F 84077,c1(C(N2CCC(NC(c3c(CC)onc3)=O)C2)=O)c[nH]c(C)c(Cl)c1=O 84078,CC(C)CCC(C(=O)NC1CNC(=O)C1)NC(=O)Cc1cc[nH]n1 84079,CC1CCC(NC(c2c[nH]nc2C(=O)OCCCCC(=O)OC(C)(C)C)=O)CC1 84080,N1(C(CC(=C)C)=O)CCC2CC(C1)CN(C(c1cc(OC)ns1)=O)C2 84081,c1(NC(C2CC3(C2)CC3F)=O)cc(-c2ccncc2)ccc1OC(F)(F)F 84082,c1(C(=O)NC(CC=C)CNC(=O)C(C2CCC2)C2CCC2)cc2n(n1)CCO2 84083,N1(C(C2N(C(C)=O)CCCC2)=O)C(C)CC2CN(C(c3ccsn3)=O)CC12 84084,C1(F)(CNC(COCc2n(C)ncc2)=O)CCC(NC(=O)CC2CCCOC2)C1 84085,C(Cn1cncn1)(C(=O)NCC(N1CCCC1)=O)NC(CC(F)F)=O 84086,c1(CN2CCN(CCC)CC2)cnc(-c2cc(F)c(O)cc2F)c(OC)c1 84087,c1(CNC(C=CC=CC)=O)ccsc1C(=O)N(CCO)CCN(C)C 84088,C1(NC(c2c(CC)non2)=O)CCOC12CCN(C(c1cnn(C)c1F)=O)CC2 84089,N1(C(C(CSC)(C)C)=O)CC2CCC(C1)N2C(C1CCCN1C(=O)OC(C)C)=O 84090,N1(C(C=Cc2cnc(C(C)(C)C)o2)=O)CC2CC(NC(c3cccs3)=O)C(C2)C1 84091,C1(c2onc(C)n2)COCCN1C(c1cc(Br)no1)C(=O)NCCC#N 84092,CC1CC(NC(c2cccnc2O)=O)CCN1C(=O)C=Cc1ccccc1Br 84093,c1(-c2cn(CC(=O)NC(C(=O)OCC)C)nn2)cccc(OCC(=O)O)c1 84094,N1(C(C2(C=C)CC2)=O)CCN(CCN(C)C(c2noc(C3CC3)c2C)=O)CC1 84095,c1(C(C(=O)NC2CC2)N(CC(C)(C)C)CCC#N)cccc(S(N)(=O)=O)c1 84096,CCCC(C(O)C(=O)N(C1CC2CC2C1)C)NC(=O)CC(C)(C)OC 84097,C1(NC(=O)Cc2csnn2)CC2CC(C1)N(C(=O)C=CSCc1ccco1)C2 84098,C1(OC(=O)NC2CN(C(C3(C(=O)OC)CC(=C)C3)=O)C2)C=CCN(C(=O)CC)C1 84099,C12CCC(CC1)C(=O)N2.C1(O)(CC(=O)NC(CC=C)CO)CCOCC1 84100,C1(C)(CC(=O)OC)CCN(C(c2ccn(C)c2)C(=O)NC2COC2)C1 84101,C(c1cccc(F)c1Cl)=CC(=O)NCC(CNC(c1c[nH]ccc1=O)=O)CO 84102,c1(C(=O)NC2(CO)CCCN(C(CCC(=O)NC)=O)C2)ccc2c(n1)CCC2=O 84103,Cc1cocc1C(=O)NC(C)CNC(=O)NC1CCCCC1 84104,c1(COC)cnc(C(=O)NCC(O)CNC(C2CCN(S(C)(=O)=O)CC2)=O)cn1 84105,c12cccc(n1)S(=O)(=O)N(C)C1CCN2C1.C(CS(C)(=O)=O)C(=O)C.CCOCC1CC1 84106,C1(S(C)(=O)=O)(C(N2CC(C)C(NC(c3c[nH]c(=N)nc3O)=O)CC2)=O)CCCC1 84107,Cc1ccnc(C)c1CNC(=O)C1=CCN(C(C2(CC3CC3)CC2)=O)C1 84108,c1(C(=O)NCC2N(C(C(C)Sc3nncn3C)=O)CCOC2)c(F)ccnc1F 84109,c1(C(=O)NCC2CCN(C(C3CC=C(C)CC3)=O)CC2)cc(F)ccc1F 84110,CC1(C)C(C)(C(=O)NC2CCCC(NC(=O)CCCCn3ccnn3)CC2)C1(C)C 84111,c1(OC)ccc(C2=NN(C(=O)C(c3ccc(C)cc3C)C3CC3)CC2)cc1 84112,CC1(C)CCN(C(=O)CCn2cnnn2)CC1C(=O)NC1CC1NC(=O)NC1CC1 84113,N1(C(C2C(=C)C2C(=O)OC)=O)CCOC(C(=O)NC(C)Cc2ccnn2C)C1 84114,S(=O)(=O)(c1cncc(F)c1)N(C1(C(=O)OC)CNC1)C 84115,C1(C2CCN(C(=O)C=C(C)C(F)F)CC2)(NC(C2CN(CC)C(=O)C2)=O)CC1 84116,N1(CC(C)OC)CCCCC1.C(C(C)CN(C)C)N 84117,c1(C(N2C(C(=O)NCc3nccs3)CC(F)C2)=O)c[nH]c2ccc(Br)cc2c1=O 84118,C1(C(=O)NCCN(C(=O)C2=NOC(C)C2C)CC)CCc2nncn2C1 84119,CC(C)(C)CCCCCC(=O)N1CCC(CN=c2ccnc(Cl)[nH]2)CC1 84120,C1(NC(C(CC#C)(C)C)=O)CC2CCCC(C1)N2C(=O)C(C)N1CCC1 84121,N1(C(C(CC=C)(C)O)=O)CC(C(=O)NC2CCC(C3CC3)C2)CCC1(C)C 84122,C#Cc1cc(F)ccc1C(=O)OCCNC(C)=O 84123,c1(C(N2CC(NC(c3nn[nH]c3Cl)=O)CC(C)C2)=O)cc(S(N)(=O)=O)ccc1Cl 84124,C1(NC(c2ccc(C#N)[nH]2)=O)CN(C(=O)CCc2cccc(O)n2)CC1C1CC1 84125,CCC(C)(C#N)C(=O)NCCN(CC(C)O)C(=O)Cn1nc(C)cc1C(F)F 84126,c1(C(N2CC(NC(CCCC(CC)C)=O)CC2(C)C)=O)cc2ccoc2cc1F 84127,N1(C(Cc2ccc(OC)cc2)=O)CCCC(NC(=O)CCc2ccnn2C)CC1 84128,C1(C(=O)NC(CCN(C(C2=CCN(C)C2)=O)C)C(C)(C)C)CCn2cnnc2C1 84129,C(=O)(N=c1ccn(C(F)F)[nH]1)C1CCCC(NC(C(CC)Cl)=O)CC1 84130,c1(C(=O)NC(C2CCN(C(CCN(CCC)C)=O)C2)C)c(C(C)C)n[nH]c1C 84131,c1(C(=O)NCC(CNC(Cc2c(C)cco2)=O)(C)F)cccn(C)c1=O 84132,c1(C(=O)NC(C(C)C)CNC(=O)CCC2CC2(F)F)ccnc(C(C)(C)C)c1 84133,c1(NC(N(CCCC(C)C(=O)O)CC)=O)nc2c(s1)CCC2 84134,c1(CC(=O)OC2C(OC)CC2)ccn2c(=O)cc(-c3ccccc3)nc2c1 84135,C(=O)(CC(CC)(C(F)F)NC(c1cccnc1O)=O)OCC 84136,C1(CC(=O)NC2C(CNC(c3ccc(C(C)(C)C)[nH]3)=O)CC2)CCCOCC1 84137,c1(CN(C(C(CCC)N(C)C)=O)C)cccc(Cl)c1C(F)(F)F 84138,CC1CCN(C(c2cnn(CCF)c2)=O)CC1CNC(C1CC1F)=O 84139,C1(C(=O)NCC(C)(O)C2CCCC2)(CC)CCN(C(C2COCC(C)O2)=O)CC1 84140,Cn1ncc(C(=O)NC(CNC(=O)CCSC(F)(F)F)(CO)CO)cc1=O 84141,N1(Cc2nc(NC(c3c(F)ncc(C)c3)=O)sc2)CCCC2(C1)NC(=O)NC2=O 84142,CC(C)CC(=O)NCCOCCOCCNC(=O)C=CC1CCCC1 84143,c1(CNC(c2ncc(NC(=O)OC)c(Cl)c2)=O)ccc(S(C)(=O)=O)s1 84144,c1(-c2cccc(OC)c2)ccc2oc(C(=O)OCCC(CO)C(C)C)c(C)c2c1 84145,N1(C(c2ccnc(OC)n2)=O)CCN(C(c2cn(C)nc2Cl)=O)C(C2CCC2)C1 84146,N1(C(C2CN(C(C)=O)C2)=O)CCC(C)N(C(c2cn3cc(C)nc3s2)=O)CC1 84147,c1(-c2cccc(OC)c2C)c(C(N2CCC(C(N)=O)CC2)=O)[nH]c2ccccc12 84148,C(C(CC(C)(C)C(=O)Nc1cccc(-c2cc(NC(C)=O)cc(Br)c2)c1)OC)OC 84149,S(=O)(=O)(c1csc(C(=O)NCC2COCCN2C(c2cccnc2)=O)c1)NC 84150,N1(C(Cn2nnc(C)n2)=O)CCOCC(NC(c2cc(NC3CC3)ncn2)=O)C1 84151,c1(C(=O)NCC(CNC(CCOCCOC)=O)CO)ccc([N+](=O)[O-])s1 84152,N1(C(CCC#C)=O)CCCC(O)(CCNC(C23CC(CN2C2CC2)C3)=O)C1 84153,c1(C(N2CCC(NC(c3ccc(C(C)=O)o3)=O)C2C)=O)ccc2nccnc2c1 84154,C12(NC(c3c(OC)oc(C)n3)=O)CCCC1CN(C(c1ccc(C)c(C)c1)=O)C2 84155,c1(C(N2CCN(C(C3C(=C)C3)=O)C3C2COC3)=O)cc(OC)cc2c1CCCC2 84156,c1(C(=O)NC23CC(C(=O)NN4CCC(F)(F)C4)(C2)C3)ccc(C(F)(F)F)cc1 84157,c1(NCc2cnc(CO)c(Cl)c2)[nH]nc2ncnc(O)c12 84158,Cc1noc2cc(N3CCC4(C=C(CO)C4)CC3)nc(Cl)c12 84159,C(=O)(C1=CNC2=NCCC2=C1)NC1(C)CCN(C(C(COC(C)C)(C)C)=O)C1 84160,S1(=O)(=O)c2cc(cs2)C(=O)C(=O)C(C#C)N2CCN1CC2.C(=O)C(F)(F)F.OC 84161,C1(C(N(CCCNC(C2C(C)C2C)=O)C)=O)CC12CC(F)(F)C2 84162,C(CC(=O)NOCCF)OCCNC(C(COCC)C)=O 84163,CCC(C)CC(=O)NCCC1(C(=O)NCC2CC(C(=O)OC)C2)CC1 84164,C1(C(=O)NCC2(CNC(C(CC#C)C)=O)CCCCC2)COc2ccccc2C1 84165,C1(NC(C2N3CCC2C3)=O)CCC(F)(F)CC1.c1(COCCC)ccn(CC)n1 84166,N1(C(CSC)=O)CCN(C(c2cn(Cc3cccs3)nn2)=O)CC(C)C1 84167,C1(C(N2CC(NC(C(C)OC)=O)C(CC3CC3)C2)=O)CC(F)(F)CCC1(C)C 84168,c1(C(N(C2CN(C(C(CC)OC)=O)CC23CC3)C)=O)ccc2nncn2c1 84169,CCCCCC(O)C(C)C(=O)N1C(CCNC(=O)C(CO)OC)C2CCCC12 84170,c1(C(N2C(CNC(Cc3ccc(OC)c(F)c3)=O)CCC2)=O)ccc([N+](=O)[O-])cn1 84171,C1(NC(C(C)OCCC=C)=O)CCCC1NC(c1cc(C(C)=O)on1)=O 84172,C1(NC)C(C)OCC12CCN(C(c1cc(Br)ccc1Br)=O)CC2.C12CCN(C1)C2 84173,C(=O)(C(C(C)CC1CCCC1)N(c1ccc(Cl)nc1C)C1CC1)NCCCSC 84174,N1(C(C(CCC)NC(N)=O)=O)CC(C(N2CCC(O)C(CO)C2)=O)CC(C)(C)C1 84175,N1(C(CCCC#C)=O)CCN(C(C2CCCN(C(C)C)C2)=O)CC1CC(C)(C)C 84176,C(=O)(C1SCCc2sccc21)N1CCC(N(C(=O)C(O)CC(F)F)CCC)CC1 84177,C(=O)(C(CC)C(F)(F)F)NC(CCCC)C(=O)NCc1cc(C)ccc1C 84178,CN1CCC(N2CC(C(=O)NCCC3(CNC(=O)CSC(F)F)CC3)C2)CC1 84179,C(=O)(C(C)(C)C(C)C)NCC1CC(NC(c2c(C(=O)OC)c(C)[nH]n2)=O)C1 84180,CC1CCN(C(=O)N(C(F)CCc2cc(N(C(C)C)Cc3ccccc3)cs2)C)C1 84181,CCC(C(=O)N(C1CC(C#N)C1)CC(=O)NC(C)Cc1ccncc1)SC 84182,c1(C(=O)NCC(CC=C)NC(=O)CN2CC3CC3C2)cnn(CC(C)(C)O)c1C 84183,C12CN(CCO1)C(=O)C13CC(C1)(C3)NC2=O.C1CC1(F)F.COC 84184,C(=O)(C1=C(Cl)CCOC1)N1CCC(O)(C(C)CNC(=O)C(F)(F)C2(O)CCC2)C1 84185,c1(C(=O)NC2(CO)CCCN(C(C(C)C(F)(F)F)=O)C2)ccc(S(C)(=O)=O)o1 84186,N1(C(CNC(CCC)=O)=O)CC(N(C(=O)C(C)Cc2ccccn2)C)C2(CC2)C1 84187,C1(NC(c2cc(C)no2)=O)COCCC1NC(=O)CCc1cc(Br)cs1 84188,Cc1onc(Cl)c1C(=O)NCC(CC(C)C)NC(c1coc(C2CCCC2)n1)=O 84189,C(=O)(CCCCCCc1cccs1)N1CC(O)CC(NC(=O)C2=CCOCC2)C1 84190,C(c1cccc(O)c1)=CC(=O)N(C1CN(C(=O)C(F)(F)CO)CC12CC2)C 84191,N1(C(CCSCCCC)=O)CCC2CN(C(=O)C(C3CCC3)OC)CC12 84192,N1(C(c2c(C)cno2)=O)CC(NC(c2cn(-c3ccccc3Cl)nn2)=O)C(O)C1 84193,C1(CNC(=O)CNS(=O)(=O)C2CC2)CCCN(C(C2(n3ccnn3)CC2)=O)CC1 84194,c1(N2CCN(C(C=C(C)C(=O)O)=O)C(C(C)C)C2)ncnc2[nH]c(C)nc12 84195,N1(C(=O)CN2CC3CC3C2)Cc2ccc(C(N3COC(CO)C3)=O)cc2C1 84196,c1(NC(C2C(NC(CC=C)=O)CCCC2)=O)ccc(C)c(CC)c1 84197,c1(OC)ccc(NC(=O)C(N2CC3CCCC23)c2nnc(C3CC3)s2)cc1 84198,c1(NCC(C2CCCC2)NC(c2ccc(OC)nc2)=O)c([N+](=O)[O-])cnn1C 84199,Cc1ccc(C(=O)NCC(O)CNC(c2c(C)noc2C(F)F)=O)cc1[N+](=O)[O-] 84200,Cc1cc(Br)cc(S(=O)(=O)N2CC3(CCC(NC(c4nccs4)=O)C3)C2)c1 84201,N1(C(c2c(C)ncnc2)=O)CCN(C(c2cc3ccccc3s2)=O)CC(O)C1 84202,C1(COC)(CNC(C2CC(=O)N(C)C2)=O)CCN(C(c2sccc2OC)=O)CC1 84203,C(=O)(C1=CC2(CN(C(=O)C(C)(C)CC)C2)OC1)N(CCn1nccn1)CC 84204,C1(CN(C(=O)CCCC2CCCC2)CC(=O)NCC2CC2)CC12CCOCC2 84205,Cc1ccc(C23CC2CN(C(=O)NCCc2noc(C)n2)C3)cc1 84206,Cc1cncnc1C(=O)NC1(CNC(=O)COc2ccon2)CC(F)(F)C1 84207,C1(NC(=O)NC(CCCOC)C)CCC2(CC1)CC2C#N 84208,Cc1cccc(F)c1CC(=O)NC1C2CC1CN(C(=O)CC1COCC(C)O1)C2 84209,c1(C(=O)NCC(N(C(=O)Cc2ccns2)C)C2CC2)cc(Cl)cn1C 84210,N1(CCOC)CC(C(N2CCC2c2cnn(C)c2)=O)CC1=O.C(=O)(C(F)(F)O)NC 84211,c1(C(N2CCN(C(C3C(OCC)C3C)=O)CC2)=O)ncc([N+](=O)[O-])c(C)n1 84212,CC1=C(C(=O)NCC2CC2NC(c2nn(C)c(C)c2Br)=O)SCCO1 84213,NS(=O)(=O)c1cccc(C(=O)NCCNC(=O)CCSCc2ccccc2)c1 84214,Cc1cc(F)sc1C(=O)NC1(CNC(c2cc(C(F)(F)F)[nH]c2C)=O)CCCC1 84215,C(=O)(CC1C(=O)Nc2cc(Cl)ccc21)NCC1(OC(C)=O)CCOC1.C1C(=O)N1 84216,C=CCC(CC=C)C(=O)NC1CN(C(=O)Cn2cnc(=N)[nH]2)C2CCCC12 84217,CC(C)C1=NOC(C(=O)N(CC(=O)NCC2CCC(=O)O2)C)C1 84218,CN=c1[nH]cc(C(N2CCCC2C2CCCN(C(=O)C=CCOCCOC)C2)=O)o1 84219,c1(C(C2CC2)NC2(C(=O)NC(C3C(=O)OCC3)CO)CCC2)ccccc1F 84220,c1(CN2C(CCC(=O)NC(C(=O)OC)C3CC3)CCC2)ccc(C#N)s1 84221,c1(C(C)=O)ccc(N2CCCC2C2(NC(=O)C(C)SC(F)(F)F)CC2)nc1 84222,c1(C(=O)NCC)cc(CC2CCC(C(=O)N(C)C(C)C)CC2)ccc1O.C1(C)CC1 84223,c1(COC)cc(C(=O)NCC2C(C)CCN2C(c2ccc[nH]2)=O)c(C)o1 84224,C1(CC)CCN(C(=O)CSCC(F)F)C1C(=O)Nc1ncncc1Cl 84225,C1(C(=O)NC(C)C(=O)NC(C)C(=O)NCC(F)CO)C=CCCC1 84226,C12(C(=O)NCCCCCNC(C3CC34CCOC4)=O)CCN(CC1)CC2 84227,N1(C(C2CCC(c3ccccc3)=NO2)=O)CCCC1C1CCCN1CC=C(Cl)Cl 84228,CC1(CCC(=O)NC)CCN(C(=O)C(=O)NC2(CO)CCCCC2)CC1.CCO 84229,C1(C(C)NC(c2c(CC)cns2)=O)CCCN(C(c2n[nH]cc2Cl)=O)C1 84230,Cn1ncc2c1CCN(S(=O)(=O)c1c[nH]c(C#N)c1)C2C(=O)OC(C)(C)C 84231,C=CC(C)CC(=O)NC1COCC1NC(c1cc(C)sn1)=O 84232,N1(C(CSC)=O)CC2(CCC(CNC(=O)CNC(=O)CCC(C)C)O2)C1 84233,N1(C(C(CO)NC(C(C)C)=O)=O)CC(O)CC1(C)C(=O)N(C)CCN1CCCC1 84234,C#CCC(C)(C)C(=O)NC1CCN(C(=O)CC(OCC)OCC)C12CC2 84235,C1(C(=O)Nc2c(C)nn(CC(N3CCN(CCF)CC3)=O)c2)CCC2C(C1)C2(F)F 84236,CCC(C)CCCCC(=O)N1CC(NC(=O)C=CC(F)(F)F)C2(CCC2)C(C)C1 84237,C(=O)(C1c2c[nH]nc2CN1C(c1cnc(C)c(C)c1)=O)NCC1(CC)CCC(=O)N1 84238,c1(CNC(c2cccc(CNC(CC3CC(=C)C3)=O)c2)=O)nnc2ccccn12 84239,C(=O)(CCCCC(F)(F)F)N1CCC(N(C(=O)C(C)(C)C)CCOC)CC1 84240,C1(C(=O)NC2CCCC2NC(c2cccnc2O)=O)(OC)CCCC(C)(C)CC1 84241,C(C1c2ccccc2CN1C(=O)CC1COCCO1)NC(C=NOC)=O 84242,N1(C(Cc2c(C)ccs2)=O)CC2CC(NC(C3CCC(C)(C)O3)=O)CC1C2 84243,N1(C(C(CC=CCC)C)=O)CCC(N=[N+]=[N-])(C(=O)NCC(C)(O)C2(C)CC2)C1 84244,Cc1cc2nc(NCC3(F)CC(NC(C4CCCOC4)=O)C3)cc(=O)n2o1 84245,C1(C(=O)NCCCC2(NC(Cc3c(C)ocn3)=O)CC2)CC2C=CC1CC2 84246,C1(CC)CN(C(C2CCCCO2)=O)CCN1C(C1CC(C(=O)OC(C)(C)C)C1)=O 84247,N1(C(CN(C2CCCS2(=O)=O)C(C)C)=O)Cc2ccoc2CC(C)(C)C1 84248,c1(C(=O)NCC(CN(C(C2(CC=C)CCCCC2)=O)C)O)cccc2sncc12 84249,c1(CNC(C2(C)CCN2Cc2cnc(Cl)cc2Br)=O)ccc(F)c(C(F)(F)F)c1 84250,N1(C(c2cncn(C)c2=O)=O)CC2CCCC2(CNC(c2cnc[nH]c2=N)=O)C1 84251,C=CCC(C)(C)C(=O)N1C2CCC(C2)C1C(=O)NC1CON(CC)C1=O 84252,c1(OCC=CC(=O)NC2CC(C)(CNC(c3c(C)cns3)=O)C2)ccc(Cl)cc1 84253,C1(O)(Cn2cc(CC(C)C)nn2)CCN(C(=O)CCC(F)F)C1 84254,C1(CC(=O)NCC2(NC(=O)CC3CC3CO)CCCCC2)CN2CCC1CC2 84255,N1(C(C=CC(C)C)=O)CCC2CCN(C(c3ccc(F)c(C(F)F)n3)=O)CC2C1 84256,c1(C)c(Cl)c[nH]c2nccc1-2.C1(C(=O)O)CNCCN1CCN 84257,N1(C(C2CN(C(C3(COC)CC3)=O)C2)=O)CCC(C#N)C1 84258,C(CC(C)(C)C(=O)NCC(CO)NC(C1(F)CCN(C(C)(C)C)C1)=O)OC 84259,C(=O)(C1CCc2nccn21)NC1C(CNC(C23CC=CCN2CCC3)=O)CCC1 84260,c1(C(=O)NCc2ccc(C(C)NC(COCC)=O)cc2)nnn2c1CCCCC2 84261,C(=O)(C(C)C1=CCCC1)NC(CCOC)CNC(c1ccc(C(=O)OC)cc1)=O 84262,N1(C(c2cc(C)[nH]n2)=O)CC2(C1)CN(C(C13CCC(C)(CC1)OC3)=O)CC2CO 84263,C(=O)(CCN=C(NCc1cccc(-c2ccncc2)c1)NCC1CC1Cl)NC 84264,CC(N=c1[nH]c2c(c(=NCc3cnns3)[nH]1)CCCC2)c1ccc(O)nc1 84265,C1(C(N2CCOC(c3cn(Cc4ccccn4)nn3)C2)=O)CCC2CCC12 84266,Cc1cc(C(N2CC(NC(c3cc(C4CCC4)nn3C)=O)C2)=O)ncc1C(N)=O 84267,C1(CC(=O)Nc2c(C)ncnc2)CC2(CC2)CN1C(=O)Cc1cc[nH]n1 84268,c1(C(=O)Nc2c(C)cc(NC(C3CCCOC3)=O)cc2)ccnc2c1cnn2C 84269,C1(C(C(=O)NCc2ccnn2C)N(CC(=O)NC)C)CCCOCC1 84270,C(C(C(=O)N1CCOCC1)NC(c1cn[nH]c1)=O)N(C)C 84271,C1(C(=O)NC2CCCN(C(c3cc(-c4ccco4)[nH]n3)=O)C2)C2CCCCCC12 84272,S(=O)(=O)(c1cc(Br)c(C)cc1F)N1CCCC(CN(CCC)C)C1 84273,Cc1ccc2c(C(N3CC(CNC(=O)C(O)C(F)F)C(C)(C)C3)=O)coc2c1 84274,N1(C(c2c(C)coc2C)=O)CC2(CCCC2NC(=O)C(C)Oc2ccccn2)C1 84275,N1(C(c2c(C)nc(Br)s2)=O)CCC2C(CCN2C(c2cc(Cl)cc(Cl)c2Cl)=O)C1 84276,CCCC(CCC)C(=O)N(C1CN(C(=O)Cc2cc[nH]n2)C1)C 84277,C1(N(C(c2cnc(CCCC)[nH]2)=O)C)CCCCN(C(c2cc(C#N)no2)=O)C1 84278,C(C(C(C)(C)C)NC(c1cc[nH]c1C(C)C)=O)NC(C=CC(C)(C)SC)=O 84279,C1(NC(c2ccc(OC(F)F)cn2)=O)C2CC1CN(C(=O)C=C1CCC1)C2 84280,N1(NCP(OC=O)(C)=O)CCC2(CC1)CCN(C(=O)C=C(C)C(C)C)C2 84281,C1(NC(CCOCC)=O)CC(C)(NC(c2cnc[nH]2)=O)C1 84282,C1(CNC(c2ncccn2)=O)CCCCN(C(=O)CCOCC2CCC2)C1 84283,N1(C(C(CC)(C)C)=O)CCC(O)(C(C)CNC(c2cc(C)c(C)nn2)=O)CC1 84284,C1(CNC(c2ccc(O)c(F)c2)c2n(CCSC)nnn2)CCOC(C)(C)C1 84285,C12(CNC(CS(=O)(=O)N(C)C)=O)CC(C1)C(NC(=O)C1=COCCO1)CO2 84286,c1(OC)cc(I)ccc1C(=O)NCC1(O)CN(Cc2ccc(O)cc2Cl)C1 84287,N1(C(c2n(C)c(S)nn2)=O)CC(CNC(=O)COCC2CCC2)CC12CCC2 84288,Cc1cccnc1CC(=O)N(C1CCN(C(=O)Cc2ccc(Cl)cc2)CC1)C 84289,c1(C(=O)NCC(CC)NC(=O)CCCCCSC)c(C)cccc1O 84290,C12COCCC1CNC2=O.Cn1ccnc1C(=O)NCC1CC1(Cl)Cl 84291,C1(CC#C)CN(C(=O)C(C2(O)CN(C(C3(C4CC4)CC3)=O)C2)F)CCO1 84292,C(C(C)CC(=O)N(C(C)C(C)(C)O)C)NC(c1c(C)nco1)=O 84293,C1(C(N2CC(CNC(=O)C(F)(F)CC3CCCO3)C2)=O)CCc2[nH]nc(O)c2C1 84294,Cc1nc(CC(=O)N(CCCC(=O)N2CC(c3cccnc3)C2)CCO)cs1 84295,CC1CC(C)N(C(c2coc(C3CC3)n2)=O)CCN1C(=O)C=CC(C)(C)C 84296,C(=O)(C(O)CC(F)(F)F)N1C(COC)(CNC(c2ccc(O)nc2C)=O)CCC1 84297,Cc1nc(CC(F)(F)F)sc1CC(=O)NCCN(C(=O)C(O)CF)C(C)C 84298,C1(C)(C(N(CC(C)N(C(=O)Cc2cn(C)nc2C(F)F)C)C)=O)CC2CC2C1 84299,C12(NC(C(C)=C3CC3)=O)CCCC1N(C(c1cnn3c1OCC3)=O)CCC2 84300,C12(NC(Cc3nc(C(C)C)sc3)=O)CC1CN(C(c1cnn(C(C)C)c1F)=O)C2 84301,C1(NC(C(C2CC(F)(F)C2)OC)=O)CCC(NC(=O)C=Cc2c[nH]cn2)CC1 84302,C12(CO)CCN(C1)C(=O)C=CCCC(=O)N2.CC=C 84303,CC(C)COCCOCCOCCOCCNCC(=O)C1CCC1 84304,C1(CNC(C(CN(CC)CC)F)=O)CN(C(C2C3CC4C(C3=O)C24)=O)CC12CC2 84305,N1(C(C(C)CN)=O)Cc2cccn2CC(C(N2CCC2C(C)(C)O)=O)C1 84306,CC1CC(CNC(=O)CCOCC(F)F)CN1C(=O)CCN1CCCC1=O 84307,C1(CCCNC(=O)COCc2ccc(F)cc2F)Cc2ccccc2C1 84308,C12(NC(c3cn(CCCC)nn3)=O)CCCC1(F)CN(C(c1ccncn1)=O)C2 84309,CC1CC2(CC(C(=O)NOCC(=O)NC3(C(F)F)CCC3)C2)C1 84310,n1(CC(N2CCC(NC(C3(C(N)=O)CC3)=O)C(F)C2)=O)ccc(=O)c([N+](=O)[O-])c1 84311,C1(NC(CC(C)(C)C#N)=O)CCCCCN(C(=O)C2=CCCC2(C)C)C1 84312,N1(C(C(CC)OCC)=O)CCN(C(=O)C=Cc2c(C)coc2C)C(CC)C1 84313,c1(C(=O)NCC(C2CCC2)NC(=O)Cc2csc(Cl)c2)ccc(F)cc1F 84314,c1(OCC)oc(C)nc1C(=O)NC1CC(N(C(=O)CC(O)c2ccccc2)C)C1 84315,C(C(F)(F)C(=O)NC1CCOCC1C(=O)NCCC(O)C1CC1)N(C)C 84316,C1(C(C)C)CCCCCN1C(=O)C(O)C(Br)c1ccccc1 84317,c1(N2CCCC(C)(CNC(C3(C)CCCC3)=O)C2)ccc([N+](=O)[O-])cc1C(N)=O 84318,Cc1nn(CC(=O)NC2CC2NC(C2(O)CC(OC3CCOCC3)C2)=O)c(=O)o1 84319,C1(NC(Cc2c(C)nc(C)s2)=O)CC2CCC(C1)N2C(C1(CF)CC2(CCC2)C1)=O 84320,c1(C(N2C3CN(C(C4(C)N(C)CCC4)=O)C(C3)C2)=O)ccc(F)c([N+](=O)[O-])c1 84321,C1(C)(CNC(C2C(C)C2)=O)CCN(C(C2CC23CC(O)C3)=O)C1 84322,C1(CNC(=O)C2CC2)(C)CC(C)(C)C1.c1(C(=O)OC)cccc(Sc2nn[nH]n2)c1 84323,c1(C(N2CC3C(C(=O)Nc4ncn(C)n4)(C3)C2)=O)c(F)cc(Br)cc1Br 84324,c1(CCC(=O)NCC(CNC(C2(CC#C)CCOCC2)=O)O)c(F)cccc1F 84325,C(CC(=O)NC1CCC(NC(=O)C(C)(C)c2cc[nH]n2)C1)(C(F)(F)F)OC 84326,C(C1=CCN(C(=O)COC(C)C)CC1)c1cncc(C(=O)OCC)c1 84327,C1(CC(C)C)(C(=O)N(C2CCCN(C(=O)CC)C2)C)CCNC1=O 84328,CC1(C)CCCC(CC(=O)NCC2(C)CCCC2NC(=O)Cn2cccn2)C1 84329,N1(CCNC(CNC(CNC(CCSC)=O)=O)=O)CCNC(=O)C1 84330,C(=O)(CCCC(F)(F)F)NC(C1CCn2ccnc2C1)C 84331,C1CCC(C)(C)C1.CCC(C)N(CCNC(=O)OC(C)(C)C)CC 84332,c1(Nc2ccc(CCCCCC)cc2)cc(C)c2sccc2c1 84333,C1(C(=O)OC)CC(C)CN(Cc2cc(C)c(-c3cnccn3)s2)C1 84334,N1(C(c2nc(OCC)oc2)=O)CCC(NC(c2coc(N(C)C)n2)=O)C(C)(C)C1 84335,C1(C(N2C(C)(C(=O)NCC3CCC3(F)F)CCC2)=O)CC2CC1CC2=O 84336,c1(C(N2CCC(n3cncn3)C2)C(=O)NCC(=C)C)cc(F)ccc1Br 84337,C(Cn1cncn1)(C(=O)N(C1C2CCCC12)C)NC(C1CC(=C)C1)=O 84338,c1(OC)ccc(C)cc1CNC(=NCC1CCCO1)NCc1ccc(SC)s1 84339,N1(C(c2c(CC)onc2C)=O)CCC(NC(=O)C=Cc2cscn2)C(C)C1 84340,c1(C(=O)NCC2C3CN(C(Cc4c(C)n(C)nc4)=O)C2C3)n[nH]c2c1CCCC2 84341,C=CC1(C(=O)NC2CCC(C(=O)NCC3CC3(C)C)C2)CCCC1 84342,C1(NC(CC2CC(OC)C2)=O)CCN(C(=O)CC(C)OC)CC1 84343,C=CC1OCCCC1C(=O)N(C)CCOCCN(C)C(c1ccc(F)cc1N)=O 84344,C1(C(N(C2CCCCC2)CC)=O)CCN(C(C2CCC=CCC2)=O)CCO1 84345,C1(NC(C=CC)=O)C2CN(C(=O)CC3(n4cccn4)CCOCC3)CC12 84346,C(=O)(C1=NOC2(CCOC2)C1)N1CCCN(C(C2N(N=O)CCCC2)=O)CCC1 84347,CCCC(F)C(=O)NC(C)(C)C(=O)NCC(C1CCOC1)SC 84348,C(CN=C(NCC1(CO)CC2CC2C1)N1CCC1)N(C1CC1)CC 84349,c1(NCCOCCNC(c2ccc(COC)c(F)c2)=O)ncc([N+](=O)[O-])c(O)n1 84350,C#Cc1cc(F)cnc1NC(C1CN(C(c2ccc([N+](=O)[O-])o2)=O)CCC1O)=O 84351,N1(C(Cc2c(C)ocn2)=O)CCC(C)C(CNC(c2cc(C(C)C)no2)=O)C1 84352,C1(CNC(C(COC)C)=O)CN(C(c2ccc(F)s2)=O)CCC12CCC2 84353,c1(CNC(N2CCCC(c3n(C)cnn3)C2)=O)cc(Br)ccc1-n1ccnc1 84354,CCC(C)CC(=O)NC1(CC(=O)NCC)CCCC1.N12CC(C1)C(OC)C2=O 84355,C1(F)(C(N(CCCCC=C)C)=O)CCN(C(C2SCC=C2C)=O)CC1 84356,Cc1cc(-c2nc(C3CCCCC3)nn2-c2cccc(Br)c2)c(C)[nH]1 84357,C(=O)(C1=NOC2(CCOC2)C1)N(C)CC1(NC(C2CCCOC2)=O)CC1 84358,C1(CN(C(C=CSC)=O)C2CC2)CCN(C(C2CC2c2nnc(S)n2C)=O)CC1 84359,C1(C2CCN(C)CC2)(C(N2CCCC(CNC(C(=O)NCCOC)=O)C2)=O)CC1 84360,N1(C(c2ccc(N)c(F)c2)=O)CC2(CCCC2NC(C2CCCC23CC3)=O)C1 84361,Cc1c(NCCCCCN2CCCC2)ncnc1N(CC#CCN(C)C)C 84362,N12CC3CC1CN3C(=O)c1cnc(o1)C2=O.c1ccc(C(C)(C)C)cn1.C1CC1 84363,c1(C(N2CC(C(=O)NC(C)Cc3ccccc3Cl)OCC2)=O)cnc(O)cc1O 84364,c1(C(C(N2CC(O)(CCNC(=O)C(F)C3CCCC3)C2)=O)O)cc(Cl)cc(Cl)c1 84365,c1(CC(=O)N(C)CC2(O)CN(C(c3cc(Cl)c[nH]3)=O)C2)c(F)cccc1F 84366,C1(C(N2CCCC2COC)C(=O)NCCC)CCCN(C(C)(C)C)C1 84367,C1(CC)C(NC(C2CC2c2cccs2)=O)CCN1C(=O)CCOc1cccnc1 84368,CC1CN(C(c2ccoc2)=O)CC2(CCN(C(c3cccc(N)c3N)=O)CC2)O1 84369,C1(NC(C(COC)(F)F)=O)CC(O)CN(C(c2ccc(Cl)nc2OCC)=O)C1 84370,C(=O)(C(CO)C(F)(F)F)NCc1cccc(NC(CCCCC=CC)=O)c1 84371,c1(C(C2CCN(C(C)(C)C)C2)C)nc(NC(=O)NCC2CCC2)[nH]c(=N)n1 84372,Cc1cc(C(=O)NCC2CC(NC(C3CC3C)=O)C2)c2c(C)c(C)[nH]c2n1 84373,CN1C2CCCC1CN(C(=O)CC(C)(C)NC(=O)C=CC1CCOC1)C2 84374,c1(OC)ccc(S(N)(=O)=O)cc1C(N1CCC(C#N)(NC(c2ccsc2)=O)C1)=O 84375,S(=O)(=O)(c1cnccc1N1CCC(C)(CO)C1)N(C(c1ncc(F)cn1)C)C 84376,C(=O)(C(C)(C)C1CCCN1CC(C1CC(=O)C1)=O)NC1(C)CC1 84377,CC(CN(C)C)CCC(=O)NCC1C=CC(NC(=O)CN2CCSCC2)C1 84378,c1(C(N2CCN(C(CC)C)CC2)C(=O)NCC(C)C)nc(Cl)cc(C)c1Br 84379,c1(C(=O)NCCCNC(c2cccc(C3CC3(F)F)c2)=O)cc(Cl)cc(Cl)c1F 84380,C(=O)(CC1=CSC2=NCCN12)N(C(CCNC(C1(C)CC(C)OCC1)=O)C)C 84381,C(CCC(C)C)(C(=O)Nc1cnc(C)c(Cl)c1)NC(CN(C(=O)OC)C)=O 84382,c1(SC)cc(C(=O)NC2CC2NC(=O)Cc2cncn2C)ccn1 84383,CCC(C)CCCCC(=O)NS(=O)(=O)c1cnccc1N1CCCN(C)CC1 84384,c1(N2C(CN(C)C(c3ccnc(F)c3Cl)=O)COCC2)ccc2nccnc2n1 84385,c1(C(C)NC(=O)C(=O)NCCc2cnn(C)c2)ccc(C(C)(F)F)cc1 84386,C1(C(N2C(CNC(c3n(C=C)ncc3)=O)CCC2)=O)CCc2nnc(O)cc2C1 84387,CC1(CCNC(C2(n3nccn3)CC2)=O)CCN(C(C2CCCC(=O)O2)=O)C1 84388,c1(C(N(C2CCCN(C(C3C(OCC)C3)=O)C2)CC)=O)cnc(CO)nc1C 84389,C1(C(C)C)N(C(c2cn[nH]c2)=O)CC12CCN(C(C1CCCCC1)=O)CC2 84390,Cc1ccc(F)cc1C(=O)NC1(C(N2CCC3(CCC3)C2)=O)CCCC1C 84391,C(=O)(C1=NOC(C)(C)C1)NC1CCCC(NC(c2c(C)ncc(C)c2)=O)CC1 84392,C1(NC(C(C)(C)NC(c2cn(C)nc2)=O)=O)CC12CC(O)C2 84393,C(=O)(CCCC=C)NCC(CC=C)NC(c1cn(CCCC#N)nn1)=O 84394,C#CCC(C)(C)C(=O)Nc1ccccc1C(n1cc(C2CCCN(CC)C2)nn1)O 84395,Cc1cc(C(=O)NCCOC2CCN(C(=O)C(O)C(C)(C)C)C2)ncc1C#N 84396,NS(=O)(=O)c1ccc(C2(CN3CCc4ccccc43)CC(F)(F)C2)cc1 84397,N1(C(CCN(CCC)C)=O)CC(c2ccccc2)(NC(c2occc2Cl)=O)C1 84398,C1(NC(C(C)Oc2cccc(F)c2)=O)CCN(C(=O)C=C2CCC2)CC12CCC2 84399,c1(C(=O)NCC2(C)N(Cc3ccc(C)cc3Br)CC2)c(Br)cc(F)c(F)c1F 84400,c1(CN(C)C(C2(CCNC(C34CCC(C3)C4)=O)CCC2)=O)ccn(C)c1 84401,c1(CN2CC(C)(CC(O)Cc3ccc(Cl)cc3)C2)cc2cc(Br)ccc2s1 84402,C(=O)(CCCCC(=O)NC1CN(C(C2(O)CCOC2)=O)CC2(CC2)C1)NC 84403,C1(NC(=O)CCCC2CN(C(C=C(C)CCc3ccccc3)=O)C2)CCOC1(C)C 84404,C(C(C)(C(=O)NCC(Cc1ccccc1)NC(C1CC(C(=O)OC)C1)=O)OC)OC 84405,n1(CC)nc(C)c(C(N2CC3CC2C3CNC(C23CCOC(C)(C2)C3)=O)=O)c1Cl 84406,N1(C(C2N(C(c3cc(C)n(C(F)F)n3)=O)CC(O)C2)=O)CCC(O)C(C)C1 84407,Cc1cc(CCC(=O)NCCNC(C2CC(=O)N(C3CCC3)C2)=O)cc(C)n1 84408,CON1CC(C(=O)NCCCN2CCC(NC(C3CC4C=CC3C4)=O)C2)CC1=O 84409,N1(C(C2CC(OC)C2)=O)CCC2(CC2)CC1C(=O)NC(CCO)C1CCC1 84410,CC1OCCC1(F)C(=O)NCC(C1CCN(C(=O)C2CC2)CC1)(C)C 84411,C1(CNC(c2ccc(C(C)(C)C)[nH]2)=O)CN(C(=O)CNC=O)CCC12CCC2 84412,c1(NC(C2CCCN(C(c3c(C)ncnc3)=O)C2)=O)ncnc2[nH]c(Br)nc12 84413,N1(C(C=CC)=O)CC(NC(=O)C(Cc2ccccc2)CC(C)C)CC2(CCC2)C1 84414,CC1CCOC1CCNC(=O)C(C1(C)CC1)NC(=O)Cc1ccon1 84415,C1(CNC(CCC#C)=O)(OC)CCN(C(c2ccc(-c3ccccc3)nc2)=O)C1 84416,c1(CC(C)C)ccc(C(=O)N(C2CCN(C(c3cc(F)c[nH]3)=O)C2)C)cc1 84417,C1(C(=O)NC2(CCC)CCOC2)CCN(C(C2C3CN(C)CC23)=O)CCO1 84418,C1(NC(CC(C)C)=O)CC2CC(NC(C3CNC(=O)N3)=O)CC12 84419,S(=O)(=O)(c1cccc(=NCC(C)C(C)C)[nH]1)N1CCC(C(C)C)CC1.CCCO 84420,N1(CCC)CCC(CNC(c2conc2CNC(=O)CCC2(C#N)CCC2)=O)C1 84421,c1(C(=O)NCC(C)(O)CNC(C2(Oc3ccccc3)CC2)=O)cccnc1Cl 84422,C(=O)(CS(=O)(=O)C1CCCC1)N1C(CNC(C2CC3CCC2C3)=O)CC(F)C1 84423,C1(=CCNC(C=CCCC(C)C)=O)CCN(C(c2c(C(C)C)cnn2C)=O)CC1 84424,C(=O)(C(F)CC(CC)CC)NCC(=C)CCNC(C1(C2CCCO2)CCOCC1)=O 84425,CC1(C(N2CCCC(F)CC2)=O)CCCN(C(=O)CNc2ncccn2)C1 84426,N1(C(c2cnn(C(C)(C)C)c2)C(=O)NC(C)C)Cc2ccccc2C(C)(C)C1 84427,CC1C(NC(=O)CNC(C2CCCCC2)=O)CC2CCC1N2C(=O)CCC1CC1 84428,c1(C(C(=O)NCC#CCNC(C2OCCN(C)C2)=O)F)ccc(F)cc1F 84429,C1(C(N2CCC(Cn3ncc(C)c3)CC2)=O)CCOC2(CCC2)C1 84430,Cc1cc(C)c(C(N2CC(CCO)(Cc3cn(CC(O)C(N)=O)nn3)C2)=O)[nH]1 84431,C(=O)(NNc1ccc(Br)c(F)c1F)N1CCC(C(=O)OC(C)(C)C)C12CC2 84432,C1(C(=O)NCCN(CCOC)C(C)=O)CCOCC1NC(=O)C=NOC 84433,CC1CN2CCN1C(C(=O)NC(CNC(c1cnc3[nH]ccc3n1)=O)C1CC1)C2 84434,C1(c2cn(Cc3c(C)nc(CC)o3)nn2)CN(C(c2ccnn2C)=O)CC1(C)C 84435,C(C(C)(O)CC(=O)NC1CCOCC1C(=O)NCCc1cn(C)nc1C)OC 84436,N1(S(CCC)(=O)=O)CC(C(=O)O)C2(CN(CC=CC=O)C2)C1.C(C)(C)(C)OC=O 84437,N1(CC23C(CN(C(c4cccc(SCC)n4)=O)C2)CC3)CCC2CN(C)CC2C1 84438,C1(NC(CNC(CCC)=O)=O)CC(C)(C(=O)OC)C1 84439,n1(CCCC(=O)NC2CN(C(C34CCCC(CO3)C4)=O)C2)cnc2ccccc12 84440,C1(C(=O)NC2C(SC)CN(C(=O)CCCn3ccnn3)C2)CC(C)(C)C(C)(C)C1 84441,C1(NC(=O)C(C2CCCCC2)O)CCCC1OCc1cccnc1 84442,FC1CC2CC1CC2NCc1cccc(Br)c1 84443,N1(C(=O)CC2CCCC2(F)F)CC2CCCC(C1)N2C(c1cncc(Cl)n1)=O 84444,c1(C(=O)NC2C(CNC(c3cc(Br)co3)=O)CC2)n[nH]cc1[N+](=O)[O-] 84445,c1(C(=O)OC)sc(-c2ccc(C(=O)NC(C)CN(C(=O)C(N)=O)C)cc2)nc1C 84446,Cn1cc(C(=O)NC2C3CC2N(C(=O)Cc2ccc(C#N)nc2)C3)ccc1=O 84447,C#CCCCCCC(=O)N1CCCC(CC)(NC(=O)C=CC(c2cccnc2)=O)C1 84448,N1(CC(=O)NCC(=O)NCCO)CCc2ccccc2C1.N12CC3CC(C3)(C1)C2=O 84449,c1(C2OCCN(C(c3c(OCC)nsc3)C(=O)NC(C)C)C2)ccc(F)c(F)c1 84450,N1(C(c2n(CC)cc(Cl)c2)=O)CCCC(CN2CCC(N(C)C)C2)CC1 84451,c1(C(=O)NCCNC(CC2C(C)C2)=O)cccc2c1NC(=O)CC2 84452,c1(C(=O)NCC2CCN(C(=O)C#CC3CC3)C23CCC3)ccnc2nccnc12 84453,N1(C(c2c(Br)n[nH]c2Br)=O)CCC2(CCCN2C(c2ccoc2)=O)C1 84454,C1(F)(CNC(c2ccoc2)=O)COCCN(C(=O)Cc2ccc(Br)cn2)C1 84455,C1(CCC)CC(C(=O)NCC(C)(C)CCNC(=O)CN(C2CCC2)C)CCO1 84456,c1(C(N2CCN(C(CC=C)=O)C(c3nccn3C)C2)=O)cc2cc(Br)ccc2[nH]1 84457,N1(CC(=O)N(c2ccc(C)c(C)n2)C2CCN(C)C2=O)CCN(C(C)=O)CC1=O.CO 84458,CC(=O)CCCC(=O)N1CCC(NC(=O)C=C(Cl)Cl)C1C1CC1 84459,C1(NC(c2cc(C(=O)OC)sc2)=O)CS(=O)(=O)CC1NC(c1c(Cl)cnn1C)=O 84460,c1(CNC(CC2N(C(c3c(OC)cncc3)=O)CCOC2)=O)cc(F)ccc1Br 84461,N1(Cc2n(C(CC)C)ncc2)CCN(C(C(=O)OC)C(C2CC2)C2CC2)CC1 84462,CS(=O)(=O)C1CC(C(=O)NCC2CCN(C(=O)CC3C=CCC3)C2)C1 84463,C1(C(C(C)C)NC(c2c(C(=O)OC)csc2)=O)CCN(C(=O)COCCO)CC1 84464,C(=O)(C1CC(=O)c2c(F)cccc21)NC(CNC(Cc1c(C)cccc1Cl)=O)C 84465,c1(SCC)c(OCCC(=O)OC)cccc1Br.n12nnnc1C(C1CC1)NCCC2 84466,C1(NC(CC2C(C)(C)C(O)C2)=O)CC(N=c2ccn3nccc3[nH]2)C1(C)C 84467,N1(C(c2ccc(C#C)c(Cl)c2)=O)CC2(C)CN(C(=O)CC(C)SC)CC2(C)C1 84468,N1(CC(=O)NCc2onc(C)n2)CCCC(n2cc(Nc3ncccn3)cn2)C1 84469,c1(C(=O)NC2CN(C(COCCC)=O)CC(C)C2)cc(Cl)cc2c1NCCC2 84470,C(C(=O)NC1CC(CNC(=O)C(F)OC(F)(F)F)C1)(C(C)C)NC(C)=O 84471,c1(NCCCN2CC(C)OCC2)ccc(O)c(-c2ccc(Cl)cc2)c1 84472,C1(OC)CC(CCNC(C23CC(NC(C)=O)(C2)C3)=O)N(C(=O)CC(C)F)C1 84473,C(=O)(C(CNC(=O)C1=CCCC1C)C(C)C)NC(COC)(C)C(N)=O 84474,CN1CCn2ncc(C(=O)NC3(C)CCCN(C(=O)COCC(C)(C)C)C3)c21 84475,N1(C(c2ccc(N)cc2F)=O)CCC2(NC(=O)CC3=CCCC3)CCCCCC12 84476,C1(C(=O)NC2C=CCN(C(Cc3scc(C)c3)=O)C2)CCc2cnnn2C1 84477,Cc1ccc(C(N2CCC(CCF)CC2)C(=O)NCC(F)F)c(O)c1 84478,CC1CC=C(C(=O)N2CCN(C(c3cccc(Cl)c3F)=O)CC2CC(F)F)CC1 84479,c1(C(=O)NCC(=O)NC2(CCNC(=O)CC3CSC3)CC2)ccccc1 84480,CN1CCCC(CC(=O)NCC2CC2NC(C2(C(N)=O)CC2)=O)C1 84481,c1(C(=O)NC2CC(NC(c3cc(C)c(Br)s3)=O)C2)cccc(Br)c1O 84482,N1(C(C(Cc2c(C)nc[nH]2)O)=O)CCC(NC(=O)CCCCCN(C)C)C12CC2 84483,O=C(C1=CS(=O)CCC1)NCC1CC(F)(F)CN1C(=O)Cn1cc(Cl)cn1 84484,N1(C(c2c(CC)cco2)=O)CC(NC(c2ccc(Cl)[nH]2)=O)C2(CCOCC2)C1 84485,N1(C(C)=O)CCCC(NC(C2CCCNC2)=O)C1 84486,c1(CC)ncccc1NC(=O)CC1CCCN1C(c1cncc(Br)c1)=O 84487,c1(C(=O)NCC2CCN(C(CC(n3ccc(C)n3)C)=O)C2)cccnc1C 84488,CC1=C(C(=O)NCc2ccnc(C(=O)NCC3COCC3(C)C)c2)SCCO1 84489,C12C=CC(C1)CC(=O)N2CC=CC1CC1.CC(C)C(=O)NC(C1CCCO1)(C)C 84490,c1(C(c2nnnn2Cc2c(OCC)cccc2)SC)cc(Cl)ccc1[N+](=O)[O-] 84491,C(CC1CCOc2ccccc21)N(C1CCN(c2cc(C)ncn2)CC1)C(C)=O 84492,c1(OC)cccc(C2CCN(C(=O)CNC(=O)CC3CCC4CC34)CC2)c1 84493,c1(C(=O)NC2CCN(CCNC(CC(C=C)C)=O)CC2)c(F)ccc2n[nH]cc12 84494,C1(C(C)C)CN(C(C2CS(=O)(=O)C2)=O)CCN1C(C1CC(=O)C1C)=O 84495,C(=O)(C(C)(C)C(=O)N1CCC(C(CO)NC(=O)C(C)c2cc[nH]n2)CC1)OCC 84496,c1(C(N2C(CC)C(NC(=O)Cc3ccoc3)CC2)=O)coc2ccccc12 84497,c1(C(=O)NCC(CC=C)NC(=O)C(C)(F)CCCC)cnc2c(ccn2C)c1 84498,N1(CCCC(=O)NC2CC(NC(C(C3CCOC3)OC)=O)C2)Cc2ccccc2C1 84499,c1(C(N(C)CCNC(=O)C(=O)N(CC(F)(F)F)C)=O)ccc2c(c1)CC(OC)C2 84500,N1(C(C2(C=C)CC2)=O)CCC2(CCC2NC(c2ccc(C)nc2)=O)CC1 84501,C=CC1(C(=O)NCCCCCN(C(=O)Cc2csc(Cl)c2)C(C)C)CCC1 84502,C1(NC(Cc2c(C)noc2)=O)CCCC(NC(=O)C(C)C=Cc2ccccc2)C1 84503,C1(C)(CCC(=O)NC2CCC(CNC(CCC)=O)C2)CCC(=O)N1 84504,C1(C(=O)NC2CC2(F)F)CC2CC2N1C(C1CCCCC1C(F)(F)F)=O 84505,c1(CCNC(C(C)N(C(C2C(CC)C2)=O)C)=O)ccnn1C 84506,c1(C(=O)NC2CC(NC(c3ncnc4sccc34)=O)C2)ccc2cc[nH]c2c1 84507,c1(C(N(CCCNC(c2cc(C)nnc2)=O)C)=O)ccc2[nH]c(=O)c(=O)[nH]c2c1 84508,c1(C(=O)NC(CC)CN(C(C23CCC(F)C2CC3)=O)CC)nc(O)nc(O)c1F 84509,C1(C)(NC(CCC2C(C)=NOC2=O)=O)CCCN(C(=O)CC(C)c2ccco2)C1 84510,C(N=c1[nH]cncc1Br)C1OCC(CNC(C(C(CC)C)O)=O)C1 84511,Cc1ccc(C)c(C(N2CC(N3CCN(C(C4CC4C#N)=O)CC3)C2)=O)c1C 84512,N1(C(C2CCC(=O)N2)=O)CCN(C(=O)Cc2cc(Cl)ccc2Cl)C(CCO)C1 84513,Cc1cc(C(=O)N(C)CC2CN(C(c3ccc(Cl)cn3)=O)C2)c(C)cc1Br 84514,C1(NC(CC=C)=O)CN(C(C2CCN(C(C)C)CC2)=O)CC12CCC2 84515,c1(C(=O)NCC(N(C(c2cc(C)ncn2)=O)C)C2CC2)ccc(Cl)cc1O 84516,C1(NC(CCCSC)=O)CCCC2CN(C(C3CCC(C)(C)O3)=O)CC12 84517,CC1CC(NC(=O)Cc2cc(F)cc(Cl)c2)CCN1C(c1cnc(Cl)n1C)=O 84518,C1(CNC(c2ccc(CSC)o2)=O)CCCCC1NC(=O)CCc1n[nH]c(=N)s1 84519,C1(C(=O)NC(CC)CCC(=O)NCCOCC(F)(F)F)C2CCC3C(C2)CC13 84520,c1(C(N2C(CCCNC(C(CCSC)N(C)C)=O)CCC2)=O)cnc2sccc2c1 84521,C12(CNC(c3cc(C(CC)CC)no3)=O)CC(C1)C(NC(C1(Cl)CC1)=O)CO2 84522,C1(CC(=O)NCCOCCC)CC2(C1)CN(C(=O)Cc1cc(C)[nH]n1)C2 84523,CCC(C)C(C(=O)NC1CCN(C2CC2)C1)N(C)C(c1sccc1F)=O 84524,C1(CC)CN(C(=O)C(O)C(C)C)CCC1NC(=O)C(C1(O)CCOCC1)(F)F 84525,N1(C(CCc2ccn(C)c2-c2ccccc2)=O)CC(S(C)(=O)=O)C1 84526,N1(C(C2CC(NC(c3ncc(C)[n+]([O-])c3)=O)C2)=O)CC2CC3CC2C1C3 84527,C1(CNC(c2c(CC)ncs2)=O)CN(CC(CC)CC(C)C)CCC1(F)F 84528,Cc1cn2c(n1)CC(C(=O)NCC(O)CNC(C1CCC(=O)N1)=O)CC2 84529,c1(OCCC)cc(OC)ccc1CC(C1CCN(C(=O)C(C(C)C)OCC)C1)C 84530,C1(CNC(C2CC(C#N)C2)=O)CCCN(C(=O)Cn2cnc(C(N)=O)n2)C1 84531,N(C(=NCCF)NC1CCCC(Cc2n(C)cnn2)C1)C.OC(F)F 84532,c1(CN2CCC(=CC(N3CCC(Br)C3)=O)CC2)ccc(-n2cccn2)c(F)c1 84533,CCCC(C(=O)NCC(CNc1ccc(Cc2nnc(C)o2)cc1)OCC)OC 84534,C1(OC)(CNC(c2ccccc2)c2nnnn2C2CCCC2)CCCCC1 84535,n1(CCC)cccc1NC(=O)NCc1ccn(CCF)n1 84536,C(=O)(CCC(C)S(C)(=O)=O)NCC1(F)CCN(C(c2nc(CC)oc2)=O)C1 84537,C1(NC(N2CCC2CC)=O)CC12CCN(C(c1cnncc1OC)=O)C2 84538,C1(S(C)(=O)=O)(C(=O)NC(CNC(C(CC)(C)OC)=O)C)CCOCC1 84539,c1(C(N(C)CC2CCN(c3nnc(C(N)=O)s3)C2)=O)cc(Br)cc2ccccc12 84540,N1(C(CCC2OCCN(C)C2)=O)CCN(C(C2(S(C)(=O)=O)CCC2)=O)CC1CO 84541,N1(C(C(C)OC)=O)CCCN(C(c2cnn(-c3ccccc3)c2F)=O)CC1 84542,C(=O)(C1=CCCC1C)NC1CCC(NC(C(c2ccc(F)cc2C)OC)=O)(CO)C1 84543,C1(NC(CNC(C=C(CC)CC)=O)=O)CCOCC1 84544,c1(C(N(C2CCN(C(C(CC)N(C)C)=O)CC2)CC)=O)ccc2occc2c1 84545,N1(CCN(C(C(CN(C)C)NC(CCOC)=O)=O)C)CC(C)(C)OC1=O 84546,C=CC(CCC)CC(=O)N1CCC(C)(NC(c2cc(S(=O)(=O)NCC)c[nH]2)=O)C1 84547,c1(CC(=O)NCC(C2CC2)NC(C(C)(O)C2CC2)=O)ccc2c(c1)OCCCO2 84548,N1(C(C=CC(CC)C)=O)Cc2[nH]nc(C(=O)NCCOC3CCOC3)c2C1 84549,C1(OC)CC(CCNC(=O)C(C)(C)CSC)N(C(=O)CN2CCCOC2=O)C1 84550,NC(=O)CCCC(=O)N(C)CC1CCC(CNC(C23C(=O)C4CC2C3C4)=O)CC1 84551,C=CC(C)(CC)NC(C1CC(NC(=O)C(C)N2CC(C)C2)C1)=O 84552,c1(N(C)Cc2c(C)nc[nH]2)nc(=NCCCCCO)[nH]c2c1SCC2 84553,C(C(CC(F)(F)F)NC(C1(c2cc[nH]n2)CCC1)=O)NC(=O)Cc1cn[nH]c1 84554,C(C)(CC(=O)NOCC(O)C(C)C)NC(CC1CC(C)C1)=O 84555,c1(C(N2C3C(CNC(c4cc(OC)no4)=O)C(C3)C2)=O)cc2n(n1)C(C)CCC2 84556,C(=O)(C#CC1CCOCC1)N1C(C(N2CC(C=C)C2)=O)CN(C)CC1 84557,C1(OC)CN(C(c2ccn(CC(C)C)n2)=O)C(C)(CNC(=O)CCC(C)(F)F)C1 84558,C(=O)(C1=CCN(C(C23CCC(CC2)CO3)=O)CC1)NCC(C1CCCCC1)C 84559,c1(OC)cnc(F)c(C(=O)NCC(C)(CNC(C2OC(C)CC2C)=O)OC)c1 84560,N1(C(c2cc(OC)c(C)cc2)=O)CCOC2(CCN(c3nnnn3C)C2)C1 84561,N1(C(c2n(C)nnc2)=O)CCC(C2CCN(C(c3cc(O)nc(Cl)c3)=O)CC2)C1 84562,c1(C(=O)NCC2N(C(C#CC3(C)CC3)=O)CC=C2)cc2c(F)ccc(Cl)c2[nH]1 84563,C1(NC(c2cnc(C)nc2)=O)C(C)(C)C(NC(=O)CC2CC2(Cl)Cl)C1(C)C 84564,c1(C(N(C)CCOCCNC(C2(CO)CCCC2)=O)=O)c(Cl)cccc1[N+](=O)[O-] 84565,C1(CNC(c2c(OC)csc2)=O)COC(C)(C)CN1C(C12CCCC1C2)=O 84566,c1(C(=O)NCC(CC)NC(c2nc(OCC)oc2)=O)cnc(CC)nc1 84567,N1(C(CC2N(C(c3ccc(C(N)=O)[nH]3)=O)CCC2)=O)CCSC2CCC12 84568,CCCCC(C(=O)NCCC(C)OC)NC(=O)COC1CCOC1 84569,C(CC(C)(C)C(=O)N1CCN(C(=O)CCCNC(c2ccsc2)=O)C(C)C1)OC 84570,c1(CC(=O)Oc2nccn2CC(F)(F)F)cnc(C2CCC2)o1 84571,C1(C(=O)NC2CCC(NC(=O)Cc3cccc(Cl)c3Cl)CC2)CCC2CC1CO2 84572,N1(C(CNC(c2[nH]cc(C(=O)OC)c2)=O)C=O)CCC(CCN(C)C)CC1 84573,CC1(C)C(C(=O)NCC(C)(C2CC2)NC(c2cc(F)cc(F)c2)=O)CCS1(=O)=O 84574,C1(C(=O)NCCn2c(CC)nnc2S)CNC(=O)CN1C(=O)C(CO)N(C)C 84575,Cc1cc(CN(C(N2CCCCC2c2ccc(C(F)(F)F)cn2)=O)CC)cc(C)c1 84576,Cc1c(CN=C(NCc2ccsc2S(C)(=O)=O)NCC2CC2)cccc1Br 84577,C1(NC(Cc2c(C)non2)=O)CCCC2CN(C(c3cnc(S)[nH]3)=O)CC12 84578,C1(C(=O)NC(C2CN(C(=O)CCCn3cccn3)C2)C)CCc2cnn(C)c2C1 84579,Cc1cc([N+](=O)[O-])cc(C(=O)NC2CCN(C(=O)C#CC3CCCC3)C2)c1Cl 84580,C#Cc1ccc(F)c(C(N2CC(C)C(NC(=O)CC3CS(=O)(=O)C3)C(C)C2)=O)c1 84581,c1(OC)cccc(CCN(C2CC(O)C2)C(C2CCN2)=O)c1Cl 84582,C1(CCC(=O)NCCNC(C(C)NC2CN(CCC(C)C)C2)=O)CCCC(=O)N1 84583,n1(C(C)C)cc(C(=O)NCCOCCCNC(C2CCCS2)=O)cn1 84584,C1(C(=O)NC(C2CCCN2C(=O)C=CC(F)(F)F)(C)C)CCC(=O)NC1 84585,C1(C#N)(C(N2CC(CN(C(c3c(C(C)C)con3)=O)C)OCC2)=O)CCCCC1 84586,c1(C(=O)OC)nn(C)nc1C(N1CC(NC(C2CN(C)C(=O)N2)=O)CC1C)=O 84587,CCC(CC(=O)N1CC(CC(N2CCCC(C(N)=O)C2)=O)(OC)C1)SC 84588,N1(C(C2C(=C)CC2)=O)CC(C2CCCCN(C(C3CCC([N+](=O)[O-])CC3)=O)C2)C1 84589,C1(C(C)C)CC(N=c2[nH]c(=NC(CF)c3cccnc3)[nH]c3c2COCC3)C1 84590,C(CSC)(C(=O)NCC=C(C)C)NC(CN(CCC)C)=O 84591,N1(C(Cc2c(C)nc(-c3ccc(F)cc3)s2)=O)CCS(=O)C(C)(C)CC1 84592,C(=O)(CC1=NNC(=O)C1)N1C(C(=O)NCC2CCC3CC3CC2)CC(OC)C1 84593,N1(C(CCCCCCC(=O)O)=O)C(C=O)C2CC(O)C1C2.N1(CC)C2CSCC1C2 84594,C(CCC)(CCCNC(c1ccn(CCF)n1)=O)NC(C(CC=C)NC(C)=O)=O 84595,c1(C(=O)NC(CC)CN(C(=O)CCC(C)C)C)cccc(F)c1C#N 84596,N1(c2snc(C)c2C#N)CCC2(NC(=O)CCCN3CCCC3)CCCCCC12 84597,c1(CC(=O)N(CC(CC)NC(C2C3CN(C)CC23)=O)C)c(C)[nH]c2ccccc12 84598,N1(Cc2cc(OC)ncc2Br)CC2CCN(C(c3nc(C)cs3)=O)C2C1 84599,c1(C(=O)NCC(C(CC)CC)C)cc(-c2nc(N3CCOCC3)no2)ccc1F 84600,n1(CC(=O)N(CCCN(C)C)C)cnc(C(=O)N)n1.C1(C(=O)OC(C)(C)C)CCO1 84601,c1(C(=O)NCC(C)NC(c2oc(Br)nc2C(F)F)=O)cn2ccccc2n1 84602,N1(C(COCCC=C)=O)CCC2(C1)CN(C(C1(C)CCN(C)CC1)=O)CCO2 84603,N1(C(C2(C)N(C(C(CC)CN(C)C)=O)CCC2)=O)CCC(CO)C12CC2 84604,C1(CC)COCCN(C(C2CCN(C(=O)Cc3cc(C)cc(C)c3)CC2C)=O)C1 84605,C1(NC(C(CC)c2ccccc2)=O)CCC(NC(=O)C(C)(C2CC2)OC)CC1 84606,c1(CCCCC)nc(C(=O)NC2CC(NC(=O)CC3C=CCC3)C2)cs1 84607,C1(C(=O)NCCc2c(C)nn(C)c2)CCN(C(=O)OC(C)(C)C)C2COCC12 84608,C1(CCN(C(CCOC)=O)C)CCN(C(C2C3CC4C(C3)C24)=O)CC1 84609,N1(C(CN(c2ccccc2Cl)C)=O)CCCC1(C)C(=O)OCc1cnsn1 84610,c1(C(N(CCNC(c2c[nH]nc2Br)=O)CC)=O)nccc(OC)c1N 84611,N1(C(c2nccc(NCC)c2)=O)CCC(C2CCN(C(C3CC3(F)F)=O)CC2)C1 84612,c1(COC(C(N(C)C)NCC)=O)c(C)nn2cc(C(F)(F)F)cnc12 84613,C(=O)(C(C)C(O)C(C)C)N(C1CC(C#N)C1)CC(=O)NC(C#C)CC1CC1 84614,C(=O)(C(CNC(C1CCCC1O)=O)C(C)(C)C)NCCSC 84615,C1(CC(=O)NC2CCC(NC(c3c(C)n(C4CC4)cc3)=O)C2)CCC(=O)NC1=O 84616,N1(C(c2c(C)oc(Cl)n2)=O)CC(CNC(=O)CCc2cccn2C)CC(C)(C)C1 84617,c1(-c2nc(CCCCCC)nn2CCN(C2CCOC2)CC)ccc(Cl)c(Cl)c1 84618,C=CCC(CO)NC(=O)C(C)CNC(=O)CCC1CC1C 84619,N1(C(c2c(CC)scc2)=O)CC(C)(C)OCC1CNC(=O)C(c1ccc(C)o1)C 84620,C=CC(CCC)CC(=O)NCCOC1CN(C(c2cn3ccnc3s2)=O)C1 84621,c1(NCc2c(O)nnc(C)c2C)nc(NCC(C)CC(C)O)c2c(n1)c(C)nn2C 84622,C1(C(=O)NCC(CC)N(C)C(C2(C)CCCOC2)=O)CCC12CCC2 84623,N1(C(C2N(C)CSC2)=O)CC2(CNC(=O)C(F)C3CCC3)CC1CO2 84624,N1(C(c2[nH]cc(C(N)=O)c2)=O)CCCC(CNC(c2ocnc2C(F)(F)F)=O)C1 84625,C1(CNC(C(C)SC)=O)CC2CCCC2N1C(=O)COCCOCCO 84626,N1(C(c2csc(C)c2N)=O)CCC(NC(C2CCC(C(N)=O)N2C)=O)CC(O)C1 84627,C1(C(=O)NC2CC(NCc3c(C(=O)OC)c[nH]n3)C2)COCCN1C1CCCC1 84628,c1(C(=O)NC(C)CNC(c2cnc(Cc3ccccc3)o2)=O)csc2nnsc12 84629,CCC(C(=O)NCC1(C(=O)N(C2(C)CC2)C2CC2)CC1)n1ccnc1 84630,Cc1sc(N)c(C(N2CC(C(N3CCC(F)(C(C)C)CC3)=O)OC(C)C2)=O)c1C 84631,N1(C(c2cccc(CC)c2F)=O)CC2(CCCN(C(c3cccc(Br)c3)=O)C2)C1 84632,N1(C(C(C2CCOCC2)OCC)=O)CCN(C(c2cc[nH]c2)=O)C2COCC12 84633,N1(C(CC)=O)CCCC(C2(NC(=O)CCCCCF)CC2)C1 84634,Cc1n[nH]cc1CNC(=O)C=CCC1(NC(=O)CCn2ccnc2)CCC1 84635,C12(CNC(CC3CC(=C)C3)=O)CC1CN(C(C13CC(c4ccccc4)C1C3)=O)C2 84636,c1(OCC)ccccc1C(C)N(C(c1csc(SC)c1)C(=O)NC(C)C)C 84637,c1(CC)nn(C)c(C(N2CC(NC(c3cnc(C(C)(F)F)s3)=O)C(C)C2)=O)c1Cl 84638,c1(C(N2C(CNC(C(C)CN(C)C)=O)CC3(CC3)C2)=O)cc2cc(N)ccc2[nH]1 84639,c1(C(=O)NC2CCCCC2CNC(=O)CC(F)(F)Cl)ccc2occc2c1 84640,Nc1ccc(Cl)c(C(=O)NCC2CC(NC(=O)CCc3cnoc3)C23CCC3)c1 84641,N1(C(Cn2cc(-c3n(CCC(C)C)ncc3)nn2)=O)CCCC(O)C1 84642,CC1(C)NC(=O)N(CC(=O)OC2C3CCC2(C(F)(F)F)C3)C1=O 84643,S1(=O)(=O)c2cc(ccc2OC)N1.C1(CC#C)CN(C(=O)OC)CCO1 84644,c1(SCC#C)cccc(C(=O)NC2CCC(NC(=O)CN3CCCC(C)C3)C2)c1 84645,N1(C(C(CO)N(C)C)=O)C2CC=C(C(=O)NC3CCC4(CCCC4)C3)C1CC2 84646,C1(NC(Cc2cc(C)no2)=O)CN(C(c2cc(O)ccc2C)=O)C(C)(C)C1 84647,CN=c1cc(C)nc(N2CCc3c(cnnc3O)C2)[nH]1.C1(OCC)(O)CCOCC1 84648,c1(CN2CCN(C(=O)CCNC(C3CC34CC4(F)F)=O)CC2)ccc(F)c(F)c1 84649,N1(C(=O)CSc2cscn2)CCN(C(C23CC4CC2C3C4)=O)C2CC12 84650,CCN=C(NCC1CCCC1OC)NCCC1CCN(C(=O)NC)CC1 84651,C1(C(=O)NC2CCN(C(C3CC(n4cnnc4)C3)=O)C2)CCC2(CC1)CC2(F)F 84652,C1(C(=O)OC)CN(C(=O)C(C2CCC2)NC(c2c[nH]nc2C)=O)CC1F 84653,c1(NCC(CC)O)cc(Br)ccc1OC(F)F 84654,C1(CC)C(=O)NCCN1C(C1CCCN1C(=O)CCCc1cnn[nH]1)=O 84655,CCCC(C)C(C)(c1nnnn1CC1CC1)NCc1sc(Br)cc1C 84656,c1(N2C3CN(C(c4cc(C)[nH]c4C)=O)C(C3)C2)ncnc2c(F)cccc12 84657,C1(NC(c2c(Br)cn(C)n2)=O)CN(C(c2ocnc2C2CC2)=O)CCC1F 84658,C1(CC)C(C(=O)NCCS(=O)(=O)NC)CCN1C(c1cccc(OC)n1)=O 84659,S(=O)(=O)(c1cccc2c1OCCO2)Nc1ccc2c(c1)N(C)CC2 84660,C=CC1OCCCC1C(=O)NCC1CN(C(=O)CNC(=O)CC)CCC1C 84661,C(C(C(=O)NCC1(O)CC(C(N)=O)C1)NC(=O)C(O)C1CCCC1)OC(C)C 84662,C(C(C)C(=O)NC(CN(C)C)C(=O)NCCCNC(C)=O)OCC 84663,Cn1nc(CC(=O)NCC(C)(C)NC(C2C(Cl)(Cl)C23CC3)=O)cc1Cl 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84976,CC(CC(C)(F)F)C(=O)NCC1CN(C(=O)CC(F)(F)C(F)F)CCO1 84977,c1(OC)ccc(C(=O)N(C(CNC(=O)C(C)(CO)OC)C2CC2)C)c(OC)c1 84978,CN1CCCC2CN(C(c3ccnc(Cl)c3Cl)C(=O)NC3(C)CC3)CCC12 84979,C1(CNC(C2C(C)(C)C2)=O)CCCCN1C(=O)Cc1cnsc1 84980,N1(C(c2c(OC(F)F)cc(C)s2)=O)CC2CCC(C1)N2C(=O)CCc1cnn[nH]1 84981,CC1=C(C(=O)NC2(C(=O)NC3CC4CCC(C3)N4C)CCCCC2)SCCO1 84982,C(=O)(C1=CCC2CCC1N2C(c1cccs1)=O)Nc1c(C)n(C(C)C)nc1 84983,C1(C(=O)NC2CC(OCC(=O)NCC3=NOCC3)C2)CC2CCC(C1)O2 84984,c1(C(N2CC(CC(C)NC(CCCC=C)=O)C2)=O)ccc(F)c(C2CC2)c1 84985,Cc1cc([N+](=O)[O-])cnc1C(=O)N(CC(C)O)CCNC(c1c[nH]c(=N)s1)=O 84986,N1(C(c2c(Cl)cc(C)nc2)=O)CC2CC(NC(=O)C(C)(C)c3ccns3)CC2C1 84987,C1(C2CCN(C(C3CC3C)=O)CC2)(NC(c2cc(C)cc(Br)c2N)=O)CC1 84988,N1(C(CCCCNC(C(CC(=C)C)OC)=O)=O)CCN(C)C(C)C1C 84989,CC1CC(NC(c2cc(C(F)(F)F)c[nH]2)=O)CN1C(c1snc(O)c1Cl)=O 84990,c1(C(N(CCCNC(=O)Cc2cc(C)on2)CC)=O)ccnc(CO)c1 84991,C1(NC(C2C(C)C2C)=O)CCC(NC(C2CC(O)C2)=O)C1 84992,Cc1ccc2c(c1)CC(NC(=O)NCC(=O)NC1CC1(C)C)S2 84993,c1(C(=O)NC(C(C)NC(N)=O)CO)ccc(NC(C2CCC2C(=O)N(C)C)=O)cc1 84994,C(=O)(C(CC1CC1F)N(C)C(C1CCCC1)=O)OCC.C1(=O)C(C)(C)N1.C(C)(C)(C)O 84995,CCC(F)(F)C(=O)N1CCC(N(C(=O)CN2CC=CC2)CCOC)CC1 84996,c1(C(=O)NC2CC(C)(CNC(CCCOCC)=O)C2)ccc2[nH]cc(C#N)c2c1 84997,CCC(C)C(C)(O)CNC(=O)CC1CCCCN1C(=O)CN(C1CC1)CC 84998,C1(CNC(c2cn(CC=C)nc2)=O)CN(C(c2cnn3c2CCC3)=O)CCN1C 84999,c1(-c2cc(OC)c(F)cc2)cc(C(=O)NCCOC2CCCC2)c2cc[nH]c2c1 85000,c1(C(N2C(C(=O)NCc3ccncc3Br)CSCC2)=O)ccc(O)cc1O 85001,C1(C(N2CC(N(C(C3=NOC(C)C3C)=O)C)C2)=O)COC2(CCC2)CO1 85002,CC1=C(C(=O)N2CCC3C(NC(=O)Cc4cc(C(F)(F)F)c(O)nn4)C23)CCO1 85003,C1(C(N2C(CNC(C(CCC)C#N)=O)C3CCC2C3)=O)CCc2nnnn2C1 85004,c1(OC)ccnc(F)c1C(=O)NCC1CCN(Cc2cscn2)C1 85005,C(CC(C)(C)C(=O)N1CCC(C)C(CC(=O)NC2(C(C)O)CC2)C1)OC 85006,c1(OC)cccc(C(F)(F)CNC(=O)NC(C)CCNC(C)=O)c1 85007,S(=O)(=O)(CCC(=O)NCCCC(C)NC(=O)COCC1CCCO1)NC 85008,CC1(C)CC(NC(C2(N3CCOCC3)CCC2)=O)CN1C(=O)C(F)C(F)(F)F 85009,C#CCCC(C(=O)OC)NC(c1ccoc1CNC(=O)C(O)CCC)=O 85010,c1(CC(=O)NCC(=O)N(C(C)C(=O)NC2CC2)C)cn(C2CC2)cn1 85011,C1(CC(=O)NC2CCN(C(c3ccc(CCC=C)cc3)=O)C2)CC(F)(F)C1(F)F 85012,C1(CCC)CN(C(C2(Cl)CC2(C)C)=O)CCN1C(=O)C=CBr 85013,N1(C(CN(C(=O)C(=O)Nc2ccccc2)C2CC2)=O)CC2CCC(CO)(C2)C1 85014,N1(C(c2cc(CC)cc(N)c2)=O)CC2(CCCC2NC(C2CCOC(C)C2)=O)C1 85015,C(=O)(C(C)S(=O)(=O)C1CCOCC1)NC1(C)CCC(NC(c2cnc(C)s2)=O)C1 85016,c1(CC(=O)NC2C(C(=O)NC(C)CC3CCC3)C2)ccc(F)cc1F 85017,N1(C(c2c(C)oc(C3CC3)c2)=O)CCCC(c2ccccc2)CC1 85018,c1(NC(=O)NC)ccc(C2=CCN(Cc3cc(N4CC(C)OC(C)C4)ncc3)CC2)cc1 85019,C(=O)(C(CCF)NC(=O)CCOC1CC1)N(CCCCC)C 85020,N1(C(C2(CNC(CNC(=O)OCC)=O)CCCO2)=O)CCC(F)(F)C(F)C1 85021,CC1CCC(C(N2CCCCC2)=O)CN1C(C12CCCN1CCC2)=O 85022,CC1OC2(CNC(C3CCCC(=O)N3)=O)CC1(NC(=O)C=Cc1cocn1)C2 85023,CCC(O)CNC(=O)C(=O)NC(COC)C1(C)CC1 85024,c1(CC)[nH]c(=N)sc1C(N1CC(NC(=O)Cc2ccnc(F)c2)C(C)C1)=O 85025,Cc1cc(NC(C2CCCCN2C(=O)NC(c2nn[nH]n2)C)=O)ccn1 85026,C(CC(C)C(=O)N1CCCC(NC(C2(CCS(N)(=O)=O)CCC2)=O)C1)=CC 85027,Cc1nc(-c2cccs2)c(CCNC(N2CC(F)CC2c2ccccc2)=O)s1 85028,Cc1ccc(C(=O)NCCC(C)N(C(=O)C(Cc2ccsc2)C2CC2)C)c(Cl)c1 85029,c1(C(N2CCC(C(C)NC(C(C)CO)=O)CC2)=O)ccc(O)c(Cl)n1 85030,N1(C(C2(C)C(C)C2)=O)CC=C(CCNC(C2CCOC23CCC3)=O)CC1 85031,C#CC1(N(C(C2CC3(CCN2C(c2cccnc2)=O)CC3)=O)CC)CCCCCC1 85032,c1(C(=O)NC2CCN(C(CCC)=O)CC2C)c(Cl)nc2cc(Cl)ccn12 85033,c1(C(=O)NCCN(CCC)C(C2(C)CCOCC2)=O)ccc(C2(C)CC2)cc1 85034,c1(CNC(CCC)(C)CC)cc(OCC)cc(OC)c1 85035,c1(-n2c(CCN3CCCC3)nc(C(CC)C)n2)ccc2nccnc2c1 85036,N1(C(C(CC)(C)OC)=O)CCCCC2(CCN(C(C3(CCF)CC3)=O)C2)C1 85037,Cn1ncn(NC(=O)C2CCCCN2C(c2occc2C2CC2)=O)c1=S 85038,c1(C(=O)NCC(CCCC)NC(C23CCN(CC2)CC3)=O)cnc2nc(C)oc2c1 85039,C(=O)(CCCCCF)NCC1C(NC(c2c(CC)ncs2)=O)C1 85040,C1(C(=O)NCC=C(C)C2CC2)CC12CCN(C(=O)CCN1CCOCC1)CC2 85041,C(=O)(C1=C(Cl)CCC(C)C1)NCC1CC(NC(Cc2ccc(OC)cc2C)=O)C1 85042,Cn1nnc2c1CCN(C(=O)C(C1(C)CC1)NC(C1CCCOC1)=O)C2 85043,C(C)(C(=O)N1CCC(CN(C(=O)Cn2ncc(O)nc2=O)C)CC1)(C(C)C)SC 85044,C(=O)(CCN(OC)C(=O)C=Cc1cncn1C)NCC1(OC)CCOC1 85045,n1(CC(=O)NCCNC(=O)Cc2ccc3c[nH]nc3c2)ccc2ccc(Cl)cc12 85046,CC1CC(NC(c2ccoc2CNC(=O)C(C)(F)c2ccon2)=O)CC(C)C1 85047,N1(C(Cc2ccc(COC)cc2)=O)CCN(C(=O)CCc2ccccc2)C2CC12 85048,Cc1cnn(C(C)C)c1C(=O)NC1CC2(C1)CC2NC(c1c[nH]c(=N)s1)=O 85049,C1(NC(C2(F)C(C)C2)=O)CCN(C(=O)C(C)(C)c2cccs2)C1 85050,C(=O)(CCCCCCCCC1CC1)N(C)CCNC(c1nc(Cl)cs1)=O 85051,C1(C(=O)NCC(C)(O)C2CCC2)CSCN1C(=O)C=CCO 85052,N1(C(C=CC=CC)=O)CCC(C)C(CNC(c2cc(C3CCOCC3)[nH]n2)=O)C1 85053,c1(C(=O)NCCOCCN(C(C2C(C)CCO2)=O)C)ccc(F)c(F)c1O 85054,N1(C(C)=O)CCC(=CC(=O)NCC(=O)NCC=Cc2ccccc2)CC1 85055,C1(COCCNC(C(C2CC2)OCC)=O)(SC)CN(C(=O)Cc2c[nH]c(CC)c2)C1 85056,C(=O)(CN=S(C)(C)=O)NC(C(C)O)C(=O)NCCCCN1CCC1 85057,C(=O)(C(CC(C)C)C(C)C)NC1C(NC(CCCCC=CC)=O)C1 85058,N1(c2cc(OC)nc(C(F)(F)F)n2)CC2CC1CN(C(=O)CC(C)C(C)C)C2 85059,C12(C(=O)NC(C)CNC(C3CCSCC3)=O)CC(CO)(C1)OC21COC1 85060,N1(C(CCCC#CC)=O)CC2(CNC(C3CCCSC3)=O)CC1CCO2 85061,C1(CNC(C=CC=CC)=O)CN(C(c2nn(CCC)nc2Br)=O)C2CC12 85062,Cc1nc(C(=O)NCCC2CN(C(c3ccn(-c4ccncc4)n3)=O)C2)co1 85063,CC1(C)CCCCC1C(=O)NC1CC(NC(c2cccc(SC(F)(F)F)c2)=O)C1 85064,CC(CC(=O)NC1CCC(CNC(C2CCOCC2)=O)C1)C(C)(C)C 85065,c1(CC(=O)NC(C2CCN(C(CCCC(C)C)=O)C2)C)ccc2cnccc2c1 85066,c1(CC)ccc(NCc2nccn2C(C)C)o1 85067,c1(C(=O)NCCCNC(C2CC(CC)C2)=O)cc([N+](=O)[O-])cnc1N 85068,Cn1nc(Cl)c(NC(=O)OCc2ccccc2)c1CCCc1ccncc1Cl 85069,CC1CC(C(=O)NCC#CCCO)CN(C(=O)Cc2csnn2)C1 85070,CC1(C)CC(C(=O)NOC(C2CCCCC2)C(=O)NC2CC(C)(F)C2)C1 85071,C(c1scnc1C)=CC(N1C(C(CNC(Cc2c(C)nc[nH]2)=O)(C)C)CCC1)=O 85072,C1(CC)C(NC(c2ncnc(C)c2C)=O)CCCN1C(=O)C=CC(=O)NC1CC1 85073,N1(C(C(COC)NC(C)=O)=O)C2CCC1C(NC(=O)Cc1nc(=N)[nH][nH]1)C2 85074,C(C(CC1CCCC1)C(=O)Nc1snc(CC)n1)Sc1ccc(N2CC=CC2)cc1 85075,Cc1nc(C(=O)NC2CN(C(c3ccc4snnc4c3)=O)C2)ccc1[N+](=O)[O-] 85076,C1(CNC(c2c(C(C)C)nns2)=O)CN(C(c2cc3occc3s2)=O)CC1(C)C 85077,N1(C(COCCCCC)=O)CC(NC(=O)CSCCC)CC2COCCC12 85078,C=CCC(C)C(=O)NCC(c1ccccc1)NC(c1cc(CCC)cnn1)=O 85079,S(=O)(=O)(c1ccc(C(=O)NCC2(CNC(c3c[n+]([O-])c(C)cn3)=O)CC2)o1)NC 85080,Cc1scc(CNc2ccc(OCC(O)CN(C)C)cc2)c1C 85081,c1(C(N(C2CCN(C(C(CC)F)=O)C2)C)=O)cc(C(F)F)ccn1 85082,C(C(=O)NNc1ncnc2c1ncn2C)N1C(C)Cc2ccccc2C1 85083,CC1(CCNC(c2cnc3ccc(F)cc3c2)=O)CCOc2ccccc21 85084,c1(CC)c(OC)cc(C(=O)NCC2CCN(C(=O)C=CC(F)(F)F)C2)cc1OC 85085,CC(C)CC(=O)NCCC(C)N(C(=O)C(n1cc(Br)cn1)C)C 85086,c1(C(N2CCCCC(NC(C(C)CC3CC3)=O)C2)=O)cc(C#N)c(O)nc1N 85087,c1(OCCO)ccc(C(=O)O)cc1.o1[nH]c(=O)o1 85088,c1(C(=O)NCC(C)N(C)C(c2cn(C3CCCCC3)nn2)=O)cccn(C)c1=O 85089,C1(CNC(CC(CC)OC)=O)CN(C(c2cc(O)n(CC)n2)=O)C2COCC2O1 85090,C1(NC(c2scc(C)c2Cl)=O)CN(C(c2ccc(=N)[nH]n2)=O)C2CCCCC12 85091,C1(CCCC)CN(C(c2cnc[nH]2)=O)CCN1C(=O)CC(CC)C1CC1 85092,c12ccc(F)cc1NCC(c1n(CC=C)nnn1)N2.C(C(Cl)Cl)NS(C)(=O)=O 85093,CC1CC(C(=O)NCC2CCCN2C(=O)CCn2cccn2)CCS1(=O)=O 85094,c1(C(N2CC3C(NC(C(C)C)=O)(C3)C2)=O)[nH]nc2ncccc12 85095,N(C1CCCc2nc(C)sc21)CC(=O)N(CC(Cl)Cl)C(C)C1CC1.CO 85096,N1(C(C(C2CCC2)NC(C2CC3CC2CC3O)=O)=O)CC2CCC(C1)O2 85097,N1(c2nnc(CC)o2)CCC(NC(C2CCCOC2)=O)C1(C)C 85098,c1(C(=O)NC(C)CNC(=O)C(c2ccccc2)C)cccc(OC(F)F)c1 85099,c1(SC(C)C(=O)NCC2CN(C(=O)Cc3cccc(N)c3)C2)ccccc1Cl 85100,c1(SC)cc(N2CCCC(C(=O)Nc3ccc(-c4cc[nH]n4)cc3)C2)ncn1 85101,c1(C(=O)NCC(CO)NC(c2c(C)nc(CC)s2)=O)nc(C)n(C)c1C 85102,C1(C(N2CCC(CC=C)(NC(=O)CC(=O)OC)C2)=O)CCc2ccccc2C1 85103,C(CCCC(=O)N1CCCC(C(=O)N(CC(C)C)C(C)C)C1)OC 85104,c1(CCC(=O)NC2CC2C(=O)NCc2cc(F)cc(F)c2)ccc2c(c1)OCO2 85105,Cc1ccc(F)c(CNC(C2C(NC(=O)OC(C)(C)C)C2)=O)c1Br 85106,C(=O)(NN1CCCC1C(=O)NC1CCCC1C(=O)NC)C1C(CC)N(C)CC1 85107,c1(CCC)nc(=NCc2ccccc2Oc2ccc(F)cc2)s[nH]1 85108,c1(C(N2CCCC(C3(C)N=N3)C2)=O)cc2cc(C#N)ncc2[nH]1 85109,Cc1cnc(C(=O)N(C(C)CNC(c2cnc(-c3ccco3)s2)=O)C)c(Br)c1 85110,c1(C(N2CC(NC(=O)CC(C)C(C)C)CC(OC)C2)=O)cc2n(n1)CCN(C)C2 85111,C(=O)(CS(=O)C(F)(F)F)N(CCNC(c1c(C)ccs1)=O)CCOCCO 85112,c1(CC(N2CCN(CCO)C(CCO)C2)=O)ccc(F)cc1F 85113,N1(C(CC=C)=O)CC(C2CCCN(C(=O)C(C)(C)Cc3cccc(Cl)c3)C2)C1 85114,Cc1cc(C(=O)NC2(CCO)CN(C(C3CC(O)C3(C)C)=O)C2)c2n[nH]cc2c1 85115,Cc1n[nH]c(C)c1CC(C)C(=O)NCC(O)CN(C(=O)CSCC(N)=O)C 85116,C1(C(C(=O)NC(C)CCNC(=O)C(C)OCC(F)(F)F)=O)CCCCC1 85117,C(=O)(C(CC(C)(C)C)OC)N(C)CCOCCCN(C)C(C1COCOC1)=O 85118,c1(OC)cc(OC)cc(C(N2CC(C(C)NC(C3CCCC3(C)C)=O)C2)=O)c1 85119,N1(C(CC(CC)(C)C)=O)CCCC2(CCN(C(=O)Cn3cc(CO)nn3)CC2)C1 85120,C1(C(N2CCC2CC2CC2)=O)C(C2CC2)CCN1C(C1CCCCCC1)=O 85121,Cc1ncc(CC(=O)NC2CC(NC(C3(n4cnnn4)CC3)=O)C2)[nH]1 85122,c1(C(N2C(CNC(c3ccoc3Cl)=O)C=CC2)=O)cc(O)c2ccoc2c1 85123,C1(CN(C(C2(CCC)CCCO2)=O)C2CC2)CCN(C(c2[nH]ccc2C)=O)CC1 85124,c1(CC2(N)CC2)cnc(O)c(Cl)c1.c12ccc(o1)C(=O)NC2 85125,CC(C)(C)CCC(F)C(=O)N1CC(CNC(=O)C=C2CCOCC2)C2(CCC2)C1 85126,C(=O)(C(C)(C)CNC(=O)CC(C)CNC(=O)C(C)=C1CC1)NCC 85127,C(C(O)C(F)(F)F)NC(C1C(NC(C2CC(C)(F)C2)=O)CCC1)=O 85128,c1(C(=O)NCC2CN(Cc3scc(C)n3)C2)ccc(I)cc1Cl 85129,c1(CC)ccc(NC(=O)CN2CC(c3ccc(F)cc3)C(N)C2)cc1 85130,c1(SC)ncc(N)c(C(=O)NC2CCN(C(=O)CN(C)C(C)=O)C2)n1 85131,c1(NCC(F)(F)Br)nc(N2CCC3OCCCC3C2)c2ccccc2n1 85132,C(=O)(C(C(C)(C)C)SC(F)(F)F)Oc1cc(C(=O)NC(COC)OC)c(N)cc1 85133,CC1(C)CN(C(c2nc(Cl)ccc2F)=O)CCC1NC(=O)C1=CCC1 85134,c1(C(=O)OC)ccn2[nH]c(=NC(=O)C3(c4cccc(O)n4)CCC3)nc2c1 85135,Cc1c(Br)ccc(NC(C2CC(NC(c3ccc(C(C)(C)C)cc3)=O)C2)=O)c1F 85136,C=CC(CC(=O)NCC12CC(CN1C(=O)Cc1cncn1C)C2)c1ccccc1 85137,c1(OC)c(F)cc(C(=O)NCC2CC2NC(=O)C(F)C2CCC2)cc1Br 85138,C1(CNC(C2CC(SC)C2)=O)CN(C(c2ccnn2C(C)(C)C)=O)CC(C)(C)C1 85139,c1(C(=O)NC(C(C)NC(C(C)Oc2cccc(C)c2)=O)C)cc2scc(Cl)c2[nH]1 85140,CC(CC(=O)NCC12CCCC(CN1C(C1CCC(C)(C)O1)=O)C2)CC(F)(F)F 85141,CC(C)C(C(=O)NC1CN(C(=O)C=CBr)CC1Cc1ccccc1F)N(C)C 85142,C(CCCCCN=c1[nH]c2ccc(F)cc2o1)NC(C(CC)SC)=O 85143,C=CCC(CNC(c1c[nH]c(C(N)=O)c1)=O)NC(c1occc1C1CC1)=O 85144,c1(-c2cccc(C(=O)NCC(CCO)C(=O)O)c2)nc2ccc(O)cc2o1 85145,CCC(CC(=O)N1CC(C(=O)NCc2ncnn2CC)C2(CCC2)C1)C(C)(C)C 85146,N1(C(COCCCC)=O)CCC(C)(C)CC1C(=O)NCc1cc(C)nc(C)c1 85147,Cc1c(S(=O)(=O)N2CCC(O)(C(N)=O)CC2)sc2ccccc12 85148,c1(C(=O)NC2CN(C(CC(C)C3CC3)=O)CC2O)cc2c(cnn2C)nc1O 85149,N1(C(C(=O)N(C)C)=O)CCN(C(C2CCC3CC23)=O)C2(CC2)C1 85150,C1(NC(Cc2cc(COC)on2)=O)CCCCN(C(C2CCCC2C(F)F)=O)C1 85151,c1(C(N2CCC(NC(c3n(CC)nnc3)=O)(CO)C2)=O)c(OC)ccnc1O 85152,Cc1cn2cc(C(=O)NCC(CC(C)C)NC(=O)C(C)n3cnnn3)sc2n1 85153,Cc1cc(C)c2c(c1)CCCC2NC(=O)Nc1ccnn1CC(F)(F)F 85154,c1(-c2nccc(NCCN(S(C)(=O)=O)C)c2)c(N=[N+]=[N-])cnn1C 85155,Cc1cc(Cl)nc(N)c1C(N1CCCC(O)(CNC(=O)CC2CCCC2O)C1)=O 85156,c12ccccc1N2.C(C(C)(C)CNC(=O)C=C1CC1)N(C(COC)=O)C 85157,c1(C(=O)NCC(C2CC2)NC(C2(C)CCCS2)=O)ncn2c1CCC2 85158,c1(NCc2cc(C)ncn2)nc(N2CC3CC3(c3ccccc3)C2)nc2sccc12 85159,C1(C)(NC(c2ncn(C)c2)=O)CCN(C(c2nnc(C(F)(F)F)s2)=O)C1 85160,N1(C(C2N(C)C(=O)CC2)=O)C2CC=C(C(=O)NCc3n[nH]c4c3CCC4)C1CC2 85161,c1(C(N(C(CN(C(c2nc(C(C)=O)sc2)=O)C)C)C)=O)ccc2sncc2c1 85162,Cn1ncc(Br)c1C(N1CCC(c2cnn[nH]2)C1)C(=O)Nc1cccc(Cl)c1 85163,N1(C(CC(C)C)=O)CCCC(CN(C(=O)Cc2ccccc2F)C)C1 85164,N1(Cc2c(CC)noc2CC)CCC(NC(=O)CC2CCCCC2C)C(C)C1 85165,C#Cc1ccc(C(N2CCCC(CCNC(=O)C(C)CS(C)(=O)=O)C2)=O)cc1Cl 85166,C1(CNC(c2c(C)nc(O)[nH]2)=O)CCC12CCN(C(=O)Cc1csc(Cl)c1)CC2 85167,C1(CC(=O)NC2(C)CCN(C(C3CCCSC3)=O)CC2)CCC2(CC1)CCC2O 85168,Cc1cc(C(=O)NC2CC(NC(c3ccc(O)nc3C)=O)CC2O)cnc1C 85169,C=C(C)CN=C(NCc1ccccc1C)N1CCC2CCCCC2C1 85170,C1(C(=O)NC(CC)CN(C(=O)C(C)C)C)CC(c2cnn(C)c2)=NO1 85171,C1(ON=C(C)C(=O)OC(C)(C)C)CN(C(=O)C(C)(C#N)CC)CC1(C)C 85172,Cc1ccccc1C(=O)NC1COCC1CNC(C1(c2ccccc2)CCOC1)=O 85173,Cc1ccc(C(=O)NC2(C)CN(C(=O)CSc3cnn(C)c3)C2)nc1C 85174,N1(C(c2onc(COC)n2)=O)CCCC(C)C1CNC(c1cnn(C)c1Cl)=O 85175,Cn1ccc2[nH]c(C(N3CC(CNC(=O)NCCCCl)C3)=O)cc12 85176,N1(C(CCC=CC)=O)CCC2(CC1)CC2CN(C(C1CC(CC)=NO1)=O)CC 85177,N1(CC(=O)N(C(=O)CCSC)CCn2ccnc2C#N)CCCc2ccccc21.CO 85178,S(=O)(=O)(c1c[nH]ccc1=NCCn1ccc2ccccc12)N1C(CC)COCC1 85179,c1(C(N2CCCC(C(C)NC(COC(CC)(C)C)=O)C2)=O)cc(C#N)oc1C 85180,C1(C2NCCN(C)C2)CCC(F)(F)CC1.n12cc(nn1)C1CCCN1C(=O)C2 85181,C(CC(C)(O)C1CC1)NC(C=C(C)CSC1(C#N)CCC1)=O 85182,c1(C(N2C(CNC(C3(COC)CC3)=O)C3CCC2C3)=O)ccc2nc(=N)[nH]n2c1 85183,C(c1ccccn1)=C(C)C(=O)N(C1CN(C(C2C(C)(C)OC2C)=O)CC1F)C 85184,C1(NC(C=Cc2cnc(C)s2)=O)C(C)CCN(C(=O)CCS(N)(=O)=O)C1C 85185,Cc1cn2cc(C(N3CC(N(C(=O)C(N4CCC(C)C4)=O)C)C3)=O)sc2n1 85186,N1(C(C(C2CCOC2)OC)=O)CCN(CCNC(c2cnc(C)s2)=O)CC1 85187,c1(OC)ncc(C(=O)N(C)CC2CCCN(C(C3CC4(C3)CC4F)=O)C2)cc1Cl 85188,C=CCCCC(C)NC(=O)CC1CCCCN1C(=O)CSCCCC 85189,Cc1cc(C(N2CCC(C(C)C(=O)NC3CC3(C)C(F)F)CC2)=O)nn1C 85190,c1(C(N2CCCCC(CNC(COCC)=O)C2)=O)cc(C2CC2)nc2onc(C)c12 85191,CC(O)C(F)(F)C(=O)NC1CCN(C(c2ccc(Br)cc2)=O)C1 85192,C1(NC(C(C)(C)OCC)=O)CN(C(c2nc(CC)ncc2Cl)=O)CC2(CCC2)C1 85193,N1(C(C(CC#C)CC#C)=O)CC2(C1)CN(C(=O)COCC1CC1)CCO2 85194,N1(C(C2(NC(C(CC=C)C)=O)CCSC2)=O)CC2CN(C)CC2C1 85195,Cc1nc(C2CC2)nc(C)c1C(=O)NCC(F)CNC(C1CC1(Cl)Cl)=O 85196,C1(C(=O)NC2CCCC(NC(=O)CCCC3CC3)CC2)CCn2nnnc2C1 85197,C(=O)(C(CO)C(C)(C)C)N(C)CC1CCN(C(C2(OCC)CCCC2)=O)C1 85198,C1(CNC(C2(CC=C)CC=CC2)=O)CCCN(C(=O)CC2C(C)C2C)CC1 85199,C12(NC(C(C)CF)=O)CCCC1N(C(c1ccnc(S)c1)=O)CC2 85200,c1(C(=O)NC2CN(C(CCN(CC)CC)=O)C3C2C3)cc([N+](=O)[O-])cnc1O 85201,C(C(CNC(C1OCCC1(C)C)=O)S(C)(=O)=O)NC(C1(CO)CC(C)(C)C1)=O 85202,N1(C(c2c(C)con2)=O)CCCC(C2CCCN2C(C2(CC3CC3)CC2)=O)C1 85203,C(CC(C)C(=O)N(C1CCCN(C(=O)COCCc2cccc(F)c2)C1)C)OC 85204,C1(NC(C)=O)CC2CC(NC(C3(CC(N4C(CO)CCC4)=O)CCC3)=O)CC12 85205,CCCC(C)(CCC)C(=O)N1CC2(CCN(C(c3[nH]nnc3C)=O)C2)C1 85206,c1(C(=O)NCC2C(NC(C(C)NC(CC)(C)C)=O)C2)ccc(NC)c(F)c1 85207,N1(C(C(C)OCCOC)=O)CC2(CC2)CC1CNC(=O)CC1CCCCC1C 85208,c1(C(=O)NCC2C(NC(C3(C#C)CCCC3)=O)C2)cc(NC(C)=O)cnc1C 85209,N1(C(CCC(=O)N(CCC)CCC)=O)CC(NC(=O)C(CSC)OC)CC1(C)C 85210,c1(C(N(CCCNC(COCC#C)=O)C)=O)ccc(NS(=O)(=O)CC)cn1 85211,c1(SCC)cc(C)ccc1-c1ccccc1.C1(OC)NCCCC1C 85212,N1(C(COC)=O)CCC2(C(=O)NCCN3CCNC3=O)CC2C1 85213,C(=O)(CC(C)(C)C)NCC(C)(C)C(C)O.C=C1CC2(C1)C(=O)NOC2 85214,C(Cc1ccccc1)(C(=O)NCCC(O)CNC(=O)CCCN(C)CCO)NC(N)=O 85215,N1(C(c2c(C(C)C)ncnc2)=O)CC2CC(NC(=O)CCCCCF)CC1C2 85216,C#CCC(C(=O)NCCCCC1CCCC1)NC(C1CCC(OC)CC1)=O 85217,C(C(C(=O)N(C1CCC(C)(C)CC1)C)C(C)C)NC(c1c(C#C)c[nH]n1)=O 85218,c1(C(N2C(NC(COc3cn(C)nc3)=O)CC2)=O)cccc(-n2cncn2)n1 85219,N1(C(CC2C(CNC(C(CCC)OC)=O)C2)=O)CCCC(C)(OC)C1 85220,C1(C(c2ccccn2)=O)(NC)CCC(F)(F)CC1.N1(C(C)=O)Cc2nc(C)sc2C1 85221,O=C1COc2cc(C(=O)NCC3(O)CCN(C(=O)C=CBr)CC3)ncc2N1 85222,c1(C(=O)NCC(CNC(c2cc(F)c[nH]2)=O)OC)cc2c(cc1Cl)CCCC2 85223,Cc1ccc(=O)n(CC(N2CCC23CN(C(C2CC24CCOC4)=O)C3)=O)n1 85224,c1(CC(C(=O)NCCN(C(Cc2cn(CC)nc2)=O)C2CC2)O)ccccc1Cl 85225,N1(C(c2c(CC)ocn2)=O)CC2CCC(C1)N2C(C1(C)CCCC1C)=O 85226,c1(-n2ccc(CN(C(Cc3c(C)cccc3)C)C=O)n2)ccc(F)cc1F 85227,Cc1cccc(C(=O)NCC2(C)CCN(C(c3nc(-c4ccco4)sc3C)=O)C2)c1 85228,c1(OC)ccc(C(=O)NCC2CCN(C(=O)C(C)=C(C)C)CC2C)c(F)c1Cl 85229,C1(C#N)(C(N2CCN(C(c3n(C)nc(C4CCC4)c3)=O)CC2)=O)CC2C=CC1C2 85230,N1(C(C2C(C)OC(=O)N2)=O)CC2CC1CN2c1ccnc(-c2cccnc2)n1 85231,c1(C(=O)OC)cc(Cl)c(C)cc1Br.c12cnn(C)c1CNC(=O)C(=O)N2 85232,N12CCC(COC)(C1)C(=O)CC(C)C2=O.C(CCO)(C1CCC1)OC 85233,c1(C(N2CC3(CN(C(c4cc(C)[nH]c4C)=O)C3)C2)=O)cc(C)c(Br)cc1C 85234,N1(C(c2cc(OC)n[nH]2)=O)C2CCC1(CNC(=O)C(C)CC1CCCO1)CC2 85235,c1(C(=O)OC(CSC2CC2)C2CC2)cc(O)nc2c(Br)cccc12 85236,c1(C(=O)NC(CC(C)NC(=O)CC2C=CCC2)C)cccc(OC2CCCC2)c1 85237,C1(C)(CC)C=C(C(=O)NC(C2CCCN2C(C2CC=CCC2)=O)(C)C)C1 85238,c1(C(=O)NCC(CNC(C2CCC(C)O2)=O)(C)C)ncccc1N 85239,Cc1cc(C)c(C(=O)NCC2CCN(C(=O)CN(C(=O)Cc3ccsc3)C)C2)[nH]1 85240,c1(CC(=O)Nc2cnn(-c3cccnc3)c2)cc(C2CC2)n[nH]1.C12CN(C1)C2=O 85241,Cc1cc(=NC2CC(C)n3ncnc32)[nH]c(NC2CCCC=C2Br)n1 85242,C(CN=C(NCc1ccc(Cl)nc1)NCC1CCCCN1C(C)C)SC 85243,CC(CCCCNC(c1ccncc1Br)=O)NC(=O)CC1(C2CC2)CC1 85244,N1(C(C2(C#C)CCCC2)=O)CC2CC(O)C1C2NC(c1c[nH]c(Br)c1)=O 85245,Cc1ccc(OCC(O)CNCCCC2CC2C)c(C)c1Br 85246,c1(NC(C2CC(=C)CN2C(C2(C)CC2)=O)=O)cccc(Br)c1OC 85247,C1(NC(C2N(C=O)CCC2)=O)CC2CCC1N(C(c1coc(Cl)n1)=O)C2 85248,c1(C(=O)NCC2CCCN(C(C(CC=C)(C)C)=O)CC2)c(Cl)nc2ccccn12 85249,c1(CS(Cc2c(OC)ccc(F)c2)=O)cc(F)c(Cl)c(Cl)c1 85250,CC1(CNC(=O)NCCNC(c2cc(C(F)(F)F)cs2)=O)CCCCC1O 85251,n1(CC(N2CC3CC(NC(C(C)NC(C)=O)=O)C3C2)=O)cc(C#N)c(O)nc1=O 85252,N12CC(C(OC)C1)NC2=O.c1(-c2scc(C(=O)OCC)n2)ccc(Cl)cc1 85253,N1(C(c2c(C)oc(C(C)(C)C)c2)=O)CCC2C(C1)CN2C(=O)C(=O)C(C)(C)C 85254,C1(CNC(=O)CC2CCC3(CNC3)O2)CC2CCCC(C1)C2 85255,n1(CC(=O)NC2CCCN(C(c3csc(C)c3N)=O)C2)cccc([N+](=O)[O-])c1=O 85256,C1(C(=O)NC(C(=O)OCC)C2CC2)CCC(C)(C)N(C(c2cccc(CC)n2)=O)C1 85257,C(=O)(C(C)(CC)CO)N(c1cn(CCCC(=O)OCC)nn1)CC1CCCOC1 85258,N1(CC=CC(=O)OC2CC2)CCCCC1CC1(Cc2cccc(F)c2)CC1 85259,c1(C(CC)C)nccc(N2CCCC2CN(C(=O)CC2CC2C)C)n1 85260,CN1CCCC2C1CCCCN2C(=O)C(N)Cc1cc(Br)cc2c1OCC2 85261,C12CC(C3OC(C)(C)OC13)CNC2=O.CCCCCC(C)(C)NC(=O)OC(C)(C)C 85262,N1(C(CCCOC)=O)CCCN(C(c2cnc(C3CCCC(C)(C)C3)[nH]2)=O)CC1 85263,c1(C(N2CCN(C(C(C=C)(C)O)=O)CC2CC)=O)n[nH]c2ccc(C)cc12 85264,N1(C(C=CC)=O)CCN(C(c2ccc(CCC)cc2)=O)C(CCCC)C1 85265,N1(CCCNC(=O)Cc2cc(CO)on2)CCCN(CCO)CC1 85266,Cc1cc(=NC2COCC2)[nH]c(Sc2cnn(CC(C)C)c2)n1.C1(N)CC1 85267,c1(NC(N(c2ncccn2)CCOC)=O)ccc2ncc(I)n2c1 85268,C1(CNC(c2onc(COC)n2)=O)CCCCN1C(c1coc(C(C)(C)C)n1)=O 85269,CCC(C)C(O)C(=O)NCC1CC(O)(CNC(c2ccnn2C(F)F)=O)C1 85270,c1(-n2c(C)cc(C)n2)ccc(C)c(C(=O)NCc2noc(C3CCCO3)n2)c1 85271,C12CCN(C(=O)CNC1=O)O2.C1(C(C)C)CCN1C(N)=O 85272,C(c1cnc(C(C)(C)C)s1)=CC(=O)NCC(CC)NC(C1(CC(F)F)CCC1)=O 85273,CCC(Cc1ccc(N)cc1)C(=O)NCCCN(C)Cc1nnc(C(C)C)o1 85274,c1(-c2c(COC)n[nH]c2)nc(C2CCCO2)nn1CC1CCSC1 85275,c1(C(CCC)NC(=O)CNC(=O)N(C2CCCCC2)C)cccc(Cl)c1.C(C)(=O)N 85276,C1(OC(=O)CC2OCCO2)CC2(CCOC2)C1 85277,c1(OC)ccc2nc(N3CCC(OC)C3)[nH]c(=NCCc3ncnn3C)c2c1 85278,C1(C(=O)NCC(C(=O)NCc2ccc(F)cc2)N(C)C)CSCC(=O)N1 85279,c1(C(C)=O)ccc(Cl)cc1NC(C1CC2(C1)CN(C(c1ccon1)=O)C2)=O 85280,CC1=NOC(C)(C(=O)NCC(C2CC2)NC(c2cc(C)c(C(F)F)s2)=O)C1 85281,c1(C(=O)NC(C)Cn2cnc3ccccc23)cnc2ncnn2c1O 85282,C1(C(C)C)CN(C(c2nc(C3CC3)cs2)=O)CCN1C(c1cc(O)nn1C)=O 85283,C1(C(=O)NC(CN(C)C(C2CCC23CCC3)=O)(CO)CO)CCCCCCC1 85284,C(CC(=O)N=c1ccn(CC(N)=O)[nH]1)(C(C)C)NC(c1cc(C)cc(F)c1)=O 85285,C1(NC(Cc2ccc(OC)cc2F)=O)CCCCN(C(C2(OC)CCC2)=O)CC1 85286,CC1(C)CN(C(=O)CCCF)CC(CCNC(=O)C(Cl)=CCl)O1 85287,C1(C(N2C(CNC(Cc3cn(CC)nn3)=O)C(C)CC2)=O)CCn2cncc2C1 85288,c1(NC2(COC)CC2(C)C)ncc(C(=O)OC)cc1Cl 85289,N1(C(C(C)C2CCOC2)=O)CCC2(CC1)CCN(C(=O)CC1CCC3CC3C1)C2 85290,Cc1nccc(C)c1CC(=O)NCC1CC(F)(F)CN1c1nnc(C(F)F)s1 85291,C1(NC(C2(CCNC(=O)CC34CCCC3C4)CCCC2)=O)CC2CC1C(O)C2O 85292,c1(CN2CCCC(C(=O)NC(CCC)=O)C2)nc2ccc(C(F)(F)F)cc2o1 85293,N1(C(c2nn(CC)c(O)c2)=O)CCCC(C(=O)NOCCC(F)F)CC1 85294,C(=O)(C(C)(O)C(C)C)NCCCC1N(C(c2cc(CSC)on2)=O)CCCC1 85295,C1(=CC(=O)NC(C2CCCC2)CNC(C(CCSC)O)=O)CCCCC1(C)C 85296,c1(CNC(=O)NC2CCCC(S(CC)=O)C2)ccc2c(c1)oc(=O)n2C 85297,Cc1cc(OCCN(C)C(=O)NCC2CC2F)cc(C)c1 85298,c1(CC(=O)NC(C2CC=CCC2)C(=O)N(CCOC)CCO)ccnc(O)c1 85299,c1(CCC(=O)NC2CCN(C(CN3CC(CC)C3)=O)C2)c(C)noc1Cl 85300,C1(NC(C2N(C(C)C)CCC2)=O)COC2(C1)CN(C(c1cncs1)=O)C2 85301,C(=O)(C1CCOc2ccc(Br)cc21)NC1C(NC(c2c(C)nco2)=O)CCCC1 85302,C1(C)(CC)CC(NC(c2ccc(C(F)F)cn2)=O)CN1C(=O)C=CC1CCCC1 85303,c1(C(=O)NCCC2(C(=O)NCc3c(C)n[nH]c3)CCCC2)csc(C#N)c1 85304,C1(CNC(CN(c2ncccn2)C)=O)CN(C(=O)CC2CCCCCC2)CCO1 85305,C(=O)(CC(C)CC(C)C)NC1CC(N(C(CNC(=O)NC)=O)C)C1 85306,CC(C)C(C(C1CCCCC1)NC(=O)CC1CCCC1)NC(c1nc(Cl)cs1)=O 85307,C1(CC=C)(C(=O)N(CC(F)(F)Cl)C)CCN(C(c2cc(Cl)ns2)=O)C1 85308,C1(N(c2cccc(O)c2F)C(c2n[nH]c3c2CCC3)=O)CCC2(CCNC2)CC1 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85327,C1(OC)CN(C(C2(NC(C)=O)CC2)=O)CC1NC(c1cccnn1)=O 85328,c1(CCNC(C(c2cccs2)NC(COCCC=C)=O)=O)c[nH]nc1O 85329,c1(Cn2c(C3C=CCCC3)nc(C3CSC3)n2)cc(F)cc(F)c1 85330,C1(NC(c2cc(CNC(=O)C3=CCCCO3)[nH]n2)=O)CCC2(CCC2)CC1 85331,C=CC(C)(CC)C(=O)NCC1C2CCC(C2)N1C(=O)Cc1ccc(F)cc1Cl 85332,C(=O)(C1(C)CCn2ccnc21)N1CCC(O)(CN(C)C(C2(C)CCCC2)=O)C1 85333,Cc1cc(=NC2C(C)C2C)[nH]c(=NCC(=O)N2CCN(C)CC2)[nH]1 85334,c1(NC(N(C)Cc2cc(C)no2)=O)cc(Cl)cc(I)c1 85335,C1(C)(C(=O)NCCC(=O)NC)CCN(C(=O)C(C(C)O)NC(C)=O)C1 85336,c1(C(=O)NCCOC2CN(C(C(CN(C)CC)F)=O)C2)cccc(COC)c1 85337,C(=O)(CC(=O)N1CC(NC(C2CN(C(C)=O)C2)=O)C1)OCC 85338,c1(C(=O)OC)cc(C(N2CCC(O)(CNC(=O)COC3CCC3)CC2)=O)cc(F)c1 85339,C1(NC(CCC#CC)=O)CN(C(c2cccc3ccoc23)=O)C2(CCCC2)C1 85340,CCCC(C)CC(=O)N1CCCC1CCCNC(C1(C(O)C(F)(F)F)CCC1)=O 85341,C12(C(=O)NC3C(NC(c4ccc(CC)[nH]4)=O)COCC3)CCC(C)(CC1)CO2 85342,n1(CC(=O)NCC(C)NC(=O)CCC2CC2)sc2cc(Br)ccc2c1=O 85343,Cc1cc(C(=O)NC(CO)C(C)NC(=O)C(c2ccc(Cl)cc2)(C)O)cc(C)n1 85344,C(C(O)C(C)(C)C)N1C(=O)C(CCOCCO)NCCC1C(C)=O.CCO 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85379,N1(C(c2c(CC)occ2)=O)CCN(C(=O)CCCc2csc(C)n2)CCC1C 85380,CC(CC(=O)N1CCCCC(NC(C2(C#N)CC2(C)C)=O)C1)C(F)F 85381,C1(CC(=O)NC(c2c(CSCC)cncc2)=O)OCCOC1(C)C 85382,C(C(C)(C)CC(=O)NC1(CO)CCN(C(c2cccc(Cl)c2)=O)C1)OC 85383,c1(C(N2CC(NC3(CC(F)F)CCOCC3)C2)=O)cc(CN(CC)CC)ncn1 85384,CC1(NC(=O)CCSCC(N)=O)CCN(C(=O)CCc2ccco2)CC1 85385,C(CCCCC(=O)NCC(C(C)C)NC(c1cc(Br)n(C)c1)=O)SC 85386,c1(CCCN(C2CCN(c3nnnn3C)C2)C)ccccc1C(=O)O.C1(C)CC1 85387,Cc1ncc2c(n1)CCC(C(N1CC(NC(C3(C)CC3Br)=O)CCC1C)=O)C2 85388,C(=O)(CC1=CCCC1)N1C(C(=O)NC2CC3CCC2O3)C=CC1 85389,C=CC(CCC)CC(=O)N(CCC(C)NC(c1cc(C2CC2)[nH]c1C1CC1)=O)C 85390,c1(CCCN(C(=O)CCNC(=O)C(F)C2CCCO2)C)ccccc1 85391,C1(C)(CNC(C(C)SC)=O)CC(F)(F)CN1C(c1cccc(OC(C)(C)C)c1)=O 85392,CN1CCC(C)(C(N2CCOC(CNC(=O)CN3CCNC3=O)C2)=O)C1 85393,N1(CCC(=O)N(C)CC2CCN(C(c3sncc3Br)=O)C2)C(=O)CCC1=O 85394,C(=O)(CCCC(C)(C)C#N)NC1CC(NC(c2c(CC)sc(=N)[nH]2)=O)C12CCC2 85395,CC(C(C)C(=O)NOCCCCF)NC(c1cnn2ccccc12)=O 85396,C#CCCCCC(=O)N1CCCC1C(C)(C)C(=O)NC(CO)C(C)(C)C 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85800,CC(CC(=O)NCc1nc(C(=O)NC(C2CCOC2)C)co1)c1ccco1 85801,CCCCCCCCCC(=O)N1CC(C)(NC(=O)Cc2ccccn2)C1 85802,N1(C(=O)NCC2CC2)CCN(c2nnc(C3CC3)n2C2(C(F)F)CCCCC2)CC1 85803,C1(N(C)C)CCCCC1NC(=O)CO.C(CCN=[N+]=[N-])N1C(C)C2CN(C2)C(=O)C1 85804,C1(n2cc(C(C3CCCC3)C)nn2)CCN(C(C2COCCO2)=O)CC1O 85805,C(=O)(C(C)C(CC)CC)N(C1CCN(C(c2c(CC)n[nH]c2)=O)C1)CCO 85806,N1(C(c2c(C)nc(C)s2)=O)CC(NC(=O)CN(CC(C)(C)C)C)C(C2CC2)C1 85807,c1(C(=O)NC(CCC)CCCNC(=O)CCC=CC(C)C)ccc(F)c(F)c1N 85808,C1(NC(c2nc(CCC)sc2)=O)CCCC1(C)NC(=O)C(C)c1ccsn1 85809,c1(C(=O)NCC2CC(O)(CNC(C3(COC)C=CCC3)=O)C2)ccc(C)nc1C 85810,Cc1[nH]c(C)c(C(N2CC3CC(CNC(=O)CC(C)c4ccco4)C3C2)=O)c1C 85811,c1(C(=O)NC2(CNC(Cc3ccc(OC)cc3)=O)CCC2)c(Cl)nc(C)nc1Cl 85812,C12CCN(CC1)C2=O.Cn1ccc(-c2cn(CC3CC(NC=O)C3)nn2)n1 85813,n1(CC(=O)NCC2C(CNC(c3n(C(CC)CC)ncc3)=O)C2)nc(C)cc1C 85814,N1(C(CC)=O)CCCC(OCc2n(C3CN(C(C4CCC(=O)O4)=O)C3)ncc2)C1 85815,N1(C(CN2CC(C)C2)=O)CCN(C(=O)C(Cl)=CCl)CCC1C 85816,C1(NC(c2ccc(C)nn2)=O)CN(C(=O)Cn2ncc(Cl)c2C)C2(CCCCC2)C1 85817,N1(C(c2ccc(C3CC3)s2)=O)CCN(C2CCCN(C(C3CC3F)=O)C2)C(=O)C1 85818,C(C(C)(C)CC(=O)N1CC(C(=O)NCC(C)(C)OCCSC)OC(C)C1)OC 85819,C(CCCC(F)(F)F)(c1ccc(NC(C)=O)cc1)Oc1ccc(C(=O)OC)cc1 85820,N=c1nc2c(C(N3CCCC3C3(NC(=O)Cn4cccc4)CC3)=O)cccn2[nH]1 85821,N1(C(c2c(C)nc(Br)s2)=O)CCN(Cc2cccc(Cl)c2O)C2CC12 85822,C12(CCNC(C(C)=CC3CC3)=O)CCC1CN(C(=O)C(O)c1ccco1)C2 85823,CCCC(CNC(C1C=CCCN1C(c1ccccc1C)=O)=O)CCO 85824,c1(C(=O)NC2CN(C(CC(C)OC)=O)C2)sc2nccnc2c1N 85825,C=CCC(C(=O)Nc1cccc(NC(C2C(C)(C)OC2(C)C)=O)c1)C(C)(C)C 85826,N1(C(C(CC)NC)=O)CC(NC(c2ccnc(OC)n2)=O)C2CCCCC12 85827,N1(C(c2c(C)cco2)=O)CCC(N=[N+]=[N-])(C(=O)N(C)CC2CCOC2)C1 85828,c12cncc(c1)C(=O)N2.c1(C(N)=O)cc(C(=O)NCC2CCC(=O)N2)n[nH]1 85829,C12(CNC(C3CC(C)(CC)C3)=O)CCCC1N(c1ncncc1C)CCC2 85830,CCN=C(NCC(C)(C)S(C)(=O)=O)NC1CC1c1ccc(C(F)(F)F)cc1 85831,Cc1ccc(C(=O)NC(C(=O)N(C)Cc2cnco2)C(C)C)c(C)n1 85832,C1(CNC(=O)C2=CCCS2)CCC2(CO1)CC(NC(=O)COc1cn[nH]c1)C2 85833,N1(C(c2cnc(C(C)C)nc2)C(=O)Nc2c(C)cccc2)CC2CC3CC2C1C3 85834,c1(C(=O)NCC2(OC)CN(C(=O)Cc3c(C)noc3C)C2)cc[nH]c(=N)n1 85835,c1(OC)ccc(CCC)cc1C(=O)NCC(C)(C)NC(=O)C=CCF 85836,Cc1cc(C(=O)NCC(C2CCCCC2)NC(=O)CC23CC(C2)C3)ccc1[N+](=O)[O-] 85837,c1(OC)ccc(C=CC(N2CCC(O)(CNC(=O)C(C)(O)C(C)C)C2)=O)cc1F 85838,c1(C(N2CCCCC(NC(C3C(C)C3)=O)C2)=O)cccnc1S(=O)(=O)C(F)(F)F 85839,c1(CC)ncccc1C(=O)N(C1CCC(NC(c2cccnc2)=O)C1)C 85840,c1(SC)ncc(C(=O)NC2CC(NC(C3(n4ccnn4)CC3)=O)C2)c(O)n1 85841,c1(C(=O)NC(C(=O)NC2CC(C(C)C)OC2)CC2CCC2)ccn2ccccc12 85842,c1(CC(N2CCC(NC(CC(C)OC)=O)CC2C)=O)coc2c(C)c(C)ccc12 85843,C=C(C)CC(C(=O)NCC(C1CCCC1)OC)NC(c1cc(O)sc1C)=O 85844,CC1CC(NC(=O)Cc2ccccc2)CN1c1ccnc(-c2nccs2)n1 85845,N1(C(CCCOCCOCC)=O)CC(NC(c2c(N)cccc2F)=O)CC(O)C1 85846,Cc1ccc2sc(N3CC4C(CNC(=O)C(F)(F)C(C)O)C4C3)nc2c1 85847,c1(C(N2CC3C(CNC(CC(C)(C)C4CC4)=O)(C3)C2)=O)cc(O)ccc1Cl 85848,S(=O)(=O)(c1cnc(NCC23CCCC2OCC3)c(Cl)c1)NC(COCC)C1CC1 85849,c1(C(=O)NC2CCN(C(CCC(=O)NCC)=O)CC2F)cccn2c(C)nnc12 85850,c1(C(N2CC(SCC)OCC2)=O)c[nH]ccc1=NC(=O)CC1CN2CCC1CC2 85851,CC(F)(F)CCN(C(=O)CC1(CCN2CCCC2)CC1)C1CC1.C12CCN(C1)C2=O 85852,CC1(NC(=O)Cn2ccccc2=O)CCN(C(c2coc(Br)c2)=O)C1 85853,N1(C(CCC(=O)OCC)=O)CCC(CO)C(NC(=O)CCCn2ccnc2C)C1 85854,N1(C(C(CC)O)=O)CC2CC3CC2C1C3NC(=O)CCc1cscn1 85855,N1(C(CC(C)n2cccc2)=O)CC(NC(=O)CCc2ccncc2Br)C(O)C1 85856,N(C(=NCCC(C)OC)NCc1cccs1)Cc1noc(C2CC2)n1 85857,c1(C2(N(C=O)Cc3ccc(OCC)nc3)CCCC2)cc(C)cc(C)c1 85858,N1(C(C(C=C)(C)O)=O)CC2CC(NC(c3ccc(CC)c(Br)c3)=O)C1C2 85859,C1(N(C(C2C(=C)C2)=O)C)CCCC(NC(c2occc2COC)=O)C1 85860,c1(C(=O)NC2C(CNC(c3cccc(C(=O)NC)c3)=O)C2)ccc(Cl)c(N)c1Cl 85861,N(C(=NCCF)NCc1cc(Cl)ccc1Br)C(C#C)C(C)OC 85862,c1(CC)ncncc1C(=O)NCCC(C)NC(=O)CCS(C)=O 85863,CC(C)(CCCO)C(=O)NCC(O)CNC(=O)CC1COCCOC1 85864,c1(OC)cc(C(=O)NC2CC3CC(NC(=O)C(C)SC)C2C3)ccc1F 85865,c1(N2CCC(CC=C)C2)nccc(=NC(C)CN(C(C)C)CC)[nH]1 85866,N1(C(=O)OC(C)(C)C)CCC(O)(C(F)(F)C(=O)N2CCC(n3ccnc3)C2)C1 85867,CN(Cc1c[nH]c(=N)s1)N1CC=C(C(C)(C)C(C(F)F)c2ccccc2)C1.O1CS1 85868,N1(C(C2C(CC)CC2)=O)CC2CC2(NC(C2CC(OC(F)(F)F)C2)=O)C1 85869,c1(C(N2C(C)C(=O)NCC2)C(=O)NCc2ccco2)cc2ccccn2n1 85870,N(C(=NCCCC(C)(F)F)NC(C)C1CC1)C(c1cccnc1)C 85871,C1(CC(=O)NC(C=C)(C)C)CN(C(C2CC3CC2CC3O)=O)CCC1C 85872,c1(OC)cc(CNc2nc(C(CC)CC)nn2-c2c(F)cccc2Cl)ccc1C 85873,C(N=c1ccn(CCF)[nH]1)(c1ccn(CCCC)n1)C1CCCSC1 85874,FC1(F)CCC2C(CCCN2C2CC(=O)NC3(CCC3)C2)C1 85875,c1(CC(C(=O)O)OC(N=[N+]=[N-])F)cccc2ccsc12.C(=O)(CC(N)CC1CC1)N 85876,C(=O)(C1=COc2ccccc2O1)N(C1C2CN(C(=O)Cc3ccccn3)CC12)C 85877,N1(C(c2c(CC)nn[nH]2)=O)CCC(CC(=O)NC2CCOC2CC(C)C)CC1 85878,c1(C(N2CC(CCNC(C3C(C)C3C)=O)C(C)C2)=O)cc2c(cn1)OCCO2 85879,C=C(Br)CCC(=O)NC1CCC(CNC(c2ccc(C(F)F)nc2)=O)C1 85880,Cc1c(O)c(=O)ccn1CN1CCC(NC(N2CCN(CCO)CC2C)=O)C1 85881,c12c(cccc1[N+](=O)[O-])C(=O)N2.C1(NC(C2C(C(=O)OC)C2)=O)CC(CO)C1 85882,Cn1c(O)ncc(C(=O)NCC23CCC2CCN3C(c2ccc(CO)s2)=O)c1=O 85883,C(CC(C(C)(C)C)NC(=O)C(C)OC1CCOC1)N(C(c1c(C)noc1N)=O)C 85884,CC(C)(CC(=O)N1CC(NC(C2CCCCN2N=O)=O)CC(F)C1)CC(F)F 85885,C1(NC(C(C)O)=O)CC2(C1)CC(NC(c1c[nH]cc(F)c1=O)=O)C2 85886,c1(C(N(C(C)CNC(C2CCCN2C2=NN=COCC2)=O)C)=O)ccnnc1S 85887,C1(NC(C(CCCCCC)C)=O)Cc2ccccc2C1NC(C1(O)CCOC1)=O 85888,CC(Cc1ccccn1)N=c1[nH]c(=NCCN2CCC(O)C2)c2sccc2[nH]1 85889,N1(C(c2cnc(OCC)nc2)C(=O)NC(C)(C)C)CCN(C)C(CC)C1 85890,c1(NCC2OCC(CNC(=O)CC34CCC(CC3)CC4)C2)ncnc2sccc12 85891,c1(C(=O)NC2C(NC(CCn3ncn(C)c3=O)=O)CCC2)c(N)ccc(F)c1F 85892,C(C(C(=O)N1CC2CCC1C2NC(c1ccc2c[nH]nc2c1)=O)C(F)(F)F)OC 85893,c1(NC(CCCn2ccc(C)c(Cl)c2=O)=O)ccc2nc(O)n(C3CC3)c2c1 85894,C1(ONC(C2CC(C)O2)=O)CCC2CN(C(c3c(C)nn(C)c3)=O)CC2C1 85895,c1(CC(=O)NCCCCC(C)NC(=O)C(C)(C)C(N)=O)ccc(Cl)cc1Cl 85896,N1(C(C2(C(=O)OCC)CC2)=O)CC(C(=O)NC2CCCC(C)C2C)C(C)(C)C1 85897,C1(CCNC(CN(C)C2CC2)=O)CC2CCC(C1)N2C(C1(C)CNC(=O)C1)=O 85898,N1(C(c2cnc(C)o2)=O)CC=CCC1C(=O)NCC1CC1 85899,c1(CN(C)CC2CCCN2C(=O)CN2CCOC2=O)c(F)cccc1Cl 85900,c1(OC)ccc(C(=O)NCCC2CCN(C(C3(CF)CC3)=O)CC2)nc1 85901,C(=O)(C1=CCCOCC1)N1CCC(COC)(NC(c2cnc(C(C)O)s2)=O)C1 85902,C1(CC(=O)NCC2N(CC)CCC2)N(C(c2cccnn2)=O)CCC1(C)C 85903,C(=O)(C1=NNC(=O)CC1)NC(CC)(CNC(=O)C(C)Cc1ccccc1Cl)CC 85904,N1(C(c2cc(CN(C)C)on2)=O)CCC2CN(C(=O)Cn3ccnn3)CCC2C1 85905,N1(C(c2c(CC)n(CC)nn2)=O)CC(O)(C2(CNC(C3CC(C)CO3)=O)CC2)C1 85906,c1(C(N(CC(N2C(C(=O)OCCSC)COCC2)=O)C(C)C)=O)cc(C)ccc1O 85907,CC(C)C(CNC(=O)COc1ccsn1)NC(C1CC1C(F)F)=O 85908,C1(C(=O)NCC2CC(CNC(C(C)OCC)=O)C2)CCc2nnnn2C1 85909,c1(C(C(=O)NC(C(C)Sc2ccccc2)C2CC2)C)cn(C)nc1C(F)(F)F 85910,C1(C)(C(=O)NC2(CC=C)CCOC2)CCCN(C(c2cn(CC)nn2)=O)C1 85911,C1(NC(CC(=O)N(C)C)=O)CCC2CN(C(=O)Cc3nc([N+](=O)[O-])n[nH]3)CC2C1 85912,Cc1cccc(C)c1C(C)NC(c1cc(Br)sn1)C 85913,N1(C(C(CC)OCC)=O)CCC2CCCC(C1)N2C(c1cc2c(nn1)CCC2)=O 85914,c1(CC(=O)NCC(C)N(C)C(c2cc3sccc3n2C)=O)cc(F)c(F)cc1F 85915,N1(C(C(COC)OC)=O)CC(C(=O)N(CCCO)C(C)C)C(C)C1 85916,C1(C(=O)NCC2C(CNC(Cc3ccn(CC)n3)=O)C2)C(C)(C)C1(C)C 85917,N1(C(CCCCC(C)C)=O)CC=C(C(C)(C)C(=O)NCC2CCC(F)C2)C1 85918,c1(C(N2C(CC)CN(C(=O)C3=NNC(=O)C3)CC2)=O)cc2n(n1)CCCC2=O 85919,c1(CC(N2C(CNC(C=CC(CC)C)=O)CC(OC)C2)=O)ccc(F)c(Cl)c1 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85955,C1(C(N(CCN(C(c2cc(C(C)(C)C)on2)=O)CC)CC)=O)CCc2nnnn2C1 85956,CC1CN(C(=O)Cc2n[nH]cc2Br)CC1CNC(=O)Cc1cnccn1 85957,c1(C(N2C(C)C(C)N(C(C3CC(=O)CCO3)=O)CC2)=O)cn2cc(Cl)cnc2n1 85958,c1(C(=O)NCC(=O)NC(C(=O)NC2CC(OC)C2)C2CCCO2)cc(C)n(C)c1C 85959,c1(-c2c(NC(c3csc(N4CCNCC4)n3)=O)nccc2)nc2ccccc2s1 85960,C(=O)(CCCC(=O)OC(C)(C)C)NC(CNC(C1CN(C(C)C)C1)=O)(C)CO 85961,C1(C(=O)NCCC2(O)CN(C(C3(OCC)CCCC3)=O)C2)CCOC(C)(C)C1 85962,CCC(F)(F)CC(=O)N(C)CC1CCCC(NC(=O)CCc2ccoc2)C1 85963,c1(C(N2C3CCC(NC(C=CC=CCC)=O)C(C3)C2)=O)cnn2ccc(O)nc12 85964,c1(NC(C2CC3CC3N2C(=O)CC2CCCCO2)=O)ncc(Br)nc1Br 85965,Cc1cc(=NCCNS(C)(=O)=O)[nH]c(NC2CCC3CC23)n1 85966,c1(CC)cc(N2CCC(CNC(=O)C(F)(F)c3cscn3)C2)ncn1 85967,c1(C(=O)NC(CC)C)ccc(=NCc2ccc(Br)c(F)c2)[nH]c1 85968,C1(Cn2cc(CN3C(C(c4cnns4)=O)CCC3)nn2)CCC2CC2C1 85969,C1(NC(=O)CC2CCC2)CCCC(NC(=O)CC23CCCC2C3)C1 85970,N1(C(C2N(c3nc(SC)c(Br)cn3)CCOC2)=O)CCc2ccccc21 85971,c1(N(c2ccncc2Br)C(=O)C(=O)N2CCC2CCC(O)O)ccc2nc(O)sc2c1 85972,CC1NC(=O)CCC1NC(c1cc(CNC(c2ccn(C(F)F)n2)=O)no1)=O 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85991,N1(CC(=O)N(CC#C)CC=C)C(C)CN(C(=O)CCCCC(C)C)CC1C 85992,CCCC(CNC(=O)C=CC(F)(F)F)C(=O)N1CCCC1CN(C)C 85993,N1(C(c2c(N)c(F)ccc2)=O)CCn2c(cc3cc(Cl)ccc23)C1 85994,c1(C(N2C(CNC(=O)CCC(C)C)CC(OC)C2)=O)nccc2c(F)cccc12 85995,C1(C2CCCCC2)(C(=O)NCC(C)N(C(c2ncn(C)n2)=O)CC)CCCCC1 85996,c1(C(N2CCN(CC)C(=O)C2C)=O)ccc2cc(F)ccc2n1 85997,c1(C(N2CCN(c3c(OC)cc(Cl)cc3)CC2)=O)ccc2[nH]nc(Br)c2n1 85998,N1(C(C(n2ccc(Cc3ccccc3)n2)C)=O)CCOC2CCNCC12 85999,Cc1nn(C)c(=O)c(C(N2CC(C(=O)O)C3(C2)CN(C(=O)CC2CC2)C3)=O)c1C 86000,Cc1c(C(=O)NC(CNC(c2ccsn2)=O)CO)cnc2ncnn12 86001,C1(NC(C=CC(=O)N(C)C)=O)C=CC(C(=O)NCC(F)Br)C1 86002,c1(SC)cnn(C)c1C(=O)N(CCCNC(=O)C(c1ccc(C)s1)C)C 86003,c1(C(N2CCN(C(=O)C(F)C3CCC3)C(CC3CC3)C2)=O)cc2n(n1)CCC2 86004,C12(CNC(c3c(CC)ncs3)=O)CCC1CN(C(=O)CN(C)C(=O)OC)C2 86005,CC(C)(CO)C(=O)NC1CCC1NC(c1ncoc1-c1ccon1)=O 86006,C=C(Cl)CC(C(=O)NC1CCC(=O)NC1)NC(=O)C(F)CCC 86007,Cc1c(C(=O)NCC(C)(CO)NC(C2CC2F)=O)cnn1C(C)C 86008,C1(NC(c2c(C)n(C3CCC3)nc2)=O)CC2(CCN(c3ccnc(C#N)n3)C2)C1 86009,Cc1nc(N(CCC(C)C)Cc2ncccn2)cc(=NC(C)C2CC2)[nH]1 86010,Cc1cccc(C(O)C(N2CC=CC(NC(c3cncc(N(C)C)c3)=O)C2)=O)c1 86011,N1(C(C(C(C)(C)C)O)=O)CCN(C(=O)CC2=NNC(=O)C2)C2COCC12 86012,c1(C(=O)NC2C(CC)CN(C(=O)CCc3cc[nH]n3)CC2)c2c(co1)CCOC2 86013,N1(C(C2N(CC)CCC2)=O)C2CCC1CC(C(=O)NCC(F)C1CCC1)C2 86014,c1(C(=O)NCC2C(NC(C(CC)SCC)=O)CC2)c[nH]nc1[N+](=O)[O-] 86015,C12(NC(CCN3CCN(CC)CC3)=O)CC1CN(C(=O)C(O)COC)C2 86016,Cc1nncn1NC(=O)C1C2CC1N(C(=O)CC1CCC1)C2 86017,CC1CCN(C(c2c(F)ccc(F)c2F)=O)CCC1N1CCC(C(=O)O)C(O)C1 86018,c1(C(=O)OC)cc(C(=O)N(C)CCN(C(=O)C(C(C)C)SC)C)c(C)o1 86019,C1(C(N(CC(C)NC(c2ccncn2)=O)C)=O)C(C)CCN1C(=O)OC(C)(C)C 86020,C(=O)(CCN(C)N=O)N1C(CN(C(C=CSC)=O)C2CC2)CCC1 86021,N1(C(C2CCCN(C(=O)CCc3ccoc3)C2)=O)C2C=CCC1CCC2 86022,c1(-c2cn(CCSCC(=O)NC3CC34CC(O)C4)nn2)ccnc(F)c1 86023,c1(C(=O)NC2CC(C(C(N3CCC(CC#C)C3)=O)F)C2)cc(C#C)ccn1 86024,c1(NCC2C(C)(C)COC2)[nH]c(=NCc2ccc(S(C)(=O)=O)s2)nc2scnc12 86025,CCCC(C(O)C(=O)NC1CCN(CCF)C1)NC(=O)CC(C)(C)COCC 86026,CN1CCC(C(N2CC(NC(=O)COc3cccc(CO)c3)C2)=O)C1=O 86027,c1(CNC(=O)NCC(O)COc2ccc(I)cc2)cn2ccsc2n1 86028,O=C1CS(=O)(=O)CC(C(=O)NCC2(CCNC(=O)C(F)F)CC2)N1 86029,c1(CN(C(C2(CC#C)CCCC2)=O)C)ccc(Cl)nc1.c1(C(C(=O)O)=O)cnn(C)c1 86030,N1(C(C(CCC)N(C)C)=O)CC2(CNC(=O)C(=Cc3cccnc3)C)CC1CO2 86031,Cc1cnc(C)c(NC(C2CCCCN2Cc2csc([N+](=O)[O-])c2)=O)n1 86032,c1(C(N(C)C)=O)ccnc(C(=O)NC2(C)CC3CC3C2)c1.C1(=O)OCCN1 86033,C(=O)(C(C)C(O)CC(C)C)NCC(C(NOC(CC)C)=O)OC 86034,C(=O)(C1=CCCN(Cc2cccc(F)c2Br)C1)Nc1ccc(OC)nc1OC 86035,c1(OC(=O)NC(C=CC(=O)NC(c2noc(C)n2)CC)C)cccc(F)c1 86036,C1(NC(c2c(C)cncn2)=O)C(C)CCN(C(c2cnc3sccn23)=O)C1C 86037,c1(NC(CN2CCN(Cc3c(C)ncc(Br)c3)CC2)=O)cc2ccoc2cn1 86038,C(C(C(=O)N1CCCC1CNC(c1cc(C)ns1)=O)C(C)(C)C)OCC=C 86039,C(=O)(C1=CCCCC1)N(CC(C)NC(C1CC(F)CN1C(=O)OC(C)(C)C)=O)C 86040,N1(C(C)C)CCCCC1C(=O)NC1(C)CN(C(C2(S(C)(=O)=O)CC2)=O)C1 86041,CC(CN(C)C)CCC(=O)NCc1ccc(C(=O)NCC2C3COCC23)o1 86042,N1(C(N)=O)CCCC(C(=O)NCC2CCN2C(=O)CCCc2ccsc2)C1 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86060,c1(C(N2CCCC(N(C(Cn3c(C)ncc3)=O)C)CC2)=O)cc2ncccc2[nH]1 86061,C12CCS(=O)(=O)C13CN(C3)C(=O)CN2C.C(C)(C(=O)OC)OCCSC 86062,N1(C(c2cnc(COC)[nH]2)C(=O)NCC2CC2)CCc2c3cc-3cc21.O(C)OC 86063,C(=O)(CCS(=O)(=O)CC(C)C)N1CC(NC(C2=C(C)S(=O)(=O)CC2)=O)C(C)C1 86064,Cc1cc(C(N2CCOCC(NC(c3ncc(Cl)s3)=O)C2)=O)c(N)c(Cl)c1 86065,C(=O)(C(F)(F)CCn1cc(CN(C)C)nn1)NC(C1CCS(=O)(=O)N1C)C 86066,C(=O)(C1=C(C)N(C)c2nnnn2C1C)NC(CC)CN(C(c1ccoc1)=O)CC 86067,C(=O)(C1=CC(O)CCC1)NCC1CC(OC)CN1C(=O)C(c1ccc(F)cc1)=O 86068,n1(CC)nc(C)c(C(=O)NC2CCCN(C(C3CC3(C)C)=O)C2)c1Cl 86069,c1(N(CC)Cc2ccc(Br)nc2)cc2c(C(F)(F)F)cc(N)nc2cn1 86070,c1(C(=O)NC2(CCCNC(C(=O)N(C)C)=O)CC2)cn2c(Br)cnc2s1 86071,N1(c2ccc(C=C(C)C)o2)CCC(C23CCC(C2)C3C(=O)O)C1 86072,CC1Cc2sc(C(=O)NCC3(F)CN(C(c4ccncc4O)=O)C3)cc2C(C)C1 86073,C1(NC(C(CNC(CCCOCCOC)=O)O)=O)CCC(C)(C)C1 86074,c1(C(N2CCC2CNC(CN(C(=O)CC2CCCN2C)C)=O)=O)ccncc1 86075,N1(C(c2ccc(C)cc2Cl)=O)CCN(C(c2nn(C)c3c2CCC3)=O)CC1C#N 86076,c1(C(=O)NCC23CC(C(=O)NC4(C)CCCS4)(C2)C3)ccc(C#N)c(F)c1 86077,C1(OCC)CCN(C(C2CN(C(c3cnc[nH]3)=O)CCO2)=O)CC1 86078,C1(C(N2CC(C(C)NC(c3c(OC)c[nH]n3)=O)C2)=O)C2CCCCC12 86079,c1(C(=O)NCCC2CCN(C(C(C)=CC3CC3)=O)CC2)c(F)ccnc1Cl 86080,CC1(C)CC(CNC(=O)COC2CCCCC2)CN1C(c1cccc(F)c1N)=O 86081,C(=O)(C(O)CC(N)=O)NC(C(N1CCC(CCOC)CC1)=O)CC1CCOCC1 86082,c1(C(=O)NCCN(C(=O)CCCC(C)=O)CCOC)ccc2cccc(F)c2n1 86083,c1(CC)ccc(C(=O)NCC2(NC(=O)Cc3c(C)nn(C)c3C)CCC2)cc1N 86084,N1(C(CSCCC(C)C)=O)CCC2CC1CN2C(=O)C(c1cncc(F)c1)C 86085,N1(C(C2N(C(c3c(C(C)C)n[nH]c3)=O)CC2)=O)CC2(C)COCC2(C)C1 86086,C1(OC)CC(NC(=O)CC(C)F)CN(C(C2CCN(CC3CCCC3)CC2)=O)C1 86087,c1(OC(C)C)ccsc1CC(=O)OCC.C12(CC1)C(=O)NC2.C(C)(C)(C)O 86088,C1(CC)CN(C(c2cnc[nH]2)=O)CCC1NC(c1cc(N(C)C)ccc1N)=O 86089,C(=O)(C(C)(O)C(C)(C)C)N1CC(C(N2C3CC(=C)CC2CC3)=O)C(C)C1 86090,Cc1cc(C(=O)NCCCN(C)C(C2(C)CC(=O)N(C)C2)=O)cc(C(F)F)c1 86091,CC1(C)CCN(C(C2C3CCOCC23)=O)CC1NC(c1cccc(Cl)c1)=O 86092,c1(C(N2CCC(C(CNC(CC(C)OC)=O)F)CC2)=O)cc(N)c(F)cn1 86093,Cc1cc(C(N2CC3(CCN(C(=O)C4=CCC4)CC3)C2)=O)c2cc(F)ccc2n1 86094,N1(C(CCCCCC#C)=O)CCc2[nH]nc(CNC(=O)C(C(C)C)N(C)C)c2C1 86095,N1(C(C(C)NC(c2c(C)occ2)=O)=O)CC2CC1C2NC(C1CC1C)=O 86096,c1(C(=O)NCC(C(F)(F)F)NC(Cn2c(C)ncc2)=O)ccc(C(F)F)cc1 86097,N1(C(CCCNC(C2CN(C(=O)NC)C2)=O)=O)CC(C)C(C)C1C 86098,N1(C(C2CC(=C)C2)=O)CCC2(CCCC(CNC(=O)COCC3CC3)O2)CC1 86099,C1(NC(C(C(C)C)O)=O)CC2CCC(C1C)N2C(=O)Cc1c[nH]c2cccnc12 86100,C1(NC(c2csc(CO)n2)=O)CCCC2CN(c3ccc([N+](=O)[O-])c(O)n3)CC12 86101,c1(C(C)C(=O)NCCCN(C(C2CC(C)(C)O2)=O)C2CC2)ccc(F)cc1F 86102,C1(C(=O)NCC2(OC)CN(C(C3CCS(=O)(=O)N3)=O)C2)(CCF)CNC(=O)C1 86103,C(CC(C)(C)CBr)(n1nnnc1C(C(C)(C)NCCNC(C)=O)SC)CC 86104,C1(CC=C)(NC(=O)C(O)C=CC)CCN(C(c2cccc(=O)o2)=O)C1 86105,Cc1cc(C)n(C(C)C(N2CC(C)(NC(C3OCCOC3C)=O)C2)=O)n1 86106,C1(NC(COC2CN(C(CNC(C3C(C)C3)=O)=O)C2)=O)CCOC1C 86107,Cn1cnc2cc(NC(N3CCC(C)(C)C(CO)C3)=O)cnc12 86108,N1(C(CC(CC)OC)=O)CCC(NC(=O)CCCOc2ccc(Cl)c(Cl)c2)C(C)C1 86109,N1(C(Cc2c(C)nc(S)s2)=O)CCCN(C(C2C(C)C2C)=O)CC1 86110,c1(C(=O)NCC2CCC(CNC(C(C)C(C)(F)F)=O)CC2)cccc2[nH]ccc12 86111,C1(CC(C)C)CCN(C(C2(CNC(=O)CCn3cnnn3)CCCC2)=O)C1 86112,CN1CCC(NC(=O)CCC2(NC(=O)Cn3c(O)nnc3O)CCCC2)C(C)(C)C1 86113,c1(C(=O)NCCC(=C)CNC(=O)CCc2ccco2)ccc(Cl)cc1 86114,c1(C(=O)NCCC(CCC#C)O)nn(CC)c2c1COCC2 86115,N1(C(c2c(CCC)nco2)=O)CC2CCC(C1)C2NC(=O)COC(C)C 86116,C1(Nc2ncc(C(=O)OC)c(F)c2)CCCC12CCN(C(C1CC(O)C1)=O)C2 86117,N#Cc1ccc(C(=O)NCCn2cc(NC(=O)CC3CC34CC4(F)F)cn2)c(O)c1 86118,C1(CCN(C)CC2CCN(C(=O)OCc3ccccc3)C2)NC(=O)NC1=O 86119,C(=O)(C(C(=O)N1CCC(OCC(=O)NCC(F)CO)CC1)OC)OC 86120,CCC1=NOC(CC(=O)N(CCCN(C)C)CCNC(=O)C(F)C(C)C)C1 86121,CC(CC(=O)NC(C)(C)C(C)NC(c1cnc(C(N)=O)s1)=O)N1CCCC1=O 86122,Cc1cc(=NCCc2cnc(O)nc2)[nH]c(NC2CC(=O)N(CCCC3CC3)C2=O)n1 86123,C1(C(=O)NCc2cccc(C)n2)CCCCCCN1C(C1CCC(C(N)=O)C1)=O 86124,N(C(=NCc1cc(C2CCCC2)on1)NC1CC(=O)N(c2ccccc2)C1)C(C=C)C 86125,c1(CN(C)C)cccc(C(=O)NCCCCCCNC(c2cc(Cl)n(C)n2)=O)c1 86126,c1(C(=O)NC2(C)CCCN(C(C3N=C(C)SC3)=O)C2)cc2cccc(C)n2n1 86127,c1(C(N2CC(C(=O)OC)OCC23CC3)=O)[nH]nc2c1COC2(C)C 86128,C12CCc3nc(sc3C1)NC(=O)C(=O)N2.CN1CCN(CCCN)CC1=O 86129,c1(C(=O)NCCN(C(c2n(CC(C)C)ncc2)=O)C)ccn2cnnc2c1 86130,c1(C(=O)NC2C3CN(C(c4c(C=C)cnn4C)=O)C2C3)c[nH]c2c(C)cccc12 86131,n1(CC)nc(C)cc1C(N1CCCC1C(C)NC(=O)C(COC)OC)=O 86132,C1(C(=O)NCC(CCN)O)CCN(CC2CC3CCC2C3)CC1 86133,N1(c2ncc(CCC)cn2)CC(F)(F)CC1(C)CNC(c1occc1C1CC1)=O 86134,Cc1nc(Cl)c(C)c(=NCC2(C)CCCN(C(c3coc(C(F)F)n3)=O)C2)[nH]1 86135,c1(CC2C(NC(=O)NC(c3ccc(C)o3)CC)CC2)n[nH]c2c1CCC2 86136,N1(CCC#C)CCC(C(N2CC(O)(CNC(c3ncoc3C3CC3)=O)C2)=O)CC1 86137,CN(C1CCSc2ccc(Br)cc21)C(N1CCC(CO)CC1)=O 86138,C1(C(=O)NC(c2nc(C)sc2)C)CCCN(CC2(O)CCC2)C1 86139,C1(C(=O)NC(C)C(C)(C)NC(=O)CSCC(F)(F)F)COC2(CCC2)CO1 86140,C(CSC)(C(=O)N1CC(CC(C)NC(=O)COC2CCOC2)C1)OC 86141,c1(C(N(C(C(=O)NC(CO)CO)C)C2CC2)=O)ccc(=O)n(C)c1.C=CCCC=C 86142,c1(CC)ccc(C(=O)NCCCNC(c2cc(=O)c(C)c[nH]2)=O)c(N)c1 86143,c1(CC)ncncc1C(=O)NCc1ccc(C(=O)N(C2CCOC2C2CC2)CC)o1 86144,CCC(C)(C(=O)NCC1CC(NC(=O)Cc2cccnc2F)CC1O)OC 86145,n1(C)cc(C(=O)NC2(CC(=O)N)CCC2)cn1.CC(C(=O)N(C)C)C1CCC1 86146,C1(C=O)CC2(CCC2)CO1.S(=O)(=O)(CC(=O)NCCC1(CO)CC1)NC 86147,CCCC(CCC)=CC(N1CC(C(=O)NC2CCC=CCC2)C(F)C1)=O 86148,c1(C(N2CC3C(CNC(CCN(C)CCO)=O)(CC3)C2)=O)nc[nH]c2ncnc1-2 86149,C1(NC(c2ccc(-c3ncon3)cc2)=O)C2CCC1N(C(=O)CC1=CCCC1)C2 86150,c1(C(=O)NCC(C)(C(C)C)NC(c2ccn(CCC)n2)=O)ccnc(F)c1N 86151,C1(CC(=O)NCCNC(=O)C2CC2)(CO)CCN(C(C2CC(=O)CS2)=O)C1 86152,c1(CC(=O)NCC(CO)NC(C2CCC3(CCC3)C2)=O)c[nH]c2ncccc12 86153,n1(CC(=O)N(C2CCN(C(c3scnc3Cl)=O)C2)CC)cc(C#N)cn1 86154,C#CC(C)N=C(NCC(C)(C)C)NC(c1ccc(C(C)C)cc1)COC(C)=O 86155,C1(C)(C(=O)NCCCC(C)NC(C2CC3CCC2C3)=O)CCN(C)CC1 86156,C1(NC(C(C)=C(CC)C)=O)CN(C(=O)CSCc2ncc[nH]2)CCC1C(F)(F)F 86157,Cc1nc(=N)[nH]c(C)c1C(N1CCC(NC(c2ocnc2C)=O)C(C)C1)=O 86158,c1(C(=O)NCC2C(NC(c3c(C)c(N)cnc3)=O)CC2)cnc2[nH]cncc1-2 86159,N1(C(CN(C)C)=O)CCCC(N2CCN(C(=O)CC3CCCC34CC4)CC2)C1 86160,C(=O)(CCCCN(C(C(=O)NC1(C)CC1)C1CCOC1)C)OC 86161,N1(CC(=O)NCCC(C)NC(=O)CCc2cncnc2)CCC(NC(N)=O)CC1 86162,C(=O)(C1COc2ccc(Cl)cc21)NC(CC=C)CNC(c1ccsc1OC)=O 86163,N1(C(C2CCCN(C)C2)=O)CC(C2CCCN(C(c3cc(Cl)on3)=O)C2)C1 86164,c1(NC(c2c(F)ccc3c2OCO3)=O)ccc2nc(OC(F)F)[nH]c2c1 86165,C1(CC)CN(C(C2CC(F)C(=O)N2)=O)CCN1C(=O)Cc1cc(C)ccc1F 86166,O(NC(=O)CC(C)(C)NC)CCCCC.C1(=O)CC(C)CC1 86167,c1(SCC2(C(=O)NC(C(C)O)(C)C)CCCC2)cccc(C(F)(F)F)c1 86168,Cn1nc2c(c1C(=O)Nc1cnccc1I)CN(C(C1CCCCO1)=O)CC2 86169,CC(C)C1=NOC(C(=O)NCC=C2CCN(C(C3CC(C4CC4)C3)=O)CC2)C1 86170,c1(-n2cc(C3CN(C(=O)CC4CSC4)CC3O)nn2)cc(F)cnc1Br 86171,CCC(C)(C)C(=O)NCC1(F)CC(NC(c2ccc(C(F)(F)CF)cc2)=O)C1 86172,C1(NC(C(c2ccc(C)cc2)=O)=O)CN(C(=O)CC23CCCC2C3)CC1(C)C 86173,c1(C(=O)NC2CC2CNC(c2cc(C(=O)OC)[nH]c2)=O)c(C)[nH]c(C(C)=O)c1C 86174,C(=O)(C(C)CC(F)(F)F)NC1COCCN(C(c2c(OC(F)F)cc(C)s2)=O)C1 86175,N1(C(C2CC(OC)C(OC)C2)=O)CCOC2(C1)CN(C(=O)C=Cc1cscn1)C2 86176,Cc1c(CC(=O)NC(C)(CNC(=O)CN(CC(C)(C)C)C)C(C)C)cnn1C 86177,c1(-n2cc(C(C)NC(c3ccccn3)=O)nn2)ccc(S(N)(=O)=O)cc1 86178,C1(C)(CC)CC(C(=O)NCCCN(C(=O)CC(=O)NCC(F)(F)F)CCO)C1 86179,c1(C(N(CC(CNC(C(CC)CCOC)=O)O)C)=O)occ2c1CCCC2 86180,c1(C(=O)NCC#CCNC(C(COC)C)=O)cc(Cl)c(OC)c(Cl)c1 86181,C1(C(=O)NC(C)CNC(c2cnc3cccnc3c2)=O)CCCCC1P(C)(C)=O 86182,S(=O)(=O)(c1cccc(C(F)(F)F)c1)N1CCC(O)(CC)C1 86183,N1(C(c2c(C#N)ccs2)=O)CCCCCCC1C(=O)NCC12CC(CCO1)C2 86184,N1(C(C(=O)NC2CC2)=O)CCC2(N(C(=O)Cc3ccsn3)C)CC2C1 86185,c1(OC)ccc(C(=O)NC2CCC(NC(c3ccncn3)=O)C2)c2ccccc12 86186,Cc1cccc(C(F)C(=O)N2CCC2CNC(=O)CNc2ccc(F)cc2)c1 86187,C1(n2c(CC(C3CC(C)C3)NCc3cnn[nH]3)nnn2)CCCCCC1 86188,c1(C(N(CC(CC)NC(C2C(C)(C)C2(F)F)=O)C)=O)ccc2ccnn2c1 86189,N1(C(c2n(C)c(S)nn2)=O)CCC2(CC1)CN(C(C1(C)CCC(=O)C1)=O)C2 86190,C(C)(C)(CC(=O)NCCN(CCCN(C)C)C(=O)Cn1cc(C2CC2)nn1)SC 86191,C=Cn1ncc(C(=O)NCC2(C(=O)NC3(C)CC3)CC23CCC3)c1N 86192,N1(C(c2cc(C)on2)=O)C2CCCC1CC(NC(c1ncc(Br)cc1O)=O)C2 86193,N1(C(c2n(COC)ncc2)=O)CCC2CN(C(c3ncoc3C(F)(F)F)=O)C2C1 86194,C1(C)(C(N2CC(F)(C(=O)NCC3(CC=C)CCCC3)C2)=O)CC(C)=NO1 86195,C(=O)(C(CCSC)SC)N(C(CNC=O)C)CC.C1(CCC)(OC)CCOCC1 86196,N1(C(c2c(C)nncc2)=O)CCC(C)(CN=c2[nH]nc(C(N)=O)s2)CC1 86197,C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC(C)C(CNC(C2CN3CCCC3CO2)=O)C1 86198,C1(C(=O)OC)CC2(CCCCCCC2)CN1C(=O)CSc1cc(C#N)ccc1Br 86199,C1(C(=O)NC2C(NC(c3c(C)cccc3C)=O)COC2)CC2CCC1C21CC1 86200,C1(C(=O)NC2CC(CNC(c3ccc(OCCO)cc3)=O)C2)CCC(F)(F)CC1 86201,c1(-c2nn(CC(C)C)c(-c3cccc(OCCOCCF)c3)n2)cccc(C#N)c1 86202,C1(CN(C(CCC)=O)CC)CC(F)(F)CN1C(=O)C(O)Cc1ccccn1 86203,c1(N2CCC(CCNC(C)(C)CNC(=O)NCCCO)CC2)cc[nH]c(=N)n1 86204,Cc1nn(CC(=O)NCC(C)(O)CNC(=O)CN2CC3CC3C2)c(=O)n1C 86205,C1(C(=O)NCCC(=O)OC)C2CCC(C2)N1C(c1ccc(C)nc1O)=O 86206,c1(C(=O)OCC)c(C)ccnc1CNCCc1cc(CC)no1 86207,N1(C(C(C)c2cccs2)=O)CC(C2CCCN(C(C3(C4CCC4)CCC3)=O)C2)C1 86208,c1(OC)ccc(C(N2CCC2CNC(c2nc(C)n(C)c2C)=O)=O)cc1F 86209,C(=O)(CS(=O)(=O)C1CCCC1)NCC1N(C(c2ccc(N=[N+]=[N-])cn2)=O)CC=C1 86210,CC(C)(CNS(C)(=O)=O)C(=O)NCCO.C1(N(C(=O)CNC=O)C)CCCCCC1 86211,C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCC(NC(C(CCC)OC)=O)C1C 86212,C(=O)(CC(=O)NC(C)(C)C)OCC1CCCN1C(c1csc(-c2ncc[nH]2)n1)=O 86213,CC(C)C(O)C(F)(F)C(=O)N1CC2CCC1C(CNC(=O)CCOCC(F)F)C2 86214,C1(C(=O)NC2(CO)CN(C(C(CC#C)C3CC3)=O)C2)CC2(C1)CC2(F)F 86215,C1(C(=O)NC(C)(C)CCNC(=O)C(F)(F)C2(O)CCC2)CCCC(N(C)C)C1 86216,CCC(CC(=O)NCC1(O)CCN(C(c2ncoc2Br)=O)C1)C1CCC1 86217,c1(CC)cc(C(=O)NC2CN(C(C3CC(n4cccn4)C3)=O)CC2C)oc1CC 86218,C(=O)(C(CC1CCCO1)C(F)(F)F)NCCCNC(CSc1n(C)cnc1)=O 86219,c1(C(=O)NCCC2N(C(C(C=C)OC)=O)CCOC2)cc(C)c2occc2c1 86220,CCC(C(=O)N(C)CCn1cc(C2CCCOC2)nn1)N(C)C 86221,c1(OCCC(=O)N(C2CCS(=O)(=O)C2)CC)ccc2c(c1CSC)OCO2 86222,Cc1ccnc(CNC(C2COCCC2NC(=O)CC2C=CCC2)=O)c1 86223,c1(CNC(=O)C(=O)Nc2cc(CCO)ccn2)cc(F)c(NS(C)(=O)=O)c(F)c1 86224,C1(NC(CCC(=O)NCC)=O)CN(C(c2ccc(N)c(F)c2)=O)CCC1(C)C 86225,c1(CCn2cc(CCC(C)O)nn2)cncc(NC(C2(C)COCCO2)=O)c1 86226,C=C1CC2(C1)CN(C(=O)C(CCCOC)NC(C1CCCOCC1)=O)C2 86227,C1(NC(C2CN(C)C(=O)C2)=O)CCS(=O)(=O)C12CN(C(C1(CO)CCCC1)=O)C2 86228,C1(NC(C2C(OC)C2)=O)CCCCC1C(=O)NCc1ccccc1OC(F)(F)F 86229,c1(C(N2CC(NC(CC(C)(C)C)=O)C3(C2)CC3)=O)cc2ccc(F)cc2[nH]1 86230,C=CCC(C)(C)CC(=O)N1CCC(C)CC1CNC(C1CCCO1)=O 86231,c1(C(N2CCCC2CNC(C2CC(F)(CO)C2)=O)=O)ccc2c[nH]nc2n1 86232,c1(C(N2C(CN(C(CS(CC)(=O)=O)=O)C)CCC2)=O)cc(Cl)c(C)cc1[N+](=O)[O-] 86233,c1(C(=O)NCCCC(=O)NCC2CC=CCC2)cc(O)ncc1F 86234,CC(C)CC(C)C(=O)NCC(C)(Cn1cccn1)NC(c1csnc1Cl)=O 86235,Cc1cnc(C(=O)NC(C)(C)CN(C)C(c2ccc(C(C)(F)F)nc2)=O)cc1C 86236,N1(C(C2C(NC(c3c(C)cco3)=O)C2(C)C)=O)CCCC(C)(F)C1 86237,c12cccnc1NC2.c1(C2N(C(C)C)CCC2)ccc(N2CCOCC2)cc1 86238,C1(NC(CC(C(=C)C)OC)=O)CN(C(=O)CC2(O)COC(C)(C)C2)CCC12CCC2 86239,C1(c2nn[nH]n2)(NC(c2ccsn2)C2CC2)CC2COC1C2 86240,C1(CNC(c2[nH]cc(C)c2)=O)(NC(=O)CCSCC(N)=O)CCCCC1C 86241,C(=O)(C1CCCc2ncnn21)NCC(C)NC(c1cnoc1-c1ccccc1)=O 86242,c1(OC)ncc(C(=O)NC2COCCC2NC(c2cc(C3CC3)cs2)=O)c(C)n1 86243,N1C(NCC(C2(O)CCCOC2)(C)C)=NCNCC1C=C.OC 86244,n1(CC)nnc(C(=O)NCC(CNC(=O)C=CCNC(N)=O)CO)c1C.C(C)(C)(C)O 86245,c1(CCC(=O)NC2C(SC)CN(C(=O)C3=CCSC3)C2)ccc(C)cc1C 86246,c1(Cc2cn(C3CCN(C(C=COCC)=O)C3)nn2)c(Cl)cc(Br)cc1Cl 86247,c1(-c2c(C(C)NC3(c4ccccc4)CCOCC3)nccc2)ccc2c(c1)CCCC2 86248,c1(COC)ncsc1C(=O)NCC1CN(C(=O)C(F)CC2CCOCC2)C1 86249,c1(NC(=O)Cc2csc(C)n2)nccc(=NC(C)c2ccccc2CC)[nH]1.CC 86250,C1(NC(CC(C)(C)O)=O)CC2CC(C1)N(C(c1cnncc1C(F)(F)F)=O)C2 86251,CCCC(C(=O)NCC1CCN(C(C2CC2CN(C)C)=O)C12CC2)S(N)(=O)=O 86252,c1(C(N2CCN(C(C3=CCCCC3C)=O)CC2C)=O)coc(S(C)(=O)=O)c1 86253,CC(CNC(c1c[nH]nc1CCNC(C1CC(=O)C1)=O)=O)CC(C)O 86254,C1(NC(c2cc(Cl)on2)=O)CN(C(C2CCC=CCCC2)=O)CCC12CCC2 86255,c1(C(N(CCCOCCN(C(C2C(CCC)C2)=O)C)C)=O)nc(OC)ccc1F 86256,c1(C(=O)NC2CC2)ccncc1N.C1(=O)C(C2CCCC2)N1CC(=O)NCC(C)C 86257,C1(NC(c2ccc(OC)nn2)=O)(CNC(=O)C(C)(C)C(N)=O)CC2CCC1CC2 86258,C1(C(=O)NC(c2ccc(F)cc2)C)COCCN(CC2COC(=O)N2)C1 86259,c1(NC(=O)NCCc2nc(CCOC)cs2)ccccc1C(C)=O 86260,c1(C(=O)NCCN(CCC)C(C2CC2(C)Br)=O)cn[nH]c1 86261,c1(C(N(CCNC(C2(C)CCC(=O)C2)=O)CC2CC2)=O)ccc2ccccc2c1 86262,C1(CNC(C=C(C)C(C)(C)C)=O)CC2CN(C(C3CC3C(=O)NCCO)=O)CC12 86263,c1(N2CCCC(NC(c3cncc(Cl)c3Cl)=O)CC2)ncnc2ccc(O)cc12 86264,CN1CCc2[nH]nc(C(=O)Nc3ccc(C(F)(F)F)nc3)c2C1 86265,c1(C(N2CCC(NC(C(C(C)C)OC)=O)C23CC3)=O)ccc2c(C)noc2c1 86266,CCC(CCC(=O)N(c1ccccc1)CC)NC(=O)CC1CCCSC1 86267,N(C1COc2ccc(Cl)cc21)C(=O)NC(Cc1ccccc1Br)CO 86268,c1(C(=O)NC(C)CC2CN(C(=O)C=Cc3cocn3)C2)cnc(OC(F)F)c(C)c1 86269,c1(C(=O)NCCN(C)C(c2ccc(F)nc2)=O)cnc(O)c(Br)c1 86270,C(C1C(C(=O)NCCC(C)NC(c2cccnc2C(F)F)=O)C1(C)C)=C(C)C 86271,c1(OC)ccc(C)cc1C(=O)NC1CC12CC(NC(=O)Cc1csc(S)n1)C2 86272,C12(CNC(CN(C)C)=O)CC1CN(C(c1ccccc1Cn1cccc1)=O)C2 86273,N1(C(c2cncc(SCC)n2)=O)CCC(COC)(NC(=O)CCC(=O)NC)CC1 86274,C1(=CC(=O)N(C(C)Cc2ccccn2)C2CC2)CCN(Cc2cnc(Cl)nc2)CC1 86275,C(CCC(=O)N(C)CCN(C)C(c1ccco1)=O)NC(C1C(=C)CC1)=O 86276,N1(n2ccncscc2)CC(F)(F)CC1CNC(=O)C=CC(C1(O)CCOC1)=O 86277,C(=O)(CCC(=O)NC1CC(C(=O)C=CC(N2CCC(CC(=O)OC)C2)=O)C1)OC 86278,C(C)(C)(CCCC(=O)NCc1cn[nH]c1)NC(c1n(CC#C)ccc1)=O 86279,C=C(Cl)CCC(=O)N(CC(C)NC(=O)C(c1ccc(O)cc1)OCC)CC 86280,c1(C(N(CC(CC)NC(=O)C(C)SC(F)(F)F)C)=O)ccc(OC)c(OC)n1 86281,c1(C(=O)NC(C)CC(C)NC(=O)C(C)CC(F)(F)F)ccc2nnc(S)n2c1 86282,c1(C(=O)NC(CNC(c2cocn2)=O)C2CCC2)cc(Cl)nnc1O 86283,c1(C(=O)NC2(CN(C)C(c3cn[nH]c3)=O)CC2)cccc(O)n1 86284,c1(-c2ccc(C(N3CCC(c4nncs4)CC3)=O)cc2)nc(C2=NOCC2)no1 86285,c1(N(C)C)cn(C)c(C(=O)NCC(C2CCOC2)NC(c2cocn2)=O)n1 86286,C=C(CNC(c1ccoc1CC)=O)CCNC(c1occc1C(C)C)=O 86287,N1(C(c2[nH]cc(C)c2)=O)CC(CC(=O)N(C2CCOC(C)C2)C)CC1(C)C 86288,c1(N2CCCC(CC)CC2)nc2ccc(Cl)cc2c(=NCCN2CCC(C)C2)[nH]1 86289,C1(NC(C(CSC)(C)C)=O)CN(C(=O)CN(C(=O)COC)C)CC1O 86290,c1(OC)cc(C(=O)OCC2CCCN2Cc2cc(C)on2)ccc1N 86291,c1(C(=O)NC2CCC2NC(=O)C2CC2)csnc1Cl 86292,n1(CC)nnc2cc(C(N3CCCC(C)(CNC(c4ccc[nH]4)=O)C3)=O)ccc12 86293,CCCCC(C(=O)NC1CN(CCN(C)CCCOCCNCC)C1)N(C)C.CC 86294,CC(CCCc1cn(Cc2n[nH]cc2C2CC2)nn1)C(=O)N(CC(=O)O)C1CC1 86295,C(=O)(C1=C(C)Oc2ccccc2C1)N1CCC(CNC(CC(=O)NCC#C)=O)C1 86296,N1(C(C(C2N(C(C(CC(C)C)OC)=O)CCC2)(C)C)=O)CC2(CCNC(=O)O2)C1 86297,N1(C(CCCC#C)=O)CCCC(C2CCN(C(c3cscc3Cl)=O)C2)C1 86298,C1(C)(CCC(=O)N(CC(C)N(C(=O)C(c2ccn(C)n2)C)C)C)OCCO1 86299,N1(C(c2c(CC)occ2)=O)CCC(C(=O)NCC(=O)N(C)C)C12CCC2 86300,N1(C(C23CC(C2)C3)=O)CCC12CCN(Cc1cccc(F)c1O)CC2 86301,N1(C(c2c(CC)c(F)ccc2)=O)CCCN(C(=O)C(c2cccnc2)C)CC1CO 86302,c1(OC)ccc(CCn2nc(-c3cccc(F)c3)nc2CCS(C)=O)cc1 86303,C1(C(=O)NCCCC2N(C(C(C)=CC)=O)CCC2)C(C=C(C)C)C1(C)C 86304,c1(C(=O)NCCN(C2CCCC2)C(c2ccccc2F)=O)ncccc1Br 86305,c1(C(N2CCN(C(C(C)SC)=O)CC2C)=O)ccnc2c1CC(=O)N2 86306,C(=O)(C(CC1CC1)NC(C1CCNC1=O)=O)NC(c1ccco1)C 86307,c1(C(N2CCN(c3cnc4cccnc4n3)CC2)=O)cccc2ccccc12 86308,N1(C(C(C)(C)OC(C)=O)=O)CCC(CO)(CNC(C2CCC3CCC23)=O)C1 86309,c1(NC(=O)NCC)cccc(C(N2CC3CC3(CNC(=O)C#CCOC)C2)=O)c1 86310,c1(CNc2ccc(NC3C(C)CN(CC(F)(F)F)C3)cc2)cc(Cl)cc(Cl)c1.OC 86311,c1(C2N(CC(N3C(N4C(=O)OCC4)COCC3)=O)CCC2)ccc(F)c(Br)c1 86312,N1(C(C=Cc2n(CC)ncc2)=O)CC2CC(C1)CN(C(c1cnc(C)cn1)=O)C2 86313,CC1(N(C(C2(F)CN(Cc3cccc(F)n3)C2)=O)C2CC2)CCCCC1 86314,C1(SCC(=O)Cc2cccc(F)c2)COc2ccc3ccccc3c2C1 86315,Cc1c(C(=O)NCCC(C)NC(c2nc(F)ccc2Cl)=O)cc(F)cc1Br 86316,CCCCCCCS(=O)(=O)CC(=O)N(C)CCN(C(=O)C1=C(CC)OCCS1)C 86317,N1(C(C(=O)NC)C#N)CCN(C(=O)COc2ccc(-c3nnc(C)o3)cc2)CC1 86318,n1(CC(=O)NCC2OCCN(C)C2)ccc(=NC(=O)C2CC2F)nc1O 86319,C1(C(N2C(CNC(CC3(S(N)(=O)=O)CC3)=O)CCC2)=O)COc2ccccc2O1 86320,c1(OC)cc(O)ncc1C(=O)NC(CNC(c1nc(C)oc1C)=O)CC(C)C 86321,C(=O)(CC(O)C(C)C)NC1(CC=C)CCN(C(=O)C=CC2CCCO2)C1 86322,C(C(CNC(=O)CCNC(=O)OC)S(C)(=O)=O)NC(C=CC(CC)C)=O 86323,CCC(C(=O)NC1CN(C(C2(c3cccc(Cl)n3)CC2)=O)CC1O)C(C)(C)CC 86324,C1(NC(c2c(C)csc2Cl)=O)CCN(C(=O)CSCc2ccncc2)CCC1CO 86325,N1(C(C2C=CCCC2)=O)CCC2(CC1)CCN(C(C1CCC(F)(F)CO1)=O)C2 86326,c1(C(=O)NCCC(C)(C)NC(c2cc(=NC)[nH]cc2)=O)csc(=NC2CC2)[nH]1 86327,CS(=O)(=O)c1ccc(F)c(C(=O)NCC2CN(C(=O)NS(C)(=O)=O)C2)c1F 86328,C1(CN(C)C(c2cnn(C3CCC3)c2)=O)CN(C(C2CC(F)C(=O)N2)=O)CCO1 86329,c1(NC)ccc(C(=O)NC(C(=O)NCc2cccc(Cl)n2)C(C)C)nc1 86330,CC1OC2(CNC(=O)C(=O)NCC(F)F)CC1(NC(C1CCN(C)C1)=O)C2 86331,C1(NC(CC(C)(C)OC)=O)CCN(C(C2CCC(F)(F)CC2)=O)C12CC2 86332,C=CCC(C)(C(=O)NC1(CCNC(=O)C(C)CC)CCC1)N(C)C 86333,C(=O)(C1Cc2ccccc21)NC1CN(C(C=C(C)C)=O)CC12CCC2 86334,c1(C(=O)NC2C(NC(c3c(C)noc3C3CC3)=O)CC2)onc2ccccc12 86335,C1(C(=O)NC(C(=O)NCc2n(C)ncn2)c2ccoc2)CCCC(C#N)C1 86336,c1(C(N2CCC(NC(CC(=O)N(C)C)=O)CC2)=O)noc2c1CCCC2 86337,CC1CCCCCCN1C(C(=O)NCCOC)C1CC1.CCC1CC1 86338,S(=O)(=O)(CCC(=O)N1CCCC(N2CCN(C(C3CC=CCC3)=O)CC2)C1)NC 86339,N1(C(CSCC(=O)OC)=O)CCC(C)(F)C1.C1(Cc2ccco2)C(=O)N1 86340,C1(CNC(C(CSC)(C)C)=O)CC(C)CN(C(=O)CC2CC(F)C2)C1 86341,C(CC(=O)NOCC1(O)CCC1)(C(F)(F)F)NC(C(C)NC(CC)=O)=O.SCC 86342,C(=O)(C1=CCCC1(C)C)NC(C)CCNC(c1cc(OCC(F)F)ccn1)=O 86343,C1(OC)(OC)CCCC(NC(=O)C2=CCN(CC(F)(F)F)CC2)C1 86344,C1(CNC(C2CC(C)N(C)C2)=O)CC2(CCN(C(c3ccnn3C)=O)CC2)CO1 86345,Cc1nnc(NCC2CCC(NC(=O)Cc3nc(C)c(C)s3)C2)c(C#N)c1C 86346,O(NC(=O)C(C)(C)CCCNC(=O)CCC(C)CC)C(C=C)C 86347,c1(CN2C(C(=O)NCc3ncc(-c4ccccc4)[nH]3)CC3CC32)ccc(I)cc1Cl 86348,C1(C)(NC(C2(C(C)C)CC2)=O)CN(C(=O)OC(C)(C)C)C1.C1(=O)CN1 86349,C1(F)(C(N(C)CCOCCNC(c2cc(C3CC3)ns2)=O)=O)CCS(=O)(=O)C1 86350,c1(OC)ccnc(N2CCCC(CN(S(=O)(=O)C(F)(F)F)C(=O)CNC(=N)N)C2)n1 86351,C1(CC(=O)NC(C(=O)NCC(N2CCCCC2)C)CO)CCC(C)(C)C1 86352,Cc1ccc(CN2CCOCC(C(=O)NCC3=CCCCC3)C2)c(C)c1 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86686,c1(C(=O)NCC(=C)CCNC(c2cc(CC3CCC3)c[nH]2)=O)oc(C)cc1C 86687,C1(C(=O)NC2CCC(C)N(C(c3csc(Cl)c3)=O)C2)CCC2(CC1)CC(O)C2 86688,C1(CN(C(=O)CC2CC(C)(C)CO2)C)COCCN1C(=O)CC1CSCCS1 86689,Cc1nn(C)c(C)c1C(=O)N(C(C)CN(C(=O)Cc1ccsc1)C(C)C)C1CC1 86690,Cn1c(C(=O)NCC(CNC(=O)CC2CSC2)C(F)(F)F)cc2ccccc12 86691,N1(CC)CCOC(C(=O)NC(C)CNC(=O)C(c2ccc(F)cc2)C2CC2)C1 86692,C=C1COc2c(NC(=O)C(C)C(F)F)cnn2C1.N12CC3(CCC(CC3)C1=O)C2 86693,C1(NC(CCC#CC)=O)C2CCN(C(=O)CCn3c(C)csc3=O)CCC12 86694,n1(CCC2(OC)CCC2)c(N(C)CCOC(C)C)nnc1Cc1nc(C)no1 86695,C1(CNC(C=CC(CC)C)=O)CCCCN1C(=O)CCNC(=O)COCC(C)C 86696,c1(C(=O)NCCC(=O)NCC2CC2C(=O)N)cccnc1S.c1(C)ccsc1 86697,C1(F)(CNC(C2CC=CCC2)=O)CN(C(=O)C(F)(F)c2csc(Cl)c2)C1 86698,c1(NC(C2CCN(C(=O)CCF)C2)(C)C)cnc(C(=O)OCC)s1 86699,N1(C(C(CNC(C2CCCC(F)C2)=O)N(C)C)=O)CCn2cncc2C1 86700,c1(SC)ccc(NC(=O)NCCC2COC(C)(C)CO2)c(N(C)C)c1 86701,c1(CC(C)C)ccc(C(N2CC(N(C)C(C3CSCCS3)=O)C(F)C2)=O)cc1 86702,c1(C(C(N2CCC(CNC(C(CC)(C)C)=O)C2)=O)(C)C)ccc2ccccc2c1 86703,N1(C(C(C)=C(CC)C)=O)CCN(C)C(C(=O)NC2COCCO2)C1 86704,C1(C(N2CC(CC)N(C(=O)COCCOCCO)CC2)=O)CCC12CCOCC2 86705,C=CC1CN(C(=O)C(C(C)C)NS(C)(=O)=O)CC1NC(C1CC(C#N)C1)=O 86706,n1(CCCSCC)nnnc1C(c1cnccn1)NCC(C)C(C)C 86707,C(=O)(C#CC1CCCOC1)N1CCC(C)C(NC(c2cc(O)cnc2N)=O)C1 86708,C1(C(=O)OC)CCC(C)(C)N(C(=O)NCC2CCP(C)(=O)CC2)C1 86709,c1(C(N2CC(NC(CS(=O)(=O)N(CC)CC)=O)C(C)C2)=O)nn(C)c(=O)cc1C 86710,N1(C(COCc2cc(C)on2)=O)CC(O)CC1(C)C(=O)N(CCCF)CCO 86711,c1(CCC(=O)NCC(C)(C)NC(c2cncc(F)n2)=O)ccc(C#N)cc1 86712,O=C(C1=NOC2COCC12)NCCCCCC(=O)N1CC(O)(c2cnn[nH]2)C1 86713,N1(C(c2ccc(CNC(Cn3ncc(C)c3)=O)cc2)=O)CC(O)CC12CCC2 86714,c1(CC)cc(C(=O)NC2COCCN(C(C3CCCC(C)(C)C3)=O)C2)c(C)nn1 86715,C1(C(N2CC(C#C)(F)C2)=O)CC2C=CC1N(C(=O)CC1C(C)(C)C1(C)C)C2 86716,O=C(CCS(=O)(=O)c1ccccc1)NCC1CN(C(=O)Cn2ccnn2)C2CC12 86717,c1(CNC(c2cnn(C)c2)CC)cccc(CC(F)(F)F)c1 86718,C(=O)(C(CCCCCCO)N1CCC1CC(C)C)NCCC 86719,c1(C(=O)NCCN(C(c2[nH]c(O)nc2C)=O)CC)oc(COC)cc1C 86720,C1(NC(CC)=O)CCCC(NC(c2cc(OC)cc(OC)c2)=O)CC1 86721,N1(C(c2cnc(CC)nc2)=O)CCCC(C)(C)C1C(=O)NCC(F)C(C)(C)O 86722,c1(N2C(N(C)Cc3ccccc3)CC(O)C2)ncnc2ccnn12 86723,c1(NCC(N2CCC(CC(C)NC(CSCC)=O)CC2)=O)cc(C)c(Cl)c(C)c1 86724,C1(CNC(C(CC)NC(c2n[nH]cc2Cl)=O)=O)C2CCCCCC12 86725,N1(C(C(CC)(C)OC)=O)CCC2(C1)CN(C(c1ccc3nn[nH]c3n1)=O)CCO2 86726,N1(C(COC(C)(C)C)=O)CCC(CCNC(C2C=CCCC2)=O)C(F)(F)CC1 86727,c1(C(N2CCCC(OC3CCCC4CCCN34)C2)=O)[nH]c2ccc(Cl)cc2c1Cl 86728,C1(F)(C(=O)NCCCN(C(C(C)OCCC(C)C)=O)CCO)CC1(F)F 86729,CC1(C)CCOC1CC(=O)NCC1(O)CCN(C(=O)CCCN2CCCCC2)C1 86730,c1(C(=O)NCC(CCOC)NC(=O)C(C)OC)cncc2nc(C)[nH]c12 86731,C(C)(C)(C(C)CC(=O)NCC(C#N)CC)NC(CC(C=C)(C)O)=O 86732,C(C(=O)NCc1cccc(C)c1)(C(=O)OC)OC(C1C(OCC)C1)=O 86733,c1(C(=O)NC2C(OC)CN(C(c3csc(CC(C)C)n3)=O)C2)cnc(C)c(C)c1 86734,CP(C)(=O)c1cncc(C(N2CCCC(NC(=O)COC3CCOC3)C2)=O)c1 86735,N1(C(C2CNC(=O)N2)=O)CC(CNC(c2cnccc2Cl)=O)C2(CCC2)C1 86736,C1(NC(CCc2cc(C(=O)OC)sc2)=O)CCCC(NCCOC(C)C)C1 86737,c1(CN2CCCC(CC(=O)Nc3cc(F)ccc3I)C2)ccc(F)cc1[N+](=O)[O-] 86738,N1(C(c2ccnc(F)c2)=O)CCC2C1CCN2C(c1cc2cccnc2[nH]1)=O 86739,c1(OC)cc(F)c(C)cc1NCc1ccnc(Br)c1Br 86740,C(CCCC(=O)N1CCC(O)(CN(C)C(C2CCCN2CC)=O)C1)OCC 86741,N1(C(C2(C#N)C(C)C2)=O)CC2CCC1CN2C(c1nc(-c2ccccn2)cs1)=O 86742,C(C(CC(=O)N1CCC(CC2CC2)C1)NC(C1CCC(C)(C)C1)=O)OC 86743,C1(O)(C(C)NC(CCN(CCC)C)=O)CCN(C(=O)CNC(=O)C(F)(F)F)C1 86744,Cn1cnc2c1CCNC2C(=O)NCC12CCC(C1)C(O)C2O 86745,C1(NC(=O)C=CC(N2CCCC2)=O)CC(O)CN(C(c2csc(C3CC3)n2)=O)C1 86746,Cc1cc(=O)c(C(=O)NC2CCC2NC(=O)Cn2nc(C)ccc2=O)c[nH]1 86747,C(=O)C(S(C)(=O)=O)C1CC1.CC(O)CCN(C1CC1)Cc1ccco1 86748,C1(C2C(CC)CCN2C(c2coc(C(F)F)c2)=O)(CNC(N)=O)CC2CCCC12 86749,C1(CNC(c2c(CC)oc(C)c2)=O)CCCC2CN(C(c3sccc3Cl)=O)CC12 86750,CC(C)CC(O)C(=O)NCC1(F)CCCN(C(c2ccc(Br)c(F)c2)=O)C1 86751,Cc1ccc(O)cc1C(=O)NCCC1CC(C(=O)NC2CCCCC2(C)O)C1 86752,C#CCCCC(C)C(=O)N1CC2CCC(CNC(c3cnc(N(C)C)o3)=O)(C2)C1 86753,N12CCC(C13CC3)C2=O.c1(C(C)NC(c2c(COC)cco2)=O)cncc(F)c1 86754,N1(C(C2(CNC(Cn3nnc(C)n3)=O)CC=CC2)=O)CCC(C)(CCO)C1 86755,N1(C(C(Br)=C(C)C)=O)CC2CCC(NC(=O)Cc3cccc(F)c3F)CC2C1 86756,c1(C(=O)NC(C2CCCCN2C(=O)Cc2ccccc2)C)cc2c[nH]cnc-2n1 86757,c1(CC(=O)NCCN(C(=O)C=C2CCN(C)CC2)CC)cc(F)cc(Br)c1 86758,C12(NC(C(C)OCC(F)(F)F)=O)CCCC1CN(C(c1cc([N+](=O)[O-])c[nH]1)=O)C2 86759,N1(C(C(C)=CC)=O)CCC2CCC12CNC(c1c(O)cccc1Cl)=O 86760,C(CCCC(=O)NCC(C)(Cn1cccn1)NC(=O)CCF)SC 86761,C(=O)(CCCCCCC)NCc1c(C(N2C(C=C)CCC2)=O)cco1 86762,c1(C(=O)NC(CNC(CC(=C)Br)=O)C)cn(C)nc1OCC(F)F 86763,C=CC(C)(CC)C(=O)NCCC1(CNC(c2[nH]c(C3CC3)nc2C)=O)CC1 86764,N1(CCOC)CC(C(=O)NC2CCCC2NC(C23CC(CCO2)C3)=O)CCC1=O 86765,C1(NC(CCC2C(C)C2)=O)CCC2(CC1)CN(C(=O)CC1CC3(CCC3)C1)C2 86766,C1(C(=O)NC2CCCN(C(CCn3ccc(C)n3)=O)C2)CN2CCC1(C)CC2 86767,Cc1oc(CNC(c2c[nH]ccc2=O)=O)nc1C(=O)NC1(O)CCSC1 86768,C(=O)(C(C(C)C)NC(C)=O)NCCCN(C(C(C)=CC)=O)C 86769,c1(C(N(CC(CNC(CC2(C(=O)OCC)CCC2)=O)O)C)=O)cc(C)ncc1Cl 86770,N1(C(c2n(CC#C)ccc2)=O)CCC2CC1CN2C(c1n[nH]cc1CC)=O 86771,C(c1ccc(C(C)(C)C)cc1)=CC(=O)N(CCCNC(=O)C(N)=O)C 86772,N1(C(c2c(C)cn(C(C)C)c2)=O)CCN(C(c2ccc([N+](=O)[O-])o2)=O)C2CC12 86773,N1(C(c2cc(OC)ns2)=O)CCSCC1C(=O)N(C)Cc1ncccn1 86774,C1(C(=O)OC(C)C(=O)NCc2cccs2)CCCN1C1CCCCC1 86775,[N-]=[N+]=NC1CCN(C(=O)CC2CCCC2O)C1C(N1CCCN(C(N)=O)CC1)=O 86776,c1(NC(C2CCN(Cc3cncnc3)CC2)=O)cc2cc(Cl)cc(Cl)c2[nH]1 86777,N1(C(C2C(C)CC2)=O)CCN(CC(=O)NCCCc2cnnn2C)CC1 86778,N1(C(C(CC)C)=O)CCC(NC(c2cn(CC3CC3)nn2)=O)C(CO)C1 86779,c1(C(=O)OC)ccc(CC(N2CCC(Nc3cccc(C(C)=O)c3)CC2)=O)nc1 86780,CC(C(=O)N(C)CCN(C)C(C1CC(=O)N(c2ccccc2)C1)=O)C(F)(F)F 86781,C(=O)(C(C)S(C)(=O)=O)N(C(C)C(N1CCCC(CN=[N+]=[N-])C1)=O)C1CC1 86782,C#CCC(CC(=O)N(CC(C1CC1)OC)C)NC(=O)CCn1cccn1 86783,C1(CC(N2CCC(NC(C3(F)CCOC3)=O)C(F)C2)=O)CN2CCN1CC2 86784,c1(C(N2CCN(C(C3CC(C#C)(O)C3)=O)CC2)=O)cc(Cl)c(Cl)n1C 86785,c1(OC)c(C(N2CC3CCN(c4ncncc4Br)C3C2)=O)cccc1[N+](=O)[O-] 86786,c1(C(N(CC(O)CNC(=O)CC23COC(C)(C2)C3)C)=O)c(N)cccc1Cl 86787,C1(CC)C(C(=O)N(CC(C)CNC(=O)C=Cc2ccco2)C)CCN1C 86788,CC1=NNC(=O)C1CCC(=O)Nc1cn(-c2ccc(F)cc2)nn1 86789,N1(C(CN(C(C)=O)C)=O)CCN2CCOCC2(CNC(=O)CCc2cn[nH]c2)C1 86790,C(C(=O)NNC(=O)C#CC1(C)CCCO1)SC.C1CCCCC(=O)Nc2cn1nn2 86791,Cc1noc(C(=O)NCCCC2CCCCN2C(=O)COC2CCOC2)c1C 86792,C1(C(N2C(CNC(C3(OCC)CCSCC3)=O)CCCC2)=O)CCN(C)S1(=O)=O 86793,c1(C(N(C2CCCCC2NC(=O)COCC2CCOC2)CC)=O)cnc(OC)cn1 86794,C#CCCN=C(NCC(C(C)(C)C)OC)N1CCC(CNC(N)=O)C1 86795,Cc1n[nH]c2cc(C(=O)NC(CNC(=O)CCC3CCCO3)C(C)C)ncc12 86796,C(=O)(C(=O)N)NCCNC(C1C(CC(C)C)C1)=O.C(C1CC1)C1CC1 86797,c1(CN(C(C(=O)Nc2ccon2)c2csnn2)CC)ccc(OC)cc1 86798,N1(C(c2ncoc2C(F)(F)F)=O)C2CCCC1CC(NC(C1(O)CCCC1)=O)C2 86799,C(C)(C)(CCCNC(=O)CC1OCCC1C)NC(Cc1cn(CC)nn1)=O 86800,C1(C(C)C)CN(C(=O)C2=NNC(=O)C2)CCCN1C(c1ccc(Cl)cc1)=O 86801,Cc1ccc2c(C(=O)NC(CNC(c3nnccc3C)=O)C(C)(C)C)c[nH]c2c1 86802,c1(C(N(CC(C)N(C(C(CC)OCC)=O)C)C)=O)ccc(-n2ccnc2)nc1 86803,C#CC(CNC(=O)C(C(C)(C)C)n1cc(C2(O)CCCC2)nn1)CC(C)(C)C 86804,S(=O)(=O)(c1ccc(C)c(C(=O)OC(C)C(N2CC(C3CCCC3)C2)=O)c1)NC 86805,n1(CC(=O)NC2CC(NC(CCCn3c(C)ncc3)=O)C2)ncc2ncccc12 86806,N1(C(c2nc(Cl)cs2)=O)CCN(CC2CCCN(C(C34CC(O)C3C4)=O)C2)CC1 86807,CC(C(=O)N1CC(n2cc(-c3c(F)cccc3Cl)nn2)CO1)C1CC1 86808,c1(C(=O)NC2CC(C(CC)NC(C3CCCCS3)=O)C2)cccn2cc(C)nc12 86809,c1(NC(C2N(C(N)=O)CC(O)C2)=O)n[nH]c2c(F)cccc12.C12CCN(CC1)C2 86810,N1(CCC(C)(C)CC(=O)O)CCC2(CCC(Cc3ccccc3)O2)CC1 86811,N1(C(C(C)n2cnnn2)=O)CCCC2(CCCN2C(c2cc3occc3s2)=O)C1 86812,CCC(COC)C(=O)NCCC(C)N(C)C(C1CC=CCC1)=O 86813,C1(O)(CNC(C=CC(=O)N(C)C)=O)CCN(C(C2CC(=O)CO2)=O)CC1 86814,O(NC(=O)C(c1ccoc1)NC(c1cc(C)sn1)=O)CCCC=C 86815,C1(NC(C2CCN(C(C)=O)C2)=O)CC2(CCN1C(=O)CSCC(F)F)CC2 86816,C(c1c(F)cccc1F)=CC(N1CCC(NC(c2c(C)csc2)=O)C1C1CC1)=O 86817,c1(C(N2C(C(=O)Nc3ncccn3)CC3CC32)=O)ccc2nccc(Cl)c2c1 86818,N12CCOC(C)C1NC2=O.C(CCF)OC(C)=O 86819,CCC(CCC(=O)N1CCC(C)(N(C)C)C1)NC(=O)C(c1ccnn1C)C 86820,C(=O)(C#CC1CCCCO1)N1CCCC(CNC(c2c(C)cn(C)c2)=O)CC1 86821,Cc1nccc(CNCC2CCCCN2C(c2cnc(Cl)nc2)=O)n1 86822,C1(NC(C(CC#C)C2CC2)=O)CC12CCN(C(c1ccc(Cl)c(C)c1N)=O)CC2 86823,c1(C(=O)NCCN(C(=O)CCc2cnoc2)CC(C)O)cccc2ccccc12 86824,C=CCCC(C(=O)NC1CCOC(C)(CC)C1)NC(c1ccc(CC)o1)=O 86825,Cc1cnccc1C=CC(=O)NCC1CCCCN1C(c1cnc2n1CCC2)=O 86826,C12(C(=O)NC(c3cccnc3O)C)CCC(NC(=O)Cc3cncs3)(CC1)C2 86827,N1(C(CN2C(C)CCC2)=O)CCCC2(CC(NC(c3cnn(C4CC4)c3)=O)C2)C1 86828,C(=O)(C(COC)CC(C)C)N(CC(CC)NC(c1sccc1C(C)(C)C)=O)C 86829,CC(CC(C)(F)F)C(=O)OCC1OCCCO1 86830,N1(C(CCc2cc(C)no2)=O)CC2CCC(C1)N2C(c1cc(C)c(Cl)cc1C)=O 86831,N1(C(C(CCC)C)=O)CCC2(CC2C(=O)Nc2ccc(O)c(Cl)c2)C1 86832,C12(C(=O)NCc3c(C)nn[nH]3)CCC(CC1NC(C1CC3(C1)CC(O)C3)=O)C2 86833,c1(C(N2C(C)(C)CC(O)C2)C(=O)NCc2cccs2)ccc2c(c1F)CCC2 86834,C(=O)(CCCCN(C)C(c1ncccc1Cl)=O)NCC(CC1CC1)OC 86835,C(C(=O)Nc1ccccc1C)(C(C)CC1CCCC1)N(CC(=O)NC)C 86836,c1(C(=O)NC(C(=O)NC2CCCN(CC)C2)(C)CO)cc(CC)nnc1C 86837,c1(CC)c[nH]nc1C(=O)NCC1(CCNC(C2(C3CCCCO3)CC2)=O)CC1 86838,C#Cc1ccc(C(N2CCC(C)C2C(N2CC3C=CC2CC3)=O)=O)nc1 86839,CS(C)(=O)=Nc1cccnc1C(N1CCC(O)(c2ccccc2F)CC1)=O 86840,Cc1nc(O)nc(C)c1CC(=O)NCCOCCCNC(=O)CCC1CCC(C)O1 86841,c1(NC(CC2(C)CN(C(=O)Cc3ccccc3I)C2)=O)ncnc2occc12 86842,c1(N2CCC(C(C)NC(c3nc(C(C)C)oc3)=O)CC2)ncnc2cccnc12 86843,C(C(C)C(F)C(=O)N(c1cn(C)nc1C)C(C)C)NC(Cc1cc(C)on1)=O 86844,c1(COC)ccnc(NC(C2CCCC(NC(c3cscc3C)=O)C2)=O)c1 86845,C12(C(N3C(C)(C(=O)NC)CC3)=O)C(NC(=O)C(C)C#N)C3CC1C2C3 86846,C1(CC(N2C(CCC=C)CCC2)=O)CCCCN1C(c1ccc(C)s1)=O 86847,C1(NC(C2(CC(C)=O)CC2)=O)CCN(C(C2CCC(C)C2)=O)CC1(C)C 86848,c1(CN(C)C)ccccc1C(=O)N(C)CC1CN(C(C23COCC2C3)=O)CCO1 86849,Cn1nccc(C(=O)NC2CN(C(=O)Cn3ncc(Br)n3)CC2O)c1=O 86850,N1(C(C(=Cc2ccccc2)OC)=O)CC(NC(=O)C(C)c2cccs2)CC(F)C1 86851,N1(C(c2n(C)ncc2)=O)C2CCCC1CC(NC(c1ccc3nnnn3c1)=O)C2 86852,c1(C(=O)Nc2ccc(NC(=O)C3CC3)cc2)cncc(O)c1Cl.c12ccc(cc1)o2 86853,C1(C)(C(=O)NCC(=C)CCNC(C2(c3ccnn3C)CC2)=O)CC(O)CN1C 86854,C1(c2n(CC)nnn2)(NCC2(c3nnn(C)n3)CC2)CCC(c2nc(C)no2)C1 86855,C12(C(N3CCCCC(NC(CC4N(C)CCC4)=O)C3)=O)CCC(CO)(CC1)CC2 86856,N1(C(C2N(CCCC)CCCC2)=O)CCC(C)(C)C(C(=O)N(C)C)C1 86857,C(C(C(=O)NC(c1nn(C)cc1O)C)C(C)(C)C)NC(C(C(=O)OCC)F)=O 86858,c1(CC2(C(=O)NC(CC(C)NC(=O)CC3CCCC3)C)CC2)ccc(O)cc1 86859,c1(CC)cccc(C(=O)NC2CC(N(C(=O)Cc3c(Cl)cnn3C)C)C2)c1F 86860,[N-]=[N+]=NC1CN(C(=O)NCc2cnc(C#N)s2)C1 86861,N1(C(CCSCC)=O)CCN(C(c2cccc(C(F)(F)F)n2)=O)C(C)C1 86862,CC1(C)CCCC(CC(N2CCN(C(c3ccnc(S)c3)=O)CC2C2CCC2)=O)O1 86863,c1(C(N2C(COC)CN(C(=O)CCCC#N)CC2)=O)c2c(nn1C)CCC2 86864,C(=O)(CC(C)C)N(C1(C(=O)OCC)CC1)CC.C12(CSC1)C(=O)N2 86865,c1(C(N(C2CCN(C(c3cc(OC)n[nH]3)=O)C2)C)=O)cc(Br)sc1C 86866,N1(C(C(CC)(C)C(N)=O)=O)CCCCC2(C1)CN(C(c1c[nH]cc1C)=O)C2 86867,C1(C(=O)NCC2(C#C)CCOCC2)CC2(CCC2)CN1C(c1ncccn1)=O 86868,Cc1scc(NC(=O)NCC(C(C)(C)C)NC(=O)OC(C)(C)C)c1N 86869,C(=O)(C(CSC)(CC)CC)NC(C(C#C)NC(=O)C=CCF)C 86870,C1(NC(c2c(C)cnnc2)=O)CCCCN(C(=O)CCOc2ccccc2Cl)C1 86871,Cc1nc(N)cnc1C(=O)N(C)CCOCCNC(=O)CC(C)n1ccnc1 86872,C1(NC(c2ccc(C)[nH]2)=O)CN(C(C2CC23CCOCC3)=O)CC2(CCC2)C1 86873,c1(CCCC)cc(N2CCC(NC(=O)C(O)CC3CC3)C(C)C2)n2ncnc2n1 86874,C(=O)(C#CC1(C)CCCO1)N1CCC(N(CC#C)C(C2CCC3(C2)N=N3)=O)CC1 86875,C=C=C(C)CC(=O)N1CCCC1(C)CNC(=O)C(C)COCC 86876,C1(CC)CN(C(c2cc(C)c[nH]2)=O)CC1C(=O)NCCC1CC(F)C1 86877,CC1CCN(C(=O)CC(C2CC2)NC(=O)CS(C)(=O)=O)CCS1 86878,c1(SCCNC(C=Cc2cc(C)c(=N)[nH]c2)=O)cc(Cl)ccc1[N+](=O)[O-] 86879,C1(NC(CN2C(C)CCC2)=O)CCC2(CC1)CC2NC(C1C2CC3C(C2=O)C13)=O 86880,c1(OC)ccc(C(=O)NCC#CC(=O)NCC(=O)NC2CCCC2)s1 86881,N1(C(C2CN(C)C2)=O)CCOCC(C)(CNC(=O)CCC2CCCCN2C)C1 86882,c1(C(=O)NCC2CCC(F)(CNC(=O)CC34CCCC3C4)C2)ccc(F)cc1Cl 86883,c1(OCCNC(N2CC(CCC)OCC2)=O)c(CO)cc(Br)cc1C 86884,N12CC(CC1=O)C(=O)N(CC)C2.c1(C2(NC(=O)C=CC3CCC3)CC2)ncc(C)o1 86885,C(CN=c1[nH]c(=NCCC2CCCCO2)[nH]c2cc[nH]c12)c1ccc(SC)cc1 86886,c1(CN2C(C(=O)Nc3ccc(Br)nc3I)C(O)CC2)cc(F)c(Cl)c(Cl)c1 86887,N1(C(C(N(C(C(C)OCC(C)C)=O)C)C2CC2)=O)CCCC[Si](C)(C)C1 86888,CCCCN=C(NCc1c(C)cccc1F)NCC1CCC(CC(N)=O)CC1 86889,c1(C(N2CC=CC(NC(=O)C=C3CCSCC3)C2)=O)c[nH]cc(Br)c1=O 86890,N1(C(C(C)OCC=C)=O)CCC2CCCC12C(N1Cc2[nH]nc(C(=O)OC)c2C1)=O 86891,Nc1sc2c(c1C(N1CCC3(CC(NC(c4csnc4Cl)=O)C3)C1)=O)CCC2 86892,[N-]=[N+]=NCCCCCC(=O)N1CCOC(CC=O)C1.C1(N2CCC2)CC(O)C1O 86893,c1(C(=O)NCC2C3N(C(C4C(CCC)C4)=O)C(CC3)C2)ccc2oc(O)nc2c1 86894,c1(SC)ccccc1C(N1CCC(CNC(=O)C(N2CCOCC2)C2CC2)C1)=O 86895,C1(NC(=O)C=CC=C(Cl)Cl)CCCCC12CCN(C(=O)C=Cc1cccs1)C2 86896,c1(NC(C2C(C)(C)C2CN)=O)ccc(CC(N)=O)cc1.N1(C(N)=O)CCC1 86897,C(=O)(CCC=CBr)N(CCCNC(c1ccc(C2CC2)s1)=O)CC 86898,Cc1nc(C(=O)NCC2(CN)CC2)c(C)s1.N1(CCC(=O)N(C)C)CCNC(=O)C1 86899,N1(C(c2cc(C)c(C)s2)=O)CC2CC1CN2C(C1CC(C2CC2)=NO1)=O 86900,N1(C(C2CNC(=O)N2)=O)CC(C2CC2)(C(=O)NC2C3C=CC(C3)C2CO)C1 86901,c1(CNC(CN2C(C)(C(=O)OC)COCC2)=O)c(F)ccc(Br)c1F 86902,c1(C(=O)NCCCCN(C)C(C2CC2F)=O)csc(C2CCC2)c1 86903,N1(C(Cn2ncc(CC)c2)=O)CCCC(NC(c2nnc(O)nc2O)=O)CC1 86904,C(C1=CCN(C(c2cc[nH]c2C2CCC2)=O)CC1)NC(C(F)OC)=O 86905,c1(C(N(C(CNC(c2sc(C(=O)OC)c(N)c2)=O)C)C)=O)cn(C)c(=O)nc1O 86906,C1(F)(CNC(C(C)OCC=C)=O)CCN(C(c2cccs2)=O)CC1 86907,N1(C(C2N(C(CCC)=O)CCCC2)=O)CC2(CCCCN(C(=O)C(C)CO)C2)C1 86908,C1(NCC(c2ccc(F)c(F)c2)C(C)C)CC2CCC1C(N)C2 86909,C(=O)(CC(O)CC(C)(C)C)NCC(=O)NCC(=O)NCCCOCC=C 86910,C1(CNC(C(C)c2cncs2)=O)CC(O)CN1C(=O)CCc1cc(Cl)no1 86911,N1(C(=O)NCC(CC)C)CCC2CN(C)CC2C1 86912,C(=O)(CCCCCOC)N1CC(CCC)C(C(N2CCCCC2C2(O)CC2)=O)C1 86913,c1(NC(CCC)CCCNC(=O)Cn2cc(C)cn2)c([N+](=O)[O-])c(CC)nn1C 86914,CC1(C(N2CCCC2CNC(=O)CC2CCCC2O)=O)CC1(F)F 86915,N1(C(CN(C)S(N)(=O)=O)=O)CCC2(CC1)CC2NC(=O)CCN1CCC(F)C1 86916,N1(CC(CC(=O)OC)NC(C)=O)CCCN(Cc2noc(C3CC3)n2)CC1 86917,C1(C(=O)NC(=O)CC(C)NC(=O)N(C)C2CC2)CCCCC1O.CC(C)CC1CC1 86918,c1(OC)ccc(CC(=O)NC2CC(C(=O)NCC3CCC(=O)N3C)C2)cn1 86919,CC(C)(CCC(=O)N1CCC(C(C)(O)CNC(=O)C#CC2CCC2)C1)[N+](=O)[O-] 86920,CC(CC(=O)N1CCC(O)C(N(C(=O)COCc2cccc(Cl)c2)C)C1)C(F)F 86921,c1(C(C(=O)N2CC(F)C2)NC(CCOC(C)C)=O)cnn(C)c1 86922,C12(NC(c3c[nH]c(=O)cn3)=O)CCC1CN(C(=O)COc1ccc(Cl)nc1)C2 86923,c1(C(N(CCC)CCNC(=O)COC2CCCC2)=O)cc2occc2s1 86924,N1(C(c2cn(CCCF)nn2)C(=O)NC)CCCC(OCCSC)C1.C(C)C 86925,C(CN=c1cc(C)nc(C)[nH]1)C1(O)CCN(C(C=CC=CC=CC)=O)CC1 86926,C1(NC(=O)Cc2cnn(C(F)F)c2)C2CC1CN(C(=O)C(F)C1CCOC1)C2 86927,CC1c2ccc(F)cc2CCN1C(c1cncs1)C(=O)Nc1cccc([N+](=O)[O-])c1 86928,c1(CNC(c2n(CCCSCC)nnn2)C23CCCC2C3)c(OC)ncnc1Cl 86929,CC(CC(C)NC(=O)CCC1CCC(=O)N1)NC(c1scnc1C(F)(F)F)=O 86930,c1(CC(N2C(C(COC)(C)C)CCC2)=O)nn(C)cc1NC(CC1CC(=C)C1)=O 86931,c1(C(=O)NCC(=O)N(CCC(=O)NC(CC)C)C)c[nH]nc1C(F)F 86932,C1(C(=O)NC(c2ccccc2O)C)CC2(CCC2)CN1C(=O)C(CO)C(F)(F)F 86933,C1(CC(N2C(C)(c3cn(CC(=O)NCC)nn3)CCC2)=O)CCC(=O)NC1=O 86934,C1(C2CCCN(C(=O)C(C)(C)CC(F)F)C2)(NC(C(c2ccncc2)C)=O)CC1 86935,CC1CN(C(c2cnn(CCNC(C3C4CCC(=O)C34)=O)c2)=O)c2cnccc21 86936,C(=O)(C(CNC(C1CNC(=O)N1)=O)CC1CCCC1)NCC(COC)C1CC1 86937,c1(C(N2CCC(N(C)CC)CC2)C(=O)NC(CC)C)cc(C)c(Cl)c(C)c1 86938,CC(CNC(=O)CC(CNC(c1cc(C(F)F)no1)=O)C1CCC1)CC(F)(F)F 86939,N1(Cc2nc(CCOC)sc2)CC2CC1CN2C(c1ccc(O)c(F)c1)=O 86940,c1(COC)nc(OC)cc(NC2CC(CNC(c3c(C)noc3C)=O)C2)n1 86941,c1(C(=O)NCC2N(C(C(CC)OC3CCCCC3)=O)CC2)cc2ccccc2s1 86942,C1(NC(C23OCC(C)(C2)C3)=O)CC2CC1N(C(=O)CCCCc1cnn[nH]1)C2 86943,C1(CC(=O)NCC2(O)CN(C(COCC=C)=O)C2)CCOC(C)(C)C1 86944,C1(N(C(CC=C)=O)CC)CN(C(=O)C(CC)=CCOC)CCC1(C)C 86945,c1(C(N(C2CN(C(c3cc(Cl)cnn3)=O)C2)C)=O)cncc2nc[nH]c12 86946,CN1CC2(CN(C(c3ccc(Cl)cc3-c3sccc3C#N)=O)C2)OC1=O 86947,C1(NC(NC(C(C)C)C)=NCC2CC(=O)N(c3ccccc3)C2)CCOC(C)(C)C1 86948,CON(CCCO)C(=O)C1(CO)CCCN(C(c2cnnc(C)c2)=O)C1 86949,C1(CC(C)NC(C2(CSC)CC2)=O)CCCN1C(=O)C=CC1CC1 86950,CC1CN(C(=O)Cc2ccn(C)n2)CC1(C)C(=O)NCC1NC(=O)NC1=O 86951,c1(N(C(=O)CC(F)(F)F)CCC)ccc(OC(C)C)cc1Br 86952,C=C(C)C1CCC(C)(O)C(NC(=O)NCc2cccc(Br)c2Cl)C1 86953,c1(CC)oc(C(=O)NC2(C(=O)NCCCN3CCC(O)C3)CCN(C)C2)cc1C 86954,C1(CC)CCN(C(=O)CC2(C)CCC2)C1C(=O)NCCS(=O)(=O)NC 86955,c1(NC(C(C)CN(C)C(C2CCOCC2)=O)=O)ncccc1OC(F)F 86956,c1(C(N2CCC3CN(C(C(CCCOC)C)=O)C3C2)=O)cc(C#N)c(O)nc1N 86957,C1(C(C)NC(C(C)N(C(C)=O)C)=O)CCN(C(=O)C(C)Cc2cccnc2)CC1 86958,N1(C(C2N(C)CCCC2)=O)CC2CC1CC2NC(c1cc(Cl)ncc1F)=O 86959,C1(CN(C)C(c2scc(Cl)c2Cl)=O)CN(C(=O)Cc2cncs2)CCO1 86960,N1(C(C2(CC=C)CCCC2)=O)CC(NC(=O)C(C)Oc2ccccn2)CCC1C 86961,C1(C(=O)NC2CCCC(CNC(=O)C(C)(F)C(C)(C)F)C2)(OC)CCC(F)(F)CC1 86962,Cc1c(C(=O)NCC2COCCN2C(=O)Cn2cnnc2)cncc1Br 86963,C1(C(N2CCC(C(CNC(C3C(=C)CC3)=O)(C)C)CC2)=O)CN2CCC1CC2 86964,c1(C(N2CCC(F)(CNC(COCCC=C)=O)C2)=O)cccc(S(N)(=O)=O)c1 86965,C(=O)(CCCCNC(=O)C(C)(F)c1ccon1)NCC1C(N(C)C)C1 86966,c1(OC)ccc(CCC(=O)N(C2CN(C(=O)CC3CC(C)C3)C2)C)cn1 86967,CC(CC(=O)N(C)CC1(O)CCN(C(=O)C(F)(F)CO)C1)C(F)(F)C(F)(F)F 86968,c1(C(N)=O)ccc(C=CC(=O)NC2CCC(CCNC(c3c[nH]nc3F)=O)C2)o1 86969,N1(CC2(NC(C=COCC)=O)CCCC2)CCN(C(c2[nH]ccc2CC)=O)CC1 86970,Cc1cc(C(=O)NCC(=C2CN(C(=O)Cc3ccn(C(F)F)n3)C2)F)n(C)n1 86971,C(CO)(CCCCCNC(C1(C)CCCC1)=O)NC(C=CC=CC)=O 86972,C1(CNC(CC2(C=C)CC2)=O)(CNC(=O)CCNC(=O)CC(C)C)CC12CCC2 86973,CC(C)CCCCC(=O)NC1CC1CNC(c1ccnc(OCC(F)F)c1)=O 86974,CC1(C)CC(C)(C(=O)NCCCC2CN(C(c3cc(=O)cc[nH]3)=O)CCO2)C1 86975,Cc1cc(C(N2CC=CC2CNC(c2ccc(=N)[nH]c2)=O)=O)ccc1Br 86976,c1(C(C)NC2C(OCC)CN(C(=O)OC(C)(C)C)CC2)nnc2ccccc2n1 86977,C12(C(=O)NCC#CCNC(Cc3cc(C(C)C)no3)=O)CCCC1CC2 86978,c1(C(=O)NCC(Cc2cccc(C)c2)CO)c2c(nn1C)CCCC2 86979,C(C)(C(C(=O)NC1CN(C)NC1=O)NC(=O)C(O)CCN(C)C)OC 86980,N1(C(C(C)Cc2ccco2)=O)CCC2CN(C(c3cn4c(n3)COCC4)=O)CC12 86981,c1(CC(=O)N(CCCN(C(COCCOCC)=O)C)C)ccc(C)nc1 86982,c1(C(=O)NCC2C(CNC(CCN(C)CC)=O)C2)ccc(S(C)(=O)=O)c(C#N)c1 86983,CS(=O)(=O)CC(=O)NC1CCCCC1NC(=O)CCNC(C1CCOCC1)=O 86984,C12(CNC(c3n(C)cnc3)=O)COCCN1CCN(C(c1cnsc1)=O)C2 86985,CCC(C)CCC(=O)NC1(C)CN(C(C2(F)CCCN(C)C2)=O)C1 86986,c1(OC)ccoc1CNC(=O)Cn1cc(CNC(=O)C(C)Cc2ccccc2)nn1 86987,N1(C(CC23CC(C)(OC2)C3)=O)CCCC(C2CC2NC(C2CCCCC2)=O)C1 86988,C1(C(=O)OCC2C(=O)OCC2)CCc2nncn2C1 86989,C(=O)(C(C)(C)CCCNC(=O)Cc1ccnc(O)c1)NC1C(C)(CC)C1 86990,N1(C(C(C)n2cccc2)=O)CCCC(c2nncn2C)C1 86991,c1(C(=O)NC(C2CCN(Cc3cccnc3Br)CC2)C)cc(Cl)cnc1Br 86992,C1(C(=O)NC(C(C)(C2CC2)OC)C)C=CCCN1C(=O)CCNC(=O)OC 86993,N1(C(CCCC=C)=O)CC(C2CC2)(C(=O)NC2CCCOC2)C1 86994,Cc1ccc2c(c1)C(C(=O)N(CC(C)O)CCNC(=O)Cc1c(C)n[nH]c1C)C2 86995,c1(OC)ncccc1CC(=O)NC1CCN(CCn2cccn2)CC1 86996,C(=O)(NNc1ncc(Br)c2ccccc12)C12CC(SCCCCCC=C)(C1)C2 86997,C1(C(N(CC(=O)NCCCC2CCCO2)CCOC)=O)CCCN1C 86998,C12(C(N(C3CCN(C(=O)CC45COCC(C4)C5)C3)CCO)=O)CCC(CC1O)C2 86999,N#CCCCC(C(=O)NCCOCc1ccccc1)NC1CC1 87000,c1(C(=O)NC2CC(F)(CNC(C3(CC=C)CC3)=O)C2)ncnc2c(C)csc12 87001,c1(C(N(C(CC(=O)N2C(C(C)C)CC2)C)C)=O)nnn(C)c1N 87002,C=CC1(C(N2C3C=CCC2CC3)=O)CCN(C(=O)C(C)COC(C)=O)C1 87003,c1(CC(=O)NCCCCC(CO)NC(=O)C=C2CC2)ccc2n[nH]cc2c1 87004,C1(NC(Cc2ccc(CCC)cc2)=O)CC2CCC1N(C(c1cc(Cl)c[nH]1)=O)C2 87005,C(CCCCCO)n1cc(CCC(C)(C)NC(CN2CCC(C)C2)=O)nn1 87006,C(=O)(C(C)C(C)NC(C1(NC(C2CN(C(N)=O)C2)=O)CCN(C)C1)=O)OC 87007,CN1CCOC(CC(=O)NC(CCN(C)C(c2ccco2)=O)c2cccs2)C1 87008,Cc1cc(S(=O)(=O)NC(C2COC3CNCC23)=O)sc1C 87009,N1(C(C#CC2(CC)CC2)=O)CCCN(C(c2cccc(C3(C)CC3)c2)=O)C(C)C1 87010,C12(n3cc(C(C=C)(C)O)nn3)CCC(NC(c3cc(Cl)ns3)=O)(CC1)C2 87011,Cc1cc(Cl)cc(C(N2CCCC(NC(c3cncc(O)c3Cl)=O)C2)=O)c1C 87012,CN1CCOC(C(=O)NCC(O)CCNC(=O)C(F)(F)c2ccccc2)C1=O 87013,c1(CC)ccsc1C(=O)NC(C(=O)NCc1cncn1C)C1CC1 87014,Cc1ncc(N)cc1C(=O)NCCC1(NC(C2CC(C3CCC3)C2)=O)CCC1 87015,c1(C(=O)NCC2N(C(C(CC)C(=O)OC)=O)CCCC2)noc2c1CC(C)CC2 87016,c1(C(=O)NC2COCCC2(F)F)cnc2sccn12 87017,c1(CCC(=O)NCC(C(C)C)NC(=O)C(C)NC(C)(C)C)cncc(F)c1 87018,c1(CN(c2nc(OCC)c(OC)cn2)C2CCCNC2)ccc2c(c1)ncn2C 87019,c1(OC)cc(C(N2CC(NC(=O)Cc3nc[nH]n3)C2)=O)cc(NC(C)=O)c1OC 87020,C(=O)(C(C)(C)C(N)=O)N1CC(NC(C2C(C)OCCC2)=O)C1 87021,CN1CCN(C(=O)C(O)CCN(C)C)CC1CO.c12cccc(c1)NC2=O.C1(C)CC1 87022,c1(SCC(=O)NC2CCN(C(CC(CCC)C)=O)C23CC3)nnc2ccccn12 87023,c1(C(=O)NCCN(C(=O)C(C2CCC(=O)N2)C)C(C)C)ncc(F)cn1 87024,Cc1cc(=O)n(CC2CCCN2C(=O)C(C)OC)cn1 87025,C1(NC(C=CCC)=O)CCC12CN(C(=O)C(CC)NC(=O)OC(C)(C)C)C2 87026,N1(C(=O)NCCCCCC#C)CCCN(C)C(=O)C1 87027,Cc1cccc(C(O)C(=O)N(C)CCNC(c2nn(C)cc2Br)=O)c1 87028,N1(C(C(C)=C(CC)C)=O)Cc2occ(C(=O)NC3CN(C)CC3OC)c2C1 87029,C#CCCCC(C)C(=O)NCC1(C)CN(C(=O)CCOCCCCC)C(C)(C)C1 87030,C(CCCCCNC(C1(c2ccno2)CC1)=O)N(C(=O)CC1CCC(=O)C1C)C 87031,n1(CC)ncnc1C(N1CCC(C(=O)NC)C1)C(=O)NCC1CC1 87032,CC1CN(C(=O)C=Cc2ccncc2)CC(C(=O)NCc2ccon2)O1 87033,c1(C(=O)NC(C(=O)Nc2cn(CC(=O)NC)nc2)C2CCCC2)ccnn1C=C 87034,Cn1cc(C(=O)NC23CC2CN(C(c2cc(C(F)F)ccn2)=O)C3)ccc1=O 87035,CN1CCCCC(C(=O)NCC(C)(C)NC(c2cnc([N+](=O)[O-])n2C)=O)C1=O 87036,C(=O)(CCCCN(C)C)N1CC(CN(C(C(C)NC(c2cccs2)=O)=O)C)C1 87037,c1(C(=O)NC2(CCNC(C3(CC)CC(O)C3)=O)CCCC2)cc(O)n(C)n1 87038,N1(C(c2c(Cl)ccc(C#C)c2)=O)CCCC2(NC(C3CC(=C)C3)=O)CC2C1 87039,Cc1cc(C)n(C(C)CC(=O)N(C)CC2CCN(C(c3ccc(F)o3)=O)C2)n1 87040,C1(NC(c2cncc(NC)c2)=O)C2CC3C1C3C2C(=O)NOCC=CCl 87041,Nc1c(C(N2CC(NC(=O)CCc3nc[nH]n3)CC(F)(F)C2)=O)ccc(Cl)c1Cl 87042,S(=O)(=O)(c1c[nH]ccc1=NCC)C1C(c2nc(C)sc2)C1.c1(CCN)cn2c(n1)SCC2 87043,c1(CCNC(CN2CCCC(NC(C(C)(C)CO)=O)C2)=O)ccc2occc2c1 87044,C(=O)(C(C)(C)C(C)(F)F)N1CC2C(C(N(C3CCC3(C)C)C)=O)C2C1 87045,N1(C(C2(SC)CC2)=O)CCC(C)C(NC(=O)C(C)(c2ccccc2)N(C)C)C1 87046,C(=O)(C(CC)C(C)(C)CC)N1CCCC(N(C(CCCC(=C)C)=O)CCF)C1 87047,C(CC(C)C)(C(=O)NCCCCS(C)=O)NC(C1C(C=C)OCC1)=O 87048,c1(OC)cc(C)c(C(C)Nc2cc(NCCc3nc[nH]n3)nc(C)n2)cc1C 87049,S(=O)(=O)(c1cccnc1NCCc1cc(Cl)sc1Cl)NC(CCC)CCC 87050,C(=O)(C(CC(C)C)OC)N1C(C(=O)NOCC(N)=O)(CC=CCOCC)C=CC1 87051,CCCCCC(O)C(C)C(=O)NC1CCCC1NC(c1nncn1C1CC1)=O 87052,CN1CC2C(CCCN2C(=O)CCc2nc(-c3ccco3)n[nH]2)C1 87053,CC1(C)OCCC1C(N1CCC(C2CCCN2C(=O)Cc2cnsc2)CC1)=O 87054,CCC(C)(COC)C(=O)N1CSCC1C(=O)NCc1nn(CC)nc1C 87055,C(=O)(C=C1SCC(=O)N1C)N(CCC(C)NC(=O)CC1CC(=O)NC(=O)C1)C 87056,C1(CNC(c2c(C(C)C)con2)=O)CN(C(C2CCOC(=O)CC2)=O)CCCO1 87057,N1(C(C=C)=O)CCCCC1C(C)(C)CNC(c1ccc(N(C)C)cn1)=O 87058,C1(F)(CNC(C(C)OCC=C)=O)CN(C(=O)CCOCC2CCC2)C1 87059,N1(C(CNC(c2cc(C)on2)=O)=O)CCN(C(=O)Cc2ccco2)CC1.C(N)(=O)N 87060,c1(OC)cc(-c2nc(C(C)O)nn2C2CC3CCC2C3)c(Br)cc1C 87061,C1(C(=O)NC(C2CCCN2C(c2ccc[nH]2)=O)C)COC(=O)C1 87062,c1(CC(=O)NC(CC)(C)CNC(C2C(C(F)F)C2(C)C)=O)ccc(C2CC2)cc1 87063,C1(C(=O)NCC=Cc2ccccc2)CN(C(c2ccc(Cl)cn2)=O)CC1(C)C 87064,c1(C(N2CCC(N(C(C3C(C=C)C3)=O)CC)C2)=O)cc(Cl)ncc1N 87065,C=C=CC(C)C(=O)N1CCC(N(CCC)C(c2ccc(CC(C)(C)C)cc2)=O)C1 87066,c1(C(=O)NCC2CCCN(C(CNC(C)=O)=O)C2)noc2c1CN(C(C)=O)CC2 87067,O=C(C1=CCCCCC1)NCc1cc[nH]c1C(=O)NCC1OC(=O)CC1O 87068,CC(C)S(=O)(=O)CC(=O)NC1CCN(C(C2CCCCCS2(=O)=O)=O)CC1O 87069,c1(C(N2CCC(c3nn[nH]n3)(C(=O)Nc3ccc(F)cc3)C2)=O)cccc(Cl)c1 87070,Cc1cncc2cc(C(N3CCOCC(CNC(=O)C(C)C4CCC4)C3)=O)sc12 87071,c1(CCCC(=O)N2C(CNC(c3cccc(C)n3)=O)CC2)c(F)cccc1F 87072,CC(C)CCCC(=O)N1CCC(NC(=O)C=CC2CCCCC2)C(O)C1 87073,CC(C)C(C)(CNC(c1ccc(C2CC2)nn1)=O)NC(C1CCC(=O)C1)=O 87074,C1(C)(C(=O)N)CCCOC1.C12(CCC1)C(=O)NCC2.C(C)(CNC)OC 87075,c1(CNC(=O)C(c2ncccc2Br)N2C3CNCC3C2)ccc2nonc2c1 87076,Cc1nnc2c(C(N3CCCN(C(=O)C(O)Cc4cnc[nH]4)CC3)=O)nccn12 87077,O=C(CC1NC(=O)c2ccccc21)NCCC1CCN(C(C2SCCS2)=O)C1 87078,C(CCC(C)CC(=O)NCCN(C(C1(C(F)(F)F)CC(F)(F)C1)=O)C1CC1)=C(C)C 87079,c1(CC)cc(Br)ccc1C(=O)NCC(C)CN(C(=O)Cc1ccoc1)C 87080,C1(C)(CNCC2(O)COC2)CN(Cc2c(C)non2)CCO1.C1(=O)C2=NOC(C2)N1.OCCC 87081,N12CC(CCC1C)C2=O.c1(C2N(CC)CCC2)ccncn1 87082,CC(CN=c1[nH]cnc2c(C(F)(F)F)cccc12)N(C)C(c1cc(Cl)no1)=O 87083,C(=O)(C1=CCCCO1)NC(c1ccc(F)cc1)CNC(c1c(C)c[nH]n1)=O 87084,C(CNC(=O)C(C)NC(N)=O)(C(C)(C)C)NC(C(C)C1CCC1)=O 87085,c1(C(=O)NC2CC(N(C)C(C3CCCSC3)=O)C2)cccc(N(C)C)n1 87086,C(=O)(C1Cc2ccc(F)cc21)NC1(CNC(CC(C)C2CCCO2)=O)CCCC1 87087,Cc1cccc2nc(NC(C3CCCN3NC(=O)C3CC3(F)F)=O)[nH]c12 87088,N1(C(C2N(C)CCOC2)=O)C2CCC1CN(C(c1ccc(C(F)F)c(F)c1)=O)C2 87089,N1(C(C)=O)CCC(CC(=O)NCCCN(C(c2cncn2C)=O)C(C)C)C1 87090,C=CCCC(=O)N(CC(C)NC(c1cscc1Cl)=O)CC 87091,C1(C(=O)O)COC2CN(C(c3ccccc3-n3cc(C4CCCC4)nn3)=O)CC12 87092,N1(C(C(C(C)O)C)=O)CCCCC(NC(=O)CCc2ccsc2)C1 87093,C1(NC(C(C)OCCOCC)=O)CCOCC1NC(C1CCCN(C)C1)=O 87094,C#Cc1cnc(C(N2CCOCCC2C(=O)NCC(=O)NOCC)=O)c(C)c1 87095,c1(OCC(=O)N(CCNC(C2(CC(C)C)CCCC2)=O)C(C)C)cccc(O)c1 87096,Cc1nc2ncnn2c(NC2CCC(NC(c3cnn(C)c3)=O)CC2)c1C 87097,c1(N2CC=CC(NC(c3cccc(OCC)c3)=O)C2)ncnc2cc(C3CC3)nn12 87098,C12(C(=O)NC(C(C)C)CNC(C3CC4(CCO4)C3)=O)CC3CC1(CSC)CC3C2 87099,c1(CC)nc(C(N2CCCC2CN(C(=O)C(F)=C(C)C)C2CC2)=O)c2ccccn12 87100,C12CCC(CC1)N2.C(C(=O)NCC(=O)NS(C)(=O)=O)OCCSC 87101,C(CN=C(NCc1cccc(Br)c1OC)N1CCC2(CCOC2)C1)OC 87102,C1(COC)CC(CNC(=O)C=C2CCSCC2)N(C(C2CSCN2C(C)=O)=O)C1 87103,c1(SC)ccccc1CC(N1CC=CC(NC(=O)C=C(C)C(F)F)C1)=O 87104,C1(C(N2CCCC2CNC(C2ON=C(C)C2C)=O)=O)(CC)CC(F)(F)C1 87105,C(=O)(C1=C(c2ccccc2)CCC1)NCCC(CNC(CCCC=C)=O)O 87106,C1(OC)(OC)CCN(Cc2ccc(Cc3ccccc3)cc2)CC1O 87107,c1(C(N2CC(C(=O)NCC3C(C)C3C)C(F)C2)=O)cccc(C#N)c1 87108,c1(CC)ncc(C(=O)NCC2CC2NC(C2CC2(C)C(F)F)=O)cn1 87109,C1(OC)CCCCN(CC(=O)N(C(CNC(c2csc(Cl)c2)=O)C2CC2)C)C1=O 87110,N1(C(CCCCCC#C)=O)CCC2(CC1)CN(C(=O)C(C(C)C)OC)CC(C)O2 87111,Cc1cc(=NCc2cc(Br)ccc2Cl)[nH]c(N2CC3CC2CO3)n1 87112,C1(CNC(C2(C)CCC2)=O)C2CN(C(=O)CCc3cccs3)CC12 87113,C1(C)(CNC(CCC2(NC(CCc3cnc(C)s3)=O)CCC2)=O)CCC(C)CC1 87114,CC1=C(C(=O)N2CC(NC(c3ccc(C(N)=O)c(Cl)c3)=O)C(F)C2)CCO1 87115,C(c1cc(Cl)c2c(c1)OCO2)=CC(N1CCC(C)C(NC(=O)C(C)N(C)C)C1)=O 87116,C(c1ccc(C#N)cc1)=CC(=O)NC1(CNC(C2CC=C(C)CC2)=O)CC1 87117,Cc1cc(O)cc(C)c1CC(=O)NCCCN(C(C1(C)CCNC1=O)=O)C1CC1 87118,C(=O)(C(C)(C)CC(C)C)N1CC(C(N2CCC(C=C)(O)C2)=O)OC(C)C1 87119,C1(OC)CC(NC(=O)C(CC(C)C)OC)CN(C(c2cccc(F)c2F)=O)C1 87120,C(N=c1cccc(S(=O)(=O)NC2CC(F)(F)C2)[nH]1)c1ccc(C(C)OC)o1 87121,N12CCC3(CC1)CC3(C)CNC2=O.Cc1nccn1CC1CCOCC1 87122,Cc1cc(Cl)c(CN(C)Cc2ccoc2)cc1O 87123,c1(OC)cc(C(N2CC(CNC(=O)C3=NOCC3)C(O)C2)=O)ccc1O 87124,c1(CCC(N2CCC(Cc3ccccc3)(NC(=O)NC)C2)=O)ccc(Br)cc1.O=COC 87125,C1(NC(CC(CC2CCC2)NC(C2CCN(C)CC2)=O)=O)CC2(C1)CC2(F)F 87126,CC1(C)CC(CO)CN(C(CCSc2ccccc2)C(=O)NCC(F)F)C1 87127,N1(CC#C)CCN(C(C2CSCCN2C(=O)Cc2cncnc2O)=O)CC1=O 87128,c1(CNC(C(C2CC(CF)C2)N(C)C(C2(CCO)CC2)=O)=O)cc(Cl)ccc1F 87129,C(=O)(C#CC(C)(C)CNC(=O)CC1CC2CC2C1)NC(CC=C)CC(F)F 87130,N1(C(C(C)OCC#C)=O)CCN(C(c2cnn(CC)c2C)=O)C2CS(=O)(=O)CC12 87131,C1(NC(=O)CSc2ccccn2)CN(C(=O)CC2CC(n3cnnc3)C2)C2CC12 87132,C(=O)(CCCS(C)(=O)=O)NC1(C)CCN(C(C2CCCC(=O)C2)=O)C1 87133,C1(NC(C(CNC(C2C(C)(C)C2(F)F)=O)O)=O)CCC2(CC1)N=N2 87134,N(S(=O)(=O)N(C)C)CC(=O)N(CC(CNC(C1(COCC)C=CCC1)=O)(C)C)C 87135,C(COC)(CC(=O)NCC1(CC)CC1)NC(C(C)=CC=C)=O 87136,c1(C(N2CCCC(C)(NC(C(C)=C3CC3)=O)C2)=O)ccn2cc(C)nc2c1 87137,C1(F)(C(N2CCN(C(C(C(C)C)SC)=O)CC2)=O)CCC(F)(F)CC1 87138,c1(N2CCCN(CCC)CC2)nc(=NCc2cnn[nH]2)[nH]c2cc(C)ccc12 87139,CCCCC(O)CC(=O)NCC(C1CCCC1)NC(c1ncccc1Cl)=O 87140,C1(n2cc(CN(C)CCC(C)(C)C)nn2)CCCCCC1O.OC 87141,N1(C(C(CO)N(C)C)=O)CC2CC1CCN2C(=O)CCC1CCCCC1 87142,C(=O)(CC(C)(C)C(F)F)NC(CCCC)CNC(c1cc(C2(O)COC2)on1)=O 87143,C(c1cn(C)cn1)=C(C(=O)N(CCCOCCNC(C1C=CCCC1)=O)C)F 87144,Cc1nc[nH]c1CC(C)NC(=O)COCC(=O)OC(C)(C)C 87145,c1(C(N2CCCC2Cc2ncncc2I)=O)cccc2ncsc12 87146,Cn1cc(NC(C2CCN(C(=O)CCCCC(N)=O)CCO2)=O)c(O)nc1=O 87147,c1(NC(C2CN(C(CC(CC)C)=O)C2)=O)ncc(F)c(OC)n1 87148,C#Cc1ccc(CC(N2CCC(NC(=O)Cc3c(C)noc3Cl)C(CO)C2)=O)cc1 87149,c1(C(=O)NC2CCN(C(=O)CCn3ccccc3=O)C2)ccnc(C(F)(F)F)c1F 87150,C1(N(C(=O)C=CCc2ccc(Cl)s2)CC)CCCN(C(=O)CCOCC2CC2)C1 87151,N1(C(c2cc(C)ncn2)=O)CCN(C)CC1CNC(c1ccoc1CC(N)=O)=O 87152,c1(C(N2C(CN(C(C3COC(=O)C3)=O)CC)CCC2)=O)cccc(O)n1 87153,Cc1cnc(NC2(C)CC2)c(S(=O)(=O)NCCC(C)c2cn[nH]c2)c1 87154,c1(C(=O)O)cc(-c2cn(-c3cccc(-c4ncon4)c3)nn2)c2ccccc2n1 87155,C1(CN(C(c2c(CC)csc2)=O)C2CC2)CCN(C(=O)CCC2CCCO2)CC1 87156,c1(CNc2ccc(SCC)cc2)cc(=NC(=O)OCC)[nH]o1 87157,c1(C(N2CC(NC(C3(F)CC=CC3)=O)CC3(C2)CC3)=O)ccc2c(c1)OCCO2 87158,C=Cc1cncc(C(N2CC(O)(C(F)C(=O)NCC(c3ccncc3)O)C2)=O)c1 87159,N1(C(CC(CC)N(C(=O)CC2CCCOCC2)C)=O)CCC(O)C(CO)C1 87160,C(=O)(CC(C)(C)N(C)C(C1(CO)CCCCO1)=O)NC(C#C)C1CC1 87161,CC(CN1CCCC1=O)N=c1cccc(S(=O)(=O)NCCCN2CCOCC2)[nH]1 87162,C(=O)(CC1=CCCC1)NCCC(C)NC(=O)CCc1cnccn1 87163,c1(C(=O)NCC2C(NC(C(C=CC)O)=O)CCCC2)cc(C2(C)CC2)ccc1C 87164,Cc1c[nH]c(C(=O)NC(c2cncc(F)c2)c2cnc(-c3ccccc3)s2)c1C 87165,N1(C(C2(C(=O)NC)CCCCC2)=O)CCC(C)N(C(=O)C(c2ccccc2)C)CC1 87166,c1(OC)ccc2nc(S(C)=O)[nH]c(=NCc3cnn[nH]3)c2c1 87167,c1(CC(=O)NCCN2CCN(C(c3c(C)onc3)=O)CC2)ccc(Cl)cc1Cl 87168,C(=O)(C(C)(C)CS(N)(=O)=O)N1CC(NC(CSc2n(C)ccn2)=O)C(C(F)F)C1 87169,Cn1cncc1C=CC(=O)NC1C2CN(C(=O)C(N3CCSCC3)F)CC12 87170,Cc1ccc(NC(C2CC(C)N(C(c3cnn4c3CCC4)=O)C2)=O)cc1C 87171,C#Cc1cnn(C)c1C(N1C(CNC(C2C3CCC2(c2cscn2)C3)=O)COCC1)=O 87172,C1(CCNC(C2(COC)CC2)=O)CC(C(N2CCCC(OC)C2)=O)C1(C)C 87173,c1(C(=O)NC(C(C)NC(c2ccc(CC)cc2)=O)CO)cnn2c1CCC2 87174,CN1CCc2ccc(C(N3CCC(CCNC(=O)CC4CCC4)C3)=O)cc2C1 87175,CCC(C)C(C(=O)NCC1CN(C(C23CC(C)(C2)C3)=O)CC1(C)C)OC 87176,C(=O)(C(C)CC(F)(F)F)NC(CC=C)CNC(=O)Cc1cn[nH]c1 87177,C(=O)(CCS(C)(=O)=O)NC1(C(=O)NCC(CC)N(C)C)CCSC1 87178,c12ccc(nc1)CNC2=O.C(c1cc[nH]n1)=CC(=O)N(C1CC(C)(C(N)=O)C1)C 87179,N1(C(c2c(C)n(C)cc2)=O)CCC(NC(=O)C(O)C(F)F)C2(CCC2)C1 87180,c1(OC)ccc2nc(N3CCC(C)C3)[nH]c(=NCC3CCCn4ccnc43)c2c1 87181,N1(C(c2c(C)n(C3CCC3)nn2)=O)CCC(CNC(=O)Cn2cncn2)C12CC2 87182,c1(CC(=O)NC2CC2NC(c2csc(-c3ccccn3)n2)=O)ccc(O)cn1 87183,c1(C(=O)NC2C(OC)CC(C(=O)NCC(CCOC)OC)C2)ccn2ncccc12 87184,O=C(C1=CS(=O)CCC1)NCC1CCCN1C(C1COCCO1)=O 87185,O=[N+]([O-])c1ccc(Br)c(Cl)c1N(C)Cc1nccs1 87186,c1(CC=CC)ccccc1C(=O)NCC(C)CNC(c1snnc1C1CCC1)=O 87187,Cc1cc(O)nc(NC(N2CC(O)(CCNC(=O)OC(C)(C)C)C2)=O)n1 87188,N1(CC(=O)NCC2CCCC2C(N2CC(O)(c3cnn[nH]3)C2)=O)CCOCC1=O 87189,C(N=c1ccnc(C)[nH]1)C1(NC(c2c(C)ncnc2C)=O)COC1 87190,c1(C(=O)NC2CCCN(C(C3(CC(C)C)CC3)=O)C2)coc(S(=O)(=O)N(C)C)c1 87191,N1(C(C(c2ccc(OC)nc2)(F)F)=O)CCC2(NC(=O)CC(C)(C)O)CCCC12 87192,N1(C(c2cc(C)c(C)s2)=O)CC2(CC(NC(=O)CS(=O)(=O)N(C)C)C2)C1 87193,N1(C(=O)C=Cc2ncc[nH]2)CC(CO)C2(C1)CN(C(c1cc(Cl)cnn1)=O)C2 87194,C1(C(=O)NCC2CCC(CC)O2)CN(C(=O)COc2cccnc2)CCO1 87195,c1(NC(=O)NC)ccc(N(CCC(=O)Nc2ccc(F)cc2)C)cc1 87196,O([Si](C)(C)C(C)(C)C)CC(=O)NC1(C(=O)OC)CC(C(F)(F)F)(OC)C1 87197,CCC(CNC(=O)C(C)OC(C)=O)(CC)C(=O)Nc1ccc(O)cc1Cl 87198,C(=O)(C#CC1(C(F)(F)F)CC1)NC(C1CCCN(C(c2ccncc2Br)=O)C1)C 87199,N1(C(c2c(-c3c(CC)cccc3C)ncs2)=O)CCCC2(C1)CN(CC)C2 87200,CC1CN(C(=O)C(O)C(C)(C)C)C(C)CN1C(=O)C=Cc1cccnc1 87201,CN1CCN(C(C2CC(C3CC3)=NO2)=O)C(C(=O)NC2(CCF)CCC2)C1 87202,CCCCN=C(NCCc1ccc(Cl)c(Br)c1)NCCc1cccs1 87203,C1(C)(C(=O)NCC(C#C)CC2CC2)CCCN(C(C2CCC2(OC)OC)=O)C1 87204,c1(C(N(C2CCCCN(C(C3(C)CC=CC3)=O)C2)C)=O)cc(Br)cnc1O 87205,N1(C(C)=O)CCCCC1C(=O)NC(C)CCNC(c1cnc(NC(C)C)cn1)=O 87206,c1(OC)cc(NC(=O)C(N2CC3CC2CN3S(C)(=O)=O)=O)c2ccccc2c1 87207,C12(C)CCN(CC1)C(=O)C=CC2.C1(C(=O)NCC2CC(OC)C2)C2CCCC(=O)C12 87208,N1(C(C=CCN(C(CCCN(C(C)C)C)=O)C)=O)CC2NC(=O)OC2C1 87209,C1(C(=O)NCC2CC(F)CN2C(=O)C=Cc2ccco2)C2CCCOC12 87210,c1(CC)sc(=N)[nH]c1C(=O)NC1(CCCCNC(=O)C(C)CSC(F)(F)F)CC1 87211,c1(C(=O)NC(CN(C(c2c(CC)nns2)=O)C)C)cc[nH]c(=NC)c1 87212,C(=O)(C#CC1CCCOC1)NC(CNC(c1ccc(C(=O)NCCC)cc1)=O)C 87213,C12(C(N3CCC(NC(=O)C=CC=C(Cl)Cl)C3)=O)CCOCC1C2 87214,C(C1CCCCCC1)=CC(=O)N(C1CCN(C(c2ccc(C(F)F)s2)=O)CC1)C 87215,Cc1cccc2[nH]cc(C(N3CC(NC(c4ccsc4Br)=O)C(C)C3)=O)c12 87216,c1(C(N2C(CNC(c3ncc(OC)nc3)=O)COCC2)=O)c(OC)ccnc1F 87217,N1(C(C(c2cccnc2)OC)=O)CC(NC(c2ccc(F)s2)=O)CCC1C 87218,C1(CCNC(C2CCC(C)S2)=O)(OC)CN(C(=O)CC(C2CCC2)C2CCC2)C1 87219,N1(C(CCC2(C)CC2)=O)CC2CC1C2C(=O)NCC1CC(CF)C1 87220,C1(CNC(C2(OC)CCN(C(=O)CC3(CO)CC3)C2)=O)Cc2nccn2C1 87221,c1(OC2CCCN(c3cc(Br)cc(OC)c3I)C2=O)nc2c(s1)COCC2 87222,C1(C(=O)NC(CCCCNC(C(C)OCCOC)=O)(C)C)COc2ccccc2C1 87223,c1(C(=O)NCC2(F)CCC(CNC(COC)=O)CC2)sc2nnc(S)n2c1C 87224,N#Cc1cccc(OCC(=O)NCCCCCCNC(C2CCC(F)(F)C2)=O)c1 87225,CC1(C)NC(=O)CC1N(C1CCCC1)C(CN(C(=O)CCN1CCCC1)C1CC1)=O 87226,C1(C(C)C)CN(C(c2cc(O)n(CC)n2)=O)CCCN1C(c1nc(=O)n(C)[nH]1)=O 87227,c1(Nc2cc(NC(CCC)CCCN(C)C)ncn2)c(C)nc(=N)[nH]c1C 87228,C1(CC(=O)N(CCNC(c2nc(C)sc2)=O)C)CCCC(C)C1 87229,C(CC1=CCN(C(c2cccc3c2NCC3)=O)CC1)NC(CC1C(C)CCO1)=O 87230,c1(C(=O)NCc2ncc(C(C)(C)C)cn2)cc(Cl)c(Cl)cc1Br 87231,N=S1(=O)CCCC(NC(=O)NCc2nc(Cc3ccccc3Cl)no2)C1 87232,CCC(C)(O)C(=O)N1CCCC1C1(NC(C2(c3cnn(C)c3)CCCO2)=O)CC1 87233,C1(C(=O)NC(C2CCOC2)C)CCCN(C(=O)C(Cl)Cl)C1C 87234,N1(C(c2c(C)noc2C)=O)CCC2(CC1)CC2C(=O)Nc1c(C)ncnc1C 87235,C1(COC)C=CCCN1C(=O)C(CNC(=O)C(n1ccnc1C)C)N(C)C 87236,C1(NC(c2cc(SC)oc2)=O)CCC2(CC1)CN(C(c1cncc(F)c1)=O)C2 87237,N1(C(c2c(CNC(C3(C(=O)NC)CC3)=O)cco2)=O)CC(C)CCCC1C 87238,N1(C(CN(C2CCC2)C)=O)CCCC1CNC(=O)CC1CCC1 87239,Cc1cc(C(=O)NCC2CCN(C(c3cn(CCO)nn3)=O)C2)nn1C(C)C1CC1 87240,N1(C(CC)=O)CCOCC(NC2CC=C(C)CC2)C1.c12cncc(c1)C(=O)N2 87241,N1(C(C2(CC#C)CCCC2)=O)CCN(C(=O)CCN2CCC(O)CC2)C(CO)C1 87242,N1(C(C(C)=C2CCCC2)=O)CCN(C(c2cc(-c3ccccc3)no2)=O)C(C)C1 87243,Cc1nc(NCCCCC(N)=O)cc(=NCc2cnn(C)c2Br)[nH]1 87244,N1(C(c2oc(C)c(Br)c2)=O)CC(C)CN(C(=O)C(F)=C2CCC2)C(C)C1 87245,N1(C(C2(C#C)CC2)=O)CC2COCC(C1)C2NC(C12CCCN(CCC1)C2)=O 87246,C(CCCCC(=O)N1CCC(O)(C(C)NC(c2cc(Cl)c(Cl)n2C)=O)C1)OCC 87247,c1(C(=O)N(C(C2CCCN(Cc3ncccc3O)C2)C)CC)cccc2nccn12 87248,C(C(C)(C)CNC(c1nnnn1C1CCOC1)C1(CC2CC2)CC1)OC 87249,c1(-c2cnc(OCC)c(C)c2)cnc2[nH]cc(C(=O)NCC3CCCN3C)c2c1 87250,c1(C(=O)NCC2CCCCN2C(=O)CC2CCCCO2)cncc2nc[nH]c12 87251,CCCCCC1n2nnnc2C(COC)N1.C1(CCNC)(COC)CCOCC1 87252,N1(C(CN2C(C)COCC2)=O)CC2CC(C(=O)NCc3ncc(F)cc3F)(C2)C1 87253,Cc1cc(OCC(=O)NC(CNC(=O)CC(C)(C)C#N)CO)cc(C)c1 87254,N1(C(C(C)=CCC)=O)CC=CC(C(=O)NCc2ccccc2C)C1 87255,c1(C(=O)NC2CN(C(CC(C)c3ccco3)=O)CC2(C)C)cc2c(o1)CCCC2 87256,c1(C(=O)NCC2(C)CCN(C(CCCCCSC)=O)C2)cc2nc[nH]c2cc1F 87257,CC(C(C)(C)C#N)NC(C1C2CC1N(C(C1C=CCCC1)=O)C2)=O 87258,CCCCC(C(=O)NC(C)CCCNC(c1csc(O)n1)=O)c1ccc(Cl)cc1 87259,Cc1cc(C(=O)N(CC(O)CNC(c2ocnc2C(F)(F)F)=O)C)sc1Cl 87260,C1(C(F)F)(NC(c2nnc(C3CC3)n2C2CCS(=O)(=O)C2)=O)Cc2ccccc2C1 87261,C(CCCCn1cc(CNC(=O)Cn2nnc(CCO)n2)nn1)N(C(C)C)C 87262,N1(C(C(CCCC)NC(c2n[nH]c3c2CCC3)=O)=O)CC2CCCC(O)C2C1 87263,CC1CC(NCc2nn(C)c3c2COCC3)c2ncnn21 87264,N1(C(C2CCN(CC)C2)=O)CCC2(C(=O)NC(CO)CC(C)C)CCCC12 87265,n1(CC(N2CCC(CNC(=O)C(F)(F)C3CC3)C2)=O)[nH]cc2c(=O)ncnc1-2 87266,C1(O)(CNC(CCC(C)NC(c2ncnc(O)c2F)=O)=O)CC2C=CC1C2 87267,CC1(C)CC(CC(=O)NCC2CC2CNC(c2cc([N+](=O)[O-])on2)=O)NC1=O 87268,c1(C2C(CC)C2)ccccc1NNC(=O)Nc1cccc(CO)n1 87269,N1(C(CCOCC#C)=O)CCC2(CC1)CCN(C(c1ccc(F)c(O)c1F)=O)C2 87270,N1(C(C2(C)N(C(CC(C=C)CCC)=O)CC=C2)=O)CCOCC2(CCC2)C1 87271,C12(NC(C3C(COC)C3)=O)CCC1CN(C(c1ccc(Cl)cc1Cl)=O)C2 87272,C(CCC(C(=O)NCC1CC(C)C1)OC)NC(=O)Cc1cncnc1 87273,CC(CC(=O)N1CC(NC(c2cnoc2Br)=O)C1)c1ccccc1 87274,CC(C)C(C)C(=O)NC1(CCNC(=O)Cc2coc(-c3ccccc3)n2)CC1 87275,C1(NC(C2CCC3(CC3)N2C(c2cocn2)=O)=O)CC2C=CCC(C1)C2 87276,C1(CNC(CCCC)=O)CCC(F)(CNC(=O)C(C)CCN(C)C)CC1 87277,c1(NC(C23CCC2CN(C(C2CC=CCC2)=O)C3)=O)ccc2ccccc2n1 87278,C(=O)(CCCN(C)C)N(C1CCC(NC(C2(F)CCC2)=O)C1)C 87279,C1(F)(CNC(C(COC)N(C)C)=O)CCC(CNC(c2cnccn2)=O)CC1 87280,C1(Nc2ncc(OC)cn2)C(C)CN(C(c2occc2C(C)C)=O)CC1C 87281,C1(NC(c2ccnc(F)c2Cl)=O)CCN(c2ccnc(Br)n2)CC1F 87282,N1(C(CCCC)=O)CCCC(CCNC(c2sc(F)cc2C)=O)CC1 87283,C(C(=O)N1OC2CCC1C2)C1(C)N(C=O)CCC1.C(CCCC=O)N(C)C 87284,CC1OC2(C(N3CCC3CNC(=O)CCN3CCN(C)CC3)=O)CC1C2 87285,N1(C(C2CCC(C)O2)=O)CCCN(C(c2cncc(Br)c2)=O)CCC1 87286,N1(C(C2N(C(CC(C)(C)N(C)C)=O)CC(=O)NC2)=O)CCC2(CCC2)CC1 87287,c1(C(=O)NC(c2cnc[nH]2)C)coc(CNC(c2ccsc2Cl)=O)n1 87288,Cc1cc(C(=O)NCCN(C(=O)Cc2cncc(C#N)c2)C2CC2)ccc1Cl 87289,O=C1CC(C(=O)NC23CCN(C(c4cccc(Cl)c4F)=O)CC2C3)CC(=O)N1 87290,c1(C(N2C(C)CC(NC(c3cnc(O)nc3O)=O)C2)=O)cc(Cl)c(Cl)cc1N 87291,C1(CNC(=O)OCC)(NC(=O)C=CS(C)=O)CCNCC1 87292,Cc1cn2cc(C(=O)N(CC(C)NC(c3cnc(Cl)c(F)c3N)=O)C)nc2s1 87293,N1(C(C(CCC)O)=O)C2CCCC1CN(C(=O)C(C)(C1CCOCC1)OCC)C2 87294,c1(CNC(C2(CC)CCN(C(C(C=C=C)C)=O)C2)=O)ccc(C#N)c(C)c1 87295,N1(C(C2N(C(C)=O)CSC2)=O)CCCC(O)(CNC(c2ccn(C3CC3)n2)=O)CC1 87296,Cn1cnc2cc(C(N3CC(CNC(C4CCCSS4)=O)C3)=O)ncc12 87297,C=CCC(C(=O)N1CC(N(C)C(c2ccn(CCC)n2)=O)C1)c1ccccc1 87298,C=CCCCCCCCC(=O)N(C)CC1CCCC(CNC(=O)CCSCC)C1 87299,c1(OC)cccnc1CNC(C1(CCNC(=O)CC2CC2C)CCCC1)=O 87300,CC(C)CCC(O)C(=O)NCCCC(C)C.C12CCN(CC1)CC(=O)NC(=O)N2 87301,c1(CCC)n[nH]c(=NC(=O)N2CCc3cc(Br)sc3C2)s1 87302,N1(C(C(CC)COC)=O)CCCC(C)(C(=O)NCc2nocc2C(C)C)C1 87303,c1(CC(N2CCC(N(C(=O)Cc3cncnc3)CC)C2)=O)ccccc1S(C)=O 87304,C1(C(=O)NCCN(C(=O)CC(C)(F)F)CCOC)CCc2cncn2C1 87305,C1(NC(c2occ(C)c2)=O)COC2C(NC(=O)C(F)F)COC12 87306,C1(N2CCOCC(C(=O)NC3(c4nc[nH]n4)CC3)C2)COC2C(O)COC12 87307,c1(C(=O)NC2(COC)CCN(C(c3ccccc3F)=O)C2)cc2cccnc2o1 87308,c1(C(=O)NC2(CNC(c3n[nH]cc3F)=O)CCOC2)cnn2c1OCCC2 87309,c1(C2CCC2)cc(C(N(CCN(C(=O)CCC2(C)CC2)CC)CC)=O)ccc1F 87310,N1(C(c2n(C)ncc2)=O)CC2CC1(C(N1CCC(C(F)F)CC1)=O)C2 87311,C1(C(=O)NC2(CNC(c3occ(C)c3)=O)CCOC2)COC(C)(C)CO1 87312,C1(N(C(=O)CN(c2ccccc2)CC(=O)O)C)CCN(CCO)CC1 87313,c1(CC)ccc(C(N2CC(CNC(=O)CCc3n[nH]c(=N)s3)C(C)C2)=O)c(F)c1 87314,C1(NC(CCN(C)CC)=O)CC2CN(C(=O)CC3CCCCC3(C)C)CC2C1 87315,CC1CN(C(c2ccc(C3CCOC3)s2)=O)CCN(C(=O)C=C2CCOCC2)C1 87316,n1(CCC(=O)NCC(C2CCC2)NC(C23CCC2CC3)=O)ccc(O)nc1=O 87317,N1(C(c2c(OCCC)cccc2)=O)CC(NC(=O)C(C)c2ccco2)CC(C)C1 87318,C=CCC(CC(C)C)C(=O)N1CCOC(CN(C(=O)CCc2cnn[nH]2)C)C1 87319,C1(CC)CN(CC(c2c(C)noc2CBr)C)CCN1CC(C)O 87320,c1(C(=O)NCCCC(C)NC(=O)CC2CCCC(C)(C)O2)nn(C)c2c1CCC2 87321,Cc1nn(C)c(O)c1CNC(=O)NC(c1ccnn1C)C 87322,C1(CNC(CCCCSC)=O)CCN(C(=O)Cc2cncc(F)c2)CC1C 87323,N1(C(C2(C#N)C(C)(C)C2)=O)CCC(C=CC(=O)NC2CC(=C3CC3)C2)CC1 87324,C1(C)(C(=O)NCCC2CCCN(C(C(=O)N(C)C)=O)C2)CCS(=O)(=O)CC1 87325,C1(O)(CN(C)Cc2ccc(C(=O)NC)cc2)C2CC3CC(C2)CC1C3 87326,C(CN=c1[nH]c(NCC(CO)C2CC2)nc2cc[nH]c12)C1(COC)CC1 87327,C1(CNC(CC)=O)CN(C(=O)C(C)(C)COC(C)C(=O)OC(C)(C)C)CCCO1 87328,N1(C(CC2N(C)C(=O)CC2)=O)CC(C(=O)NCCn2cc(C#N)cn2)CC1(C)C 87329,c1(OC)ccccc1C=CC(=O)NCC(C)(CO)NC(c1cc(F)ccc1C)=O 87330,C1(C(=O)OC)CCC(C)N(CC#CC(OC)OC)C1.C(C(C)C)O 87331,c1(NCC(=O)NCCCC2(NC(CSCCC#N)=O)CC2)ccc2ccoc2c1 87332,c1(OC)nc(NC(C2CC2NC(c2scc(C)c2Cl)=O)=O)cnc1C#N 87333,c1(COc2c(OCC)cccc2)ccc2c(c1)OCCO2 87334,N1(C(C2(C)CCOCC2)=O)CC2CC(NC(=O)C=CC3CC3)CC2C1 87335,C1(CNC(C=CC(N)=O)=O)CCN(C(=O)CCNC(C2CCC2)=O)C1 87336,N1(C(CC(C)(C)SC)=O)CC2(CCCN(C(=O)CCc3ccccc3Cl)C2)C1 87337,C1(C(=O)NC(C2(O)CN(C(c3nc(OC)oc3)=O)C2)C)CC(C)(C)C(C)(C)C1 87338,c1(N2CCC(OC)(CO)C2)nc(NCC2(CF)CCC2)c2cnn(C)c2n1 87339,C1(NC(=O)CC2CCC(C3CC3)O2)CCCN(c2ccccc2)C1=O 87340,c1(CNC(NCC(=C)Cl)=NCCC2CCOCC2)ccc(OC)c(F)c1F 87341,CC1CC(C(=O)NC(C2CN(C(=O)CCCc3ccc(F)cc3)C2)C)CCO1 87342,N1(c2nccc(CC(=O)OC)n2)CC2(CCCC2NC(=O)CCC(C)C)C1 87343,Cc1cc2ccc(C(N3CCC(CNC(C4CC(C)OCC4)=O)C3)=O)cn2c1 87344,Cc1cnc(NC2CC(NC(=O)Cn3nc(O)ccc3=O)C2(C)C)nc1O 87345,c1(C(N(CCN(C(c2cccc(C)c2F)=O)C(C)C)C)=O)ccc2nn[nH]c2n1 87346,C12CN(CCN(C(=O)CO)C1)C2=O.CC1CN(C(=O)OC(C)(C)C)CC1CO 87347,C1(NC(C(C)SCC)=O)CC(O)(CNC(C2(n3cnnn3)CC2)=O)C1 87348,N1(C(C(=O)Nc2ccc(OC)cc2)CCC2CC2C)CCC(S(=O)(=O)C(F)F)C1 87349,c1(NC(C2CCCC3CC23)=O)c(F)cccc1F.CC1C(=O)N(C)CCN1C 87350,c1(OC)cc(CN2CC(C(N3CCC(C(F)F)CC3)=O)CC(F)C2)cc(I)c1O 87351,C12(CNC(C3CN(C(C)=O)C3)=O)CC1CN(C(C1CN(C)CCO1)=O)C2 87352,Cc1cccc(N(c2ccnn2-c2ccccc2)C(=O)C(=O)NC(C)C)c1 87353,CCC(CC(=O)N1CCN(C(=O)CCSc2ccc(C)cc2)CC1CC)C(F)F 87354,c1(OC)cccc2c(CC(=O)NCCCN3CCC(O)CC3)c[nH]c12 87355,Cc1cccc(N)c1C(=O)NC1CCN(C(C)C)CC1C 87356,c1(CC)onc(C)c1C(N1CC2CC2(NC(=O)CCc2cccc(OC)n2)C1)=O 87357,c1(C(N2CCCC(OC(C)(C)C)C2)C(=O)NC(CC)(C)C)ccc2c[nH]nc2c1 87358,c1(C(N(CC(C)NC(c2cnc(C(C)O)s2)=O)C)=O)cnn(C)c1C1CC1 87359,C1(C(N(C2CCC2O)C)=O)CC(O)C(O)CC1CNC(C1(N(C)C)CC1)=O 87360,C(=O)(C1=COCCC1)NC(C1CCCCC1)CNC(c1noc(CC)c1C)=O 87361,Cc1cc(N)c(C(=O)NCC2CN(C(c3ncccc3Br)=O)CCO2)cc1F 87362,c1(C(=O)NCC2(OC)CCN(C(=O)C=C(Cl)Cl)C2)ccc2c(c1)OCC2 87363,C1(NC(C(CC#C)C)=O)CC2(C1)CN(C(c1ccnc(OCC)c1)=O)C2 87364,c1(CC(=O)NCC(C(C)C)N(C(COC)C)C)cc2ccccc2o1 87365,c1(SCCC(=O)NC(CNC(C(CC)OC)=O)C)ccc(C)cc1 87366,c1(OC(CC)C)cc(N2CCC(C3CC(N)CCO3)CC2)nc(C)n1 87367,C1(CNC(c2ccc(C3CCCNC3)cc2)=O)CCNCC12CC2 87368,CC(CCCN(C1(N(C)C)CC1)C(c1ccccc1)=O)C1CCCO1 87369,C(C1=CCCN(C(C2C3CCC(F)(F)C23)=O)C1)NC(=O)CC(C1CC1)C1CC1 87370,c1(C(=O)NCC2CCC(C)CN2C(=O)CC(C)(C)C#N)ccnc(P(C)(C)=O)c1 87371,C1(CC(=O)NC(CC(=O)NCCCn2c(C)ncc2)C2CC2)CCCCN1C 87372,c1(C(=O)NCC2C(C(=O)NCC(=O)N(C)CC)CCC2)ccccc1CC#N 87373,C1(C(=O)NC2CCC(NC(Cc3ccc(C)o3)=O)CC2)CC2CCCCCCC12 87374,c1(C(=O)NCCC(=O)N(C2(C(N)=O)CCOC2)C)ccc(CC#N)cc1 87375,c1(CCC(=O)NCCOc2ccc3cccnc3c2)cccc2c1OCCO2 87376,C1(CNC(=O)CC2(c3nn[nH]n3)CCCC2)C=CCOC1 87377,N1(C(C2CCC(=O)N2)=O)CC2(CCCC2NC(c2ccc3nc[nH]c3c2)=O)C1 87378,c1(C(=O)NCCCC(C)(C)O)cccc(C2CC2)c1.C(=O)(C(F)(F)CN1CCCC1)N 87379,C1(C(N(C2CCN(C(C3(C)CC(C(F)(F)F)C3)=O)C2)C)=O)CC2C=CC1CC2 87380,N1(C(CNC(CC)=O)=O)CCC(CC(C)NC(c2sc(C)nc2CC)=O)CC1 87381,C(=O)(C1=NOC2COCC12)N(CCNC(C(C)SCC)=O)C1CC1 87382,C=CCCCCC(=O)NC1COCC1CNC(c1c[nH]c(Br)c1)=O 87383,N1(C(c2occ(C)c2)=O)CC2OCCN(C(=O)CCCc3ccncc3)C2C1 87384,C(C1=CCCOC1)NC(C#CCNC(C1C(C#N)C1)=O)=O 87385,Cc1cc(C(=O)NCc2cc[nH]c2C(=O)NCC(F)C2CCC2)[nH]c1C 87386,c1(NC(C(=O)N(C(C)(C)C)C)=O)cncc(SC2CC3CCC2C3)c1 87387,N1(C(C(C(C)C)O)=O)CC2CN(C(=O)COCC3CCCCC3)CC2C1 87388,c1(C(C)(F)F)ccccc1C(N1CC(CNC(=O)CCC2CC3CCC2C3)C1)=O 87389,C1(NC(CC(C)(C)C)=O)CC2(C1)CN(C(c1nc(Br)cnc1N)=O)C2 87390,Nc1cccnc1C(=O)NCC1COCCN1C(=O)CN1CCOC1=O 87391,C1(CNC(c2cnc(OCC)nc2)=O)CN(C)CCN1C(c1csc(=N)[nH]1)=O 87392,N1(C(c2n(CC)ncc2)=O)CC(CNC(=O)CC2CCCCN2C)C(O)C1 87393,c1(CCC(=O)N(C2CCN(C(CCC(=C)C)=O)C2)C)cn2ccccc2n1 87394,c1(OC)cc(OC)[nH]c(=NC2CCC(C)N(C(C3CCC4(CCC4)O3)=O)C2)n1 87395,c1(CNC(NC(CC)C)=NCC2CN(C)CCO2)ccc2c(c1)CCCC2 87396,c1(NC(C2CCC(NCc3c[nH]c(Br)c3)CO2)=O)cccc(O)c1F 87397,C=Cn1nccc1C(=O)NC(C1CCN(c2nnc(C(N)=O)s2)C1)C 87398,CCCCCCCCC(=O)NCc1n[nH]cc1C(N1CCC2CCC12)=O 87399,c1(OC)ncc(S(=O)(=O)N(CC(c2ccccc2C)O)C)cc1C 87400,c1(NC(c2n[nH]cc2NC(c2cc(Br)cnc2O)=O)=O)cccc2c1OCC2 87401,C1(C(=O)NCC2CN(C(c3cnc[nH]3)=O)CC2O)CN2CC3CC2(CO1)C3 87402,N1(C(C(C2CC2)SC)=O)CCC(CNC(c2ccc(Cl)c(C(F)F)c2)=O)C12CC2 87403,Cc1csc2ncnc(N3CCCC(CCNc4cnnn4C)C3)c12 87404,c1(CC(=O)NCC(CC)NC(c2csc(-c3ccoc3)n2)=O)c[nH]c(=N)nc1O 87405,C12(CNC(c3cc(C)c(F)cc3)=O)CCCC1N(C(C1COC(C)C1)=O)CC2 87406,C(CC(F)F)(C(=O)NC(C)C(=O)N(C)C)NC(C(C)OCC=C)=O 87407,C=CCC(C(=O)N(CC(O)CF)C)NC(=O)CCCN1CCCC1 87408,Cc1nc(N2CCC(NC(=O)C=Cc3cncn3C)C2)c2scc(C)c2n1 87409,C1(C(N(CCOC)CCNC(=O)CC=C(C)C)=O)CCCCC1C(F)(F)F 87410,c1(C2C(C(=O)NCCOCCCNC(=O)CC3CC=CC3)C2)nc(S)n[nH]1 87411,c1(NC(C)=O)ccc(CC(N2CCCC(NC(C3CCCSC3)=O)C2)=O)c(Cl)c1 87412,c1(C(=O)NCC2(CC(=O)NC3C=CC(CO)C3)CCCC2)coc2c1COC2 87413,N1(C(C2CC(C)(C)C2)=O)CC2CC1(C(=O)NCC1CC3CCC1C3)C2 87414,c1(C2CCN(C(c3cnn(CCC)c3Cl)=O)C2)cc(F)cc(Cl)c1 87415,c1(OCCCC(=O)NCCN(C(c2cccc(SC)c2)=O)C)ccc(C#N)cc1 87416,c1(CC)nn(C)c(CC)c1CC(N1CC(C)C(NC(C2CCC(=O)N2C)=O)C1)=O 87417,N1(C(C2CC=C(C)CC2)=O)CCC2C(C1)CN2C(c1cc(C)cnc1C)=O 87418,C(c1c(C)nn(C)c1Cl)=CC(=O)NC(CC)(C)CNC(C1CN2CCC1CC2)=O 87419,C1(CCN)CCN(C(C2CCCCC2OCC(C(CNC(CC)=O)=O)=O)=O)CC1 87420,N1(C(C2N(C(CCC(C)NC(C)=O)=O)CCC2C(C)C)=O)CCC2(CC1)CN(C)C2 87421,c1(C(=O)NC(C(C)C)C(C)NC(=O)Cc2cncs2)cccc2c1OCC2(C)C 87422,CC1CCN(C(C2CCC=CO2)C(=O)Nc2ccc(Cl)cc2F)CCS1 87423,FC1(F)CCCC(CCNc2ccnn2-c2ncccc2Br)CC1 87424,C(=O)(C1CCCc2ccccc21)NC(CN=c1[nH]nc(C(=O)OC)s1)C 87425,CCC(C)C(O)CC(=O)N1CCC(CC(=O)NCC=C(Cl)Cl)CC1 87426,C(CO)(CCCNC(c1ccc(=N)[nH]c1)=O)NC(c1c(C(C)(C)C)c[nH]c1)=O 87427,c1(NCC(=O)N(C2CCN(C(C3(CC)CC3)=O)C2)CCO)ccccc1[N+](=O)[O-] 87428,C1(NC(CCc2cnc(C)o2)=O)CCCC(C(=O)NC2CC(CC(N)=O)C2)CC1 87429,Cc1cnn(C)c1CC(=O)NCC1(CNC(C2CC2C)=O)CCCC1 87430,CCC(C)(C(=O)O)n1cc(Br)cn1.n12cc(nn1)C1(CC1)C(=O)N1CCC21 87431,c1(C(C(=O)NCC2(CN(C(=O)C(C)NC(N)=O)C)CCC2)OC)ncc(NC)s1 87432,C(CNC(=O)C(C)(C)OC(C)C)(CC(C)C)NC(C(Cn1ccc(C)n1)C)=O 87433,c1(NC(C2(CC)CN(C(=O)Cc3ccoc3C)C2)=O)cnccc1CO 87434,C(C)(CCCCNC(=O)C(F)CC1CCOC1)NC(c1ccc(C)o1)=O 87435,C1(CC(=O)NC(Cc2ccoc2)C(=O)NCc2nocc2C2CC2)CCCSC1 87436,Cc1cc(C)c(C(=O)NCC(C)(C(C)C)NC(C2CCNC2=O)=O)o1 87437,C1(C(=O)NCCCO)CC=CCN1C(C1CCN(CCOC(F)F)C1)=O 87438,c1(N(C23COC(COC)(C2)C3)C(N(C)CC)=O)cccc(Cl)c1 87439,CC1(C(=O)NC2CCC(NC(=O)CCOC3CCCC3)C2)CCc2ccccc21 87440,N1(CC(C)C)CC2C3CCC(C2C1)N(C(=O)CO)C3.S1(=O)(=O)c2c[nH]c(c2)N1 87441,N1(C(c2c(CC)nccc2)=O)CCC2(CCCN2C(C23CCC2CC3)=O)C1 87442,N1(C(c2c(C)c[nH]n2)=O)CCC(CN(C(=O)COC2CCCCC2C)C)CC1 87443,CC1(C)CC(NC(c2coc(C3CC3)n2)=O)CN(C(=O)Cc2n[nH]c(=N)s2)C1 87444,c1(OC)ccc2cc(C(N3CCOCC(NC(=O)C(F)C(C)(C)O)C3)=O)sc2c1 87445,C1(CNC(Cc2c(C)cnn2C)=O)CCCCN(C(c2cnn(C3CC3)c2)=O)C1 87446,Cc1ccc(C#N)cc1C(=O)NCc1ncoc1CCNC(C1OCCC1C)=O 87447,CC#CCC(C(=O)N1CCCC(CC)(CO)C1)NC(=O)C=CC(C)OC 87448,c1(OC)ccc2c(c1)c(C1CC1)c(C)n2CCNS(=O)(=O)c1nn(C)nc1Br 87449,c1(C(=O)NCCN2C(NC(c3cnc(S)[nH]3)=O)COCC2)cc(F)cc(F)c1 87450,C1(C(=O)NCC(O)CO)(OC)CCN(Cc2ccc(F)cc2)CC1 87451,C1(CCC)CN(C(C2CCC(=O)NC2)=O)CCN1C(=O)CC1CCC1 87452,c1(C(N2C(CCNC(c3c(CC)nn(C)c3)=O)COCC2)=O)ccc(F)cc1Cl 87453,C1(N(C(c2c(CC=C)cccc2)=O)C)CC2CC1N(C(c1cn(C)cc1C)=O)C2 87454,CN1CC2CCN(C(=O)C(CCF)NC(c3c[nH]cc3C3CC3)=O)CC2C1 87455,c1(NC(C23C(CN(Cc4ccc(OC)nc4)C2)C3)=O)cccc2c1OCC(=O)N2 87456,C1(C(N2CCC(C(C(=O)NCC3(CC(=O)OC)CC3)C)C2)=O)CCC(O)CN1C 87457,N1(C(CS(CC)(=O)=O)=O)CCCN(C(C2CC(F)C(=O)N2C)=O)C(C(C)C)C1 87458,C(=O)(C1OCCn2ccnc21)NC1C(CNC(c2c(C)cccc2Cl)=O)CC1 87459,c1(NC(C23C(CN(C(c4cccc(C#C)c4)=O)C2)C3)=O)ccc2c(c1)OCO2 87460,N1(C(C2(C(=O)OCC)CC2)=O)CCC(C)(NC(C=C(CCC)C)=O)CC1 87461,N1(C(CC(C(=O)OC)C)=O)CCC(C)(C)CC1C(=O)NCC(CC(C)C)OC 87462,c1(CN2CCCOCC2)ccc(Br)nc1.C(C(=O)N)S.N(CCSC)(CC)CC 87463,C1(C(=O)NC(COCCOC)C)COCCN(C(=O)C=CC(C)(C)C)C1 87464,c1(CC)cccc(C(N2CCC(C)C2CNC(=O)C=CC2CC2)=O)n1 87465,c1(-c2c(C(=O)NCC3(C(=O)OCC)CCOCC3)nco2)cccc(F)c1 87466,Cn1c(NC(=O)C(O)Cc2ccccc2Cl)nnc1C1CCOC1 87467,C(C)(C)(CC(F)C(=O)N(C1CCC2(CC1)CC2)C)NC(C(CCCC)O)=O 87468,CC1(C)CC(CNC(C2OCC3CCCC23)=O)CN1C(c1cnc(Cl)c(N)c1)=O 87469,C1(C(=O)NC2(C)CN(C(=O)CC3(O)CCOC3)C2)Cc2c(F)cccc2O1 87470,N1(C(c2c(C)c[nH]c2)=O)CCN(C(=O)CCc2cncnc2)CC(C)C1 87471,C1(CC(=O)NC2(CNC(=O)CC3CCCC3)CCC2)CCCOC1c1cn[nH]c1 87472,C=CC1(O)CCN(C(=O)CC(C(C)OC)NC(c2cncnc2CC)=O)C1 87473,C(=O)(C(C1=CCSC1)N(CCS(=O)(=O)C(C)(C)C)C1CC1)NC1(C)CCCC1 87474,CCCCCCCCC(C)(C)C(=O)NC1CCCCN(C(=O)CC2CCC3CC23)C1 87475,C(C(C)(C)CC1CN(C(=O)C(C)(C)C)C1)OC.C12(CCC1)C(=O)NC2 87476,c1(SCC(N)=O)cccc(C(N2CC(F)CC2c2ccc(F)cc2)=O)c1 87477,C(C(CC(=O)NCC(C)(O)C1CC1)NC(c1cscn1)=O)OC.C(C)(=O)N 87478,c1(NC(CCC)=O)cncc(CCC(N2CCN(CC(F)(F)CO)CC2)=O)n1 87479,c1(C(F)(F)F)ccc(CNC2CCC(Sc3ccccc3)C2)cc1 87480,C1(C(=O)NC(c2ccc(OC)cc2)C)CC12CCN(c1nc(Cl)ncc1F)CC2 87481,CC(C(=O)Nc1cnc(F)nc1)C(C)NC(c1ncc(F)cn1)=O 87482,CCCC(C)(C)C(=O)NCC(CNC(c1cnn(C)c(=O)c1)=O)OC 87483,CC1C(NC(C2CCN(c3ccncc3)CC2)=O)CCCN1C(=O)CCCF 87484,N1(C(CCc2ccc(C)cc2)=O)CCC2C(CCCN2C(C2CCSCC2)=O)C1 87485,N1(C(CCSCCC)=O)CCC2CCN(C(c3nc(C)c(N)cc3C)=O)C2C1 87486,N1(C(CCOc2ccc(C)cc2C)=O)CCN(C(=O)CNS(C)(=O)=O)CC(O)C1 87487,CC(C)C(CNC(=O)CC1CCCC(=O)C1)C(=O)NCc1c(F)cccc1F 87488,c1(CCC)ccc(CC(N2CC=CC(N(N3CCC(F)C3)C(=O)CC)C2)=O)cc1 87489,c1(CCC=O)cccc(CC)c1.C(=O)(CN(C)CC)OCCC 87490,C1(C(N(CCC#C)C(C)C)=O)CC(C)CN(C(C2(SC)CC2)=O)C1 87491,C1(N(C(=O)CCN2CC=CC2)C)CN(C(=O)CC2CCC(F)(F)CO2)CC1(C)C 87492,C(N=c1[nH]c(=NCC(C(C)C)N(C)C)[nH]c2c1CCCCC2)c1snc(C)n1 87493,CC1(CC(N2CCC(CNC(C3(CCF)CC3)=O)C2)=O)CC1(F)Cl 87494,c1(C(=O)NC2CCN(C(C3CC4C(C3)C4(F)F)=O)CC2F)occ2c1CCOC2 87495,C(c1cccc(C#N)c1)=CC(N1CC(OC)C(NC(C2CCCOC2)=O)C1)=O 87496,N1(C(CC2C(C)(C)CCO2)=O)CC2COCC(C1)C2NC(=O)C1=C(Cl)CCC1 87497,N1(C(COCC)=O)CCCC2CN(Cc3ccc(S(C)(=O)=O)c(C)c3)CCC12 87498,c1(CC)nc2n(n1)CC(C(N1CC3(CCNCC3C(=O)NC)C1)=O)CC2 87499,c1(SC(CC(=O)NCC2(NC(C3C(CC(C)C)C3)=O)CC2)C)cccc(F)c1F 87500,C1(NC(c2nnc(S)s2)=O)CCCC1Cc1ccccc1 87501,c1(C(C(=O)NCCC(C)F)NC(C2CC(=C3CC3)C2)=O)cccnc1 87502,CCC(C)(O)C(=O)NCC1CC(OC)CN1C(=O)CCc1ccco1 87503,N1(C(CCCCCSC)=O)CCC2(CCOCC2)C(NC(C2CC(SC)C2)=O)C1 87504,C1(C#CC(=O)NC2CCCC(N(C)C(c3cc(C)c(C)[nH]3)=O)C2)(CC)COC1 87505,N1(C(COCCSC)=O)CCC(CNC(C2(CCF)CC2)=O)C1 87506,C(CCCCCC(=O)NC(C1CCN(C(c2ccc(C(N)=O)cc2)=O)C1)C)SC 87507,N1(C(C(NOC)=O)=O)CC(C(=O)NC2(c3cc[nH]n3)CC2)C(C)(C)C1 87508,Cc1ccc(C=CC(=O)NCC(C)CN(C(=O)CCSCC(N)=O)C)cc1 87509,CCS(=O)(=O)CC(=O)N1C2CCC(C2)C1CNC(=O)C(c1cnccc1C)(C)C 87510,C(CC(C)(C)C)(C(=O)N1CCC(C)(C(N2CCCCC2)=O)C1)OC 87511,C12(C(N3CCC(CNC(c4c(C)nc(CO)s4)=O)C3)=O)CCC(CC1)CC2 87512,C(=O)(CCC(C)N(C)C)OC.C12CCC(CC1)N(C(C)=O)C2 87513,C=CCCCCCCC(=O)NC(C1CCCCC1)CNC(C1(C#N)CCCC1)=O 87514,N1(C(c2ccc(F)c(C)c2Cl)=O)CCC2(CC1)CN(C(=O)C(C)(C)F)C2 87515,c1(C2(NC(N(C)CC34CC(C(=O)OC)(C3)C4)=O)CC2)ccc([N+](=O)[O-])cc1 87516,C1(NC(c2cn3nc(C)sc3n2)=O)CC(N=c2ccnc(S(C)(=O)=O)[nH]2)C1 87517,c1(C(=O)NC2CCC(C)N(C(=O)Cn3nccn3)C2)ccn2c1CSCC2 87518,C1(NC(C(=C(C)C2CC2)F)=O)CCN(C(=O)C=Cc2cccnc2)CCC1CO 87519,c1(OC)ccc(Br)cc1S(=O)(=O)NCCC1CCCC(C)C1 87520,C(CCCC#N)(C(=O)NC(C)C)N1CC(C)CC(C(=O)NC)C1 87521,c1(NC(C(n2cc(C(C)OC)nn2)C)=O)ccccc1[N+](=O)[O-] 87522,C(c1ccccc1)=CCN(CC(=O)N(C1CN(C(=O)CC2(C)CC2)C1)C)C1CC1 87523,c1(C(=O)NCC(CN(C(C(=O)NCC)=O)C)C)n[nH]c(CC)c1[N+](=O)[O-] 87524,C(=O)(C1=C(Cl)CCC1)N1CC(CNC(c2c(CC)n(C)nc2)=O)C(C(F)(F)F)C1 87525,N1(c2ccnc(SC)n2)Cc2nccn2CC(NC(=O)CCc2ccn(C)n2)C1 87526,C=CCC(C)(CC)C(=O)NC1CCCC1CC(=O)NCCc1cnnn1C 87527,c1(OCCC)nc(C)ccc1C(=O)NC(CNC(=O)CCC(C)C)C1CC1 87528,c1(C(=O)NCC(CCNC(C(CC)SC)=O)OC)c(-n2cccn2)cccc1F 87529,C1(C(N2CCC2c2nncn2C)=O)(OC)CN(C(C2CCC2C(=O)OC)=O)C1 87530,Cc1nc(C(C)C)ccc1C(=O)NC1CCCC(NC(c2cc(F)n(C)n2)=O)C1 87531,C1(NC(=O)CCCCCF)CCC2(CCN(C(c3csc(C(F)F)n3)=O)C2)C1 87532,c1(C(C(=O)OC)NC(=O)COC2CCCOC2)ccccc1F 87533,CC1(C)CN(C(=O)NCc2snc(C(F)(F)F)c2Cl)Cc2cccc(Br)c21 87534,C(=O)(CS(=O)(=O)C1CCCC1)NCC(C(C)(C)C)NC(C1CC2(C1)CC2(F)F)=O 87535,Cc1ccc2snc(C(N3CC(C)(NC(C4CC5CCCCN5C4)=O)C3)=O)c2c1 87536,C1(NC(Cc2ccn(C(C)C)n2)=O)COC2(C1)CN(C(C1CCCOCC1)=O)C2 87537,CC1OCCCC1C(=O)NC1(C(F)(F)F)CC(C(F)F)(NC(=O)CC2(C)CCC2)C1 87538,Cc1ncnc(C)c1C(N1CCCC1CNC(c1ccc(I)c(C(F)(F)F)c1)=O)=O 87539,CCC(C(=O)NCCCOCCNC(=O)CC1(C)CC1)n1ccnc1 87540,C(CN=C(NCCc1cnnn1C)NCC1CCCC1C1CC1)SC 87541,C(=O)(C1=CCCOCC1)N1CC(CCc2cn(CC(C)O)nn2)C1 87542,N1(C(CC(C)N(C(C)=O)C)=O)CCCC(C(N2CCC(N3CCC3)CC2)=O)C1 87543,c1(CC#N)cc(Br)ccc1C(=O)NC1CC1C(=O)N=c1cc[nH][nH]1 87544,CC1(C(=O)NCCc2cscn2)CCCN1Cc1cccc(F)c1 87545,C1(O)(Cn2cc(C(C)C3CC3)nn2)CCN(C(c2cccc(F)c2)=O)C1.c1ccsc1 87546,C1(CC(=O)NC2(CC3CC3)CC2)(C(=O)NC(C)CC2CCC2)CCC1.COC 87547,N1(C(c2c(C)ncnc2)=O)CCC2(CCSCC2)CC1 87548,CC1(CNC(C2(F)CCCN(C(c3coc(CO)c3)=O)C2)=O)CC2CCC1C2 87549,C1(CC(=O)OCC(C)(C)C)(C(=O)OC(COC(C)=O)C(C)C)CCCCC1 87550,c1(C(=O)NC(C(=O)NC)Cc2cc(Br)ccc2Br)coc(C2=CCCCC2C)n1.CCO 87551,C1(C(=O)NCC2(NC(=O)Cc3csc(S)n3)CC2)CCCC1(F)F 87552,N1(C(CC(C)(C)OC)=O)CC2CC1CN2C(c1cccc(-n2ccnc2)c1)=O 87553,Cc1cc(Cl)ncc1C(N1CCOCC1c1noc(-c2ccoc2C(C)C)n1)=O 87554,C1(CCNC(C2N(C(C)C)CCC2)=O)CCCN(C(C2CCCN2C(C)C)=O)C1 87555,C#Cc1cc(F)c(C(=O)NC(CO)C(C)NC(c2cnnn2C2CC2)=O)cc1F 87556,C12(C(=O)NCCCOCCNC(c3c(C)nns3)=O)CCC(C1)C2(C)C 87557,C(CCC(=O)N1CCCC1C(=O)N(C1CCC1)C)OC(C)C 87558,CP(C)(=O)C(O)C(=O)NCCOC1CCN(C(=O)CCC2CCCC(=O)N2)CC1 87559,c1(C(=O)NC(C)CCNC(C2(CCF)CC2)=O)cc([N+](=O)[O-])ccc1OC(F)F 87560,c1(C(=O)NC(CNC(C(CC=C)C)=O)(C)C(C)C)cc2c(s1)CCC2=O 87561,c1(OC)ccc(Cl)c(C)c1C(N1CCC2CN(C(=O)C(C)CC3CC3)CC12)=O 87562,Cc1cc(C(=O)NC(C2CCN(C(=O)C=Cc3cncs3)C2)(C)C)no1 87563,CC(C(F)F)N(C)N1CCC(C(N2CCOCC2)=O)CC1 87564,N(C1COc2ccc(F)cc21)C(C1COC2(CCC2)OCO1)=O 87565,Cc1cncc(C)c1C(=O)NC(CCNC(c1cc(C(F)(F)F)c[nH]1)=O)C(C)C 87566,N1(C(C(C=C)C)=O)CCN(CO)CC1.c1(C)ccc(Cn2cc(C)cn2)cc1 87567,c1(C(=O)NC2(CNC(C3C(C)CCCO3)=O)CCOCC2)ncc(F)cc1F 87568,Cc1nc(NC(CNC(=O)CC(C)n2ccnc2)C(C)C)c2c(C)c(C)sc2n1 87569,CC1=C(C(=O)N2CC=CC(NC(C3CCCSC3)=O)C2)CCCO1 87570,c1(SCCOCCCCC=C(C)C)ccccc1.C12(CC1)NC(=O)N2 87571,C1(C(N2CCCC(N(C)C)C2)=O)CCC2(CC2)N1C(C1(N(C)C)CCCCC1)=O 87572,N1(C(COc2cccc(C#C)c2)=O)CCC2(CCCN(C(=O)CCC(C)(C)C)C2)C1 87573,N1(C(c2cc(OC)c(O)cc2)=O)CC2(CCOCC2)CC1CNC(C1(C)CC1)=O 87574,C1(N(C)CC2CCN(c3sc(C(=O)OC)c(Cl)n3)CC2)Cc2cccnc2C1 87575,C1(N(C(C(C=CC)O)=O)C)CCCC(NC(C2CC(=O)N(CC)C2)=O)C1 87576,c1(C(=O)N(CC(C)NC(=O)CN2CCOCC2)C)cc2c(F)c(F)ccc2s1 87577,c1(C(N2CC(CNC(c3cnn(C)c3F)=O)OCCC2)=O)cccc2cncn12 87578,C1(CNC(COCC#C)=O)CCCC(C#C)C1.C1=CCNC(=O)C1 87579,c1(OCC(=O)NC(C2CC2CNC(=O)CC2CCC2(C)C)C)ccc(C#N)cc1 87580,C1(CCNC(c2cc(C)n(C)n2)c2n(C(C(=O)OC)C)nnn2)CCN(C)CC1 87581,c1(Nc2c(C(=O)NCC(C)(C)C(N)=O)cc(OC)nc2)ncc2[nH]ncc2n1 87582,c1(C(=O)NCC(C)C)cc2n(n1)CCN(C(c1cc3c(o1)CCCC3)=O)C2 87583,C(=O)(C(F)CCC(C)C)N(C(C(=O)NCC(CC(C)C)OC)C)C(C)C 87584,C1(C(=O)NC(C(C)C)c2cccs2)(CN)CC12CCCC2 87585,c1(C(=O)NCCOCCNC(c2c(C)nncc2)=O)cccc(CO)c1C 87586,c1(OC)cc(S(=O)(=O)N2CC(O)(CNC(c3cc4cccnc4[nH]3)=O)C2)ccc1Br 87587,n1(CC(=O)NCC(=C2CN(C(C3CCC(=O)O3)=O)C2)F)c(=O)oc2ccccc12 87588,c1(C(=O)NC(C2CCCC2)CNC(c2n(CC#C)ccc2)=O)ncccc1SC 87589,C=CC1(C(=O)NCC(c2ccc(F)cc2)NC(C2CC2C)=O)CCOCC1 87590,C12(C)CCN(CC1)C2.C1(C(N(CC=C)C)=O)(CC)CC1 87591,CC1CCCC(C(N2CCOCC2CN(C)C(c2cn(C)nc2C2CC2)=O)=O)C1 87592,c1(C(=O)NC(C(=O)NC(C2CCOC2)C#C)SC)cncnc1 87593,N1(C(C(CCC)N(C)C)=O)CCC2(CC1)CN(C(=O)Cc1ccc(CC)cc1)C2 87594,N1(C(CN(c2ncccn2)C)=O)CCCCC12CC(NC(=O)CCC(C)(C)C)C2 87595,C1(CCNC(c2c(C)cc[nH]2)=O)CC2CCC(C1)N2C(=O)CCCc1cncs1 87596,CCC(CC)C(C)C(=O)NCCCNC(C1(CO)CCCCO1)=O 87597,Cn1cnc2nc(N3CCN(S(C)(=O)=O)CC3)nc(NCc3cc(Cl)ccn3)c12 87598,CN1CCC(NC(=O)COC2CCCCC2)C1c1cccnc1 87599,N1(C(c2nccc(OC)c2)=O)CCCC(O)(CNC(C2CC3(CCC3)CO2)=O)C1 87600,C12(CC(N3CC(N(C(C(C4CC(F)(F)C4)OCC)=O)C)C3)=O)CCC(CC1)CC2 87601,n1(CC(=O)NCC(CC)NC(C2CC2c2nccn2C)=O)cnc([N+](=O)[O-])c1 87602,CC1CC(NC(c2cn(CC3CCCO3)nn2)=O)CCN1C(C1CCCSC1)=O 87603,c1(C(=O)NCC(CNC(c2ccnnc2S)=O)F)cc(Cl)ccc1[N+](=O)[O-] 87604,C(=O)(C(CO)C(F)(F)F)NC1C2C(C(=O)NC(C(=O)NC)CC3CC3)C3C(C2)C13 87605,C1(CC(=O)N(c2nn[nH]n2)CC#C)NC(=O)N(c2ccccc2)C2=C1C(=O)OC2 87606,c1(CNC(C(=O)N(CCCCO)CC)=O)cc(Cl)ccc1OC(C1CCCO1)C 87607,c12ccc(cc1)o2.c1(C(N2CCC(OC)C2)C(=O)NC)c(C)cnn1CC(F)F 87608,c1(C(=O)NCC(=CC(=O)NCC#C)C)cccc(C)c1C 87609,c1(CN(CCOC)C)cn(CCC(=O)N(CCC(C)(C)O)CCO)nn1 87610,Cc1c(N(C)CC2CCCC(C)C2)ncnc1N1CCC(C(N)=O)CC1 87611,C1(C(=O)NC2CCN(C(c3c(C)snn3)=O)C2)CCOC2(CCCCC2)C1 87612,c1(C(=O)NCC2(COC)CN(C(=O)CC(C)(C)C)C2)cc(F)ncc1OC 87613,C1(C)(CC(=O)N(C2CCCC2)CCC)CCN(C(c2cc(Cl)no2)=O)C1 87614,CCCCC(C)CCC(=O)N1CCC12CN(C(=O)C(COC)CC(C)C)C2 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87633,C1(C(=O)NCCCOCCC(=O)NC2CN(C(C)=O)C2)SCC=C1C 87634,C(=O)(CCCC(F)(F)F)NCCCCC(C)NC(c1ccc(N)cn1)=O 87635,C1(NC(c2ccc(CNC(c3ccc(C#C)o3)=O)s2)=O)CCC(C)(C)CC1 87636,c1(CNC(=O)NCc2c(OC)n(C)nc2)cc(F)ccc1C 87637,C1(NC(C(C)(C)SC)=O)CN(C(=O)C2=CS(=O)CCC2)CC2(CC2)C1 87638,CN1CC(CC(=O)NCc2ncoc2C2CN(C(=O)CC3(CO)CC3)C2)C(O)C1 87639,N12CC(C)N(CC1C)C(=O)c1cccc(c1)SCC2=O.n1(COC)nnc(=N)[nH]1 87640,C(=O)(C(C)(C)C(F)F)N1CC2C(NC(c3nn(CC)c(O)c3)=O)(C2)C1.c12ccc(cc1)s2 87641,O=C(CCCCC1CC1)NC1CN(C(C2(c3cc[nH]n3)CC2)=O)C1 87642,C1(CNC(c2n(CC)nnc2)=O)CN(C(c2cc(C(C)=O)cs2)=O)CC12CCC2 87643,N1(C(c2n(CCOC)ncc2)=O)CC2CN(C(c3cnc(C(C)=O)s3)=O)CCC12 87644,c1(OC)c(C(N2C3CCC2CC(NC(c2ccnn2C)=O)C3)=O)ccc(Cl)c1C 87645,C1(C(=O)NC2C(CC(=O)NC(C#C)CCC)C(O)C2)NC(=O)OC1C 87646,C1(N(C)C2CC2)CCN(C(=O)NCCCCCC2CCCC2)CC1 87647,C#CC1(C(=O)NC(c2nc[nH]n2)C)CNC1 87648,Cc1nc2ccc(C(N3CC(NC(C4(C)COC(=O)C4)=O)C3)=O)cc2o1 87649,C12(C(=O)NC3C(CN(C)C(c4ccc(C(N)=O)nc4)=O)CCC3)CCC(CC1)C2 87650,C(=O)(C(C)(C)CCS(C)(=O)=O)NCc1nc(OC)nc(O)c1 87651,N1(C(CCCN=[N+]=[N-])=O)CC2CC(C1)CN(C(=O)CCc1cccnc1Cl)C2 87652,CC1(C)CCCCC(NC(=O)C(O)C2CN(C(=O)CNc3ncccn3)C2)C1 87653,CC1CN(C(=O)C=C2CCCCC2)CC1CC(=O)NC1CC2CCCC12 87654,C1(C(=O)NCC#CC(=O)NCc2cc(OC)no2)CCC(C2CC2)C1 87655,C12(NC(CCc3cc(C)on3)=O)CC1CN(C(c1cnn(C)n1)=O)C2 87656,N1(C(c2csc3cc(Cl)cnc23)=O)CC2CCCC(NC(C3(C4CC4)CC3)=O)C2C1 87657,C1(CC)CCCC1(C)C(=O)OCC1CC1.C12CC(=O)N(C1)C1CN(C1)CC(=O)N2 87658,C1(CP(C)(C)=O)CCCN(CC(O)CNCc2ccccc2)C1 87659,c1(CNC(c2nnc(C)s2)c2nnnn2C2(C)CC2)ccc(F)nc1 87660,Cc1ncc(C(N2CCC(C)C(CNC(c3ccc(O)nc3)=O)C2)=O)c(C)n1 87661,c1(C(=O)NCC(CCNC(C2(C#N)CC(C)C2)=O)(C)C)ccc2sccc2c1 87662,n1(CC(N2CC(NC(C3CCC34CCOCC4)=O)C2)=O)ncc(=O)c2ccccc12 87663,Cc1ncnc(C)c1OCC(N1CCN(C(C2CC2F)=O)C(C(C)C)C1)=O 87664,c1(CC)cnc(C(N2CCC(NC(c3ncccc3C(F)F)=O)C2C)=O)cn1 87665,C=CCC(C(=O)N(C)Cc1nccn1C)NC(C1CCCC1CN=[N+]=[N-])=O 87666,c1(CC(=O)OC)cccc(NC(=O)N(CC(C)C)C)c1.C12C3CN(CC13)C2 87667,c1(C(=O)NCC(CNC(c2c(C)onc2)=O)(C)C)nn2c(c1Br)CCC2 87668,CCCC(CCCNC(c1ccnn1C1CC1)=O)NC(C1CC1c1cccs1)=O 87669,c1(C(C(=O)NCCOCC)N(CCCCCCCO)C)cc(NC(C)=O)nc(Cl)c1 87670,C1(NC(CSCC)=O)CCCC(N(C(=O)CC2CN(C)C2)C)C1 87671,N#Cc1cnn(CC(N2CC3C(CNC(c4cnc(C5CC5)nc4)=O)C3C2)=O)c1N 87672,c1(C(N2CCCC(C)(NC(C3ON=C(C)C3)=O)C2)=O)cccc2c1OCCN2C 87673,Cc1ncnc(C(N2CCSCC2C(=O)N(CCCCC(C)C)C)=O)c1C 87674,Cc1cc(-c2nnnn2C(C)C)ncc1COC(C)(C)C.C12CCC(CC1)N2 87675,N1(C(CN2CCN(C(CC3N(C)CC=CC3)=O)CC2)=O)CC(=O)NCC12CC2 87676,N1(C(c2n(C)cnc2)=O)CC2C(NC(=O)C(c3cccc(Br)c3)(C)O)C2C1 87677,c1(NC(c2cc(Cl)cc(Br)c2)c2n(CCSC)nnn2)ccc2c(c1F)CCC2 87678,C1(NC(C2(C)CC(=C)C2)=O)CCCN(C(c2ccc(C#N)c(O)c2)=O)CC1F 87679,Cc1cc(NCCCNC(=O)CS(=O)(=O)C2CC2)ccc1S(C)(=O)=O 87680,c1(C(C)NCc2cccc(P(C)(C)=O)c2)ccc2c(c1)CC(C)O2 87681,C1(NC(c2ncc(C)nc2)=O)CC2CC1CC2C(=O)N(C1CC1C)C 87682,C(=O)(CC(C)c1cnn(C)c1)NC1CN(C(COCCCCC)=O)C1 87683,C1(C(C)C)N(C(c2cnc3ccsc3c2)=O)CC12CCN(C(C1CC1C)=O)CC2 87684,c1(CC(=O)NCCC(C)CCNC(c2ccc(F)cc2)=O)cccc(Cl)c1Cl 87685,N1(C(C=CSC)=O)CCCC(C)(C)C1CNC(C1C2CCCOC12)=O 87686,CC(C)CCC(C(=O)N1CC(CN(C)C)C1)NC(=O)CC1CCCC(=O)N1 87687,CC(CCCNC(c1cnc[nH]1)=O)NC(=O)CCc1nccn1C 87688,C1(CC)CCN(C(c2cn(CC)nn2)=O)C1C(N1CCC1c1ccccc1)=O 87689,C1(C(=O)NCC=CCNC(C(n2ccc(C)n2)(C)C)=O)CC(C2CC2)=NO1 87690,C1(C(C)C)CC(CO)CN(CC(=O)NC2CCSC2)C1 87691,c1(CN2CC(N(c3ncnc4ncccc34)C)C2)cccc2nccnc12 87692,CC(C)CC(C)(O)C(=O)N(C)CC1CCN(C(c2ccc(CN(C)C)[nH]2)=O)C1 87693,N1(C(CCCCOC)=O)CC(NC(C2(C(=O)N(C)C)CC2)=O)CC(F)(F)C1 87694,Cc1ccc(O)c(C(N2CCC(O)C(NC(C3CC4(C3)CC4F)=O)C2)=O)n1 87695,C1(NC(c2ccc(=NC)[nH]c2)=O)CC2CN(C(=O)C=C3CCC(C)C3)CC2C1 87696,N1(C(CCC)=O)CCC2(C=C(C(=O)N(C)Cc3cn[nH]c3)C2)C1 87697,C1(C(=O)NC2(CCN(C)C)CN(C(C3CN(C(C)C)C3)=O)C2)CC2CCC1O2 87698,C1(C(=O)Nc2nnco2)CN(Cc2ccnc(-c3ccccc3CO)c2)CCN1 87699,CP1(=O)CCN(CC(=O)NCCCc2nn[nH]n2)CC1 87700,c1(C(N2CC=CC(NC(CCCCOC)=O)C2)=O)cnc2n1CCCCC2 87701,CC1(C)CCCN1CCNC(=O)Nn1cc(CCc2ccccn2)nn1 87702,c1(SCNC(C(c2ncc(COC)o2)N(C)Cc2ccco2)=O)ccc(Br)cc1 87703,c1(C(N2C3CC(NC(=O)C(CO)c4ccccc4)(C3)C2)=O)cnc2ccsc2c1 87704,C=C(C)CC(C)C(=O)NC1CN(C(c2cc(CC)c(C)s2)=O)CC1O 87705,c1(C(=O)NCC(N(C)C(C2C=CCC2)=O)C2CC2)ccc(Br)cn1 87706,C(c1ccc(Cl)c(Cl)c1)=CC(=O)NC(CC)CN(C)C(c1c[nH]c(=O)cn1)=O 87707,c1(C(C(=O)NC2CC2)N(CCOC)CC2CCOC2)cc(C(C)(C)C)on1 87708,N1(C(C=C(C)C(C)C)=O)CCCN(C(=O)C=CSCC2CCCO2)C(C)C1 87709,C(=O)(C1=C(C)CCCC1(C)C)NC1C2(CN(C(c3n(CC)ccn3)=O)C2)CCC1 87710,c1(C(N2C(C(N(CC(=O)N(C(C)C)C)C3CC3)=O)CCC2)=O)c[nH]c(=O)cn1 87711,C=C(Cl)CCC(=O)N(CC(C)NC(=O)C(C)(C)c1cscc1Cl)C 87712,Cc1cccc(C(C)(C)C(=O)NCCCC(C)NC(c2nc(C(C)C)cs2)=O)c1 87713,C1(C(N(C)CC2CN(C(C(C)OCC)=O)C2)=O)CN(C(=O)CC)CCO1 87714,Cc1ncccc1CC(=O)NCC1(CCCNC(c2cnsc2)=O)CCCC1 87715,N1(C(=O)C2=NOCC2)CCN(C(=O)CC2CCOCC2)C(CC(F)(F)F)C1 87716,c1(C(N2CC3C(CNC(CC4CC(OC)C4)=O)C3C2)=O)ccc(Cl)nc1C 87717,c1(COC)ccc(C(N2CC(NC(=O)Cc3ccsc3)C(C#N)C2)=O)cc1OC 87718,c1(C(N(CCNC(=O)CCN(CC(C)C(C)C)C)CC)=O)cccc(F)c1OC 87719,Cc1ccc(C(C)C)c(C(N2CCSC(C)(C)C2)=O)c1 87720,N1(C(C=C(C)C(C)(C)C)=O)CCN(C(c2cc3ccsc3[nH]2)=O)CC1C 87721,c1(C(N(C2CCCN(C(=O)Cc3ccccc3)CC2)C)=O)cnc2ccnn2c1 87722,C1(C)(C(=O)NC(CNC(CCCN(C(C)=O)C)=O)C)CCOCC1 87723,c1(C(N2CCC(NC(C3(CC=C)CCCC3)=O)C(C)C2)=O)cc(O)cc(C#N)c1 87724,C=CC(CC)CC(=O)N(C(C)C(=O)NCCc1ccns1)CCOC 87725,N1(C(C(C(C)O)(C)C)=O)CC2CCC1CN2C(=O)Cc1ccccn1 87726,C12CCCCN1C(=O)OCC2.N1(C(C2CC2(F)Cl)=O)CCCC1.O=C1CN1 87727,c1(C(N2CC(C(=O)Nc3ccc(CO)cc3)NCC2)=O)cc(Br)cc(Br)c1O 87728,Cc1nc(O)nc(C)c1CC(N1CCCCC(CNC(=O)C(N)=O)C1)=O 87729,c1(OCC(=O)NCC23CCC(NC(C(C)C)=O)(C2)CO3)ccccc1[N+](=O)[O-] 87730,N1(C(C(CC(=O)C(c2cn(-c3n(C)ccc3)nn2)=O)O)=O)CCOCC(CO)C1 87731,C(C)(C)(C(=O)NC(C)C)NC(CN(C(=O)C=CC(F)(F)F)CC)=O 87732,c1(C(=O)NCC2C(C(=O)NCc3cn(CC)nc3)CCO2)cncc(OC)n1 87733,C(=O)(C1COc2ccccc21)N1CCC(NC(CC2(CSC)CC2)=O)C12CC2 87734,C1(CC)(NC(=O)CC(O)C2CCCC2)CCN(C(c2n[nH]c3c2CCC3)=O)CC1 87735,c1(C(=O)NC(C)CCN(C(=O)C(C)(C)C)C)ccc(P(C)(C)=O)cc1 87736,CCCCN=C(NCc1ccc(F)cc1F)NCC1CCCN1S(=O)(=O)CC 87737,CC(C)C(C(=O)NCC1C(C)(C)C1(F)F)C(C)NC(C1CCC(F)(F)C1)=O 87738,Cc1csn1CC(=O)NCCN(C(=O)CC1CCCC1)C1CC1 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87983,N1(C(C(CCC)F)=O)CC(CNC(c2c(C)coc2C2CC2)=O)CC(C)C1 87984,C(CO)(C(C(F)(F)F)C(F)(F)F)NC(C(C)C)(C)c1nnnn1Cc1ccco1 87985,c1(OCC(N2C(CO)CC(NC(C3N(C)C(=O)OC3)=O)C2)=O)ccc(Cl)cc1F 87986,C(C(C(C)(C)C)NC(=O)C(C)OC1CCOCC1)NC(COCCCC#C)=O 87987,CCC(C)C(=O)NC(C)CCCNC(c1cnoc1-c1ccco1)=O 87988,CCCCCC(C)Cc1nc(-c2c(I)c(C)nn2C)cs1 87989,C(=O)(C(F)C(F)(F)C(F)(F)F)NC1C(NC(C(=O)NCCOC)=O)CC1 87990,N1(C2CN(C(CNC(C)=O)=O)C2)CC(C(C2CC2)N(C)C)CC1=O 87991,C12(CCN(C(=O)CCc3cc(C)no3)C1)CC(=O)N2.CSC=CC=C 87992,c1(C(=O)NCC2CN(C(C3C(C(=O)NCC#C)C3)=O)C2)n[nH]c2c1CCCCC2 87993,C1(C(C)OC(c2c(-c3nc(COC)on3)cccc2)=O)Cc2ccccc2O1 87994,C1(NC(C2C(CNC(C(OCC)OCC)=O)OCC2)=O)=NOC(C)(C)C1 87995,c1(OC)cnncc1C(=O)NC(C)CNC(=O)CCOC1CCOC1 87996,CC(CCC(C)(C)C)C(=O)NCC1CC2COCC2N1C(=O)CSC(C)(C)C 87997,C1(C(N2C3C(NC(C4CSCCS4)=O)C(C3)C2)=O)Cc2ccccc2CO1 87998,CCC(CC)CCCC(=O)NC(Cc1cc[nH]n1)C(N1CCCC(N=[N+]=[N-])C1)=O 87999,C1(NC(c2nn(CC)c(C)c2)=O)CC2CCC(C1)N2C(=O)Cc1ncc(C)s1 88000,C(=O)(C1c2c[nH]nc2CN1C(=O)C#CC1(C)COC1)N(CC(C)O)C1CC1 88001,c1(C(=O)NC2CN(C(CC3CC(OCC)C3)=O)CC2F)c[nH]c2ccc(Cl)cc12 88002,O=C1CCCC(C(N2CCOC(C(N3CCC(C4CCCO4)C3)=O)C2)=O)CC1 88003,CON(C)C(=O)C(C)NC1CCCCC1n1cccc1 88004,N1(C(c2c(C)nc[nH]2)=O)CC2(CCC(C(=O)NC(c3ccc(Cl)cc3Cl)C)O2)C1 88005,c1(C(N2CC(CC)C(NC(C3(C)CCCC3)=O)C2)=O)ccc2n[nH]c(C)c2c1Cl 88006,N1(C(c2nn(CC)c(C)c2)=O)CCOC2(C1)CN(C(c1cc(C)cc(Cl)c1)=O)C2 88007,CC1CCc2[nH]c(C(N3CC(C)CCC3c3cccc(OC(F)F)c3)=O)cc2C1 88008,N1(C(CC)=O)CCOCC2(COCCN2C(=O)C(O)C(C)c2ccccc2F)C1 88009,CC(C)C(C)CCNC12CCCC1C2 88010,c1(C(N(CCC(=O)N(C2CCSC2)C)CC=C)=O)ccnn1C 88011,c1(CN)ccc(C2CN(C(C34CC(CC(F)F)(C3)C4)=O)CCO2)cc1 88012,N1(C(CC(=O)OCC)=O)CC(NC(=O)CCc2nccn2C)CC1(C)COC 88013,CN1CCC(NC(N2CCCC(C)(N3CCCC3)C2)=O)C(C#N)C1 88014,c1(N(C2CCN(C(c3ccccc3Cl)=O)CC2)C)cnc(C#N)cn1 88015,C12(NC(CCCNS(C)(=O)=O)=O)CCC1CN(C(=O)CCc1cccnc1)C2 88016,N1(C(Cc2cc(C)cc(C)c2)=O)CCC(NC(C2CCC2)=O)CC(C)(C)C1 88017,CC(C(C)(C)C)=CC(N1CCC(N(C(=O)CC(O)C2CCCC2)C)C1)=O 88018,CCC(CO)C(=O)NCCC1(O)CN(C(=O)C(C)CC2CCC2)C1 88019,N1(S(CC(=O)OC)(=O)=O)CCC(F)(F)C(NC(=O)Cc2ccc(F)cc2Br)C1 88020,C(CCC(=O)NC1CCOCC1(C)C)(C(C)C)NC(Cn1c(C)nc(C)n1)=O 88021,c1(CC(=O)NCC2CCCC(NC(c3csnn3)=O)C2)nc([N+](=O)[O-])n[nH]1 88022,N1(C(C=C2CCC(C)CC2)=O)CCN(C(=O)CCCN=[N+]=[N-])C(C2CCC2)C1 88023,c1(NCCCC)ccc(C(N2CC(F)(CNC(C3CC3C#N)=O)C2)=O)cc1 88024,C1(NC(CC2N(CC)CCOC2)=O)CCC2CN(C(c3cc(O)ncn3)=O)CC12 88025,n1(CCN(C(=O)CC2CCCCO2)CC)cc(C2CCCOC2)nn1 88026,O=C(CC1=CCCCC1)N1CCC(O)(CNC(=O)C(F)(F)CC2CC2)C1 88027,C1(C(=O)NC(CC=C)CNC(c2cnn(C3CCC3)c2)=O)CCCC12CCC2 88028,C1(CC)(NC)CCN(C(C2CCC(CO)CC2)=O)CC1 88029,CC(O)(CNC(c1conc1CNC(C1(CO)CCC1)=O)=O)C(F)(F)F 88030,c1(CC(=O)NC(c2ccc(C)cc2)CNC(C2C(C=C)C2)=O)cc(F)c(N)cc1F 88031,c1(NC(C2CC(NC(C3(C#N)C(C)C3)=O)C2)=O)ccccc1OCC(F)(F)F 88032,C1(OC)CCCCC1OC(c1cn(-c2ccc(N)cc2)nn1)=O 88033,C1(C(=O)NCc2scc(C)c2)C2CC1N(C(=O)Cc1nc(=N)[nH][nH]1)C2 88034,c1(C(=O)NCC2CC(NC(c3cc(SC)n(C)n3)=O)CC2O)cc2sccc2[nH]1 88035,CN1CCN(c2cc(O)ccn2)CC1.c1(C(=O)N(C2CCOC2)C)ccc(C)cc1 88036,c1(C(=O)NCC2CN(C(C(C=C)O)=O)CC2(F)F)ccc2c(c1)C(CC)C(=O)N2 88037,N1(C(CCOCC#C)=O)CCC2CN(C(C3OCCN(C)C3=O)=O)CC12 88038,C1(CC)CCCN(C(c2cccc(CO)c2)=O)C1C(=O)NCCC(C(C)C)N(C)C 88039,c1(N2C(=O)CC(C(=O)NCC(CN(C(=O)C(C)(C)O)C)O)C2)ccc(F)c(F)c1 88040,C1(C(=O)NCC(CNC(C2CC(N(C)C)C2)=O)O)COCCN1CC1CCCC1 88041,C1(CC#C)(C(=O)NCCOCC2CC2CNC(c2cc(OC)cs2)=O)CCCO1 88042,C(=O)(CS(=O)(=O)C1CC1)NC1C(C2CCN(C(C(C)=C(C)C)=O)CC2)OCCC1 88043,CN1C2CCCC1CN(C(C13C4CC1C1C(C(=O)Nc5cnsc5)C4C31)=O)C2 88044,c1(N(C(c2cnc(C)[nH]2)=O)CC2CC2)ccc(Cl)cc1 88045,C(CCC(C)(C)NC(c1cnc[nH]1)=O)NC(c1cn(CC(CC)O)nn1)=O 88046,CC1(C(=O)Nc2cncc(Br)c2Cl)CCCN(C(=O)CCc2cnccn2)C1 88047,c1(C(=O)NC2CCN(C(CSCCCC)=O)CC2)ccnc2ncccc12 88048,N1(C(Cc2c(C)nccc2)=O)CCC2CCC12CNC(c1c(C)nc(C)n1O)=O 88049,C(=O)(CS(=O)(=O)CCO)NCC1(C(C)(C)C)CCN(C(C(F)OC)=O)C1 88050,C(CCCC(C)NC(c1cnn(CC)n1)=O)NC(C(C)(C)OCC)=O 88051,c1(NC(C)CCc2ccccc2F)nccc(=NCc2nnc(CO)s2)[nH]1 88052,c1(CN(CCCCCC)C)nc(-c2cncnc2)nn1CC(c1ccccc1)(C)O 88053,N1(CC(=O)NCC(C)(C2CC2)NC(CCCCC#C)=O)CCc2ccccc21 88054,C1(CC=C)(NC(=O)C(F)C(F)(F)F)CCN(c2cc(OCCC)ncn2)CC1 88055,N(C(=NC1CCS(=O)(=O)C1)NCC1CC(C)(C)C1)C1CC(OC)C1 88056,C#CCCCCCC(=O)NCC1C2CN(C(=O)CC(C)N(C)C)CC12 88057,S(=O)(=O)(CC(=O)NC1CCCC1NC(c1nccn1CC(F)F)=O)N(C)C 88058,C1(N(C(CSCC=C)=O)CCF)CCCN(C(c2cn(CC)nn2)=O)C1 88059,C(=O)(C1CCCc2c1ncn2C)N1CCN(C(C(=O)NCC)=O)C(C)C1 88060,Cc1nn(CC(=O)NC2C3CN(C(=O)C(C)CC4CC4)CC23)c(C)c1Cl 88061,Cc1cc(C(=O)NC2CCC(N(C(=O)CN(C3CCCC3)C)C)C2)ncc1CO 88062,c1(C(=O)NC)cccnc1NC(C12CC1CN(C(c1ccc(CO)nc1)=O)C2)=O 88063,C12(C(=O)OCc3c(C)cc(C)nc3Cl)CCCCC1NC(=O)C2 88064,Cc1n[nH]c(C)c1CC(=O)N(C)CC1CN(C(C2CCOC2C)=O)CCO1 88065,N1(C(COC(CC)C)=O)CC(NC(c2cn[nH]c2)=O)C(C2CC2)C1 88066,C1(CC)CC(C(=O)N(CC)Cc2cccc(Cl)c2)CCN1C(=O)CCC1CC1(F)F 88067,N(C1CCCc2sc(Br)cc21)C(=O)NCCc1c(F)cc(Br)cc1 88068,C1(OC)(OC)CCC12CC(Cn1cc(-c3cnn(C)c3Br)nn1)C2 88069,C(=O)(C(=O)CCC(C)(C)C)N1C(C)CN(C(c2cc([N+](=O)[O-])n[nH]2)=O)CCC1 88070,N1(C(c2n(C=C)nnc2)=O)CCN(C(c2cc(O)nc(O)n2)=O)CC1COCC 88071,N1(C(CCC(=C)Cl)=O)CCC2(CC1)CN(C(C1Cc3nc(C)cn3C1)=O)C2 88072,c1(C(N2C(C(N(CCCO)CC#C)=O)CC2C)=O)ccc(CC)cn1 88073,C12COCCC1C21N=N1.C1(NC(=O)OC(C)(C)C)CCCC1 88074,Nc1ccc(C(N2CCC(O)(CNC(C3CCS3(=O)=O)=O)C2)=O)c(O)c1 88075,C1(NC(CCNC(C)=O)=O)CC(F)CN(C(C2(C)CC=CCO2)=O)C1 88076,CC(CC(F)(F)F)C(=O)Nc1ncc(C(F)F)s1 88077,c1(N(C2CCN(C(=O)CC3CC3)CC2)C)c(C#N)cnc2ncccc12 88078,c1(NC(C2CC(C)(NC(=O)C(F)CC3CC3)C2)=O)cc(C(F)(F)F)ncn1 88079,C1(OCCCN(C)C(=O)NCC2(C(C)CCO)CCC2)CCC(F)(F)CC1 88080,c1(C(N2CCC2NS(=O)(=O)C)=O)ccc(CNCCC(c2ccccc2)O)s1.CO 88081,N1(C(CC=C)=O)CCCN(C(=O)Cc2n[nH]c(C)n2)CC1 88082,CC1=C(C(=O)N2CCC(CNC(C34CC(F)C3C4)=O)CC2C)C(=O)OC1(C)C 88083,c1(CC(=O)NC(CN(C(c2csc(Br)n2)=O)CC)C)cc(OC)no1 88084,C1(OCC)CN(C(C2(CO)CCOC2)=O)CC1CO.c1(C(=O)NCC)ncccc1CC 88085,CCC(CC(F)F)C(=O)N1CCN(C(c2cscc2C(N)=O)=O)CC1 88086,N12C3CCC(C1CC3)C(N1CC3CC1CN3C)C2=O.CCCC(F)C(=O)OC 88087,CC(Cc1cccs1)N=c1[nH]c2c(c(=NC(C)c3c(F)cccc3Cl)[nH]1)CCC2 88088,n1(C(C(=O)N(CC#C)C(=O)OC(C)(C)C)C)cc(Br)cn1.C1=CC2C(C2)NC1=O 88089,c1(CNC(C2(OC)CCN(C(C3OCCCC3(C)C)=O)C2)=O)ccnc(F)c1F 88090,c1(C(C)C)[nH]nc(C(N2CC(NC(C3(C)C=CCC3)=O)C2)=O)c1[N+](=O)[O-] 88091,N#CC1(C(=O)NCC2CC(C(=O)NCc3nnc(O)o3)C2)CCOCC1 88092,Cc1cc(-c2cn(C3CC(NC(c4c(C)cnn4C)=O)C3)nn2)n(C)n1 88093,Cc1cnc2c(C(=O)N(C3CCN(C(=O)C(C4CCCCC4)C)C3)C)cnn2c1 88094,Cc1c(F)cc(C(N2CCCC(N(C)C(C34CSC(C3)C4)=O)CC2)=O)c(F)c1N 88095,Cc1nc(C(N2CCCC(n3cc(CNC(=O)C(F)C4CC4)nn3)C2)=O)c(C)o1 88096,c1(SCC)ccc(C(=O)NC2CCN(C(=O)CN(C)C(=O)OC)C(C)C2)c(F)c1 88097,c12ccc(cc1)CN2CCC.C1(CNC(=O)NC2CC2)SCCS1 88098,C(C(=O)NCC1NC(=O)CC1(C)C)(C(C)(C)C)NC(C1C(C)=CCS1)=O 88099,Cc1nc(CO)sc1C(=O)NCC(C)NC(c1nc(=N)cc[nH]1)=O 88100,c1(C(N(CCOCCNC(C(C(C)O)C)=O)C)=O)ccc(F)c2ccoc12 88101,Cc1nc[nH]c1CC(=O)NC1(C)CN(C(C2CCC(C)C2)=O)C1 88102,C1(NC(CCC=C)=O)C=CCN(C(=O)C(C)NC(C2CCCCC2)=O)C1 88103,Cc1[nH][nH]c2ncnc(=NCC3(O)CN(C(c4csc5cncn45)=O)C3)c1-2 88104,C1(O)(CN(C(C(C2CC2)SC)=O)C)CCCN(C(c2ccn(C(C)C)n2)=O)C1 88105,C=CCC(C)(C)CC(=O)NCCCCNC(c1c(C)ncnc1O)=O 88106,C1(NC(C(C=C)(C)O)=O)CN(C(c2cc3ccccc3o2)=O)C2(CCC2)C1 88107,Cc1cnc(Cl)c(S(=O)(=O)N2CCCC2(C)C(=O)Nc2ccnc(Cl)c2I)c1 88108,C=C(C)C1CN(C(C23COC(C2)C(NC(=O)CSCC(C)C)C3)=O)CCO1 88109,c1(N2CCCC(C)(CO)C2)cc(Br)ccc1S(=O)(=O)NCCCC#N 88110,Cn1cnc2cc(C(N3CCCC(NC(=O)C4=CCCOC4)C3)=O)ccc12 88111,C1(C(C)C)CN(C(=O)CN2CCNC(=O)C2)CCN1C(=O)Cc1cccnc1 88112,C1(COC)(NC(c2cc(C(N)=O)co2)=O)CCN(C(c2cc(=O)cc[nH]2)=O)CC1 88113,c1(C(F)F)cccc(-c2nc(NC3CC3(F)F)cs2)c1 88114,N1(C(CNC(=O)NC)=O)CCN(C(c2cn(CCOC)nc2C)=O)CC(C)(C)C1 88115,c1(C(N2CC(NC(C(CC)n3cccn3)=O)C2)=O)cc(C(F)(F)F)cc(N)c1 88116,C12(CNC(=O)Nc3c(NC(C)=O)cccc3C)C3CC(CC13)C2(F)F 88117,CC1CN(C(=O)CN(C)C(c2ccccc2)=O)CC1NC(C1(F)CC=CCC1)=O 88118,N1(C(c2c(CCC)occ2)=O)CC(S(C)(=O)=O)CC1(C)C 88119,N1(C(Cc2ccc(SC(C)=O)cc2)=O)CC2CN(C(=O)Cn3ccnc3)C2C1 88120,Cc1cc(F)ccc1C(=O)NCC(C1CCCN1c1ccncc1)(C)C 88121,C(CC(F)F)(C(=O)NC1CCCC1C#N)N(C)C.C1CCC(=O)NCCO1 88122,c1(C(=O)NC2CCCC2NC(C23CCCN2CCC3)=O)ccc2nccn2n1 88123,CC1COCCN(C(=O)CCNC(=O)COC2CCCO2)C1 88124,N1(C(C=NOC)=O)CCC2(CCOC2)C(CNC(=O)CNC(c2cscn2)=O)C1 88125,N1(C(C(CC2CN(C(C(CCOC)OC)=O)C2)F)=O)CCNC(=O)C1C 88126,c1(C(=O)NCC2CC(NC(C(C)c3ccsn3)=O)C2)n[nH]c2ccc(Cl)cc12 88127,c1(C(N(CCCNC(=O)C(F)C2CC2)C2CC2)=O)nnsc1C1CCC1 88128,C(C(=O)NC(c1ccc(C)cn1)C)(C(C)CC)NC(C1(C=C)CCCC1)=O 88129,CC1(C)CCOC1CS(=O)(=O)NC(c1cnc(CN2CCCC2)o1)=O 88130,Cc1cccc2c1CCOC2C(=O)NC1COC2CN(C(=O)C3=CCOC3)CC12 88131,C(=O)(CC(C)(C)C(=O)OC)N1C(CNC(CCC=C)=O)CCC1 88132,C=Cn1ncc(C(N2CCC(C)(C)C2CC(=O)NC2(C)CC(C)C2)=O)c1N 88133,C1(CNC(C(CCC)C)=O)CN(C(=O)C=C(C)c2cccc(Cl)c2)CCC1(F)F 88134,C1(c2cn(-c3ncccc3F)nn2)(CNC(Cc2cn(C)nn2)=O)CCCOC1 88135,C(CC(C)(C)C)(C(=O)N1CCC(C)(C(=O)N(C)CC2(CO)CC2)C1)OC 88136,C#Cc1cccc(C(=O)NCCN(CCCCCC)C(c2cnn(C)c2Cl)=O)c1F 88137,c1(C(N(CC(CN(C(=O)CCC2CCCO2)C)O)C)=O)nccc2cccnc12 88138,CCCCCC(F)C(=O)N1CC(NC(=O)CCCCCn2cnnn2)C(C)(C)C1 88139,C1(N(C(c2cn(CC)nn2)=O)C)CCCN(C(c2cc(C)c(CC)o2)=O)C1 88140,N1(c2ncnc(N3CC(COCC)OCC3)c2C)CC(CCO)OC2(CCC2)C1 88141,c1(C(=O)NCCC2(O)CN(C(C3CC(=O)OC3)=O)C2)cc(C2CCC2)ccn1 88142,C(=O)(CC(C)(C)CC(=O)OC)NCC1OCCCN(C(c2ccc(SC)o2)=O)C1 88143,C1(NC(C(CC)NC(N)=O)=O)CCC2CC1CN2C(=O)C(C)OC(C)(C)C 88144,N1(C(C(CC)(F)F)=O)CCc2ccccc2C(NC(c2ccncc2Cl)=O)C1 88145,C1(C)(NC(CC2C=CC(NC(c3cc(C(C)C)on3)=O)C2)=O)CC(F)(F)C1 88146,c1(C(C)=O)[nH]c2ccccc2c1C(=O)NCC1CC1(Cl)Cl.C12CCCC1NC2=O 88147,Cc1ncnc(C(=O)NCC(CC2CC2)C(=O)NC2(c3nn[nH]n3)CC2)c1C 88148,C12(NC(C(C)O)=O)CCC(CNC(=O)CCCN3C(=O)CN(C)C3=O)(C1)OC2 88149,C(=O)(C(O)CC(C)(C)C)NCC1C(CC)CN(C(=O)Cc2cccc(C)c2)CC1 88150,C1(CC2(O)CCSC2)CCc2cccnc2C1.n12cc(nn1)CNC(=O)CC2 88151,N1(C(=O)OC2CCC(n3ccnc3)C2)CCCc2cc(OC(F)F)ccc21 88152,CC(C(=O)NC1CC(CC(N2CCOCC23CC3)=O)C1)S(N)(=O)=O 88153,C1(C)(c2cn(-c3ncn(C)n3)nn2)COCCN1C(c1nc(I)cs1)=O 88154,C(=O)(C1CCCc2ncnn21)N1CC(N(C)C(c2csc(S)n2)=O)C1 88155,C1CC(C(C)(C)C)NC(=O)C=CC(=O)N1.C(C(C)(C)N(C)C(=O)C1CC1)N(C)C 88156,c1(C(=O)NCC(C)N(C(=O)Cc2ccnc(F)c2)C)cnn2ccn(C)c12 88157,C(=O)(C(C)(C)C(C)C)N(CCCN(C(C)=O)C)C.C1CCC(=O)N1.C(N)=O 88158,c1(CN2C3(CC(F)(F)C3)CC2)ccc2c(c1)CCCO2.C1CN1 88159,c1(OC)ccc2c(c1)CC(C(=O)NCC(C)(C)NC(=O)C1=CCOC1)O2 88160,c1(C(=O)NCCC2CC(C(=O)NC3CC(F)(F)C3)C2)cc(Cl)ccc1Cl 88161,C(=O)(CCC(=O)N1CC(CC(C)NC(=O)CCCc2cccnc2)C1)NCCC 88162,Cc1cc(C(N2CCCC2(C(=O)NC(C(C)O)C2CC2)C(C)C)=O)nc(O)n1 88163,c1(CSCC(=O)NCC(=O)NC(C2(C(C)(C)C)COC2)C)ccccc1 88164,N1(C(CCNC(C)=O)=O)CCC(O)C(NC(=O)CCN(C)CCO)C1 88165,CCCCC(C)(F)C(=O)NCC1CN(C)CCN1C(=O)CCc1ncc(F)cn1 88166,S(=O)(=O)(c1ccc(NC(C2CCCCC2)CO)cc1Cl)NC(c1c(C)ncs1)C 88167,N1(C(C(CC)OC)=O)CCCC(CNC(=O)CCn2ccnc2C)C1 88168,N1(C(CCCOCCC)=O)CC(C(=O)NC(CF)C(F)(F)F)C(C)C1 88169,C1(NC(=O)CCCc2cccs2)CCN(C(=O)Nc2ccc(O)c(O)c2)CC1O 88170,C12(NC(CN(C(C)=O)C)=O)CCCN(C(c3cn(C)c(C(F)F)n3)=O)CC1C2 88171,C1(NC(c2ccc(Cl)s2)=O)C=CCN(C(=O)CCOC2CCCCO2)C1 88172,C1(NC(CNS(CC)(=O)=O)=O)CC12CCN(C(c1cnccc1N(C)C)=O)C2 88173,C1(N)CCC2(CC1)CCN(CCc1c(F)cc(F)cc1F)C2.[N-]=[N+]=NCC1CCC1 88174,C1(NC(CC(C)(C)C2CC2)=O)CCCN(C(c2ccc(Br)c(O)n2)=O)CC1 88175,Cc1cnccc1CN(C(=O)CCSc1nccn1C)C.N12CCC(C1)C2=O 88176,c1(C(=O)NCC2(NC(C(C)C#N)=O)CCCC2)cc2nccc(Cl)c2s1 88177,C1(CC)C(NC(c2cncnc2)=O)CCN1C(=O)CCCc1cnn[nH]1 88178,C(=O)(CCC(F)(F)C(=O)N1CCN(C(C2C=CCCC2)=O)CC1COC)OCC 88179,Cc1cccc2c1OCC2C(=O)N1CC(CCCCNC(=O)CCOC(C)C)C1 88180,c1(CC)cccc(C(N2CCCC(CNC(=O)CSC3CCOC3=O)C2)=O)c1F 88181,C1(C(=O)NCC2N(C(CCCCCOCC)=O)CCC2)Cc2ccncc2N1 88182,C(C(CC(C)C)NC(c1occ(C)c1C(=O)OC)=O)NC(CCN(CCC)C)=O 88183,C1(C(=O)NCC(C(C)(C)C)NC(C2ON=C(CC)C2)=O)Cc2cc(C)ccc2S1 88184,N1(Cc2cncc(C)c2)C(C(N2CCC3(CCCO3)C2)=O)CC2CCCCC12 88185,c1cccc(C#N)c1C.C(CCC(C)C(=O)NC(=O)COC(C)=O)OC 88186,C(=O)(C1CCCc2nccn21)NCC12N(C(c3scc(OC)c3)=O)C(CC1)CC2 88187,C(CC1CC1)(C(=O)NC(C)(CNC(C1CCCSC1)=O)C1CC1)OC 88188,N1(C(CC(CC)O)=O)CCC2CC(NC(C3(OC)CCC3)=O)CCC2C1 88189,Cc1cn2c(n1)CC(C(=O)NCC13CC1CN(C(C1(C(N)=O)CC1)=O)C3)C2 88190,C1(OCC(=O)NC2(CC(=O)OC)CC2)CCN(C(C2(C)CCOC2)=O)C1 88191,c1(C(N2CCC(C)(NC(CN(CCOC)C)=O)C2)=O)[nH]c2ccc(Cl)cc2c1Cl 88192,CCC(C(=O)Nc1cn(C)nn1)NC(=O)CC1CCN1C(=O)C1CC1 88193,c1(C(=O)NCC2C(NC(C3(OCC)CCCC3)=O)CCC2)cc(C#N)ccc1Cl 88194,c1(OC)ccc(S(=O)(=O)N2CC(SC(F)(F)F)C2)c(C)n1 88195,C(CC(CCC)CCC)NC(C1N(C(CCC#C)=O)CC(O)C1)=O 88196,C1(CNC(CC(COC)C)=O)CN(C(=O)COc2cccc(C#N)c2)C2(CCC2)C1 88197,C1(CC)(NC(c2cc(CNC(C3CC(C)(C)C3)=O)on2)=O)CCCC1 88198,c1(C(=O)NC(CNC(CC(C)OC)=O)(C)Cn2cccn2)cccc(N)n1 88199,c1(CC)c(C(N2CCC(C(F)C(=O)N(CCCO)C)C2)=O)cnn1C 88200,C(=O)(C(CC=C)CC(C)C)NC1(CC=C)CCN(C(c2cccnn2)=O)CC1 88201,Nc1ccc(C(N2CCOC(c3ccncc3)C2)=O)c(OCCO)c1 88202,CCC(C)(CNC(C1CC(N(C)C)C1)=O)C(=O)NCC1COCC(C)O1 88203,c1(OC)ccc(NC(=O)CCC2CCN(C(C3CC3F)=O)CC2)cc1C 88204,N1(C(C(COC)C)=O)CCN(C(c2nc(Cl)c(Cl)s2)=O)CC(C)(F)C1 88205,Cc1cc(C(N2CC(CCNC(C3CCCCC3C)=O)OC(C)C2)=O)nc(Cl)c1 88206,C#CC1(O)CC(C(N2CCOC(CC(=O)NC(c3nccc(O)n3)C)C2)=O)C1 88207,Cc1cc(C(=O)NCCC2(O)CCCN(C(C3CSCC(=O)N3)=O)C2)ncc1N 88208,C1(CNC(c2c(Cl)cn(CCC)n2)=O)CN(C(C2C(C#N)C2(C)C)=O)CC12CC2 88209,c1(C(=O)NC(Cc2ccc(CC)cc2)CO)ccc(NC(C)C)c(S(N)(=O)=O)c1 88210,C(=O)(CCCC(C)(C)NC(=O)COC1CCCOC1)NCC1(CCC)CCC1 88211,N1(C(CNC(N)=O)=O)CCN(CCNC(C2(CCn3ccnc3)CC2)=O)CC1.C(=O)NC 88212,N1(C(C2CC(CC(=O)NCC=C(Cl)Cl)C2)=O)CC2(CC2)C1 88213,C1(C(=O)NC(CC)CNC(=O)CCc2ccccc2OC(C)C)CC12CCOC2 88214,c1(OC)cc(F)c(CC(=O)N(CC(C)NC(c2csc3nccn23)=O)C)c(Cl)c1 88215,c1(C(=O)Nc2ccc(-c3ccncc3)cc2)ccn2cccc2c1 88216,N1(C(c2cccc(C3(CC)CCOCC3)c2)=O)C(C)C2CC1(CO)C2 88217,C1(C(=O)NCc2cncc(CC)c2)CC12CCN(C(C1CC1(F)Cl)=O)C2 88218,C1(NC(COCCN(C)C)=O)CN(C(=O)CC2C=CCCC2)CCC1(F)F 88219,Cc1cc(C(=O)NCC23CCC(CC2)N3C(=O)C(c2ccnn2C)C)cc(C)n1 88220,N1(C(CSCCC)=O)CCC2(CC1)CN(CC1COCCO1)C2 88221,C1(CC(=O)NCC2C3CCC(=O)C23)CCN(C(c2cn(C3CC3)nn2)=O)CC1 88222,c1(C(=O)OC(C(=O)OC)C2CCCC2)cc(C(F)(F)F)nc2c1CCCC2 88223,C1(CCOC)(NC(C2CCCN2C(C)C)=O)CCN(C(C2(C(C)C)CCC2)=O)C1 88224,C(=O)(CCC(F)(F)CN=[N+]=[N-])N(CC(C)NC(C1CCc2nn[nH]c2C1)=O)CC 88225,n1(C(CC)(C)C)nnnc1C(C(C)(C)SC)N(C1CCNC1)CC 88226,c1(C(C(=O)Nc2ccccc2)N(C2CCNCC2)CC)cc2cc(F)ccc2o1 88227,C1(C)(OCCOC)CN(C(=O)CCCF)C1.C1=CCNC1=O 88228,C(=O)(CC(C)CC(=O)NC(C)C(F)C(=O)N(C)Cc1cnco1)OC 88229,c1(C(=O)NCC(CCC)NC(c2cncc(Cl)c2Cl)=O)cccn2nncc12 88230,C12CCCC1NC(=O)C2.c1(C(=O)NC2(CC=C)CC2)ccsn1 88231,n1(CC(=O)NCCCOCCCN(C(C)(C)C)C)cccc1C=O.CC(C)(O)COO 88232,N1(C(C(CC)C)=O)CC2(CCN(C(C3CCOCC3)=O)CC2)C1 88233,Cc1cc(C(=O)NC2(CCCCNC(=O)CC3CC3C(F)(F)F)CC2)cc(O)n1 88234,c12ccc(c(C)n1)CN(CC)C2C(=O)NCCC1CC1.C1(CN(C)C)CCOC1 88235,CN1CC2(CCCN(C(=O)CCc3c(Cl)cccc3Br)C2)CC1=O 88236,S(=O)(=O)(C1CCCCC1)N1CCC(C(=O)NCCNC(=O)NC2CC(F)C2)CC1 88237,C(CCC(=O)NCC(O)C(=O)NCC1(SC)CC1)OCC 88238,N1(C(c2ccc(C)cn2)=O)CCN(C(c2csc3nccn23)=O)CC(C)(F)C1 88239,C1(C(N(C2CN(C)CC2O)C)=O)CC(O)CCN1C(c1nccnc1N)=O 88240,C1(C(N(CC(C)N(C)C(c2cc3cccnn3n2)=O)C)=O)CCc2cnnn2C1 88241,c1(C(COC(=O)Cc2nc(C(F)(F)F)n[nH]2)NC)ccc(C(F)(F)F)cc1 88242,N12CC(CC1(C)C)CC2=O.C(=O)(C(F)C(C)(F)F)NCC1CC(C(C)C)C1 88243,Cc1[nH]nc(C(=O)NC(C(=O)N2CC(C(C)(C)C#N)C2)c2cccs2)c1O 88244,C1(NC(C(C(C)C)n2cnnn2)=O)CN(C(c2nscc2Br)=O)CC12CC2 88245,C(=O)(CCCC(C)(C)C)NCC1CCN(C(c2c(N)ccc(C(=O)OC)c2)=O)C1 88246,C(=O)(C1=CCCCC1)N1C(C(N)=O)CC(NC(CC(c2ccc(F)cc2)C)=O)C1 88247,CN1CCOC(C(=O)NCC(C2CCCN2C(=O)Cc2cnoc2)(C)C)C1=O 88248,C1(CNC(c2cccc(SCC)c2)=O)CC2(CO1)CN(C(=O)C(C)CC1CC1)C2 88249,c1(N(CC(C)C#N)C)nc(NCC2COC(=O)O2)c2cnn(C)c2n1 88250,C1(NC(c2c(C)nn[nH]2)=O)CN(C(c2ccc(-c3ccc(Cl)cc3)o2)=O)CC1C 88251,CC(C)C(CCNC(C12CC(CN1C1CC1)C2)=O)NC(C1(C)CCCC1O)=O 88252,Cc1cnc(N)c(C(N2C3CCC2C(NC(=O)CC(=O)NC2CC2)C3)=O)c1 88253,C1(CNC(C2CCC2)=O)CC2(CCN(C(c3cccc[n+]3[O-])=O)CC2)CO1 88254,C(=O)(C1=CCOC1)NC(C)CCCNC(c1cn(C2COC2)nn1)=O 88255,C(CCC1CCC1)(C(=O)NCC(Cc1ccc(Cl)cc1)CO)NC(C)=O 88256,C#CCCCC(C)C(=O)N1CCN(C(=O)Cc2cnoc2)CC1C1CC1 88257,Cn1nc(C(N2CCCC(F)(F)CC2)C(=O)NC2(C)CC2)c2c1CCC2 88258,c1(OC)ccccc1OCCC(=O)NCC1CC(NC(C2COCC(C)O2)=O)C1 88259,c1(C(=O)NC2(C)CCN(C(c3cccc(OCC)c3)=O)C2)nc(C)c(Br)c(Cl)n1 88260,N1(C(C2C(C)C2)=O)CCCC(N(C(=O)CCC2CCCOC2)CCO)C1 88261,c1(NC)ccc([N+](=O)[O-])cc1NC(=O)C(N1CCN(C)C(C)C1C)=O 88262,C1(C(N2CC(CCCCC)C2)=O)CCC(C)N1C(c1ncccc1Cl)=O 88263,n1(CC(=O)O)cccc(NC(=O)NC2CCC=CCC2)c1=O 88264,c1(C(C(=O)NC)NC(N2CCC(O)CC2C(C)C)=O)cccc(F)c1F 88265,CCCC(C)(CCC)C(=O)NCC1(O)CCN(C(=O)CC2CCCC(=O)N2)CC1 88266,C(c1ccsc1Br)=CC(=O)NC1CCC(CNC(C2(Br)CC2)=O)C1 88267,N1(C(Cc2c(C(C)C)con2)=O)CCN(CCNC(C2(C)CC(F)C2)=O)CC1 88268,N1(C(C(C(C)C)n2ccc(C3CC3)n2)=O)CCN(C(=O)C(N)=O)C2(CCC2)C1 88269,C(C(C)(O)CC(=O)NC1CCCN(C(c2cc(C#N)cs2)=O)C1)OC 88270,c1(NC(Cn2c(C)cc(C)n2)=O)ccc(NC(c2cnc(C(N)=O)cn2)=O)c(F)c1 88271,C=Cc1ccc(C(N2CCSCC2C(N2CC3CC3(CC)C2)=O)=O)cc1 88272,N1(C(c2cc(OC)ncc2)=O)CCN(C(=O)CC2CCCN2C(C)C)C(CO)C1 88273,C(=O)(CC(CC)CC)NCC1CN(C(C2(OCC)CCC2)=O)CC1C 88274,N1(C(=O)Cn2cc(C(F)(F)F)nn2)CCN(C(C2CC2(Cl)Cl)=O)CC1 88275,C12(NC(c3c(C)con3)=O)CCC(CN(C(C3(CO)CCOCC3)=O)C1)C2 88276,C12(C(N3CC(NC(CSC(C)C)=O)C(CC4CC4)C3)=O)CCCCCC1OCC2 88277,C(CC(CC)C(=O)NC1CCCN(C(c2ncccc2C(F)F)=O)C1)=CC 88278,C(C(=O)N1CCC(C2CCCN2C(=O)CC2CC2)CC1)(C(C)C)OC 88279,C1(CNC(c2n(CC)ncn2)=O)(OC)CCN(C(c2ccn(C(C)(C)C)n2)=O)C1 88280,N1(C(CP(C)(C)=O)=O)CC2(CCCN(C(=O)Cc3cccc(C(F)F)c3)C2)C1 88281,C1(C(N(CC#CC)CC)=O)C2CC3C(C2NC(=O)CC2CC(CC)C2)C13 88282,C1(F)(C(N2CCC(OCCNC(C3(n4cccn4)CC3)=O)C2)=O)CC=CCC1 88283,c1(N2CCC(NC(c3cncc(C)n3)=O)C2)ncnc2ncc(Br)cc12 88284,N1(Cc2cc(OC)c(C)cc2)CCCC(C2CCCN(C(c3cn[nH]c3)=O)C2)C1 88285,Fc1ccc(CN(C(F)(F)C(F)Cl)CCN2CCCCC2)c(F)c1C(F)(F)F 88286,Cc1ccc(CCN=C(NCc2cccc(C#N)c2)NCC(C)(C)C)c(Cl)c1 88287,CCC(CC)(c1nnnn1CCCC1CC1)NCC(C1CC1)C1CC1 88288,O=C(C1=C(F)CN(C(=O)CC2CCCC2)CC1)N(CC(F)CO)C1CCC1 88289,n1(CCCC)nccc1C(=O)NC(C1CCN(C(=O)C(O)C2CC2)C1)C 88290,N1(C(C(N2C(C(C)C)CCCC2)=O)=O)CCCN2CCCC2C1 88291,c1(CC(C)N(C(C(=O)NCC2CCOCC2)C2CCOC2)CC=C)ccc(C)o1 88292,C1(CNC(c2cnc(SC)[nH]2)=O)CN(C(=O)Cc2nnc(S)n2C)CC12CC2 88293,C(C(C)(C)CC(=O)N1CCCC(NC(=O)CC2CCC(C)(C)C2)CC1)OC(C)=O 88294,CC(C)(O)C(F)(F)C(=O)N1CC2CN(C(=O)CSc3cccc(C#N)c3)CC2C1 88295,N1(C(C2OCCN(S(CC)(=O)=O)C2)=O)CCN(C(=O)CSC2CC2)C(C(C)C)C1 88296,N1(CCC(=O)NC(CNC(=O)CC(F)F)Cc2ccccc2)CCC(O)CC1 88297,CCC(C)C(O)CC(=O)NC(C)(C)CNC(=O)COCCc1ccccc1 88298,CC1CCC(NC(c2cc(C(C)(C)C)ccn2)=O)CN1C(=O)CC1(O)CCCC1 88299,c1(OCCCN(CCCc2cn(C(C(=O)OCC)(C)C)nn2)C)ccc(F)cc1 88300,C1(NC(Cc2nc(C)oc2)=O)CC2CCC(C1C)N2C(C1CN(C(=O)CO)C1)=O 88301,Cc1ccc(CC(=O)NCC2CC3CN(C(C4CCCCC4O)=O)CC23)c(Cl)n1 88302,c1(COC)ccc(CNC(c2n[nH]cc2CNC(=O)CCc2nc(O)n[nH]2)=O)o1 88303,N1(C(c2cn(CC)nc2)=O)CC(C2CC2)(C(=O)NC(c2cccc(C)n2)C)C1 88304,Cc1cc(C)c(C=CC(=O)N(CC(C)NC(c2cnc(Cl)[nH]2)=O)C)cc1C 88305,N1(c2nc(OCC)c(C)cn2)CCC2(CC1)CN(C(=O)CC(C)SC)CC2CO 88306,C1(CCOC)CN(C(=O)C(C)(CO)NC(c2ccnc(C)c2)=O)CCN1C(C)=O 88307,C1(C(N2CC(NC(c3ccc(CCC)[nH]3)=O)C2)=O)C2CCC(F)(F)C12 88308,c1(N(C)C)ccc(C(=O)NC2C=CC(CNC(=O)CCc3ccc[nH]3)C2)nn1 88309,N1(C(C2(N=[N+]=[N-])CC2)=O)CC2CCC1C1CN(C(c3cccc4sccc34)=O)CC21 88310,N1(C(c2cc(COC)[nH]n2)=O)CCCC(C)(C(N2CCCC(OC)C2)=O)C1 88311,c1(C(=O)NCC(C)NC(CCCN(C(C)=O)C)=O)ccc(C#N)c(C)c1 88312,c1(C(N2CCC(NC(COCC(=O)NC)=O)C(O)C2)=O)n[nH]c2c1NCCC2 88313,C12(C(=O)NC(CNC(CNC(C)=O)=O)C3CC3)CC(C1)C(C)(C)O2 88314,CCCCC(CNC(c1scc(C)c1OC)=O)NC(c1cc(Cl)c[nH]1)=O 88315,c1(CN(CCNC(c2c(C)ocn2)=O)C(C2CC(F)CN2C)=O)cc(F)cc(Cl)c1 88316,Cn1ccc(CC(=O)NCCCCNC(C2CCOC2)=O)n1 88317,C(=O)(C(CN=[N+]=[N-])NC(c1cc(Cl)n[nH]1)=O)N(CCCN(C)C)C 88318,O=C1Cc2c(NC(c3csc(NC(c4cc(Cl)ccn4)=O)n3)=O)cccc2N1 88319,CC1(C)CCCCC1CC(=O)NCC(C)(C)OCC1CCC1.C1CC(=O)N1 88320,N1(C(c2cnc(CC)nc2C)=O)CCC(CNC(=O)C(C)C(C)(C)C)C(F)(F)C1 88321,N1(C(c2c3cccc(CC)c3[nH]c2)=O)CCN(C(=O)C(F)F)C(C)CC1C 88322,C1(C(=O)NCC(C)Cn2cccn2)(CO)CCN(C(=O)CCCC2CCC2)C1 88323,Cc1cc(NC(N2CCCC2CCC(=O)NC2(C#N)CCOCC2)=O)c(C)cc1Br 88324,C1(NC(CCCOCC=C)=O)CCN(C(C2(C3CCCCO3)CC2)=O)CC1F 88325,C1(OC)CN(C(c2sccc2C)=O)CC1NC(=O)CCNC(C)=O 88326,C1(C(=O)NC2CCCC(CNC(c3ccc(SC)s3)=O)C2)CCC(C)(F)CC1 88327,N1(C(C(CC)(C)C)=O)CC(C)CN(C(C2CCCCN2N=O)=O)C(C)C1 88328,Cc1cc(CNC(=O)C(CNC(C2(C)CCNC2=O)=O)CC2CCCC2)sc1C 88329,C(N=c1[nH]c(Cl)nc2c1SCC2)C1(CNC(C2COC3COCC23)=O)CCC1 88330,C(N=c1[nH]cc(C#N)c2ccsc12)C1OCC(CNC(=O)C=Cc2cocn2)C1 88331,C1(CC#C)(C(=O)N(C)CCN(C)C)CCN(C(=O)Cn2ccc(C)n2)C1 88332,CC1CCCC(CC(=O)NC(C)CCCNC(=O)Cc2cnccc2Cl)O1 88333,c1(C(=O)NCCC2N(C(COCCC)=O)CCC2)ccc(Cl)c(C)c1Cl 88334,C#CC1CCN(C(=O)CCC2CCN(C(c3cc(C)c[nH]3)=O)CC2)C1 88335,c1(C(N2CCOC(CO)C2)=O)cccc(Br)c1.C12CC(C1)C(=O)N2 88336,N1(N(c2[nH]nnc2C2CC2)C)CCC(C)(C2CCCN2C)C1 88337,C1(CNC(C2(C(C)(F)F)CC2)=O)CC2(CCN(C(=O)CSC3CCCO3)C2)CO1 88338,c1(CC(=O)NCC(CNC(CC2(C=C)CC2)=O)CO)nccc(OC)n1 88339,c1(NC(=O)NC2(C=C)CC(C(=O)O)C2)cccc2c(F)ccnc12 88340,C1(C(NOCC(=O)NCC2C(C)CCC2)=O)CC2CC1CC2O 88341,Cc1cc(C(N2CCOCC2CNC(c2cc(O)ccc2F)=O)=O)c(O)c(Br)c1 88342,C1(C(=O)NC(C2CCCCC2)C)CC2(CCN1C(c1csnn1)=O)CC2 88343,N1(C(c2c(N)ccc(C(C)C)c2)=O)CCC2(CCC2)C(NC(c2cnsc2)=O)C1 88344,C12(NC(CCC(=O)NCC)=O)CCC(CC1NC(=O)CCn1ccnc1C)C2 88345,C=CC(CC)CC(=O)NCC1CC(OC)CN1C(C1CC1c1sccc1C)=O 88346,c1(C(=O)NC2C(OC)CN(C(c3ccc(C#C)o3)=O)C2)cnc2occc2c1 88347,C(=O)(CC(C)CC(=O)NC(C)(C)C(C)NC(c1cnccc1C(F)(F)F)=O)OC 88348,C12(NC(CC3(C)CCC3)=O)CCC(Nc3nccc(C(OC(F)(F)F)=O)c3)(CC1)C2 88349,S(=O)(=O)(CC(=O)N1CCN(C2CN(c3ccccc3)C2)CC1)N(C)C.C1CO1 88350,c1(CCC(=O)NCC(C)N(C(=O)CCNS(=O)(=O)CC)CC)cncn1C 88351,c1(SCCNC(c2cncs2)=O)ccc(C(=O)NCC(CNC(C)=O)F)c(F)c1 88352,C1(C(=O)NCCCC2CCCO2)(CC)CN(C(=O)CCOC2COC2)C1 88353,N1(C(C(CCOC)(C)C)=O)CCC2(CC1)CCN(C(c1cn3ccsc3n1)=O)C2 88354,c1(C(N2CCN(c3cc(C)[nH]c(=O)c3)CCC2=O)=O)cc(=O)c2ccccc2o1 88355,CCCC(C)C(=O)NC(C)CCCNC(c1cnn(CCN(C)C)c1C)=O 88356,CC(C(C)C(=O)NCCc1cnc[nH]1)NC(=O)C=Cc1cccnc1 88357,c1(NCC(=O)N(C(CN(C(CC2ON=C(C)C2)=O)C)C)C)ccc(F)cc1 88358,c1(C(=O)NCC(CNC(CCNC(C(C)(C)C)=O)=O)CO)ccnc(O)c1F 88359,CC(CF)CC(=O)NC(C1CCN(C(c2[nH]nnc2-c2ccccc2)=O)CC1)C 88360,C(C#CCN=c1[nH]c2c(c(=NCC3(c4ccccc4)CCSC3)[nH]1)SCC2)OC 88361,Cc1cc(C#N)cnc1C(N1CCOCC(NC(=O)C2=C(Cl)CC2)C1)=O 88362,C1(F)(C(N(C2CC(C)OCC2)C)=O)CCCN(C(C2COC(=O)NC2)=O)C1 88363,c1(CC(=O)NC(CN(C(C(C)SCCCC)=O)C)C)ccc([N+](=O)[O-])cc1 88364,Cc1cn(C)nc1C(N1CCCC1CCCNC(c1cc[n+]([O-])cc1)=O)=O 88365,C1(NC(CCC)=O)(CC)CCCN(C(=O)C(C)C(O)CC)C1 88366,Cc1nn(CC)c(C)c1C(c1ccccc1)NC(C1CN(C(=O)C(C)O)CC1C)=O 88367,CC1(C)CC(O)CN1C(C1CC(NC(c2ccccn2)=O)C1)=O 88368,C(=O)(C1=CCCN(C(=O)C)C1)NC(CC=C)C(=O)OCCC(C)C 88369,N1(C(c2nc(C)c(C)s2)=O)C2CCCC1CN(C(C1CC1(C)C)=O)C2 88370,Cc1scnc1C(=O)N(CCC(C)NC(C1CSCCS1)=O)C 88371,c1(C(N2CC(C)CC(NC(C(C)SC)=O)C2)=O)c[nH]c2nccc(Cl)c12 88372,c1(C(=O)NC(CC(C)NC(=O)CCCF)C)nccc2nn[nH]c12 88373,N1(C(CCCC=C)=O)CCC2CCN(C(=O)Cc3ccc([N+](=O)[O-])cc3F)CC12 88374,CCC(C(=O)NCc1cc[nH]c1C(=O)NC1(c2ccccn2)CC1)OC 88375,N1(C(c2n(CC)nnc2)C(=O)NC)CCC2(CCN2)CC1 88376,C(N=c1cc[nH]c(=NCCC2CC(F)C2)[nH]1)c1ccc([N+](=O)[O-])cc1 88377,C(C(C)(O)C(=O)NCC1CN(C(=O)C(F)n2cccn2)CC1C)OC 88378,C(N=c1nc(C2CCCC2)[nH]s1)C1CCN(C(C2(COC)CCCCO2)=O)C1 88379,c1(CC)cc(C(=O)N(C)CC2(O)CCN(C(=O)CN3CC4CC4C3)C2)c(C)nn1 88380,c1(C(N2CC(C)(C)C(c3cn(CCO)nn3)C2)=O)csc2ccc(F)cc12 88381,C(=O)(CCCN(C)N=O)N1CCN(C(CNC(C(=O)NC)=O)C)CC1 88382,N1(C(C2(c3c(C)cccc3)CCOCC2)=O)CCCn2nccc21 88383,N1(C(c2n(CC)cc(Br)c2)=O)CC2CCCC(NC(c3cnn(C)c3)=O)C2C1 88384,c1(C(=O)NC2CC2NC(C2CCCO2)=O)nccc2ccccc12 88385,C(=O)(C1=NOC2(CCC2)C1)OC(C)CCNC1CCCC1 88386,C1(C(=O)NCC2(C)CCN(C(CCc3cncc(C)c3)=O)C2)CN2CCC1CC2 88387,c1(C(=O)NCCOC(CNC(c2cnc(CC)[nH]2)=O)(C)C)nnccc1C 88388,N1(C(CN2CC(=O)NC2=O)=O)CCC(C2CCN(C(=O)Cc3ccsc3)CC2)C1 88389,C1(OC)CN(C(C2CC2F)=O)CC1NC(=O)CCN1CCOC1=O 88390,C1(S(=O)(=O)C(N2CC=CC2C(=O)NCc2nc(C(=O)OC)on2)=O)(CC=C)CC1 88391,N1(C(C2(CCC=C)CC2)=O)CCOCC(C(=O)NOCC2(C3CC3)CC2)C1 88392,CC(C)CC(O)C(C)C(=O)NCCNC(c1nnn(C(C)C)n1)=O 88393,C1(NC(c2c(C)cc[nH]2)=O)CCN(C(=O)Cn2ncc(Br)c2C)C(C)C1 88394,CC(C)CCC(O)C(=O)N1CC(CNC(=O)CN2CC=CC2)CCC1C 88395,c1(CC)nc(C)c(C(=O)NCC2(NC(c3cnnn3C)=O)CC2)o1 88396,c1(C(N2CC(CNC(C(CCC)C)=O)C(C)C2)=O)cc(C)cc(Br)c1 88397,C12(C(=O)NCC3(CCNC(C(N4CCCC(O)C4)C)=O)CC3)CCOC(C)(C1)C2 88398,C(C(C)(CC(C)C)NC(c1cnc(N)cn1)=O)NC(CC1(COC)CCCC1)=O 88399,c1(OC)ccc(OCCC(=O)NC(C)CCNC(=O)C(C#N)C2CC2)cc1 88400,C1(N(C)C)CCC(C(=O)NCCC(=O)N(CCCO)C2CCC2)C1 88401,c1(C(N2C3CN(C(CSc4ccc(C)cc4)=O)C(C3)C2)=O)cnc2occc2c1 88402,CCC(O)C(C)C(=O)NC(C)CCN(C(=O)CNC(c1ccccn1)=O)C 88403,CC(C(=O)N1NC2CCC1C2)C(F)(F)c1ccc(Br)cc1 88404,N1(C(C(C(CC)CC)C)=O)CCN(C(c2ccc(C(F)F)o2)=O)CC2(CC2)C1 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88423,NC(=O)CC(C(=O)NCC1C=CCCC1)NC(C1CC(C2CC2)C1)=O 88424,CC1=C(C(=O)NCCC(C)NC(=O)CCC2=CCCCC2)S(=O)(=O)CCO1 88425,C1(CNC(COCCC)=O)CC2CCC1N(C(=O)C(F)CC1CCCC1)C2 88426,CCC(C)C(O)CC(=O)NCC1CCCC1C(=O)NCC12CCC(CC1)CC2 88427,c1(C(=O)NCC(CN(C(=O)CC2CCCCC2O)CC)(C)C)cc(C)cc(C#N)c1 88428,CCCCCCCCC(C)CC(=O)N1CC(NC(=O)CS(=O)(=O)C2CC2)C(O)C1 88429,C1(C(N2CC(NC(CCSC)=O)C(CO)CC2)=O)C(C)(C)CCCC1(C)C 88430,C1(C(=O)NC)CCCC2CN(C(=O)C(N3CCC(c4cc(F)ccc4F)C3)=O)CC12 88431,n1(CCC(=O)NC(CCC)CNC(c2ccnc(CC)c2)=O)cc([N+](=O)[O-])cn1 88432,N1(C(Cc2nc(C)oc2)=O)CCC(NC(c2nc(C)nn2C)=O)C12CCC2 88433,C1(NCCNC(C2CC(C)(F)C2)=O)CCN(Cc2ccno2)CC1 88434,c1(C(=O)NCCN(C(c2c(CC)onc2C(F)(F)F)=O)C)cc(C)cnc1N 88435,C(=O)(C1CCCc2nn[nH]c21)N(C1CCCN(C(C(=O)NCCOC)=O)CC1)C 88436,c1(CC(=O)NC2C(NC(CC(C=C)C)=O)COC2)ccc(Cl)c(Cl)c1 88437,c1(C(N2CC(CNC(C(CC#C)(C)C)=O)C(C)C2)=O)ccc2cc(C)ccc2n1 88438,c1(C(=O)Nc2c(C(=O)Nc3ncncc3Br)scc2)ccc(C(F)(F)F)c(I)c1 88439,N1(C(C(CC)COC)=O)CCC(C)(C)C(NC(c2ccncc2OC)=O)C1 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88457,CCCC(CC)CCC(=O)NCC(C)CC(=O)N(C1CCNC1=O)C 88458,C1(NC(C2C(C(=O)OCC)C2)=O)CCN(C(=O)Cc2cnn(C)c2C)C12CCC2 88459,C(=O)(C1=CCCC1P(C)(C)=O)NC1(C)CN(C(c2ncncc2Cl)=O)C1 88460,N1(C(CC2N(C)CCC2)=O)CCC2(CCC2)C(CNC(=O)C(F)CC(C)(C)C)C1 88461,C(CCS(=O)(=O)c1ccc(F)cc1)NC(=NCCSC)NCc1cnnn1C 88462,N1(C(c2c(C)onc2)=O)CCC(O)(CCNC(=O)CCC2CCCCN2C)CC1 88463,Cc1cc(C(N2CCC(C)N(C(=O)CC3(O)CCC3)CC2)=O)c(C)cc1Br 88464,C(C(F)(C(=O)NCC1(C#N)CC1)C(C)C)NC(c1c(C)scn1)=O 88465,C(=O)(C1=NOC(C)(C)C1)N1CC(OC)C(NC(c2cnc3n2CCC3)=O)C1 88466,CN1CC(O)CC1CNC(=O)CCC1CC1.C1(=O)C(C)(C)CN1 88467,C(CO)(CCCCNC(=O)CN1C(=O)CCC1=O)NC(=O)Cc1cnoc1 88468,c1(C(N2CC(C)(NC(C(C)C(C)N(C)C)=O)C2)=O)cccc2cncn12 88469,c1(OC)cccc(Cl)c1NC(=O)C(=O)NCCNC(C)Cc1ccc(Cl)c(Cl)c1 88470,Cc1c(C(N2CCSCC2C(=O)NC(c2cccnc2)C)=O)oc2ccccc12 88471,c1(C(=O)NC2C(C)CN(C(C3(C(F)F)CCC3)=O)CC2)cccc2c1ncn2C 88472,C(=O)(C1=NN(C)C(=O)CC1)NC(C(C(N1CCCC(C#C)(O)C1)=O)(C)C)C 88473,c1(C(=O)NC(C2CC(NC(C34CC(CO)(C3)OC4C)=O)C2)C)cc2occc2s1 88474,C(CNC(=O)CCCCN(C)C)(C(C)C(C)C)NC(c1cc(C)c(Cl)s1)=O 88475,N1(CCCNC(C(CNC(c2c(CC)con2)=O)C)=O)C(=O)CNC1=O 88476,N1(C(c2c(SC)cnn2C)=O)CC(C(=O)NCC2CC23CCOCC3)CC(C)C1 88477,N1(C(C2CC(O)(CNC(c3cn(C4CC4)nn3)=O)C2)=O)CC2CC3CC2C1C3 88478,Cc1coc(C(N2C(C(N3CC(CC(F)(F)F)C3)=O)CC2C)=O)c1 88479,N1(C(c2ccccc2O)=O)CC2(CCC2C(N2CCCCC2c2ccccc2)=O)C1 88480,CC(CN=c1ncc2ccccc2[nH]1)N(C)C(=O)NC1(O)CCCCC1 88481,c1(C(N2CC(C(=O)OC)C(F)C2)=O)cnc2c(C(=O)O)cnn2c1 88482,c1(C(=O)NCCCN(C(=O)Cc2cc[nH]n2)C(C)C)cccc2c1OCC(=O)N2 88483,C1(CC)CN(C(C2C=CC(NC(=O)CCc3cn[nH]c3)C2)=O)CCN1C 88484,C1(N(C(CC(C)NC(N)=O)=O)C)CCCCN(C(=O)COCP(C)(C)=O)C1 88485,c1(C(N2CC(C)CC(NC(CN(C(C)=O)C)=O)C2)=O)ccc2ccc(Cl)cc2n1 88486,C1(N(C(Cc2c(C)cccn2)=O)C)CN(C(C2CC3CCC2CC3)=O)CCC1C 88487,N1(C(c2cc(OC)ns2)=O)CCCC(N(C(=O)CN2CCC2C)CCF)C1 88488,C1(C)(OC)CC(NC(c2ccc(CNC(=O)C(C)NC=O)nc2)=O)C1(C)C 88489,C(C(CO)C(C)(C)C)NC(C(N(C(c1c(C)nncc1)=O)C)C1CC1)=O 88490,c1(O)ccc(F)c(F)c1.C1(NCC2C(NC(C(C)O)=O)C2(C)C)CCN(C)CC1 88491,C=C=CCCN=c1[nH]c(N2CCC(C)(CN(C)C)C2)nc2c1COCC2 88492,C1(CC(=O)NCCCC2(NC(=O)C=CC(C3CCOCC3)=O)CC2)COCC1O 88493,N1(C(CS(=O)(=O)NCC)=O)CC2CCN(C(=O)C(C(C)(C)C)N(C)C)C2C1 88494,C(=O)(C=CC(=O)N(CC(C)NC(=O)C=CC(N)=O)C)N(C)C 88495,c1(C(=O)NC2CC(NC(C(COC)(C)C)=O)C2)cc(OC(F)F)cc(F)c1 88496,N1(C(CC(C)N(C(c2cncc(C)c2)=O)C)=O)CC(C(C)C)CCC1C 88497,C(CN=c1[nH]c(=NCC2(F)CC2)c2sccc2[nH]1)CN(CC)CC 88498,N(C(=NCC=CC(C)C)NC1CCC2(CC2)C1)C(CC)C 88499,C1(CC(=O)NC2C(C(N)=O)CC=C2)C2CN(C(c3ccns3)=O)CC12 88500,Cn1ncc2c(=O)n(CN3CCC(O)C(F)(F)CC3)cnc12 88501,C(CCCCc1ccccc1)(c1nnnn1C)N(C)C1CC1 88502,c1(N(CCCC)C(=O)NCC#CC)c[nH]c2cccc(C)c12 88503,c1(-c2cn(CC)nn2)cccc(C(N2CCOC(NC(CSCCC)=O)C2)=O)c1 88504,C(c1ccccc1)=CC(=O)NCCOCC(=O)NCCCCN(C)C 88505,C1(N(C(CCCC#N)=O)Cc2ccccc2)CCCC12CN(Cc1cccc(=O)o1)C2 88506,Cc1nc2cc(CO)cc([N+](=O)[O-])c2[nH]1.C12CCN(C(=NCC3CC3)NC1)CC2 88507,c1(SC)ccccc1CC(=O)OC1CC(=O)N(C(C2CCOC2)=O)C1 88508,n1(COC)nccc1C(=O)NC(C)CC(C)NC(=O)CC1CCCC1 88509,Cc1n[nH]cc1C=CC(=O)NCCCN(C(=O)C(CN(C)C)CC1CC1)C 88510,CC1CCc2[nH]nc(C(=O)N(CC(C)NC(c3cc(O)cs3)=O)C)c2C1 88511,C12(NC(C3N(C)CCCC3)=O)CCC(C(=O)NCC3CCC(O)CC3)(CC1)C2 88512,C1(C(N(CCC(=O)NCC#CCCC)C)=O)CC12CCOC2 88513,N1(C(C2(C#N)CCCC2)=O)CCC2CCN(C(C3CC3C(N)=O)=O)CC2C1 88514,c1(C(=O)NC(CC=C)CNC(=O)CC23CCC(CC2)OC3)cn2ccccc2n1 88515,N1(C(C(CSCC)C)=O)C2CCC(C(N3CCC(OCCO)CC3)=O)C1CC2 88516,C1(C(=O)NCCc2nccs2)CCCN1C(=O)C=Cc1ccc[nH]1 88517,N1(C(CCC)=O)CCCC1Cc1cn(CCCNS(=O)(=O)C2CC2)nn1 88518,C1(C#N)(C(=O)NCc2c(C(N(C)Cc3c(C)cco3)=O)[nH]cc2)CC1(C)C 88519,C(=O)(C1=NOC2COCC12)NCC1C(C(N2C(CC)COCC2)=O)C1 88520,C(CN=c1[nH]cc([N+](=O)[O-])cc1C(N)=O)(N(C)C(C1(C2CCC2)CC1)=O)C1CC1 88521,CC1CN(C(C2C3CN(C(c4ccncc4F)=O)CC23)=O)CC(C)O1 88522,N1(C(CC2CC(=C)C2)=O)CCN(C(C2(C)CC3CCC2C3)=O)CC(O)C1 88523,N1(C(C2(OC)CS(=O)(=O)C2)=O)CCCCC(CNC(c2cc[nH]n2)=O)C1 88524,C1(C(=O)NCCN(C2CC2)Cc2ccccc2)CNC2(CCC2)C1 88525,c1(OCC(N2CCC(n3cc(CC=C)nn3)CC2)=O)c(F)cccc1Cl 88526,C1(C(=O)NC(C(C)NC(c2c(C)c[nH]n2)=O)C)C(C)(C)C1(C)C 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88599,c1(C(CN(C(C(C2CC2)SC)=O)C(C)C)CC)ccccc1.C12(CC1)CC(=O)N2 88600,CC(C)(C)CCC(F)C(=O)NC1CCCC(NC(c2ccc(N)c(Cl)n2)=O)C1 88601,C12(C(=O)NC3CN(C(Cc4ccc(C)cc4C)=O)C(C)C3)CCCN(CCC1)C2 88602,c1(C(=O)NCC2(O)CCN(C(COC(C)C)=O)C2)cc2cccnc2s1 88603,CC(O)C(C(=O)NCCC(C)NC(c1ccccc1CO)=O)N(CC(F)(F)F)C1CC1 88604,C1(C(N(CC(COC)(F)F)C)=O)CCN(C(C2CCC2C#N)=O)C(C)(C)C1 88605,C1(CNC(CNC(=O)OC)=O)(OC)CCN(C(C2CC(C)(O)C2)=O)C1.C1(C)CC1 88606,C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CCC(C(C)NC(c2csc(C(F)F)n2)=O)C1 88607,C(C1CCC1)=CC(=O)NCC=CC(=O)N(C(C)CC1CC1)C 88608,CP1(=O)CCN(C(=NCc2ccccc2)NCC(C)OC(F)F)CC1 88609,C1(C(=O)NC(CC)(C)CSc2ccccc2)CC2(CN)CC1C2 88610,c1(NC2CCN(C(=O)NCC=CC(C(C)C)C)CC2)ccc(Cl)c(Cl)c1Cl 88611,c1(C(N2CCC(N(C)C(C3CC(F)C3)=O)C2)=O)ccc2nn(C)cc2c1 88612,C1(NC(Cc2cc(C)ns2)=O)CCCC(N(C)C(c2cccc(C3CC3)c2)=O)C1 88613,CCC(C)C(C)C(=O)NCC1(F)CC(CNC(c2c(Br)c(C)nn2C)=O)C1 88614,C(=O)(C#CC(C)(C)CNC(c1cccnn1)=O)NC(CC)C(C)CN(C)C 88615,N1(C(C2CN(c3c(C)cccc3)C(=O)C2)=O)CCC2(CCOCC2)C1 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88634,C(=O)(C1=COCCO1)N1C(COC)(CNC(c2[nH]cc(C)c2C)=O)CCC1 88635,n1(CCC(=O)NC2C(NC(C(N3CCOCC3)C)=O)CC2)cc(Br)cn1 88636,C(C(C)(C)C(=O)NCC1(C2CCC2)CC1)N(C)C.C12CCCC1NC2=O 88637,CC(C)CC(C)(C)C(=O)NCC1CCCN1C(C12CC(CO1)C2)=O 88638,c1(N2CC(SC)(Nc3c(F)ccc(C(=O)NC(C)CC)c3)C2)nc(C)nc(C)c1F 88639,C(=O)(CCC(C)(C)NC(C1CN(C(C)C)C1)=O)N(C(C(C)C)CO)C 88640,C(C(=O)NOCCc1ccncc1)(c1ccc(Cl)cc1)NC(C(C)(OC)OC)=O 88641,C1(NC(CCSCCCC)=O)CCCC(CN(C)C(C2COC2)=O)C1 88642,C(=O)(C(COC)CC(C)C)N(CCC)CCNC(C1CCCCC1(F)F)=O 88643,C(c1ccc(OC2CC2)cc1)=CC(=O)NCC(C1CC1)NC(C12CCC1CC2)=O 88644,c1(C(N2C(CNC(c3n[nH]c4ncccc34)=O)CCC2)=O)c(F)ccc(O)c1F 88645,C12(CNC(CC3(N(C(c4c(C)cns4)=O)C)CC3)=O)CCCCC1C2 88646,C1(C(N2CCCC(C)(N(C)CC)C2)=O)(NC(Cn2c(C)ccn2)=O)CCC(C)(C)C1 88647,C1(NC(=O)CC2CC2)CCOC12CCN(C(c1csc3c(Cl)cccc13)=O)CC2 88648,c1(C(=O)NCCCCCNC(C(C)C)=O)nc(C(F)(F)F)n2c1CCCC2 88649,C(CCC(=O)NCC1CNC(=O)C1)NC(C1CC(C(C)(C)C)C1)=O 88650,Fc1cc(CC2CCC2)cc(-c2nc(-c3ccoc3)nn2C2CCCOC2)c1 88651,C(=O)(C1CCCn2ncnc21)N1CCN(C(CNC(C2(C)CCOC2)=O)=O)CC1 88652,c1(CNC(C(C2CCCO2)NC(=O)CNc2cnsc2)=O)cccc(F)c1 88653,N1(c2ccnc(=O)[nH]2)CCCN(C(=O)CN2CCCC2=O)CC1 88654,Cc1c(C(=O)N(C)CC2C3CN(C(c4sccc4Cl)=O)CC23)cnn1C 88655,c1(C(=O)NC2C(CNC(c3c(CC(C)C)ncs3)=O)C2)cc(=N)[nH]c(Cl)n1 88656,CN1C2CCC1CC(C(=O)NCC1CCCN(C(C3CCC(C)(F)CC3)=O)C1)C2 88657,C1(C(NOCC(=O)OCC)=O)CCOCC1(C)NC(=O)OCc1ccccc1 88658,N1(C(CN(C(=O)C=CCN2CCCC2)CC)=O)CC2(C1)CC(C)(F)C2 88659,c1(OCC(=O)NCCCCC(C)NC(CC2CC(SC)C2)=O)ccc(C)cc1F 88660,N1(C(CSCC2CC2)=O)CCC(O)C(C)(C)C1.c1(OC)cccc(C(=O)NCC)n1 88661,C(=O)(N=c1[nH]c(Br)cnc1Cl)C1N(Cc2ccc(OCC)c(C)c2C)CC(F)C1 88662,c1(C(N(C)CC2N(C(C3(C)CC=C(C)CC3)=O)CCC2)=O)c(C)nc2sccn12 88663,c1(C(=O)NCCCC(C)NC(C2CC3CC3C2)=O)cc(O)nc(Cl)c1 88664,n1(CCC(=O)N(C2CCC(NC(=O)CC(O)C3CCCC3)CC2)C)ccccc1=O 88665,N12CCOCC1CC2=O.N1(Cc2cnc(CCCC)[nH]2)CC(=O)N(C)C1 88666,N1(C(COCCOC)=O)CCCN(C(=O)CN2CCC(F)(F)C2)C(C)C1 88667,c1(C(N2CCC(O)(C(=O)NC(CCCOC)CO)CC2)=O)cc2cccnc2[nH]1 88668,Cc1cccn(CC(N2CC3CC3(NC(C3CN(C)CCO3)=O)C2)=O)c1=O 88669,C12CCN(CC1)n1cc(cn1)N2.C1(C(=O)OC)CCCN(C(c2nccs2)=O)C1 88670,C1(NC(COCC(=O)NC)=O)COC2(C1)CN(C(=O)C(C(C)C)NC(N)=O)C2 88671,C1(C(=O)NCC=CCNC(=O)CCC2CCCC2)C2CCC(=O)C12 88672,C1(NC(C=CCC)=O)CN(C(c2cc(OCC)no2)=O)C(C)(COC)C1 88673,CC1(C)CN(C(=O)CCOCC2CCCO2)CCC1NC(c1cnc[nH]1)=O 88674,C(=O)(Nn1cnnc1)C1C(NC(C2OCC(C)(C)C2)=O)CCOC1 88675,CC12CCC(C(=O)NCC34CC(NC(=O)CN5CCOCC5)(C3)C4)(CO1)C2 88676,c1(CNC(CN(C(=O)OCC)C)=O)cc2n(n1)CC(NC(=O)CC1CCOC1)CO2 88677,C1(c2ccc(Br)cc2)(OC(C2CCS2)=O)CCCCC1 88678,Cc1cc(C(=O)NC2CC(O)CN(C(c3cc(CO)cc(Cl)c3)=O)C2)ncc1F 88679,Cc1cc(N)c(C(N2CCN(C(c3sc(F)cc3Cl)=O)CC2CCO)=O)cc1C 88680,C(=O)(C1CCCc2ccccc21)NC(C(C)C)CNC(C12CC(C)(C1)C2)=O 88681,C1(NC(C(C(=O)OC)C)=O)CN(C(=O)CCN2CCCS2(=O)=O)CC12CC2 88682,N1(C(c2c(C)cco2)=O)Cc2ccccc2C1C(=O)Nc1cncc(C(N)=O)c1 88683,N1(C=O)CC2CCC1CN2C(=O)C(C(C)(C)C)S.c1(CC)cccnc1C(F)(F)F 88684,c1(-c2nc(NC(CC3(C(=O)OCC)CC3)=O)sc2)cccc(C#N)c1 88685,c1(C(N2CCC3C2CC3)=O)ccc(O)cc1.c1(COC)ccc(-c2nc(C)on2)o1 88686,C1(CC(=O)NCC(=O)NCC(=O)NCC(N)=O)(N(C)C)CC1.C(CO)N 88687,c1(NCC2CCC(C)(CC)O2)nc2c(F)cc(Cl)cc2s1 88688,c1(C(=O)NC2(CC=C)CN(C(=O)Cc3ccoc3C)C2)cccc(C(=O)C2CC2)c1 88689,C(=O)(C(CC)CC(C)C)NCCOCCCNC(COCCC#C)=O.C1CCS1 88690,CN1CC(C(=O)NC(CC2CCC2)C(=O)NCC2(C(C)(F)F)CC2)CCC1=O 88691,c1(C(=O)NC2CCC(CNC(C(C)(C)C)=O)C2)cc2sc(Br)cc2[nH]1 88692,N1(C(COC(CC)C)=O)CC(CCNC(c2ccc(C3CC3)cc2)=O)C(C)C1 88693,C1(C(N2C(CNC(C3N(C)C(=O)CC3)=O)CCC2)=O)CCC(=C(F)F)CC1 88694,C1(CC(=O)NCC2(NC(CNC(C3CC34CCC4)=O)=O)CCOC2)CC2(CC2)C1 88695,c1(C(=O)NCC(CNC(Cn2cc(C(C)=O)nn2)=O)O)csc(C#N)c1 88696,C1(C(=O)NC2CC3(C(NC(CCc4ccn(C)n4)=O)C3)C2)CC2(CCOCC2)C1 88697,Cn1cc(Cl)c(C(=O)N(C2CC3CC2CN3)C2CCC(O)C2O)n1 88698,c1(OC)ccc(CN(C)C(=O)OCCC(=O)OC(C)(C)C)c(F)c1.C12CCC1N2 88699,C1(CNC(C2(CC)CC2(F)F)=O)COCCN(C(=O)C#CC2(C)CC2)C1 88700,C12(CNC(C(C)NC(CC)=O)=O)CCC(C1)N(C(=O)Cn1nc(C)ccc1=O)C2 88701,C(=O)(N=c1cc(Cl)cn[nH]1)C1C(NCc2cc(C)ncc2)C1 88702,N1(C(C2CCCN(CC)C2)=O)CC2(C)CC1(C(=O)N(CC(C)(C)N(C)C)C)C2 88703,c1(OCC)cc(N2CCC(C(C)NC(=O)C=CSC)C2)ncn1 88704,C1(CC(=O)NCC)C2CN(C(=O)CC3(NC(=O)CC4CC5CCC4C5)CC3)CC12 88705,N1(C(c2ccc3nn[nH]c3n2)=O)CC2(C1)CN(C(c1cc(=O)cc[nH]1)=O)CCO2 88706,C1(CNC(C(C)C2CCC2)=O)(CNC(C2(C)COC2)=O)CC1(F)F 88707,c1(C(=O)NC(C2CCN(C(CC(C)C)=O)C2)C)oc(Br)nc1C(F)(F)F 88708,C1(C(N2CCCN(C(Cc3ccc(C)s3)=O)CC2)=O)CCCCN(C)C1=O 88709,CS(=O)C=CC(=O)NCC1CC(NC(=O)Cn2cc(Br)cn2)C1 88710,Cn1cc2c(CN3CCC4CN(c5ncnc6n[nH]cc56)CC4C3)cccc2n1 88711,N1(C(C(C)NC(CC)(C)C)=O)CCC(O)(CNC(C2CCCN2S(C)(=O)=O)=O)C1 88712,c1(NC(CCC(C)ONC(C(C)NC(C)=O)=O)=O)cc2ncccc2[nH]1 88713,C1(C)(COC)CC(NC(c2c[nH]c(=O)cn2)=O)CN1C(=O)C#CC1CC1 88714,C12CC(NC(C)=O)CCN1C2=O.C1(OCC(=O)NC)CC(CF)C1 88715,c1(OC)cncc(C(=O)NC2CC(NC(C3CC(n4ccnn4)C3)=O)C2)c1 88716,C1(CNC(C2C(C)C2)=O)CC2(CO1)CN(C(=O)CNC(=O)C1CC1)C2 88717,N1(C(COCC(C)C)=O)CC2CC(NC(c3cnc(O)c(Cl)c3)=O)CC1C2 88718,c1(C(=O)NCC2(CNC(C(C)(C)CF)=O)CC2)cc(O)nc(C2CCCO2)n1 88719,c1(C(N(CCOC)CCNC(=O)CN2CCSCC2)=O)ccc(F)c(COC)c1 88720,c1(CNC(C(CCCC#C)C)=O)ccc2c(c1)CN(C(C1CCC1C(=O)OC)=O)C2 88721,c1(C(CF)NC(=O)NC2CC(C)(C(=O)OCC)C2)cccc(OCC)c1 88722,CC(CC(=O)NCC1CCN1C(=O)C(C)(C)C(N)=O)C(F)(F)F 88723,n1(CC)c(C(=O)N(C(c2ccccc2)CNC(C2(F)CC2C)=O)C)cnc1O 88724,C#CCC(CC(=O)Nc1cc(OC)cc(Cl)c1)NC(=O)C=C(C)C(C)(C)C 88725,CN1Cc2ccc(CNC(c3coc(N4CCOCC4)n3)=O)cc2C1=O 88726,C(=O)(CCN=C(NCc1cc(C)on1)NC1CCOC(C)(C)C1)NCC 88727,c1(COC)nc(C(N2CC(N(C(=O)C(C)N3CC(C)C3)C)C2)=O)cs1 88728,c1(C(=O)NCCC2N(C(C3CCC(C)CC3)=O)CCCC2)nccc2occc12 88729,C1(CCNC(CC(=O)OCC)=O)CCCN(C(C2CC(C)CCO2)=O)CC1 88730,C1(C(N2CCC(OC)(CNC(=O)CC3(CO)CCC3)C2)=O)CCC(C)(C)OC1 88731,c1(OCC(=O)NCC(CCNC(C2CC(C)(F)C2)=O)O)c(F)cccc1F 88732,N1(C(C(C=CCCC)O)=O)CCCC12CCN(C(C1CC(=O)CCO1)=O)C2 88733,c1(C(=O)NCC2C3CN(C(Cn4c(C)cc(C(F)F)n4)=O)CC32)ccc(F)c(F)c1 88734,S(=O)(=O)(c1ccc(NCC2(C)CCC(=O)N2)c(F)c1)N1CCC(CC=C)C1 88735,C1(NC(C(C2CCC2)NC(C2CC(C)(C)C2)=O)=O)CCCCNC1=O 88736,C#CC1CCC(CNC(=O)C(C2CCN(C(c3cn(C)nc3C)=O)C2)C)CC1 88737,N1(C(C(N2CCOCC2)C)=O)CC(CO)C2(CCN(C(C3COC(=O)N3)=O)CC2)C1 88738,CC1(C)CC(C(=O)NC2CCCCN(c3nnc(CO)s3)C2)=NO1 88739,C1(CC)CN(C(=O)CCc2cc(C)n(C)n2)CCN1C(=O)COc1ccncc1 88740,Cc1csc(C=CC(=O)NCC2(C)CCCN2C(C2C=CCCC2)=O)n1 88741,Cc1n[nH]cc1C(=O)NC1CC(C(C)NC(=O)CCSc2nccn2C)C1 88742,CCCCC(CNC(=O)CCOCc1ccccc1)NC(=O)C(O)CC 88743,c1(CCNC(COCCCC#C)=O)n[nH]cc1C(=O)N(C12CC(C1)C2)C 88744,C1(CNC(C(C(CC)O)C)=O)CCC2CN(C(c3nc(C)sc3C)=O)CC12 88745,C#Cc1cccc(C(=O)NC23CC2CN(C(c2ccc(CC#N)cc2)=O)C3)c1F 88746,N1(C2(CC(N3CC(C(=O)OC)(CNC(C)=O)C3)=O)CC2)CCCC(C(=O)COC)C1 88747,C(CCC(=O)NC(Cc1ccccc1)CCNC(=O)COC1CCOC1)OCC 88748,CC(C)(CCF)C(=O)NC1CC(O)(CNC(C2CC(CC3CC3)C2)=O)C1 88749,c1(C(N2C(CCNC(=O)Cc3cccnc3)COCC2)=O)ccn2ccnc2n1 88750,N1(C(C(c2ccc(C)o2)C)=O)CC(N(C)C(c2nc(C3CC3)oc2C)=O)C(O)C1 88751,O=C(CCn1cc(C2CCCO2)nn1)NNC(=O)c1ccc2cc[nH]c2c1 88752,c1(CC)nc(CNC(C2(NC(C3CC(=O)CS3)=O)CC(O)C2)=O)n[nH]1 88753,C(CO)(C(F)(F)F)NC(C12CC(NCc3ccc(C)o3)(C1)C2)=O 88754,C(CC1=CCN(C(C2CCc3ccnn3C2)=O)CC1)NC(C(C)(O)C1CC1)=O 88755,C(=O)(CCC(=O)NN(C)C)NCC(CC(=O)NCCOCC=CC)C 88756,c1(C(=O)NC)ccc(F)c(C(N2CCN(C(c3cc(Cl)c[nH]3)=O)CC2CF)=O)c1 88757,c1(C(=O)NCCC2(CNC(C3C4CC5C(C4)C35)=O)CC2)ccc2c(n1)CCO2 88758,Cc1c(C(=O)OC(C(F)(F)F)C2CCCOC2)cccc1Cl.C1CO1.CCO 88759,c1(C(=O)NC(CCNC(c2cnn(C)c2)CC)(C)C)cc(C)n(C(C)(C)C)n1 88760,N1(C(CCc2scc(C)c2)=O)CCOC(CCNC(C2(C)CNC(=O)C2)=O)C1 88761,C(=O)(C(CC(N)=O)NC(c1cc2n(n1)CCO2)=O)NCC(C(=O)OC)C 88762,N1(C(CSc2nc(C)[nH]n2)=O)C(CNC(=O)OC(C)(C)C)CC2COCC12 88763,C(=O)(CC(C)C(F)(F)F)NC(CCN(C(CCCCOC)=O)C)C 88764,C1(O)(c2cn(C3CC(NC(C4CCC(C)(CC)O4)=O)C3)nn2)CCOC1(C)C 88765,Cn1c(C(N2CC(CNC(C3CC(C)(C)CO3)=O)C2)=O)cc2sccc12 88766,C(=O)(C(CCNC(C1C2CCCOC12)=O)OC)NCC1(CN(C)C)CCC1 88767,c1(N2CC(CC)(CC)S(=O)CC2)nc(C)cc(=NCC2CCCN2C(C)C)[nH]1 88768,N1(C(c2c(C)nn(C(C)C)c2)=O)CC(NC(=O)CC=C(Cl)Cl)CCC1C 88769,C(c1c[nH]c2ccccc12)=CC(N1C(CCC(N2CCCC(C)CC2)=O)CCC1)=O 88770,C1(NC(CCN(C)CC)=O)CCN(C(=O)C(C(C)C)c2cnc(C)s2)C1(C)C 88771,c1(C(C)C(=O)NC2(CC(=O)NC(C)COC(N)=O)CC2)cnn(C)c1 88772,C(=O)(C(C)(CCF)NC1(c2ccn(-c3c(F)cccc3F)n2)CCC1)OC 88773,C1(NC(Cc2c(CC)cccc2)=O)CC2(C1)CN(C(=O)Cn1cnnc1O)C2 88774,N1(C(c2c(C)ncn2C)=O)CCC2(CCCN2C(c2cncc(Cl)c2)=O)C1 88775,CC1CN(C(=O)COc2ccccc2)CC(C)C1NC(=O)CCCN=[N+]=[N-] 88776,C1(NC(c2c(C)nco2)=O)CC2CCCC(C1)C2.C12(CC(F)(F)C1)C(=O)N2 88777,c1(C(N(CCC)CCNC(c2sccc2Cl)=O)=O)ccc(F)c(C)c1C#N 88778,c1(NC(CCC)C)ncnc(NCCc2ncccc2C)c1C 88779,Cc1ncc(C(=O)NCC2CCCCN(C(c3cnc(C)s3)=O)C2)cc1N 88780,c1(C(=O)NC(CC)CN(C)C(C2CCCO2)=O)c[nH]c2c(Cl)cccc12 88781,N1(C(C2ON=C(C(=O)OC)C2)=O)CCOCC(C)(CNC(c2cnc(Cl)[nH]2)=O)C1 88782,Cc1cc(NC(=O)NC2(C(N)=O)CC2)ccc1[N+](=O)[O-].C12CC1C(=O)N2 88783,C1(CNC(c2c(OCC)oc(C)n2)=O)COC(C)(C)CN1C(c1ccns1)=O 88784,C1(NC(c2cnc(COC)s2)=O)CC2CC1CN2C(c1cn(C)c(C)n1)=O 88785,Cc1csc2ncc(C(=O)N(C)CC3CC(F)CN3C(=O)CC3(C)CC3)n12 88786,C=Cc1cc(C(=O)NCCOCCN(C(=O)CSCCC(C)C)C)cc(F)c1 88787,Cc1cc2c(C(N3CCSCC3CCNC(=O)OC(C)(C)C)=O)cccc2o1 88788,C(=O)(CC(C(F)(F)F)NC(=O)OC(C)(C)C)NCC1(NC(CSC)=O)CC1 88789,Cc1nc(C)n(CCC(=O)NC(C)CC2CN(C(=O)CC(F)(F)F)C2)n1 88790,N1(C(c2c(CC)oc(C)c2)=O)CC2CCCC(C1)N2C(C1CC2(C1)CC(F)C2)=O 88791,n1(CCOC)nnc2c(N3CCCCC3CNC(=O)C(C)CC(N)=O)ncnc12 88792,N1(C(C(COCC)(C)C)=O)CC2(CC)CC1(CNC(C1CCCCC1O)=O)C2 88793,C1(C(=O)NCC2(F)CC(NC(C3(CF)COC3)=O)C2)CCCCCC1 88794,c1(C(=O)NCC(C)(CNC(=O)CCC2CCCOC2)OC)cncnc1C 88795,C1(CC#C)CCN(C(=O)CC2(NC(c3c[nH]c(=N)o3)=O)CC2)C1 88796,N1(C(c2cccnc2O)=O)CCCC2C1CCN2Cc1ccc(F)c(F)c1Cl 88797,C(CC1CC1)(C(=O)NC1CC1)NC(CN(C)C(c1n[nH]c(C2CC2)n1)=O)=O 88798,C1(NCCc2ccc(C(F)(F)F)cc2)CCC2COCCC2C1 88799,CC1(C)CC(C(=O)NCCNC(=O)CCc2ccc(Cl)cc2)C(C)(C)O1 88800,CC(C)C(CNC(=O)CP(C)(C)=O)C(=O)NC(C)(CO)C(C)(C)O 88801,c1(CC)nn(C)c(Cl)c1C(N1CCC(O)(CNC(=O)C(CO)N(C)C)C1)=O 88802,CC12CC(C(=O)NCC(CNC(c3cc(O)cs3)=O)C(F)(F)F)(CCO1)C2 88803,c1(C(=O)NC2C(C)CCN(CCC(=O)Nc3nccs3)C2)ccc(Cl)cc1F 88804,C(C)(C)(CCC(=O)N(C)CC1CN(C(=O)C(c2ccc(Cl)s2)C)CCO1)OC 88805,c1(OC)cc(C(=O)NC2CC2C(=O)NCc2cc(CO)ccc2O)ccc1F 88806,c1(CCNC(C2C=CCN(C(=O)CC34CCC(CC3)C4)C2)=O)cc(O)ncn1 88807,Nc1cc(Cl)cc(Cl)c1C(=O)NCCC(O)CNC(c1cnc(C2CC2)[nH]1)=O 88808,c1(C(N2CCN(C(=O)NCc3cccc(C)c3)CC2)=O)cc(Br)cc2ncoc12 88809,c1(C(=O)Nc2c(OC)occ2)ccc(OC)c(OC)c1.C1(C2CC2)CNC(=O)N1 88810,c1(C(=O)NC2CC(OCC(=O)N(C3CCN(C)C3)C)C2)cnnc(O)c1 88811,C(=O)(CCCCN(C)C(C)C)NCCc1c(C(=O)N)c[nH]n1.C1(OC)CC(C(C)CC)C1 88812,C1(C(=O)OC2CC3C(C2)C3(F)F)C2CC(C(O)C2O)S1(=O)=O 88813,CCC(C)N(OC)C(=O)C1CC=CCN1C(C1CC2(C1)CC2(F)F)=O 88814,c1(C(C)C)nccn1CC(=O)NCC(O)CN(C)C(C1CC1C(C)(C)C)=O 88815,CC(C)C(C)C(CNC(=O)COCC1CC1)NC(c1c(Cl)n[nH]c1C1CC1)=O 88816,C(C(=O)NNC(=O)CC1CCN1)(c1ccoc1)OCC 88817,CC(C)C(C)(CNC(=O)C(C)Oc1ccc(Cl)cc1)NC(=O)C=Cc1cocn1 88818,N1(C(c2c(CC)nc(C)o2)=O)CC(C(=O)NCc2nccc(C)n2)CCC1(C)C 88819,Cc1cccc(CCCNC(c2nc[nH]n2)C)c1 88820,c1(C(=O)NC(C2CCCCN2C(=O)C(C)(C)C2CC2)C)ccc2ocnc2c1 88821,C(=O)(C1=CCc2ccccc21)NCC1C(NC(C(c2ccc(Cl)cc2)C)=O)CC1 88822,C(CNC(c1c(C)coc1C)=O)(C(C)(C)C)NC(CCNC(=O)NC)=O.C1CO1 88823,C1(S(N)(=O)=O)(C(=O)NC(C(C)NC(C2CCCC(=O)N2)=O)CO)CCC1 88824,C(=O)(CC(O)CC(C)(C)C)N1CCC(CN(C(CCCn2ncc(C)c2)=O)C)C1 88825,c1(OC)ccc(O)c(N(C(=O)CCCCCN(C)C)Cc2ccsc2C)c1 88826,C1(CCOC)CN(C(=O)Cn2cncc2C)CCN1C(=O)CN1CCC1C 88827,c1(C(=O)NC(C2CCCN(C(=O)C=CS(C)=O)C2)C)cc(C(F)(F)F)ccc1Cl 88828,C1(NC(=O)Cc2ccccn2)CCC2CN(C(=O)CCCCC(F)(F)F)CC2C1 88829,c1(C(=O)NC2(CC)CN(C(C3(OC)CCOCC3)=O)C2)cnc(S(C)(=O)=O)s1 88830,c1(CC)n[nH]c(CC)c1CC(=O)NCC(C(C)C)NC(=O)Cc1ccc(Cl)nc1 88831,N1(C(CSC(C)C)=O)CC2(C(N3CCOC(CC(N)=O)C3)=O)CCC1CC2 88832,N1(C(c2ccc(C#C)cc2)=O)CCC2CN(C(c3ccc(C)cc3C)=O)CC12 88833,C1(N(C(CC=C=C)=O)CCF)CCCN(C(=O)CN2CSCCSC2)C1 88834,N1(C(c2cn(CC)nn2)=O)CC(NC(C2(OC3CCOCC3)CC2)=O)CC(O)C1 88835,CC1C(NC(C2CCCCC2)=O)CC2CCC1N2C(C1(CO)CCCC1)=O 88836,Cc1cn2cc(CC(=O)NC(C3CC3F)=O)nc2s1.N12CCCC(C1)N2C 88837,N1(C(C(C)NC(N)=O)=O)CC=C(CNC(c2ccnc(C(C)(C)C)c2)=O)CC1 88838,C1(N(C(c2ccc(CC)o2)=O)C)CCCCC1N(C)C(C1CCCC1C(=O)OC)=O 88839,C(CC(C(C)(C)C)C(=O)NC(=O)Cc1cnsc1)N(C(=O)CSc1cccnc1)C 88840,C1(CNC(Cc2cccc(OC)n2)=O)CCC2(CCC2)C1NC(=O)CC=C(C)C 88841,N1(C(c2cc(F)ccc2F)=O)CC2CC(C1)CN(C(C1CC=CCO1)=O)C2 88842,C1(CCNC(CNC(COC)=O)=O)CCCN1C(c1cnoc1)=O 88843,c1(C(C)C)cc(C(=O)NCCOCCNC(C2COC(C)(C)CO2)=O)ccc1F 88844,C1(CC#C)C=CCN1C(C1CCC1CN)=O.C123CC1(C2)C3 88845,c1(C(=O)NC23C(CCN(C(C4(CC)CC4)=O)CC2)C3)cc(O)nc2c1CCCC2 88846,CC(C)=C=CC(=O)N(C(C)C(=O)NCCC(C)O)C 88847,C1(NC(C(C)c2ccsc2)=O)C2CN(C(=O)CCc3ccc(N)cn3)CC12 88848,Cc1cc(F)c(C(=O)NC2CC(C)(NC(c3ccnc4c3CCC4)=O)C2)cc1F 88849,C12CCN(C1)C(C1CC1c1ccco1)C(=O)N2.N1(NC(C)=O)CCOCC1.C(C)C 88850,c1(C(N(C(CCNC(c2nc(C)oc2)=O)C)C)=O)cnc2n1CCC(C)C2 88851,N1(C(CSCCCC)=O)CCC(C2(O)CN(C(C3CCCC3OC)=O)C2)CC1 88852,c1(C(=O)NC(C)CNC(=O)CN(C)C2CC2)ccc(CC2CCC2)c(F)c1 88853,c1(C(N2CCC(NC(C3(OC)CC3)=O)C(C(C)C)C2)=O)ccnc2c1ncn2C 88854,Cc1c(CC(=O)NC2(C)CN(C(=O)CCCC3CCCC3)C2)cccc1Br 88855,c1(C(=O)NCC(CNC(Cc2c(C)ccc(F)c2)=O)F)cccc2c1OCCO2 88856,Cc1c[nH]cc(C(=O)NC(C(C)NC(=O)Cc2cncs2)C(C)C)c1=O 88857,c1(C(N(C2CC3CCC(C2)N3C(c2nncs2)=O)C)=O)cccc2c1ncn2C 88858,N1(C(CC(=O)OC)=O)CCC(CC(N)=O)(NC(=O)Cc2ccsn2)CC1 88859,C(=O)(C1CCc2cccc(F)c21)NCC(C1CC1)NC(c1c(C)noc1C)=O 88860,CCC(CCCC(=O)N(CC(O)(CC)CC)C)NC(=O)CC1CCCC(=O)C1 88861,N1(C(CCc2cnc(C)o2)=O)CCC(C(N2CC(F)(F)C2C2CC2)=O)C(C)(C)C1 88862,N1(C(C2(C(C)C)COC2)=O)CCC2CCC(C1)N2C(=O)CCn1cccn1 88863,N1(C(CCOCCC)=O)CCCC(C2CCN(C(=O)CC(F)F)CC2)C1 88864,N1(C(c2ccc(C3(C)CC3)o2)C(=O)Nc2ccccc2)CCC(C)(CC(O)C(F)(F)F)C1 88865,N(C1CCCc2ccoc21)C(C(C(CCC)NC(=O)C(C(C)C)NC(C)=O)O)=O 88866,Cc1cc(=NC(=O)N2CC(C)CCC2c2ccccc2)[nH]n1-c1ccccc1CO 88867,c1(C(N2CCC(NC(C=CCC)=O)(CO)C2)=O)nc2ncccn2n1 88868,C1(C)(CNC(c2cn(CCOCC)nc2)=O)CCCN1C(=O)CC1CCCN1C 88869,C1(CNC(C=C(CCC)C)=O)C=CC(NC(c2coc(COC)c2)=O)C1 88870,N1(CC2CCC(C)O2)CCc2cnccc21 88871,C1(C(=O)NC(C(C)NC(C=Cc2ccc(CC)o2)=O)CO)CCn2nnnc2C1 88872,N1(C(c2ccccc2Cl)=O)CCCCC2C1CCCN2c1nnc(C2CC2)s1 88873,N1(C(=O)CCc2cnn[nH]2)CCC(NC(=O)COC2(F)CC2)CC1 88874,c1(CN2CCC(N)C2)ccc(OC(F)(F)F)cc1F.CC(CCO)C1CCNC1 88875,N1(C(CCC(CC)OC)=O)CC2CCCC2(NC(c2c[nH]nc2Cl)=O)C1 88876,c1(CNC(CCC2C(C)C2)=O)cc(NC(=O)CC(N2CCCCCC2)C)ccn1 88877,c1(C(=O)NCC2(NC(C(C(CC)C)O)=O)CC3CCC2C3)c[nH]c2nccc-2c1 88878,C(=O)(CCC(C(C)C)NC(=O)CC1CC(=O)C1)Nc1ccc(C#C)nc1 88879,C1(CNC(C=CC=CC)=O)CCN(C(C2COC(Cn3cccn3)C2)=O)C12CC2 88880,C1(CN(C(C)C(=O)NCCCCCNC(c2cn[nH]c2)=O)CC)CCCC1(F)F 88881,N1(C(c2cn(C)nc2C(F)(F)F)=O)CCC(F)C(NC(=O)CSC2CC2)C1 88882,c1(C(C)NC(=O)C(=O)N(C)CC2CCOC2C)cccc(Cl)n1 88883,N1(C(c2c(C(=O)OC)cccc2)=O)CCN(C(=O)CC2CC2C)CC(O)C1 88884,c1(C(=O)NC2CCCC(NC(C3(C)CC(=C)C3)=O)C2)cnn2cc(C)cnc12 88885,O=CN1CCCC1C(N1CC2C(CNC(c3csnc3Cl)=O)C2C1)=O 88886,Cc1c(Cl)sc(Cl)c1C(N1CC2CC(CNC(=O)CCC3CCCC3)C1C2)=O 88887,C1(NC(c2ccnnc2O)=O)CC2CCC1CN2C(=O)Cc1cnccn1 88888,c1(CC)c(N2CCC(O)(CNC(C3CCCCC3C)=O)C2)nc(C2CCC2)nc1Cl 88889,CCCCCCC(C)C(=O)NCC(CNC(=O)CCSCCCC)OC 88890,N1(CC(=O)N(CCNC(CN(C2CCOC2)CCC#C)=O)Cl)CCCCCC1.C(CO)N 88891,CC1CCCn2c(C(N3CCC(n4cnc5ccccc45)C3)=O)cnc21 88892,C1(NC(c2n(C)ccn2)=O)CCCCC1NC(c1ccncc1F)=O 88893,N1(C(C2C(CC)CCC2)=O)CC2CCCC(C1)N2C(c1ccc2cnsc2c1)=O 88894,C12(C(=O)NC3CCCN(C(c4ccc(NC)c(F)c4)=O)C3)CCCCN1CCC2 88895,N1(C(C(=O)NCC=CCSC)=O)CC(O)CC(F)(F)C1 88896,C1(NC(CC2(N(C(c3nccc(C)c3N)=O)C)CC2)=O)C2CCC3C(C2)CC13 88897,c12nc(cc(Cl)n1)N2.C1(NC(=O)CCc2cccnc2)(CO)CCCN(OC)C1 88898,N1(C(C(c2cncc(F)c2)C)=O)CC2CCC(C1)N2C(=O)Cn1cc(Cl)cn1 88899,CC1CCN(C(C2CN(C)CCN(C)C2)=O)CCN1C(=O)CC(C)(C)C1CC1 88900,c1(C(N(C2CCCCN(C(CC3(COC)CC3)=O)C2)C)=O)cc2ccccc2o1 88901,CC1CN(C(=O)NCCc2ccc(F)cc2F)CC(C)S1(=O)=O 88902,C1(NC(C2(C=C)CC2)=O)CN(C(=O)CC2CC=CCN2C)CC2(CCC2)C1 88903,c1(C(N(C)CC2C3CN(C(C(C=C)(F)F)=O)CC32)=O)noc2ccc(F)cc12 88904,N1(C(C#CC2(C)CC2)=O)CCCC1C1CCCN1C(C1CCc2nc[nH]c2C1)=O 88905,C1(C(=O)NCCNc2cc(N)cnc2)CCCN(C(=O)CC2COC(C(=O)O)C2)C1 88906,Cn1cnc2cc(C(=O)NC3CC4(NC(=O)CC5(CO)CC5)COC3C4)ccc12 88907,C1(NC(C(C)C(C)(F)F)=O)COC2(C1)CN(Cc1cnn(CC(F)F)c1)C2 88908,C(C#Cc1cn(CCn2cccn2)nn1)NC(c1ncccc1F)=O 88909,C(=O)(C1=NNC(=O)CC1)N1CCN(C(C=Cc2cc(OC)ns2)=O)C2C1C2 88910,C1(C(N2CC(OCCC(=O)NCC(CCC)N(C)C)C2)=O)CCCCNC1 88911,O=C(CC(C(F)F)NC(C1CCC2(CC2)C1)=O)Nc1cnsc1 88912,c1(C(=O)NC2CC(NC(CC(C=C)C)=O)C2)cnc(O)n(C2CC2)c1=O 88913,C1(NC(C=COCC)=O)CN(C(=O)Cc2ccc(O)cc2)CC1N=[N+]=[N-] 88914,C1(C(=O)NCC2(CNC(C(C(C)C)C)=O)CC2(F)F)CC(F)(F)C1(C)C 88915,c1(C(N(CCCN(C(c2nccc(C)c2O)=O)C)C)=O)cc2cccc(F)c2o1 88916,C#CCC(O)C(=O)N(CCNC(=O)C(=Cc1ccccc1)C)C1CC1 88917,C12(NC(c3c(C)nns3)=O)CCC(CC1)N(C(c1c(C3CC3)noc1C)=O)C2 88918,c1(C(N(C)CC2COCCN2C(C2SCCCS2)=O)=O)cccc2nc[nH]c12 88919,CC(C(=O)NCCCN(C(=O)C(c1ccc(Br)s1)C)C)C(F)(F)F 88920,c1(C(=O)Nc2cc(OC)c(F)cc2)ccc2c(c1)CN(C(=O)CSCC(=O)O)C2 88921,C1(CC(=O)NC2CN(C(C(c3ccccc3)C)=O)C2)SC2=NCCN2C1=O 88922,Cc1c(C(N2CCC(N3CCCC3=O)CC2)=O)cc([N+](=O)[O-])cc1[N+](=O)[O-] 88923,C1(CC)CN(C(c2ccc(C(F)F)nc2)=O)CCC1NC(=O)CC(C)(C)OC 88924,c1(C(N2CC(NC(C(COC)(C)O)=O)C(O)C2)=O)ccc2c(c1)nc(CO)n2C 88925,c1(OCC(=O)NCC2CC2NC(c2ccnn2CC2CCC2)=O)cccnc1 88926,N1(C(CCN(CCC)C(C)=O)=O)CCC(O)(C(C)C)C1 88927,N1(C(=O)Nc2cc(-n3ccnc3C)ccn2)CCC(NC(COC)=O)CC1 88928,C1(CC(=O)NC2(C#C)CC2)CN(C(C2CCC(C)CC2)=O)CCO1 88929,n1(CCOC)cc(C(=O)NOC(C)(C)COC(C)C)c(C(=O)OC(C)(C)C)n1 88930,n1(CC(=O)NC(CC)CN(C)C(c2cnn(C)c2OC)=O)cc(C)ccc1=O 88931,C1(NC(CC(C)OC)=O)(COC)CCN(C(=O)C(c2cccc(Cl)c2)C)C1 88932,C1(C(=O)NC(C2CC(NC(C=C(C)C)=O)C2)C)C2CCCC12 88933,c1(C(=O)NC2(CCNC(C3CCOC3)=O)CCCC2)cnc(-n2cccn2)cn1 88934,C1(CC(N2CCOC(CCNC(=O)CN3CCC3C)C2)=O)(OC)CCCCC1 88935,c1(N(CC(C)NC(=O)CN(C)C(C23CCCCC2C3)=O)C)ccc(Cl)cc1 88936,C(CCC(C(=O)N1CC=CC1CN(C)C)NC(c1ccc(=O)n(C)c1)=O)OC 88937,C1(C(N2CCN(CC3CCCC3)CC2)=O)(CN)CC2(CC(F)C2)C1 88938,c1(C(=O)NC(CC(C)NC(c2nnn(C)c2C(F)(F)F)=O)C)cc2n(c1)CCC2 88939,C1(N(C(C(CC)Oc2cccc(C)c2)=O)CC)CCN(Cc2csc(C)n2)CC1 88940,C1(ONC(C2CC=CC(NC(Cn3ncc(C#C)c3)=O)C2)=O)CCC12CCCC2 88941,C#Cc1cnn(C)c1C(N1CCCC(N(C(=O)Cc2cn(C)nc2Cl)CC)C1)=O 88942,C1(C(=O)NC(C23CCC(CC2)C3)CNC(=O)Cc2ccns2)COCC1C1CC1 88943,c1(N2C(C(C)OC(C)C)CCC2)nc(NCc2nnc(O)n2C)c2ncsc2n1 88944,c1(C(=O)NCCC(CNC(c2ccc(C)cc2Cl)=O)(C)C)ccn2nncc2c1 88945,c1(C(=O)NCC(CC=C)NC(=O)C(C)(CC)CO)ccc(CC)c([N+](=O)[O-])c1 88946,c1(CC(=O)NCC(C)CN(C(=O)CC2(N3CCCC3)CCC2)CCO)cnn(C)c1 88947,c1(CCC(c2c(C)ccnc2)NCCC2CCC3(CC3)C2)ccc(F)cc1 88948,C12(C(=O)OCC)COC(C(=O)NC(C3CN(C(=O)C(C(C)C)SC)C3)C)(C1)C2 88949,c1(-c2c(C)occ2)csc(=Nc2cccc(CC3CC3)c2)n1CC1CCCS1 88950,C(=O)(C(C(C)O)NC(=O)CCCCN(C)C)NCCOCCC=C 88951,c1(C(C)(C)C)cc(C(N2CCCC2C2(NC(=O)CCc3cn[nH]c3)CC2)=O)co1 88952,CC1CCC(C)(C(N2CCC(O)(C(C)NC(=O)CC3(C)OCCO3)C2)=O)C1 88953,Cc1cc([N+](=O)[O-])ccc1CNC(c1nn(CC(F)(F)F)cc1I)=O 88954,C1(OC)CC(N=c2[nH]c(=NCc3ccc(F)cc3)[nH]c3ccc(Cl)cc23)C1 88955,N1(C(CNC(c2ccoc2)=O)=O)CCN(C(c2cc(O)ncn2)=O)C2COCC12 88956,n1(COC)cc(Br)c(C(=O)Nc2ccc(OCc3ccccc3Cl)cc2)n1 88957,c1(C(N2C(CC(=O)NCCOC(C)=O)CC3(CC3)C2)=O)ccc2c(c1)OCCCO2 88958,Cc1cc(C(=O)NCC2CCCC2NC(=O)C=Cc2nnn(C)n2)n(CCO)n1 88959,CC(C(=O)NCC1(NC(C23CCCC2C3(F)F)=O)CCC1)C(C)S(C)(=O)=O 88960,C1(CNC(C2(C(N(C)C)=O)CC2)=O)CN(C(C2COCCC2(F)F)=O)CC1(C)C 88961,C1(C)(C(N2CC(C(C)OC)C2)=O)CCN(C(=O)C=C(C)C(C)C)C1 88962,c1(C(=O)OC)ccc(O)nc1NCC(C)NC(c1c[nH]c(C)cc1=O)=O 88963,N1(CCOC)CC(C(=O)N(CC(C)NC(c2cccn2C2CC2)=O)C)CC1=O 88964,c1(C(=O)Nc2c(-c3cc(=NC)[nH]cc3)cncn2)c(F)ccc(O)c1F 88965,c1(C(=O)N)ccc2occc2c1.N12CC(CC1=O)C(=O)N1CC2C1.CNS(=O)(=O)NCCl 88966,CC1(C)CCCC(C(=O)NCC(C2CC2)NC(=O)Cn2ccc(C(F)F)n2)C1 88967,C12(CNC(C(C)C)=O)CN(C(=O)CC3CC4(CCC4)CO3)CC(F)(C1)C2 88968,c1(-n2cc(CC3CCCN(C(CCC(=C)Cl)=O)C3)nn2)ccc(C)cc1Cl 88969,C1(C(=O)NC(C2CC(NC(=O)C(C)Cc3cccnc3)C2)C)CCC(CO)CC1 88970,C(=O)(C(CCOCC)OC(C)(C)C)NC(c1ccc(SCC)o1)C(=O)OCCC 88971,CC(C)C1CCNC(=O)CC2CC2C(=O)N1.c1(SCCn2cncn2)ccc(F)nc1 88972,N1(C(C(C)OCC#C)=O)CCOC(CCCNC(=O)Cc2ocnc2CC)C1 88973,c1(OC)c(C)ccc(C(N2CC3CC3(CNC(=O)CS(N)(=O)=O)C2)=O)c1F 88974,c1(C(=O)NCC2C(C)CCN(C(CC(CC)(C)C)=O)C2)c(N)cc(Cl)cc1F 88975,c1(OC)cc(C)c(C)cc1C(N1CC2(CCC(NC(c3sccc3I)=O)C2)C1)=O 88976,C1(C(=O)NCCCN(C(C23CCC(OC)C2C3)=O)CC)CC2(C1)CC(C#N)C2 88977,C1(CCNC(=O)CC2CCNC2)CN(C(C2CCCCCC2)=O)CCO1 88978,N1(Cc2cc(C)cc(F)c2)CCCC2(CCCN(C(=O)C(Cl)(Cl)Cl)C2)C1 88979,Cc1cccc(Br)c1C(N)C(N1CCC2(CC1)CC2)=O.N12CCC1C2 88980,N1(C(C2(NC(C)C)CC2)=O)CCCC1C1CCCCN1C(=O)C=CC1CCC1 88981,N1(C(C2C3CN(C(CC(CC)C(F)F)=O)CC32)=O)CCc2ncccc2C1 88982,N1(C(C(c2cncnc2)C)=O)CC(C(=O)NCCn2cnccc2=O)C(C)(C)C1 88983,c1(C(=O)NC2CCCCC2F)c(Cl)ccc2cccnc12 88984,N1(C(CC2CC(C)C2)=O)CCNC(=O)c2c(Br)cccc21 88985,Cc1c[nH]nc1CNC(=O)CC1CCC(NC(=O)C(C2CCOCC2)O)C1 88986,C(=O)(C(C)C(O)C(C)C)NC1CN(C(c2c(C)nc(CCC)o2)=O)CC1CO 88987,CC(CO)C(C)N=c1ccnc(NCc2cccc(Cl)c2Br)[nH]1 88988,N1(C(c2c(C)scn2)=O)CCCC(COC)(NC(=O)COCC2CC2)C1 88989,N1(C(C2=NOC(C)C2)=O)CCCN(C(=O)C(C)Cc2ccncc2)C(C)C1 88990,CC(C)(O)C(C)(C)C(=O)N1CC2(CCN(C(c3sccc3CC#N)=O)C2)C1 88991,N1(C(CC(CCC=C(C)C)C)=O)CCC(O)(C2(NC(=O)CS(N)(=O)=O)CC2)CC1 88992,[N-]=[N+]=NC1CCN(C(C2CN(C(=O)COCC(F)F)CC23CC3)=O)C1 88993,N(C(=NCC1CCC(=O)NC1)N1CCC(C(F)(F)F)CC1)C(COC)C 88994,C1(c2n(CCCSCC)nnn2)(NCCC(N)=O)CCN2CCCC2C1 88995,c1(C(CO)NC(C2N(C(c3cn(CC)nc3)=O)CC=C2)=O)cc(Cl)cc(Cl)c1 88996,C1(NC(c2c(NC)cncc2)=O)CC2COCC1N2C(=O)COCCC(C)C 88997,N1(C(c2c(CC)ocn2)=O)CCC2CN(C(c3ccc(N)cc3O)=O)CCC2C1 88998,C(=O)(C1=CCCOCC1)NC1(CNC(c2cc(N)cc(F)c2)=O)CCCC1 88999,N1(C(Cc2nc(CC)sc2)=O)CC(NC(C2CCC(C)(C)OC2)=O)C2(CC2)C1 89000,N1(C(c2c(N)ccc(C)c2F)=O)CC(NC(=O)Cc2cnoc2)C(S(C)(=O)=O)C1 89001,c1(CC)ncc(C(N2CCCC(N(C(c3snnc3C)=O)CC)C2)=O)c(C)n1 89002,Cc1nc(C(=O)NCCC2CCCN2C(=O)C(C2CCC2)C2CCC2)c(C)o1 89003,c1(SCC)cc(O)nc(SC)n1.CCC(C(C)C)N1CCOCC1 89004,C=CC1OCCC1C(=O)NCC=CCNC(c1cc(-c2ccoc2)[nH]n1)=O 89005,S(=O)(=O)(CCC(=O)NCC(C)(C)CNC(c1cnn(CCC(F)(F)F)c1)=O)NC 89006,N1(C(NC)=O)CCC2OCCCC2(CNC(CCNS(=O)(=O)CBr)=O)C1 89007,c1(C(N2C(C)CCC(NC(C(COC)C)=O)C2)=O)cc2c(OC)[nH]c(=N)nc2s1 89008,c1(C(=O)NCC2CN(C(CC(C)(C)OC)=O)CC2O)cc(=O)c2ccccc2o1 89009,c1(C(N(C2C(C)CCN(C(CCCCOC)=O)C2)C)=O)ccc(=O)n2c1CCC2 89010,N1(C(c2ccc(SC)cc2)=O)CCC2(C)CN(C(=O)CCc3cnc[nH]3)CC12 89011,Cc1ccc(NC(=O)NC2CCN(C(=O)OC(C)(C)C)C2)cc1N=[N+]=[N-] 89012,N1(C(c2c(SCC=C)cccc2)=O)CC2(C1)CN(C(C1CCC3CC3C1)=O)C2 89013,N1(C(CCC=C)=O)CCN(C(=O)Cn2cc(Br)ccc2=O)CC1CC1CC1 89014,C1(C(N2CCC(CC#C)C2)=O)CN(C(=O)C(C)CSC)C(C)(C)C1 89015,CCC(C)(C)CNC(=O)C(C1CCC1)NC(c1cnns1)=O 89016,C=CCC(CNC(=O)C=NOC)NC(C1CC1CSc1ccccc1)=O 89017,c1(C(N2CCC(CNC(=O)CC(O)C3CCCC3)C2)=O)cc([N+](=O)[O-])cnc1O 89018,N1(C(C2C(C)=C2)=O)CC2(C1)CN(C(=O)C(C)Oc1ccc(F)cc1)CC(C)(C)O2 89019,C1(OCC)CN(C)C(C)(C(N2CCC(CN(C)CCc3ccccc3)CC2)=O)C1 89020,C=C(CNC(=O)Cn1ccc(NC(=O)Cc2cc(OC)no2)n1)CCNC(C)C 89021,CCC1=C(C(=O)NCC2CN(C(C3CCCN3C(C)=O)=O)CCN2C)CCCO1 89022,N1(C(C)Cc2cc(F)ccc2F)CCC2(CC1)CCN(c1ncnc(=N)[nH]1)CC2 89023,c1(OC(C)=O)nc(O)n[nH]1.c12nnnn1CCSC2NCC1CC(OC)C1 89024,c1(C(=O)NCC2C(CNC(c3ccc(C#C)nc3)=O)C2)ccc(C)c(C)c1Cl 89025,Cc1cc(C(=O)N(C2CN(C(c3ccccc3F)=O)C2)C)c2ccccc2n1 89026,N1(c2cc(NCCn3ncc(COC)c3)ncn2)CC(C2=NOCC2)C1 89027,n1(CC(N2C(CNC(=O)COCCOCCO)CC2)=O)cc([N+](=O)[O-])cn1 89028,N1(C(C(=O)NCC)=O)CCC2OCCN(C(=O)CCSCc3ccccc3)C2C1 89029,N1(C(C(CO)NC(N)=O)=O)CC2CC1CN2C(c1cc(Cl)ccc1Cl)=O 89030,CCC(O)C(C)C(=O)NCC1CCN(C(=O)CCC2CCCO2)CC1 89031,C(=O)(CCCCC(=O)OC(C)(C)C)NC1CN(C(Cc2nc(C)[nH]n2)=O)C(C)C1 89032,c1(N2C3CN(C(c4c(OC)ccs4)=O)C(CC3)C2)ccc([N+](=O)[O-])c(OC)c1 89033,C#Cc1ccc(C(=O)NCC2(O)CCN(C(C3(C#N)CCC3)=O)C2)cc1 89034,C(CCCCC(=O)N1CC2(C(=O)N(C(C)CO)C)CC1CO2)SC 89035,C#CCCC(C(=O)N1CCC(N=[N+]=[N-])C1)NC(C1CC(=O)C1(C)C)=O 89036,Cc1nc2ccnn2cc1C(=O)NCCC(C)N(C(=O)C(C)NC(N)=O)C 89037,C(C(C)(C)C(=O)N1CC(F)CC1CN(C(=O)C(C)Oc1ccc(Cl)cc1)C)OC 89038,C1(NC(CC)=O)CN(C(c2ccc(CC(C)C)s2)=O)CC1C(F)(F)F 89039,C1(COC)(NC(=O)C=C2CCC2)CCN(C(=O)Cn2nccc2C)C1 89040,N1(C(c2cc(OC)n[nH]2)=O)CC2CC1(C(=O)NC1CC13CC(O)C3)C2 89041,c1(C(N2CCC(O)(CN(C(C(C=C)(C)O)=O)C)C2)=O)ccn(C)c(=O)c1 89042,C1(O)(CNC(c2cccc(-c3ccccc3)c2)=O)CCN(C(C2OCCO2)=O)CC1 89043,N1(C(c2c(CC)ocn2)=O)CCCC(NC(c2c(C)nnn2CC)=O)CC1 89044,CC1(C)C(CNC(C2CCNC2=O)=O)CCN1C(=O)Cc1nc(C2CC2)n[nH]1 89045,c1(CCC(=O)N(C2CCCC(NC(=O)C3CC3)C2)C)ccc2c(c1)NC(=O)CO2 89046,N1(C(C2(CCCC)CC2)=O)CCC2CC(OCCOc3cc(C)on3)CCC2C1 89047,c1(OC)cnc(N2C3CN(C(c4cccc(C(F)(F)F)c4Cl)=O)CC23)nc1C 89048,C1(NC(C2N(C(C)C)CCC2)=O)CCC2CN(C(c3cnnc(O)c3)=O)CC2C1 89049,C(C1c2ccsc2CCN1C(C1CCCOC1)=O)NC(Cc1nc(CC)sc1)=O 89050,Cc1cn(CC(=O)NC2CC23CC(NC(=O)CC(F)(F)F)C3)c2ccccc12 89051,C(C)(CO)(C(F)(F)F)NC(c1cn(CCNC(c2cc(OC)n(C)n2)=O)nc1)=O 89052,C1(C(C)C)CCN(C(c2cc(-c3ccccc3)n[nH]2)=O)C1C(=O)NO 89053,C1(NCCCCC(F)(F)F)CC2(CC(NC(N3CC(CN(C)C)C4C3C4)=O)C2)C1 89054,c1(COC)nccc(=NCC23CC(CNC(c4n[nH]c(C)c4O)=O)(CO2)C3)[nH]1 89055,C1(C(N(c2ccc(C(=O)OC)cc2)C)=O)CC(=O)N(C)C1c1cnn(C)c1 89056,C(=O)(C1=CC2(CCOC2)C1)N(CCCNC(C1(C)C(C)CCCC1)=O)C 89057,N1(C(C(F)=C(C)C)=O)CCOC(CCNC(=O)CCc2nccn2C)C1 89058,C12(C(N(CCC#C)C)=O)C(NC(c3ncncc3C)=O)C3CC1C2C3 89059,N1(C(CC(CC)CN(C)C)=O)CC2CCOC2(CNC(=O)CSC(F)(F)F)C1 89060,Cc1c(C(N2CC(CF)OC(CF)C2)=O)[nH]c2cc(Cl)ccc12 89061,CCS(=O)(=O)c1ccccc1-c1cn(CC2CCN(C(=O)C(C)(CO)CO)C2)nn1 89062,C1(CNC(C(Cc2ncn(C)c2)O)=O)CCC(NC(c2cnc(O)n2C)=O)CC1 89063,N1(C(C(C#C)(C)C)=O)CCC2CCN(C(C3CN(C)C(=O)N3)=O)CC2C1 89064,c1(CNC2CCC(C(=O)NCC(C)O)C2)c(Cl)cc(F)cc1Cl 89065,Cc1cc(C(=O)N(CC(C)NC(C2CCOC(=O)N2)=O)C)c2c(n1)CCCC2=O 89066,N1(C(C(C)NC(C)=O)=O)CCN(C(=O)CCCc2nccs2)C(c2cn[nH]c2)C1 89067,N1(C(c2cccc(NC)n2)=O)CCC2(CCCCC2NC(=O)CC(C)C2CC2)C1 89068,S(=O)(=O)(c1ccc(NCc2cnccn2)c(Br)c1)N1C(C)C(C)(C)CC1 89069,C12(C(=O)NCCCNC(C3CCCO3)=O)CC3CC1C2C3O 89070,c1(CC(C)NC(c2n(CCOCC)nnn2)(C)COCC)ccc(F)cc1 89071,C1(CNC(=O)COc2cccc(Br)c2)CN(C(=O)C2=COCC2)CCC1(C)C 89072,Cc1c(C(=O)NCC(C)(CO)NC(=O)CCn2cnc(=N)[nH]2)nn(C)c1C1CC1 89073,c1(C(N2CCN(C(C3CC4CCCCCC34)=O)CC2)=O)cc(O)ccc1Cl 89074,C(C(C)(C)C(=O)NCCC1CCCN1C(=O)C(C1CCCCC1)F)OC 89075,C(=O)(CC(C)(C)C(F)F)N1CCCC(N(C(C2(OC)CCCCCC2)=O)CC)C1 89076,c1(C(N(CC(CC)NC(=O)C(CC)SC)C)=O)cc(C)c2c(O)n[nH]c2n1 89077,C(CC1=CCCCCC1)N.C1(C(=O)O)(CC)CCN(CCc2ccccc2)C1 89078,c1(C(N2CCC(C)(CNC(=O)C3CC3)CC2)=O)cc2c(s1)-c1ccccc1CC2 89079,N1(C(C(CC=C)(C)O)=O)CC(C(N2CCC(C)(CCO)C2)=O)C2(CCC2)C1 89080,C(=O)(CC1=CCCC1)NC(C1CCN(C(c2cn(C)nc2CN(C)C)=O)CC1)C 89081,CC1(C)CCC=C1C(=O)N1CCCN(C(=O)Cc2ccc(F)c(Cl)c2)CC1 89082,c1(C(=O)NC2CCCC(NC(c3cnc(C)o3)=O)C2)ccc2cccc(F)c2n1 89083,N1(C(C(CCC)C)=O)CCOCC(C(N2CC(C#N)(SC)C2)=O)C1 89084,c1(C=O)ccn(CCO)c(=O)c1.C1(CC#N)CCC(C(=O)NC2C(C)CC2)CC1 89085,c1(C(=O)NCc2cccc(C(N(CCC(=O)OC)C)=O)n2)c(O)cccc1F 89086,N1(C(CC(CNC(=O)C(=CC2CCCC2)C)OC)=O)CC2CC1CC2CF 89087,c1(C(=O)NC(CCNC(c2ccc(CC)[nH]2)=O)C)ccc2c(=O)n(C)cnc2c1 89088,Cn1ncc(C(N2CCC3CC23C(=O)NCC2(n3cccn3)CC2)=O)cc1=O 89089,c1(C(N2CC3C(N(C)C(C4(C)CC4(F)F)=O)C3C2)=O)cc(=O)c2ccccc2[nH]1 89090,C(CCNC(C1(NC(C2C(C)(C)C2(C)C)=O)CC(O)C1)=O)(C(C)C)OC 89091,C(CC(=O)NCc1cscn1)(C(F)(F)F)NC(=O)CC1COCCOC1 89092,C1(C(CNC(C2(CC)COC2)=O)C)CCN(C(c2c(C)nsc2C)=O)CC1 89093,Cc1ccnc(CNC(c2n[nH]cc2CNC(c2cn(C)nn2)=O)=O)c1 89094,c1(N2CC(CCCCNC(C(CC)OC)=O)C2)ccc2cnccc2c1[N+](=O)[O-] 89095,Cc1cn2cc(C(=O)NC3CC(C)(NC(C4CCC=CCCC4)=O)C3)ccc2n1 89096,N1(C(C(C)Cc2cnn(C)c2)=O)CC2(CCCCN2C(c2coc(CO)c2)=O)C1 89097,CC(C)C(CNC(C1CCCCO1)=O)C(=O)Nc1cccc(OS(C)(=O)=O)c1 89098,N1(C(c2c(Cl)cnc(-c3ccc(C)cc3)n2)=O)CCCC2NC(=O)CCCC12 89099,C1(C)(CNC(C=CCCC)=O)CCCN(C(=O)C=Cc2nc(C)cs2)C1 89100,C(=O)(C(CC)C(F)(F)F)NC(CC(=C)C)C(=O)NC1CCC(C(C)C)CC1 89101,c1(CC)c(C(=O)NCCNC(=O)C(C2CCC2)C2CCC2)nnn1C 89102,c1(C(N2CC(C3N(C(=O)CCC4CCCO4)CC3)C2)=O)csc(-c2ncc[nH]2)n1 89103,Cc1ccccc1NC(=O)C(N1CCOC(C(=O)N(C)C)C1)c1ccc(Cl)s1 89104,c1(-c2cccc(C(N3CC(CO)C4CC34)C(=O)NC)c2)ccccc1C(F)(F)F 89105,c1(OC)ccc(C(=O)N(C)NC(CCCn2cc(CC34CCCC3C4)nn2)=O)cc1 89106,Cc1cc(C#N)ccc1C(N1CCC2CC12C(N1CC(CC(N)=O)C1)=O)=O 89107,C1(CC)(NC(c2occc2C(C)C)=O)CCCN(C(c2cncc(N)c2C)=O)C1 89108,c1(C(=O)NC)cccc(S(=O)(=O)N)c1.C(C(N)=O)(C1CC1)NC(C)C1CC1 89109,N1(C(CCOC(C)=O)=O)CCC(F)(CNC(c2ccn(CC(F)F)n2)=O)C1 89110,CC(C)CC(CNC(=O)C=Cc1cncn1C)NC(C1CN(C)CCO1)=O 89111,c1(OC)ccc(C(C)C(=O)NC(C)CCN(C(=O)C2=CCCCC2)C)cc1OC 89112,C=CCC(C(=O)N1CC(O)CC1C(=O)NCC(c1nncn1C)C)NC(C)=O 89113,CC1C(C=CC(N2CC(O)(CNC(c3cc(C(N)=O)c[nH]3)=O)C2)=O)C1(Cl)Cl 89114,C(CC(C)C(=O)NCC(C)NC(c1cccc(NC(C2CCCC2)=O)c1)=O)OC 89115,C1C(C)CCC(CC)N(C(=O)NCC)C(=O)OCCN(CC)C1 89116,CCC(CC)C(F)C(=O)NC(CCCC)CC(=O)NCC#Cc1cnn(C)c1 89117,C1(C(=O)NC(C2CCCN2C(=O)C=Cc2cc[nH]c2)(C)C)CCC(CCO)CC1 89118,CCC(C)(CNC(C1CC1F)=O)NC(c1cc(CF)on1)=O 89119,c1(OC)ccc(CCC(=O)NC2CCCC(NC(=O)C(C)SC3CC3)C2)c(F)c1 89120,c1(C(=O)NCCOC2CCN(C(=O)CC3CC3(Cl)Cl)C2)cccc2c1CCCN2 89121,c1(OC)cc(F)c(-c2ncccc2C(=O)N(C)Cc2cccc(CO)c2)c(F)c1 89122,C1(C(=O)NCCN(C(CC(C)(C)O)=O)C2CCCCC2)C2CCCCCC12 89123,C1(C)(Nc2ccc(CNC(CCC(=O)OC)=O)cc2)CCCS1(=O)=O 89124,C1(CN2C(CNC(c3cncc(Br)c3)=O)CC(F)C2)CCCCCCC1 89125,N1(C(C(COC)C)=O)CCC(C(=O)NCC2CC23CCOC3)CC1C 89126,N1(C(=O)NC(C2CCCO2)C)CC(CO)(NC(C2CC(=O)N2)=O)C1 89127,C=C1Cn2c(C(=O)NCC(C)CNC(C3CCN(C)C3=O)=O)nnc2S1 89128,c1(N(S(=O)(=O)C(F)(F)F)C(c2ccco2)=O)ccc(Br)c2c1CNCC2 89129,c1(CC)occc1C(=O)N(CC(C)O)CCNC(c1cc(COC)on1)=O 89130,c1(C(N(C2CCN(C(c3cc(COC)on3)=O)C2)CC#C)=O)cn2ccsc2n1 89131,CN1CCOCC2(COCCN2c2nnnn2CC2CCC3(CNC3)O2)C1 89132,C1(C(=O)NC(CNC(C(CCC)NC(C)=O)=O)C)COc2ccccc2C1 89133,C1(CNC(C2C(C)OCCC2)=O)CC(F)(F)CN1C(=O)Cc1ccc(O)cc1 89134,c1(CNC(c2cnn(C3CNC3)c2)=O)ccc(N2CCCC(O)C2)cc1 89135,C1(C)(CN(C(c2ccc(CCN(CC=C)C)nc2)=O)CCOC)C(C)(C)C1(C)C 89136,c1(OCCC(=O)NC2CC(c3ccccc3)CO2)ccc(Br)cc1 89137,N1(CC(N2CCC(OCCNC(C=C3CCC(C)C3)=O)C2)=O)CC(=O)NC1=O 89138,C1(C(=O)NC(C2(CNC(=O)C(F)OC(F)(F)F)CC2)C)CCC2(CC1)CC2(F)F 89139,C1(C(=O)NCCCCC(C)NC(CC(C=C)(C)C)=O)CN(CP(C)(C)=O)C1 89140,C(CC(C)CCNC(C1CCN(C(C)=O)CC1)=O)NC(CCCOC)=O 89141,c12c(cccc1C)S2.C=CC(O)C(=O)N1CCCC1Cn1cc(C2CCC2)nn1 89142,C1(C(=O)NC(CC)CCOC)CC(N=[N+]=[N-])CN1C(=O)CCc1cncn1C 89143,C(=O)(C(CCSC)SC)NCCCCCN(C(CC)=O)C 89144,CCC(CC)CC(F)C(=O)NC(CNC(C1CCC1)=O)CCOC 89145,CN1CCCC1C=CC(N1CCOC(CCNC(=O)CSc2n[nH]c(=N)s2)C1)=O 89146,C1(C(=O)NCC(CCNC(CN(S(N(C)C)(=O)=O)C)=O)O)CN2CC3CC2(CO1)C3 89147,c1(C2(NC3CC(=O)NCCn4c3nnn4)CCC2)ccc(Br)cc1.CCCOCC 89148,N1(C(c2c(C(=O)OC)scc2)=O)CC2CN(C(=O)CSCC(N)=O)CC2(C)C1 89149,c1(C(=O)NCC2N(C(CCOCC#C)=O)CC(C)CC2)cccc2nonc12 89150,N1(CCCC)CCN(C(=O)CC2CCCCN2C(=O)Cn2cccn2)CC1 89151,C1(NC(C2(C(=O)Nc3cccc(C)c3)CC2)=O)COCCN(C(N)=O)C1 89152,C12CC3CCC(C1)N3ONC2=O.c1ccc(F)nc1.c1(C=O)ccncc1 89153,c1(C(C(=O)NCCCCCC)N(C)CC2CCOC2)cc(C)nc(C)n1 89154,Cn1cc(C(=O)NCC2CC2NC(=O)CC2(C)CC2)c(C2CCCO2)n1 89155,Cc1c(CNC(=NCCC2CN3CCN2CC3)NCC(C)(C)C)c(Cl)nn1C 89156,c1(N2C(C)C(NC(c3ccc(CO)cn3)=O)CCC2)ncc(C#N)cc1Cl 89157,C(C)(CC(=O)NC1C2CC1N(C(c1ccc(CO)s1)=O)C2)(C(F)F)N(C)C 89158,c1(CC)ccc2cc(C(=O)NCC(C)CNC(=O)C=CCOC(C)(C)C)[nH]c2c1 89159,CC1(C)CN(C(c2cnco2)=O)C1C1CCN(C(C2CCCSC2)=O)CC1 89160,C1(NC(c2cn(CC3CCOC3)nn2)=O)CC12CCN(C(c1cnns1)=O)CC2 89161,c1(CC2(C(=O)NCCNC(C3CCC4CC34)=O)CC2)ccccc1SC(F)(F)F 89162,C#Cc1ccc(CC(=O)N(CC(C)O)CCNC(=O)C(=Cc2cccnc2)C)cc1 89163,C1(CC(=O)NCC(C(C)C)NC(=O)CC2CCCCC2)CCCCN1C 89164,CCCC(C)CCCC(=O)NCCC1(CNC(C2(c3cc[nH]n3)CC2)=O)CC1 89165,C1(CNC(CSCC)=O)Cc2ccccc2CN1C(c1cc(C2CC2)ns1)=O 89166,c1(C(N2CC(CC=C)(NC(=O)Cc3ccsn3)C2)=O)c(C)cccc1[N+](=O)[O-] 89167,N1(C(COCC(C)C)=O)CC(NC(=O)CCCn2ccccc2=O)CC2(CC2)C1 89168,N1(C(C(C(C)C)OCC)=O)CCc2ccc(C(=O)NCCC(O)C(C)C)nc2C1 89169,c1(C(N2CC(O)CC(NC(C=CCC)=O)C2)=O)ccc2ncnn2c1 89170,N1(C(C(CO)NC(CC=C)=O)=O)CC(F)(F)C(F)(F)C1 89171,Nc1cc(Cl)ccc1C(N1CC2CC(NC(c3ccc(F)s3)=O)C2C1)=O 89172,C1(NC(=O)C2=CCCCC2)CCCC12CN(C(c1ccn(CC(F)(F)F)n1)=O)C2 89173,C(=O)(C#CC(C)(C)CN(C)C)N1CCOCC(n2cc(CCCC=C)nn2)C1 89174,c1(C(=O)NCC2N(C(Cn3ncc(C)c3)=O)CCN(C)C2)cccc2c1CCC2 89175,c1(C(=O)NC2CC(NC(c3c(C)c(F)ccc3)=O)C2)cnc2[nH]c(=N)sc2c1 89176,C1(C)(CCC)CCN(C(COC(C)(C)C)C(=O)NC(c2ccccc2)C)C1 89177,CC1(CNC(C2CC(F)C(=O)N2)=O)CCCN1C(c1nc(Cl)cs1)=O 89178,C1(C(=O)N(C(C)CN(C)C(C)=O)C)(CC)CCNC1=O.C1C(CCO)O1 89179,c1(CC)cccc(C(=O)NC2CCCC(CNC(c3c[nH]c(=NC)s3)=O)C2)c1O 89180,c1(C(=O)NCCOCCCNC(C(C)OC)=O)ccnc2c(C(=O)OC)cnn12 89181,c1(C(N2CCC(F)(CO)CC2)C(=O)NCC(=C)C)cccc(C2CC2)c1F 89182,CN1CC(O)(CN(C)C(C2(OC3CCOCC3)CC2)=O)C1.C(=O)(C)NC 89183,CC1CCC(O)C(NC(c2ccc(CNC(c3csc(Cl)n3)=O)nc2)=O)C1 89184,N1(C(C(CC)N(C)C)=O)CCCC(CN(C)C(c2ccn(CCOC)n2)=O)C1 89185,c1(C(=O)NCCN(C(CCC2C(C)C2)=O)C2CC2)cnc2nc(O)nc-2[nH]1 89186,c1(CC(=O)NC2C(OC)CN(C(c3ccsc3OC)=O)C2)cc(F)ccc1O 89187,C1(CNC(c2c(C)snc2)=O)CN(c2nc(C3CC3)ns2)CCC12CCOC2 89188,N1(C(C2(CC=C)CC2)=O)CCC(C(=O)NC2CC(C#N)C2)CC1 89189,c1(C(N(CC(CNC(C2(CC)CC2(F)F)=O)O)C)=O)nn(C)c2c(=O)[nH]cnc12 89190,c1(C(N2C(C)CCC(NC(C3C(=C)C3)=O)C2)=O)cnc2ncccc2c1 89191,c1(CNC(C(F)=C(C)C)=O)ncoc1C1CN(C(C2CC(C)CO2)=O)C1 89192,C1(CNC(CCn2c(C)csc2=O)=O)CN(C)CCN1C(c1cccc[n+]1[O-])=O 89193,c1(C(C)C)ccc(N)c(C(N2C3CCC2C(NC(C2CCCOCC2)=O)C3)=O)c1 89194,c1(C(C(=O)NNC(C(=O)NCC(C)CCNC(C)=O)=O)C)cccnc1.C1(N)CC1 89195,Cc1nn(C)c(N(C)C)c1-c1cn(CC(N2CCCN(C3(C)CC3)CC2)=O)nn1 89196,N1(C(CN2CCCC(CC)C2)=O)CC2(CCCC2NC(C2C=C2C)=O)C1 89197,N1(C(C2C(C)C2)=O)CCC(OCCNC(C2CC2c2ccoc2)=O)CC1 89198,C(CC(C(=O)NC1CCCCC1)N(C)Cc1cnn(C)c1)SC 89199,C1(C(=O)NCC(C)N(C(=O)CSCc2ccncc2)C)C=CC=CC=C1 89200,C(=O)(CCN=C(NCC1CN(C(=O)C2CC2)C1)N1CCCC1)Sc1ccccc1 89201,Cn1cc(C(=O)NC2C=CC(C(=O)NC3(n4ccnn4)CC3)C2)c(=O)n(C)c1=O 89202,C1(CC(=O)NC(CN(C(CCSCC)=O)CC)CC)OCCC1C 89203,N1(C(c2cc(C)[nH]c2C)=O)CC2CC(C(=O)NCC#CCCO)C(C2)C1 89204,Cc1ccc(C2CCCC2NC(c2ccc(Br)cc2)CO)c(Br)c1 89205,C12(NC(C(C)CC3CCCC3)=O)CCCC1CN(C(=O)CC1(CO)CC1)C2 89206,N1(C(C)=O)CCCC(C(c2nnc(C(C)(C)C)s2)NC2CCCC2C(=O)NC)C1 89207,N1(C(c2c(CNC(c3c(CC)noc3)=O)occ2)=O)CC2CCC2(OC)C1 89208,C1(C(=O)NCC2CC(NC(c3cccc(OCC(F)F)c3)=O)C2)C(F)(F)C12CCC2 89209,C1(CNC(Cc2n(C)ncc2)=O)CC(F)CN1C(=O)CSC(C)(C)C 89210,c1(C(C)C(=O)NC2CCN(C(c3cc(C4CCC4)[nH]n3)=O)C2)cc(F)cc(F)c1 89211,C1(NC(C(C)S(C)(=O)=O)=O)CN(C(=O)C(CSC)c2ccccc2)CCC12CCC2 89212,c1(OCCONC(C2(n3cc(C(C(C)C)O)nn3)CC2)=O)cccc(C#N)c1 89213,O=C(CCCC1CCCO1)NCC1(CO)CCC1.n12cc(nn1)C(=O)NCC2 89214,N1(C(c2ccc(CC#N)cc2)=O)CCC(NC(C2COCC2C(F)F)=O)C(O)C1 89215,C1(C(N(C2CCN(c3ncccn3)C2)C)=O)CCS1(=O)=O 89216,C1(C(N(C(CC)CCC(=O)N(C)CCNC(=O)C(C)C)C)=O)CCCC(C)(C)CC1 89217,N1(C(CC)CO)CC(=O)N(CC(N)CF)C1 89218,c1(C(=O)NCC(CC)N(C(=O)Cn2cnnc2O)C)cccc(C(C)(C)C)n1 89219,N1(C(C(C)OCC(C)C)=O)CCOCC(C=O)C1.C(C)(C)(C)NC(C)C 89220,N12C(CCC1C1CC1)C2=O.C1(C(N)=O)CCC(C(=O)NC2CCC(O)C2)C1 89221,C(=O)(C(O)CC(C)C)NC(CC)(C)CN(C(=O)CC1CNC(=O)C1)C1CC1 89222,Cc1cc(C(=O)NCC2CC(F)(CNC(=O)CC(C)F)C2)ns1 89223,C1(C)(C(=O)NCCCOC)CCCN(C(=O)Cn2nc(C)cc2C)C1 89224,C1(NC(C(COCC)N=[N+]=[N-])=O)CC(N=c2[nH]cnc3cnccc23)C1 89225,c1(C(=O)NCC2N(C(C3CC(C#C)(O)C3)=O)CCC2)ccc(F)cc1SC1CC1 89226,C12(N(CCI)Cc3cccc(Br)n3)CCCCCC1NCC2 89227,Cc1cncc(C)c1C(=O)NCCCCNC(C1CCC1C)=O 89228,C12(NC(C(n3cc(CC(C)O)nn3)C)=O)CCC(C1)C(O)C2O 89229,CCCC(O)CCN=c1nc(N2CCC(C(C)(C)C)C2)c2sccc2[nH]1 89230,Cc1cc(CC(=O)NC23CC(C2)N(C(=O)CC(C)n2cccn2)C3)cc(C)c1 89231,c1(CNC(C2CCc3ccccc3O2)=O)ccccc1C1CCCCc2ccccc21 89232,c1(C(C(N2CC=CC(NC(CCS(C)=O)=O)C2)=O)C2CC2)cc(F)cc(F)c1 89233,C1(C(=O)OC)CC(C(=O)OC)C12CCCC2.N12CC(C(C#N)C1)NC2=O 89234,C(=O)(C1=CCSC1)NC(CC)CN(C(=O)CCc1ncco1)C 89235,C=CC(CC)CC(=O)N(C)CC1CCN(C(=O)C(COC(C)(C)C)N(C)C)C1 89236,C(C)(C(O)C(F)F)NC(C(C)(C1CCC1)NC(C(CC)O)=O)=O 89237,C1(n2cc(C3CCOC3)nn2)(C(N(CCC2CC2)CC)=O)CCOCC1 89238,C1(CNC(C(C2CCOC2)OC)=O)CC(C)N(C(=O)C=Cc2cncs2)C1 89239,C(=O)(C(C)C(C)S(C)(=O)=O)NC(CNC(CC(=O)NCC)=O)(C)CO 89240,N1(C(CC2CC(C)(O)C2)=O)CCC(C(=O)NCCC(O)C(F)F)C(O)C1 89241,C(CC(=O)N(C1CCCC(C)(C)C1)C)(C(F)(F)F)NC(c1c(CC)onc1C)=O 89242,C#CC1(C(N2CCOC(COC)C2)=O)CN(C(=O)CC(F)(F)F)C1 89243,CC1(C(N2CCC(CF)(NC(c3coc4c3COC4)=O)C2)=O)CC2CCC1C2 89244,c1(C(C(=O)N(CC(C)NC(C)=O)CC)NC(=O)CCOCCF)cnn(C)c1 89245,c1(CC(=O)NCCCN(c2ccccc2)C(c2cc(Cl)no2)=O)nnc(O)nc1O 89246,N1(C(c2c(C)cc(C)[nH]2)=O)CCC(NC(c2cnc(C(F)(F)F)nc2)=O)C12CC2 89247,N1(C(C2(C)CCC(C)C2)=O)CC(CNC(=O)C(C)(C)N(C)C)C(F)(CO)C1 89248,N1(C(CCc2onc(C)n2)=O)CCC(O)C(N(C(=O)CSC(C)C)C)C1 89249,c1(C(=O)NCCC(C)NC(C=C(C)c2cccs2)=O)cnc(O)cc1C 89250,c1(C(=O)Nc2cc(OC)c(Br)cc2C)c(Cl)nc2cc(Cl)ccn12 89251,O=C(CCCC1CC1)NCCCCC1CN(C(c2ncoc2C2CCC2)=O)C1 89252,C1(CC(=O)NC2(C)CC(NC(C(C)Cn3ccnc3)=O)C2)CCC(C)(C)C1 89253,N1(C(c2ccn(C3CCC3)c2)C(=O)NC)CCC(F)(C(=O)OC)C1 89254,O=[N+]([O-])c1ccc(-c2cccc(OC(F)F)n2)c(Cl)c1 89255,N1(C(COC(CC)(C)CO)=O)CCC(c2cn(CCCCOC)nn2)CC1 89256,C1(NC(=O)COC2COC2)CCC2CC1CN2C(C1CC1CF)=O 89257,c1(-c2nc(CCC)nn2C2CCC(C(F)(F)F)CC2)cc(Br)ccc1OC 89258,c1(NCCN(CC)CC)ccnc(N2CCC(N3CCC(O)CC3)CC2)n1 89259,CCC(C)(CSc1nc(CS(C)(=O)=O)nn1CCc1cccs1)C(N)=O 89260,C(=O)(CC(F)F)NCCOCCCN(C)C(c1ncccn1)=O 89261,c1(CC)nc(C)cc(=NCCC2CCC(NC(C3CCCC(O)C3)=O)C2)[nH]1 89262,C(C(=O)OCc1cn[nH]c1)(C(=O)NC(C1CCN(c2ccccc2)CC1)C)OC 89263,Cc1ccc(=N)[nH]c1C(N1CC(NC(=O)CC2CCC2)C2(CC2)C1)=O 89264,Cc1ccc(C(C)NC(C2CC2CNC(=O)C(F)C2CCC2)=O)nc1 89265,c1(C(N2CCCCC(CNC(c3ccc[nH]3)=O)C2)=O)ccc2c(=O)ccoc2c1 89266,[N-]=[N+]=NCCCCC(=O)NCCOC1CCN(C(=O)CC2CCCC2(F)F)C1 89267,C#CC1(C(N2CCC(OC)C2)=O)CCN(C(=O)C(C)CCC)C1 89268,C#CC1(CC)COCCN1C(=O)NC1CC1c1n[nH]c(C)n1 89269,c1(OC)ccc(CCC(=O)NC2CCC(NC(c3cnc(S)n3C)=O)C2)cc1F 89270,c1(N2CCC(C=C)C2)nc(=NC(Cc2ccccc2)CCO)[nH]c2ncn(C)c12 89271,N1(C(Cn2c(C)cnc2)=O)CCC12CN(C(=O)CCc1cccc(C(C)C)c1)C2 89272,Cc1noc(C)c1C(C)(C)C(=O)N(CCCNC(=O)C(C)NC(C)(C)C)C 89273,C(C(=O)NN1CCCC1C(=O)N(C)CCc1cnnn1C)OCC=C 89274,C1(CNC(=O)C(=O)NC2CCN(c3cc(F)cc(F)c3)C2)CCCC2OCCC12 89275,C1(NC(CC2CC(C(=O)OCC)C2)=O)C=CCN(C(c2ccnc(C3CC3)c2)=O)C1 89276,C#Cc1ccc(C(=O)NC(Cc2cn[nH]c2)C(=O)NCCN2CCOC2=O)o1 89277,CP(C)(=O)c1ccc(C(=O)NC2CC3CC2N(C(C2(C#N)CC2)=O)C3)s1 89278,CC#CCC(C)N=c1[nH]c(=N)[nH]c(=NCc2ccc(C)cn2)[nH]1 89279,c1(C(=O)NC2(CCNC(C3C(C)C3C)=O)CC2)ccc(Cl)c(O)c1 89280,c1(C(=O)NCC2N(S(CCC(=O)OC)(=O)=O)CCOC2)ccc(S(N)(=O)=O)c(Cl)c1 89281,C1(CCC(=O)NCC(C)(C)F)CCN(C(c2cc(Cl)ncn2)=O)CC1 89282,CC1Cc2ncccc2CN1S(=O)(=O)c1cc(-c2ccccc2)ns1 89283,c1(C(C(=O)NCC(CNC(=O)C(CO)C2CCC2)OC)C)ccc(C(F)F)cc1 89284,Cc1ccc(C(CNC(c2nccnc2C)=O)NC(C2CCC(C)(C)C2)=O)cc1 89285,C(=O)(C(C)(C)CCCN=[N+]=[N-])NC1CC(C)(CNC(C2CCOC2)=O)C1 89286,CC1(C)COCCC1C(N1CC2CC2(NC(c2csc(-c3cnc[nH]3)n2)=O)C1)=O 89287,c1(C(=O)NC2C(CNC(Cc3cc(C)sc3C)=O)C2)c[nH]c2ccccc2c1=N 89288,c1(C(C(F)F)NC(CCn2cc(CCCOCC)nn2)=O)c(F)cccc1F 89289,C1(C(=O)NCC23CC(CO2)N(C(c2cccnc2)=O)C3)Cc2cncn2C(=O)N1 89290,c1(OCC)cc(NCC(Cc2ccc(F)cc2F)C(C)C)ccc1Br 89291,CCCCC(C)CCC(=O)N(CCCN(C(=O)CCc1c(F)cccc1F)C)C 89292,c1(C(N2CC(SC)C(NC(c3csc(Cl)c3)=O)C2)=O)ccc2cc[nH]c2c1 89293,Cc1coc(OCCOCCNC=O)c1-c1ccccc1.C(=O)(CN(C)C1CC1)NC 89294,Cn1c(COCC(=O)NCCC2CN(C(c3cnn[nH]3)=O)CCO2)nnc1S 89295,Cc1c(C(C(=O)NC2CCCC2)N(C)Cc2ncon2)cnn1CCO 89296,C1(C2CCCN(C(c3ccc(C)cc3)=O)C2)(NC(C(C(COC)C)C)=O)CC1 89297,n1(C(C)C)cnnc1CC(=O)NC1(C(=O)O)CC1 89298,N1(c2nnc(COC)s2)CCC(NC(=O)CC2CCOC2)CC(C)(C)C1 89299,N1(C(C2C(c3c(C)occ3)C2)=O)CCN(C(=O)C(Cl)=CCl)C2CCCC12 89300,N1(C(C(CC)CN(C)C)=O)C2CCC(C(=O)NC(C(C)C)C3CCC3)C1CC2 89301,c1(OC)noc(C)c1C(=O)NC(C1CC(NC(c2cnn(C3CC3)c2C)=O)C1)C 89302,c1(C(=O)NCCNC(Cc2cnc(C)s2)=O)csc(=NC2CCCCC2)[nH]1 89303,N1(CCN2CCOCC2)CCOCC1NC(c1cccc(NCC)c1)=O 89304,N1(CC(=O)NCCN(CCC)C(c2snc(O)c2Cl)=O)CCC(CO)CC1 89305,N1(C(c2cccc(C)n2)=O)CCCC2CN(C(=O)C(c3cccnc3)O)CCC12 89306,N1(C(COC(C2CCN(c3ccncc3)C2)=O)=O)CCCN2CCCC2C1 89307,Cc1ccc2[nH]nc(C(=O)NC(C)(CNC(C3CCC4CC3CO4)=O)C3CC3)c2c1 89308,CC1=C(c2ccccc2)CN(c2cccc(S(=O)(=O)N3CCSC(C)C3)n2)CC1 89309,N1(C(C2(CC)CCCCO2)=O)CC(NC(=O)CCC2(C)COC2)C2(CC2)C1 89310,N1(C(C(CC)COC)=O)CCC2(CC1)CCN(C(C1(C)COC(=O)C1)=O)C2 89311,c1(C(CO)NC(=O)NCC(C2CCCN(CC)C2)=O)ccc(F)c(C)c1F 89312,C12(CNC(c3cc(CC)on3)=O)CCC1CCN2C(=O)C=Cc1ccc(C)nc1 89313,Cc1ncc(C(N2CCC2(C)C(=O)N(C2CCCC(O)C2)C)=O)cn1 89314,C1(NC(C2(C=C)CCCC2)=O)CC2CC(NC(C3(CF)CC(F)(F)C3)=O)CC12 89315,c1(C(N2CCC(C(Cc3c(C)nccc3)C)CC2)=O)ncc(Cl)cc1C(=O)O 89316,Cc1ccc(C(=O)NC(C)C(C(C)C)NC(=O)CSc2c(C)n[nH]c2C)cc1 89317,N1(C(C2(C)N(C)CCC2)=O)CCC2(CC2C(N2CCOC3(CC3)C2)=O)C1 89318,C(=O)(CC(O)C(C)C)NC(COCC)C(=O)NCCc1[nH]cnc1C 89319,C(=O)(C(F)(F)CC(F)(F)F)N(CCNC(C1CC1CF)=O)C1CC1 89320,c1(C(=O)NCCOC2CN(C(c3n(CC)cnn3)=O)C2)ccnc(C)c1Cl 89321,C(=O)(C1=C(C)OCCC1)NCCCN(C(c1cccc(OC)n1)=O)C(C)C 89322,Cc1c(C(=O)NC2CC(CNC(=O)CC(=O)NC3CC3)C23CCC3)ccn1C1CC1 89323,C(=O)(CCC(F)(F)C(F)F)NCC1C(C(N2CCC(C(N)=O)CC2)=O)CC1 89324,CCC(C(=O)Nc1n[nH]cc1C(N1CCC(C(C)OC)C1)=O)N(CC)CC 89325,CN1CCN(C(C2CC3(CCO2)CC3)=O)C(C(N2CCCC(C#N)C2)=O)C1 89326,C(=O)(C(C)(C)C1=CCN(C(c2cnc(OC)nc2)=O)C1)N1CCCC(CCC)C1 89327,CCCC(C(=O)NCCN(C1CCCC1)C(c1ccsc1)=O)OC 89328,Cc1cnc2cc(C(N3CCN(C(C4CC=CC4)=O)C(CO)C3)=O)ccn12 89329,C#Cc1ccc(Br)c(C(=O)NC(C)CN(C)C(C2(C)C=CCCC2)=O)c1 89330,C1(C(=O)O)CN(C(c2cnco2)=O)CC12CN(C(c1ccccc1O)=O)C2 89331,c1(CN(C)C(=O)NC2NCCC2C2CC2)c(F)c(F)c(F)c(F)c1F 89332,N1(C(C(C)CSC(F)(F)F)=O)CCN(C(C23CCC2CC3)=O)CCC1C 89333,c1(C(=O)NCC(CO)NC(C(c2ccc(C)o2)C)=O)n[nH]c2c1CCCC2 89334,N1(C(C(=O)NC)N(C(CNC(=O)OC(C)(C)C)C)CC)CCC(CCOC)C1 89335,c1(C(N2CCN(C(CC=C)=O)CC2CC2CC2)=O)cc2ccc(F)cc2cn1 89336,CCC(CC)(CCNC(=O)Cc1ccon1)NC(=O)C(Cc1ccccc1)N(C)C 89337,C1(NC(CC(C)c2ccccc2)=O)CN(C(c2ccc(O)nc2Cl)=O)CC12CC2 89338,c1(OC)ccc(C(C)CNC(N2CC3(CC3)CC2CC2CCCC2)=O)cc1OC 89339,C1(N(C)CC=CC=O)(C(=O)N(CC)Cc2c(C)cnn2C)CC(F)(F)C1.CC 89340,CC(C(=O)N1CC(NC(C2CN(CC(F)(F)F)C2)=O)C(O)C1)C(F)F 89341,N1(C(CC(C)(C)C(F)F)=O)CCC2CCN(C(C3CNC(=O)N3)=O)C2C1 89342,c1(OC)cccc(C=CC(=O)NCC2(O)CN(C(=O)CC(C)(C)CN(C)C)C2)c1 89343,C1(c2cccc(C)c2)CCCN1NC(=O)c1cnn(C2CCCCC2)c1C 89344,C(=O)(C(C)(C)c1cccs1)N(CCOCCNC(CSCC)=O)C 89345,C1(C(=O)NC2(C)CN(C(=O)C3=CCC(F)(F)CC3)C2)CC12C1CC3CC(C1)CC2C3 89346,C1(CC)CN(C(c2cccc(Cl)c2)=O)CCN1C(c1cc(O)nc(OC)n1)=O 89347,CCC(COC)C(=O)N1CCCC(NC(=O)C=Cc2cncn2C)C1 89348,C1(NC(c2cn(CCCC)nc2)=O)CN(C(=O)C(C)(C)OC)CCC12CCC2 89349,C(=O)(C(O)CCC(C)C)N1CCN(C(CNC(C2(C#C)CC(=O)C2)=O)C)CC1 89350,c1(SC)cccc(NC(N2CCCC2c2cc(C)ccn2)=O)c1 89351,c1(C(=O)NCCC(C)(C)NC(C=CC(CC)C)=O)ccccc1O 89352,c1(N2CCC(C)(NC(=O)C=CCOCc3ccccc3)C2)cncc(C#N)n1 89353,c1(C(N(C)CCOCCCN(C)C(C2CCCC2O)=O)=O)cc2ccccn2c1 89354,C1(CCNC(C2C(c3n(C)ccn3)C2)=O)CCCCN1C(C1COCC1(C)C)=O 89355,C(CC(=O)N1CC(S(N)(=O)=O)C1)(C(F)F)NC(C1(C)COCCO1)=O 89356,c1(NC(C2N(C(=O)OC)CC3(CC3)C2)=O)cccc(NC(=O)C(F)F)c1C 89357,N1(C(c2cnn(CC)c2C)=O)CCCC(NC(=O)CC2(CO)CC2)C(F)C1 89358,c1(C(N2CCC(NC(c3c(C)ncn3C)=O)C2)=O)ccc(N)cc1C(C)(C)C 89359,N1(C(C(C2(O)CN(C(CN(C)C3CC3)=O)C2)F)=O)CCCC12CCNC2=O 89360,N1(C(C2CSCCN2C(c2cccs2)=O)=O)CCc2ncncc2C1 89361,C(CN=c1cccc(S(=O)(=O)NCc2ncccc2N)[nH]1)c1ccc(C)nc1 89362,Cc1c(C(=O)NC2COCCN(c3nc(Cl)ncc3C(N)=O)C2)c(C(F)F)nn1C 89363,c1(C(=O)NCC2C(CNC(C3(C)C(C)(C)C3)=O)C2)cc(O)cc(O)n1 89364,N1(C(C)C)C(=O)NC(CSc2ccccc2)C(C(=O)OC(=O)C2CC2)=C1C1CC1C 89365,C1(CN(C)C(C2CC(CC3CC3)C2)=O)CCCN(C(C2C3CC(=O)CC23)=O)C1 89366,C(=O)(C1CCCn2cncc21)NC1(C)CN(C(=O)Cc2c(Cl)ccc(O)c2Cl)C1 89367,C#CCC(C)(CC)C(=O)N1CC(NC(c2ccc(CC(C)C)cc2)=O)C(C)(C)C1 89368,C1(NC(C2OCC(CNC(CCCNC(=O)OC)=O)C2)=O)Cc2ccccc2C1 89369,N1(C(C2OCCN(C(CC(C)OC)=O)C2)=O)CCC(C2CCC2)C1 89370,Cc1c(C(C)NC(=O)NCCSc2ccccc2)cnn1CC1CCCO1 89371,C(C(C)N=c1ccc(C(F)(F)F)n[nH]1)NC(c1c(C)nc(CO)nc1)=O 89372,C1(C(C(=O)N(C(CN(C(COCCCC)=O)C)C)C)OCC)CCCCCC1 89373,C(CN=c1[nH]c(CCO)cs1)(c1ccccc1)N(c1ccccc1)C 89374,O=C1CC(n2cc(NC(=O)C(=O)NC(c3cccc(Cl)c3)CO)cn2)C(=O)N1 89375,C1(CNC(c2cc(C)ccc2NC(C)=O)=O)CN(C(=O)C(C)N(C)C)CCC1(F)F 89376,N1(C(C#CC(=O)N(C)C)=O)CCCC2(NC(=O)CN3CCCCCC3)CC2C1 89377,c1(CNCC(C)CF)ccc2nonc2c1 89378,c1(C(N(CC(O)CNC(C2CC=CC2)=O)C)=O)cnn(CCC2CCCCO2)c1 89379,c1(CCCCn2cc(-c3ccc(C=C)cc3)nn2)c(C)cc(NC(C)=O)cc1C 89380,CC(O)(C(=O)NC1CC2CCN(C(=O)Nc3ccc(F)c(F)c3)CC12)C(F)(F)F 89381,C1(C#N)(C(N2C(C)C(C(=O)NCC(c3cccnc3)O)CC2)=O)CC12CCC2 89382,Cc1nn(C)c(Cl)c1C=CC(N1CCC(O)C(NC(C2(O)CCC2)=O)C1)=O 89383,c1(C(N(C)CC2CN(C(C3C=CC(=O)N=N3)=O)CCO2)=O)ccc2[nH]ccc2n1 89384,c1(CNC(C2CC(=C)CN2C(=O)CCC(N)=O)=O)cccc(Cl)c1F 89385,C#Cc1ccccc1CC(=O)NCC1CC(CNC(C2C=CC=CC=C2)=O)CO1 89386,C(=O)(C1CCCc2sccc21)NC1CCC(CNC(c2ccc(N)c(F)n2)=O)C1 89387,n1(CC(N2CCCC(NC(=O)C(F)(F)C3(O)CCC3)C2)=O)cc2ccccc2n1 89388,N1(C(=O)OC(C)(C)C)CCCCC(NC(=O)NC(CO)C2CC2)C1 89389,C1(C(C(=O)NCCCCN(C(C)C)C)C)CCCN(C(=O)C=CC2CC2)C1 89390,C(=O)(C1=CCC(F)(F)CC1)N1C(CNC(=O)CNC(=O)OC)CC(COC)C1 89391,C=CCC(F)(F)C(=O)N1CCC(CCCNC(=O)C(CCOC)OC)CC1 89392,c1(C(=O)NCCN(C=O)C2CC2)ccc(C2CC2)cn1.C1(n2ccnc2)(CO)CCCC1 89393,C1(OCCNC(C2CC(C3CC3)C2)=O)CCN(C(C2(C(F)F)CCCO2)=O)CC1 89394,N1(CCCOCC)CCN(C(c2nc(C(F)(F)F)c(Cl)[nH]2)C(=O)NC)CC1 89395,c1(C(N2CCCC(CC(=O)NC(C)CCc3cn[nH]c3)C2)=O)cncn(C)c1=O 89396,C(C)(CNC(=O)C(c1cccs1)NC(C1CCSCC1)=O)(CO)OC 89397,C#Cc1cccc(C(N2CCC(O)(C(C)NC(=O)CCC3CCCOC3)C2)=O)c1 89398,Cn1cnnc1CCC(N1CC(CO)(NC(c2ccc(-c3cc[nH]n3)s2)=O)C1)=O 89399,c1(NC(C2N(C(c3c(C)nc4sccn43)=O)CCOC2)=O)cccc2nc(O)oc12 89400,C(=O)(C1=C(Cl)CCCC1)N(CCCNC(C(C)NC(CC)=O)=O)C(C)C 89401,N1(C(CCC2(C)CC2(F)F)=O)CC(C2CN(C(C3COCCC3(F)F)=O)C2)C1 89402,N1(C(CS(=O)(=O)N(CC)CC)=O)CCCC2CCCC12.c1(C(=O)NCC)cnco1 89403,C1(C(=O)NC2CCN(C(C3C(CCC)C3)=O)CC2)CC2(CCCC2)CO1 89404,c1(CC)cnccc1C(N1CCC(N(C)CC2N(C(COC)=O)CCCC2)C1)=O 89405,C(=O)(N=c1ccnc(C(F)(F)F)[nH]1)C1N(Cc2n(C)cnc2)C2C(C1)C2 89406,C1(C(N2C(C(=O)NCC3(O)CC3)(CC)CCC2)=O)C2CCC(C2)C1C 89407,CC(CC1CCC1)C(=O)N(C)CC1CCCN1C(C1CC1C(C)(F)F)=O 89408,C=CC1(C(=O)NC(CC)CC(F)(F)F)CCN(C(c2cc(C)ccc2O)=O)C1 89409,Nc1cc(C(N2CCCC2CNC(C2CCCC23CC3)=O)=O)cnc1Cl 89410,Cc1cnn(C)c1CC(=O)NC(c1ccccc1C(F)(F)F)C(F)F 89411,c1(C(=O)NCC(CC)NC(c2c(C)csc2C(=O)OC)=O)cccc2c[nH]nc12 89412,CCCC(C(=O)N(CCCNC(C12CC(c3ccccc3)(C1)C2)=O)C)N(C)C 89413,N1(C(CC2C(C)OCC2)=O)CCC(NC(=O)Cn2cncn2)C(C)(C)C1 89414,c1(OCCCCC)ccc(NC(=O)C(c2cccc(OC)n2)(F)F)cc1 89415,c1(C(=O)NC(CCC2CCC2)C(=O)NCC2(F)CC2)n[nH]c2ccccc12 89416,C=C(C)c1ccnc(NC2C3CCC4C(C3)CC24)n1 89417,n1(CC)cc(Cl)c(C(=O)NC2CCCC(CNC(=O)CC3CCS(=O)(=O)C3)C2)n1 89418,N12CCC3(CC1)CC3C2=O.c1(CNC(=O)OC(C)(C)C)ccoc1C(=O)O 89419,c1(C(N2CC(C)C(NC(c3cc(N)c(Cl)cn3)=O)C2)=O)ccc(C2CC2)nc1O 89420,O=C1NCC2CN(C(c3cccc(N4CCCOC4=O)c3)=O)CCC12 89421,c1(C(N2C(C(C)C)C(C(=O)NCC3CC(F)(F)C3)CC2)=O)ccc2c[nH]nc2c1 89422,C1(CC(N2CCC(CC)C2CNC(=O)C=CCOC)=O)CCC(C)(C)CO1 89423,c1(COCC)cccc(CNC)c1.C12CCCCC1CNC2=O 89424,CN1C(=O)CN(CC(=O)NCCC2(NC(=O)Cc3ccsn3)CCC2)C1=O 89425,C1(C(N2CC(NC(c3c(Cl)cn(CCC)n3)=O)C(O)C2)=O)CC2CCCC(C1)C2 89426,c1(C(N2CC(C3(NC(c4c(SC)ccs4)=O)CC3)C2)=O)c(C)ccc(C)c1O 89427,n1(C(C)C)cc(C(=O)NC2CN(C(C3(F)C4CCCC34)=O)C2)c(O)nc1=O 89428,c1(N2C(C(=O)NCc3c(OCC)ccs3)CSC2)nc(C)cc(C#N)n1 89429,c1(C(=O)NCCN(C(=O)C(C)(C)C2CCOC2)CCC)cccc(S(C)(=O)=NC)c1 89430,C1(C#N)(NCC(=O)NCC(CNC(C=CC(c2cccnc2)C)=O)(C)F)CC(=O)C1 89431,c1(OC(C)C)nc(NC(C2CCN(Cc3cc(Br)ncc3Br)CC2)=O)cc(O)n1 89432,C1(CNC(c2cc(C)n(C3CC3)c2C)=O)CN(C(=O)C(N)=O)CCC12CCC2 89433,n1(CC(N2CCC(COC)(NC(C3CCC3(C)C)=O)C2)=O)cc(S(N)(=O)=O)cn1 89434,Cn1nc(C(=O)NC(CNC(c2csc(C(F)F)n2)=O)C(C)(C)C)cc1CO 89435,N1(C(CCC2N(C(C(C=C)OC)=O)CCCC2)=O)CCC(C)(OC)CC1 89436,C(=O)(C#CC1CCOC1)N(C(C(CC)C)C(=O)NC1(CC2CC2)CC1)C 89437,C1(CNC(C(C(C)O)Nc2ccncc2C(F)(F)F)=O)CN(C(N)=O)CCN1C 89438,C=CC1(C(=O)NCC2(O)CC(NC(=O)CNc3cccnc3)C2)CCC1 89439,C1(CNC(C2(F)C(C)OCC2)=O)CCCCN(C(=O)C=CCn2cncn2)C1 89440,N1(C(C(N2C(CC)CCSC2)=O)C)CCC(C)CC1 89441,CCCCC(C)(F)C(=O)N1CCCC(Cc2cn(C3C(=O)OCC3(C)C)nn2)C1 89442,CCCC(C)C(=O)N(CCCNC(=O)CC1CC=CCN1C)C(C)C 89443,C(N=c1[nH]c(=NCCOC)[nH]c2c1CSC2)C1C(CNS(NC)(=O)=O)C1 89444,c1(CC(N2C(CNC(=O)CC3CNC(=O)O3)CCC2)=O)c[nH]c2cccnc12 89445,N1(C(c2c(C)ccs2)=O)CC2(C1)C(Nc1nccc(C)n1)CCS2(=O)=O 89446,CC(O)(CC(=O)N1CC2CC1CC2NC(=O)Cc1ccc(Br)nc1)CC(=O)O 89447,c1(C(N(C(CCNC(CCC(CC)C)=O)C)C)=O)ccc(=NCCOC)[nH]c1 89448,Cc1cc(CNC(=O)CCCCCn2cc(-c3cncc(C)c3)nn2)cc(F)c1 89449,C1(CCC)(NC(=O)C(C)CCOC)CCCN(C(c2sccc2C(F)F)=O)C1 89450,Cc1cc(Br)ccc1CCC(N1CCOC(C(C)NC(=O)C2=C(Cl)CC2)C1)=O 89451,C(=O)(CCCC(=O)NCC(C)NC(=O)Cc1ccc(OC)c(Br)c1)NC 89452,C1(CCNC(C(CC)n2cncn2)=O)CCCN(C(c2oncc2C)=O)C1 89453,c1(C(=O)NCCOCCNC(C2N(N=O)CCCC2)=O)ccc2[nH]nc(Cl)c2c1 89454,C(=O)(C1=C(Cl)CCOC1)N1CCC(NCC)CC1.n1(CC=O)nc(O)ccc1=O 89455,c1(C(N2CCN(C(CNC(C(C)SC)=O)=O)CC2)=O)ccc(Cl)c(F)c1O 89456,C1(C(=O)NC(CC)CN(C(=O)C2=CCC2)C)CC(C)(C)CCO1 89457,C12(NC(COc3cncc(C)n3)=O)CCC1CN(C(=O)CC1CNC(=O)C1)C2 89458,c1(CC(C)C)cc(C#N)c(NC(=O)CNC(C2(F)COC2)=O)s1 89459,CCC(C(=O)NC1CN(C(c2nccn2C)=O)CCC1C)C(C)C 89460,C(C(N=[N+]=[N-])C(=O)NC1CC(C(=O)NC(C)CC(=O)OC)C1(C)C)OCC 89461,O=C(C(Cl)=CCl)NC1(CO)CN(C(=O)C=Cc2ccoc2)C1 89462,c1(CC(=O)N(C)CC2CCN(Cc3cccnc3Br)C2)cccc(O)c1 89463,N1(C(c2c(Br)ccc(N)c2)=O)CCC(NC(C2CCCS2)=O)C2(CCC2)C1 89464,N1(C(C(CC)SC)=O)CCC(CNC(=O)C=Cc2cccc(OC)c2)C(C)C1 89465,CC1(C(=O)NCC2CCN(C(=O)C(C)(C)c3cnc[nH]3)C2)CC(F)(F)C1 89466,CS(=O)(=O)c1cc([N+](=O)[O-])ccc1NCC(c1cc(Br)ccc1Cl)O 89467,N1(C(C2CCCC(=O)CC2)=O)CC2CCC(C1)N2C(=O)CSCc1cccnc1 89468,CC1=C(C(=O)NC2(C(=O)NCCCO)CC2C)COCC1 89469,CC(C)(C)CCC(=O)N1CC(C)(C)CC1CNC(=O)Cn1ccc(C2CC2)n1 89470,N1(C(C(CC)C2CCOCC2)=O)CCCN(C(C23CCC(C2)OC3)=O)CC1 89471,N1(C(Cc2ccc(CC)s2)=O)Cc2ccccc2C(NCc2ccc(Cl)cc2)C1 89472,N1(c2ccnc(CN(C)CC3CC4(C3)OCCO4)n2)CCc2c(Cl)cccc21 89473,N1(C(CC2CCCN(C(C(C(=O)OC)(C)F)=O)CC2)=O)CCC(C)C(C)(C)C1 89474,c1(C(N2CCCC3CC23)CC)ncc(C)cc1-c1ccc(CN2CCCC2=O)s1 89475,CN1CCC(C(=O)NCC=CCNC(=O)CCC(=O)c2ccccc2)CC1=O 89476,c1(C(=O)NCC2(F)CC(CN(C)C(C3(C)CCCCO3)=O)C2)ncn2c1CCC2 89477,N1(C(C(=O)N(C)C)=O)CC2(CCC2)CC1C(=O)NCC(C)(O)C(=O)OC(C)(C)C 89478,N1(C(CSCCOC)=O)CC(C)(C(N2CC(F)(F)CCC2C)=O)CC1(C)C 89479,Cc1cncc(C(N2CC(CC(C)NC(=O)C(C3CCC3)C3CCC3)C2)=O)n1 89480,CC1CC2(CO1)CC(F)(F)C2N=c1[nH]c(=N)[nH]c(=NCc2ccc(N)cc2F)[nH]1 89481,CCC(CC)=CC(=O)N(C1CCCO1)CCCC(C)C 89482,C#CC1CCCC(NC(=O)CC2(NC(C3CN4CCC3CC4)=O)CC2)C1 89483,C(=O)(C(C)(C)CS(N)(=O)=O)NCC1C(NC(c2cnc(OC)s2)=O)CC1 89484,C(CCC(C)(C)C(=O)NNc1ccc(S(=O)(=O)NCC2CC2(F)F)cc1Br)OC 89485,C1(C(=O)NC2(C)CCC(CNC(c3n(C)cnc3)=O)CC2)C2CCC3C(C2)CC13 89486,Cc1nc(Cl)ncc1CN(CCC(N1CCCCCC1)=O)C 89487,N(C1CC2CCCc3cccc1c32)C(C(C(CCC)NC(C)=O)O)=O 89488,C1(NC(c2c(CC(C)C)nc(C)s2)=O)CC2(CCN(C(C3C4CCC(=O)C34)=O)C2)C1 89489,c1(C(=O)NCC2CC(NC(C3C(C4C(C)C4)C3)=O)C2)cnc2c(c1)nnn2C 89490,c1(C2C(Cn3ncc(C)c3)C2)cc(C)ccc1O.C1C(CO)CNC(=O)N1 89491,C1(NC(CC(C)O)=O)CCCCC1N(C)C(c1cc(C(=O)NC2CC2)ccn1)=O 89492,c1(C(CC)C)nc(N2CCC(NC(=O)COCC(=O)N(C)C)C(C)C2)cc(C)n1 89493,Cc1nscc1CC(N1CC(NC(c2cn(C3CCOCC3)cn2)=O)C1)=O 89494,C=CC(C)(C)CC(=O)N1CCOCC1CNC(C1CCCCN1CC(F)(F)F)=O 89495,c1(CNC(=O)OCC)nc(=NC(C)C(=O)c2ccc(OC)cc2C)s[nH]1 89496,C12(NC(C=C(CCC)C)=O)CCCC1N(C(c1ccc(F)c(C)c1N)=O)CC2 89497,C1(C(C=O)F)CC2(CCN(C(=O)C3CC3)CC2)C1.c1(COCC)cc(C#N)n(C)c1 89498,C(=O)(C(C)(C)C(=O)N1CCC(NC(=O)COC(F)(F)F)C(F)C1)NC 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89535,c1(C(=O)NC2C(NC(C(C)(C)C#N)=O)CCC2)ccc(Br)c(N)n1 89536,c1(C(N2CC3C(NC(c4n(C)ncc4C#N)=O)C3C2)=O)ncn2c1CCCCC2 89537,C1(NC(c2c(COC)ncs2)=O)(CO)CCN(C(C2CCCC2)=O)C1 89538,CCCCC(O)C(=O)N1CC2C(C1)N2C(c1cc(I)ccc1Br)=O 89539,C(C(=O)NC1(C(=O)NCc2cccs2)CC1C)(C1CC1)OCC 89540,C=CCC(C)(C)CC(=O)N1CC(CNC(C2CCN(C)C2=O)=O)OC(C)(C)C1 89541,C1(C(N2CCC(N(C(=O)CCCN(C)C3CC3)CC#C)CC2)=O)OCCCC1(C)C 89542,CCCCCC(O)CC(=O)NCC(C)NC(=O)C(c1ccc(Cl)cc1)O 89543,CCC(C)CC(C(=O)NCC(C)(O)C(C)C)NC(=O)CCOCC1CC1 89544,Cc1cnc(CCN)nc1.C1(C(C(=O)CCC2CCC2)=O)COCCC1C 89545,N1(C(C2CC(F)(F)C2)=O)CCCC(C2(NC(C3(c4ncco4)CC3)=O)CC2)C1 89546,C1(C(=O)NCCCC(=O)OCC)CCN(C(=O)c2c[nH]c(=N)c(C)c2)O1 89547,c1(N2C(CCC3CCCN(C(C=CCC)=O)C3)CCC2)nc2ccccc2o1 89548,C1(CN2CC(C)(CC)OCC2)CC2CCC(C1)N2C(CC)C(=O)Nc1nn[nH]n1 89549,c1(C(=O)NCC(CC(C)C)NC(=O)CCc2cnco2)cn2c(n1)CCC2 89550,C1(CNC(=O)CCc2cncnc2)CC2CN(C(=O)Cc3ccnnc3O)CC12 89551,N1(C(c2cc(C)nn2C)=O)CCC2(CC1)CCC2(C)C 89552,c1(NC(=O)OC)cnc(NC(=O)C(=O)NC2CC2c2ccc(F)cc2F)c(Br)c1 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89571,c1(C(N(C(CNC(=O)CSC(F)(F)F)C2CC2)C)=O)cccc(N2CCCC2)n1 89572,c1(OC)ccc(NC(=O)C(C2CCC2)N(CC(F)(F)Cl)C)c(OC)c1 89573,c1(C(=O)NCC(CC)NC(C(C(=O)OCC)(C)C)=O)cc2ccc(C)cn2c1 89574,C1(NC(c2n[nH]cc2-c2ccncc2)=O)CCCN(C(c2ccc(Cl)s2)=O)C1 89575,C1(CCNC(CCCC)=O)CCCN(C(=O)CN(C2CCSC2)C)C1 89576,C(C(C)(C)CNC(=O)C1CC1)N(C(C)C)C(=O)OC(C)(C)C.C1CC1Cl 89577,C1(NC(=O)CCCSc2ccccc2)CC(F)CN(C(=O)Cc2cnsc2)C1 89578,c1(C(=O)NCC(C)(CO)NC(c2cc(CO)ccn2)=O)cncc(Cl)c1 89579,Cc1cc(C(=O)NCC(C)(CO)NC(=O)CNc2ccccn2)ccc1O 89580,c1(C(N(C2CCN(CC3CC3)CC2)CCc2cn(CC)nc2)=O)cnn(C)c1Br 89581,C1(C)(C(N(C(C)C(=O)NC)CC)=O)CC(NC(=O)Cc2ncc(C)o2)C1 89582,C#CC1(C(=O)NCCC(C)(C)CC)CCN(C(C2CC3CCC3C2)=O)CC1 89583,n1(CC#C)cccc1CNc1ccccc1.c1(C2c3nnnn3C2)ncoc1C 89584,c1(CC(N2CC(C(C)NC(C=CC=CCC)=O)OCC2)=O)c[nH]c2ncccc12 89585,C(=O)(C(C)(C)CCCNC(C1CCOC1)=O)N(CCc1ccccc1)CC 89586,c1(C(=O)NC2C=CC(CC(=O)NC3(C)CC(C)(C)C3)C2)ccnc2[nH]cnc12 89587,c1(CCC(=O)NCC(C)NC(C2(C)CC2(F)F)=O)nc2ccccc2[nH]1 89588,Cn1ccc2sc(C(=O)NC3CCN(C(=O)CSCC4CCCO4)C3)cc12 89589,N1(C(CCc2c(OC)nccc2)=O)CC2(CCN2C(C2(C)CCCC2)=O)C1 89590,CCCCCCC(C)(CC)C(=O)NCC1CN(C(c2sccc2Cl)=O)CC1(C)C 89591,Cc1nc(CO)sc1C(=O)NC1COCC1CNC(C1CC(=O)N(C)C1)=O 89592,C1(NC(CC2(C=C)CCCCC2)=O)COC2(C1)CN(C(C1CCCC1(F)F)=O)C2 89593,N1(C(C2(C)CCC(C)CC2)=O)CCCC2CN(C(C3CC(=O)C3)=O)CCC12 89594,c1(N2C3CCN(C)C3CCC2)nc2c(c(=NCNC3CCCCCC3)[nH]1)CCC2 89595,C(=O)(C1=CCCOCC1)NCC1(O)CCN(C(C(C2CCCCC2)N(C)C)=O)C1 89596,C1(C(C)NC(C2(C(=O)NC)CCC2)=O)CCN(C(=O)CCc2nncs2)C1 89597,N1(C(C2(CC(=O)OC)CC2)=O)CCC(O)(C(C)NC(=O)C(C2CCCCC2)F)C1 89598,c1(CC)nc(C#N)cc(=NCC2CN(C(=O)C=CCF)CC2C(F)F)[nH]1 89599,C1(NC(C2C(NC(CC3CCC(OCCC)CC3)=O)CCO2)=O)CCCC(F)(F)C1 89600,N1(C(C2(SC)CC2)=O)CC(NC(=O)C(CC)c2ccccc2)CC2(CC2)C1 89601,N1(C(=O)NC2CC(CS(C)(=O)=O)C2)CC(O)(Cc2cnccn2)C1 89602,n1(CCOC)ccc(C(N2CCC(NC(=O)C(O)C3CCCC3)C2C)=O)c1C 89603,Cc1cc(C(N2CCC(N(C(=O)C(n3ccnc3C)C)CC3CC3)C2)=O)c(C)o1 89604,CCCCC(CC)CC(=O)NCCCOCCNC(=O)C=Cc1cscn1 89605,c1(OC)c(F)ccc(C)c1C(=O)NCCOCCN(C)C(c1cc(F)n[nH]1)=O 89606,C12(CCNC(CCC=C)=O)CCC1CN(C(c1csc(O)n1)=O)C2 89607,CCCCCCCC(O)C(F)(F)C(=O)OCc1noc(-c2cnn(C)c2)n1 89608,CC1CC(=O)NC1C(=O)NCCCN(C(=O)C=C1CCSCC1)C 89609,CC(O)(C(=O)NCC1CCC(CNC(c2ncccn2)=O)C1)c1ccccn1 89610,N1(C(C(CC)OC)=O)CCC2(CCCN(C(=O)C3=CSCS3)C2)CC1 89611,C1(C)(CNC(C2(CCN(C)C)CC2)=O)CN(C(=O)CC2CCCO2)CCO1 89612,c1(CNC(C2COCCN2Cc2c(C)n[nH]c2C)=O)ccc(C#N)cc1 89613,CN1CC=C(CC(=O)N2CC3(CCC3NC(c3csc(Cl)c3)=O)C2)CC1 89614,N1(C(c2ccc(C)nn2)=O)CC2CC(NC(=O)CCOCC3CC3)CC2C1 89615,N1(C(c2c(CC)occ2)=O)CCC2(CC(NC(=O)CS(=O)(=O)CCOC)CO2)C1 89616,n1(CC)cc(C(=O)NCC2CC(COC)CN2C(=O)Cc2cnsc2)c(C)n1 89617,C1(NC(c2c(OC)n[nH]c2)=O)CC2CN(C(=O)CC34CC(F)(C3)C4)CCN2C1=O 89618,C=Cc1ccc(C(N2CC3CC2CC3NC(=O)COc2ccc(F)cc2)=O)cc1 89619,N1(C(CC2CCN(C)C2=O)=O)CCC(NC(c2cc(C3CC3)no2)=O)C(CO)C1 89620,C1(CC)(CC)CC(NC(=O)C(C)C(C)C)CN1C(c1cccc(OC(C)C)c1)=O 89621,C=CC1(CC(=O)NC(C)(CNC(C2C(C)C2C)=O)C2CC2)CC1 89622,Nc1ccccc1O.c1(N(CC(O)COCC(F)F)CO)cccc(F)c1 89623,c1(C(=O)NC(CNC(C(CC)(C)CO)=O)CO)ccc2c(c1)OCO2 89624,N1(C(c2c(OC)nccc2)=O)CC(C(=O)N(C2(C)CC2)C)OC(C)C1 89625,c1(SCC(=O)NC(CNC(C2CC3C=CC2O3)=O)CO)ccc2ccccc2c1 89626,Cc1cccc(Cl)c1C(N1CCC(C(N)=O)C(C(=O)C(F)(F)F)C1)=O 89627,C1(CNC(C(=O)NCC=C(C)C)=O)CC(CN(C)C)CO1 89628,c1(CC)ccc(C(=O)NC(CNC(=O)CCc2cnn(C)c2)CC)cc1Cl 89629,c1(OC)cnccc1C(=O)NCCc1n[nH]cc1C(=O)NCC(C)(O)CCO 89630,c1(C(=O)NC2CN(C(c3cccc4c3OCO4)=O)C2)noc2ccc(Br)cc12 89631,N1(C(c2c(C)nn(C)c2)=O)CC2CCCCC2(NC(=O)Cc2cncn2C)C1 89632,C1(C(N(C)CC)=O)CCCN1NC(=O)c1cc(N(C)C)no1 89633,CC1CCc2[nH]c(=NCc3ccns3)nc(N3CCC4(CC3)CC4(F)F)c2C1 89634,N1(C(CNC(CC)=O)=O)CC(C(=O)NCC2CC=CCC2)C2(CC2)C1 89635,C1(C(N(CCNC(c2cn(C)cn2)=O)CC)=O)CCn2c(O)nnc2C1 89636,C1(NC(c2n(C)ccn2)=O)CCN(C(C2OCC2(C)C)=O)C12CCC2 89637,CC(F)(F)CC(=O)NCc1ccoc1C(=O)NCc1ncsn1 89638,C1(C#CC(=O)N2CCC(NC(C3(n4nccn4)CC3)=O)C(O)C2)(CC)CC1 89639,c1(NC(CC(CC)C2CC2)=O)c(Br)c(C)nn1C(C)(C)C.c12cn(nn1)CCOC2 89640,C1(CC(=O)NC2CCN(C(C3(CF)CC3)=O)C2c2ccccc2)CCC(=O)NC1 89641,C#CCC(C)(C(=O)N(C)Cc1ccncn1)NC(=O)COCCSC 89642,N1(C(CCOCC(C)C)=O)CCCC(C2(NC(C3CCNC3=O)=O)CC2)C1 89643,S(=O)(=O)(c1ccc(=NCC2CCCCCC2(F)F)[nH]c1)NC1CC(=O)NC1 89644,c1(C(N2CCC(N(C(CC=C=C)=O)CC3CC3)CC2)=O)cc(C)ncc1C 89645,c1(C(=O)NCC2C=CC(NC(C(C)=C(CC)C)=O)C2)c(C)ccoc1=O 89646,N1(C(C(c2ccccc2)OC)=O)CC(NC(c2cc(C)cc(C)c2)=O)CC(F)C1 89647,CCC(C(=O)N1CCOCC(C(=O)NCC2(F)CC(O)C2)C1)C(F)(F)F 89648,c1(OCCNC(C(N2C(CCC)CCC2)c2ccn(CC)n2)=O)ccccc1Cl 89649,N1(C(c2c(C)c[nH]c2)=O)CCC2CN(C(c3cccc(CCO)c3)=O)CCC2C1 89650,CC1Cn2nc(C(=O)NCCNC(C3CCCC(F)(F)C3(F)F)=O)cc2C(=O)N1 89651,c1(C(=O)NCC(C)NC(=O)CNC(=O)C2CC2)cccc(-c2ccccc2)c1O 89652,N1(C(C(CC(=O)OCC)(C)C)=O)C2CCC1CC(NC(c1nscc1C)=O)C2 89653,N1(C(CC=CC(C)(C)C)=O)C2CCC(C2)C1C(=O)NCC1(F)CCOC1 89654,C(C(F)(F)CO)(c1ccccc1)N(C(=O)CNc1cccc(OC(F)F)c1)C 89655,N1(C(C(c2ccccc2)OCC)=O)CCN(C(C2CC(CC3CC3)C2)=O)CC1 89656,N1(C(C(C(=O)OCC)C)=O)CCN(C(=O)COC)CC1C(C)C 89657,C1(NC(C=CC(C)C)=O)CCCN(C(=O)CC2(C)CC2(F)F)CC1 89658,N1(C(c2cc(CNC(c3[nH]cc(C)c3)=O)sc2)=O)CCC(C)(N(C)C)C1 89659,C1(C(C(=O)NCC(=C)C)N(C)C(c2cnn(C)c2)C)CC2(C1)C(F)(F)C21CCC1 89660,c1(C(N2CCC(C)(NC(C3CCC(CC)C3)=O)CC2)=O)[nH]nc2c1CCC2(C)C 89661,C1(C(=O)NCC(CN(C(c2cnc(C(=O)OC)s2)=O)C)C)Cc2ccccc2N1 89662,c1(C(=O)NC2C(C#N)CN(C(c3cc(Br)cnc3Br)=O)C2)ccc(F)c2ccoc12 89663,C(=O)(C(O)CCCNC(=O)Cn1[nH]cnc1=N)N1CC(C#C)(N(C)C)C1 89664,Cc1cscc1NC1CCC(NC(c2cnn(CC)c2)=O)C1.C(C)(C)(C)O 89665,C1(NC(CC(C)c2cccnc2)=O)CN(C(=O)CSc2n[nH]c(O)n2)CC1C 89666,N1(C(CSCC)=O)CCN(C(=O)C(O)CC(N)=O)C(C(C)C)C1 89667,c1(C(=O)NCC2(C)CCN(C(C(C)(C)CC(F)F)=O)C2)cc(C#N)c(O)nc1N 89668,c1(C(CC)C)ccc(=NCCCOCCc2ccccc2)[nH]n1 89669,C(=O)(CCCC(F)(F)F)NCC=CCNC(=O)C=Cc1ccc(Br)s1 89670,c1(C(N2CCC(C)(NC(CCN(CCC)C)=O)C2)=O)cc(C)c2ncn(C)c2n1 89671,CN1CCN(C(C2CCOC2(C)C)=O)C(C(=O)NCC2CCN(CCO)CC2)C1 89672,Cc1cn2cc(C(N3CC(NC(=O)NCc4ccn5ccnc5c4)C3)=O)nc2s1 89673,N1(C(Cc2cccc(OC)c2)=O)CC2(CC(NC(=O)CCC(C)OC)C2)C1 89674,c1(C(=O)OC)nc(NC(C2CN(C(C)=O)CCO2)=O)cnc1C 89675,N1(C(c2c(C)noc2)=O)CCCC(CCC(N2CC=CC2C(N)=O)=O)C1 89676,c1(OC)nn(C)cc1C(=O)NCC1(NC(=O)C=CS(C)=O)CCOC1 89677,Cc1c(CC(N2CCOCC(C)C2)=O)sc2ccccc12 89678,C1(C)(CNC(C2CC(NC(C(C3CCOCC3)OCC)=O)C2)=O)CCCCCC1 89679,C(=O)(CC(C)CNC(C1CCS(=O)CC1)=O)NC(C#C)CC1CCC1 89680,c1(NCC2CCN(C(c3cc(C4CC4)ncn3)=O)C2)c(F)cccc1[N+](=O)[O-] 89681,Cc1ccc(C(=O)NCC(C)(Cn2cccn2)NC(=O)CCC2CC2(F)F)n1C 89682,N1(S(CC)(=O)=O)CCCC(C(N2CC3CC3(NC(=O)CCCCC3CC3)C2)=O)C1 89683,c1(C(N2CC3C(NC(C4C(C)C4C)=O)C(CC3)C2)=O)csc2c(Cl)cccc12 89684,c1(C(N2CCC(F)(c3nn[nH]n3)CC2)=O)ccc(-c2ccc(Cl)cc2CO)cc1F 89685,C(=O)(C1=NOC(C)(C)C1)N1C(C(=O)NC(C#C)CCC)CSCC1 89686,C1(C(N(C)CC2CCN(C(=O)CC(C)(C)O)CC2)=O)CCc2cnn(C)c2C1 89687,C#CC1CCCCN1C(=O)CSCCNC(=O)C(=O)CC(C)C 89688,c1(C(=O)NCCC2(C)CCN(C(COCCC=C)=O)C2)cccc2c1OC(C)C2 89689,C(=O)(C#CC(C)(C)O)NC1CCN(C(c2sc(C)c(O)n2)=O)CC1 89690,N1(C(c2cc(COCC)on2)=O)C(C(N2CCC(OC3CC3)C2)=O)CC2CC12 89691,c1(C(=O)NC(C2CC=CCC2)C(N2CCC(=C)C2)=O)cnc(O)cc1C 89692,c1(CC)nc(C)c(CC(=O)NC(C)(C)CCNC(=O)C(F)C2CC2)c(C)n1 89693,C1(NC(CC(CCC)C)=O)CCSC12CN(C(=O)COCc1cccnc1)C2 89694,N1(C(Cc2cccc(C)n2)=O)CCCC(N(C(c2cccs2)=O)C(C)C)CC1 89695,C=CCCC(C(=O)NCC1(C2CC2)CCC1)NC(=O)CC1COC(=O)C1 89696,c1(C2(C(N3CCC(N(C(C(CSC)C)=O)C)C3)=O)CCC2)cccc(Cl)c1 89697,C1(C(=O)NC(c2cnccn2)C)C=CCN(C(=O)CC2(N(C)C)CCC2)C1 89698,c1(C(=O)NC(C)CCCNC(C2CCCSC2)=O)cnc2occc2c1 89699,N1(C(C(CCOC)C)=O)CCC(CNC(=O)Cc2nnc(C)o2)C12CCC2 89700,C(C)(C(C)(C)C(=O)NCC(=O)NC1CC1)NC(CC(C)C)=O 89701,Cc1cc(NC(=O)CCN2CCC2)ccc1NC(C1CCCC1n1cccc1)=O 89702,N1(C(c2cnc(CC)[nH]2)C(=O)NCCCC(=O)OCC)CCN(C(C)C)C(C)C1 89703,CC1CCN=C2C=CNC=C2S(=O)(=O)NCC(CCCC2CC2)OCCC1 89704,C1(CNC(C#CC(C)C)=O)CCCC12CCN(C(=O)CC1OCCC1C)CC2 89705,C1(NC(C2(SC)CC(O)C2)=O)CN(C(=O)CCc2ccc(F)cc2)C2(CCC2)C1 89706,N1(C(C(CC)C)=O)CC(CO)C2(C1)CN(C(=O)C(c1cccc(Cl)c1F)(C)C)C2 89707,c1(C(=O)NCC2CCN(C(c3c(N)cc(F)cc3)=O)C2)cc2ccccc2cc1O 89708,CC(C)C(C(C)NC(=O)CCn1cncn1)NC(=O)Cc1ccc(O)cc1 89709,C1(C(N(CCC)C(C)C)=O)CN(C(=O)C(C)NC(C)(C)CC)CCO1 89710,CCC(C(=O)N(C(C)CCNC(c1ccc(S(N)(=O)=O)o1)=O)C)C(F)(F)F 89711,CN1CCC(O)C(NC(C2CCC(NC(c3cnn4c3OCC4)=O)C2)=O)C1 89712,c1(C(N(CCCNC(C(C)c2cncs2)=O)CCO)=O)cc([N+](=O)[O-])ccn1 89713,C1(NC(C2(CC)CCCO2)=O)CC2(C1)CC(NC(=O)CCc1ccc(=N)[nH]c1)C2 89714,CN1CC(C(=O)NCCC2(C(=O)NC(C)(C)C(O)CO)CC2)CCC1=O 89715,C1(C)(c2ccc(NC(CCCn3c(C)ncc3)=O)cc2)NC(=O)NC1=O 89716,c1(-c2nc(C(c3cc(C)nc(N4CCS(=O)(=O)CC4)n3)C)on2)cc(F)c(Cl)cc1Cl 89717,N1(C(c2ccnc(OC)n2)=O)CCN(Cc2cc[nH]n2)C(C(=O)O)C1 89718,C1(NC(CC(CC)O)=O)CN(C(c2cc3c(s2)CCC3)=O)CCC1C 89719,C1(CNC(=O)CN(C2CCOC2)C)COCCN(C(=O)CCOC2CCOC2)C1 89720,C12(C(=O)NCn3cc(C(=O)NC(COC)C)nn3)C3C4C1C1C2C3C41C(N)=O 89721,c1(C(N(CCN(C(c2c(C)noc2N)=O)C)C)=O)cc2c(F)c(F)c(F)cc2[nH]1 89722,CC1(C)CN(C(C2(Cl)CC2)=O)C1C1CCN(C(C2CCS(=O)(=O)N2)=O)CC1 89723,c1(C(=O)NC(CCNC(C(CCC)C)=O)(C)C)cc([N+](=O)[O-])c[nH]1 89724,C1(NC(c2c(C)c(F)ccc2)=O)CN(C(=O)CCCC2CC2)C2(CCC2)C1 89725,CC(C)(CS(C)(=O)=O)C(=O)NCC(CO)NC(c1cnc(N)c([N+](=O)[O-])c1)=O 89726,Cc1cc(F)sc1C(=O)NC1(C(=O)Nc2cnn(C)c2)CCCCC1 89727,Cc1cccc(C(O)CNC(c2cc(C#N)no2)c2ccccc2)c1 89728,Cc1cc(=NCCCNS(C)(=O)=O)[nH]c(N2CCCC(O)CC2)n1 89729,c12cccc(c1)O2.O=C(COC(F)F)NOC1CN(C(=O)Cc2ccno2)C1 89730,c1(OC)ccc(-c2ccccc2)cc1CNCC(O)C1(C)CC1 89731,C=CCC(CC(F)F)NC(=O)COC1CCN(C(=O)C(C2(O)CCCC2)F)C1 89732,Cc1ccn2ncc(C(N3CCC4CC3CN4C(c3ccc(Cl)nc3)=O)=O)c2c1 89733,C(=O)(CCC(CF)CF)NCC1C(C(=O)NCc2cc(C)ns2)CCO1 89734,c1(CC)nc(Cl)[nH]c(=NC2CC(NC(=O)Cc3ccc(C)cc3C)C2)c1Cl 89735,C(C(CC(=O)NC1CC(CNC(N)=O)C1)C1CCC1)NC(C(CC)N(C)C)=O 89736,C12(C(=O)NC3CCN(C(C4(CC)CCOC4)=O)CC3)CCC(N(C)C)(CC1)CC2 89737,C1(C(C)C)CN(C(=O)CC(C)(C)F)CCN1C(=O)CC1CCC(=O)N1 89738,Cc1cc(C(=O)N(C2CCN(C(c3ccc(C#N)cc3)=O)C2)CCO)ccc1Br 89739,C1(CNC(c2cnc(OC)s2)=O)CC2(CCN(C(C3SCCC3C)=O)CC2)C1 89740,N1(C(C(CC2CC2)NC(CCc2ccn(C)n2)=O)=O)CCn2nncc2C1 89741,N1(C=O)CCCCC(C2CN(c3ncccn3)C2)C1.Cc1c2cc(Cl)c(Cl)c1-2 89742,c1(C(C)(C)O)cc2n(n1)CCN(CC(=O)NC1CC3(C1)CC(F)C3)C2 89743,CCC(C)C(C)C(=O)N1CC(O)CC1CNC(C1C2CN(C)CC12)=O 89744,CC(C)CC(O)C(=O)NC(C)CC1CN(C(=O)CCCn2ccccc2=O)C1 89745,C(=O)(CC(C(F)(F)F)NC(c1ccc(C#N)cc1)=O)NCc1c(C)occ1 89746,N1(C(C2CC(C)(C)N(C(C3CCCC(=O)N3)=O)C2)=O)CCC(F)(F)C(O)C1 89747,N12CC=CC(C1)C2=O.C1(C2C(=O)N2)CCCN1C.CC(C)COCCC(C)(C)C 89748,C1(CC)CCC(C(=O)NC2CCCCC2C(=O)NCC(c2ccncc2)O)CC1 89749,c1(C(N2C(C(C)NC(C3C4CC5C(C4=O)C35)=O)CCC2)=O)ccc2c(c1)CCO2 89750,C(=O)(C(C(C)C(C)C)N(C)C)NCCC(=C)CNC(=O)CNC(=O)CC(C)C 89751,c1(C(N2C(c3ccn(C)n3)CCC2)=O)cnc2cnc(Cl)cc2c1 89752,CC1(C)CN(C(c2c[nH]cc(F)c2=O)=O)CC1NC(=O)Cn1ccc(O)nc1=O 89753,c1(C(=O)NC2CC(CC(=O)NCc3n[nH]c(O)n3)C2)cccc(F)c1F 89754,c1(N2C(CNC(CS(CCOC)(=O)=O)=O)CCC2)cc2c(cn1)C(=O)CCC2 89755,N1(C(=O)OC(C)(C)C)CC(c2ccccc2)(NC(C2CCCS2)=O)C1 89756,c1(C(=O)NC(CC)CNC(=O)C(C)(C)N2CCCC2)ccc(Br)cn1 89757,N1(C(CCc2cc(C)sc2C)=O)CCCN(C(c2cc(C#N)c[nH]2)=O)C(C)C1 89758,CCC(C)(CCNC(=O)Cc1ccccc1F)NC(=O)CC1CCCCO1 89759,Cc1ncc(C(=O)NCC2(F)CCN(C(c3cn4c(n3)SCC4)=O)CC2)c(O)n1 89760,C(=O)(C1=CCCCCC1)NC1CCN(C(CC2CC(=O)NC(=O)C2)=O)C1C(F)(F)F 89761,N1(C(CCCC(=O)OC)=O)CC2CN(C(C3CCC(C)CC3)=O)CC2(C)C1 89762,c1(C(N)=O)cccc(C(=O)NCC2CN3CCC23)n1.c1ccccc1 89763,c1(C(N(CC(C)O)CCNC(c2ccc(C3CC3)nn2)=O)=O)cc(Cl)nnc1O 89764,C1(NC(C2CSCN2C)=O)CCN(C(C2CC(C)C2)=O)CC1 89765,c1(OCCC)cccc(-c2cccc(OCC3(C)CC3)c2)c1 89766,CC(C)(C(=O)NC1CCC(CNC(C2(CO)CCCO2)=O)C1)S(C)(=O)=O 89767,c1(C(C(=O)N(CCC)CCNC(=O)Cc2ccno2)N)ccccc1.C(C)=C 89768,CC1(CNC(c2c[nH]c(=N)s2)=O)CCCC1NC(c1cccc(C(F)(F)F)n1)=O 89769,C1(N(C(CCC=CC(C)C)=O)C)CN(C(=O)C(C)CN2CCCCC2)CCC1O 89770,N1(C(CCCOCC=C)=O)CC2CC(NC(c3cnsc3C)=O)CC2C1 89771,N=c1nc(CCNC(=O)C(N2CCCC(C(=O)O)C2)=O)cc[nH]1 89772,C1(C2CCCN(C(=O)C3=CCC(C)CC3)C2)(NC(C=C(CCC)CCC)=O)CC1 89773,c1(C(=O)NCC2OCCN(C(CC3(C=C)CCC3)=O)C2)cc(C#N)c(O)nc1N 89774,Cc1cccc(NC(C23CC2CN(C(c2ccc(CO)cc2)=O)C3)=O)n1 89775,N1(C(C2(CC)CC(C)(C)C2)=O)CC(C)OC2(CCN(C(=O)CSC(C)C)CC2)C1 89776,C(=O)(C1=NOC(C)C1C)NC1(CN(C(c2c(C)ccnn2)=O)C)CC1 89777,N1(C(c2ncncc2Cl)=O)CCN(C(c2nc(Cl)cs2)=O)CC(O)C1 89778,N1(C(C(c2cnn(C)c2)SC)=O)CCc2ccccc2C1CNC(C1(C)CC1)=O 89779,C1(=O)C(CC(C)C)N1.Cc1nsc(Br)c1C(NOC(=O)CN1CCCCC1)=O 89780,C(C(C(=O)NCCC(C)CO)C(C)(C)C)NC(C(CC)(C)CC)=O 89781,C1(NC(CC(C=C)(C)O)=O)CC2CCC(C1F)N2C(c1ccccc1F)=O 89782,c1(C(N(CC(C)NC(=O)C=Cc2ccoc2)CC)=O)cnc2[nH]ncc2c1 89783,C1(NC(C=CC(C)NC(C2CC(F)(CSC)C2)=O)=O)COCC1F 89784,N1(C(C2C(CC)OCC2)=O)CC2CCC(C1)N2C(C1CCC(C)(C)O1)=O 89785,C1(CNS(c2cccc(OC)n2)(=O)=O)CCCC2(CC(C(=O)O)C2)O1 89786,C1(C(CNC(CN(CC)CC)=O)NC(C2CN(C)C2)=O)CCCCC1 89787,C(=O)(C1Cc2ccccc21)Nc1cccc(C)c1C(=O)NC(COC)(C)CO 89788,CCC(C)CCC(=O)N1CCOC(CNC(c2ncoc2-c2cnn(C)c2)=O)C1 89789,Cc1nn(C)c2cc(NC(C3CC4CC4N3C(c3cc[nH]c3)=O)=O)ccc12 89790,C(Cc1cnc[nH]1)(C(=O)NCCSC(F)F)NC(=O)Cc1ccon1 89791,c1(C(=O)NCCCC(C)NC(CCC=C=C)=O)cc2c(nc1O)CCCC2 89792,C1(CC(=O)N(C2CN(C(C(C)CSC(F)(F)F)=O)C2)C)CCCC1(F)F 89793,Cc1cncc(C=CC(N2CCCC2CCNC(=O)CC2CCC3CC3C2)=O)c1 89794,c1(C(N2CCCC(CNC(c3sccc3I)=O)C2)=O)cccc(F)c1I 89795,Cc1cc(C(=O)NCC(C)(C(F)(F)F)NC(=O)CN(C)C)cc(C)c1N 89796,N12CC3CCCC3CCCCC1c1ccc(c[nH]nnn1)C2=O 89797,c1(N2CCC=C(C)C2)[nH]c(=NCCc2cccs2)nc2c1ncn2C1CC1 89798,C1(CNC(C(C(C)C)OCC)=O)CN(C(c2snnc2C)=O)CCCO1 89799,c1(C(N2CC(C)C(CNC(=O)COc3cn[nH]c3)C2)=O)nc2ccc(Cl)nn2n1 89800,N1(C(CC2CC(C)N(C(C3CCOC(=O)CC3)=O)C2)=O)CCC2(CCC(O)C2)C1 89801,N1(C(c2c(C)cnnc2)=O)CCC(C)(C)C(CNC(C2CCOC(C)(C)C2)=O)C1 89802,N1(C(C(COC)O)=O)CCC(C2CCN(C(=O)C(C)(C)C(C)(F)F)C2)CC1 89803,CCCC(C)(C)CC(=O)N1CCC1(C)CC(=O)NC(c1cn(C)nc1C)C 89804,c1(C(N2CC3C(NC(C(F)=CCC)=O)(CCC3)C2)=O)c(C)[nH]c2ccc(Cl)cc12 89805,C1(CC)CN(C(c2cscc2CC)=O)CCN1C(=O)C=Cc1nccs1 89806,c1(C(=O)NC(CCOC)CNC(C2(C#N)CC2)=O)ccc(SC)c(OC)c1 89807,c1(C(N(C)CCO)=O)cccc(S(=O)(=O)N(C(C2CCCOC2)(C)C)C)c1 89808,N(C(=NCC(C)(C)CC(=O)OC)N1CCN(C)C(=O)C1)C(C=C)C 89809,c1(NC(N2CC(C(C)C)OCC2)=O)ncc2c(n1)CCNC2=O 89810,C1(C(=O)NCCC(C)NC(=O)C(C)(C)Nc2ccccn2)CC2CC1CC2(F)F 89811,c1(C(=O)NCCC(CCNC(C(C)N(C)C)=O)C)cnn2c1S(=O)(=O)NCC2 89812,c1(C(=O)NCCC2CC(NC(CC(C)(C)OC)=O)C2)cc(F)cc(N)c1F 89813,C1(NC(c2ccoc2)=O)CCC2(CCCN(C(C3CCCOCC3)=O)C2)C1 89814,c1(CC(C)NC(=O)Cc2cccc(Cl)c2Cl)ccc([N+](=O)[O-])nc1 89815,C1(NC(CCN(C(COCCC#C)=O)C)=O)CC2CC2C1 89816,c1(C2(NCC(C3CCC(O)CC3)(C)C)CCC2)cccc(F)c1 89817,CCC(C#N)(CC)C(=O)NCC1CCN(C(=O)C(c2ccccc2)OC)CC1 89818,C1(F)(C(=O)NCC2N(C(C3CCCN(C)C3)=O)CC2)CCC(F)(F)CC1 89819,C=CCC(CC(C)C)C(=O)NCC1CCCC1NC(c1cc(COC)[nH]n1)=O 89820,C=CC(C)(C)CCCNC(=O)C(CC1CCOCC1)NC(=O)C(F)CC 89821,C12(C(C)=O)CCC(C(=O)NCC3(NC(C4CC(C)=NO4)=O)CCOC3)(CC1)CC2 89822,c1(C(N2C(CNC(CN=S(C)(C)=O)=O)CC2)=O)cc(Cl)ccc1[N+](=O)[O-] 89823,C#CC1CC2(CC2)CN1C(c1cc(CCN(C(=O)C(Cl)Cl)CC)on1)=O 89824,C1(C(=O)NCC(CC)NC(C(CO)CCCCCC)=O)CS(=O)(=O)CC12CC2 89825,C(=O)(CCC(C)(C)NC(C1C(C)C1C)=O)NC1(CC(=O)OC)CC1 89826,c1(CC(=O)NCC=CCNC(C2CCC(CO)CC2)=O)ccccc1Br 89827,N1(C(C2CCC(=C)CC2)=O)CC2CCOCC2(NC(=O)CCC(C)C)C1 89828,C(C(C)(O)CNC(=O)C(C)Cc1cnn(C)c1)NC(COCCC=C)=O 89829,C=CC(CCC)CC(=O)N1CC(NC(=O)C(c2ccc(F)cc2F)(C)C)C(F)C1 89830,c1(C(=O)NCC(CNC(C2C(CC)CC2)=O)O)nccc(C)c1N 89831,c1(CN(CC(=O)NC(c2ccc(-c3cccnc3)cc2)C)C)ccc(Br)cc1F 89832,N1(C(C=O)=O)CC(N(CC(F)(F)F)CCO)C2(CC2)C1.CC(C(C)C)=C1CCC1 89833,c1(Oc2ccnc(NC(=O)NC3CC(OC)C34CCC4)n2)ccc(C)c(CO)c1 89834,C=C(C)CCC(C)NC(=O)CC1CN(C(=O)CN2CCSCC2)CCO1 89835,c1(NC(c2c(Br)cn(CC)n2)C)cc(NC2CC3CCC2CC3)ncn1 89836,CC(CNC(=O)CCC1(NC(=O)CC2(N(C)C)CC2)CCC1)C(C)(F)F 89837,c1(NC(C(N2CCC(Oc3ccc(C)cc3)C2)=O)=O)c(F)cc(I)cc1F 89838,c1(C(N2CCCCC2c2cccn2C)C(=O)NCC)nc(Cl)c(C)cc1[N+](=O)[O-] 89839,C1(NC(CNC(C2C(C)C2)=O)=O)CCC2(CC1)CN(CC1CCCCS1)CCO2 89840,CCCCC(C)C(=O)NC1CCCCCC1C(N1CC[Si](C)(C)CC1)=O 89841,N1(C(CCC#C)=O)CCCCC(C(=O)NC2CC23CCCCC3)C1 89842,S(=O)(=O)(c1cccc2ccccc12)N1C(C(C)(O)CO)COCC1 89843,C(=O)(C(O)CC(F)(F)F)NC1CC2(CN(C(c3c(C(C)=O)cc(F)cc3)=O)C2)C1 89844,N1(C(C(C)OC)=O)CC2(CCCCN2C(c2cnc3c(c2)CCCC3)=O)C1 89845,N1(C(CC(=O)OCC)=O)CCCC(CC)C1C(N1CCCC(OC)C1)=O 89846,N1(C(c2ncc(Cl)cc2F)C(=O)NC(C)(C)C)CCC12CCSCC2 89847,c1(N(C(C)C)C)ccc(C(C(=O)NCCC#N)N(C)CC2CCCCC2O)cn1 89848,c1(CNC(=O)CC2CCN(Cc3ccc(C#N)s3)C2)cnc2ccc(F)cn12 89849,C1(N(C)C(C2CC(F)(CF)C2)=O)CCCN(C(=O)COCCCF)C1 89850,c1(C(C(=O)N(C(C)C(c2cnn(C)c2)=O)C)=O)ccc([N+](=O)[O-])cc1 89851,C(=O)(C(C)C1=CCCC1)N1CC(NC(c2cc(SC)oc2)=O)C1 89852,C1(CC)CN(C(C2(SC)CCOCC2)=O)CCN1C(c1occ2c1CCC2)=O 89853,CC1(NC(c2cc(Cl)cc(Cl)c2)=O)CCC(NC(C2CC(C)(O)C2)=O)CC1 89854,c1(CC(=O)NC(C)CNC(C2CCCCN2C)=O)csc2ccc(Cl)cc12 89855,c1(C(N2CCC(C)(NC(c3c(OC)cccc3)=O)C2)=O)nc(Cl)ccc1F 89856,Cc1c(C(=O)NCC2CCC(NC(C3CCCN(C)C3)=O)C2)nnn1C(C)C 89857,Cc1c(C(=O)NC(C)C(C)NC(c2ccc(F)o2)=O)cncc1Br 89858,N1(C(c2c(C)nc(-c3ncc[nH]3)s2)=O)CCC(C)C(NC(=O)C(F)=C2CCC2)C1 89859,C1(C(N(CCN(C(=O)C(F)(F)c2ncccn2)CC)CC)=O)CCCC(C)C1 89860,C(C1C(C(=O)NCCn2cc(CCC3CCCCO3)nn2)C1(C)C)=C(C)C 89861,C1(CNC(c2c(C)cno2)=O)N(C(C2CCN2C)=O)CCC1(C)C 89862,c1(CC(=O)N(C2(C)CN(CCOC)C2)c2ccccc2)ccc(Cl)c(C)c1F 89863,c1(C(=O)NCCCCN(C(C(C(C)C)OC)=O)C)ncn2c1COCC2 89864,C1(C(C)NC2(CN3CCCC3)CSC2)CCN(C)CC1 89865,C12(C(=O)NCCCCC3(NC(CCCC)=O)CC3)CCC(CC)(C1)OC2 89866,C(C1=NOC2CN(C(=O)CCC3OCCO3)CC12)NC(CCCN=[N+]=[N-])=O 89867,C#CCC(C)(C(=O)N1CC(F)CC(F)C1)NC(=O)CC1CSCCO1 89868,C1(NC(C(CC)SC)=O)CCCCC12CCN(C(C1(C#N)CCCC1)=O)CC2 89869,C1(C(=O)NCCCCCCC2CC2)COCCN(C(=O)CNc2ccccc2Cl)C1 89870,C1(C(=O)NCC2(F)CN(C(c3c(NC)nccc3)=O)C2)CCc2c[nH]nc2C1 89871,N1(C(C)=O)CC2(CCCC(CNC(c3cnsc3C)=O)O2)C1 89872,c1(C(=O)O)ccnc(C(F)(F)F)c1F.c12ccc(cc1)C(=O)NC1(CC1)NC2=O 89873,c1(N2CCC(CNC(c3ccc(C(C)C)cc3)=O)C2)ncc2ccsc2n1 89874,C1(CC(=O)NCC2(F)CC(CNC(C(C)c3ccsc3)=O)C2)C(C)(C)C1(C)C 89875,CCC(CC(=O)N1CCC(C(=O)NC(C23CCC(CO2)C3)C)C1)C(C)(C)C 89876,CC1(C)COC(C)(c2cn(CCCC(=O)NC3CCCC3N=[N+]=[N-])nn2)CO1 89877,c1(CC(=O)NCC2C3CN(C(C=C(C)C(F)F)=O)CC32)ccc([N+](=O)[O-])cc1F 89878,N1(C(C(CC)=CC)=O)CC2CC2C1C(N1CC(NC(C)=O)C1)=O 89879,c1(CC)nocc1C(=O)N(CC(CNC1CC(C)(C(=O)OC)C1)C)C 89880,CCC(c1ccc(C)cc1)=CC(=O)Nc1cncc(OC)c1 89881,c1(OC)cccc(CC(=O)NC(C2(O)CCN(C(=O)CP(C)(C)=O)C2)C)c1Cl 89882,C(=O)(CCC(C)(C)C(=O)NCC1CCCCC1C(F)(F)F)OCC 89883,C#CCC1C(=O)NN2CCCC2C(=O)N1.c1(SCCOC)cn[nH]c1 89884,N1(C(c2c(N)c(Br)cc(F)c2)=O)CCc2c(Cl)cccc21.C1C(=O)N1 89885,N1(C(CN2C(C)CCCC2)=O)CCC2CCC12CNC(=O)CSC(F)(F)F 89886,c1(CC=C)cccc(C(=O)N(C(C)C(=O)NCC2=NOC(C)C2)C2CC2)c1 89887,c1(C(C)=O)cnc(N2CCC(F)(CNCc3csc(Br)n3)C2)nc1 89888,Cc1cc2c(cc1Cl)C(N(CC(C)C)C(C1CCC(c3ccccc3)O1)=O)CO2 89889,C1(C2CN(C(C=C(COC)C)=O)C2)CCN(C(C2C=CC2COC)=O)C1 89890,Cc1ccc(C(=O)NC2CCCC(NC(=O)C(F)(F)c3nccn3C)C2)n1C 89891,C1(NC(=O)CCN2CCOCC2)CN(C(C23CCC2C3)=O)CC1O 89892,C1(CNC(C(C)Cc2cnn(C)c2)=O)(NC(=O)C(C)OC2CCOC2)CC(F)(F)C1 89893,Cc1nc(O)ccc1C(=O)NC(C)CCNC(c1ccc(-n2cccn2)cc1)=O 89894,c1(C(=O)NCC(CC)NC(c2snc(Cl)c2Cl)=O)cnc(OC)cn1 89895,c1(NC(N(CC=C)CC=C)=O)ccc(OCCCCc2ccc(Cl)s2)cc1 89896,C1(CC)(CC)CC(NC(=O)CC2CCC(=O)N2)CN1C(=O)Cc1ccsc1Cl 89897,S(=O)(=O)(c1ccsc1)N1CC(F)(C(N2CCC(O)(c3cc[nH]n3)C2)=O)C1 89898,CC1C(NC(=O)CCn2cccnc2=O)CCCN1C(c1ccc(C#N)s1)=O 89899,N1(c2ncc(C)cn2)CCN(Cc2cnn(C)c2C)C2CC12 89900,Fc1ccc2scc(CNC3CCCCC3c3cccc(Cl)c3)c2c1 89901,C1(NC(CC2CCN(C)C2)=O)CC2CC(C1)N(C(=O)CCC1CCCN1C)C2 89902,N1(C(c2cc(C(C)C)on2)=O)CCCCC1CNC(=O)CCN1CCCC1 89903,c12cc(ncn1)C2.N1(C(N)=O)CC(CNC(=O)Cn2cc(C3CC3)cn2)C1 89904,CC#CCCC(=O)N1CCC(CC(N2CC(C)C2)=O)CC1 89905,CC(C)CC(CNC(c1csc(O)n1)=O)C(=O)N(CC(O)CF)C 89906,N1(c2n(CCC#C)c(C(CC)N(C)C(=O)OC)nn2)CCC2(CCOCC2)C1 89907,N1(C(CCSCC)=O)CCC(C(C)(C)C)CO1.C1(=O)C(CCO)N1 89908,c1(CC)ccc(F)c(C(N2CC(NC(c3cn(C)nc3COC)=O)C2)=O)c1 89909,c1(C(=O)NC2CC(CC)(CC)N(C(=O)CNC(C)=O)C2)cc2cnc(Cl)cc2s1 89910,C1(NC(=O)Cc2ccc(Cl)cc2)CC2CC1N(C(c1cnc(N(C)C)s1)=O)C2 89911,c1(C(=O)NC2CCC(CNC(c3coc(Br)n3)=O)C2)nc(O)[nH]c(=O)n1 89912,C1(C(=O)Nc2cnn(C3C=CCC(SCCC(C)(C)CO)C3)c2)(OC)CCCCC1 89913,c1(CC=C)ccccc1C(=O)NC(C1CC(NC(C2OCCC2C)=O)C1)C 89914,c1(OC)cc(C(C)CC(=O)N(C)CCN(C)C(N2CC3CC3C2)=O)ccc1C 89915,C(CCC(CCC)NC(=O)Cn1cccnc1=O)NC(C=C(CCC)C)=O 89916,c1(C(N2CC(O)CC2CNC(C23CCCC2CCC3)=O)=O)ccc2c[nH]nc2n1 89917,Cc1ncc([N+](=O)[O-])cc1C(=O)NC1CN(C(=O)CC(C)N(C)C)CC1C 89918,CN1C(=O)CCCC1C(N1CC(F)(F)CC1CNC(=O)COC(F)F)=O 89919,C(CCC(O)C(=O)NCCN1CCOCC1C)NC(c1cc(C)oc1)=O 89920,C(=O)(CS(=O)(=O)N1CCC(O)(C(=O)Nc2ccc(SC)cc2)C1)OCC 89921,C(C)(C)(CCCC(=O)NC(c1nccc(C)n1)C)NC(c1ccc(C=C)cc1)=O 89922,C1(CNC(=O)COCCF)CCCCC1NC(C1CCCOC1c1cn[nH]c1)=O 89923,c1(C(N2CCC(C)(C(=O)OCC)C2)C(=O)NC)cc(C2OCCO2)ccc1Br 89924,C12(OC)CN(C1)C(=O)Cn1cc(nn1)C2.C1(C(=O)OC(C)(C)C)CC=CCC1 89925,N1(c2cncc(C#N)n2)CCC2(CCC(CNC(C3CC=CCC3)=O)OC2)CC1 89926,Cc1cc(C(N2CCOC(C(N3CCOCC3CN(C)C)=O)C2)=O)ccc1C#N 89927,N1(C(c2c(NC(C)=O)cncc2)=O)CC2CCCC2(NC(=O)C=CC2CCCC2)C1 89928,CCS(=O)(=O)c1ccc(F)c(C(=O)NCC2(F)CCC(NC(=O)C(O)CF)C2)c1 89929,CC1CC(CCNC(c2cc(C(C)(F)F)n[nH]2)=O)CCN1C(=O)CCNC(N)=O 89930,c1(OC)cc(C(=O)NC(C)(CNC(c2ccc(C)cc2C)=O)C(C)C)c(F)cn1 89931,Cc1cccc(NC(C)CCNC(=O)OC(C)(C)C)c1C(F)(F)F 89932,c1(C(c2nnnn2C2CCOC2)NCCC(=O)NC)cc(OC(C)=O)nc(Cl)c1 89933,C1(NC(c2ccc(C)c(C)n2)=O)CC2CC1CN(C(=O)C=Cc1csc(C)n1)C2 89934,C12(C#CC(=O)O1)COC2.C1(C(=O)NCC)(N(C)C(=O)OC(C)(C)C)CC1 89935,C1(C(=O)NCC2C(NC(c3ccc(C(F)F)s3)=O)CC2)CC(F)(F)C1 89936,CC1CCC(C)N(C(=O)CCOC2CN(C(c3cc[nH]c(=N)n3)=O)C2)C1 89937,c1(C(=O)NCC2(C)CN(Cc3ncn4ccccc34)C2)ccc2nccnc2c1 89938,c1(CNC(C2N(C(c3c(C)ocn3)=O)CCCC2)=O)ccc(F)c(Cl)c1 89939,C(C(C)C(F)C(=O)NCC(F)F)NC(C=C=C(C)C)=O 89940,c1(CC)conc1CC(=O)N(CCCNC(=O)CC1COC(=O)N1)CCO 89941,N1(C(C(c2ccc(C)cc2)F)=O)CCC(O)C(C(=O)NCC2CCN(C)CC2)C1 89942,C12=NC=CC(=NCCNCC1)N2.C(c1cccnc1)=CCN(C(CC)C)C 89943,C1(NC(CS(C)(=O)=O)=O)C2CCN(C(=O)Cc3coc(-c4cccs4)n3)CCC12 89944,C1(c2nc(C(C)OCC)nn2-c2ccc(Br)nc2)CCc2nncn2C1 89945,c1(C(=O)NC(C(C)C)CNC(c2nnc(S)n2C)=O)ccc2cncn2c1 89946,c1(COC)cccc(OCC(=O)N(CCCN(c2ccccc2)C)C)c1 89947,C1(CCOC)(NC(=O)Cc2csc(COC)n2)CCN(C(=O)C(O)C(C)C)C1 89948,CC#CC1CCN(C(=O)COC2CC(NC(c3cc(CC)sn3)=O)C2)C1 89949,C1(NC(=O)C2CC2)CC(C)N(C(=O)CC(=O)Nc2cnc(C(=O)OCC)s2)C1 89950,Cc1cc(C(=O)NC(C)CN(C)C(C23CC(CO2)C3)=O)c2c(c1)C(C)CCN2 89951,N1(C(CC=CC(C)(C)C)=O)CCOCC1CCCNC(=O)CSc1n[nH]c(O)n1 89952,c1(OC)ccc(C(=O)N(C(C)CNC(c2ccc(C(F)F)cn2)=O)C)c(F)n1 89953,C1(NC(C(C=C)O)=O)CCN(C(=O)C(C)NS(=O)(=O)CC)CC1(C)C 89954,C(=O)(C(C)(C)CC(=O)OC)NCCC1CN(C(C2C(C(N(CC#C)C)=O)C2)=O)C1 89955,c1(C(=O)NC(CCNC(CCCCCC)=O)C)c[nH]c2c(C)cccc12 89956,C(C(F)C(=O)NCC(C)F)C1CN(C(COC(C)=O)=O)C1 89957,C1(CC)CCCC(CNCc2cc(Br)cs2)C1 89958,N1(C(C2(NC(CCOC)=O)CCCC2)=O)CCC(NC(=O)CN2CCC2C)CC1 89959,c1(OC(c2c(C)cc(F)c(Br)c2)=O)nc(O)c2cnn(C)c2n1 89960,C(=O)(C(C(C)C)NC(C1CCC(=O)C1)=O)N(C1(COC)CC1)C 89961,C(=O)(C(C)(CNC(=O)COCCOCCO)CC)NC1CC(SC)C1 89962,CC1(C)CCC(C(=O)NCCC2(O)CN(C(C3CCC34CCC4)=O)C2)COC1 89963,S(=O)(=O)(c1ccc(S(=O)(=O)NCCC)cc1)N(CC(C)(C)N)CC#C 89964,C1(C(N2CCC(CCNC(c3c(OC)c[nH]n3)=O)C2)=O)CCN(C)CC1 89965,C1(C(N2CCCC(CC)(NC(c3cccn3C)=O)C2)=O)CCCC1P(C)(C)=O 89966,N1(C(C(F)OC)=O)CCc2ccccc2C1CNC(c1nccn1C)=O 89967,C1(N(C)C)CCCN(C(C23CC(CCNS(=O)(=O)Cc4ccccc4)(C2)C3)=O)C1 89968,N1(C(c2cccc(CC)c2)=O)CCC2CCC(C1)N2Cc1ccc(C(=O)OC)cc1 89969,C1(C(=O)NC(C(C)C)(C)CNC(c2cnc[nH]2)=O)CCC2(CCC2)CC1 89970,c1(CCC)ncoc1C(=O)NC(C(N1CCC(CF)C1)=O)C1(C)CC1 89971,Cc1cc(C#N)cnc1C(=O)N(CC(C)CNC(C1CCCC(O)C1)=O)C 89972,c1(C(=O)NC23C(CN(C(CC(C(C)C)O)=O)C2)CCC3)ccc2c(c1)COCC2 89973,CC1(C)C=C(C(=O)N2CC(CNC(C3C4COCC34)=O)CC2(C)C)C1 89974,c1(OCC)nc(N2CCC(C)C(NC(c3cc(C)c(C)s3)=O)C2)ncc1Cl 89975,C1(C)(CNC(c2cccc(C)c2)=O)CCCN(C(=O)Cc2c(O)ncnc2O)C1 89976,C1(O)(CCNC(=O)COCCF)CCN(C(c2ccc(C(F)(F)F)o2)=O)C1 89977,Cc1cc(=O)ccn1CC(N1CC(F)(F)CC1CNC(=O)CN(CC(C)(C)C)C)=O 89978,Cc1cc(C(N2CC(CC(C)NC(=O)Cn3cc[n+](C)c3)C2)=O)[nH]c1C 89979,C(CC(C)(C)C(=O)NCC1CC(NC(c2ccc(C(C)C)nc2O)=O)C1)OC 89980,C1(C)(C2CCN(CCNC(=O)C(=O)NC)C2)NC(=O)NC1=O.C12CCCC1CN2.CO 89981,C(=O)(C1=NN(C)C(=O)CC1)NC1CC2CC(NC(c3ccc(OC)s3)=O)C1C2 89982,c1(C(C)C)cc(=NCC2CCCN(C(=O)CSc3ccccc3C)C2)[nH]c(Cl)n1 89983,N1(C(c2n(C)nnc2)=O)CC2CC(NC(=O)CCc3c(Cl)cncc3Cl)C(C2)C1 89984,C1(C(=O)NC2CC(C)CN(C(=O)Cc3cnsc3)C2)Cc2ccccc2C1 89985,N1(C(CCNC(=O)OC)=O)CC(C(=O)N(CC(C)O)CCF)CC1(C)C 89986,CCC(C)(O)C(=O)N1CCC(N2CCN(C(=O)Cc3ncc(C)o3)CC2)C1 89987,N1(C(CCCCCC)=O)CC2(C1)CN(C(=O)CC1CCC1OC)CC2CO 89988,CCC(C)CC(C)C(=O)NCCN(C)C(c1ccc(CN(C)C)nc1)=O 89989,N1(C(COCC=C)=O)CC(NC(C2CC2CF)=O)C(C)C1 89990,N1(C(COCCC(C)C)=O)CCC(C)(C)C(NC(=O)CC2CCC(=O)N2)C1 89991,O=[N+]([O-])c1cccc2[nH]nc(-c3nc(-c4cccc([N+](=O)[O-])c4)no3)c12 89992,c1(N2CCOCC(CNC(CCSC)=O)C2)ncc([N+](=O)[O-])cc1Br 89993,N1(C(C2(C#N)CCCC2)=O)CC(C2CN(C(C3CC(=C4CCC4)C3)=O)C2)C1 89994,c1(C(N2CC3N(C(C(CCSC)N(C)C)=O)C3C2)=O)c(C)ncnc1C 89995,N1(C(c2c(CC)con2)=O)CCOCC1CC(=O)NCC(C)CN(C)C 89996,c1(C(=O)NCC(C(=O)OC)Oc2cccc(F)c2)ccn2c1CSCC2 89997,C1(C(=O)NCc2cn(C(C)C)cn2)(N)CC1(C)C.N1(C(C)C(=O)CC)CCOC1=O 89998,C1(C)(COC)CC(NC(=O)CC2CC2)CN1C(c1c(Cl)cccc1Cl)=O 89999,C1(OC)CC(CNC(=O)Cc2cncs2)(NC(=O)COC(F)F)C1 90000,n1(CC(=O)NC(C)CC(C)NC(=O)CCCn2cccc2)nnc2c1CCCC2 90001,Cc1ccc(C(C)C)cc1C(=O)N(C(C)CCNC(=O)C(c1cnn(C)c1)O)C 90002,CON(CCC(=O)N1CC2C(C1)C2(F)F)C(=O)C1COC(=O)N1C 90003,N1(C(C(COC)C)=O)CCN(C(=O)CNC(c2nccc(C)n2)=O)CC1 90004,N1(C(CC)=O)CCC(C(=O)NCc2cnn(C)c2)CC1C 90005,C1(C(=O)NCC2(F)CN(C(C3CCCCCC3)=O)C2)CCC2(CCC2)OC1 90006,c1(C(=O)NCC(C)C(=O)NC(C)(C)CCCF)ccc(C#N)cn1 90007,C=C1CCN(C(C2CC(OC(C)=O)C2)=O)C(C(=O)NC(C)C(F)(F)F)C1 90008,c1(CC(=O)NC2CC(F)(CNC(=O)Cc3cnoc3)C2)c[nH]c2cccc(F)c12 90009,c1(C(=O)NC(CCCNC(C(CC)N2CCCC2=O)=O)C)cnc(C(N)=O)cn1 90010,CC1OC(=O)NC1C(=O)NCC1CCCCN1C(c1cn(-c2ccccc2)nn1)=O 90011,c1(CCC(N2C(C)CN(C(C3CC3(Cl)Cl)=O)CC2)=O)nc2cnccc2[nH]1 90012,c1(C(=O)NCCN(C(=O)CCC2(C#N)CCC2)CCC)cncc(C(N)=O)c1 90013,Cc1ncc(Br)cc1C(N1CC2C(C(=O)Nc3cc(C(=O)N)no3)C2C1)=O.C(N)=O 90014,C12(C(=O)NCC3CCN(C)C3)CC(CO1)N(C(=O)CC1CCCC1)C2 90015,C1(CC)CCN(C(=O)CCCC2CC2C)C(C(=O)NCc2nnnn2C)C1 90016,C1(C(N(CC(C)NC(=O)CC2CNC(=O)C2)C)=O)CCC(=O)N(C)C1 90017,CON1CC(C(N2CCN(C(=O)COc3nscc3Br)CC2)=O)CC1=O 90018,c1(C(C)C(=O)NC2CCCCC2NC(=O)CSCCCO)cccc([N+](=O)[O-])c1 90019,C1(C(N2CC(N(C(=O)CCC3CCC(C(N)=O)O3)C)C2)=O)CCOC(C)(C)C1 90020,c1(CN2CCC(F)(C(N3CCC4COCC4C3)=O)C2)c[nH]c2ncc(Br)nc12 90021,C(C1CCCCCC1)=CC(=O)N(C1CCN(c2cccnn2)C1)C.C1CCC1 90022,c1(NC(C)CCCC(F)(F)F)cc(=NCc2nc(Cl)cs2)[nH]cn1 90023,C(=O)(CCC1=CCCCC1)N1CCC(C)(C=O)CC1.C1(CCC=O)CCC(=O)N1 90024,N1(C(CCOC(C)C)=O)CCCC(NC(C2CC(=O)CS2)=O)C1 90025,C1(NC(CCCC#C)=O)CCN(C(c2ccc(C(C)C)nc2)=O)C(C)C1 90026,CN1CC2CCC(C1)N2C(C1CCCCN(C(=O)Cc2ccon2)C1)=O 90027,CP(C)(=O)c1cccc(C(=O)N=c2[nH][nH]cc2Br)c1 90028,C1(CC(N)=O)(NC(CC2N(CC)CCC2)=O)CCN(C(=O)CCC2CC2(Cl)Cl)CC1 90029,c1(C(=O)NCC(CC)NC(=O)CCC(C)CC)nccc2[nH]nc(C(C)C)c12 90030,N1(C(C(CC)(C)CO)=O)CC23CCCC2(C1)CN(C(c1c[nH]cc(C)c1=O)=O)C3 90031,c1(SC)cc(C(=O)N(C(C)CNC(c2cn(C(C)C)cc2C)=O)C)nn1C 90032,C(=O)(C1=CCc2ccccc21)N1C(CNC(C2=CC(C)(C)C2)=O)C(C2CC2)CC1 90033,N1(C(c2c(C)nc(CC)o2)=O)CCC(C)(C)C1C(=O)NCC1CCCN(CC)C1 90034,C1(=CC(=O)N(C2CC(NC(C3CCC(OC)C3)=O)C2)C)CCCCCC1(F)F 90035,N1(C(C(CCC)CC2CCCC2)=O)CC2(CCN(C(=O)Cc3cccn3C)C2)C1 90036,n1(CC(=O)OCC)nc(C)c([N+](=O)[O-])c1NCC1CC(OC)C1 90037,N1(C(c2nc(C)nn2C)=O)CC(C)(CNC(=O)C=CC(F)(F)F)CC1(C)C 90038,CCCC(C)(C)C(=O)NCC(=O)NCCC1(C)CCC(O)CC1 90039,C(=O)(C(C)(C)CCC#N)N1CC(CNC(C(CC)N2CCCC2=O)=O)C(C)C1 90040,c1(C(=O)NC(C)CNC(C2CCC2(F)F)=O)ncn2ccccc12 90041,c1(OCC)cnc(N2CCC(C3CCCN3C=O)CC2)cn1.C1(C(=O)OC)CC12CC2 90042,c1(C(N2C(COC)CN(C(=O)Cc3cccs3)CC2)=O)c(Cl)nc2ccccn12 90043,CC1(C)CN(C(C2CC3CCC3C2)=O)CCN1C(c1cc(Cl)c(Cl)c(Cl)c1)=O 90044,N1(C(Cc2c(CC)csc2)=O)CCC(NC(c2scc(C)c2Cl)=O)C1C 90045,CC#CCC(C)N=c1[nH]c(=NCC2(C3CC3)CC2)[nH]c2c1CCCCC2 90046,CC(C(=O)NCC1(F)CC(NC(=O)Cc2cc[nH]c2)C1)C(C)(F)F 90047,c1(CC(=O)NC2CCC(NC(=O)C(O)C3CC3)C2)ccnc(O)c1 90048,C(=O)(C(C)(C)N=[N+]=[N-])N1CCC(C=C)(C(=O)NCCCOCC#C)C1 90049,CC1CC(CNC(c2ocnc2-c2ccccc2)=O)CN1C(C1CC(=O)N1)=O 90050,Cn1cc(N)c(C(=O)NC2CCC2NC(c2ncsc2Br)=O)n1 90051,C1(NC(c2cc(C(C)=O)on2)=O)CCC2(CCCN2C(=O)C2=CCCSC2)CC1 90052,C(=O)(C(C(C)(C)C)NC(C)=O)NC12CC(NC(C3(OC)CC3)=O)C(OC1)C2 90053,C(C(C)C(=O)N(CCCNC(c1sccc1Cl)=O)Cc1ccccc1)OC 90054,c1(CC)ccc(O)cc1O.C12(CC)CCCN1CC(=O)NC2=O 90055,C(N=c1cc[nH]c(=NCCn2cc(Br)cn2)[nH]1)C1(C)CC2CC2C1 90056,c1(C(N2CC(C(N3CC(c4nc[nH]n4)C3)=O)CC2CO)=O)cnc(O)cc1O 90057,CC1Cc2cc(Br)ccc2N(C(=O)Cc2cn(C)nc2C(F)(F)F)C1 90058,N1(C(C(=O)NC2CC(CCC)C2)=O)C2(CCCC2)OCC1CC#N 90059,N1(C(c2c(C)cco2)=O)CC(NC(C2CC2c2cnc[nH]2)=O)C(C)(C)C1 90060,C(C(C)(C)C(=O)NC1CC2(C1)CC2C(N1CCC(F)(C(N)=O)C1)=O)OCC 90061,C(=O)(C1=CCC2(COC2)OC1)NCC1C(CNC(=O)Cc2ccon2)C1 90062,c1(C(=O)NCC2N(C(C3C(=C)C3)=O)CC=C2)cc(O)ccc1[N+](=O)[O-] 90063,C1(NC(=NCC)NCC2CC(=O)N(CC(F)(F)F)C2)CCC2(CCCCC2)C1 90064,CCC(C)CC(C(=O)NCCC1NC(=O)NC1=O)NC(c1cc(F)ccc1F)=O 90065,c1(C(=O)NC(CC)(C)CNC(=O)Cc2ccc(O)c(C)c2)cc(F)cc(F)c1F 90066,CC(C)C(O)C(C)C(=O)NCC1(C)CCN(C(C2(CC(F)F)CC2)=O)C1 90067,C(C)(C(C(C)C)NC(c1cn(C)[nH]c1=N)=O)NC(COC(CC)(C)C)=O 90068,c1(NC(C2(C)N(Cc3ccc(C#C)s3)CC2)=O)ccc(F)c(C(N)=O)c1 90069,C(CCC(=O)NC(c1nocc1C(=O)N(c1ccccn1)C1CC1)C)C1C(C)C1 90070,N1(C(C2(OCC)CCC2)=O)CCCCC1CN(C)C(c1csc(C(C)(C)C)n1)=O 90071,c1(C(N(C(CNC(c2ncc(C)c(C)c2)=O)C)C)=O)cc(Br)c(O)nc1C 90072,C1(C2CCCN(C(=O)Cc3nncn3C)C2)(NC(COCCC(C)C)=O)CC1 90073,C(CCCCCN=[N+]=[N-])NC(CCC1CCN(C(C(C)NC(=O)NC)=O)C1)=O 90074,c1(OC)ncccc1C(=O)NCCCCC1CCN(C(c2ccoc2)=O)CC1 90075,C1(NC(C=CC)=O)CCC2(CCN(C(=O)CC3CCC(C)C3)C2)C1 90076,c1(OC)ccc(CN2CCC(O)(C(=O)NCC3CCC3)C2)c(Br)c1 90077,Cc1cc(=NCCCNc2ccccc2)[nH]c(=NCc2ccc(C)c(Cl)c2)[nH]1 90078,c1(C(=O)NCC2(C)CCC(NC(Cc3c(C)con3)=O)C2)cnc(O)n(C)c1=O 90079,C1(C(=O)NC(C#C)CC)C2CCN(C(=O)C(OCC)OCC)CC12 90080,S(=O)(=O)(c1ccc(-c2cccnn2)cc1)NC(C)CN(C)C 90081,N1(C(C=C(C)C)=O)CCC(NC(=O)CCn2c(C)csc2=O)CC(O)C1 90082,Cc1ccn2nc(C(=O)N(N3CCN(C(=O)C(C)(C)C)CC3C#N)C)nc2n1 90083,CC(C)(O)CC(=O)NCCC1CCCN1C(c1occc1C1CCC1)=O 90084,c1(CCC(=O)NC(C)CCc2ccc(F)c(Br)c2)cccc2c1OCCO2 90085,c1(C(N(CCC(C)NC(c2ccc(=N)[nH]c2)=O)C)=O)cc2ccccc2c(O)n1 90086,N1(C(Cn2c(C(F)F)cc(C)n2)=O)CC(NC(C2CC(=C3CC3)C2)=O)C(C)(C)C1 90087,C(N=c1cc(F)nc[nH]1)C1CCC(NC(c2ccc(C(N)=O)c(F)c2)=O)C1 90088,c1(C(=O)Nc2cccc(OC)n2)ccc2c(C(=O)Sc3nc[nH]n3)n[nH]c2c1 90089,Cc1ccc(F)c(N)c1C(N1CC(CC(C)NC(C2CC2(F)Cl)=O)C1)=O 90090,Cc1nc(C(N2CC(C3(NC(=O)C(O)P(C)(C)=O)CC3)C2)=O)c2ccccn12 90091,C1(CN(C(CC=C)=O)CC2CC2)CCN(C(=O)C(O)C(C)c2ccccc2)CC1 90092,C12(CNC(CC3(C)CCCO3)=O)CC(CO1)N(C(C1CCCN1C=O)=O)C2 90093,O=S(=O)(C1=CCS(=O)(=O)C1)N1CCN(c2csc(Cl)n2)CC1 90094,S(=O)(=O)(c1ccc(NCCC(C)C)c(F)c1)NCC(CC)(C)CO 90095,C1(C(N(C(C)CNC(=O)CN2CCN(C3CC3)C2=O)CC)=O)CC2(C1)CC2F 90096,C(=O)(CCP(C)(C)=O)N1CC(C)C(C(=O)NC2CCN(CCF)C2)C1 90097,C1(NC(c2n(CC#C)ccc2)=O)CC2CCCCN2C1.N12CCC(C1)OCC2=O 90098,CCCCC(C)CCC(=O)NCCC(C)N(C)C(C1CCC(c2cc[nH]n2)O1)=O 90099,C12(NC(c3n(C)nnc3)=O)CCCC1CN(C(C1CCC=CO1)=O)C2 90100,C1(C(N(CCN(C(c2ccc(COC)s2)=O)C)C)=O)CCCCC1F 90101,c1(C(N2C(CCCNC(C(C(C)C)F)=O)CCCC2)=O)cccc2nc[nH]c12 90102,c1(NCC(=O)NCC(CNC(CS(CC)=O)=O)(C)O)cc(C)ccc1OC 90103,Cc1cc(Cl)c(NC(C2CCN(C(=O)C(C)c3cccs3)CC2)=O)c([N+](=O)[O-])c1 90104,C(=O)(C(C(C)C)OC1CCCCC1)NCCCC(C)NC(CN(S(C)(=O)=O)C)=O 90105,C12(NC(c3ccc(OC)nc3)=O)CCC(C1)N(C(C1(C#N)CCCO1)=O)C2 90106,C(C1CCc2ccccc21)Cc1onc(C(C)(C)C)n1 90107,c1(N(C(=O)CCCn2c(O)nnc2O)C)ncnc(Cl)c1C(=O)NCCNC1CC1 90108,C1(C(=O)NCCC2(NC(C(CC=CC)C)=O)CC2)CC2(CCCCO2)C1 90109,c1(C(=O)NC(CNC(c2c(C)nncc2)=O)C)ccc2ncn(C)c(=O)c2c1 90110,C(c1ccc(Cl)cc1F)=CC(=O)NC(C(C)C)CNC(=O)CCC1CC1(Cl)Cl 90111,CCCCC(CC(=O)NCC1(COC)CCCC1)NC(c1cc[nH]c1C)=O 90112,C12(C(N3CCOCC(NC(C4CC(C5CC5)=NO4)=O)C3)=O)CCC(CC1O)C2 90113,N1(C(C23CCCCC2C3)=O)CC(N=c2[nH]c(Cl)nc(C3CC3)c2F)C2(CCC2)C1 90114,CN1CCC2(CCN(C(=O)C(c3ccccc3)NC(=O)CC3CNC(=O)O3)C2)C1 90115,C(=O)(C(O)CC1CC1)NCC(C)=CC(=O)NC(CO)C1(O)CC1 90116,c1(C(=O)NC2CN(C(CCSC)=O)CC2C(F)F)cc(C)nc(C)c1 90117,C1(C(=O)NCC(CNC(=O)C=CSc2ccccc2)O)CCc2nnc(O)n2C1 90118,n1(CC)ncc2cc(C(=O)NCc3ccnc(-n4cc(CO)nn4)c3)cnc12 90119,c1(C(N(CCNC(c2c(CC)cccn2)=O)C)=O)cnc2ccnn2c1 90120,N1(C(C)C)CC2(CN(C(C3C(NC(C4(C)CCCC4O)=O)C3(C)C)=O)C2)C1 90121,N1(C(CCN(C(C)C)C(CCc2ccc(O)nc2)=O)=O)CCC2(CCC(C)C2)C1 90122,c1(C(=O)NC2CCC(NC(c3cccc(SC)c3)=O)C2)c[nH]c(=N)c2[nH]ccc12 90123,c1(N2CCC(OCCN(C)C)C2)nccc(=NCc2nccn2CC2CC2)[nH]1 90124,Cc1csc2ncnc(NC(C3CCC(n4cc(CN5CC(F)C5)nn4)CC3)=O)c12 90125,C1(C(N2CC(CNC(C=C(C)C)=O)N(C)CC2)=O)CCC2(CC1)CC2(F)F 90126,N1(Cc2c(CC)n(CN3CCCC3)nc2)CC2CCC(N)C2C1 90127,CCC(C(=O)NCC(C)(C)CNC(=O)C=CCN(CC)CC)OC 90128,Cc1cnccn1.C1(SC)CCN(CC2CC2)C1.C12CCC(O1)c1ncsc1CN2 90129,c12c(cccc1C)CN2.C(C(C)CC(F)F)c1c(-c2n(CC#C)ncc2)nn[nH]1 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90182,C(CCC(=O)NC1CCC(CCNC(c2coc(Cl)n2)=O)C1)N(C(C)C)C 90183,C1(NC(=O)Cc2cc(C3CC3)on2)CC2CCCC(C1)N2C(c1coc(Br)c1)=O 90184,C1(C(N(C2CCCCN(C(c3cnccn3)=O)C2)C)=O)CCCC(C)(C)CC1 90185,c1(N2CC(OC)C3(C2)CC3)nc2cccnc2c(=NCCC2CCOC2)[nH]1 90186,C1(NC(C2CN(Cc3nc(Br)cs3)CCC2O)=O)CCc2ccccc2C1 90187,CC(CS(C)(=O)=O)NC(=O)C(CN(C)C)NC(=O)C=Cc1cncn1C 90188,C1(O)(c2cn(CC(CC)C)nn2)CCN(C(c2cnc(C(F)(F)F)nc2)=O)CC1 90189,N1(C(C=CCC)=O)CC2CCOCC2(NC(c2csc(S)n2)=O)C1 90190,N12CCCC(C1)C2=O.N1(C(C2(COCC)CC2C(=O)NC)=O)CCC(COC)C1 90191,Cc1ccc(F)cc1C1(CNS(=O)(=O)N(C)CCSc2ccccc2)CCOC1 90192,N1(C(CC(=O)NCC#C)=O)C2CCCC1CC(NC(c1cc(F)n[nH]1)=O)C2 90193,c1(C(=O)Nc2sncc2C(F)F)n[nH]c2ccc(-c3ccccc3F)cc12 90194,N12CC(NC(c3ccon3)=O)CC1C2=O.C1(C(=O)OC(C)(C)C)(CC2CC2)CCC1 90195,N1(C(c2cc(SC)oc2)=O)C(C(=O)NCc2cnoc2)CCC1C 90196,C(=O)(C(C(C)(C)C)NC(N)=O)NC(C1CN(C(c2c(C)nccc2Cl)=O)C1)C 90197,c1(C(N2CCN(C(C(c3cccc(Cl)c3)N(C)C)=O)CC2)=O)ccc(O)c(Cl)c1 90198,N1(Cc2c(OCCC)ccc(Br)c2)CCCC2CN(c3ncnc(C)c3Br)CC12 90199,c1(OC)ccccc1NC(=O)C(C1CCCN(C(=O)CC2CCCCC2O)C1)C 90200,C12CCCCC1NC(=O)CC1(CC1)N2C.C1(NC(C2CN(C(N)=O)C2)=O)CCCC1 90201,C1(NC(=O)NCCC(CNc2cccc(C)c2C#N)OC)CCOC2(CCC2)C1 90202,c1(CN2CCC(F)(C(=O)NCc3ccnc(F)c3)C2)cc(Cl)ccc1Cl 90203,C(C(C(C)(C)C)NC(c1ccn(C)c1)=O)NC(CCCOC(C)C)=O 90204,O=C1CCCCC(C(=O)NCCCCC(=O)NCC2CC3(CCC3)CO2)C1 90205,Cc1nc(C(N2CC(F)(CNC(C3(CO)CC3)=O)C2)=O)c(C)s1 90206,N1(C(C=C(C)C(F)F)=O)CCC2(CCCC2NC(C2CCC2)=O)C1 90207,c1(N2CC(CC(C)C)C2)nc(NC2(N3CCCC3)CC2)c2c(ncn2C)n1 90208,c1(C(N2CC(O)(CC(=O)NCc3cccs3)C2)=O)ccncc1F 90209,C1(CCOC)(C(N2CC(CO)CC2CO)=O)CCN(C(=O)Cc2cc[nH]n2)CC1 90210,CC1CCCCC1C(N1CC(CNC(c2cccc(C(C)(F)F)c2)=O)C1)=O 90211,Cc1n[nH]c(=NCCC2CCC(NC(C34CC(CO)(C3)OC4C)=O)C2)s1 90212,N1(C(N2CCN(CCN(C(CS(CC)=O)=O)C)CC2)=O)C(C)CCCC1C 90213,Cc1ncnc(O)c1C(=O)NC1C2CN(C(c3c(C4CC4)cnn3C)=O)CC12 90214,N1(C(C(=O)Nc2cc(OC)n[nH]2)CCc2ccc(Cl)cc2)CCC(C)C1(C)C 90215,C1(COC)(CNC(c2cc(C#N)cs2)=O)CCN(C(c2cccc(O)n2)=O)C1 90216,N1(CCN(C2CCOC2)C(CSCC(N)=O)=O)CC2CCC(C1)O2 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90253,N1(C(C2(Cc3cnn[nH]3)CCCC2)=O)CCC(CC(C=O)NCC2CC2Cl)CC1 90254,CCC(C)(C)CC(=O)N1CCCC(O)(CNC(c2cc(C3CC3)ccn2)=O)C1 90255,c1(N(C(C)C(=O)N(C(C)CNC(=O)CNC(N)=O)C)C)ccc(F)cc1F 90256,N1(C(C)=O)CCN(CCN2C(=O)NC(CC(F)F)C2=O)CC1C 90257,Cc1cc(C(N2CC(C(N)=O)(CNC(C3CN(CC(C)C)C3)=O)C2)=O)nnc1O 90258,N(C(=NCc1cccc(OC)c1)NCC1(C#N)CCCC1)C(CC)C 90259,c1(CNc2ccc(-c3ccc(OC(C)C)nc3)cn2)c(F)cncc1F 90260,c1(NC(=O)NCC(C(F)(F)F)c2ccon2)nccc(C(F)(F)F)n1 90261,c1(C(=O)NC2(c3cn(-c4cn(C)nc4)nn3)CCC2)cc(Br)cnc1C1CC1 90262,c1(CC(=O)NCC2C(NC(C3C(C)(C)C3)=O)CC2)c(Cl)cccc1Br 90263,C(=O)(C(CC(C)C)CC(C)C)NCC1CCN(C(CCC(=C)Cl)=O)C1 90264,C1(CC)CN(C(c2ccc(C(C)C)s2)=O)CCN1C(C12CC(F)(C1)C2)=O 90265,c1(C(=O)NCC2C(CNC(C(C)O)=O)C2)cccc(Oc2ccccc2)c1 90266,c1(CCNC(CC2C(N)CCC2)=O)ccc(Br)c(F)c1 90267,c1(C(CCN(C)CC2CCCC(O)C2)=O)ccc2ncsc2c1 90268,c1(OCC)n[nH]c2cccc(-c3nc(CS(C)(=O)=O)nn3C(C)C)c12 90269,C(=O)(CC1=CCCC1)N1CCN(CCNC(=O)C(C2CCOCC2)O)CC1 90270,C1(n2cc(-c3ncc(C)cn3)nn2)CC2CCC1(NC(=O)CC1CCC(=O)N1)C2 90271,C12CC13CCC(CC3)C(=O)N2.C1(CC(=O)OC(C)(C)C)CCCOC1 90272,N1(C(CC(=O)OC)=O)CCC(NC(c2cc(-c3csc(C)n3)c[nH]2)=O)C12CC2 90273,c1(CNC(=O)NCCC(C)N(CCC)C)sccc1OC 90274,C1(C(N2CCC(N3CCN(C(C(CC)(C)O)=O)CC3)C2)=O)Cc2cc(F)ccc2O1 90275,C1(C)(CCNC(C2CC(OCC)C2)=O)CCN(C(C2(C)CCC(=O)N2)=O)CC1 90276,Cc1nc2c(s1)C13CC(C1)NC(=O)NC1(N2C(=O)CO3)CCCN(C)S(=O)(=O)C1 90277,N1(C(c2cncc(C)c2)=O)CCCC(NC(=O)C2=CCC2)C(F)C1 90278,C(c1cc(Cl)cc(Cl)c1)=CC(=O)NC1(CF)CCN(C(c2[nH]c(=N)sc2)=O)C1 90279,Cc1cc(NC(=O)C(CC(C)C)N(C(=O)C(=O)C(C)C)C)c(C)cc1F 90280,N1(C(C2CCC(=C)CC2)=O)CC(NC(c2nc(OC)ccc2Cl)=O)CC1(C)C 90281,CN1CCC(C)(C(N2CC(=O)NCC2C(=O)N(C)OCc2ccccc2)=O)CC1 90282,N1(C(CC)C)CCN(C(C2COCC2NC(=O)Cc2cncn2C)=O)CC1 90283,CN1CCCC1c1cc(C(=O)NC2CCN(C(=O)COC3CC(F)(F)C3)C2)n[nH]1 90284,c1(SCC)ccc2c(c1)OCCO2.c12cc(ccn1)OC(=O)N1CCC(C1)NC2 90285,C(=O)(C#CC1(C)CCCO1)N1C(C(N2CCC(COC(C)=O)C2)=O)CCC1 90286,n1(CC(=O)N(C(C)C(C)(C)N(C)C)CCO)cc(C(N2CCOCC2)C2CC2)nn1 90287,CS(=O)(=O)c1csc(C(=O)NC2CC(C)(NC(C3CC3C#N)=O)C2)c1 90288,N1(C(c2c(CC)con2)=O)CC(NC(c2cnn(C(C)C)c2)=O)C(F)C1 90289,C(=O)(CC(C)C(C)(C)NC(c1cnn(C)n1)=O)N1CC=C(C)CC1 90290,CC1(C)CC(NC(C23CC4CC2C3C4)=O)CCN(C(c2ccccc2CO)=O)C1 90291,C1(CCOC)(NC(C2CCCC2)=O)CCN(C(c2ccccc2SCCO)=O)C1 90292,c1(CN2CCN(C(C3CCCS3(=O)=O)=O)CC2)ccccc1SC(C)C 90293,C(C(=O)NOC(C)(C)CO)=CC(C)(C)SC.C1(C)C=CCC1 90294,c1(C(=O)NC(C2(O)CCCN(C(c3cnoc3)=O)C2)C)cnn2c1N(C)CC2 90295,c1(C(=O)NC2CC(C)(NC(CN3CCC(OC)C3)=O)C2)ncccc1C 90296,C1(NC(c2scc(C)c2)=O)C2CCC1CC(NC(=O)C=CCCC(C)C)C2 90297,C1(C(=O)NCC2(C=C)CCC2)CCC2(CC2)N1C(=O)CN=[N+]=[N-] 90298,N1(C(c2c(C)ocn2)=O)CCC2CCCC12CNC(c1ccc(N)c(Cl)c1)=O 90299,c12nc(ccc1C#N)C(=O)N2CCC.c1(C(=O)NCC)ccc(C)cn1.C(C)C 90300,c1(CN(C2C(C)CCNCC2)C(=O)C(F)n2cccn2)cncc2ccccc12 90301,CCCC(C(O)C(=O)NCc1csnc1C)NC(C1(C)COC(=O)N1)=O 90302,C1(C(C)C)CCC(C)N(C(=O)C(=O)NC2C(F)(F)C23CCC3)C1 90303,Nc1cc(O)nc(CCNC(C2CCN(c3ncccn3)CC2)=O)n1 90304,c1(C(=O)NC2CCCC(NC(C3(C)CC4CC4C3)=O)CC2)ccn2nccc2c1 90305,N1(C(c2c(Cl)cn(CC)n2)=O)CCCC(NC(C2(C)CC(F)(F)C2)=O)C1C 90306,C1(C(N2CC3(CC(NC(c4cn(CCF)nn4)=O)C3)C2)=O)CCC(C2CCC2)CC1 90307,c1(OC)ccc(Br)cc1C(CO)NC(C1CC1NC(c1coc(C)n1)=O)=O 90308,c1(C(N2CC(CN(C(=O)CCCN(C)C)C)OCC2)=O)cnc2c(c1)NC(=O)CN2 90309,C1(C(=O)NCC(N2CCC(O)C2)(C)C)C(C#N)C1(C)C.C12CCC(O1)NC2=O 90310,N1(CC(C)NC(C2(CO)COC2)=O)CCN(C(=O)CC2CCCCC2)CC1 90311,C1(N(C(C(CCC)S)=O)Cc2ccc(C(F)(F)F)cc2Br)COC2(CCNCC2)C1 90312,N1(C(CC2CC(=C)C2)=O)CC(C2CN(C(c3cnn(CCOCC=C)n3)=O)C2)C1 90313,Cc1cnc(CNC(C2CCCN(C(C3CCCCC3O)=O)C2)=O)nc1 90314,N1(C(C2(Cc3cccc(C)c3)CC2)=O)CCC2C(C1)CN2C(=O)CN=S(C)(C)=O 90315,C(C(C(C)C)C(C)C)NCC(CCCC)Sc1ccccn1 90316,C(=O)(C(CC)C(F)(F)F)N(CC(=O)NCC1C2C(C2CC)C1CO)CCC 90317,C(CC(=O)NCCCNC(=O)C(C)C1CCOC1)N(CCOCCOC)C.C(CO)O 90318,C(=O)(C1=CCCCC1C)N1CCCC(CN(C(c2sc(C)c(Br)c2)=O)C)C1 90319,Cc1nc(NCC2CCN(C(C3CCC(=O)N(C)C3)=O)C2)c(C)c(C)n1 90320,C(c1cccnc1C)=CC(=O)NCC(CNC(c1nncc(CCC)c1)=O)OC 90321,C12(C(=O)NC(CC#C)CO)CCCC1N(C(=O)Cc1cc(C)[nH]n1)CC2 90322,N1(C(c2c(C(C)C)nns2)=O)CCN(C(C2CCCN2C2CC2)=O)CC1C 90323,N1(C(C2N(CC)CCC2)=O)CC2COCCC2(NC(=O)C=Cc2nc(C)cs2)C1 90324,N1(C(CC(=O)OCC)=O)CCC(O)(CN(C)C(C2CSCN2C(C)=O)=O)C1 90325,CC1(C)CN(C(C2CCS(=O)(=O)C2)=O)CCC1C(=O)N=c1ccn(CC2CC2)[nH]1 90326,CCC(C)C(O)C(C)C(=O)N1CC2CC1C2NC(C1(c2ccccc2)CC(C)=NO1)=O 90327,C1(CNC(C2CC=CC2)=O)CCC2(CCC2)C1NC(=O)Cc1ccnn1C1CC1 90328,c1(CC(=O)N(CC(CNC(c2c(CC)[nH]cc2)=O)(C)C)C)ccc(C)c(F)c1 90329,c1(OC)cc(OCC(N2CCC(CNC(=O)Nc3ccccc3O)C2)=O)ccn1 90330,Cc1ccc(C(C)C(=O)NCC2CCC2C(=O)NC2(CF)CCC2)o1 90331,c1(CNC(C2(CC=C)CN(C(c3cc(C)nn3C)=O)C2)=O)sc(C)nc1C 90332,N1(C(C2CC(OCC)C2)=O)CCC(NC(C2CCCC(F)(F)C2)=O)C(C)(C)C1 90333,C=CCC(CNC(c1cnco1)=O)C(=O)NC(c1cnccc1C)C 90334,C(C(O)CC(C)C)NC(c1ccc(Cn2cc(C(CC)(C)C)nn2)o1)=O 90335,CC(CN(C)C)CN=c1nc(N2CCCC(C#N)C2)c2cccc(F)c2[nH]1 90336,N1(C(c2ncc(NC)nc2)=O)CC(C)(C)CC1C(N1CCC(c2cc[nH]n2)C1)=O 90337,C(=O)(C(O)CC[S+](C)C)N(CCCCNC(=O)C(C1CCCCC1)F)C 90338,c1(C(N2C(CNC(c3ccc4sncc4c3)=O)CCC2)=O)noc2c1COCC2 90339,C(=O)(C#CC1CCCO1)NC1(CO)CN(C(C2C(c3cn(C)nc3)CC2)=O)C1 90340,Cc1cc(C(=O)NCC2(O)CC(Nc3ncc(I)cn3)C2)c2ccc(F)cc2n1 90341,C1(C(=O)NC2(CO)CCCN(C(=O)Cc3ccco3)C2)CCc2nccn2CC1 90342,c1(C(=O)NC(CCCCNC(=O)OC(COC)C)C)c(OC)ccnc1F 90343,C1(C(N(C)CC2CCCN2C(C2CCC23CCC3)=O)=O)CCc2cn(C)nc2C1 90344,c1(N(CC(=O)NC2CC(NC(C=C(CCC)C)=O)C2)C)ccc2nncn2n1 90345,C1(C)(CNC(c2nc(CC(C)C)sc2)=O)CN(C(=O)C(O)CC2CC2)CCO1 90346,CC(C)CC(O)C(C)C(=O)N1CCC(N(C(=O)CC(=O)N(C)C)CCO)CC1 90347,C(=O)(C(C)CC(N)=O)N1C(CNC(c2cnc(C)n2C)=O)CCC1 90348,c1(C(=O)NCCCCC(C)NC(=O)Cn2cc(C(C)O)nn2)ccc(=O)n(C)c1 90349,C1(C(=O)NC2(CNC(c3cn(C)nc3)=O)CC2)CCCCN1CC1C2COCC12 90350,C1(CNC(Cc2ccn(C)n2)=O)CC(NC(=O)CN2C(=O)CNC2=O)C12CCC2 90351,c1(C(=O)NCC(C)CNC(C2COC(=O)N2)=O)cc(Cl)c(F)cc1Cl 90352,c1(C(C(C)C)NC(C2CCN(C(c3ccco3)=O)C2)=O)ccccc1F 90353,CN=c1nc(C(N2CCC(F)(CNC(=O)C(C)=C(C)C)CC2)=O)cc(C)[nH]1 90354,C1(C(=O)NC(C#C)CC)CSCCN1C(c1cccc[n+]1[O-])=O 90355,C(C(C)(C)C(=O)N1CC(NC(C2CCOC2)=O)C(C)C1)SC 90356,C#CC(C(C)(C)OC)NCc1cc(Cc2cc(COC)on2)on1 90357,CC(C)CC(CNC(c1ncccc1F)=O)NC(=O)CC1(C(F)F)CCCCC1 90358,C1(C(=O)OCC)(CNC(C2CC(F)CN2C(=O)CC#N)=O)CCOCC1 90359,CC(C)CCCCCC(=O)N1CC(N(C)C(C2CC3CCC2C3)=O)C1 90360,Cc1cc(O)nc(C)c1C(=O)N(CC(C)NC(C12CC(C)C1C2)=O)C 90361,C=CCC(CNC(=O)Cn1nnnc1C)NC(=O)CCNC(=O)C=CCl 90362,CCCCCS(=O)(=O)CC(=O)N1CC2=C(C1)CN(C(=O)C(c1cnn(C)c1)C)C2 90363,N1(C(C2C(CNC(C3(C#N)CC(C)C3)=O)CCC2)=O)CC2CCC2(C(N)=O)C1 90364,C1(C(=O)NCc2ccc(C3CCCCC3)s2)CCCN1CC1CCCCO1 90365,CC(N=c1[nH]c(=NCC2CCOCC2)[nH]c2c1SCC2)c1nc(O)n[nH]1 90366,Cc1nc2ccccn2c1C(=O)NCC1CCN1C(=O)CC1(O)CCOCC1 90367,C1(CC(=O)N(CCC[N+](C(=O)C(F)F)([O-])OC)C)(C(=O)OCC)CCC1 90368,CCCCCC(O)C(=O)NCCN(C(=O)C(=Cc1ccc(Cl)cc1)C)CC 90369,c1(C(=O)NC(C2CCCN2C(=O)C(=Cc2cscn2)F)C)c[nH]nc1OC(F)F 90370,C(=O)(C1=COCCO1)NC(C)CCCNC(C12CC(CCO1)C2)=O 90371,c1(C(C(=O)NC2CCOC2)N(CC(COC)C)C)cc(S(C)(=O)=O)co1 90372,c1(CC(=O)N(C(CNC(=O)C(F)(F)F)CO)CC(=O)NCCF)ccc(Cl)nc1 90373,C(CCN(C)C)(C(=O)NC1(CSC)CC1)NC(c1c(CCC)[nH]cc1)=O 90374,O=C(C=C[SH](C1CC1)c1cccc(Cl)c1)NC1C2C3CCC(C3)C12 90375,Cn1ccc2cc(C(=O)NC34COCCC3CN(C(C3(Cl)CC3)=O)C4)cnc12 90376,c1(C(=O)NC(CCN(C(CCN(CC(C(C)C)C)C)=O)C)C)csc2cncn12 90377,C(CC(C)C)(C(=O)NCc1ccc(CC)o1)NC(c1c(CC)c[nH]n1)=O 90378,C1(C(=O)NC23CC(CNC(c4cc(C)[nH]n4)=O)(C2)C3)Oc2ccccc2OC1C 90379,N1(C(CCCOCCOCC)=O)CC(C)CN(C(C2(SC)CC2)=O)CC1C 90380,C(=O)(C1=NOC(CNC(=O)C(C)(F)c2ccon2)C1)N1C(CC)CC(O)C1 90381,c1(CN(CCCCCC(=O)NC)C)ccc2[nH]ccc2n1.C12CCCN1C2=O 90382,C1(CC)CN(C(=O)C2=NOCC2)CCC1CNC(=O)CC1CCC(=O)NC1 90383,C1(NC(c2c(C)nc(C)o2)=O)COC2(CCN(C(c3sccc3C)=O)C2)C1 90384,C12(NC(=O)CCSC(F)(F)F)COCCC1CN(C(c1ccns1)=O)C2 90385,c1(C(N(S(CC=C)(=O)=O)C(C)C)=O)cn(CC(=O)OC)c2ccccc12 90386,C1(S(C)(=O)=O)(C(=O)NCC2(CNC(CN(CCC#C)C)=O)CC2)CCCC1 90387,c1(OC)ccc(NC(=O)CNc2ccc(-c3nc(C)cs3)cc2)c(C)c1 90388,C1(CNC(C(C(C)C)OCC)=O)CN(C(=O)C=Cc2ccc(C)s2)CCCO1 90389,CON=CC(=O)NC(CC1CCCC1)C(=O)NCCOC1(C)CCCC1 90390,Cc1nc2c(N3CC(O)(CNC(c4ccc(Cl)nc4)=O)C3)ncnc2[nH]1 90391,O=C(NNc1ccc(C(=O)NC2CCS(=O)(=O)C2)cc1F)C1CC12CC2 90392,c1(C(N2CC(C)C(C)(CNC(=O)CC3CCOC3)C2)=O)nccc2ncccc12 90393,C1(C(N(CCC(C)(C)NC(C2CCCCC2)=O)C)=O)CCCCC1F 90394,N1(C(CC(=O)NCC)=O)Cc2nccn2CC(NC(C2CCCSC2)=O)C1 90395,O=C1NCC2(CCCN(c3nccc4[nH]ccc34)C2)O1 90396,C1(C)(NC(c2ccn(CC)n2)=O)CCCN(C(=O)CCc2nc(C(C)C)no2)C1 90397,C1(N(C)C)CCC(C(=O)NCC=CCNC(c2coc(CO)c2)=O)CC1 90398,C(CCC(=O)NC(c1ncc[nH]1)C)(C(C)C)NC(C(COC)N(C)C)=O 90399,c1(C(=O)NCC(C(C)C)(C)NC(=O)C(O)C2CCC2)cnc(Cl)cc1N 90400,Cc1cc(C(=O)NCC(C)C(N2CC(F)(F)C2C2CC2)=O)cnc1F 90401,c1(C(=O)NCCCCC(C)NC(c2c(CC)noc2C)=O)cn2c(n1)SCC2 90402,CC1(C)NC(=O)CC1C(=O)NCCC1CC1 90403,Cc1cccc2c(C(=O)NC3CC(F)(CNC(C4CC45CC5(F)F)=O)C3)n[nH]c12 90404,C12(NC(C(CC=C(C)C)c3ccccc3)=O)CCC(CC1)N(C(=O)CCN(C)C)C2 90405,CN1C2CCC1CC(C(=O)NC13CC(NC(=O)C#CC4CCCO4)(C1)C3)C2 90406,C=C(C)C1OCCCC1C(N1CC2OCC(NC(=O)CCc3cnc[nH]3)C2C1)=O 90407,C12(CNC(CC=CC(C)(C)C)=O)CC1CN(C(=O)C(CC1CC1)CC1CC1)C2 90408,N1(C(CS(C)(=O)=O)=O)CC(O)(C2(CNC(=O)CC=C(Cl)Cl)CC2)C1 90409,Cc1csc(CCC(=O)N(CC(C)NC(=O)CCn2cc(Cl)cn2)C)c1 90410,N1(C(C(C)Cc2cnn(C)c2)=O)CCN(C(C2(O)CCCC2)=O)CC1CC1CC1 90411,C1(C(=O)NCC(C(C)C)NC(=O)C=CCO)CCCN(c2ccccc2)C1=O 90412,C1(NC(C2(NC(C)=O)CCC2)=O)CC(O)CN(C(C23CC4CC2C3C4)=O)C1 90413,C1(CC(=O)NC2C(C(=O)NC(C3CCCO3)CC)CC2)CCC(C(N)=O)CC1 90414,C1(F)(C(N2C(C)CC(CNC(C=CC=CC)=O)C2)=O)CCC(F)(F)CC1 90415,c1(CC)cccnc1C(=O)NCC(C)CN(C)C(c1ccc(C(F)F)nc1)=O 90416,c1(C(=O)NC(C)CNC(C2CC3CC3CC2C)=O)cc2c(cn1)OCCO2 90417,C1(NC2CCCC(C(C)(C)C)C2)CC2CC3CC(C2)C1C3 90418,C1(CNC(N)=O)CCCN(C(C2CSCN2C(c2cccnc2)=O)=O)C1 90419,C(C(CC(=O)NCC1CCC(F)(F)C1)OC)NC(CC(=O)NCC#C)=O 90420,c1(N2CC(NC(=O)Nc3c(F)cccc3Br)C(O)CC2)nc(C)nc2c1CCC2 90421,C(=O)(C(F)CC(C)(C)C)N(CC(C)C)CC(=O)NC12CC1COC2(C)C 90422,C1(CC(=O)NCc2c(C(N(C)Cc3cc(C)on3)=O)occ2)CCCC(C)C1 90423,C1(N(C(C2C(C)CC2)=O)C)CCC2CN(C(=O)CN3CCNC3=O)CC12 90424,CC(=O)CC(C)(C)C(=O)N1CCN(CCNC(c2cc(F)n(C)n2)=O)CC1 90425,c1(OCC(C)C)ccc(CCNC(=O)CCn2ncn(C)c2=O)cc1 90426,CCC(C)C(O)C(=O)NCCCOCCN(C(c1cnn(C)c1SC)=O)C(C)C 90427,CC(C)CCCCC(c1nnnn1CCC1CCCC1)NC(CC)C1CCC1 90428,C1(NC(N2CCC(COCc3nn[nH]n3)C2)=O)CC(O)(c2cccnc2)C1 90429,c1(C(=O)NC(CNC(CN(CC)CC)=O)(C)CC)cccn2c(C)nnc12 90430,CC1(CNC(=O)COCC2CCOC2)CCN(C(=O)C(C2CC2)C2CC2)CC1 90431,N1(C(c2nc(C)[nH]c2C(F)(F)F)=O)CC(NC(=O)Cn2ccsc2=N)C(C)(C)C1 90432,C1(CCOC)CN(C(c2cncc(OC)c2)=O)CCN1C(c1cc(C)sc1C)=O 90433,CC(C)C(C)(O)C(=O)NCCCCCNC(=O)Cn1cnccc1=O 90434,CC(=O)C(C)(C)CC(=O)NC1(C)CCN(C(C2CCC(C)(C)C2)=O)C1 90435,C1(CC(=O)NCC(CNC(c2cn(C(C)C)nn2)=O)C)COC2CC1C2 90436,N1(C(c2n(CCC)ccc2)=O)CCC(CO)(NC(=O)CCCCOCC)C1 90437,CC(CNC(c1ccoc1)=O)C(=O)N(CCN(C)C)C1CC1 90438,N1(C(C2CC(SC)C2)=O)CC2C(CC(=O)NCC(F)Br)C2C1C 90439,Nc1c(C(=O)OCCSCc2ccccc2)cc(Br)cc1Br 90440,CCS(=O)(=O)C=CC(=O)NCCN1CCC(NC(c2cc(Cl)nc(Cl)c2)=O)CC1 90441,C(C)(C(C)(C)C(=O)NC1CC(O)C(O)C1=O)NC(CN(C(=O)OCC)C)=O 90442,C1(O)(C(C)NC(=O)Cc2ccoc2)CCN(C(C2(C#N)CC(F)(F)C2)=O)CC1 90443,C1(NC(CCC)=O)CCN(c2nnnn2Cc2cccc(I)c2)CC1 90444,C1(C(=O)NCCn2cc(CNC(C(CC)C)=O)nn2)Cc2cccnc2C1 90445,c1(CC(C)SC2CCCO2)ccc(C(=O)NOCC2CCCCC2)cc1 90446,Cc1nn(C)c2c(NCC3CCC(F)(F)CC3)nc(N(CC(Cl)Cl)C)nc12 90447,C1(C(=O)NCC(CCC)NC(C2C3CCC2CC3)=O)COC(C)(C)C1 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90690,c1(OC)ccccc1OCC(=O)NCC1(CO)CCOC1.c12ccc(cc1)[nH]c2=O 90691,C#CCCCC(C)C(=O)NCCC1(O)CN(C(=O)C(C)N2CCCC2)C1 90692,C1(COC)(NC(=O)CCn2ccc(C)n2)CCN(C(C2CC(C#N)C2)=O)C1 90693,C1(C(=O)NCCC(=C)CNC(C2CCN(C)C2=O)=O)CCCc2ccccc2C1 90694,N#Cc1cc(F)c(C(N2CC(F)CC2C(=O)NCC2CCC(=O)NC2)=O)c(Cl)c1 90695,CCC(F)C(=O)NC1CCC1NC(=O)Cn1cc(C(=O)NC)nn1 90696,N1(C(C2C(=O)NCC2)=O)CCC2(CC1)CC(NC(C1CC3(C1)CC3F)=O)CCO2 90697,C1(C(N2C(C)(C)CCC(C(=O)OCC)C2)=O)CCc2ncc(Br)n2C1 90698,C1(C(=O)NC(C)CN(C(=O)CN2SCCCCC2)C)CC2OC(C)(C)OC2C1 90699,c1(C(N(CC(Cl)Cl)C)=O)cc(CNC(c2cnn[nH]2)=O)cs1 90700,C1(C(=O)NCC2N(C(c3nc(CC)oc3)=O)C3C(C2)C3)CCC(C)(F)CC1 90701,C1(CC(=O)NCC#CCNC(C2CC23CCC3)=O)CCc2ccccc2C1 90702,N1(C(Cc2c(C)n(C)nc2)=O)CC(CO)C2(C1)CN(C(c1ccc(N)cn1)=O)C2 90703,C1(NC(CN(CC)Cc2ccccc2)=O)CN(C(c2sccc2F)=O)C2CC12 90704,C1(C)(C(=O)NCC(C)N(C)C(c2csc(-c3ccncc3)n2)=O)CCCN(C)C1 90705,N1(C(CC2N(C(C3=CCC(C)CC3)=O)CCC2)=O)CCc2nnnn2CC1 90706,N1(C(CNC(=O)CC2CCCC2)=O)CC2CN(C(=O)CC3CCC(=O)N3)CC2C1 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90759,C1(C(C)C)CCC(C(=O)NCC(O)CC2CCCC2)N1C(=O)CC#N 90760,N1(C(C(F)=CCC)=O)CCCC(C)(C)C1CNC(=O)CC1C=CCC1 90761,C1(C(CO)NC(C(C)OC2CCCC2)=O)CCN(C(=O)Cc2ccc(F)nc2)CC1 90762,C1(C(N(C2CCC(NC(=O)C=C3CCCC3)C2)C)=O)SCCCS1 90763,c1(CC)conc1C(=O)NCCCNC(=O)CC1CC1(C)C 90764,c1(NC(C(c2cccc(Cl)c2)NC)=O)nc2cccc(Br)c2[nH]1 90765,C(=O)(CCCC(C)CC)N(C1CCCN(C(=O)CSC(F)(F)F)CC1)CC 90766,Cc1[nH]c2ncnc(N3CCC(C4(NC(c5ccc[nH]5)=O)CC4)C3)c2c1C 90767,C(c1ccc2occc2c1)=CCC(N1C(C)CN(C(=O)OC(C)(C)C)C(C)C1)=O 90768,c1(OCCOC)ccc(COC(=O)COc2ccc(O)cc2I)c(Cl)c1 90769,c1(OC)cncc(C=CC(N2CCC(NC(=O)Cc3ccns3)C2(C)C)=O)c1 90770,c1(CC)ccc(C(=O)NC2CC(CCNC(=O)C=CSC)C2)c(O)c1 90771,c1(C(=O)NCCc2c[nH]c(=NCc3cc(F)cc(Cl)c3Cl)s2)[nH]nc2ccncc12 90772,N1(C(CCOC2CCN(C)CC2)=O)CC2(CNC(=O)C3=CCSC3)CCC1C2 90773,CC(C)(CCC#N)C(=O)NCC1(CNC(C2CCCN2C)=O)CC(=C2CCC2)C1 90774,Cc1coc(C)c1C=CC(=O)N(C)CC1CCCCN1C(=O)CCc1nncs1 90775,c1(C(N2C(CNC(C(C)C#N)=O)CC2)=O)cc(Cl)ccc1O 90776,N#Cc1ccc(CS(=O)(=O)NC2CN(c3ccccc3F)C2)cc1 90777,Cc1cc(C)c(C(N2CCOC(C)(CNC(c3cnsn3)=O)C2)=O)c(C)n1 90778,N1(C(c2n(C)ccc2)=O)CCC2(CC(NC(c3cncc(Cl)c3Cl)=O)CO2)C1 90779,c1(N(C2CCCCC2=O)CCN(C)C)ccc(Br)cc1 90780,C1(N(C(CC(C)SC)=O)C)CCN(Cc2oc(C)nc2C)CC1 90781,N1(C(C2(COC)CCOC2)=O)CCCCC(NC(c2ccc(C(N)=O)o2)=O)C1 90782,N1(C(C=CCN(C(=O)CCCCN(C)C)C)=O)CCC2OCCC2C1 90783,CC1(C)CN(C(=O)CN2CCOCC2)CCC1C(=O)NC1CCCC1O 90784,Cc1cc(NC(c2cccc(F)c2)=O)ccc1NC(=O)CC(=O)NCC(F)(F)F 90785,N1(C(c2[nH]n(C)c(=O)n2)=O)CC(F)(F)CC1CNC(c1cncnc1C1CC1)=O 90786,c1(CC)nc(C(=O)NCC2C(C)CCN2C(=O)CC2CC2C(F)(F)F)c(N)s1 90787,CC(C)CC(CNC(c1ccn(C(F)F)n1)=O)NC(C1(CN(C)C)CC1(F)F)=O 90788,N1(C(Cn2c(C)ccn2)=O)CCCC12CCC(NC(=O)C=Cc1cnc[nH]1)CC2 90789,CC1CCC(C(N2C3CCC2C(NC(C2CC24CCOCC4)=O)C3)=O)CC1C 90790,C1(NC(=O)Cc2cnoc2)CCCN(C(=O)C(O)Cc2cnc[nH]2)C1 90791,C(=O)(C(C)(C)C(F)F)N1CC(N(C(=O)CN2CCCCCCC2=O)C)C1 90792,c1(CC)oc(C)cc1C(N1CC(C(=O)NC2CCNC(=O)C2)C(C)C1)=O 90793,c1(C(N(C(CNC(CCc2ccc(C)o2)=O)C)C)=O)cc(C(F)F)ccc1F 90794,n12c3c(cc(cc3)c1=O)CC2.C1(C)(C(=O)NCCCNC(C)=O)CC(C)=NO1 90795,c1(C(=O)NC(C(=O)N(CC(C)OC)C)C)cncc(O)c1 90796,C1(NC(=O)CSC(F)(F)F)CN(C(=O)Cn2ncccc2=O)C2(CCCOC2)C1 90797,c1(C(N2C(C)CCC2)=O)cn2c(n1)CN(C(c1c(Cl)cnn1C)=O)CC2 90798,c1(C(N(CCCNC(C2COCC(C)O2)=O)C2CC2)=O)cc2cccn2c(O)n1 90799,c1(CNC(N2CCC(NS(=O)(=O)C3CC3)CC2)=O)ccc2nonc2c1 90800,c1(C(N2CC(C)C(CNC(=O)C(CO)N(C)C)C2)=O)c[nH]c2c(F)cccc12 90801,C1(NC(c2c(C)sc(Cl)n2)=O)CCN(C(=O)COCC2CCCOC2)CC1F 90802,c1(OC)cc(C)cc(C(=O)NC2CC(C(=O)NC3CCCC3N(C)C)C2)c1N 90803,CCCCCCC(C)CC(=O)N(C1CCN(CCOc2ccccc2Cl)CC1)C 90804,C1(C(=O)NCC)(CC2CC(NC(c3onc(COC)n3)=O)C2)CCCNS1(=O)=O 90805,C(=O)(CS(=O)(=O)CCO)NC(C)CNC(=O)CC1(NS(C)(=O)=O)CCCCC1 90806,CN1C(=O)CN(CC(=O)NC2CCCC(NC(C3CCOCC3(C)C)=O)C2)C1=O 90807,C(c1nc2ccccc2o1)=CC(=O)NC1C(CNC(C(C)(C)CO)=O)CCCC1 90808,CCCCC(C(=O)NCCCCn1cc(CNC(=O)OC(C)(C)C)nn1)N(C)C 90809,c1(OC)ccc(C(=O)NC(CNC(c2cnc(C(C)(C)CF)o2)=O)C(C)C)cc1 90810,C1(C(N2C(C(=O)OCC)CN(C(=O)C(F)(F)F)CC2)=O)CC(=O)CC12CCC2 90811,c1(C(=O)C2CC2)ccc(S(=O)(=O)N2CCCN(C(=O)NC3CCCCC3)CC2)s1 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90830,C1(NC(c2c(SC)scc2)=O)CCN(C(c2[nH]nnc2C)=O)C(C)C1 90831,C1(N(C)C(c2ccccc2N2CCOCC2)=O)CN(C(C2COC2)=O)CC1(C)C 90832,c1(C(=O)NCCN(C(c2n(CC)cnn2)=O)C2CC2)ccc(S(=O)C(C)C)cc1 90833,Cc1ccncc1CNC(=O)C(Cc1cn[nH]c1)NC(c1cocn1)=O 90834,O=C(C1=C(c2ccccc2)CCO1)NC1(C2CN(C(=O)CC3CCOC3=O)C2)CC1 90835,N1(C(c2cn(CCOC)nc2)=O)CC2CCC(N(c3cnc(C#N)cn3)C)C2C1 90836,Cc1cccc(C(=O)N(CC(=O)NCCc2cnnn2C)CC2CC2)n1 90837,C1(NC(=O)Cc2cc[nH]n2)CCCC(NC(=O)Cc2nc(C3CC3)cs2)C1 90838,C1(OC)CN(C(=O)C(C(C)C)NC(=O)C2CC2)CC1NC(c1cccn1C)=O 90839,c1(C(=O)NC2CCC2NC(c2nsnc2O)=O)cc2nccn2c(O)n1 90840,N1(C(c2c(COC)cc[nH]2)=O)CCC(C)C(CNC(=O)C=Cc2cncn2C)C1 90841,C1(C(=O)NCc2cn(CC(N3C(CC(C)O)CCCC3)=O)nn2)CC12CCOCC2 90842,O=C(CC1CC2(C1)CN(C(=O)CC1CCOC1=O)C2)Nn1cncn1 90843,C1(NC(c2ccsn2)=O)CCN(Cc2ncc(Cl)cc2Cl)CC1F 90844,C1(CC)CCC(O)(C(=O)N(CCCNC(c2cc(C(=O)OC)cn2C)=O)C2CC2)C1 90845,c1(C(C)O)ccc(NNC(=O)NCCc2ccc(NC3CCOCC3)cc2)cc1 90846,C(CC1CCC1)(C(=O)N(C(C)C(=O)NCC(C)(C)O)C)OC 90847,c1(NCCOC)ccc(S(=O)(=O)N2CCC(c3ncno3)C2)c(Br)c1 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91057,N1(c2onc(C)n2)CC(C(N2CC(NC(=O)COCC(C)(C)C)C(C)C2)=O)CC1=O 91058,N1(C(C(C(C)C)C(C)NC(c2ccc(F)s2)=O)=O)CCC2CN(C)CCC12 91059,c1(CN2C3CCN(C3)CC2)ccc(Br)c(OC)c1.n1(CC)ncc(Br)n1 91060,CC(C)CCCOCC(N1CC(O)(N(C(=O)C(C)CC2CCCO2)C)C1)=O 91061,N1(C(C(C)NC(C2CCCC2)=O)=O)CCN(C(c2cnsc2)=O)CC(O)C1 91062,Cc1csc2ccc(CC(=O)NCCC(C)(C)NC(=O)CC3CCC4CC34)cc12 91063,C1(NC(c2c(C)cno2)=O)CCC2(C1)CN(C(=O)Cc1cccs1)C2 91064,C1(C(N2CC(CO)C(CO)C2)=O)CC12CCN(Cc1cnn3ncccc13)CC2 91065,N1(C(CC2C(C)CC2)=O)CC(NC(C2CC3(CCC3O)C2)=O)CC12CCCCC2 91066,C1(CN(C(C2CC(C)CO2)=O)CC)CCC(N(C(=O)CN2CCCC2)C)CC1 91067,CS(=O)c1ccccc1C(=O)NCC1(O)CN(C(=O)C=CC2CCCO2)C1 91068,CC(C)CC(CNC(=O)CC(C)(C)C(F)F)C(=O)NCC(C)CCCO 91069,c12n[nH]c3ccc(cc13)-c1ccc(nc1)CN2C.CC(C)CCN1CCCC1 91070,C1(C(N2CCN(C)CC2CCO)=O)CC2(CCC2)CN1C(=O)CN1CCNC1=N 91071,c1(C2(C(N(C3CCN(C(=O)C(C)(C)CF)C3)CC)=O)CC2)ccc(C#N)cc1 91072,CCCCCC(O)C(=O)NC(C)(CNC(c1cc(C)ccc1C(C)C)=O)C1CC1 91073,N1(CCCN(C)C(c2cncs2)=O)CCN(C(=O)CC2(N(C)C)CCOCC2)CC1 91074,Cc1nc(C)c(C(N2CCC(C)(CNC(C3(CF)COC3)=O)C2)=O)nc1C 91075,C1(C(=O)NC2CCN(C(c3cc(C)cc(O)c3)=O)C2)(OCC)CCC(C)(C)C1 91076,Cc1nn(C)cc1C(O)C(=O)NC1CCN(C(=O)C(=Cc2cccnc2)F)C1C 91077,c1(NC(=O)NC(c2ccc(OC)nc2)(C)C)cc(SCCF)cc(F)c1 91078,c1(CCC(=O)NC(CNC(=O)COC2CCCOC2)C2CC2)ccc(F)c(F)c1 91079,c1(CN2CCCC(C(=O)NC3CC(CC(=O)OC)C3)C2)cccc([N+](=O)[O-])c1 91080,C12(F)CC(C1)NC2=O.C1(COC)CCN(C(c2ccc(CNC(C)=O)o2)=O)C1 91081,C(=O)(C(F)C(F)(F)C(F)(F)F)N(c1c(OC)c(Cl)ccc1)C 91082,c1(C(=O)NCC2(C(=O)NCC(C(C)C)(C)F)CC(C)(C)C2)cc(C#N)ccc1N 91083,Cc1cc(C)n(CC(=O)NCC(C)(CO)NC(c2cn(C)cn2)=O)n1 91084,Cc1cc(-n2cc(-c3ccc(F)cc3Br)nn2)ncc1Br 91085,CN1CCN(Cc2ccc(N(C(CCCSCc3nc(CO)no3)=O)C)cc2)CC1 91086,C1(OC)CC(NC(N2CCN(c3cccc(C(F)(F)F)c3)C(=O)C2)=O)C12CCC2 91087,C1(NC(=O)COc2ccc(Cl)cc2)CCN(C(C2CCOCC2)=O)CCC1CO 91088,C1(C(=O)NCCCSC2CCCC2)CCCCS1.C1(=O)CCCOCCN1C 91089,C(=O)(C1=CCCSC1)NC(C(N1CC=C(C)C1)=O)CN(C)C 91090,C1(C)(NC(C(C)N=[N+]=[N-])=O)CC=CCC1.N12CCCC1CCC2=O 91091,C1(N(C)C(c2cccnc2)=O)CC2CCC(C1)N2C(C1C2CCC(=O)C12)=O 91092,c1(CC)c(C(=O)NC2CC2CNC(=O)Cn2nnnc2C2CC2)ccn1C 91093,c1(C(C#C)NC(=O)N(c2cnn(C)c2)C2CC2)cccc(Br)c1 91094,CCC(CCC(=O)N(CCC(=O)NCC(O)C(C)(C)C)CCCO)OC 91095,c1(CCCCC)nc(C(N2CC(=CCNC(=O)C(C)=C(C)CC)C2)=O)cs1 91096,c1(C(=O)NCC(N(C(CCOC)=O)C)C2CC2)ccc(S(C)=O)cc1 91097,CCCCC(C)C(=O)NC1CN(c2ncccc2Br)C1 91098,c1(OC)cc(N2CCC(NC(c3cncc(C)c3C)=O)C2)nc(CN(C)C)n1 91099,C(CNC(c1n[nH]cc1Br)=O)(CC)(CC)NC(c1cc(COC)on1)=O 91100,N1(C(C(CC)C(C)C)=O)CCC2(CCCCC2NC(=O)CN2CCCCCC2)C1 91101,c1(C(N(C2CCCCN(C(c3ccccc3Cl)=O)C2)C)=O)cncc2sccc12 91102,Cc1cn2c(C(=O)NC(C)C(CO)NC(C3(F)CCOCC3)=O)c(Cl)nc2s1 91103,C(=O)(C1=CC2C=CC(C1)C2)NCC1CCC(C(=O)NC(CCCCCC)C)CC1 91104,c1(COC)ccnc(C(=O)NCCCCCN(C)C(c2cn[nH]c2)=O)c1 91105,c1(SC)ncc(C)c(N2CCN(CCC(C)C)CC2)n1.c12cccc(c1)C(=O)N2 91106,C(=O)(CCC(C)(C)C#N)NCCC(C(C)(C)C)NC(c1ccc(OC)c(C)c1)=O 91107,C(=O)(CCCCCN=[N+]=[N-])NCC1C(CCC(=O)N(OC(F)F)C)C1 91108,CN1CCC(C(N2CCC(OCCNC(=O)CCC3CCC(=O)N3)C2)=O)C1 91109,N1(C(CC2C(C)=NOC2=O)=O)CCN(C(c2cnccc2C(F)F)=O)CC1CF 91110,C=CCCCC(=O)N1CC(CNC(c2cncn2C(C)C)=O)CC1C 91111,N1(C(C2(CC)CCC2)=O)CCC(CNC(c2ccnc(F)c2Cl)=O)C(C)C1 91112,C=CCCCC(N(C)C)NC(=O)C(c1ccco1)OC 91113,c1cnc2ccc(-n3nc(C4CCCO4)nc3CC3CC3)cc2c1 91114,N1(C(c2cnc(CC(C)C)s2)=O)CC(CNC(C2(CC(F)F)CCC2)=O)C2CC12 91115,C1(CC(=O)NC(C(N2CCC(SC)C2)=O)(SC)SC)CCCC(F)(F)C1 91116,N1(CC)CC2CCC1CN2N1CC(c2ccccc2)C1C(N)=O 91117,c1(C(=O)NCC2(C(N3CCSC4CCC34)=O)CC(=C)C2)cc2cnccc2[nH]1 91118,c1(C(N(CC(CC)NC(c2cncnc2)=O)C)=O)ccc(C)c(C)c1F 91119,C(CC1C(=O)N1)SC.C1(C)(NC(N)=O)CCN(C(=O)CC(N2CCCC2)C)C1 91120,C12(CC)CC1CN(N1CCCC1Cc1ccco1)C2 91121,C#CCC(C)(C)C(=O)N(CCC(C)NC(c1ccccc1OC(C)CC)=O)C 91122,c1(C(=O)NC2CN(C(c3cc(C)nn3C)=O)CC2(C)C)nn2c(c1C)CCCC2 91123,C(=O)(C(C)(C)CNC(=O)C(C)CO)NCc1nc(OC)oc1 91124,CC1(C)CN(C(=O)CS(C)(=O)=O)CC1C(=O)NCC1C(CO)C1(F)F 91125,N1(C(c2cc(C)nc(O)c2)=O)CC(NC(c2cn(C)nc2C)=O)CC12CCC2 91126,N1(CC(=O)N(C(CNC(CSCC)=O)C)C)C(C)=CC(C)=NS1(=O)=O 91127,c1(CCC(=O)NCCN(C)C(C2CC2(C)C)=O)ccccc1[N+](=O)[O-] 91128,C1(CNC(C(CN(C)C)NC(C2CC2C(C)(C)C)=O)=O)CCCC12CC2 91129,Cc1c(C(N2CCCCC2C2CCCC2O)=O)c(C)n2ccncc12 91130,C1(NC(c2c(CC)csc2)=O)CC2CC(NC(c3cnccc3N(C)C)=O)C2C1 91131,N1(C(c2cnn3c2N(C)CC3)=O)CCCC12CCC(NC(C1CC1F)=O)CC2 91132,c12ocnc1C2.c1(OCCNC(C(C)OCC#C)=O)ncc(C(C)C)s1 91133,Cc1nc(C)c(C(=O)NCC(O)CCNC(c2occc2Cl)=O)nc1C 91134,c1(C(N2CC(CNC(c3n(C=C)ncc3)=O)(OC)C2)=O)cccc(C(C)C)c1N 91135,CN1CCN(C)CC(C(=O)N(CCCNC(C2(n3cncn3)CC2)=O)C2CC2)C1 91136,CC(=O)CCN=C(NCC(=O)NC(=O)NC1CCC1)NC1CSC1(C)C 91137,N1(C(CC(CNC(=O)Cn2cncn2)O)=O)CCC(CO)=C(F)C1 91138,C(c1cncc(C)c1)=CC.C1(N)CCN(c2nnnn2C2C3CC4C(C3)C24)CC1O 91139,C1(CNC(C(C)(C)CO)=O)CCN(C(C2CCN(c3ncccn3)C2)=O)C12CC2 91140,c1(C(=O)NC2(CNC(CCC=C)=O)CCOCC2)cc2c(s1)CCC2 91141,C(=O)(CCS(=O)(=O)c1ccc(C)cc1)N1CC2C(N(C(C(CC)C)=O)C)C2C1 91142,N1(C(CCCC=C)=O)CCCOC(CNC(=O)C(C(C)C)N2CCCCC2)C1 91143,C1(C)(C(=O)NCC(CC)NC(=O)Cc2ccsc2Br)CCCC1O 91144,N1(CC(=O)N(C)Cc2cccc3c2OCCO3)CC=C(c2ccc(F)cc2)CC1 91145,c1(CNC(C2(NC(C(C3CCOC3=O)C)=O)CC(O)C2)=O)ccc(C#N)o1 91146,CCCCS(=O)(=O)CC(=O)N1CCCC2CN(C(c3cc[nH]c3C3CC3)=O)CC12 91147,CCS(=O)(=O)c1cccnc1C(=O)NCC1CCN(C(C23COCC(C2)C3)=O)C1 91148,c1(C(C2CCOCC2)C(=O)NCC(C)(CO)NC(C(C)SCC)=O)ccccc1Cl 91149,C1(CC(=O)N(C)CCn2cccn2)C2CCCC2N1C(c1ccc(C#N)o1)=O 91150,N1(C(CC2CN(C)C2)=O)CCCC2(CNC(c3ccc(C#N)cc3)=O)CCCC12 91151,C1(CNC(CC2CC(OC)C2)=O)CC(C)(C)CN1C(C1CCCOC1)=O 91152,c1(NC(=O)NCC2COC3(CO)CC2C3)c(C(F)(F)F)nc2ccccn12 91153,N1(C(C=CCC)=O)CC(NC(C2CCN(C(=O)OC(C)(C)C)C2)=O)C(O)C1 91154,C#CC1(CCOC)CN(C(=O)C(CCSC)NC(=O)OC)C1.C(=O)(C(C)OC)NC 91155,Cc1cc(C)c(C(=O)NCCCC2CCCCN2C(=O)C(c2ccnn2C)O)o1 91156,C(=O)(C(CC(C)(C)C#N)N1CCNC(=O)C1)NC(CC)(C)C 91157,CC(C)(C(=O)NC1CN(C(=O)Cc2ccoc2)C(C)(C)C1)C(N)=O 91158,C1(NC(C2C(C(C)C)CCC2)=O)CN(C(=O)C2=CCCC2C)C2CCCC12 91159,c1(SCC)cc(C(=O)NC2(CNC(=O)CN(C)CCOC)CCCC2)no1 91160,C1(C(CNC(C2N(CC(C)C)CCC2)=O)(C)C)CCCCN1C(=O)COC(F)F 91161,CC1CCN(C(c2cc3ccsc3[nH]2)=O)CCN1C(=O)C=C1CN2CCC1CC2 91162,c1(C(N2CC(C)(NC(c3ccccc3)=O)C2)=O)cc(F)cc(N)c1F 91163,c1(C(N(C2CCN(C(=O)COCC3CCOC3)CC2)C)=O)cccc2sccc12 91164,c1(OC)c(C(=O)N(CCC(=O)N(C2CCOC2C)C2CC2)C)cnn1C 91165,c1(OC)ccccc1C=CC(=O)NC1CCCC1CNC(c1cc(Br)n[nH]1)=O 91166,CCC(CC)C(C)C(=O)NC12CCOC(CNC(c3cc(Cl)cnc3O)=O)(C1)C2 91167,Cc1ccc2c(C(=O)N(C(C)CCNC(=O)C(CN(C)C)C(C)C)C)csc2c1 91168,C1(OC)CCCC(CNCc2cn(C(C)(C)CC(=O)OC)nn2)C1.c12conc1C2 91169,CCCC(CCCNC(=O)CC1CCN(C)CC1)NC(=O)CN(C1CCC1)C 91170,Cc1ccc2[nH]c(=NCC3CC(CNC(c4cnc(C)o4)=O)CO3)sc2n1 91171,C#CC1CN(C(=O)CNCCC)CCN1C(=O)Cc1n[nH]c(=N)s1 91172,N1(c2cc(C)nc(CO)n2)C2CCC1CC(CNC(c1cc3c(s1)CCC3)=O)C2 91173,CCCC(C(=O)NCCCNC(c1ccc(N)c(C(=O)OC)c1)=O)S(N)(=O)=O 91174,C=C=CC(C)C(=O)N(CCCN(C)C(c1ccn(-c2ccc(F)cc2)n1)=O)C 91175,C1(CNC(C(C2CCCCCC2)C)=O)C2CC1N(C(=O)CSc1nc[nH]n1)C2 91176,CCCCCCC(F)C(=O)N1CCC(CN(C(=O)CC2(O)CCOC2)C)CC1 91177,N1(C(c2cn(-c3cnnn3C)nn2)CC(=O)NCCCC)CCCCCC1 91178,c1(C)ccc(C#N)cc1.C12CC(=O)N(C1)CC1CCN(C1)C(=O)NC2C.CCS 91179,c1(CC(=O)NCC(CNC(CCC(C)N(C)C)=O)O)cc(Cl)cc(Br)c1 91180,c1(NC(C2CC(=C)CN2Cc2cc(C)[nH]c2C)=O)ccc(Br)cc1OC 91181,CCC(C)CCC(O)CC(=O)NC1CCN(C(=O)CCS(N)(=O)=O)CC12CCC2 91182,C12(CNC(Cc3cccc(C)c3)=O)CCC(C1)N(C(C1CCCCCCC1)=O)C2 91183,Cc1nnc2ccc(C(=O)NC3CCCC(NC(C4CC(F)C4)=O)C3)cn12 91184,C(=O)(CC1C(=O)Nc2ccccc21)NC1CCN(C(c2ccc(C)[nH]2)=O)C1(C)C 91185,Cc1ccc(C(=O)NC2CCC(NC(=O)CNC(=O)C(F)(F)F)C2)nc1F 91186,c1(NCC=C)[nH]c(=NCC2C(F)(F)C23CCC3)nc2c1ncn2C 91187,CS(=O)(=O)CCC(=O)NC1CC(CCNC(c2cn3ccnc3s2)=O)C1 91188,N1(C(CCC2CC(C)C2)=O)CCc2nc(CNC(=O)C(C)(C)C(C)(C)C)sc2C1 91189,N(C(=NCCNC(=O)CC1CCOC1)NC(C1(C#N)CCC1)C1CCC1)C.S(C)(=O)(=O)N 91190,C12(C(=O)NC3CN(C(C(C=C)(C)O)=O)CC3C)CCCN(CCC1)C2 91191,C(=O)(CCC(C)(C)C#N)NCC1CC(NC(Cc2c(CC)con2)=O)C1(C)C 91192,N1(C(C2C(=C)CC2)=O)CC(O)CC1CNC(c1cc(C2CC2)cs1)=O 91193,C(=O)(CCCCCN(C)C(C1CCC2(CC2)C1)=O)N1CC(OC)C(OC)C1 91194,N1(C(C=Cc2nc(C)c(C)[nH]2)=O)CCCC12CCN(C(=O)CC1COC(C)C1)C2 91195,N1(C(C(=O)NCCCCc2cccc(F)c2)=O)CCCCC(C2CCOC2)C1 91196,C(=O)(C1=CC2CCCCCCC12)NC1C(C)(C)CN(C(=O)C=CC2CCCO2)C1 91197,N1(C(c2cn(CCOC)nn2)=O)CCN(C(=O)C(C)CC=C)C2COCC12 91198,c1(C(=O)NCC(CC)NC(c2ncnc3sccc23)=O)cnc2ncnn2c1C 91199,c1(CCCC(=O)NCCN(C(C2(F)CCOCC2)=O)CC)ccccc1F 91200,C1(CC(=O)NC2CC3CN(C(C(CC)C)=O)CC32)CCCC2(CCC2)O1 91201,c1(CC)c(C(=O)NC2CCN(C(C3CC34CCCCC4)=O)C2)cnc2ncnn12 91202,C=CCN=C(NCCNS(C)(=O)=O)N(C)CC1CCCS1(=O)=O 91203,c1(C(N(CCCNC(=O)C(C(C)O)N(C)C)C(C)C)=O)ccc(S(=O)(=O)CF)nc1 91204,Cc1nc(C=CC(=O)NCC(CO)NC(=O)C=Cc2nnn(C)n2)cs1 91205,Cc1cnn(CC(=O)NCC2CC(F)(CNC(c3ccc(C(C)C)o3)=O)C2)c1 91206,N1(C(CC(C)c2ccco2)=O)CCC(C(=O)Nc2nn[nH]n2)CC1 91207,C1(NC(N2C(c3cn(CC4CCN(C)C4=O)nn3)CCC2)=O)CCc2nccn2C1 91208,c1(OC)c(O)cc(C(N2CC(NC(=O)CC3CCCC3O)C2)=O)cc1C#N 91209,c1(N2CC(C(=O)NCc3ccco3)SCC2)ccn2ncc(I)c2n1 91210,CCC(CC)(CCNC(=O)C(C)(CO)OC)NC(=O)C(CSC)N(C)C 91211,C(=O)(C(C)(C)ONC(=O)CNC(=O)CS)OC.c1(C(C2CC2)C2CC2)ccccc1 91212,C(=O)(C(F)C(C)(C)O)NCCOC1CCN(C(CC2(C(=C)F)CCC2)=O)CC1 91213,C1(C)(CC)CCC(N=c2[nH]c(=NCC3CC3(Cl)Cl)[nH]c3c2SCC3)CC1 91214,N1(C(c2cc(OCC)ncc2)=O)CCN(C(=O)CN2CCC(C)C2)CC1C(C)C 91215,CC1CN(C(C2(C)CCCN2C(=O)Cc2cncnc2)=O)CC1N=[N+]=[N-] 91216,C1(NC(c2cc(CC)[nH]n2)=O)CCN(C(c2cccc(C)c2O)=O)C(C2CC2)C1 91217,Cc1nn(CC(=O)NCC2(O)CN(C(=O)CSCc3ncc[nH]3)C2)c(=O)n1C 91218,C1(C(C)(C)C(=O)NCCNC(C2C(NC(=O)NCC)C2)=O)(CC2CC2)CC1 91219,C1(C(=O)NC(CNC(CCCC)=O)C=C)(OC)CCC(F)(F)CC1 91220,N1(C(c2cccc(S(C)(=O)=O)c2)C(=O)NC)CCCC2(CC1)CNC(=O)N2 91221,N1(C(CC(C)(C)C)=O)CCN(C(c2cnn(CCF)c2)=O)C(C2CCC2)C1 91222,Cn1nc(C(F)F)cc1C(=O)NC(c1ccccc1)CNC(C1CC2CC1CO2)=O 91223,C(=O)(CCC[N+](=O)[O-])N1CCC(C)C1CNC(=O)CC1(c2ccccc2)CCC1 91224,c1(C(N2CCCC(CNC(CCCN(C)C)=O)CC2)=O)cnn2c1OCCC2 91225,c1(NC(C(C)C(=O)Nc2cn(C)nc2C#N)=O)ncc2ccccn12 91226,c1(NC2CCCC(NC(C3CC4CC4C3)=O)C2)ncnc2sccc12 91227,N1(C(C(C(CC)CC)F)=O)CCC2(CCN(C(c3cccc(F)c3)=O)C2)C1 91228,c1(N(C)CC2CSCCO2)ccc(S(=O)(=O)N2CCCC2CN(C)C)cc1Cl 91229,C(=O)(C1=CCCSC1)NC(C1CCCN(C(CCOC(C)=O)=O)C1)C(C)C 91230,c1(NC(C2N(c3nc(C)c(F)cn3)C3C(C2)C3)=O)cc(F)c(C)c(Br)c1 91231,c1(C(=O)NC2C3(CN(C(CC(=O)OCC)=O)C3)CC2)cccc2c1OC(F)(F)O2 91232,CCCN=C(NCC1CN(C2CCCCO2)C1)N1CCC2(CC1)C(OC)CC2OC 91233,N1(C(C=CCOC)=O)CCC(NC(c2ncnc(OC)c2Cl)=O)CC1C1CC1 91234,C(=O)(C(C)(C)C(C)NC(c1sccc1C)=O)N(CCCCCOC)C 91235,c1(C(N2CC(N(C(C3(C)N(C(C)=O)CCC3)=O)C)C2)=O)ccc(P(C)(C)=O)cc1 91236,C1(C(N2CCC(O)(C(CNC(CCN(CC)CC)=O)(C)C)C2)=O)CCCCS1(=O)=O 91237,C=CC(CC)CC(=O)N1CCCC1C(C)(C)NC(=O)C(=Cc1c[nH]cn1)F 91238,c1(-n2cc(NS(CC)(=O)=O)nn2)ccc(OCCN(C)C)cc1 91239,c1(C(=O)NCCc2cc(C(N3CC(C(=O)OC)C3)=O)no2)nccnc1N 91240,c1(CCNc2cccc(OC)c2C)ccc2cn(C(F)F)nc2c1 91241,CC(C)(C)C1=NOC(C(N2CC(C)(C)OCC2CNC(=O)C2=CCCCC2)=O)C1 91242,CCCCC(C(=O)NC)NC(C1CC(O)(CNC(=O)CCC(=O)C2CC2)C1)=O 91243,N1(C(CCCCOC)=O)CC(F)(F)CC1CC(=O)NC1CC(=O)N(C)C1 91244,C(CCCCC(=O)NCc1ccnc(C(=O)NCC(O)C2(Cl)CC2)c1)OC 91245,C1(C)(C(N2CC(C(C)NC(=O)NCC3CC3)C2)=O)CCOC(C)C1 91246,C1(CNC(c2c(SCC)cncc2)=O)CCCCN(C(=O)CN2CCSCC2)C1 91247,C1(O)(CC)CCCN(C(C2(C)CC(NC(=O)C#CC(C)(C)O)C2)=O)CC1 91248,c1(C(=O)NCC2CCN(C(CC(C)(C)OC)=O)CC2)cccc(C)c1C#N 91249,C1(CC(=O)N(CC(CNC(CSCC(C)C)=O)C)C)CCC(=O)C1 91250,C1(C(C)C)CC(C(=O)NCC(=O)NC(c2ccccc2)C(C)(C)C)=NO1 91251,C1(NC(c2c(N(C)C)nccc2)=O)CN(C(C2NC(=O)NC2=O)=O)CCC1O 91252,C(=O)(C1=NOC(C)C1)NCc1occ(C(N(CC#C)CC)=O)n1.C1(O)CC1 91253,c1(CN2CCOCC(C(=O)OC)C2)cc(C)c(OCC#C)cc1C 91254,N1(C(c2c(OCC)[nH]cc(C)c2=N)=O)CC(NC(=O)COCCSC)CC(C)(C)C1 91255,c1(N(CC(CC)C)C(C2CCCCN2C2CCCC2)=O)nc(C(C)C)nc(C)c1Br 91256,C1(NC(CS(C)(=O)=O)=O)CC1C1CCCN(C(c2ncnc3c2CCCC3)=O)C1 91257,c1(N(CC(CC)C)C)nc(=NC2CC2F)[nH]c2cc(OC)ccc12 91258,C1(NC(C(N2C(=O)CCC2=O)C)=O)C2CC1N(C(N)=O)C2.C12(CC1)C(=O)N2 91259,C1(C(=O)NCC(CC(C)C)NC(=O)Cc2cc(Cl)ccc2O)CC(C2CC2)=NO1 91260,N1(C(C)C)CCN(C(=NCC2CCCCC2)NCc2ccc(F)cc2)CC1=O 91261,N1(C(C(CC)SC)=O)Cc2n[nH]cc2C1C(=O)N1CC(C)(C)C1 91262,N1(C(CSCCCC)=O)CC(N(C(=O)C(C)CC)C)C(C)(C)C1 91263,N1(C(C2C(C)OC(=O)N2)=O)CC(NC(=O)CCc2ccccc2Cl)CC(C)C1 91264,CCC(O)CC(=O)NCCCCCN(C(=O)C(c1ncccc1C)(F)F)C 91265,c1(C(=O)NCC2CCN(C(=O)COC3CCOCC3)C2)cnc2[nH]cnc2c1 91266,C(C(CNC(C1CCC1c1nc[nH]n1)=O)C(F)(F)F)NC(COC(C)C)=O 91267,C1(=O)CCCC(=O)N1.C1(N(C)C)CC(F)(C(=O)NCCNC(=O)OC(C)(C)C)C1 91268,c1(OCCOCCOC)ccc(NC(C2CNC(C)(C)C2)C)cn1 91269,c1(C(N(C)CC2CCCC(NC(=O)Cc3cscn3)C2)=O)cc2cc(F)ccc2[nH]1 91270,Cc1cc(C(=O)NC2CC(CCNC(C3(CO)COC3)=O)C2)c(C)c(C)c1 91271,C12(C(=O)NCC(C)(C)NC(c3c(C)c(O)ccc3)=O)CCCN1CC(O)C2 91272,N1(C(CCC2(NC(C(CC)C(=O)OC)=O)CCC2)=O)CCC(F)(F)C(C)C1 91273,c1(NC2C(C)(C)COC2)c(C#N)cnn1C1CC1CO 91274,N1(C(C(C(C)O)C)=O)CCOC2(CCS(=O)(=NC(=O)C3CCCCC3O)CC2)C1 91275,Cc1cc(C(=O)N(C)CC2CCCN(C(C3CCC3(C)C)=O)C2)cc(O)c1 91276,c1(C(N2CC(CCCCNC(COC(C)C)=O)C2)=O)ccc2ncnc(O)c2c1 91277,Cc1cc(=O)c(C(=O)NCCCCNC(C2CCCC23CCC3)=O)c[nH]1 91278,N1(C(C(C)O)=O)CCC(C2(O)CN(C(=O)CC3CCC4(CCC4)O3)C2)CC1 91279,C1(C(=O)NCC2CC(CC)C2)CN(C(=O)CCCCCF)CC(C)(C)C1 91280,N1(C(CCC(C)C)=O)CCCC2CN(Cc3cc(Cl)ccc3F)CCC12 91281,c1(OC)ccccc1OCC(N1CCCC(COC(C2CCCC(=O)C2)=O)C1)=O 91282,c12[nH]c3ccccc3c1NC2=O.c1(CC)ncc(CNC(C2(CC)CCC2)=O)s1 91283,N1(C(C2(c3c(C)n(C)nc3)CC2)=O)CCCCC(N(C)C(C2CCCO2)=O)C1 91284,C1(NC(C2C(C(C)O)C2)=O)CCCN(C(=O)CC2(C(F)(F)F)CCC2)CC1 91285,C1(NC(C23CC(CCC)(C2)C3)=O)CCN(C(c2cc3sc(C)cc3s2)=O)CC1(C)C 91286,c1(C(N(C2CN(C(C3C(OC)CCC3)=O)CC23CC3)C)=O)cc2sccc2n1C 91287,C12(CNC(C(C)OC)=O)CC(NC(=O)CSc3n[nH]c(O)n3)C(CO1)C2 91288,C(=O)(C1=CC2CCCCCC12)NCCCC(C)NC(c1cc(CC(C)C)on1)=O 91289,N1(CC)CCCC(C(N2CC=CC2CNC(=O)C=Cc2ccc(Br)s2)=O)C1 91290,c1(OC)cccc2c1C(C(=O)NC(C1CCCN1C(=O)COCCF)(C)C)CC2 91291,C1(C(NC(=NCCC2CCSC2)NCCS(C)(=O)=O)C)Cc2ccccc2O1 91292,c1(C(N2CC(N(C(=O)CC3CSC3)C)C(O)CC2)=O)nccn2ccnc12 91293,N1(C(Cc2ccn(CC)n2)=O)CC2CN(C(=O)C=Cc3cccnc3C)CCC12 91294,N1(C(C=C(C)C(F)F)=O)CCC(NC(=O)CNC(C2CCCN2C)=O)C1 91295,C(C)(C(C)(C)C(=O)NCCC(O)C(F)(F)F)NC(C1(CC)CCCCO1)=O 91296,N1(C(C2=NNC(=O)C2)=O)CC2CCCC(NC(c3noc4c3CCCC4)=O)C2C1 91297,Cc1ncnc(C)c1C(N1CC(CNC(C2CC(Cc3ccccc3)CO2)=O)C1)=O 91298,N#Cc1c(F)cc(C(=O)NCc2ccc(CNC(=O)CCC(F)F)cc2)cc1F 91299,C1(COC)CC(CNC(=O)CC2CC(=O)NC2=O)N(C(c2cc(Cl)c[nH]2)=O)C1 91300,N1(C(C(CC(C)C)F)=O)CCN(C(c2ncc(F)cc2F)=O)CCC1C 91301,C1(C#N)(OC)CC(C(=O)NC2(C(=O)NCCC#CCO)CCC2)C1 91302,C(=O)(C(F)CCC(C)(C)C)N(CCN(C(C(N1CCCC(C)C1)=O)C)C)C 91303,N1(C(C(COC)N(C)C)=O)CCN(C(c2cn(C)c(=O)n2C)=O)C2COCC12 91304,N1(C(C(CN)N)=O)CCC2(CC1)CC2NC(c1cc2ncccc2[nH]1)=O 91305,CC1(C)CC(CNC(=O)COCCCF)CN1C(=O)C1=NNC(C(F)(F)F)C1 91306,N1(C(C(C)=C2CC2)=O)CC2C(NC(c3c[nH]nc3F)=O)CS(=O)(=O)C2C1 91307,CC(C)(C)C(=O)N1CC(C)(CCC(=O)NCc2cscn2)C1 91308,C(C(=O)N1CC(CN(C)C(c2ccc(-c3cc[nH]n3)s2)=O)C1)(C(C)C)OCC 91309,c1(C(=O)N(CC(=O)Nc2cccnc2)C2CC2)ccc2nonc2c1 91310,c1(C(=O)NCCC2(O)CCCN(C(c3c(C)nsc3)=O)C2)nc2c(s1)CCCC2 91311,CC1(CNC(CCCOC(C)(C)C)c2nnnn2C2CC2)COc2ccccc2O1 91312,O(NC(=O)C(Cc1cnc[nH]1)NC(c1ccc(F)cc1)=O)Cc1ccc(Cl)cc1 91313,O=[N+]([O-])c1cccc2c1CCN2S(=O)(=O)CCCCS(=O)(=O)Nc1ccon1 91314,C1(O)(CNC(C(c2cccc(OC)c2)C)=O)CCCN(C(C2(SC)CC2)=O)CC1 91315,c1(N2C(CN(C)C(C3CSCN3C)=O)CCC2)ccc(C#N)c(C(F)(F)F)n1 91316,C=CC(C)(CCOC)C(=O)NCC1=CCN(C(=O)CCC2CCN(C)CC2)CC1 91317,N1(C(c2c(C)coc2)=O)CCC(CN(C(=O)CC2CCC3CC23)C)CC1 91318,c1(NC(C23CCC(c4ccccc4)C2C3)=O)cccnc1Br 91319,N1(C(c2c(CC)cns2)=O)CC(C2CN(C(C3CCCC3c3cnn(C)c3)=O)C2)C1 91320,N1(C(=O)Cc2nc3c([nH]2)CCCC3)CCC=C(C(=O)O)C1 91321,c1(C(N(CC(C)CNC(=O)COC2CC2)C)=O)ccc(C=C2CCCCC2)o1 91322,C12(NC(C3(C)NC(=O)NC3=O)C)CCC1CS(=O)(=O)C2 91323,c1(OC)cc(OC)c(C(=O)O)cc1F.C(=O)(C(C)CN1CCOCC1)NCC 91324,CC1(C)C(NC(c2ccc[nH]2)=O)C(C)(C)C1NC(=O)CCc1cncnc1 91325,c1(CNC(c2nnsc2C2CC2)=O)nccn1-c1ccccc1 91326,c1(CC)cc(N)ccc1C(N1CCC(F)C(NC(=O)Cc2c(C)nn(C)c2C)C1)=O 91327,N1(C(C(C)C)=O)CCC(CC(C)NC(C2CCCN2C)=O)CC1 91328,N1(C(C2CC(=C)C2)=O)CCCC1C(=O)NCc1ccnn1C 91329,C1(NC(CC2C(C)(C)N(C(=O)Cn3cncn3)CC2)=O)CCC(C2CC2)CC1 91330,C1(NC(C2(COCC)CC2)=O)CC1C1CN(Cc2ccccc2)C1 91331,c1(C(C(=O)NCC(CCC)NC(c2cnn(C)c2F)=O)=O)ccc(F)c(F)c1 91332,c1(C(c2ccccc2Cl)C(N2CCC(c3ccco3)C2)=O)cc(Cl)cc(Cl)c1 91333,c1(C(=O)NC2CCC(CCNC(Cc3n(C)nnc3)=O)C2)cc(=O)c(O)c[nH]1 91334,C(C)(CNC(=O)Cn1cc(C(C)O)nn1)(CC(C)C)NC(C(CCOC)OC)=O 91335,Cc1coc(C)c1CNC(C)C(c1ccccc1)NCC1CCCN1C 91336,C1(C)(CCNC(C(CC=C)C)=O)CCN(C(c2ccc3c(c2)CC3)=O)CC1 91337,Cc1cc(O)nc(C)c1C(N1CCN(C(c2onc(C)c2C)=O)CC(C)C1)=O 91338,C=C(CC)CN=C(NCc1cccs1)NCC(C)C(F)(F)F 91339,CC1CCc2[nH]nc(C(N3CCC(NC(=O)Cc4ccno4)C3C3CC3)=O)c2C1 91340,C1(NC(c2cccc(-n3cccn3)n2)=O)CCOC(CNC(C2CC=CC2)=O)C1 91341,c1(C(C)CNC(=O)NCC(C2CCOC2)OC)ccccc1Cl 91342,C1(CNC(C(CCCC)(C)F)=O)CN(C(c2coc(CO)c2)=O)CCC12CCC2 91343,CCS(=O)CC(=O)NC1(C(=O)NCCOCC(F)(F)F)CCSC1 91344,c1(OCC(=O)NCC2C(NC(COCC)=O)C2)cccc(C(N)=O)c1 91345,c1(C(c2n(C3CCC3)nnn2)NC2CS(=O)(=O)C2)ccc(F)c(Cl)c1Cl 91346,C1(NC(c2c(C(N)=O)nccc2)=O)CCCC(NC(=O)CCCn2ccnn2)CC1 91347,C(c1ccncc1)=CC(N1C(C(=O)NCC(C)OCC=C)CC1C)=O 91348,Cc1cnc(C=CC(=O)NCCC(C(C)C)NC(c2ccccc2N)=O)[nH]1 91349,C12(NC(C(C(C)C)SCC)=O)CCCC(NC(c3ccc(C)cc3N)=O)(C1)C2 91350,C=CC(F)(F)C(=O)N(CCNC(c1ccccc1N(C)C(C)=O)=O)CC 91351,N1(C(C(C(C)NC(C(=O)NC)=O)C)=O)CCCC2CN(C)CC12 91352,C1(N(C(=O)CC2CC(F)(F)C2)CC)CCCN(C(=O)C(C)CNC(N)=O)C1 91353,N1(C(=O)OC(C)(C)C)CCCC(c2cn(CCNC(C3C4CCCC34)=O)nn2)C1 91354,C1(NC(CC(=C=C)C)=O)COC2(CCCN(C(c3cc(NC)ccc3Cl)=O)C2)C1 91355,N1(C(C=CCC)=O)CCC2(CCCC2NC(=O)Cc2c[nH]c3cc(Cl)ccc23)C1 91356,N(C(=NCCCc1cccs1)NC(c1ccc(F)c(F)c1)C)C(C#C)CCC 91357,N1(CCCC)CCN(C(c2cc(CNC(=O)Cn3nccn3)ccn2)=O)CC1 91358,C1(NC(C(C)O)=O)CCCC1NC(=O)Cc1cncs1 91359,c1(C(=O)NCC23OCCC(NC(C(C(C)C)C)=O)(C2)C3)nnn2c1CCCCC2 91360,c1(OC)cc(N)c(F)cc1S(=O)(=O)Nc1cc(S(=O)(=O)F)c(Cl)cc1F 91361,c1(-c2onc(-c3ccc(-c4ccc(C)cc4)cc3)n2)ccc2ncccc2c1 91362,C1(C(C)C(=O)NCC(C)(C)F)CCN(C(=O)C(C)(C)n2ccnn2)C1 91363,C(C)(CO)(C(=O)NCC1(O)CN(C(=O)COc2cncc(Cl)n2)C1)OC(C)=O 91364,CC1CN(C(=O)C(=O)Nc2ccncc2Cl)CCN1CCN1CCOCC1 91365,Cc1cc(Cl)cc2cc(C(=O)N(CC(O)CNC(C3CS(=O)(=O)C3)=O)C)[nH]c12 91366,C(=O)(C1=CCCOCC1)NCC1OCCN(c2ncc(C(C)=O)cc2C)C1 91367,N1(C(C(OCC)CC(=O)N(CCCF)CCl)=O)CC(C)(OC)C1 91368,CC(C)C(C)CC(=O)N1CC(C(=O)NCCCCn2ccnc2)CC(C)C1 91369,N1(C(c2c(NC(C)=O)c[nH]c2C)=O)CC(NC(=O)CC(C)(C)F)C2(CCC2)C1 91370,N1(C(C(C(=O)OCC)CC)=O)CCC2(CC(C(N3CC(O)C(O)C3)=O)C2)C1 91371,C=CC(C)(O)CC(=O)N1CCC(CC)CC1.n1(CC)cc(C(C)(C)CC)nn1 91372,C1(C(=O)OC)CCN(C(=O)NC(c2ccc(Cc3nn[nH]n3)cc2)=O)C1(C)C 91373,c1(CC)ccc(C(=O)NC)s1.C1(=O)C(CC2CC2)N2CCC(C2)N1 91374,N1(C(c2c(C)cc[nH]2)=O)CCC(C2(NC(C3C4COCC34)=O)CC2)CC1 91375,C=CCCCCCCC(=O)NCC(=C)CCNC(C1CCCCC12CCC2)=O 91376,c1(Cn2cc(C3CCN(C(c4ccc(C(C)=O)s4)=O)C3)nn2)ccc(Cl)nc1 91377,c1(NC(C(C(C)NC(=O)C(C)(Cl)Cl)C)=O)cc(O)cc(F)c1 91378,N1(C(c2cc(C(N)=O)[nH]c2)=O)CCCC2(CCCN2C(c2cc(O)ncn2)=O)C1 91379,c1(C(N2C(C(N)=O)C=CC2)=O)ccc(S(=O)(=O)N2CC3CCC(C2)NC3)cc1 91380,c1(NC(N(Cn2c(C)cc(C)n2)CC2CC3CCCC23)=O)ccc(Cl)cc1O 91381,c1(C(=O)Oc2ccnc(C(=O)N(CC(C)NCCC)C)n2)ccc(C)c(C)c1O 91382,C(=O)(C1CCCc2scnc21)NC1(CN(C(C2C(C)C2)=O)C2CC2)CCC1 91383,c1(C(C(=O)N(CCCN(C(=O)CSCc2cccnc2)C)C)=O)ccc(Cl)s1 91384,C1(C(=O)NCCNC(C(CC)c2ccccc2)=O)CCC2(CCOCC2)CO1 91385,C1(COC)CN(C(c2ccc(Br)nc2F)=O)CCN1Cc1scnc1Cl 91386,c1(CNC(c2cc(C)on2)=O)ccnc(C(N2CCC(C(C)O)C2)=O)c1 91387,C#CCCCC(=O)N1CC(F)(C(=O)NC(C(=O)OC)C2CCC2)C1 91388,Cn1nc2c(c1C(N1CC3=C(C1)CN(C(c1c[nH]ccc1=N)=O)C3)=O)CSCC2 91389,S(=O)(=O)(c1cccc([N+](=O)[O-])c1C#N)NC(COCC)CC 91390,N1(C(C(=O)Nc2snc(C(C)(C)C)n2)=O)CC2CCC2(C(=O)O)C1 91391,Nc1cc(C(=O)NCc2cc(O)nc(CNC(=O)C=CCO)n2)cc(O)c1Cl 91392,C1(C(=O)NCC(C)(CO)NC(c2cc(F)c[nH]2)=O)CC2CCCC(C1)C2 91393,C(=O)(C1=CC2(CCOC2)C1)N(CCNC(C1(C)CC2CCC1O2)=O)CC 91394,CC1(C)CCCC(CNC(=O)CC2CCCC(NC(c3scnc3Cl)=O)C2)O1 91395,C1(NC(c2c[nH]cc2C2CC2)=O)CCCCCC1NC(C1CCSCC1)=O 91396,c1(CC(N2CC(n3cc(-n4nc(C)c(Cl)c4)nn3)C(C)C2)=O)cccc(Cl)c1C 91397,C=C(Br)CC(C)(C)C(=O)NCCC1CCC(NC(c2cnnn2CC)=O)C1 91398,CC(C)(O)C(C)(C)CNC(=O)NCC1COC2(CCC2)C1 91399,N1(C(COC)=O)CCC2(CC1)CC(NC(=O)NC(C)(CCBr)c1nn[nH]n1)CCO2 91400,C1(C(c2n(C(c3ccccc3)C)nnn2)NCCC2CCC2)(OC)CCSCC1 91401,C(=O)(CCCCC(C)CC)NCC(CCC)C(=O)NCc1nnsc1C 91402,c1(CC)ccc(NC(=O)NCCC(=O)NCC2CCCCN2C)cc1 91403,CCCCC(O)C(C)C(=O)N1CCCCC1CC(=O)NC1CC(OC(C)C)C1 91404,c1(C(=O)NC2CN(C(C(COC)OC)=O)C3(C2)CCC3)cc2nc(Cl)ccc2s1 91405,C1(CNC(c2nc(COC)sc2)=O)C2CCC(C2)N1C(=O)CC1C=CCCC1 91406,C(C)(C)(CC(F)C(=O)NOC1CCCCC1)NC(CC(CCC)C)=O 91407,C(=O)(c1c(C)[nH]c(=O)[nH]c1=O)NC1CCC(NC(c2cc(OC)c(C)cc2)=O)C1 91408,Cc1nc2c(C)cc(C(=O)N(CC(C)NC(=O)CCC3CC3)C)cn2n1 91409,N1(C(C(=O)NCCc2cccc(F)c2)=O)CCc2nc(O)cc(Br)c2C1 91410,C1(CS(=O)(=O)NC(C2(CC=C)CCCCN2)=O)CCCC2(CCC2)O1 91411,c1(CNC(C2C=CC(NC(c3cnc(Cl)s3)=O)C2)=O)cccc(O)c1 91412,C(CC(C(=O)NC1C(C)C1(C)C)NC(=O)CC1CCSC1)=CC 91413,c1(C(N2CC(C)(NC(c3cn(CC(CC)O)nn3)=O)C2)=O)ccc([N+](=O)[O-])[nH]1 91414,C=CCC(C)C(=O)NOC(CC(C)C)C(=O)N1CCCC1CC1CCC1 91415,CC1(NC(=O)CCCc2csc(=N)[nH]2)CCCN(C(c2csc3cncn23)=O)C1 91416,C12(C(=O)NCCCCNC(C3(c4ccccc4C(=O)O)CC3)=O)CCN(CC1)C2 91417,C=CCCC(F)(F)C(=O)N1CC(C(=O)N(CC(C)O)C2CC2)C2(CCC2)C1 91418,CC1(C)C(C(=O)NC(CC(N2CCC(F)(F)C2)=O)C2CC2)C1(F)F 91419,S(=O)(=O)(c1ccc(Br)cc1NC(c1ccc(C2CC2)cn1)C)NC(CC)CO 91420,N1(C(C(=CC2CCCC2)C)=O)CC2CCOC2(CNC(c2cncc(C)n2)=O)C1 91421,N1(C(C(C=CCCC)O)=O)CCOCC(CNC(=O)C(F)(F)CN(C)C)C1 91422,Cc1ccc(F)c(CNC(C2CCC(CNC(C3CC4CCC4C3)=O)C2)=O)c1 91423,c1(C(=O)OCC)ccc(C(=O)NCC#CCNC(C2(C)CCCC2C)=O)nc1 91424,CCCC(CCC)C(=O)NC1CC(O)CN(C(=O)C(C2CCOCC2)F)C1 91425,N1(C(CC=CC(C)(C)C)=O)CCC2(NC(=O)Cc3ccn(C4CC4)n3)CCCC12 91426,C(=O)(C(CC(F)F)C1CCC1)N(CCNC(C(C=C)(C)O)=O)CC 91427,N1(C(C(C)=CC(C)(C)C)=O)CCC(C)(C)C1C(=O)NCc1nc(C(N)=O)no1 91428,CC(C)CCC(O)C(=O)N(C1CCN(CCCO)C1)CC1CCCCC1 91429,C1(C(=O)NCc2c(C(=O)NC(c3cnccn3)C)scc2)CC(=O)CCO1 91430,C1(N(C(=O)CC2CSCCS2)CC)CC2CCC(C1)N2C(=O)Cc1ccsc1 91431,N1(C(C2C(NC(C=CCN(C(C)(C)C)CC)=O)COCC2)=O)CCOCC2(CC2)C1 91432,c1(C(N2CCC(O)(NC(=O)OCC)CC2)C(=O)NCCC)nc(Br)c(C)cc1Cl 91433,C#CCCN=C(NCC(C)Cc1cccs1)NC1CN(CC(=O)OCCOC)C1 91434,C1(CC(=O)N(CCNC(C2CCN(CC(F)(F)F)C2)=O)CC)CCCOCC1 91435,Cc1cc(-c2nn[nH]n2)cc(C)c1CC(=O)Nc1c(Cl)cc(Cl)cc1Cl 91436,c1(C(CC)C)ccc(C#N)c(NC2CCN(C(c3cc(C)nc(Cl)c3)=O)CC2C)n1 91437,CCN=c1[nH]c(C)c(C(N2CCCCC2C2CCN(CC(N)=O)C2)=O)s1 91438,c1(C(N2CC(C)N(C(c3cnc(C(F)F)nc3)=O)CC2)=O)cccc2ccsc12 91439,CC1CC(CNC(C2(C(F)F)CCC2)=O)CN1C(=O)COc1ccccc1Cl 91440,Cc1cc(=NC(=O)C(=O)N2CCN(C(c3nnc(S)n3C)=O)CC(O)C2)[nH]o1 91441,Cc1ccc(C)c(CC(=O)NCCCC(C)NC(C2CC2CC(C)(C)C)=O)c1 91442,C1(C(N2CCC(N(C(CN(C(C)=O)C)=O)C)C2)=O)COCCN1C 91443,N1(C(C=CCCC)=O)CCC(NC(c2csc(CC)n2)=O)CC1C 91444,C=CC(CCC)CC(=O)N1CCOC(CN(C(=O)CCNS(C)(=O)=O)C)C1 91445,n1(CC)cc(Br)c(C(N2CC(NC(=O)C=Cc3cncn3C)C3CC23)=O)n1 91446,c1(COC)nc(C)c(C(N2CC(CNC(=O)CC3CCC(=O)C3C)C2)=O)s1 91447,N1(C(Cn2ccc(C)n2)=O)CC2CN(C(c3ccc4ncnn4c3)=O)CC2C1 91448,c1(C(=O)NCCC2CC(NC(C3CC(O)C(F)C3)=O)C2)cncc2c1CCCC2 91449,c1(C(=O)NCCC(CCNC(CC=CC)=O)C)c[nH]cc(Br)c1=N 91450,N1(C(c2nc(C(=O)OC)sc2)=O)CC(OC)C(NC(C23CCCC2C3)=O)C1 91451,C(CCC(C)(C)CN=C(NCc1cccs1)NCc1cccs1)N(C)C.C1CCCCC1 91452,Cc1cccc(C=CC(=O)NC2CC(NC(=O)C3=CCCCC3)C23CCC3)c1 91453,C(=O)(C1CC=Cc2ccccc21)NC(C1CCCN1C(=O)CSCC(F)F)C 91454,N1(C(C(COC)C)=O)CC(NC(=O)C2=CSCCO2)CC12CCC2 91455,C(=O)(C1=CCCCC1C)N1CC(O)(CN(C(CCCOC)=O)C)C1 91456,C1(C(N)=O)CCCN(C(=O)CC2(CNC(c3c(CN(C)C)cco3)=O)CC2)C1 91457,C1(CNC(C(CC)SC)=O)CCCN(C(=O)CSc2ncccn2)CC1 91458,N1(C(=O)Nc2c(C(=O)NC)n(C)nc2)CCC2NC(=O)NCC2C1 91459,N1(C(C(CC)C(C)O)=O)C2CCCC1CN(C(=O)C(C)CC1CCCCC1)CC2 91460,C1(CNC(COCCC)=O)CC2COCC2N1C(c1c(F)ccnc1F)=O 91461,c1(C(N2CC3CC2(c2nc(C)no2)C3)C(=O)NC(CC)C)ccc(C)c(Cl)c1 91462,C(=O)(C(O)C1=CCCCC1)N.C1(OC)CC2N(C1)C(=O)CCCC1(CCC1)NC2 91463,C1(NC(C2(CC)CCCCC2)=O)CN(C(=O)CC2CCN(C)C2)CC1N=[N+]=[N-] 91464,N1(C(C(C(CC)O)C)=O)CC=C(CCNC(c2ccnn2CC2CC2)=O)CC1 91465,CC1(C)CCN(C(=O)CC2CCC(=O)NC2)C1C(=O)NC1CC2CCC1O2 91466,CC(O)(CC(=O)NC1CC1C(=O)NCc1cc(F)c(Cl)cc1Cl)CC(=O)O 91467,C(=O)(CC(C(C)CC)NC(C1CC(CF)C1)=O)NCC(C=C)(C)C 91468,C1(CCOC)(NC(=O)CCn2cncn2)CCN(C(C2CCC(C)O2)=O)CC1 91469,Cn1ncc2ncnc(NCC3CC(F)(CNC(C45CC4COC5(C)C)=O)C3)c12 91470,c1(C(=O)OC)cc(F)cc(Br)c1NC(=O)CNc1n[nH]cc1-c1ccc(F)cn1 91471,C1(OC)(OC)CCC1C(=O)NC1CCCC1C(=O)NCCc1ccccc1 91472,c1cc2[nH]c(=NCc3ccc(C(F)(F)F)s3)[nH]c(=NCC3CCCSC3)c2[nH]1 91473,n1(CC)nccc1S(=O)(=O)N1CCCC1c1cn(CC2CCCO2)nn1 91474,C1(n2cc(CC(COC)O)nn2)CON(C(=O)C2(c3csnn3)CC2)C1.C(C=C)=CC 91475,CC(C)(C)CC(O)CC(=O)N1CC=CC(C(=O)NCc2ccncc2)C1 91476,C1(C(N2C(CCC(=O)N(C3CC3C3CC3)C)CCC2)=O)OC2CCC1C2 91477,CCC(C)(CC)C(=O)NC(CC(=O)NCCC(C)(C)OC)C1CC1 91478,CCCC(O)C(=O)NCCSCC(=O)NCc1cnn(C(C)C)c1 91479,c1(CC(=O)NCCC2CCN(C(C(CSC)OC)=O)C2)ccc(CC(C)C)cc1 91480,N1(CC(N2C(CNC(Cc3cc(C)ns3)=O)C=CC2)=O)CCNC(=O)C1 91481,Cc1ccc(C#N)c(NC(C2C3CC2N(S(=O)(=O)c2ccncc2)C3)=O)c1 91482,c1(C(=O)NCc2cc(F)ccc2-c2ccc(Cl)cc2)n[nH]c2c1COCC2 91483,Cc1c(F)cccc1S(=O)(=O)N1CC(NC(=O)C2=COCC2)CC(C)C1 91484,N1(C(COC2CCCC(C)C2)=O)CCN(C(=O)Cc2ccc(F)nc2)CCC1C 91485,n1(CCC(N2C3C(NC(C(C)(C)F)=O)CC(C3)C2)=O)ccc2ccccc12 91486,c1(C(=O)OC)sc2ccccc2c1CC(N1CC=CC(NC(=O)C(C)(C)O)C1)=O 91487,C1(CCNC(C=CC(=O)OCC)=O)CCCCC1C.C1(C)(C)CC=CC(=O)N1 91488,c1(C(=O)NCC2CN(C(CC3(C)CC3)=O)CC2O)coc2ccc(F)cc12 91489,C=CC(C)(CC)C(=O)N1CCN(CC(N2CCCN(C(=O)CO)CC2)=O)CC1 91490,c1(C(N2CC3C(CNC(CC(CC)OC)=O)C3C2)=O)nn(C)c2c1CCC2 91491,C(=O)(C(O)CC(C)(C)C)NC(CC)CC(=O)NC1CC2COCC(C1)C2 91492,N1(C(C=CC(C)NC(COCC(=O)NC)=O)=O)CCCN(C)C(=O)C1 91493,N1(C(CC=C)=O)CC(CNC(=O)C(C2CC2)SC)CC12CCC2 91494,c1(OCCOC)cc(C(=O)NC2CCCC2C(=O)Nc2nc(C)cs2)ccn1 91495,C1(C(=O)NCCOCCC(=O)NC2(C(N)=O)CC2)C2CCC(F)C12 91496,C#CC1CN(C(=O)C(COCc2cn(CC(=O)OCC)nn2)C(F)(F)F)CCN1C 91497,C1(OCC)CC2(C1)CC2C(=O)NCC(C)NC(c1cncnc1)=O 91498,C(=O)(C(CC)CCCC)NCC1N(C(c2cccc(SCCCC)c2)=O)CC=C1 91499,C12(CNC(c3cncc(OCC(F)F)c3)=O)CCC(CC1)N2C(=O)C=C1CCC1 91500,Cn1[nH]c(=NC(=O)NCCC2CCC3(CCCC3)O2)cc1C1CC1 91501,C1(OC)CC2CC1CN(C(=O)CC1(NC(c3cnncc3C)=O)CC1)C2 91502,c1(C(=O)NCCCOCCCNC(C2CCC(C)S2)=O)cccc(Cl)c1 91503,C(C(=O)N=c1c(Cl)c[nH]cc1I)c1c(C#N)scc1.c1cc2cc(F)ccc2[nH]1 91504,c1(N(CCC(=O)NC)C)[nH]c(=NC(C)c2cc[nH]n2)nc2c1ncn2C 91505,c1(CC(=O)NCC(C)N(C)C(C2CN3CCC2CC3)=O)ccc(Br)cc1F 91506,c1(C(N(CCNC(C2CCCCC2F)=O)C2CC2)=O)ccccc1F 91507,C1(NC(C(N)=O)=O)CCCC(NC(c2cc(Cl)cc(Cl)c2)=O)CC1 91508,C(=O)(C(C)(C)C(=O)N1CC(NC(C2C3CN(CC(F)(F)F)CC23)=O)C(F)C1)NC 91509,c1(C(=O)NC(CN(C)CC2(CCC=C)CC2)C)n[nH]c(C)c1[N+](=O)[O-] 91510,Cc1cc(O)ncc1C(=O)NC1CC1CNC(c1ccc(O)c(Cl)n1)=O 91511,C1(C(=O)NCCCC(C)NC(c2nn(C)cc2Cl)=O)CC12CC(C)(C)C2 91512,N1(C(CONC(c2cncc(C)n2)=O)=O)C2CCC1CC1(C2)N=N1 91513,N1(C(CC(=C)C)=O)CCC2(C1)CN(C(c1ccnn1C(F)F)=O)C2 91514,Cc1nsc2ncc(C(N3CCCC4(C3)CN(C(C3CCCOC3)=O)C4)=O)cc12 91515,c1(CC)ccc(C(=O)NCC(CO)NC(=O)COCCCC(C)C)c(OC)c1 91516,CC1CCC(C)(C(=O)NC2CC(NC(c3cnc(Br)s3)=O)C2)C1 91517,c1(NC(C2N(S(CC=C)(=O)=O)CCSC2)=O)c(F)cc(F)cc1[N+](=O)[O-] 91518,c1(C(=O)NCCOCC(=O)NCC=CCNC(C2CC(C)(O)C2)=O)ccc(N)cc1 91519,c1(C(=O)NCC(C(C)C)NC(c2cc(OC)ncn2)=O)sc2cccnc2c1Cl 91520,C(CC(=O)NC12CC1CN(C(c1cn(C)nc1O)=O)C2)(C(C)C)OCC 91521,C(CCCCCNC(C1CC(CN(C)C)C1)=O)NC(C)=O 91522,c1(C(NOCC(CC(=O)OC)C(F)(F)F)=O)cc2cc(Cl)cnc2[nH]1 91523,c1(CC)ncncc1C(N1CCC(CNC(C23COC(CF)(C2)C3)=O)C1)=O 91524,c1(C(c2n(CCCC)nnn2)N=Cc2ccccc2C)c(F)cnc(Cl)c1C 91525,N1(C(c2cc(C)oc2C)=O)CC23CCCC2(C1)CN(C(=O)C(O)CC1CC1)C3 91526,CN1CCc2cc(C(=O)NC3CN(C(C4CC5CCCCN5C4)=O)C3)ccc2C1 91527,c1(CN2CC(F)(C(=O)NCC(F)CO)C2)csc2ccccc12 91528,C(N=c1[nH]c2cc(Br)ccc2o1)C1C(C)CN(C(C2CCOC2)=O)C1 91529,c1(OC)ncnc(N2CCC(O)C(C(=O)OCCC(F)(F)F)C2)c1C 91530,N1(C(c2c(C)cc(Cl)cc2)=O)CCCC(C2CCN(C(=O)C(O)C(C)C)CC2)C1 91531,N1(C(c2ncncc2Cl)=O)CC2CCC(C1)N2C(C1CCN(C(F)(F)F)C1=O)=O 91532,c1(C(N(CC(c2ccccc2)CC)CC)=O)ccc(C(F)(F)F)s1 91533,N1(C(CC(C)SC)=O)CCOCC1CC(=O)NOC1CCC(O)C1 91534,CCC(C(=O)N1CC(C)C(C)(CNC(C2CC(O)C(O)C2)=O)C1)C(F)(F)F 91535,C1(NC(C2(CC)CCN(C(=O)Cc3ccon3)CC2)=O)CC2CCC(C1)C2O 91536,C1(NC(c2cc(C)[nH]n2)=O)CC(O)CN(C(c2ccc(-c3ccncc3)o2)=O)C1 91537,c1(NCCOCC=C)cc(=NC2CCOc3ccccc32)[nH]c(COC)n1 91538,C1(CNC(C(C)C2CC2)=O)CCC(NC(=O)CN2CCOC2=O)C1 91539,c1(C(=O)NCC2CC(NC(C=Cc3n(CC)ccn3)=O)C2)c(Cl)ccc(F)c1F 91540,c1(OC)c(C(=O)NCC(C)N(C(=O)COC2CCOC2)C)cc(Br)cc1F 91541,CN1CCOCC1CC(=O)NC12CC1CN(C(c1ccc(-c3cccs3)[nH]1)=O)C2 91542,C1(CCOCCN(C(COC2CN(C(C)=O)C2)=O)C)CC(F)(NC(C)=O)C1 91543,c1(C(=O)NC(CCNC(c2cc(C(C)C)no2)=O)(C)C)cc2c(ccn2C)[nH]1 91544,C1(CC(N2CCCC(C3N(C(c4c(C)cco4)=O)CCC3)C2)=O)CCCCC1(F)F 91545,C1(C(=O)NCC(CC)(C)Cl)COCCN1C(c1cc(=O)cc[nH]1)=O 91546,C=CCC(C)(C)CC(=O)N1CC=CC1CNC(c1ncnc(C)c1C)=O 91547,C1(CNC(CSCCC(C)C)=O)CN(C(=O)CC(C)F)CC2(CCC2)O1 91548,N1(C(C2CCCN(C3CN(c4nnc(C)s4)C3)C2=O)=O)CCN(CCO)CC1C 91549,CC1=NOC2(C1)CC(C(N1CC(NC(C3CCS(=O)CC3)=O)C(C(F)F)C1)=O)C2 91550,C1(CC)(NC(=O)CC(C)COC)CCN(C(c2ccc(C(C)(F)F)cc2)=O)CC1 91551,N1(C(C(CCC)OC)=O)CC2(C1)SCCC2NC(=O)Cc1cnoc1 91552,c1(C(=O)NC(CC(C)NC(COCCC(=O)OCC)=O)C)ccc(C)c(Cl)c1F 91553,C1(NC(c2cc(C)nnc2)=O)CCC(C)(NC(c2cc(Cl)ncc2O)=O)CC1 91554,Cc1noc(C)c1C(=O)NC1(CNC(C2CC23CC3(F)F)=O)CCC1 91555,N1(CC2CCN(C(COC(C)C)=O)CC2)CCC2(CC1)OCCc1ccccc12 91556,c1(NC(CCC)CCCNC(=O)CC#N)ccc(S(C)(=O)=O)cc1[N+](=O)[O-] 91557,C1(C(=O)NC2(CO)CN(C(c3sccc3C(F)(F)F)=O)C2)CCc2ccnn2C1 91558,Cc1ccc2[nH]c(C(N3CC(C)(NC(=O)C#CC4CC4)C3)=O)cc2c1F 91559,n1(CC)cc(Br)cc1C(=O)NC(C1(O)CN(C(C2CC23CCC3)=O)C1)C 91560,C1(CC=C)(NC(c2nnnn2CCC2CC2)(C2CC=CC2)C)CCCC1 91561,CC(CN(C(=O)C(C)NS(C)(=O)=O)C)N=c1[nH]c2cc(Br)ccc2o1 91562,C1(F)(C(=O)OCC)CN(C(c2cncc(N)n2)=O)CC12CCC2 91563,O=C1NCCOC2CCCN(Cc3ccc(C(F)(F)F)c(Cl)c3)C12 91564,C1(NC(C2CCCNS2(=O)=O)=O)CCN(C(C2CCCSC2)=O)CC12CCC2 91565,CC(CNC(C1OCCC1NC(=O)C=CCN1CCC1)=O)(CO)CO 91566,C=CCC(C(=O)N1CCCC1CC(C)C)NC(=O)COCC(=O)NC 91567,C1(C(=O)NC(CCC)CCO)CN(C(C2CCCN2C)=O)CCC1(C)C 91568,c1(C(=O)NCC(=O)NCC(CN(C2CCC2)C)O)c[nH]cc1C(C)(C)C 91569,c1(NC(C2CC(CN)CO2)=O)cc(Cl)cc2c1OCC(=O)N2 91570,N1(C(c2cc(F)c(Br)cc2F)C(=O)NCC)CCc2nc(C)n(C)c2C1 91571,N1(C(c2cc(CC)[nH]n2)=O)CCC2C(C(=O)N(C3CCCC3O)C)C2C1 91572,CCCCCCCC(O)C(F)(F)C(=O)NC1CN(C(=O)C(F)F)CC(C)(C)C1 91573,c1(N2CC(C)(CC)OCC2)ccc(S(=O)(=O)NCCCCCn2cccn2)cc1Br 91574,c1(OC)c(Cl)nc(Cl)[nH]c1=NC1CN(C(c2ccc(Cl)c(F)c2)=O)CC1F 91575,c1(C2(F)CC(C(=O)NC(C)CCN(C)C(C3CC3C)=O)C2)cccc(F)c1 91576,Cc1cccc(CC(CNC(N2CCCC2CCCO)=O)C(=O)O)c1 91577,N1(C(CNC(N)=O)=O)CCC2(C1)CN(C(c1n[nH]c3c1CSCC3)=O)CCO2 91578,C(=O)(C(C)(CNC(=O)C(C)SCC)CC)N1CCC(OCC)C1 91579,c1(OC)cccc2cc(COC(c3csnc3C(F)(F)F)=O)oc12 91580,C1(N(C(=O)NC)CCO)CCN(C(=O)CC2CC2(Cl)Cl)CC1.C1C(=O)N1 91581,N1(C(C(CC=C)OC)=O)CC(C)(C)OCC1CNC(c1c[nH]c(=N)s1)=O 91582,c1(C(=O)NC(C(C)C)CNC(=O)C(c2ccnn2C)O)ccnc(C2CC2)n1 91583,c1(OC)cccc(C)c1C(N1CCC(CC(=O)NC2CCS(=O)(=O)C2)C1)=O 91584,C1(CC)(NC(=O)CNC(=O)C(C)CC)CCN(C(C2CC3(CCC3OC)C2)=O)CC1 91585,CC1CN(C(c2csc(Cl)c2F)=O)CC1NC(C1CC1F)=O 91586,c1(C(=O)NCC(=O)NC2(C)CC(O)(CO)C2)cccc2occc12 91587,C(=O)(C(=O)CC(C)C)NC(C(=O)NCC(CC)C#N)(C)CO 91588,C12(C(c3nnnn3CCN(CCO)C3CC3)NC(=O)C(Cl)=CCl)CCC(CC1)C2 91589,N1(C(CC#CC)=O)CCCC(C(=O)NCc2cc(C)sc2C)C1 91590,C1(CC(=O)OC)CCCN(C(=O)CC2(NC(=O)Cc3cn(C)nn3)CC2)C1 91591,Cc1cc(NC(C2CC(C)(C)CN2C(c2cccc(CC#N)c2)=O)=O)cnc1Cl 91592,c1(C(N2CCC(OCCNC(C(C)OCCC=C)=O)CC2)=O)ccc(C)nc1C 91593,c1(C(N2CC(C)CC(NC(C3(OCC)CCCC3)=O)C2)=O)c(C)nc(=N)[nH]c1C 91594,C1(C(=O)NCC(CC(F)(F)F)NC(c2cnco2)=O)CCc2c[nH]nc2C1 91595,C1(C(=O)NC(C(=O)OC)CSC)CCCN(C(=O)COC(C)C)CC1 91596,N1(C(C(C2CC2)SC)=O)CCCC(O)(CCNC(=O)CCC2CC2(F)F)C1 91597,N1(C(c2c(C)onc2)=O)CCCCC(CNC(=O)CC2(C)CCCO2)C1 91598,C(=O)(C(CNC(c1c[nH]c(=NC)s1)=O)CC(C)C)NC(CCC)C(C)(C)C 91599,c1(CCC)ccc(CC(=O)N(C)CCNC(=O)C(C)Cc2ccc(Cl)cc2)cc1 91600,C1(NC(c2c(C)ncn2O)=O)CN(C(C2CC23CCC3)=O)C2(CCCC2)C1 91601,c1(C(=O)NCC(C)CO)c(Cl)nn(C)c1Cl 91602,c1(CC)cc(C(=O)N(C)CCN2CCN(C(=O)C(O)C(C)OC)CC2)ccc1F 91603,C(=O)(C(C)NC(C)=O)N(C(C)CNC(C1CN(C(C)=O)C1)=O)CC 91604,CCC1=NOC(CC(=O)N(CCCN(C)C(C2C(Cl)(Cl)C23CC3)=O)C)C1 91605,c1(CC)ccc(N2CC(C(N3CCCC(CNC(=O)CO)C3)=O)CC2=O)cc1 91606,c1(C(N(C2CN(C(C(C)SC(C)C)=O)CC23CC3)C)=O)cnc2c(c1)ncn2C 91607,Nc1cccc(C(=O)NCC2CCC2NC(c2ccnnc2O)=O)n1 91608,c1(C(N2CC(C)C(C)C2)C(=O)NC(CC)C)c(Cl)nc(Cl)n1C 91609,Cc1ccc(C(CNC(=O)Cc2ccncn2)NC(=O)CC(C)(F)F)cc1.C(C)(C)(C)O 91610,C1(CN(CCCNC(c2c(C)onc2)=O)C2CC2)CCC(C)(C)CC1 91611,N1(C(C=Cc2ccc(OC)cc2)=O)CCN(C(=O)CCC(C)OC)CCC1C 91612,C1(CO)CCN(CCOc2cccc(OC(F)(F)C(F)c3ccccc3)c2)CC1 91613,C(CC(=O)NCCCC1CCC1)(C(F)(F)F)NC(=O)CCc1nccs1 91614,N1(C(CC2(C)CC2)=O)CCC(C2(NC(=O)CNc3ccc(CO)cn3)CC2)CC1 91615,CC(C)C(C=O)C(C)C.c1(C2CCCN(Cc3ccccc3)C2)ccc(F)cc1O 91616,c1(CCCC(N2CC(C)C(CNC(=O)C(C)C(C)(C)O)C2)=O)ccc(F)c(F)c1 91617,N1(C(C(=O)NC2CCCN(CCF)C2)=O)CCOC2(CCCC2)C1 91618,N1(C(CCN(C(CN(CCC#C)C)=O)C)=O)CC2(C1)CC(C)(O)C2 91619,n1(CC#N)nc(-c2cc[nH]n2)nc1-c1ccccc1OCC(F)F 91620,Cc1ccc2cc(C(=O)NCCC(C)NC(=O)CN(C)C)c(C)nc2c1 91621,N1(C(=O)C=CCOc2ccc(F)cc2)CCN(C(=O)Cc2cccnc2)C2CC12 91622,C#Cc1cccc(C(=O)NCc2cccc(CNC(c3cnc(S)[nH]3)=O)c2)c1F 91623,C(=O)(CC(C)C(C)C)NC1(C(=O)NCc2ncc(CC)s2)CCCCC1 91624,Cn1cc(C#N)cc1C(=O)NC(CC1CCOCC1)C(=O)NCc1nnc(O)o1 91625,C1(CNC(C2CC(=C)CN2C(C2CC3CC(=O)C2O3)=O)=O)CCCC2(CC2)C1 91626,CC(C(=O)NCC(CO)NC(c1cncc(F)c1)=O)C(=O)N1CCOCC1 91627,N1(C(CCOC(CC(C)C)C)=O)CCCC1(C)CNC(C1CN(C)C(=O)N1)=O 91628,c1(C(N2CC(OC)C2)=O)ccc(C(N2CC(C)(CS(C)(=N)=O)C2)=O)cc1 91629,c1(C(=O)NCC2CC(O)(CNC(C(C(C)C)NC(C)=O)=O)C2)c(C)nc(C)n1O 91630,C1(C(=O)NC(C(=O)OCC)CC)CC(F)CN1C(C1SCCS1)=O 91631,C1(CNC(C(C2CN(C(=O)CSC3CC3)C2)OC)=O)CC2CCC2C1 91632,N1(C(C(Cc2cn(C)nc2)O)=O)CCOCC(NCc2cccc(O)c2Cl)C1 91633,C12(NC(C3CCN(C)CC3)=O)CCCN(C(=O)Cc3cc(F)cc(Cl)c3)CC1C2 91634,n1(CC(=O)NC2C(NC(CC(=O)N(C)C)=O)CC2)ncn(C)c1=O 91635,c1(C(N2CCC(CNC(C3(C=C)CCCCC3)=O)C2)=O)nnn2ccccc12 91636,C(CCCCCN=c1[nH]c2ccc(F)cc2o1)N(C)C(C1CC2(CCC2)C1)=O 91637,N12CCC3(CC1)CC23C(CCC(F)(F)F)=O.NC1Cc2ccccc2C1=O 91638,Cc1c(NC2CC(F)C2)ncnc1N1CCC(C)=C(Br)C1 91639,CC1C(C)N(C(=O)C(c2cnccn2)C)CCN1C(c1cnc(F)c(F)c1)=O 91640,N1(Cc2nc(N(c3ccc(Br)cc3Br)C(C)=O)sc2)CCOC(C#N)C1 91641,C=C(C)C1CCC(C)=CC1C(C(=O)NC(C)(C)C)N1CCC1C1CCCCC1 91642,N1(C(C(C2CC2)OC)=O)CCC(C2(NC(c3ccccc3C#N)=O)CCC2)CC1 91643,C(CNC(=O)CC(=O)N(CC(O)CO)C)(CC(=O)N1CCCC1)OC 91644,c1(C(=O)NC2CCCN(C(C(CCC)O)=O)CC2)cc(S(=O)(=O)NC2CC2)cs1 91645,c1(C(N(CC(C)CNC(C2CN(c3ccn(C)n3)C2)=O)C)=O)cc2n(n1)CCO2 91646,C12(C)CC(CCO1)NC(=O)C(C)(C1CC1)N(C)C2=O.C1(CC)CC2(C1)CC(C)C2 91647,C1(C(N2C(NC(C(OC)OC)=O)CC2C)=O)CCCN(C(=O)N(C)C)C1.C(C)(C)O 91648,C1(NC(=O)C(F)C2CCCC2)(CNC(C23CCC(C2)C3)=O)CCCC1 91649,C1(CNC(C2CC3(CCOCC3)C2)=O)CCC2CN(C(C3CCCS3)=O)CC12 91650,S(=O)(=O)(CCCN=c1nc2scnc2c(NCc2ccc(OC)cc2OC)[nH]1)CC 91651,C1(C(=O)NCCNC(=O)CC2CCCSC2)CCCCC1(F)F 91652,c1(C(=O)NCC2(CNC(c3ccc(C)cc3O)=O)CCC2)cc2cn[nH]c2cn1 91653,c1(C(=O)NC2(CC(N3CCCC(CCO)CC3)=O)CCC2)cc2n(n1)CCCC2 91654,c1(C(=O)NC2CC(NC(C3(CCC=C)CC3)=O)C2)ccnn1C1CCC1 91655,N1(C(c2c(CC)n(CC)nn2)=O)CCN(C(c2cncc(C)c2)=O)C(CC2CC2)C1 91656,Cc1cnc(N(C2CCCNCC2)C(c2ncccc2C)=O)nc1 91657,C1(C(=O)NCCSC)(COC)CCCN1C(=O)C(C)SC.C(=O)N(C)C 91658,N1(C(C(COC)(C)O)=O)CCN(C(=O)CCOC2CCCC2)C2CCCC12 91659,c1(CC(=O)NCC2(F)CC(NC(C3CC3F)=O)C2)cc(Cl)ccc1Cl 91660,N1(C(C2(CCC)CCC2)=O)CCC2(CC2C(N2CC(F)(C#N)C2)=O)C1 91661,c1(C(=O)NC2(CNC(C3(S(N)(=O)=O)CC3)=O)CCC2)ccc(=O)n(CC(=O)O)n1 91662,C1(NC(Cc2c(C)nn(CC)c2C)=O)CCCN(C(c2cnc(C3CC3)s2)=O)C1C 91663,Nc1nn2ccccc2c1C(=O)NC1CCC(CO)C1 91664,C1(C)(CC)CC(C(=O)NCc2cc(C(=O)NCCc3cnc(C)[nH]3)no2)C1 91665,C(=O)(CCCCCN=[N+]=[N-])N(C)CCNC(C1(n2ccnn2)CC1)=O 91666,c1(CC(=O)NCC2=CCN(C(COC(C)=O)=O)CC2)c(C)[nH]c2ccnn2c1=O 91667,CN1CCC(N(C)C(CC(=O)NC2(C)CC(NC(C3CCCCC3)=O)C2)=O)C1 91668,Cc1cc(N)c(C(N2CC3CC3(NC(=O)CCN(C)CCO)C2)=O)c(F)c1 91669,C1(C#N)(C(=O)NCC(CNC(C(C)=C(CC)C)=O)OC)CCCC(=O)C1 91670,C1(C(C)C)CN(C(c2cccc(CO)c2)=O)CC1C(=O)NC(C)C(C)(C)C 91671,c1(N(CCC(=O)NC2CC(C)(CNC(=O)CC3CCCCO3)C2)C)ccc(Cl)cc1 91672,C(c1ccc(F)c(F)c1)=CC(=O)NC(C)CCCNC(C1CCC1C)=O 91673,C1(NC(C(CC)SC)=O)CCN(C(=O)CCC(C)(C)C#N)CCC1CO 91674,C12(NC(CCc3nc(C)sc3)=O)CCC1CN(C(C1CCCN1N=O)=O)C2 91675,Cc1cc(=O)n(CC(N2CC(NC(c3cn(CC4CC4)nn3)=O)C(O)C2)=O)cn1 91676,Cc1ccc(C(N2CCN(C(=O)C(C)(C)n3cnnn3)CC2CO)=O)c(N)n1 91677,c1(C(N(CC(CN(C(C23CC(C)C2C3)=O)C)O)C)=O)ccnc2c1ncn2C 91678,C(c1csc(Br)c1)=CC(=O)NC1CCCC(NC(=O)CCC2CCC2)C1 91679,N1(C(C2(C)CCCCC2)=O)CC(C(=O)O)C2(C1)CN(C(c1ccc(N)cn1)=O)C2 91680,c1(CCCN(CCCNC(C2CCCC2)=O)CC)cncc(CO)c1 91681,c1(C(=O)NCc2c(COC)n[nH]c2)ncn2c1COc1ccccc1-2 91682,c1(C(N)=O)ccc(CC(=O)NCC(F)(F)F)cc1Cl.c12nccn1C2 91683,CC1CC(NC(C2(C(F)(F)F)CC(F)(F)C2)=O)CN1C(c1ccoc1)=O 91684,c1(C(C(=O)N(CCC(=O)OCCC(C2CCOC2)O)CC=C)C)ccccc1 91685,C(=O)(C1=CCCC1C)NC1CCC(NC(Cc2c(C)cccc2)=O)C1 91686,CC1C2C(CCN2C(c2cn3c(n2)CCC3)=O)CN1C(=O)C(N1CCNC1=O)C 91687,C1(C(N(C)CC2CCN(C(COCc3onc(CC)n3)=O)C2)=O)OC2CCC1C2 91688,N1(C(C2(OCC)CC2)=O)CCN(C2CCC(NC(c3cncc(C)c3)=O)C2)CC1 91689,Cc1nc(Nc2ccc(C#N)s2)sc1C(=O)NC(c1ccnc(F)c1)C 91690,N1(C(CCn2ncc(C)c2)=O)CCCC1(C)CC(=O)NCC1CC(=C2CC2)C1 91691,Cc1cc(C(=O)NCC(O)CNC(=O)CCC2CCCCN2C)ncc1F 91692,c1(C(=O)NCC2N(C(C(C=C=C)C)=O)CCN(C)C2)cc2sccc2n1C 91693,CC1COCC(C(=O)NC(C2CCCN2C(=O)CC2CCSCC2)C)O1 91694,c1(C(=O)NC2(CN(C(c3cnc(OC)c(C)n3)=O)C)CC2)noc(C)c1[N+](=O)[O-] 91695,N1(C(C(COC)OC)=O)CC(C(N2C3C=CCC2CC3)=O)C2(CCC2)C1 91696,N1(C(C(C)N(C(CC(C=C)CCC)=O)CC)=O)CC2(CCOC(=O)N2)C1 91697,N#CC1CN(C(C2(S(N)(=O)=O)CC2)=O)CCN1C(=O)OCc1ccccc1 91698,C1(NC(c2cc(C3CC3)ccc2Cl)=O)CC2CN(C(=O)C=C3CCCC3)CC2C1 91699,N1(C(c2c(C)nc(C)o2)=O)CC2CCN(C(c3c[nH]cc3C(C)(C)C)=O)CC2C1 91700,c1(SC)cncc(C(=O)NCC(C)NC(=O)CCc2ccc(C(F)F)cc2)c1 91701,CC(C(=O)NC1(N(C(=O)CC2(O)CCCC2)C)CC1)C(C)n1cccn1 91702,CC1(C)CC(NC(C2(CO)CCCCC2)=O)CN(C(c2ncc(F)cc2N)=O)C1 91703,N1(C(c2n(C)nc(Cl)c2)=O)CCC=C(C(=O)N2CCC(O)C2)C1 91704,c1(C(=O)NC2(CNC(c3cc4n(n3)CCCC4=O)=O)CC2)cc2nc(Cl)ccc2s1 91705,C12(C(N3CC(NC(c4cc5n(n4)CCO5)=O)C(O)C3)=O)CCC(CO)(CC1)C2 91706,c1(CCC(=O)NC2(C3CCCN3C(C3CCC(C(N)=O)O3)=O)CC2)ccc(O)nn1 91707,C1(OC)CN(N2CC(c3ccccc3)OC(C)C2)CC1c1cccc(F)c1 91708,C1(NC(CCCNC(C=Cc2ncn(C)c2)=O)=O)CC2(CCOC2)C1 91709,N1(CC)CC(C(=O)NC2CN(C(c3ccccc3C(F)(F)F)=O)CC2C)CC1=O 91710,N12CC(C1)C(O)C(=O)NCC2=O.C1(CNC(C2(CC=C)CC2)=O)CCCO1 91711,N1(C(c2cc(C)no2)=O)CCc2ccccc2C(NC(=O)C(C)n2cncn2)C1 91712,c1(C(=O)Nc2c(C#N)cccc2Cl)cnn2c1CN(C(=O)Nc1cc[nH]n1)CC2 91713,C=CCC(CC=C)c1nc(-c2cccc(F)c2)nn1C(c1ccccc1)C 91714,Cc1nc(N2CC(CNC(C3CC34CCC4)=O)(OC)C2)cc(O)n1 91715,C1(C)(Cn2cc(CC(C(C)C)O)nn2)CCN(C(=O)CCC2CCN(C)CC2)C1 91716,C(=O)(CCc1nccs1)NCCN(C(CNC(C)=O)=O)C 91717,C1(NC(c2cn(CCC)nc2)=O)CN(C(c2ccc(C3CC3)o2)=O)CC12CCC2 91718,C(=O)(C(O)(C(F)(F)F)c1ccccc1)NCCCC1OCCN(C(COC)=O)C1 91719,Cn1cc2ccc(NC(C3CC34CCN(C(=O)CCc3cccs3)CC4)=O)cc2n1 91720,c1(C(C)NC(=O)Nc2cncc(-c3csc(=N)[nH]3)c2)c[nH]c2ccc(F)cc12 91721,C1CC(F)Cn2cc(nn2)S1.C1(C(C)(C)C)CCC1C(N1CCCC1)=O 91722,CC1CCC(NCC(C)(C)CNS(=O)(=O)c2ccccc2)Cc2ccccc21 91723,c1(CC2C(C(=O)NCC=CCNC(c3ccsc3)=O)CCCC2)ccc(Cl)nc1 91724,N1(C(CCc2ccc(C)cc2)=O)CC(N(C)C(c2ccnnc2O)=O)C2(CC2)C1 91725,C(CC(C(C)C)(c1nnnn1CCCSCC1CCCO1)NC(=O)CO)N(C)C1CC1 91726,C(N=c1ccc2nnc(-c3ccccc3)n2[nH]1)c1ccc(OC(F)F)cc1 91727,C1(CN(C(=O)C(C)(C)Cc2cnn[nH]2)C)CCCC(NC(c2cnn[nH]2)=O)C1 91728,C1(NC(C=CCN(C)CC)=O)CC(NC(c2coc(CC3CCC3)c2)=O)CC1O 91729,N1(C(c2[nH]cc(C)c2)=O)CCC(CC(=O)NCCSC(C)C)CC1 91730,Cc1nc(O)nc(C)c1CC(=O)NCC1CC1NC(c1sc(C(C)C)nc1C)=O 91731,CCC(CCOC)C(=O)N1CCCC(C)(C(=O)NCCCO)C1 91732,N1(C(c2c(OC)n[nH]c2)=O)CCC(CNC(C2COCCN2CC)=O)(OC)C1 91733,C1(NC(CC2CCN(C)CC2)=O)C2CC3CN(C(=O)CC4CS(=O)(=O)C4)C1C3C2 91734,C1(N(C(C2(CC(F)F)CC2)=O)CC)CCCN(C(=O)Cc2ccccc2Cl)C1 91735,Cc1cccc(C2(C(N3CCC(CC(=O)N(C)C)C3)=O)CC2)c1 91736,c1(CC)ccc(Br)cc1NC(C1CCN(C(=O)Cc2cc(C)n(C)n2)CC1O)=O 91737,c1(CC(=O)NCCNC(=O)CC2CC(F)C2)cn2c(n1)CCCC2 91738,CC1(C)CN(C(=O)C(=O)NCC(F)F)CCC1NC(C1(c2cccc(Cl)c2)CC1)=O 91739,CCC(F)(F)C(=O)NC1CCC(NC(=O)Cn2cc(C3CCOC3)cn2)C1 91740,c1(C(=O)NCC2(CNC(C(C(=C)Cl)(C)C)=O)CC23CCC3)nnn2c1CCCC2 91741,c1(C(N(C2CCN(C(=O)CNc3cccnc3)C2)C)=O)cc(O)c(F)cc1N 91742,c1(CC(=O)NC23C(CN(C(c4cc(OC)ns4)=O)C2)C3)c(C)cccc1C 91743,C(CC1=NC(=O)C(C)C(=O)Nc2ccccc21)SCC.c12nnc(o1)CN2C 91744,CN=c1ccc(C(=O)N(CCC(C)NC(=O)CNS(=O)(=O)NC)C)c[nH]1 91745,C(C(C)CC(F)(F)F)NC(=O)NC(c1ccc(C)cc1)CCc1ccccc1 91746,CS(C)(=O)=NC(=O)NC(c1ccc(F)cc1)c1ccc(F)cc1 91747,N1(C(C(CC2CCC2)OC)=O)CCC(C(=O)NCC2CCSC2)=C(F)C1 91748,CCCC(C)(CC)C(=O)NCCN1CCN(C(c2cc(C)n(C3CC3)n2)=O)CC1 91749,N1(C(CS(CC)(=O)=O)=O)CC2CN(C(=O)COCCCF)CC(F)(F)C2C1 91750,c1(C(=O)NCCCCCCNC(C2N(CC)CC2)=O)ccc(Cl)c2occc12 91751,C(CO)(C(=O)NCC1CCC(NC(C2CCN2C2CCCC2)=O)C1)OC 91752,C1(C(C)O)CCN(C(c2nn(Cc3ccccc3)cc2Br)=O)CC1 91753,c1(CCC(=O)NC(C2C(NCC3C(C)(C)C3)C2)=O)c(F)cccc1F 91754,c1(C(=O)OC)ccc(C)c(C(=O)NCCC2(O)CCN(C(=O)CC(C)F)C2)c1 91755,c1(C2(C(=O)NCCCN(CC(F)CNC(C3CCC3)=O)C)CC2)ccnc(Cl)c1 91756,Cc1cccc2c1CC(C(=O)NCC1CC13CCN(C(=O)CCC(F)F)CC3)N2 91757,c1(NC(=O)NCC(CC(=O)O)c2ccccc2)cc(O)nc(CCCSC2CC2)n1 91758,N1(C(CSCC)=O)CC(C)OC2(CCN(C(=O)C=C(C)C(F)F)C2)C1 91759,C1(C(=O)NCC(CN(C)C(C2(C(F)(F)F)CCC2)=O)O)CC(C)(F)C1 91760,C1(CC2=NOC(C(=O)OC)C2)CN(C(c2cc(Br)co2)C(=O)NC2CC2)CCO1 91761,C1(C)(CC)CC(NC(c2cc(OC)cc(Cl)c2)=O)CN1C(c1cc(C)on1)=O 91762,C1(C)(NC(CCOCCN(C(c2c(C)cco2)=O)C)=O)CC(C)(C)OC1=O 91763,c1(CC)nnc(C)cc1C(N1CCN(C(=O)CNC(=O)NC)C(CO)C1)=O 91764,c1(C(N2CC(N(C(C(=O)OCC)CCO)C)C2)=O)ccc2c(C)cc(O)nc2c1 91765,C(=O)(C(C(C)(C)NCC1CCCC1(C)C)SC)OC 91766,CC(C)CC(O)C(C)C(=O)N1CC(C(=O)N(C2CC2)C2CC2)C(C2CC2)C1 91767,CCC(Cc1ccccc1)CC(=O)NC1CN(C(=O)CS(C)(=O)=O)C(C)(C)C1 91768,C1(NC(CSCC#N)=O)CC(NC(C2CC2[N+](=O)[O-])=O)C(O)C1 91769,C(=O)(C1=CCCOC1)NC(C(CO)NC(c1c(C)sc(Cl)n1)=O)C 91770,C1CCCC(C)NC(=O)C2(CC(C)(C)C2)C(=O)N1.C1(OCC)CC(CC(=O)OC)C1 91771,c1(NC2CCC(C(=O)OC)C2)ccc(C2(C(=O)O)CC2)cc1 91772,C(=O)(C1CCc2cccnc21)NCC1(C(C)(C)C)CCN(C(C=COCC)=O)C1 91773,c1(CNC(CC2(C)CCN2C(=O)CC2CCOC2=O)=O)cncc(O)c1 91774,C#CC1(C(=O)NC(CC)C2CC2)CN(C(C2CCSC2)=O)C1 91775,C1(C)(C(N2CC(OC)(CNC(=O)CCNC(c3cccs3)=O)C2)=O)CCCCC1 91776,c1(C(=O)NCCN(C)C(c2cnns2)=O)cn(CC(F)F)cn1 91777,c1(C(=O)NCC2CCCN2C(C2CC2[N+](=O)[O-])=O)cnc2ccc(Cl)cn2c1=O 91778,Cc1csc2ccc(C(=O)NNC(=O)C(C)C)cc12 91779,c1(CC)cc(C(N2CCC3(NC(=O)CN(C)CCOC)CC3C2)=O)ccc1OC 91780,C1(N(C(=O)CNC=O)C)CCCN(C(c2sccc2-n2cccc2)=O)CC1 91781,Cn1ccc2cccc(NC(C3C4CCC3CN(S(=O)(=O)CCBr)C4)=O)c12 91782,C1(CNC(=O)CCF)CCN(C(=O)CCOc2cc(F)cc(F)c2)CC1(F)F 91783,N1(C(C2N(C(c3n(C)nc(O)c3)=O)CCCC2)=O)CC(=O)NC(=O)C1 91784,N1(C(CC(C=C)CC)=O)CC2CCC1C(CNC(=O)C=Cc1csc(C)n1)C2 91785,CC1(CCNC(C2(C#N)CC3CC3C2)=O)CCN(C(=O)CC2(N(C)C)CC2)CC1 91786,N1(c2ccnc(N3CCCC(C(C)C)CC3)n2)CCc2nncn2CC1 91787,c1(-c2c(C)noc2C)cnc2[nH]cc(C(=O)Nc3cccc(OC(F)F)c3)c2c1 91788,C1(C)(C(=O)NCC(CNC(C(CC)F)=O)O)CNC(=O)C1 91789,C1(O)(CC2CC2)CCN(C(c2nnnn2NC(=O)C(C)(C)c2ccsc2)C)CC1 91790,Cn1nnc2c1C(C(=O)NCC#CCNC(C1CCOCC1(C)C)=O)CCC2 91791,CC1(C)CCC(n2cc(C3CCOC3)nn2)CN1C(c1ccn2cncc2c1)=O 91792,N1(CC(CN(C)C)O)CCCC(C(N(CC(c2ccccc2)OC(C)C)C)=O)C1 91793,N#Cc1ccc2c(c1)CCCN2C(=O)COc1cc(C#N)on1 91794,c1(OC)cccc(C(=O)N(C)CCNC(C2(O)CCC(C)C2)=O)c1OC 91795,C1(CCC)CN(C(C2CC2(C)C(F)(F)F)=O)CC1NC(c1cc(Cl)cs1)=O 91796,c1(CC)ncncc1C(N1CCCC1C(C)(C)NC(=O)C(C)Cn1ccnc1)=O 91797,c1(C(=O)NCCN(C(=O)CCCCC(N)=O)C(C)C)ccc2[nH]cc(C#N)c2c1 91798,c1(C(=O)NC2(CCCNC(c3nnn(C)n3)=O)CC2)cnc(OCF)nc1 91799,CC1(C(=O)NCCc2ccsc2)CCCN(C(c2c[nH]c(=N)o2)=O)C1 91800,N1(C(C(N2CC(C)C2)C)=O)CCN(C(c2ccncn2)=O)CC1c1nccn1C 91801,Cc1cc(CN2CCN(c3ccc(C4CC4)c(C)n3)CC2)ccc1F 91802,C1(CNC(CCNC(CCC=C)=O)=O)CCOC1C=C 91803,N1(C(C2C(C)=CCS2)=O)CC2(C(=O)N(CCCC(F)(F)F)C)CC1CO2 91804,C(C)(C)(S(C)(=O)=O)CNC(N(C)CC1COC(c2ccccc2)C1)=O 91805,C(=O)(C(O)CCCn1cnnn1)N1CC(C)C(NC(=O)CCc2ccc(N)cn2)C1 91806,C(=O)(CCCS(C)(=O)=O)NCC1(CNC(C(CO)N(C)C)=O)CC12CCC2 91807,C=CC(CCC)CC(=O)N(C1(C(=O)N(C)CCO)CCC1)C1CC1 91808,C(C)(C)(CC(F)C(=O)N(C)CC1COC(=O)N1)NC(c1c(C)c[nH]n1)=O 91809,C(=O)(C(C)(C)C(C)O)NC1(CC(N2CCC(C)(N(C)C)C2)=O)CC1 91810,C(N=c1nnc(C)c(C)[nH]1)C1C2N(C(C3(CCOC)CCC3)=O)CC(CC2)C1 91811,c1(NC2CCN(S(C)(=O)=O)C2)[nH]c(=NCc2c(Br)nnn2C)nc2scnc12 91812,c1(C(=O)NC(CC=CC)C(=O)N2CCC(C(=O)NC)C2C)c[nH]c(=N)c(C)c1 91813,N1(c2cc(NCc3c(CC)nn[nH]3)ncn2)CCCOC(CO)C1 91814,CC(C)C(C(=O)NC1CC(CO)C12CCC2)C(C)NC(c1coc(CO)c1)=O 91815,C12CC(C)CN(C1)C2=O.Cc1cncc(-c2cn(CC34CC(CO3)C4)nn2)c1 91816,N(C(=NCc1ccccc1)N1CCC2(CCOC2)C1)CC1CCC(C)(C)CO1 91817,c1(SCCC(=O)NC2C=CC(CNC(c3c(C)ccs3)=O)C2)ccccc1Cl 91818,c1(C(=O)NCC(CNC(c2n(CCC)nc(C)c2)=O)O)cc(C#N)c(N)cc1O 91819,C1(C(N2CCC(COC)C2)=O)CC2(CCN1C(=O)CCS(C)(=O)=O)CC2 91820,c1(OCC(=O)N(C(CNC(c2c(CC)nco2)=O)C)C)ccccc1C#N 91821,Cc1cccc(OC2(C3CCCO3)CC2)c1.N12CCC(C1)N(C)CCC2=O 91822,C1(CC(=O)NC2CC(NC(c3c(C)nc(C4CCC4)s3)=O)C2)CC2(CCC2)CO1 91823,C1(NC(c2nc(C(C)NC(C(C)N3CCCC3)=O)oc2)=O)C(O)C2CCCC12 91824,C(C(O)C(C)(C)C)NC(C(C)NC(Cc1c(C)ocn1)=O)=O 91825,N1(C(c2c3c(sc2)CC(C)CC3)=O)CCOC2(C1)CN(C(c1cnn(C)n1)=O)C2 91826,C=C(C)CCN(CC(C)NC(=O)NCC)C 91827,CC1CC(NC(c2ccsc2)=O)CN1C(=O)CC12COCC(C1)C2 91828,Fc1cc(Cl)cc(Br)c1CN(c1ncc2cn[nH]c2n1)C1CNCC1(F)F 91829,C1(CC(N2CC(NC(c3coc(C4CCC4)n3)=O)C(O)C2)=O)CC2(CCC2)CO1 91830,c1(CC)cc(C(=O)NCC(O)CCNC(C2CCSC2)=O)cc(C)c1 91831,C(=O)(CC1=CCCCC1)NC1C(C)(CN(C(C2(OCC)CCC2)=O)C)CCC1 91832,C1(NC(c2nc(CC)oc2)=O)CC2(CCCN(c3ncc4ncn(C)c4n3)C2)C1 91833,C#Cc1cc(C(=O)NCC2(C)CCCN2C(=O)CCC2CCOC2)ccc1Cl 91834,C1(CN(C(c2scnc2C2CC2)=O)C2CC2)CCCCN1C(=O)CCC1CC1 91835,C12(C(=O)NCc3c(C(=O)OCC)nns3)CNCC1COC2 91836,c1(-n2cc(C34N(C(=O)C(F)F)CC(C3)C4)nn2)ccc([N+](=O)[O-])cc1F 91837,c1(C(N(CCCC(=O)NCc2nccs2)C)=O)c[nH]c(C#N)c1 91838,N1(C(c2nc(C(C)C)oc2)=O)CC(C2CN(C(C3CCCCC3F)=O)C2)C1 91839,C(=O)(C(CNC)CC)NCc1c(C(=O)NC(C(=O)NCCC)C)[nH]cc1 91840,C(=O)(C(C)S(C)(=O)=O)NCCn1ncc(C(N(CC(CC)C)C)=O)c1 91841,N1(C(C2(OC)CC2)=O)CCCC2(CC(NC(=O)C=C3CCC(C)CC3)CO2)C1 91842,C1(C2CC2)(CNC(c2cn(CC)nc2)=O)CCN(C(c2c(Br)noc2C)=O)C1 91843,Cc1nc(O)nc(C)c1C(=O)NCC(C)(O)CNC(=O)Cn1cc(C(C)O)nn1 91844,CC(C)CC(F)C(=O)NCC1CCCCN1C(c1cc(C(N)=O)on1)=O 91845,c1(CNC(=O)CNC(=O)CNC(C2CCCS2)=O)ccncn1 91846,N1(C(c2c(C)ncs2)=O)CC(CNC(=O)C(C(C)O)N(C)C)CC1(C)C 91847,C#CC1(O)CN(C(=O)CSCCNC(C2(CF)CC2)=O)C1 91848,CC#CCCC(=O)N1CC(OC)C(NC(=O)CCCSCCOC)C1 91849,C1(O)(CN(C(=O)CCC2CCC(=O)N2)C)CN(C(=O)CCc2cn[nH]c2)C1 91850,c1(CC)ccc(C(=O)NCC2(F)CC(CNC(=O)C=CC3CCOCC3)C2)cn1 91851,C1(CC(=O)NCC(C)(CO)NC(C(C)=C2CCC2)=O)COC(C)(C)C1 91852,N1(C(CNC(C(C)(C)C)=O)=O)CCOC(C)(CNC(C2CC2(Cl)Cl)=O)C1 91853,C1(NC(C(COC)(F)F)=O)COC2(CNC(=O)COC(C)=O)CC1C2 91854,C#CC1COCCN1C(C1(CNC(=O)C#CC2CC2)CC1)=O 91855,CCC(CC)CC(F)C(=O)N1CCC2(CC1)CC2C(N1CCC1C1CCC1)=O 91856,N1(C(C2(C)CC(F)C2)=O)CC2(C)CC1(C(N1CCC3(CCC3)C1)=O)C2 91857,c1(C(=O)NC2CC(CCNC(CSC)=O)C2)ccc(N2CCCC(O)C2)cc1 91858,C(C1=CCN(Cc2cc(Cl)ccc2O)CC1)NC(c1cccc(F)c1C1CC1)=O 91859,C1(C(N(CCNC(C2(OC)CCCC2)=O)C(C)C)=O)C2CCN(CC2)S1(=O)=O 91860,N1(C(C(C)OCC=C)=O)CC(C(N2CCCC(C(C)(C)O)C2)=O)C(C)(C)C1 91861,N1(C(C2(N(C(c3n(C(C)C)ccn3)=O)C3CC3)CCC2)=O)CC2(CC(CO)CO2)C1 91862,C=CCCCCCCC(=O)N1CCN(C)C(C(C)C)C1.C12CC(C)(C1)C(=O)N2 91863,c1(OCC)c(NC(=O)CC2CNC(C(F)(F)F)CO2)cc(F)cc1Br 91864,C1(S(C)(=O)=O)(C(=O)NC(CC(C)NC(c2ccncc2F)=O)C)CCC1 91865,c1(CC(=O)NC2(CCNC(c3ccon3)=O)CCC2)cc(F)c(F)c(F)c1 91866,C(=O)(CC(C)C(=O)NC1(C)CN(C(=O)CCSc2ccccc2)C1)OC 91867,Cc1nc(C2CC2)ccc1C(=O)NCC1(C)CC(NC(c2cc(Cl)c[nH]2)=O)C1 91868,N1(C(C2CC=C(C)CC2)=O)CCCC2CN(C(=O)CC3CC=CCC3)CC12 91869,N1(C(CSc2c(C)ccc(C)c2)=O)CCN(C(C2CC3CC2C3)=O)C2(CCC2)C1 91870,Cc1ccc(CC(N2CC(F)CC2CN(C)C(C2CCCCCC2)=O)=O)c(F)c1 91871,CCC(CCC(=O)N(CC(=O)OC)C1CCC1)NC(=O)CCF 91872,CC1CCN(C(=O)C(=O)NCC(F)F)C1CNC(c1c(Br)ncn1C)=O 91873,C(=O)(C(C)S(=O)(=O)C(C)C)NC(CC(C)C)CNC(=O)CC(C1CC1)C1CC1 91874,N1(C(C(C)=C(CC)C)=O)CC(CNC(=O)CCC(CC)CCC)OC2(CCC2)C1 91875,c1(NC2C(OCC)CCC2)ccc(S(=O)(=O)Nc2ccccc2[N+](=O)[O-])cn1 91876,C(CCCC(=O)N(C)Cc1nnnn1C)NC(C1C(CC)OCC1)=O 91877,C1(CC(=O)N(C2CCN(C(=O)COCCF)C2)C)COC(C)(C)CO1 91878,N1(C(C(=O)NC2C(C(C)(C)C)C2)=O)CCOC2c3ccccc3OCC12 91879,C1(N(C(C(c2cccc(Cl)c2)CC)=O)C)CCC(NC(=O)CC2CCSC2)CC1 91880,O(NC(=O)C(F)C1CCOCC1)CCNC(c1ccc[n+]([O-])c1)=O 91881,CC1CN(C(C2(CC(C)C)CCCC2)=O)CCN1C(C1CCC(=O)NC1)=O 91882,C1(NC(CCn2c(C)cc(C)n2)=O)CN(C(C2CCC2C)=O)C2(CCC2)C1 91883,C1(CC(=O)NCC2N(C(C3(CN(C)C)CC3)=O)CCOC2)COCC(C)(C)O1 91884,N1(C(C(OC)OC)=O)CCN(C(C2(C)CCC(OC)C2(C)C)=O)CC12CCC2 91885,C1(CNC(c2ccc(CC)o2)=O)(CC)CCN(C(=O)CNC(=O)CNC(C)=O)C1 91886,C1(C(C)NC(c2c(-c3ccccc3)cnn2C)=O)CCCN(C(C2CCNC2)=O)C1 91887,C1(CNC(C2C(C=C)C2)=O)COCCN1C(=O)CC1CCSCC1 91888,c1(C(N2C(C)C(C)N(C(C3(C)CC(C)(C)C3)=O)CC2)=O)cnn2c1CN(C)CC2 91889,O=C(C=Cc1ccccc1Cl)NNc1ccccc1S(C)(=O)=O 91890,C1(NC(C2C(NC(=O)CC3(O)CCC3)CCO2)=O)CC2COCC(C1)C2 91891,C1(C(N2CCN(CCNC(=O)CC3=CCCC3)CC2)=O)CC2CCCCN2C1 91892,c1(C(=O)NCCC(N2CC(NC(C(C3CCOCC3)C)=O)C2)=O)c[nH]c(=O)cn1 91893,Cc1nc(C(=O)N(C)C)ncc1NC(=O)C=Cc1ccsc1 91894,C1(C2C(C(C(=O)NC(C(=O)NC)C3CCOC3)N(C)CC3CCC3)C2)(C2CC2)CCC1 91895,C1(CN(C(C(c2cccc(O)c2)C)=O)C)CCN(C(=O)C=CC2CCCC2)CC1 91896,CCC(C)(CC)C(=O)NC(C1CCN(C(=O)C(C)Oc2cccnc2)C1)C 91897,c1(CC(=O)C(C2CC2(F)Cl)=O)c(Cl)cnn1C.C(CCNCCO)N 91898,c1(CNC(C2CCCC(NC(C(C)(F)F)=O)C2)=O)ccc(F)c(C(F)(F)F)c1 91899,c1(C(C)C(=O)NC(C2(O)CN(C(c3ncccc3Cl)=O)C2)C)c(F)cccc1F 91900,C(=O)(C#CC1CC1)NCC1CC(C(=O)NCC#CCOC)C1 91901,c1(C(=O)OC)coc(C=CC(=O)N(CC(C)NC(=O)Cc2ccon2)C)c1 91902,N1(C(c2scc(C(C)=O)c2)=O)CCN(C(C2CC2(F)Cl)=O)CC(C)(C)C1 91903,c1(C(N2CC3(NC(CCOCCC)=O)C(C2)C3)=O)ccc2ncn(C3CC3)c2c1 91904,C1(C(=O)NCC(=O)N(CC)Cc2ccncc2)CCC(OC)CC1 91905,C1(CNC(C2CC=CC2)=O)CCCC12CCN(C(C1(F)CC1)=O)CC2 91906,c1(OC)n[nH]c(C(=O)NC2(CNC(=O)CC3(O)CCCOC3)CCOC2)c1Cl 91907,N1(C(C(CC(N)=O)NC(C(C2CCC(=O)N2)C)=O)=O)CC(C#N)C2(CCC2)C1 91908,C1(CNC(C(C=C)O)=O)CC(F)CN1C(C1CNC(=O)C1)=O 91909,C(=O)(CC1=CCN(C(c2c(F)cccc2F)=O)CC1)Nc1ccc(C)nc1C 91910,c1(C(N2CC=CC(NC(C3(CC=C)CCOCC3)=O)C2)=O)onc2ccccc12 91911,c1(NCC(=O)NC(CN(C)C)CC(=O)N(C)C)ccccn1 91912,N1(C(C(n2cnc(C#N)n2)CC)=O)CC(CNC(=O)CCC#N)C(C(F)(F)F)C1 91913,C(=O)(CCCCC(C)CC)NCC1N(CC(=O)N(C(CCCC)C)C2CC2)CCC1 91914,C1(NC(C(CCCOC)(C)C)=O)CCC2CN(C(C3CCCO3)=O)CC2C1 91915,C(CC(F)CN=[N+]=[N-])NC(c1cc(CNC(C(C)NC(CC)=O)=O)ncc1)=O 91916,Cc1nn(CC(N2CC3CCC3(CNC(c3cc[nH]n3)=O)C2)=O)c(C)c1C 91917,C1(NC(C2CN(C(=O)NC)C2)=O)COCCC1NC(c1cc(C)sn1)=O 91918,c1(N2CCC(COC)(CO)C2)ncnc(N2CCC(c3ccccn3)C2)c1C 91919,c1(C(C)NC(=O)C(=O)NC(C2CCCS2(=O)=O)C)c[nH]c2ccccc12 91920,Cc1ccc(Cl)cc1NC(=O)CCCCCN(C(=O)Cn1nc(C)cc1C)C 91921,CCCC(CCCNC(C1CC1(c1ccccc1)C)=O)NC(=O)CSC(F)F 91922,c1(OC)ccc(C(N2CC(CNC(=O)CC3CCOCC3)CC2(C)C)=O)c(F)c1 91923,CCC(O)CC(=O)NCCC1(CNC(=O)CCc2nc(-c3ccco3)no2)CC1 91924,CC1(C)CC(NC(=O)C=CCO)CCN(C(=O)CC2CCNC(=O)C2)C1 91925,C1(C(C(C)C)NC(=O)CC2CNC(=O)C2)CCN(C(C2CC2[N+](=O)[O-])=O)CC1 91926,c1(NCC(CNC(C2(C=C)CCOCC2)=O)C)ncnc2c1nnn2C 91927,Cc1c[nH]nc1C(=O)NC1CC(C)(C(=O)NC(C)CCCO)C1 91928,C(CCC(C)C)(C(=O)NCCOC)NC(CNC(CCCC)=O)=O 91929,C1(C(N(CC(=O)NC)CC)=O)CCCN(C(=O)C2=C(Cl)CC2)C1 91930,c1(C(=O)NCCCCNC(Cc2cn(C)nc2)=O)ccc2c(c1)COC2 91931,c1(C(=O)NC(C2(C(=O)NC3CCCC3(F)F)CC2)C)ccc([N+](=O)[O-])o1 91932,C=CC1CN(C(=O)Cc2ccno2)CC1NC(=O)Cc1ccc(C(C)C)c(F)c1 91933,c1(C(=O)NC(C(C)NC(Cc2ccc(OC)cc2)=O)C(C)C)c(F)cccc1F 91934,C1(CCC(=O)N(CCCO)CC#C)CCCN1C(=O)CCn1cccn1 91935,c1(C(N2CCN(C(C34CC3CNC4=O)=O)CC2)=O)ccc(Cl)cc1 91936,CCC(CC(=O)N1CCC1CNC(C1(OC)CC1)=O)c1ccccc1 91937,C1(O)(C(C)NC(=O)CC2CC=CCC2)CCN(C(c2cc[nH]c2)=O)C1 91938,c1(OCCN(C=O)Cc2cnn(C3CCOC3)n2)cccc(Br)c1I 91939,c1(C(=O)NCCC(=C)CNC(c2c[nH]ccc2=O)=O)cn2ccc(C)cc2n1 91940,c1(N(C(C(C(C)C)SC)=O)CC(C)OC)c(F)cccc1[N+](=O)[O-] 91941,c1(C(=O)NCC(C2CCCCC2)NC(C(C)N(CC)CC)=O)ncc(Cl)cc1Cl 91942,c1(OC)ccc(Cl)c(F)c1C(=O)NCC(C(C)C)NC(=O)CSc1ccncc1 91943,c1(OC)ccnc(N(CC(C)CNC(C2(C)CCCC2C)=O)C)n1.C1C(=O)N1 91944,C1(C(F)F)(OC)CCCN(C(c2nc(Cl)cs2)C(=O)NC2COC2)C1 91945,N1(C(C(C(C)C)C)=O)CCn2ncc(CNC(C3C4CCCCC34)=O)c2C1 91946,Cc1c(C(=O)NCCC(C)CCNC(=O)C(C)C2CCC2)cccc1Cl 91947,C1(NC(Cc2ccc(C)s2)=O)CN(C(=O)C(F)n2ccnc2)C2CCCC12 91948,c1(C(=O)Nc2ccc(-n3c(C)cc(C)n3)nc2)cc(F)c2nc(C)cn2c1 91949,CCCCC(O)C(=O)NCC1(C)CCN(C(c2cccnc2OC)=O)C1 91950,c1(CCC)ccc(F)cc1C.C1C(CC(C)C)S1 91951,C(CO)(CC(C)(C)C)NC(C1C(CNC(Cc2nc(C)[nH]n2)=O)C1(C)C)=O 91952,C1(C(N2CC3CC2C3C(C2(C3CC3)CC2)NC(=O)C2CC2)C)CC(C)OC1C 91953,c1(C(N2CC(O)(CN(C(CSC(C)C)=O)C)C2)=O)cc(Cl)c(Cl)[nH]c1=N 91954,C=C=CCC(=O)N1CCC(CCNC(c2nnc(CO)s2)=O)C1 91955,C(C(CC1CCCC1)C(=O)NCC1CCN(C2CC2)C1)NC(C=CCC)=O 91956,N1(C(CC(C)(C)C)=O)CCN(C(c2coc(O)n2)=O)CC1CCO 91957,CC(C)CCC(=O)C(=O)N1CC(CC(=O)NC2CC(F)C2)C(C)C1 91958,C1(O)(CNC(Cn2cc(CNC(CCC=CCC=C)=O)nn2)=O)CCC(C)C1 91959,C#CCC(C)C(=O)NCCc1ccc(-c2cn(CC)nn2)cc1.N12CCCC1C2 91960,c1(OCC(C(=O)NC(CNC(C=C(COC)C)=O)(C)CO)C)ccccc1Cl 91961,CC(CC(=O)N1CCC(O)(CNC(=O)CC2CN(C)C2)C1)C(F)(F)F 91962,c1(CC)cc(C(N2C(CNC(=O)CCC3CCCCO3)CC3CC23)=O)ccc1F 91963,C(C1CCCO1)=CC(=O)NCCC(C)N(C(=O)CCC1CCC1)C 91964,C(=O)(CCCN=[N+]=[N-])NCCC(C)(C)NC(C(C1CCCOC1)OC)=O 91965,CCC(C(=O)NCCCCC1(NC(=O)Cc2csc(Cl)n2)CC1)C(F)(F)F 91966,CC(C)(C#N)CCCC(=O)NCC1C=CC(NC(c2c(F)cccc2F)=O)C1 91967,C1(NC(C(C=C)CC)=O)(CNC(c2csc3cncn23)=O)CC2CCC1CC2 91968,C12(C(N(CCCN(C(CSC)=O)C)C)=O)CCC1CN(C(=O)OC(C)(C)C)C2 91969,c1(C(=O)NC2(C)CN(C(COCCC)=O)C2)cc(C(=O)OC)ccn1 91970,C1(CNC(c2c(OC)scc2)=O)C(C)CCCN1C(c1cc([N+](=O)[O-])c[nH]1)=O 91971,Cc1cc(C(N2CCOCC2C(=O)N(C)CC2CCOC2)=O)oc1C 91972,N1(C(C2CC(C)N2C(C2CC3CCC(C2)O3)=O)=O)CCc2ccccc21 91973,N1(C(c2cc(OCC)n[nH]2)=O)CCC2(CCCN2C(C2CCCCC2(C)C)=O)C1 91974,c1(C(N2CCC(C(CO)NC(c3c(C)onc3)=O)CC2)=O)ccc2nonc2c1 91975,C1(NC(C2(NC(=O)NC)CCCC2)=O)CN(C(c2cnc(S)nc2)=O)CCC1O 91976,C1(NC(CC(C)OC)=O)CCS(=O)(=O)C12CN(C(C1CCN(C(C)C)CC1)=O)C2 91977,c1(C(N2CC(NC(c3c(C)ccs3)=O)C(C)(C)CC2)=O)cnn(C)c1S(C)(=O)=O 91978,C1(C(=O)NC(c2ccc(C)nc2)C)CCN(C(c2ccccc2F)=O)C(C)(C)C1 91979,C(=O)(C1=CCc2ccccc21)NC(C)CC(C)NC(c1cnc(Cl)cc1Cl)=O 91980,C(c1c(F)cccc1F)=CC(=O)NC(CC)CNC(c1ccc(C(N)=O)[nH]1)=O 91981,C1(NC(CCC(N)=O)=O)CCC2CCN(C(=O)C(C3CC(F)(F)C3)O)C1C2 91982,N1(C(C(CC(C)C)=O)=O)CCC2CN(C(C3(C4CC4)CCC3)=O)CC2CC1 91983,n1(C(C)C)cnc2c(N(C)Cc3nc[nH]n3)[nH]c(=NCC3CC(F)C3)nc12 91984,N1(C(C(c2ccccc2)OC)=O)CCCOC(CNC(C2(SC)CC2)=O)C1 91985,c1(C(=O)NCCCN(C(C2CC(C)(F)C2)=O)CC)cc2n(n1)CCCNC2=O 91986,n1(CCNC(C2(CCC=C)CC2)=O)cc(C(=O)N(CCCO)CCCO)nn1 91987,N1(C(C2C(C)(C)CO2)=O)C2CCC1CN(C(C1CC3C=CC1C3)=O)C2 91988,C1(NC(C=C(CCC)C)=O)CC2CCC(C1)N2C(=O)C(F)(F)C(O)CC 91989,c1(NC(C)=O)cc(C(N2CC(CC(=O)NC3(C#N)CCC3)C2)=O)c(F)cc1F 91990,c1(C(N2CC(OC)C(NC(c3cccnn3)=O)C2)=O)ccc(F)c(C(F)(F)F)c1 91991,C1(O)(C(=O)NC2C(NC(Cc3ccn(CCN(C)C)n3)=O)C2)CCC(C)(C)CC1 91992,Cc1ncc(CCNC(=O)CCN(C(=O)C=CC2CCOC2)C(C)C)[nH]1 91993,N1(C(C(CC)(F)F)=O)CC2CCN(C(=O)CCOCC3CCCC3)CCC2C1 91994,c1(C(N2C(C)(CNC(C(C)OCC#C)=O)CCC2)=O)ccc(Cl)cc1O 91995,c1(C(=O)NC(C(C)C)CNC(=O)CC(C)(C)C)coc2c1C(O)CCC2 91996,c1(C(N2C(CNC(C(C)(C)C#N)=O)CC(F)C2)=O)cc(F)cc([N+](=O)[O-])c1 91997,CC1CN(C(=O)Cc2cc(O)nc(O)n2)CCN1C(c1coc(Cl)c1)=O 91998,c1(CNC(C(=O)NC2N(C(=O)OC(C)(C)C)CCCCC2)=O)cnc2n1CCCC2 91999,c1(C(=O)NCC2CN(C(C3(C)CC(=C)C3)=O)CC2O)nc2n(c1Cl)CCCC2 92000,c1(CC(=O)NC(C2CCOC2)CC)cccnc1Oc1ccsc1 92001,N1(C(CCOC(C)C)=O)CCCC2(C1)C(NC(c1cc(F)n[nH]1)=O)CCN2C 92002,c1(C(=O)NCC(CC)(C)NC(c2csc(COC)c2)=O)nc(O)sc1C 92003,N1(C(CN(C)C(=O)OC)=O)CCCC(CO)C1.C#CCCNC(C1CC1N)=O 92004,c1(C(N2CCN(C(C3CC3(F)F)=O)C(C3CCCC3)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 92005,C1(C(=O)NC(CC)(C)C(F)(F)F)CCN(C(c2ccc(NC)s2)=O)C12CCC2 92006,C1(CC(=O)NC2C(CNC(CNS(NC)(=O)=O)=O)CC2)COC(C)(C)CO1 92007,Cc1cccn2c(C(=O)NC3CCN(C(c4ccnn(C)c4=O)=O)C3)cnc12 92008,c1(NC)cc(Cl)ccc1C(N1CCC(CO)C(NC(C2(C)CCCCO2)=O)C1)=O 92009,C(c1ccccc1F)=CC(=O)NC1(C)CCN(C(CN2C(C)CCC2)=O)C1 92010,C1(NC(=O)NCC2(N(C)C)CCC2)CSC(CCC(F)(F)F)C(=O)N1 92011,CCC(=O)CCC(=O)N1CCCN(CCNC(=O)C(F)C2CCOC2)CC1 92012,c1(C(=O)NCCC2CC(NC(C3(C)COCCO3)=O)C2)cnn2c1OCC2 92013,C1(CC(=O)NCC2CCN2C(=O)C=CCNc2ccccc2)CCCCC1(F)F 92014,Cc1ccc(C(=O)NC2(CNC(=O)CC3CC4(CC4)CO3)CCCC2)cc1F 92015,c1(C(=O)NCC(CNC(Cc2c(C)ncs2)=O)(C)C)cnc2nc(O)ccc2c1 92016,N1(C(CC2CCC(C)C2)=O)CC23CCCC2(C1)CN(C(c1coc(CO)c1)=O)C3 92017,c1(C(N(C2CN(C(C3(C)CC3(C)C)=O)CC23CC3)C)=O)cc(F)cc2cc[nH]c12 92018,C1(C(=O)Nc2n(C3CN(C)C3)nnn2)CCCC(NC(C2CC2C2CC2)=O)C1 92019,c1(CNC(C(C2(C)CC2)NC(C(C)=CCC)=O)=O)ccn(C)n1.CC 92020,CN1CCN(C(=O)C(C)(O)C2CCOCC2)CC1CNC(C1(C)CCSCC1)=O 92021,c1(CNC(C(=O)NCc2ccc(SC)cc2)=O)ccc2c(c1)CCO2 92022,Cc1cc(C(=O)NCC2CC(NC(c3ccsn3)=O)C2)n2nc(C)cc2n1 92023,N1(C(C2CC(=O)NC2)=O)CC(NC(=O)Cn2cnc(C(N)=O)n2)C2CC12 92024,CC1(C#CC(=O)NC2CN(C(=O)CCS(C)=O)CC23CC3)CC1 92025,Cc1onc(C)c1C(=O)NC1C2CC(NC(C3CCCC3C)=O)CC12 92026,CN1CCC(CNC(C2CC(NC(c3ccncc3)=O)CCO2)=O)CC1 92027,N1(C(CC2N(C(c3occ(C)c3)=O)CCCC2)=O)CCCC(O)(CN(C)C)C1 92028,C1(NC(Cn2c(C)ncc2)=O)CN(C(C2(C)CCCO2)=O)CC(C)(C)C1 92029,C(F)(F)(C(=O)NNC(=O)CC1CCC(O)C1)c1cccc(C(C)(C)C)c1 92030,N1(C(c2c(C)n(C)nc2)C(=O)NCCC2CC2)CCCC2CCCC12 92031,N1(C(C(C)(C)C2CC2)=O)CC2(C=C(C(=O)NOCCCN3CCC3)CO2)C1 92032,C1(CC(C=CCCC(CN)C)CNCCn2nnnc2OC)CCC2(CCCCC2)CC1.C(C)(C)=CC.OC 92033,c1(C(=O)NCC(CC)NC(c2cc(C3CCC3)nn2C)=O)cc(C)nnc1O 92034,C1(CNC(C2(C)CCN(C)C2)=O)CC2(CC(NC(=O)CC3CC3(C)C)C2)C1 92035,C1(SC)CN(C(=O)CSc2nncs2)CC1NC(C1CC(C)C1)=O 92036,C1(NC(C=Cc2ncc(C)[nH]2)=O)CN(C(=O)C(C2CC2)C2CC2)CC1C1CC1 92037,N1(C(C23N(C(c4ccn(C)c4)=O)CC(C)(C2)C3)=O)C2CCC1CC(C(N)=O)C2 92038,c1(N(C(CCNC(C2(OC)CCS(=O)(=O)C2)=O)C)C)ccc([N+](=O)[O-])cc1Cl 92039,N=c1nc2c(c[nH]1)CC(C(=O)NCC13CC(CN1C(C1COCCO1)=O)C3)CC2 92040,C1(CC(=O)NCC(C2CC2)NC(c2cncc(C=C)c2)=O)CCC2(CCC2)CO1 92041,C1(C(N2CCC(O)(CCNC(C(C)O)=O)CC2)=O)CC(c2cn(C)nc2C)=NO1 92042,C12CCCCN(C1)C2=O.C1(CC)CCCN1C(=O)C(=O)N(C1(CO)CC1)C 92043,CC1(C)NC(=O)N(CC(=O)NC2CC(NC(=O)C(CO)NC(N)=O)C2)C1=O 92044,C1(C(N2C(CNC(c3nccc4cc[nH]c34)=O)CCC2)=O)CCCN2CCCC12 92045,c1(C(N(C)CC2CN(C(C34CC(F)(C3)C4)=O)C2)=O)cc2n(n1)CCNS2(=O)=O 92046,c1(C(N2CC(CNC(C(CC(C)C)NC(N)=O)=O)C2)=O)cnn2c1NCCC2 92047,C1(NC(Cc2c(C)con2)=O)CCCCN(C(=O)C(F)C(C)(F)F)C1 92048,c1(C(=O)OC)cnn(C)c1S(=O)(=O)NCC1OC(=O)CC12CCC2 92049,Cn1ncc(Cl)c1NC(C1(CO)CCN(C(C2OCCC2(C)C)=O)C1)=O 92050,N#Cc1cccc(CNC(=O)CC2(CNC(c3ccc(C(N)=O)o3)=O)CC2)c1 92051,C1(OC)CCC2CN(C(=O)CC=CCNC(C3CC3(Cl)Cl)=O)CC12 92052,C#CC1(C(=O)NC(c2ccc(O)nc2)C)CCN(C(C2C=C(C)CS2)=O)C1 92053,C1(NC(CCC(=C)Cl)=O)CC(C(=O)NC(C)(C)CC(F)(F)F)C12CCC2 92054,C(CN=c1[nH]c(Cl)nc2ccc(Cl)nc12)C1(C(C(=O)N)=O)CC1.CC(C)CC(C)N 92055,Cc1cc(F)cnc1C(=O)NC(CC1CC1)C(=O)NCC1CC2(CCC2O)C1 92056,N1(C(C=C(C)C)=O)CCC(N(C(c2cnco2)=O)CC2CC2)C1 92057,C1(OC)CN(C(=O)COC2(C)CCCC2)CC1CNC(C1CCCN1N=O)=O 92058,C(N=C(NCCSc1ccccc1)NCC(F)(F)CO)C1CC(=C)C1 92059,C1(C(=O)NCC(C2CCC2)NC(C(c2cccnc2)C)=O)CCC2CC1C2(C)C 92060,C(CC1CCc2ccccc21)OC(=O)Cc1cnc(C(N2CCCC2)=O)s1 92061,C1(NC(C2N(C(CCC)=O)CCCC2)=O)CCN(C(=O)CCCC(F)F)C1(C)C 92062,c1(C(=O)NC(C)CNC(=O)CC(C)N(C)C)cc(Cl)cc(F)c1N 92063,N(C(=NCc1ccc2cnccc2c1)N1CCN(CC)CC1)C(CC)C 92064,C=C=CC(C)C(=O)NC1CCN(CCNC(=O)C(C)CC=C)CC1 92065,c1(C(=O)NCc2cn(CCOC(C)=O)nn2)ccc(-n2cc(Br)cn2)cc1 92066,C=CCC(CC)C(=O)N1CC(CNC(=O)CC(C)SC)CC1(C)C 92067,c1(CNC(=O)NC(C2CC2(F)F)C)ccc2c(c1)NCCS2 92068,c1(C(=O)NCC2C(CNC(C(CC(C)C)F)=O)C2)cc2ccc(Cl)c(F)c2[nH]1 92069,N1(C(C(C2CCOC2)OC)=O)CC2(CCN(C(c3cc(N)c(F)cc3C)=O)C2)C1 92070,N1(C(c2ncc(C(C)=O)cn2)=O)CCN(C(=O)CCCC(C)C)C(C2CCC2)C1 92071,c1(C(=O)NCC(C)N(C(c2cc(C(=O)OCC)n[nH]2)=O)C)nccn2nccc12 92072,C(=O)(CC1CCc2ccccc21)N1CCC(NC(c2cscn2)=O)CC(C)(C)C1 92073,C(=O)(C(COC(C)=O)C(F)(F)F)NC1C2(NC(C(CCCC)C)=O)CCC(C1)C2 92074,Cn1ncc(C(=O)NC2CCC(Sc3ccccc3)CC2)c1-c1ccccn1 92075,N1(C(C2C(NC(c3ccc(OC)s3)=O)C3C=CC2C3)=O)CCC2(CCOC2)C1 92076,c1(CC)ccc([N+](=O)[O-])cc1C(=O)NC1CCN(C(C2CSCC(=O)N2)=O)CC1 92077,CC(CC(=O)NC1(C)CCN(C(c2ncccc2O)=O)C1)C(F)(F)C(F)(F)F 92078,N1(C(C2CCCN(CC)C2)=O)CC2(CCN(C(c3ccoc3Cl)=O)CC2)C1 92079,N1(c2ncc(C#C)cn2)CC2(CN(C(C3CCCCN3C(C)=O)=O)CCO2)C1 92080,C1(C(=O)NC(CCOC)CNC(=O)Cc2ccc(C)s2)CC(=O)N(C)C1 92081,c1(C(N2C(C)C(C)N(C(c3cncnc3)=O)CC2)=O)ccc(S(=O)(=O)CF)cc1 92082,CC1C2CCC(C2)C1C(N1CCC(C(C)(C)C(=O)NCC2CC2(F)F)C1)=O 92083,C1(CC(=O)N(CCCCCO)CC)CN(C(=O)Cc2cccc(O)c2)CCO1 92084,c1(OC)cc(F)c(NC(=O)COC2CN(C(=O)C=CC3CCOC3)C2)c(F)c1 92085,c1(C(CS(C)(=O)=O)NCCC(=O)NCCCN(CC)CC)ccc(F)cc1 92086,N1(C(=O)Cc2cncnc2)CCOC2(C1)CN(C(c1cc3c(s1)COCC3)=O)C2 92087,C(=O)(C1CNCc2n[nH]cc21)OC.C12CC3(CCC(CC3)CNC1=O)C2 92088,C(=O)(CC(C)(O)C(F)(F)F)N1CCN2CC1SCC2=O.CN(C)CCO 92089,N1(C(CO)=O)CCC(N(C(=O)C(O)C(C)C)C)CC1.CCCCCOCCOC 92090,C1(C(=O)OCC)CCN(C(C2(C(C)(F)F)CCOCC2)=O)CC1C 92091,C1(C(=O)NCC(CC)(CC)NC(C2C(F)(F)C23CC3)=O)(CC)CCNC1=O 92092,c1(C(C)C)cc(C(=O)NC(C)CCNC(=O)CSc2ccncc2)n(C)n1 92093,c1(C(=O)NCC(CC)NC(=O)CN(C)C(C)=O)csnc1C 92094,c1(NC(CC2N(C(CCn3c(C)ncc3)=O)CCC2)=O)cc(Cl)ncc1Br 92095,N1(C(C=Cc2c(C)ccs2)=O)CCC2CN(C(C3CC34CCSCC4)=O)CCC12 92096,C#Cc1cn(C)nc1C(=O)NCC1CN(C(c2cnc(S)n2C2CC2)=O)CC1C 92097,c1(CNC(C2N(C(C3CC(OCC)C3)=O)CCC2)=O)ccc(O)c(C)c1 92098,c1(CCC(=O)NC2CC(C)(C(=O)NCCN(C)C3CC3)C2)cccc(C(F)(F)F)c1 92099,C1(C(=O)NC2C(C)(C)CN(C(=O)Cc3ccsc3)C2)CCc2nccn2CC1 92100,C#Cc1ccc(C(=O)NCCC(C)NC(C2CC(C#N)C2)=O)c(F)c1 92101,C(c1cnc(OC)nc1)=CC(=O)N(CCC(C)NC(C=NOC)=O)C 92102,N1(C(C2OCCN(CC)C2)=O)C2CCCC1CC(NC(c1nc(O)n[nH]1)=O)C2 92103,CCC(C)C(O)C(=O)N1CC(n2cc(-c3ccnc(C)c3C)nn2)C1 92104,CC1(CC(=O)NCC2CN(C(=O)Cn3nccn3)C3CC23)CCOCC1 92105,c1(C(=O)OCC)cccc(C(=O)NC(C)CN(C(=O)C(F)CSC2CC2)CC)c1F 92106,c1(OC)cc(C)ccc1OCC(c1nc(CC(F)(F)F)no1)CCN(C)CC 92107,NC1CCN(C(c2csc(-c3cccnc3)n2)=O)C(c2ccccc2)C1 92108,N1(C(C2CCN(CC)CC2)=O)CCN(C(C2CCSCC2)=O)C(CC#N)C1 92109,N1(C(Cc2n(C)nc(C3CC3)n2)=O)CCOC2(CCN(C(C3(C)CC3(F)F)=O)C2)C1 92110,C(C(C)(C)CC(=O)N1CCC(N(CCO)C(c2cnnc(C)c2)=O)C1)OC 92111,C1(NC(c2nc(C)n(C)n2)=O)CC2CC(NC(=O)C3=CCOCC3)CC2C1 92112,Cc1cn(C(C)C)[nH]c1=NC(=O)c1csc(Nc2ncncc2F)n1 92113,C1(CNC(CN(C)C)=O)CCN(C(c2csc(NC3(C)CCC3)n2)=O)C1 92114,CC1Oc2c(C(=O)NC(CNC(=O)C(C)(F)F)C3CC3)cccc2NC1=O 92115,CC1(C)CCC2(CC1)CC2C(N1CC2=C(C1)CN(C(C1CC1(Cl)Cl)=O)C2)=O 92116,N1(C(=O)CC2CCS(=O)(=O)CC2)CCN(C(=O)C2=CCCOC2)CC(O)C1 92117,C1(C(=O)NC(CC)CNC(c2cnc(O)c(OC)c2)=O)CCc2nc(C)ncc2C1 92118,c1(OC)ccc(CO)cc1NC(C1CCN1C(=O)CC1C=CCC1)=O 92119,CN1CC2CCC(C1)N2C(C1CCCCCN1C(c1cc(CO)on1)=O)=O 92120,Cc1cccc2c(CCC(N)C(c3ccc(F)nc3)=O)c[nH]c12 92121,C(C(C)(C)CN=c1[nH]c(=N)[nH]c(=NC(C)Cc2cccc(Br)c2)[nH]1)OC 92122,c1(C(=O)NCC2CCN(C(C3(OC)CCCOC3)=O)CC2)cnc(Cl)cc1N 92123,c1(N(C(C2N(C(c3cc(C)c(F)cc3)=O)CCCC2)=O)CC)cc(C#N)ccc1Cl 92124,C1(N(C)C)CCC(C(N2CCCC(C(O)C(F)(F)F)C2)=O)CC1 92125,C=C(C)C(C)(O)C(=O)NNC(=S)NC1CCC12CCC2 92126,Cc1ncnc(C(=O)NC(CNC(=O)CCCN2CCCCC2)C2CCC2)c1C 92127,c1(ONC(=O)NC(C(N2CC(C)OC(C)C2)=O)(C)C)ccc(Cl)cc1[N+](=O)[O-] 92128,C(=O)(C(CC(C)C)NC(c1cc(OC)ccc1F)c1nnnn1C)NCCOC 92129,CC1CN(C(=O)C(C)(CO)NC(c2ccc(CC#N)cc2)=O)Cc2nncn21 92130,N1(C(C(C(C)C)N2CCCC2=O)=O)CC2CCCN(C(c3cc(O)no3)=O)C2C1 92131,N12CCC(O)(CC1)CC(=O)NCc1cccc(n1)C2=O.C(C(F)F)(C(C)(C)C)OC 92132,c1(C(N2CC(CNC(C(CCC)C)=O)C(O)C2)=O)ccc2cc[nH]c2n1 92133,c1(NC(CC2(C)CN(Cc3c(OC)c(F)ccc3)C2)=O)nccc2[nH]ccc12 92134,c1(CC(N2C(CNC(C=CCC)=O)CN(C)CC2)=O)ccc2c(c1)COC2 92135,Cc1cccc(C=O)c1.c1cccc(C2CCN(N3CCCC(F)C3)C2)c1 92136,c1(C(C(O)C2CC2)OC)cn(C(C)(C)C(C)C)nn1 92137,CP(C)(=O)c1ccc(C(=O)NC2C3CN(C(C45CCCC(C4)OC5)=O)CC23)nc1 92138,N1(C(=O)CCCC(F)F)CCC2(CCN(C(=O)C(F)(F)C(O)C3CC3)C2)C1 92139,N1(C(c2ncnc(C)c2C)=O)CCCC2(CCN(C(=O)CSCC(F)(F)F)C2)C1 92140,c1(C(N2CCC(C(C)NC(C(F)OC)=O)C2)=O)cccc2ccc(O)nc12 92141,C1(C(=O)Nc2nnc(CC3CCCC3)s2)CCCN1CC(F)F 92142,C1(C(=O)NCCOCCN(C)C(C2C3CC3C3CC23)=O)CC(N(C)C)CCO1 92143,c1c(C)noc1Cl.Cc1cc(C(=O)NC2(CO)CN(C=O)C2)on1 92144,Nc1ncnc2c1ncn2CC(=O)NCC1CCC2(CCCC2)C1 92145,c1(CC)nc(C)c(C(=O)NCCCCC(=O)N(CC2N(C(C)=O)CCC2)CC)o1 92146,c1(C(=O)NC(C)CCCNC(C2(C)CC2(Cl)Cl)=O)ccccc1Br 92147,c1(C(=O)NC2C(C(=O)NCCn3ncc(C)c3)COC2)cncc(F)c1 92148,C(=O)(C(C)C(F)F)N(C(=O)CCN(c1cccs1)CCCO)CC.CC(C1CC1)OC 92149,CC(C(=O)N(C(C)CCNC(c1ccc(C2CCOC2)cc1)=O)C)C(C)(F)F 92150,C12CCCN1N(CCC)CCNC2=O.c1(C(=O)NC)ccc(CO)s1.C(=O)NC 92151,C1(C)(CNC(c2ccn(COC)n2)=O)CCCN1C(=O)COC1CCCCC1C 92152,n1(C(CC)CC)ccc(C(N2CCC(CNC(=O)C(C)COC)C2)=O)n1 92153,C1(C(=O)NCC2C(NC(CSCCC#N)=O)CCCC2)CCC2CCCCN12 92154,C#CCCCCC(=O)N1CCN(C(=O)CC(C)c2ccccc2)CC1CCO 92155,C(CC(CC)C(=O)NCC1CCCN1C(C1CCCC(CF)C1)=O)=CC 92156,S(=O)(=O)(c1c[nH]c(C(N2CC(CCNC(=O)C(O)C(C)(C)C)(OC)C2)=O)c1)NC 92157,N1(C(C(CC)(C)F)=O)CC(NC(c2ccc(CO)nc2)=O)C(N=[N+]=[N-])C1 92158,C1(CCOC)(NC(c2cn(C)nn2)=O)CCN(C(=O)CC(C)(F)F)C1 92159,Cc1cc(C(=O)NCc2nc(C(=O)NCC3CCCCC3(C)C)co2)nc(C)c1 92160,N1(C(C(CC)=CC)=O)CCCC(CNC(C2CCCCC2C)=O)C1 92161,C(=O)(C1=CC2(CCOC2)C1)NCc1ccc(COC)cc1.C12CCC1C2 92162,c1(C(=O)NC2(CO)CCN(C(C(CC)C)=O)C2)cnc2[nH]c(C(F)(F)F)nc2c1 92163,c1(NC(C2(F)CN(S(Cc3cccc(C#N)c3)(=O)=O)C2)=O)ccc(Br)cc1[N+](=O)[O-] 92164,c1(C(=O)NC2CN(C(CCCOC3CCCC(C)C3)=O)C2)cc(OC)cc[n+]1[O-] 92165,C1(NC(c2ccc[nH]2)=O)COCC1C(=O)Nc1ccccc1.C12(CC1)C(=O)N2 92166,C1(NC(c2csc(C)c2N)=O)CCCC(NC(C2CC3CC3C2)=O)CC1 92167,c1(CC)nn(C)c2ncnc(NOCc3n[nH]c(C)n3)c12 92168,N1(C(C2N(C(C3(CC)CCCC3O)=O)CCCC2)=O)CC(C2CCCCC2)C1 92169,c1(C(=O)NC2CC(N(C)C(c3cnc(O)c(F)c3)=O)C2)cccc2nccnc12 92170,c1(NC(CC)C(O)c2ccccc2)ncccc1S(=O)(=O)NCCC(F)(F)Br 92171,N1(C(C(CC)=CCCC)=O)CC(NC(C2(COC)CCCC2)=O)C(COC)C1 92172,N1(C(CS(CC)=O)=O)C2CCC1C(CNC(c1c[nH]cc(Cl)c1=O)=O)C2 92173,N1(C(C=CC=CC)=O)CCC(CC(=O)NC(CN2CCCC2)CC)C1 92174,N1(C(C(CC)CO)=O)CC2CCCC2(NC(c2cc(C)no2)=O)C1 92175,CCC(C)C(=O)N1CCC(C(=O)Nc2occc2C)C1 92176,c1(-c2c(N3CCN(C(CC)=O)CC3)nccc2)ccc2[nH]c(C(=O)OC)cc2c1 92177,C=CCCN=C(NCC(C)C(F)(F)F)NCc1ccc(C2CC2)cc1 92178,C1(C(N2C(C(C)NC(=O)C3=CCCO3)CCC2)=O)CC2CCC(C1)N2C 92179,CCC(C)(C(=O)N1CCC(F)(C(=O)N(C(C)C(C)(C)C)C)C1)OC 92180,c1(C(N2CCN(C(C(CC=C)C)=O)C(C)C2)=O)cc(C#N)ccc1Cl 92181,C1(C(=O)NC(C)C(C)(C)NC(c2cncc(Cl)c2)=O)OCCOC12CCC2 92182,Cc1ncc(C(F)(F)F)cc1C(=O)NCC1CCC12CN(C(C1CC1F)=O)C2 92183,C1(NC(=O)C=Cc2cocn2)CCCCCN(C(C2(C3CCCCC3)CC2)=O)C1 92184,c1(C(=O)NCC(CN(C(=O)C2=CCOCC2)C)O)cnc2c(Br)cccn12 92185,N1(Cc2cn(CCC)nc2C)CCOCC(C(N2CCOCC2CC(C)C)=O)C1 92186,C(=O)(CCCC(=O)NCC(CO)NC(=O)C(O)CC1CCOCC1)N(CC)CC 92187,c1(-c2cn(CCC3CN(C(c4cc(Br)n[nH]4)=O)C3)nn2)cc(F)cc2c1OCC2 92188,N1(CC(=O)NCC2CCC(NC(C=C(C)C)=O)CC2)CCCCC(O)C1=O 92189,N1(C(C=NOC)=O)CC(NC(c2cnc(C)c(CC(C)C)c2)=O)CC(O)C1 92190,C1(CC(=O)N(CCCCNC(C23CC(CC)(C2)C3)=O)C)CCCN(C)C1 92191,CCC(C)(C)C1(C(=O)NCC(=O)NCCN(CCOC)C(C2CC2C)=O)CC1 92192,C1(CC)C(C(=O)NCC(C)(O)C2CCC2)CCCN1C(C1CCC(C)(C)OC1)=O 92193,n1(C(C)C(N2CCCC2C(C2CC2)NC(=O)CNC=O)=O)ccc2ccccc12 92194,Cn1cnc2c1CCC(C(=O)NC1CCCN(C(=O)COc3ccccc3)C1)C2 92195,C12(C(=O)NCC(=C)CCNC(=O)C(N3CCN(C)CC3)C)CC(C)(C1)OC2C 92196,C1(CNC(CSCCC(C)C)=O)C2CCC(C2)N1C(C1CC(=O)N(C2CC2)C1)=O 92197,C1(C(N2CC(O)(CN(C(C3C(C(=O)OC)C3)=O)C)C2)=O)C(C)(C)C1(C)C 92198,N1(C(=O)NCC(O)CN2CCOCC2)CC2CCC1C1CNCC21 92199,C1(NC(C(CC2CC2)NC(CC2OCC(C)(C)C2)=O)=O)CCCN2CCCC12 92200,Cc1ccccc1C(C)CC(=O)N(C1CN(CC(N2CCC(C)C2)=O)C1)C 92201,Cc1cccc2c1CCOC2C(=O)Nc1ccc(F)c(C#N)n1 92202,CC1CC(C(=O)NC23CC(CNC(C4CCN(C)S4(=O)=O)=O)(C2)C3)CCS1(=O)=O 92203,CC(CF)CC(=O)N1CCC(C(C)CNC(c2ccn(C3CC3)n2)=O)CC1 92204,c1(N2CC(C)C(NC3CCCN(c4ccccc4CO)C3=O)C2)nccc(C#N)n1 92205,c1(OC)cc(NC(C2CC2NC(c2cccc(O)c2O)=O)=O)ccc1C 92206,CC(CCCCN=c1c(C#N)c[nH]c2ccccc12)NC(C1CC1C)=O 92207,Cc1cc(F)ccc1C(O)C(N1CCN(C)CC1CNC(=O)C=CC(C)(C)C)=O 92208,C1(C(=O)NCc2c(C(N(C)CC3CCN(C)C3)=O)occ2)CCC(=O)NC1 92209,Cc1c(C=CC(=O)NCCCCC(C)NC(C23CCC(CC2)CO3)=O)cnn1C 92210,C(C(C)(CC(C)C)NC(C1CCOCC1(C)C)=O)NC(c1cccc(C)n1)=O 92211,N1(C(CCSC)=O)CC2CCCC(CNC(=O)CN3CCn4nccc43)C2C1 92212,C(C)(C)(CC(=O)N1C(C(=O)N(c2ccc(F)cc2)C)CC2CC12)OC 92213,S(=O)(=O)(c1c[nH]ccc1=NCc1ccc(N(C)C)o1)N(CC(=C)Br)C(C)C 92214,N1(C(CC(C=C)C)=O)CCN(C(C2CCC(CC)CC2)=O)CC1C1CCC1 92215,n1(CC(=O)N(CC)Cc2cc[nH]n2)ccc(=NC(=O)C2(O)CCOCC2)nc1O 92216,N1(C(C2CC(=C)C2)=O)Cc2n[nH]cc2C1C(=O)N1CCOC(CC(C)C)C1 92217,c1(C(=O)NCCC(=C)CNC(=O)C=CCO)[nH]c(O)nc1C 92218,Cc1nc2sccn2c1C(=O)NCC(O)CNC(C1C2CCC1CC2)=O 92219,C12(NC(C3C(NC(C)=O)C3)=O)CC(CNC(C3(C)CCCCO3)=O)(C1)OC2C 92220,C(=O)(CC(C)C(F)(F)F)N1CCCC(CC=C)(NC(=O)C(C)=CCC)C1 92221,N1(C(C2OCCN(C(=O)CC3CCOC3)C2)=O)CCC2(CCCO2)C1 92222,C1(C(=O)NCC(CCC)NC(=O)C2=NNC(=O)C2)CCc2nccn2C1 92223,S(=O)(=O)(c1ccc(Br)cn1)NC1C(C(=O)Nc2c(F)cc(C(F)(F)F)cc2F)C1 92224,Cc1c(C(=O)NCCSc2ccccc2)cnn1C(C)C.N12CCC(C)(C1)C2=O 92225,C1(C(C(=O)N(CCCCCCNC(C2CCC(=O)N2C)=O)C)O)CCCCCCC1 92226,C1(C(N2CC(C)C(CNC(=O)C3=C(Cl)CC3)CC2)=O)CN(C)CCN(C)C1 92227,c1(OCC)cccc(C=CC(=O)NCC(c2ccccc2)NC(=O)C=NOC)c1 92228,C(=O)(CCS(C)=O)N1CC(CNC(c2nc(C(=O)OCC)sc2)=O)C1 92229,N1(C(CC(C=C)(C)C)=O)CCC2(C1)CN(C(C1CS(=O)(=O)CC(=O)N1)=O)CCO2 92230,N1(C(c2ccc(C)nc2C)=O)CC2CCCC2C1C(=O)NCCCC(F)F 92231,C1(NC(c2c(C)ncs2)=O)CC12CCN(C(=O)CCN1C(=O)C=CC1=O)CC2 92232,C(=O)(C(C)(O)C(C)(C)C)NC(C)CNC(c1ccc(C(C)(C)C)cc1)=O 92233,N1(C(c2[nH]c(=NC)sc2)=O)CCCOC(CNC(=O)CCc2ccc(Cl)nc2)C1 92234,CCC(CCOC)C(=O)NC1CC(C(=O)N2CCCCC2CC)=CC1O 92235,N1(C(CN(CCOC)C)=O)CC2(CCCC2)C1C(=O)NC1(C2CC2)CCC1 92236,CC(CC(=O)NCC1C2CCCOC12)C(C)(C)NC(c1cscc1Cl)=O 92237,C1(NC(c2cc(C)sn2)=O)CC(NC(c2ccsc2C)=O)C12CCC2 92238,CC1(C)CN(C(C2CCOC2C(F)(F)F)=O)CCC1NC(C1(COC)CCC1)=O 92239,c1(C(=O)NCCC(=O)NC2(CO)CC2)cc(Br)ccc1Cl 92240,Cc1cc(C)c(C(N2CCC(CNC(C3CC4(CC4)CO3)=O)CC2)=O)cc1C 92241,C1(N(C)C(c2ccc(F)s2)=O)CCCN(C(=O)CC2CC(C(C)(C)C)C2)C1 92242,C1(CNC(CN(C(C)C)C(C2CC2(F)Cl)=O)=O)CNC(=O)CO1 92243,CC1CCCC(=CC(N2CCC(NC(=O)CN(C)S(N)(=O)=O)C2C)=O)C1 92244,N1(C(C2(SC)CC2)=O)CC2COCC(C1)C2NC(C1CCC2(CCOCC2)O1)=O 92245,N1(CCC)CC2(CN(C(c3c[nH]cc3Br)=O)C2)C1 92246,C12(C(=O)NC(CC#C)CC)CC1CCN2C(c1nccs1)=O 92247,C(=O)(CCC(CC)CCC)NCCC(=O)NC1C2(CCN(S(CC)(=O)=O)CC2)C1 92248,C1(C)(C(=O)NC)CCN(C(C2CC2C(C)NC(=O)COC)=O)C1 92249,c1(C(N(c2ncc(C3CC3)s2)CC)=O)c(C)cc(C)cc1C 92250,C(c1ccccc1F)=CC(=O)NCCCCCCNC(=O)C(O)Cc1ccccc1 92251,CN1CCC(CC(=O)NC2(C)CCN(C(C3CCOC3)=O)C2)C1=O 92252,N1(C(C)C)CC(C(N2CCC(N(C(=O)CCN(C)CCO)CCO)C2)=O)CCC1=O 92253,CC1OCCOC1C(=O)NCC1(C(=O)NC2CC(CO)CC3CC23)CCC1 92254,C1(C(=O)NCCC(CNC(C(C)Oc2ccccc2)=O)O)CCCC(=O)N1 92255,C1(CCCC)CCN(C(N2C(C)(CC(=O)OC(C)(C)C)CC2)=O)CC1.C(C)C 92256,c1(C(=O)NCC(CNC(c2c(CC)sc(=N)[nH]2)=O)(C)O)cnc2ncnn2c1C 92257,C1(CN)CN(C(C(N2CCC(N3CCCCC3)CC2)=O)C2COC2)CCO1.CC(=O)N(C)O 92258,N1(C(CCCC)=O)CCCC(c2nc(-c3ccc(CC)nc3)nn2C2CCSC2)C1 92259,CC(C)(C#N)CCC(=O)NC1CCN(C(c2cc(Br)c(F)cc2F)=O)C1 92260,C1(O)(Cc2nnc(S)n2C)CCNCC1.C1(CC)CC12CCOC2 92261,N1(C(CC(=O)NCC#C)=O)CCCN(C(=O)COCC2CCCC2)C(C(C)C)C1 92262,c1(N(C)CCOCCC2CC2)cc2cn[nH]c2cn1.c1ccc(Cl)nc1C#N 92263,C1(C(C)NC(CC2(OC)CC2)=O)CCCCN1C(C1CCCN1C1CC1)=O 92264,Cc1ccc(Cl)cc1CNCC1(C(=O)Nc2cccc(-n3ccnn3)c2)CC1 92265,N1(C(c2cccc(N(C)C)n2)=O)CCC(C2(NC(C3CC3C(F)(F)F)=O)CC2)C1 92266,C1(CNC(C(C2CC2)NC(c2c(C)nn(C)n2)=O)=O)CC12CCCCC2 92267,CC1(C(N2CCN(CCNC(=O)CC3CCSCC3)CC2)=O)COC(=O)N1 92268,C(c1ccc(C)cc1C)=CC(=O)NC1C(CNC(C2=CC(C)(CC)C2)=O)CC1 92269,C1(C(=O)NCC(CC)NC(=O)C=CCN2CCCC2)(CC)CC1(F)F 92270,CCCCCS(=O)(=O)NC(c1cncc(-c2ccncc2)c1)=O 92271,Cc1cc(N)c(F)c(C(N2CCC=C(CNC(=O)CC3CCCCO3)C2)=O)c1F 92272,Cc1cc(C(=O)NCC(O)CNC(C2COCCN2CC2CCC2)=O)ncc1F 92273,C1(C(=O)NCCN(C(=O)CC2CCCN2C(C)C)CCC)CCC(=O)N(CC)C1 92274,c1(C(N2CCC(O)(CC(=O)NCC3(O)CC(C)(C)C3)C2)=O)ccc(F)c(F)c1 92275,C(=O)(C#CC1CCCOC1)NCC1CC2N(C(c3cc(OC)n[nH]3)=O)C(CC2)C1 92276,C1(NC(C2(CNC(COC)=O)CCC2)=O)CCC(C(N)=O)C1 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92399,c1(OCCC)ccc(C(N2CCC3C(C2)O3)=O)cc1OCC 92400,N1(C(C(CC)O)=O)C2CCC1CC(NC(c1cccc(N)c1C)=O)C2 92401,N1(NC(=O)CC2CC(C(F)F)C2)CCCC(C(=O)NCC(n2cnc(C#N)n2)C)C1 92402,c1(C(N2CC(NC(c3cc(CC)on3)=O)C2)=O)c(Cl)cc(C)cc1Cl 92403,N1(C(C23CC(C)(C2)C3)=O)CCC2CN(C(C3(c4ccno4)CCC3)=O)CC12 92404,CN=c1nc(NC2CCCn3nc(C)nc32)[nH]c(=NCC(C)c2ccsc2)[nH]1 92405,c1(OC)ccc(Br)c(C(=O)NCC2CCCN(C(C3CNC(=O)C3)=O)CC2)c1 92406,c1(N(CCOCC#C)C)nnc(C2CCCCO2)n1CC1CCCO1 92407,C1(N(C(=O)CNC(C2CCCCC2)=O)C)CCCCC1NC(=O)C(CCO)N(C)C 92408,N1(C(C(C)OCC=C)=O)CC=CC(C(=O)NCC2CCOC2(C)C)C1 92409,CCC(C)C(C(=O)N1CC=CC1(C)C(=O)NCCc1cn[nH]c1)OC 92410,C(=O)(CCCCCCn1cc(-c2csc3nccn23)nn1)NCCC1(C)N=N1 92411,c1(C(N(CCCNC(c2csc(Cl)c2)=O)C2CC2)=O)ccc(-c2cc[nH]n2)s1 92412,N1(C(=O)CCOc2cc(F)ccc2F)CCC2(CCN(c3cnc(F)cn3)C2)C1 92413,Cc1cccc(N(C(C=CC(=O)OC)=O)C)c1C.c1(CC2CCCC2)cnn[nH]1 92414,Cc1sc(Cl)nc1C(N1CC(CN(C(=O)C(C)Cn2ccnc2)C)C1)=O 92415,N1(C(c2c(C)cns2)=O)CCC2CCC12CNC(C1CC(OC(F)(F)F)C1)=O 92416,C1(NC(C(C(=O)NC)(C)C)=O)COC2(CCN(C(C3CCC(C)(C)O3)=O)CC2)C1 92417,C1(C)(NC(c2scc(OC)c2)=O)CCN(Cc2nccn2C(C)C)C1 92418,c1(C(C=O)O)ccc(Cl)c(Cl)c1.c1(NC2CC(NC(=O)C)C2)cccc(C(F)(F)F)c1 92419,C1(C(=O)NCC=CCNC(c2cnc(O)s2)=O)(CF)CC(F)(F)C1 92420,Cn1cccc1C(=O)NCCCCCNC(C1(C)CC1Br)=O 92421,C(=O)(C(C)(C)C(C)C)NCCCCC1(NC(CC(=O)NCC)=O)CC1 92422,CC1(C)C(C(c2nnnn2C2CCCC2)NCCn2ccnn2)C1(C)C 92423,CCN=C(NCc1ccc(C2(C)OCCO2)cc1)NC(C1CCCC1)C 92424,c1(CC(=O)NCC(C)(O)NC(=O)COc2ccon2)ccc(C(F)(F)F)c(F)c1 92425,C1(C2CC2)(C(N2C(CC(N)=O)CCC2)=O)CN(C(c2ncn3c2CCC3)=O)C1 92426,c1(C(N2C(CNC(C34C(C)OC(C)(C3)C4)=O)COCC2)=O)scc2c1CCCC2 92427,O=S(=O)(c1c[nH]ccc1=NC1CCCC(C2CC2)C1)NCC(O)Cn1cccn1 92428,c1(C(=O)OC)[nH]ccc1Cn1cc(C2(N(C)C)CC2)nn1.N1CC(C)(C)C1 92429,C1(NC(Cn2ncc(CC)c2)=O)CCCC2CN(C(c3cc(F)n(C)n3)=O)CC12 92430,c1(C(=O)NC2C(NC(c3nn(C)c(Br)c3)=O)C2)ccn2ccsc12 92431,C12(C(N3CCC(O)(CNC(C=C(CC)C)=O)C3)=O)CCC(C1)C(C)(C)O2 92432,c1(NC(C2CC(F)CN2C(=O)C(c2cccc(Br)c2)O)=O)ccn2ccnc2c1 92433,C(CNC(=O)C=CC(=O)NC1CC1)(CC(F)(F)F)NC(CSc1n[nH]c(=N)s1)=O 92434,N1(CCN2CCCCC(C)C2)CC2CN(C(=O)C(c3ccccc3)=O)CC2C1 92435,C12(C(=O)NCC3(CNC(=O)C=Cc4cncs4)CCCC3)OCCCC1C2(F)F 92436,C1(NC(c2n(C)nnc2)=O)CCN(C(=O)Cc2c(F)cccc2Cl)CC12CCC2 92437,c1(NC(N2C(C)(CCC(=O)OCC)CCC2)=O)cc2occc2n1C 92438,N1(C(=O)NCCc2csnn2)CCCC(Cc2ccccc2)C1 92439,C=C1CC2CCCC(C1)N2C(C1(F)CN(C(=O)C(CC)NC(C)=O)C1)=O 92440,C12(CNC(CSC)=O)CCC1CN(C(=O)C=Cc1ccoc1)C2 92441,c1(NC2CCN(C(Cc3nc(C)[nH]n3)=O)CC2)ncnc2c1ncn2C1CC1 92442,N1(C(c2ccc(C)s2)=O)C2CCC1CC(CNC(=O)CC13CNC(=O)C(C1)C3)C2 92443,Cc1[nH]nc2c1CCC(C(=O)NCCc1coc3ccccc13)C2 92444,c1(C(N2CCCC(NC(C3(CC=C)CC3)=O)C2)=O)c[nH]c2cc(Br)ccc12 92445,CC1=CCSC1C(=O)N(C1CCN(C(c2cnc(Cl)s2)=O)C1)C 92446,CCC1=NOC(C(N2CCC(C(C)C(=O)NCCCc3cnc[nH]3)C2)=O)C1 92447,c1(COC)nc(C(=O)NCC2CC2CNC(c2cc(Cl)cs2)=O)cs1 92448,N1(C(C(C)N2CCCC2)=O)CC2C=CC1C(C(=O)NCCc1cn(C)cn1)C2 92449,O=C(C1=CS(=O)CCC1)NCC1CCCCCN1C(c1cc(=O)cc[nH]1)=O 92450,N1(C(C=CCC(C)(C)OC)=O)CCN(C(c2cc(C)nc(C)c2)=O)C(C2CC2)C1 92451,C(=O)(CC(C)CNC(=O)C(C)(C)CC1CCOC1)N(C)Cc1ncc(C)o1 92452,N1(C(C2(SC)CC(=O)C2)=O)C2CCC1CC(N(C)Cc1ccc3c(c1)OCO3)C2 92453,C1(NC(C(CC)(F)F)=O)CS(=O)(=O)CC1NC(=O)C(C)(C)OCC(F)(F)F 92454,N1(C(CCCCCC#C)=O)CC2CCCC(NC(C3CCNC3=O)=O)C2C1 92455,c1(C(=O)NCC2(CCNC(c3conc3C3CC3)=O)CC2)cccc(F)c1Cl 92456,c1(CC(=O)NC2(C)CN(C(COCc3cc(C)no3)=O)C2)ccccc1S(C)=O 92457,c1(C(C(F)(F)F)OC(C(c2n(C)cnc2)O)=O)cccc(C(F)(F)F)c1 92458,c1(C(=O)OC)ccc(C(N2CCSC(C)C2C)=O)cc1Br 92459,c1(NC(c2c(C(=O)NC3CC3CC3CC3)cc[nH]2)=O)cc(O)nc(O)n1 92460,c1(C(C(=O)NCC2(CO)CC2)N(C(=O)CC(F)(F)F)C)ccc2c(c1)sc(=O)n2C 92461,c1(OC)ncc(C(F)(F)F)cc1C(=O)NCC=CCNC(=O)C(O)CC1CC1 92462,C(=O)(CCC(C)C#N)NCC1(F)CC(NC(c2c(CC)nn(C)c2)=O)C1 92463,C1(C)(NC(CO)=O)CCC(C)C1.C1(C(N(c2ccccc2)CC)=O)(C)CCCC1 92464,C(=O)(CCC(C)(C)NC(=O)C(C)CC#N)NC1(C(=O)OC)CCC1 92465,Cc1ccc(O)nc1CNC(=O)CC(C)(C)CNC(C1OCCC1C(C)C)=O 92466,C(C(C)C(F)C(=O)NCC1COCC1N(C)C)NC(C(CC)C)=O 92467,CC(C)C1C(=O)N1.c1(NC2C(CNC(=O)OC(C)(C)C)CC2)ncccn1 92468,Cc1cc(C)c(C(N2CCCC(NC(=O)CN(C)S(N)(=O)=O)C2)=O)cc1N 92469,c1(CN(CCCSC)C)cc(Cl)cc([N+](=O)[O-])c1.C1(OC)COCCC1C 92470,c1(C(N(CCN(C(=O)C2=NOC(C(C)C)C2)CC)CC)=O)cc(C)nnc1O 92471,c1(C(=O)NCC2N(C(C(C)Cn3ccnc3)=O)CCC2)cc(N)ccc1O 92472,C(=O)(C(C)(C(C)C)OC)N1CCC(N(C(CCCN(CCC)C)=O)C)CC1 92473,c1(C(=O)NC2CC(CC(=O)N(CCCC)CCOC)C2(C)C)cc(C#N)cn1C 92474,C1(NC(C(CC)CO)=O)CC2(CCN(C(=O)CC3C=CCCC3)C2)C1 92475,C1(CNC(Cn2c(CCC)nnc2S)=O)CCN(C(=O)C2=CC(C)(C)C2)C12CC2 92476,c1(C(N2CCN(C(C3CC(C)SCC3)=O)CC2C)=O)cccc2c1C(=O)CC2 92477,C(=O)(C(C)(C)CS(C)(=O)=O)NCC(C)(CO)NC(c1cc2ncccc2[nH]1)=O 92478,c1(OC(C2(C)ON=C(C(C)C)C2)=O)ccnc2cc(Br)ccc12 92479,Cn1nc(C(C)(C)C)cc1NC(C1C(CNC(C2CCCSC2C)=O)C1)=O 92480,CC1CN(C(C2(C(F)(F)F)CCOCC2)=O)CC(C)N(C(c2csc(Cl)c2)=O)C1 92481,c1(C(=O)NCC2C(NC(C3(C(N)=O)CCC3)=O)C2)cccc(F)c1F 92482,C=CCCCCC(=O)NC(C)C(C)NC(c1cc(C2CCCCC2)on1)=O 92483,C12(N(CCN(C(C)C)C(c3ncccn3)=O)C)CC(C)(C1)OC2C 92484,N1(C(C(CC)F)=O)CCN(C(C2CC(N(C)C)C2)=O)CC1c1cnn(C)c1 92485,c1(CC(=O)NCC2CCC(C)CN2C(C2CC=CCC2)=O)nnc2n1CCOC2 92486,Cc1cc(CNC(c2[nH]ccc2C2CC2)=O)oc1C(=O)NCc1cnc(O)[nH]1 92487,C1(CC)N(C(C2(C(C)C)CCN(C(c3cccnc3O)=O)C2)=O)CC1(C)C 92488,N1(CCNC(CSS(C)(=O)=O)=O)CCCN(C(=O)C=Cc2cn[nH]c2)CC1 92489,C(=O)(C(CC(=O)NCC)N(C)C)NC1CC(NC(C2(c3ccc(C)cc3)CC2)=O)C1 92490,C1(CCC)CC(NC(=O)C(N2CC(c3ccc(Br)cc3)C2(C)C)=O)CCO1 92491,C1(CS(=O)(=O)CC(N2CCC(C(=O)O)C2c2ccco2)=O)CC2(CCC2)CO1 92492,c1(SCC#C)cccc(C(=O)NC(C)CCCNC(=O)C(C)OCC(C)C)c1 92493,N1(C(C(c2ccc(F)cc2)(C)F)=O)CCC(C2(NC(=O)C(O)C3CCC3)CC2)C1 92494,CC1=CCN(C(c2cc(CCNC(C3(N(C)C)CC3)=O)on2)=O)C1 92495,c1(C(=O)NCCOCCNC(C2(CO)CCCO2)=O)n[nH]c2c1CCC2 92496,c1(C(=O)NCCCC2(NC(COCCCOC)=O)CC2)ncnc2sccc12 92497,Cc1cnc(F)c(CNC(=O)C(c2cccs2)NC(=O)C2=CCCCC2)c1 92498,N1(C(CN(C2CCC2)C)=O)CCCCC12CN(C(C1(c3ccno3)CC1)=O)C2 92499,c1(NC)cnc(Cl)cc1C(=O)NC(CNC(C1CCCC(=O)N1)=O)C1CCC1 92500,c1(SC)nc2nc(C)c(CC(=O)NC3COC4(CCN(CCF)C4)C3)c(C)n2n1 92501,C1(C(N(C)CC2CCSC2)=O)C2CC3C(C2NC(c2cc(=O)n(C)cn2)=O)C13 92502,N1(C(C(F)=C(C)C)=O)CCc2ccccc2C1CNC(=O)CC1NC(=O)NC1=O 92503,C1(C(N2CCC(c3ccccc3)C2)=O)CN(C(C2CC2C2CC2)=O)CCC1(F)F 92504,c1(NC2CN(C(=O)O)C2)cccnc1.C1(CN)CCCO1.CC(C)(C)N1CC1=O 92505,Cc1cc(CC(N2CCC(NC(=O)Cc3cc(-c4ccco4)on3)C2)=O)cs1 92506,N1(C(C2CCC(NC(C3CC(C)(F)C3)=O)C2)=O)CC(C(N)=O)C(C(C)C)C1 92507,N1(C(COc2cc(C)cc(C)c2)=O)CCN(C(=O)C=Cc2cocn2)C(C)C1C 92508,C=CCCCCC(=O)N1CCCOC(CCNC(=O)CC(C)NC(N)=O)C1 92509,c1(C(N(C2CCC(NC(=O)CCCn3cncn3)C2)C)=O)cnc2ccsc2c1 92510,N1(C(CC(=O)NC)=O)CCCC1(C(=O)NCC=Cc1ccco1)C(C)C 92511,C1(O)(C(C)CNC(C2(C)CC2)=O)CCN(C(C2(CF)CC2)=O)C1 92512,C1(CNC(COCCCC(C)C)=O)CN(C(C2CC2(C)C(F)F)=O)CCO1 92513,Cc1nnc2cc(N3CCCC(CCNC(=O)CC=C(Cl)Cl)CC3)ncn12 92514,c1(C(N(C=O)Cc2csc(C)n2)C)cnccn1 92515,c1(NC(CCN(C(C2CN(CC)C(=O)C2)=O)C(C)C)=O)ccc(F)c(C)c1 92516,c1(C(c2nnnn2C2CCOC2)NCC2(COC)CC2)cc(Br)c[nH]1 92517,CC1CCN(C(=O)C(C)N(C)C)C1CNC(=O)C(=Cc1cccn1C)F 92518,c1(N2CCN(C(CSC)=O)CC2)nc(N2CCC(C(C)C#N)CC2)cc(C)n1 92519,Cc1ccc(C(N2CC(CC(F)C(=O)N3CC(C4CCCO4)C3)C2)=O)[nH]1 92520,C1(CC(=O)NC2CCCC2C(=O)NC2CC2c2cccnc2)CC(O)C12CCC2 92521,C1(C2CCN(C)CC2)(C(=O)NC(CC)CNC(=O)CCC2CC2(F)F)CC1 92522,C(=O)(C1=C(Cl)CCCC1)NC12CCCC(NC(Cc3cc(C)c(F)cc3)=O)(C1)C2 92523,O=S(=O)(c1cccc(=NCc2ccoc2)[nH]1)NC1CC1Cl 92524,CC(C)CC(C)C(=O)NC1CCN(C(C2(C(F)(F)F)C=NC=C2Cl)=O)C1C 92525,c1(C(=O)NC(CC=C)CNC(=O)CCc2nncs2)c(Cl)cccc1Cl 92526,C(=O)(C(C)(O)C(C)(C)C)NCC(CN(C(=O)CSc1ccccc1[N+](=O)[O-])C)O 92527,Cc1cccc(CNC(C2CCCCN2C(=O)C(O)CC2CCCC2)=O)c1 92528,n1(CCC(=O)OCc2c(NCC)nccc2)nc(C)c(C)c1C 92529,N1(C(C(=O)NC(c2ccccc2)C)c2cnsc2)CCC(C)(CC2COC2)CC1 92530,N1(C(C2(COCC)CCOCC2)=O)CCC(C(C)(C)O)(CNC(=O)CCF)CC1 92531,c1(C(C(=O)NCC2CN(C(C(c3ccc(F)cc3)OC)=O)C2)C)cccc(F)c1 92532,c1(C(N2CCC(C(C(=O)NCC3C4CCCC34)F)C2)=O)cnn2c1CCC2 92533,N1(C(Cn2ncn(C)c2=O)=O)CCCC1C1CCCN1C(=O)OC(C)(C)C 92534,c1(C(=O)NCC2N(C(CN3CC(C)C3)=O)C3C(C2)C3)ccn(CC(F)F)c(=O)c1 92535,C1(C(=O)NC(CCNC(C2(C(F)F)CC(=C)C2)=O)C)CN=C2N=CNN2C1 92536,C12(C(=O)NN3CC(C(C)N(C(=O)CCCN(C)C)C)C3)CCCCC1C2 92537,Cc1c(C(=O)NC2CCC(C(C)NC(c3cccnc3O)=O)C2)nnn1C 92538,C1(NC(c2ccc(C(C)C)s2)=O)CCC(NC(=O)CCC2CCCCN2C)CC1 92539,N1(CCN2CCC(C)CC2)CC(NC(N2CCCS2(=O)=O)=O)CCC1C 92540,N1(C(CC2(C)CCCO2)=O)CC2CCCC2(NC(c2cc[nH]c2C2CC2)=O)C1 92541,N#Cc1cncc(C(=O)NCC2(C(=O)NCc3cc(CO)ccn3)CC2)c1 92542,c1(SCC)ccc(-c2cc(C(=O)Nc3ccc(Br)nc3C)ccc2OC)cc1F 92543,C1(C(=O)NC(c2ccccc2)COC)CCC(NC(c2ccncn2)=O)CC1 92544,c1csc(C(=O)OC)c1.C(C(=O)NCC(=O)N(C)CCOC)SCC 92545,C1(CC)CN(C(c2ccsc2C#N)=O)CC1C(N1CCOC(C)C1)=O 92546,C1(C(=O)NCC(C)(C)NC(c2nnc(C)s2)=O)CCCC(F)(F)CC1 92547,C(=O)(C(C)(F)C(=O)NC1COCC1NC(c1sccc1SC)=O)OC 92548,c1(C(N2C(CCCNC(C3(C)CC3(Cl)Cl)=O)CCC2)=O)ncc(F)cn1 92549,C1(C(C)C)CN(C(c2cnnn2C(C)C)=O)CCN1C(C12CCC(F)(CC1)C2)=O 92550,c1(C(=O)NCCC(O)CCc2ccccc2)cc(O)c(C(F)(F)F)cc1I 92551,C1(C(=O)NCC(CC=C)NC(=O)C=CCN2CCOCC2)CC2C=CC1O2 92552,c1(C(=O)NCCCCC(C)NC(=O)CCCCCC#N)nc[nH]c2ncnc1-2 92553,c1(C(N2CC(NC(C(F)OC)=O)C(F)C2)=O)ccc2c(N(C)C)ncnc2c1 92554,c1(C(=O)NCCCN(C(C(C)OC)=O)C)c2c(c[nH]c1=N)CCC2 92555,C1(NCCc2c(F)cccc2)Cc2cscc2C1 92556,N1(C(c2c(NCC)scn2)=O)CC(NC(=O)CCOc2cccnc2)C2CC12 92557,C=CCC(C(=O)NCC(=O)NC(C)C)NC(c1cnn(C)c1)=O 92558,C1(C(=O)NCCN(C(=O)OC)C)(NC(C2CC(F)C2)=O)CCOCC1 92559,C12(C(=O)NC(CNC(c3nc(C(C)OC)sc3)=O)(C)CO)CCCC1CCC2 92560,C1(C(=O)NCC(CO)NC(c2cnc(Cl)n2C)=O)(OCC)CCCCCC1 92561,C(CCCCC(=O)N1CCC(NC(c2cn(C)c(C)n2)=O)CC1C1CC1)SC 92562,N1(C(C(C)CSC(F)(F)F)=O)CCC2(CC1)CC(NC(=O)CSc1nc[nH]n1)C2 92563,c1(C(N2CCN(C(Cc3n(C)cnc3)=O)C3C2C3)=O)nccc2ncccc12 92564,c1(OC)c(C(N2CCN(CC3CN(C(=O)CC4CCC4)C3)CC2)=O)c(C)nn1C 92565,C1(C(=O)Nc2c(C)cc(NC(C34CC(C)(CO3)C4)=O)cc2)CCCC(F)(F)CC1 92566,c1(C(N2CCC(C)(NC(CC(C)OC)=O)C2)=O)cc(S(=O)(=O)N(C)C)cnc1O 92567,C1(CN(C(C(C)c2ccsc2)=O)C)COCCN1C(c1sccc1Br)=O 92568,C(=O)(CC1=CCOCC1)NCC(CC(C)C)(C)NC(=O)Cn1ncnn1 92569,CC1(NC(=O)C=CC(=O)N(C)C)CCCCC1CO.c12ccc(cc1)NC(=O)C2 92570,c1(CCC(=O)NCC(CC)NC(C2CC2F)=O)cccc(OC(C)C)c1 92571,N#Cc1ccc(C2(NC(=O)Cn3cc(-c4cccnc4Cl)nn3)CCC2)cc1 92572,Cn1ncc([N+](=O)[O-])c1C(=O)NCCC(C)(C)NC(C1CC1c1cccnc1)=O 92573,N1(C(C=Cc2c(C)ccnc2)=O)CC2CCC1CC2NC(C1CC12CCOC2)=O 92574,C1(C(C)(C)Nc2nc(C)[nH]n2)CCN(C(=O)COC2CCCC2)CC1 92575,c1(SC)ccc(C(N2CC(OC)C(O)C2)=O)cc1.C12CC(COC(C)=O)CN1C2=O 92576,Cc1ncc(C=CC(=O)NCC2(F)CC(NC(=O)C(C)c3ccsc3)C2)c(O)n1 92577,N1(C(CC2C(=O)NCCC2)=O)Cc2occ(C(N3CCC3C3CCC3)=O)c2C1 92578,C1(CNC(C(C)OCCOCC)=O)(COC)CCCN(C(=O)C(C)N(C)C(C)C)C1 92579,C1(C(=O)NCC(CCCC)NC(=O)Cc2nccs2)CNc2ccccc2O1 92580,CCCCC(CC(=O)NC(C)CCF)NC(C1CC2CCC1O2)=O 92581,C(=O)(C(C)(C)CCCC1CCCCC1)NC(c1nnc(C2CCCN(C)C2C)o1)C 92582,c1cc(C2CC2)c2c(c1)C(Nc1nnnn1Cc1ccccc1)CCC2 92583,Cc1c(C(N2C3CCC2C(NC(=O)C(c2ccc(F)cc2)F)C3)=O)cccc1O 92584,CON1CCC(CC(=O)NC2COCCN(C(c3n[nH]c4c3COC4)=O)C2)CC1 92585,C1(C(=O)NCC(CC)NC(=O)Cn2nc(C)cc2C(F)F)CC(=O)N(CC(C)C)C1 92586,c1(C(N2CC(OCCNC(C3(C=C)CCOCC3)=O)C2)=O)ccc2cnoc2c1 92587,c1(C(=O)NCC(C(C)C)NC(C2(OC)CCOCC2)=O)cnc(C(F)F)c(C)c1 92588,Cn1cccc(C(=O)NCC2CCN(C(C3CC3CC(C)(C)C)=O)CC2)c1=O 92589,c1(-c2scc(C(=O)NC(C(C)NC(CC=C)=O)C)n2)ccccc1OCC 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92607,CC1C(C(=O)Oc2cccc(-c3ccncc3)c2)CCCCC1C=O 92608,C12(C(N(C)CC3CN(C(=O)CC4=CCCC4)CCO3)=O)CCCC(C)(C1)OC2 92609,N1(CCCO)CCCC(CCOc2cc(NC)ncc2)C1.C1(O)CCOC1 92610,C(=O)(CCCC(=O)N(C)C)NCC(C1CCCC1)NC(c1[nH]c(CC)c(Cl)n1)=O 92611,CC1CCC(C(=O)NCCCNS(C)(=O)=O)C1.C1(C)(C)C(=O)N1 92612,C(=O)(C(CC(F)F)C1CCC1)NC(CNC(=O)COc1cccc(F)c1F)CO 92613,C1(NC(C2N(C(CCC)=O)CCC2)=O)C2CC1N(C(C1CC3CCCC13)=O)C2 92614,C12(NC(c3snc(O)c3Cl)=O)CCC1CN(C(=O)CCOc1cccnc1)C2 92615,N#Cc1ccc(CCC(=O)N)c(F)c1.c1(C(CO)=O)cccc2sccc12 92616,CC1=NOC(C)(C(=O)NC(C2CN(C(C3COC(=O)N3)=O)CCO2)C)C1 92617,N1(C(c2ccnc(Cl)c2)C(=O)NCC2CC2)CCC2(CC1)OCc1ccncc12 92618,N1(C(C(c2c(C)ccc(F)c2)(F)F)=O)CCCC2(CCCC2)CC1 92619,c1(C(N2C3(CNC(CC(C=C)C)=O)CCCC(C2)C3)=O)ccc2oc(C)nc2c1 92620,C(=O)(CS(=O)(=O)CC(C)C)NC(C1(O)CCN(C(C(CC)C)=O)CC1)C 92621,S(=O)(=O)(c1cnc2ncc(Cl)cn12)N1CCC2(CCC(C)CC2)C1 92622,N1(C(c2cnc(CC)[nH]2)=O)CC(C)N(C(=O)Cc2coc3ccccc23)CC1C 92623,Cc1noc(C)c1CCN(C(C1(F)CN(NCCC(C)C)C1)=O)CC1CCCC1 92624,N1(C(c2n(C(C)C)cnc2)=O)C2COCC1CC(NC(=O)C(C)CC(N)=O)C2 92625,c1(C(=O)NC(CNC(CC2(C)CC2)=O)(C)C2CCC2)csc(-c2ccccc2)c1 92626,C1(NC(C=CC)=O)CS(=O)(=O)C2CN(C(c3nnn(C4CCOC4)c3C)=O)CC12 92627,C(=O)(C(C)NC(=O)OC(C)(C)C)NC1CN(C2(C(=O)NC)CC2)C1 92628,C(CN=c1ccn2c(Br)cnc2[nH]1)C1CCN(C(c2c(C(=O)OC)cn(C)n2)=O)C1 92629,C1(CNC(C2(CC=C)CC2)=O)C2CN(C(c3ccsc3Br)=O)CC12 92630,CCCC(O)C(CO)NC(C1OCCC1NC(=O)CC1CCCC1)=O 92631,N1(C(C(C=C)OC)=O)CCN(C(c2c(SCC)cccc2C)=O)CC1C1CC1 92632,c1(OC)ccc(CN2CCC(CC(N3CCCC3C(N)=O)=O)C2)c(Br)c1 92633,C1(CNC(c2n(CC)cnn2)=O)CCN(C(=O)CC23CCCC2C3)C1(C)C 92634,c1(CC(N2CC(NC(C3CCC3)=O)C3C2C3)=O)cc(F)cc(Br)c1 92635,CCC(O)C(C)(C)C(=O)N1CC2CC1C2NC(=O)CCCN(C)N=O 92636,S(=O)(=O)(CC(=O)N1CCCC(N(C)C(C2CCCCN2CC(F)F)=O)C1)NCC 92637,CC1(C(N2CCC(CNC(C3(C(F)(F)F)CCOCC3)=O)C2)=O)CC=CCO1 92638,c1(CC(=O)NCC2CN(C(CNC(C)=O)=O)C2)csc(NC=O)n1 92639,Cc1ncc(Br)cc1-n1cc(C2CCCN(C(c3sc(Cl)nc3C)=O)C2)nn1 92640,c1(C(=O)NCCCNC(CN2CCN(CC(C)C)CC2)=O)cccc2nc[nH]c12 92641,Cc1cc(N)cc(C(=O)N(CCCNC(=O)C(c2ccccc2F)C)C)c1F 92642,c1(C(C)C)cccc(C(N2CCCCC2CNC(=O)C(C)(C)c2cscn2)=O)c1 92643,C(CN=c1[nH]c(=NCc2nn(C)c(SCCO)c2Br)[nH]c2c1COC2)OC(C)C 92644,c1(C(=O)NC2C(NC(=O)Cn3ncnn3)C2)cccc(OCCCF)c1 92645,N1(C(C2CCCC2)=O)CCN(C(=O)C=CC2CCCCC2)C(c2ccncc2)C1 92646,c1(C(=O)NC2CN(C(C3(C#C)CCCC3)=O)CC2O)ccc(Cl)c(C)c1Cl 92647,N1(C(C(C)SCC)=O)CC(CNC(=O)Cc2ccc(C)c(OC)c2)C(F)(F)C1 92648,C1(C(=O)NC2C(CNC(=O)Cn3cnc([N+](=O)[O-])n3)C2)CCC2(CCCCC2)C1 92649,c1(C(=O)NC2(CC=C)CCN(C(=O)C(C)(CC)CO)C2)ccc(O)c(OC)c1 92650,c1(C(=O)NC2CC(F)(CNc3c(C)c(Cl)ncn3)C2)c(C)cc(=O)oc1C 92651,N1(C(c2c(C)noc2)=O)C2CCC1CN(C(=O)C(C)NC(=O)C1CC1)C2 92652,O(NC(=O)CC(C)NC(C1CCCN(C(C)C)C1)=O)CCOC(C)C 92653,N1(C(C2(N(C)C)CCCCC2)=O)CCCN(C(C2CSCN2C)=O)C(CO)C1 92654,C1(NCc2c(C)scc2OC)CC2(C1)CC(C(=O)OC1CCCCC1)C2.C(CO)S 92655,C=C(C)C(CC(=O)N1CCCC(N(CC2CC2)CC)C1)OCC.C(C)(C(=O)NC)C 92656,c1(C(=O)NCCC2(OC)CN(C(c3ncc(CC)cn3)=O)C2)c[nH]cc(C)c1=O 92657,CCC(CCOC)C(=O)N1CCOC(C)(CNC(=O)CCC(=O)NCCCOC)C1 92658,c1(OC)nc(C)ccc1C(=O)NCC1(CCNCC2(c3cnn(C)c3)CC2)CC1 92659,Nc1nonc1C(=O)NCC=CC(C1CN(C(=O)Cn2ccnn2)C1)N1CCCC1 92660,N1(C(c2cn(CCOC)nn2)=O)C2CCC1C(CNC(C1CC(O)C1)=O)C2 92661,CC1OCCN(C(C2CCCN2C(C2CC3(CCC3O)C2)=O)=O)C1CO 92662,N1(C(CCSCCCC)=O)CC2CCCN(C(c3ncoc3C)=O)C2C1 92663,C1(NC(CC2C(C)(C)C2)=O)CC2(CCCN(C(c3c(Cl)csc3Cl)=O)C2)C1 92664,c1(OC(C)=O)ccc(C(=O)OCC(=O)C2(Cl)CC2)c(F)c1F 92665,c1(C(=O)NC2C=CC(CNC(C3CN(OC)C(=O)C3)=O)C2)ccn2c1CCCC2 92666,Cc1cccc2[nH]cc(CCC(=O)NC3CCN(C(=O)C(C)S(N)(=O)=O)C3C)c12 92667,N1(C(C(CCC)NC(C)=O)=O)CCCC(F)(CNC(C2SCCCS2)=O)C1 92668,c1(CC)ccc(F)c(C(=O)NCC2COCCN(C(=O)CC(C)C(F)F)C2)c1F 92669,C(=O)(C1CSc2ccccc21)N1CC(OCCNC(C2CN3CCN2CC3)=O)C1 92670,C1(CNC(CC2(C)OCCO2)=O)CC(C(F)(F)F)CCN1C(=O)CCCN=[N+]=[N-] 92671,C(=O)(C1=NN(CCO)C(=O)CC1)N1C(CNC(COCC#C)=O)C(C)(C)CCC1 92672,C(C(C(=O)N(C)Cc1nccn1CC)C(C)(C)C)NC(c1oc(CC)c(C)c1)=O 92673,N1(C(c2c(SC)cn(C)n2)=O)CCC(NC(c2ccccc2C(F)F)=O)C(C)C1 92674,CC(C)(C(=O)N1CC2CC1C2NC(=O)CN1C(=O)NC(C2CC2)(CO)C1=O)C(F)F 92675,C(=O)(C(C)CCCC(C)C)NC(CC=C)CNC(=O)C=CC(=O)N(C)C 92676,N1(C(C2(COC)COC2)=O)CCC(CO)(NC(=O)CN2C(=O)CNC2=O)C1 92677,c1(C(N2C(CNc3cc(OCC)ncn3)CCCC2)=O)ccc(C#N)nc1C 92678,N1(C(c2cnc(C)nc2C)=O)CCCC2(CCN2C(c2cnc(Cl)c(I)c2)=O)C1 92679,CCC(O)C(C)(C)C(=O)NCCCN(C(=O)CCNC(C1CCCCCC1)=O)C 92680,c1(C(=O)NCCC(CCNC(c2ccc(C#C)cc2)=O)C)c(C)cc(C)cc1C 92681,c1(OC(C)C)cccc(NCC(=O)NCC#CCNC(=O)CCC2CCCC2)c1 92682,C1(CNC(C(C)c2cc[nH]n2)=O)(CN(C)C)CCN(C(=O)Cc2nc[nH]n2)CC1 92683,N1(C(COCC)=O)CCCCC1C(C)NC(c1cnn(C(C)C)c1F)=O 92684,Cc1ccc(F)c(N)c1C(N1CC(NC(=O)C=Cc2c[nH]nc2C)CC(F)C1)=O 92685,c1(OCC(=O)NC(CNC(C(C)CO)=O)C(C)(C)C)ccccc1C(F)(F)F 92686,CCCCC(O)C(=O)N1CCCC1(C)CNC(=O)CCSc1n[nH]c(C)n1 92687,c1(OC)cc(F)cc(F)c1C(C)Nc1ncnc(N2CCC(OCCO)CC2)c1C 92688,N1(C(c2c(C)cc(C)o2)=O)CCC(NC(=O)C(C)CN2CCOCC2)C12CC2 92689,C1(NC(c2cc(SCC)on2)=O)CN(C(=O)C(C(C)C)N(CC)CC)CCC1(C)C 92690,c1(C(C)C)cnc(C#N)c(Oc2ccc(=O)n(-c3ccc(F)cc3)n2)c1 92691,S(=O)(=O)(c1ccc(C=CC(=O)NC2CCSC3(CCC3)C2)cc1)OC(C)(C)C 92692,C(=O)(CCCC(=O)NC(C)C(CO)NC(C1NC(=O)OC1C)=O)NCCC 92693,c1(CC)nn(C)cc1C(=O)NCC(n1cc(CC2CCCCC2)nn1)C 92694,Nc1cccc(C=CC(N2CCOC(CNC(C3CCCCCCC3)=O)C2)=O)c1 92695,c1(C(N2C3CC(NC(C4CCS(=O)(=O)CC4)=O)C2CC3)=O)ccc2nnnn2c1 92696,C1(CNC(NC(C)C)=NCCC2C(C)C2(F)F)C(F)(F)C12CCOCC2 92697,c1(C(=O)NCC2(COC)CN(C(C3CN(C)C3)=O)C2)cc(Cl)cnc1OC 92698,c1(N)ccccc1F.C1(N(C(=O)CCOC)CC)CCN(C(=O)CC(C)COC)CC1 92699,C1(C(=O)NCCN(C(=O)CCc2nccs2)C)CC(N(C)C)CCO1 92700,C(=O)(CCC(C)(F)F)N1CCC(CN2CCN(C(C3C(C)C3)=O)CC2)CC1 92701,c1(C(N2CCC(N3C(=O)C3C3CCOC3)C2)=O)cc2cscc2s1.COOC 92702,c1(C(=O)NCC2(C(N3CCN(C)CC3C(F)F)=O)CC2)cc2ccc(Cl)cc2s1 92703,C1(C2CCCC2)(NC(C2C3CN(C(C(CCC)F)=O)CC32)=O)CC1 92704,N1(c2cc(OC)ncn2)CCC2(CCN(C(=O)C(C)S(=O)(=O)C(C)C)CC2)CC1 92705,c1(C(N2CCN(C(c3sccc3C3CC3)=O)C3C2C3)=O)cccc2scnc12 92706,N1(C(C=CCC)=O)CCC2CCN(C(c3c(C)[nH]c4ccc(O)cc34)=O)CC2C1 92707,C1(C2CC2)(NC(c2c(C)nccc2)=O)CCN(C(=O)COc2cccnc2)CC1 92708,C(=O)(CC(C)(C)CNC(C1(C)CC(=O)C1)=O)NC(C(=O)N(CC)CC)C 92709,C1(NC(c2ccc(C(C)C)cn2)=O)CCN(C(C2CC3(CSC3)C2)=O)C12CCC2 92710,CC1OC2(C)CC1(C(=O)N(C1CCN(CCOCC(F)(F)F)CC1)C)C2 92711,c1(CCC(C(=O)C(C)(C)C2CCOC2)=O)nnc(S)nc1O.C1(NC)CNC1 92712,n1(CCC)ccc(=NC(=O)C23COCC2CN(C(=O)Cn2nccn2)C3)[nH]1 92713,Cc1ncc(NC(=O)CC(O)C2CN(C(=O)CC=Cc3ccccc3)C2)cc1Cl 92714,C(=O)(C(C)(C)Cc1ccccc1)NCC(C)NC1CC(F)(CC2C3CCCC23)C1 92715,Cc1ccc(C(=O)NCC2(C(C)(C)O)CN(C(C3CCOC3)=O)C2)nc1F 92716,c1(OC)cc(Cl)ccc1C(N1CC(CO)(NC(=O)CC2(C(F)(F)F)CC2)C1)=O 92717,C(=O)(C1=CCc2ccccc21)NC(C)CNC(c1csc(CCC(F)(F)F)n1)=O 92718,C(=O)(CC1=CCN(C(=O)CN2CCCC2)CC1)NCCc1nccc(C)n1 92719,N1(C(Cc2c(C)ccs2)=O)CC(NC(=O)CN2CCC2)CC1C 92720,N1(C(c2c(C)cccc2C)=O)CC2CCC1C(CNC(C1(C(F)F)CCC1)=O)C2 92721,CC(CC1CCC1)C(=O)NCC1CCN1C(=O)CN1CC=CC1 92722,C=C=C(C)CC(=O)N1CC=CC(C(=O)N(CCCC)CCO)C1 92723,C(=O)(CC(CC(C)C)NC(=O)OC(C)(C)C)NC1(CNC(CC(C=C)C)=O)CCC1 92724,c1(OC(C(=O)NCC2C(NC(C(C)(C)OC(C)C)=O)CC2)C)ccc(Cl)cc1 92725,c1(C(N2CCC(CNC(C3CCN(C(C)=O)C3)=O)C2)=O)ccc2c(c1)COC2(C)C 92726,c1(C(C(=O)C2CC2)=O)cnc2nc(NCc3ccc(I)cc3Br)ccc2c1 92727,CC1CCc2ncc(C(N3C4CCC3CN(C(C3CCCN3C=O)=O)C4)=O)n2C1 92728,C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)N(CC(C)NC(CC(CC)C)=O)CC 92729,N1(C(c2c(C)cnn2C)=O)CCCN(C(=O)CCNc2cccnc2)CC1 92730,C(=O)(N(NC(=O)C1CCOC(C)(C)C1)C(=O)N(C)C)OC 92731,c1(OC)nccc(C(N2CC3(C2)CN(C(C2CCCCNC2=O)=O)C3)=O)c1F 92732,CCC(CNC(=O)C(CCOC)NC(c1ncc[nH]1)=O)(CC)C(N)=O 92733,c1(C(c2n(C(C(=O)NC)C)nnn2)NC2CCC(CO)O2)ccc(C#N)cc1F 92734,c1(OCC(=O)NC2CC(NC(c3ccn(CC)n3)=O)C2)cccc2cccnc12 92735,C1(C(=O)NCCCN(C(C(C2CC2)OC)=O)C)CCc2[nH]nc(O)c2C1 92736,CCC(F)(F)CC(=O)NC(C(=O)NCc1[nH]c(C)nc1C)C1CCCC1 92737,C1(NC(C(N2CCCCCC2)C)=O)CC2CCC1N(C(=O)CCC(N)=O)C2 92738,C1(CNC(C(C)(C)SC)=O)CCN(C(c2nnn(C)n2)=O)CC1C 92739,c1(-c2ccc(NCCCn3c(C)cc(C)n3)cc2)cc(C)c(C)nn1 92740,C(c1cccc(O)c1)=CC(=O)NC1CN(C(CCCOC(C)=O)=O)C2C1C2 92741,CC(C)(C)S(=O)(=O)CC(=O)NCCC1CN(C(c2csnn2)=O)CCO1 92742,CC1OC2CCC1(C(=O)N(CCCNC(=O)COCC1(F)CC1)C)C2 92743,N1(C(c2c(=N)[nH]cnc2)=O)CC(NC(=O)C2=CCCSC2)CC12CCOC2 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92761,c1(C(=O)NC2CCCN(C(=O)C(O)CCn3cncn3)C2)cccc2c1CCCC2 92762,C1(C(N2CC(C)C(CNC(c3csc(S)n3)=O)C2)=O)CCc2nnc(O)cc2C1 92763,c1(C(=O)NCC(C)CNC(C2CC3(C2)CC(F)C3)=O)cccc(C(N)=O)c1N 92764,c1(C(=O)NC2CN(C(C(CC)n3nccc3C)=O)C2)cc(C)cc(Cl)c1 92765,C1(SC)CCN(C(=NCc2nnn(C)c2C(F)(F)F)NCC2(OC(C)C)CCC2)C1 92766,C1(F)(CNC(C(N2CCOC2=O)C)=O)CCN(C(=O)C(C)N2CCC2)C1 92767,c1(C(C(=O)NCCC2N(C(C(C3CC3)SC)=O)CCC2)O)cccc(F)c1 92768,C1(N(C)C(C2(NC(=O)C(C3CCOCC3)F)CSC2)=O)CCCCC1O 92769,N1(CC)CCN(CC(N2CCCC(N(C(=O)C(C)CF)CCO)C2)=O)CC1 92770,c1(C(=O)NCC2C(NC(c3c(CC)oc(C)c3)=O)C2)cnc(OC)c(Cl)c1 92771,C1(CCNC(CC=CC)=O)CC(F)(F)CN1C(=O)C(C)Oc1ccncc1 92772,C(C(N=[N+]=[N-])C(=O)N1CCOCC(NC(c2ccc(Cl)nc2Cl)=O)C1)OCC 92773,c1(CC)cnc(O)c(C(N2CCC(O)C(NC(C3SCC=C3C)=O)C2)=O)c1 92774,C(=O)(CC(C)(C)CCCCC)N1CCCC(CCOC)(NC(C2C(=C)C2)=O)C1 92775,C1(CCOC)(NC(C2CC2(Cl)Cl)=O)CCN(C(c2cccc(F)c2)=O)C1 92776,c1(CNC(N(CC2C(CC(C(=O)OCC)F)CC2)CC)=O)n[nH]c2c1CCCC2 92777,C1(O)(C(CC)C(=O)N(CC(C)(C)CNC(=O)CCc2ccco2)C)CCCCC1 92778,C(CC(C)(C)C(=O)N(CCCNC(=O)C(C1CCCC1)N(C)C)CCO)OC 92779,c1(CC(=O)N(CCN(C(=O)Cn2cncn2)CC)CC)ncc(Cl)s1 92780,C(=O)(CC(N(C)C)NC(=O)C(C)(c1cccs1)NC(=O)CC(C)C)OCC 92781,C1(N(C(=O)Cc2nc(-c3ccco3)oc2C)CC)CCCN(C(=O)C(C)O)C1 92782,CC1(C)CC(O)C(O)CN(C(=O)Cn2cc(-c3cc(C(=O)O)ccc3F)nn2)C1 92783,CC1CCC(NC(C2CC23CCSCC3)=O)CN1C(=O)CCN1CCCCC1 92784,c1(C(N(C)CC2CCN(C(c3nc(COC)oc3)=O)C2)=O)cc(Cl)ncc1N 92785,c1(C(=O)NCC2(C)CCN(C(C(CC)NC(C)=O)=O)CC2)cc2c(s1)CCOC2 92786,C1(NC2CCN(c3nc(C)cc(OC)n3)CC2F)CCCC1S(C)(=O)=O 92787,c1(CCNC(N(CCCO)C)=O)csc2ccc(Br)cc12 92788,N1(C(c2cc(OC)n(C)n2)=O)CCCC(CO)(CNC(C2COCCC2C)=O)C1 92789,C1(CN(CC)CC)CCN(C(=O)CCCCC(=O)NC(C)C(=O)OC)CCC1(F)F 92790,C1(C(=O)N(C)CCc2cnc[nH]2)(COC)C=CCN1C(=O)C(F)OC(F)(F)F 92791,c1(NCCC(C)(C)NC(c2cc(CCC)[nH]n2)=O)ncnc(Cl)c1Br 92792,CONc1cccc(C(=O)NCCOCCNC(c2c(S(N)(=O)=O)cnn2C)=O)n1 92793,C=C(C)C1OCCCC1C(N1CCCCC1CCCNC(=O)CC1CC1)=O 92794,C1(CNC(C2CC3CC3C2)=O)CC2(CCOCC2)CN1C(C1(O)CCSCC1)=O 92795,Cc1nc2n(n1)CC(C(=O)N(C)CC1CCCN1C(=O)CCCC(C)C)CC2 92796,Cc1cnc(O)c(CNc2ccc(OCc3cccc(F)c3)cc2)c1 92797,C1(O)(CNC(CN(C)C)=O)CCCN(C(=O)C(CC(F)F)C(=O)OC(C)(C)C)C1 92798,c1(C(N2C(C)CC(NC(C=C(C)C)=O)C2)=O)ncnc2c1c(Br)cn2C 92799,N1(C(c2cc(NC)nc(Cl)c2)=O)CC2CCCN(C(c3cnsn3)=O)C2C1 92800,C1(CNC(C2C(c3n(C)cnn3)C2)=O)CN(C(=O)CCNC=O)CCC1C(F)(F)F 92801,N1(C(C2N(C(CNC(=O)OCC)=O)C(C(C)C)CC2)=O)CC2CCCC(O)C2C1 92802,C1(NC(C2OCCN(CC)C2)=O)CCCN(C(C2CN3CCC2CC3)=O)CC1 92803,N1(C(CN(CCC)C)=O)CC(OC)CC1C(=O)NCC(C)N(CC)CC 92804,C1(NC(C2(CO)CC2)=O)CCCCC12CCN(C(=O)C=C1CCCC1)CC2 92805,C(c1cc(F)c(O)c(F)c1)=CC(=O)NC(CC)CNC(C1C2CN(CC)CC12)=O 92806,C1(OC)CCCC(C(=O)NCC(C)(C)CN(C(=O)CC2CC=CCC2)C)C1 92807,N1(CC(C)(C)NC(C23CCC(CC2)O3)=O)CCN(C(c2cc(C(N)=O)c[nH]2)=O)CC1 92808,c1(C(=O)NCC#CCNC(c2cc(OC)no2)=O)cc(Br)c(C)nc1O 92809,c1(C(=O)NCC(C)(CO)NC(c2c(C(C)C)cco2)=O)cc2oc(Br)cc2[nH]1 92810,c1(C(=O)NCC(CNC(C2(C(F)F)CC(=C)C2)=O)(C)O)cncnc1C 92811,N1(C(c2c(C)nn[nH]2)=O)CCN(C(C2CC3CCCCC23)=O)CC12CCC2 92812,C=C1CCN(C(c2cc(CO)n(C)n2)=O)C(C(N2CCC=C(Cl)C2)=O)C1 92813,Cc1cc(=NCCC=CBr)[nH]c(N2CCC(Cc3ccnn3C)C2)n1 92814,C1(NC(CC2CC(=O)NC2)=O)CN(C(=O)CC2C=CCCC2)C2(CCCCC2)C1 92815,C(=O)(C(O)C(C)(C)C)NC(CSCC)C(N1CCN(CC)C(C)C1)=O 92816,N1(C(C2CCN(C)C(=O)C2)=O)CCC2(CCCN2C(c2ccc(F)c(Cl)n2)=O)C1 92817,C1(CCCNC(=O)CCc2cn[nH]c2)CCN(C(C23CCCC2CC3)=O)CC1 92818,C12CCCC1N=C1C=CNC=C1S(=O)(=O)NC2.CC(CS(C)(=O)=O)N(C)C 92819,c1(CNC(C(CO)NC(CCCSC)=O)=O)ccc(C)nc1O 92820,C1(CC(=O)NCCNC(C(C)C2CCCC2)=O)CN(C(=O)C(CO)N(C)C)CCO1 92821,CC(CC(N)=O)C(=O)N1CCCCC(NC)C1.c1(C=O)cc(C2CC2)ccc1F 92822,C(=O)(CCCC(=O)N(C)C)NCC(CNC(C1CC(C(=O)OC)C1)=O)(C)O 92823,c1(NC(C(N2C(C(CC)O)CCC2)=O)=O)cccc(-c2ccccc2O)c1 92824,C1(CN(C)C(C2CSCC(=O)N2)=O)CCCN(C(C2CC(CC3CC3)C2)=O)C1 92825,c1(OC)cc(N2CCCC(C(C)NC(=O)C(O)Cc3cnc[nH]3)C2)nc(C)n1 92826,CC(CCO)N=c1[nH]c2c(c(=NCCC3(C)CC3)[nH]1)SCC2 92827,C1(C(N(CCCCNC(C2CN3CCC2CC3)=O)C)=O)CN(CP(C)(C)=O)C1 92828,c1(C(=O)OC)ccc(CCC(=O)NCCNC(=O)CSC(C)=O)cc1 92829,c1(OC)ncc(C=CC(N2CC3C(C(=O)NC4(C)CCCS4(=O)=O)C3C2)=O)cn1 92830,Cc1cccc(C(CNC(C2C3CCCC23)=O)N(C)Cc2ccccc2)c1 92831,C(=O)(C(C)CN(C(=O)CCc1ccn(C)c1)C)NCC(=O)NC(C)C 92832,C1(CC(=O)N)(C(=O)O)CCCCC1.c1(CC(C)NC=O)cn(CC2CCCCC2)nn1 92833,C1(c2ccccc2)(C(=O)NC2(CNC(C3CC4CCCC34)=O)CC2)CC2(CC2)C1 92834,n1(CCC(=O)NC2CN(C(=O)C=CCO)CCC2C(F)(F)F)cnc([N+](=O)[O-])c1 92835,C1(NC(C2OCCN(C)C2=O)=O)COC2(C1)CN(C(=O)CN1CCC(O)CC1)C2 92836,C12(C(=O)NCC(=C)CCNC(=O)C3CC3)CCC(CC1)C(C)O2 92837,C1(NC2C(NC(COc3c(C)cccc3)=O)CCCC2)CCC(C2CCCO2)O1 92838,N1(C(C(C)OCCOCC)=O)CC(NC(C2CC2C(C)(C)C)=O)C(F)C1 92839,C1(OC)COC(C(=O)OC(C)(C(C)C)c2nnnn2C2CCCC2)C1 92840,C1(CC(F)=CC(=O)NCCNC(CCCC(C)(F)F)=O)CCS(=O)(=O)C12CCC2 92841,c1(C(N2CC(CNC(c3cc(C(=O)OC)[nH]n3)=O)C2)=O)cc(OC)ccn1 92842,C1(C(=O)OC)CCCCN1C(=O)NCc1c(CNc2cc(Cl)ccn2)cccc1 92843,CN(C)C1CCc2ccc(NC(c3ccc(F)cc3)c3nnnn3CCCF)cc21 92844,c1(CC)ccc(C(N2CCC(CN(C(c3cnc[nH]3)=O)CC)C2)=O)nc1 92845,C1(O)(CCNC(c2ncoc2Br)=O)CN(C(C2(c3ccno3)CCC2)=O)C1 92846,c1(C(n2nc(-c3cnn(C)c3)nc2CC(C)CC)C=C)ccc(Cl)cc1 92847,C1(C(N(CCC#C)C)=O)CC12CCN(C(c1cc(CC)sn1)=O)C2 92848,C(=O)(C1CCCc2nn(C)cc21)NC1CC(F)(CNC(c2c(C)cc(C)[nH]2)=O)C1 92849,C1(NC(CC)=O)CC(=O)N(C2CN(C(=O)CN3CCOC3=O)C2)C1 92850,C(=O)(C(C)(O)CCC)NCC(C)(C1CCC1)NC(c1c(CC)n(CC)nc1)=O 92851,Cc1nc(C)n(CCCC(=O)NC(C)CCCNC(=O)CN2CCCCCC2)n1 92852,c1(C(N2CCN(C(c3nnn4c3CSCC4)=O)CC2)=O)cccc2c1COC2 92853,C1(C(=O)NCC2(NC(C=CC3(C)COC3)=O)CCC2)CC2C(C1)C2(C)C 92854,Cc1cn2cc(CC(=O)NC3CCN(C(=O)Cc4cc[nH]c4)CC3F)nc2s1 92855,N1(C(c2c(-c3c(CC)n(C)nc3)ncs2)=O)CCN(C)C(=O)C1 92856,c1(C(N(CC)CC2CCCN2C(=O)C(C)SC(C)C)=O)cc2n(n1)CCC2 92857,Cc1cc(SCC(=O)NCC(O)CNC(c2ccc(CF)cc2)=O)cc(C)c1O 92858,c1(CNC(CC2(C)CCN2C(=O)CC2COCCOC2)=O)ccc2c(c1)CC2 92859,N1(C(CC2(COC)CC2)=O)CC2CCC1C1CN(C(C3CCC34CCC4)=O)CC21 92860,c1(CC)n[nH]c(CC)c1CC(=O)NC(C1CN(C(c2coc(O)n2)=O)CCO1)C 92861,c1(C(=O)NCCC2N(C(CC(C=C)C)=O)CCOC2)c[nH]c2c(F)cccc12 92862,c1(C(=O)NCC(CC=C)NC(C2C3CC4C(C3)C24)=O)ccccc1SCCO 92863,CC1COCC(CC(=O)NCC2(C(N3CC4CC4(CO)C3)=O)CCC2)O1 92864,CCCC(C(O)C(=O)NC(C)C(=O)NC1CC1)NC(c1c[nH]c(C#N)c1)=O 92865,N1(c2ccnc(CN(CCCCN(C)C)C)n2)CC(O)CC2(CCCC2)C1 92866,Cc1ccccc1OCCC(=O)NCC(C)(C1CC1)NC(C12CCN(CC1)C2)=O 92867,c1(OC)c(C(=O)N(CC(C)(C)NC(c2csc(C)c2C)=O)C)sc(Cl)c1Cl 92868,N1(C(CCCN(C(C)C)C)=O)C(C(=O)NC2(CC3CC3)CCC2)CCC12CC2 92869,c1(Nc2nc(SC)nc(C)c2)cc(C)cc(Br)c1C.C12(C)CN(C1)C2=O 92870,C1(C(C)NC(=O)CC2CC(F)C2)CCN(C(C2OCCOC2C(F)(F)F)=O)CC1 92871,CC1(C)CN(C(=O)CC2(C)CC(F)(F)C2)CC1CNC(C1CC2CC1C2)=O 92872,N1(C(N2CCC(OC)C2)=O)CCC2C1CCN2C(c1cccc(C2CC2)c1)=O 92873,c1(C(N2CC(CNC(C(C(=C)C)(C)O)=O)(OC)C2)=O)ccc(C#N)cc1O 92874,N1(C(CCCOC)=O)CC2CC1CN(C(c1nccc3ccsc13)=O)C2 92875,c1(C(N2CCC(C(C)NC(=O)Cc3cnn(C)c3)CC2)=O)cc2c[nH]nc2s1 92876,CCCCC(C(=O)NCC1CCC(C(=O)N(CC(C)(C)O)C)C1)C(C)C 92877,S(=O)(=O)(c1cccc(Cl)c1Br)N(C)CCNCC(F)F 92878,Cc1nn(C)c(C)c1CCC(=O)N(CC(O)CNC(=O)C(C)(C)NS(C)(=O)=O)C 92879,c1(OC)ccc(C(=O)NC(C2CN(C(=O)CC3CC4(CC4)C3)C2)C)c(Br)n1 92880,N1(C(=O)COC2CCCC2)CC2COCC(C1)N2C(=O)CC1CC1 92881,CCCCCCOCCC(=O)NCCC1(O)CN(C(c2n[nH]cc2OC)=O)C1 92882,c1(C(N(CCCNC(=O)CCC2CCCC2)C)=O)ccc2nc(S)oc2c1 92883,C1(NC(C=C(C)C)=O)CN(C(c2sc(-n3cccc3)nc2C)=O)CC1C 92884,Cc1cc(N2CCC(C)C(NC(c3ccc(C)s3)=O)C2)c(C#N)cn1 92885,C12CCC(CC1)C(=O)N2.Cc1ccsc1C(=O)NCCCC(C)O 92886,C1(C(=O)NCC(CNC(C=Cc2c(C)ccs2)=O)C)CCc2nnc(O)cc2C1 92887,C=C1c2ccccc2C(=O)N1CC(=O)NC1CC(C)N(C(c2cc[nH]c2)=O)C1 92888,Cc1cc2[nH]c(C(=O)NCC3CCN(C(=O)C(O)CC(N)=O)C34CCC4)cc2s1 92889,C1(C)(CNC(C=C(CC)C)=O)CCCN1C(=O)CC1CCOC1=O 92890,C(=O)(C1=COCCC1)NC1CC(N(C)C(c2ncoc2C2CCCO2)=O)C1 92891,C1(O)(C(=O)NCC2(NC(C3CC(=C)C3)=O)CC2)CC2CCC1C2 92892,C(=O)(C1=CC(N)C1)C(=O)CCC1CCC(C)O1.C1(CCN)(OCC)CCC1 92893,C=CCC(CNC(=O)CCn1cc(C)cn1)NC(c1n[nH]cc1Br)=O 92894,CC(C)(C)S(=O)(=O)CC(=O)N1CCCC1C(C)(C)NC(c1cc(O)nc(O)c1)=O 92895,C(=O)(C(O)CC(F)(F)F)NC1CC(F)(CNC(C(c2c(OC)cccc2)C)=O)C1 92896,N1(C(C(C)=CC)=O)CC(CNC(c2nc(C)nn2C)=O)OC(C(F)(F)F)C1 92897,C1(=O)C(C)(C=C)CCN1.C1(=O)C#CCN1.C=CCC1CC1 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92967,C1(C)(CNC(COCC=C)=O)CCN(C(c2ccnc(C(F)(F)F)c2F)=O)CC1 92968,c1(C(C)(C)C)cccc(C(=O)N(CCCNC(C2CCCN2C(N)=O)=O)C)c1N 92969,S(=O)(=O)(c1ccc(NC2CCCOC2)c(C#N)c1)NCC1(C)CC1(Cl)Cl 92970,N1(C(CCCC)=O)CC(NC(C2CCN(C)C2C)=O)C2(CC2)C1 92971,c1(CCC(=O)NC(c2ccc(C)cc2)CNC(=O)C(C)C(F)F)c(Cl)cncc1Cl 92972,c1(C(N2CC(COC)(NC(=O)C(F)F)C2)=O)cc(C)c(C)c(Br)c1 92973,c1(NC(C2C(NC(C(CCC)CCC)=O)C2)=O)cc(F)cc2cc[nH]c12 92974,CCCC(CCC)CC(=O)NCC1CCCN(C(C23CC2COC32CCC2)=O)C1 92975,C1(C)(CC)CC(NC(c2ccc(OC)s2)=O)CN1C(C1CCSC(C)C1)=O 92976,C1(C(N2CCCC(CNC(C3CCC(F)CC3)=O)C2)=O)CC2(C1)CC1(CC1)C2 92977,CC(C(F)F)NC(=O)CCOCCN(C(=O)Cc1cncs1)C 92978,C1(NC(CC(=O)OC)=O)CC2CC(NC(=O)C(c3cnn(C)c3)C)C2C1 92979,Cc1cc(CNC(=O)C(=O)Nc2ccn(CCC(F)(F)F)n2)cnc1F 92980,C(=O)(C1CCCn2c(Br)cnc21)N1C(CNC(c2cnn[nH]2)=O)C2CCC1C2 92981,C(=O)(Nn1cnn(CC)c1=O)C1CN(C(C(C#C)(C)C)=O)CC1(F)F 92982,c1(OC)cccc(CN2CCCC(NC(C3CCC=CO3)=O)C2)c1O 92983,C1(C(=O)NC(C)CC(C)NC(=O)COCCN(C)C)CCOC2(CCCCC2)C1 92984,c1(NC(=O)NC(C(c2ccc(OC)cc2)O)C)cc(OC)cc2ccoc12 92985,CC1c2cc(Br)ccc2OC1CNC(=O)N(CC1CC1)CC1CC1 92986,C(=O)(CCN=C1NS(=O)(=O)c2ccccc21)N1CCC(C)(NC(c2cnc[nH]2)=O)C1 92987,C1(F)(CNC(c2ccc(-c3ccc(F)cc3)s2)=O)CCC(CO)CC1 92988,CCC(C)CC(C(=O)NCC(C)(C)OC)NC(C1(OCC(C)C)CCC1)=O 92989,CN1CCCC(C(N2CC(O)(C(=O)NCCOc3cccc(Br)c3)C2)=O)C1 92990,c1(C(=O)NC(C2CCCN(C(=O)Cc3nc(=N)[nH][nH]3)C2)C)[nH]nc([N+](=O)[O-])c1Cl 92991,N1(C(c2sc(Br)cc2C)C(=O)Nc2cccc(OC)c2)CC(F)(F)CCC1C 92992,c1(C(N2CCCN(C(C3C(C)(C)C3(C)C)=O)CC2)=O)n[nH]c2nccc(Cl)c12 92993,Cc1ncc(CCC(=O)NC(CNC(C2CC2c2ccccc2)=O)C2CCC2)o1 92994,N1(C(C(C=C)c2ccccc2)=O)CCN(C)C(C(=O)NCC2CCNC(=O)C2)C1 92995,C(=O)(C(C)(C)CCCC(=O)NC(C)(C)CNC(c1cncc2sccc12)=O)OC 92996,N1(C(CC2(OC)CC2)=O)CC2CN(C(=O)C(C(C)O)CNC(C)=O)CC2C1 92997,c1(C(=O)NC(C(C)NC(C2=NOC(C)C2)=O)C)cccc2sccc12 92998,c1(N2C(C)CC(CNC(=O)CSCC(F)(F)F)C2)ncnc2sc(Cl)cc12 92999,Cc1c(C(=O)N(C)CC2(NC(=O)Cc3cnccc3Cl)CC2)cccc1CO 93000,N1(C(C(CC)(C)O)=O)CC(NC(C2CC3(CSC3)C2)=O)CC2(CCC2)C1 93001,N1(C(c2ccc(C#C)cc2C(F)(F)F)=O)CCN(NC(=O)C2CC(O)C2)CC1 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93125,CC(C)CC(C(=O)N1CC2CC1(CNC(=O)CSC(F)(F)F)C2)C(C)C 93126,C#Cc1cn(C)nc1C(N1CCC(CC(=O)NCc2ncc(C)cc2C)C1)=O 93127,C1(NC(c2ccnc(F)c2)=O)CCCN(C(C2CCN(C(=O)C3CC3)CC2)=O)C1 93128,c1(OCC)cc(N)ccc1C(N1CC(Cc2ccc(F)cc2)C(C(F)(F)F)C1)=O 93129,C(=O)(CCCN(C)N=O)N1CC(C)C(C)(CNC(C2(C)CSC2)=O)C1 93130,c1(NC(C2CCCN2C(=O)Nc2cccc(Cl)c2)=O)ccc(=O)n(CCO)c1 93131,C1(NC(c2ccc(COC)o2)=O)CCN(C(c2oc(Br)nc2C)=O)CC1C 93132,c1(C(C(=O)NCC(C)N(C(C=CCCC)=O)OCC=C)OC(C)=O)ccccc1 93133,C1(CC=C)(NC(=O)C(O)CSC)CCN(C(=O)Cc2ccc(Cl)cc2)C1 93134,CC(C)(O)CCC(=O)NC1CN(C(=O)CC(=O)NCC(F)(F)F)CC12CC2 93135,c1(OC)ccc(CNC(c2csc(C)c2C)c2nnnn2C2(C)CC2)c(C(N)=O)n1 93136,C12(C(C)(C)C)CC(C(=O)NC3(CO)CN(C(C4COC(=O)O4)=O)C3)(C1)C2 93137,c1(NC(C(=O)N(CCCCN(c2cnn(C)c2)C)C)=O)ccc(C2CC2)cc1F 93138,C(=O)(C1=CCSC1)NC(CC)CNC(=O)C(c1ccccc1Br)F 93139,Cc1c(C(=O)NCCNC(c2ccc3nn[nH]c3n2)=O)oc2ccccc2c1=O 93140,C1(NC(COCCCCCC)=O)CCCCC1NC(C1(OCC)CCCCC1)=O 93141,O=S(=O)(c1ccc(Br)cc1N1CCC=C(F)C1)NCCc1cccs1 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93388,c1(C(N2CC(C)N(C(=O)CC3CCCCN3C)CC2)=O)cnc2ccnn2c1O 93389,Cn1nc(C(N2CC(O)CC2C(N2CC(O)(c3nn[nH]n3)C2)=O)=O)cc1C#N 93390,c1(C(N2CC(C(C)NC(c3coc(C(F)F)c3)=O)C2)=O)cccc2ccoc12 93391,C1(CCNC(C(CO)N(C)C)=O)CCN(C(C2(CO)CCCO2)=O)CC1 93392,N1(C(CCOC2CCN(C)CC2)=O)CCNCc2cc(F)c(F)cc21 93393,C1(NC(c2cc(C)sn2)=O)CCN(C(=O)Cc2cscn2)CC1(C)C 93394,CCC(CN(C)C)S(=O)(=O)Nc1nc(-c2ccccc2)no1 93395,C1(C(N(CC(CN(C(=O)Cc2cc[nH]n2)C)O)C)=O)CCc2ccc(F)cc2C1 93396,Cc1cc(C(=O)NC(CO)C(C)NC(=O)CC(C)C2CCCCC2)nnc1O 93397,c1(OC)cc(C#N)ccc1NC(=O)Nc1cc(Sc2ccccc2C)cs1 93398,c1(C(=O)NCCNC(c2c(CC)nc[nH]2)=O)cc(C)nn1C1CCC1 93399,C1(NC(c2cc(CC)oc2C)=O)CC12CCN(C(=O)Cc1coc(C)n1)C2 93400,N1(c2nc(C)nc(C#N)c2)CCCC(C2(NC(C3C4C5CCC(C5)C34)=O)CC2)C1 93401,C1(C(N(CC(Cc2ccccc2)NC(c2cnns2)=O)C)=O)CCCC(=O)O1 93402,C=CCC(C(=O)N1CCCC(C(N)=O)C1)NC(=O)Cc1ccsc1Cl 93403,c1(C(N2CC(O)(C(CNC(C3CCCC(C)C3)=O)(C)C)C2)=O)cc2scc(Cl)c2[nH]1 93404,C(N=c1[nH]cnc2cccc(Br)c12)C1CCCN(C(C2(CC=C)CCC2)=O)C1 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93459,NS(=O)(=O)c1n[nH]cc1C(N1CCN(C(=O)C2=NOCC2)C(CC(F)(F)F)C1)=O 93460,N1(C(c2c(CC)non2)=O)CC2=C(C1)CN(C(c1ccn(C(C)C)n1)=O)C2 93461,N1(C(CSCC=C)=O)CCCN(C(c2c(C(F)(F)F)cccc2F)=O)CC1C 93462,CC1=C(C(=O)N2CCCC(CNC(=O)C(c3cn(C)nc3C)(F)F)C2)CCO1 93463,C(CSC)(C(=O)N(CCC(=O)NCC1CC1(Cl)Cl)C(C)C)OC 93464,C1(C(=O)NCC2CC(CNC(=O)OC(C)(C)C)OC2)CC2CC(C1)C2 93465,CC1CC(C(=O)NC2(CC(=O)NC3CC4(CC4)C3)CCC2)CCS1 93466,CC(C)CC(C(=O)N(C(C)CCNC(=O)CCCN=[N+]=[N-])C)C(C)C 93467,CC1=CCC(C(=O)N(CCC(=O)NC2C=C(C)CCC2)C(C)C)CC1 93468,c1(CCNC(=O)NCc2ccc(-c3ccnc(F)c3)cc2)cc(F)c(Br)cc1Cl 93469,C1(C(=O)NC(C(C)C)CNC(=O)C(C)CN2CCCCC2)CCCCC1C(N)=O 93470,CC1CN(C)CC1C(=O)N(C)CC=CCC(=O)NC1CC1n1cc(CO)nn1 93471,c1(CN(C)CC2NCC(OC)C2)cc([N+](=O)[O-])ccc1Cl 93472,C12(COC)CC(NC(c3cc(Cl)n(C)n3)=O)(CN1C(C1CSC1)=O)C2 93473,C=CC(CCC)CC(=O)NCCOC1CCN(C(c2coc(C(C)OC)n2)=O)C1 93474,CC(C)C(F)(CNC(=O)CCCC1CC1C)C(=O)N(C(CO)C(C)C)C 93475,N1(C(C(C(C)C)C)=O)CCCN(C(c2cc(-c3ccccc3F)[nH]n2)=O)CC1C 93476,Cc1ccc(C(C)C(=O)NCCCN(C(=O)CN2CCC2C)C(C)C)s1 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93615,C(=O)(C(CCC(C)(C)C)OC(c1c(C)cccc1O)=O)OC 93616,N1(C(c2ccc(COC)[nH]2)=O)CC(C)CCC1CNC(c1nccc(C)n1)=O 93617,C1(CNC(c2ccc(C(C)(C)C)s2)=O)CN(C(=O)C2CC2)CC1C(F)(F)F 93618,C1(NC(c2cc(CC)on2)=O)CC(CNC(c2cc(C)c(C)o2)=O)C1(C)C 93619,C(=O)(C(O)CCCNC(C1CC(F)C1)=O)N1CC(CC(C#C)C)C1 93620,N12CCCC3(CC3C1)NC(=O)C=CC2=O.c1(SCC=CCC)ccncc1 93621,c1(SC(C)C(=O)N(C)CCN(C)C(C2(C)CCCC2C)=O)ccc(Br)cc1 93622,C12CCN(CC1)C(=O)N2.c1(C(=O)OC)ccc(CNC(=O)COC2CC2)s1 93623,CCCC(O)CN(C)C(c1cn(CCNC(=O)Cc2cc[nH]c2)nn1)=O 93624,C1(NC(C2(C)CC2)=O)CCCCC1NC(=O)CSc1ccccc1Cl 93625,C1(C(=O)NCCC(C)NC(C(C)Cc2cccc(F)c2)=O)CC(C(C)(C)C)=NO1 93626,c1(NC(c2c(CNC(C(C3CCC3)OCC)=O)ocn2)=O)ccc(O)c(C)c1 93627,N1(C(C2(CC(C)C)CCC2)=O)CCOC(C)(CNC(c2cncc(Cl)c2C)=O)C1 93628,CN1CCC(N(C)C(c2c[nH]nc2CNC(=O)CCC2OCCO2)=O)C1 93629,CC1(C)CC(NC(=O)C(O)C2CCC2)CCN(c2nc(Cl)nc(C3CC3)c2F)C1 93630,c1(CC)cc(N)ccc1C(=O)NCC1CCCCN1C(=O)CCc1cnc(O)[nH]1 93631,c1(C(N(C2CCCN(C(=O)CSC(F)F)C2)C)=O)cc2cccc(F)c2cn1 93632,c1(-n2ncc(C(=O)NCC3(c4cccc(Br)c4F)CC3)c2)ccc([N+](=O)[O-])cc1 93633,c1(C(=O)OC)cnc(C)[nH]c1=NCCC(C)NC(=O)C1CCCc2nccn21 93634,CCCC(CNC(=O)C(=O)C(C)(C)C)C(=O)N1CC(N2CCCC2=O)C1 93635,C1(NC(C2N(C(c3ccc(CSC)o3)=O)CCOC2)=O)CC2(C1)CN(C(=O)CO)C2 93636,C1(NC(C2CCS(=O)CC2)=O)CCCN(C(=O)CCC2CCCCC2)CC1 93637,N1(C(c2c(CC)cccc2)=O)CC(CN(C)C(C23C4C5C6C4C2C6C35)=O)CC(C)C1 93638,Cc1cc(F)c(C(N2CCCC2CN(C)C(C2CC=CC2)=O)=O)cc1F 93639,n1(CC)cc(CCNC(C2CN(C(c3ccc[nH]3)=O)CCO2)=O)c(C)n1 93640,c1(OCC)ccc2cc1OCc1c(cccc1)NC(=O)N2.C1(N(C)C)CC1 93641,c1(OC)ccc(C(N2CC3CCC2C3NC(=O)C#CC(=O)N(C)C)=O)c(N)c1F 93642,N1(Cc2cc(COC)no2)CCC(=O)N(CCC(C(F)(F)F)OC)C1=O 93643,C1(NC(=O)C=Cc2cscn2)CC2CCC1(CNC(c1cc(Cl)c[nH]1)=O)C2 93644,c1(C(=O)NC(CNC(C2(COC)CCCO2)=O)C)ccc(Cl)c(N)c1 93645,N1(C(c2nc(CC)oc2)=O)C2CCC1C(NC(c1cnc(C(F)(F)F)nc1)=O)C2 93646,C(CCSC)(C(N)=O)NC(C1C(NC(C(CC)N(C)C)=O)COC1)=O 93647,c1(C(N2CCC(NC(CCCNC(COC)=O)=O)CC2)=O)ncc(F)c(OC)n1 93648,Cc1oc(C#N)cc1C(N1CCOCC1CC(=O)NC(c1cn[nH]c1)C)=O 93649,Cc1nc2ccc(C(N3CC(NC(=O)CNC(=O)C4CC4)CC3(C)C)=O)cc2[nH]1 93650,CC1CSc2ccc(Br)cc2C1NC(c1c(N)sc2ccccc12)=O 93651,c1(C(=O)NCC2(F)CC(C(N(C3(CCN=[N+]=[N-])CC3)C)=O)C2)cccc(F)c1F 93652,N(C(=NCC1CCOC1)NCC(=O)Nc1nc(C(C)NCCSC)cs1)OC 93653,CC(CCc1ccccc1)CC(=O)NCC1CCN(C(=O)CC2CCCO2)CC1 93654,n1(C(C)C)nccc1C(=O)NC(C1CCCN1C(C1CCC1C)=O)C 93655,C(=O)(CN=c1cc[nH]cc1)NCC1CCN(C(c2c(C(C)C)noc2)=O)C1(C)C 93656,c1(C(=O)NC(CNC(c2n(CCC)nc(C)c2)=O)C)cc2ccccc2oc1=O 93657,c1(C(N(C2CCC(NC(CCOCCOC)=O)C2)C)=O)csc2cccnc12 93658,C1(C(N2CC3C(CNC(c4c(C)ccs4)=O)(C3)C2)=O)C(O)C(=O)N(C)C1C 93659,N1(C(C2(CC3CC3)CCCN2)=O)CC2CC23CC13 93660,CC(C)(O)CC(=O)NCc1ccc(C(=O)NCc2ccc(Cl)nc2)nc1 93661,c1(CC)ccc(C(=O)NCC2CCCCCN2C(C2CCC(=O)C2)=O)cc1Cl 93662,Cc1snnc1C(N1CC(CO)(NC(c2cc(CO)on2)=O)C1)=O 93663,C(=O)(CS(=O)(=O)c1ccccc1Cl)NC(CNC(C1N2CC(C)N(CC2)C1)=O)C 93664,CCC(CCC(=O)NCCCC(C)NC(=O)C(C)(Cl)Cl)OC 93665,N1(CCC(=O)NCCCN(C(=O)CO)CC)c2ccccc2Sc2ccccc21 93666,Cc1ccc(O)cc1C(=O)NC1CC1CNC(c1c[nH]nc1-c1ccccc1)=O 93667,C1(C(=O)NC(CC(C)(C)NC(CNC(CC)=O)=O)C)CCc2ccc(F)cc2O1 93668,Nc1ccc(C(=O)OCCOC2CC(C(F)(F)F)C2)nc1F 93669,C1(CNc2nc(C)cc(CC)n2)CC2CCC1N(C(=O)C(C(C)C)NC(C)=O)C2 93670,N1(C(C2C(=C)CC2)=O)C2CCC1CC(CNC(c1c(C)ccnc1Cl)=O)C2 93671,c1(-c2c(C(=O)OCC)n(C)nc2)ccc2c(c1)COC21CN(CC2CCC2)C1 93672,N1(C(c2cc(C)cc(F)c2)=O)CC(NC(c2cccc(C)n2)=O)C2CCCC12 93673,C1(NC(C2CC(OC)C2)=O)C2CC(NC(=O)CC3NC(=O)NC3=O)CC12 93674,c1(C(=O)NC2(CNC(C(C(C)C)F)=O)CCCCC2)nccc2n[nH]cc12 93675,c1(CN(C(C)C)C(c2ccnn2CC(F)(F)F)=O)cn(C(C)(C)C2CC2)nn1 93676,N1(C(c2ccc(C)c(O)c2)=O)CC2CC1CCC2NC(c1n[nH]cc1C(C)C)=O 93677,CCC(C)(C)C(=O)N1CCCC(CCNC(=O)C(C)COc2ccccc2)C1 93678,c1(CNC(CC2CCCN(C(C3(CC)CC3)=O)C2)=O)cc2cnccc2[nH]1 93679,CN1CC(C)(C(=O)NCC2CC(NC(c3cccc(OC(F)F)n3)=O)C2)CC1=O 93680,C1(CNC(C=C2CCC(C)C2)=O)CN(C(=O)CC2(C)CC(F)(F)C2)CC1O 93681,c1(SC)cccc(C(=O)NC(C)(C)CCCNC(=O)Cn2cnnn2)n1 93682,c1(C(=O)NCC2N(C(c3c(CC)nccn3)=O)CC2)c(F)ccc(Cl)c1F 93683,c1(NC(CN2CC(C(C)(C)C)OCCC2)=O)ccc(F)c(N)c1 93684,C(=O)(C(CC)N(C)C)N(CCCC1CC(CC)C1)C.n1(CNC(C)=O)cc(C)nn1 93685,C1(C)(C(=O)NCCN2CC(OC)C2)CCN(C(=O)CN2CCOCC2=O)C1 93686,C1(=O)C(C)(O)C(C)N1.C1(C(=O)OC)CC12CC2C(=O)O 93687,C(=O)(C(C)(C)C(=O)N1CC(O)(C(F)C(=O)NCc2cccc(F)c2C)C1)NC 93688,C#Cc1cccc(CC(=O)NC2CCOCC2C(N2CCOCC2CO)=O)c1 93689,CC(C)C(C)C(CNC(=O)Cc1cnn(C)c1)NC(=O)C=Cc1cncn1C 93690,N1(C(CCc2cccc(C)c2)=O)CCN(C(=O)COC2CC=CC2)C(C(F)F)C1 93691,N1(C(CC(C)CF)=O)CC2CCN(C(C3C4CC5CC(C4)CC3C5)=O)C(C2)C1 93692,C(CC(=O)NCC(C)CN(C(=O)CCSC(F)(F)F)C)NC(COC)=O.C(C)=O 93693,c1(-c2scc(CC(=O)NCC(C3CCCCC3)NC(C)=O)n2)cccc(Cl)c1 93694,c1(C(=O)NC(CCCNC(C(CC)C(C)O)=O)C)ncn2ccccc12 93695,C1(F)(C(=O)NCC(C)(C)O)CCOC1.c1(CCOCC(=O)NCCS)ccccc1 93696,Cc1cncnc1C(=O)NC(CCC1CC1)C(=O)NCC(F)Br 93697,C1(N(C(C(N2CCNC2=O)C)=O)C)CN(C(=O)CCC(C)(C)N(C)C)CC1(C)C 93698,C1(CNC(C(c2ccccc2)C)=O)CN(C(=O)CC2COC(=O)C2)CCO1 93699,CC(CC(=O)NC(CNC(C1CC1F)=O)CO)n1ccnc1 93700,C=CCC(C(=O)N1CCC(CN(C(=O)C(CC)NC(N)=O)C)CC1)C(C)C 93701,C1(CN(C)C)CCCN(C(=O)CN(C)C(=O)OC2CC(C)(C)C2)CC1 93702,C1(C(=O)NCc2onc(N(C)C)n2)CC(=O)CN1C(=O)C=Cc1cncs1 93703,C1(OC)CC(C(N2CC=CC2CF)=O)N(C(c2cccc(N3CCCC3)n2)=O)C1 93704,C1(O)(C(N2CC3(C(=O)OCC)C(C2)CCO3)=O)CCc2ccccc2C1 93705,N1(C(c2cc(C(C)C)nc(O)c2)=O)CC2CCC1CN2C(=O)C=CC1CCOC1 93706,C1(NC(=O)Cc2ccc(F)c(F)c2)CCN(CC2CC(=C3CC3)C2)CC1O 93707,C1(NC(CC2CC(=O)OC2)=O)CCOCC1C(N1CC=CC1)=O 93708,Cc1ccccc1NC(C1CCCC(NC(=O)Cc2c(C)n[nH]c2C)C1)=O 93709,c1(Oc2ccc(N(C(CC)=O)C)cc2)ccc(NC(=O)NC2CC2)nn1 93710,Cc1cccc(-n2cc(CO)nn2)c1C.C1(=O)C(C(C)C)CNC2CCC(C2)N1 93711,C1(CC)CN(C(=O)C=C2CCCC2)CCN1C(=O)Cc1ccnc(F)c1F 93712,C(C(CC(C)C)C(=O)N1CCC1CNC(c1cc(Cl)cc(Cl)c1OC)=O)OC 93713,C1(NC(c2cnsn2)=O)CC2CC(NC(c3ccn(CCF)n3)=O)C2C1 93714,N(C1CCc2sc(C(=O)OC)cc21)CC1(CS(C)(=O)=O)CCC1 93715,C1(CNC(c2[nH]cc(C(C)(C)C)c2)=O)CC2CCC1N2C(C1CC2(C1)CC2F)=O 93716,CCC(C(=O)N1CCC1CNC(c1cnn(CCF)c1)=O)OC 93717,c1(C(=O)NCC2C=CC(NC(=O)CCSC3CC3)C2)sc([N+](=O)[O-])cc1Cl 93718,N1(C(CCCCCCC)=O)CCC2(CC1)CC(C(=O)N(C)CC1CC1)CO2 93719,CC1CN(C(=O)C(=O)N(C)C)CCCN1C(=O)CCC(=O)c1cccs1 93720,N1(C(c2c(C(F)(F)F)ccc(OC)c2)=O)CCC(CO)CC(N)C1 93721,c1(C(=O)NC2CC(CNC(c3cnc(OC)c(C)n3)=O)C2)c[nH]nc1S(N)(=O)=O 93722,O=C1NCc2cc(NC(C3CN(C(c4cccc(F)c4OC4CC4)=O)C3)=O)ccc21 93723,CC1(C)OC2CCC(N(C)CC3CCO3)C2O1 93724,N1(C(c2c(OC)cc(C)s2)=O)CCCOC(CNC(C2CCN(C)C2)=O)C1 93725,C1(CNC(=O)CN2CC3CCC2C3)(NC(c2cc(Cl)c(Cl)[nH]2)=O)CC2CCC1C2 93726,C(=O)(C(CC=C)C(C)C)NC(CC#C)C(=O)NCc1ccc[n+]([O-])c1 93727,C1(NC(C2CC(=C)C2)=O)CCC2CCN(C(c3ccc(C4CC4)c(N)c3)=O)C1C2 93728,c1(C(=O)NCCN(C(=O)CC(C)P(C)(C)=O)CCOC)cc(C)c(C)c2ncsc12 93729,N1(C(C(CCC)C#N)=O)CCC(C)(C)CC1C(=O)NC(c1ncc(C)cn1)C 93730,N1(C(c2c(CC)ccs2)=O)CCC2CN(C(c3nnn4ccccc34)=O)CCC12 93731,C1(COC)CN(C(c2ccsc2S(C)(=O)=O)=O)CCN1C(=O)C#CC1(C)CC1 93732,C1(C(N2CC(NC(c3c(OCC)ncnc3OC)=O)C2)=O)CCN2CCCC2C1 93733,CC1CN(C(c2ccnc(C(F)(F)F)c2)=O)CC1NC(c1cc(Cl)c(Br)s1)=O 93734,C1(CC)CCN(C(=O)C(COC)NC(=O)CC2CC3(C2)CN3C)O1 93735,N1(C(CN(C(C(C)C)=O)C)=O)CCOC(CNC(=O)CCC2CCCCN2C)C1 93736,N1(C(CC2CC(OCC)C2)=O)CC2OCC(NCc3ccc(C)cn3)C2C1 93737,C1(NC(c2cc(C)on2)=O)CN(C(=O)CC(C2CC2)C2CC2)CC1C(F)F 93738,C(C(=O)NC1CCCCC1NC(=O)CCOC1CCOC1)(C(C)C)OCC 93739,C1(CNC(CC(c2ccccn2)N(C)C)=O)C(C(F)(F)F)C2CCC1N2 93740,C(=O)(C(C)CC(F)(F)F)NC1COCCN(C(CCCCOC)=O)C1 93741,N1(C(C(C)C(C)(C)C)=O)CC(NC(c2nccc(Cl)c2O)=O)CC12CCCCC2 93742,C12(CC)CCC(C(N(C(C3CCc4nncn4C3)=O)C3CC3)=O)(CC1)CC2 93743,Cc1c(NS(=O)(=O)Cc2cccc(F)c2)ncnc1N1CCC(C)(C(C)C)CC1 93744,C(=O)(CCCCC(C)=O)N1CCC(C(N2CCC(F)(CO)CC2)=O)(CC)C1 93745,c1(C(N2C(C)CC(CNC(C(C=CC)O)=O)C2)=O)cc(Cl)ncc1F 93746,c1(C(=O)CSC2CCOC2=O)cc(N2CCCC2=O)ccc1O 93747,c1(OC)c(F)ccc(NC(=O)Nc2c(C)cncc2C)c1F 93748,c1(C(N(C)CC2CN(C(c3c(C(=O)OC)c(C)on3)=O)C2)=O)cc2n(n1)CCO2 93749,C1(C(=O)NCCNC(CC2(OC)CCC2)=O)OCCC1C(C)C 93750,Cn1cc([N+](=O)[O-])c(C(=O)NCC(C2CC2)NC(=O)Cn2ncc(C#N)c2N)n1 93751,C1(C#N)(C(N2CC(CC=C)(C(=O)NC(CO)C(=O)NC)C2)=O)CCCCC1 93752,C1(C(C)C)(C(=O)NCCCCC2CN(C(=O)CCF)C2)CCC1 93753,CNS(=O)(=O)N1CCC(C(N2CCCC2CNC(=O)CC(C)COC)=O)CC1 93754,c1(CCC(N2C(C3(N(C)C(c4cnn(C)n4)=O)CC3)CCC2)=O)cc(F)cc(F)c1 93755,Cc1[nH]c(C#N)cc1C(=O)NC1CN(C(=O)C2=CC(C)(C)C2)CC1CO 93756,CCCCC(C(=O)Nc1ccc(Br)cc1F)NC(=O)NCCCC(=O)OC 93757,c1(OC(C)C(=O)NCCC(C)(C)NC(c2coc(Cl)c2)=O)ccccc1Cl 93758,C1(NC(c2cc(CNC(=O)Cn3ccnc3)no2)=O)CCCC(O)C1 93759,c1(OC)ccn2cc(C(=O)NC3(C)CN(C(=O)C4=CCCCC4)C3)nc2c1 93760,n1(CC)cccc1C(N1CCC(C(C)C(=O)N(C)CCN2CCCCC2)C1)=O 93761,C12(C(=O)NC3(CSC)CC3)C(NC(c3cnc(S)nc3)=O)C3CC1C2C3 93762,C1(CC(=O)NCC(CNC(C2CCN(CC)C2)=O)CO)COC(C)(C)CO1 93763,C(c1cccc(O)c1)=CC(=O)NCCC1CCCN(C(c2ccnc(C)n2)=O)C1 93764,c1(N2C(=O)c3ccc(nc3)C2)ccc(Br)cc1C.C1(CC(=O)N)C(=O)ON=C1C 93765,C1(CNC(CN2CC(CC)C2)=O)(CNC(=O)CSC(C)C)CCCC1 93766,C1(NC(=O)CCSC2CCCO2)CCCCN(C(=O)CSc2cn[nH]c2)C1 93767,c1(C(=O)NCC=Cc2n(C)ncc2)n[nH]c2c1CN(C(=O)Cc1ccsc1)C2 93768,N1(C(C(C)(C2CC2)OC)=O)CCC2(CCCCC2NC(=O)C(C)C2CC2)C1 93769,C12(C(=O)NC3CC(CNC(C(CC=C)(C)C)=O)C3)CCCCC1C2(F)F 93770,c1(N2C(C3CN(C(CCN(c4ccnc(Br)n4)C)=O)C3)CCC2)ccc(Cl)cc1 93771,C(c1ccc(Br)o1)=CC(=O)NCC(C)(C)NC(c1ccc(=N)[nH]n1)=O 93772,N1(C(Cc2cc(CC)no2)=O)CCN(C(=O)C(c2ccccc2)C)C2CCCC12 93773,C(C)(C)(C#CC(=O)NCC1(O)CC2C=CC1C2)NC(CNC(=O)OCC)=O 93774,C1(CC)CN(C(=O)C=CC(C)C)CCC1NC(=O)C(c1cccc(C)c1)(F)F 93775,CCC(C(=O)NC1CC(CO)N(C(C2CNC(=O)N2C)=O)C1)C(C)C 93776,N#CC1(Cc2cnn(Cc3ccc(Cl)cc3)c2)CCCC2(CCCOC2)O1 93777,c1(C(=O)Nc2ccc(NC(C3CC(=O)NCC3)=O)nc2)cn2ccccc2n1 93778,CC(C)CC(CNC(c1cnn(C(C)C)c1)=O)C(=O)NC1CCSCC1 93779,N1(C(c2c(Br)ccc(OC)c2)C(=O)NCCC2CC2)C2CCC1CN(C)C2 93780,Cc1cccc(CC(=O)NCC(CC2CC2)C(=O)NCP(C)(C)=O)c1 93781,C1(OC)CC(CNC(c2cncc(C(C)C)c2)=O)N(C(=O)COCC(F)(F)F)C1 93782,Cc1cc(Cl)ccc1OCC(=O)NCCC(C)N(C)C(C1CC12CC2)=O 93783,c1(C(=O)NCC2(C)CCC(NC(C=CC(C)C)=O)C2)cccc2c1nc(O)n2C 93784,C1(C(N2CC(C)(CCC(N3CCOCC(O)C3)=O)C2)=O)CC(=O)CC12CCC2 93785,c1(C(C(=O)NC(c2c(Cl)cccc2Cl)CC(=O)OC)C)nc(F)ccc1Cl 93786,CC1C(C)N(C(C2CCCS2)=O)CCN1C(c1cc(C2CCOCC2)[nH]n1)=O 93787,c1(C(C(=O)NC)N(CC=C)C)cn(C)nc1OC(F)F.C1(O)CCC1 93788,C(=O)(C(CCC1CC1)NC(=O)CC1CCCN1C)N(C)Cc1cscn1 93789,CC(C(=O)N1CCC(CC2CCC2)C1)S(C)(=O)=O 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94033,C(=O)(C(C)CCCOC)NC(c1nnnn1C)CCC 94034,c1(C(=O)NCC(CC)(C)NC(c2ccc(CO)o2)=O)c(C)cc(C#N)cc1C 94035,n1(CC)nc(C)c(C(=O)NC(CNC(c2sccc2Cl)=O)CO)c1C(F)F 94036,c1(OC)cc[n+]([O-])c(C(=O)NCC(C(C)C)NC(C2CNC(=O)C(C)(C)C2)=O)c1 94037,c1(NC(C(=O)NCCCCNC(c2c(SC)csc2)=O)=O)ccc(C2CC2)cc1 94038,C1(C(N2C(CC(=O)NCCOC3CCOC3)COCC2)=O)Cc2ccccc2C1 94039,[N-]=[N+]=NC1CC(C(=O)NCCc2cscn2)N(C(=O)C2=COCCC2)C1 94040,N1(C(CC(CNC(CC=C=C)=O)(C)C)=O)CC(=O)N(C)CC1CC 94041,CC1CN(C(C2CN(C(=O)CCC3(C#N)CCC3)CCO2)=O)Cc2c[nH]nc21 94042,c1(C(=O)NC(C(C)C)Cc2ccc(F)cc2)ccc(N2CCCC2=O)c(Cl)c1 94043,Cc1ccc(-n2nc(C(C)C)nc2C2CC(=O)N(CCS(C)(=O)=O)C2)c(C)c1 94044,CC1(C(=O)NCC2OCCC2C(=O)NCC2CCC2C(=O)N(C)C)CC(C#N)C1 94045,Cc1cccc(Br)c1C(C(=O)NCC(C)C(C)(C)C)NC(=O)CC1CSCCO1 94046,C=CC(CC)CC(=O)NCC12CC(CN1C(=O)C(C)(C)CO)C2 94047,C=CCCCCCC(C)(c1nnnn1CCCC)NC(C)CCC(=O)OC 94048,C(C)(C)(CN=c1[nH]c2ccccc2s1)C1N(C(C2(COC)CC2(F)F)=O)CCCC1 94049,C1(C(N(C2CC(NC(C3CSC3)=O)C2)C)=O)Cc2nn(C)cc2C(=O)N1 94050,C12(C(=O)NC(C3OCCN(C(C=C4CCC(C)C4)=O)C3)C)CC(C)(C1)OC2(C)C 94051,CCC1=NOC(C(N2CC(F)(C(=O)NC(C)(CO)C3CCCC3)C2)=O)C1 94052,C1(C(=O)NC2CC(NC(c3c[nH]c(=NC)s3)=O)C2)CCc2c[nH]nc2C1 94053,Cc1cc(C(F)F)oc1C(N1CC(NC(C2CCC(F)(F)C2)=O)C(O)C1)=O 94054,CN1CCOC(C(=O)NCCC2COCCN2C(c2csc(Cl)c2)=O)C1=O 94055,C1(CC(N2C(CNC(COC(CC)(C)C)=O)CCC2)=O)COCCN1CC(F)F 94056,Cc1csc(C(N2CCCC(C(C)NC(C34CC(CCO3)C4)=O)C2)=O)c1C 94057,C1(N(CC=CC=O)C)CCOC(C)C1.C(C(=O)NCC=CC=CC)=CC=CC 94058,c1(OC)ccc(C(C)(C)C(=O)N(O)Cc2cn(C(C)C(C)O)nn2)cc1OC 94059,C1(NC(CC2CC(C)(C)OCC2)=O)CC2(CCCN(C(C3(C)CCCOC3)=O)C2)C1 94060,C1(CCC)CN(C(=O)CC(C)CC)CCN1C(=O)CN1CCC(C)CC1 94061,C1(C(=O)NCC2(O)CN(C(CC=CC)=O)C2)(C(F)F)CCN(C)CC1 94062,c1(C(N2C(CNC(c3cc(OCC)ns3)=O)CC2)=O)cc(CC)nn1CC 94063,N1(C(C2CC(CF)C2)=O)CCC(Cn2cc(C3COCC3O)nn2)C(F)(F)C1 94064,CCCC(CC)C(=O)NC1(CO)CCCN(C(c2cc(C(C)=O)cnc2C)=O)C1 94065,N1(C(c2cc(C)n(C)c2)=O)CCCC2(CC(NC(=O)CCc3nccs3)C2)C1 94066,C(=O)(CCC(F)(F)F)N(CC(C)NC(=O)C(C)CC1CC1)CC 94067,C1(C(=O)NC(C)(C)CNC(c2ccccc2)=O)CC1CCS(C)(=O)=O 94068,C1(NC(C2(NC(C)=O)CCC2)=O)C2CCC(C2)C1C(=O)NC(C)COC(F)F 94069,c1(SC)ccccc1-c1cn(CCCN(C)C(C2CC3CC3C2)=O)nn1 94070,C1(CC(=O)NCC(C)C2CC2)CC(NC(C2CCCC2)=O)C1 94071,n1(CC(=O)N(C)CC2CCN(C(C3(F)C(C)OCC3)=O)CC2)cccc(N)c1=O 94072,c1(C(N2CC3CC2CCC3Nc2n[nH]c3c2CCC3)=O)cccn2ccnc12 94073,N1(C(CCCNC(=O)OC)=O)CCC(C2CC2)(CCNC(=O)C(C)S(N)(=O)=O)C1 94074,C1(CNC(c2[nH]cc(C(C(C)C)=O)c2)=O)CN(C(C2C=CCC2)=O)CC1C 94075,O=C(C1CCCOc2ccccc21)NC1COCC1N1CCCC1 94076,c1(CNC(c2c(C)cnn2C)=O)ccc2c(c1)CCC2NC(=O)CSC(F)(F)F 94077,c1(C(=O)NCC(C)(C)NC(C2(COC)CCOC2)=O)cc2cc(Cl)ccn2n1 94078,N1(C(COC(CC)C)=O)CC2CC2(NC(c2oncc2C)=O)C1 94079,C12CCN(CC1)NCC(=O)N2.c1(CSCCNC(C2C3CCC23)=O)cccnc1 94080,N1(C(=O)C(N2CCCC2CO)C)CCCCCC1.C=CCC(=O)NC1(CNC)CC1 94081,c12nc(ncc1Br)NO2.C1(NC(C)C)C2CN(C(=O)CCc3ccco3)CC12 94082,C1(C(=O)NC2CCCC2OCC(F)(F)F)CCC(F)(CO)C1 94083,c1(C(=O)NC2(c3ccccc3)CN(C(c3cnn(C4CC4)c3)=O)C2)n[nH]c(O)n1 94084,c1(C(=O)NC2CC3(C(NC(CC4ON=C(C)C4)=O)C3)C2)ccnc2[nH]c(O)nc12 94085,n1(CC(=O)NC2(CC(=O)NC3CCCCC3CO)CCC2)[nH]cc2c(=O)ncnc1-2 94086,C1(C(=O)NCC(CNC(CC(C)OC)=O)O)CC(=O)N(C(C)C2CC2)C1 94087,CCCCC(CC)C(=O)NCCNC(c1sccc1C(C)(C)C)=O 94088,Cc1cc(C(N2CCNC(C(=O)NCC3CC(=O)N(C)C3)C2)=O)cc(C#N)c1 94089,c1(C(=O)NCCC2(O)CN(C(CSCC)=O)C2)sc2cncn2c1C 94090,c1(C(=O)NCC(CCC)NC(c2cc(C3(C)CC3)on2)=O)ccc(F)c(O)c1 94091,N1(C(C(Cn2cccn2)NC(C2CC(C(C)C)C2)=O)=O)CCCC(C)(O)C1 94092,C1(NC(C(CC)N(C)C)=O)CCCC12CCN(C(c1oc(C)nc1CC)=O)CC2 94093,c1(NC(C)=O)cccc(F)c1-c1cnc(F)c(C(N2CC3C(C2)C3(C)C)=O)c1 94094,c1(C(=O)NC(c2cccc(N)n2)C)cnc2n1CCOCC2 94095,C(=O)(C(C)(C)CC(F)(F)F)N(CC(CNC(c1c(OC)n(C)nc1)=O)C)C 94096,CCC(C)(O)C(=O)NC1C=CCN(C(C2(O)CCCCC2)=O)C1 94097,c1(CCCNC(CCN(C(CCCOC)=O)CCO)=O)ccc(O)cc1 94098,CCC(CC)C(C(=O)N1CC(NC(c2cc3scnc3[nH]2)=O)C(CC2CC2)C1)OC 94099,C1(CC(=O)NCCOCCN(C(=O)CCCCc2cnn[nH]2)C)COCCN1C 94100,C12(C(=O)NC3CC(NC(c4c(C)nc(Br)o4)=O)C3)CC(C)(CCO1)C2 94101,C(CN=c1[nH]c2c(c(=NC3CC4CC4C3)[nH]1)CCCCCC2)c1ccc(C)o1 94102,Cc1cc2ncc(C(=O)NCC(C)NC(=O)CN3CCCC3C)cc2[nH]1.C(=O)O 94103,N1(C(CCC=C)=O)CCC(CO)(NC(c2cnn(-c3ccccc3)n2)=O)C1 94104,C1(CNC(=O)C(O)CN2CCCC2F)CCN(C(c2cc(CF)on2)=O)CC1 94105,N1(C(C(C)NC(C)=O)=O)CCC(C(C)(C)C)(CNC(=O)CCCc2cccnc2)C1 94106,c1(CNc2ccc(OC)c(Br)c2F)cnc2c(c1)c(C)nn2C 94107,C1(=O)C(C2CCC2)OCCN(CC)CCNCCCCN1C.C=CCOC 94108,C(=O)(C1=Cc2ccccc2C1)N1C(C)(CC(=O)N(C)CC2CCCCCC2)CC1 94109,c1(CNCCCN(C(=O)OCC)C)cccn1Cc1ccccc1 94110,c1(NC)cccc(C(N2CC(CN3CCN(C(=O)C(C)CO)CC3)C2)=O)n1 94111,C12(C(N(CC(C)CNC(=O)C(c3cnn(C)c3)O)C)=O)CC1CNC2=O 94112,N12CCCC1C2=O.c1(CNC)nnc(O)o1.C1(CCOC)CC1C=O 94113,c1(C(=O)NCC2(O)CN(C(C(C)Sc3nncn3C)=O)C2)nn(C)cc1N 94114,c1(OCC)ncc(C(=O)NC2CC(N(C(=O)C(c3cccnc3)=O)C)C2)s1 94115,c1(NC2CCC(CNC(COc3c(C)ccc(Cl)c3)=O)C2)ccc(F)cc1[N+](=O)[O-] 94116,c1(N(CCCCN(C)C(C2CCC3CC3CC2)=O)C)c([N+](=O)[O-])cnn1C 94117,c1(C(N(C)CC2N(C(c3cnc(OCC)s3)=O)CCC2)=O)ccc(F)c(F)c1 94118,n1(CCNC(=O)OC)nnnc1C1C2CC(C2)N1.c1(SC)ccccc1.C(C)O 94119,C1(CCNC(C(COC)C)=O)CN(C(=O)C(F)=C(C)C)CCCO1 94120,c1(OC)cccn2ncc(C(=O)NC(C)CNC(=O)Cn3nnc(C4CC4)n3)c12 94121,c1(OC)cc(CC(=O)NCC2(C(C)NC(=O)CC(C)(F)F)CC2)cc(F)c1 94122,c1(C(=O)NCC(CCNC(C2(CCCC)CCC2)=O)O)ccc2c(c1)OCCO2 94123,c1(C(N(CCC)CCN)=O)ccc(F)c2c1OCC2.c1(C=O)cc(CC(C)C)cs1 94124,C12(CNC(c3cn(CCC)nc3)=O)CC1CN(C(=O)CC1CCC1(F)F)C2 94125,C1(C(N2CCN(C(CNC(=O)CC(F)(F)F)=O)CC2)=O)CCc2nc(O)[nH]c2C1 94126,Cc1c(C(=O)NC(C2(O)CN(C(C3CC34CCC4)=O)C2)C)[nH]c2c(Cl)cccc12 94127,Cc1noc(C)c1C(=O)Nc1ccsc1C(=O)NC1CC1(F)F 94128,c1(OC)ncc(Br)c(=NC(=O)C2(O)CCN(S(=O)(=O)c3ccc(Cl)cc3)C2)[nH]1 94129,CC1(C(=O)NS(=O)(=O)CCCC2CCOC2)Oc2ccccc2NC1=O 94130,N1(C(C)C)CC2C3CCC(C2C1)N(C(c1cc(O)nc(C2CC2)n1)=O)C3 94131,c1(CNC(c2n(C)ccn2)CC2CCOC2)cc(F)ccc1Br 94132,N(C(=NCCc1cncn1C)NCCN1CCCC1)CC1(C)CCCCO1 94133,C1(O)(C(N(C(C)CCNC(=O)CC2(C)CCOC2)C)=O)CC2CCC1C2 94134,C1(CNC(=O)CCC2CCCN(C(C3C4CCC3CC4)=O)C2)CCCC2CC12 94135,C(=O)(C1=CC2(CCOCC2)C1)N(CCCNC(C1(C)CCCNC1=O)=O)C 94136,C1(CCC)CN(C(c2nc(C)oc2OCC)=O)CCN1C(c1cc(=O)cc[nH]1)=O 94137,c1(C(=O)NC(C)(CNC(c2cn[nH]c2)=O)Cn2cccn2)cccc2scnc12 94138,c1(NC(=O)NC2CC3CC(C(=O)O)CC23)cc2cc(Br)ccc2s1 94139,c1(C(CC(c2cccs2)NC(=O)CC(C)C)C)ccc(F)c(F)c1 94140,c1(C(=O)NCC(=C)CCNC(=O)Cc2occc2C)ccccc1SCC 94141,C1(C(=O)OCC)(C(c2cccc(Cl)c2)Nc2nc[nH]n2)CCCCC1 94142,N(C1CN(c2nc3ccccc3s2)CCc2ccccc21)C(C(C)CC(F)F)=O 94143,C(=O)(C(C)(C)C(=O)NC1CCCC(C(=O)Nc2ncnc(Cl)c2Br)C1)OC 94144,c1(C(=O)NCCN(C(=O)C(Cc2ccsc2)NC=O)CC)ncc(Cl)n1C 94145,c1(SCC)ccc(C(=O)N(C2CN(C(=O)CCCNC(=O)OC)CC2O)C)cn1 94146,c1(C(=O)NCC(CC)(CC)NC(=O)C(F)(F)COC)ccc2cccnc2n1 94147,C12(NC(C3CCCCS3)=O)CC(C(=O)NCc3snnc3C3CC3)(C1)C2 94148,C(C)(C)(CCNC(=O)Cc1cc(C(C)C)no1)NC(COCC(=O)NC)=O 94149,CCCC1=C(C(=O)N(C2CC(NC(=O)C(C(C)C)OCC(C)C)C2)C)CCCO1 94150,CC(=O)CCC(=O)NCC1CCC(N(C(=O)CC2OCCC2C)C)CC1 94151,C1(NC(c2cc(C(=O)OCC)no2)=O)CN(C(c2cc[nH]c2)=O)C2CC12 94152,c1(C(=O)NCCN(C(=O)CCOCC2CCCO2)C)cc2cccc(F)c2s1 94153,C(C(C(=O)NOCCCC)NC(c1ccc(C)nn1)=O)SCC 94154,c1(C(=O)NC2C(NC(C(C)(C)CF)=O)CC(F)(F)C2)cnc2c(F)cccc2c1 94155,N1(C(C(C(=O)OCC)(C)F)=O)CC2(C1)CN(C(=O)C(C)(C)C(C)C)CC2CO 94156,Cc1cc(C(N2CC3C(C(N4CCC=C(F)C4)=O)C3C2)=O)n(C)n1 94157,c1(CC)ccc(C2(C(=O)OC)CCCC2)cc1.c1cn(CC(=O)Nc2nccs2)nn1 94158,Cc1cc(F)ccc1COCCN(C(=O)NCC1CC1)CCNC(=O)COC(C)C 94159,c1(C(N2CCC(c3nncs3)C2)C(=O)NC)cccc(CNC(C)(C)C)n1 94160,Cc1ccc(C(=O)N(CC(N2CC(CN(C)C)CC2C)=O)C(C)C)cn1 94161,c1(C(=O)NCCC2CN(C(C3CCCCC3)=O)CCCO2)cc2ccncc2[nH]1 94162,c1(C(N2CCCC(C3N(C(CC=C)=O)CCC3)C2)=O)ccc(CC)cc1Cl 94163,CCCCC(O)CC(=O)NC(CC)CC(N1CCC2(CCCO2)C1)=O 94164,c1(C(N2CC(NC(CCC#C)=O)C(C)C2)=O)ccc(NC(C)C)cc1Cl 94165,c1(C(=O)NC2(CNC(C(C)OCCCC)=O)CCOC2)ccc2occ(C)c2c1 94166,N1(C(CN(C(CC)C)C2CC2)=O)CCCC2C1CCN2c1ccncn1 94167,C(=O)(C(F)C(=O)NC1CCCC1CNC(c1ccncc1Br)=O)OCC 94168,C1(C(=O)NCCCn2cc(CC3CCNC3=O)nn2)C2Cc3cc(Cl)ccc3C12 94169,c1(C(N(C)CC2CCCN(C(c3c(C)cn(C)n3)=O)C2)=O)cc2sccc2s1 94170,N1(C(c2cncc(OC)c2)=O)CCCC(C)(C(N2C(C)CCC2(C)C)=O)C1 94171,C1(NC(CCOCC(C)C)=O)CCCC(NC(=O)CCc2nc(N(C)C)no2)C1 94172,C=CC(C)(O)C(=O)N1CC(NC(=O)CCSCC)C(C(F)(F)F)C1 94173,CN1CCN(C(=O)C(CC2CC2)NC(c2cc[nH]c2)=O)CC1CO 94174,C=C(C)CC(C(=O)NC1(c2cccc(F)c2)CC1)NC(C1CC(C)C1)=O 94175,c1(C(=O)NC2CC(NC(c3ccn(CC(=O)OCC)n3)=O)C2)ccc(F)c(Cl)c1 94176,c1(CC)nc(=NC2(CNC(C3CCC4(CCOCC4)O3)=O)COC2)s[nH]1 94177,c1(N(CCCc2cc(Cl)ccc2Cl)C)nc(NCC2CC(F)C2)c2[nH]ccc2n1 94178,C1(OC)(CNC(C2(C(F)(F)F)CC2)=O)CCN(C(c2sccc2Cl)=O)C1 94179,c1(C(N(C(CNC(C2CCN(C(CC)=O)C2)=O)C)C)=O)cc([N+](=O)[O-])cc(C)n1 94180,C1(NC(c2ccc(N3CCC3)nc2)=O)CN(C(C2CC(CF)C2)=O)CC1C(F)F 94181,c1(N2CC(CN(C)C(c3c[nH]cc3Br)=O)C2)nc(Cl)nc2c1ncn2C 94182,c1(N2CC=C(C)C2)ccc(S(=O)(=O)N2CCCC3(CCCCC3)C2)c(Cl)c1 94183,c1(C(=O)Nc2c(C)n(-c3ccc(OC(F)F)cc3)nn2)cn2cc(F)ccc2n1 94184,CC1CC2(CC(C(=O)NC3CC=C(C(=O)N(C)Cc4ncco4)C3)C2)C1 94185,CC1=C(C(=O)NCC(C)(F)CNC(C2(C(C)C)CNC(=O)C2)=O)C(C)(C)CCC1 94186,c1(C(N2CCN(C(C(CC)CC)=O)C(CCCC)C2)=O)ccc2c(c1)COCO2 94187,C(=O)(CCC(=O)NCC(C)(C)OC1CCC1)NC.N12CCC(C1)OCC2=O 94188,Cc1cc(N)c(C)nc1C(=O)NCC(O)CNC(=O)C(c1ccc(F)c(Cl)c1)O 94189,CN1CCN(C(C2C(C)(C)C2(C)C)=O)C(CNC(C2CCCC(O)C2)=O)C1 94190,c1(C(N(CCOCCN(C(Cn2c(C)ncc2)=O)C)C)=O)cnn2c1N(C)CC2 94191,n1(C(C2CCCN(C(C(COCC(C)C)(C)N(C)C)=O)C2)=O)nnc2ccccc12 94192,N1(C(c2scc(C)c2)=O)CC2(CCCC2NC(c2cccc3nonc23)=O)C1 94193,c1(C(=O)NC(C(=O)OC)CC2CCCO2)cccc2nccn12 94194,C1(CNC(C=CS(C)=O)=O)CN(C(=O)C=Cc2cccc(F)c2)CCCO1 94195,C(CCCCCNC(c1cccc(C(F)(F)F)n1)=O)NC(=O)C(Cl)=CCl 94196,c1(C(=O)NCc2c(C)c(Cl)ccc2)n[nH]c2c1CN(C(C13CC(C1)C3)=O)CC2 94197,c1(NCC(CNC(C(CCCOC(C#CC)C)C)=O)F)cc(O)c2ccsc2c1 94198,c1(N2CCC(NC(c3c(C(C)C)ocn3)=O)C2)ncnc2c1[nH]c(=N)n2C 94199,C1(CNC(C2CCCO2)=O)CC2CC2N1C(=O)CC1CC(n2cnnc2)C1 94200,C(=O)(CCS(C)(=O)=O)N1C(C)(C(=O)NC2(COCC)CC2)C=CC1 94201,N1(C(C(CCC)OCC)=O)CCN(C(=O)C(C)(C)CCOC)CC(CO)C1 94202,C(=O)(C(CNC(C1CC=CCC1)=O)C(C)C)N1C(CC(=O)OCC)CCC1 94203,C=C1CC(C(N2CCCC2CCCC)=O)(CNC(C2CCCSC2)=O)C1 94204,O=C1CCOC(C(=O)NCC2CC(F)(CNC(=O)C(F)n3cccn3)C2)C1 94205,C1(COC(c2ccn(C)n2)=O)CC(=O)N(C(C2CCCC(=O)O2)=O)C1 94206,N1(C(C23OCC(C)(C2)C3)=O)CCC2(CC1)CCN(C(=O)C=C1CCSCC1)C2 94207,CCC(CCC(=O)NCCC1CCC1)NC(c1cn(CC)nn1)=O 94208,C1(OC)CC(C(N2CCCCC2c2cccc(C)c2)=O)CC1OC 94209,c1(C(N2CCC(C(CNC(C(C)CO)=O)(C)C)CC2)=O)ccc2scnc2c1 94210,N1(CN(C2CC(N)C2)C)CCCCCC1=O.N1(CC(=O)NS(C)(=O)=O)CCC(F)(F)C1 94211,Cc1ccc(CNC(c2n[nH]cc2CNC(C2C3CN(C)CC23)=O)=O)cc1C 94212,N1(C(n2c(CC)nnc2S)=O)CC(C(N)=O)CC(C)C1 94213,Cc1nccc(C(=O)N(C(CC(F)F)C(=O)NCCCC2CCOCC2)C)c1C 94214,c1(N(C(C2(CC#C)CCOC2)=O)CCCO)cc(C)cc(C)c1 94215,CC1CCCC=C1C(=O)NCC(C)(C1CC1)NC(=O)C=CC(=O)N(C)C 94216,N1(C(CC=CC=C)=O)CCC(OCCC(=O)OCCSC(C)CC)C1 94217,c1(OC)n[nH]c(NC(C2CC23CCN(c2cc(C(F)(F)F)ncn2)C3)=O)c1C#N 94218,CN1CCN(C(C=CC(=O)NC2CC2)=O)C(C(=O)NOC2CCCC2)C1 94219,c1(C(N2CCC2CNC(C2(C(F)F)CCC2)=O)=O)coc2c1CS(=O)(=O)C2 94220,N1(c2ncc(C(=O)OC)s2)CCOC(C)(CNC(=O)CNc2nccs2)C1 94221,N1(C(C(=O)NC(C)=O)C)CCN(C(=O)C(c2cccnc2)O)CC1 94222,C(=O)(C1CCCn2cncc21)N1C(CNC(c2c(Cl)cncc2Cl)=O)CC1 94223,c1(C(=O)NCCCNC(=O)C2=CCSC2)ccc([N+](=O)[O-])c(C(F)(F)F)c1 94224,c1(C(CCOC)NC(c2n(C(CC)C)nnn2)C2(C3CC3)CCC2)nc(Br)cn1C 94225,c1(C(=O)NC2CC(CNC(C3CC(CC)OCC3)=O)C2)nc(N(C)C)nc(=N)[nH]1 94226,c1(C(=O)NC(COCC)C(=O)N2CCC(SC)C2)ccc([N+](=O)[O-])[nH]1 94227,N1(C(C(C)(C2CC2)OC)=O)CCC2(CC1)CC(NC(=O)C=CC(N)=O)CCO2 94228,C1(F)(C(N2CCCC(CCC=C)C2)=O)CCN(C(C2CCCC(CF)C2)=O)CC1 94229,C(=O)(CCCCCF)NC(C)(CNC(=O)C=Cc1nnc(C(C)(C)C)o1)C1CC1 94230,c1(C(=O)NCC(C)(C2CCC2)NC(CC(CC)C)=O)cccc(C(=O)OC)c1O 94231,C1(NC(C2C(C)N(C)CC2)=O)CCC12CCN(C(c1cnccc1CO)=O)CC2 94232,N1(C(c2[nH]c(CC)c(Cl)n2)=O)C2CCCC1CN(C(C1(CO)CC(C)(C)C1)=O)C2 94233,C1(c2ccccc2)(NC(=O)CNC(=O)CCc2cncc(Br)c2)CC2CCC2C1 94234,c1(OC)cccc(C(=O)NC(C)CN(C(=O)COCC2CCC2)C)n1 94235,C(CCC(C)(C)NC(=O)C(c1ccc(C)s1)C)NC(C(C)NC(COC)=O)=O 94236,C(=O)(C1=C(Cl)CCC1)NCC(C)(C(=O)O)OC 94237,N1(C(C2N(C(C)C)CCC2)=O)CC2(C1)CN(C(c1ccc(C(F)(F)F)nn1)=O)C2 94238,c1(C(=O)NCC(CC)(CC)NC(=O)CCC2CC2C)sc2nccc(C)c2c1C 94239,C1(C(N2CC=CC(NC(C3N(C)C(=O)CC3)=O)C2)=O)CC2(C1)OCCO2 94240,N1(C(C(CCF)NC(CCCC)=O)=O)CC2(CO)CC1(CO)C2 94241,CCC(CN=c1[nH]c(=N)[nH]c(=NCC2(c3ccccc3)CCC2)[nH]1)OC 94242,c1(OC)cc([N+](=O)[O-])ccc1C(=O)NCC(C)NC(C1CCCN1CC(C)C)=O 94243,C1(N(C(C(C)NC(C)=O)=O)C)CCN(C(c2ccnn2C2CCC2)=O)C1 94244,C(=O)(C(C)C(F)(F)F)N1CC(NC(C(c2c(OC)cccc2)O)=O)C(SC)C1 94245,CC1CC(NC(C2CCCN2C(C2CCCC2)=O)=O)CN(C(C2(C)CC(=O)C2)=O)C1 94246,CC1(C#N)CN(CC2(c3c(F)cccc3F)CC2)CCO1 94247,C(=O)(C#CC1CCCCO1)NC(CNC(C(CCCC)O)=O)(CC)CC 94248,C1(C(=O)NC2C(C(=O)NC(c3ccncc3F)C)CC=CC2)CC(=O)CC12CCC2 94249,C(=O)(C(C)(CC)CC)N1CCC(N(C(C=CC)=O)C(C)C)CC1 94250,Cc1ccnc(C(=O)N(C2CC2)CC2CCN(C(=O)CC3CN(C)C3)CC2)c1 94251,C1(C(N2CC(O)(CNC(c3nc[nH]c4ncnc3-4)=O)C2)=O)CN=C2N=CNN2C1 94252,N1(C(c2c[nH]c(=NC)s2)=O)CCCCC(CNC(c2coc(C3CC3)n2)=O)C1 94253,CC(COC(c1c(O)noc1C)=O)CC(=O)N1CCCC1 94254,N1(C(C2CC(CNC(C3(CC)CCCC3)=O)OC2)=O)CC(F)(F)C(F)(F)C1 94255,CC1(C)CC2(CC(NC(C3(CC(c4cccc(F)c4F)=O)CCCCC3)=O)C2)C1 94256,c1(OCC)nc(C)ccc1C(N1CC(NC(c2cnc(CC)s2)=O)C(O)C1)=O 94257,N1(C(c2ncnn2CCCF)=O)CCC2C(C1)C2(F)F 94258,c1(C(=O)Nc2c(C)nc(CO)cc2)cnn2ccc(C(F)(F)F)nc12 94259,CS(=O)(=O)CCCC(=O)NCC1(F)CC(CNC(c2cc(CO)on2)=O)C1 94260,C1(CC(N2CCN(C(CC3OCC(C)(C)C3)=O)CC2)=O)COc2ccccc2O1 94261,C1(NC(C(C)SC)=O)CCN(C(c2cnn(CC(F)F)c2C)=O)CC1 94262,c1(C2(C(=O)NC(C3CN(C(C(=O)NC(C)C)=O)C3)C)CCC2)ccccc1 94263,c1(C(=O)NCC(C)N(C(=O)CC2CCCC(=O)C2)C)cccc(N)c1 94264,Cc1cc(Br)c(C)c(S(=O)(=O)N2CCC3(CCN(C(=O)CN(C)C)CC3)CC2)c1 94265,C(=O)(C1=C(C)CCC1)N1C(C(N2CC3CCC3C2)=O)(CC)CCC1 94266,C1(C(=O)NC2CN(C(c3csc(-c4ccco4)n3)=O)C2)CCC(CC2CC2)CC1 94267,C1(NC(c2cc(C(F)F)no2)=O)CC2CN(C(=O)Cn3nccn3)CCN2C1=O 94268,CCCCCCCNC(C1COCCC1NC(c1cc(CC)[nH]n1)=O)=O 94269,CC(CC(C)(C)C)C(=O)N(CCCN(C)C(c1cc(C(F)F)no1)=O)C 94270,N1(CC(=O)NCCSC)CCC2(CCOC2)C(C(=O)NCCOCC=C)C1 94271,N1(C(CC2C(NC(c3ccc(OC)nc3)=O)CCC2)=O)CC2(CN1CO)CCC2 94272,C(=O)(C(CP(C)(C)=O)C(F)(F)F)Nc1cc(C)c(Br)cc1F 94273,O=C1NCc2ccc(-c3ccc(N4CCN(c5cccc(Br)c5)CC4)cc3)cc21 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94851,C1(NC(CCOCCC)=O)CCSC12CN(C(=O)C(C(C)C)n1cnc(C)c1)C2 94852,C(=O)(CC1=CCCC1)N1C(C)(CNC(c2ccc(SC3CC3)cc2)=O)CCC1 94853,C1(CNC(C23N(C(c4ccccc4)=O)CCC2C3)=O)CC2(CCCO2)C1 94854,c1(C(=O)NCCC2N(C(CSCCC)=O)CCOC2)c(C)nc(O)nc1C 94855,C=CCC(C)C(=O)NC1COCCC1C(=O)NCC(F)C1CCC1 94856,Cc1ccc(C(N2CCCC2CN(C(=O)C(=O)NC(C)C)C)=O)c(N)n1 94857,C1(C)(C(=O)NC(=O)C2CC2)CC2CN1c1ccc(nc1)C(=O)N2.C1(N)CC1.C(F)F 94858,C1(CN(C(=O)C(C)NC(C)=O)CC)CCCN1C(C1CC(C(F)F)(OC)C1)=O 94859,Nc1ccc(Cl)c(C(=O)NCC2CCCCN2C(=O)C(F)C2CCOC2)c1 94860,C1(NC(CCCC(=O)OCC)=O)COC2(CCN(S(C)(=O)=O)C2)C1 94861,CC1(C)CCN(C(C2OCCC2(C)C)=O)CC1C(=O)NCC(F)F 94862,CN=C(NCC(C1CC1)OC)NC1CC(OC)C1 94863,c1(C(=O)NCC(N2CCC2C(=O)Nc2nccnc2Cl)=O)cnc2cccnn12 94864,C1(CCCNC(C2CN(C(=O)C(CO)NC(=O)C(F)(F)F)C2)=O)CC2(C1)CC2F 94865,CC1(C)CCCC(O)(C(=O)NCC2(C)CCN(C(C3CC(=O)CO3)=O)C2)CC1 94866,Cc1c(CC(=O)NCC=C2CCN(C(=O)CCCCN(C)C)CC2)cnn1C 94867,CC1CCC(C(=O)NC2CC2CNC(c2ccnnc2O)=O)CC1 94868,c1(C(=O)NCCCOCCCNC(C2CCN(C)C2=O)=O)c[nH]c2ccncc12 94869,Cc1cc(N2CC(CN(C(=O)CC(C)c3cnn(C)c3)C)C2)c(Br)cc1[N+](=O)[O-] 94870,Nc1cc([N+](=O)[O-])ccc1C(=O)NC1COCC1SCc1cn(C23CC(C2)C3)nn1 94871,c1(C(N2CCCC(C)(NC(=O)CCC3CC3CC3CC3)C2)=O)ccc([N+](=O)[O-])cc1 94872,N1(C(C(C)(C)NS(C)(=O)=O)=O)CC2CCN(C(c3cc(F)cc(Cl)c3N)=O)C2C1 94873,c1(Nc2cc(C(C)(C)NC(=O)NC(C3CCOC3=O)C)[nH]n2)cnc(O)c(F)c1 94874,C(=O)(C(F)(F)CC(C)C)N1CC(CNC(c2c(CC)cns2)=O)C1 94875,Cc1cnccc1C=CC(=O)NCCC(C)NC(=O)C=CCn1cncn1 94876,c1(CCC(=O)NCC2N(C(c3occ(C)c3C)=O)CC2)c(Cl)cncc1Cl 94877,C1(NC(c2n(CC)ncn2)=O)C2CC3CN(C(=O)CN(S(=O)(=O)CC)C)C1C3C2 94878,c1(C(=O)NCC(CNC(CCNS(CC)(=O)=O)=O)(C)C)cc(Cl)nnc1O 94879,c1(-c2ccnc(CN3C(C(F)(F)F)CCC(C(C)C)C3)n2)cnc2cccnn12 94880,c1(C(=O)NC(CC)CN(C(=O)C(C)(C)NS(C)(=O)=O)C)ccc(CSC)c(F)c1 94881,CCCC(C(O)C(=O)N1CC(N(C)CCO)C1)NC(=O)Cn1cnc(=N)[nH]1 94882,CC(C)(CNC1CCC(Cc2ccccc2)C1)CO 94883,C(=O)(CC1COCc2ccccc21)NC(C1CN(C(=O)C2=CCOC2)CCO1)C 94884,CC1CCC(C(=O)NC2(CC(=O)NCCNC(=O)CC(C)(C)C)CC2)OC1 94885,CC1C(C(F)(F)F)NCCN1C(c1cc(-c2cccc(F)n2)no1)=O 94886,C12(C(N3C4C(NC(CC5(OCC)CC5)=O)CC(C4)C3)=O)CCC(CO)(CC1)CC2 94887,n1(C(C)(C)C)c(O)nc2cc(C(=O)NCC3CCC3NC(=O)C3CC3)ccc12 94888,C1(CC)COC(C)CN1C(c1nc(F)ccc1Br)C(=O)NCC1(C)CC1 94889,C12(NC(CC)=O)CCCCC1N(C(=O)Cc1csc(N3CCCCC3)n1)CC2 94890,N1(CC(=O)NCC(CNC(CCOC(=O)CO)=O)C)CCCCC1C 94891,CC1OC2(C)CC1(C(N1CCC1CNC(c1ccc(SC3CC3)o1)=O)=O)C2 94892,C1(C(C)NC(=O)C(F)C2CCC2)CN(C(c2cc[nH]c(=N)n2)=O)CCO1 94893,C(=O)(C(O)C(F)(F)F)N1CC(C(N2CCC2C)=O)(COC)C1 94894,c1(OC)ccc2c(ccn2CC(=O)NC2CCCC2CNC(=O)CCC(C)O)c1 94895,c1(C(=O)NCC2N(C(C3CCC3)=O)CCN(C)C2)nnc(O)c(Br)c1O 94896,C1(C(=O)NC2C(C)(C)C(Nc3ncc(Br)cn3)C2)CC2CCCCCCC12 94897,CC1CC(C(N2CC(CCO)(NC(=O)CCn3cccnc3=O)C2)=O)CCN1C 94898,O=C1CC2CCCC2(C(=O)NC(CNC(C2CCn3cnnc3C2)=O)C2CC2)C1 94899,C(=O)(C(=O)N=S(C)(C)=O)N1C2C(NC(C(C(C)C)N3CCCC3=O)=O)CC(C2)C1 94900,C1(NC(Cc2ccc(SC)cc2)=O)CCN(C(=O)CN2CC(C)C2)CC1C.N(C)C 94901,C(N=c1[nH]c(-c2ccc3occc3c2)cs1)(C(F)(CC)CC)c1n(CC)nnn1 94902,C12CCCC1C(=O)NCCOC1CCN(C1)C2=O.C1(N2CCCC2)(CC)CCCC1 94903,C1(NC(CC2(NC(C3CNC(=O)N3)=O)CC2)=O)CC2CC(O)C1C2 94904,C1(C(=O)OC(C)(C)C)(CC)CCCN(C(=O)CCSC)C1 94905,N1(C(C(c2n(C(C)C)ccn2)(F)F)=O)CC(NC(=O)C(C)C(C)(F)F)C(C)(C)C1 94906,CC(C)CCC(C(=O)N(C)CC1(O)CCC1)NC(=O)C(C)CC(F)F 94907,C(CC(N)=O)(C(=O)NC(c1ccccc1O)C)NC(C(F)OC)=O 94908,CC1(C)Cc2ccc(S(=O)(=O)N3CCCC(c4ccno4)C3)cc2C1 94909,C1(OC)CN(C(=O)CCN2CCCC2=O)CC1NC(C12CC1CNC2=O)=O 94910,c1(OC)cccc(CC(=O)NC2CC(CO)N(C(=O)CC(C)OC(C)=O)C2)n1 94911,c1(C(=O)NCCC2CC(NC(C3N(CC)CCC3)=O)C2)cccc2sccc12 94912,C(=O)(C1CCCc2nn[nH]c21)N1CC2CCN(C(=O)CC34CC(C3)C4)CC2CC1 94913,c1(C(N2CC(NC(c3cn(CCC)nc3)=O)(COC)C2)=O)sc2cncn2c1C 94914,c1(-c2c(OC)ccnc2)cn2cnc(C(=O)Nc3nc(C)ccc3F)c2s1 94915,N1(C(=O)OC(C)(C)C)CCCCC1CCC(=O)NC(C1CC2CCC12)=O 94916,C1(NC(C23CCC(NC(C(CCCC)F)=O)(CC2)C3)=O)CCOC2(CCC2)C1 94917,c1(COC)cccnc1C(=O)NCCC1CCCN(C(c2cc(C)co2)=O)C1 94918,C1(C2C(=O)N2C2CC2)CC=CCC1.C=C(C)COCC(=O)NCCNC(N)=O 94919,c1(C(=O)NCCNC(c2cc(C(C)(C)C)n[nH]2)=O)cccc2c1CCC2 94920,C1(NC(C(CC)OC)=O)CC2CCC(C1)N2C(c1cnc(-c2ccoc2)s1)=O 94921,N1(C(C(CSC)(C)O)=O)CC2(CC(NC(=O)CN(C3CCS(=O)(=O)C3)C)C2)C1 94922,C1(CC(=O)NC(C)CCOC)(OC)CN(C(C2(OC)CC2)=O)C1 94923,C1(C(N(CC(CN(C(C(CC)CO)=O)C)O)C)=O)CCn2c(O)nnc2C1 94924,N1(C(c2cnc(C(C)OC)s2)=O)CC2C(CN(C)C(c3cccnc3)=O)C2C1 94925,CCCC(C(F)(F)F)NC(=O)C=C(C)CNC(c1ccc(OC)s1)=O 94926,C=C(C)CCCC(=O)NCCN(C(=O)CC1CCCC(=O)C1)CC 94927,N1(C(C(C(C)C)C)=O)CCCC2(CCN(C(C3(C)CC(C)(C)C3)=O)C2)C1 94928,c1(NC(C(C)OCc2cccc(C)c2)=O)cccc2c1CC(=O)N2 94929,C1(NC(CSc2n(C)nnn2)=O)CN(C(=O)CC2CC(=O)C2)CC1n1cccn1 94930,c1(OC)cc(C)nc(N2CCOC(C(=O)Nc3cc(C)cc(C)c3)C2)n1 94931,C(=O)(C1CCc2ccccc21)N(CCCN(C(CCc1cc(C)on1)=O)C)C 94932,C12(NC(C3(C)CC(=C)C3)=O)CCC(NC(c3c(C)coc3C(C)C)=O)(CC1)C2 94933,N1(C(C(C(=O)OCC)F)=O)CC2(CCN(C(c3ccc(F)cc3O)=O)C2)C1 94934,c1(NC(C23C(C(=O)OC(C)(C)C)C2CC3)=O)cnc2[nH]cc(C#N)c2c1 94935,N1(C(CC2ON=C(C)C2)=O)CCC2(CCN(C(c3sc(C)cc3Cl)=O)CC2)C1 94936,Cc1cc(C(=O)NCC(C2CC2)NC(=O)Cc2ncc(Cl)s2)c(C)n1C 94937,c1(C(N(CCCCNC(C2CC2(C)C)=O)C)=O)ccc(OCC(F)F)nc1 94938,C1(S)CCN(C)C1.c1(N(CC)CC)nnnn1CCCc1ccccc1 94939,C(=O)(C(O)CCCCC)N1C(CCNC(C2(C=C)CC2)=O)CCC1 94940,CC(C)(C)S(=O)(=O)CC(=O)N1CCN(C(=O)CCN2CCCC2=O)C(C(F)F)C1 94941,C1(CNC(c2cc(C)n(C)n2)=O)CN(C(=O)CC2C=NN(C)C2=O)CC12CCC2 94942,c1(OC)ccc(CC(=O)NC2CC(C)N(C(=O)CN3CSCCSC3)C2)cc1F 94943,N1(C(C(c2cnn(C)c2)C)=O)CC(CC(N)=O)OC(C)(C)C1 94944,C(=O)(CCC(=O)N1C(C(=O)Nc2ccnc(SC)c2)CC2CC12)OCC 94945,C12CCC3CN(CCC3C1)C(=O)C1(CCCC1)c1cn2nn1.C1(C(=O)OC)CCN1 94946,C1(C(C)NC(CCSC)=O)CN(C(=O)CNC(=O)C2CC2)CCO1 94947,C1(CCNC(CN(CC)CC)=O)CCC(NC(c2ccc(C)o2)=O)C1 94948,C(=O)(C1CCc2c[nH]nc21)N(C(CC)CC(=O)N1CC(c2ncc[nH]2)C1)C 94949,c1(OC)ccc(F)c(C(=O)NCCC2CCN(C(=O)CC3(OC)CC3)C2)c1F 94950,Cc1ccc(C(=O)NC2CCC(CNC(=O)CCC(=O)N(C)C(C)C)C2)nc1C 94951,c1(CCCC(=O)NC2CCCC(CNC(C=CCOC)=O)C2)c(F)cccc1F 94952,CC1(C)CC(CC(=O)NC2CN(C(c3cccc(F)c3O)=O)CC23CC3)C(=O)O1 94953,c1(C(=O)NC2CC(CCNC(C3(C)CC=CC3)=O)C2)ccn2nccc2n1 94954,N1(C(c2scc(C)c2C)=O)CCN(C)CC1C(=O)NC(CO)C1(C)CC1 94955,N1(C(c2c(C)nccc2)=O)CCC2(CC1)CCN(C(=O)C(C)CC1CCCO1)C2 94956,C(CCSC)(C(=O)NCCF)NC(C1(N=[N+]=[N-])CC1)=O 94957,N1(C(=O)NCc2nc(CC)sc2Br)CCCN(S(C)(=O)=O)CC1 94958,C1(C(=O)NC2CCC(CCNC(CSC(C)(C)C)=O)C2)CC12CCOCC2 94959,c1(-n2cnc(NC(c3ccc(CN(C)C)o3)=O)n2)ncc(Cl)cn1 94960,N1(C(c2c(C)nc(CO)s2)=O)CC=C(CNC(C23CCC2C3)=O)CC1 94961,c1(C(=O)NCCN(C(CCc2cnc(C)o2)=O)C)cnn(C(C)C)c1C 94962,N1(C(C(C)C2CC2)=O)CCCC(CC(=O)N(C)CCc2cc[nH]n2)CC1 94963,C1(F)(CNC(C2(CC#C)CC=CCC2)=O)CCN(C(=O)C=C(C)C)CC1 94964,C(C(=O)N1CC(CO)(NC(=O)C(c2cnn(C(C)(C)C)c2)=O)C1)(C(C)(C)C)SC 94965,c1(CC)nc2n(n1)CC(NC(=O)NCCC1CCCN(C)C1=O)CC2 94966,C1(CC)C(C)CCN1CC(O)CNC(=O)CC1(OC)CCC1 94967,C(=O)(C(CNC1CN(c2nccc(C#N)n2)C1)CC(C)C)N(C1C(C)=NNC1=O)C 94968,N1(N2CCC(C)(CO)C2)CCC2CCN(C(C)=O)CC12.CCC(C)C=CC=O 94969,C1(C(C)(C)NC(Cc2cc(C)[nH]n2)=O)CCN(C(C2CCOC(=O)N2)=O)CC1 94970,C(N=c1cc(C)[nH]c(=NCC2CC3(CCCC3)CO2)[nH]1)c1c(CC)noc1 94971,N1(C(c2cccc(CNC(c3nn(CC)c(O)c3)=O)n2)=O)CC2CC2C2CC12 94972,CC1CCN(C(c2cccc(Cl)c2)C(=O)Nc2ccccc2)CCS1(=O)=O 94973,CN1C(=O)OCC1C(=O)NCC1CN(C(=O)CN2CCC(C(N)=O)CC2)CCO1 94974,c1(C2N(C(C3COCC4(CCN4)C3)=O)CCC2)c(F)cc(Br)cc1F 94975,c1(C(=O)NC(CNC(C2C(F)(C(=O)OC)C2)=O)(C)C(C)C)cc(C)c(C)cc1N 94976,c1(C(N2CC(CNc3ncc(C(C)=O)nc3)C2)=O)ccc(Br)c2ccncc12 94977,C(C)(CCC(=O)N1CC=CCC1C(N1CCC2CC12C)=O)OCC 94978,CCC(CC)C(C(=O)NC(C)C(N1CCN(C)C(C2CC2)C1)=O)OC 94979,c1(C(=O)NC2(CNC(=O)CCCCSC3CC3)CCC2)cccc(C=C(F)F)c1 94980,C1(C(N2CCOC(=O)C2)=O)(OC)CCN(Cc2cnc(F)c(C)c2)CC1 94981,C12(C(=O)O)CCCCC(CN(S(=O)(=O)c3cnn(-c4ccc(F)cc4)c3)C1)C2(F)F 94982,N1(C(c2cc(CNC(=O)Cc3ccns3)on2)=O)CCn2cnnc2C1 94983,N1(C(c2cc(OC)cc(O)c2)=O)CCCC12CCCN(C(=O)C(C)O)C2 94984,N1(C(C(CC(=O)OCC)C)=O)CCC(C)N(C(=O)CCc2cn[nH]c2)CC1 94985,Cc1ccc(C=CC(=O)NC2CN(C(=O)OC(C)(C)C)CC2C(F)(F)F)nc1 94986,C(C1=CCCN(C(c2cnnc(O)c2)=O)C1)NC(CC1C(C)CCCC1)=O 94987,C(=O)(C1=CC(O)C(NC(=O)CCC2CC2(F)F)C1)N1CC(C#N)(SC)C1 94988,C(=O)(CC(O)C(C)C)N1C(C(N2C(CCC=C)CCC2)=O)CC(=O)C1 94989,c1(OC)cc(-c2ccc(NC(=O)CC(C)SC)cc2)nc(C)c1 94990,c1(C(C)NC(c2nnnn2C2CC2)SC(F)F)c(F)c(F)cc(Br)c1F 94991,N1(C(C2CC(C#N)(OC)C2)=O)CCC(O)(CNC(c2cc(Cl)ns2)=O)CC1 94992,c1(CN2CCC(N(C)C(C)C)(CC)CC2)cccc2c1NC(=O)CO2 94993,C1(CNC(c2noc(CC)c2C)=O)CC(C)(C)CN1C(C1COC(=O)N1C)=O 94994,CCC(C(=O)N1CCC(C(C)N=c2[nH]nc(COC)o2)C1)C(C)C 94995,C(C(C)(C)CN(C)C(C1CC1(Cl)Cl)=O)NC(C(C1CC(F)(F)C1)OC)=O 94996,CC(C)(C#CC(=O)NCc1nnc(O)o1)CNC(C1CCC(O)C1)=O 94997,C(=O)(CCCC(=O)N1CCCCC1CCCNC(=O)Cc1ccc(C)cc1)OC 94998,c12ccc(c(C(C3(C)CC=CC3)=O)c1OC)C(=O)N(C)CC1(CC1)CS2.OC 94999,c1(NC2CC=CCC2)cc(N2CCC(CCn3ccnn3)C2)ncn1 95000,C1(C(N2C(C(C)(C)NC(=O)C3=CCCSC3)CCCC2)=O)CCn2nncc2C1 95001,N1(C(c2cccc(C(C)=O)c2)=O)C2CCCC1CN(C(c1cn(CC)cn1)=O)C2 95002,C1(SC)CCN(C(C2(NC(c3cc(Cl)on3)=O)CC2)=O)C1 95003,C(=O)(CS(=O)(=O)CC(C)C)NCC(CNC(c1cc(C)c(C)s1)=O)O 95004,C1(C(=O)NCC2C(C(N3CCC(COCC)C3)=O)CCC2)CCS(=O)CC1 95005,N1(C(C2C(C(=O)OC)C2)=O)CCC2(CC1)CN(C(C1(O)CCCC1)=O)CC2CO 95006,C1(O)(CC(=O)NCC(C)(C2CC2)NC(c2n(CC)ccc2)=O)CCOCC1 95007,c1(NCC(=O)OC)ccc(C#N)c(OC)c1 95008,C(c1ccccc1Br)=CC(=O)NC1CN(C(c2ccc(C(N)=O)[nH]2)=O)C1 95009,c1(C(N(CCN(C(=O)C(C)NS(C)(=O)=O)CC)CC)=O)nn(C)nc1C 95010,c1(SC)c(C(N2CCC(NC(=O)Cc3cc[nH]c(=N)c3)C(C)C2)=O)cccc1F 95011,CC1CC(C(=O)NCC(F)C2CCC2)CCN1C(c1occ2c1CCC2)=O 95012,C1(CC(=O)N(CCO)CC2CCCCN2C(=O)CC2CCCC2)CCCOCC1 95013,C(=O)(CC(C(F)F)NC(C1OCCO1)=O)N(CC=C)CC 95014,C1(CC(=O)NC2CNCCC2O)CCC(F)(F)CO1 95015,C(N=c1nc2c(cnn2C(C)C)c(NC2CC3CC(O)C2C3)[nH]1)c1c(C)ocn1 95016,C(CC1c2ccccc2CCN1c1nc2ccc(F)cc2s1)NC(C(C)CF)=O 95017,C1(NC(c2cn(CC)nn2)=O)CN(C(C2C(F)(F)C23CCC3)=O)CCC1O 95018,CC(C)CC(CNC(=O)CCOCC(F)(F)F)NC(C1CC(=O)CCO1)=O 95019,Cn1cnc2c1C(C(=O)NCC=CCNC(=O)CCCn1ccnc1)CC(=O)N2 95020,c1(CCOC(c2sc(Br)c(Br)c2Br)=O)c(Cl)cccc1Cl 95021,C(C1=NOC2CN(C(=O)C3=CCSC3)CC12)NC(c1ccc(SC)cc1)=O 95022,C1(C(C)NC(=O)CC2CCCC2)CCN(C(=O)Cc2ccnc(F)c2)CC1 95023,O=C(CCCCCF)N1CCC(NC(c2ccnn2CC(F)(F)F)=O)C1C1CC1 95024,Cn1nc(C(=O)NC2(CO)CCN(C(C3CCC(OC)CC3)=O)C2)cc1C(F)F 95025,C(=O)(C1=C(C#N)CCC1)N1CC(C(C)(C)C)N(CC2(S(C)(=O)=O)CCCC2)CC1 95026,C1(C(=O)NCC(=C)CCNC(c2cnn(CC3CC3)c2)=O)(CC)CCC(C)(C)CC1 95027,CC1CN(C(=O)C=Cc2ccccc2)CCC1NC(C1SCCCS1)=O 95028,C(=O)(CC(O)C(C)(C)C)NCc1ccc(CNC(c2c(OC)nccc2)=O)cc1 95029,Cn1cnnc1CCC(=O)NCCn1cc(CO)nn1.c12ocnc1CC2.N 95030,CC1Oc2ccccc2N(CC(=O)N2CCN(c3ccc(Br)cc3)CC2)C1=O 95031,N1(C(C2(CC=C)CCCN2C(C2CC(C)=NO2)=O)=O)CCC2CN(C)CC2C1 95032,C(CCC(=O)NC(C1CCOC1)CNC(=O)CC(C)F)CCCC(=O)NOCC#C.O.CC.CCC 95033,CCC(CCC(=O)NCc1cccc(C#N)n1)NC(=O)CC1CCCN1C 95034,C(C)(C)(CC(F)C(=O)NC1COCC1CO)NC(C(C)=CC1CC1)=O 95035,Cc1cnc2c(CN3CC4CN(C(=O)Cc5cccnc5)C4C3)cnn2c1 95036,c1(C(=O)NC(CNC(c2cc(C)c(N)cn2)=O)C2CC2)ccc2sc(C)nc2c1 95037,C(CCCCC(=O)N1CCC(C(C)(C)CNC(C2C(=O)ON=C2C)=O)CC1)SC 95038,c1(OC)coc(C(N2CC(C)C(C)(CNC(=O)C(C(C)C)N(C)C)C2)=O)cc1=O 95039,c1(C(=O)NC23C(CN(C(C(C(C)C)O)=O)C2)CCC3)c[nH]c2nc(F)ccc12 95040,N1(C(c2ncn(C(C)(C)C)c2)=O)CC(NC(c2ocnc2C2CC2)=O)C(C(F)F)C1 95041,C#CCCCCC(=O)N1CCC(C(C)C(=O)N(C(C)C(=O)OC)C)CC1 95042,N1(C(CCOC(C)=O)=O)CCCC2(C1)CN(C(c1ncn3c1CCC3)=O)CCO2 95043,C1(C(N2C(CN(C)NC(c3cn(CC4CC4)nn3)=O)CCC2)=O)CC2CCC2C1 95044,c1(CC(=O)NCC(C)N(C)C(c2cc(CO)on2)=O)nc2ncccn2n1 95045,Cc1ncc(C(=O)N(C)CC2CCCCN2C(=O)C=CC(F)(F)F)n1C 95046,C(CNC(C1COCCO1)=O)(C(C)(C)C)NC(C(CC1CC1)NC(C)=O)=O 95047,C#CC1(NC(c2csc(CNC(C3CCSC(C)C3)=O)c2)=O)CCCCC1 95048,c1(OC)cc(C(C(=O)NCC(C)C)N(C2CCSC2)C)c(Br)cn1 95049,c1(C(N2C(CNC(c3n(C=C)ncc3)=O)C(C)CC2)=O)c(Cl)cc(C#N)cc1Cl 95050,C1(NC(CCC)=O)CCN(C(=O)C(C(=O)OC)OC(C)(C)C)C12CC2 95051,c1(C(N2CC(N(C(c3scc(C)c3C)=O)C)C2)=O)ccc2c(c1)CCC=C2 95052,CCC(O)C(C)C(=O)NC1CC(c2ccccc2)(NC(c2cc[nH]c(=N)c2)=O)C1 95053,C1(C2CCN(C(C3CCNC3=O)=O)CC2)(NC(C2=NOC(C)C2)=O)CC1 95054,n1(CC(=O)NCCOCCNC(=O)CC2CC(F)(F)C2)cnc(Br)c1 95055,c1(C(N2C(CC(=O)NC(c3ccccc3)C)CCC2C)=O)cc(CO)ccc1F 95056,Cc1ccccc1OCC(N1CCC(CN(C)CC2C3CCCC23)C1)=O 95057,c1(C(N(C)Cc2ccc(OC)c(OC)c2OC)=O)ccc2c(C)noc2c1 95058,Cc1ccc(C(N2C(C(=O)NCC3(C)CC(O)C3)CC2C)=O)cc1 95059,N1(C(C(C)C2CCC2)=O)CCC2C(C1)NC(=O)CN2C(=O)C(=O)N1CCCC1 95060,c1(CN(CCCOC)C2CC2)cc(C(=O)O)ccc1I 95061,c1(CO)cccc2c1CC(NCc1cn(-c3ccccc3)nc1-c1cccs1)C2 95062,C(CCCCCNC(=O)C(C1CC1)N(C)C)N(C(C(n1cc(Br)cn1)C)=O)C 95063,C1(c2c(OC)cccc2Cl)CCN1N1CC2CCC(O)CC2C1 95064,CC12CCC1CN(C(C1CCC(CNC(c3cc(Cl)n[nH]3)=O)C1)=O)C2 95065,C1(C(=O)NCC(C)(C2CCC2)NC(CCC=CC)=O)CCCC(OC)C1 95066,c1(C(=O)NC(C2CCCN2C(=O)COCCCF)C)cc(Cl)cc(Cl)c1 95067,c1(CC)cnc(Cl)[nH]c1=NCC1CCC(NC(=O)CCc2cc[nH]n2)C1 95068,C(=O)(C1=NN(c2ccccc2)C(=O)CC1)C(=O)Cn1cncn1.C1(N)CN(C=O)C1 95069,C(=O)(CC(F)(F)C(C)C)NC(C)CNC(=O)C=Cc1c[nH]nc1C1CCCCC1 95070,N1(C(c2ccc(OC)nc2)=O)CC2CC(NC(c3cc(C)nc(C)n3)=O)C(C2)C1 95071,c1(OC)cc(O)c(CNC2CC2C(=O)Nc2ccc(Br)nc2F)c(Br)c1 95072,N1(C(C=C(CCC)C)=O)CCC(NC(c2cnn3cc[nH]c23)=O)C12CCCC2 95073,CCC(C(C)(F)F)NC(=O)CN(C1CC(C#N)C1)C(c1cc(C)c(C)[nH]1)=O 95074,c1(OC)cc(C(N2CCCC2CNC(=O)C(C)C(C)C)=O)cc(Br)c1 95075,Cc1c(CN(c2ccc(Cn3cccn3)o2)CCn2ccnn2)cccc1Cl 95076,O=C(N=c1ccn(C2(CO)CCC2)[nH]1)C1CC1C1CN(C(=O)Cn2nccn2)C1 95077,c1(CNC(C(CC)C)c2nnnn2CC(F)F)ccc(F)c(F)c1C 95078,CC1(CNC(C2CC3CC2CO3)=O)CCN(C(c2cnc(C(N)=O)cn2)=O)C1 95079,C1(NC(c2coc(Cl)n2)=O)CCC2CCN(C(C3CCC(=O)N(C4CC4)C3)=O)C12 95080,c1(CC)nn(C)c(CC(=O)NC2CCN(C(=O)COC3CCC3)C2C(C)C)c1Cl 95081,n1(CC(=O)NCCC(C)N(C(c2c(C)n[nH]c2)=O)C)cc(Cl)c(O)nc1=O 95082,c1(CC(N2C(COC)CN(C(c3ccoc3C)=O)CC2)=O)cc2ccccc2o1 95083,N1(C(c2c(C)[nH]cc2)=O)CC(NC(c2cnns2)=O)C2CCCC12 95084,C1(C(=O)NC(CCCNC(Cc2c(C)scc2)=O)(C)C)CC2(CCOC2)C1 95085,C(=O)(CC(C)(O)CC(=O)O)NC1CCCN(C(c2ccc(C)cc2C(F)(F)F)=O)C1 95086,c1(CC)cc(C(=O)N(CC(C)NC(=O)C(F)(F)c2cncs2)C)cc(O)n1 95087,c1(C(NOCC(=O)OCC)=O)c(CNC(=O)Cn2nnc(C)n2)cnn1C 95088,Fc1ccc(C2(C(c3nnnn3C3CC3)Nc3cnn[nH]3)CCCCC2)cc1Cl 95089,c1(C(=O)NCC2CCN(C(=O)C3=CC4(CCOC4)C3)CC2)cccn2nccc12 95090,C(=O)(C1OCC(C)c2ccccc21)NCCN(C(c1cc(CCC)on1)=O)C 95091,N1(CCC(=O)N(C(CNC(C(C=C)(C)O)=O)C)C)Cc2ccccc2C1 95092,N1(C(C(C=C=C)C)=O)CC2N(C(C3CC(n4ccnc4)C3)=O)CCC2(C)C1 95093,C1(C(=O)NC2C3CC(NC(C4COCCO4)=O)CC32)CCCC12CCC2 95094,C1(C(=O)NCCC2(NC(C=Cc3ccc(C)o3)=O)CCCC2)CCCC(C#N)C1 95095,N1(C(c2cc(C)c(C)nn2)=O)CC(C)CN(C(c2ccn(C)c(=O)c2)=O)C(C)C1 95096,C1(NC(C(C)N(CC)CC)=O)CC(O)CN(C(=O)CCS(=O)(=O)NC)C1 95097,N1(C(Cc2c(C)cc(C)s2)=O)CCN(C(C2(C)CCCNC2=O)=O)CC12CCC2 95098,CCCC(C)(O)C(=O)N1C2CCC1C(NC(c1ccccc1OCCF)=O)C2 95099,C(=O)(C1CCCn2ncnc21)N(C(CNC(c1cccc(C)c1O)=O)C)C 95100,C(=O)(C1=CCCCC1P(C)(C)=O)N1C(C(O)CCn2cc(C(C)=O)nn2)CCC1 95101,N1(N2CC(C#C)(NC(C3CC4OC3C3CC43)=O)C2)CC2CC(C)C2C1 95102,C#Cc1ccc(C(=O)NCC(C2CC2)NC(c2ccc(C(C)(F)F)nc2)=O)cc1 95103,Cc1cc(C(=O)NC2C=CCC(C(=O)N(C3CCSC3)C)C2)ncc1F 95104,C1(C(=O)OCC(C(C)C)(C)C)Sc2ccccc2NC1=O 95105,C1(COC)(NC(C2CCCCS2)=O)CCCN(C(c2cc(Cl)no2)=O)C1 95106,Cc1cc(C#N)cc(C)c1C(=O)NC(CNC(=O)C=Cc1cncn1C)C1CC1 95107,CCCCCC(O)C(=O)N1CC(COC)(NC(C2(C)CC(C)=NO2)=O)C1 95108,CC1=C(C)CC(C(=O)NC(C)(CNC(c2sc(C3CC3)nc2C)=O)C2CC2)CC1 95109,C1(C(=O)NC2(CCNC(Cc3ccc(C)cc3)=O)CCC2)CCC=CCCC1 95110,c1(CC)ccc(CSCC(=O)Nc2cncc(C)n2)c(Br)c1 95111,N1(C(C2(C)CCN(S(=O)(=O)C3CC3)CC2)=O)CCC2(CCNC(=O)O2)CC1 95112,O=C1CCCCC(C(=O)NC2CC3CCC2(C(=O)NC2CCC(OCF)CC2)C3)C1 95113,CCC(O)C(F)(F)C(=O)NCc1cc[nH]c1C(=O)NC(C)CCO 95114,C1(c2nnc(C3(C#C)COC3)o2)CC(F)(F)CN1CC 95115,C1(COCCCCCC)(C(F)F)CCN(C(C2(Cl)CC2)=O)C1.C1(C)C(=O)N1CC 95116,C12(C(N(CCCNC(c3cc(Cl)ns3)=O)CCO)=O)COCC1C2(F)F 95117,C12(NCc3ccc(CCCCC)cc3)CCC(CO)(CC1)OC2 95118,c1(C(N2CCC(C(=O)NC3CC(C)C3)C(O)C2)=O)ccc(C#N)c(F)c1 95119,c1(CCC(=O)NC2C(NC(C3(C)CCCO3)=O)C2)ccc(O)nc1 95120,N1(C(C2COCCN2C)=O)CCC2CC1C(=O)N2C.C12(CC)CN(C1)C2=O 95121,Cc1ccc(C#N)cc1C(N1CCC(NC(C2(C)CC(C)(C)C2)=O)C(C)C1)=O 95122,N1(C(C=C(COC)C)=O)CC(N(C)C(c2ccc(CF)cc2)=O)C(C)(C)C1 95123,C(=O)(CC(C)(C)C(C)(F)F)NC(CNC(C1(C)CCN(C)C1)=O)(C)C 95124,C(C(C(=O)NC1CC1)NC(c1nocc1C)=O)OC 95125,N1(C(C(C)(C)O)=O)Cc2ccccc2CC1CNC(=O)Cc1c[nH]nc1O 95126,CCCCCC(C)(C)CNC(c1sc(-c2ccc(OC)cc2)nc1C)=O 95127,c1(C(N2CCC(CN(C(CC(=O)OCC)=O)C)C2)=O)cnc2occc2c1 95128,N1(C(c2ccsn2)=O)CCc2sc(CNC(C3(c4cc[nH]n4)CC3)=O)nc2C1 95129,CCCCC(O)C(=O)NCCN(C(c1ccc(CF)cc1)=O)C1CC1 95130,CN1CCCC(CCNC(=O)CC2CCCC(NC(=O)Cc3ccsc3)C2)C1 95131,C(=O)(CC(C(C)(C)C)NC(=O)CC1=CCCCC1)NCc1c(C)noc1 95132,c1(C(N2CC(NC(CC(n3ccc(C)n3)C)=O)C2)=O)n[nH]c2c1CN(C)CC2 95133,c12cccnc1S2.C#CCCC(=O)N(CCCN(C(=O)CC1CCC(=O)N1)C)C 95134,n1(CCC)cc(C(N2CC(C(C)NC(C3(CC)CCOC3)=O)C2)=O)nn1 95135,C12CC3CC1CC3C(=O)N2.N1(C(C2C=CC(N(C)C)C2)=O)CCOC(C(=O)NC)C1 95136,C1(C)(CC)CC(NC(C2CC(F)(CO)C2)=O)CN1C(c1cnc(C2CC2)s1)=O 95137,C1(OC)(CNC(c2ccc(Cl)cc2)=O)CCN(C(=O)CCC2CCCN2C)C1 95138,N(S(=O)(=O)N1Cc2ccccc2C1)C(C(c1ccccc1)N(CCC)CC)=O 95139,c1(C(N2CC3CCN(C(C4CC(N(C)C)C4)=O)C3C2)=O)cnc2c(c1)nnn2C 95140,N1(C(c2c(C)nsc2)=O)CCN(C(=O)C#CC(C)(C)O)C(CC(F)F)C1 95141,S(=O)(=O)(c1cc(Br)c2ccccn12)NC(c1ccc(F)c(F)c1)(C)C 95142,N#CC1CCC(NC(C2CSCCN2C(c2cc(C(N)=O)co2)=O)=O)CC1 95143,C1(NC(c2ccc3c(c2)CCO3)=O)CCC2CN(C(c3cnns3)=O)CCC2C1 95144,C1(CNC(c2n(CC)ncn2)Cc2cccc(Cl)n2)CC12CCC(F)(F)CC2 95145,N1(C(C)=O)C(C)CN(C(=O)CCn2cnc(C)cc2=O)CC1C 95146,c1(NCCCC(=O)OCC)ncnc(Cl)c1C#N 95147,c1(OCC)ccc(-c2cc(CNCc3c(C)cccc3O)ccn2)cc1NC 95148,c1(C(C(=O)NCCSC)N(C(C)C)Cc2cncs2)cccc(C(F)(F)F)c1 95149,Cc1cccc(C(=O)NC2(C)CC(NC(=O)C(C3CC(F)(F)C3)O)C2)c1 95150,C1(CNC(c2n(C)cnc2)=O)CN(C(=O)CC2CC(n3cnnc3)C2)CC12CCC2 95151,N1(C(C2(OC)CC2)=O)CC2ON=C(CNC(c3cnn4c(C)ccnc34)=O)C2C1 95152,c1(C(=O)NCCC(=O)NCCCOCCCC)cncn(C)c1=O.C(C)(=O)O 95153,c1(CC(=O)NCCC(C)N(C(C(COC)C)=O)C)c(C)cccc1F 95154,N(C1CCC(NC(=O)Cc2cccs2)c2ccccc21)C(CC=C(C)C)=O 95155,N1(CC(=O)O)CCN(c2ccccc2)CC1C.CCC(CSC)(CC)O 95156,c1(NCC2CCC(O)C2)nccc(N2CCOC(c3cccnc3)C2)n1 95157,N1(CC(=O)NCC2CN(C(C(OC)OC)=O)C(C)CC2)C(=O)CC(C)(C)C1=O 95158,c1(CC)cc(NC(c2cccc(OCCO)n2)=O)sc1C(=O)NC 95159,N1(C(CNC(=O)OCC)=O)CCOCC(C)(CNC(=O)C(C)C2CCCO2)C1 95160,C1(CC(N2CCCC(CNC(c3nncs3)=O)C2)=O)CC(c2ccccc2)=NO1 95161,C=CCC(C)(C)C(=O)NC.c1(C(=O)NC(C2(OC)CCC2)C)cnc(CC)s1 95162,CCC(C(=O)NCC(C)NC(c1ccc2nccn2c1)=O)C(C)(F)F 95163,c1(CC(N2CC(OCCC(=O)NC3C(OC)C(O)C3)C2)=O)cncnc1O 95164,c1(CN(C(=O)CCCC2CCCC2)C(C)C)cncc(C(=O)OC2CCCOC2)c1 95165,C1(C(=O)Nc2cccc(C3(C)CC(=O)C3)c2)CC2CCCCN2C1=O 95166,C(C1=CCN(C(=O)C=Cc2cn(C)cn2)CC1)N(CC)CC.C1=CCNC1=O 95167,c1(OC)ccccc1-c1cnc(NC(c2ccc(C#N)s2)=O)nc1.C1C(=O)N1 95168,C(=O)(C(F)(F)c1ccccn1)NCCCCN(C)C(C1CC1C(F)(F)F)=O 95169,CCCC(C)CC(=O)N1CC(NC(c2ccnc(Cl)c2O)=O)C(C)C1 95170,Nc1ccccc1-c1cn(CCCC(=O)NCc2csc(O)n2)nn1 95171,c1(C2(C(=O)NC(C)CN(C(=O)CCSCC(N)=O)C)CCCC2)cccc(Cl)c1 95172,C(CCSC)(C(=O)NC(c1ccccc1)CCO)OC 95173,c1(OC)cc(N2CCCC(NC34CC(C3)N(C(=O)COC(C)(C)C)C4)C2)ncn1 95174,O=S(=O)(c1ccc(NCCC2CCCOC2)cc1Br)NCC1CC12CC2 95175,N1(C(c2cnc(F)c(CO)c2)=O)CCc2c(O)ncnc2C1 95176,c1(C(C(=O)Nc2ccccc2Cl)N(CCOCC#C)CC)ccc(F)c(OC)c1 95177,C1(C(=O)NC(C=C)(C)C(=O)OC)C2Cc3ccccc3C12 95178,C1(CN(C(C(=O)NCC=C)C2CC2(C)C)CCN(C)C)CCCCO1 95179,C1(C(=O)NC(C2CCCN2C(=O)CCc2cccc(O)c2)C)OCCN(C)C1=O 95180,N1(C(C(=O)NCc2cccc(OC)c2)C(C2CCC2)OC)CCCCC(C)C1 95181,c1(OCC(c2nc(CCC)nn2-c2ccc(C#N)cc2)C)cc(C)cc(C)c1 95182,CCC(CC(=O)N1CCC(C2CC2)(CNC(c2cnsc2)=O)C1)C(F)F 95183,Cc1ncc2n1CCC(C(N1CC(C)(C)OCC1CNC(=O)C(C)(C)C#N)=O)C2 95184,C1(CC(N2CC(N(C(CN(C3CCC3)C)=O)C)OCC2)=O)OCCCC1(C)C 95185,N1(C(C2(C)CCN(C(CCC(C)C#N)=O)C2)=O)CCN(C)C(=O)C1C 95186,c1(C(N2CCCC(C(C)NC(CCC(=O)OCC)=O)C2)=O)nnn2c1CCCC2 95187,C(=O)(C(O)CC(N)=O)NC(C(=O)NC(C)Cn1cncn1)CCC1CCC1 95188,Cc1cc(C)c(C(N2CCCCC2C(=O)NC(c2nnc(O)o2)C)=O)s1 95189,Cc1nc(N2CCOCC2)ccc1NC(=O)NC(C1CC=CCC1)C(=O)O 95190,CC(CCN=c1nc(-c2ccccc2)[nH]s1)NC(C1CC=CCO1)=O 95191,N1(C(c2ccc(CSCCC)o2)=O)CCCC2C1CCN2C(C1CC1C#N)=O 95192,Cc1cn2ccc(C(=O)NCC(C)(C(C)C)NC(c3cnnc(O)c3)=O)cc2n1 95193,C1(C(=O)NC(C)CN(C)C(c2n[nH]cc2C(F)(F)F)=O)CCc2nncn2C1 95194,N1(C(C(C)OC)=O)CC2C(C(=O)NC3CC(C(C)(C)C)C3)C2C1 95195,N1(C(Cc2ccc(OC)c(Cl)c2)=O)CC2(CCC2)CCC1C 95196,c1(C(N2C(CCNC(CC(C)OC)=O)CSCC2)=O)c(F)cc(OC)cc1F 95197,c1(C(C)C)ncc(C(N2CC(NC(c3cccn3C)=O)C3CC23)=O)n1C 95198,c1(Cn2cc(CSC(C)C)nn2)cccc(OC)n1.C12(C(=O)OC)CC(CC)(CO1)C2 95199,C12(C(N(CC(CO)(CO)NC(=O)CC3OCCO3)C)=O)CC1CCC2(F)F 95200,C1(CC(=O)N(CCNC(C(CC)=CCCC)=O)CCOCC)CCCC2(CCC2)O1 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95219,C1(CNC(c2c(CC)occ2C)=O)CC(C)(C)CCC1NC(=O)CC(C)(C)N(C)C 95220,C1(CNC(COc2cc(C)on2)=O)CN(c2nc(C)nc(C)c2C)CCC1(F)F 95221,CC1(CNC(C2CN3CCN2CC3)=O)CCN(C(c2cccs2)=O)CC1 95222,c1(OC2CCN(C(C3CCOC3)C)C2)ccccc1F.C(CN(C)C)O 95223,Cc1cnc2nccc(C(=O)NCCNC(=O)C(C(C)C)n3cc(C)cn3)c2c1 95224,N1(c2nc(N3CCC(F)(CF)CC3)cc(C)n2)CCc2c(C)nccc2C1 95225,c1(C(=O)NC23C(CN(C(C(C)C4CCCC4)=O)C2)C3)cccc2ccn(C)c12 95226,C(=O)(C(C)CC(F)(F)F)N1CCC(NC(C(C)=C(CC)C)=O)C(CC)C1 95227,c1(C(=O)NCC2(NC(C(C3CCC3)OC)=O)CCC2)c(C)ccc(Cl)c1O 95228,N1(C(C(=O)NCc2scc(C(=O)OCC)n2)C2CCC2C(F)(F)F)CC(C)C(C)C1 95229,N1(C(CCSc2n(C)nnn2)=O)CCN(C(=O)C=CCN(C)C)CC12CCC2 95230,C1(C(N2CC(C)(CCC(N3CC(N(CC=C)C)C3)=O)C2)=O)CCCCNC1=O 95231,Nc1cc(C(=O)NC2CCN(C(C3CC(=O)N3)=O)C2)cnc1N 95232,CC1CCC(O)(C(=O)NCC2CC(C(=O)NCc3ncn(C(C)C)n3)=NO2)CC1 95233,c1(C(=O)NCC2N(C(c3n(CC)ncn3)=O)CC2)n[nH]c2c1CC(C)CC2 95234,C1(CNC(C2CCCN(C)C2)=O)CN(C(=O)CNS(C)(=O)=O)CCC12CCC2 95235,C1(C2(NC(C3CC3F)=O)CC2)CCCCN1C(c1ccccc1O)=O 95236,c1(C(=O)NC(C(C)NC(C(C=C)(C)C)=O)C(C)C)c[nH]c(=N)nc1CC 95237,c1(OC)cnc(C=O)c(F)c1.C1(=O)C(C)(C)C(=O)N2CCC3C(C23)N1.OC 95238,C1(C(N2C(C(=O)N(C3CC3)CC3CCOC3)CCC2)=O)C2(CC2)C12CC2 95239,C1(c2nnc(N3CCC(OC)C3)n2-c2ccccc2)CC2CCCCN2C1 95240,C(CCCC(C)(C)OC)NC(CC1(C=C)CN(C(=O)OCC)C1)=O.C(C)(C)C 95241,Cc1nc(O)ccc1C(N1CCC(CCNC(=O)CC2(C(F)F)CC2)C1)=O 95242,C1(COCC(=O)NCC2(N(C)CC3CCCCO3)CC2)CCn2nccc2C1.COC 95243,C=CC1COCCN1C(C1(NC(=O)CCC(C)CN(C)C)CCSC1)=O 95244,N=c1[nH]nc(CCCC(=O)NCCC(O)CNC(C2C=CCC2)=O)s1 95245,c1(C(=O)NCCCNC(C(C(CC)O)C)=O)ccc2sccc2c1 95246,N1(C(c2cc3c[nH]cnc-3n2)=O)CCC2C1CCCN2C(C1CCC(O)CC1)=O 95247,N1(C(=O)Cc2ccc(F)c(F)c2)CC2(CCC(C(N3CCC(CO)C3)=O)O2)C1 95248,CCCCCC=O.C1(C(=O)OC)CCNC1C(C)(C)C 95249,CN1CCC(C(=O)NC2(CNC(c3cc(C(F)(F)F)ns3)=O)CCOC2)C1=O 95250,C1(C(=O)NCCCCCCNC(c2cn3ccnc3s2)=O)COC2(CO)CC1C2 95251,c12ccc(cc1)[nH]c2=O.N1(C(CSCCC)=O)CCCC1COC(C)CC 95252,C(=O)(C1CCc2ccccc21)N1C(C(=O)NCc2c(C)ocn2)C(C)CC1 95253,C(=O)(CC1CCc2ccccc21)N1CC2(C(CO)CN(C(C3C(=C)CC3)=O)C2)C1 95254,Cc1c(C(=O)NCCC2CCCN(C(=O)CC(C)CN(C)C)C2)ccn1C(C)C 95255,C1(NC(C2COC2)=O)CC(CNC(=O)C(c2cccc(F)c2F)(F)F)C12CCC2 95256,CCCC(C)CC(=O)N1CCC(NC(C2(c3ccc(OC)c(OC)c3)CC2)=O)C1 95257,C1(NC(C2(COC)CCOCC2)=O)CC2CCC1CC2NC(=O)CCF 95258,C1(OC)CC2CC1CN(C(C13C4CC(CC14)C3(F)F)=O)C2.O=C1CC2=NN(C2=O)C1 95259,C1(NC(CC2(OC)CCC2)=O)CCC(C(N2CC(C(C)NC)C2)=O)CC1 95260,CC1CC(C(=O)NCCOC2CCN(C(c3ccc(O)nn3)=O)CC2)C1(C)C 95261,CC1=CCC(C(=O)NC2CC(F)CC2NC2CC2C(=O)OC(C)(C)C)C(C)CC1 95262,C12(CNC(CNC(CCC(C)C)=O)=O)CCC(CC1)N(C(C1(C)CC1(F)Cl)=O)C2 95263,C1(NC(COCCSC)=O)CCN(C(C2COC3(CCC3)CO2)=O)CC(C)(C)C1 95264,C1(C(N(C(CC)C(=O)N2CCC(SC)C2)C)=O)CCCN(C(C)=O)C1 95265,C1(N(CCC)C(C2CC(C)C2)=O)CCN(C(=O)COC)C1 95266,C1(CNC(=NCC)NC2C(C)(C)C2(C)C)CCCC2CCCCC12 95267,C1(NC(C=CCN(CC)CC)=O)CC(O)CN(C(c2cnc(-c3ccsc3)s2)=O)C1 95268,C(=O)(C1=NN(C)C(=O)CC1)N1C(C)CN(C(c2ncoc2-c2cccs2)=O)CC1 95269,c1(C(=O)OC)cc(OC)cc(C(=O)NC2CC(NC(C3(C)CC(C#N)C3)=O)C2)n1 95270,C1(CNC(COC)=O)CC2(CO1)CN(C(c1cc3scnc3[nH]1)=O)C2 95271,C12(NC(c3ccc(=N)[nH]c3)=O)COCCC1CN(C(C1(CF)CCOCC1)=O)C2 95272,N1(C(c2c(CC)scn2)=O)CCCC(N(C(=O)C=CC(C)C)CCO)C1 95273,Nc1ccc(C(=O)N(CC(F)(F)F)Cc2cccnc2)c(F)c1F 95274,C1(CNC(CSCCCC)=O)CC(F)CN1C(=O)COCC(C)C 95275,C1(=O)CCCC(C)(C)N1.C(C(C)(O)C1CC1)N(C(=O)Cc1nc[nH]n1)C 95276,N1(C(CC(C)SC)=O)CC2CCOC2(CNC(=O)CSc2cn[nH]c2)C1 95277,C(CCCCCNC(C1CCCN1CCC(C)C)=O)N(C(c1c(C)con1)=O)C 95278,c1(C(=O)NCCC(C)NC(c2coc(C(F)F)c2)=O)cn2ccnc2s1 95279,N1(C(Cc2c(C)scc2)=O)CCOCC(CNC(C2CC(OC(C)(C)C)C2)=O)C1 95280,N1(c2ccc(C#N)nn2)CCCCC(NC(c2cccc(C(N)=O)c2)=O)CC1 95281,C(C(CC(F)(F)F)NC(C1CCCOC1)=O)NC(=O)CCc1ncc[nH]1 95282,C(=O)(C1=NNC(=O)C1)N(CC1CC(NC(c2cc(N(C)C)ncc2)=O)C1)CCO 95283,c1(CC)cnc(O)c(NC(c2c(NC(=O)C(C)C(C)(C)C)cccc2F)=O)c1 95284,C(=O)(C1=NOC(C(N2CCC(CNC(=O)CC3CC3)C(O)C2)=O)C1)OC 95285,C1(C(=O)NC(C(=O)NC(C(C)SC)C)CC2CC2)CCCCC(=O)N1 95286,N1(C(C(C)NC(C(C)SC)=O)=O)CCOC(n2cc(C(C)(C)C)nn2)C1 95287,c1(C(=O)NC(CC)CNC(c2c[nH]nc2NC)=O)cc(S(=O)(=O)NCCO)c[nH]1 95288,c1(C(N(CCCNC(CCCCOC)=O)C)=O)cccc(C2CC2)c1Cl 95289,Cc1cc(C(N2CC(NC(C3(Cc4nccs4)CC3)=O)CC(F)C2)=O)ccc1I 95290,c1(C(=O)NCCN(C(=O)CCc2cc(C)nc(C)c2)CC)cnn2ccn(C)c12 95291,C1(NC(c2c(CC)ocn2)=O)CCCC(NC(=O)CCN2CCC(O)CC2)CC1 95292,n1(CC(=O)N2CC(=O)NCC2)cc(C2CC2)nn1.C1(SCC)CCC=CO1 95293,CCCS(=O)(=O)C(C)C(=O)NCCCCNC(=O)CC1CCCC(=O)N1 95294,CCC(C(=O)N1CC(N(C(=O)Cc2ccc(Cl)nc2C)C)C2(CC2)C1)C(F)(F)F 95295,c1(C(N(CC(C)C#N)C)=O)ncccc1CNC(=O)C(C1CCC(=O)N1)C 95296,c1(NC(c2n(C(CC)(C)C)nnn2)C2CC2)cc(CSC)cc(C)c1 95297,c1(NC(=O)NCC(=O)NCC(CC=C)NC(c2ccccc2)=O)cc(O)nn1C 95298,n1(-c2n(C)ncn2)nc(C2CC(=C3CC3)C2)nc1-c1ccc(CS(C)(=O)=O)cc1 95299,c1(CC)ccc(C(=O)NC2CCCCC2CNC(=O)C=Cc2cn(C)nn2)cn1 95300,c1(NC(=O)CC2CCN(CCCO)C2)cccc(CNC(c2ccncc2)=O)c1 95301,C1(C(=O)NC2C(CN(C)C)CCC2)CCOCC1NC(=O)CCn1cccn1 95302,Cc1cc(N)ccc1C(N1CC(CCO)(NC(=O)CC2CC3C=CC2CC3)C1)=O 95303,C1(C(=O)NCC(C)(C)CCO)CC2(CCN1C(c1ccn3nccc3c1)=O)CC2 95304,c1(NC(N(CC(CC)(O)CC)C)=O)cccc(Cl)c1OC(C)C 95305,C(=O)(C1CCCc2nn[nH]c21)NC1C(NC(=O)COc2cccnc2)CCCC1 95306,Cc1ccc(C)c(C(N2CCC2C(=O)N(C)CC2CC2)=O)c1 95307,N1(C(CCOCCC)=O)CC(OC)CC1NC(=O)CSCc1ncc[nH]1 95308,C1(C(N2CCC(N(C)C(C3CC3c3cncn3C)=O)C2)=O)CCCCC1(C)C 95309,C=CCCCCCCNC(C12CC1CN(C(=O)CCC(C)CN(C)C)C2)=O 95310,N1(C(C=CC)=O)CCCC(C)(C)C1CNC(c1cc(S(C)(=O)=O)co1)=O 95311,C(=O)(CC(C)C=C)NC(C(=O)NCC(=O)OCC#C)CC1CCC1 95312,CCCCC(C(=O)N(C1CCCC1)CCNC(=O)Cc1ccc(Cl)cc1C)C(C)C 95313,C1(CCCCNC(CC2N(C(C)C)CCC2)=O)CCN(C(=O)CC(C)N(C)C)CC1 95314,N1(C(c2cc(C)n(C)c2)=O)CCC(NC(=O)CCCC(=O)N(C)C)C(F)(F)CC1 95315,CC(C)(C)C(CO)C(=O)N1CCC1CNC(C1CCCN1C(=O)OC)=O 95316,c1(NC(C2C(C)(CC)C2)=O)cccc(NC(C23CC(CO)(C2)OC3C)=O)c1 95317,N1(C(COCC(C)C)=O)CCN(C(=O)CCC2CCCN(C)C2)C(CC(C)(C)C)C1 95318,N1(C(C(C(C)(C)C)=O)=O)C2CCC1CC(CNC(C1(Cc3ccsc3)CC1)=O)C2 95319,C1(c2nc(COCCS(Oc3ccc(C)s3)(=O)=O)no2)CC(=O)CC(=O)N1 95320,C(=O)(C(F)(F)C(F)(F)C(=O)O)NC1C2CN(C(C(CN(C(C)C)C)(C)C)=O)C(C2)C1 95321,c1(C(=O)NC23CCN(C(c4cccc(C)n4)=O)CC2C3)cnc2ccnn2c1C 95322,N12CCCC1(C(C)C)C(=O)N(C1CC1)c1cscc1C2=O.C1(CC)CCOC1 95323,C1(C)(C(=O)NCC(CC)NC(=O)CC2CC2(C)C)CCCCNC1=O 95324,C1(C(=O)NCCCOC(=O)NC)CCOCC1NC(c1n[nH]c(C)c1O)=O 95325,Cc1noc(CSCC(=O)NCCCC2CCCN2C(=O)CC2(CO)CC2)n1 95326,N1(C(CCN(CC#C)C(C2CC(O)(C#C)C2)=O)=O)CCOC2C(O)CC12 95327,C1(C(N)=O)CN(C(=O)CCF)CCC1NC(c1ccccc1-n1cccc1)=O 95328,c1(C(=O)NCC(C)(C2CC2)NC(C(C2CC2)OC)=O)ccccc1C#CC1CC1 95329,C1(C(N2C(C(=O)NCCCc3cn[nH]c3)C=CC2)=O)C2CCC(F)C12 95330,c1(CNC(CC2CN(c3ncc(CC)cn3)C2)=O)cc(C(=O)O)ccc1F 95331,C1(C(=O)NCCOCCC=C)CSCN1C(=O)CCc1ccnn1C 95332,CCCC(C)CC(C(=O)NCCCF)N1CCC1(C)CCO 95333,c1(C(N2CC(C)(NC(C3CC(C)N(C)CC3)=O)C2)=O)ccc2ccncc2c1 95334,C(CC(C(C)(C)C)NC(c1cnn(C)n1)=O)N(C)C(C12CCCN1CCC2)=O 95335,Cc1cccc(CC(C2CC2)NC(c2cc(C3CC3)n(C)n2)=O)c1 95336,C1(NC(C(CC)C(=O)OC)=O)CC(C(=O)N2CCCOC(CCO)C2)=CC1O 95337,C1(C(N(C(C)C(N2CCC(C(=O)OC)C2)=O)CC)=O)CCCSC1C 95338,CCC(C)CCC(=O)NCC1(NC(C2CC23CCOCC3)=O)CCOCC1 95339,CC(F)(C(=O)N1C2CCC1CC(CNC(=O)C(F)(F)c1nccs1)C2)C(F)(F)F 95340,N1(C(C(CC)C)=O)CC2=C(C1)CN(C(=O)C(=CC1CCCC1)C)C2 95341,C1(Cn2cc(C(C)NC(c3ccc([N+](=O)[O-])o3)=O)nn2)CC2(CCC2)C(=O)O1 95342,c1(CC(N2C(C)CCC(CC)C2)=O)sc2ccccc2c1C 95343,C1(N(C2CN(C(=O)OC(C)(C)C)C2)CC(F)F)C2CCC(=O)C12 95344,C#CC(CC(C)(C)C)NC(=O)C(CC=C)NC(=O)Cc1cc(C)on1 95345,c1(C(=O)NC2CC(NC(C3CCCC(C(=O)OC)C3)=O)C2)cc(O)nc(N(C)C)n1 95346,c1(C(=O)NCC2(C)CCN(C(C(C3CCC3)OC)=O)C2)ccc(Cl)cc1F 95347,C1(CC(=O)OC)(C(=O)OC)CCN(C(C2CCC(n3ccnn3)CC2)=O)C1 95348,C1(NC(C(C)Cn2ccnc2)=O)CC2(C1)CC(C(=O)NC1CN(C3CCC3)C1)C2 95349,C1(CCC(=O)N(CCC(C)NC(=O)CCn2ccccc2=O)C)CC2(CC2)CO1 95350,C1(C(N2CCC(CNC(CCC(C)C)=O)CC2)=O)CCCC1S(C)(=O)=O 95351,C=CCC(CC(C)C)C(=O)NC1CCC1CNC(=O)CN1CCCOC1=O 95352,N1(C(CC(C)CN(C)C)=O)CC(CNC(c2ccc(CO)cc2)=O)OC(C)(C)C1 95353,CC1(C)CN(C(c2cccc(C(F)F)n2)=O)C(CNC(=O)CCCC(F)F)CO1 95354,C(=O)(CCCc1ccccn1)NC(CCN(C(C(C1CCC1)OCC)=O)C)C 95355,CC1c2ncc(C(=O)NC3C4COCC34)n2CCN1C(c1cnon1)=O 95356,Cc1cc(C(=O)NC2CCCC2NC(=O)Cc2cnsc2)cn1C(C)C 95357,c1(C(N2CCC(C(C)NC(COCCC#C)=O)CC2)=O)cnc2c(ccn2C)c1 95358,C=C=CC(C)C(=O)NC1(C2CCCCN2C(=O)C=Cc2ccncc2)CC1 95359,N1(C(c2c(C)c[nH]c2)=O)CCC2(C(=O)Nc3nc(Br)ccc3C(N)=O)CC2C1 95360,c1(C(=O)NC2CC(NC(CN=S(C)(C)=O)=O)CC2O)cncc2nc(O)[nH]c12 95361,N1(C(c2scc(CNC(C3C(C)CCO3)=O)c2)=O)CCC(F)(F)C1 95362,C(C(F)(F)CCC(=O)NCCc1ccncn1)n1cc(C2C(C(=O)OC)C2)nn1 95363,N1(C(c2c(CC)c[nH]n2)=O)CCC2CN(C(c3ccc4cnoc4c3)=O)C2C1 95364,c1(OCC)cc(C(=O)NCCN(C(=O)C=CC=C(Cl)Cl)CC2CC2Cl)ccc1F 95365,Cc1nc2cc(CC(=O)NCCN(C(=O)CC(C)CC(C)(C)C)C)ccc2o1 95366,CC(=O)CCCCC(=O)N(CC(C)O)CCNC(=O)C(C)CC=Cc1ccccc1 95367,C12(C(N3C(CNC(CCC4(C)N=N4)=O)CC3)=O)CC(C)(C1)OC2C 95368,N1(C(c2c(OC)csc2)=O)CCC(NC(=O)C(C)P(C)(C)=O)C2(CCC2)C1 95369,Cc1cc2cc(-c3cccc(C(F)F)c3)[nH]c2cc1Cl 95370,C1(C(=O)NCc2nnc(C(F)F)s2)CC2(CC2)CN1C(=O)Cc1ccsc1 95371,C(CCC(C)CC(=O)NC1CCN(C(C2CCN2S(C)(=O)=O)=O)CC1)=C(C)C 95372,C#CC1CCCC(NC(=O)CCN(CCO)C(C2CCCC(NC)CC2)=O)C1 95373,c1(N(C(C2CN(C(=O)COC(F)(F)F)C2)=O)C2CC2)cccnc1 95374,c1(C(=O)NCC=CCNC(c2ccn(CC)n2)=O)ccnc2[nH]ncc12 95375,N1(C(C(C(=O)OC)C)=O)CCN(C(=O)CC2CC(C)(C)C2)C(C2CC2)C1 95376,C1(C(=O)Nc2cncc(CC)c2)CCOCCN1C(C1CCCN1C1CC1)=O 95377,N1(C(C(CC(C)C)NC(c2ccc(CC)cc2)=O)=O)CCC2(CNC(=O)O2)C1 95378,c1(NC(C2CCCN(Cc3ccc(F)cn3)CC2)=O)cnc(Br)c(Br)c1 95379,c1(C(=O)NCC(N2CC3C(NC(C4N(C(C)=O)CC4)=O)C3C2)=O)cc(C)ccc1C 95380,C1(C(N(C)CC2(NC(C(CC)CC(F)F)=O)CC2)=O)CC12CCS(=O)(=O)CC2 95381,N1(C(CC2C(C)=NOC2=O)=O)CC(NC(=O)CC2CSCCO2)CC(O)C1 95382,S(=O)(=O)(c1ccc(NC(C)C)nc1)NCC(=O)N(CC(C)C#N)CC 95383,c1(C(N2CCC(OCCNC(C3C(=C)C3)=O)C2)=O)c(F)ccc(O)c1F 95384,c1(C(=O)NCC(CCOC)NC(c2cccnc2C)=O)cc(C(C)(C)C)n(C)n1 95385,c1(C(=O)NCCC2OCCN(C(CCC(N)=O)=O)C2)cc(O)cnc1Cl 95386,c1(C(=O)NCCCCCNC(c2ccn(CC)n2)=O)cnn2cc(OC)ccc12 95387,C1(CN(C(C=CC(=O)NC(C)C)=O)C)CN(C(C2CC2CF)=O)CCO1 95388,C1(C(=O)NCC(C2CCOC2)NC(CCOC(C)=O)=O)CC2CCC2C1 95389,c1(SCC#N)ccc(NC(C2C3CN(C(c4cnoc4C4CC4)=O)CC23)=O)cc1 95390,c1(C(N(CC(=O)N(CC(CC)(F)F)C)C2CCC2)=O)cc(C)nc(O)c1 95391,c1(OCC)nccc(=NC(=O)c2ncc(-c3c[nH]c4ncccc34)cn2)[nH]1 95392,C(CC(C)(C)C)(C(=O)NC1CN(C(=O)CCOCC(F)F)C1)OC 95393,c1(C(=O)NC2(CC)CCN(C(C3(Br)CC3)=O)CC2)ccc2scnc2c1 95394,C(=O)(C(C(C)C)C(C)C)NC1CCN(C(C(C)OCCCC)=O)C1(C)C 95395,c1(C(N(C(C)CNC(=O)CC2CC23CC3)C)=O)cc2c(cc1Cl)NC(=O)C2 95396,C1(C#N)(C(=O)NCC2C(CNC(Cc3c(CC)con3)=O)C2)CCCOC1 95397,C(C1CCN(C(=O)CC2CCCCO2)CC1)=CC(N1CC(O)(C(C)(C)C)C1)=O 95398,C=C(C)CC(C(=O)N(C)CC1CCC1)NC(c1cncc(C)n1)=O 95399,N#Cc1ccc(OCCOC)c([N+](=O)[O-])c1.c1(CN2CCNCC2)cccc(F)c1[N+](=O)[O-] 95400,N1(CC(N2CCCC(C)(N(C)C)C2)=O)CCc2ccccc2C1 95401,C1(C(=O)NC(c2ccc(F)cc2F)COC)COC(C)(C)CN1 95402,Cc1ccc2cc(C(N3CC(C)C(C)C3)C(=O)NC(C)C)ccc2n1 95403,C(=O)(C(C)(C)C(C)(C)C)N1CC2C(CNC(c3c(C)n(C(C)C)cc3)=O)(C2)C1 95404,c1(C(N(CCCN(C(C(CC)C(=O)OC)=O)C)C)=O)cccc2cc(F)ccc12 95405,c1(CC(=O)NC2CC(CNC(Cc3cc(C)[nH]n3)=O)C(O)C2)cc(Cl)ccc1Cl 95406,N1(C(C=CC(C)C)=O)CC2CCC(CNC(=O)Cc3cc(O)ncn3)(C2)C1 95407,CC1C=C(C(=O)NC2CN(C(C3(Sc4ccccc4F)CCCCC3)=O)C2)C1 95408,N(C(=NCCCCl)NC1CCCCC1)Cc1nnn(C)n1 95409,C1(C)(C(=O)NC2CC(NC(c3ccc(CNC(C)=O)s3)=O)C2)COCCO1 95410,N=C1NC(=O)C(CC(N2CC(CNC(=O)CC3(O)CCC3)C2)=O)S1 95411,CCC(F)(F)CC(=O)N1CC2C(CNC(c3ccc(C(N)=O)cn3)=O)C2C1 95412,C(=O)(C1c2c[nH]nc2CN1C(c1snc(C)c1N)=O)N(CC#C)CC1CC1 95413,CC1CC(NC(c2ccc(C#N)o2)=O)CCN1C(=O)CCc1cnccn1 95414,C1(CC)(CNC(=O)C=CCO)CCCN1C(c1sc(C)nc1-c1ccccc1)=O 95415,c1(C(N2C3(CNC(CSCCOC)=O)CC(C2)C3)=O)cc(OC)c(F)c(C)c1 95416,C#Cc1cccc(C(N2CCC(C(=O)Nc3c[nH]ccc3=O)C2C)=O)c1C 95417,C1(C)(C(=O)NCCC2(O)CN(C(C(C)c3cccs3)=O)C2)CCC(=O)N(C)C1 95418,Cc1cccc(C(N2CCCC2C2(NC(=O)Cc3cccc(Cl)c3)CC2)=O)c1N 95419,N1(C(c2cc(CC)no2)=O)CCCC2C(CCCN2C(=O)Cc2nnc(C)s2)C1 95420,C1(C(N(C(C#C)CC)C2CC2)=O)COCCC1NC(=O)CCCOC(C)(C)C 95421,N1(C(C2C(CC)C2)=O)CCCC(C(=O)NCCOCCSC)CC1 95422,c1(OC(C)(C)C)cnc(C(N2CCC(NC(c3coc(Br)n3)=O)C2)=O)cn1 95423,C1(CNC(CCN(CC(C(C)C)C)C)=O)C2CCC(C2)N1C(=O)Cc1ccncc1 95424,Cn1cnc(C(=O)NC2CC2CNC(C2(F)CCCCC2)=O)cc1=O 95425,c1(C(CNC(CC)=O)NC(=O)CCOC2CC(NC(C)=O)C2)ccc(F)cc1 95426,C#CCC(C)(C)C(=O)N1CCC1CC1=CCCN(C(C2CCC(COC)O2)=O)C1 95427,Fc1cc(N2CCCC2c2cccc(I)c2)cc(Br)c1 95428,C1(CNC(c2nn(C(F)F)cc2Cl)=O)CN(C(C2CCOC(C(F)F)C2)=O)CCO1 95429,Cc1nn(C(C)(C)C)cc1C(=O)NC1CCC(C)(CNC(=O)CC(F)(F)F)C1 95430,Cc1cc(=NC(=O)C(=O)N2CCCC2CCN=c2nc3[nH][nH]cc-3c(O)n2)[nH]o1 95431,c1(C(=O)NCC(c2ccccc2)CNC(C23CCC(C2)C3)=O)cccc(Cl)c1Cl 95432,C(=O)(C1=CC2C=CC1C2)NC1C2CC(C(=O)NCCC(C(=O)OC)C)C(C2)C1 95433,c1(C(N2CCC(Cc3cn(C(COC)COC)nn3)C2)=O)oc(C2CC2)nc1C 95434,c1(C(N2CC3C(NC(C4C(OC)CCC4)=O)C3C2)=O)sc2ncccc2c1N 95435,CC1(CN2C(C(=O)NCc3cnc(O)c(F)c3)CC(=O)C2)CC2C=CC1C2 95436,C1(NC(c2c(OC)cccc2)=O)CN(C(C2(CCO)CC2)=O)CCC1C 95437,C(C)(C)(CC(F)C(=O)N(CC(C)O)C)NC(CNC(C(C)C)=O)=O 95438,n1(CCC(=O)NCC2N(C(C3C(=C)C3)=O)CC2)c(=O)nc(O)c2ccccc12 95439,C1(C(=O)NC2(C)CCN(C(CN(c3cnccn3)CC)=O)C2)CCC2(CCC2)O1 95440,Cc1ccnc(O)c1C(=O)NC1CCCCCC1NC(=O)Cc1sc(O)nc1O 95441,C1(C(=O)N(C2CCCC2)Cc2ccncc2Cl)CNCCC1(F)F 95442,C1(NC(CC2(OC)CN(C(C3ON=C(CC)C3)=O)C2)=O)CCCCCC1C(N)=O 95443,C(=O)(C(CN(C)C)C(C)C)NC(C1CCN(C(C(COC)NC(C)=O)=O)C1)C 95444,c1(CNC(CCCCCOC)=O)cccc2c1CCN(CC1C(Nc3cocn3)C1)C2 95445,CC1(C)CC(C)(C(N2CCC2(C)CCO)=O)CN1NC(C1CC2(CC2)C1)=O 95446,CC(CC(=O)NCC(c1ccccc1)N(C(=O)CN1CC2CC2C1)C)NC(N)=O 95447,C1(CC(=O)NC(C2CCC2)C)CCCN(C(=O)CCCCNC(N)=O)C1 95448,C(=O)(CCCC(F)(F)Br)N(C1CCN(CC2CC(C)(C)CO2)C1)C 95449,N1(C(C(CC2CC2)OC)=O)CC2CCC1CN2C(=O)Cc1ccc(C)s1 95450,N1(C(CNC(C)=O)=O)CCN(C)C(C(=O)NCc2cccnc2C)C1 95451,C1(C(=O)NC2CCC(NC(C3(C#N)CC(C)C3)=O)CC2)CCOC(C)(C)C1 95452,N1(C(C(C)=NOCC#N)=O)CCN(C(c2n[nH]c3ccccc23)=O)CC(O)C1 95453,CCCCCCC(O)CCC(=O)NCC1(OC)CN(C(=O)C=CS(=O)(=O)CC)C1 95454,CC1CC(C(=O)NCC(O)COC(c2cncs2)=O)N(CC(C)(C)C)C1 95455,C(Cc1ccccc1)(CCNC(=O)C=C(C)C(C)(C)C)NC(C(C)c1cccs1)=O 95456,N1(C(C(COC)(F)F)=O)CC(NC(c2cccc(OC(F)F)c2)=O)CC(O)C1 95457,CC1CN2CCN1C(C(=O)N(C)CCN(C)C(c1nccn3nccc13)=O)C2 95458,N1(c2ncnc(OC)c2C)CCC2(C(=O)O)C(C1)C2(F)F 95459,c1(C(=O)NCCCC(C)NC(C2C(C(C)O)C2)=O)ccc([N+](=O)[O-])c(O)c1 95460,N1(C(c2nc(CC)sc2)=O)CC2CCC(NC(=O)Cc3c(C)noc3Cl)CC2C1 95461,C=CCC(CC(=O)N1CC(=O)NCC1C)NC(c1cnn(CC)c1C)=O 95462,C(C(C)(O)C(F)(F)F)NC(CC(CNC(CCCNC(=O)OC)=O)C)=O 95463,C1(CNC(C(C)NC(c2ccccc2)=O)=O)COCCN(C(N)=O)C1 95464,CC1(C)OCCCC1CNC(=O)CC1CCN(C(=O)Cc2ccccn2)CC1 95465,N1(C(=O)OC)CCC(NC(=O)CC2CC2CNC(=O)C(C)n2cccn2)C1 95466,c1(CC(=O)NC2C(CNC(C=COCC)=O)COC2)csc2sc(C)cc12 95467,C1(N(C(C(CCC)OC)=O)CC)CCCN(C(=O)C=Cc2nnc(C(C)C)o2)C1 95468,CC1CN(C(=O)CN(C)C(N)=O)CC(CCNC(=O)C(c2ccccc2F)O)O1 95469,c1(C(=O)NCC2(CNC(CSc3n(C)ccn3)=O)CCCC2)cc2n(n1)CCO2 95470,c1(C(C(=O)NC2C=CCN(C(CN(C(COC)=O)C)=O)C2)(F)F)ccc(C)c(C)c1 95471,Cn1cc(C(=O)NCC2OCCC2C(=O)Nc2cc(C(N)=O)cc(O)c2)n(C)c1=O 95472,N1(C(C2(F)C(C)OCC2)=O)CCCC2(CCN(C(=O)CC3CCC(O)C3)C2)C1 95473,c1(C(N2CC(CNC(C3COC(=O)O3)=O)C2)=O)ccc2cncnc2c1 95474,c1(C(=O)NCC(C)NC(=O)C2=CCSC2)c[nH]c2cccc(C#N)c12 95475,N1(C(c2cc(C3CC3)ccc2F)=O)CCC2(CCN(Cc3ccc(O)cc3)C2)C1 95476,N1(C(COCCC=C)=O)CCN(C2CCC(NC(=O)C(C)(C)C3CC3)C2)CC1 95477,C1(C(N2CC(C(C)NC(=O)C(c3ccc(F)cc3)(C)C)C2)=O)CCCCS1(=O)=O 95478,c1(C(C)(C)C(=O)NCC(O)CCNC(c2n[nH]cc2Cl)=O)ccc(F)cn1 95479,C(=O)(C(CC(F)F)C1CCC1)NCCN(C(C1(C)ON=C(C)C1)=O)C 95480,CC(C)(C(=O)NCC(CO)NC(C1CCOC1)=O)C1CCC1 95481,C1(NC(=O)Nc2c(C(C)C)cccc2)C2CC3CC1CC(O)(C3)C2 95482,CNS(=O)(=O)N1CCC(C(=O)NCCNC(C2CN3CCC2(C)CC3)=O)CC1 95483,C1(c2cccc(F)c2)(NC(=O)C=CCO)CCN(C(=O)CCCC2CCOCC2)C1 95484,CC1CCC(Cl)=C(C(=O)N2CCN(C(=O)COCC(C)(C)C)CC(O)C2)C1 95485,N1(C(c2c(C)csc2)=O)CC2CC(C1)CN(C(C1CC(C)(C)C(C)(C)C1)=O)C2 95486,c1(C(N(CCCNC(C2COCCO2)=O)C)=O)cc2ccc(F)cc2cn1 95487,c1(SCC(N2CCC(NC(c3c(C)nns3)=O)CC2)=O)ccc(F)c(F)c1 95488,C1(NC(c2cc(C(C)(C)C)no2)=O)CCCC(NC(C2(CC3CC3)CCOC2)=O)C1 95489,c1(CCC(=O)NC(CC)(C)CNC(C2CNC(=O)N2)=O)nc2ncccn2n1 95490,Cc1cccc(F)c1CNC(C1C(C)CCN1C(=O)CC1CC(=O)NC(=O)C1)=O 95491,N=c1cc[nH]cc1C(=O)N(CC1CCN(C2CCOC2)CC1)Cc1cccnc1 95492,C1(CNC(Cc2cccc(OCC)c2)=O)CN(C(c2scnc2C)=O)CC12CC2 95493,CN(CCCC(=O)N1CCC(N(C(=O)C(O)C(F)(F)F)CC2CCCO2)CC1)N=O 95494,c1(SC)cccc(C(=O)NC2CN(C(c3cccnc3O)=O)CC2C)c1O 95495,O=C1CCC(C(=O)N2CC3(NC(=O)CC4CCCC(=O)N4)CC2C3)=NN1 95496,Cc1onc(C(N2CCCC(NC(c3cc(Br)no3)=O)C2)=O)c1[N+](=O)[O-] 95497,c1(C(=O)NCC(=O)NCC(=O)NC2CC(N(C)C)C2)ccnc(C2CC2)c1 95498,c1(N2CCCC3C4C=CC(C4)C2C3)nc2cccnc2c(=NCC2CCCS2)[nH]1 95499,N1(C(C(CC#C)(C)C)=O)CC(CNC(=O)C(C)n2cccn2)C2(CCOCC2)C1 95500,C1(C)(CC)CC(C(N2CC(C)(CO)C2)=O)CN1C(=O)CCS(=O)(=O)N(C)C 95501,C12(C(N(C)Cc3ccncn3)=O)CCCC1CN(C(C1(C#N)CCCCC1)=O)C2 95502,c1(CNC(N(C(C)C(=O)O)CC#C)=O)cccc(-c2nnco2)c1 95503,N1(CC2(O)CCN(Cc3ccccc3)C2)CCc2sccc2C1c1ccccc1 95504,c1(COC(c2nnn(C)c2C2CCC2)=O)oc2ccccc2c1CS(C)=O 95505,C1(C(N2CC3C(NC(C(C)N(C(C)=O)C)=O)C3C2)=O)CCC([N+](=O)[O-])CC1 95506,c12ccc(o1)CN(C1CC1)C2C(=O)NCC(=O)OC.CCC(C)(C)OC 95507,C(CC(=O)N1CC2CCC(C1)N2C(=O)C=Cc1ncc[nH]1)(C(F)(F)F)OC 95508,C1(C(N(C)CC2CC(=C)C2)=O)CCC(C2CC2)N1C(C1CCCC1F)=O 95509,N1(C(C(C(C)(C)O)F)=O)CC2(CCN(C(=O)Cc3ccncc3Cl)CC2)C1 95510,c1(C(N(CC(CC)NC(c2csc(C3CCCO3)n2)=O)C)=O)ccc(O)c(Cl)n1 95511,N1(C(C2(C)COC2)=O)CCCC2(CCCCC2NC(C2CC3CC3C2)=O)C1 95512,Cc1cn(C)cc1C(N1CC(=O)CC1C(=O)NCCC1CCCN1C)=O 95513,N1(C(C(C)NC(CC)=O)=O)CC2C(CN(C(=O)CCN3CCC(O)CC3)C)C2C1 95514,N1(C(Cc2c(C)nn(C)c2)=O)CC2CCCCCC2C1.C12(CCCCC1)C(=O)N2 95515,Cn1nc(CNC2CN(C(c3nc(Br)cs3)=O)C2)c2ccccc12 95516,C(=O)(CC(C)(C)C)N(C1CCC(Oc2ccncc2)C1)CCCN(C)C 95517,CC(C)(C)CC(O)C(=O)N1CC=CC1CNC(c1ncc2[nH]ncc2n1)=O 95518,N1(C(C(CC=CCC)C)=O)CCN(C(=O)C=CC(C)(C)SC)CC1C1CCCC1 95519,C(CC(C(=O)N(CC(N1CCCC(C(C)O)C1)=O)CC(C)C)OC)OC 95520,c1(C(N(C2(C(N3CCCC(C)(C)C3)=O)CC2)C)=O)ccc2[nH]ccc2c1 95521,CCC(CC)C(C)C(=O)N1CCCC(C)(CNC(=O)CC2COCCN2C)C1 95522,c1(C(N2C3(CNC(CC4(C)CCCO4)=O)CC(C2)C3)=O)cccc2c[nH]nc12 95523,N1(C(c2c(COC)ccs2)=O)CCN(C(=O)C=Cc2cscn2)C(CC(F)F)C1 95524,c1(NC2CC(N)C2)cc(C)ccc1[N+](=O)[O-].c1(CSCC)cc(C(=O)N)no1 95525,Cc1nc(N(C)C)sc1C(=O)N(C(C)CN(C1CC1)C(C1CC2CC2C1)=O)C 95526,C(CC(C)(C)C)(C(=O)NC1CCCCC1C(=O)NC(C)Cc1cnccn1)OC 95527,c1(OC)ccc2c(c1)CCCC2C(=O)N(c1ccc(N)c([N+](=O)[O-])c1)C 95528,c1(CC)cc(C(N2CCCC2C(C)NC(c2cc(F)cc(F)c2)=O)=O)ccc1Cl 95529,c1(C(=O)NC(C(=O)OC)Cc2cccs2)noc2c1CC(C)(C)CC2 95530,C#CCC(C)(C)C(=O)NCC(CO)NC(c1c[nH]c(=N)nc1C)=O 95531,c1(OCC)cnnc(NC(C2(NC(=O)CN3CCN(C)CC3)CC2)=O)c1 95532,O=C(CN1C(=O)Cc2ccccc21)NC1C2CCCN(C(=O)CSC(F)F)C2C1 95533,C1(C(N(CCCNC(CC(C)N(C)C)=O)CCO)=O)CCN(S(=O)(=O)N(C)C)C1 95534,CC(CC(F)F)C(=O)NCC(N=c1[nH]nc(-c2ccccc2)o1)c1ccccc1 95535,C1(C(C)NC(=O)CC2CC(N(C)C)C2)C2CN(C(=O)NCc3ccc(F)cc3)CC12 95536,C(=O)(CC(C)CC(F)(F)F)N1CC2(CN(C(C(C3CCOCC3)C)=O)C2)C1 95537,n1(CCCOC)nc(-c2ccc(N)cn2)nc1-c1nc(C(F)(F)F)cs1 95538,C1(C(N)=O)CCCN(C(c2cncc(CNC(c3cc(C(F)(F)F)c[nH]3)=O)c2)=O)C1 95539,N1(C(CCC)=O)CCCC(C)C1CNC(=O)CCc1cn(C)nn1 95540,C1(NC(CC(C)F)=O)CN(C(=O)CCOc2cccnc2)C2(CCCC2)C1 95541,C(CCC(O)CO)NC(CONC(c1cc(OC)no1)=O)=O 95542,C1(SCCOC(c2cc(OC)c(Br)nc2)=O)OC(=O)CC12CCC2 95543,c1(C(=O)NC(CNC(CCOc2c(C)cccc2)=O)CO)cccc([N+](=O)[O-])c1 95544,c1(SC)ccc(Cl)c(C(N2CCN(Cc3cn(CCF)nn3)CC2)=O)c1 95545,CC(C)C(C)CC(=O)N1CC(O)CC1CNC(=O)COc1ccon1 95546,C1(OC)CN(C(=O)C(C)N(C)C(C)=O)CCC1NC(C1CCCCN1C)=O 95547,N1(C(c2cccc(C(C)C)c2N)=O)CC2CN(Cc3sc(Br)nc3Br)CC12 95548,C1(NC(C2CC(CC)(CC)C2)=O)C=CCN(C(=O)C(N2CCOCC2)C)C1 95549,c1(CC(=O)Nc2c(OCC)cccc2)ccc(S(C)(=O)=O)c(F)c1 95550,Cc1c(C(N2CC3CC3(CNC(=O)CCOC3CC3)C2)=O)cccc1C(F)(F)F 95551,N1(C(C(C)(C)OCC)=O)CCCC(C(=O)NCc2nc(CO)n[nH]2)C1 95552,C1(C)(C)CC(=O)N1.C1(C(=O)OC)CCN(C(c2ccccc2)CC)CC1 95553,c1(OC(C)C)cc(CNCCCNC(C2CCN(C(C)=O)C2)=O)ccn1 95554,c1(C(=O)NCC2C(CNC(C(F)=CC)=O)C2)ccc(-c2cccnc2)s1 95555,c1(CCNC(c2cn(CCO)nn2)=O)cncc(C)n1.C(C(=O)OC)N1CC1 95556,c1(NC(C(C)n2ccnn2)=O)cccc(CNC(c2ccoc2Br)=O)c1 95557,c1(OCC(F)(F)F)c(F)cc(NCCCC(F)F)cc1F 95558,C1(CC(=O)NCCC2CC(NC(=O)CCc3ccoc3)C2)CC1(Cl)Cl 95559,N1(C(CCC=C)=O)CCOCC(C(C)(C)C)C1.c12ccccc1C(=O)N2 95560,C1(NC(C2(N(C)CC)CCC2)=O)CCC(C)(C)C1.C1C(C)NC(=O)N1C 95561,C(=O)(CC(C)(C)CC(F)F)NC1CC(C)N(C(C2CC2C2CCCCC2)=O)C1 95562,Cc1cccc(C(=O)NCC2(C)CCC(NC(c3ncncc3F)=O)C2)c1 95563,C1(C#N)(CC(=O)N(C2CC(O)CN(C(C3(C)CCOCC3)=O)C2)C)CCOCC1 95564,C1(C(=O)NCC(C)N(CC)CC)CCC(C(C)C)N1C(=O)CC1(C)OCCO1 95565,C12(NC(CSCCCC)=O)CC(CNC(=O)CCC(C)(C)OC)(C1)OC21CCC1 95566,c1(C(=O)NC(CN(C(=O)Cc2ccno2)CC)C)ccnn1C1CC1(F)F 95567,N#Cc1cc(Br)ccc1N1CCN(C(C2CC(c3ccncc3)CN2)=O)CC1 95568,N1(C(C2(C)C(C)C2)=O)CCOCC(CNC(c2ccc(Cl)c(Cl)c2)=O)C1 95569,n1(CCC)ccc(C(=O)NC(C)C(C)NC(=O)CNC(=O)CSC(C(C)(C)C)=O)n1 95570,N1(CC(=O)N(CC(CC)NC(=O)C(C)C2CC2)CC)C(=O)NC2(CCCC2)C1=O 95571,N1(C(c2ccc(SCc3ccc(C)cc3)o2)CCCO)CC2C3C=CC(O3)C2C1 95572,C(C(=O)N=c1ccn(CCF)[nH]1)(C1CC1)NC(c1c(C)cns1)=O 95573,c1(C(=O)Oc2cccc(C3CC3)c2)ccc2nccn2n1 95574,CN=c1[nH]cc(C(=O)NC2CC(C(F)C(=O)NCCC#CCO)C2)o1 95575,C#CC(C(C)(C)C)NC(c1cccc(CNC(=O)OC(C)(C)C)c1)=O 95576,C1(=O)C(C)Cc2cn(nn2)CCNC(=O)N2CC(C2)O1.CCCOC 95577,C(CC1C(=O)Nc2ccccc21)NC(=NCC(C)C)NC1CCCC1 95578,C1(C(=O)NC2CCCCN(CC)C2)COC2(C1)CN(C(C1CCCS1(=O)=O)=O)C2 95579,C1(C(C)C)CN(C(C2CCCCCC2)=O)CCN1C(c1cccn1C)=O 95580,C(=O)(C1=NOC2(CCN(C(c3cc(C#N)ccn3)=O)C2)C1)NC(C)CN(C)C 95581,c1(N2C3C(CNC(C4(C)CC4Br)=O)C(CCC3)C2)nc(O)c2ccc(Cl)cc2n1 95582,c1(OCC)cnccc1C(=O)NCC1(NC(=O)Cn2ccnc2C)CCCCC1 95583,c1(C(C(C)NC(=O)CCc2cnc[nH]2)NC(c2ccon2)=O)ccccc1 95584,C1(CNC(CCC(CC)C)=O)CC2(CO1)CN(C(=O)CC1CCCCC1)C2 95585,N1(C(c2c(C)ccnn2)=O)CC(C(=O)NOC2CCOC2)C2(CC2)C1 95586,C=CCN(OC)C(=O)C(C)N1CCCC1.C1(=O)CCC(CC)N1 95587,c1(CN(c2n(CCCC)c(-c3cncc(CO)c3)nn2)C)cnc(OC)c(F)c1 95588,C(=O)(C(C)CCCOC)NC1CC(C)(CNC(c2c(CC)c[nH]n2)=O)C1 95589,C1(NC(C=CCC(C)(C)NC(Cc2cccc(C)n2)=O)=O)CC2CC1CC2CO 95590,CCN=C(NCc1ccc(CN(C)C)cc1)N1CCC(S(C)(=O)=O)CC1 95591,C#CCCCCC(=O)NCC12CC(NC(C3CCCC3(F)F)=O)(C1)C2 95592,C1(CNC(C(C2CCOC2)NC(C=CCOC)=O)=O)(CO)CCOCC1 95593,c1(C(N2CC(OCCNC(C(C=C)OC)=O)C2)=O)cc(O)cc(=O)o1 95594,C(=O)(C(CCC(N)=O)NC(=O)CC1(O)CCCCCC1)OCCC 95595,c1(CCC=CC(=O)NCC2CN(C(C3(F)CCOC3)=O)CCO2)ccc(F)cc1 95596,CC1CCN(C(C2CCCC(=O)CC2)=O)CCN1C(C1CC=CCO1)=O 95597,N1(C(c2c(CCC)occ2)=O)CC(NC(c2cc(C)c(C)[nH]2)=O)CC2(CCC2)C1 95598,C(=O)(CCC(F)(F)F)N1C(C(=O)Nc2ccc(C(=O)OC(C)(C)C)nc2)CCC1 95599,CC(=O)CCCC(=O)N1CCCC1CN(C(=O)C(C)Cc1cccc(Br)c1)C 95600,C1(C(N2CC(CNC(=O)CCCCCO)C(F)(CO)C2)=O)Cc2ccncc2C1 95601,Cc1nc2c(s1)CC(NC(=O)NCc1ccn(-c3cccc(Br)c3)n1)CC2 95602,c1(C(=O)NCCCN(C(=O)CCC2CC2)C2CC2)c(F)ccc2c1OCO2 95603,N1(C(C(c2ccccc2F)C)=O)CCC2C(NC(=O)CSc3ccc(Cl)cc3)C12 95604,c1(C(=O)NCCC(CNC(c2ccc(SC)o2)=O)O)c(Cl)ccc(Br)c1N 95605,C1(CC(=O)NC2C=CCN(C(c3c(C)nco3)=O)C2)CC(=O)CC(=O)N1 95606,c12ccc(s1)C(=O)N(CC(C)O)CCNC2=O.c1(NC(C)=O)ccn(C(F)F)n1 95607,N1(C(c2c(C)c[nH]n2)C(=O)NCCCF)CCN(c2cccnn2)CC1 95608,C1(O)(c2cn(CNC3COC4COCC34)nn2)CCN(C(C)CCOC(F)F)CC1 95609,c1(C(=O)NC2(COC)CCN(C(CC(=C)Br)=O)C2)cn2cnnc2cn1 95610,C1(CNC(=O)C=CC(F)(F)F)CCCC1NC(c1cc(COC(C)(C)C)on1)=O 95611,CC(C(C)(C)C(N)=O)NC(=S)NCC(C)CCc1ccccc1 95612,N1(C(C(C)CC(N)=O)=O)C2CCC1CC(N(C)C(c1cccc(C(N)=O)c1)=O)C2 95613,c1(C(N(C(C)CC(=O)Nc2ccc(CO)cc2)C)=O)ccc2c(c1)C(=O)OC2 95614,C1(N(CC=C(C)C)C(C2CCN(C)C2)=O)CCN(C(c2ccccc2)=O)C1 95615,C1(C(=O)NCC2(C(N)=O)CN(c3snc(CCC)n3)C2)CCSC(C)C1 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95651,C1(NC(C(CCC)O)=O)CCCN(C(=O)CCc2ccc(F)nc2)CC1 95652,C1(CNC(=O)C=CC(C)(C)SC)C2CC1N(C(=O)COc1cnn(C)c1)C2 95653,C(CC(=O)NC1CCn2ccnc2C1)(C(C)(C)C)NC(C(=CC1CCCC1)C)=O 95654,c1(-c2c(C)occ2)nc(CC2CCC(O)C2)n(C2CCC2)n1 95655,c1(C(=O)NC2C(NC(CC=CC)=O)C2)cnc2ccccn12 95656,C(=O)(C1=CCOCC1)NCC1(C)CCN(C(=O)CC2C=CCCC2)C1 95657,N1(C(CCOCC(C)(C)C)=O)CC2CCC(C1)N2C(c1ccc(F)c(N)c1F)=O 95658,CC1COCC(C(N2CCC(C(=O)NCC(C)(O)C(F)F)C2)=O)O1 95659,c1(OC)nccc(=NC(=O)C2COCCN2C(c2ccc3[nH]c(=N)sc3c2)=O)[nH]1 95660,C1(C(=O)NC(CNC(CSCC#C)=O)(C)C)CC(=O)N(CCN(C)C)C1 95661,c1(CCC(=O)NC2CC3CCC2N3C(c2ccnnc2)=O)ccc(O)c(F)c1 95662,CC(C)C(C(=O)NC1(CCC(C)O)CC1)n1cncn1 95663,C1(N(C(Cc2cc(C)sc2C)=O)C)CCCCN(C(C2CC2C(F)(F)F)=O)C1 95664,c12ccc(C)cc1CC(=O)N1CCC(CC1)CC(C)N2.n1(CC)cc(CO)nn1 95665,N1(C(N2CCC(Cc3cscc3Br)C2)=O)CCC(O)(c2cnccn2)CC1 95666,CCC(CN(C)C)CC(=O)NCCC(C)NC(c1cnn(C2CCCCC2)c1)=O 95667,c1(NC(C2CCN(C(c3cc(F)ccc3O)=O)C2)=O)ccc2c(F)n[nH]c2c1 95668,C(=O)(CC(C)P(C)(C)=O)NCCC(CNC(C1(n2cnnn2)CC1)=O)OC 95669,C1(C(F)(F)F)(SCCNC(C2CC2N(C(=O)OC(C)(C)C)CC)=O)CC(F)C1 95670,C1(CC)CCC(C2COCCN2C(=O)C(=O)NCCOc2nccs2)O1 95671,N1(C(C(C=C)O)=O)Cc2ccccc2CC1CNC(c1cc(C2(C)CC2)on1)=O 95672,c1(C(=O)NC2CN(C(c3cscc3Cl)=O)C2)cc(F)cc2cc[nH]c12 95673,C1(CC)CN(C(=O)C(C)n2ccnn2)CCC1CNC(=O)Cc1cc(C)ns1 95674,N1(C(c2n[nH]c(C)c2O)=O)CC(=O)NCC1C(=O)NCCCn1ccnn1 95675,C1(CNC(=O)C=CCF)CN(C(c2ccc(N3CCCC3)nn2)=O)CCO1 95676,CC(C)(C#N)CC(=O)NC1CCN(C(=O)CCNC(=O)OC(C)(C)C)CC1(C)C 95677,C(=O)(CC(C)c1ccco1)NCCCN(C1CCCCC1)C(CSCC)=O 95678,Cc1sc(Cl)c(C(=O)NC(C)(CNC(C2CC(OC(F)F)C2)=O)C(C)C)c1C 95679,C(=O)(C(C(C)C)S(=O)(=O)C1CCCCC1)NC1CN(C(c2cc(C)nn2C)=O)C1 95680,C1(CSC)CCCN1C(=O)C(=O)NCCCCC1CCCCO1 95681,N1(C(=O)COC2CC2)CCCN(C2CCN(C(c3cc(N)cc(F)c3)=O)C2)CC1 95682,C1(NC(c2c(SCC)cccn2)=O)CC2CC1CN(C(=O)CC1CC3CC3C1)C2 95683,C1(CNC(c2cc(C)no2)=O)CN(C(c2sccc2C#N)=O)CCO1 95684,c1(C(=O)NCCN(CC(C)O)C(=O)CSc2nnnn2C)cccc2nsnc12 95685,c1(OC(C(=O)NCC=CCNC(CCC)=O)(C)C)ccc([N+](=O)[O-])cc1 95686,c1(-c2ccc(NCCN(C(c3cc(C)c(O)nn3)=O)CC)s2)ccc(Cl)c(Cl)c1 95687,C1(NC(C=C(C)C(C)C)=O)CCN(C(c2c[nH]c(C(F)(F)F)c2)=O)CC1F 95688,c1(CCC(=O)NCC(CC)(C)NC(=O)C(C)O)cccnc1Br 95689,C1N2C(=NCCCCCCS(N)(=O)=O)NCC1=CC=COC(CCC)CC2 95690,C1(CCC(=O)NC(C2(C(N(CCCOC)C)=O)CC2)C)CCC(=O)C1 95691,c1(C(=O)NCCOC2CN(C(C3(S(C)(=O)=O)CC3)=O)C2)cc2sccc2[nH]1 95692,N1(C(c2c(C)ccc(F)c2)=O)CCC(F)(F)C(NCc2cc(Br)c(Br)s2)C1 95693,C1(CNC(C)=O)C(C)CCN1C(c1cnn(C2CC2(F)F)c1)=O 95694,N1(CCCCO)CCC(N=c2ccc3nnc(-c4cccc(Br)c4)n3[nH]2)CC1 95695,N1(C(C=CCN(C)CC)=O)CC(CCNC(=O)C(CCO)N(C)C)C(C)C1 95696,C1(C)(C(=O)NC2(CCCC(=O)NCC(c3ccsc3)C)CCC2)CC(=O)N(C)C1 95697,C1(C(N(CC(O)CNC(c2coc(CO)c2)=O)C)=O)CC12CC(C)(C)C2 95698,N1(CC#C)CC2CCC(C1)C2NS(=O)(=O)CCC.c12ccc(cc1)c(=O)o2 95699,c1(C(N2CCC(OC(F)F)CC(C)(C)C2)=O)cnc2ccccc2c1 95700,C1(C)(CC)CC(NC(C23CC(CO)(C2)OC3C)=O)CN1C(=O)CSC(F)F 95701,C1(NC(c2ncccc2CO)=O)CN(C(c2cnc(S)nc2)=O)CC2(CCC2)C1 95702,C1(NC(=O)NC2CC23CCC3)CCOCC1O 95703,c1(C(=O)OC)ccc(C(=O)NCCCCNC(C2(O)CCC2)=O)cc1O 95704,C1(C)(C(=O)NC(CC)CN(C)C)CCCN(C(=O)Nc2cccc(C)c2)C1 95705,N1(C(Cc2c(C)scc2)=O)CCCC2(CC(NC(c3ncccc3F)=O)CO2)C1 95706,c1(-c2n(C(CC)C)nc(-c3nccs3)n2)nc(C)n2c1CCCC2 95707,C(CCC(C)(C)NC(=O)CC1CC1)N(C)CC1CCOC1.c12c[nH]nc1CNC2=O 95708,N1(C(C(=O)Nc2c(C)c3c(cn2)cccc3)=O)CC2(COC(C)(C)C2)C1 95709,c1(CC)nc(=N)[nH]c(=NCC2CC(C)N(C(c3cccc(C4CC4)c3)=O)C2)[nH]1 95710,Cn1cc(Cl)c(CC(=O)NCc2occc2C(=O)NCC(C)(C)CO)n1 95711,C1(N(C(C=CC(CC)=CC=CC)=O)C)CCN(C(C2CN(C3CCC3)C2)=O)CC1 95712,C1(CCC(=O)N(C(C(C)SC)C)C)CCN(C(c2cnc(O)o2)=O)CC1 95713,c1(OC)nccc(C(N2CCCCC2CNC(c2ncccc2C2CC2)=O)=O)n1 95714,N1(C(CC(CCCC)O)=O)CC2(CCN(C(c3cc(C)nc(O)c3)=O)CC2)C1 95715,C1(C)(CC(=O)NCC2(CSC)CC2)CCN(C(C2C3CN(C)CC23)=O)C1 95716,C1(F)(C(=O)NCC2N(C(c3c(CC)ncs3)=O)CC=C2)CCCN(C)C1 95717,c1(-c2nc(C(CC)CC)nn2-c2ccn(CCOC)n2)cnn2c(C)ccnc12 95718,Cn1cc(C(N2CCC(O)(CNC(=O)C(C)(C)F)C2)=O)c(Cl)n1 95719,N1(C(C(C2CCN(Cc3cc(Br)c[nH]3)CC2)C)=O)CCC(C)(CO)C(O)C1 95720,C#CCCC(O)CCNC(c1cccnc1CNC(=O)C(C)C1(O)CCC1)=O 95721,C1(C(N2CC(SC)C(n3cc(C(C)(C)CO)nn3)C2)=O)CCCCN1N=O 95722,Cc1cnc2nccc(C(N3CC(CNC(C4CC4F)=O)CC3C)=O)c2c1 95723,c1(NC(C2C(NCc3ccc(OCC)c(C#N)c3)C2)=O)nccc2scc(Br)c12 95724,N1(C(CCC(=O)NC)=O)CCC2CN(C(c3coc4c3C(O)CCC4)=O)CC2C1 95725,N1(CC(C)C)CCN(C(=NCCCCl)NCc2noc(C(C)(C)C)n2)CC1 95726,C(=O)(C(O)P(C)(C)=O)N1CC2C(NC(C3CC(C)(N(C)C)C3)=O)C2C1 95727,C1(C(=O)NCC(CCC)(C)O)CCCN(C(=O)C(C)CC(C)C)CC1 95728,C1(CN(C)C(c2ccoc2C(F)(F)F)=O)CCCN1C(=O)CCC#N 95729,C1(C(=O)NC(c2cnn[nH]2)C)CC(O)CN1C(C1CN(C(N)=O)C1)=O 95730,c1(C(N(CC(CNC(c2c(C)scc2)=O)C)C)=O)cccc(OCC(F)F)n1 95731,c1(C(C)=O)ccc(C(=O)NC2CCC(C)N(C(c3[nH]c(C)cc3C)=O)C2)cc1F 95732,C(=O)(C1=NOC2COCC12)NC(c1cccnc1)C.C12CC1NC2=O 95733,C(=O)(C#CC1CCCOC1)N1C(CS(C)(=O)=O)CN(C(c2cnn[nH]2)=O)CC1 95734,Cc1ccc(C(=O)NCC2CCCC2C(=O)NCC=C(Cl)Cl)nc1 95735,c1(CC)cc(C(=O)NCC(C(C)C)NC(C2CN(C)CCO2)=O)cc(F)c1 95736,C1(NC(CCCCCSC)=O)CN(C(C2OCCCO2)=O)CC1N=[N+]=[N-] 95737,c1(C(N2CCC(C)(CNC(C3(CC)CCOCC3)=O)C2)=O)cc(C#N)ccc1F 95738,c1(C(=O)NC(CC)CN(C(=O)C=CCO)CC)cccc2c3c([nH]c12)CCC3 95739,N1(C(CCCOC)=O)CC2CCC(NC(c3cccc(S(C)=O)c3)=O)(C2)C1 95740,C1(C(=O)NC2CC3CC(NC(CCSCC)=O)CC32)CC(C(C)(C)C)=NO1 95741,CCC(F)(C(=O)OC)C(=O)N1CC(O)(C(C)NC(C2CN(S(C)(=O)=O)C2)=O)C1 95742,CC1CN(C(=O)C=Cc2cnccn2)CC(C)CN1C(C1COC1)=O 95743,Cn1ccc(C(=O)NC2CC2C(=O)Nc2ccc(C(F)F)cc2F)cc1=O 95744,C1(CCC)CCCN(C(=O)C(CNC(=O)C(C)(C)C2CCCO2)CCC)CC1 95745,C12(CNC(CC3(COC)CC3)=O)CCCC(CN1C(c1cncc(C)c1)=O)C2 95746,c1(NC(C2CCCC(C(=O)OC)C2)=O)nn(C)c2ccccc12 95747,c1(OC)ccc(NC(C2CN3CCC2C3)=O)c(OCC2CCOCC2)c1 95748,C1(C(=O)NC(C)CN2CCCC2)CCN(C(C2CC23CCC3)=O)C12CC2 95749,C1(C(N)=O)(CNC(=O)CN2CCOCC2)CN(C(c2cc(C(C)(C)C)c[nH]2)=O)C1 95750,C1(CC(=O)NCC(C(C)C)NC(C2CCC(C(=O)OC)C2)=O)CCCC(C)(C)O1 95751,C(CC(=O)N1CC2(CCOC2=O)C1)(C(C)(C)C)NC(C(CCC)(C)O)=O 95752,C=CCC(F)(F)C(=O)NC1CN(C(c2cc(CC)ccn2)=O)CC1OC 95753,N1(C(C2C(OCC)C2C)=O)CCCCC(NC(c2cccnc2C2CC2)=O)C1 95754,CC1CN(C(c2ccnn2CCF)=O)CCC1CNC(C1CC2(CCOC2)C1)=O 95755,CC1CN(C2CCC2)CCC1C(c1ccccn1)CCNC(=O)CC(C)(C)O 95756,Cn1ccc2ccc(C(=O)NC(C)(CNC(=O)CCN3CCCCC3)CO)cc12 95757,c1(NC(N(CCCC)CC2CCN(Cc3ccccc3)C2)=O)ccc(C)c(OC)n1 95758,N1(C(C2N(S(c3cccc(C)c3)(=O)=O)CC2)=O)CC(S(=O)(=O)C2CCCCC2)C1 95759,N1(C(C2N(CC)CCOC2)=O)CCCC(O)(CCNC(=O)Cc2ncoc2C)C1 95760,Cc1cnc2nccc(C(=O)NCC3CCCCN(C(=O)C(C)CN(C)C)C3)c2c1 95761,C(C(C(C)(C)C)NC(C1(C(F)(F)F)CC1)=O)NC(C=CC(C)C)=O 95762,c1(C(N2CCC(N3CCC(NC(C(C)O)=O)C3)CC2)=O)ccc(C#N)c(Cl)c1 95763,C(CCC(C)CC(=O)NC1(CF)CCN(C(=O)CN(C)C(C)C)C1)=C(C)C 95764,n1(CCOC)cc(CNC(=O)C(Cc2cn[nH]c2)NC(c2cccs2)=O)nn1 95765,CC(C)CCC(=O)NCC(O)C(=O)N(CCNS(C)(=O)=O)C1CC1 95766,C1(NC(C2CCC(C(F)F)CC2)=O)COC2(C1)CN(C(C1(F)CCCC1)=O)C2 95767,N1(C(C(c2cncnc2)C)=O)C2CCC1C1CC1(NC(=O)CC1CCC1)C2 95768,C(=O)(C(C)(C)C(=O)N1CCCCC1C(=O)NCC1C2CCCOC12)OCC 95769,Cc1ccc(C2CC2C(=O)NCC(C2CCC2)NC(c2cocn2)=O)o1 95770,C(=O)(CC(F)(F)F)N1CC(N(c2ncccn2)C(C(C)NC(=O)OC(C)(C)C)=O)C1 95771,c1(C(N2CCCCC(CN(C(C(=O)NC)=O)C)C2)=O)ccc2nn[nH]c2c1 95772,Cc1ncc(Br)c(N2CCCC(CNc3ccc(-c4ccccc4C)nc3)C2)n1 95773,CC(C)(CCNC(=O)Cc1csc(-c2ccsc2)n1)c1nn[nH]n1 95774,C(=O)(C1=CCCN(C(C2CC(O)C2)=O)C1)N(CC(C)O)CC(C)O 95775,C1(Nc2ccc(NCC=CC(C)(C)C)cc2)OC2CCC1CC2 95776,CC1CC(NC(=O)CCc2ccon2)CN1C(c1ncccc1C(F)(F)F)=O 95777,N1(C(COC(C)C)=O)CCCC(NC(c2ccn(C)c(=O)c2)=O)C(F)C1 95778,CC(C)C(O)C(=O)NC1CCC1CNC(c1ccccc1C(N)=O)=O 95779,c1(C(=O)NC(C2(O)CN(C(=O)C(O)C(C)(C)C)C2)C)cc2ccc(Br)cn2c1 95780,C1(CC=C)(NC(=O)C(C)CO)CCCN(C(=O)CS(=O)(=O)NC2CC2)C1 95781,N1(C(c2c(C)cno2)=O)CCN(c2nc(C(C)C)ns2)C(CCO)C1 95782,c1(NC(C23C(CN(C(C(CC=C)C)=O)C2)C3)=O)cc(F)cc2[nH]ccc12 95783,C1(C)(C(N(C(C)C(=O)N(C)C)CC)=O)CCN(C(C2CC(=C3CC3)C2)=O)CC1 95784,c1(CC(=O)NC(C)CC(=O)NCCC(O)c2cccs2)ncccc1F 95785,C1(C(N(C(C(N)=O)C2CCCC2)C)=O)CCC1NC(C1(CC2CC2)CC1)=O 95786,N1(C(=O)Cc2ccc(C)o2)CCC(NC(C2(C(=O)OCC)CC2)=O)C(C)C1 95787,N1(C(CCCc2ccc(C)s2)=O)CCCC(C2(NC(c3cnc(O)s3)=O)CC2)C1 95788,c1(NC(C(N2CCC(C3(C)OCCO3)CC2)C)=O)nc(C(F)(F)F)ccc1I 95789,c1(OC)ccncc1C(=O)NCc1nocc1C(N1CCC1(C)C(N)=O)=O 95790,CC(C)CC(C)(O)C(=O)N1C2CCC(C(=O)NCc3cnns3)C1CC2 95791,N1(C(Cc2cc(C)ns2)=O)CCC2(NC(=O)CCn3cccn3)CCCCC12 95792,c1(OC)cc(C=CC(=O)NCCCCCCNC(=O)CC(C)N(C)C)ccc1O 95793,N1(C(CC(COC)(C)O)=O)CCC(N=[N+]=[N-])(C(=O)NOCC=CCl)C1 95794,Cn1ccc2[nH]c(C(N3CCC(NC(C4(n5cccn5)CC4)=O)C3)=O)cc12 95795,c1(CNC(CCC2N(C)CCC2)=O)ccc(C(=O)NCC(N2CCCC2)C)nc1 95796,C(C(=O)N=c1cc(C)n(C2CC2)[nH]1)=CCN(CCC)C.C12CCCCC1NC2=O 95797,N1(C(c2c(C)cccn2)=O)CCC2CCC(NC(=O)C(F)(F)Br)C12 95798,Cc1nscc1NC(C(CC1(C#N)CC1)N(CC(=O)OC)C1CC1)=O 95799,c1(C(N2CC3C(CNC(C=COCC)=O)(C3)C2)=O)cc(Cl)cc(Cl)c1OC 95800,CC1(NS(C)(=O)=O)CCCC1(F)F.c12ccc(cc1)c(=O)n2C(c1ccco1)=O 95801,c1(C(N(CCCn2cncn2)C)=O)ccc(CNC(=O)C=C2CCC2)nc1 95802,CN1CCC(C(=O)NC(C)(C)CCCCNC(=O)C(F)CC2CCC2)C1=O 95803,c12cc(c(F)cc1F)C(=O)CN2.C(CCCC(=O)OC(C1CCOC1)=O)SC 95804,Cc1ccc2c(Cl)c(C(=O)NC3CCC34CN(C(=O)Cc3cnc[nH]3)C4)sc2c1 95805,c1(NC(C2CC2NCc2csc([N+](=O)[O-])c2)=O)cccc(Cl)c1I 95806,c1(C2CN(C(C3CC3(F)c3ccon3)=O)C2)nc2c(s1)C(CCCN)CCCC2 95807,N1(C(COCCOC)=O)CCC2(CNC(=O)C3=NNC(=O)CC3)CCCCC12 95808,c1(NC2CN(C(c3nc(COC)sc3)=O)CC2C)ncnc(N(C)C)c1[N+](=O)[O-] 95809,c1(CN2CCC(F)(C(N3CCC(F)CC3)=O)C2)cnc(Cl)cc1Cl 95810,c1(C(=O)OC)cccc(NC(=O)C(c2ccc(OCC(F)F)cc2)C)n1 95811,Cc1c(C(=O)NC2CC(CNC(=O)CSC3CC3)C2)[nH]c2c(F)cc(F)cc12 95812,c1(C(=O)NCC2CN(C(C(F)(F)C3(OC)CCC3)=O)CC2C)cccc(Cl)c1F 95813,N1(C(CC2(C=C)CCC2)=O)CCC(C2(NC(=O)C(C)O)CC2)C1 95814,c1(OC)cc(-c2ccc(Cl)c(C(C)=O)c2)ccc1O 95815,c1(CC)nn(C)cc1C(N1CCOCC1CN(C)C(c1cccnc1NC)=O)=O 95816,N1(C(c2c(O)ncc(NC(C)=O)c2)=O)CCC2(CCN(C(=O)C(O)CSC)C2)C1 95817,c1(C(N(CC(CNC(c2c(O)ccc(CC)c2)=O)C)C)=O)cc(S(N)(=O)=O)co1 95818,c1(OC)cc(CC(=O)NOCc2ccccc2)cc(Br)c1OCc1cccc(F)c1 95819,C1(OC)CCC(C(=O)NCC2CCCCC2NC(=O)CSC2CC2)CC1 95820,Cc1ccc(Cl)c(N)c1C(N1CCC(CNC(=O)C(C)C(F)F)C(F)(F)CC1)=O 95821,C=CCCC(C(=O)NCCCOCCN(C(=O)CC(=C)Br)CC)c1ccccc1 95822,C1(CNC(C(C)(C)C#N)=O)CCCCN(C(=O)CC2SC(=N)NC2=O)C1 95823,c1(C(CNC(c2ccc(F)cc2F)C(=O)OC)=O)cccc2nsnc12 95824,C1(C(=O)NC2(C(N(CCC#C)CCOC)=O)CC2)CC1C#N 95825,CCC(C)(O)C(=O)N(C)CCN(C)C(c1cnn(-c2ccc(Cl)cc2)c1C)=O 95826,C1(NC(c2cnn(C)c2F)=O)CCC2CC1CN2C(c1cc([N+](=O)[O-])c[nH]1)=O 95827,c1(CC(=O)NCCOCCNC(C2ON=C(CC)C2)=O)n[nH]c2ccc(Cl)cc12 95828,Cc1csc(CC(=O)N(CC(C)N(C(=O)Cn2ccnc2C)C)C)c1 95829,CCCCCCCCN(C(=O)C(CC1CCC1)OCC(C)SC)C.C1(=O)C(C)O1 95830,C1(C(=O)NCCC(C)NC(c2cscc2C(F)F)=O)CC(c2ccccn2)=NO1 95831,N1(C(C(CCOCC)NC(=O)C(C)n2cnnn2)=O)CCn2nc(C)nc2C1 95832,Cc1cc(C(=O)NCCN2CCN(C(C3CCNC3=O)=O)CC2)cnc1O 95833,N1(C(C(C=CC)O)=O)CCCC2(CCN(C(=O)C=CSc3ccccc3)CC2)C1 95834,C1(C(CNC(c2c(C)occ2)=O)F)CCN(C(=O)CCC2CCCCO2)CC1 95835,C(=O)(C(F)(F)C(O)C1CC1)NCC(C)NC(=O)CCc1cc(Cl)cs1 95836,C1(C(N2CC3CC(NC(C(C)OCCOC)=O)C3C2)=O)CN2CCCN1CC2 95837,CC(C)CN=C(NCC1(CCOC)CCCC1)N1CC(C)N(CCO)C(C)C1 95838,CCC(CC(C)C)C(=O)NCC1CC2(CC2)CN1C(c1cc(CSCC)on1)=O 95839,C(CC(C)C)(C(=O)N1CC2CC(NC(c3ncc[nH]c3=O)=O)C2C1)NC(C)=O 95840,C1(CNC(CC(C)N(C)C)=O)CN(C(c2n[nH]c3c2COCC3)=O)CC(C)(C)O1 95841,CCCC(C(C(=O)NCC)N1CC(O)C2(CCC2)C1)OC 95842,c1(NC(C=CC(N2CC(=C(CNC(C(CC)OC)=O)F)C2)=O)=O)ccc(F)cc1C 95843,C(=O)(C(F)(F)C(F)(F)F)NCCC1CN(C(C2CC(OC(C)(C)C)C2)=O)C1 95844,N1(C(C=CC(CC)C)=O)CC(O)(C(C)(C)CNC(C23CCC2C3)=O)C1 95845,N1(C(C2(C)CCCCO2)=O)CC2(CCCC2NC(C2(C3CCC3)CC2(F)F)=O)C1 95846,c1(C(=O)NC2C(NC(CCc3n(C)cnc3)=O)CCC2)c(F)cc(F)cc1Cl 95847,C1(CNC(COCC)=O)CCN(C(=O)COCc2ccccc2)CC1 95848,Cc1cc(C(N2CCN(C(=O)CCC3CC3CC3CC3)C3CCC23)=O)ccc1C#N 95849,CC(C(=O)N1CCC(n2cc(-c3ccc(Br)cc3)nn2)CC1)C(F)F 95850,N1(C(=O)CC2(O)CC2)CC2(CCN(C(c3ccc(Br)cc3F)=O)CC2)C1 95851,N1(C(C(Cn2ccc(C)n2)C)=O)CC2CN(C(c3ccc(C)c(O)c3)=O)CCC12 95852,N1(C(C=CC=CC)=O)CCCC2(NC(=O)C=CC(CC(F)(F)F)=O)CCCC12 95853,c1(C(N2CC=CC(NC(CC3(COC)CCCC3)=O)C2)=O)cn2ccncc2n1 95854,N1(C(Cn2cnc(=N)[nH]2)=O)CCC2(NC(c3ccc4nc[nH]c4n3)=O)CCCC12 95855,c1(OC(C(=O)OCCCC(C)O)Cc2ccccc2)ccc(Cl)cc1 95856,c1(C(=O)NC(CC(C)C)CNC(C2(C)CCCCO2)=O)ccc([N+](=O)[O-])s1 95857,c1(C(=O)NC(CNC(C=CC(CC)=CC)=O)C2CC2)nc(Cl)sc1C 95858,c1(C(N2CCC(CCOC)C2)=O)n[nH]c2c1CN(C(=O)CCc1cccnc1)C2 95859,N#Cc1ccc(F)c(C(=O)NCC2C3CN(C(=O)Cn4cc(Br)cn4)CC23)c1 95860,CC1C(NC(=O)CC2=CCCC2)CC2CCC1N2C(=O)CC1CCC2CC12 95861,C12(CNC(c3ccc(C)c(F)c3)=O)CCCCC1N(C(=O)C=CC1CC1)CCC2 95862,c1(COC)cc(Cl)ccc1S(=O)(=O)N1CC(Cn2cc(Br)cn2)C1 95863,C(N=c1[nH]c(=N)[nH]c(Cl)c1[N+](=O)[O-])C1CC2(CC(NC(C=CCN(C)C)=O)C2)C1 95864,c1(OC)ccccc1C(=O)NCC1(Nc2cc(Cl)ncn2)CC1 95865,CCCS(=O)(=O)CC(=O)NC1CCC(NC(=O)CC2OCCC2(C)C)CC1 95866,C1(N(C)C(c2cc(C(C)(C)C)on2)=O)CCC(NC(=O)CCCC#N)CC1 95867,c1(C(=O)NC(CNC(c2c(CC)c[nH]n2)=O)C(C)C)ccc2c(c1)C(C)C(C)O2 95868,C1(CNC(c2ncn(CC)n2)=O)CC12CCN(C(c1c(C)nnn1CC)=O)CC2 95869,CN1CCOCC1CC(=O)NC1CCN(C2CCN(C(=O)C(F)=CC3CC3)C2)CC1 95870,C1(NC(c2ccn(CC)n2)=O)CCCCC12CCCN(c1cc(C)nc(C)n1)C2 95871,N(C(=NCCOC(F)F)NCC(Cc1ccccc1)C(C)C)CC(CC)(C)C 95872,c1(C(=O)NNC(=O)C2CC(O)CN2CC(F)(F)F)cc(F)cnc1Br 95873,C1(C(=O)NCC(C)NC(c2c(CCC)n[nH]c2)=O)CC12CCC1(CC1)CC2 95874,Cc1cc(C(=O)NC2(c3cc(Br)ccc3Cl)CC2)cc(C)c1N 95875,c1(C2(C(N3CCC(C)(NC(c4snc(Cl)c4Cl)=O)C3)=O)CC2)ccc([N+](=O)[O-])cc1 95876,CC(F)(CC1CCCC1)C(=O)NCC1C=CCN1C(c1nc(=N)cc[nH]1)=O 95877,N(C[Si](C)(C)C)C(CCC1(NC(C2(Cl)C(C(C)=O)C2)=O)CCC1)=O 95878,C1(CNC(C2N(Cc3cnc(OC)nc3)CCOC2)=O)C2CCCCCC12 95879,C1(C(N(C2CCN(C(Cn3ccc(C)n3)=O)C2)C)=O)CCC(CCC#N)CC1 95880,CC(CC=Cc1ccccc1)C(=O)NCCC1CCCN(C(=O)C2CC2)C1 95881,N1(C(C(=Cc2ccncc2)C)=O)CCN(C(c2cn(C)nc2Cl)=O)C(C2CC2)C1 95882,c1(N(C2CNCC(F)(F)C2)C(C(c2cccc(C)n2)(F)F)=O)nccc(C#N)n1 95883,C1(C(=O)NCC(CCOC)OC)CC2C=CC1N(C(c1ccccn1)=O)C2 95884,C1(CNC(c2c(CC)nn(C)c2)=O)N(C(=O)CC2CC(C)=NO2)CCC1(C)C 95885,N1(C(c2c(CNC(CC(C)C3CCCO3)=O)n[nH]c2)=O)CCC2(CCN(C)C2)C1 95886,c1(NCC(CC2(CC)CC2)(C)C)ccc(S(=O)(=O)N2CCCC(C)C2C)c(Cl)c1 95887,c1(C(N2C(C(=O)Nc3c(C)cnc(F)c3)CNCC2)=O)cc(Br)cc(Cl)c1Cl 95888,C1(CNC(C=CCN(C)C(N)=O)=O)CCCN1C(=O)Cc1ccccn1 95889,c1(OC(C)C(=O)OCC2CON(C)C2=O)cccc(Br)c1 95890,N1(C(COCC(=O)NC)=O)CC(C(=O)NC2CCC(=O)NC2=O)C(C)(C)C1 95891,c1(C(=O)NC2COCC2NC(=O)C(F)(F)C2CCCO2)c(F)cccc1Cl 95892,C1(C(N2C(C(=O)NC3(C)CC(O)(CO)C3)CC3CC32)=O)C2CCCC(=O)C12 95893,N1(C(CCC(=O)NC)=O)CC(C)CN(C(c2cc(CO)ccn2)=O)C(C)C1 95894,C(c1csc(C)n1)=CC(=O)NC(CCNC(c1n(CC)cnn1)=O)C 95895,c1(OC)cncnc1C(N1CC2CC2(CNC(=O)CCc2ccc(C)cc2)C1)=O 95896,c1(C(=O)NCC(O)CC2CCOC2)cc(Cl)sc1Br 95897,c1(OCC)ccc(OCC(N2CC3C(CN(C(=O)COC)C)C3C2)=O)cc1 95898,N1(C(C2(CCCC)CCC2)=O)CC(N=[N+]=[N-])CC1C(=O)NC(COC)C1CC1 95899,C1(CCNC(c2c(CC)con2)=O)CN(C(C2CC(F)CN2C)=O)CC1C 95900,c1(C(=O)NC2CCCN(C(c3cc(CCC)[nH]n3)=O)C2C)c(C)ccc(C)c1N 95901,c1(C(N(CC(C)(C)CNC(=O)CSC(C)C)CC)=O)cnc2c(C)cccc2c1 95902,CC(CCNS(=O)(=O)Cc1ccnc(Cl)c1F)P(C)(C)=O 95903,N1(C(C2(CC)CC2(F)F)=O)CC(C)(C)OC2(C1)CN(C(=O)C1=CCS(=O)(=O)C1)C2 95904,C1(C)(C(N(CC(C)O)CCNC(=O)Cc2ccno2)=O)CCC(=O)N1 95905,c1(C(=O)OC)nc(I)cnc1NC(C1CC(NC(c2conc2C)=O)C1)=O 95906,N1(C(=O)CCSC2CCCC2)CC2(CCN2C(c2ccccc2C(F)F)=O)C1 95907,C(c1scnc1C)=CC(=O)N(CC(C)(C)NC(c1c(CC)occ1)=O)C 95908,c1(C(=O)NC2C(NC(c3cc(Cl)cs3)=O)COCC2)ccc(F)c2c1CCC2 95909,C(=O)(CC1=CCOCC1)N1CCC(O)(C(C)NC(=O)Cc2c[nH]nc2O)C1 95910,Nc1ccc(C(=O)NCC2CN(C(c3scnc3Cl)=O)CC23CC3)c(Cl)c1 95911,C(CCC)(C(O)C(=O)NC(CC(=C)C)C(=O)OC)NC(C(C=C)(C)CC)=O 95912,n12nc3n(c1=O)CCN(C3)C(=O)NCC2C.C(C(=O)OCC(F)F)C(C)(C)C 95913,CC1CC=C(C(=O)NC(C2CCCC2)CNC(=O)CSC(C)(C)C)CC1 95914,Cc1ncc2cc(C(N3CCC(Cn4cc(C5CC5CO)nn4)C3)=O)nn2n1 95915,c1(CC)nn[nH]c1C(=O)N(CCC(C)NC(C1CC1CCOC(C)=O)=O)C 95916,CCC(C)CCC(O)CC(=O)NCC(O)CNC(c1cc(Cl)ccc1Cl)=O 95917,N1(CC)CCOC(C(N2CC(OC)C(C(=O)NCC(C)CC3CCCC3)C2)=O)C1 95918,c1(CC(=O)N(C)CC2CC(F)CN2C(C2OCC2(C)C)=O)nc([N+](=O)[O-])n[nH]1 95919,C1(C(=O)NCC(CC)(CC)NC(=O)CCNC(C2CCC2)=O)OCC2COCCC12 95920,Cc1cc(=NCc2cnc(C(F)F)s2)[nH]c(NC2CCS(=O)(=O)C2(C)C)n1 95921,C1(C(=O)NC(CN(C(=O)CCSCC(N)=O)C)(C)C)CN2CCC1CC2 95922,C1(NC(CCCN(C(=O)CCC(F)(F)F)C)=O)CC2CCC(C1)N2C 95923,C1(C2CCOCC2)(C(N2CC3(CN(C(C4CC4F)=O)C3)OCC2)=O)CCOCC1 95924,CC1CCc2onc(C(=O)N(CC(C)NC(c3ccc(Cl)cn3)=O)C)c2C1 95925,C(C(N=[N+]=[N-])C(=O)NC(CSCCOCC)=O)NC(CNC1(COC)CCC1)=O 95926,C1(C(N2CCC(NC(C(CCC)NC(C)=O)=O)C2)=O)CC(F)(F)C1(F)F 95927,C=CCCC(O)CN(C(=O)C(CC1CCCC1)NC(C1CCCN1CC)=O)C 95928,C#CCC(C)(C)C(=O)N1CC(C(N2CC(C(F)(F)F)C2)=O)C2(CC2)C1 95929,C1(CCC=C)(NCc2cc(Br)cs2)CN(C(=O)OC(C)(C)C)C1 95930,C(C(C)N(C)N1CCCC1C1CCCCN1Cc1ccccc1)n1c(C)ncc1 95931,O(N=c1ncnc2[nH][nH]c(Br)c1-2)Cc1ccc(-c2c(Cl)c(C#N)c(F)c(F)c2)s1 95932,c1(OC(CCN(CC)CC)=O)ccc(F)c(C(F)F)c1F.C12CC(C1)NC2=O 95933,c1(N2CC(=O)N(CC(C)C)CCC2=O)nnccc1C#N 95934,N1(C(CCCOCC)=O)CC(C)C(C)(CNC(=O)CCc2ncc(C(C)C)o2)C1 95935,c1(C(=O)NC2CC(NC(CCc3c(OC)cccc3)=O)C2)nc(Cl)ccc1N 95936,N1(C(CC(C(C)C)O)=O)CC2CC(NC(=O)COCP(C)(C)=O)CC2C1 95937,N12CCC(C(C)C1)NC(=O)C2.c1(C(=O)OC)ccsc1OC 95938,C1(C(=O)NC2CC(C(C)C)OC2)CN(C(C2(C(C)(F)F)CC2)=O)CC1F 95939,C1(C(=O)NC23CC(NC(C(C)c4ccsc4)=O)(C2)C3)CN2CCN1CC2.C1(C)CC1 95940,Cc1nc2ccc(C(=O)NC(C)C(C(C)C)NC(=O)CC(C)C)cc2c(=O)n1C 95941,C1(C(N2CC(C(C)NC(C3(C)CC3)=O)OCC2)=O)CC2CC(=O)C1O2 95942,O=C(NNC(=O)C12CCCC1C2)c1ccccc1 95943,CC(C)CCCC(C)C(=O)NCC1CN(C(c2ccc(CO)o2)=O)CCCO1 95944,N1(C(CNS(CC)(=O)=O)=O)CC2CN(C(c3cnc(OC)nc3C)=O)CC12 95945,c1(C(=O)NC2(C)CCCN(C(c3cc(C(N)=O)[nH]n3)=O)C2)cc(F)c(F)c(F)c1 95946,C12(NC(C3CCS3(=O)=O)=O)CCCN(C(c3cc4ccsc4s3)=O)CC1C2 95947,c1(N2CC(NC(C(C3CC3)OC)=O)(CO)C2)nc2ccc(Br)cc2o1 95948,C1(NC(C2(COC)CC2)=O)CC(O)CN(C(c2c(OC)ccnc2O)=O)C1 95949,CCCC(C(=O)N1CCCC1C(C)NC(=O)C=Cc1cccc(F)c1)S(N)(=O)=O 95950,C(=O)(CC(C)C(C)C(C)C)N1CCC(NC(c2cn(CC)nn2)=O)C(C)C1 95951,C(CC(C)C)(C(=O)NCCN(C(C)C)C(C)C)NC(c1c(C)nccn1)=O 95952,CC(C)CC(CC(=O)NC(C(N)=O)C1CC1)NC(C1COCCC1C)=O 95953,C(=O)(CCC(=O)c1cccnc1)NCCCC(C)NC(=O)C(F)n1cccn1 95954,CC(C)(C#N)C(=O)NCCOCCNC(C1CC(O)(c2ccncc2)C1)=O 95955,N1(C(CCCC(=C)C)=O)CC2(CCN(C(=O)C(C(C)(C)C)N(C)C)CC2)CC1C 95956,C1(F)(CNC(CSCC)=O)CCN(C(c2ccc(Oc3cccnc3)cc2)=O)C1 95957,C1(NC(CCCCNS(C)(=O)=O)=O)CCCCN(C(C2(C3CC3)CCC2)=O)C1 95958,N1(C(c2nc(COC)oc2)=O)CCOC(CN(C)C(C2COCCN2C)=O)C1 95959,C1(NC(CCC(C)C)=O)CN(C(C2CCCN(S(C)(=O)=O)C2)=O)CCC1C 95960,c1(C(=O)NCC2(NC(=O)C(O)CF)CCCCC2)ccc2nc(O)[nH]c2c1 95961,c1(C(N2CCC(OC)(CNC(c3ccc(C)nc3O)=O)C2)=O)ccc(N)c(O)c1 95962,C1(NC(C(C2CC2)SC)=O)CCCC(NC(=O)CNC(=O)CNc2ccsn2)C1 95963,C(C(=O)N1CCC(Cn2cc(-c3cnsc3)nn2)C1)(C(C)C)SC 95964,C(CN=C1NC2CCCCC2N1)NS(CCCC)(=O)=O 95965,N1(C(c2cncc(C)c2C)=O)C2CCC1CN(C(=O)Cn1nnnc1C)C2 95966,N1(C(C(CC)(C)F)=O)CC(CNC(=O)COCCOCCO)OC(C)(C)C1 95967,C1(N(C(=O)CCC2CCC(=O)C2)C)CCCN(C(=O)CN2C(=O)CNC2=O)CC1 95968,C1(COC)CCCCN(c2nnnn2CCc2ccc(O)nn2)C1 95969,C1(C2CCC2)(C(=O)NCC(CC)(C)NC(c2cccc(C(C)C)n2)=O)CC1 95970,c1(C(=O)NC2CC(CNC(C(C=C)(C)C)=O)C2)sc2ccc(C(C)=O)cc2c1C 95971,C1(CNC(C2(C(CC)=O)CC2)=O)(NC(c2cnc(OC)s2)=O)CCCC1 95972,c1(OC)ccc(F)cc1CC(=O)NCC1CC(C)N(C(c2cnncc2O)=O)C1 95973,Cc1cccc2[nH]c(C(=O)NC3CC3CNC(C3CCCC(C)(C)C3)=O)cc12 95974,C1(NC(C2C=CCC2)=O)CC2CC(C1)N(c1nccc(CO)n1)C2 95975,C(c1nc2ccccc2s1)=CC(N1C(CNC(c2c(C(N)=O)scc2)=O)CC1)=O 95976,C1(C(=O)NCc2c(C)nns2)CCN(C(C2CC2(Cl)Cl)=O)C12CCC2 95977,N1(C(C2CCCC(C)(C)C2)C(=O)NCC)CCOc2ccccc2C1C(=O)OC 95978,Cc1nn2c(c1C(=O)NC(C)CCNC(C1(O)CCC1)=O)CCCC2C 95979,N1(C(c2ccc(OC)c(C)c2)C(=O)NC2CCCC2)CCC2(CC(=O)N(C)C2)C1 95980,c1(OC)ccc(C(N2CC(NC(=O)CC(C)F)C(C)C2)=O)c(OC)c1 95981,Cc1ccc2sc(=NCC3CCN(C(=O)Cn4ccnc4C4CC4)C3)[nH]c2c1 95982,N1(C(c2c(C)c[nH]n2)=O)CC(NC(C2(c3ccccc3)CCCC2)=O)CC1(C)C 95983,CC1CCC(C(C)(O)CNC(=O)COC(C)(C)CNC(c2cnnn2C)=O)CC1 95984,c1(CCCC(N2CCOCC(NC(CCCOC)=O)C2)=O)cccc2sccc12 95985,CC1=C(C(=O)NC(C)CN(C(=O)C(C)N(CC(F)(F)F)C)C)S(=O)(=O)CCO1 95986,C1(CN(C(C2C3(CC3)C23CC3)=O)CC)CCCN(C(C2CCC(=O)N2)=O)C1 95987,C1(OC)CCC2(C(=O)NCCCN(C(=O)CN3CCOCC3)C)CC12 95988,C(=O)(C1Cc2ccccc21)N1CCC(C)(CC(=O)N(C)Cc2c(C)nsc2)C1 95989,c1(C(=O)NCC(CCC=C)O)nc2c(s1)CC(=O)CC2 95990,S(=O)(=O)(c1ccc(Cl)cc1F)N1CC2N(C(C3CCC(=C)CC3)=O)CC(C2)C1 95991,c1(NC2CC(C(=O)OC(=O)NC(C(=O)NC(C(=O)OC)C)C)C2)ccc(C#N)cc1 95992,N1(C(c2c(OC)nsc2)=O)CCN(C(=O)CCN2CCCC2)C(CC(C)(C)C)C1 95993,c1(CN2CC3(CCN(C(CC(=O)OC)=O)CC3)C2)cccc2cccc(C)c12 95994,c1(C(C(=O)NCC2CC(NC(CSCC(N)=O)=O)C2)=O)ccc(Cl)cc1Cl 95995,C1(CC(=O)NC(C=C)COC)C=CC(N(C(=O)C=Cc2ccsc2)CC)C1 95996,c1(C(N2CCC(C)(NC(CC(=C=C)C)=O)C2)=O)cc(OC)ccc1OC 95997,C#Cc1cccc(C(=O)NCC(N2CCN(C(C3CCCOC3)=O)CC2)=O)c1C 95998,c1(OC)nccnc1CNC(c1csc(C(=O)NCCc2ccc(Cl)s2)n1)=O 95999,Cc1ccc(C)c(C(=O)NCCCOCCN(C)C(c2nccnc2C)=O)c1 96000,C#CCC(C(=O)NCC1CCN(C(=O)CC(OCC)OCC)C1)C1CC1 96001,C1(CCC)(NC(=O)CCCCN(C)C)CCN(C(=O)CNC(=O)C2CC2)CC1 96002,C1(COC)(CNC(=O)CC(C)SC)CCN(C(=O)C(C)CC(C)C)CC1 96003,CC1(C)CC(NC(C2CC=CCO2)=O)CN1C(=O)CCC(=O)N(CCO)CCO 96004,c1(C(=O)NC2CN(C(C)=O)C2)ccc2cccnn12.N12CC(C3CC13)C2=O 96005,c1(OC)ccc(C(N2CCCC(CNC(=O)CCc3ccoc3)C2)=O)c(Br)c1 96006,c1(-n2cc(C3CCN(C(=O)Cc4cnc(Cl)s4)C3)nn2)ccncc1Cl 96007,N1(C(C=CC(C)(C)SC)=O)CCCN(C(c2c(F)ccc(Cl)c2F)=O)C(C)C1 96008,c1(C(=O)N)cnn(C)c1.c1(CC2(C(=O)NC(C(C)OC(C)C)C)CC2)ccccc1 96009,CC1(C)OC(=O)CC1C(N1CCC12CN(C(=O)CCc1ccc(Br)nc1)C2)=O 96010,C1(OCC(=O)NC2CC(C(=O)OC)C2)CCN(C(c2ccnnc2)=O)CC1 96011,c1(CC)oc(C)cc1C(N1CC2CC2(CNC(c2cc(OC)n(C)n2)=O)C1)=O 96012,C1(NC(c2ccc(C(n3cncn3)=O)o2)=O)CCCC1n1cc(CCCO)nn1 96013,C1(CNCC(CN(C(C)=O)C)C)C2CC3CC(C2)CC1C3 96014,c1(NCC)cnc2scnc2c1.N12CCCCC1CCCNC(=O)SCCC2=O 96015,CC(CC(F)F)C(=O)NCC(CO)NC(=O)Cn1ccc(Br)cc1=O 96016,C(=O)(CCCCC(N)=O)NCC(S(C)(=O)=O)CNC(C1CC1C#N)=O 96017,Cc1cccc2ncc(C(N3CCC(C)CC3CNC(c3c[nH]c(=N)o3)=O)=O)n12 96018,C1(CNC(CC(=C)C)=O)CCC2(CO1)CC(NC(=O)C=CC1CCC1)C2 96019,N1(C(Cc2ccc(C(=O)NC)cc2)=O)CC(CNC(=O)Cc2cncs2)C2CC12 96020,CCCC(C)(CC)NC(C1(CO)CCN(C(=O)CCc2ccoc2)C1)=O 96021,C(C(CNC(C1CC(OC)C1)=O)S(C)(=O)=O)NC(CCCC=C)=O 96022,C(=O)(C1CCCc2c[nH]nc21)NC(C1(CNC(=O)C(C)C(C)n2cccn2)CC1)C 96023,Cn1nc(CNC(C2(C)C=CCC2)=O)c2c1CCN(C(c1ccc(O)cc1)=O)C2 96024,C1(NC(=O)C=Cc2cnc[nH]2)CC2(C1)CC(C(=O)NCC1CCC(F)(F)C1)C2 96025,c1(C(N2C(C(N(CC)Cc3nccn3C)=O)CCC2)=O)cc(O)cc(F)c1 96026,c1(C(N2C(C(=O)NC3CCN(C4(C)CC4)C3=O)CCC2C)=O)cnc(S)nc1 96027,N1(C(CCC2CCN(C(C(c3ccccc3)C)=O)C2)=O)CC2COC(=O)C2C1 96028,N1(C(C(c2n(C)ncc2)NC(=O)CSc2ccc(O)cc2)=O)CCC(F)(F)C(O)C1 96029,C1(OC)CN(C(c2ccc(F)cc2)=O)CC1C(N1CCC(F)(CO)C1)=O 96030,Cc1cc(F)c2nc(O)cc(C(=O)NC3CCCN(CC(F)F)C3)c2c1 96031,c1(C(=O)NC2C(F)CCN(C(CCC(C)C)=O)C2)ccc(Cl)c(C)c1F 96032,C(=O)(NN1CCCN(C)CC1)Nc1c(-c2c(C)ccnc2)nc(C(C)C)s1 96033,c1(C(=O)NC2CC(C)N(C(=O)CNC(C3CCCC3)=O)C2)csc2nccn12 96034,c1(C(=O)NC2C(NC(=O)Cn3ncnn3)CC(F)(F)C2)cnc2c(F)cccn12 96035,N1(C(Cc2cc(CC)no2)=O)CCC(C2CC2)C1CNC(=O)C(C)(C)NC(C)=O 96036,c1(C(N2C(C)CC(C(N3CC(CC)N(C)CC3)=O)C2)=O)cccc2[nH]ncc12 96037,C1(NC(=O)C(F)n2cccn2)C2CC(O)C1N(C(=O)CCc1ccc(O)nc1)C2 96038,C1(NC(CC(=C)C)=O)CC2C(NC(C3CC(=O)N(C4CC4)C3)=O)C2C1 96039,C(C(C)(C)C(=O)N1CCC(C)C1)OC(C1CC(C(=O)OCC)C1)=O 96040,c1(NC(N2C(CNC(C3N(CC)C(=O)CC3)=O)CCC2)=O)cccc([N+](=O)[O-])c1 96041,c1(C(=O)NCC2CN(C(COCCCCC)=O)CC2O)onc2c1CCCC2 96042,c1(NC(C2CCCN2C(c2cnccc2C#N)=O)=O)ncc(F)cc1Br 96043,N1(C(CCC=C)=O)CCn2cc(C(N3CCC4(CCCO4)C3)=O)nc2C1 96044,N1(C(C2C(c3nc(CC)sc3)OCC2)=O)CCOc2c(F)cccc2C1 96045,N1(C(CNC(C(C)Cc2ccccc2)=O)=O)CCN(C2CCN(CC#N)C2)CC1 96046,C1(O)(CNC(c2ccsn2)=O)CN(C(=O)C(F)(F)C23CC(C2)C3)C1 96047,N1(C(c2c(Cl)cnc(C)n2)=O)CC2(CCC2)CC1CNC(=O)CCc1ccon1 96048,C1(NC(c2cnccn2)=O)CCC2(CC1)CN(C(c1ccoc1Cl)=O)CCO2 96049,c1(CNC(=O)NCC2(C)CC(OC)(OC)C2)ccc2nsnc2c1 96050,n1(CC(=O)NCC2CC(NC(CC(C)CF)=O)C2)nnc2c1CCCC2 96051,C1(CCC)CN(C(=O)Cn2cnc(=N)[nH]2)CC1NC(C1(C)CCCO1)=O 96052,C12(CNC(CSCC=C)=O)CC1CN(C(c1cc(C3CC3)nn1CC)=O)C2 96053,N1(C(C2CCC(OCCCC)CC2)C(=O)NC)CC2C3C=CC(C3)C2C1 96054,C#CCCCC(=O)NCCCN(CCCNC(=O)C(C)(C)NC(=O)C=COC)C 96055,C1(NC(C=C(CC)CC)=O)CCC2CC1CN2C(=O)CC1(C)CC1(Cl)Cl 96056,c1(NC(N2CCC(CCC)(CO)C2)=O)cc(O)nc2cnccc12 96057,C(=O)(CC(O)C(Cl)(Cl)Cl)N(C(c1cnn(C)c1)C(=O)NCCNN(C)C)C 96058,C1(C(=O)NCC(CC)O)CCCN(C(c2nnn(C(C)C)c2C)=O)C1 96059,O=C1CN(C(C2CCC3(CC3)C2)=O)C(C(N2CC(CO)(CF)C2)=O)CN1 96060,C(=O)(C1CSc2ccccc21)NC(CNC(c1cccc(S(C)=O)c1)=O)(C)C 96061,C1(C(=O)NC2CC3(C(NC(CSCCOC)=O)C3)C2)CCc2nn[nH]c2C1 96062,c1(OC)ccc(F)c(C(=O)NC2CC2CNC(=O)CCOC(C)CC(C)C)c1Cl 96063,C1(CN(C)C(C2CCOC2)=O)CCC(CNC(=O)Cc2cccn2C)CC1 96064,CC1(C(=O)NCCC2(O)CCN(C(=O)CC3CSC3)C2)CCC(F)(F)CC1 96065,C1(C)(C(=O)NC2(C(=O)NC3CC(OC)C3)CSC2)CCCCC1 96066,C1(C(=O)NCCCC(C)(C)NC(CN(C(=O)OC)C)=O)CCC2(CC1)CC2(F)F 96067,c1(-n2cc(C(C)N(C)C)nn2)ccccc1C(=O)NC(C)CCO 96068,CCC(C(=O)OC)C(=O)N1CCCCC1C(=O)N(CC)Cc1ccc(C)nc1 96069,C(C)(c1ccc(F)cc1F)=CC(=O)N(CC)CC1CCN(C(=O)C=CCF)CC1 96070,C#CCCCCC(=O)NC1CC(C(F)C(=O)NC(CCC)C(=O)N(C)C)C1 96071,C12(C(=O)NCC3C(C)CN(C(C4CCC5(CC5)C4)=O)C3)CCC(CC1)OC2 96072,C1(OC)CC(C(=O)NC2(n3cc(C)cn3)CC2)N(C(=O)CC(C)n2cccn2)C1 96073,c1(OC)cc(F)c(Br)cc1S(=O)(=O)N1CCOCC1C 96074,N1(C(CC(C(=O)OC)C)=O)CCC(C)(C)CC1C(=O)NCC1CC1(C)C 96075,C1(NC(C)=O)CC(NC(c2ccc(OC(F)F)cn2)=O)C1(C)C 96076,C(=O)(CC(C(F)(F)F)c1nccn1C)N1CCN(C(C(CC)CC)=O)C2C1C2 96077,S(=O)(=O)(CCCCF)C(NNC=O)=O.NC1(CO)C2CC3C(C2)C13 96078,CC#CCC(C)N=c1[nH]c(=NC)[nH]c(=NCc2sccc2S(C)(=O)=O)[nH]1 96079,c1(NC(C(CCC)NS(=O)(=O)c2ccc(C)s2)=O)cc2cccnc2c(Br)n1 96080,N1(C(c2ncoc2C2CCCO2)=O)CC2CCC1CN2C(C1CC2CC1CO2)=O 96081,C1(COC)C2CCCC2CN1C(=O)C(CC)C(=O)OC(C)(C)C 96082,N1(CCC(=O)NC(CC(C)NC(Cc2ccn(CC)n2)=O)C)CCN(C)CC1 96083,N1(C(c2n(CC)ncc2Cl)=O)CCC(C2CCN(C(=O)C=CC3CC3)C2)C1 96084,Cc1coc(C(C)C)c1C(=O)NCC1CN(C(=O)C(C)OCCC(C)C)CCO1 96085,N1(C(C2C(OC)CC2)=O)C2CCC1C(F)C(NC(=O)Cc1cnccn1)C2 96086,CC1C(=O)CCC(C(=O)NCCCOCCCNC(=O)C(C)(F)F)C1(C)C 96087,c1(COC(c2cc(F)ccc2F)=O)ccc2c(c1)OCCCO2 96088,CC1(C)C(NC(=O)C2=CCSC2)CCN1C(=O)CCc1ccc(F)nc1 96089,Cc1ccc(OC(C)C(=O)OCc2coc(-c3ccccc3F)n2)c(F)c1F 96090,c1(NC(=O)Cc2ncccn2)ccc(CCN(C)C)cc1.C12CN(C1)C(=O)CO2 96091,C(C1C(C(N2CC(CCO)(NC(=O)C(=CC3CCCC3)C)C2)=O)C1(C)C)=C(C)C 96092,C(C(C)C(=O)NC1CCC1NC(=O)C(C)(C)C)OCC 96093,N1(C(C2CN(C(N)=O)C2)=O)CC(O)(CNC(=O)COC2CCOC2)C1 96094,Cc1ccc(C)n1C(N1CCC(CC(=O)NCCOc2ccc(F)cc2)C1)=O 96095,c1(C(=O)NC(CC(C)C)CNC(C2CC2C#N)=O)c[nH]c2c(F)cccc12 96096,N1(C(C(c2cccc(O)c2)NC(CCC=CCC=C)=O)=O)Cc2cccnc2C1 96097,N1(C(CC(C)CNC(=O)C(=O)N(C)C)=O)CCn2nccc2C1 96098,C#CCCCC(=O)NC1(CNC(c2ccc(CCC(N)=O)cc2)=O)CCOC1 96099,c1(C(N2CCC(CN(C)C(C3(CO)CCCC3)=O)C2)=O)cc(C(F)(F)F)ncn1 96100,C1(OC)CC(NC(C2CSCCS2)=O)CN(C(=O)CCN2CCP(C)(=O)CC2)C1 96101,C(=O)(C1CCc2cc(Cl)ccc21)NC1C2CN(C(CSCCN(C)C)=O)C1C2 96102,Cn1nc(C(N2CCCCCC2CNC(=O)CC(F)(F)Cl)=O)c2c1CCC2 96103,O=C(CCCOc1cccnc1)NCC1CNC(=O)C1.c12csc(n1)CNC2=O 96104,c1(C(=O)NCC(CNC(c2c(C)ccn2C)=O)C)cccc2[nH]cc(Cl)c12 96105,CC1(C)CC(CC(=O)NCC2(O)CC(C(=O)NC3(C4CC4)CCC3)C2)CO1 96106,Cc1cc(C(=O)NC2(C)CN(C(c3cc(C4CC4)nnc3O)=O)C2)cc(O)n1 96107,N1(C(CN(C(C)CC)CCC)=O)CCN(C(=O)CCCCC#N)CC1C 96108,C1(CNC(C2C(CC)C2)=O)C2CN(C(=O)Cc3c(N)cnn3C)CC12 96109,c1(C(N2CCC(NC(C3CC(C(C)C)OCC3)=O)CC2)=O)c(F)cc(O)cc1F 96110,C(=O)(C(C)(C)CSC)NCC1C(C(N(C(CC)CC)C2CC2)=O)CC1 96111,N1(C(CCC(=O)OC)=O)CCC(C2(N(C(C)C(C)C)CC(C)C)CC2)CC1 96112,C1(C(=O)NCC2C(NC(CCOCc3ccc(C)cc3)=O)CC2)CCC2(CCC2)C1 96113,n1(CC(=O)NCC(C)(C2CC2)NC(c2cc(C)no2)=O)[nH]cc(C(=O)OCC)c1=O 96114,C1(CNC(C2(CCC)CC2)=O)CN(C(=O)C(=O)NOC)CCN1C 96115,C12(CNC(C=CC=CC)=O)CC1CN(C(=O)Cn1cc(Br)c(=N)[nH]1)C2 96116,Cn1c(NC(c2c(Br)ncn2C)c2nnnn2C)cnc1Br 96117,C(=O)(C(C)CC(F)(F)F)N1CC(C)(C(=O)NCCCc2cc(C)no2)C(C)C1 96118,CC1(C)CC(C(N2CC3CCC3(CNC(c3cscc3Cl)=O)C2)=O)C(C)(C)O1 96119,CCCC(C)CC(=O)NC(C)(C)CNC(C1SCCS1)=O 96120,N1(C(C(C(CC)CC)C)=O)CC(CNC(c2csc(C)n2)=O)OC2(CCC2)C1 96121,C1(C(=O)NC(C(C)C)CNC(C2(S(N)(=O)=O)CCC2)=O)CC2(CCCCC2)CO1 96122,n1(C(C)(C)C)cnc(C(N2CC(O)(CCNC(=O)C(F)=C3CCCC3)C2)=O)c1 96123,c1(C(N2C3(CNC(C(C)OCC#C)=O)CC(C2)C3)=O)ccc2nc(C)cn2c1 96124,N1(C(CN(CCCCCC)C)=O)CC(NC(=O)COCCCCC)CCC1C 96125,C1(C(C)NC(=O)CCc2ncccn2)CCCN(C(c2cn(C)nc2C(F)F)=O)C1 96126,N1(C(C2(C)N(C(C=C(C)C(F)F)=O)CCC2)=O)CC2CC1CN2CCO 96127,CC1CCc2[nH]c(C(=O)NCCNC(C3(CCO)CC3)=O)cc2C1 96128,C(C(=O)N(OC)C(C)CC)C1CC(NC(CC2ON=C(CC)C2)=O)C1 96129,C1(CNC(C2(CC#C)CC2)=O)(OC)CCN(C(c2ccc(CC)cc2O)=O)CC1 96130,c1(SCC(=O)N(CCCNC(c2cc(C)no2)=O)CC)ccccn1 96131,c1(C(=O)NCC2N(C(CCC(C)(C)C)=O)CC(F)C2)ccc(Cl)c2ccccc12 96132,C(=O)(C(C(C)C)c1cnc(C)s1)NC(CC(C)NC(C=CC)=O)C 96133,Cc1c[nH]cc(C(=O)NCCC2(O)CCN(C(c3ccc(Cl)cc3N)=O)C2)c1=O 96134,c1(C(=O)OCC)c(NC(=O)NC2(CF)CC(=O)C2)nc(C)n1C 96135,CC1(C)C(CO)CN1C(=O)CCN(CC(F)(F)F)C(=O)C(O)C1CCC1 96136,CCCCC(C(=O)NC1(C(=O)OC)CCC1)NC(C1CC1(C)C(F)F)=O 96137,N1(C(CCCC)=O)CCCC2(C1)C(NC(c1ccsn1)=O)CCN2C 96138,CCCCN=C(NCCc1ccc(NS(N)(=O)=O)cc1)N1CCC(C)C1 96139,c1(C(=O)NC2CC(F)(CNC(c3cc(CC)nn3C)=O)C2)cc2ccccc2o1 96140,CC(C)CC(C)(CNC(C1CC(CCO)C1)=O)NC(=O)C(N1CCCCCC1)C 96141,C12CC(C1)C(=O)N2.C(=O)(CCn1ccnc1)NCCNS(C)(=O)=O 96142,N1(C(n2cnnc2)=O)CCN(C(=O)CCC2CCC(C(C)(C)C)O2)C(CF)C1 96143,c1(C(=O)NC(CNc2nccc(OCC)n2)C2CC2)[nH]c2ccc(F)cc2c1C 96144,c1(CNC(=O)CC(C)NC(=O)CC2CCC2)ccccc1O 96145,C1(NC(C(CCC2CC2)NC(C(COC)C)=O)=O)CCCCC12CC2 96146,C#CCC(CC#C)C(=O)NC(C)(CC)CCNC(c1ccc(Br)c(C)n1)=O 96147,C(CCC=O)OCC.n1(C(C)NC(C2CC2NC)=O)cc(NC(=O)C(C)O)nn1 96148,CCCC(C)(C)C(=O)NCC1CCCN1C(c1cnn(C2CCOCC2)c1)=O 96149,C(=O)(C(O)C(C(C)C)OC)N1C(C(=O)NC2CCN(C(CC)=O)C2)CC(F)(F)C1 96150,C(CO)(C(C)(C)CO)NC(C(C)CNC(=O)C(F)CC1CCOC1)=O 96151,N1(C(C(CSC)CC(C)C)=O)CCC(C2CC(NC(=O)C(C)(C)N(C)C)C2)CC1 96152,C1(C(N(CCCC)CC(C)C)=O)COC2COCC2N1C(=O)CS.C(C)(C)C 96153,c1(C(c2ccc(OCCC(CO)CCF)cc2)=O)c(F)ccc(Cl)c1F 96154,C1(C(=O)NC(C2CCCO2)CO)(CC)CCN(C(c2ccc(C)c(C)n2)=O)CC1 96155,C1(CC(=O)NC2C=CCN(C(c3c(C#N)scc3)=O)C2)CCn2cncc2C1 96156,C1(F)(C(=O)NCC2C3CN(C(c4cc(C)n(C)n4)=O)CC32)CCN(C)CC1 96157,c1(C(=O)NCC2N(C(CC(C=C)C)=O)CC(F)C2)c[nH]c2cc(C)ccc12 96158,N1(C(CC2CC(=O)NC2=O)=O)CC(NC(=O)COCCN(C)C)C2CCCC12 96159,c1(NC(C2CCN(C(C)C(=O)Nc3nccs3)CC2)=O)cc2ccccc2[nH]1 96160,c1(OCC)c(CNC(=O)C=CC(C)(C)NC2(C)CCCCC2)cc(C)cc1Br 96161,Cc1ccccc1C(C)C(=O)NCCOCCN(C1CC2CC2C1)C 96162,C1(C(=O)N(C(CC)C(=O)O)C)CCN(CCn2cc(CCC)nn2)CC1O 96163,c1(COCC)nc(NCCOCCC2CCC2)cc(=NC2CCS(=O)(=O)C2)[nH]1 96164,c1(C(=O)NCC(CCC)NC(c2cc(=O)cc[nH]2)=O)nccc(C)c1F 96165,C12(NC(CS(=O)(=O)NC)=O)CCCCCC1N(C(c1ccc(C)o1)=O)CC2 96166,C1(CNC2(C(=O)Nc3ccccc3)CC2)CC(OC)CN1C(C1C(CC)C1)=O 96167,C1(C(=O)Nc2cc(C)[nH]n2)CCN(C(c2ccc(N3CCNC3=O)cc2)=O)CC1 96168,c1(NCC(c2ccccn2)N(C)C)ccc(S(=O)(=O)NCCS(C)(=O)=O)cc1Br 96169,C(C(C)(F)C(C)(C)F)OCCC(N1C(C)CC(CC(=O)NCCO)C1)=O 96170,CC1CC(NC(C2CC(F)(F)C2)=O)CCN1C(c1cc(CO)ccn1)=O 96171,N1(c2ncnc(OC)c2C)CC2CN(CNC3CCC(F)C3)CC2C1 96172,N1(C(=O)C(F)(F)c2cscn2)CCOC2(CCS(=O)(=NC(=O)C=CCF)CC2)C1 96173,CCC(C)(CNC(=O)C(C1CCCCC1)C)C(=O)NCC1COCCN1C 96174,c1(CCCC=C)cn(C(c2ccccc2)C2CC2)nn1.C12CN(C1)C2=O 96175,C1(CNC(Cc2cc(C)sc2)=O)(NC(=O)CC2CCCN(C)C2)CCN(C)C1 96176,c1(C(N2CC(CSCCN(CC)CC)C2)=O)cnc(C(C)(C)C)[nH]1 96177,C1(CC(=O)N(CCCNC(C=CCOCCOC)=O)C(C)C)CCCCN1C 96178,c1(C(=O)NCCC(C)N(C(CC(CC)O)=O)C)[nH]nc2ncnc(O)c12 96179,N1(C(C(CSC)C)=O)CCCCC1CC(=O)N(C(C)C(=O)NC1CC1)C 96180,N1(CCC(=O)NCC)CC=C(C(=O)N(C)CC2CCCC3CC23)C1 96181,CC(CC(=O)N1CCCCC1C1(NC(=O)C=Cc2c[nH]cn2)CC1)C(C)(C)C 96182,c1(N(C)Cc2ccccc2)nc(=NCC2COCC(C)(C)O2)[nH]c2c1CCCC2 96183,C(C(=O)NCc1ccncn1)(C(C)O)NC(c1c(CC)cco1)=O 96184,CC(C)CC=O.C(C)(CC(=O)NC1CCC1CNC(=O)C(CC1CCC1)SC)OC 96185,NC(=O)CC(O)C(=O)N1CCOC(CCNC(C2CCCCC(=O)N2)=O)C1 96186,CC1CCn2ncc(C(N3CCC(C)C(CNC(=O)C(C)(O)CCCl)C3)=O)c2C1 96187,C(=O)(C(F)(F)C1(O)CCC1)NCCNC(C(N1CC(C)C1)C)=O 96188,c1(C(N2C(CNC(C3COCCO3)=O)CC2)=O)cnc2[nH]cnc2c1 96189,CCCCC(O)C(C)C(=O)N1CCC(OCC(=O)Nc2c[nH]ccc2=O)C1 96190,N1(C(CC(CC)C)=O)CC2CC(NC(=O)CC3CC(C(F)F)C3)CC2C1 96191,c1(C(N2CC(C(C)NC(CCC(=O)NCC)=O)OCC2)=O)cc(Cl)c(N)c(Cl)c1 96192,C(N=c1nc2c(ncn2C)c(NCCOC(F)(F)F)[nH]1)C1CC(OC)C12CCC2 96193,N1(C(CC2C(C)OC(C)C2)=O)CC2(CCCCN(C(C3CCCS3=O)=O)C2)C1 96194,c1(N2CCN(C(c3cc4ncc(C)n4cc3)=O)CC2)cc(C)c([N+](=O)[O-])cc1Br 96195,CC(C(C)(C)C(=O)NCc1sccc1Cl)NC(=O)Cc1cccn1C 96196,c1(C(=O)NCC2CC(CNC(C=COCC)=O)OC2)ccc2ncnc(C)c2c1 96197,c1(C(C(=O)N(C2CCN(C(=O)C(C)(C)C3CCC3)CC2)CC)C)c(C)noc1C 96198,c1(CCC)c(C(N2CC(NC(C3CN(C(C)=O)CCO3)=O)C(C)C2)=O)cnn1C 96199,Cc1cnc2ccc(C(N3CCC(C)C(CNC(C4(CCF)CC4)=O)C3)=O)cn12 96200,C1(NC(CCOCC(C)C)=O)CN(C(=O)CCC=CC(C)C)C2(CCOC2)C1 96201,N1(CCCCC)CCCN(Cc2cn(C3CCC3)nn2)CC1 96202,C(=O)(C#CC1CCOCC1)N1CC(C(=O)NC)C(Cn2cc(COC)nn2)C1 96203,C1(NC(CC(C)=C(C)C)=O)CC2CN(C(=O)Cn3cccc3)CC2C1 96204,N#Cc1ccc(Cl)c(C(N2CCC(OCCNC(C3CCCS3)=O)CC2)=O)c1 96205,C(=O)(CC(CC1CC1)N(C)C)OCCCC=C.n1(C2(C=O)CC2)ccnc1 96206,C12(C(=O)NC(C3CCCC3)CNC(=O)CCc3nc(O)n[nH]3)CSCC1C2(F)F 96207,Cc1ccc(C(=O)NCC2CCN2C(=O)C(c2ccc(Cl)s2)C)cn1 96208,CC1CCCCN1CCC(=O)NC(CNC(=O)C(C)(C)CF)C(C)(C)C 96209,C(CN=c1nc(Cl)[nH]c(C)c1C#N)C1CCN(C(c2c(OC)ccnc2)=O)C1 96210,N1(C(CC(CC)OC)=O)CCCCC12CC(NC(=O)CC1CCCC(=O)N1)C2 96211,Cc1cn2cc(C(N3CC4C(NC(=O)C(C5CCCCCC5)O)C4C3)=O)sc2n1 96212,C(=O)(C(C)(C)CC(=O)NC1CCCCC1NC(=O)C(C(C)C)NC(C)=O)OC 96213,CCC(CC)(CO)C(=O)NCCOCCCN(C)C(c1cn(C)ccc1=O)=O 96214,C1(CC)COC(C)CN1C(=O)NC1(c2nnc(C3CCS(=O)(=O)CC3)o2)CC1 96215,c1(-n2ncc(CNC3CC(NC(C(C)C4CCOC4)=O)C3)c2)ccccc1F 96216,N1(CCOC)CCCC(NC(=O)C(CCOC)OC)C1C.C1CCS(=O)(=O)C1 96217,c1(C(N(CC(C)O)CCNC(=O)CC2(C)CCOCC2)=O)cnc2[nH]nc(O)c2c1 96218,N1(C(C)=O)CC2CCCN(C(=O)Nc3c(C)nn(C)c3Sc3ccccc3)C2C1 96219,N1(C(C2C(NC(C3(C=C)CCCC3)=O)CCO2)=O)CCc2nc(O)[nH]c2C1 96220,C(=O)(C1=CCCOC1)N1C(CCNC(C2CC2(Cl)Cl)=O)CSCC1 96221,C1(C(=O)OCC(c2ccccc2)=O)CCCCC12CCC2 96222,c1(COC)nc(NCCS(=O)(=O)N(C)C)cc(N2CC3C(C2)C3(C)C)n1 96223,N1(C(C2=CC(C)(C)C2)=O)CCN(C(=O)CCCCN2CCCCC2)C2COCC12 96224,Cc1cc(=NCC2(C)CSCCO2)[nH]c(=NCc2nccc3c2CCCC3)[nH]1 96225,c1(C(N2CCN(C(=O)NC(c3ccco3)C)CC2)C(=O)OC)cc(F)cc(Cl)c1 96226,CN1CCC(C(=O)NCCCN2CCN(C(C3(C)CC3(F)F)=O)CC2)C1=O 96227,C1(NC(Cc2ccc(OCC)cc2)=O)CC(C)CN(C(c2cscc2C#N)=O)C1 96228,N1(C(CC(=O)NCC#C)=O)CC2CCCC(CNC(=O)CSCC=C)C2C1 96229,N1(C(CCNC(=O)NC)=O)CCC(CNC(c2ccc(C(N)=O)cc2)=O)C(C)C1 96230,C1(C(=O)NC2CCN(C(CCCSCC)=O)C2)CCCN(C(=O)NC)C1 96231,c1(C(=O)NC(CC)CN(C(=O)CSc2cccs2)CC)cccc2c1OCO2 96232,C(=O)(C1=CCCC1C)N.C12CCC(C1)NC2=O.C1(C(=O)OC)CC(CC)C1 96233,c1(C(N2CCC(CCNC(C=COCC)=O)CC2)=O)oc2c(c1C)C(=O)CCC2 96234,n1(CCOCC=C)c(N2CCC(C)(C(=O)OC)C2)nnc1CO 96235,C1(CC(=O)NC(CNC(CC=C)=O)Cc2ccccc2)(COC)CCOCC1 96236,c1(NC(CNC(C2(OC(C)C)CC2)=O)=O)cnn(C2CCC2)c1 96237,c1(C(=O)N(CCCNC(C2CC23CCC3)=O)CCO)cc(Br)cc2c1OCC2 96238,C1(CNC(C(C)n2cccn2)=O)CCCCN(C(C2(C(F)(F)F)CC(O)C2)=O)C1 96239,N1(C(CCCOCC=C)=O)CC(C)(C)CC1CNC(c1[nH]nnc1CC)=O 96240,N1(C(CC)=O)CCCC1C1CCCCN1C(c1c(C)n(C)c2ccc(OC)cc12)=O 96241,N1(N2CCCC(OC3(C)CCCC3)C2)CCC(C)(C=O)CC1.C(C=O)(OCC)OC 96242,c1(C(=O)NC2CC(CNC(C(CCCC)O)=O)CC2O)ccc2nn[nH]c2n1 96243,c1(CC(=O)NC2CCCCC2NC(C2CC3C=CC2C3)=O)cccnc1Br 96244,C1(OC)CC2CC(C(=O)Nc3cccc(CNC(=O)C=CCF)c3)CC12 96245,c1(C(N2CCC(OCCNC(C(CC#C)C)=O)C2)=O)n[nH]c2c(C)cccc12 96246,c1(-c2ccc(C(=O)NCC=CC)s2)cccc(F)c1.CON=CC(=O)N1CCC1 96247,Cc1ccc2c(C(N3CCC(O)(c4ccc(Br)cc4)C3)=O)noc2c1 96248,C(c1cccnc1)=CC(=O)N(C(C)CN(C)C(c1cnc(C2CCCO2)s1)=O)C 96249,C(=O)(C1=CC2C=CC1C2)N1CCC(CC=C)(NC(C2CCC(=O)CC2C)=O)C1 96250,c1(NC(C23C(CN(C(c4c(C)c(F)ccc4)=O)C2)C3)=O)cccc2nsnc12 96251,c1(CNC(=O)C(=O)Nc2cc(C(=O)NC)cc(F)c2)cccc2c1OC(F)(F)O2 96252,n1(CCCC)cc(C(=O)NCCOCCCN(C(=O)C(C)n2cccc2)C)c(C)n1 96253,C1(C(=O)NCC2CCCC(NC(c3ccncc3F)=O)C2)(SC)CC(F)(F)C1 96254,CCCC(CCC)CC(=O)NC(C)(CO)C(=O)NCC(O)C1CCC1 96255,CP(C)(=O)CCC(=O)N1CCCCC(C(=O)NC2CC3(CC3)C2)C1 96256,CCC(C)(F)C(=O)Nc1ccnnc1C 96257,N1(C(CSCC(C)C)=O)CCC(CC(=O)N(C2CCC2)CC2CC2)C1(C)C 96258,c1(CNC(C(c2cc(C)sc2)N(C)C(=O)O)=O)cnc2ccccc2c1.C1(C)CC1 96259,N1(C(CC2CC(=C)C2)=O)CCOCC(CNC(c2c(C(C)C)cccc2C)=O)C1 96260,C(=O)(C1CC(=O)Nc2ncn(C)c21)NCCNC(COC(CC)CC)=O 96261,c1(C(=O)NC2C(C)N(C(c3cnc(C4CC4)nc3O)=O)CC2)cc(Cl)cc(Cl)c1 96262,C1(C(N2CC(CCNC(=O)C(C)N(C)C(C)=O)(OC)C2)=O)CCNC(=O)C1 96263,c1(SC)ncc(C(=O)NCC2CCCC2NC(=O)C(F)C(C)(C)O)c(O)n1 96264,c1(CC)ccc(C(N2CCC(N(C(=O)CC3CCC(F)(F)C3)CC)C2)=O)cc1 96265,N1(C(C2(OCC)CCC2)=O)CCCCC(Nc2ncc(C)c(C)n2)C1 96266,C(=O)(C1OCCn2ccnc21)NCCCN(C(C(CC)(C)O)=O)C 96267,C(=O)(CCC1=CCCCC1)NC(C)CC1CN(C(c2sccc2C#N)=O)CCO1 96268,c1(-c2ccc(NC3CCCC(CC(=O)OC)C3)cc2)cc2cc(Cl)cnc2[nH]1 96269,Cn1cc([N+](=O)[O-])c(CC(N2CCC(O)(CNC(=O)C#CC3CCCC3)CC2)=O)n1 96270,c1(C(=O)NCC2(CNC(C(C)SCC)=O)CCCC2)ccc(P(C)(C)=O)nc1 96271,N1(C(CCC(C)=O)=O)CC2CC(C1)N(C(c1cc(-c3cccnc3)[nH]n1)=O)C2 96272,c1(CC(=O)NCC(CC)NC(=O)C(C)SC(F)(F)F)coc2c(C)c(C)ccc12 96273,N12CCCCC1C(=O)N2.C(C)(C(=O)NC)NC(=O)NC.C(CN1CCCC1)(CO)N 96274,C=CC(O)(C(=O)N1CCC(C)(NC(c2cc(C3CC3)no2)=O)C1)C(F)(F)F 96275,c1(C(=O)NC(C)(CNC(=O)CCc2ccc[nH]2)C2CC2)ncsc1Br 96276,c1(N2CC=CC(NC(C(CC)OC3CCCCC3)=O)C2)cc(C)ncc1C#N 96277,C12(C(=O)NC(CNC(c3cc(C4CC4)no3)=O)C3CC3)CC(C1)C(C(F)(F)F)O2 96278,c1(C(N2CCCCC(NC(C(CC=C)(C)C)=O)CC2)=O)cnn2c1CC(C)CC2 96279,C#CCCCC(=O)NC1(CNC(=O)Cc2cc(C(F)(F)F)n[nH]2)CC1 96280,CCC(C(=O)N(CCCCNC(c1cn(C)cn1)=O)C)NC(C)=O 96281,C1(CCNC(COCC(=O)OC)=O)CCN(C(C23CC(C)C2C3)=O)CC1(F)F 96282,c1(C(=O)OC)cc(C2CCC2)ccc1C.C1(c2cn(C3(CC)CC3)nn2)CN2CC12 96283,c1(C(=O)NC2C(NC(C(C)O)=O)C2)cc2ncccc2[nH]1 96284,C(=O)(C(CN(C)C)c1ccccc1)NCCC(C)N(C(=O)COCCF)C 96285,C(=O)(CC1OCc2ncccc21)N(CC(C)NC(CCC(=C)Br)=O)C 96286,C1(C(=O)NCC2(C)CCN(C(C)=O)C2)CC2(CCOCC2)CN1 96287,N1(C(C(C)NC(C)=O)=O)CCC2CN(C(=O)C=C3CCOCC3)CC2C1 96288,CC(C)CCCCC(=O)N1CCN(C(=O)CCCCc2cnn[nH]2)C2CC12 96289,C(=O)(C1CCc2nnc(C)n21)Nc1cccc(NC(CCCCCC=C)=O)c1 96290,C1(C(N2CCC(Cn3ccnn3)C2)C(=O)NC(CC)(C)C)CC12CCCCC2 96291,Cc1ccc(C=CC(N2CC3CC3(C(N3CCCC(C(C)(C)O)C3)=O)C2)=O)s1 96292,N1(C(CC2CC(=O)C2)=O)CC(F)(COC(=O)CCc2cncnc2)C1 96293,CCCCCC(O)CC(=O)NC(CCC)CC(N1Cc2ccccc2C1)=O 96294,C1(CC)CN(C(=O)Cn2cnnn2)CCN1C(=O)CCn1cc(Br)c(C)n1 96295,C(=O)(C(O)CC(F)(F)F)N(C)CC1(C)CC(NC(=O)C(c2ccnn2C)O)C1 96296,C(=O)(CCCCC(C)(C)OC)N1CCCCC(CNC(CS(CC)(=O)=O)=O)C1 96297,c1(C2C(C(=O)NC(CC)CNC(c3nc(Cl)sc3C)=O)C2)ccc2c(c1)OCO2 96298,C(=O)(C1CCCc2nncn21)NC(CC)(CC)CCNC(=O)CCS(C)(=O)=O 96299,CC1(C)CCCC(C(N2CCCC2CNC(C2(C(N)=O)CC2)=O)=O)C1 96300,CON(C(=O)C=CC1CCN(C(=O)CC2COCC(C)O2)CC1)C1CCCC1 96301,C(=O)(C(C)(CC)C(=O)NCC1(CNC(C2CNC(=O)N2)=O)CC1(F)F)OCC 96302,C(=O)(C(CC(C)C)C(N)=O)N1CC(CC(=O)NC(c2ccccc2)CC)(SC)C1 96303,n1(CC=C)cc(Cl)c(=NC(=O)N2CC(C)C(N)C2C2CCOCC2)[nH]1 96304,C(=O)(CCC(C(C)C)NC(=O)C1=C(C)OCC1)N1CC=C(COC)CC1 96305,CCS(=O)(=O)CC(C)NC(=O)C(N1CCCC(C(F)(F)F)CC1)=O 96306,C1(CC(=O)N(CCN(C(=O)C=Cc2ccco2)C(C)C)C)CC2(CCC2)CCO1 96307,c1(C(=O)NC2C(NC(C(CCC)OC)=O)C2)c2c(c[nH]c1=N)CCC2 96308,c1(C(N(CC(CNC(CC2C(CC)C2)=O)(C)C)CC)=O)cc(=O)cc[nH]1 96309,c1(OC)cccc(C(F)(F)C(=O)N(CC(O)CN(C(=O)CC2C=CCC2)C)C)n1 96310,Cc1noc(C(=O)N(CC(C)N(C(=O)C(C)Cc2c(C)n[nH]c2C)C)C)c1C 96311,c1(NC(C2CCN(C(C(c3ccccc3)C)=O)C2)=O)cccnc1OC(F)F 96312,N1(C(C=NOC)=O)CCOC(C2(NC(=O)CNC(c3nnc(S)n3C)=O)CC2)C1 96313,C12(C(N3CC(Cn4cc(C(CC)O)nn4)OCC3)=O)CCCCC(=O)N1CCC2 96314,c1(C(C(=O)NCC2CC2)N(C2CC(OCC)C2)C)cc(N(C)C)ccc1OC 96315,C1(CC(=O)NCCCC(=O)NCCSC(F)F)CCC(O)C1 96316,C1(C(c2sccc2Cl)NCc2nnnn2CC2CC2)(COC)CCCO1 96317,C1(C(=O)NCC(CCC)OC)(NC(C2CC3C=CC2C3)=O)CCC(C)(C)C1 96318,c1(C(C)C(=O)NCCCNC(C2CCCN2C(=O)OC(C)(C)C)=O)ccccc1Br 96319,CCCCCC(C)(CC)C(=O)N1CC2(CCC2NC(=O)CSC(F)(F)F)C1 96320,n1(CC(=O)NC2(C)CN(C(C(CC)O)=O)C2)[nH]cc2c(=O)ncnc1-2 96321,N1(C(CCN(C(CC2CCC(C)C2)=O)CCO)=O)CCN(C(C)(C)C)CC1 96322,C1(C(=O)NC2C=CCN(C(c3cc(F)ccc3Cl)=O)C2)CCn2c(O)nnc2C1 96323,c1(CCN(C)C)ccccc1.c1(S)ccc(OC2CCCC2)nc1 96324,Cc1cc([N+](=O)[O-])c(S(=O)(=O)NC2CCC3(CCCC3)CC2)cc1C(=O)O 96325,C1(c2n(C(CC)C3CCC3)nnn2)(NCCS(=O)(=O)CC)CCC(C)(CC)CC1 96326,c1(C(=O)OC)c[nH]ccc1=N.c12ccc(cc1)NC(=O)NC1CCCN1C(=O)C2 96327,N1(C(c2ccc(CC)o2)=O)CCCN(C(c2cn(C)[nH]c2=N)=O)C(CO)C1 96328,C(=O)(CC(C(F)(F)F)N1CCOCC1)OCC(COC)NCOCC(F)(F)F 96329,CC1CCN(CC(=O)N(CCC(C)(C)NC(=O)C(F)CC2CCC2)C)C1 96330,C=CC(C)(C)CC(=O)NC(C)CCNC(c1cc(Cl)ncc1NC)=O 96331,C(C(C(=O)NOCC(=O)NC)NC(C1CC(=C2CCC2)C1)=O)CC=C 96332,N1(C(CCc2cc(C)[nH]n2)=O)CCOCC1C(=O)NCC(O)COC(C)C 96333,Cn1ccnc1C(=O)NC(C(=O)NCC1(O)CCSC1)C1(C)CC1 96334,C=CCCC(C)(c1nnnn1CCCC1CC1)NCCC1COCCO1 96335,CC(O)C(C(=O)NCC=CBr)NC(C1CC(=O)C1(C)C)=O 96336,Cc1nc(NC2CCC(CCNC(=O)CNC(=O)CC(C)(C)C)C2)c(C)c(C)n1 96337,C12(CNC(CC(C)SC)=O)CCCC1N(C(c1cc(CC(C)C)on1)=O)CC2 96338,CC(C)(C(=O)NC1CC(F)(CNC(=O)CN2CCCCS2(=O)=O)C1)C(F)F 96339,C1(CNC(CCC(C)(F)F)=O)CN(C(c2cnc3c[nH]nc3c2)=O)CCC1(C)C 96340,C1(CC)=NC=C1CN(C)CCn1cc(C(c2nccs2)=O)nn1 96341,c1(CC)ccc(C=CC(=O)NC2CCCN(C(=O)CN3CCCCC3)C2)cc1 96342,c1(C(c2nnnn2CC)Nc2c(C(=O)NCC)csc2)cccnc1S(C)(=O)=O 96343,C(=O)(CC(C)(C)C(=O)N1CC(C(=O)NCC)C(C(C)C)C1)OC(C1(O)CCC1)C 96344,C1(C(=O)NCCN(C(C(C(=O)OC)C)=O)Cc2ccccc2)CCC(C)(C)CO1 96345,CCCCN=C(NCCCC1CCCOC1)NCc1cc2ccccc2[nH]1 96346,C1(CC)CCCN(C(=O)Cn2cc(C(=O)N(C3CC4CCC3CC4)C)nn2)CC1 96347,C(C)(C)(CCC(=O)N1CCCC(C(N2CCC(C)(C(N)=O)C2)=O)C1)OC 96348,N1(C(c2c(C#C)c[nH]n2)=O)CCC(F)CC1C(N1CCC(C)CC1)=O 96349,C(=O)(C(C)CC(F)(F)F)NCC(=C)CCNC(=O)C(CCCC)N(C)C 96350,C=C(C)CCCC(=O)NCC(C)(C(C)C)NC(=O)CCOc1ccccc1C 96351,CC1CN(CCO)CCN1C(=O)C(=O)NCC1CC(F)C1 96352,C(=O)(CC(C)CC(F)(F)F)NCC1N(C(c2cnc(SC)s2)=O)CC(O)C1O 96353,N1(C(C2C(CC)C2)=O)CC(C)(C)CCC1CNC(c1cc(C)nc(C(F)F)n1)=O 96354,C1(C)(C(N2CC(C)(NC(=O)CN3CCSCC3)C2)=O)C2Cc3ccccc3C12 96355,N1(C(CCNC(CNC(N)=O)=O)=O)CCC(OC)C(CNC(C2CCC2)=O)C1 96356,N1(C(c2cccc(C)n2)=O)CC2CCC1(CNC(c1[nH]c(O)nc1C)=O)CC2 96357,c1(NC(CCCNC(CCCCOC)=O)=O)ccc(Oc2ccc(F)cc2)c(F)c1 96358,CC1(C)C2CC(C(=O)NC3(C)CN(C(=O)CNS(=O)(=O)C4CC4)C3)CC12 96359,c1(C(=O)NC(C)CCCCNC(=O)CCSC(F)(F)F)cc(=O)cc(Cl)[nH]1 96360,N1(C(c2nccc(N)c2Cl)=O)CCC(NC(c2ncc(F)cn2)=O)C(CO)CC1 96361,C(C#CC#CCO)NC(C(C1CCCN(C(c2ccns2)=O)C1)C)=O 96362,C1(CC(N)=O)(NC(c2cc(OC)ns2)=O)CCN(C(C2CSCCS2)=O)CC1 96363,N1(C(c2cc(OC)nn2C)=O)CCN(C(=O)C(O)CC(C)C)C(C(C)C)C1 96364,c1(N2CCN(CCCC)CC2)nc(N(CCC(C)CCO)C)nc2c1CCC2 96365,CCC(C)(C)C(C(=O)N1CCC(CN(C)C(c2cc(C3CC3)sn2)=O)C1)OC 96366,Cc1ccc2nc(C)c(C(=O)NC3CC3CNC(c3nnn(C)c3N)=O)cc2c1 96367,c1(NC)c(C(=O)NCCCNC(c2cc(F)c(F)cc2Cl)=O)sc2nccnc12 96368,N1(C(CC(C)N(C)C(c2ccc(=O)n(C)n2)=O)=O)CCC(C2CCC2)C1 96369,C1(CNC(C(CNC(=O)Cc2ccn(CC)n2)OC)=O)CCCCCN1C 96370,C1(C)(C(=O)NCCCCC2CCN(C(CNC(CC)=O)=O)CC2)CCC(F)(F)CC1 96371,C1(NC(C=C(CCC)C)=O)CC2CC1N(C(=O)CC1(O)CCCCC1)C2 96372,c1(CC(C(N2C(CNC(c3cnc(C)[nH]3)=O)C=CC2)=O)C)cccc(Br)c1 96373,c1(NCC2(CC)CCOC2)ncc(S(=O)(=O)NCC2CS(=O)(=O)CCO2)cc1Cl 96374,C#CC1(O)CC(C(=O)NCCCOCCC(N2CC=CC2(C)CO)=O)C1 96375,C(=O)(C1=COCCC1)N1C(CN(C(c2ccc(OC)nn2)=O)C)CCCC1 96376,CCC1=NOC(C(=O)NC23CC2CN(C(=O)CCOC2CCCC2)C3)C1 96377,Cc1cc(CO)ncn1.N12CCC(CC1)NC(=O)C1CC(C1)C(=O)N1CCC2CC1 96378,CC1(C(N2CCN(C3CCCN(C(C4(C(N)=O)CC4)=O)C3)CC2)=O)CCNC1=O 96379,c1(C(=O)NCC(C2CCOC2)NC(c2n(C(C)C)nnc2)=O)cnc2n1CCC2 96380,N1(C(C=C(COC)C)=O)CC(C2(NC(c3ccc(C(=O)NC)cc3)=O)CC2)C1 96381,C1(NC(c2c(C)cccc2)=O)CCN(C)C12CCCN(CC(C)O)C2 96382,c1(C(N2CC3C(NC(c4c(CC)n(CC)nn4)=O)C3C2)=O)cnc(O)n(C)c1=O 96383,C1(C)(NC(c2n(CCC)nnn2)C2CC2(Br)Br)CCC(=O)N(C)C1 96384,CC1(C(=O)NCc2ccoc2C(=O)NC2CC(O)C2)CCC2CC2C1 96385,c1(CC(=O)NCC2(NC(c3cnn(CCF)c3)=O)CC(F)(F)C2)ccc(O)cc1 96386,c1(C(N(CC(C)(C)NC(C23CCCCC2C3)=O)C)=O)cc2c(cc1Cl)NC(=O)C2 96387,O(NC(=O)N(c1nn[nH]n1)C1CC1)CC(=O)OCC 96388,C1(C(=O)NC2C(NC(CC(C(C)C)O)=O)CC2)CC12C1CC3CC(C1)CC2C3 96389,C(=O)(C(C)(O)CCN(C)C)NCC(CC)N(C)C(c1cccc(SC)c1)=O 96390,c1(OC(C(=O)NC(c2ccc(C(F)(F)F)o2)CC)C)cccc(C)c1C 96391,N1(C(Cc2c(C)noc2C)=O)C2CCC1(CNC(c1ccco1)=O)CC2 96392,c1(C(N2C(CNC(CC(=O)NCC)=O)CC(OC)C2)=O)cc2c(=O)[nH]ccn2n1 96393,c1(NC(CC2CC(C)(C)N(C(c3sccc3C#N)=O)C2)=O)cnc2[nH]cnc2c1 96394,C1(C(=O)NCCCOC=C)C2CCCC2CN1C(=O)CN1CCCCC1=O 96395,N1(CC(=O)NCC(=O)N(CC(C)NC(=O)CC2CCCC2)CC)CCC(C)C1 96396,c1(NC(C2C(N)CCC2)=O)c(Br)cc(Br)c2cccnc12 96397,Cc1cc(CC(=O)NC2CCCCC2NC(c2ccc[nH]2)=O)nn1C(F)F 96398,N1(C(CC(CCC)O)=O)CC2(CCN(C(=O)CCCC(C)C)CC2)C1 96399,CC1=C(C(=O)N2CC(NC(c3ccsc3CN)=O)C(C)C2)CCO1 96400,CCC(C(=O)NC1CC(CNC(=O)C=CCN(C)CC)C1)n1ccnc1 96401,N1(C(C(CC)C=CC)=O)CCC2(CCCN2C(c2cnc(CO)nc2C)=O)C1 96402,c1(C(=O)NCC(C2CC2)NC(C2CC23CC(O)C3)=O)ccc(Br)cc1Br 96403,N1(C(CC(CCC)C)=O)CC(CNC(c2ccnnc2C)=O)OC(C)(C)C1 96404,Cc1ccc(C(=O)Nc2cc(F)cc([N+](=O)[O-])c2)c2c1NCCC2 96405,c1(CC(=O)NCCCC2(NC(=O)Cc3ccncc3Cl)CC2)ccc(Cl)cn1 96406,CC(C)C(CCNC(=O)Cc1cc(C(C)C)no1)NC(C1CCC(O)CC1)=O 96407,Cc1cc(=NCC2CCSC2(C)C)[nH]cc1S(=O)(=O)N1CCOC(CCO)C1 96408,C(=O)(C1=CC2CCCC12)NCC1N(C(CSC(C)C)=O)CCN(C)C1 96409,c1(C(N(CCNC(c2ccc(C#C)cn2)=O)C2CC2)=O)ccc(P(C)(C)=O)cc1 96410,CC1CCC(C(=O)NCCCCC2(NC(c3ccco3)=O)CC2)O1 96411,C1(C(N(C2CNC(=O)C23CC3)C)=O)CCN(C(=O)CCC2(C)CCCO2)O1 96412,CCC(CCC(=O)NC(CC(=O)NC)C1CC1)NC(C1CCCSC1)=O 96413,C12(C(=O)NCC3C(CNC(c4ccc(CC)nc4)=O)C3)CC3CC(C(=O)N1)C2C3 96414,N1(C(C=C2CCC(C)(C)CC2)=O)CCC2(CCC(NC(C3CCCO3)=O)CC2)C1 96415,CCCCCC(O)C(=O)NC(C1(O)CN(C(c2cncc(Cl)c2)=O)C1)C 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96611,Cn1cc(C(=O)NC2(c3nnnn3C3CCOC3)CCCCC2)c(C(F)F)n1 96612,CCCCC(O)CC(=O)NC1CN(C(c2ccccc2C(N)=O)=O)CC2(CC2)C1 96613,N1(C(C=CC)=O)CC2CCC(C1)N(C(c1cnn(-c3cccc(F)c3)c1N)=O)C2 96614,NC12CN(C(c3cnn(-c4ccccc4S(C)(=O)=O)c3)=O)CC1CS(=O)(=O)C2 96615,C1(CNC(=O)Cc2cscn2)CC(O)CN1C(C1CC(=O)N(c2nccs2)C1)=O 96616,C(=O)(CC(C)(C)C=C)N1CCCC(N(C(=O)Cc2cccc(F)c2O)CC)C1 96617,c1(CNC(=O)NC(c2ncc[nH]2)CC)n[nH]c2c1COCC2 96618,O=C1Nc2cccc(-c3ccc(F)c4ccncc34)c2CO1 96619,C(=O)(C1=CCC(NC(C2CC3C=CC2CC3)=O)C1)NCCCC1(C)CC1 96620,N1(C(C2(F)CCN(C(CCCC=C)=O)C2)=O)CCC(CO)C(C)C1 96621,c1(C(=O)NC(CNC(C=C(C)C(F)F)=O)(C)C2CC2)cc(C)n(C)n1 96622,C(CC)(CC)(CCNC(=O)C(C)c1ccsn1)NC(c1c(CC)cco1)=O 96623,Cc1cc(C(N2CCCC(F)(CNC(c3ccon3)=O)C2)=O)cnc1C(F)F 96624,c1(OC)cc(OC)c(C(N2CCC(NC(C3CCC3(F)F)=O)C2C)=O)cn1 96625,C(CCCCC(=O)N1CCC(CF)CC1)NC(c1n(C)ccc1)=O 96626,c1(C(N2CCC(F)(CNC(C(CCC)C#N)=O)CC2)=O)cc(F)c(N)cc1F 96627,C(C)(CC(=O)NCC(C)(C)CN(C(=O)CCC1CCCN1C)C)N(C(C)=O)C 96628,c1(NCCc2ccc(OC)cc2C)[nH]c(=NCC2CCC=CO2)nc2scnc12 96629,N1(C(C2C(CC)CCCC2)=O)CCC(NC(=O)CCC2CCOC2)C(C)(C)C1 96630,c1(C2C(C(=O)NCCCCCNC(C(C)OC)=O)C2)cccc(F)c1Br 96631,CC1(C(N2CCC(n3cc(CNC(=O)C=CCO)nn3)C2)=O)CCOC1 96632,c1(OC)cc(C(=O)O)ccc1NC(C1CCCC(N(C)C)C1)=O 96633,c1(C(=O)NC(CC(=C)C)C(=O)NCCN2CCCCCC2)ccc2[nH]ccc2c1 96634,C=CC1CCCN(C(=O)NCCCNc2ccc(OC)cc2Cl)C1 96635,N1(C(CCCC#N)=O)CCN(C(=O)CC2CCC3CC23)CC1Cc1cccc(F)c1 96636,c1(CC)sc(C(=O)N(CC(C)NC(c2ccc(C(N)=O)nc2)=O)CC)cc1C 96637,N1(C(C(C)NC=O)=O)CCC2(CCC(N(C)C(c3cnc4sccn34)=O)CC2)C1 96638,CCC(C)CCC(=O)NCCC1(NC(c2sccc2OC)=O)CCC1 96639,C12(CNC(c3c(C)nc(O)[nH]3)=O)CCCCC1N(C(=O)Cn1cncn1)CC2 96640,c1(NCC#CC)cc(N2CCN(CCN3CCCCC3)CC2)nc(C)n1 96641,C1(NC(C(C2CCCCC2)C)=O)COC2(C1)CN(C(c1scnc1C(F)F)=O)C2 96642,N1(C(CC2(C)CN(Cc3ccc(OC)nc3)C2)=O)Cc2cccc(F)c2C1 96643,N1(C(C2(CC)CCCO2)=O)CC(CNC(c2cc3scnc3[nH]2)=O)OC(C)(C)C1 96644,C(=O)(C1CCCc2nncn21)NC(C1(O)CN(C(=O)Cc2csc(S)n2)C1)C 96645,C(=O)(CCC(=O)NN(C)C)N1C(CN(C(C2C(CN(C)C)C2)=O)C)CCC1 96646,N1(CCN(C(=O)C(c2cccs2)NC(=O)Cc2cnn(C)c2)C)CCN(C)CC1 96647,c1(C(=O)NC(CN(C(=O)C(C(C)C)NC(N)=O)CC)C)cncc2ccc(F)cc12 96648,C1(C)(CN(C(C2CCN(CC)C2)=O)C)CCCC1NC(=O)C(F)=CCCF 96649,C1(c2nnc(C(C)C)o2)CN(C(c2cnncc2C(F)F)=O)CCO1 96650,C1(NC(CC2CN(C(C)=O)C2)=O)CCCCC1NC(=O)C(c1cnn(C)c1)OC 96651,CC1CN(C(=O)C=CC2CCCN2C)CC(=O)N1 96652,c1(C(=O)NC(CC(C)NC(C(C2CCC(=O)N2)C)=O)C)cc(O)n(C)n1 96653,C(=O)(Nn1cnnc1C)C1CN(C(c2ccc(OC)o2)=O)CC1C 96654,c1(C(NNC(C2CN(C(=O)OC)CC2F)=O)=O)c(C)nn(C)c1C 96655,N1(C(c2c(C)nn(C)c2)=O)CCOC2CN(C(=O)CC3CC3C(F)(F)F)CC12 96656,C=CC1(C(=O)NCC(C2CC2)N(C)C(c2cccc(F)c2)=O)CCCCC1 96657,c1(CC(=O)NCC2C(NC(c3n(C)ncc3)=O)CCC2)ccc(Cl)cn1 96658,N1(C(C=C(CCC)C)=O)CC(CNC(c2cnc3cc[nH]c3c2)=O)C2(CCC2)C1 96659,C1(C(N2CCCC2CC)C(=O)NCC)CCCC(F)C1 96660,C=CC(C)(C)CC(=O)NCC(O)CC(=O)N(C1CCCC1O)C 96661,c1(C(=O)NCCNC(c2cnn(CC(F)(F)F)n2)=O)snc(O)c1Cl 96662,c1(C(N2CCC(C)(CCNC(C(CSC)C)=O)C2)=O)ccnc2ccsc12 96663,c1(C(N(C(CN2CCOCC2)C(C)C)CC)C)c(F)ccc(Br)c1OC(F)F 96664,C1(NC(CCCC(C)=O)=O)CCC2(CCCN(C(C3(C=C)CC3)=O)C2)C1 96665,Cc1nc(C(C)C)[nH]c(=NC(C(C)NC(=O)C(n2cc(Cl)cn2)C)C(C)C)c1C 96666,C1(C(=O)NCC2COCCN(C(=O)CCCOCF)C2)CC(=O)C12CCCC2 96667,C12(C(=O)NCC3CN(C(c4cnc(C5CC5)o4)=O)CC3O)COCC1C2(F)F 96668,c1(CCC(=O)NC(C(C)C)CNC(C2CSC2)=O)nc2ccccc2o1 96669,CC1=C(C)CC(C)(NC(=O)C(C(C)O)NC(c2c(C)cnnc2O)=O)CC1 96670,CC1=NS(=O)(=O)N(C)C=C1C(=O)NCC1C=CC(NC(=O)C(C)CC2CC2)C1 96671,C1(C(N2CC(NC(CSCC)=O)C2)=O)CCC2CCC1O2 96672,C1(NC(=O)CNCCC)CN(C(C2CCN(C(=O)OC(C)(C)C)C2)=O)C(C)(C)C1 96673,c1(CC(C)C)ccc(C(N2CCC3CC23C(=O)O)=O)cc1Br 96674,N1(C(C(CC)C#N)=O)CC(C)(C)C(NC(C2CCCOC2)=O)C(C)(C)C1 96675,CN1CC(C(=O)NCC2CCCCN(C(=O)C(=O)C(F)(F)F)C2)CCC1=O 96676,N1(C(C(C(=O)OC)C)=O)CC2CN(C(=O)CCN3C(=O)C=CC3=O)C2C1 96677,c1(OCc2ccc(OC(F)F)cc2)cc(C(=O)OC)nc(CC23CC(C2)C3)n1 96678,C1(CNC(CN(C(C)C)C)=O)CN(C(=O)C(C)Oc2ccccc2Cl)C(C)(C)C1 96679,c1(C(=O)NC2CN(C(CC3C(C)(C)C3)=O)C(CO)C2)cc2c(s1)CCCC2 96680,C(C(CC(C)(C)C(=O)OCC)OC)OC(N=c1cc(CC(=O)OC)s[nH]1)=O 96681,N1(C(Cc2c(C)nc(S)s2)=O)CCCN(C(c2nocc2Cl)=O)C(CO)C1 96682,c1(C(C(=O)N(CCC)CCNC(C2CCCO2)=O)(C)C)cccc2ccccc12 96683,c1(C(=O)NC2(C)CN(C(=O)CC3(O)CC3)C2)cc2c(cc1[N+](=O)[O-])OCCCO2 96684,Cc1cc(N)cnc1C(=O)NC1CC2CC(NC(c3csc(C(N)=O)n3)=O)C1C2 96685,N1(C(C(C2CCCC2)OCC)=O)CC2CCC1CN2C(=O)C(c1ccccc1)O 96686,c1(C(=O)NCC(CNC(=O)Cn2cnnc2O)O)cc2cccc(F)c2s1 96687,c1(N(C(C2C3CN(c4ncc(C(=O)OC)cn4)CC32)=O)C)ccc(C)c(Br)c1 96688,C1(CC(=O)NCC(C)N(C(=O)CCc2conc2C)C)(CC=C)CCCCC1 96689,c1(C2(C(=O)NC(C)CN(C)C(C3CC(F)C3)=O)CC2)ccc2c(c1)OCO2 96690,C1(C(=O)NCCc2c(C)n[nH]c2C)(NC(Cc2cc(C)on2)=O)CCN(C)C1 96691,c1(N(C(C)(C)C)CC(N2CCCCC2)=O)cccc2c1C(=O)CC2 96692,C(=O)(C1Cc2ccc(Cl)cc21)NC1(CO)CCCN(C(c2c(CC)cno2)=O)C1 96693,CC1(C)CCC(C)(NC(=O)CC2CCCN(C(=O)CCP(C)(C)=O)C2)C1 96694,Cc1cc2ccc(C(N3CCC(NC(=O)C(C)C4CC4)C(F)C3)=O)cn2c1 96695,C1(C(N(C)CC)=O)CCN(C(=O)CC2CCCN(CCOC)C2)CC1 96696,c1(C(C(=O)NC2CC2)N(CC(CC)C)CCOC)ccc2c(c1)oc(=O)n2C 96697,Cc1nc(CCC(=O)NC2CCN(C(c3ccc(C)n3C)=O)C2C2CC2)[nH]c1C 96698,Cc1ccn2ncc(C(=O)NC3(C)CCCN(C(C4CCSC4)=O)C3)c2n1 96699,c1(C(=O)NC2C(CNC(C(C)OCC(C)C)=O)CC2)cccc2nccnc12 96700,C1(CNC(=O)CC2CCCCC2)CCN(C(C2C3CCCC23)=O)CC1O 96701,N1(C(C=CC(CC)=CC)=O)CCC(NC(c2cc(C)[nH]n2)=O)CC1C 96702,c1(C(N2CCC(C3N(C(=O)OC(C)(C)C)CCC3)C2)=O)ccc(F)c(Cl)c1 96703,Cc1cccc(NC(=O)C(=O)N(c2cncc(F)c2)CCCC(C)O)c1 96704,C1(CCNC(CC=C=C)=O)CCCN(C(c2cncc(N)n2)=O)CC1 96705,C12(C(=O)NC3CC(N(C(CCn4c(C)csc4=O)=O)C)C3)CCC(=O)N1CCS2 96706,Cc1cc(Cl)c(C(=O)NC2CC(C)N(C(C3CC(CF)C3)=O)C2)s1 96707,c1(C(=O)NCC(C(C)C)NC(C2CCCC(OC)C2)=O)cncc2[nH]ccc12 96708,C1(C(N(C2CCN(C(c3cnns3)=O)C2)CCC)=O)CCC(C(F)(F)F)O1 96709,CC1CN(C(C2CC2F)=O)CCCN1Cc1ccc(CNN2CCCCC2)cc1 96710,c1(C(N2C(C)CN(C(=O)C=CCBr)CC2)=O)ccc(O)cc1[N+](=O)[O-] 96711,c1(CNC(=O)NC2CC(C)SC2)ccccc1C(F)F 96712,N12CCn3ncc(c3C1)SCC2=O.N1(C(=O)OC(C)(C)C)CC(F)C1 96713,N1(C(CSC)=O)CCC2CCC(C1)N2C(c1cc(OC)c(N)cc1F)=O 96714,C1(NC(C(CCOC)C)=O)C2CCN(C(=O)C(C)(C)COC(C)C)CC12 96715,C1(C(=O)NCC2(CN(C)C(c3cc(C#N)cs3)=O)CC2)CCc2ccccc2C1 96716,C1(NC(C(=Cc2cn[nH]c2)C)=O)COC2(C1)CN(C(c1ncc(F)cc1C)=O)C2 96717,N1(C(c2cccc(Cl)n2)=O)CCC2CCC(C1)N2c1ncnc2ccsc12 96718,c1(C(=O)OC)cc(CCOC(C)C)cc(S(=O)(=O)NC(c2ccc(Br)cc2)C)c1 96719,C12(C(=O)NCCC(C)OC)CC(CO)(CN1C(=O)CC1CCCC(=O)N1)C2 96720,c1(COC2C(=O)N(c3cccc(Cl)c3)CC2)cc(I)c(Cl)cc1Cl 96721,c1(C(=O)NC2C(NC(C(C)OCC#C)=O)CC2)cc(N)ccc1O 96722,CC(CNC(=O)OC(C)(C)C)C(=O)N1CCC(n2cc(CNC(=O)CO)cn2)C1 96723,Cc1cc2c(cc1C)C(C(=O)NCC(C)CNC(=O)CC1(C#N)CC=CC1)CO2 96724,C(=O)(C1=C(C)N(C)c2nnnn2C1C)NCCN(C(C(CC)OCC)=O)CC 96725,N1(C(CCCSC)=O)CCOC2CCN(C(C3CCCOC3C)=O)CC12 96726,c1(C(=O)NCCC2(C)CCN(C(c3c(C)nc(SC)o3)=O)C2)cc(C)cc(O)n1 96727,c1(CC(=O)NCC2N(C(C34CC(OC)C3C4)=O)CCC(C)C2)c[nH]c2cccnc12 96728,c1(CC(=O)N(CCC(C)NC(C(CC)N(C)C)=O)C)coc2c(C)c(Cl)ccc12 96729,CC1NC(=O)OC12CN(C(=O)CCOCCN(C)C(c1cnsn1)=O)C2 96730,C(CCC(CCC)NC(c1c[nH]nc1-c1ccncc1)=O)NC(C(C)OCC)=O 96731,C(=O)(C1CCc2nccn21)NC(C(C)C)CNC(c1ccc(C(=O)N(C)C)cc1)=O 96732,C1(NC(c2cncc(OC)c2)=O)CCCN(C(C2C=CCS2)=O)C1C 96733,Cc1cn2c(n1)C(C)CC(C(=O)NCC1CCN1C(=O)C#CC(C)C)C2 96734,Cc1cc(N2CCC(NC(c3cn(C)cn3)=O)C23CCC3)ccc1[N+](=O)[O-] 96735,N1(CC(CC)C(C)C)C(=O)CN(CCCc2nccs2)C1=O 96736,c1(NC(C(=O)NC2(COC)CCOCC2)=O)ccc2c(c1)N(C)C(=O)CO2 96737,c1(CCN=C(NC(C#C)C)NCCC(=O)NC)ccc2[nH]ccc2c1 96738,C(=O)(C(CC(C)C)C(C)C)NC(C(=O)NCc1c(OC)ccnc1)CCF 96739,C(=O)(CC(C)(C)C)N1CC(NC(C2CCN(C(C)=O)C2)=O)(CO)C1.C1(=O)C(C)N1 96740,C12(C(=O)NCCN(C(C3C(C=C)C3)=O)CCC)CC1CCC2(F)F 96741,c1(C(=O)NCC2(C(C)NC(C3C(CC)C3)=O)CC2)cnc(C)o1 96742,c1(CC(=O)NC(C)CNC(C2CCC2)=O)ccc2ccncc2c1 96743,N1(C(c2cc(C)cc(Cl)c2)=O)C2CCC1CC(CNC(C1CCCSC1)=O)C2 96744,C1(NC(C(CC)n2ccnc2)=O)CC2(C(=O)N(CC)Cc3cc(C)on3)COC1C2 96745,Cc1cc(O)ncc1C(=O)NC(c1ccccc1)CNC(c1ccc(SC)s1)=O 96746,c1(NC(C2CN(S(=O)(=O)C(F)(F)F)CCC2O)=O)cc(Cl)ccc1I 96747,O=C1CN(CC(=O)NCCNC(c2csc(C(F)(F)C(F)(F)F)c2)=O)CCN1.C1(SC)CC1 96748,CC(C)C(O)C(F)(F)C(=O)N1CCCC(n2cc(CNn3ccsc3=O)nn2)C1 96749,CC(C)(C)CC(C)(C)C(=O)NC1CN(C(=O)C(C)(C)Cc2ccccc2)CC1O 96750,N1(C(Cc2cn(C)nc2)=O)CCC2CN(c3ccc([N+](=O)[O-])cc3F)CC2C1 96751,Cc1cc(N2CCCC(C)C2)nc(=NCCc2ccc(Br)cc2F)[nH]1 96752,c1(C(=O)NC(C(=O)NC2C(OC)C3(C2)CCC3)CC(C)C)cccc2cncn12 96753,C(=O)(C1=CCN(C(=O)C(C)(C)n2cccn2)C1)NC(C1CCN(C)C1)C 96754,Cc1nsc(N)c1C(=O)NCC1(O)CCN(C(c2ccoc2Cl)=O)C1 96755,CC1C(NC(=O)CCCC(N)=O)CC2CCC1N2C(=O)C(F)(F)CO 96756,C1(C)(CC)CC(C(=O)NCCCC(CO)NC(=O)CN2CCCC2=O)CCO1 96757,CN1CCN(C(N2CCOCC2C(N2CCCC(CO)C2)=O)=O)CC1 96758,C(=O)(CC(F)(F)C(F)(F)F)NCC(C)(C1CC1)NC(CCOCC#C)=O 96759,C1(NC(=O)C=C2CCCC2)CC2C(NC(=O)CN3CCCS3(=O)=O)C2C1 96760,N1(C(c2c(C)cncc2)=O)C2CCC(C2)C1CNC(=O)CSCC1CCCCO1 96761,C1(C)(CC(=O)N(C)CCNC(c2csc(C3CC3)n2)=O)CCS(=O)(=O)N1 96762,C(CO)(CO)(CO)NC(C1(NC(C(C)n2cncn2)=O)CCC1)=O 96763,N1(C(C(N2CCN(C(=O)OC)CC(C)C2)=O)=O)CCC2(CC1)CNC(=O)C2O 96764,N1(C(C(C)c2cc[nH]n2)=O)C2CCC1CC(CNC(C1(CF)CCC1)=O)C2 96765,N1(CCN(C)C)CC(C(=O)NCC(C)(C)CNC(C2CCCC(=O)O2)=O)CC1=O 96766,C(=O)(CC(F)(F)C(F)F)NCC1(C)CCN(C(C)=O)C1.c12ccc(cc1Cl)[nH]c2=O 96767,c1(SC)ccc(O)c(C(=O)NCC2C3CN(Cc4cnn(C)c4)CC23)c1 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96785,CC1(C)C(C(=O)NCC2(O)CCSC2)CCN1C(c1ocnc1C1CC1)=O 96786,CC12CN(C(c3ccc[nH]3)=O)CC1CN(C(C1(C3CCCO3)CCC1)=O)C2 96787,N1(C(C(OCC)SC)=O)CCCC(C)(C(N2CCCC(F)(F)C2)=O)C1 96788,c1(N(C)CC2(CNC(C(C)(C)C)=O)CC23CCC3)ncncc1I 96789,CC1(C)NC(=O)N(n2cc(C3CCCN(C(=O)CSCC(C)(C)C)C3)nn2)C1=O 96790,Cc1cc(N2CCC(F)(CO)C2)ncc1S(=O)(=O)NC1CCCOC12CCC2 96791,c1(OC(C)(C)C)cccc(C(=O)NCC2(OC)CCN(C(c3ccon3)=O)C2)n1 96792,N1(C(c2c(CC)c[nH]n2)=O)CC(NC(=O)C(C)c2cncs2)CCC(O)C1 96793,c1(OC)cc(N)cc(C(N2CCC3(NC(=O)COCC(C)C)CC3C2)=O)c1OC 96794,N1(C(=O)OC(C)(C)C)CCc2[nH]nc(C(N3CCC(F)(F)C(O)C3)=O)c2C1 96795,c1(OC)c(Cl)cc(C(=O)NC2CC(NC(c3nccc(C)n3)=O)CC2O)nc1Cl 96796,N1(C(CC(C)F)=O)CCN(C(=O)CC2CCC(F)(F)CC2)CC12CCC2 96797,C(=O)(C(Cc1ccoc1)CC1(NC(=O)Cc2cncs2)CCC1)N(C)OCC 96798,C1(NC(c2nc(C)sc2)=O)CN(CCCCS(C)(=O)=O)CCC1C 96799,CC1(C(=O)NCC2CCC(F)(CNC(c3ccc(C(N)=O)o3)=O)C2)CCC(=O)N1 96800,Cc1cc(C)c(C(N2CC(C(=O)NCC(O)CF)C(C)C2)=O)cn1 96801,c1(C(N(C)CC2OCCN(C(C3(CC)CCCC3)=O)C2)=O)cc(F)c(O)c(F)c1 96802,C=C=C(C)CC(=O)NCCN(CC(C)O)C(=O)CN(C1CC1)CC 96803,c1(CNc2c(C)nc(Br)cc2)cnc2c(c1)CN(S(=O)(=O)c1ccc(I)cc1)CC2 96804,C1(NC(CCc2cc(OC)no2)=O)(CO)CCN(C(C2COCCO2)=O)C1 96805,N1(C(CCC(N)=O)=O)CC2CCCCN2CC1CNC(=O)CC1CCOCC1 96806,N1(C(c2cnc(C)s2)=O)CCC(C)(C(=O)NCCC2CCCC2(C)C)C1 96807,C1(NC(C2C(=C)C2)=O)(CO)CCN(C(=O)C(c2ccc(F)c(F)c2)O)CC1 96808,N1(C(CC2ON=C(CC)C2)=O)CC(F)(F)CC1C(=O)NCC(F)C(C)(C)O 96809,C1(NC(C(=O)Nc2cc(C(C)C)sn2)=O)CCCN=C(I)CC1 96810,CC1(C)CC1(C)C(=O)NCCC1CC(C(=O)NCc2csnc2C2CC2)C1 96811,CC(C)C(O)CC(=O)NCC1(NC(c2ccc(C3OCCO3)cc2)=O)CCCC1 96812,N1(C(c2c(OC)nccc2)=O)CCCC(C)(NC(c2cn3ccsc3n2)=O)C1 96813,C1(CCCNC(=O)CCOC2CCC2)CCOC1.CC(C)=CC(=O)NC(C)(C)C 96814,c1(OC)cccc(CC2CNC2=O)c1.N1(C(C)=O)CCN(C(=O)CCBr)CC1 96815,c1(C(=O)NC2C(CNC(C(C)(C)c3ccsc3)=O)C2)ccc(SC(F)F)nc1 96816,C#Cc1ccc(C(=O)NCC(O)CN(C)C(C2CC2C(N)=O)=O)cc1 96817,CCC(C)(COC)C(=O)NC(CNC(c1ccc(OC)nc1Cl)=O)C(C)(C)C 96818,Cc1cccnc1C(C(C)C)NC(C1CCCC1n1cc(CO)nn1)=O 96819,C1(n2cc(C(=O)NCC3(F)C(C)C3)nn2)CCCN(C(C2CCC2)=O)C1 96820,N1(C(Cc2c(C)nn(C)c2C)=O)C2CCC1CN(C(C1CC(=C3CCC3)C1)=O)C2 96821,c1(COC(CC)C)ncccc1CNC(=O)CSC(C1CN(C)C(=O)N1)=O 96822,C1(NC(C(CCC(C)(C)C)NC(Cc2c(C)n(C)cn2)=O)=O)CCNC(=O)CC1 96823,C1(CC)CN(C(c2cn3c(n2)SCC3)=O)CCC1NC(c1coc(C(C)C)n1)=O 96824,c1(N(C(c2ccnn2CC)C(=O)NC(CC)C)C)ccc(C)c(F)c1 96825,C1(C2CCN(C(c3cnc(OCC)s3)=O)CC2)(NC(C=C(CCC)CCC)=O)CC1 96826,CC1(C)CCC(F)(F)CC1C(=O)NC1CCN(C(=O)CC2CC=CC2)CC1F 96827,C1(C(=O)NC2CCCC(NC(C3CCC(N(C)C)CC3)=O)C2)(OC)CCCCC1 96828,C(=O)(C1=COCCO1)NCC1C(NC(c2n[nH]c(C)c2Cl)=O)CCCC1 96829,N1(C(c2c(CC)ccs2)=O)CCCC2CN(C(c3cccc(C)c3N)=O)CCC12 96830,CS(=O)(=O)c1ccc(NC(C23CC(NC(=O)Nc4cncnc4)(C2)C3)=O)cc1 96831,c12ccc(cc1)NC1CCC21.n1(CC)cncc1CNCC 96832,CON(C(=O)C=CCNC(C1CCCCO1)=O)Cc1ccc(C)cc1 96833,C1(c2cn(C3CCN(C(C(C)(C)OC(C)=O)=O)C3)nn2)C(C)(C)C1(C)C 96834,N#CC1CCC(C(=O)NC(CC2CC2)C(=O)NC2CCCC(C(N)=O)C2)C1 96835,C1(NC(c2scc(C(C)=O)c2)=O)CC(NC(c2cncc(C(F)F)c2)=O)CC1O 96836,C1(C)(CN(C(=O)CC2C=CCC2)C)CCCC1NC(c1sccc1Cl)=O 96837,Cn1ncc2c(C(=O)NC3CCC3NC(c3cnc4c(c3)CCC4)=O)ccnc12 96838,N1(C(C)C)Cc2ccc(C(=O)NCC3CC4CCC(C3)N4C)cc2C1=O 96839,c1(NC)ccc(C(N2CC(NC(=O)CCc3ccc(O)nc3)C(F)C2)=O)cc1F 96840,N1(C(C=C2CCC(C)CC2)=O)CC2CCC(CNC(C3CCCCN3C)=O)C2C1 96841,N(C(O)=C1C=CC(C(=O)NCC2CCCC(=O)N2)=NNC=C1)C(C)(C)C 96842,c1(OCCC)ccccc1C(=O)NCC(O)CN(C(=O)CNC(C1CC1C)=O)C.SCC 96843,c1(OC)ccc2[nH]c(C(N3CC(C)(NC(c4cnc(S)[nH]4)=O)C3)=O)cc2c1 96844,N1(C(CCNC(N)=O)=O)CCC(CCC(=O)NCCC(O)C(F)F)CC1 96845,C1(C(=O)NC2CC3(CN(C(COCC)=O)C3)OC2)CCC2(CC1)CC2(F)F 96846,c1(C(N2CCCCC2C)C(=O)NCC=C)cc(OC)ccc1Cl 96847,C(c1cn[nH]c1)=C(C)C(=O)NCCCn1cc(C(=O)NCC(=O)NCCO)nn1 96848,C(=O)(C(F)(F)C1=CCOCC1)N1CC2C(CNC(=O)CCCCC(F)F)(CC2)C1 96849,N1(C(C=C(C)C)=O)CCCC1C(C)(C)C(=O)N1CCC(OCC2CC2)C1 96850,C(=O)(C(C)(C)n1cc(Cc2ccccc2)cn1)OCC.C(C)(CN(C)C)S 96851,c1(C(=O)NCCC2CCN(C(C(COC)O)=O)C2)ccc(OC)c(SC(C)C)c1 96852,c1(C(=O)NCC2C(NC(c3c(C)c[nH]n3)=O)CCCC2)cc(Cl)ncc1Cl 96853,C1(CNC(C2C(=C)CC2)=O)CC2(CCN(Cc3cc(C)sc3C)C2)CO1 96854,C1(C(C)C)CCCN(C(c2cc(CNC(=O)COCCN(C)C)on2)=O)C1 96855,C(C)(CSC)(C(=O)NCc1noc(C)n1)NC(C(C=C)O)=O 96856,c1(C(C(=O)NCc2cccc(Cl)c2)N(C(CSC)C)C)ccnc(S(C)(=O)=O)c1 96857,c1(CNC(C(C2CC=CCC2)NC(c2ccc(C)s2)=O)=O)ccccc1N=[N+]=[N-] 96858,C(=O)(CC(C1CC1)NC(C1CCCN1C(c1cccs1)=O)=O)NC 96859,c1(OC)ccc(C(=O)NCCC2CN(C(C3C(C)(C)C3(C)C)=O)CCO2)nc1N 96860,N1(C(c2c(CC)cno2)=O)CCOCC1CC(=O)N(C1CCN(C)C1=O)C 96861,c1(C(=O)NCC(C2CC2)NC(c2n(CCC)ncc2)=O)cc(OC)ccc1OC 96862,C1(C(N2CCCCC2Cc2cn(-c3ccc(F)cn3)nn2)=O)CN2CCC1C2 96863,N1(C(C2CCCSC2)=O)CCN(C(=O)CSCc2ccccc2)C(C2CC2)C1 96864,n1(CC)ncnc1C(C)NC(=O)C(C1CCOC1)NC(=O)CN(CC(C)(C)C)C 96865,N1(C(CC2(C)CC2(Cl)Cl)=O)CC2CCC1C1CN(C(=O)Cn3cccc3)CC21 96866,N1(C(c2c(OC)nn(C)c2)=O)C(CNC(c2ccccc2O)=O)CC2COCC12 96867,C(=O)(C1CCCc2cccnc21)NCC1CN(C(C2C(C)C2C)=O)CC(C)(C)O1 96868,N1(C(c2c(CC)ocn2)=O)CC(C(=O)NCC2CCCC23CCC3)C(F)(F)C1 96869,C(=O)(C1=C(Cl)CCC(C)C1)NCC(C1CCCC1)NC(C1(C(C)C)CC1)=O 96870,C1(C(N2CCCC(CN(C(=O)CCC3CC3(F)F)CC)C2)=O)CCC2(CCC2)CO1 96871,c1(C(=O)NC2CCN(C(CSCCC(C)C)=O)CC2F)cc2cc(Cl)ccc2s1 96872,C(=O)(CC1=NN(C)C(=O)C1)NC12CC(CNC(C(CC=C)(C)C)=O)(OC1)C2 96873,S(=O)(=O)(c1ccc(N2CCC(C(N3CCC3)=O)C2)c(Br)c1)N(C)CCN(C)C1CC1 96874,N1(C(C2(CC#C)CC=CCC2)=O)CC2CCCC2(NC(c2cc(C(N)=O)c[nH]2)=O)C1 96875,Cc1cccc(C(C(C)C)NC(=O)NCCc2nc(C(C)(C)C)no2)c1 96876,C1(CNC(CCCC=C)=O)CCC(C)CN1C(c1ccc(-c2cn[nH]c2)cn1)=O 96877,CCC(CC(C)C)C(=O)N(C1(C(=O)NC)CC1)C.C12CCCC1C(=O)NC2 96878,C1(C(=O)NCC(C(=O)NC)(C)C)CN(C)CCN1C(=O)CN1CCC(OC)C1 96879,c1(OC)ccc(C(N2CCC(NC(c3cnc(C)nc3C)=O)C2)=O)cc1OC 96880,Cc1ccc(F)c(C(N2CC3CCC2C3NC(=O)Cc2n[nH]c(C)n2)=O)c1 96881,Nc1cc(C(N2CCN(C(=O)C(F)C3CCC3)CC2C2CC2)=O)c(F)c(F)c1F 96882,C1(C(=O)NCCC(CNC(=O)Cc2cncnc2O)O)CCC12CCOCC2 96883,C1(CNC(C2C=CCC2)=O)C2CN(C(c3cc(CC(F)(F)F)[nH]n3)=O)CC12 96884,N1(C(C2CN(OC)C(=O)C2)=O)CCC2CN(C(=O)C=CCO)C(C)C12 96885,C1(CC#C)(C(N2CC(O)C(O)C2)=O)CCN(C(c2coc(CCC)c2)=O)C1 96886,N1(C(C(C)NC(N)=O)=O)CC(NC(=O)C(F)(F)c2nccs2)C(C)C1 96887,C1(OC)(CNC(C2(c3ccccc3)CC2(F)F)=O)CN(C(C2CCO2)=O)C1 96888,CCC(CC)C(C(=O)N1CCC(CC(=O)NCC(C)COC)C1(C)C)OC 96889,c1(NCC=C)nc(N2CCCC(C(F)F)C2)c2c(n1)CCCCCC2 96890,C12(C(N3C(C)CN(C(=O)COc4cncc(Cl)n4)CC3)=O)CCOC1CCOC2 96891,C1(C(CC(=O)NCCN(C(CNC(CCC)=O)=O)C(C)C)C)CCCC(O)C1 96892,C(C(N)CC(F)(F)F)NC(C1CCCN(c2snc(CC)n2)C1)=O 96893,c1(C(C#C)N(CC(=O)C=CC2(OC)CC2)C)ccn(C)c1 96894,c1(CN2CC3C(C(=O)NCCC#C)C3C2)ccc(NC(C)=O)c(F)c1 96895,c1(CCCC(=O)N(CCN(C(C2(CC=C)CC2)=O)C)C)ccc(F)cc1F 96896,CCCCC(CC)C(=O)NCC(CCNC(c1c(CC)nn(C)c1CC)=O)OC 96897,CC(CC(=O)NCC12CC(NC(C3CNC(=O)N3)=O)(C1)C2)C(F)(F)F 96898,c1ccc(C(C)=O)cc1O.C(c1ccccc1)=CC(=O)NC(COCC)CC.C(C)C 96899,c1(NCC(CCNC(=O)NCC2(C(=O)OC(C)(C)C)CC2)O)c(F)cccc1F 96900,C1(C(=O)OCC)CCC(C(N2CCC(NC(C3CC(F)C(=O)N3)=O)CC2)=O)CC1 96901,c1(C(N(CC(C)(C)CNC(=O)CNC(=O)CC(C)(C)C)C)=O)c(F)c(F)ccc1F 96902,CC(C)P(=O)(CC(=O)NCCCC(C)(C)NC(N)=O)C(C)C.C1(=O)CCN1 96903,C1(C(N2C(CCNC(c3c(C)nc[nH]3)=O)CCCC2)=O)CNC(=O)CC1(C)C 96904,C1(CNC(C(COCC)n2cc(-c3ccccc3Cl)nn2)=O)COCCN1C=O 96905,C1(O)(C(=O)Nc2c(OCCOC)cccc2)CCCN(C(=O)Nc2ccsc2)C1 96906,Cc1ccccc1OCCCC(=O)NC1CCCC1NC(C1(O)CC(CF)C1)=O 96907,N1(C(CNC(N)=O)=O)CC(NC(C2(C3CCC3)CCC2)=O)CC12CCCOC2 96908,N1(C(Cc2ccn(CC)n2)=O)CC(C)C(N=c2[nH]c(SC)nc(Cl)c2C)C1 96909,C(C(C)(C)C(=O)NCCNC(N)=O)N(C(=O)C=C1CCCCC1)C 96910,Cc1cccc(O)c1C(=O)NCC1(CNC(=O)CC2CCOC2)CC12CCC2 96911,c1(C(N2CC(OCCNC(C(CC=C)OC)=O)C2)=O)cc2n(n1)CCCN2 96912,CCCC(CNC(c1cc(Cl)n(C)n1)=O)C(=O)NCC(O)C=O.OCC 96913,Cc1ccc(CC(C)N(C(C(n2cc(CN3CCCC3)nn2)C)=O)C)cc1 96914,N1(C(C(C)Cn2cccn2)=O)CCC(C)(C)C1CNC(=O)COCCCF 96915,C12(CNC(CS(CC)=O)=O)CCC(CC1)CN2C(c1cn2ccccc2n1)=O 96916,c1(C(C(N2CCC(NC(c3ncc(F)cc3Cl)=O)C2)=O)O)cc(Cl)cc(Cl)c1 96917,N1(C(CCC2CC(OC)C2)=O)CC2(CCN2C(=O)Cn2cnnn2)C1 96918,C1(CNC(=O)CCOC2CCC2)(NC(c2cc[n+]([O-])cc2)=O)CCOCC1 96919,Cc1cn(C)nc1C(N1CC(n2cc(Cn3cncn3)nn2)C(O)C1)=O 96920,C(=O)(CC1C(=O)Nc2ccc(F)cc21)NCCC1(C)CCN(C(=O)CNC=O)C1 96921,c1(CC)ccc(C(N2CCOCC2CN(C(=O)CCc2ccoc2)CC)=O)nc1 96922,C1(CC(=O)N(CC(C)NC(c2cccc(CCO)c2)=O)C)CCC(=O)N1C 96923,N1(C(c2cnc(NC(C)=O)o2)=O)CCN(C(=O)CCN2CCCC2=O)C2CCC12 96924,CC1C=C(C(=O)N(CCCNC(=O)Cc2ccccc2CC(N)=O)CCO)CC1 96925,CN1CCN(CCC(N2CCC(NC(=O)CNC3CC3)CC2)=O)CC1.C(C)(C)(C)C 96926,c1(C(=O)OCC)cnc(N2CCN(c3ccnc(C)n3)C3CC23)nc1C 96927,c1(NC(C2CC(NC(=O)OC(C)(C)C)C23CCC3)=O)ccncc1N=[N+]=[N-] 96928,C1(C(=O)Nc2c(C)cno2)CCC(C)(CNC(=O)C(C)COc2ccccc2)CC1 96929,c1(NC(C(=O)N(C(C)COC)CCOC)=O)cccc2cnnn12 96930,c1(C(=O)NC(c2ccc(S(C)=O)cc2)C)cnn2c1N(C)CCC2 96931,O=C(C1CCCc2nn[nH]c21)N1CCC2(C1)CN(C(c1coc(O)n1)=O)CCO2 96932,N1(C(C(C=C)(C)C)=O)CC2CCCC(NC(c3nn(C)cc3C(C)=O)=O)C2C1 96933,N1(C(C(CC)CN(C)C)=O)CCCC(F)(C(=O)NC(C)CN(C)C2CC2)C1 96934,CC1CN(C(C2CC2(Cl)Cl)=O)CC1CCNC(C1CCCCCC1)=O 96935,c1(C(=O)NC(C)CCCNC(=O)CCC2CCCN2C)nccn2ncnc12 96936,c1(CNCCN(C(=O)CN2CCC2C)CC)nccn1C(C)(C)C 96937,C1(CC(N2CCC(C)(CCC)C2)=O)CC2(C1)CN(C(C1(C)COCCO1)=O)C2 96938,C(=O)(CCCCCF)N(CC(C)(C)NC(C(C(=O)OC)C1CC1)=O)C 96939,c1(OCC(C)(C)NCCS(N)(=O)=O)ccccn1 96940,CC(C(=O)OC(C)(C)C)C(=O)NCCC1CC(NC(C2CCCN2N=O)=O)C1 96941,C(C(C)C(=O)NC(Cc1ccco1)C(=O)N(C1CC(CO)C1)C)SC 96942,c1(CC(=O)NCC2CCC(NC(C3CC3c3cccc(Cl)c3)=O)C2)ncccc1F 96943,c1(C(C(=O)NCC2CC(NC(C=CC=CC)=O)C2)C)ccc([N+](=O)[O-])cc1 96944,c1(NC(C(CC)n2nccc2C)=O)ccc(Br)c2c1CCO2 96945,C=C(C)C1CN(C(=O)C(C2CCOC2)NC(=O)CNC(=O)CN(C)C)CCO1 96946,c1(OC)cc(OC)nc(N2CC3CN(Cc4cc(Br)ccc4O)C3C2)n1 96947,C(CC(C)C)(C(=O)NCC(n1ccnn1)C)ONC(c1c(CC)nco1)=O 96948,c1(NC(c2ccc(F)cc2Cl)C)ccc(C=NO)cc1 96949,CC1CCCC1(C)C(N1CCOC(CNC(=O)Cn2ccnn2)C1)=O 96950,CC1(C)CCCC(CCNC(c2ncc(Cl)s2)C(=O)NCCCOCC2CC2)C1 96951,C1(NC(CCCn2c(C)ncc2)=O)CCN(C(=O)COCC2CCCC2)CC1O 96952,CCCCC(O)C(=O)N1CCN(Cc2cnc(OC)cn2)C2CC12 96953,C1(NC(C(C)N(CCOC)CC)=O)CCN(Cc2cnc(C(C)(C)C)s2)CC1C 96954,CC(Cn1cccn1)C(=O)NCc1n[nH]cc1C(=O)N(C1CCCC1C)C 96955,C1(CC)CCCCC1C(N1CCCCC1CCNC(c1cnccc1Cl)=O)=O 96956,C1(NC(c2ccc(O)cc2)=O)COCCN(C(C2CCN(C3CC3)C2=O)=O)C1 96957,C(CCO)(C(F)F)NC(C1(C)N(Cc2n(C(C)(C)C)ncc2)CC1)=O 96958,C#Cc1cc(OC)cc(C(=O)OC)c1.C1(=O)CN1CCF 96959,c1(OC)ncccc1C(N1CCC(CC(C)NC(=O)CCCn2ccnc2)CC1)=O 96960,c1(CCC(=O)N(CCNC(CCNC(C)=O)=O)C)ccc(Br)nc1 96961,c1(N2CCN(C(=O)C=Cc3ccc(Cl)cc3Cl)CC2)ncnc2ccc(Cl)cc12 96962,c1(OC)cccc(NC(=O)C(c2c(C)noc2C)NC(c2cc[nH]c2C(C)C)=O)c1 96963,C1(C(N2C(CNCc3cncc(N(C)C)c3)CCC2)=O)CC(=O)N(C)C(=O)N1 96964,Cc1ccc(C(N2CCN(C(C3(c4ccc(F)cc4)CC3)=O)C3CC23)=O)cc1Cl 96965,Cc1cc(C(=O)NCC(C)(Cn2cccn2)NC(C2CN(C)C2)=O)n[nH]1 96966,CCC(C#N)C(=O)N1CCN(CCCNC(C2CC2C(F)(F)F)=O)CC1 96967,C1(C(N2CCN(C(c3nc(CC)oc3)=O)CC(CO)C2)=O)CCc2nnnn2C1 96968,c1(OC)cc(C(N2CCC(O)C(C(=O)Nc3c(Cl)cccc3I)C2)=O)ccc1Cl 96969,C(=O)(C(CCc1ccccc1)N1CCOC(CN(S(C)(=O)=O)C)C1)NCCOC 96970,N12Cc3[nH]nc(c3C1)C2=O.Cc1ccc(CSCC(=O)NCC(N)C(N)=O)cc1 96971,N1(C2CN(C(CCc3cnc(C)o3)=O)C2)CC(C(=O)NCc2cn[nH]c2)CC1=O 96972,c1(C(N2CC(CCOC)N(C(=O)CN(C)CCO)CC2)=O)cc2cccnc2s1 96973,c1(SCCn2c(COCC)nnc2N(C)C)cccc(S(F)(F)(F)(F)F)c1 96974,CC(C(=O)NC1(C2CCCN2C(c2ccc(CCC3CC3)cc2)=O)CC1)C(C)(F)F 96975,C1(C(=O)NCc2ccc(SC)cc2)CCN(CC2CCCN(C)C2)CC1O 96976,C12(C(=O)NC(c3cnc(C4CC4)o3)CNC(=O)CC3CCCC3)CCCN1CCC2 96977,N1(C(c2cccc(F)c2F)C(=O)NCCCOC)CCC(O)CC(C)(C)C1 96978,Cc1nc(NCCC2=CCCCC2)cc(N2CCCN(CCC(F)F)CC2)n1 96979,c1(C(=O)NC(C(c2ccccc2)NC(CC2CC(=C)C2)=O)C2CC2)ncc(C)s1 96980,C=C(C)CC(C(=O)NCc1ccc(C(=O)NOCC2(O)CCCCC2)o1)OC 96981,C(C(=O)Nc1noc(C2(C)CC2)n1)(C(C)C)OC 96982,C=C=C(C)CC(=O)N(CC(=O)NC1CC(OC(C)C)C1)CC 96983,C(Cc1cc[nH]n1)(C(=O)N(CCCF)CC)NC(C=CC=CCC)=O 96984,Cc1cc(Br)ccc1C(=O)NCC(C(C)C)NC(C1(C)CC(C)(C)C1)=O 96985,CCCC(C)(O)CC(=O)NC(c1ccc(NC(=O)C(C)COC)cc1)C 96986,Cc1cc(=NC2CCCCC2C)[nH]c(N2CCc3nc(-c4ccsc4)sc3C2)n1 96987,CC(C)C(C)CC(=O)NCC1(C)CC=CC1.N12CC(CC1=O)C(=O)N(C)CC2C 96988,c1(C(=O)NC2CCCC2C(=O)Nc2ncccc2Br)c(Br)cccc1Br 96989,c1(C(N2C(CNC(CC)=O)CC(C(F)(F)F)C2)=O)cc2c(cc1F)NC(=O)CC2 96990,c1(C(C)CC(=O)Nc2cn[nH]c2)cccc(I)c1 96991,CCC(C)CC(C)n1c(N(C(C)C)Cc2cccc(F)c2)nnc1C1CCOC1 96992,c1(C(=O)Nc2cnccc2[N+](=O)[O-])cc(-c2ccc(CO)o2)cc2c[nH]nc12 96993,CC(C)C(C)CC(=O)N(C1CC(C(=O)NCC(O)(C2CC2)C2CC2)C1)C 96994,c1(C(=O)NC2(C)CN(C(C3CCc4n[nH]cc4C3)=O)C2)cc2n(n1)CC1(CC1)C2 96995,Cc1ccc(CN2CC(F)(C(N3CCOC(C#N)C3)=O)C2)cc1Cl 96996,CC(CN(C)C)CCC(=O)N(CC(C)NC(=O)CC1CCC(=O)C1)C 96997,C(CC(C)(C)C)(C(=O)NC(C)(CNC(=O)CSc1cnn(C)c1)CC(C)C)OC 96998,C1(C)(C(=O)NC(CC)C(F)(F)F)CCCN(C(c2cc(C)n(C)c2)=O)C1 96999,C(C)(CC(C)(C)C)(c1n(CCOC)nnn1)NC1CC(F)(F)C1(C)C 97000,c1(C(=O)NCCN(C)C(c2ccc(Cl)c(Cl)c2)=O)cc2sccc2[nH]1 97001,c1(-c2cccc(COCC(C)C)c2)nc2c(s1)CCN(CC1CNC(=O)C1)C2 97002,C1(c2cn(CC3CC(CNC(c4n[nH]cc4Cl)=O)C3)nn2)CCOCC1.CC 97003,Cc1cc(=NC2CCCn3ccnc32)[nH]c(N2CC3C(CO)C3C2)n1 97004,N1(C(C2C(c3c(C)cccc3)C2)=O)CCN(C(c2nc(O)c(C)s2)=O)CCC1C 97005,C1(C(=O)NC(CNC(Cn2cnc(C(C)=O)n2)=O)C(C)(C)C)CCCC2(CC2)C1 97006,C#Cc1cccc(C(N2CCCC2CCC(=O)N(C)CCc2cccs2)=O)c1C 97007,Cc1cnn(C)c1C(=O)NCC(CC(=O)NC(C)(C)CC(C)C)C1CCC1 97008,c1(C(N2C(CC=C)(C(=O)NC3CC(F)(F)C3)CCC2)=O)cc(C)cc(C#N)c1 97009,c1(CCC(=O)NC(C(C)NC(C2(C(=O)N(C)C)CC2)=O)C)ccc2ncccc2c1 97010,c1(C(=O)NCC2(C)N(C(C(CCC)OC)=O)CCC2)sc2ncccc2c1Cl 97011,c1(C(=O)NCCC(C(C)C)NC(c2cccc(O)n2)=O)ccc2c(c1)CCOC2 97012,C1(NC(c2cc(C)nc(O)n2)=O)C2CCCCN(C(=O)Cc3c[nH]nc3C)C12 97013,C(=O)(C1=C2CCN=C2NC=C1)NCC(CNC(C1N(C)CC(C)(C)C1)=O)O 97014,C(=O)(C1=COCCC1)N1C(C)CC(NC(=O)Cc2ccccc2CC2CC2)C1 97015,C(=O)(C1OCCn2ccnc21)N(CCCCNC(C1(C(=O)NC)CCC1)=O)C 97016,C1(CNC(C(=O)Nc2ccc(C)cc2)=O)CCC2CN(C(C)(C)C)CC12 97017,c1(-c2onc(-c3cccc(OC)c3)n2)cccc2cc(OC)ccc12 97018,C12(CNC(c3cccc(CCC)c3)=O)CCC(C1)N(C(=O)C(C)N(C)C)C2 97019,CC(F)(F)CCCC(=O)NC1CC(F)CN(C(c2c(F)cccc2Br)=O)C1 97020,CC1=C(C(=O)NCCN(CC(C)O)C(N2CCN(C(=O)C(C)C)CC2=O)=O)CCO1 97021,C1(C(N2C3C(CNC(C(C(C)O)C)=O)CC(CC3)C2)=O)CCc2cnn(C)c2C1 97022,N1(C(C(C)(C)O)=O)CC2CCC1CN2C(C1(C#N)CCC1)=O 97023,C1(C(=O)NC2CC(C)(CNC(CC(=O)OCC)=O)C2)CC2(CCCO2)C1 97024,C1(C)(C(=O)NC23CC(NC(CCSC)=O)(C2)C3)C2CCC(C2)C1(C)C 97025,N(C1COc2ccc(F)cc21)C(C1=C(C)OCC1)=O 97026,N1(C(C(N2C(C)CN(c3ccncc3)CC2)=O)=O)CCC(C2(O)CCC2)CC1 97027,CN1CCC1CNC(=O)NOCC1CC1 97028,CC1Cc2sc(C(=O)C(N(CCNO)CC(F)F)=O)cc2C(C)C1.C(=O)C(O)C(C)(C)C 97029,c1(CNCC2C(OC)(CO)CC2)sccc1S(N)(=O)=O.n12cc(nn1)CNC(=O)C2 97030,C(=O)(C1CC(C)(C)Oc2ccccc21)N1CCC(NC(c2n(C)cnc2)=O)C1 97031,N1(C(c2cccn(C)c2=O)C(=O)NC2CCCC2)CCc2c(ncn(C)c2=O)C1 97032,O=C(C1CCCc2nn[nH]c21)N1CCCC(N(c2ncnc(Cl)n2)CCO)C1 97033,Clc1ccc(-c2nc(CC3CC4CCC3C4)n(C34CCN(CC3)C4)n2)cc1Cl 97034,N1(C(c2ccnc(OC)n2)=O)CC(CNC(=O)OC(C)(C)C)CS(=O)(=O)C1 97035,Cc1ccc(CC(=O)NC23CC2CN(C(=O)CN2CCCC2=O)C3)c2ccccc12 97036,c1(C(=O)NC(c2ccc(F)cc2)CNC(CC(C)CF)=O)cnn2ccccc12 97037,c1(C(=O)NCC2COCCN2C(c2ccnnc2O)=O)c[nH]c2ncnc(O)c12 97038,Cc1ccc([N+](=O)[O-])cc1C(=O)Nc1cnc(Br)c(Cl)c1.c12cccnc1NC2 97039,C1(C(=O)NCC2CC(NC(COC(C)(C)C)=O)C2)CCC(n2cccc2)CC1 97040,c1(C(N(CC(C)NC(=O)CC2CCC2(C)C)C)=O)nsc2ccccc12 97041,Cc1[nH]nc(C(=O)NC2CN(C(=O)C=CCF)CC2C(F)F)c1C 97042,N1(C(C(C(=O)OCC)(C)C)=O)CCc2ccccc2C(NC(=O)C(O)C2CC2)C1 97043,CON(C(=O)C=C(C)CNC(=O)C(C(C)C)NC=O)C1CCC1 97044,CC1(C)CCOC1C(N1CCCCC1C1CCN(C(=O)C(O)C2CCCC2)C1)=O 97045,C(=O)(CC(O)CC(C)C)NCC(C1CCCCC1)NC(C(CC)(CO)OC)=O 97046,C(=O)(CC(O)C(C)C)NC(C(=O)NCC1(C(=O)OCC)CC1)(C)CO 97047,C(=O)(C1=NOC(C)(C)C1)N(C1CCCN(C(=O)Cc2cc(OC)no2)C1)CC 97048,Cc1cc(C(N2CCCN(C(=O)CCCN3CCC3)CC2C)=O)cc2c1CCC2 97049,CCC(C)(O)C(=O)N1CC(NC(=O)Cc2sccc2-c2ccccc2)C(SC)C1 97050,Cc1noc(C)c1CC(N1CCC(N(C(=O)CCc2ccccc2F)C)C1)=O 97051,c1(C(=O)NC(CCCC)CNC(=O)CC(C)C2CC2)cc(C)c(C)c(Br)c1 97052,c1(NCC(C)N(C)C(C2CC(F)(CO)C2)=O)cc2nn[nH]c2cc1[N+](=O)[O-] 97053,N1(CCNC(C2CCC2)=O)CCN(C(=O)CC2CCC(=O)N2)CC1 97054,C1(C(N(C2CCSCC2)C)=O)CCCC(NC(=O)Cc2ccc(Cl)s2)CC1 97055,c1(OC)cc(C(N2CCC(CO)(NC(=O)C(CCO)N(C)C)C2)=O)cc(F)c1F 97056,C1(NC(C(C(CC)C)OC)=O)CC2CCC(C1)N2C(C1(C)CCOCC1)=O 97057,c1(C(C)NC(=O)CNC(N)=O)c[nH]c2ncc(C(=O)NC3CC=CCC3)cc12 97058,c1(C(C(=O)NCCC(CNC(C(C)(C)OCC)=O)O)CC)c(C)noc1C 97059,C(C)(CO)(C(F)(F)F)NC(CC1(CNC(C(COCC)C)=O)CC1)=O 97060,Cc1cc(Cl)cc(Br)c1NC(C1CC(F)CN1Cc1cnc(O)c(Cl)c1)=O 97061,C(=O)(CS(N)(=O)=O)NC12CC(NC(CCc3cc(C)on3)=O)(C1)C2 97062,N1(C(c2ccc(OC)s2)=O)CCC2CN(C(C3CCCC3C(F)F)=O)CC12 97063,N1(C(C2(C)CC2(Cl)Cl)=O)CCC(C)(NC(=O)CN2CCS(=O)CC2)C1 97064,N1(C(c2occ(C)c2)=O)CC2(NC(c3c(-c4ccsc4)noc3C)=O)CCC1C2 97065,CCC(C)(O)C(=O)NCCCN(C(=O)CC1CCCS1(=O)=O)C(C)C 97066,C12(C(=O)NCCC(C=C)C)CC(CN1C(C1C=CCCC1)=O)C2 97067,C(=O)(C1CCCc2nncn21)N(C(C(C)CO)Cc1ccccc1)C(=O)C(F)F 97068,n1(CCC)cc(C(=O)NCC2CCCC2NC(=O)C(C)SC(F)(F)F)cn1 97069,c1(-c2c(C(=O)Nc3n(C)nc(O)c3)csc2)c(Cl)cc(F)cc1Br 97070,c1(C(N2CCC(C)C2CNC(=O)OC(C)(C)C)=O)cc(O)nc(O)n1 97071,c1(C(=O)NCC2ON=C(C)C2)ccccc1NC(=O)C(CC1CCC1)NC(C)=O 97072,c1(C(=O)NOCc2ccccc2)ncn(Cc2cc(C(F)F)no2)n1 97073,C1(C(=O)NCC(C)(C2CCC2)NC(C=COCC)=O)CC2(C1)CC(O)C2 97074,CCCCC(CNC(C1OC(C)CC1C)=O)NC(=O)C(C)CSC 97075,CC1=C(C(=O)NC2CCN(C(c3c(F)ccc4nc[nH]c34)=O)C2)C(=O)OC1(C)C 97076,N=c1[nH]c(=NCC2CCN(CC(F)F)CC2)[nH]c(=NC2CCOC3(CCCC3)C2)[nH]1 97077,c1(C(=O)NCC2CCCN(C(C3(CO)CC3)=O)C2)ccc2c(O)nnc(O)c2c1 97078,CC(C(=O)NCC(c1ccc(Cl)cc1)N1CCOCC1)C1=CCCC1 97079,c1(NC(C2(C)CCN(C(Cn3c(C)cc(C)n3)=O)CC2)=O)ccc(C#N)c(Cl)c1Cl 97080,Cc1cc(C(=O)NCC(O)CNC(C2(O)CCCC2)=O)ccn1 97081,CCC(CCC(=O)NC(CN(C)C)C(=O)NCC1CCC(=O)NC1)OC 97082,Cc1nc(C(=O)NCCCCN(CCCNC(c2cnc(C)o2)=O)C)c(C)s1 97083,S(=O)(=O)(c1ccc(C(N)=O)cc1)NC1CC(CC(N2CCCC(F)C2)=O)C1 97084,CCCCCC(F)C(=O)N(C(C)C(N1CCOC2(CC2)C1)=O)C 97085,N1(C(c2nn(CC)nc2C)=O)CC(C)OC2(CCN(CC3CCC3)C2)C1 97086,N1(C(C2CC(=C)C2)=O)CC2CC(C1)CN(C(=O)CN(C)C(=O)OC)C2 97087,C1(C(=O)NC(CCO)C2CCCC2)C2CCC(C2)N1C(=O)CC1CSCCO1 97088,N1(C(C(CC)Oc2ccccc2C)=O)CCCC(C)(Cc2cc(C)on2)C1 97089,N1(C(C2CCN(C(C(C)CC3CCCC3)=O)C2)=O)CCC2(CCCCC2)C1 97090,c1(OC)ccc(C=CC(=O)NC(C)CCNC(=O)CC2CCCC(C)C2)cc1Cl 97091,C(CC(O)C(=O)N=c1ccn(C2CCC2)[nH]1)NC(=O)C=CC1CCOCC1 97092,c1(NC(C(N2CC(C=O)C2)=O)=O)cc2c(s1)CCC2C(=O)OC(C)(C)C.CNC 97093,C(=O)(C1=NOC(C(C)(C)C)C1)NC(C1CN(C(c2ccc(CF)cc2)=O)C1)C 97094,c1(C(=O)NCC2OCCN(C(C(CC)(C)F)=O)C2)cc(OC)c(OC)c(F)c1 97095,C(=O)(CCCCC(F)(F)F)NCC1CCCC(CNC(C2C(CC)C2)=O)C1 97096,C1(N(C(C(CC)CC(C)C)=O)C)CCCC2CN(C(c3csc(=N)[nH]3)=O)CC12 97097,c1(CC(=O)NC2CN(C(c3ccc(Cl)cc3)=O)CC2O)ccc2ncccc2c1 97098,C(=O)(C(C)C(C)C(C)(C)C)N1CC(CCNC(c2c(OC)cc(F)cc2)=O)C1 97099,CC1(C)CC(CC(N2CC(C)(O)C2)=O)C(=O)O1.C1(C(=O)NC)C2CCC3C(C2)CC13 97100,CC(C)(CN(C)C)C(=O)N1CCC(=CCNC(c2cncc(F)n2)=O)CC1 97101,N1(C(c2cn(CC(C)O)c(=O)cc2)=O)CCC2CN(C(C3(O)CCOC3)=O)CC12 97102,N1(C(c2ccc(C)cn2)=O)CCC(CNC(=O)CN2CCCCC2)CC1C 97103,c1(CC(=O)NCC(C)(CO)NC(C(F)=CC)=O)cccc(OC(F)F)n1 97104,c1(C(=O)NCC2N(C(c3c(C)cc(Br)cc3)=O)CCOC2)ccc2c(c1)NC(=O)C2 97105,C1(C(N2C(C)(CNC(C(C(C)C)NC=O)=O)CCC2)=O)CCCCN(C)C1=O 97106,c1(N(C(CCNC(C=COCC)=O)C)C)cc2c(cn1)C(=O)CCC2 97107,C1(CNC(c2cc(OC)no2)=O)CCN(C(c2c(Cl)cc(Cl)nc2N)=O)CC1C 97108,C1(C(C(=O)NCCOCC(C)(C)C)F)CCCN(C(=O)CCCn2cncn2)C1 97109,Cc1cc(C(=O)NCCN(C(C2CCC(=O)NC2)=O)C(C)C)cc(C)c1O 97110,C1(CC(=O)N(CC(C)(O)CO)C2CC2)C2CN(C(=O)CCCN(C)C3CC3)CC12 97111,C1(C(N2CCCC(CCNC(c3c[nH]cc(Cl)c3=O)=O)C2)=O)OC2CCC1CC2 97112,N1(C(C2C(=C)C2)=O)CC2(CNC(c3cc(Cl)ncc3OC)=O)CC1(COC)C2 97113,c1(OC)nc(N2CCOCC2CNC(c2ccc(F)c(C(F)F)n2)=O)cc(C)n1 97114,C=C(C)CCCC(=O)N1CC(C(=O)NC(C)(C)CCCF)OC(C)C1 97115,C1(C(=O)NC2CCC(N(C)C(c3cccc(C(F)F)n3)=O)C2)C2CC3C(C2=O)C13 97116,CC(C)(CCNC(C1(c2cccs2)CC1)=O)CN=c1[nH]c2cc(Br)cnc2s1 97117,C1(NC(C(N2CCSCC2)C)=O)CN(C(c2ccc(N)cc2O)=O)CC12CCC2 97118,C1(C(N2C(CN(C(CCC3C(C)C3)=O)C3CC3)CCC2)=O)CCCC1C1CC1 97119,N1(C(C2C(=C)C2)=O)CC2(C1)CN(C(=O)C(=O)NNC(=O)c1ccccc1)C2 97120,Cn1cnc(CC(O)C(=O)NCC(C)(C)NC(=O)CCc2cnoc2)c1 97121,C(CN=c1[nH]n(C)cc1[N+](=O)[O-])C12CC(NC(C3CCC(=C)CC3)=O)(C1)C(C)O2 97122,c1(C(=O)NCc2cc(C(N(C(CO)C3CC3)C)=O)sc2)cnn(C)c1Cl 97123,C(=O)(CCCC(=O)N1CCOCC1C(=O)NCC1(C)CC(O)C1)OCC 97124,c1(C(=O)NC(C)C(C)(C)NC(C2CCCCO2)=O)cc2n(n1)CCNC2=O 97125,C(=O)(C(C)(C)C(C)(C)O)N1CCCC(F)(C(N2CCC(OCC#C)C2)=O)C1 97126,CC(=O)C(C(C)C)c1nc(C(C)(CC)NCC(c2ccc(Br)cc2)=O)no1 97127,c1(C(N(CC(C)NC(=O)C(c2cccn2C)=O)C)=O)ccc(Br)cc1O 97128,c1(CC)nnc(C=CC(=O)NCCN(C(C2CC3(C2)CC3F)=O)CC2CC2)o1 97129,O=C1COc2cc(C(N3CCN(C(=O)C(F)C4CC4)CC3CO)=O)ccc2N1 97130,c1(C(C)=O)cc(=NCCC2CCCN(C(=O)CCC3CCC3)C2)[nH]cc1[N+](=O)[O-] 97131,C#CCC(C(=O)NCC(C)CNC(c1ccn(CC(C)C)n1)=O)C1CC1 97132,C1(CNC(C2(COC)CCOCC2)=O)CC2(CCN(C(=O)C(CO)C(C)C)C2)CO1 97133,C1(C(=O)NCC2(C#C)CCCC2)CCC2(CC2)N1C(c1ccc(C)n1C)=O 97134,C1(CNS(C)(=O)=O)CN(C)CCN1C(=O)CN(C)CC.c12cnccc1C(=O)N2 97135,C1(C(N(CC(=O)OCC)C)=O)(CNC(=O)CN2CCCC2=O)CC12CCC2 97136,C(=O)(N=c1[nH][nH]c2c1CN(C(c1occc1Br)=O)C2(C)C)c1ccc(OC)c(Cl)n1 97137,c1(C(C(=O)Nc2cncc(OC(C(=O)OC)C)n2)(F)F)cc(Cl)nc(Cl)c1 97138,c1(C(=O)NC(C2CCN(C(c3ccc(F)nc3)=O)C2)C)cc2cc[nH]c(=O)c2s1 97139,C(C(CC)(CC)Sc1ccccc1)NC(C1C(CC)COC1)=O 97140,C(=O)(C(C)(C)C(N)=O)NCC1C(NC(C2N(C(=O)NC)CCC2)=O)CCCC1 97141,N1(C(C(C(=O)OCC)OC)=O)CCC(C(C)C)CC1C(=O)Nc1cccnc1C 97142,C1(NC(C(C2CN(C(CC)=O)C2)OC)=O)CCN(Cc2coc(C)c2)C1 97143,C(=O)(CC1=CCN(C)CC1)N1CC(NC(c2cc(C(=O)OC)no2)=O)C1 97144,C1(NC(C(F)(F)C2(OC)CCC2)=O)CCC(NC(=O)C(C)OCCC(C)C)CC1 97145,c1(C(=O)NCC2C(C)CN(C(=O)C(C)(Cl)Cl)CC2)cnc2ncc(Cl)cn12 97146,CCC(CC(=O)OCc1ccccc1)C1CC1.n12cc(nn1)C(C)CNC(=O)C2 97147,N1(C(c2c(C)nc(C(C)C)s2)=O)CCN(Cc2ccncc2C#N)C2CC12 97148,N1(C(C=CC(C)(C)C)=O)CCC=C(C(=O)NCc2ncccn2)C1 97149,C1(C)(NC(C)=O)CCN(C(=O)CSCCN(c2ccccc2C)C)C1 97150,c1(OC)cccc(CCC(=O)NC(C)(C)CN(C)C(c2nncn2C2CC2)=O)c1 97151,C1(C(N2C(CCNC(C(N3CCNC3=O)C)=O)CCCC2)=O)CC2(CC2)CN1C 97152,Cc1ccc(SCC(=O)NCC2C3CN(C(C4CCCSC4)=O)CC23)cc1C 97153,c1(C(=O)NCC2CN(C(C3CC3[N+](=O)[O-])=O)C2)c[nH]nc1C.N1(C=O)CCCC1 97154,N1(C(c2nc(CC)oc2)=O)CC2(CC2)CC1C(=O)NCC1CC12CCOCC2 97155,C1(C(=O)NC(C2CCCCC2)CNC(Cc2c(C)occ2)=O)CCCC(=O)O1 97156,Cc1cnc(F)cc1C(N1CCC(Nc2nccnc2C#N)C1C)=O 97157,N1(C(CNC(CC)=O)=O)CCCC2CCN(C(c3cnc(C)cc3C)=O)CC12 97158,CN1CCCC(NC(=O)CSCCNC(C23CCC(C2)C3)=O)C1 97159,C1C(C)(C)C(=O)N2CCCC2C(=O)N1C(C)C.c1(C(CO)SC)ccc(F)cc1 97160,N1(C(C(C(C)C)NC(c2ccc(COC)[nH]2)=O)=O)CC(CN(C)CC)CC1(C)C 97161,N#Cc1ccc(NC(=O)CN(C2CCCO2)Cc2ccccn2)cc1F 97162,C(=O)(C#CC1CCC1)N1CCCC(N(C(c2ccc(N(C)C)nn2)=O)C)C1 97163,c1(C(N2CCC(=Cc3ccccc3)CC2)=O)cc(Br)c2occc2c1 97164,C1(NC(c2cc(C)nn2-c2ccccc2)=O)CC(N=c2[nH]cnc3cnccc23)C1 97165,C1(NC(CCC=CC)=O)C(C)(C)CN(C(=O)CC2CCNC(=O)C2)CC1(C)C 97166,C1(C)(CNC(c2c(CC)nc(C)[nH]2)=O)COCCN(C(C2CC(C(F)F)C2)=O)C1 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97376,Cc1cc(Cl)ccc1NC(=O)C(C)(C1CCC1)NC(C1CC(CF)C1)=O 97377,N1(C(c2c(C)nc(Br)s2)=O)CCC(C)(NC(C2CCC(=O)NC2)=O)CC1 97378,c12nc(cs1)CC(=O)N2.c1(C(C(=O)NCC(C)CSC)OC)csc(SC)c1 97379,N1(C(CCc2cncc(OC)c2)=O)CCN(C(C2CCCO2)=O)C(CO)C1 97380,N1(C(CCNC(=O)OC)=O)C(CNC(=O)Cn2cc(CO)nn2)CC2COCC12 97381,N1(C(c2cncn(C)c2=O)=O)CCC2(CCC2NC(=O)CN2CCOCC2)CC1 97382,Cc1cc(=NC2CCc3cc(Br)cnc32)[nH]c(NCc2ccc3nc(O)[nH]c3c2)n1 97383,c1(C(=O)NC2(C)CCN(C(C(C)NC(C)=O)=O)C2)cc2cc(Cl)cnc2[nH]1 97384,c1(C(N2C(C(N3CC(C#C)C(O)C3)=O)COCC2)=O)cccc2c[nH]nc12 97385,C(=O)(C1CCc2c[nH]nc21)NCCC(CC)(CC)NC(C(C)OCCOCC)=O 97386,n1(CC)nc(C)c(C(=O)NC2CC(NC(C3(OC)CCC3)=O)C(O)C2)c1Cl 97387,C(CCC(C)(C)C(=O)NCC(O)CC(C)C)NC(C(C)=CC(C)(C)C)=O 97388,CCCCCCCCC(C)C(=O)N1CCN(c2nc(Cl)nc3ccccc23)CC1 97389,C1(CNC(CC(C=C)C)=O)CC2CCC1N2C(c1ccc(CO)s1)=O 97390,Cc1cccc(Cl)c1C(N1CCC(C)C1CNC(=O)CCNC(c1ccco1)=O)=O 97391,CCC(C)C(C(=O)Nc1ccccc1)N(C(C)C)Cc1cc(C)sc1C 97392,C1(C(=O)NC2CCCC2)CCCN1C1CC1.C12(CC1)N(C)C2=O 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97516,C1(NC(C2(CO)CCCC2)=O)CCCCN(C(C2CN3CCC2CC3)=O)CC1 97517,N1(C(C2(OC)CCC2)=O)CC2CC1C2CNC(C1(c2ccc(OC)nc2)CCC1)=O 97518,Cc1ccc(F)c(C(F)(F)C(=O)NCCC(C)N(C(=O)CN2CCCC2=O)C)c1 97519,c1(NC(C2C(NC(C=C(C)c3ccco3)=O)C2)=O)c(O)cccc1O 97520,c1(OCC)cccc(CC(N2CCC(CCNC(C3(C)CC(O)CN3)=O)C2)=O)c1 97521,c1(C(=O)NCc2cc(C(F)F)on2)c(C2CC2)cccc1N 97522,n1(CC)cnc2c(NC3CC(NC(=O)COC4CCC4)C3)ncnc12 97523,C1(C2(C(=O)N(C)C)CCC2)CN(C2C(c3ccc(C)cc3)C2)CC1(C)C 97524,C1(CC)CN2CCCC2CN1C(c1cnn(CCF)c1)C(=O)NCC(C)C 97525,c1(CC(N2CC(CNC(C(CC)(O)c3ccccc3)=O)C2)=O)ccc(F)c(F)c1 97526,c1(C(=O)NC(CN(C(C(C)OC2CCCC2)=O)CCO)(C)C)ccc(=O)n(C)n1 97527,C1(C(=O)NCC2(OC)CN(C(c3cocn3)=O)C2)Cc2c[nH]cc2S1(=O)=O 97528,Cc1cc(CNC(c2cccc(Cl)c2)c2nnnn2C2CCC2)c(C)o1 97529,c1(C(=O)NCCC(CC)(CC)NC(=O)C(F)=C2CCC2)nn2cccnc2c1Cl 97530,N1(CCCNC(c2nnc(C)s2)=O)CCN(C(C2CC2C(=O)OC)=O)CC1 97531,C#CC1(NC(=O)C(CC(C)CC)NC(c2coc(C)n2)=O)CCCCCC1 97532,N1(C(CNC(C(CC)C)=O)=O)CC2C(NC(=O)CCCCN3CCCCC3)C2C1 97533,c1(C(=O)OCC)c(NC(=O)CC2CCN2CC)cccc1F.C1(C=O)CC(C)=NO1 97534,C1(NC(c2ccc(C)nc2)=O)C2CC3CN(C(=O)CN4CCC(C)(O)C4)C1C3C2 97535,c1(C(=O)NC(c2cn(CCOC(C)=O)nn2)CCC)cc2cccc(Br)c2o1 97536,c1(CC(=O)OC(C)(C)C)cc(C(=O)NC2CCC2NC(c2csnn2)=O)no1 97537,C(=O)(C(C#N)CC1CC1)NCC(C)(C)NC(C1CC(CCC)C1)=O 97538,c1(CC(=O)NC2C(NC(Cc3cc(C)ns3)=O)COC2)cccc(C(C)C)c1 97539,C1(NC(C2C(c3c(OC)cccc3)C2)=O)C(C)CCN(C(C2CCO2)=O)C1C 97540,C1(C(CNC(COCC)=O)F)CCN(C(c2nnsc2-c2ccccc2)=O)CC1 97541,c1(C(=O)NC2CC(CNC(C3(n4nccn4)CC3)=O)C2)ccc2c(n1)OCCO2 97542,C1(C(=O)NCc2scc(C(N(CC(CC)O)C)=O)c2)CCC(C)(C)C1 97543,Cc1cccc(F)c1CNC(C1CCCN(C(C2CC2C)=O)C1)=O 97544,CCC(C)(C#N)C(=O)NCCC1(NC(C2CC3(C2)CC3(F)F)=O)CC1 97545,c1(OC)ccc(S(=O)(=O)N(c2noc(C3CCC3)n2)C2CCCC2)cc1[N+](=O)[O-] 97546,CC1CC2(CCN(CC3CCC(F)C3)CC2)CN1C(=O)CCS(N)(=O)=O 97547,N1(C(C(C)CF)=O)CC2CC(NC(=O)CSCc3ccccc3Cl)C1C2 97548,N1(C(c2c(C)cnnc2)=O)CCCN(C(=O)CC2(C)CCS(=O)(=O)N2)C(CO)C1 97549,C(=O)(C(=O)N(O)C(C)C)NCC(C)N(C(c1cnc(C)nc1C1CC1)=O)C 97550,CC(c1ccccc1)=CC(N1CCC(C)(CNC(C2CC(C)(C)CN2C)=O)C1)=O 97551,c1(COC)csc(C(=O)NCC2(CO)CN(C(=O)C(F)=C(C)C)C2)c1 97552,C(=O)(CCC(=O)CCC(=O)N1CCC2OCC(=O)NC2C1)OC(C)(C)C 97553,C12(CCNC(C3CC(F)C3)=O)CCC1CN(C(c1coc(O)n1)=O)C2 97554,C1(CC)CCCCCN1Cc1cccc(-c2noc(C)n2)c1 97555,CC1CN(C(C(=O)NCC2CCCN2CC2CCCC2)=O)CCN(CCO)C1 97556,S(=O)(=O)(c1ccc(NCC2(C)CC2Br)c(Cl)c1)N1CCCC2(CC(OC)C2)C1 97557,C1(NC(C2C(COC)C2)=O)CCC(N(C(=O)Cc2cnn(C)c2C)C)CC1 97558,c1(C(N(CCC)CCNC(C2CC(OC)C2)=O)=O)cnc(C2CCCC2)nc1 97559,C12(NC(C(c3ccc(C)cc3)C)=O)CCC1CN(C(=O)CN(C)C(C)C)C2 97560,CC(=O)CCCC(=O)N(CC(O)CN(C(C)C)Cc1noc2c1CCC2)C 97561,c1(C(N(CCN(C(=O)C(C)(CC)CC)CC)CC)=O)ccc(Cl)nc1OC 97562,N1(C(c2cc(OC)n[nH]2)=O)CCC2(CCCCN(C(C3CCCS3(=O)=O)=O)C2)C1 97563,c1(OC)cc(N(C)CC2CCN(C(=O)CC3C=CCCC3)C2)nc(OC)n1 97564,c1(C(=O)NC(CC)CNC(c2ccc(C)cn2)=O)ccc2oc(O)nc2n1 97565,C1(C(N2CC(CC)(CC)C2)=O)(CCF)CCN(C(=O)CC2(COC)CC2)C1 97566,C1(CC=C)(NC(=O)CCCNC(C)=O)CC2CCC(C1)N2C(c1cnn(C)n1)=O 97567,CC(C)C(F)(F)CC(=O)N1CCN(C(C2CC(CC(F)(F)F)C2)=O)C(C)C1 97568,N1(C(=O)CC(c2ccccc2)N2CCCC2)CCN2C(=O)NCCC2C1 97569,C(=O)(CCN=C(NCC1CCCCO1)NC1CC1c1cccc(C)c1C)NC 97570,CC1CN2CCCC2CN1C(=O)C(=O)NC1CC=CCC1C(F)(F)F 97571,C(=O)(CCCS(C)(=O)=O)N(CCCCCNC(C1(C)CC=CC1)=O)C 97572,N1(C(C2(c3ccc(C)s3)CC2)=O)CC2CCC(C1)C(NC(=O)C=CCN(C)C)C2 97573,Cc1ccc(C(N2CCC(CNC(=O)Nc3ccccc3C(F)(F)F)C2)=O)cc1 97574,c1(C(C)C)ncncc1C(N1CCN(CC(C)NC(=O)CC2(C#N)CC2)CC1)=O 97575,C1(CN(C(c2cn(CCC(C)C)nn2)=O)C)C2CN(C(=O)C(CO)N(C)C)CC12 97576,C1(OC)CC(CNC(C2CCC=CCC2)=O)N(C(=O)Cc2ccon2)C1 97577,C1(NC(=O)CCN2CCOCC2=O)CN(C(C2CC3(C2)CC32CC2)=O)CC12CC2 97578,c1(C(=O)NC2CN(C(c3c(C)cc(N)cc3)=O)CC2F)cccc2c[nH]nc12 97579,C1(C(=O)NCC#C)CCN(C(c2ccc(-n3cc(Cl)cn3)cn2)=O)CC1C 97580,c1(C(=O)NCC(N2CC(NC(CSC(=N)N)=O)C2)=O)ccc(N=NC(N)=O)cc1 97581,CC(C)C(C(=O)NCCOCCO)C(C)NC(C1CC(F)(CF)C1)=O 97582,C=CCC(C)(C)CCNC(C1CCC(C)CN1C(=O)CCc1ccc(C)o1)=O 97583,N1(C(CNC(C)=O)=O)CCOC2(CCS(=O)(=NC(=O)C3(C)CC(C)=NO3)CC2)C1 97584,C1(C(N(C(C)C(=O)NCCCC(C)CO)C2CC2)=O)CCC(=O)N(C)C1 97585,C(C)(CC(=O)N(CC(C)C(=O)N(C)CC1(OC)CCC1)C)OC 97586,CC(C)C(F)(CNC(c1cccc(O)c1F)=O)C(=O)Nc1cncnc1O 97587,C#Cc1ccc(CC(N2CC(NC(=O)C(C)COCC)C(C=C)C2)=O)cc1 97588,C1(N2CCC(C#N)(NC(=O)Cc3cc(Br)ccc3Br)C2)CCc2ccccc2C1 97589,CC(=O)CCC(=O)N1CC(CC(N2CC(F)(C3CC3)C2)=O)CC1C 97590,c1(SC)cncc(-c2cn(CC(C)NC(=O)Cc3ccccn3)nn2)c1 97591,C1(C(=O)NCC2N(C(C(C)(C)C(N)=O)=O)CCC2)CN2CCCC2CO1 97592,C1(C(=O)NCCn2c(CC)nnc2)C(C)CCN1C(c1cncc(F)c1)=O 97593,N1(C(C(CC)n2cncn2)=O)CCC(OCCNC(=O)C=CC(C)CC)CC1 97594,C(=O)(C1CCCn2nccc21)N1CC(CNC(c2ccc(=O)n(CCF)c2)=O)C1 97595,N1(C(c2cc(C)c(C)nn2)=O)CC(NC(c2cnn(C)c2)=O)CC12CCCOC2 97596,C1(NC(C(N(C)C(c2nnc(O)nc2O)=O)C2CC2)=O)CNC(=O)C12CC2 97597,N1(C(c2c(CC)ncs2)=O)CCC(C(N2CC(OC(C)C)C2)=O)CC1C 97598,C(CC)(CCC(=O)N1CC(O)CC(O)C1)NC(C(C=C)OC)=O 97599,c1(COC)cc(N2CCCC(C3CCCCN3C(C3CC3C(C)O)=O)C2)ncn1 97600,N1(C(COC)=O)C2CCC1CC(C(N1CCCC(CF)C1)=O)C2 97601,Cc1noc2ncc(C(N3CC(NC(c4cc(F)cc(Br)c4)=O)C3)=O)cc12 97602,C12(C(=O)NCCC3CN(C(COCC=C)=O)CC3C)CCC(N(C)C)(CC1)CC2 97603,C1(NC(C2(C(C)(C)O)CC2)=O)CN(C(=O)CSc2cccs2)CC(C)(C)C1 97604,C1(C(=O)NCC(C)CNC(C2CCN(c3ccccc3)C2)=O)CC(C)OC1C 97605,N1(C(c2cc(C)nc(O)n2)=O)CC2(C(=O)N(C(C)C(C)C)C3CC3)CCC1CC2 97606,N1(C(c2cccc(C)c2)=O)CCC2(CC1)OCCC2NC(c1ncc(Cl)s1)=O 97607,N1(C(C2C(C)(C)C(O)C2)=O)Cc2cc(Cl)ccc2CC1CO 97608,C1(CNC(=O)CCn2cc(Cl)cn2)(CO)CCCN(C(C2COCCO2)=O)C1 97609,c1(C(=O)NC2(CF)CCN(C(C(C)(C)c3cc[nH]n3)=O)C2)cc2c(s1)CCC2 97610,O=C1OC2CCC1CN(C(=O)C(CC(F)F)NC(=O)CC1COCCO1)C2 97611,c1(C(N2C(CNC(COCC(C)C)=O)C=CC2)=O)cccc(-n2cnnn2)c1 97612,C1(NC(C(C)n2cncn2)=O)(CO)CCN(C(=O)CC2(CN(C)C)CCC2)C1 97613,C(=O)(CCC(F)(F)Cn1cc(CC(O)C2CC2)nn1)N(C)Cc1cc(Cl)sc1Cl 97614,C12(CNC(Cn3c(C)nc(C)n3)=O)CCCC1N(C(=O)COCC1CC1)CCC2 97615,C1(C(=O)NC(CC(=O)NC)C2CC2)CCCN(C(=O)CNC(C)=O)CC1 97616,C=CC1(C(N2CCC(O)(C(N)=O)C2)=O)CCN(C(c2ccc(Cl)o2)=O)C1 97617,c1(C(=O)NCCCC(C)NC(C2(CCF)CC2)=O)c(Cl)csc1Cl 97618,C(=O)(C1=CC2(CCN(C(c3cc(C)cnn3)=O)C2)C1)N1CCC(CC)CC1 97619,C1(C(=O)NC2CCN(c3nnc(-c4ccon4)s3)C2)CCOC2(CCC2)C1 97620,C(CCNC(C1COCCC1C)=O)(C(=O)N(C)CP(C)(C)=O)OC 97621,CCCC(CCCNC(=O)C=Cc1cocn1)NC(=O)CC1(C)CCC1 97622,c1(C(=O)NC2CC(C(C(=O)N(CC(C)(C)O)C)F)C2)cc(=N)[nH][nH]1 97623,C(=O)(C(C)C(F)(F)C(F)F)NCC(CNC(c1ccc(C(C)C)nc1)=O)(C)O 97624,c1(C(=O)NCC(CN(C)C(C2CC23CC(O)C3)=O)O)ccc(O)c2c1CCCC2 97625,c1(C(C(=O)N(C)C)N(CC)C(C)C)ccc(S(=O)(=O)N(C)C)cc1 97626,N1(C(c2csc(Cl)c2Br)C(=O)NCCCSCC)CC2CCC(CC2)C1 97627,N1(CC2N(C(C(n3cc(CC4(C)CC4(C)C)nn3)C)=O)CC2)CCCCCC1 97628,C1(COC(c2cccc(SC)c2)=O)CC2CCC(C1)N2C 97629,CCC(C)(C)C(C)CC(=O)N1CC(NC(c2cc(C(F)(F)F)n(C)n2)=O)C(F)C1 97630,C(=O)(CCCN(C)N=O)N1C(C(C)NC(C2CC3C(C2)C3(F)F)=O)CCC1 97631,CC(C)(CN=c1ccnc(-c2cccc(Cl)c2)[nH]1)NC(c1cnn(C2CCC2)c1)=O 97632,c1(OC2CCN(CC(C)(C)N)C2=O)ccc(Cl)c(Cl)c1.C(C)(C)(C)OC(=O)NC(=O)C1CC1 97633,O(S(=O)(=O)c1cc(Br)ccc1Br)c1ccc(OCC)c(Br)c1 97634,N1(C(c2n(C)ccc2)=O)CC2CCCCC2(CNC(c2cnco2)=O)C1 97635,N12CCCC1C1(CC1)C2=O.C(c1cc[nH]n1)=CC(=O)NC(C1CCCO1)C 97636,Cc1c(Br)noc1C(N1CCC(O)(CN(C(=O)C(O)C2CC2)C)C1)=O 97637,S(=O)(=O)(c1c[nH]ccc1=NCC1CCS(=O)(=O)N1C)NC(C)Cn1ccnc1 97638,C1(C(=O)NC(C)CF)C2CCC(C2)N1C(c1ncccc1Cl)=O 97639,c1(C(=O)NC2C3(CC(NC(C4CCC(=O)NC4)=O)C3)C2)ccc2oncc2c1 97640,C1(CC)CN(C(c2cc(C)ccc2I)=O)CCN1Cc1cnc(C)cn1 97641,C1(C(C)(C)NC(CN(C(C)=O)C)=O)CCCN1C(=O)Cc1ccccn1 97642,c1(C(N2CCOCC(C(F)(F)F)C2)C(=O)NC)ccc(Cl)c(Cl)c1F 97643,c1(C(=O)NCC(C)CNC(C2CC(F)(CF)C2)=O)c(C#N)ncn1C 97644,C1(NC(c2cc([N+](=O)[O-])c[nH]2)=O)CC2CCC1N(C(=O)Cc1ccno1)C2 97645,c1(C(N(CCC(C)NC(c2ccc(C3(C)CC3)o2)=O)C)=O)ncccc1Br 97646,C(CNC(=O)CC1C=NN(C)C1=O)(CC(=O)NOCCOC(C)C)OC 97647,c1(OCC(=O)NC2CC(NC(C3CS(=O)(=O)C3)=O)C(O)C2)cccc(F)c1 97648,C1(CC(N2CCC(CCNC(=O)CN3CCCNC3=O)C2)=O)CC2C=CC1CC2 97649,N1(C(CCOCC#C)=O)CCCC(CCNC(c2cc(CC)[nH]n2)=O)C1 97650,Cc1nc(C(C)C)sc1C(C)N(c1nccc(-c2ccccc2)n1)C 97651,C=CC1(CC(N2CC(CO)(CF)C2)=O)CN(C(C2CCC(=O)C2)=O)C1 97652,C1(CCC#C)CCCN1C(=O)C(CC1CCOCC1)NC(=O)CCSCCCC 97653,Cn1ncc2c(NCc3nc(Br)n[nH]3)nc(N3CC4C5C=CC(O5)C4C3)nc12 97654,C#CCCCC(=O)NC1CC=CCC1C(=O)NCc1nnn(CC)n1 97655,c1(C(=O)NC2C(C)N(C(=O)Cc3cnn(C)c3)CC2)cc2cccnc2nc1N 97656,c1(CC(=O)NCC(CC=C)NC(c2nccn2CC)=O)ccc(CO)c(F)c1 97657,Cc1cc(C(=O)NC2CC3(C2)CC(C(=O)Nc2cc(I)ccc2C)C3)cc(O)n1 97658,CC1CC=C(C(=O)N2CC(C)(C)CC2CNC(c2sccc2C(C)(C)C)=O)CC1 97659,C1(CNC(c2c(OC)nccn2)=O)CCC2(CN(Cc3csc(C)n3)C2)O1 97660,N(C(=NCCC1(O)CCC1)NCC1C2(CC2)C12CC2)C(C)Cc1ccccc1 97661,C1(CNC(CC2(C)CC2(F)Cl)=O)CC2(CO1)CN(C(=O)COCCCN=[N+]=[N-])C2 97662,C1(CNC(c2cc(C)ns2)=O)CCC2(CCN(C(C3(C)CC(F)C3)=O)CC2)O1 97663,Cc1ccc(C(=O)NC2CN(C(c3ccccc3OC(F)(F)F)=O)CC2O)n1C 97664,N1(C(c2cn(CC)nn2)=O)CC(C(N2CC(F)(C#N)C2)=O)C2(CC2)C1 97665,C1(CNC(C2C(C)C2)=O)CCCCCN1C(=O)C=Cc1cc(Cl)sc1Cl 97666,C1(C(=O)NC(C)C(C)(C)NC(c2cnc3occc3c2)=O)CCc2nnnn2C1 97667,c1(OC(c2ncccc2Br)c2n(CCOC)nnn2)ccc(C)c(C)c1 97668,CC1CC2(CO1)CN(C(c1coc(CNC(C3CC=CCC3)=O)c1)=O)C2 97669,c1(C(=O)NC(CN(C(c2n(CC)ncn2)=O)C)C)cc2c(cc1N)OCO2 97670,c1(C(N2CCCC(NC(CCCC#C)=O)C(F)C2)=O)c(C)nn2c1CCCC2 97671,c1(N2CCCC(C(N(C)C)=O)C2)nc2ccsc2c(=NCc2ccc[nH]2)[nH]1 97672,C=CCCC(C)(C)C(=O)N1CC2CC2(CNC(c2ccnc3[nH]nnc23)=O)C1 97673,c1(CC(=O)Nc2ccc(C(CC)OC)cc2)c(F)cccc1F 97674,c1(OC)cc(CNC(COc2ccc(NC(=O)NC3CC3)cc2)=O)nc(Cl)c1 97675,C1(NC(C(C)O)=O)CCCCC12CCCN(C(=O)CC1(O)CCC1)C2 97676,C(=O)(CC(C)C(C)(C)C)N1CCC(CCNC(c2nc(COC)oc2)=O)C1 97677,c1(OC)cc(C(=O)NCCC2(O)CN(C(c3cc(Cl)ccc3O)=O)C2)cc(Cl)n1 97678,C1(CC)C(NC(=O)NCC(c2ccccc2)(C)F)C1(C)C 97679,CC1CC(C(=O)NCCCN(CCO)C(c2cncc(F)c2)=O)C(=O)O1 97680,N(C1CC(C)C(=O)c2ccccc21)C(C(=O)N(N1CCc2ccccc21)C)=O 97681,C1(NC(c2cnn(C(C)C)c2Cl)=O)CC(F)CN(C(c2ccc(F)cc2)=O)C1 97682,c1(-c2c(C)csc2)cnc2ccc(C(=O)NC(c3cc(F)ccc3OC)C)cn12.C1CC1 97683,N1(C(C=CC(CC)C)=O)CC(CC(=O)NCC(Cl)C(C)(F)F)CCC1C 97684,CC(CN(C)C)CC(=O)NCCc1ccc(F)cn1.C12CC(C1)C(=O)NCC2 97685,N1(C(CCC#CC)=O)CCC(CNC(=O)CSS(C)(=O)=O)C(F)(F)CC1 97686,N1(C(CCCNC(=O)OC(C)(C)C)=O)C2CCC1CC(NC(=O)CC1=CCCC1)C2 97687,C(C(C)(C(=O)N1CC(C(N)=O)(CNC(C2CCN(C)C2)=O)C1)OC)OC 97688,c1(CC)ncncc1C(N1CCN(C(CNC(C2CC2F)=O)C(F)(F)F)CC1)=O 97689,c1(C(C(=O)NCCCC(=O)OC)NC(c2cn(C(C)C)nn2)=O)ccc(Cl)cc1 97690,C(CCCC(=O)NC(C)(C)CN=[N+]=[N-])N(C(=O)C=Cc1ccccc1)C 97691,C(C(=O)Nn1cnn(C)c1=S)N(CCC)C(C1(C(C)(C)O)CCC1)=O 97692,N1(C(C(CC(C)C)(C)C)=O)CCC2(CCC2NC(c2ccsc2Cl)=O)CC1 97693,CC1CN(C(C2(O)CCN(c3nnc(C(N)=O)s3)CC2)=O)CCC1CO 97694,C1(C(N2CC3=C(CN(C(c4c(C)nc(C)[nH]4)=O)C3)C2)=O)CC2(CCCCC2)CO1 97695,C1(CNC(C(CC2CCC2)NC(c2c(COC)noc2)=O)=O)NC(=O)NC1=O 97696,c1(CC)nnc(N2CCC(OCCNC(=O)Cn3cnnn3)C2)o1 97697,N1(C(c2cnco2)=O)CCOC(C(F)(F)F)C1.n1(C)cc(CCOCCO)nn1 97698,C(C)(CO)(C(=O)NC1CCN(CCNC(=O)CC2CCCCC2C)CC1)OC 97699,C1(O)(C(N2CC(NC(c3cnc(SC)s3)=O)C2)=O)CCCCCC1 97700,CC1(C#N)CC2CCC1N2C(N1CCC(N)C1)=O 97701,C1(CNC(CN(C(=O)CCc2cnn(C)c2)CC(C)C)=O)CCNC1=O 97702,CCOC(C)(C(=O)OCc1ccccc1C(=O)NC(=O)OC(C)(C)C)C1CC1 97703,N1(C(C(C)CC2CC2)=O)CCOC2(CCN(C(=O)COCC3CC3)C2)C1 97704,C=CCCC(C)(C)C(=O)NC1CCCC1NC(=O)C(CC)NC(N)=O 97705,c1(CC)cc(C(=O)NCC2CN(C(C3COCCN3C)=O)C2)ncn1 97706,N1(C(CC)C(=O)O)CCC(C(N2CC(SCC(C)C)C2)=O)CC1 97707,C1(N(C(=O)CCC2CCC2)C)CCCN(C(C2(CNC3CC3)CCC2)=O)CC1 97708,C(=O)(CCCS(N)(=O)=O)NC1C(C)N(C(c2cnc3c(c2)CCC3)=O)CC1 97709,C(=O)(C1CCc2c[nH]nc21)N1CC(COC)(NC(c2cnn(C(C)C)c2)=O)C1 97710,CC(c1ccccc1F)=CC(=O)NCCOC1CCN(C(=O)C(C)SC(C)C)C1 97711,N1(C(C)=O)CC2(NCC(c3nccc(Oc4ccccc4)n3)C)CC1CO2 97712,Cc1cc(C(N2C(C(=O)NCC3(CO)CC4CC4C3)CCC23CC3)=O)nc(C)c1 97713,CC1=C(C(=O)NCC2CCCN2C(=O)Cc2nc(=N)[nH][nH]2)CC1 97714,c1(NCC2C3CN(C(C(C)NC(=O)C4CC4)=O)CC32)c(C#N)c(=O)n(C)c(=O)n1C 97715,C1(CCNC(C2(OC)CCOC2)=O)CCCN(C(c2noc(C3CC3)c2C)=O)C1 97716,C1(NC(C2C(CNC(c3ccc(C#C)o3)=O)CCCC2)=O)CCc2nncn2C1 97717,Cc1csc2cc(C(=O)NC3CC3NC(c3cc(F)cc(F)c3)=O)[nH]c12 97718,Cc1cc(Cl)c(C(=O)NC2CCN(c3ccc(Br)cc3)C2=O)cc1C 97719,c1(CC(C)C(=O)NCC2(NC(=O)Cc3ccc(F)nc3)CCC2)ccc(N)cc1 97720,N(C1CCCc2n[nH]cc21)C(=O)COCCCN=[N+]=[N-].CCC1CCC(=O)N1 97721,c1(NC(C2C(N(C)C)COC2)=O)ccc(CNC(=O)CN2CC=CC2)c(F)c1 97722,N1(C(C(C)=C(C)C)=O)CCN(C)CC1CNC(=O)C(O)C(F)(F)F 97723,c1(C2(C(=O)NCC3CCN(S(C)(=O)=O)C3)CCCC2)cc(F)ccc1F 97724,C12(C(N3CC(C(=O)N(C)Cc4cc[nH]n4)(CC)C3)=O)CCCC1C2(F)F 97725,c1(CC(N2CCCC(C(CO)NC(=O)CN3CCCCC3)C2)=O)cc(F)cc(F)c1 97726,N1(C(CCC(N)=O)=O)CCCCCC1CNC(C1CCCC1(F)F)=O 97727,C(c1ccc(Cl)cc1)(C(F)(F)F)=CC(N1CCN(C(C(C)O)=O)C2(C1)CCC2)=O 97728,C1(NC(C=CCN(C)CC)=O)CCCCCN(C(c2cnccc2C)=O)C1 97729,CCC(CNC(c1cccnc1CNC(C1(C)CCCN(C)C1)=O)=O)(CC)CO 97730,N1(CC(=O)N(CC(C)(C)C)C(C)C)CCN(n2c(CC(C)(C)C)ncn2)CC1.ON 97731,C1(CC#C)(C(=O)NCc2ocnc2C(=O)NC2CCCCC2O)CCCCC1 97732,c1(C(=O)ON2C(Cn3cc(C)nn3)CCC2)cnc2c(c1)c(C)nn2C 97733,C1(C(N2CCC(CCNC(C3CN(C(C)=O)C3)=O)C2)=O)Cc2cc(Cl)ccc2O1 97734,c1(CCC)nc(=NC2CCCN(C(=O)CN3CC4CCCC(C3)N4C)C2)s[nH]1 97735,Cc1csc2c(C(=O)NC3CCC(CNC(c4snnc4C4CC4)=O)C3)ncnc12 97736,CC1CN(C(=O)CC2COC(=O)C2)CC(C)CN1C(=O)CN(c1cnccn1)C 97737,c1(C(N(CCCCNC(Cn2c(C)ncc2)=O)C)=O)cc(F)cc([N+](=O)[O-])c1 97738,Cc1ccc(N)c(C(N2CCC(NC(=O)Cc3c(F)cncc3Cl)CC2)=O)c1 97739,Cc1ccc(CC(=O)NC2CCC(C(=O)NC(c3ccccc3)C)OC2)cc1F 97740,C1(NC(C2C(C=C)(C(F)(F)F)C2)=O)CCCN(CC=Cc2cncc(C)c2)C1C 97741,Cc1nccnc1CNC(=O)CCN(C(=O)C(C)CC#N)C 97742,c1(C(N2CC3(CN(C(c4ccc(N(C)C)cc4)=O)C3)C2)=O)cccc2[nH]ncc12 97743,C(c1ccccc1)=C(C(=O)NCC(CC)NC(=O)Cc1ccsc1)C 97744,CC(CN(C)C)CC(=O)NC1(C(N2C3CCC2C3)=O)CCOCC1 97745,CCC(C(=O)NCC(C1CCC1)NC(=O)CCCNC(N)=O)N(C)C 97746,C1(C(=O)NC2C(CC)N(C(=O)CN3CCC(F)CC3)CC2)CC2CC(=O)C1C2 97747,CCC(CC)(C(=O)N(CC(C)NC(=O)C(C)C(C)C)C)c1ccccc1 97748,C1(C(N2C3CCC(N(C)C)C(C3)C2)=O)CCCC1C1CCCC1 97749,C(C(=O)N1CCCC(CNC(C2(C(F)(F)F)CC2)=O)C1)(C(C)O)NC(C)=O 97750,C1(CC(N2C(CNC(CCC(=O)NCC)=O)CC(O)C2)=O)CC2(CCC2)CCO1 97751,C1(NC(c2c(C)ncnc2)=O)C2CCCN(C(c3nccn3C)=O)C2C1(C)C 97752,Cc1cc(NC(c2conc2C(C)NC(C2COCC2(C)C)=O)=O)cc(F)c1 97753,c1(CC)ccnc(C(N2CC(N(C)C(c3cc(Cl)c(Cl)s3)=O)C2)=O)c1 97754,C12(NC(c3c(C)ccs3)=O)CCN(C(c3cccc(C(F)F)n3)=O)CC1C2 97755,C1(NC(=O)CCF)CC(F)(F)CC1NC(=O)CCC1CCCO1 97756,N12Cc3n[nH]cc3C1C2=O.CC12CCOC(C(N3CCC(CCO)C3)=O)(C1)C2 97757,C=CCC(C(=O)NC1CC2(CCN(C(=O)CN3CSCCSC3)C2)C1)C(C)(C)C 97758,N1(C(c2c(Cl)cc(C)s2)=O)CCC(NC(C2SC3C=CC2CC3)=O)C(CO)CC1 97759,C1(C(F)F)(OC)CC(C(=O)NCC2CN(C(=O)CC3(C(F)F)CC3)C2)C1 97760,c1(C(=O)NC2(C)CN(C(C3CCCCC3C3CC3)=O)C2)cccc2[nH]ccc12 97761,N1(C(c2ccnc(C)n2)=O)C2CCC1CC(O)(CNC(c1cc(Cl)c[nH]1)=O)C2 97762,c1(C(C)NC(=O)COC(C)(C)CNC(=O)CC2(O)CCC2)cccn1C 97763,C1(NC(=O)C(=O)Nc2ccccc2)CCCC(NC2CCCNCC2)C1 97764,N1(C(c2c(CC)ccc(F)c2)=O)CC2CCC(C1)N2C(c1cc(Cl)c(Cl)s1)=O 97765,Cc1nn(CC(=O)NC2CN(C(c3nc(O)sc3C)=O)CC2CO)c(=O)o1 97766,c1(N2CCC(NC(=O)OC(C)(C)C)CC2)nc(C2=CCCCC2)cs1 97767,C1(C(=O)NCCn2c(C)ncc2)CC(C)CN(C(c2cccc(Br)c2F)=O)C1 97768,c1(OCCCC(=O)NCC(CNC(CC2CCC(C)O2)=O)(C)C)ccc(O)cc1 97769,C(=O)(C(C)CS(C)(=O)=O)NCCC(C)NC(=O)C(c1ccccc1F)C 97770,n1(C(C)C)cnc2cc(NCC3CCC4(CCOCC4)O3)ccc12 97771,N1(C(c2cn(C)c(O)n2)=O)CCC2CCCC12C(N1CCOCC1)=O 97772,c1(C(=O)NC2CCC(CNC(C3N(CC)CC3)=O)C2)c(C)ccc(Br)c1F 97773,c1(CC(=O)NC(CC=C)CNC(=O)C(c2cncn2C)O)ccc(Cl)c(C)c1 97774,Cc1cccc(C(CNC(c2nnc(S)n2C)=O)NC(=O)CCSC(F)(F)F)c1 97775,c1(C(N2CCN(C(C#CC3(C)CC3)=O)C3C2C3)=O)cccc2c1OC(F)(F)O2 97776,C1(C(N2CC(O)(C(C)NC(C3CCC(CF)C3)=O)C2)=O)(CCF)CCOCC1 97777,C=CC1CCCN(NC(=O)c2cc(COC)cnc2OC)C1 97778,N1(C(C2CC(O)(CC#C)C2)=O)CCOCC1CNC(c1c[nH]nc1F)=O 97779,CN1CC=CCC1CC(=O)NC1CCCCC1NC(c1ccsc1C(F)(F)F)=O 97780,c1(C(N2CCC(C)CC2C(=O)NOC(C)(C)CO)=O)c[nH]c2ccccc12 97781,c1(C(=O)NC2CC(NCc3cc(C)[nH]c3C)C2)c(F)c(F)c(O)c(F)c1F 97782,c1(NC(=O)CC2CCN(Cc3ccc(C(=O)O)cc3)C2)ncc(F)cc1O 97783,NC1COC2(C(=O)NCC3CN(CCCO)CCO3)CC1C2 97784,C1(C(N2C(C)CN(C(c3cnc(O)s3)=O)CC2)=O)CCn2ncnc2C1 97785,C=C(C)C(CC(=O)N1CCN(C(=O)CC(C)(F)F)CC1CCOC)OCC 97786,c1(C(N2CC(NC(CC(CCSC)O)=O)C2)=O)nc[nH]c2nccc1-2 97787,C12(CNC(c3nccc(C)c3N)=O)CCCCC1CN(C(c1ccccc1)=O)C2 97788,C(=O)(CC(C)CC(F)(F)F)N1CCC2(CC(NC(COCCCOC)=O)C2)C1 97789,C(=O)(CS(=O)(=O)CCC(F)(F)F)NCCN(C(c1onc(C)c1C)=O)C1CC1 97790,N1(C(C(C(C=C)O)(C)C)=O)CC2CCC(C1)N2C(=O)Cc1ccccc1Br 97791,C(=O)(CC(C)(C)CNC(=O)C=CC1CCCCC1)N(CC)Cc1ccn(C)n1 97792,CC(CN(C)C)C(=O)N(C)CC1CCCN1C(c1ccc(C(F)(F)F)o1)=O 97793,N1(C(c2cc(C)oc2)=O)CC2CCCC2(Nc2ncncc2I)C1 97794,c1(C(N(CCCNC(C2C(CCC)CCC2)=O)CCO)=O)c(C)n[nH]c1C 97795,CC1(C)C(C(=O)NCCN(C(=O)CC=CC(C)(C)C)CCO)CC1(F)F 97796,C1(NC(c2cncc(C)n2)=O)CCSC12CN(C(c1cc(C(F)F)ccn1)=O)C2 97797,C12(CC)CC(C(=O)NCCC3CCC(NC(=O)C=CC4CCCCC4)C3)(CO1)C2 97798,C1(C(=O)NC(CCC)(C)C)CN(C(=O)C(C)(C)C(C)O)CC1(F)F 97799,C(C(C)(C)CN=c1cccc(S(=O)(=O)NCC2CCC(C)(C)CO2)[nH]1)OC 97800,N1(C(c2c(CC)cns2)=O)CCCC2(CCCN2C(c2cc([N+](=O)[O-])ccn2)=O)C1 97801,C(=O)(C(C)(C)C)NCCC(=O)N(C)CC1(NC(CSC(C)C)=O)CC1 97802,c1(C(=O)OCC)cccc2cc(CN3CCOC(c4cccc(CC)c4)C3)oc12 97803,c1(C(N2C(CN(C)C(c3cc(Cl)no3)=O)CCC2)=O)cnc(Cl)cc1N 97804,c1(C(=O)NC2CCN(C(CCN(CCCCOC)C)=O)CC2)cnc(F)cc1C 97805,C(C(C)C(C)CC)NC(C1N(C(c2c(CC)cns2)=O)CCC1)=O 97806,Cc1ccc(CNC(C2OCCC2NC(C2CCCOC2C)=O)=O)nc1 97807,CN1CCN(C(C2CCCN2C(C2CC(C)(O)C2)=O)=O)CC1CO 97808,c1(NCC2CCC(NC(Cc3ccc(C(N)=O)cc3)=O)C2)ccnc(C#N)n1 97809,C1(O)(C(N2CCC(N(C(=O)COC(F)(F)F)CCC)C2)=O)CCC(CCC)CC1 97810,N1(C(C(=O)N(C)C)=O)CCOC2CCN(C(C3SCCCS3)=O)CC12 97811,Cc1ccc(C(N2CC(CNC(=O)C(C)NC(C)(C)C)C2)=O)c2cccnc12 97812,c1(C(N2CCN(C(C3C(C)(C)C(=O)C3)=O)CC2CCO)=O)cnn2cccnc12 97813,N1(C(C(C)n2cncn2)=O)CC2(C=C(C(=O)NC3CC(CCO)C3)CO2)C1 97814,C1(CNC(c2ccnc(S)c2)=O)CC12CCN(C(=O)CS(=O)(=O)C1CC1)CC2 97815,C(=O)(C(C)(CNC(C1CC=CCC1C)=O)CC)NC(CC#CC)C 97816,Cc1cc(CN(C)C)ccc1N=c1[nH]c(N(C)C)nc2c1CCCCCC2 97817,C1(CCNC(CC=C=C)=O)CCCN(C(=O)CC2(C#N)CCOCC2)CC1 97818,C(=O)(CC(C)(C)C(C)(F)F)NC1C(NC(CCC(C)C#N)=O)CCCC1 97819,C1(CCNC(CC2(OC)CN(C(C3(C4CC4)CCC3)=O)C2)=O)CCCC1(C)C 97820,C1(C(N(CCNC(C(n2ccc(C)n2)C)=O)C)=O)C2CCC(F)(F)C12 97821,C1(CC(=O)NCCN(C(C(C2CCCCC2)OC)=O)C(C)C)COCCN1C 97822,C#Cc1ccc(OCC(=O)NCC(C)NC(C2CCCN2S(C)(=O)=O)=O)cc1 97823,C1(C(N(CCOCCNC(COC)=O)C)=O)(C(=O)OC(C)(C)C)CCN(C)CC1 97824,C(C1CCCCC1)=CC(=O)NC1CC(C)(CNC(c2coc(C(F)F)n2)=O)C1 97825,CC(C)(F)C(=O)N1CCC(C(F)C(=O)NCC(C)(C)O)C1 97826,CC(CN=c1[nH]c(=NCC2CC(F)C2)c2[nH]ccc2[nH]1)S(N)(=O)=O 97827,c1(C(=O)NC(C2CN(C(C=CCCC(C)C)=O)C2)C)cc2scnc2[nH]1 97828,C1(C(=O)NCc2cc(C)no2)CC2CC1CC2O.C1(C(NOCC)=O)CCC(C)C1 97829,c1(CNC(=O)NC(C(=O)OCC)C(C)CC)ccc2nc(C)ccc2c1 97830,c1(C(=O)NCCN(C(C(C=C)(C)C)=O)CC)cc(=O)n2nccc2[nH]1 97831,C1(C2(NC(c3c(C)cc(C)s3)c3nnnn3C3CC3)CCC2)CCC12CCCO2 97832,CCCC(C(=O)NCCCCCN(C(=O)C(C)OC(C)(C)C)C)OC 97833,C1(NC(CN(C(C)C)C)=O)CCCC(C(=O)NC(C)(C)CCN(C)C)C1 97834,C(C(CCO)N=c1[nH]c2c(c(=NCCCn3ccnc3)[nH]1)CCCCC2)N(C)C 97835,c12ccc(Cl)nc1on(C1CCN(C(=O)CN(C)CCO)C1)c2=O.CC=CC 97836,C=Cc1cnn(C)c1C(N1CC(NC(=O)CC2CCCCC2(F)F)C2(CC2)C1)=O 97837,C1(CNC(CN2CC(CC)C2)=O)CN(C(c2cc[nH]c2C)=O)CC12CCC2 97838,c1(C(=O)NC(C)CCNC(=O)C(c2ccccc2)O)cccc2c1OCO2 97839,Cn1cc(Br)cc1C(=O)NCC1(CNC(=O)CSCCC#N)CC12CCC2 97840,c1(C(=O)NC(CC)(C)CNC(=O)C2=C(C)OCC2)cc2c(Cl)c(F)ccc2[nH]1 97841,c1(C(=O)NCC2CC2NC(C2CC(C(F)(F)F)C2)=O)ccc(F)c2c1OCC2 97842,C1(C(=O)NC(CC)CN(C)C(c2cc(CO)[nH]n2)=O)OCC2CCCC12 97843,C(=O)(CS(=O)(=O)C1CCCC1)NC1C(NC(C(C(CC)CC)OC)=O)C1 97844,C1(NC(CC(C)(C)SC)=O)CC(O)CN(C(c2cccc(O)c2Cl)=O)C1 97845,C1(NC(c2c(C)nc(O)[nH]2)=O)CC2CCC1N(C(c1csc(Br)n1)=O)C2 97846,c1(C(=O)NC2CCOC2C(N2CC(SC(F)F)C2)=O)cncc(O)c1 97847,Cc1nc2cc(C(=O)NC3CN(C(C4C5CCCCC45)=O)CCO3)cnc2[nH]1 97848,c1(C(=O)NCCN(C(=O)C(F)(F)C2CC2)CCOC)c[nH]cc(C)c1=O 97849,C=C=CC(C)C(=O)NC1(C(N2CC(N3CCCCC3)C2)=O)CC1(C)C 97850,c1(C(N2C(CNC(c3c(C)cn(C)c3)=O)C(C)CC2)=O)cnc(Cl)cc1N 97851,c1(C(=O)NCCC2(CNC(CC(C)c3ccco3)=O)CC2)nccc2ccsc12 97852,Cc1cc(=O)c(NC(=O)C(CNC(=O)CC2OCCOC2C)CC2CC2)c(C)[nH]1 97853,C1(C(=O)OCC2CC2)(C(=O)NCCNC(c2nc(CC)oc2)=O)CCOC1 97854,c1(CC)noc2ncc(C(=O)NCC(F)CNC(C3CC3CC)=O)cc12 97855,c1(CN(C(=O)C(CC2CC2)CC2CC2)C)ccc(O)cc1.C(=O)(C(F)(F)CO)N 97856,c1(NC(C(Cc2cc[nH]n2)NC(C(C)=C2CC2)=O)=O)ccc2c[nH]nc2c1 97857,N1(C(CN2CCN(C(c3c(C)nc(C)s3)=O)CC2)=O)CC2C(C1)C2(F)F 97858,c1(C(=O)NC2CCC(NC(=O)C=C3CCOCC3)C2)cc2sc(Cl)cc2[nH]1 97859,Cc1cc(O)ccc1C(N1CCC(NC(=O)C(=O)Nc2c(F)cccc2F)C1)=O 97860,C(=O)(CCCCCCNC(c1cnccc1C)c1nnnn1CCCF)OCC 97861,N1(C(C=CC)=O)CC(NC(c2ncsc2CC2CCCCC2)=O)C(CC(C)(C)C)C1 97862,N1(C(C(C)OC)=O)CCC(O)(CCNC(C2(CSC)CCC2)=O)C1 97863,C1(OC)CC(C(N2CCCCC2CNC(=O)CC2CCCSC2)=O)CC1OC 97864,c1(OC(=O)NCC(N2CCC(CN(c3ccccc3)C)C2)=O)ccccc1 97865,c1(CCC(=O)NC2C(NC(C3CC(N(C)C)C3)=O)C2)ccc(Cl)cc1.C(C)(=O)O 97866,N1(CCC)CCCC1CCCc1ccccc1.c12nccn1NC(=O)N(C)C2 97867,C(=O)(C1=NOC(CNC(=O)CSC(F)(F)F)C1)NCC1(C)N=C(C)SC1 97868,N1(C(C2N(C=O)CCC2)=O)CCN(C(=O)C=CSc2ccccc2)CC(CO)C1 97869,C1(C(=O)NCc2cc(C(=O)NC(COC)CO)n[nH]2)CC(=O)C12CCC2 97870,c1(N(C(C(C2CCN(C(c3c(C)csc3C)=O)CC2)C)=O)C)cccc(F)c1C 97871,O(NC(=O)CC(CNC(=O)C(C)C1CC1)OC)C(C(=C)Cl)=O 97872,c1(C(C)C(=O)NCCNC(c2cnn(-c3ccccc3F)c2)=O)cncc(F)c1 97873,O=C(CS(=O)(=O)Nc1ccccc1)NC1CCCC1CNC(=O)Cn1nccn1 97874,C(=O)(CCC(C)(C)F)N1CCC(NC(c2c(OC(F)F)cc(C)s2)=O)C1 97875,N1(C(c2n(C(C)C)ncn2)=O)CC(NC(c2ccccn2)=O)C(CC(C)(C)C)C1 97876,Cc1cc(=NCc2ccoc2)[nH]cc1S(=O)(=O)NCC1CCCC(C2CC2)O1 97877,C=CCC(CNC(C1CC(C)(O)C1)=O)NC(c1cc(OC)no1)=O 97878,N1(CCOC)CC(C(=O)NCC2CCC2NC(c2cc(C)ns2)=O)CC1=O 97879,c1(C(=O)NC2(C)CC(NC(C(c3cc(C)sc3)(C)C)=O)C2)cc(C)c(N)cc1F 97880,N1(C(C=CC(C)C)=O)CCC2(CCC2)C(CNC(C2(C)COC(C)(C)CO2)=O)C1 97881,CC1(C)CCc2nc(CNC(=O)C(=O)NCC3(CCO)CCCCC3)sc2C1 97882,n1(CC(CN2CCC(C#CC)CC2)O)nc2ccccn2c1=O.C12CN(C1)C2=O 97883,C(=O)(C(C(C)CC)N(C)Cc1ccccc1Br)NCC(=C)C 97884,N1(C(C2CC3OC2C2CC32)=O)CCC2CN(C(c3ccnc(C(F)F)c3)=O)C2C1 97885,C(CC(C)(C)C(=O)NC1CCC1NC(=O)Cc1ccc(C)cc1)OC 97886,C1(C#N)(C(=O)NC2CCCN(C(c3nc(N(C)C)nc(=N)[nH]3)=O)C2)CC12CCC2 97887,N1(C(c2c(OC)nccc2)=O)CCN(C(C2CCN2C(C)(C)C)=O)CC2(CC2)C1 97888,C1(NC(CC2N(CC)CCOC2)=O)CCN(C(=O)C(C)OC)C(C)C1 97889,C1(C(N(c2cccc(C)c2)C)=O)C2CCN(C(c3ccc[n+]([O-])c3)=O)CC12 97890,c1(C(N(CC(=O)N(CC(CC)(O)CC)C)C2CCC2)=O)ccc2[nH]ccc2n1 97891,c1(C(=O)NCC(CNC(=O)CN2CCCC(CO)C2)F)c(O)cccc1F 97892,c1(C(C)NC(C(CC)O)=O)ccc(CNC(=O)Cc2csc(=N)[nH]2)cc1 97893,C1(CNC(c2c(C(C)C)nns2)=O)C2CN(C(C3CCCN3S(C)(=O)=O)=O)CC12 97894,C(=O)(C(CC)C(C)(C)CC)NCC(C)(C1CCC1)NC(CC=C)=O 97895,CCCC1C(O)C(=O)N1.C1(NC(=O)OC(C)(C)C)OC(=O)NC1(C)C 97896,C1(NC(C(CC)C)=O)CCCCCC1C(=O)NCc1ccc(Cl)cc1 97897,N1(C(C=CC)=O)CCC2CN(C(=O)CCCN(c3ccccc3Cl)C)CCC2C1 97898,C1(C(N(C)CC2CC(=C)C2)=O)CCCN1C(c1coc(C)c1)=O 97899,C(=O)(C1CCCc2nc[nH]c21)N1CCC(NC(C(CC)(F)F)=O)CC1 97900,C1(C)(C(=O)NCC2=CCN(C(C3CCCC(C)(C)O3)=O)CC2)CCCCNC1=O 97901,N1(C(Cc2c(C)ocn2)=O)CC(NC(C2CC3CC3C2)=O)CC(C)C1 97902,C(=O)(C#CC(C)(C)CNC(C1COCCN1C)=O)NCC1(C)ON=C(C)C1 97903,c1(OC)ccc(F)nc1NC(C1CCCC1NC(c1c(O)cccc1F)=O)=O 97904,C1(CNC(C=CC=CC)=O)CCN(C(c2ncc(C)cc2F)=O)C1(C)C 97905,N1(C(COCCCC)=O)CCN(C(=O)CC2COC(C)(C)CO2)C(C2CCC2)C1 97906,C1(C2CCC2)(C(N(CCCNC(C(C(C)C)CO)=O)C)=O)CC1(F)F 97907,c1(CC(N2CC(C)N(C(=O)Cn3cccn3)CC2C)=O)cc2cc(Cl)ccc2[nH]1 97908,c1(C(=O)NC2CCN(C(C(c3ccc(F)cc3)CC)=O)C2C)ccc([N+](=O)[O-])o1 97909,c1(C(N(C(CC)CNC(=O)C(C)n2cnnn2)C)=O)ocnc1C1CC1 97910,c1(CN2CCC(CC(=O)N(CC=C)CC3CCOC3)C2)c(F)cccc1F 97911,C1(CC(=O)NC2C3CN(C(C(CC=C)C(C)C)=O)C2C3)CCC2(CC1)CCC2O 97912,c1(C(N2C(CNC(c3nncc(C)c3)=O)CC(C)(C)C2)=O)cncc2nc[nH]c12 97913,CCC1=C(C(=O)NC2C=CC(C(=O)NC(C)CCn3cncn3)C2)CCCO1 97914,c1(C(N(CCCNC(=O)CCCc2cnn[nH]2)C)=O)ccc2oc(O)nc2n1 97915,N1(C(c2ccc(CC)o2)=O)CCCN(C(c2cscc2C(F)(F)F)=O)CC1CO 97916,C1(CC)CN(C(c2cn(CCC(C)C)nn2)=O)CCN1C(=O)C(=O)NCC(F)F 97917,c1(NC(=O)NC2C(OC)COCC2)c(C#N)ccc2c1CCCC2 97918,Cc1nc(C(=O)NCc2csc(C(=O)N(C)Cc3cnn[nH]3)c2)cn1C 97919,CC1(C(=O)Nc2ncc(F)cn2)C=CCN1C(c1sccc1Cl)=O 97920,C(=O)(C1CCCc2cccnc21)NC1CCC(NC(c2cnc(SC)n2C)=O)C1 97921,C1(C(=O)NCCN(C(C)C)C(c2c[nH]c(-c3ccncc3)n2)=O)CCCC(F)C1 97922,CCCN=C(NCCN1CCCCC1)NC1CCCC1CNS(C)(=O)=O 97923,c1(OC)cc(CCC(=O)NC2CCCN(C(C3CCOC3C)=O)C2)ccc1Cl 97924,Cc1ccnc(CNC(=O)CC2C3CN(C(c4cnc(O)o4)=O)CC23)c1 97925,c1(C(N(C2CCCN(CCC(=C)C)C2)C)=O)cnc(O)c(Cl)c1 97926,c1(CCCC(=O)NCC(C(C)C)NC(C(CC)OC)=O)cc2ccccc2o1 97927,CCC(CC)C(C(=O)NC1(CCO)CCN(Cc2ccc(F)cc2)CC1)OC 97928,C=CC(C)CC(=O)NCC(CNC(=O)CCC1CC(NC(=O)OC(C)(C)C)C1)CO 97929,c1(Sc2ccc(OCC(=O)NC3C4CN(OC)CC34)cc2)cccc(C)c1C#N 97930,C1(NC(CCC2(C#N)CCC2)=O)CCN(C(c2cnc(O)o2)=O)CC1CO 97931,c1(NCCN(C)C(c2cccc(F)c2F)=O)nc(Cl)nc2nc(Cl)n(C)c12 97932,N1(Cc2c(Br)ccc(C)n2)CC2CC(NC(=O)C3=CCCCO3)CC2C1 97933,C1(C(N(CC(=O)OC)C)=O)C(C2CC2)CCN1C(C12CC(CO)(C1)C2)=O 97934,C1(NC(C2(COC)CC2(F)F)=O)CC(CO)N(C(=O)CC(C)(C)O)C1 97935,C1(NC(c2c(C(C)(C)OC)cccc2)=O)CC(O)CN(C(=O)C(C)=CC2CC2)C1 97936,Cc1c(Br)ccc(F)c1C(=O)NC12CCC1CN(C(=O)C#CC1CC1)C2 97937,Cc1[nH]c(C#N)cc1C(=O)NCc1cccc(C(N2CC(C)(C)C2)=O)n1 97938,C1(F)(CNC(COCCC=C)=O)CCN(C(c2nnn(-c3ccccc3)n2)=O)C1 97939,C1(NC(CC2OCCN(C(C(C)OCC(C)C)=O)C2)=O)CC2CC1CC21CC1 97940,C12(NC(=O)COC3CCC3)CCCN(C(=O)CCCC(F)(F)F)CC1C2 97941,Cc1cc(=NC2CC3CN(C(=O)CC4(C)CCCC4)CC23)[nH]c(Cl)n1 97942,C(=O)(C(C)(C)CC(C)(C)C)N1CC(C2(NC(CC(C)C)=O)CC2)C1 97943,c1(N2CCc3c(cnc(C)n3)C2)nc(=NCC(C)CCO)[nH]c2ccccc12 97944,C1(NC(=O)C(C)n2cccc2)(CC)CCCC1.N(CCOC)(C(=O)C1CC1)CC 97945,c1(CC(=O)NC2C(CNC(C3(C#C)CCCC3)=O)C2)cc(Cl)cc2c1OCC2 97946,C1(CC(=O)OCC)(C(=O)NCC2CCC2NC(c2cc(Br)c[nH]2)=O)CCCC1 97947,C(=O)(C(C)(C)CS(N)(=O)=O)NC1(C)CCCC1NC(c1ccc(F)cc1C1CC1)=O 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97966,C1(c2nnnn2CC2CCOC2)(NC(CC)COC)CC2CC1CC21CC1 97967,n1(CC(N2CC(CNC(C(C(C)C)OCC)=O)C(C)C2)=O)cnc2ccccc12 97968,c1(N2CC(C)(CCC#N)OCC2)ccncc1S(=O)(=O)NCC(C)(C)c1cccs1 97969,c1(C(NOCC(=O)NC(CC#C)C)=O)ccc(O)nn1 97970,N1(C(C)=O)CC2COCC(C1)N2C(c1ccc(C(=O)NC)cc1)=O 97971,CC(O)(Cn1ccccc1=O)C(=O)NCC1(CNC(C2CC=CCO2)=O)CCC1 97972,Cc1ccc2c(=NCc3ccccc3)[nH]c(=NC3CCCC3C3CCC3)[nH]c2c1 97973,c1(NCC(COC)(C)CO)[nH]c(=NCCc2ncccc2C)nc2scnc12 97974,N1(C(C(=O)NC(C)C)=O)CCC(C)(CCNC(C2C=CCCC2)=O)CC1 97975,c1(C(N2CC3C(C(=O)NC(COCC)(C)C)(C3)C2)=O)ccc2c(c1)C(=O)CC2 97976,N1(C(CCC(=O)OC)=O)CCN(C(=O)C(O)CC(N)=O)C(C)C1 97977,N1(C(C2(CC(F)(F)F)CC2)=O)CC2(C1)CN(C(=O)C(CC)OCC)CC2CO 97978,N1(C(C2CN(C)C2)=O)CCC2C1CCN2C(C1C2C=CSC12)=O 97979,C1(NC(CSCCOC)=O)(SCC(=O)NC(C2CCCCO2)C)CCCCC1 97980,CC(C)C(C)C(=O)NCC1CCN1C1(c2ccc(OC(F)F)cc2)CC1 97981,C(C(=O)NC(CNC(=O)CC1CCCC1)CO)(SC)SC 97982,c1(C(=O)NC2CN(C(=O)C(F)CC3CCCC3)CC2C(F)F)ncc(Cl)cc1O 97983,N1(C(C2(C#C)CN(C(=O)C=CCN3CCCC3)C2)=O)CCN2CCCC2C1 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98036,CCC(CC)CC(=O)N1CC=CC(C(=O)NCC=CC(=O)NC(C)(C)C)C1 98037,N1(C(c2n(C)nc(C3CC3)c2)=O)CCC(NC(C2CCC(O)C2)=O)C12CCC2 98038,N1(C(CCCC(=C)C)=O)CCCC(C2CCN(C(C3CN4CCN3CC4)=O)C2)C1 98039,c1(C(=O)NCCCn2cc(C3CCCC3O)nn2)cnn2cccc(Br)c12 98040,c1(N(C(=O)OCC)C)ccc(C(=O)NC2(c3ccccc3Cl)CCOCC2)cc1 98041,c1(C(=O)NCCCCC(C)NC(C(CC)O)=O)c(C)sc(C)c1Br 98042,CC1CCCN(C(=O)COc2ccccc2Cl)C1CNC(c1ccc(Cl)cc1)=O 98043,C(C(C)CC(F)(F)F)NC(C(c1ccnn1C)NC(CSCCOC)=O)=O 98044,C1(CNC(c2sc3cc(C)sc3c2)=O)Cc2ccccc2CN1Cc1nnsc1Cl 98045,Cc1cc(Br)cc(CN2CCC(O)(C(=O)NC3CCC(O)C3)CC2)n1 98046,c1(C(=O)NCCCN(C(C2CC(O)C2)=O)CC)cncc(-c2ccoc2)c1 98047,c1(CC=C)cccnc1-c1csc(NC(C2CC(CNS(C)(=O)=O)CC2CC)=O)n1 98048,O(P(C)(=O)CNC(=O)C=C(C)CNC1C(NC=O)C(O)C1)CC.C(C)(=O)O 98049,C1(NC(c2ncn(COC)c2)=O)CCOCC1NC(=O)C=CC(=O)N(C)C 98050,C1(C(C)NC(=O)C(F)(F)c2cscn2)CCN(C(c2ccnnc2Cl)=O)CC1 98051,c1(C(C)CC(=O)NCC2CCN(C(c3c[nH]c(Br)c3)=O)C2)ccc(F)cc1 98052,C#Cc1cccc(CC(=O)NCC2(NC(c3ncccn3)=O)CCCCC2C)c1 98053,C1(C(N(C2CCN(C(C(CC)C)=O)C2)C)=O)CCn2c(cnc2C)C1 98054,O=C(CCCNC(c1cc(C2CC2)no1)=O)NCC1C=CCC1 98055,c1(CCN=C(NC2C(C)CC2)NC2CC2)ccc2c(c1)OCCO2.OC(F)(F)F 98056,N1(OC(C(C)(C)C)=O)CCN(C(N2C(C)CC(C)C2)=O)CC1C 98057,c1(C(=O)NC2CC(F)(CNC(c3cc(C)on3)=O)C2)cc(N)cnc1C 98058,O=C(N=c1cc(Br)[nH][nH]1)C1CC2(CCN(C(c3cnccc3Br)=O)CC2)C1 98059,O=C(C1=CCCC1)NC1CN(c2cc(-n3cncn3)ncn2)CC1F 98060,C(c1c(F)cccc1F)=CC(N1CC(OCCNC(C(C(C)OC)O)=O)C1)=O 98061,N1(CCC)CCCC1C(=O)NC(C)CNC(C1(C(=O)NC)CC1)=O 98062,Cc1cc(C(N2CCCC(C(C)NC(=O)CCF)C2)=O)cc(I)c1 98063,c1(OC)ccc2c(c1)CCN(C(C(=O)NCC1CCCC1)C1CC1c1ccsc1)C2 98064,N1(C(c2ccon2)=O)CCC2CN(C(c3cc(=O)cc[nH]3)=O)CC2C1 98065,C1(C(N(CCCCCNC(C(COC)N(C)C)=O)C)=O)OCCOC1(C)C 98066,c1(C(=O)NC2CC3(C(NC(c4c(N)cc(Cl)nc4)=O)C3)C2)n[nH]c2c1CCSC2 98067,C1(C(=O)NCc2cccc(CNC(CCCC#C)=O)c2)CCn2c(C)cnc2C1 98068,c1(C(N(C2CN(C(C3CCC(CC(F)(F)F)CC3)=O)C2)C)=O)cc(C#N)ccc1F 98069,C(CCCCCC(=O)N1CCC(O)C(F)(F)C1)NC(=O)CC1CC2CCC1O2 98070,CCCCC(C)CCC(=O)NCC1(NC(c2cccn2C2CC2)=O)CCOC1 98071,n1(CCOCC=C)c(N2CCOC(CSc3cccs3)C2)nnc1CCOCC 98072,C(N=C(NC1CC1)NC1CC(C)(C)Oc2cc(F)ccc21)c1c(C)ncs1 98073,C1(CNC(c2cc(CC)[nH]n2)=O)CCCC2CN(C(=O)C=CN3CCCC3)CC12 98074,n1(C2CN(C(CSc3cn(-c4c(OC)scc4)nn3)=O)C2)nc(C)c(Cl)c1C 98075,C(=O)(CCC(C)(C)F)NCC1C(C(=O)NC(CC=C)C)CCO1 98076,CC1(C)CN(C(c2ccccc2F)=O)CC1CNC(=O)CCCCO 98077,CC(C)(C)CC(C)(C)C(=O)N(CCO)CCO.C(C(C(F)(F)F)C(F)(F)F)N 98078,Cc1ccc(C(=O)NCC2CC2)c([N+](=O)[O-])c1 98079,Cc1cccc(COC(C)C(=O)NC2COCC2NC(=O)C#CC2CC2)c1 98080,CCC(C)CCC(=O)NC1CCCCC1NC(=O)Cn1ccc(C(=O)OC)n1 98081,C1(NC(CCCOCC=C)=O)CCCCC(C)(C)C1 98082,c1(-n2c(C(C(C(=O)OC)NC3CC3)OC)nnn2)c(Cl)nc2ccccn12 98083,c1(C(=O)N(C2CC2)CC2CCCN2C(c2csnn2)=O)coc2c1CS(=O)(=O)C2 98084,C1(C(N2C3C(NC(C(C)OCCOC)=O)C(C3)C2)=O)CCCC2(CCOC2)O1 98085,N(C(=NCCN1CCOCC1)NC(C)Cc1ccncc1)CC(C)(C1CC1)OC 98086,C(=O)(C#CC1CCCC1)NC(CC=CC)C(=O)NC(c1nn(C)cc1O)C 98087,N1(C(c2cc(SC)oc2C)=O)CCC2(CCC2NC(c2occc2C)=O)CC1 98088,C=CC1CN(C(c2ccon2)=O)CC1NC(=O)CCC1CC1 98089,Cc1nn(C(C)C)c(C)c1C(=O)NCC(C1CC1)NC(=O)Cc1ccn(C)n1 98090,C1(CCOC)(NC(c2ccc(OC)o2)=O)CCCN(C(C2C(C)C2(F)F)=O)C1 98091,c1(C(N2C(CNC(C(CCC)C)=O)CCCC2)=O)c(C)cccc1C 98092,C(=O)(C(O)CC(C)C)N(CC(CC)NC(c1ccc(OCC2CC2)nc1)=O)C 98093,C12(NC(c3c(COC)ncs3)=O)CCN(C(=O)COc3ccon3)CCC1C2 98094,c1(Nc2ncc(-c3cccc(CC#N)c3)s2)nccc(Br)c1O 98095,C1(NC(C2CC(C)(CC)C2)=O)CN(C(C2C3CCC(=O)C23)=O)CCC12CCC2 98096,C=CCCC(C(=O)NCCCC(N)=O)NC(=O)CC1C=CCC1 98097,N1(C(c2occc2Br)=O)CC2CC(C1)N(C(c1coc(Cl)c1)=O)C2 98098,C(C)(C)(C(C)CC(=O)NC1C2C3CCC(C3)C12)NC(CC(C(=O)OCC)C)=O 98099,N1(C(C(CCC#C)O)=O)CCN(C(c2ccc(CC)c(F)c2)=O)CC2(CC2)C1 98100,C(C1=CCN(C(=O)CC(F)(F)F)CC1)NC(C(C)Sc1nncn1C)=O 98101,C(=O)(CCCC(F)(F)C(F)(F)F)NCC(C1CC1)NC(c1nc(C#C)sc1)=O 98102,C1(CC)CCC(NC(=NCc2cncc(O)c2)NC(C)CC)CC1 98103,N1(C(C)=O)CCCCC1CN=C(NCc1nnn(C)n1)NC1CCC1 98104,C1(C(N2C(CCC)C(=O)NCC2)=O)CC2CCN(Cc3n[nH]c(C)c3C)CC12 98105,c1(C(=O)NC2CC3CN(C(c4c(CC)nccc4)=O)C2C3)cc2cccnn2c1 98106,C12CN(C(C3(C)CC3(F)F)=O)CC1N2.C1(O)(NCC(SSC)(C)C)CC(F)(F)C1 98107,C1(NCc2cccc(-c3nnc(C)o3)c2)CCC(C)(C)CC1CN=[N+]=[N-] 98108,Cc1oc(C)c(C(N2CCC(NC(=O)CN3CC(C)(C)C3)CC2)=O)c1C 98109,C(c1cccc2cccnc12)=CC(=O)NC1CN(C(C2CC(C)(O)C2)=O)CC1O 98110,Cc1cccc(C)c1NC(=O)C(N1CCC(C)(CNC(C2CCCCO2)=O)C1)=O 98111,c1(C(=O)NCC(F)CNC(c2cccc[n+]2[O-])=O)cc(C2CC2)ncn1 98112,c1(C(=O)OCC)cccc(C(=O)NCC(C)CN(C(=O)COC(C)(C)C)C)c1 98113,CCCC(C)(O)C(=O)NC1CC(CC(=O)NC2CC(C)(C(N)=O)C2)C1(C)C 98114,N1(C(c2ccc(C(N)=O)[nH]2)=O)CCOCC1CC(=O)NCC1(C)CCCC1O 98115,N1(C(C(C2CCCO2)NC(CCCCOC)=O)=O)CCC2(C1)CN(C)C2 98116,CC(F)(F)CCCC(=O)NCC(N1CCN(C(C2CCC2)=O)CC1)=O 98117,C1(NC(CC2(C(=O)OC)CCC2)=O)CCC(n2cc(-c3csc(C)n3)nn2)C1 98118,c1(C(=O)NC2COCCN(C(C3CC4(CCC4)CO3)=O)C2)ccc2ccnn2c1 98119,N1(C(CC(CC(C)(C)C)O)=O)CCCC(C2CN(C(=O)CC(C3CC3)C3CC3)C2)C1 98120,c1(C(N(C2CCN(CC)C2)C)=O)cnc(CNC(=O)Cn2nccn2)nc1 98121,CC(C)C(CCNC(=O)COC(F)F)NC(c1cnn(C(C)C)c1)=O 98122,c1(OC)cc(OC)cc(N(CCO)Cc2n[nH]c(Br)n2)c1 98123,c1(OCCC)ccccc1C(=O)NC(C)CCCNC(c1cc(C)[nH]n1)=O 98124,N1(CC)CC(C(=O)N(C)CCNC(c2ncn(C(C)C)n2)=O)NC1=O 98125,CN1CCN(C(C2(C)CC2(C)C)=O)CC1CNC(=O)CCc1ccc(F)cc1 98126,N1(C(c2c(CC)nn[nH]2)=O)CCCN(C(=O)C#CC2(C)CC2)C(C)C1 98127,c1(C(N2CC(N(C(=O)C3=COCCO3)C)C(C)(C)C2)=O)ccnc2ccncc12 98128,c1(C(N2CC(NC(C3CC(=C)C3)=O)C3C2C3)=O)ccc(C(=O)OC)cn1 98129,CS(=O)(=O)CCC(=O)NCC(CC1CCCC1)C(=O)N(C1CCOC1)CCO 98130,C1(CNC(C2(OC)CCCC2)=O)CCCN(C(c2ccccc2Cl)=O)C1 98131,N1(C(CC(COC)COC)=O)C(C)CN(C(c2cn(C(C)C)nc2C)=O)CC1C 98132,O=C(C1CCc2nccn21)NCCC1CCCCN1C(c1cnc(C(F)F)s1)=O 98133,CC(C)CC(O)C(=O)N(C(CNC(=O)CCC(=O)c1ccc(Cl)cc1)C1CC1)C 98134,N1(C(c2cc(C)cc(F)c2)C(=O)NC2CCC(SC)CC2)CCCC(C)C1CO 98135,N1(C(CS(CC)=O)=O)CCC2(CCCCN(C(C3(Oc4ccccc4)CC3)=O)C2)C1 98136,C(=O)(C(C)C(=O)OC(C)(C)C)N1C(CN(C(CC(C)n2cccn2)=O)C)CCC1 98137,c1(OC)ccc(CCC(=O)NCC(C)N(C)C(c2cccs2)=O)cn1 98138,C(CC1(O)C(=O)Nc2ccccc21)NC(=O)Cc1cc(F)c(Cl)cc1Cl 98139,Cc1nc(C(=O)NCC2(CNC(C3CC34CCCC4)=O)CCC2)cn1C 98140,C1(CC)(CC)CC(NC(=O)Cn2nccc2C)CN1C(=O)CSC1CC1 98141,C(=O)(C(O)CC(C)(C)C)NCCCCNC(C(c1c(C)n[nH]c1C)C)=O 98142,Cn1ncc2c(C(N3CCC(C4(NC(c5cc(O)no5)=O)CC4)C3)=O)ncnc12 98143,CC12CC(NC(c3csc(O)n3)=O)(C1)C1(CN(C(=O)CC3=NNC(=O)C3)C1)O2 98144,Cc1cc(Br)cc(C(=O)NCC2CCN(C(=O)C(F)(F)CO)C2)c1C 98145,C(C)(COC)(CO)SCCCNC(=O)C1COCC(=O)N1.C(C)(C)O.OC 98146,C1(COC)CCCC(C(=O)NCC(F)F)C1 98147,c1(C(=O)Nc2ccnn2C)ccc(S(=O)(=O)N(C)C)cc1.Cc1ccc2c(c1)S2 98148,C(CC(C(=O)N1CCCC1CCO)NC(C1CC=CCC1)=O)OCC 98149,CCCCCCC(F)C(=O)NC1CCN(C(=O)Cc2cnc(C)nc2O)C1 98150,c1(C(=O)NCC(C)NC(=O)CNC(C2CCC2)=O)ccn2ncc(Br)c2n1 98151,N1(C(CC=C=C)=O)CCC2(NC(=O)C(=Cc3cccnc3)F)CCCC12 98152,N1(C(c2ccc(C)o2)=O)CCC(O)CC1NC(c1[nH]nnc1C)=O 98153,N1(C(C(CC)O)=O)CC2CCCC(CNC(c3ncccc3F)=O)(C2)C1 98154,N1(C(C(CC(=C)Cl)NC(=O)C(O)CN2CCCC2)=O)CCc2nc[nH]c2C1 98155,c1(C(CNC(Cc2c(C)ocn2)=O)NC(=O)CC2CC3CC3C2)cccc(Cl)c1 98156,c1(OCC)cncc(C(=O)NCC(C2CCC2)NC(=O)CC2CCN(C)C2=O)c1 98157,c1(CCC(=O)NCC2C(CNC(C3(C(=O)OC)C(=C)CC3)=O)C2)ncccc1C 98158,CC1CC(NC(c2cnn(CCNC(c3ccncc3Cl)=O)c2)=O)CCS1 98159,c1(CC)cc(N2CC3C(CNC(c4n[nH]cc4Cl)=O)C3C2)nc(CC)n1 98160,CCC(O)CC(=O)NCC(c1ccc(C)cc1)NC(c1c(C)nsc1C)=O 98161,N1(C(C2CCN(C3CC3)CC2)=O)CC2CN(C(C3(C4CC4)CC3)=O)CCC2(CO)C1 98162,N1(C(C(C2CCCC2)OC)=O)CCC(NC(c2nc(C3CC3)ncc2Cl)=O)C(F)C1 98163,Cc1ccncc1CC(N1CC2C(NC(c3cn(CCO)nc3C)=O)C2C1)=O 98164,C1(C(=O)NC(C)C(=O)NC2CC2)CC2(CCC2)CN1C(c1cc(=O)cc(Cl)[nH]1)=O 98165,CCCCS(=O)(=O)NC(C)C(=O)NC1(CCNC(c2nnn(C)c2C)=O)CC1 98166,N1(C(C2C(C)(C(C)C)C2)=O)CCN(C(=O)CC(C)(F)F)C2(CCC2)C1 98167,C1(C(N2C(C(C)CNC(c3cccnc3)=O)CCCC2)=O)CC(C)(C)CN1C 98168,C1(NC2(c3n(CCOC)nnn3)CC3CCCC23)CCC2(CCOC2)O1 98169,N1(C(c2cnc(CC)s2)=O)CC(C)CCC1CNC(=O)CNS(=O)(=O)NC 98170,C1(CNC(=O)C(F)Cc2ccccc2)CN(C(=O)C=Cc2cc[nH]n2)CCCO1 98171,C(CN=c1[nH]n(C)cc1[N+](=O)[O-])C1N(C(c2cc(C)nc(Cl)c2)=O)CCCC1 98172,N1(C(c2c(SC)snn2)=O)CCCCC1CCCNC(C1CCS1(=O)=O)=O 98173,c1(C(=O)NCC2(C)CCCN2C(c2cccc[n+]2[O-])=O)ccc2scnc2c1 98174,C1(C(=O)OC)COC(CCC(=O)NC(C)CCNC(=O)C(N)=O)C1 98175,CCC(C)C(C(=O)NC1C(C#N)C1(C)C)N(c1ccccc1)Cc1cccc(O)c1F 98176,C(=O)(C(CC(C)(C)C)OC)NCC(CNC(C1CCC(=C)CC1)=O)OC 98177,c1(C(N2CCC(O)(C(N3CCOC(CO)C3)=O)C2)=O)c(F)cncc1F 98178,C#CCC(CC#C)C(=O)NCC1CCN(C(C2(C)CCN(C)CC2)=O)C1 98179,CC1CN(CC(=O)CCc2c(F)cccc2F)CC2(CCCOC2)O1 98180,CCC(O)CC(=O)N1CC(CC(C)NC(c2cc(-c3ccc(Cl)s3)on2)=O)C1 98181,C1(N(C(=O)CCCSC2CC2)CCNC(C=CCOC)=O)CCC2(CCC2)OC1 98182,C1(C(=O)NCC(C(C)C)NC(CC(C(F)(F)F)OC)=O)COc2ccccc2O1 98183,N1(C(c2ccc(N(C)C)cc2)=O)CCN(C(=O)CNC(=O)NC2CC2)C2CC12 98184,CN1CCOc2ncc(C(=O)NCC3CC3CNC(C3(F)CCC3)=O)cc21 98185,CC1CC(C(=O)NCC(C)(O)C2CC2)N(C(C2CC(CF)C2)=O)C1 98186,C(CC(F)F)(C(=O)N(C1CC1C1CC1)C)N(C(=O)CC1CC(C2CC2)C1)C 98187,N1(C(=O)NC2CN(CC(=O)OC)C(=O)C2)CCC(NC(SC(F)(F)F)=O)C1(C)C 98188,C1(c2cn(CC3CCC3CN)nn2)(NCC)CCCOC1 98189,C(=O)(CCCC(C)(C)NC(=O)C=Cc1cnn(C)c1)N1CC(O)(CC(C)C)C1 98190,C1(C(=O)NC2CCN(C(c3c(S(N)(=O)=O)n[nH]c3)=O)C2)CCCCC12OCCO2 98191,N1(C(C2C(C)C2C)=O)CCOC(CNC(=O)CO)C1.C12CCCN(C1)C2=O 98192,C(=O)(C(CNC(c1csc(F)c1)=O)CC1CC1)N(C(C)(C1CC1)C1CC1)C 98193,C1(CNC(COCc2n(C)ccn2)=O)CN(C(C2C3CCCCCC23)=O)CC1(C)C 98194,c1(CC(=O)NCC2CCC(NC(C3CC(=C)C3)=O)C2)cc(Br)ccc1F 98195,C1(NC(C=CC(C)C)=O)CCC(C)N(C(c2cnn(C3CC3)c2Cl)=O)C1 98196,N1(C(=O)CCCc2ccccc2)CCN(C(=O)C(O)C2CC2)C(CCO)C1 98197,N1(C(C2CC(C#N)C2)=O)C2CC1CN(C(=O)CC(=O)NCC1CC1)C2 98198,O=C(CCCCCCNC(C1CCOC(=O)CC1)=O)NC1CCC(F)(F)C1 98199,C(CCN=c1[nH]c(N2CCN3CCOCC3C2)nc2c1SCC2)OC(C)(C)C 98200,CCCC(C)(CC)C(=O)NC(C)CNC(c1ncccc1-n1cccn1)=O 98201,c1(C(=O)NCCC2N(C(CCCC(C)C)=O)CCOC2)ccc2c(c1)C(C)CO2 98202,C1(C(N(C2CCN(C(c3cc(C(F)(F)F)on3)=O)C2)C)=O)CCCS(=O)(=O)N1 98203,C1(C(=O)NC(CC)CO)CC(NC(C2(C)CC(C)=NO2)=O)C(O)C1 98204,c1(C(N2CC(CN(C(C(CSC)OC)=O)C)OCC2)=O)cn2cc(Cl)cnc2n1 98205,c1(CNC(c2nccc(CNC(C(CC)(C)O)=O)c2)=O)cc(C)cc(F)c1 98206,Cc1cc(C(F)F)n(CC(N2CCC(NC(=O)CC3(C)CCCC3)C2C)=O)n1 98207,N1(C(c2cn(C)nc2)=O)CCOC2(CCN(C(c3cc4n(n3)CC(F)C4)=O)C2)C1 98208,C1(C2(NC(=O)C=CC(C)(C)N(C(=O)CCCC(C)=O)C3CC3)CC2)(OC)CCC1 98209,c1(CC(=O)NC23N(C(COCCCOC)=O)CC(C2)C3)c[nH]c2cccnc12 98210,CCCCCC(C)CC(=O)NCCN(C(=O)C(F)CC1CCCC1)C 98211,N1(C(c2cccc(C(C)C)n2)=O)CC(CNC(=O)COC2CC2)N2CCC1C2 98212,C(CC(F)F)(C(=O)NCc1cc(O)ccc1F)N(C)C(c1ccnc(CO)c1)=O 98213,C12CCC(CC1)CNC2=O.C(=O)(C(C)CC1CCCC1)NCC(=O)OC 98214,n1(CC(=O)NC2C3N(C(c4c(C)cn(C)c4)=O)C(CC3)C2)cc2ccccc2n1 98215,N1(C(Cc2scc(C)c2)=O)CCC2CN(C(c3cnc([N+](=O)[O-])n3C)=O)C(C)C12 98216,C1(CNC(C2N(C(N)=O)CC(O)C2)=O)CC2(CC2)CN1C(=O)CC(C1CC1)C1CC1 98217,N(CP(C)(C)=O)(C(c1cc(C)oc1C)C(=O)NCCCF)CC(=O)OC 98218,c1(C(=O)NC2CCN(C(c3c(CC)cno3)=O)C2C)ccc2ncccc2n1 98219,N1(C(C(C)(C)CF)=O)CCN(C(c2cc(F)c(CO)c(F)c2)=O)CC(O)C1 98220,c1(CCC(=O)NCC2(N(C)C(C3CCC3)=O)CC2)nc(-c2ccccn2)no1 98221,N1(C(C(C=CC)O)=O)CCN(C(=O)CNC(C2(c3cccnc3)CC2)=O)CC1 98222,Cc1cc(OCCC(=O)N(CCCNC(C2CC23CCSCC3)=O)C)cc(C)c1 98223,CC(C)C(C)COCC(=O)NCCC(C)N1CCC1.C1(CC(=O)N)CC=CC1 98224,c1(C(=O)NCCN(C)C(c2ccc(C(F)C(F)(F)F)cc2)=O)ccnc(Cl)c1N 98225,c1(C(=O)NCC#CC(=O)NCC2CN(C(C)=O)C2)c[nH]c(=S)cn1 98226,c1(C(N2CC(N(C(C3N(C)C(=O)CC3)=O)C)C(F)C2)=O)cncc2c1CCCC2 98227,C(=O)(NNC(=O)c1c(C(F)(F)F)cnn1C)N(C)C 98228,Cc1c(Cl)ccc(Cl)c1NC(C1C=CCN1C(c1ccc(Br)cc1I)=O)=O 98229,C(=O)(CC(C)c1cnn(C)c1)N(CCCCN(C(C1(SCC)CC1)=O)C)C 98230,c1(COC)csc(C(=O)N(CCNC(C2CCCC2F)=O)C2CC2)c1 98231,N1(C(CCC#C)=O)C2CCC1CN(C(=O)Cc1ccc(Cl)nc1F)C2 98232,C12(C(=O)NC3C(NC(C(C)(C)SC)=O)CCCC3)CCCC(CCC1)C2(F)F 98233,C(C)(CCC(F)(F)F)(C(F)(F)F)NC(CNc1ccc(OC)cc1)=O 98234,C(=O)(CCC(C)(C)F)N(CC(Cc1ccccc1)NC(C1CC(O)C1)=O)C 98235,CC1CCC(NC(=O)Cn2cnnc2)CN1C(=O)CCCC1CCCC(=O)N1 98236,C1(NC(c2cnns2)=O)CC12CCCCCC2.C12(CC1)C(=O)NCC2 98237,c1(C(N2CCC(N(C(C=C(CC)CC)=O)C)C2)=O)c(C)c[nH]c1CC(N)=O 98238,C1(C#N)(C(N2CC(OC)(CNC(C3CCCC(N(C)C)C3)=O)C2)=O)CC12CCC2 98239,C(=O)(CCS(C)(=O)=O)NCCCCC(C)NC(C1COCC1(C)C)=O 98240,N1(C(CCN(C)CCO)=O)CC(O)(C2(CNC(C3(C)COCCO3)=O)CC2)C1 98241,c1(C(N2CCCC(N(C(C34COCC3C4)=O)CC)C2)=O)cccc(F)c1C#N 98242,c1(CNC(Cn2cc(CNC(C3(C)C(C)(C)C3)=O)nn2)=O)ccncc1F 98243,c1(C(N(CC(C)NC(=O)C(c2ccc(C(F)F)cc2)C)C)=O)cc(Cl)cn1C 98244,C1(CNC(Cc2c(C)nc[nH]2)=O)CN(C(=O)CC2CCC(C)C(C)C2)CCCO1 98245,Cc1nc2c([nH]1)CN(C(C1CCCCCN1C(C1COCC(C)O1)=O)=O)CC2 98246,CC(C)CC(CNC(c1cc(C#N)n(C)n1)=O)C(=O)NCc1ncsn1 98247,N12CC(C(C)C1)Cc1cc(n(C)c1)C(=O)OC(C1CN(OC)C1)C2=O.O(C)CC 98248,C12(C(=O)NC3(C)CC(N(C)C)C3)CC1CN(C(=O)CN(c1ccc(Cl)cc1)C)C2 98249,C1(C(=O)NC23CC(NC(=O)C=Cc4cnccn4)(C2)C3)CC2CCCCC2O1 98250,C1(CNC(C2(NC(C(CC3CC3)OC)=O)CC2)=O)CCCCC1(C)C 98251,c1(C(=O)NCCCCN(C(Cc2cc(C)sc2C)=O)C)cc(O)nc(O)n1 98252,c1(C(=O)OC)cc(C)nc(N(C(C)CNC(=O)Cc2cc(C)ns2)C)n1 98253,C1(NC(C=C(C)C(C)(C)C)=O)CCC(NC(=O)CC(O)c2ccccc2)CC1 98254,Cc1c(C(=O)N(C)CCOCCN(C)C(C2CC2Cl)=O)cccc1N 98255,Cc1cc(C(=O)NC2CCC2CNC(c2ncc(Cl)s2)=O)cc(C)c1Cl 98256,C1(NC(C(C)C2CCC2)=O)CCOC12CCN(c1ccc(F)cc1[N+](=O)[O-])CC2 98257,C(=O)(C1=C(C)S(=O)(=O)CC1)N(CCN(C(=O)Cc1ccc(OC)cc1)CC)CC 98258,c1(OCC=C)c(NC(C2(C)CCN2C(=O)CC(F)(F)F)=O)cccc1C 98259,CC1(C)Cc2c(Br)cccc2C1NC(=O)N(c1ccc(Cl)cc1)CC(F)F 98260,C1(CCNC(CCCNC(N)=O)=O)CCN(C(=O)Cc2ccsn2)CC1 98261,O=C(C1=CCCOC1)NC1CCN(C(=O)Cc2cnc(C3CC3)[nH]2)CC1F 98262,CCCCS(=O)(=O)CC(=O)N1CC2C(CNC(c3cn(C)cn3)=O)C2C1 98263,n1(CCC(N2CC(NC(c3cnco3)=O)C(O)C2)=O)ncc2c1CCCC2 98264,N1(C(C2(NC)CCC2)=O)CCC(N(CCS(N)(=O)=O)C(=O)NC(C)C)CC1 98265,C1(NC(C(c2ccc(C)o2)C)=O)CC2CCC1N2C(C1(C)CC1)=O 98266,N1(C(CC2CC(=C)C2)=O)CCC(CCNC(C2CCOC2C(C)C)=O)CC1 98267,C1(CC)CN(C(=O)Cc2ccnc(Br)c2)CCN1C(c1nc(O)cs1)=O 98268,C1(CNC(CCCOCC)=O)CCC(C)(C)CN1C(=O)CCSC1CCCCC1 98269,N1(C(CC(C=C)C)=O)CC2CCC1C(CNC(c1cccc(F)c1CC)=O)C2 98270,C(CC(F)(F)F)(c1ccc(Cl)cc1)NC(C1CC(=O)N(CC2CCCC2)C1)=O 98271,c1(C(N2CCCC(C)(NC(=O)C=C3CC3)C2)=O)cccc2c1C(=O)NC2 98272,c1(NC)cnncc1C(=O)NC1COCC1O 98273,C(c1cccnc1)=C(C)C(=O)NCCOCCNc1ccnc(N2CCCC2)c1 98274,N1(C(C2(SC)CCC2)=O)CCC(C=CC(=O)Nc2ccn(C(C)C)n2)CC1 98275,C1(C(N2C(C(N(CC(C)(C)N(C)C)C)=O)COCC2)=O)CC2(C1)CC2(F)F 98276,c1(C(=O)NCC(C)NC(c2c(CC)nc[nH]2)=O)ccc(F)c(Cl)c1N 98277,N1(CC2CC(C(=O)OC)CN(C(C3CCCO3)=O)C2)CCC(O)C(C)(C(F)(F)F)C1 98278,c1(NC(N2CCOC(C3CC3)CC2)=O)ccnc2c1CCC2 98279,c1(CC(=O)N(CC(C)NC(=O)CCNC(N)=O)C)cccnc1Br 98280,c1(CC(N2C(CNC(C(C3CC3)SC)=O)CC2)=O)cccc(C)c1F 98281,C12(CNC(CSCC)=O)COCCN1C(=O)CN(C(c1cnc(=N)[nH]c1)=O)C2 98282,c1(CC)ocnc1C(=O)NC(C)C(CO)NC(c1cc(F)n[nH]1)=O 98283,C12(NC(C(CC)CC)=O)CC3CCC(C1C2)N3C(c1cnc(N)s1)=O 98284,c1(N2C3CN(C(C4(CC)CCOCC4)=O)CC2CC3)ncnc2cc(C#N)ccc12 98285,N1(C(Cc2c(C)ncnc2C)=O)CCC2CN(C(=O)CC3NC(=O)NC3=O)C2C1 98286,c1(N2CCCC3(NC(c4ccsc4)=O)C(C2)C3)nc2cc(F)ccc2o1 98287,C(=O)(C(C)(C)C(C)O)NCC1(C(C)NC(c2nc(CC)sc2)=O)CC1 98288,c1(OC)cc(OC)cc(CCNC(=O)NC(c2cc(Br)ccc2C)C(F)(F)F)c1 98289,C(C)(C)(CC(=O)NC1CC(CC(N2CCCC(O)C2)=O)C1)OC 98290,N1(CC)CCOC(C(N2CCC(CNC(C3(COC)CC3)=O)C2)=O)C1 98291,Cc1cc(C(=O)NC2CC2CNC(=O)C(C)C#N)c(C)n1-c1ncc(Br)cn1 98292,C1(CC(=O)N(CCCNC(=O)CC2(O)CCC2)C)CCOC(C)(C)C1 98293,C1(NC(C2C(C(=O)OC)C2)=O)CCN(C)C12CCCN(C(c1sccc1Cl)=O)C2 98294,c1(C(CCC(c2nnnn2C(C)(C)C)C(c2ccsc2)C)N)cc(Cl)n(C)n1 98295,c1(C(N(CCN(C(=O)CCCc2cnn[nH]2)C)C)=O)cnn2cccc(Cl)c12 98296,C1(CCCNC(C2(C)CC2)=O)CN(C(c2ccc(-c3ccco3)s2)=O)CCO1 98297,C1(C(=O)NC2C(CNC(c3c(C(C)C)ocn3)=O)C2)CC12CC(F)(F)C2 98298,c1(C(=O)OC)cc(C(N2CC(CCNC(C3CC3F)=O)(OC)C2)=O)nn1C 98299,n1(CCC)ncc(C(=O)NCC2(NC(c3cc(C)cs3)=O)CCC2)c1C1CC1 98300,CC(CCN(C)C)C(=O)NCC1CC(F)CN1C(=O)Cc1cc(C(F)(F)F)co1 98301,C1(CN(C(c2n(CC)nnc2)=O)C)COCCN1C(c1nncs1)=O 98302,C#CCC(C)(C(=O)NC1CC(O)CC1O)NC(C1(CC(=O)OC)CC1)=O 98303,C(=O)(CC(CC)NC(=O)C(O)C1CC1)NCC(=O)OCC=C 98304,C1(NC(C2C(C(C)(C)C)C2)=O)CC2CC1N(C(C1CN3CCC1CC3)=O)C2 98305,c1(CC)nc(C(=O)NC(C2CCN(C(=O)CC3(N(C)C)CC3)C2)(C)C)co1 98306,N1(C(COCCCOC)=O)CCCC(C2CCN(C(=O)COCCF)CC2)C1 98307,C=CCCCC(=O)NCC1CCCC(CNC(c2cnc(-c3ccsc3)s2)=O)C1 98308,C1(C)(NC(CC2(C)CCC2)=O)CCCN(C(C2CC(C)(F)C2)=O)C1 98309,C=CC1(NC(=O)C(F)CC2CN(C(c3cccc(CO)c3)=O)C2)CCOCC1 98310,c1(NCC(CNS(N(C)C)(=O)=O)O)cc(S(=O)(=O)NCCSCCO)ccc1C#N 98311,CC#CCC(C)NC(=O)CN(C(c1cccnc1)=O)CC1CC1 98312,C1(CNC(CCNC(=O)NC)=O)CCC(C)N(C(c2nc(OC)ccc2Cl)=O)C1 98313,C(=O)(C(CN=[N+]=[N-])NC(c1n[nH]c2c1CCC2)=O)NCC1CCCN(C)C1 98314,N1(CCc2cn(C3CN(C(C(COC)(C)OC)=O)C3)nn2)CC(O)CCC1=O.C(C)=O 98315,CN=c1ncc(C(=O)NC2CC(C(=O)Nc3cc(N(C)C)ccn3)C2)c[nH]1 98316,CCC1=C(C(=O)NCCC2CCCN(C(c3cnncc3OC)=O)C2)CCCO1 98317,N1(CCC(=O)NC23CC(C2)N(C(c2cncc(F)c2)=O)C3)C(=O)CCC1=O 98318,c1(C(N(CC(C)NC(C2C=CCC2)=O)CC)=O)ccc(P(C)(C)=O)s1 98319,C1(C(N2CC(C)N(C(C3C(C)(C)C3(C)C)=O)CC2)=O)CC2(C1)NC(=O)NC2=O 98320,c1(C(=O)NC2CCC(NC(C3C(C)=C3)=O)C2)c(C)c(C)nn(C)c1=O 98321,c1(C2C(C(=O)NCCN(C(c3cnn(C)c3OC)=O)CC)C2)ccccc1C 98322,c1(-n2c(C3CN4CCCC4CO3)nc(CCN(C)C)n2)cn(C)c(=O)n(C)c1=O 98323,C(=O)(C#CC1CCOC1)N(CCOCCCN(C(c1cnc(COC)s1)=O)C)C 98324,N1(C(c2n(CC=C)ccn2)=O)CCCC(CC)(CNC(=O)C#CC2CC2)C1 98325,c1(CC(=O)NCC2N(C(C3C(COC)C3)=O)CCCC2)cc(C(N)=O)ccc1Cl 98326,c1(CC(C)C(=O)N(C)CCN(C)C(c2cc(F)c[nH]2)=O)ccccc1F 98327,C1(CNC(C2(CF)CCC2)=O)CCCC1C(N1CCC1c1cscn1)=O 98328,c1(C(C)O)ncc(C(=O)NC2CN(C(=O)COCc3nccs3)C2)s1 98329,CC(CCN(C(=O)CCSC(F)(F)F)C1CC1)NC(=O)C=CCN1CCCC1 98330,N1(C(c2c(OCC)ccs2)=O)CC2(CCCN2C(=O)Cc2cc(Cl)ccc2Br)C1 98331,c1(C(=O)NCC2CCCN2C2CCCCC2)cccc2c1OCCC(=O)N2 98332,N1(C(C)C(=O)Nc2cccc3ccccc23)CC2(CCCC(C)(C)O2)C1 98333,c1(OC)cc(CC(N2CC(NC(c3coc(C)n3)=O)C3CC23)=O)ccn1 98334,c1(NC(C(N2C(CC=C)CCC2)=O)=O)cccc(F)c1C 98335,C(=O)(CS(=O)(=O)C1CCCC1)NCC1CN(C(C(CSC)OC)=O)C2(C1)CCC2 98336,N1(C(C=NOC)=O)CC2CN(C(=O)Cc3cc[nH]n3)CCC2(CO)C1 98337,C#Cc1ccc(C(=O)N(C(C)CCNC(=O)C(CC)CCOC)C)cc1 98338,C1(NC(=O)NCc2nc(Cc3cccc(Br)c3)cs2)C2CCOCC12 98339,C(c1c(C)cccc1C)=CC(=O)NC(CCC)CNC(C1(n2cnnn2)CC1)=O 98340,c1(C(=O)NC(CC=C)CNC(C2CCCCCN2C)=O)cc2cc(C)ccc2o1 98341,C1(C)(CNC(C2N(C(C)C)CCC2)=O)CCN(C(=O)CCn2ccnn2)C1 98342,c1(CN2C(CC(=O)Nc3cccc4c3CCC4)COCC2)cccc2sccc12 98343,C(CC(F)F)(C(=O)NC(c1ncc(OC)cn1)C)NC(C(COCC)C)=O 98344,Cc1nc2cc(C(N3CC(CCNC(=O)CC(C)P(C)(C)=O)C3)=O)cc(O)c2[nH]1 98345,C1(C(=O)NCCN(C(C2(COC)CCCCO2)=O)C)CC(=O)N(OC)C1 98346,c1(CC)cn(C)nc1C1CC1.c12sccc1CC(=O)NC(CSC)CNC2=O 98347,c1(C(=O)NCC(CNC(=O)Cc2cc(C(F)(F)F)no2)O)cccc(OC(F)F)c1 98348,c1(C(=O)NCC(CNC(CCCNC(N)=O)=O)F)sc([N+](=O)[O-])cc1Cl 98349,c1(C(N2CCN(C(=O)C(O)C3CCCC3)CC2CF)=O)ccn2nccc2c1 98350,C(C(C(=O)NC(C1CCCC1)CNC(c1ccn(C)n1)=O)N(C)C)N(C)C 98351,c1(OC)ccc2[nH]cc(NCC(=O)Nc3ccc(Cl)c(F)c3)c(=N)c2c1 98352,c1(CC(=O)NCC2CN(C(C3N(CCC)CCC3)=O)C2)c(C)oc2ccccc12 98353,CC(CC(=O)N1CCOC(CC(=O)NCC(F)Cl)C1)C(C)(C)C 98354,CC1(C)CC(C(=O)NC(C)(C)C(C)(C)CO)CN(C(C2C3CCCC23)=O)C1 98355,Cn1nc(C2CC2)c(Br)c1C(N1C(CO)CCC12CCC2)=O 98356,Cc1nc(C(C)(C)C)nc(O)c1C(N1CCCC(C)(NC(C2CC2CF)=O)C1)=O 98357,C(=O)(C(C(C)(C)C)N1CCCC1=O)NC1CCN(C(c2ccc(OC)cn2)=O)C1 98358,N1(C(COCCCC(C)C)=O)CC(CNC(C2CCC(N(C)C)CC2)=O)C(C)C1 98359,N1(C(CCCC=C)=O)CCC(CC)CC1C(=O)N(CCC1CCC1)CC 98360,Cc1ccc(C(N2CC(NC(c3ncoc3C(C)C)=O)CC(C)C2)=O)c(N)c1C 98361,N1(C(CC2CC(SC)C2)=O)C(C)CN(C(=O)CC2CCC(=O)N(C)C2)CC1C 98362,C(=O)(C#CC1CCOCC1)NC1C(NC(c2c(C)noc2C)=O)CCCC1 98363,C1(CC)CCN(C(=O)OC(C)(C)C)C(NC(=O)NCCN2CCC(C(C)(C)C)C2)C1 98364,C#Cc1cccc(C(=O)NC(CNC(c2ccc[nH]2)=O)CCOC)c1F 98365,C=CCCCCC(=O)NC(c1ccccc1)CNC(=O)C=C1CCCCC1 98366,C(=O)(C(C)(C)CC(C)(C)C)N(C1CCC(CNC(C(C)C(C)(C)C)=O)CC1)C 98367,c1(CN2CCC3(C(C(=O)Nc4ncc(C#N)cn4)C3)C2)ccc([N+](=O)[O-])c(Br)c1 98368,c1(C(=O)NC(CC)CNC(=O)C(c2cccn2C)=O)ccc(N)c(C)c1C 98369,c1(C(N2CCCCC(NS(CC=C)(=O)=O)C2)=O)cccc(C(F)(F)F)c1O 98370,c1(C(=O)NC2CCN(C(C(CC)(C)O)=O)CC2CO)cccc2c1CCO2 98371,N1(C(c2ccc(OC)cc2)=O)CCN(C(=O)Nc2cc(Br)ccc2OC)CC1C 98372,c1(C(N(C)CC2(O)CCN(C(Cc3nc(CC)sc3)=O)C2)=O)cccc(N)c1C 98373,N1(CCN2CC(C)OC3(C2)CCC3)CCC2(CC1)OCCc1ccsc12 98374,c1(C(=O)NCCN(C(=O)C(F)n2ccnc2)CCC)cc(F)c(Cl)cc1Cl 98375,c1(C(N2CCC(NC(CC(CCCC)CC)=O)C2)=O)ccc2c(=O)n(C)c(C)cc2n1 98376,c1(C(CN(CC(C)Cc2ccc(Cl)cc2)C(C)=O)=O)cc(C(C)C)cc(Br)c1 98377,C1(C(N(CCCCNC(c2c(SC)ccs2)=O)C)=O)Cc2ccccc2CO1 98378,N1(C(C=C(C)C(C)(C)C)=O)CC(O)CC1CNC(=O)C(O)C1CC1 98379,c1(C(=O)NCC(C(=O)NC(CCC)C(=O)N(C)C)O)cc(C)c(C)nn1 98380,N1(C(c2cccc(CC)c2)=O)CC2(C1)OC1(C)CC2(NC(C2CCCOC2)=O)C1 98381,Cc1cnn(C)c1CNC(C1C(C)CCN1C(=O)CC(C)(C)C)=O 98382,C1(CC=C)(C(=O)NC(C)Cc2ccnn2C)CCN(C(c2ccnn2C=C)=O)C1 98383,N1(C(CC2CCC(C)O2)=O)Cc2ccccc2C(CNC(C23CC(C)(C2)C3)=O)C1 98384,CCCC(C)CC(C(=O)NC)N1CCN(C2CCC2)CC(C)(F)C1 98385,C1(SC)CN(C(=O)C(O)Cc2ccccn2)CC1NC(=O)COc1cn[nH]c1 98386,C(C)(C)(CC(=O)N1CC2CC1C2C(=O)NCc1cncs1)N(C)C 98387,C1(CNC(=O)CN(C(c2ccccn2)=O)C2CC2)CC(CNc2cnco2)CO1 98388,C1(NC(=O)NCCCOc2c(C)ccc(C)c2)CC(C)c2ccccc2N1 98389,N#Cc1cnc(N2CCC(F)(F)C(CNC(c3cccc(Cl)n3)=O)C2)c(Cl)c1 98390,N1(C(c2sc(C)c(Br)c2)=O)CCC2CN(C(c3c(F)cccc3Br)=O)CC12 98391,C1(NC(C(C2CC2)OCC)=O)(CF)CCN(C(=O)CC2COCC(C)O2)C1 98392,Cc1cn2ccnc(C(=O)NC3CCCC3CNC(c3cn(C)nn3)=O)c2n1 98393,CC(=O)CCCCC(=O)NCC(CNC(=O)CCc1cc(Cl)no1)CO 98394,CONC(=O)C(=O)NCC1CN(C(c2ccc(C3CC3)o2)=O)CCO1 98395,C(CC(=O)N1CCC(NC(=O)COc2ccccc2F)C1C)(C(N)=O)NC(C)=O 98396,c1(CC)cc(C(N2CCCC(NC(=O)CCc3cc(C)no3)CC2)=O)ccc1O 98397,C(=O)(CN1C(=O)Cc2ccccc21)OC1CCCC(OC(C)(C)C)CC1 98398,C1(NC(C(C(C)C)(C)C)=O)COC2(CCN(C(=O)CN3CC=CC3)C2)C1 98399,c1(CN2CC(OCC)C(CC(=O)NS(C)(=O)=O)C2)c[nH]c2cc(Br)ccc12 98400,c1(C(N2CC(C(=O)Nc3ccns3)OCC2)=O)ccc2occc2c1 98401,C1(CC(=O)N(C(C)C(=O)NCCCc2cc[nH]n2)CC)CCC(CC)O1 98402,N1(C(C(C(C)C)SCC)=O)CCC2(CCCC2NC(=O)CC2CSCCS2)CC1 98403,C1(C(=O)NCCn2c(C)ncc2)CCC(O)CN1C(c1cccc(F)c1O)=O 98404,c1(C(=O)NCCCN(C(C2CCC(CC)O2)=O)C)cccc(C2CCOCC2)c1 98405,C1(CC#C)(C(=O)NC2CCCCC2CO)CCN(C(C2CCOC2C(C)C)=O)C1 98406,C12(NC(=O)CCC3CCCO3)CC3CCC(C1C2)N3C(=O)C(O)c1ccsc1 98407,N1(C(CCCOC(C)=O)=O)CCCC(NC(c2nnc(S)n2C)=O)C(F)C1 98408,c1(C(N(C)CC2(NC(c3cc(C(=O)OC)on3)=O)CC2)=O)noc2c1CCCC2 98409,c1(SC)cccc2c1N(C(C(=O)NC(=O)OC(C)(C)C)c1ccoc1)CCC2 98410,c1(CCC(=O)NC2CCC(NC(C(CC)OCC)=O)C2)ccc(OC)cc1F 98411,C(=O)(CCS(C)(=O)=O)N(C1CCN(C(c2c(C)onc2)=O)CC1)CCOC 98412,c1(NC(C(C(=O)N(CC)CC2C3CN(C(=O)NC)CC23)F)=O)cc(C#N)cn1C 98413,n1(C(C)(C)C)ncc2c(N)[nH]c(=NC3C=CCCCC3)nc12 98414,C1(C(=O)NCc2n(CC)ncn2)CC2CC1CC2NC(c1cc(C)nnc1C)=O 98415,C1(CC(C)NC(C(C)=CC2CC2)=O)CCN(C(=O)CSCC(F)F)CC1 98416,C(=O)(C(C)C(=O)NC1(CO)CN(C(C2(C(C)(C)C)CCC2)=O)C1)OC 98417,C(=O)(C1c2c[nH]nc2CN1C(=O)CCNC(C)=O)NCCOCCC 98418,C1(NC(COC2CCCN(C)C2)=O)CN(C(=O)CCc2ncnn2C)C(C)(C)C1 98419,c1(C(N2C(C3(OC)CC3)CCC2)=O)cc(C)cnc1C.C12CCC(CC1)NC2=O 98420,C1(CC)CN(C(c2cnns2)=O)CC1NC(c1ccc(CN=[N+]=[N-])cc1)=O 98421,CC1C(C(N2CCC(CCNC(=O)C(C)(Cl)Cl)C2)=O)C(O)C(=O)N1C 98422,C#Cc1cnn(C)c1C(N1CCC(CCN(C(=O)COC(C)C)C)CC1)=O 98423,c1(CC)cccc(C(=O)N(C(C)CCNC(c2cncc(C)n2)=O)C)c1O 98424,N1(C(C2(C)CSC2)=O)CCC2(COC(CNC(C3(C)CCSCC3)=O)C2)C1 98425,c1(C(=O)NC(CNC(c2cc(CC)n(C)n2)=O)C)c[nH]cc(Br)c1=N 98426,c1(CNC(C2(C(=O)NCC)CC(O)C2)=O)ccncc1OCC(F)F 98427,c1(NC(=O)NCC)nccc(=NCC(NCC2CC2Br)N)[nH]1.CC 98428,C1(CCSNC(C(=O)NC(c2ccccc2F)C(C)C)=O)CCNCC1(F)F 98429,C1(C(C(=O)NCCOCC=C)C)CCNCC1 98430,C(=O)(C1=C(C)CCOC1)N1CCC(C(=O)N(C)Cc2ccoc2C)(COC)C1 98431,c1(C(=O)NC(CNC(C2CC(C)(CC)C2)=O)C)cc(C)ccc1[N+](=O)[O-] 98432,CC(C)C(F)(F)CC(=O)NC1CCC(C)N(C(c2cc(N)c(Cl)cn2)=O)C1 98433,C1(c2nc(C)on2)CCN(C(=O)CCCCNC(=O)OC(C)(C)C)CC1 98434,c1(C(=O)NCCN(C(=O)CNC(c2ccc(Cl)s2)=O)C)cc(C#N)c[nH]1 98435,c1(C(=O)NCC(CN(C(C(CCCC)O)=O)C)C)coc2cc(F)cc(F)c12 98436,C1(NC(c2n(CCSC)nnn2)C2CC(F)(F)C2)C(C)CCC1C 98437,c1(CC)cccc(C(N2CCC(CCNC(C3(C)C=CCC3)=O)C2)=O)c1N 98438,c1(C(CC)NC(=O)C(C2CC2)NC(=O)CCOCC(F)F)cccnc1 98439,C1(C(=O)NCCNC(CC2(C)CC(F)(F)C2)=O)COC2(CCC2)CO1 98440,c1(CC)cc(C(=O)NCCCNC(=O)CCc2cccnc2F)cn(C)c1=O 98441,c1(C(=O)NC2(C#N)CCC(C)C2)ccc(S(=O)(=O)N2CCCCCCC2)cc1 98442,N1(C(CC(C)CNC(=O)Cc2cnoc2)=O)CC2CCN(C)C2C1 98443,C(S(=O)(=O)C(C)C(=O)NC)c1n(CC)c(N(C(C)C(CC)CC)C)nn1 98444,Cc1c(C(N2CCC(CNC(C3CC4CC3C4)=O)CC2)=O)oc2c(C)cccc12 98445,c1(C(=O)NCC(CNC(c2c(C(C)C)con2)=O)F)cc(F)ccc1N 98446,c1(NCCOC)cc(=NCC2CN(C(=O)CO)CCO2)[nH]cn1 98447,N1(C(C2CC=C(C)CC2)=O)CCCC(C2CC2NC(=O)C(C)(C)C(F)F)C1 98448,CC1C(=O)N(C)CN1C(=S)NC1CCCC(F)(F)C1 98449,c1(C(N2CCC(C(=O)N3CC(O)CCO3)(C(C)C)C2)=O)cccc([N+](=O)[O-])c1 98450,C12(C(C)C)CCC(NC(=O)C(CC3CCOCC3)NC(=O)CN(C)C3CC3)C1C2 98451,c1(C(=O)NC(C2CCCN2C(=O)Cn2cnnc2O)(C)C)ccc2nn[nH]c2c1 98452,C(C)(C)(CC(F)C(=O)NC(c1cccnc1)CO)NC(c1ccc(C)nc1O)=O 98453,c1(C(N2CC3C(CNC(C(C)CC(F)F)=O)C3C2)=O)nnc2ccccc2c1N 98454,CN=c1[nH]cc(C(N2CCCC(C3CCCN3C(=O)COc3ccsn3)C2)=O)s1 98455,C1(C(N(CC(O)CF)C(C)C)=O)COCCN(C(c2ccc(C#N)o2)=O)C1 98456,Cc1cc(C(C)C)nc(N2CCN(C)C(CNC(=O)Cc3ccoc3)C2)n1 98457,C1(S(C)(=O)=O)(C(=O)NC2CC(C)(NC(CC3C(C)C3(F)F)=O)C2)CC1 98458,N1(C(Cc2c(C)ocn2)=O)CCC(C)(C)C1C(=O)NCCCN1CCC(O)C1 98459,c1(C(=O)NCC23C(CN(C(C4(C)CS(=O)(=O)C4)=O)C2)CC3)cnc2nccn2c1 98460,c1(C(=O)NC)ccnc(CN(C2CCCSC2)C)c1 98461,C1(NC(c2ccc(Cl)cc2F)=O)CCC(O)CN(CC2CC(=C3CCC3)C2)C1 98462,c1(OC)ccc(C=CC(N2CC=CC(NC(=O)CSC(C)C)C2)=O)cc1F 98463,c1(CC(N2CCC(N(C(C=C(COC)C)=O)CCO)C2)=O)cccc2nsnc12 98464,Cc1cc(-c2cn(Cc3csc(C(F)(F)F)n3)nn2)ccc1N(C)C 98465,N1(C(=O)NC(C)Cc2cccc(F)c2F)CC(C)(C)CCC1CO 98466,C1(NC(CCN(C)CC)=O)CCN(C(C2(n3cnnn3)CCCCC2)=O)CC1OC 98467,Cc1sccc1C(=O)NCCN(C(=O)CCCc1cncs1)CC(C)O 98468,c1(C(COC(C)=O)NC(=O)CCN2CCCC(C(F)F)C2)ccc(F)cc1C 98469,C(C(C(=O)N1CCC(CN(C)C)C1)n1cc(-c2csnn2)nn1)OCC 98470,CC(C(=O)NCc1cccc(CNC2CCOCC2)c1)C(C)(C)C 98471,C(=O)(CCCCN(C)C(C)C)N(CCCN(C(=O)C(c1ccccc1)C)C)C(C)C 98472,C1(C)(C(C)(C)C)CC(C(=O)NCC(O)CNC(C2CSCCS2)=O)C1 98473,C1(NC(C2(CO)COC2)=O)CCC2CN(C(c3cc4c(s3)CCC4)=O)CC2C1 98474,C12CCCN(C1)C(=O)C(=O)N2.C1(C(C2CCC2)NC)CCC1 98475,Cc1c(NC(c2csc(C(=O)NC(C3CCOCC3)(C)C)n2)=O)cc(F)cc1Br 98476,N1(C(C(C)OCCCC)=O)CC(NC(=O)Cc2ncoc2C)C(C(F)F)C1 98477,C1(COC)CCCC1NC(=O)CC1(C)CCN1C(C)=O 98478,CCC(CC)(CC)C(=O)N(C)CCN(C(=O)CN1C(=O)NC(C)(CCC#N)C1=O)C 98479,c1(CC)cc(C(=O)NC2CC(NC(c3noc(CC)c3C)=O)C2)cc(C)c1 98480,C1(CNC(c2c(C(C)C)csc2)=O)CCCCN(C(=O)COc2ccsn2)C1 98481,C(C(C)CC(=O)N=c1ccn(C(C)C)[nH]1)NS(CCCC)(=O)=O 98482,N1(C(C2CCN(C(c3nc(C)c(C)s3)=O)C2)=O)CCC(C)C2(CCC2)C1 98483,C1(F)(CNC(c2c(CC)noc2)=O)CCC(CNC(=O)OC(C)(C)C)CC1 98484,C1(NC(c2c(C)n(C)nc2)=O)CC12CCN(C(C1CC3CCC3C1)=O)CC2 98485,n1(CCc2cc(C(N3CCC(CCC)(OC)C3)=O)on2)nc(C)c([N+](=O)[O-])c1C 98486,C1(C)(NC(Cc2c(CC)noc2CC)=O)CCCN(C(c2cnn(C)n2)=O)C1 98487,c1(OC)cc(C(=O)N(C(CNC(C2(CO)CCCCC2)=O)C2CC2)C)cnc1C 98488,C1(CNC(c2cc(OC)no2)=O)N(C(=O)Cc2cc(C)cc(F)c2)CCC1(C)C 98489,N1(C(C=NOC)=O)CC(F)CC1C(=O)NCc1cnc(S)nc1 98490,c1(OC)ncccc1C(=O)NCC(C)(C1CCC1)NC(c1ccoc1Cl)=O 98491,CCCCCC(O)CC(=O)NC(CN(C(=O)CC(C)C)CC)Cc1ccccc1 98492,c1(C(=O)NCC2N(C(c3c(Cl)ccc(C#C)c3)=O)CC2)coc2cc(F)ccc12 98493,C12(NC(c3cc(CN4CCOCC4)c[nH]3)=O)COCCC1CN(C(=O)C1CC1)C2 98494,C(=O)(C(C(C)C)n1cc(C)cn1)NC1(CNC(CCCNC(C)=O)=O)CCCC1 98495,c1(CNC(C(CC)n2ccnc2)=O)cnn2c1CN(c1nnc(C3CC3)s1)CC2 98496,Cc1ccc(N(C(=O)C(=O)N(CC(C)CNC(=O)CSC(F)F)C)C)cc1 98497,C1(NS(c2c(NC(C3CCOC3)C)nccc2)(=O)=O)COc2ccc(F)cc2C1 98498,N1(C(CCC)=O)CCCC(C(N2CCCC2c2cc(Br)cs2)=O)C1 98499,S(=O)(=O)(c1c(C)cc(C)cc1C)N1C(C(=O)N(CC)Cc2nccs2)CC(=C)C1 98500,c1(NC(C2CC3(CCN(C(=O)CCBr)C3)C2)=O)cc2c(Cl)cccc2s1 98501,c1(CC(C)Nc2c(C)n(C(C)C)nn2)ccc(Cl)c(-c2nn[nH]n2)c1 98502,N1(C(=O)C2=CCCCC2)CC2OCCN(C(C3CC3(F)F)=O)C2C1 98503,N1(C(CCC=CC)=O)CC(N=[N+]=[N-])CC1C(=O)NCCN1CC=CC1 98504,C(=O)(CCC1=NNC(=O)CC1)NC1CN(C(CN(CCC)C)=O)C2(C1)CCOC2 98505,CC(C)(C)C(O)C(=O)NC1CN(C(=O)CC23CCCN2CCC3)CC12CC2 98506,N1(C(C(=O)NC(C(=O)NCC)c2ccoc2)C)CCOCC1 98507,C1(C(=O)NCC(C)CNC(C2(n3cnnn3)CCOCC2)=O)(CC)CCCOC1 98508,N1(C(Cc2ccc(C)s2)=O)CCC2CN(C(C34CCC(=O)N3CCS4)=O)CC2C1 98509,C(=O)(CCCCNc1sccc1C(N1CC(N(C(C)=O)C2CC2)C1)=O)OCC 98510,c1(NC(N2C(C(=O)NC)CCOCC2)=O)cccc(S(F)(F)(F)(F)F)c1 98511,CCCC(CCC)=CC(=O)N(C(C)CCNC(=O)C(C)(C)n1ccc(C)n1)C 98512,CC(=O)C(C)CC(C)C(=O)NC1CC2(C1)CC2C(=O)NCc1cnn(C)c1 98513,C1(NC(C(CCSC)NC(C)=O)=O)C2CCC1N(C(c1ccsn1)=O)C2 98514,c1(C(=O)NCCN(C(C2CCN(CC)C2)=O)Cc2nonc2C)cccc(Cl)c1 98515,N1(C(CC(C)(C)F)=O)CCN(C(=O)C=Cc2nccs2)CC1C1CCC1 98516,C1(NC(c2c(CC)n[nH]c2)=O)CCC12CCCN(C(=O)CC1COCCN1C)C2 98517,c1(CC(=O)NC(C(=O)N(C)Cc2cn(CC)nc2)CO)ccc(C)cc1 98518,C1(C(N(C)Cc2cnc(CCC)s2)=O)CC(=O)N(OCc2ccccc2)C1 98519,N1(C(C(C)OCCC(C)C)=O)CC2CC(NC(c3coc(C(F)(F)F)c3)=O)C1C2 98520,c1(N2CCC(SC(F)F)C2)[nH]c(=NCc2cn(C3CCC3)nn2)nc2sccc12 98521,C1(N(C(=O)Cc2cnc(-n3cccn3)s2)C)CN(C(=O)Cn2cnnn2)CC12CC2 98522,C1(C)(C(=O)NCC#CCNC(C2(CC#C)CCCO2)=O)CNC(=O)C1 98523,C(=O)(CCC(=O)c1ccncc1)NC(C)(C)CNC(=O)Cc1cc(C2CC2)on1 98524,C(=O)(C(C)(C)CC(=O)N1C(C(=O)Nc2cncc(C(C)C)c2)CC2CC12)OC 98525,c1(C(=O)NCCN(C2CC2)CCF)cc(C2CC2)n(C)n1.C1(C(=O)C=O)CC1(Cl)C(F)F 98526,C1(F)(CNC(C2CCC(C)O2)=O)COCCN(C(=O)C2=C(C#N)CCC2)C1 98527,C=C(C)CC(C)(c1ccccc1)NCc1cc(C2CC2)no1 98528,C(=O)(CC(C)c1cccnc1)NCCCC1(NC(C(C)C)=O)CC1 98529,c1(C(C)NC(=O)Cc2nncs2)nc(=O)o[nH]1 98530,C1(C(=O)NC2(C)CN(C(N)=O)C2)(COC)CCCN(C(C2CCN(C)C(C)C2)=O)C1 98531,N1(CC(=O)NCCC2CC(NC(C3C(C)(CC)C3)=O)C2)CCCNC1=O 98532,C1(C(=O)NCC(c2cnccn2)(C)C)COC2(CCN(C(=O)CC3CC3)C2)C1 98533,N1(C(C2(SC)CC(=O)C2)=O)CC2CC1CN2C1CCCCC1 98534,C(=O)(C1=CC2C=CC(C1)C2)N1CCC(NC(c2scc(C)c2C)=O)C(C)C1 98535,c12ccc(cc1)NC(=O)C2.Cc1cnn(C)c1.C1(COC2CCC2)CCCC1.C(C)C 98536,N1(C(Cc2sc(C)c(C(C)C)n2)=O)CCCC(C)(NC(c2sccc2C#N)=O)C1 98537,c1(CC)cnn2ccc(CN3CCC(C(=O)O)C(C)C3)nc12 98538,c1(CC(=O)N(C2CN(C(=O)C=C3CCC3)C2)C)cccc2ccccc12 98539,N1(C(c2ccc(C(C)=O)o2)=O)CCCC(NC(=O)CCOC2COC2)C1C 98540,C1(C(N2C(C)CC2)=O)CCCC(NC(=O)COCC2CC2)C1 98541,C1(C2(O)CCC2)(CNC(CC2(C)N(C(C=Cc3ccc(C)o3)=O)CC2)=O)CC1 98542,CC1=NS(=O)(=O)N(C)C=C1C(=O)NC12CC(C1)N(C(=O)C=CC1CCOC1)C2 98543,N1(C(CC(C)OC)=O)CC2CC(NC(=O)Cc3ccnc(Br)c3)C2C1 98544,CCCC(C(=O)NCCOC(=N)O)NC(=O)CCOC1CCCC1 98545,C(=O)(C(O)CC(F)(F)F)N1C(C(=O)NCCCOCCCC)(COC)CCC1 98546,c1(OCC#C)ccc(CCCN(c2cccc(Br)c2)C2CCC2)cc1.C(=O)OC 98547,Cc1nnc(Br)cc1C(N1CCCC(O)(CNC(C2CC23CCC3)=O)C1)=O 98548,c1(C(N2CC(CC(=O)NCC3C(CCC)C3)C(C)C2)=O)cn2c(n1)CCC2 98549,N1(C(CC#C)=O)CCC2(CCCN(C(c3cc([N+](=O)[O-])ccc3I)=O)C2)CC1 98550,S(=O)(=O)(c1ccc(C#N)cc1)NC(CC)C(=O)N(CC)CC1CCCO1.O 98551,C(CCCCC(=O)N1CC(C(N2CCOC(SC)C2)=O)(CC)C1)OCC 98552,C=CCCCCCC(=O)NCC(C)(CC)NC(C1CNC(=O)N1C)=O 98553,CC1CCCC=C1C(=O)N1CCCC1C(C)(C)CNC(=O)CCCC(F)(F)F 98554,C1(C(N2CC(NC(c3c(C)cc(F)cn3)=O)CC2(C)C)=O)CC2(CCC2)CCO1 98555,C1(C(=O)NCC2COCCN(C(C(C)O)=O)C2)C2CC3CC(C2)CC1C3 98556,c1(COC(=O)NCC(=O)Nc2ccc(C(F)(F)F)cc2)ccccc1Br 98557,C1(C(=O)NCC2(CCNC(C(CN(C)C)N(C)C)=O)CC2)CC(=O)N(O)C1 98558,C=CC(C)(C)CC(=O)NCC1(C(=O)NC(C(C)(C)O)C2CC2)CCCC1 98559,C=CC(CCC)CC(=O)NC1CN(C(=O)Cn2nc(C)c(C)c2C)CC(F)(F)C1 98560,C(=O)(C(C)CC(C)(C)C)N(CCCC(N1CCN(C(=O)CSC2CC2)CC1)=O)CC 98561,C(CC1c2ccccc2CN1C(c1ncc(C)cc1C)=O)NC(CCC=C)=O 98562,C1(C(N(CCC(C)NC(C2N(CC)CCCC2)=O)C)=O)CCC2(CCCC2)CC1 98563,N1(C(COC)=O)CC(CNC(c2cc(C(N)=O)[nH]n2)=O)N2CCC1C2 98564,c1(CC)cc(C(=O)NCCC2CCN(C(=O)CCC3(C)CC3)C2)c(C)o1 98565,N1(C(CSCC=C)=O)CCCC2(CNC(c3ccns3)=O)CCCC12 98566,n1(N(C)C)nc(C(F)F)nc1-c1ccn(-c2ccc(C(F)(F)F)cc2)n1 98567,c1(C(=O)NCC2N(C(C=CC)=O)CC(C)(C)CC2)cc(Br)cc([N+](=O)[O-])c1C 98568,c1(OC)ccc(C(C)C(N2CCCC2CNC(=O)CC2(C(F)F)CC2)=O)cc1F 98569,c1(C(N2CC3CC(NC(C4(COC)CC4)=O)C3C2)=O)ccc2ncnn2c1 98570,c1(C(=O)NC2(COC)CN(C(CCCOC)=O)C2)sc(C(C)C)nc1C 98571,c1(CCCC(=O)NCC(O)CNC(c2ccccn2)=O)ccccc1F 98572,C(=O)(C(CC(C)C)N(C(C#CC)(C)C)C)Nc1sccc1C 98573,C(=O)(C(C)(C)CCCF)NCC1(C)CCC(NC(CN(CC)CC)=O)C1 98574,C(=O)(C1CC(=O)Nc2ncccc21)N(CCCNC(=O)C1CCc2nccn21)C 98575,C(CC(C(C)C)NC(=O)CCc1cncc(O)c1)NC(c1c(C)cns1)=O 98576,C(=O)(CCC(C)(C)F)NCC(CC)NC(c1ccc(F)cc1)=O 98577,C1(COC)CN(C(=O)C(c2ccnn2C)O)CCN1C(c1cc(Cl)cs1)=O 98578,C1(C#N)(C(=O)NCc2ncc(C(N3C(C=C)CCC3)=O)cn2)CC(F)(F)C1 98579,c1(C(=O)NCC(CNC(CCN(C)CCO)=O)O)c(F)c(F)cc(O)c1F 98580,c1(C(=O)NCCCCNC(C(C(=O)OCC)CC)=O)ccccc1[SH](=O)=O 98581,C1(COC)(OC(c2cc(C(=O)Nc3ccccc3)on2)=O)CCCS(=O)(=O)C1 98582,c1(C(=O)NC(C2(O)CCN(C(c3c(C)nn[nH]3)=O)CC2)C)nnn2ccccc12 98583,CC1CC(=O)NCC1C(=O)NCC1CCCN1C(c1csc(-c2ncc[nH]2)n1)=O 98584,c1(NC(C(C(C)(C)C)NCC#CC2CC2)=O)ccc2c(c1)CCC2 98585,N1(C(COCCNC(c2c(C)cns2)=O)=O)CCC2CN(C)CC12 98586,C1(C(=O)OCC(=O)OC(C)(C)C)CNC(=O)CC12CCN(S(C)(=O)=O)CC2 98587,c1(C(C(=O)NCCN(C(CC(C)OC)=O)C2CC2)(C)C)ccc(Cl)nc1 98588,C1(NC(C2C(=C)C2)=O)C2CC(O)C1N(C(c1ccccc1-c1ccncc1)=O)C2 98589,c1(C(=O)NC(CNC(C(C)C(C)(F)F)=O)CO)cnc(N)c(Cl)c1 98590,C1(CNC(COCCNC(C(C=C)OC)=O)=O)CCCC12CCC2 98591,C(=O)(C(C)(C1CCCCC1)NCCCOC(=O)C1CC1)OC 98592,N1(C(C2(CC#C)CC2)=O)CC2COCC2(C(=O)NCCCc2cnn(C)c2)C1 98593,C1(CCNC(CC(C)c2ccncc2)=O)CCCN(C(=O)C(F)=CC2CC2)C1 98594,C12(C(=O)Nc3nc(-c4ccc(C)cn4)sc3)CCC(N)(CO1)C2 98595,C1(CCC(=O)NC2CC(N(C(c3ccc(CSC)o3)=O)C)C2)C(=O)NN=C1C 98596,c1(C(=O)NCC(C)N(C)Cc2ccc(C)nc2)n[nH]c2c1CCOC2 98597,Cc1cnccc1C=CC(=O)NC1CCCC(NC(c2c(C)nn(C)c2Cl)=O)C1 98598,Cc1oc(Br)cc1C(=O)NC1CC2(C1)CC2NC(=O)CN1CCCNC1=O 98599,N1(C(c2ccc(CC)cn2)=O)CC(CC(=O)NC2(C(N)=O)CCC2)CC1(C)C 98600,CC1C(NC(=O)CN(C2CCCC2)CC)CCCN1C.C(=O)(CCC1CCCN1)N 98601,C(c1c(Cl)nc2sccn12)=CC(=O)NC(c1ccccc1C)C(=O)OC 98602,C(C)(CN=c1[nH]c(Cl)ncc1C1CC1)NC(C(C)Sc1cc([N+](=O)[O-])ccc1Cl)=O 98603,c1(C(=O)NCC2N(C(C(C(C)C)O)=O)CCN(C)C2)cccc2c1COC2 98604,C1(CNC(c2ccsc2F)=O)CCC(NC(c2[nH]nnc2C2CC2)=O)C1 98605,C(CNC(c1ccccc1)C1(O)CC1)(CC(F)(F)F)NC(C(C)CC1CC1)=O 98606,c1(CNC(c2n(CCSC)nnn2)c2cscc2C)ccncc1Cl 98607,CC1CCN(C(C2(CO)COC2)=O)CC1NC(=O)CC(F)(F)Br 98608,c1(OC)ccc(C)c(C(=O)N(C2CCN(C(=O)CCC(C)SC)C2)C)c1 98609,c1(CC)ccc(F)cc1C(=O)NCCCC1CCCCN1C(c1[nH]ccc1C)=O 98610,C1(CCC(=O)NC(C)C(=O)NCC(C2CCOC2)OCC)(N(C)C)CCCCC1 98611,c1(C(N2CCC(C(C)(C)NC(C3N(C(C)C)CCC3)=O)C2)=O)ccc(CO)cn1 98612,c1(CC)ccc(C=CC(=O)NC2COCCN(C(=O)CC3CC(F)C3)C2)cc1 98613,c1(CC(=O)NCC2N(C(C(C)SC)=O)CCCCC2)coc2ccc(F)cc12 98614,CN1CC(O)CCC1C(N1CCCCCC1C(=O)NC1CCCC1C(C)(C)C)=O 98615,C1(N(C(C=CCCC)=O)C)CCN(C(c2cc(Cl)ncc2OC)=O)CC1C 98616,CC1(C)CC(C(=O)NC2CC(C)(NC(C3CCC(=O)NC3)=O)C2)CCO1 98617,C1(NC(C2(SC)CN(C(C(CCC)CC)=O)C2)=O)CC(C)(C)OC1(C)C 98618,CC(C)(O)C(C(=O)NC1CCCC1O)NC(c1cnn(C2CC2)c1)=O 98619,C(C(C)CC(=O)NCC1(n2ccnc2)CN(C(C2(CC(C)C)COC2)=O)C1)OC 98620,N1(C(C(C)C(F)F)=O)CC(C2CC2)(C(=O)NCC2(C#N)CCC2)C1 98621,C=C(C)CC(C(=O)N1CC(NC(c2cn(C(C)C)cn2)=O)C1)NC(C)=O 98622,N1(C(C(C)OCC(C)C)=O)CC(NC(c2coc(Cl)n2)=O)CC12CCCCC2 98623,C1(CC)(NC(=O)CSc2ccc(C)cc2)CCN(C(C2CC3CC3C2)=O)CC1 98624,C(=O)(CCCN(C)C(=O)NC1CC(=C2CCC2)C1)OCC1CCCN1C(N)=O 98625,c1(CN(C)CCC2CCC2)ccn(CC(=O)NCC(=O)NCC2CC(CF)C2)n1 98626,N1(C(=O)CC2CCC3CC23)CCOC2(CCCN(C(c3ocnc3C3CC3)=O)C2)C1 98627,c1(C(C(=O)NCCOC)N(CC=C)C)ncc(Cl)n1C 98628,C12(CC(=O)NCCCCCN(C)C(C3C4CCC(=O)C34)=O)CCCCC1C2(F)F 98629,Cc1n[nH]c(C)c1CCCNC1CCN(c2ccnc(N3CCC3)n2)C1 98630,C(=O)(CC(c1ccccc1)C1CCCCC1)N(C1CCCNC1)C(=O)C(N)CO.CC 98631,c1(C(=O)NC2(CNC(C(C)N3CCC3)=O)CCCC2)c(Cl)c([N+](=O)[O-])nn1C 98632,C12(C(=O)NC3CCCCN(C(c4cccc(C)n4)=O)C3)CCC(CO)(CC1)CC2 98633,N1(C(c2nn(CC)c(C)c2)=O)CCC(N(C)C(c2cc(OC)nn2C)=O)C(C)C1 98634,N1(C(Cc2cccc(SC)c2)=O)CCN(CC2(C(=O)N(C)C)CC2)CC1C 98635,C1(C(=O)OCC(=O)C2CC2C(F)F)CSC(c2ccccc2O)=N1 98636,N1(C(CC=C)=O)CCC2(CCCC2C(=O)NCc2cccc(C#N)c2)C1 98637,Cc1ccc2c(C(=O)NCC3(F)CC(NC(C4CCC4(F)F)=O)C3)cnn2c1C 98638,c1(C(=O)NC(C)CN(C(=O)CC(C)CN(C)C)C)ccc2oc(N(C)C)nc2c1 98639,c1(C(=O)NCC(CNC(C2CCC(=O)N2)=O)CO)c[nH]c(=O)c2ccncc12 98640,c1(N2CCC(CC(=O)Nc3cc(OC)ncc3)CC2)ccnc(S(C)(=O)=O)n1 98641,C1(N(C(=O)CCOCCN(C)C)C)CN(C(c2cc(F)cs2)=O)CC1F 98642,c1(OCCC(N2CCCC2CCNC(C2(c3cnno3)CC2)=O)=O)ccccc1 98643,c1(NC(C)=O)ccc(C(=O)N(CC(O)CNC(=O)C(F)n2ccnc2)C)nc1 98644,c1(C(=O)NC2CN(C(c3nn(C(CC)C)c(C)c3)=O)CC2C)cc(Br)ccc1O 98645,c1(CC)cnc(C(=O)NCC2CC2NC(c2cccnc2C)=O)cn1 98646,c1(C2(C(=O)NCCN(C(c3cn(CCC=C)nn3)=O)C)CC2)ccc(F)cc1Cl 98647,N1(CC(=O)NC(C2(O)CCN(C(c3ccns3)=O)C2)C)CCC(F)CC1 98648,c1(C(=O)Nc2ncncc2-c2c(F)cccc2F)cccc2scnc12 98649,N1(C(c2cn(C)[nH]c2=N)=O)CCCC(NC(C2(CO)CC(F)(F)C2)=O)CC1 98650,N1(C(Cc2c(C)ccnc2)=O)CC(F)(F)CC1CNC(C1CCCOC1)=O 98651,c1(C(=O)NCC2(F)CCN(C(C(=CC3CCCC3)C)=O)C2)cccn2cncc12 98652,c1(C(=O)NC(c2ccccc2)C(C)NC(C=CCOC)=O)cnc2sccn12 98653,C1(F)(C(=O)Nc2nccnc2Br)CCN(C(c2occc2Br)=O)CC1 98654,N1(C(C(F)OC)=O)CC(O)(CCNC(c2ccncn2)=O)C1 98655,C1(C(=O)NCCCN(C)C(C2C(Cl)(Cl)C23CC3)=O)CCc2ccccc2C1 98656,N1(C(=O)Nc2c(CC)ccc(C(F)(F)F)c2)Cc2ccccc2SCC1C 98657,c1(NC(C2(F)CN(Cc3ccc(O)c(Br)c3)C2)=O)nc2ccccc2[nH]1 98658,N1(C(c2c(C)n(C)cc2)=O)CCN(C(C2CCCO2)=O)C2(CCC2)C1 98659,C(=O)(CC1CCc2ccccc21)NCCN(C(C=CSC)=O)C1CCCCC1 98660,N1(c2cc(NCC3CC(CC(C)(C)C)C3)nc(COC)n2)CC2CC(F)CC2C1 98661,c1(N(C(CCNC(C(C(C)C)N(C)C)=O)C)C)nc(C(C)(C)C)nc(=N)[nH]1 98662,C1(C(=O)NC)CN(C(=O)OC)CCN(C(=O)CC2(C)CCC2)C1 98663,C1(C(=O)NC2CN(C(C3C(C)C3c3ccccc3)=O)C2)CCc2nn[nH]c2C1 98664,C(=O)(CCC(C)(F)F)NCCNC(=O)CN(C)C(C1(OCC)CCC1)=O 98665,N1(C(c2cncc(N)c2)=O)CCCC(C2(NC(C3(CF)CC3)=O)CC2)C1 98666,C1(C(N2CCC(N(C)C(C3CCCS3)=O)CC2)=O)CCC12CCNCC2 98667,c1(C(=O)NCC2(OC)CN(C(C(CC)O)=O)C2)nc2n(c1C(C)C)CCCC2 98668,C(=O)(CCCCNC(=O)CC12CCCC1C2)OCC1(C)CSC1 98669,C(CCN(C)C)(C(=O)NCCOC)NC(C(C)OCCC=C)=O 98670,Cc1ccc(F)c(C(=O)NC2CCC(N(C)C(c3cccnc3)=O)CC2)n1 98671,C(=O)(CCCC(=O)C1CC1)C(N(C)CC1(CNC(=O)Cc2cc[nH]n2)CC1)=O 98672,c1(C(=O)NC2(C)CC(NC(c3c(C)cn(C)c3)=O)C2)cc2c(s1)CC(C)CC2C 98673,S(=O)(=O)(c1cc(C)ccc1C)NCCC(=O)N(C1CCNCC1F)CCCC 98674,N1(C(C(=O)NC2Cc3c(cn(C)n3)CC2)=O)CCS(=O)(=O)Cc2ccccc21 98675,C(=O)(C(C(C)(C)C)n1cc(CCS(N)(=O)=O)nn1)NC(CCCc1c(C)ccs1)=O 98676,c1(NC(=O)NC2CC3(CSC3)C2)c(Br)cnn1CC1CC1 98677,N1(C(C2N(C)C(=O)OC2)=O)Cc2ccccc2C1CNC(C1CCCCC1)=O 98678,c1(C(N2CCCC(C(C)NC(=O)COC(C)(C)C)C2)=O)cc(C#N)cn1C 98679,CC1C(NC(=O)C(C)(O)C2CC2)CC2CCC1N2C(c1cc(Br)c[nH]1)=O 98680,Cc1ccc(C(C)(C)C(N2CCC(C)(NC(=O)CC(C)O)C2)=O)cc1 98681,CCC(C)(C)CCCC(=O)N1CCCC1CNC(C1COCCO1)=O 98682,Cc1[nH]nc(C(N2CCCC2C2(NC(C3CSCN3C)=O)CC2)=O)c1[N+](=O)[O-] 98683,CN1CCCC1CC(N1CC(CN(C(C2(C3CCCCO3)CC2)=O)C2CC2)C1)=O 98684,C(=O)(CCCC(C)(C)CC)N1CCC(CCNC(c2nc(CC)oc2)=O)(CO)C1 98685,N1(C(C(CCCCC)C)=O)CC2(C=C(C(=O)Nc3cccc(C)n3)CO2)C1 98686,C(=O)(C(O)CCC(C)C)NCCN(C(=O)CN1CC2CCC1C2)CCC 98687,CCC(CC(=O)NC(C)CN(C(=O)CC1(OC)CCC1)C)c1ccccc1 98688,c1(OC)ccc(OC)c(C(=O)NCC2CCN2C(=O)Cc2c(F)cccc2F)n1 98689,CC1CCCN(C(c2ncccc2C(C)(C)C)=O)C1CNC(c1cnc(Cl)s1)=O 98690,C=CC(C(=O)NC(CNC(=O)CN(C)C1CC1)CCCC)OC 98691,C(=O)(CC(C)C(=O)NC1CC(CNC(=O)CC2(CO)CCOCC2)C1)OC 98692,C1(C(=O)NCc2ccc(C(=O)NC(COC(C)C)(C)C)o2)COC(=O)N1C 98693,c1(C(=O)NCC(O)CC(N2CCCC(O)(CC3CC3)C2)=O)ccn2cncc2c1 98694,C1(CNC(CC2(N(C(=O)CCc3cncnc3)C)CC2)=O)CC12CCOCC2 98695,Cc1ccccc1-n1ccc(C(=O)NC(C)CCNC(=O)CSC2CC2)n1 98696,c1(CC(=O)NCC(CNC(=O)CC2(C(F)(F)F)CC2)F)ccsc1Cl 98697,C1(NC(CC(CC)C)=O)CCc2nc(NC(=O)C(C)CC(N)=O)sc2C1 98698,N1(Cc2cc(OC)cc(F)c2)CCn2c(cnc2Br)C1.c12ccccc1C(=O)N2 98699,c1(CN2C(c3c(C4(CO)CC4)ccnc3F)CCC2)cccc2[nH]ncc12 98700,N1(C(C(CCSC)NC(=O)OC(C)(C)C)=O)CC2CCC1CN2C(c1ccon1)=O 98701,N1(C(C2CCC(NC(c3ccc(C4CC4)cc3)=O)C2)=O)CC2CCCCCC2C1 98702,c1(CC(N2CC(NC(CCN(CCC)C)=O)C2)=O)cc(C(F)(F)F)cc(F)c1 98703,C1(CC)CN(C(=O)C=C(C)c2cccs2)CCC1NC(=O)CCc1ccncn1 98704,N1(C(c2ccc(CC)s2)=O)CCCC2(NC(c3cccc4cnnn34)=O)CCCC12 98705,c1(NC(C(C)OC(C(CCOC)C)=O)=O)c(F)cccc1F.C1CC(=O)O1 98706,CCCC(C)(O)CC(=O)N(CCNC(C1CCN(CC)C1)=O)CCOCCO 98707,c1(C(=O)NC(c2nc[nH]n2)C)conc1CNC(=O)CCc1cncn1C 98708,[N-]=[N+]=NC1CC(C(=O)NC2CC3(CCCO3)C2)N(C(c2ccc(F)cc2F)=O)C1 98709,C(c1ccc(C)cc1C)=CC(=O)NC1C2CCN(C(c3ncn(CC)n3)=O)C21 98710,c1(C(N(CC)Cc2cccs2)=O)c(Br)nnn1C 98711,C(CC(C(=O)N(C)CC1CCN(C(c2[nH]ccc2C)=O)C1)N(C)C)SC 98712,c1(N(C)C)cncc(C(=O)N(C2CC(NC(c3c[nH]cc3Br)=O)C2)C)c1 98713,Cc1cc(N(C)C)cc(C(=O)NCC2CCN(C(c3ccc(Br)c(Cl)c3)=O)C2)c1 98714,N1(C(c2n(C)nnc2)=O)CCCC(C(=O)NC2(C(C)(F)F)CC2)C1 98715,N#Cc1ccc(CNC(=O)C(=O)NCc2sc(Cl)cc2Cl)nc1 98716,C1(NC(C(CC)F)=O)CC2CCC1N2C(=O)COCC1CCOC1 98717,c1(C(=O)NC2(CO)CCCN(C(C(C3CC3)SC)=O)C2)cccc2[nH]ncc12 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99062,C1(C(=O)NC(CNC(CCc2onc(C(C)C)n2)=O)(C)CO)CCN(C)C1C 99063,C1(NC(=O)CONC(C2CCCCC(=O)N2)=O)CCCCCC1CO 99064,c1(CCC)cc(C(=O)N(CCC(C)NC(=O)C(C)Cc2ccncc2)C)n[nH]1 99065,C#CC1CCC(C(N2CCCC(F)(CNC(C3OCCC3CC)=O)C2)=O)CC1 99066,CCC1=C(C(=O)NCCC(C)(C)NC(=O)CCc2ccco2)CCCO1 99067,C1(CC(=O)NCC2N(C(c3ccc(C)s3)=O)CC=C2)COC2CC1C2 99068,Cc1cc(C(N2CC(NC(c3nc(O)c(C)s3)=O)C3CC23)=O)n2nc(C)cc2n1 99069,N#CCC(CC(=O)NC1CCCC1NC(C1(O)CCOCC1)=O)c1ccccc1 99070,c1(NC(=O)NC)ccc(C(=O)NCC2CCCC2NC(C2(CC)COC2)=O)cc1 99071,C1(NC(C(C(=C)Cl)(C)C)=O)CCC2CCN(C(=O)CCNC(=O)OCC)C1C2 99072,C1(C)(CNC(C(COC)C)=O)CCC(NC(c2ccncc2C(F)F)=O)C1 99073,c1(C(=O)NC(CC)(C)CNC(=O)C(C)NC(c2cccs2)=O)sc(CO)nc1C 99074,C1(C(=O)OC)CC12CCN(C(=O)CC1(C)CN(C(=O)Sc3ccccc3)C1)C2 99075,N1(C(C=CC(=O)OCC)=O)CCC(C(=O)NCC2CCSC2)(CC)CC1 99076,Nc1cccc(C=CC(N2C3CCC2C(CNC(=O)COC2CC=CC2)C3)=O)c1 99077,C(=O)(C1Cc2ccccc21)N1CCC(C(=O)NCC(C)CO)CC1(C)C 99078,c1(C(N2CCC(C(C)NC(C3CCN3C)=O)C2)=O)ccc(CC(N)=O)cc1 99079,c1(C(=O)NC(C)CCCNC(C2COCCO2)=O)cnc2c(F)ccc(F)c2c1 99080,CC(C)(C)CC(=O)N1CC(NC(C2(c3cncc(Br)c3)CC2)=O)C2CC12 99081,N1(C(c2ccc(C(=O)NC)cc2)=O)CC(N(C)C(c2conc2C)=O)C2(CC2)C1 99082,N1(C(Cc2cccc(COC)c2)=O)CCN(C(c2nc(O)sc2C)=O)C2CC12 99083,N1(C(CC(C)n2ccnc2)=O)CCCCC1CNCc1cnn(-c2nccs2)c1 99084,c1(C(=O)NC2CC(CNC(CN3C(C)CC3)=O)C2)cc(F)ccc1N1CCOCC1 99085,Cc1cccc(C2=CCN(C(=O)NCC3C(CN)C3(C)C)CC2)c1 99086,C(CN=c1nc(O)c(Cl)c[nH]1)NCc1ccc(Cl)cc1Cl 99087,N1(C(CC2C=NN(C)C2=O)=O)CCC(C(=O)Nc2cnc(Cl)nc2)CC1(C)C 99088,CC1COc2c(C(=O)NCC=CCNC(=O)Cn3[nH]cnc3=N)cccc21 99089,c1(C(N2CCCN(C(CC(C)C3CCCO3)=O)CC2)=O)ncccc1N=[N+]=[N-] 99090,C(CC(=O)N1CC(OC)CC1CNC(c1cc(C)ccc1C)=O)(C(C)C)NCC 99091,C(=O)(C1=C(Cl)CCOC1)NCC12CN(C(C(CCC)OCC)=O)C(C1)CO2 99092,C1(NC(C(OC)OC)=O)CCCC(CNC(=O)C(C)(C2(C)CC2)N(C)C)C1 99093,c1(C(C)NC(N2CCCN(CCO)CC2)=O)cc(OC)c(OCC2CCCO2)cc1O 99094,N(C(=NCCc1cccs1)NCCCN1CCCC1)C(c1nn(C)cc1C(F)F)C 99095,c1(C(=O)OCc2ccc(C)c(Cl)c2)cc(P(C)(C)=O)n(C)c1 99096,CCC(CC(F)F)C(=O)N1CCCC1C(=O)NC1(c2ccc(F)cc2)CC1 99097,CS(=O)(=O)CC(F)(F)CCNC(=O)Nc1nn[nH]c1C(F)(F)F 99098,N12CCC(C)(C)C1CC(=O)N(CC(=O)OC)C(CC#C)C2=O.C(C)(C)OCC 99099,c1(C(N2CCC(NC(C3CCCS3)=O)C2)=O)cc(F)c2cc[nH]c2c1 99100,N1(C(CC(=O)OC)=O)CC(NC(=O)C(C)c2ccco2)CCC1C 99101,c1(COC)nn(C)cc1C(=O)N(CCNC(c1cc(C)n(C)c1)=O)C1CC1 99102,N1(CC(=O)NCCCN2CCN(C(C(CC)(C)O)=O)CC2)C(=O)NC(C)(C)C1=O 99103,C(=O)(C1=CC2(CCOC2)C1)N(CC(C)(C)CNC(=O)CCCn1ccnc1)C 99104,CC(C)(CCCCNC(c1csc2cncn12)=O)NC(=O)CCN1CCCCC1 99105,CC(C)C(C)C(CNC(c1ccnc(F)c1N)=O)NC(=O)CCCCNC(N)=O 99106,S(=O)(=O)(c1ccc(Br)cc1SCCCCCCCC)N1C2CC(=C)C(C2)C1 99107,C1(NC(CCSC)=O)COCC1NC(C1CN(C2CCOC2)C1)=O 99108,N1(C(C(CCC#C)O)=O)CCCN(C(c2cnoc2C)=O)C(C(C)C)C1 99109,CC(C)(O)C(F)CNC(C1(C2CCCN2C(C2CCCO2)=O)CC1)=O 99110,CC1CC(C(N2CC(NC(C3C=CC(NC(=O)OC(C)(C)C)C3)=O)C2)=O)CC(C)C1 99111,CC1C(NC(c2cnccc2Br)=O)C(C)CCN1C(c1coc(N(C)C)n1)=O 99112,c1(OCC)ccc2c(c1)C(NC(=O)NCCNc1nc(C)cs1)CCO2 99113,N1(CC(=O)NCC(=O)N(C)CCN(C)C(c2ccccn2)=O)CCCCS1(=O)=O 99114,c1(C(=O)NCCCCCNC(=O)Cc2cncs2)cnn2c1CCC2 99115,c1(C(=O)NC2(C)CCN(C(C34COCC3C4)=O)CC2)ccc(Cl)c([N+](=O)[O-])c1 99116,C1(NC(c2cc(C)oc2)=O)CCCCN(C(C2CC(OCC(C)C)C2)=O)C1 99117,CCC(C)(O)C(=O)NCCCN(C(=O)CCC1CC(C)(C)CO1)C1CCCC1 99118,CC(C)CCCC(C)CNC(=O)CC1CCCN(C(=O)CC(C)N(C)C)C1 99119,N1(C(c2c(Nc3ccccc3)cnc(Cl)c2)=O)CCCC2(CCC2O)C1 99120,c1(-n2c(C(c3n(CC#C)ccn3)NCC3CC(O)C3)nnn2)ccc(Cl)cc1F 99121,Cc1ncc(Br)c(N2CCOC(CNC(c3sccc3Cl)=O)C2)n1 99122,c1(CNC(C(=O)NCC)=O)ccc(Oc2cc(F)cc(Br)c2)c(F)c1 99123,Cc1csc(Cl)c1C(=O)NCC1CC1CNC(=O)CNS(=O)(=O)C1CC1 99124,N1(C(C2(SC)CN(C(CC(CC)O)=O)C2)=O)CCOC(C)CC1 99125,c1(COC)cncc(C(=O)N(C(C)CN(C(=O)CCc2cncs2)C)C)c1 99126,c1(CC)cc(C(=O)NCC(C)(C2CCC2)NC(c2cc(C)[nH]n2)=O)ccc1O 99127,CC1SCCCC1C(N1CCC2CC12C(=O)NCCNC(=O)CO)=O 99128,Cc1cn2ccc(C(N3CCC(Cc4cn(CCO)nn4)C3)=O)cc2n1 99129,N1(C(C2ON=C(C)C2)=O)CCN(C(c2ccnc(SC(F)(F)F)c2)=O)C(CF)C1 99130,Cc1nc(Cl)ncc1NC(C1CCCN(C(C2CC(C)(C)C2)=O)CC1)=O 99131,N1(C(C(C)S(N)(=O)=O)=O)CC(NC(=O)C(F)(F)C2CC2)CC12CCCCCC2 99132,C(c1ccccn1)=C(C)C(=O)NC1CCC(C)(CNC(c2ccns2)=O)C1 99133,c1(C(=O)NC(C)C(=O)NC(C)CC2(O)CCC2)sccc1SC(C)(C)C 99134,CC1CCN(C(c2ncsc2C2CC2)=O)CC1NC(=O)CSc1cn[nH]c1 99135,C(=O)(C(C(=O)NCCN(C(=O)CC1(O)CCOC1)CC)OC)OCC 99136,C=C(C)CC(C(=O)NCC1(C)CNC(=O)O1)NC(=O)Cc1cnnn1C 99137,N1(C(C)C)CC(C(=O)NCCN2CCC2)(C(=O)N)C1.C1(OC(C)C)CC1C=O 99138,C1(NC(c2cnn(C)c2Cl)=O)CCN(C(=O)COc2ccon2)CCC1(F)F 99139,c1(C(=O)NCCCCNC(C(n2ncc(C)c2)C)=O)cnc(O)cc1C 99140,C1(C(=O)OC)CCC(F)(F)CN1C(=O)NCC(c1ccccc1F)N1CCCC1 99141,C1(CNC(C(COC)OC)=O)CCCC2(CN(C(=O)C(CC(C)C)OC)C2)O1 99142,S(=O)(=O)(c1c[nH]ccc1=NC(C(C)(C)C)C[N+](=O)[O-])NC1CN(C)C(C)(C)C1 99143,C(=O)(C1c2c[nH]nc2CN1C(C1CCC1C)=O)N1CCCC(C)(OC)C1 99144,N1(C(C(C)n2ccnc2)=O)CC2CCC(C1)N(C(=O)CCc1cc(F)ccn1)C2 99145,N1(C(C(C)CF)=O)Cc2ccccc2CC1CNC(=O)C(c1ccccn1)O 99146,N1(C(CCc2[nH]c(=N)sc2)=O)CCC2(CCCN2C(=O)CC2CCCC(O)C2)C1 99147,c1(OCC)cc(C(=O)NCC(C)NC(=O)C(C)NC(C2CCC2)=O)[nH]n1 99148,C1(C(N2C(CO)CC(NC(C3C4COCC34)=O)C2)=O)CC2C=CCC(C1)C2 99149,Cc1c(C(N2CC(NC(C3CN(C)C3)=O)C(O)C2)=O)c(Cl)nn1C 99150,C1(CNC(C(c2cccnc2)OC)=O)CCN(C(=O)C(C)(C)CO)CC1C 99151,CCC1=NOC(C(=O)N(C2(C(=O)NC3CCNC(=O)C3)CCC2)C2CC2)C1 99152,C(CC(C)OC(=O)NC1CCCC1)OCC.C1(=O)CO1 99153,N1(C(CC(C)(C)SC)=O)C2CCC1CC(N(C)C(C1CC3CCC(C1)C3)=O)C2 99154,C(=O)(CC(COC)NC(=O)CCc1cccn1C)NCC1CC(CC)C1 99155,C1(OCCNC(CC2(SC)CC2)=O)CCN(C(c2cncnc2)=O)CC1 99156,C(=O)(CCC(C(C)O)NC(c1ccc(Br)cc1F)C(=O)Cc1ccccc1)OC 99157,C123CCC(C1)N(C2)C(=O)C(C(C)C)N(NC(C(C)=C(CC)C)=O)C3.CC 99158,CC1CN(C(c2cnc(C(F)(F)F)nc2)=O)CCCN1C(C1CC(C)(F)C1)=O 99159,Cc1ccc(S(=O)(=O)NC(c2cccc3nnn(C(C)(C)C)c23)=O)cc1C(=O)O 99160,N1(C(CN(C(C(C)C)=O)C)=O)CCC(CNC(=O)C(C(C)C)N(C)C)C12CC2 99161,C(=O)(CCCC(C)(C)C)N1CC(CCC)N(C(c2cc(CCCO)on2)=O)CC1 99162,C1(C(C)NC(C(CC)SC)=O)CCCN1C(C1(CO)CCCCC1)=O 99163,c1(C(N(CC(CC)NC(c2nc(=N)cc[nH]2)=O)C)=O)ccc(NC)c(F)c1 99164,Cc1nc(Cl)nc(N2CC=C(CNC(c3cc(Cl)cnc3C)=O)CC2)c1[N+](=O)[O-] 99165,Cc1c(C(=O)NCC2CC2NC(=O)CCn2cnc(=N)[nH]2)[nH]c2c1CCCC2 99166,c1(C(=O)NCC(C)N(C(C2CCC(C)O2)=O)C)nc(C(C)C)ncc1Br 99167,C(C)(CC(C)(C)C)(c1nnnn1C(C)(C)C)NCc1nccc(C)c1 99168,c12ccc(cc1)CNC2=O.N1(CCC#N)CCCC1CN1CCCC1 99169,c1(C(C)=O)c(NCc2ccc(F)c(Cl)c2F)c(C#N)cn1C 99170,CC(C)C(C)(O)CNC(=O)C(CC1CCC1)NC(=O)CC1CCCCO1 99171,c1(CC)cnc(C(=O)NC(c2cccc(C)c2)CNC(=O)C(=O)C(C)C)nc1 99172,n1(CCC(=O)NC(CN(C(C(C2CCCC2)OCC)=O)C)CC)ncn1C 99173,Cc1cc(C(c2nc(C(C)C)no2)C)ccc1Br.SC