SMILES O=C(CC=Cc1ccccc1)C(=O)c1sccc1Br C12(C(=O)NCCCC(C)NC(c3ccc(OC)cc3)=O)CCCC1C2(F)F c1(C(N(C)C)=O)ccc(C(=O)N(CCNCC(=O)NCC(O)CF)C)cc1 C1(NC(C2CC(SC)C2)=O)CCC2(CC1)CCCN(C(=O)CCN(C)CCO)C2 C1(C(N2CCOC(C)(CNC(C=COCC)=O)C2)=O)CCc2cc(C)ccc2O1 C1(C(=O)Nc2cncc(C)c2)CCCCC1(C)NC(=O)C(C)n1ccnn1 C=CCC(CC=C)C(=O)N1CCN(C)C(CNC(=O)C(C)(C)C(=C)C)C1 c1(CC)ccc(F)c(C(N2CC3CCC3(CC(N3CCC(C)C3)=O)C2)=O)c1 S(=O)(=O)(c1cccnc1)NCC(=O)NC(CNC(c1c(CC)ncnc1)=O)CO [N-]=[N+]=NCC(C(=O)O)NC(C1CCC(c2ccccc2)N1)=O N1(C(=O)CC2CSCCO2)CCN(CC(=O)NOCC2CCCC2)CC1 C(=O)(CCCC(=O)c1ccccc1N)N(C1CN(C(=O)CC2CCC(=O)N2C)C1)C c1(OCC)ccccc1NC(C1COCCN1C(=O)COC(F)F)=O C(N=c1[nH]c(=NC(C)c2c(F)cccc2F)c2ccccc2[nH]1)c1cnc(C)o1 C1(NC(CCCCCCC)=O)COC2(CCCN(C(=O)Cc3cnn(C)n3)C2)C1 N1(C(C=CC=CCC)=O)CCC(CCC(=O)NC2(C(O)CO)CC2)CC1 n1(CC)cnc2c(NCCCC(C)C)nc(N3CC4COCC4(C(N)=O)C3)nc12 Cc1ccc(F)cc1CN1CC(Cc2cccc(Cl)c2)OC(C)C1 N1(C(C(C)NC(c2cccs2)=O)=O)CC2CCN(C(C3CC=CC3)=O)C2C1 CC1(NC(c2cc(C(N)=O)[nH]n2)=O)CCCN(C(C2CCC(C3CC3)C2)=O)C1 C(=O)(C1=CCCCC1)NC(CC=C)CNC(c1sccc1C1CC1)=O CC1=C(C)CN(C(C2CCCCN2C(=O)Cn2c(O)nnc2O)=O)C1 C(C1CCc2cc(F)ccc21)NC(c1c(C)nn(CC(C)C)c1Cl)=O c1(C(=O)NCC(C)NC(C(C)C2CC2)=O)cccc2sccc12 n1(CC)c(C)cc(C(=O)NC2CC2NC(=O)CN2C(=O)CCC2=O)c1C C=CC1CN(C(=O)C=Cc2ccn(C)c2)CC1NC(=O)CC12CCCC1C2 c1(C(=O)NC2C(CNC(c3ccc(=N)[nH]n3)=O)C2)c[nH]c2cc(Br)ccc12 C(CCCCCCCCC(=O)N(C)C)N(CCCN(C(=O)C=CCl)C)C C1(NC(C2CCCC(F)C2)=O)CCCCC12CCN(C(=O)CCCC1CCC1)C2 c1(C(=O)NCC(CCCC)NC(C2CC3(CC(=O)N3)C2)=O)cccc(F)c1C C1(CC(=O)NC(C2CCN2C(=O)CCc2nnnn2C)C)NC(=O)CNC1=O C(=O)(CCC1N=N1)N(CC(O)COCC(F)F)CC(N)=O CC(CCc1nc[nH]n1)N(CC(c1nn[nH]n1)C)C c1(OC)cc(CC(N2CC(C(=O)NCCc3cccs3)CC(F)C2)=O)ccc1O c1(NCC2(C)CCCC2)cc(F)c(CNC2C3CCC2CN(CC(=O)O)C3)c(F)c1 C(=O)(C(CCC(N)=O)NC(N)=O)N(C(C)CN(C)C(c1cncc(N)n1)=O)C C(CCN(C)C(C1(c2cc[nH]n2)CC1)=O)(C(C)C)NC(c1cn(CC=C)nc1)=O C(=O)(C(C(C)(C)C)NC(c1cccc(C)c1)=O)NCC(CC)C c1(CC(=O)NC2(CNC(=O)CN3CCS(=O)CC3)CCC2)c(F)cc(F)cc1F Cc1cccc2sc(CN(C(=O)CC3CCC3C(F)(F)F)C)nc12 c1(C(=O)NC2CN(C(C(C=CC)O)=O)CC2N=[N+]=[N-])nn2c(c1C)CCCC2 Cc1ccc(CC(=O)NC2C3CC2N(C(c2cn(CCCF)nn2)=O)C3)c(C)c1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CC(=C)Cl)C(=O)N(CCO)CCOC N1(CC(CC)(C)Nc2cnc3c(ccn3C)c2)CCCc2cc(OC)ccc21 N1(C(CC(CC)CN(C)C)=O)CCCN(C(c2cnnc(O)c2)=O)C(C)C1 N1(C(c2ccc(NCc3cn(C4CCC4)nn3)cc2)=O)CC2CCC1C(O)C2 C(=O)(C(O)Cc1cnc[nH]1)NCCOCCCN(C)C(C1COCCO1)=O C(CNC(=O)CCCOC(C)C)(C(C)(C)C)NC(c1ccc(CC)[nH]1)=O C(=O)(C(F)C(C)(C)O)N(C(C)C)CCNC(=O)C(C)(C)CNC(=O)C1CC1 c1(OCCOC)cccc2c1CCCC(N1C(=O)Cc3nccnc3NC1=O)C2 NS(=O)(=O)c1ccc(NC(C23CC2CN(Cc2cscc2Br)C3)=O)cc1 C1(C(=O)NCCCC2OCCN(C(CCN(CC)CC)=O)C2)CCOC(C)(C)C1 C(N=C(NCc1snnc1C)NC1CC1C)c1cc(C)sc1 C(=O)(CS(=O)(=O)CCO)N(C1CCCCN(C(c2c[nH]c(C#N)c2)=O)C1)C c1(C(=O)NCC2C(NC(Cc3c(C)non3)=O)CCC2)c(Cl)n[nH]c1C N1(C(C(C)OC(C)(C)C)=O)CC=CC(NC(=O)Cc2ccn(C(F)F)n2)C1 C1(CNC)CC(F)CN1C(=O)Cc1ccc(C)o1.C1(C=O)CC(N(C)C)C1 c1(C(N2CCCC3(CCN3C(=O)CC3CCCC3)C2)=O)ccc2[nH]nc(Br)c2c1 C12(C(N3CC(C)C(N=[N+]=[N-])C3)=O)CC3CC(C1)CC(C(F)(F)F)(C3)C2 C(CCC)(C(=O)NCC1CC(C(=O)NCC2COC(=O)N2)C1)=CCC CC1CN(C)CC1C(N1CCN(CCNC(=O)CCn2cnccc2=O)CC1)=O N1(C(C(CO)N(C)C)=O)CC2CCC(N)C2C1 CC1CCN(C(c2ccc(C#N)[nH]2)=O)CCN1C(=O)CN(c1ccc(Cl)nn1)C c1(CC)cnn2ccc(C(=O)NC(C3CCN(C(=O)C(C)CN(C)C)C3)C)nc12 N1(C(C)C)CCCN(C(c2cnc(C(C)O)s2)C(=O)NC2CCC2)CC1 C1(CNC(C2CC23CC3)=O)CCC12CCN(C(=O)Cc1nnc(O)s1)CC2 C1(C(=O)NCC(CC)N2CCCC2)CCN(C(C2CC(C)(C)CO2)=O)CC1 c1(-c2cn(CC(=O)NCCN(C)C)nn2)ccc(C2CCC2)nc1 c1(C(=O)NCC2CN(C(CSCCOC)=O)CC2(C)C)cccc(Cl)c1[N+](=O)[O-] C(CC1CCOCC1)(C(=O)NC1CCN(C(C)=O)C1)NC(C=CC=CCC)=O N1(C(C=CCCC)=O)CCCC(CCOC)(N(C(C2(N(C)C)CC2)=O)CC)C1 CC1CC(CNC(c2cc(Cl)no2)=O)CN1C(c1cc(F)n[nH]1)=O c1(OC)ccc(Cl)c(C(N2CCC(C)C(CNC(=O)C3=CCCC3)C2)=O)n1 C12(C(=O)NC(C3CCCCC3)CNC(C3(C)CCCS3)=O)C3CCC(CC13)C2(F)F Cc1ncccc1OCC(N1CCC2C(NC(=O)CCc3ccccc3Cl)C12)=O N1(C(C)=O)CC(C(=O)O)C2(CCN(C(C3(C(=O)OC(C)(C)C)COC3)=O)CC2)C1 N1(C(C2CC(C)NC(=O)C2)=O)CC2(CCN(C(=O)CCC3CCCCO3)C2)C1 c1(C(N2CC(ON3CC(CO)C3)C2)=O)cn(CCO)cn1.C1(C=O)CC2(CC2)C1 Cc1cc(F)c(C(=O)NC2CC(C)N(C(C34CC(C3)C4)=O)C2)c(F)c1 Cc1coc(C)c1CNC(=O)C(CCOCCO)NC(=O)CN1CC(C)C1 C(=O)(C1=C2CCCN=C2NN1)NCCCC1N(C(C(C(C)C)(C)O)=O)CCCC1 N1(C(CNC(C(c2cnc[nH]2)NC(C2N(CC(=C)C)CC2)=O)=O)=O)CCOCC1 C12(SCC)CCC(CC1)N(CN)C2.C(=O)CC(C)C(=O)OC(F)(F)F c1(NC(c2cc(C3CCOC3)[nH]n2)=O)cccc(NC(c2ccoc2Br)=O)c1 C1(CCCc2c(C)ncs2)(C(=O)N)CCN(C(C2CC2F)=O)C1.CO c1(C(=O)NC2CC2c2cn(CCNC(COCC)=O)nn2)csc2ccccc12 c1(C(=O)NCC(C(C)C)(C)NC(c2ccsn2)=O)ccn2c1CSCC2 c1(CN2CCC(N(C(C(c3ccc(OC)cc3)C)=O)C)C2)ccc(Cl)nc1C C12(CNC(=O)COC(F)(F)F)CCCC1N(C(=O)Cc1cccnc1)CCC2 C12(NC(C(C)OCCCCCC)=O)COCCC1CN(C(c1ccoc1)=O)C2 CC1CCOC(C(=O)NC(C2CCCN(CC(=O)N(C3CCCC3)C)C2)C)C1 c1(C(C2CC2)NC(C(=O)NC(c2nccn2C)C(C)C)=O)cccc(F)c1 N1(C(CC2CCCC(C)(C)C2)=O)CC2CCC(N=c3cnc(F)c[nH]3)CC2C1 C1(NC(c2c(C)scn2)=O)CN(C(=O)Cc2ccc3nn[nH]c3c2)CC(C)(C)C1 C1(C(=O)NC(c2ccccc2)C)(CC)CCN(C(c2csc(C(=O)O)n2)=O)C1 C1(NC(C(c2ccccc2)OC(C)C)=O)CC(O)CN(C(c2cc[nH]n2)=O)C1 CN1CC(CC(=O)NCCCN(C(=O)CN(C)C(c2ccoc2)=O)C)C1 N1(C(COCC(=C)C)=O)CCN(C)CC1CNC(C1CCCN1C)=O Cc1cn[nH]c(=NC(=O)c2ncc(C(F)(F)F)cn2)c1.C1(C)(CNCC)CCCN1 C1(F)(C(N(C(C(=O)NCC2(C)CCCO2)C2CCCO2)C)=O)CCCCC1 c1(CC(C(=O)NC(c2cn(Cc3ccoc3)nn2)C)C2CC2)ccc(O)cc1 c1(CN(CCCN(C)C(=O)Nc2nnnn2C2COC2)C)conc1C1CCCO1 N1(C(C2(N(C)C(c3cccc(Br)c3)=O)CC2)=O)CCC2(C=Cc3ccccc3O2)C1 N1(C(C(CC)N(CC)CC)=O)CCC(C)(C)C(C(=O)NCC2C(C)C2C)C1 c1(N(C(=O)CCN(S(C)(=O)=O)C)CCNC(CCOCCC)=O)cccnc1 Cc1cc(F)ccc1-n1nnnc1C1(NCC2CCCOCC2)CCOC1 N1(C(c2c(C)[nH]nc2Br)=O)CCN(C(C2CCCCS2)=O)CC(O)C1 C1(C(=O)NC(CNC(C(C)(C)OC)=O)(C)C(C)C)CCc2cnnn2C1 c1(SCC)ccc[n+]([O-])c1.C(CC(CN)NC(C1CN(C2CCCCC2)C1)=O)OC C(=O)(CC(CC)C1CC1)NCC(CCC)OCC.c1(C=O)cc(C(N)=O)c[nH]1 C1(C)(COC)CCN1C(=O)C(ONC(=O)Cn1cnnc1)C c1(OC)ccc(F)c(N)c1C(=O)NCC1CCC(CNC(c2cn[nH]c2)=O)CC1 N1(C(c2cc(C)[nH]n2)C(=O)NCCCC)Cc2ccc(OC)cc2CC1C Cc1nc(C2CCCO2)sc1C(N1CCC(CNC(=O)C(F)=CCCF)CC1)=O c1(N2Cc3c(nc(N(C)C)s3)CC2)nc(N2CCC(O)CC2)c2c(ncn2C)n1 Cc1cc(C(=O)N(CCCCCCNC(c2ccc(F)cn2)=O)C)c(N)cc1F N1(C(c2cc(C(C)C)[nH]n2)=O)CC(NC(c2ccncc2C2CC2)=O)CC(C)C1 Cc1cnc(C(=O)N(CC(C)(C)NC(C2CC2c2ccnn2C)=O)C)c(C)c1 c1(C(N2CCCC(CNC(c3ccc(C)nc3)=O)C2)=O)cccc2ccsc12 C1(CCNC(C(COCC)NC(c2cn(CCO)nn2)=O)=O)CC(C)(C)CO1 Cc1cccc(OC(C)CN2C(=O)CN(CC3CN(C)CCO3)C2=O)c1C C12(OC)CCC(C(N3CC(N(C)C)C3)=O)(CC1)C2.c12cn(nn1)CCCN(C)C2 C=CCC(C)(C)CCNC(=O)CCCC1CCCCN1C(C1CC(C)(F)C1)=O N1(C(C(C)O)=O)CC2(CCC2)CC1CNC(=O)CN1C(=O)CNC1=O C#CCC(C)(C)C(c1nnnn1CCC1(C)CC1)Nc1cnc(C)nc1C N1(C(C2(OCC)CCOCC2)=O)CCC(NC(=O)CCCOCC)CC(C)(C)C1 Cc1cc2[nH]c(C(N3C4CCC3C(NC(=O)C(F)(F)C(F)F)C4)=O)cc2s1 c1(CCCSCC(=O)NC(CC)CNC(C)=O)cc(Sc2ccccc2)n(C)n1 c1(C(C(=O)NCC(C)C)N(C)CC2(C=C)CC2)ccc(-c2cccs2)cc1 c1(C(C)C)c(Br)cc(F)c(F)c1F.C12CCCN(C1)C(=O)CCCn1cc2nn1 c1(OC)cc(C(=O)NC2CCOC2C(N2CCSCC(C)C2)=O)ccc1C(C)=O c1(C(C(=O)N)(F)F)ccc(F)cc1.C1(C(=O)N(CCC2CCOC2)CCO)CS(=O)(=O)C1 C(=O)(C1=CCN(C)C1)NCC(C1CCN(C(C2COC(=O)O2)=O)CC1)C N1(C(c2n(CC)nnc2)=O)CCCCC1CNC(C1CCCN1C=O)=O N1(C(CCCCC#C)=O)CC2CCC1CC2NC(c1ncnn1CC)=O C(=O)(C(C)CCC)N(CC(CC)NC(c1cnn(Cc2ccccc2)c1)=O)CC Cn1ccc2cccc(C(N3CC4(C3)CN(C(c3csc5cncn35)=O)C4)=O)c12 N1(C(C(CC(F)F)N(C(c2c(CCC)nco2)=O)C)=O)CCCC2(CCCO2)C1 c1(C(c2n(CCCOC)nnn2)NC(CC)C2CC2)cccc(OC)c1 Cc1nn(C)cc1C(O)CNC(=O)NC1CC1.c12ccc(cc1)c(=O)[nH]2 C1(C(=O)NC2CCC2N)OC2CCC1CC2.CC1(C)CN(CC(=O)C(CN)=O)C1 C(c1cccc(Br)c1)=CC(=O)NC(C)C(C)NC(c1cnc(C(F)F)o1)=O c1(C(N2CCC(NC(C(CC)NC(C)=O)=O)C2)=O)sccc1S(N)(=O)=O.C(C)(C)(C)O C=CCCC(C(=O)NC1CC(NC(=O)CC2CCC(C)(C)O2)C1)c1ccccc1 c1(C(N(CCNC(=O)Cc2nc(=N)[nH][nH]2)CC)=O)cc2c(Cl)nccc2o1 C1(CNC(COC(CC)(C)C)=O)COCCN(C(c2n[nH]cc2C(F)(F)F)=O)C1 Cc1sc(-c2nc[nH]n2)nc1C(N1CCC1CNC(=O)C=Cc1cn[nH]c1)=O N1(C(C(C)OCCOC)=O)CCC(CCOC)(NC(=O)CN2CCOC2=O)C1 c1(C(N(CC(C)NC(=O)Cn2ccnc2)C)=O)ccnn1C(C)(C)C CC1CN(C(=O)C(c2ccc(F)cc2F)C)CCCN1C(c1cnc(O)[nH]1)=O N1(C(C=C(COC)C)=O)CCC(CO)(CNC(=O)C(O)CCSC)CC1 C(=O)(C1=CCCCCC1)NCC1C(OCC)CN(C(C2(C)CCN(C)C2)=O)C1 C(=O)(C(C)CC(=O)OC1CC1)NCCOCC(N1C(C#C)CC1)=O c1(CCC(=O)NCC(=C)CCNC(=O)CN2CCC(C)C2)cccc(C(N)=O)c1 CC1(C)CCC(CNC(=O)C=CCC(C)(C)NC(c2cnc(S)nc2)=O)C1 C1(NC(CCc2scc(C)n2)=O)CCN(C(=O)C(O)Cc2cnc[nH]2)C1(C)C c1(C2N(C(=O)NC(CCCC)COOCN)CCC2)ccc(Cl)c(Cl)c1 c1(C(=O)NCC(CC)NC(c2ccc(C)c(C#N)c2)=O)cc(F)cc2cc[nH]c12 CCCCC(C(=O)OC(C1CN(C(=O)Cn2cncn2)CC1C)=O)c1ccccc1 c1(N2CCC(NC(CC)=O)CC2)nc(=NCCC(C)N(C)C)[nH]c2c1COCC2 C=CCCCC(C(=O)N1CC(=O)NCC1CC)NC(C1CCS(=O)CC1)=O c1(NCCCC(C)NC(c2c(CC)ocn2)=O)cc2nnc(C(C)(C)C)n2cn1 N1(C(CC2(C)CC2(F)Cl)=O)CCC2(CCOCC2)C(CNC(c2ncc[nH]2)=O)C1 CC1(C)CC(CC(=O)NCCOCCNC(c2c(CO)cccc2F)=O)CCO1 CCC(CC)(CO)C(=O)NCC1(NC(c2ccncc2Cl)=O)CC2CCC1CC2 N1(SCc2cn(CC3CC(=O)OC3)nn2)CCN(C(=O)CN2CCCNC2=O)CC1 c1(CCC(=O)NCCNC(C(C(CC)CC)C)=O)c(C)nc2ncnn2c1C C=CC(C)CC(=O)NCC(=O)Nc1ccccc1OC(F)(F)F N1(C(C(COC)OC)=O)CC(CNC(=O)C(CC2CCC2)OC)CC1(C)C CC1(C#CC(=O)N2CC(C3CN(C(C4CCC4)=O)CCO3)C2)CC1 c1(C(=O)OCc2ccc(-n3cncn3)cc2)cc(C2CCN2)ccc1Br c1(N2C(=O)OCC2)ncccc1C(=O)OC(C)(C)C.Cn1nccc1-c1nn[nH]n1 C1(C)(C(N(CCCC)CCCO)=O)CCN(C(c2cc(C)no2)=O)C1 N1(C(c2cc(C)ns2)=O)CCN(C(c2cnc(C3CC3)nc2)=O)CC1C N1(C(CSC)=O)CC2(CC(NC(=O)CCOC3CCOCC3)CO2)C1 c1(NC)ccc(F)cc1C(=O)NC1CCCC(NC(c2ncn(C3CC3)n2)=O)C1 C1(C(=O)NCC=CC2CC2)CC2(CCN1C(c1ccnc3cc[nH]c13)=O)CC2 c1(-c2cn(C(CC)CC(=O)NCc3ccc(O)nc3)nn2)n[nH]c2c1CCCC2 C1(C)(C(N2CCC(NC(CCCCC)=O)C(O)C2)=O)CC(C(F)(F)F)=NO1 N(C(=NC(C)CSC)NCC1C2CCCCC12)CC1(C(=O)OCC)CCC1 N#CCS(=O)(=O)CC(=O)NC1CCC1CNC(c1ccc(Br)o1)=O C(C)(C(=O)N1CC(n2cc(CCC3CCCO3)nn2)C1)(OC)OC N1(C(CCC2(C)CN(C(C(CCC)(C)C)=O)C2)=O)CCOCC(F)(F)C1 C1(NC(c2cccc(F)c2)=O)CCN(C(=O)Cc2ccnc(F)c2F)CC1F N1(C(CC=C(C)C)=O)CC2CCCC1(CNC(=O)CC1CCNC(=O)C1)C2 N1(C(C(C)OCCOC)=O)CCN(C(c2ncn(C(C)C)n2)=O)CC(C)(C)C1 S(=O)(=O)(c1ccc(NCC2(C3CC3)CCC2)cc1Cl)N1CCN(CC)C(C)(C)C1 c1(C(C)NCC(C2CC3CCC2C3)O)cc2c(s1)CCC2 c1(C(=O)NC2C(C)N(C(=O)CCc3ccc(F)cc3)CC2)csc(=NC2CC2)[nH]1 CCCCC(C)CCC(=O)NC(CCOCC)C(N1CC2CCC(C1)C2O)=O c1(NC(=O)NC(C2CCN(C(C3CCCC3)CO)CC2)C)c(Br)cc(C)cc1Br C1(OCC)CN(C(=O)CCc2cc(C)no2)CC1CNC(=O)CC(C)(C)O O=C(C1=CCCCC1)NCC1CN(C(c2cn(CC3CC3)nn2)=O)CC1(F)F N1(C(C(C2CCC(C)(C)CC2)C)=O)CCC2CN(C(=O)CCC(=O)N(C)C)CC12 C(C(C)C)(C(O)C(=O)N(C1CN(C(c2ccc(C)c(O)c2)=O)CC1(C)C)C)OC C=CCC(CC(F)F)C(=O)NC(C1CCOC1)CNC(=O)C(CC(C)C)OC N1(C(COCCC(=O)OC)=O)CC2CCC1C(CNC(=O)C(C)C1CCC1)C2 N1(C(C2(CN(C)C)CC2)=O)CC2CCCC2(NC(c2cccc(C#N)c2)=O)C1 c1(CC)noc(CC)c1CC(=O)NCC1CC(O)CN1C(=O)Cc1csc(C)n1 N1(C(c2c(C)nc(C)[nH]2)=O)CCOCCCC1CNC(=O)CSCC1CCCO1 n1(CC)cnc2nc(=NCC3(CF)CC3)[nH]c(NCC3COCCN3C)c12 N1(C(CCCC)=O)CCC2(CCC2CNC(C2CCCN(C)C2)=O)CC1 C1(C(N(C(C)CO)CC)=O)CC(F)(F)CN1C(=O)COC c1(CN2C(=O)NCC(=O)NCCCN2)ccccc1.C1(NC=O)COCCO1 C(CCCC(=O)NC1(CO)CCN(C(=O)C=Cc2cncn2C)C1)OCC c1(C(N2C(C(=O)NC(c3cc(F)cc(F)c3)C)C=CC2)=O)ncc(Cl)cc1Cl N1(C(C2(C)CCC(=O)N2)=O)CC(C2(NC(c3cncc(C#N)c3)=O)CC2)C1 C(=O)(CN=c1ccc(C#N)c[nH]1)N1CC(C(C)NC(COCC#C)=O)OCC1 Cc1cccc(C(=O)NC2CCCN(C(C3C=CCS3)=O)C2)c1F C=CCC(C(=O)N1CCC(C)(CCNC(c2cc(CCO)on2)=O)C1)N(C)C N1(C(C2CN(CCC)C(=O)C2)=O)CCC(NC(C2(CCC)CC2)=O)C(O)C1 N1(C(C(c2ccccc2)OC)=O)CC2CC(C(=O)NCC3CCCCCC3)C(C2)C1 C1(C(N2CC(O)(C(C)NC(CSCC(C)C)=O)C2)=O)CC(C)CCC1C(C)C N#Cc1ccc(CC(=O)NC2CS(=O)(=O)CC2NC(c2cc[n+]([O-])cc2)=O)cn1 C1(CNC(CC=CCC)=O)CCCCN(C(c2nc(Cl)c(Cl)s2)=O)CC1 c1(C(=O)NCCC(C)NC(c2[nH]cc(C)c2)=O)ncccc1C1CC1 C(=O)(C1=NNC(=O)CC1)NC(C)(C)CNC(=O)CC(F)F c1(C(=O)NCC(N(C(C(CCOC)OC)=O)C)C2CC2)c[nH]c(=N)nc1C(F)(F)F CC(C)C(C(=O)NCC(CC(F)(F)F)NC(=O)CC1CC(=O)C1)C(C)C N1(C(C2CC(CCC)C2)=O)CC(CNC(c2cc(C)n(CC)n2)=O)CC1(C)C N1(C(CSCC)C(=O)N(C(=O)CC(O)CC(C)C)C(C)C)CCC2CCCC2C1 Cc1cc(C(N2C3CCC2CC(NC(=O)C(C)(C)C(C)O)C3)=O)c(O)c(C)n1 CC1(C)CC(NC(=O)CCC2CCCCO2)CN1C(c1cc2scnc2[nH]1)=O Cc1ccncc1C(=O)NCC1CCN1C(=O)CCn1cc[nH]c(=O)c1=O c1(C(=O)ON2CCC(OCC3CC3)C2)cc(F)c(O)c(F)c1 N1(C(=O)NCCC(C)F)CCCCC1c1nccn1C c1(C(N2CC3CC(NC(c4c(C)ocn4)=O)CC3C2)=O)c([N+](=O)[O-])c(C)nn1C C1(NC(=O)CCOC2CC2)CN(C(C2CCC(=C3CCC3)CC2)=O)CCC1CO c1(C(N(C2CCN(C(=O)Cn3cccc3)C2)CCC)=O)cnc(OC)nc1 Cc1ccnc(C)c1CC(N1CCC1CNC(c1c(Br)cnn1C(C)C)=O)=O C(=O)(CC(CC(N)=O)CC(C)C)NCC(CC(C)C)NC(c1cc(C)nn1C)=O C=CCCCC(C(=O)NCCOCCOC)NC(c1cnc(O)c(C)c1)=O N1(C(C#CC(C)C)=O)CCOC(C(=O)NCC(O)CC(C)(C)C)CC1 C1(CCOC)(NC(=O)CCc2ccnc(C)n2)CCN(C(C2CCCO2)=O)CC1 c1(CC)cnccc1C(=O)NCC(C)NC(c1ncn(C2CC2)n1)=O C(N(C)N1CCc2nc(C(=O)OCCOC)ncc2C1)c1cccc(OC)c1 C1(C(=O)NCC2(c3ccncc3)CC2)CC2CC(F)(F)CC(C1)C2(F)F N1(C(=O)Cc2cccc(Br)c2)CC2(CCCN(C(C3CCCCO3)=O)C2)C1 C(=O)(C1=CC2C=CC1C2)N1CCC2(CC1)C(=O)N2.C(C)(C(C)n1cccn1)OC c1(CC)occc1C(N1CC(NC(C2(NC(=O)CNC(C)=O)CC2)=O)C1)=O Cc1ncc(C(N2CCC(C(c3nncn3C)O)C2)C(=O)NCCCC2CC2)s1 C1(NC(CNC(C)=O)=O)CC1C1CCN(C(c2cc(Cl)cc[n+]2[O-])=O)CC1 c1(CNC(C(C2CCN(C(C3(OCC)CCC3)=O)C2)C)=O)ncc(Br)c(O)n1 c1(C(=O)NC2CCC2C(N2CCOC3CC23)=O)ncnc2cc[nH]c12 C1(C(=O)NCCCCC#CC)CC12CCN(C(C1(C#N)CCCO1)=O)C2 N1(C(C2CCC(=C)CC2)=O)CC2CCCC2(NC(c2cnn(CCO)c2N)=O)C1 N1(C(CC2C=NN(C)C2=O)=O)CCC(C#N)(NC(=O)Cn2ccc(O)nc2=O)C1 c1(CN2C(CC(N3CCCC(O)(CF)C3)=O)CCC2)ccc(O)c(C(F)(F)F)c1 C(C)(C)(CCC(=O)N(CCNC(=O)C(C)Oc1ccc(Cl)cc1Cl)CCO)OC c1(COC)cccc(C(N2CCOC(Cn3cc(C(C)SC4CC4)nn3)C2)=O)n1 C1(CNC(C(C)CNC(=O)C(F)(F)F)=O)CCCC(C)(C)C1 N1(C(c2c(C)cccc2F)=O)CCCC2C1CCN2S(=O)(=O)c1ccccc1C N1(C(CC(=O)NCC#C)=O)CC=C(CNC(C2([Si](C)(C)C)CC2)=O)CC1 c1(CNCC(F)(F)N(c2ccccc2)C)cc(F)cc(Br)c1F c1(C(=O)NC(C(=O)NC(CC)CCCO)COC(C)C)ccc2cc[nH]c2c1 N1(C(c2ccc(COC)cc2)=O)C2CCC1CC(NC(=O)C(CO)NC(N)=O)C2 N1(C(NC2CCCN(c3cccnc3)C2=O)=O)CCC2C(F)(F)C2(F)C1.C(C)CC c1(OCCC(=O)NCC(C)(C)CNC(=O)CC2(CS(C)(=O)=O)CC2)ccccc1O Cc1cc(Cl)c(C(=O)N(C)CCOCCNC(C2CC2C)=O)cn1 CC1CN(C(C2CC3(CC3)C2)=O)CC(C)CN1C(=O)CC1=CCCC1 c1(NC(c2cccc(C3CCCN3)c2)=O)cccc(OCC2CCCO2)c1 C(C(O)C(=O)NC1CC=CCC1)NC(CCCOCC=C)=O CP(C)(=O)C(CC(=O)N1CCOCC1c1cn(-c2cc(F)cc(Br)c2)nn1)OC c1(CC)cc(C(N2CCN(C(=O)CC3CNC(=O)C3)CC2)=O)c(C)o1 C1(C(=O)OC(c2cccc(C)c2)C(=O)Nc2ccn(C)c2)CCC(C2CC2)CC1 C(CCN=C(NCCC1CCCCC1)N1CCC2(CCCOC2)C1)OC(=O)NC C1(C)(CCNC(c2nc(C)sc2)=O)CCN(C(=O)CCCC#N)C1 C1(c2n(C3(C)CC3)nnn2)(Nc2cc(F)cc(Br)c2)C2CCC(C2)C1(C)C c1(C(=O)NC2CC3CC(NC(c4c(C)ccs4)=O)CC32)cc2nc(=O)ccn2[nH]1 Cn1cc(C=CC(N2CCC(O)(CCNC(=O)CN3CCCC3CO)C2)=O)nn1 c1(CC)cc(C(=O)NCCC2(OC)CN(C(C3(OC)CCC3)=O)C2)sc1C c1(C(N2C(C(C)(C)NC(C3CC3C(C)(C)O)=O)CCC2)=O)n[nH]cc1F C(c1cc(Cl)cc(Cl)c1)=CC(=O)NCC(CC)NC(c1cccc(F)c1C)=O c1(C(=O)NCCCOCCNC(=O)CCC2CCOC2)conc1C1CCCO1 NC(=O)CCCCC(=O)NC1CCN(C(c2n[nH]c(C3CC3)n2)=O)CCC1CO C1(NC(C(C)CC(F)F)=O)CCCCC12CCN(C(C1CCCN1C(N)=O)=O)C2 CC1CN(C(=O)C2=CCCCCC2)CCN(C(c2cccn3ccnc23)=O)C1 c1(C(=O)NCC2CC(NC(C3(F)CCC3)=O)C2)ccc2scc(Br)c2c1 N1(C(c2n[nH]c(C)c2Cl)C(=O)NCC2CCCO2)CCCC2NC(=O)CC12 C1(C(N2CCC(C(=O)NC)CC2)=O)CC(F)CCN1C(=O)C1=NOCC1 C(=O)(C(F)(F)CCn1cccn1)N1CC(CNC(CC2CC(=O)OC2)=O)OCC1 C1(C(C)(C)C)C(C(=O)NOC(c2coc(O)n2)=O)CCN1Cc1cccnc1 c1(C(c2nnnn2C)NCC(C)Cn2ccnc2)ccc(C#N)nc1 CC1CCN(C(=O)CN2CCCCC2)C1C(=O)NCCC1CCCCO1 C1(CNC(c2c(C)n[nH]c2C)=O)CN(C(c2ncnn2C)=O)CCC1C c1(C(N2CCCCC(NC(C3C(C)CC(=O)N3)=O)C2)=O)cn2cccnc2n1 Cc1ccc(O)c(C(N2CCOC(CCCNC(=O)CC(C)N(C)C)C2)=O)c1 c1(C(=O)NCC(C)NC(=O)Cc2ccc3[nH]ccc3c2)[nH]nc2c1CCC2(C)C C1(OC)CCCC(C(=O)N=S(C)(=O)Cc2cc(F)ccc2F)CC1 CC(C)CC(F)C(=O)NCCC1CC(NC(c2ccnc(OCCO)c2)=O)C1 C=C(C)C1OCCC1C(=O)NCC1COCCN1C(=O)CCNC(C)=O c1(C(=O)NC2(C(=O)NCC(C3CCC3)OC)CC2)sccc1C1CC1 C1(=O)C(Cc2ccoc2)N1.CC(C(=O)N(C)C(C1CC1)C1CC1)N1CCCC1 c1(OCC(CN2CC(CN)OCC2)O)ccc(F)cc1.c12ccc(cc1)o2 n1(CC(=O)NC(CNC(C2N(CC)CCCC2)=O)(C)C)cnc2c1CCCC2 C(C)(C)(CC(F)C(=O)NC1CC(OC)C1(C)C)NC(c1ccc(CC)o1)=O c1(C(=O)NC(C=CC(=O)Nc2c(OC)cc(C)cc2)C)ncc(C#N)cc1C N1(C(c2c(Cl)cccc2Cl)C(=O)NC)CCn2cc(Br)cc2C1 C1(OC(F)F)CC(CNC(c2ccnc(OC(C)C)c2)=O)N(CC)C1 Cc1cc(CCC(=O)NC2CC(C)(CNC(=O)COC3CC=CC3)C2)c(C)s1 C1(C(=O)NCC2C3CC2N(C(=O)CCSC2CCCC2)C3)CCC2CCCCN12 N1(C(C(CC)C)=O)CC(OC)CC1CNC(c1ccnn1CC1CCCCC1)=O C(=O)(CC(C)C(F)(F)F)N1CC(OC)(CNC(c2cnc(F)c(Cl)c2)=O)C1 N1(C(C)C)CCCC1C(=O)NCC1CN(C(c2cnn(CC3CC3)c2)=O)C1 C(=O)(C(C1=NOC2CC12)N1CCc2cc(Br)ccc2C1)NCCOC Cc1ccc(Br)c(C(=O)NC2CC(NC(=O)C(O)C(F)F)C2)c1 C=C=CC(C)C(=O)N1CC(CC(=O)NCCc2cnc(C)s2)(OC)C1 c1(C(=O)NCCC2CCN(C(C3(C)CC4C=CC3C4)=O)C2)ccc(S(N)(=O)=O)o1 c1(C(=O)NC2CN(C(=O)CN3CCOC4CC34)CCN2)ccc(F)cc1Br C12=Nc3cccnc3C(=NCC3CCN(C3)CCN3CC4CC3CN14)N2.CC.OC C1(C(N(CC(CC=C)(F)F)C)=O)CCN(C(C2CCCN2C=O)=O)CC1(C)C CCC(CCCO)N=c1cc(C)nc(N2CCOC3(CCSC3)C2)[nH]1 c1(CC(=O)NC23CCN(C(CC(=O)NCC#C)=O)CC2C3)cnc2ccccn12 CC1(CO)C(C(=O)NC2CCC(F)(F)CC2)CCN1C(c1ccccn1)=O c1(C(N(C(C(N2CCC(C(=O)OCC)C2)=O)C)C)=O)nc(C)sc1C c1(NCC)cccc(C(N2CCC3C(NC(=O)C(N4CCOCC4=O)C)C23)=O)c1 N1(C(C2(CC)CC2(F)F)=O)CC2CN(C(c3c[nH]c(=O)cn3)=O)CC2C1 C(CC(C(C)C)NC(=O)C(C)(C)c1ccsc1)N(C(Cc1c(C)scc1)=O)C C1(NC(c2ccc(CCCCC)s2)=O)CCCCC1NC(=O)CC(O)CC c1(OCCC)ccc(C(N2CC(NC(C3(C)CCC(=O)N3)=O)C2)=O)cc1OC C1(C(=O)NC2(CC(=O)OC)CC2)COC(CNC(C2CC(OC)C2)=O)C1 c1(C(=O)NC(C)C(c2ccccc2F)NC(=O)CNC=O)cc2n(n1)CCOC2 C(c1ccccc1)=Cc1nc(C)[nH]n1.n12nnc(c1C)C(=O)NCC(O)C2 C12(CNC(c3nc(CCC)oc3)=O)CC1CN(C(c1c[nH]nc1C(F)F)=O)C2 c1(OC)ccc(C(N2CCCC2CCNC(C2CC3C(C2)C3(F)F)=O)=O)c(Cl)c1 C12CCN(C13CCC3)C(=O)CNC2=O.C(C)(C(=O)NCC)OCCOCCC C(=O)(CCC(C)(C)C#N)NC1C2(C(N(C)CC3CC3(F)F)=O)C3CC1CC23 N1(C(C(C=CC)O)=O)CCN(CC2CN(C(=O)COc3ccsn3)C2)CC1 C1(C(N2CCC(NC(C3CC3N)=O)C2)=O)Cc2cccnc2C1.N=c1cc[nH]c(C)n1 c1(C2(C(N3C(CNC(N)=O)CCC3)=O)CCC2)ccccc1Cl C(=O)(C(=O)CCC(C)(C)C)NCC1CN(C(Cc2c(OC)c(Cl)ccc2Cl)=O)C1 C1(C)(NC(C2C(=C)CC2)=O)CCN(c2nc(CCOC)ns2)CC1 C1(CC(=O)NCC2(C(N(C)Cc3ccco3)=O)CC2)CSCCO1 C1(NC(CN2C(C)CCC2)=O)CCSC12CN(C(c1ccc(Cl)nc1O)=O)C2 N1(CCOC)CC(C)N(C(=O)CNC(C2(n3cncn3)CC2)=O)CC1C C1(C(=O)NCC2C(NC(CCCC#CC)=O)C2)CN2CCCN1CC2 N1(C(C=CCCC)=O)CC(NC(c2coc(-c3ccccc3)n2)=O)C(C(F)F)C1 c1(CNC(c2ccc(OCCC)nc2)=O)cnc(C=C)c(Br)c1 CCC(C)(CO)C(=O)NC1CC(CCNC(=O)C(C)C(O)CC)C1 C1(NC(CCN(CCCCC)C)=O)CCCCC1NC(=O)C(=Cc1cccs1)C S(=O)(=O)(c1cccc(C(=O)NCC(CO)NC(c2scnc2Cl)=O)c1)N(C)C C(=O)(C1Cc2c(Cl)cccc21)NC1CCN(C(C(CCC)OCC)=O)C1C C(=O)(C(C)C(C)C)N1CC(O)(C(=O)NCC2N(C(C)=O)CC2)C1 C1(C(=O)NC2CC(O)CN(C(c3c(O)cccc3F)=O)C2)CCCCCC1(F)F C12(C(N3CCCN(C(C4CCC5(CCC5)O4)=O)CC3)=O)CC3CC(CC(C3)C1)C2 Cc1cccc(C(N2CCCC(CC(=O)N(C)CC3CCOCC3)C2)=O)c1C#N C1CC(=O)N1C.C1(C(=O)NC)(C(=O)NC(CC2CC2)C2CC2)CC1.OC c1(C(=O)NC2C(C(C)C)CN(C(C3(F)CC=CC3)=O)CC2)cnc2[nH]ncc2c1 CCC(CC)CC(F)C(=O)N(C)CC1(O)CCN(C(=O)C(C)N(C)C)C1 c1(C(C)C)ccc(C(N2CCCC2C(C)NC(C2CC23CCCC3)=O)=O)nc1 C(=O)(C1CCCc2nccn21)N1CCC(OCCNC(C(N)=O)=O)C1 N1(C(C(CCOC)OC)=O)CCC(COC)(NC(=O)Cn2nnc(C)n2)CC1 C#CCCC(O)C(=O)NC(C)CNC(=O)Cc1sc(C)nc1-c1ccccc1 CC1(C)OB(C2C3CN(C(=O)CCn4cncn4)CC3CN(C(C3CCC3)=O)C2)O1 c1(CCC(N2CC(C(C)NC(COCC(=O)NC)=O)C2)=O)ccc(Cl)c(F)c1 N1(C(C(CC=C)(C)C)=O)CCC2C1CCN2C(=O)C(Cl)CC c1(C(=O)NCCC(CNC(=O)CCc2cn[nH]c2)O)ccc(F)c(O)c1F N1(C(c2c(-c3ccn(C)n3)n[nH]c2)=O)CCCC(CO)(NC(=O)C=C2CCC2)C1 c1(CCCN(CCCNC(CNC(CC)(C)C)=O)C)ccc2nccn2c1.C(F)(F)O N1(C(CCCC)=O)CCCC2CN(C(c3cc(F)ccc3F)=O)CCC12 C1(NC(CC2ON=C(CC)C2)=O)CC2CC1N(C(c1ccoc1CC(N)=O)=O)C2 C1(C(=O)NCCN(C(C(C=C)(F)F)=O)C)CCc2c(cnn2C)C1 N1(C(=O)NC2CCCC3CN(Cc4cn(C)nc4)CC23)C(C)(C)CCCC1(C)C O=C(Cc1ccc(Cl)cc1)N=c1cc(Br)c2cccnc2[nH]1 C1(N(C(=O)C(C)Cc2ccncc2)CC)CCN(C(C2(C#N)CCCO2)=O)CC1 C(=O)(CCCCC(N)=O)N1CC(NC(c2c(NC)cncc2)=O)C(C)CC1 C12(NC(c3ncc(F)cc3F)=O)CCN(C(=O)CCCc3ccsc3)CC1C2 C1(C(=O)NC(C#C)C(C)C)(CC)CCN(C(=O)CC2CCCC2)C1 C1(CC)CN(C(=O)C(c2ccccc2C)(C)C)CC1NC(=O)C(CC)OC Cc1nc(C(C)NC(=O)C(CN(C)C)NC(=O)C=CC2(C)COC2)no1 c1(CN(CC)Cc2cc[nH]c(=N)c2)ccc(Br)cc1F C1(C(C)NC(=O)C(C)OCC(C)C)CCN(C(c2ccn(C(F)(F)F)n2)=O)C1 C1(C(=O)NC(C#CCC)(C)C)C2CCCC2CN1C(=O)CCC(=O)NCCC c1(CNC(NCC(F)=C(C)C)=NCCC2CCOC2)cc(C)c([N+](=O)[O-])cc1Br C1(C)(CNC(C(C2CC2)OCC)=O)CCN(C(=O)C(F)(F)CC2CC2)C1 C(c1cncn1C)=CC(N1CC(CCC=C)(C(=O)NC(C)Cc2nccs2)C1)=O C12(CNC(C3CC4CC4C3)=O)CC1CN(C(=O)C=CI)C2 C1(NC(c2c(OC)csc2)=O)CN(C(=O)Cc2ncccc2F)CCC1F C1(C(N(C)CC2(F)CCC2)=O)CC2(CCN(C(=O)C3=CC4C=CC3C4)C2)C1 S(=O)(=O)(c1ccc(-c2ccc(F)cc2)c2nonc12)N1C(C(=O)OC)CC(O)C1 C1(C(N2CCC(O)(C(C)C)C2)=O)COC2(C1)CN(C(=O)CCCn1cncn1)C2 CC1(C2(C)CC2NC(c2cnn(CC3CCOCC3)c2)=O)CC1 Cc1nc(C)c(C(=O)NCC2CC2CNC(c2cncc(C(F)F)c2)=O)o1 CN1CCC(C(=O)OC2(NCC3CC3)CCOCC2)C1=O N1(C(C(CCC)F)=O)C(C(=O)NC(CO)CCC(=O)OC)CCC1C C1(C(N(C)CC2CN(C(c3csc(=N)[nH]3)=O)C2)=O)Cc2cccnc2C1 N1(C(CC(C(C)C)NC(c2ccc(C#N)s2)=O)=O)CC2(CNC(=O)N2C)C1 C(=O)(CCCS(N)(=O)=O)N1CC2C(CNC(C(c3cccc(F)c3)CC)=O)(C2)C1 C#CCC(C(=O)OC)NC(=O)CC(C)NC(=O)CC(C)(F)F C1(O)(C(N2CC(C(C)CNC(=O)C(=O)N(C)C)C2)=O)CC(CF)C1 C1(C(CC)CC)CCCN(C(c2csc(C)n2)C(=O)N(C)C)CC1 N1(CC)CC(Nc2cc(NC3CC4CC4C3)nc(C)n2)CCC1=O Cc1sc(C(N2CCCC(O)(CCNC(c3cc(O)cs3)=O)C2)=O)c(C)c1C C1(C(N(CC(C)O)CCNC(C2CC(C(=O)OC)C2)=O)=O)C=CCCC1 Cc1oc2cc(C(N3CCC4CCN(C(c5ccccn5)=O)C4C3)=O)[nH]c2c1C C#CCCC(O)C(=O)N1CCC(CNC(C2(C(N)=O)CCC2)=O)C(O)C1 N1(C(C=CC)=O)CC(NC(=O)C(Cc2ccsc2)NC=O)CC1(C)C C1(CNC(C=CCN(C)CC)=O)CCCC2CN(C(c3cn(C)ccc3=O)=O)CC12 C(C)(C(=O)NC1CN(C(C2(C(C)C)CCC2)=O)C1)(C(C)C)NC(C)=O c1(C(N)=O)cccc(C(=O)Nc2ccc(N3CCC(CCO)CC3)cc2)n1 c1(OC)ccc(S(=O)(=O)Cc2ccnn2C2CCCC2)cc1Cl C=CCC(CC(=O)N1CCCC1C(O)CO)NC(c1n[nH]cc1CC)=O C1(NC(C2C(C(C)(C)C)C2)=O)CCN(C(c2cc(N)cnc2Cl)=O)C12CCC2 Cc1c[nH]cc(C(N2CC=CC(NC(c3csc(Cl)c3)=O)C2)=O)c1=O C(CC(C(C)(C)C)NC(=O)C#CC1CC1)N(C)C(c1ccc(C#N)n1C)=O Cc1nc(C(N2CCN(C(c3cccc(Sc4cnoc4)c3)=O)CC2)=O)nn1C C(=O)(CC(C)(C)CNC(c1cc(Cl)nn1C)=O)N1CC(C(C)C)OCC1 C(=O)(CC(O)C(C)C)N(CCOCCCNC(c1cc(COC)oc1C)=O)C C(=O)(C(CNC(=O)C(C(C)C)C1CCC1)CC1CC1)NCC(C(=O)OCC)O C1(NC(C2(CCC)CC2)=O)CN(C(C2CCOC2)=O)C2(CCCCC2)C1 c1(NC(C(CCNC(C2CC2C(C)(C)C)=O)OC)=O)ccc(O)cc1Cl C(=O)(CC(C)(C)CC(C)=O)N1CC2CC(NC(c3nc(COC)oc3)=O)C2C1 O=C1CC(CC(=O)NCC(O)CNC(C2(Oc3ccccc3)CC2)=O)CC(=O)N1 Cn1nnc2cc(C(N3CC(NC(c4cnc(C5CC5)[nH]4)=O)CC(O)C3)=O)ccc12 C1(C(=O)NC(CNC(=O)Cc2cc[nH]n2)C2CC2)C2C3CC4C1C1C2CC3C41 N1(C(c2nc(CC)oc2)=O)CCC(=O)NC2CN(C(=O)Cc3cc[nH]n3)CCC12 c1(CCC(=O)NC2(C)CCN(C(=O)C(F)=CCCF)C2)cccc(F)c1F C=C=C(C)CC(=O)N1CCOCC1CC(=O)NCCc1cnn(C)c1C C1(C(=O)NC2C(c3ccn(C)n3)C2)CC2(CCC2)CN1C(=O)CCC(CF)CF N1(C(Cn2c(CCC)nnc2S)=O)CCCN(C(c2cn(CC)cn2)=O)CCC1 C1(Nc2ccn(C3CCCC3)n2)(CO)CCN(C(C2CC(CC(=O)OC)C2)=O)C1 C(c1cn(C)cn1)=CC(=O)NCC(C1CC1)NC(C(C)CSc1ccccc1)=O CCCC(C)(C)CC(=O)N(CC(=O)NCc1cnco1)CC C(=O)(C1=CCC(NC(=O)CCN=[N+]=[N-])C1)N(CCCC)CC(N)=O C(CCCl)(CCCl)(c1n(C(C(=O)OC)C)nnn1)NCCSCCO N1(C(CN(C(C(CC=CC)C)=O)CCOC)=O)CCC12CC(C)(CO)C2 CC1C2CCC(C2)C1C(=O)N(CCC(=O)NCC1CSCCO1)C C1(CN(C(c2c(CC)onc2)=O)C)COCCN1C(c1c[nH]c(=O)cn1)=O Cc1cc(C(N2CC(N(C3CC3)C(C3(C)CC3)=O)CC(O)C2)=O)cc(Br)c1 N(C(=NCCCF)N1CCC2CCCCC2C1)CCCN(c1ccccc1)C c1(OC)ccc(C(=O)NCCC2CCN(C(=O)C(O)C(F)F)C(C)C2)c(C)c1 N1(C(C(CC)O)=O)CC2CCC(CNC(c3ccc4cc[nH]c4c3)=O)(C2)C1 C(CCCC(=O)NCC(F)CNC(=O)C(C)(C)Cc1ccc(Cl)cc1)NC(C)=O Cc1[nH]nc2c(C(N3CC(N(C)C(C4CNC(=O)CC4(C)C)=O)C3)=O)cccc12 C1(C)(CNC(C2C(C)(C)CO2)=O)CCCN(C(C2(C(C)(C)O)CC2)=O)C1 N1(C(CC)=O)C2CCC1C(C)C(NC(c1cccc3[nH]cc(Cl)c13)=O)C2 CN1CCC(NC(C2CC2F)=O)C12CCCN(C(c1cc(N)c(Cl)cn1)=O)C2 CCCCC(C)C(=O)NCC(O)CNC(=O)C(=Cc1ccc(C)cc1)C Cc1cc(C(=O)NC2CC(C)N(C(c3nc(=O)n(C)[nH]3)=O)C2)cnc1C(F)F c1(C(=O)NC2C(c3ccc(OC)cc3)CCNC2)ccc(Br)cc1OC(F)F C(=O)(CS(=O)(=O)CCO)NC1CC(CCNC(c2c(C)csc2Cl)=O)C1 C1(C(=O)NC23CC(NC(C4Cc5nccn5C4)=O)(C2)C3)CCc2nccn2CC1 c1(C(C(N2CCC(CN(C(=O)Cn3cncc3C)C)C2)=O)OC)cccc(F)c1 N1(C(C(CC)CCOC)=O)CC(NC(=O)Cc2cc(C3CC3)on2)CC2(CC2)C1 C1(N(C(C=CCC)=O)CC)CCN(C(=O)COCCC)CC1.C1(=O)CN1 C1(NC(CCC=CC)=O)CC(OC)CN(C(C2CCCCN2CC(F)F)=O)C1 Cc1ccc(C(N2CCCCCC2CNC(=O)C(c2ccn(C)n2)C)=O)nc1C N1(C(C)C)CCN(CCC(=O)NCC2CC2NC(=O)CCn2ccnn2)CC1 c1(C(=O)NCC2CC(F)(F)CN2C(=O)CC2CC=CC2)ccn2nnnc2c1 c1(C(N(C2CCN(C(C3C(C)CC3)=O)CC2)C)=O)ccc(SCC(N)=O)c(F)c1 C12(NC(CCCN=[N+]=[N-])=O)CCCC1CS(=O)(=O)C2 N1(C(C(C2CCOCC2)C)=O)CCC(C2CCN(C(C3(CCF)CC3)=O)C2)CC1 C123CCC(CC1)(CC2)NC3=O.C(=O)(C(C)CC(=O)N(C)C)N(C(C1CN(C)C1)C)C c1(C(N(CC(C)(C)CNC(=O)CC(F)F)CC)=O)ccc2c(ccn2C)c1 C12(C(=O)NC(C3OCCN(C(c4c(CCC)n[nH]c4)=O)C3)C)C(=O)C3CC1C2C3 O=C(C1=CCCCCC1)NCC1CC1CNC(c1ccc(C2CC2)cc1)=O C1(C(C)NC(=O)CC2CS(=O)(=O)C2)CN(C(=O)CC2(C)CC2)CCO1 CCC(O)C(F)(F)C(=O)NCC1(CNC(C2CCN2S(C)(=O)=O)=O)CCCC1 c1(C(N(C(CNC(CC(COC)C)=O)C)C)=O)c[nH]c(=O)c2ccnn12 N1(C(CC2N(C(C(CC)C(F)(F)F)=O)CC3(CC3)C2)=O)CC2CCC(C1)C(=O)N2 Cc1ccc(CC(=O)NCC(CC(F)(F)F)NC(=O)CC(C)F)cc1F N1(C(Cc2c(C)n[nH]c2)=O)CCC(F)(C(=O)NCC2CC(C)(C)CO2)C1 c1(CC(=O)N(CC(C)NC(COC)=O)C)n[nH]c2ccccc12 C1(COC)(CNC(=O)C(C)(C)C2CCCCC2)CCCN1C(=O)C(CO)N(C)C CC1COC2(C1)CN(C(C1CN(C(=O)C(C#N)CCC)CC1(F)F)=O)C2 C=C1CCC(C(=O)NC(C(=O)NCC2C(C=C(C)C)C2(C)C)C(C)OC)CC1 Cc1nc2c(CCC(=O)NC3CCC(C)N(C(=O)CCCN(C)C)C3)cccc2o1 c1(OC)ccc(CNC2CC(CC(=O)NCc3cc4ncsc4[nH]3)C2)cc1Cl CC1(C(=O)NCCC2CC2C2CC2)CCN(C(=O)Cc2c[nH]nc2O)C1 C1(CNC(c2c(C)ncnc2)=O)(NC(=O)COC2CC(F)(F)C2)CCCCCC1 C(=O)(C#CC1(C)CCCO1)NCCCC(C)NC(Cc1nc(C(C)C)sc1)=O c1(C(=O)NCC2CC(NC(c3cnn(C(C)C)c3N)=O)C2)cnc2ncccn12 N1(C(CC2CCCC(C)(C)O2)=O)CCC2(CC1)CC2NC(=O)Cn1cnnn1 C1(C(N2CCC(O)C(n3cc(CCC4CC4)nn3)C2)=O)(C)CCCNS1(=O)=O.CO C1(C(=O)OC)OCCN(C)C1.c12cnc(o1)CCC(=O)N1CC(C1)CC(OC)C2 C1(NC(c2cc(C(=O)OC)sn2)=O)CCN(C(c2cc(C)ncn2)=O)CC1F c1(C(C(=O)N(CCn2cc(C3(O)CCC3)nn2)CC)O)cccc(Cl)c1 c1(SCC(N2C(C(C)(C)CNC(=O)COC(F)F)CCC2)=O)ccc(Cl)cc1 N1(C(C(CCC)F)=O)CC2CCC2(CCN(C(C2CC3(CSC3)C2)=O)C(C)C)C1 C(C(C)(CCOC)NC(C1CCCO1)c1nn[nH]n1)OC N1(C(C=CCN(C(CC(=O)NCC#C)=O)C)=O)CCC12CCCCC2 N1(Cc2c(-c3ccccc3)nccc2)CC(c2cccs2)CC(c2ccccc2)C1 C1(C(N2CC(CC(C)NC(=O)Cc3scnc3C)C2)=O)(COCC)CCCO1 C1(CNC(CNC(C)=O)=O)C(O)C(O)CN1C(=O)CC(C)(C)C1CC1 Cc1cc(=O)oc(C)c1C(=O)NCCC1(NC(=O)CC2(O)CCCN(C)C2)CC1 C=C(C)CN=C(NCc1cc2ccccc2s1)NCC1CCC(N(C)C)CC1 Cn1nc(Cl)c(C(N2CCN(C(C3CCOC(=O)CC3)=O)C(CO)C2)=O)c1Cl N1(C(C(CC)(C)C#N)=O)CC2CCN(C(=O)CCCC(C)(F)F)C2C1 Cn1cnc2c1CN(C(c1cc(Br)cs1)C(c1ccc(F)cc1)C1CC1)CC2 Cc1ncc(C(=O)NCCN(C(=O)Cc2cnnn2C)C(C)C)cn1 c1(CC)cc(C(=O)N(C)CCOCCC(=O)N2CC(CC(C)(C)C)C2)c(C)o1 C=C1CCN(C(=O)CCn2ccc(C)n2)C(C(N2CC(=O)NCC2CC)=O)C1 CC(C)CC(CN(C)C(C1CCN(CC=C(C)C)CC1)=O)NC(=O)CC(C)(C)O CCC(C(=O)N1CCCN(C(=O)CC(=O)NCC2CC2)CC1)C(C)O CC1=CC(C)C(C(N2CC=CC2(C(=O)Nc2ccccc2)C(C)C)=O)CC1 c1(-n2cc(CN3CCC(CO)CC3CO)nn2)c(F)cccc1F N1(C(C2CCC(C(C)C)CC2)=O)CCC(NC(=O)C=CC2CCCO2)C(C)(C)C1 N1(CC2C(NC(c3ccc(OC)c(I)c3)=O)C2)CCc2c(Br)cccc2C1 CC(C)C(CN(C)C)C(=O)NCC1CC1CNn1cc(-c2ncccc2F)nn1 C1(NC(c2cc(CNC(c3c(OC)scc3)=O)[nH]n2)=O)CN(C)CCC1O c1(CCCC(=O)NCC2(CNC(=O)CC3COC(=O)C3)CC2)ccccc1Br Cc1cc2cnccc2n1CC(N1CCN(CC(=O)NC(C)(C)CO)CC1)=O c1(C(=O)NCCCCC2CN(C(C3(CCC)CC3)=O)C2)cc(C#N)ccc1N c1(C(N(CCNC(c2cc(O)n(C)n2)=O)CC)=O)nnc2n1CCCCC2 c1(CC(=O)NCC(CN(C(C2CCN(C(C)=O)C2)=O)CC)(C)C)ccc(F)cn1 C1(NC(c2ccn3ccsc23)=O)CCN(C(=O)CCc2cnc[nH]2)CC1O C1(C(N2C(C)CC(C(=O)NCCOCCO)C2)=O)CCC2(CCC2)O1 N1(C(COCCSC)=O)CC(NC(=O)CCN2CCCCCC2)CC12CCC2 C1(SCC2N(CC)CCC2)CN(C(c2c(N3CCOCC3)cccc2)=O)CCO1 c1(C(=O)NC(CC=C)CNC(=O)CC(C)C2CC2)cc2cc(Cl)ccc2n1C c1(CC)oc(C(c2nc(Cc3nnnn3C)cs2)NC(=O)OC(C)(C)C)cc1Br c1(CNC(C2CCCN(C(=O)Cc3cccnc3)C2)=O)cnc(Cl)cn1 C(=O)(C1CC(=O)c2ccccc21)N(C)CC1CCN(C(C2CC2C(N)=O)=O)C1 C(=O)(C(C(C)CC)N(C)C)NCC1(CNC(C(C=C)(C)C)=O)CCCC1 CC#CCCCC(=O)NOC(CC(C)C)C(=O)N1CCCCC1CCOC C1(C(N2CC(NC(CCNC(=O)NC)=O)C2)=O)CCS(=O)(=O)C1 C1(N(CCNC(C2(C(C)C)CCCC2)=O)C)CCCCCC1.C(=O)(C(C)OC)NCCF C12(F)CC(C1)C2.C1(C(=O)NC(=O)C2CC2)CCCN1NC(=O)CC1CCC1 Oc1ccc(N=c2scc(-c3ccc([N+](=O)[O-])s3)n2CC2CCC=CCCC2)cc1 CCCC(C(=O)NC(C)(CNC(=O)CNC=O)C1CC1)NC(c1ccccc1)=O c1(C(=O)NC(CNC(CN(C)CC)=O)CO)n[nH]c2c(OC)cccc12 C1(C(=O)NCCCN(C)C(c2ccco2)=O)CCn2c(O)nnc2C1 CC1COC(C(=O)NCC2(CNC(=O)C(C)(C)NC(=O)C(F)(F)F)CC2)C1 c1(CNC(CN(C(=O)OC)C)=O)cc(C(=O)NC2C=CCCC2)cs1 c1(OC)c(C)cc(C(=O)Nc2cc(Cl)ccc2OCC(=O)N(C)C)cc1Cl c1(C(N(C(C)C(=O)NCC=CC(C)(C)C)C)=O)ccc2cncn2c1 CC1C(=O)N(C)CCN1C(=O)CN(C(=O)C=Cc1ccsc1)CC1CC1 c1(C(=O)NC(c2ccns2)C)cc(-c2ccccc2)n2cnc(C(N)=O)c2n1 C1(NC(C(COC)C)=O)CCN(C(c2ccc(OC)cc2C)=O)CC1OC C1(C(=O)NC)CC2CC1N(C(c1cc(-c3nn[nH]n3)cc(O)c1)=O)C2 C=CCCCCCCC(=O)NC1CN(C(c2ccc(C#N)[nH]2)=O)CC1O c1(NC(C(C2CCCO2)NC(C2C(CC)OCC2)=O)=O)cccc(CO)c1 c1(NCC(=O)NC2CC(F)(CNC(CC3C(C)CCO3)=O)C2)ccccc1[N+](=O)[O-] CC1CCCC(CC(=O)NC23CC2CN(C(=O)Cc2cncnc2)C3)O1 N1(C(c2cc[nH]n2)=O)CCC2CC2(C(=O)NCC2OCC3CCC2C3)CC1 Cc1cc(=NC2C=CCCCC2)[nH]c(N2CCN(C(c3ccncc3)C)CC2)n1 C12(CNC(C3(CC#C)CC3)=O)CCC(CC1)N2C(C1CC(O)C1n1cccn1)=O CCCC(C(=O)NCCC1(OC)CN(C(=O)C(CC)N(C2CCCC2)C)C1)OC C1(NC(c2c(NC)snc2C)=O)CC(NC(=O)CCCc2cncs2)C12CCC2 N1(C(C2C(CCC)CN(C(c3cc[nH]c3)=O)C2)=O)CC(C)(C)OCC1(C)C c1(C(N2CCC(CNC(COCC(=O)NC)=O)C(C)C2)=O)cnn2c(F)cccc12 N1(C(C(n2c(C)cc(C)n2)C)=O)CCN(C)C(CNC(=O)CC(C)n2ccnc2)C1 N1(C(c2[nH]c(=NCC)sc2)=O)CCCC2(C1)CN(C(c1cc(C)nc(O)n1)=O)C2 C1(C(N)=O)CCCCC1NC(c1csc(CNC(c2cc(=O)cc[nH]2)=O)c1)=O C(=O)(C(O)CC(C)(C)C)N1CC2(CC(CC(=O)Nc3ccc(N(C)C)nc3)C2)C1 C(=O)(CC(C)(C)C(F)(F)F)N1CC(C(C)NC(C2(COCC)CCOCC2)=O)C1 CC1NC(=O)CCC1CNC(=O)C(=O)NC(=O)C(C)(N)c1ccoc1 N1(C(C2C(OC)CCC2)=O)CC(NC(=O)CCCS(C)(=O)=O)CC(F)(F)C1 C(C(CC1CC1)C(=O)N1CC(n2cnnc2)C1)NC(=O)C(C)(C)C(=O)NC C1(NC(=O)C=Cc2cocn2)CN(C(=O)Cc2cncc(O)c2)C2(CCC2)C1 Cc1cc(C(N2CC3CN(S(=O)(=O)c4cccs4)CC3C2)=O)ccc1[N+](=O)[O-] N1(C(c2ccc(C)cc2)=O)CCC(C)N(C(C2CCCC(=O)C2)=O)CC1 Cc1nc2c(N3CCC(O)(C(C)NC(C4(C)C=CCCC4)=O)CC3)ncnc2s1 C(CC(C(=O)NC(CO)C1(C)CC1)NC(=O)Cc1cc(C)[nH]n1)OC C=C(C)CCCC(=O)NCCCCN(C)C(c1ccc(C(=O)NCC(C)C)s1)=O C(=O)(C(CNC(c1cncc(C#N)c1)=O)C(C)C)N1CCC(C)(N(C)CC)C1 c1(C2C(C(N3CC(=C(C(=O)O)F)C3)=O)C2)ccc(Cl)cc1F CCCCC(C)C(=O)N(C1CCN(C(c2cncc(Cl)c2)=O)C1)CC(F)(F)CC C(=O)(C1=C(C)OCCC1)NC(C1CC1C(=O)NCC1(C)CC2CC2C1)C c1(CC=C)cnc(N(CCC)C(C2CCN(C(=O)CCC)C2)=O)s1 C1(C)(NC(C(CC2CC2)NC(c2c(OC)c[nH]n2)=O)=O)CC(O)(CO)C1 N1(C(CCC(=O)NCC)=O)CCC(C2CC2)(CNC(C2CCCCNC2=O)=O)C1 c1(CNCC(c2ccccc2)CNC(C2(C)CCC2)=O)cc2ccccc2cc1O c1(OC)ccc(C(=O)NCCCCCNC(=O)C(F)CN(C)C(C)C)cc1OC c1(C(=O)NC2CCN(C(C(COC)(C)COC)=O)CC2C)cccc2c[nH]nc12 CCC(O)C(=O)NCc1cc(CC(=O)N(CC(=O)OC)C)cs1 c1(OC)ccn2c(C(=O)NCCNC(c3cccc(C(C)C)n3)=O)cnc2c1 Cn1nc(C(=O)NCC(O)CC(=O)NCc2nccc(O)n2)cc1Cl c1(C(=O)NCC(C)COCc2ccncc2)ccc(OC(F)(F)F)c(Cl)c1 CCC(CC(F)F)C(=O)NCC1COCC1NC(=O)CCOc1cccnc1 C1(C(NOCCN(C)C)=O)CC=CC(NC(=O)C(C2CC2)C2CC2)C1 C1(C(=O)NC2(CC#C)CCCC2)CC2CCC(C1)N2C(=O)C(F)=CCCF c1(NC(C(C)NCCC2CC(CNS(CC)(=O)=O)C2)=O)c[nH]c2nccc(Cl)c12 c1(C(=O)NC2(CNC(CCC3CCC(C)O3)=O)CCC2)coc2c1CCCC2 Cc1cc(C(F)(F)F)n2nc(C(=O)NC3CCCCNC3)cc2n1 C1(C(N(C2(n3cccc3)CC2)C)=O)CC(NC(=O)Cc2cc[nH]n2)C(O)C1 C1(C(=O)NC(C2CCN(C(c3cnnn3C)=O)CC2)C)C2Cc3ccc(Cl)cc3C12 N1(C(c2ccc(CC)s2)=O)CCC(CNC(c2cc(CCO)on2)=O)(OC)C1 C(C(CC)C(C)C)(c1nnnn1C1CCCC1)NCCF.c1(OCC(C)O)ccccc1 C(=O)(CS(=O)(=O)C(C)(C)C)NC12CN(C(C(C=C)O)=O)C(CC1)C2 C1(F)(C(=O)NCC(C2CCC2)OCC)CCN(C(=O)C(COC)N=[N+]=[N-])CC1 C1(C(=O)NC2(C(=O)NOCC3CCC(F)C3)C(C)C2)CCC(O)CC1 C(C#CC(=O)N(C)CC1CC1(C)C)NC(COC(C)C)=O CCC(C)(O)CNC(=O)CCC1CCN(C(C2CCC2C(C)(C)C)=O)C1 CC(C)CCC(C(=O)N1CCCCC1)NC(c1cccc(F)c1O)=O C1(CC(=O)NCC2(O)CCN(c3ccc(C(=O)O)nn3)CC2)CCCC2(CC2)C1 CC1=CCC(C)(C(N2CCN(CCNC(=O)CNC=O)CC2)=O)CC1 c1(NC)ncc2cc(Br)ccc2n1.N1(C(CNC(N)=O)=O)CC2CC2(C=O)C1 C1(CC(C)C)NC(=O)CCN(CCC2CCCC3(CCC3)O2)C1=O c1(OC)cncc(C(=O)NCCC2(O)CN(C(C3CC3c3ccco3)=O)C2)n1 C#CCCN=C(NCc1ccc([N+](=O)[O-])cc1C(F)(F)F)N1CCC(C)C1 N1(C2CN(C(C(n3ccc(C4CC4)n3)C)=O)C2)CCN(C(C2COC(=O)N2)=O)CC1 c1(C(C)=O)ccc(-c2cn(CCCCNC(c3cc(O)nn3C)=O)nn2)cc1 N1(C(c2cc3scc(C(=O)O)c3[nH]2)=O)CCC2(CCC2)C(F)C1 C1(N(C=O)CC2(CC(O)CN3CCCC3)CCCCC2)CNCC1C1CCCC1 C1(OC)CN(C(=O)CCSc2nnnn2C)CC1NC(C1(C)CC1C)=O c1(N2CCC(C=C)CC2)nc2c(c(=NCC3CCN(CC)CC3)[nH]1)CCC2 N1(C(C(CC)(C)C)=O)CC2CCCN(C(=O)Cc3c[nH]c4cc(Br)ccc34)C2C1 N1(S(c2ccc(C)cc2Cl)(=O)=O)Cc2cccc(C3=CCOCC3)c2C1 CC1(c2cn(CCN3CCCC3)nn2)CCCN1C(c1scnc1C(F)F)=O C(CCC(F)(F)F)ONC(C1CC(C(C)C)C1)=O.C1(=O)CCCN1 c1(C(=O)NCC(C(C)C)NC(C2(CN(C)C)CCC2)=O)cc(S(=O)(=O)N(C)C)c[nH]1 CC1CC2(CC(C(N3C(C(=O)NC(C(=O)OC)C4CC4)CCC34CC4)=O)C2)C1 n1(CC(=O)NCCCC(C)NC(c2cnc(OCC)s2)=O)ccc(=O)c(O)c1C C1(C(N(CC(C)(C)C(=O)N(C)CC2CC3(CCC3)C2)C)=O)CC2CCC(C1)C2 c1(C(N2C(C(C)NC(CCOCC)=O)CCC2)=O)cnc2c[nH]nc2c1 N1(C(c2ccc(C)nc2O)=O)CC(NC(=O)C#CC2CCCO2)C(S(C)(=O)=O)C1 N1(C(C2C(=C)CC2)=O)CC(NC(c2cnnc(C3CC3)c2)=O)CC12CCC2 C(=O)(CCC(C(C)C)NC(=O)C(C)C1(O)CCC1)N1CC(OCC(C)C)C1 CC1(C)OC(C(N2CC3(C2)CN(C(c2ccc(S(N)(=O)=O)s2)=O)C3)=O)C(C)(C)O1 O=C1NC(=O)C(CC(=O)OCC2COC(=O)O2)S1 C1(NCc2c(Cc3cn(C)nc3)cc(F)cc2)CCSC(C)(C)C1 c1(CC)nncn1NC(=O)c1occc1CNC(C1CC(OC)C1)=O Cn1ncc(S(=O)(=O)N2CC3CCCC3(NC(=O)OCc3ccccc3)C2)n1 N1(C(C=C(C)C(F)F)=O)CC(F)CC1CNC(c1csc(C(F)(F)F)n1)=O CC(C)(CNC(=O)CNC(=O)CC1CCCCC1)CCNC(c1cocn1)=O N1(C(C(=Cc2ccncc2)CC)=O)CCN(C(=O)CCc2nncs2)CC1C1CC1 CCC(CC)CC(F)C(=O)N1CCC(C(=O)NCCC2CCN(C)C2)(CC)C1 c1(C(N2CCC(CN(C(c3cc(CC)no3)=O)C)C2)=O)cnc(SC)n1C c1(COC)nc(CC2CCCC2)n(-c2ccnc(O)c2)n1 CCC(CC)C(=O)N1CC(CC(C)NC(C2(c3ccc(F)cc3)CCC2)=O)C1 c1(NCC)cncc(C(=O)NCCCC(C)NC(=O)CN2CC3CCC2C3)c1 C(C(C)(CC(C)C)NC(c1cc(C)c(Cl)s1)=O)NC(C(=O)NCC)=O CCC(C)(C)C(O)C(=O)NCC1CCN1C(c1cc(C(F)(F)F)n(C(F)F)n1)=O c1(OC)c(CNN2CC=CCC2)cccc1C C1(F)(CNC(c2cccc(F)c2Br)=O)CCCN(C(C2CCC2)=O)C1 c1(C(=O)Nc2ccc(NC(C)CCC3CCC(=O)N3)cc2)cnn2ccncc12 N1(Cc2occ(C(=O)OCC)n2)CC2CN(C(=O)CC(C)COC)CC2C1 CC1CC(C(c2nccn2C)NCC(=O)N(C)C)CCC1(C)C c12ccc(o1)c(=O)[nH]2.C(C)(C)(C=CC(=O)NCC1(OC)CC1)OC Cc1c[nH]c(C(=O)NCC(C2CCN(C(C3(C)CC3(F)F)=O)CC2)F)c1C c1(C(c2nnnn2CCOC)NC(CC)CC)ccn(C(C)C)c1 c1(C(=O)NC(CNC(CCCN(CCC)CCC)=O)C)cc(C2CC2)cc(O)c1 C1(NC(C(CC)C(C)C)=O)COC2(CCN(C(c3cnn(C)c3C#N)=O)CC2)C1 C(=O)(CCN=c1[nH]c(N2CC(c3ccccc3)C2)nc(=N)[nH]1)C(C)CC1CC1 CONC(=O)C(=O)N(CC(C)NC(=O)CC(C)CN(C)C)C c1(NC(C2CCN(CCCNC(C3CN(C)CC3O)=O)C2)=O)ccc(F)c(O)c1 C1(NC(C(C)Cn2cccn2)=O)CCC(C(=O)NCCCc2nncs2)CC1 N1(C(=O)C=C2CN3CCC2CC3)CCC2CCCN(C(c3cnc[nH]3)=O)C2C1 C1(NC(=O)C=Cc2cn[nH]c2)C2CC3CC(C2)CC1(CNC(c1ccon1)=O)C3 Cc1cnc2cc(C(N3CC4CC3CC4CNC(=O)CCC(C)(C)F)=O)ccn12 CC(=O)C(C)(C)CC(=O)NCC1CC(C)N(C(c2ccc(C(N)=O)s2)=O)C1 c1(C(C(=O)NCCCC2CC2)N(CCC)CCC)ccc(Cl)cc1C(F)F Cc1cc(Br)cc(C)c1C(N1CCN(S(=O)(=O)C2CC2)C(CC#N)C1)=O c1(C(=O)NC2CCN(C(CCNC(=O)NC)=O)CC2F)cc2cncn2c(O)n1 c1(N2CCC(CC=C)C2)ncc(S(=O)(=O)N(C2CCCC2)C)cc1Cl C(CCC(C)(C)C(=O)N1CC(C(=O)N(C2CCCC2C)C)CCC1C)OC C1(C(N(CCCCNC(C2(C)CC2(Cl)Cl)=O)C)=O)CCCCN1N=O N1(C(C=Cc2ccc(OC)cc2C)=O)CCN(C(C2CC(=O)C2)=O)C(C)CC1C C=CCC(C)C(=O)N(C1CCN(C(c2nsc(OCC)n2)=O)CC1)C N#Cc1cc(F)ccc1C(N1CCN(C(c2cccc(Br)n2)=O)CC1CC#N)=O n1(CC)nnc(C)c1CNC(=O)CN(CCOC)C(c1cnco1)=O C1(CNC(C2(COC)C=CCC2)=O)CN(C(C2CCS(=O)(=O)C2)=O)CC1C C1(C)(CC)CCC(C(=O)NCC2(COC)CN(C(=O)C(c3cnn(C)c3)=O)C2)O1 C1(CNC(CSCCC#N)=O)CC2CCC(C1)N2C(C1CCC=CCC1)=O c1(C(c2cc(-c3cccs3)sn2)(C)CN(C)C)ccc(Cl)cc1 C12(CNC(C3(CC(C)C)CCC3)=O)CC(CN1C(=O)CCC1CCN(C)CC1)C2 c1(C(=O)NCC2(OC)CN(C(C3CCOC(=O)N3)=O)C2)scc(C)c1C c1(NC(C2CCS(=O)(=O)C2)=O)ccc(CCn2cc(-c3cnccn3)nn2)cc1 c1(C(C)CC(=O)N2CCC(N(C(=O)CCCc3cccs3)C)C2)ccccc1F Cc1c(C(=O)NCC2CCN2C(=O)CCn2cccn2)nn2ccccc12 c1(CCC(=O)O)ccc(F)c(F)c1F.C1(C)(C(C)(C)C)CN(C(=O)NCC)CCO1 C1(CC)CN(C(c2nccs2)=O)CCN1CC(=O)Nc1nc(C(=O)OC)co1 N#Cc1cc(C(N2CC3(CCC(C(N4CC(O)C(O)C4)=O)O3)C2)=O)c(Br)cc1F C=CC1CN(C(=O)COc2cccc(F)c2)CC1NC(C1CC(O)CN1C)=O c1(NC2C(NC(=O)NCCN(S(N(C)C)(=O)=O)C)CCCC2)c(F)ccc(F)c1F c1(C(N(CC(O)CNC(C2CCCO2)=O)C)=O)ccnn2ccnc12 N1(C(CSCCC)=O)CCOC(C(=O)NCCOCCCF)C1 c1(C(C)C)cccc(C(N2CCC(CN(C)C(C)C)C2)=O)c1 N1(C(C2(O)CCC2)=O)CCCC1C1CCCC1O.COC C1(NC(c2ccc(CC)c(C)c2)=O)CC2CCC1CN2C(C1CC2CC2C1)=O C1(CNC(CCCOCC=C)=O)CCN(C(c2cc(C)cc(F)c2)=O)C12CC2 Nc1ccc(C(=O)NCC2COCC2NC(=O)Cc2cccc(Cl)c2)nc1N C1(C(=O)NC(CC=CC(N2C(CSC)CCCC2)=O)(C)C)CCC(N=[N+]=[N-])C1 N1(c2ccc(OC)c(C#N)c2)CCC(F)(F)C(CNC(=O)C2=CCCS2)C1 c1(C(=O)NC(CNC(c2n(C=C)ncc2)=O)CO)ccc2[nH]ccc2c1F C12(CNC(c3c(C)nn(C)c3)=O)CCC1CN(C(c1ccc(C(F)F)cc1)=O)C2 Cc1cc2nc(N3CCOC(C(C)NC(=O)C=CC4CCCC4)C3)cc(=O)n2o1 CCC(CCCC(=O)NC(C)Cn1cccn1)NC(=O)C(=O)CC(C)CC C1(C(=O)NC(C)C2CC2)CCCCCCN1C(c1cccc2nc[nH]c12)=O N1(C(C=CC)=O)CCCN(CCNC(=O)CC2CCN(OCC)CC2)CC1 C1(O)(C(N2CCC(C(C)NC(c3cc(C)sc3)=O)C2)=O)CC2(CCOCC2)C1 CCCCC(O)C(=O)NCc1nc(C(=O)N(C)OC2CCCC2)c(C)o1 N1(C(=O)OC(C)(C)C)CCCN(CC(F)(F)CO)CC1 c1(-c2[nH]c(=NCC34CC(N(C)C)C3C4)sc2)ccc2snnc2c1.C1CN1 CC(C)C(C(=O)N1CCCCC1CN(C(=O)Cc1ccno1)CC)N1CCCCC1 C(c1ccoc1)=CC(=O)NCC(O)C(=O)NCC=CCl CC(CC(=O)N1CCC1CNC(c1sccc1C(F)F)=O)N(C)C n1(CC)cnc2c(NCCC(F)(F)C3CC3)[nH]c(=NCCSC)nc12 c1(C2(C(=O)NCC(CC)NC(c3cnc[nH]3)=O)CC2)ccccc1C CC(C)CCCC(=O)NCc1cn(C2CCN(C(C3COC(=O)N3)=O)CC2)nn1 Cc1ncc(C(=O)NC(C)(CNC(c2ccc(C(C)(C)C)cn2)=O)CO)cn1 c1(C(N2CCN(C(C3=NOC(C)C3)=O)CC2C2CC2)=O)ccc2c(n1)CCC2 C1(C)(C(=O)NCC(C)NC(=O)C=CCn2cncn2)CCCCO1 C1(C(=O)NCC(CCNC(C2(SCC)CC2)=O)O)CCS(=O)(=O)C1 CCCCC(CC)C(=O)NCC1(O)CCN(C(C2(N(C)C)CCCCC2)=O)CC1 c1(C(=O)NCC(C2CC2)C2CC2)n[nH]c2c1CN(C(C1CCCC1C1CC1)=O)C2 C#Cc1cnc(C(=O)NCC2CC(C)N(C(CCCCCCCC)=O)C2)c(C)c1 c1(CN(CCOC)CCO)cc(C#N)ccc1F.C1(CC(=O)O)CCN(C)C1 C1(CNC(C2C3C4CCC(C4)C23)=O)CCCN(C(c2oc(CO)nc2C)=O)CC1 n1(CC)nc(C(=O)N(CCNC(c2cc(CO)on2)=O)C2CC2)c(C)n1.C1CC1 N#Cc1cccc(C(CCc2cccc(N3CCCC3=O)c2)NC(=O)CCON)n1 Cc1ncc(C(=O)NCC(O)CNC(=O)C(C)Cc2ccc(F)cc2F)c(=N)[nH]1 N1(C(CN(CCCCCC)C)=O)CC2(C1)CN(C(=O)C1=COCCO1)CC2CO c1(C(N2CCC(C(=O)OC)(CC)C2)C(=O)NCCC)ccc(CC(=O)OC)cc1 c1(NC(c2nc(C)sc2)=O)cc(Cl)ccc1CN(C)C C1(CCNC(c2ccc(C(C)C)o2)=O)CCN(C(C2OCCC2(C)C)=O)CC1 C1(NC(c2c(C)cc(F)cc2)=O)CCN(C(c2cn[nH]c2)=O)CCC1(F)F c1(C(N2CCC(NC(c3cncnc3)=O)C23CC3)=O)cc2c(cc1O)CCCC2 c1(C(=O)NC(CNC(C2N(CC)CCC2)=O)C2CCC2)cnc(O)c([N+](=O)[O-])c1 CCC(C)(COC)C(=O)NCC1=CCCN(C(=O)CCF)C1 CN1CCN(C(C2C3CC(=O)CC23)=O)CC1C(N1CC2CC1(CO)C2)=O c1(OC)cc(C)nc(NC(=O)NCC(c2ccc(OC)cc2)(C)C)n1 N1(C(C2C(OC)CCC2)=O)CC(CNC(C2CNC(=O)N2C)=O)C(C(F)(F)F)C1 C12(NC(c3ccnc(C4CC4)c3)=O)CCOCC1CN(C(=O)C=CC(F)(F)F)C2 c1(C(N2C(CNC(=O)COCCCF)CCC2)=O)ccc(C(F)(F)F)c(Cl)c1 N1(C(COCCC(C)C)=O)CCC(O)C(C(=O)NC(C)(C)CCO)C1 C1(N(C(c2ccc(C)o2)=O)C)CCN(C(=O)Cc2csc(C(C)(C)C)n2)CC1C N1(C(C)=O)CCCC2(CNC(c3cc(C(=O)OC(C)C)c(C)nc3C)=O)CCCC12 c1(C(=O)NCC2N(C(c3c(C)nn[nH]3)=O)CC=C2)cc2cc(Br)cc(F)c2o1 N1(C(C(C)OC)=O)CC(NC(c2occ3c2CCC3)=O)CCCC1C Cc1nc2cc(C(N3CC=CC(NC(c4cnc(S)nc4)=O)C3)=O)ccc2n1C Cc1c(C(N2CCC(C(C)NC(=O)COC3CCCCC3)CC2)=O)ncn1C C1(CNC(C2CC(C)(NC(C(CCC)O)=O)C2)=O)CC12CCCCC2 c1(C(=O)NC2CN(C(CCOC(C)=O)=O)CC2C)c[nH]nc1[N+](=O)[O-] N1(C(c2nccc(OC)c2)=O)CCN(C(C2C(F)(F)C23CC3)=O)CCC1C N1(CC(N2C(CN(C(=O)Cn3ncn(C)c3=O)C)COCC2)=O)CCC(=O)NC1=O c1(C(N(C2CCN(C(=O)CCc3cscn3)CC2)CC#C)=O)cccc(C)c1C N1(C(C(CCC)CNC(=O)CC2CC=CC2)=O)CCC2(CNC(=O)O2)C1 c1(OC)cc(OC)c(C(=O)N(C)CCNC(C2CCC3CC3CC2)=O)c(F)c1 C1(CNC(=O)C=CCN2CCOCC2)CCCCC1NC(=O)Cn1cccc1 CN1CCC(C(=O)NC2CN(C(c3cc(Br)n[nH]3)=O)CC(C)(C)C2)c2ccccc21 N1(C(c2ncc(C)n2C)C(=O)NCCOCC)CCOCC12CC2 CC1CC(NC(=O)C=C(Cl)Cl)CN(C(=O)C=C2CN3CCC2CC3)C1 CC(C)CCCC(=O)N1CCC(O)(CNC(=O)Cn2cc(C(F)F)cn2)C1 c1(C2N(C(=O)OCc3cc(OC)no3)CC2)ccc(Cl)cc1F C(=O)(C1=C(F)CN(Cc2ccccc2)CC1)OC1(C)N(C)S(=O)(=O)CC1 C1(C(N)=O)CN(C(=O)C(C2CCCO2)NC(=O)C(=O)NCC2CC2)C1 Cc1cnc(C(N2CCC(=CCNC(C3CC(N(C)C)C3)=O)CC2)=O)c(C)c1 C=CCCC(=O)NCCN(C(=O)C(C)N(C)C(C)=O)CCC c1(C(=O)NCC2CCC(C(=O)NCCCOCC)C2)n[nH]c(C)c1Cl CC(C)(F)C(C)(F)C(=O)N1CCC(Nc2cc(Cl)ncn2)C1 C(=O)(C1=C2CCCN=C2NN1)N1C(C)(COC)CC(NC(=O)CSC(F)F)C1 n1(CC)nc(C(=O)NCC2CCCCC2NC(=O)CCC(F)F)c(Br)n1 C1(NC(c2ccccc2N2CCCC2)=O)CN(C(C2CSC2)=O)CCC1O C1(C)(CNC(Cc2c(C)occ2)=O)CN(C(=O)C(=O)NCC2CC2)CCO1 c1(CNC(NC(C=C)C)=NCCc2cnccn2)ccc2c(c1)cc(C)n2C C1(NC(CC(C)(C)O)=O)CCN(C(C2CC3CCC2CC3)=O)C12CCC2 C1(C2CN(C(C3(O)CC(C)(C)C3)=O)C2)(NC(C2N(C)CCC2)=O)CC1 C1(CCNC(C2CCN(C(CC=C)=O)C2)=O)CCCCN1C(=O)CCCC CC1CN(CCNC(N2CCCC2Cc2cccs2)=O)Cc2ccccc2O1 C1(C(=O)NCC2(CNC(=O)C3=CCC(F)(F)CC3)CC2)Cc2cc(Cl)ccc2O1 N1(CCOC)CCC(NC(C2(NC(c3cc(OC)ns3)=O)CC(O)C2)=O)C1 C(=O)(CS(=O)c1cc(Br)ccc1OC)N1CCC(Nc2ccc(OC)cc2)CC1 CC(O)(CNC(c1ccoc1C(F)(F)F)=O)CNC(=O)CC1NC(=O)NC1=O C#Cc1cnn(C)c1C(=O)N(C(C)CNC(c1sc(CC(F)(F)F)nc1C)=O)C C1(NC(CCc2cc(C)[nH]n2)=O)CC=CCC1C(=O)NCCSCC(C)C C(=O)(C(CC(C)CC)NC(=O)C1=C(C)OCCS1)NC(C(=O)NCCC)CC N1(C(c2c(OC)ccc(Cl)c2)=O)C2CCCC1CC(CCN1CCCCC1)C2 c1(C(CC(=O)OCC)NC(c2cscc2I)=O)ccc(Cl)cn1 C(C(C)(C)CC(=O)NC(CCN(CC)Cc1cccnc1)C(=O)NC(C)C)OC C12(CNC(c3[nH]cc(CC(C)C)c3)=O)CCCC1CN(C(=O)CN1CCC1C)C2 N1(C(C(C=C)(C)C)=O)CCc2c(CNC(C34CC3C4)=O)cccc2C1 C(=O)(CC(C)(C)CC(=O)NCC(CC(C)C)NC(=O)C1=CCCC1)OC N1(C(CSCCOC)=O)Cc2occ(C(=O)NC3CC3(C)C)c2C1 N1(C(Cc2c(F)ccc(C)c2)=O)CCC2(C1)CN(C(=O)COCCN(C)C)CCO2 CCCC(C)CCN=c1nc2scnc2c(N(CC(C)C#N)C)[nH]1 c1(OC)cc(O)c(COC(=O)C(F)(F)c2nccn2C)cc1Cl c1(NC(=O)CCC2CCCC2)nc(CC(N2CCCC2CO)=O)cs1 N1(C(C2C(OC)C2)=O)CC(C)CCC1CNC(c1cn(-c2ccccc2)nn1)=O C1(C)(CNC(C2(C)CSC2)=O)CN(C(C2CC2C#N)=O)CCO1 c1(CNc2c(C#N)n(-c3cccc(C(N)=O)c3)nc2)cc(Cl)cc(Cl)c1S(N)(=O)=O CCC(C(=O)OC)C(=O)NC(C(N1CCSC(C)CC1)=O)C(C)OC C1(C(N2CCC(C(N3C(C(C)C)CCCC3)=O)C2)=O)CC2CCCC2C1 C1(C(=O)NC(C)C(CO)NC(=O)CCn2cncn2)CCN(C2CCSC2)CC1 CCCCC(CNC(=O)CC(O)c1ccccc1)NC(c1cccc(O)n1)=O c1(-c2cc(C(=O)Nc3csc4nccnc34)c(F)nc2)ccn2ncnc2c1 C1(C#N)(C(N2CCN(C(CC3CN(C(C)=O)C3)=O)C(C3CC3)C2)=O)CC12CCCC2 O=C(CCS(=O)(=O)c1ccccc1)NC1C2CCC1N(C(=O)COCC1CC1)C2 C1(C2CN(C(c3cn(C(F)F)cn3)=O)C2)(NC(CC2C(=O)NC(=N)S2)=O)CC1 N1(C(C2(F)CN(Cc3ccc(OC)nc3)C2)=O)CCN(C)C(C)(C)C1 C1(N(C(C(COC(C)C)NC(=O)CC2CSCCO2)=O)C)CCCCC1O C1(NC(=O)CN2CC(=O)NC2=O)CC2CCC(C1)N2C(C1CC(=O)C1C(F)(F)F)=O O=C(CCC1=CCc2ccccc21)NC1CCC1NC(C1CCCC(F)(F)C1)=O c1(C(N2CC(COC)(NC(=O)C=Cc3ccnn3C)C2)=O)cccc(=O)n1O c1(C(=O)NCCCC2N(C(CCOC)=O)CCCC2)cccc2[nH]nc(O)c12 C=C(C)C(C)(C)C(=O)N1CCCC(C(C)C(=O)N(C)Cc2ccon2)C1 C1(CC(=O)OC)(C(=O)OC(C)(C)C)CCCC1.c12cc(n[nH]1)N(CC=C)C(=O)CC2 C12(CNC(c3cc(N)c(Cl)cc3)=O)CCCC1CCN2C(=O)CC1(CO)CC1 CN(C1CS(=O)(=O)c2ccc(Cl)cc21)C(=O)NCc1ncco1 C(=O)(C1=NOC2(CCN(C(c3cc(Br)cn4ccnc34)=O)C2)C1)OC C(=O)(CCCCCCCS(C)(=O)=O)NC1C(NC(C(C)C2=CCCC2)=O)CCC1 Cc1ccc(CC(=O)NCC2CC2NC(C2(C)CCC2)=O)c(C)c1 CCCCCCCCN=c1[nH]c(C)cc(=NCc2csc(C)c2C)[nH]1 Cn1cncc1CCC(=O)NCC1CC(CNC(=O)CCc2ccccc2)CO1 C(=O)(C(C)C(C)(F)F)NC(CNC(c1cn(CCOC)nc1)=O)C(C)C.C1C(=O)N1 N1(C(CC2(CC)CCC2)=O)CCC(C(=O)N(C23CCN(CC2)CC3)CC)C(C)C1 c1(C(=O)NC2CCN(C(=O)CCSc3ccccc3)CC2)cc(F)c(F)cc1Cl C1(O)(C(=O)OC)CCN(CCCCCNC(=O)COCCCOC)CC1 N1(C(CC2(CC(=O)OC)CC2)=O)CC2CCN(C(C3C=CC=CC=C3)=O)C2C1 N1(C(c2c(NC)ccc(F)c2)=O)CC(C)N(C(c2coc(C(N)=O)c2)=O)CC1C c1(CC)cn2c(C(N3CCN(C(c4ncccc4F)=O)CC3)=O)cccc2n1 C1(CNC(C(C)(C)C)=O)CN(C(c2cc(Br)ccn2)=O)CCC12CCOC2 C#Cc1cncc(C(=O)NCC2CCCN(C(c3ccc(C)nc3OC)=O)C2)c1 C1(C(=O)NCC2C=CCCC2)CC2CCC1N2C(=O)CCOC1CCCC1 c1(CC)ccc(S(=O)(=O)N2CCC(C(C)NC(c3n[nH]cc3I)=O)C2)cc1 c1(NC(C2(CNC(CN(C(C)=O)C)=O)CC2)=O)cccc2c1C1CCC2CC1 O=S(=O)(c1cccs1)NCCNCCCN1CCN(c2ccc(Cl)cc2)CC1 c1(OC)ccc(C(N2CC(NC(C3(C(C)C)COC3)=O)C(C)(C)C2)=O)c(F)c1Cl Cc1ccc(F)c(C(=O)NCC2(C)CCN(C(C3(S(C)(=O)=O)CCC3)=O)C2)c1F N1(C(CCc2cncc(C)c2)=O)C2CCC1CN(C(=O)CCC(N)=O)C2 C=C=CCC(=O)N(CC(C)C(=O)Nc1ccsc1C)C c1(CCC(=O)NCCC2(CNC(C3CC4C=CC3C4)=O)CC2)cccc(F)c1 C(C(=O)Nn1cccn1)N(C)C(C1CCC2(CCC2)O1)=O Cc1cc(=O)n(CCC(N2CCC(NC(C3CC(O)C3)=O)C(CO)C2)=O)cn1 C1(NC(C2CCCN(C)C2)=O)CCN(C(c2cc(C#N)on2)=O)CC1(C)C N(C(=NCCNc1ccc(Cl)cc1Cl)N1CCS(=O)(=O)CC1)C(COC)C c1(CC)ccc(C)cc1-c1cn(C2CC(C(=O)NC(C(C)C)C3CCC3)C2)nn1 c1(C(C)C(=O)NCCCCCN(C)C(C2(C)CC2(Cl)Cl)=O)ccc(F)cc1 S(=O)(=O)(c1ccc(Cl)nc1C)N1C2CN(C(c3ccc(C)nc3C)=O)C(C2)C1 C(=O)(C1=CC2CC=CCC12)NC1(CNC(c2n(C)c(O)nc2)=O)CC1 C(=O)(C1CCCc2n[nH]cc21)N1CCC(NC(C(CC)n2cncn2)=O)C(C)C1 C1(C(N(CCNC(=O)C=Cc2cc[nH]n2)CC)=O)CCC(O)CN1C C(C(C)(O)CC(=O)NCC1CC1)OCC#C.C1=CCOCCNC(=O)C1 C1(C(N2CC(C(N)=O)(CNC(=O)Cc3csnn3)C2)=O)COC2(CCC2)CO1 c1(C(=O)NC2C(CNC(C3N(C(CCC)=O)CSC3)=O)COC2)cc(C)nn1C C(CC(C)(C)CC(=O)N1CCC(C)(CC(=O)Nc2cc(C)cc(C)c2)C1)OC Cc1sc(O)nc1C(=O)NC1(C)CN(C(=O)C(C)n2cncn2)C1 N1(C(C(CC)CC)=O)CCC2(CC1)COC(CNC(=O)CCS(C)=O)C2 c1(CCC(C)C)ccccc1C(=O)NCC1CC(F)(CNC(=O)CNC=O)C1 C(=O)(n1ccc(C(=O)NCC2(NC(=O)CC3CCCO3)CC2)n1)OC(C)(C)C c1(CCC)ccc(C(=O)NC2CCCC2CN(C(=O)C(c2ccccc2)C)C)[nH]1 N1(CC)CCC(CNC(c2cc(CNC(=O)C(C)c3ccco3)no2)=O)C1 c1(C(=O)NCCCC(=O)NC(C2CCCCO2)CC)ccc(CO)cc1 N1(C(C2C(C)=C2)=O)CCCC2CN(C(c3ccn(C4CC4(F)F)n3)=O)CC12 CN1CC(C(=O)N2CCSC(CC(F)(F)F)C2)c2ccccc2C1=O C(CCCC(=O)N(C)CC1CCSC1)NC(C1C(CCOC)C1)=O c1(C(N2CC(NC(CN3CCN(CC)CC3)=O)C2)=O)cc(Cl)c2cc[nH]c2c1 CCCC(C(=O)OC)C(=O)NC1CCN(C(c2cn(C(F)F)c(C)n2)=O)CC1 CCCCCCCC(=O)NCC12CC1CN(C(C1CC3CC3C1)=O)C2 c1(C(=O)NCC2C(CC(N3CC(C=C)OCC3)=O)C2)cccc2ccncc12 c1(C(=O)NC(CCN(C(C(C(C)C)C)=O)C)C)cn(C(C)C)c(=O)nc1O N1(C(c2c(C)nns2)=O)CC2(CC(C(=O)NCc3ncccn3)CO2)C1 C1(O)(CCNC(CCCSCC)=O)CCN(C(=O)CC2CCC(O)C2)CC1 CC(c1cccs1)=CC(=O)OC(C)(C)C.N12CCN(CC1)C(=O)OCCC2 N1(CC(=O)Nc2cccc(SC)c2)CC2CN(Cc3ccccc3C)CC2C1 C1(F)(C(=O)NCC(C)N(CCO)C)CCN(C(=O)CC2COCCOC2)CC1 c1(C(C2CC2)OC)nc(CC2CCC(C)(C)C2)n(-c2ccnc(C(C)C)c2)n1 N1(C(C2CCN(C(CC)=O)C2)=O)CCOC2(C1)CN(Cc1ccncc1)C2 C(c1cccc(Cl)c1)=CC(=O)NCCCCCCN(C)C(C1COC(=O)O1)=O CCCCC(C)C(=O)N1CCC(NC(=O)C=CC(C)C)C1 c1(SC)ccc(C(=O)NC(CC)C(=O)NC(C2CSC2)C)o1 c1(NC(c2cc(C)n(C)n2)CC)[nH]c(=NCC2(C)CC2Br)nc2scnc12 c1(C(=O)NC2CCCN(C(C(CC)F)=O)C2)ccc2ccc(Br)c(F)c2n1 C1(C(=O)NCCC2(NC(C=CCC)=O)CCC2)CCc2nnc(C)n2C1 N1(C(CCC#C)=O)CCC(C2CCCN2C2CCOCC2)CC1 c1(C(N(CCNC(c2c(C)ccn2C)=O)CC)=O)cc2ccc(Cl)cn2c1 CCCCCC(F)C(=O)NCc1nc(C)c(C(=O)NC(C)C(C)N(C)C2CC2)o1 N1(C(Cc2cccc(OC)c2)=O)CCN(C(c2ccc(CF)cc2)=O)C(C)C1C c1(NC(c2c(C)c[nH]n2)=O)ccccc1N1CCN(C)CC1 c1(C(=O)NCC(C)N(C)Cc2cncs2)ccn2ccccc12 c1(C(=O)OCCC(c2ccccn2)C)cnn(C2CCC2)n1 c1(CC)ccc(OCCC(N2CCCC2C2CCN(C(=O)CNC=O)C2)=O)cc1 c1(COC(C)(C)C)nc(CNC(=O)C(CC2CCC2)OC(=O)C2CC2)cs1 C(=O)(CCS(C)(=O)=O)NCCN(C(C(C)C)=O)C1CC1 C(=O)(CCCC(F)(F)F)N1CC2(CC(NC(c3ccc(CO)s3)=O)C2)C1 N1(C(CN(C(C(C)OCCCCC#C)=O)CC)=O)CCC(CO)C12CCC2 C(C(=O)N1CC(=O)NC(C)C1)(C(C)(C)O)NC(C1C(OC(C)=O)C1)=O C(CCCCCC(=O)N1CCCC1(C)C1CCC1)NC(c1cnc(C)s1)=O c1(-c2c(CC)ccs2)ccc2occ(CC(=O)Nc3nc(C)c(Cl)s3)c2c1 Cc1cc(NC(=O)NC2(NC(c3ccc(Br)nc3F)C)CCOCC2)cc(C)c1Cl CC1N(C(C2(NC(c3csc(F)c3)=O)CC(CO)C2)=O)CCC12CCC2 N12CCC3CCC(CC13)CC2=O.C(C(CCO)C(C)(C)C)OC(C)(C)C C(CC(C(=O)N1CC(CO)C1)NC(c1cccc(=O)o1)=O)OC C1(C(N(C2CCN(c3nnc(C(C)(C)C)s3)CC2)CCC)=O)CCCCNC1=O c1(C(CNC(C2(C)CC2(Cl)Cl)=O)NC(CCC)=O)ccccc1Cl C(=O)(C(C)(C)C1=CCN(C(=O)C2=CC3C=CC2C3)C1)NC1C(C)CC1 n1(CC(N2CCN(C(C3(C=C)CCCCC3)=O)CC2)=O)cnc2cc(C)ccc12 c1(OC(C)C(N2CCN(C(c3ccc(Cl)s3)=O)CC2)=O)cccc(Br)c1 C1(C(=O)NC(c2c[nH]ccc2=O)C)CC2(CC2)CN1C(C1CC2C(C1)C2(C)C)=O C1(NC(CC=CCNC(CC(COC)(C)C)=O)=O)CCCCN(C)C1=O c1(OC)cc(Br)cnc1C(C(=O)NC1CCOC1)N(C)CC1CC2C=CC1CC2 C1(NC(CC2(C)CC2(Cl)Cl)=O)CCC2CN(C(c3cncc(Cl)c3Cl)=O)CC2C1 c1(C(=O)NC(C)CN(C(=O)C(C)C(C)(C)C)C)cccc(S(=O)(=O)CF)c1 c1(C(N(C(C)CNC(=O)CC(F)(F)c2ccccc2)C)=O)cccn(O)c1=O C1(NC(Cc2c(C)ocn2)=O)CCN(C(=O)CSc2ccc(O)cc2)CC1F C=Cn1nccc1C(=O)NCC(C)(C)CNC(C1CCCN1CC1CCCC1)=O C1(N(C(C(C)OC(C)=O)=O)C)CCCN(C(=O)C(O)Cn2cncn2)C1 Cc1nn(C)c(C)c1CC(=O)NCC1(CNC(=O)Cn2ccccc2=O)CC1 C1(NC(C2=CN=C(OC)CC2)=O)COC2CN(C(=O)CCC3(C)OCCO3)CC12 CCC(C)C(O)C(=O)N1CC(CNC(c2c(C)nn(C)c2C)=O)CC1(C)C C1(NC(c2csc(Br)n2)=O)CC2CCC1N2C(c1ccnnc1Cl)=O c1(CCCNC(=O)NCC2CC(Cc3ccccc3)=NO2)ccnc(C(F)F)c1 C1(NC(C(C)c2cc[nH]n2)=O)CCC2(CC1)CN(C(c1ccc(Cl)nc1N)=O)C2 c1(C(=O)NCCN(C(C)(C)C)C(C2CCCCC2O)=O)cc(Cl)ncc1Cl c1(C(=O)NC2CN(C(CS(CC)=O)=O)C(C)(C)C2)cnc(O)n(C)c1=O N1(C(C)=O)CS(=O)(=O)CC1C(N1CCN(C(c2cc(O)n(C)n2)=O)CC1)=O c1(CC(=O)N(CC(CC)NC(C2CCCN(C)C2)=O)CC)ccc(OC)cc1C c1(C(=O)NCC23C(CN(C(C=CCCC(C)C)=O)C2)CC3)cc2cccnc2[nH]1 N1(C(C(C)C2CC2)=O)CCC2(CC1)CC(Nc1ncc(I)cn1)CO2 C1(NC(C2CN(C(C3CC3c3ccco3)=O)CC2F)=O)CC1C1CCCCC1 N1(C(C2(C#N)CC=CC2)=O)CC2(C1)CN(C(c1cnn3ccsc13)=O)CCO2 C(=O)(CCC(C(C)C)NC(=O)COC1CCCC1)N1CC=C(C)CC1 n1(CCCC2(C)CC2)nc(-c2ccccc2)nc1Cc1cccnc1F C1(CC)CC(O)CN1C(C1C=CC(NC(=O)CN2CCC(F)CC2)C1)=O C1(NC(CC(C)N(C)C)=O)CN(C(=O)COCP(C)(C)=O)CC(C)(C)C1 c1(C(=O)NC(CNC(C(C)c2ccsn2)=O)C)c[nH]c2cccnc2c1=O c1(CNC(C)=O)cc(C)no1.C1(C)C(=O)N1C1CC1.C(C(=O)NCC(C)O)O C12CC3(CCC(N=C4NC5=NCN4N=CC=C1N5)CC3)C2.OC c1(C(=O)NCCNC(C2COC(=O)O2)=O)cc(Cl)c2n[nH]cc2c1 C(=O)(CCC(=O)N1CC(CNC(=O)C(C)NC(N)=O)CC1C)OCC N1(C(Cn2c(C)cc(C)n2)=O)CC(O)CCC1C(=O)NCC(=C1CCCCC1)F C(C)(C(CC(=O)NCC(C)(COC)CO)NC(C1CCC(F)CC1)=O)OC CC#CCCCC(=O)N(C)CCNC(c1cc(Br)c(Cl)cn1)=O C1(CC)CN(C(=O)COCc2ncc(C)o2)CCN1C(=O)CC1C=NN(C)C1=O c1(C(=O)NCC2OCC(CNC(c3c(C)nsc3C)=O)C2)ccc(F)c(Cl)c1 Cc1cc(C(N2CCC(NC(c3cn(C)ccc3=O)=O)C(O)C2)=O)c(C)c(C)c1 C(=O)(CCC(C)(C)N(C)C)NC1CC(C(N(C)CCN(C)C2CC2)=O)C1(C)C c1(C(N2CCC(C(C)NC(CNS(NC)(=O)=O)=O)C2)=O)n[nH]c(SC)c1Cl C1(CC=C)(NC(C2CCCCC2OC)=O)CCN(C(c2ccno2)=O)C1 c1(N2CCCCC(NCC=CC(N3CCCC3)=O)C2)ncnc2sccc12 c1(C(N(C2CN(C(c3ccn(C4CC4(F)F)n3)=O)C2)C)=O)cc2c([nH]1)CCCC2 c1(C(=O)NC2(CC(=O)NC3C(C4C(C)C4)C3)CCC2)cnn2ccc(Cl)c(F)c12 c1(C(N(c2cc(O)ncn2)C)=O)ccc(N)c(OCC(F)(F)F)c1 c1(C(=O)NCC2CCCN(Cc3c(F)cccc3I)C2)ccc2sccc2c1O N1(C(c2nc(C)sc2C)=O)CC(C(=O)NC(C)CCC(F)(F)F)CC(C)(C)C1 c1(CC(=O)NC(C)C(C)NC(=O)CCC2CCOC2)ccccc1OC(F)(F)F c1(OC)cncc(OC)c1C(=O)NCCNC(=O)C(c1cc(C)cc(C)c1)O C1(C(N2CC(NC(CC(CC)(C)C)=O)(CO)C2)=O)CCCC2(C1)CC2(F)F n1(CCC(=O)NC2CCN(C(C(CCCOC)C)=O)C2)c(=O)oc2ccccc12 N1(C(CSC(C)C)=O)CCC2CCC(NC(C3CCn4c(O)nnc4C3)=O)C1C2 CCC(C)N(OC)C(=O)C12CCN(C(c3snnc3C)=O)CCC1C2 c1(C(=O)NC2CCN(C(c3c(C(C)=O)cccc3)=O)C2C)cccc2oncc12 C1(NC(C(C(C)O)C)=O)CN(c2ccncn2)CC12CCOCC2 Cc1cc(C(=O)NC(C)(CNC(c2cnsn2)=O)C(C)C)c(Cl)cc1F C1(C(N(CCNC(CC(C)(C)SC)=O)C2CC2)=O)CCCC(C)(C)C1 c1(-c2ccc(CNC(=O)NC3CN(C)CC3C(F)(F)F)cc2)cc(Cl)ccc1F N(C(=NCC(F)F)N1CCC(C)(OC)C1)Cc1nc(CC)sc1 CN1C(=O)CCCC1C(=O)NCC1COCC1NC(=O)COCC1CCOC1 N#Cc1cc(C(=O)NCC(C2CCOC2)NC(=O)CNC(c2ccco2)=O)co1 c1(CC)ccc(C(N2CC3C(NC(C4C5CCC4CC5)=O)C3C2)=O)c(C)n1 c1(CNC(C2(F)C(C)C2)=O)cc(O)nc(CNC(c2ccc(F)cc2)=O)n1 N1(C(C23CC(C(=O)OC)(C2)C3)=O)CCOCC(NC(C2CN(CC)C2)=O)C1 C1(N(C(C(c2cccs2)NC(C=CCCC)=O)=O)CC)CCN(CC)C1 N1(C(CCNC(c2cccc(NC)c2)=O)=O)CCC(N=[N+]=[N-])C1 C1(C(=O)NC(CCN(C(=O)CCc2cccc(O)n2)C)(C)C)CC2C=CC1CC2 Cc1scc(C(=O)N(CC(C)NC(c2sccc2C#N)=O)C)c1N CC1(C)CCCCC1C(N1CCCN(C(=O)CN2CC(=O)NC2=O)CC1)=O CC(CNC(c1ccc2nc(O)[nH]c2c1)=O)CN=c1cc(Cl)nc(C(F)(F)F)[nH]1 C(CCN=C(NCCN1CCCC1=O)NCCN1CCOCC1)SC CCCC(F)C(=O)NCCC(O)CNC(c1ccc(C(N)=O)s1)=O CC1(C)CCOC(C(N2CCCC(NC(c3cc(CC4CC4)on3)=O)CC2)=O)C1 C1(CCNC(c2onc(C)n2)=O)CCCN(C(=O)CCOC2CCOCC2)CC1 c1(C(=O)NCC2C=CCN2C(C23CCC2C3)=O)c(F)cccc1Br Cc1nc(CSCC(=O)NC2CC(N(C)C(C3COCC3SC(C)C)=O)C2)cs1 c1(CN)ccnc(CC(c2nc(C3CC3)no2)C(c2ccccc2Cl)C)c1.C(F)(F)F Cc1ccnc(NC(=O)CCCCCc2ccc(F)cc2)c1Br c1(C(=O)NCC(C)CNC(C2CCC(O)C2)=O)cc([N+](=O)[O-])ccc1Cl c1(CC)nc(C)ncc1C(N1CCC(F)C(NC(=O)Cc2cn(C)nc2C)C1)=O C1(C)(CNC(c2ncn(C)n2)=O)CCN(C(=O)CC(F)(F)F)C1 Cc1nc2ccccc2c(C(N2CC(CC(C)NC(=O)C=CCO)C2)=O)c1C C1(C)(C(c2nnnn2C2COC2)NC(c2ccnn2C)C)CCCCCC1 Cn1ccn2ncc(C(N3CCN(C(=O)CC4COCC4(C)C)C4CC34)=O)c12 Cc1cc(F)c(Cl)cc1NC(C1CC2CC2N1Cc1ccc2c(c1)CCC2)=O c1(OCC)ccc(Cl)c(C(N2CC(NC(c3cccs3)=O)C(C)(C)C2)=O)n1 C1(NC(c2cc(OC)no2)=O)CN(C(C2C(C)(C)OC2(C)C)=O)CCC1F C1(NC(C2CC23CC3)=O)C2CCC1N(C(c1ccc(-n3nnnc3O)cc1)=O)C2 N1(C(C2CC(C)N(C(=O)C(=O)NOC)CC2)=O)CCC2(CCC2)CC1 c1(CC(N2CCC(NC(C3(CO)CCCO3)=O)CC2)=O)n[nH]c2cc(Cl)ccc12 N1(C(CC2(CNC(c3c(C)ccs3)=O)CC2)=O)CCC2CC1C(=O)N2C c1(C(=O)NCCC(C)NC(=O)C(C2CC2)C2CC2)ccccc1OCCF.C(N)(=O)N C1(CC(N2CC(OC3CCN(C(COC)=O)CC3)C2)=O)CCCC(C)(C)C1 C(=O)(CCCCC(C)(C)C)N(C1CC2CCC(C1)N2C(=O)COC(F)F)C c1(C(=O)NCCN(C(=O)C#CC2CCOCC2)CC(C)O)cncc(P(C)(C)=O)c1 CCC(O)C(C)(C)C(=O)NCC1CC(C(=O)NO)(NC2(O)CCCCC2)C1 N1(C(C(=O)NC(CC)(C)C)C)CC(C)OC(C)(CC)C1 C=CCC(C(=O)N1CC(O)(CNC(c2cc(C(C)(C)C)c[nH]2)=O)C1)C(C)(C)C S(=O)(=O)(CC(=O)NC1CCC(C)(CNC(=O)C(=Cc2cscn2)F)C1)N(CC)CC CC(CCC(=O)NCCCS(C)=O)NC(C1(CO)CC(C)(C)C1)=O c1(CNC(C2CC(C)(F)C2)=O)cc(C(=O)NC2CC(=C(F)F)C2)ccn1 C1(CC(=O)O)(NC(=O)C(=O)NCCc2ncc(F)cn2)CCCCC1 CC1CC(C(=O)Nc2ccsc2)CCN1CCNS(C)(=O)=O O=C(C1=CC2CC(C1)CC2O)N(CCNC(c1cn(C2COC2)nn1)=O)C1CC1 CC1Cc2c[nH]nc2C(C(=O)NCCCCCCNC(C2(O)CCOCC2)=O)C1 C1(C(N(CC(C)O)C)=O)(Nc2cccc(O)c2)CCN(C(C)CO)CC1 CCCC(F)C(=O)NC1CN(C(=O)CN2CCNC(=O)C2)CC1CC1CC1 C(=O)(CCC(F)(F)F)N1CCC(C(C)Nc2nccc(OCCC)n2)C1 c1(-c2cnc(SCC)nc2)nc2ccc(C#N)cc2[nH]1 C1(CNC(CCCCOC)=O)CCN(C(=O)Cc2ncccc2C)CC1O N1(C(C2(COC)CCC2)=O)CCC(NC(C2SCCS2)=O)C(C(N)=O)C1 N1(C(CC2CC(C)(C)OCC2)=O)CCC(C2(NC(=O)C=CCO)CC2)C1 c1(C(N2CC(CCCNC(C=CC)=O)OCC2)=O)cc(O)cc(F)c1 c1(-c2c(C)nn(CC)c2C#N)ccc2nc(C(=O)NCCC(C)CO)sc2c1 CC(C)(C(=O)NCCC1CCN(C(=O)CSCC#N)CC1)C(N)=O N1(C(c2scc(OC)c2)=O)CC(C)CN(C(c2csc(C3CC3)n2)=O)CC1C C1(C(=O)NCC2CC2NC(C2CCCN(S(C)(=O)=O)C2)=O)(OC)CCCCC1 CC(CC(=O)NCC1CCCCN1C(C1CCC(C)(C)O1)=O)C(F)(F)F N1(C(c2ccc(C(C)=O)cc2)=O)CCCCC(NC(C2CCC=CCCC2)=O)C1 c1(NC(C2C(C(=O)NCC(C)(C)O)C2)=O)c(F)cc([N+](=O)[O-])cc1Br C1(C2(O)CCN(C(N3C(NC(C)(C)C)CCC(C)C3)=O)CC2)(NC(CC)=O)CC1 N1(C(C)C)CCCC1C(N1CCC(C(=O)NCCC(C)c2cn[nH]c2)C1)=O N1(C(=O)CCc2cnc[nH]2)CC2CN(Cc3nc(Br)cs3)C2C1 c1(C(N2CCC(OCCNC(C=CC)=O)C2)=O)c[nH]c2c(Br)cccc2c1=N c1(C(=O)NCCN(C(=O)CCc2cocn2)C2CC2)ccc(-c2nc[nH]n2)cc1 c1(CNC(C(CC)(C)C(F)F)=O)n[nH]c2c1CN(C(C1(C#N)CC=CC1)=O)CC2 CCC(CC(=O)NC(CNC(c1cc(C2CC2)ccn1)=O)C1CC1)C1CCC1 CCC(CCCO)N=c1nc2sccc2c(NCCc2cccn3ccnc23)[nH]1 C(=O)(CC(C)CC(C)C)NC1CCN(C(c2ncn(CC)n2)=O)CC1O N1(C(C(C)(O)c2ccccc2)=O)CCC(C(F)(F)F)(NC2CNC2)C1 N1(C(CCC=CCC=C)=O)CC(=O)NCC1C(=O)NCC(F)(F)COC Cc1ncc(C(N2CCOCC(CNC(C3(C(F)F)CCCO3)=O)C2)=O)cc1N C1(NC(C(C=C)(C)C)=O)C2CC3C1C3C2C(=O)NOCCCCF C1(N(C(=O)C=CCN2CCCC2)CC)CCN(C(=O)CSc2nccn2C)C1 CC1CC(NC(=O)C(C)(C)Cc2ccccc2)CN(C(c2nn[nH]c2Cl)=O)C1 C1(C(=O)NCc2cnc[nH]2)C2CCN(C(C3CN(C4COC4)C3)=O)CC12 c1(OCC)c(C(N2CC(CNC(=O)CC3CCC3)C(C(F)F)C2)=O)cccc1F C12(CNC(C3(C#C)CC3)=O)CCCC1N(c1ccncc1C#N)CCC2 c1(C(N(CC(C)NC(Cn2c(C)cc(C)n2)=O)C)=O)cncc2cc(Cl)ccc12 C(=O)(C(C)(C)C(F)(F)F)N1C2CC(CNC(C=CSC)=O)C1CC2 c1(SCCNC(C2N(CC)CCC2)=O)cc(COC)ccc1O N1(C(C(CC)CCOC)=O)CCC2(CC1)CCN(CC#CC(F)(F)F)C2 N1(C(C2=C(C)CCCC2)=O)CCC2(C1)CN(C(=O)C(C)Cn1ccnc1)CCO2 C(CCS(=O)(=O)c1ccc(F)cc1)N(C(=O)C(C)(C)CCCl)C C1(NC(CCCC#C)=O)CCN(C(=O)CC(C)NC(N)=O)C12CCCC2 CCC(C)C(O)C(C)C(=O)N(CCCCNC(c1cc(C)ccc1OCC)=O)C N=c1[nH]nc(CSCC(=O)NCC2CCN2C(=O)CC2COC(=O)C2)s1 C1(NC(Cc2ccc(C(C)(C)C)cc2)=O)CCN(C(=O)CCF)C1(C)C CC1C2C(CCN2C(c2cncn2C)=O)CN1C(=O)C(C1CCS(=O)(=O)CC1)O Cc1noc2cc(C(=O)NCCCCN(C(=O)C=Cc3nccs3)C)ccc12 c1(NC(C2(COC)C=CCN2C(=O)C(CC(C)C)OC)=O)ccc(N=[N+]=[N-])cc1 Cc1nc(C)c(C(N2CCN(C(=O)C(C)c3cc[nH]n3)C(C(F)F)C2)=O)nc1C C1(C)(CCC(=O)NCC2N(C(C3CCC(N(C)C)C3)=O)CC2)CCC(=O)N1 c1(NC(C(COCC)C2CN(C(=O)OC(C)(C)C)C2)=O)cc2c(s1)CCOC2 C1(NC(CC(C2CC2)NC(C(COC)C)=O)=O)CCC2(CCC2)C1 c1(C(N2CCC(CCOCC)C2)=O)ccc2nc(NC3CC4CC4C3)sc2c1 n1(CCCNS(C)(=O)=O)cc(C(c2cccs2)O)nn1.CC1C(=O)N1C C1(O)(CN(C(C(=O)NCC2CCOC2)c2csnn2)C)CCCC1 CC1(C)CCN(C(=O)COc2ccc(Cl)cc2)CC1C(=O)NCCC1(O)CCC1 Cc1ccc(OCC(=O)NC2CC2CNC(=O)CC2(CO)CC2)c2c1CCC2 O=S(=O)(c1ccc(Br)cc1N1CCCCCC1C(F)(F)F)N1CC=CC1 CC1(C)C2CN(C(C3CCCC3)=O)C(C(=O)Nc3cccc(F)c3I)C12 N1(C(C(C=C)O)=O)CCC(NC(=O)C(F)(F)CO)C(CC)C1 C(Cc1nc(-c2cccnc2)no1)(CC(F)(F)F)NC(CCCC(OC)OC)=O CCC(C(=O)NCCCNC(C12CCCC1C2)=O)Oc1ccccc1 CC1CCN(C(C2OCCN(C)C2=O)=O)CC1NC(=O)C(C1CC(F)(F)C1)O Cc1onc(Br)c1C(=O)NCCCOCCNC(C1CN(C(=O)N(C)C)C1)=O c1(C(=O)OC)cccc(C(C23CC(CN4CC5CC4C5=O)(CO2)C3)=O)c1.O(C)OC c1(C(=O)NC2CCOC2c2ccco2)cc2n(c(=O)c1)CCS2 Cc1ccc(C(N2CC(CO)(NC(=O)CC3CC4CC4C3)C2)=O)cc1CO C(=O)(C1=CCCCCC1)N(C1CC2CCC(C1)N2C(c1ncccc1N)=O)C c1(COC(c2ccc(Br)cc2Cl)=O)cc2n(n1)CCCC2 c1(OC)ccc(CN2CCCC2CCCCC#N)cc1OCC(F)(F)F C1(SC)(CCCC(=O)N)CCCCC1.C(=O)(COCCOCCO)NC Cc1cncc(C(=O)NCC(C)(CO)NC(=O)CSCCC(C)C)n1 C(=O)(C1=CC2(CCN(C(c3ncccc3F)=O)C2)C1)NC1(C(=O)OC)CCC1 N1(C(CCc2cc(C)no2)=O)CCN(C(C2CC2C)=O)C(CCO)C1 CC1C(NC(C2CC2(C)Br)=O)CC2CCC1N2C(c1cc2ccccc2o1)=O c1(C(=O)NC2C(CNC(c3c(C)nc(C4CC4)[nH]3)=O)C2)c[nH]c2cccc(Cl)c12 N1(C(CC(=O)NC)=O)CC2CC1CN(C(=O)CC=C(C)C)C2 C1(NC(C2(CC)CC2(F)F)=O)CC12CC(NC(=O)CC(F)(F)F)C2 C1(NC(CS)=O)CC(C)(NC=O)C1.C1(CC(=O)N(CC#C)C)CC1COC(C)(C)C C1(CC)CC12CN(C(C1CCN(S(=O)(=O)C(F)(F)F)CC1)=O)C2 c1(NC)cc2ccccc2cc1C(=O)OCC(C1CCN(C)C1)=O CC1CN(C)C(=O)CN1C(=O)CC(C(F)F)NC(c1ccc(F)cc1)=O C12(C(N(CCCC)C)=O)C(NC(c3nnc(S)n3C)=O)C3CC1C2C3 C1(C(N(CC(=O)NCc2ccc(OC)cn2)C2CC2)=O)C2CCC(F)(F)C12 c1(C(=O)NCCCN(C(c2cnn(C)c2C(F)F)=O)CC)c(Cl)nn(C)c1C CC1(C)CCCCC1C(=O)NCC(C1CC1)NC(=O)CCn1ccnn1 c1(C(=O)NC(CNC(Cc2c(C)ncs2)=O)CC(C)C)csc2nccn12 CCC(C)CC(C)C(=O)N1CC(NC(=O)C(n2c(C)cc(O)cc2=O)C)CC1C c1(CC(N2CCC(NC(CNC(CC)=O)=O)C2)=O)c(C)cnn1C C#Cc1ccc(C(N2CCC2CNC(c2cc(C)cnc2OC)=O)=O)cc1C N1(C(CCSC)=O)CCC(NC(=O)CCc2cncnc2O)CC1C1CC1 c1(-c2ccc(NC(c3n(C)ncn3)=O)s2)ccc(C#N)nc1 C(C(CC(F)(F)F)NC(C1(c2ccoc2)CC1)=O)NC(=O)Cc1ccc(C2CC2)cc1 C1(C(N2CC3(CCOC3)C2)=O)COC2CN(Cc3cccc(C(F)(F)F)c3)CC12 c1(COCC)nc(NCC(c2ccccc2F)NC(C2C=C2C)=O)cc(C)n1 N1(C(c2scc(C)c2)=O)CC(N(C(=O)Cn2ccccc2=O)C)C(O)C1 Cc1c(C(=O)NCC2CCN(C(c3ccc[nH]3)=O)C2)[nH]c2ccc(C(N)=O)cc12 Cc1scnc1CNC(=O)C(c1cn(C)nn1)NC(c1cc(CO)[nH]n1)=O N1(C(N=c2nc(C)n(C)[nH]2)=O)CCC2(CC1)CC2(C)C(N1CCC(N(C)C)C1)=O c1(C(N2CC(NC(c3scc(C)n3)=O)C3(C2)CC3)=O)cccc2cc(Br)cnc12 Cc1ccc(C(=O)NCCN(C(=O)C(c2ccccc2)N(C)C)C)c(F)c1 c1(-c2nc(-c3ccncc3)nn2C2CCOC2)cc2sc(Cl)cc2s1 N1(C(CC(COC)(C)C)=O)CC(CO)C2(C1)CN(C(=O)C(F)CCC(C)C)C2 Cc1cc(=NCCc2nc(O)n[nH]2)[nH]c(NC2CN(C3CCOCC3)C2)n1 Cn1c(O)nc(N2CC(O)(CCNC(=O)CC=CC(C)(C)C)C2)cc1=O Cn1cc(Cl)c(C(=O)NCc2nc(CNC(C3CC4(C3)CC4F)=O)cs2)n1 C1(C(N(C)CC2COCCN2C(c2cc(Cl)n(C)n2)=O)=O)CCCC12CCC2 c1(CN(C)CC23CC(C=O)(C2)C3)cccc2ncsc12.C(C)(C)(C)OCC n1(CC(=O)NC2CCN(C(=O)OC(C)(C)C)C23CC3)c(O)nc2ccccc2c1=O C12(C(=O)NC(C(C)NC(=O)C#CC(=O)N(C)C)(C)C)CCCC1OCC2 C(=O)(C1=CCCSC1)N(C(c1c(OC)cn(-c2ccccc2)n1)=O)C1CC1 Cc1cc([N+](=O)[O-])cc(C(=O)NCC2COCCN(C(c3ocnc3C)=O)C2)n1 Cc1cc(=NCc2cn(C)cn2)[nH]c(NCCS(=O)(=O)C2CC2)n1 CCC(CC(=O)NCC(=CC(=O)NOC1(OC)CC1)F)CC(C)C c1(C(=O)NCC2N(C(CSCC=C)=O)C3C(C2)COC3)cccn2c(C)nnc12 C1(NC(=O)CCF)CN(C(=O)CCn2cnc3c2CCCC3)C2(CCOCC2)C1 N1(C(COCC(=C)C)=O)CCCC2(CCC2NC(C2CCC(=O)N2)=O)C1 N1(C(c2cc(OC)ncn2)=O)CCC(C2(NC(=O)C(F)CC(C)C)CCC2)CC1 c1(N2CCN(C(C3C(=C)C3)=O)C(C)C2)ncnc2ccc(C(F)(F)F)cc12 N#Cc1cc(NC(C2CN(C(c3cnc[nH]3)=O)c3ccccc3O2)=O)cc(F)c1F c1(CC=CCNC(COc2ccc(OCC)cc2)=O)cc(S(C)(=O)=O)co1 Cc1ccnc(C)c1C(=O)NCC(F)CNC(c1cc(F)cs1)=O C1(CC)OCCC1C(N1CCCC1C(C)(C)C(=O)N1CC(O)(CC)C1)=O CC(C)(C)CCCCC(=O)NC(C)(CNC(=O)COCC1CCCOC1)CO C1(C(=O)NC2C(C(=O)NCC(C)(C)n3cccn3)CC2)CC(=O)C12CCC2 c1(OCCC(=O)NCC2(NC(C=C(CCC)C)=O)CC2)ccccc1[N+](=O)[O-] C1(NC(CC2CC(SC)C2)=O)CC2CCC(C1)N2C(=O)CCC(C)CN(C)C C1(C(=O)NCC2C(NC(=O)Cn3cccn3)C2)C2CCCCC12 N(C1CN(C(C23CCC(C2)C3)=O)Cc2ccccc21)C(C(CC)SC)=O C12(CNC(c3cc(C)no3)=O)CCCC1CCN2C(=O)CN1CC2CC2C1 CC1(C)CC(C(=O)NC23CC(CNC(C45CSCC4C5)=O)(C2)C3)C(C)(C)O1 C1(NC(CCC(=O)NCCC)=O)CN(CCc2cccnc2C)CCC1C C(=O)(C(C)C(C)C)N1CC(CC=C)(C(=O)N(C)CC2(O)CCOC2)C1 C(=O)(C(C)CC(N)=O)N(C(C)C(=O)NC1CC1)CC1CC2(CC2)C(=O)O1 N1(c2ncc(C(=O)OC)c(C)c2)CCN(C(C2(C(C)(F)F)CC2)=O)CCC1C CC1(C)CCCC1C(N1CCCCC1CCNC(c1ccsc1C(F)(F)F)=O)=O c1(N2CCCC(NC(C(CC)F)=O)CC2)ncnc2sc3c(c12)CCC3 C(C(=O)N1CC(NC(=O)COc2cccc(F)c2Cl)C(C)C1)(C(F)(F)F)OC(C)=O C(=O)(CC1=CCCC1)NCCOC1CCN(C(CCN(C(CCC)C)C)=O)C1 N1(C(C=CCN(CC#C)C)=O)CCC(NC(c2ccc(CO)c(Cl)c2)=O)CC(O)C1 C(CCC(=O)NCCC(c1cccs1)NC(=O)Cn1cccn1)N(C)C N1(C(Cc2c(C)ccnc2)=O)CCCC(C)(C)C1C(=O)NCC1COCCN1C N1(C(=O)NCc2nnc(C(=O)OCC)s2)CCC(O)C12CCC2 c1(CNC(C2CCCN(Cc3ccnc(Cl)c3Cl)CC2)=O)ccc(F)c(Br)c1 c1(NC2CN(C(c3c(C)ccc(C#N)c3)=O)CC2F)ncc2cc(F)ccc2n1 C12(C(=O)NC3(CNC(C(CO)NC(C)=O)=O)CCCC3)CCC(CC1)OC2 C12(C(N3CC(NS(C)(=O)=O)C3)=O)CC1CN(Cc1ccccc1OCCO)C2 Cc1ccsc1C=CC(N1CCCC1CN(C)C(c1cnc(C2CC2)s1)=O)=O C1(C(N2CC(NC(c3cncs3)=O)C2)=O)C2CCC1(c1ccc(Br)cc1)C2 N1(C(C(c2ccc(C)s2)C)=O)CC(CCCC2CCCC2)CC1(C)C.C1(=O)CCN1 Cc1cccc2c1CN(C(=O)CC1CC3(CO1)CN(C(=O)OC(C)(C)C)C3)C2 c1(C(=O)NC(C(CC)NC(c2cnn(CCO)c2)=O)C)ccc(CF)cc1 C1(C2(O)CCC2)(C(N2CCC(C(CC)O)CC2)=O)CC1.c12ccc(nc1)[nH]2 C1(C(=O)NCC(C2CCCN2C(c2ncoc2C)=O)(C)C)(CC)CC(C)(C)C1 C1(C(=O)NCC(CN(C)C(c2cc(Cl)ncc2F)=O)O)Cc2cncn2C(=O)N1 C12(CCCC1C)C(=O)N2.C(=O)(CC(=O)NCCSC(C)C)OCCC(C)C N1(C(c2c(-c3cncc(C)n3)cncc2)=O)CCC2COCC2C1 N1(C(c2nc(CC)oc2)=O)CCN(Cc2cnn(C(F)F)c2)CC1C Cc1cc(C(N2CC(O)CC2CNC(C2CC23CC3)=O)=O)nn1CCO N1(C(c2cnn(C(C)C)c2Cl)=O)CCCCC(N(C)C(C2CC(F)C(=O)N2)=O)C1 C12(NC(C3N(C(COCCOCC)=O)CC3)=O)CCCN(CC1)C2 c1(C(N2CCN(C(C)CCC)CC2)C(=O)NCCCC)ccccc1Cl c1(C2(C(C)NC(=O)C(N3CCc4sccc4C3)=O)CC2)ccc(F)c(C#N)c1 C(=O)(CCC(=O)c1cccs1)N(CCNC(=O)CCC1CC(C)C1)CC C1(NC(c2n(C=C)nnc2)=O)C2CC3C(C2)C13C(=O)NCc1ccc(O)cc1C C1(C(N(CCNC(C(CC)(C)O)=O)C)=O)CCc2ncsc2C1 c1(NCC2CC(NC(CCC(C)OC)=O)C2)ncnc2sc(C(F)(F)F)nc12 C1(NC(CC(CC)(C)C)=O)CN(C(C2CC3(C)CCC2(C)O3)=O)C2(CCOC2)C1 CCCC(C(N)=O)NC(c1conc1C(C)NC(c1cnc(OC)s1)=O)=O c1(C(=O)NC2CN(C(c3cn(CC)nn3)=O)CC2C)ccc2nn[nH]c2c1O C1(C)(CC)CCC(C(=O)NS(=O)(=O)CC2(OC)CCC2)O1 CC1C(C)S(=O)CCN1C(c1cn(CC2CC2)nn1)=O n1(CC(=O)NC2C(NC(C(CCOC)C)=O)CC=CC2)cc(C)c2ccccc12 Cc1ncnc(C)c1C(=O)NC1CCC1CNC(C12CCC1CC2)=O C1(CNC(CSCCOC)=O)CN(C(=O)CC(C)C)CC1O C1(=O)C(C)N1.C1(OC(C)C)CC(C(=O)CNC(=O)COC(C)(C)C)C1.C(C)(=O)O c1(CC)ccc(C(=O)NCC(C)CNC(=O)C(F)(F)C(F)F)cc1F c1(SCC(=O)NCC(C)(C(C)C)NC(C(CC)F)=O)ccc(F)c(F)c1 c1(OC)cccc(C2CC2C(=O)N(C)CCNC(=O)CCc2nc(=N)[nH][nH]2)c1 C1(NC(c2ccc(SCC)nc2)=O)CC=C(C(=O)NCc2cc(C)cnc2O)C1 S(=O)(=O)(c1ccc(C(=O)N(CC(C)(C)NC(=O)C(C)NCC)C)cc1)NCC CC1(C)C(CC(=O)NCCc2ccsc2)CCN1C(C1CCCC1C1CC1)=O C#Cc1cncc(NC(C2(C)CCN(C(=O)CCOCC(C)C)CC2)=O)c1 CC(C)CC(C)CC(=O)N1CCC(CNC(=O)C=Cc2ccncn2)C1(C)C C(C)(C(=O)NNC(=O)C(C)(C)CCCCNC(C1CCCCC1O)=O)OCC Cn1ncc(CC(C(C(=O)C2=C(Cl)CC2)=O)N)c1O.c1(CN)ccccc1 C(=O)(C1=NOC2(CCC2)C1)NCCC1(NC(=O)CCc2ncc[nH]2)CCC1 C=Cn1nccc1C(N1CC(OCCNC(C2CC(C)CO2)=O)C1)=O c1(C(N2CCC(NC(CCCC#CC)=O)C(C)(C)C2)=O)ccc2c(n1)OCCO2 N1(C(c2ccc3nc(OC)sc3c2)=O)CCCC2CN(C(=O)C3=CCC3)CCC12 C1(C(N(C(C)C(F)F)C)=O)CCCN1C(C1(C)C=CCC1)=O C1(CN(CCOC)C(=O)N(C)C2CC2)CCC1 c1(NC(=O)CC2CCN(CC(O)CC3N=N3)C2)nccc(Cl)c1F c1(OCC(=C)C)ccccc1C(=O)NCCN(C(=O)CCC1CCC(=O)C1)CC CC1CN(C(C2CCN2C(C)(C)C)=O)CC1NC(c1cc(-c2cnn(C)c2)no1)=O C1(NC(CC(C)F)=O)CC2(CCC(CNC(c3cnn(C)c3C#N)=O)OC2)C1 C1(OC)CN(C(=O)CC2OCCCO2)CC1NC(c1cscc1C(F)(F)F)=O C(=O)(C(C)(O)Cc1ccccc1)NCCOCCCNC(CNC(CC)=O)=O N1(C(CCC(=C)Cl)=O)CC2C3CCC(C2C1)N(C(c1ccc(F)c(N)c1)=O)C3 n1(CC#C)cccc1C(=O)NC1CCCC1NC(=O)CNC(=O)Oc1ccccc1 C1(NC(CNC(C)=O)=O)CC2(CCC(CNC(C3(C#N)CCCOC3)=O)OC2)C1 CC(C)(C(=O)N1CC2CC(NC(c3ccc(F)nc3)=O)CC2C1)C(F)(F)F c1(C(=O)NCC2(O)CN(C(c3onc(C)n3)C)C2)cc(F)c(O)c(F)c1 CCC(O)C(F)(F)C(=O)N1CCN(C)C(CNC(=O)Cc2ccc(F)cc2C)C1 C1(C(=O)NCC(CNC(c2n(CCC)ncc2)=O)O)CCCCN1S(C)(=O)=O C(=O)(CCCCC(=O)N=c1ccc2cc([N+](=O)[O-])ccc2[nH]1)OC(C(=O)OCC)C CC(C(=O)NCC1(F)CCCN(C(=O)C(C)(C)n2cccn2)C1)S(C)(=O)=O c1(CC)cc(C(N2CCC(CN(C)C(c3ccc(F)o3)=O)C2)=O)ncn1 N1(C(CN2C(C)CCC2)=O)CC2(CC(C(=O)Nc3ccccc3CN(C)C)CO2)C1 C(=O)(CC(C)(C)CC(F)F)NC1CCCN(C(COc2c(C)cccc2)=O)CC1 C1(C(=O)NCC2C(C(=O)NC3CCN(CC)C3)CC2)OCCOC1C c1(C(=O)NCC2N(C(CC3(CC)CCOCC3)=O)CCCC2)cc(N)cnc1O n1(C(CC)(C)C)nnnc1C(C1COCCO1)NCc1ccc(C(F)(F)F)o1 C1(=CCNC(=O)C(C2(O)CCCC2)F)CCN(C(=O)Cc2ccccc2Cl)CC1 N1(C(C2(C)CCCCC2(F)F)=O)CC2(C1)CN(C(C1CC(O)C1)=O)CC2CO N1(C(c2c(C)cc(N)cc2)=O)CCN(C(=O)C2CC2)C(C)CC1C.c12nncn1S2 C1(CCC)CN(C(=O)COCc2ccccc2)CC1NC(c1ccncc1Cl)=O Cc1cnccc1C=CC(N1CCC2C(NC(c3ccc(CO)cn3)=O)C2C1)=O c1(NCc2cc(CC)no2)cc(C(C)(C)O)ncn1 N1(C(c2cc(C)oc2C)=O)CC2(CCCC(CNC(=O)CSc3nc[nH]n3)O2)C1 c1(C(=O)NCC2(CCNC(C3C(C)CC(=O)NC3)=O)CC2)cnc2nccn2c1 CCCCCC(CC)C(=O)N1CCCCC1CNC(c1nc(C)no1)=O N1(C(CC(CC)C)=O)CC2(CCOCC2)C1C(C)C CN1CCCC(C(=O)NC2CCC2NC(c2nccc(C(F)(F)F)n2)=O)C1 c1(N(C)Cc2nn(C)cc2Cl)nccc(=NCCC(CO)CC(C)(C)C)[nH]1 C1(NC(C(C)CF)=O)CCN(C(=O)CN2CCCCCC2=O)CC12CCC2 C(CNC(=O)OCC(C)OC)(CC(=O)NCCn1ncccc1=O)OC C1(C(=O)NCCOCCC)N(C(=O)CC(CC)CC)CC12CCCC2 N1(C(CCN(CC)CC)=O)CCC2(CCCCC2NC(c2cnco2)=O)C1 CC(F)(F)CCC(=O)NCCC(Cc1ccccc1)NC(=O)C=Cc1ccco1 C1(n2ncc(C)c2)CCN(C(=NCC2CCC3CC23)NCC2CCC2)C1 C1(C)(C(=O)NC(CCSCCC)=O)CC(CN2CCC(CO)C2)C1 C1(CCC)CN(C(C2CN3CCN2CC3)=O)CCN1C(C1CC12CCCC2)=O c1(CCC)ccccc1C(=O)NC1CCCC1CNC(=O)C=Cc1nccs1 N1(C(CCC(=O)NC)=O)CC2CC(NC(c3ncn(C)n3)=O)CC2C1 c1(C(N2CC(NC(=O)Cc3csc(S)n3)CC(OC)C2)=O)nc2cnccc2s1 N1(C(CCC(C)SC)=O)CCC(C)N(C(=O)CSC(=N)N)CC1 Cc1nn(C)c2sc(C(=O)NC3CC4CC3N(C(C3(C)CCNC3=O)=O)C4)cc12 C(=O)(CCCCCCC(=O)OC)NC1C2CN(C(CC=CC=C)=O)C1CC2 CC#CCCCC(=O)N1CCC1CC(=O)NC(COC)CO C=CC1CN(C(c2cccn2C)=O)CC1NC(=O)C(O)Cc1ccccc1Cl N1(C(CCC(=C)C)=O)CCCC(NC(=O)CCC(=O)NCC)C(F)C1 N1(C(c2c(CC)c[nH]n2)=O)CCc2sc(CNC(=O)C(C)C(C)C)nc2C1 c1(CN2CCC(NC(C(c3ccc(F)cc3)N)=O)C2)cc(F)ccc1F Cc1ccc(CCNC(C2CCN(Cc3ccnc(F)c3Cl)CC2F)=O)cc1C N1(C(c2c(OCC)oc(C)n2)=O)CC(NC(c2cnc(S)[nH]2)=O)C2(CCC2)C1 C1(NC(=NC)N2CCC(CC(F)(F)F)C2)COc2ccccc2C1 C1(C(N(CC(CC)NC(c2cn(C)cc2C)=O)C)=O)CC2(CCC2)C1(F)F C(=O)(CCCCC(N)=O)NC1CN(C(CCCCCOCC)=O)C2C1C2 c1(C(N2C(CC)COC(C(F)(F)F)C2)=O)cnn2cccc(Cl)c12 C1(C(=O)OCc2ccc(OC)o2)N(C(=O)CC2CCC(C)CO2)CCCC1(C)C Cc1cc(C(=O)NC2CC(CCNC(=O)CC(C)c3cnn(C)c3)C2)sc1Cl C1(C(=O)Oc2cc(OC)cc(C(F)(F)F)c2)CC2CC1C1CCCC21 N1(C(c2ccc(CCC)o2)C)CCc2c(OC)ccc(C(=O)OC)c2C1 CC1CCN(C(C)C(N2CCCC(CNC(=O)CC3NC(=O)NC3=O)C2)=O)CC1 C#CCCCCCCC(=O)NC(C1CCN(C(C2(CCOCC)CCC2)=O)C1)C C1(C(N(CC(CC)NC(=O)CCNC(C2CCCC2)=O)C)=O)CCOC(=O)N1 N1(C(CCOCCCOC)=O)CCC(C(=O)NCC2(O)CCC(C)(C)C2)C(O)C1 C(=O)(C1=NNC(=O)CC1)N(C(CNC(C1(N(C)C)CCCCC1)=O)C1CC1)C c1(NC(C(C2(O)CN(C(CC)=O)C2)F)=O)ccc(CC)cc1O C1(S(C)(=O)=O)(C(N(CCNC(c2cc(C)ns2)=O)C)=O)CCCCC1 c1(C(N2CCC(=CCNC(c3c(C)snc3)=O)CC2)=O)cc(Cl)nnc1Cl CC(O)C(C)C(=O)NC1CC(F)(CNC(c2coc(-c3ccc(Cl)cc3)n2)=O)C1 C(=O)(CC1=NNC(=O)C1)N1CC(C(C)C)C(NC(=O)C=Cc2ccncn2)CC1 n1(CCOC)ccc(=NC(=O)C2(C)C=CCN2C(=O)CC2CCC(O)C2)[nH]1 CCCCC(CC)N(C(=O)C(C)CC1CC1)C.C1(=O)CC2(CC2)CN1 Cc1nn(C)c(-n2ccnc2C)c1C(=O)NCCC1CCN(C(=O)C(C)CO)N1 CC1CC(NC(c2cn(CC(F)(F)F)cn2)=O)CCN1C(c1ccoc1)=O c1(C(N2CC3(C2)CN(C(C2CCCCNC2=O)=O)C3)=O)n[nH]c2c1COC2 CC(CC(=O)N1CC(n2cc(CC3CCCCO3)nn2)CO1)SC(C)(C)C1CC1 Nc1cc(C(N2CCCC2CNC(c2ccncc2Cl)=O)=O)cc(F)c1 N1(C(C(N2C(C)CCCC2C)=O)=O)CCC=C(C(=O)NC)C1.C(CCF)SC C(=O)(CCCCNC(=O)C(O)c1ccco1)N1CCC(OCC2CC2)C1 S(=O)(=O)(c1ccc(C(F)F)cc1F)NC1CN(Cc2ccc(C)nc2Br)CC1(F)F c1(NC(=O)NCc2nccn2CCc2ccccc2)cc(Cl)c([N+](=O)[O-])cc1F Cc1cc2cnc1OC(=O)NC2.C1(C(=O)Nc2ccccc2)CN(C)CC(=O)N1 c12cc(no1)C(=O)NC2=O.N1(CC2C(C)C2)CCCC1 O=C1CCN(C(c2c[nH]nc2CCNC(C2CC3CCCC3C2)=O)=O)CCCN1 C(C(C(=O)N1CCC(C(=O)O)C1)n1cc(-c2cncn2C)nn1)OCCOC c1(CC)ccc(C)c(C(=O)N(CC(C)CNC(=O)C(C)NC(=O)OC)C)c1 C1(CN(C(=O)C(=O)N(c2ncc(CCO)s2)C)C)CCc2ccccc2C1 c1(CC)cc(C(=O)NC2CCCC2NC(=O)CCc2cnn[nH]2)cc(N)c1 N(C(=NCCN1CCCC1=O)NC(CF)CF)CC(=O)Nc1ccccc1 C1(C)(C(=O)NC2CC(CC(=O)Nc3cc(C)no3)C2)CC(F)(F)C1 O=S(=O)(c1ccc(Br)cc1NC1C=CCC1)N1CCCC(c2nc(=N)[nH][nH]2)C1 CC(C)C(S(C)=O)c1noc(C2CCCN2Cc2ccc(Cl)cc2)n1 C1(NC(=NCCNC(C)=O)NCCc2ccccc2Cl)CCc2ccccc2C1 N1(C(c2c(OC)nsc2)=O)CCCC(O)(CNC(C2CC2(F)F)=O)C1 CC(C)C(C)C(C)CC(=O)N1CCC(C)(NC(c2cnsn2)=O)CC1 N1(C(CC(=O)NCC)=O)CCN(C)CC1CNC(c1cc(C(N)=O)cc(Cl)n1)=O Cc1ccc2[nH]cc(CC(=O)N(C)C)c2c1.N12CCN1C(C)C2.C(=O)CN(C)CC C1(CNC(c2cnn(C)c2C(F)F)=O)CC(N=c2[nH]cnc3cc(I)sc23)C1 C1(C(N2CCC(CNC(c3c(CC)cno3)=O)C2)=O)CCc2cnn(CC)c2C1 N(C1CCOc2ccc(Br)cc21)C(=O)C(c1ccccc1)Oc1ccccc1Br N1(C(Cc2ccc(C)cc2)=O)CCC(O)C(C(=O)NCc2cn(C)nc2C)C1 c1(C(=O)NC2C(NC(CN3CCC(C)C3)=O)COCC2)cnc2ccoc2c1 N1(C(CC(C(CC)(C)C)O)=O)CCC2(CCCCN(C(=O)CC(C)(F)F)C2)C1 C1(CNC(C(c2ccccc2)C)=O)CC(NC(c2ccncc2O)=O)CC1O CN1CCCC(CNC(=O)C(CO)NC(C2(C)CCN(C)C2)=O)C1 N1(C(CC=C)=O)CC(CNC(c2ccc(-c3ncc[nH]3)cc2)=O)C(C)C1 C1(SCC(=O)NC(CC2CCCC2)CO)CCCNC1 c1(N(CCNC(c2cc3c(s2)CCC3)=O)CC)ncnc2scnc12 C1(CNC(CN(C2CC2)CC)=O)CCN(C(C2CCCC3CC23)=O)CC1C CC1(C(=O)NC2COCC2NC(c2c(F)cccc2F)=O)Cc2ccccc2N1 CCCC(CC(C)C)C(=O)NC1C=CCN(C(C2(N(C)C)CCCC2)=O)C1 C1(NC(C(C)OCCOC)=O)CCCC(NC(=O)C(c2cc(C)ccn2)(C)C)C1 C(=O)(CCC(=O)N(CCNC(=O)C(c1ncccc1F)(F)F)CCOC)NCC C(=O)(C(C)CS(C)(=O)=O)Nc1cc(C)c(N2CCOC2=O)cc1 N1(C(C2(CC=C)CC2)=O)CCCC(C2CCN(C(=O)C(C)(F)C(C)(C)F)CC2)C1 C1(CNC(C2(CCCC)CC2)=O)CC2CCC1N2C(=O)C(c1ccc(C)s1)C C(=O)(C1CCc2ccccc21)NC1(CNC(c2c(C)ccc(C)n2)=O)CCC1 CC1(C)CC(C(=O)N2CC(NC(C3C4CCCCC34)=O)C3(CC3)C2)=NO1 N#CCCCCCC(=O)NC1CC(NC(C2CCCC2C2CC2)=O)CC1O C(CCC(C(=O)N1CCC(O)(C(N)=O)CC1)NC(=O)C(F)CC(C)C)OC C(=O)(C1=CS(=O)CCC1)N1CCC(CNC(C2(COC)CC2)=O)C1 C1(C(=O)NCC2CCCCN2C(c2cc(COC)c(C)o2)=O)(CC)CCNC1=O c1(OC)cnccc1C(N1CC2CC1(CNC(=O)CC1CC(C(F)F)C1)C2)=O c1(C(=O)NC23C(CN(C(C4(C#C)CC4)=O)C2)C3)ccc(N=S(C)(C)=O)cc1 C1(C(N(CCCC2CCCC2)C)=O)CCN(C(C2(N)CC2)=O)CCO1 Cc1[nH]nc(C(=O)NC2CCC(CNC(C3(O)COC3)=O)CC2)c1C(F)(F)F N1(C(C=CCOC)=O)CCC(C)(CNC(c2ccc(C)nc2C)=O)CC1 O(C=C(C#N)C(=O)NCC(O)CNC(=O)CC1CCS(=O)(=O)C1)CC c1(OC)ncc(NC(=O)CCCn2cc(C(C)O)nn2)cc1C.c12ccc(o1)C2 CCC(C(=O)N1CC(F)CC1CNC(=O)Cc1ccn(C(C)C)n1)C(C)C N1(C(C2(C)CC(C(=O)OCC)C2)=O)CC(OC)CC(NC(=O)CC2CCCC2)C1 C(=O)(N=c1cnc(Br)c(C)[nH]1)c1c(NC(Cc2cccc(OC)c2Cl)=O)c[nH]n1 S(=O)(=O)(c1nc(N2CCC(Cc3nccs3)CC2)ccc1Br)N(CCOC)C c1(C(=O)NCCNC(=O)NC2(c3ccc(Br)cc3)CC(C)C2)ccn2nccc2n1 C1(CCNC(CNC(=O)OC)=O)CC(NC(C)COCC2CCC2)C1 Cc1c(C(N2CC3(C2)CN(C(=O)CC2CC2)C3)=O)nc2sccn12 Cc1cc(C#N)cc(C)c1C(=O)NC1CN(C(c2cnn(CCO)c2)=O)CC1C c1(CNCC(CC)SCC(F)(F)F)ccn(C(C)(C)C)n1.c1(S)nnnn1CC(F)F CCC(C#N)C(=O)NCC(C)N(C(c1ccnn1C1CCC1)=O)CC S(=O)(=O)(c1ccc(C)c(C(=O)NCC2CC(O)CN2C(=O)CNC(C)=O)c1)NC c1(C(=O)NC(CCN(C(C)C(=O)NC(N)=O)C)C)cnc2c(c1)nnn2C N1(C(C2C(CC)CCC2)=O)CCC(CC2CCN(C(=O)C(O)C3CC3)CC2)CC1 c12cccc(c1)CS2.CCC(C(=O)NCCOCCNC(C1(F)CC1)=O)OC C1(NC(C(C)SC)=O)C=CCN(C(c2cccnc2N)=O)C1 c1(C(N2C(CNC(CC(=O)N(C)C)=O)COCC2)=O)c(F)cccc1Cl N1(C(Cc2cc(OC)no2)=O)CC(NC(=O)CCN2CCOCC2)C2(CCC2)C1 C1(NC(C(C=C)O)=O)C2CC3CN(C(c4cnc(SC)nc4O)=O)C1C3C2 C(=O)(CCCCC(C)(C)OC)NC1C(NC(c2c[nH]c(=NC)s2)=O)C1 N1(c2n(CCOC)c(C(C)(O)COC)nn2)CCC(C2Cc3ccccc3C2)C1 Cn1cc(C(F)(F)C(=O)N(C2CCNCC2)Cc2ccc(C#N)cc2)ccc1=O N1(C(c2n[nH]cc2Br)=O)CCN(C(=O)CN2CC=CC2)C(C2CCCC2)C1 CC(C)C(C(=O)NCC12CC(NC(=O)CC(O)c3ccccc3)(CO1)C2)C1CC1 C1(c2nnnn2C2CCC2)(NC(c2onc(CSC)n2)C)CC2CC2C1 N1(C(CCC#CC)=O)CCC(C)CC1C(=O)NC(CCOC)C(C)C C1(NC(=O)C(=O)NCC(F)F)CC(O)(CNC(=O)Cn2cnnc2)C1 c1(C(=O)NC2(C(=O)NC3CN(C(C(CSC)OC)=O)C3)CCC2)cccc(Cl)c1 C1(NC(C(CC=C)C)=O)CC2(C1)CN(C(C1CNC(=O)N1)=O)C2 C1(C(N2CCC(NC(c3cc(C(=O)OC)sc3)=O)C2)=O)CC12CC(F)(F)C2 CCCCCC(C)CC(=O)NC1CCN(C(=O)COc2cccnc2)CC1F Cn1ncc(Br)c1C(N1CC(NC(c2cc(=O)cc[nH]2)=O)C1)=O C1(C(=O)NCc2cnc(CC)s2)CC(F)(F)CN1C(c1ccc(F)cc1C)=O c1(OC(=O)NC(C(=O)OCCC(C)C)NC(=N)NC(C)(C)C)ccccc1OC N1(C(C2CCN(C(N(CCC(=O)NC)C)=O)C2)=O)CCN(C)C(CO)C1 N1(C(Cn2c(C)nc(C)n2)=O)CCC(CNC(=O)C(C(C)C)NC(C)C)C(C)C1 CC1CN(C(c2occ(SCC)n2)=O)CC1CC(N1CCC1c1cccnc1)=O N1(C(C=CCOC)=O)CC2CCCC1(CNC(C1CCS(=O)(=O)CC1)=O)C2 C1(OC)CCC2(C(N3CCCC3CN(C)C(C3CCC(=O)N3)=O)=O)CC12 c1(OCCCNC(c2coc(CSC3CCC3)n2)=O)ccc([N+](=O)[O-])cc1F Cn1cc2c(n1)CCN(C(C1CC(NC(=O)CC(C)(C)CC(F)F)C(O)C1)=O)C2 CC(C)C(CCNC(C1CC1(C)C)=O)NC(c1cc(=O)n(-c2ccccc2)[nH]1)=O C1(NC(c2c(OC)nsc2OC)=O)CS(=O)(=O)CC1NC(=O)C(C)NS(C)(=O)=O c1(C(=O)NC2(C)CC(NC(C(CCC)OCC)=O)C2)cc(S(=O)(=O)N(C)C)c[nH]1 N1(C(c2c(C)csc2)=O)CCC12CN(C(c1cccc(C)c1F)=O)C2 CN1CC2(CCN(CC(=O)Nc3cccn3Cc3ccccn3)CC2C(=O)O)C1 C(CC(O)CNC(=O)COCC(F)(F)F)NC(=O)C(O)C1CCCC(C(=O)O)C1 N1(C(CC2(OC)CCC2)=O)CC2CC(NC(=O)Cn3cc(C(=O)OC)nn3)C1C2 c1(OCC)cc(C(=O)NC2CCC(C)(CNC(=O)C(C)C)C2)ccn1 C1(=O)C(C(C)C)O1.c1(CC(C(=O)NCCCC)SC(C)C)ccccc1Cl Cc1ccccc1C=CC(=O)NCCN(C(C1CC1F)=O)CC1CC1 CCC(C)CCC(=O)NC1(C(=O)NC)CC1.C1=CCNC(=O)C1 c1(C(N(CC(C)O)CCNC(=O)C(O)CC(C)(C)C)=O)cnc2nnc(O)n2c1 C(=O)(CC(C(F)F)c1ccccc1F)N1C(c2cc(COC)on2)COCC1 C1(CC)CC(C(=O)N(C)CC2(O)CN(C(=O)CC3(COC)CCCC3)C2)CCO1 c1(C(N2CC(C)N(C(=O)CSc3ccncc3)CC2)=O)c[nH]c2nccc-2c1 c1(NCC2CCN(CCCN)CC2)cccn2nnnc12 C1(C(=O)NC2CC2)CN(C(=O)C(CCc2ccsc2)N2CCCC2)CCO1 C12CC3CC1CC3NC2=O.O=C1CN(C(C2CCSC2)=O)CCN1 C12CC(F)(C1)C(=O)N2.c1(CN(CC(=O)N(C)C)C(=O)OC(C)(C)C)ccccc1 C12(CC(=O)NC(=O)CC3(NC(=O)CCCC4CCC4)CC3)CCCC1C2 C1(NC(C2CC23CC3)=O)CCN(C(c2cc(C(F)F)[nH]n2)=O)CCC1CO CC1(CC(N2CCC(NC(=O)COC(F)(F)F)C2)=O)CCOCC1 N(C1CCCNc2ccccc21)C(=O)CNC1(n2cnnn2)CCSCC1 C1(CC)CCC(C(=O)NCCC2CN(C(=O)Cc3nncs3)C2)CC1 Cc1ccc(C(=O)NCC(CC(C)C)NC(C2C(C)CC2C)=O)c(F)c1F c1(N2CCCCC(COCC)C2)ncnc(Cl)c1NC(c1cccnc1NC)=O C(c1ccc(C)c(C)c1)=CC(=O)NCC1C2N(C(C(C)SCC)=O)C(CC2)C1 n1(CNCC(=O)Cc2coc(C(F)F)n2)cnnc1C(C)(C)C.C12CC1C(=O)N2 c1(-c2sc(NC(c3cc(C)no3)=O)c(C)n2)ccc(N2CCC(N)CC2)cc1 C1(NC(=O)CCCCC2CC2)CCC2CCN(C(C34CCC(C3)OC4)=O)C1C2 C1(CC)CN(C(=O)Cn2nnc(C3CC3)n2)CCN1C(=O)CCc1cccnc1 C(=O)(CC1=NNC(=O)C1)N1CCC(CC=C)(NC(c2ccccc2NCC)=O)C1 C(=O)(C(C)(C)S(C)(=O)=O)NCC(CNC(C(C)(C)Cc1cnn[nH]1)=O)O Cc1cc(CN(CCC#N)CC(=O)N(N2CCOCC2)Cc2cccnc2)co1 C12(NC(C(=O)NC(C(=O)NCC)CC)=O)COC(COC)(C1)C2 N1(CC)CCC(C(=O)NC(CN(C)C)C(N2CC(C)(C)C2COC)=O)CC1 CC1CN(C(c2occc2C2CC2)=O)CCC1NC(c1ncn(C)n1)=O C1(C(=O)NCC2CC(NC(Cc3ccc(C)cc3C)=O)C2)OCC2CCCCC12 N1(C(c2cn(CC)nn2)=O)CCN(C(=O)CC(C)(C)O)C(CC(F)F)C1 c1(C(N(C)CC2N(C(C(C)NS(C)(=O)=O)=O)CCCC2)=O)ccc(N)c(Cl)c1 c1(CC)cccc(OCC(=O)NCC(C2CCC2)NC(c2cc(O)n(C)n2)=O)c1 Cc1cnccc1-n1nc(C2CCCO2)nc1-c1cc(-c2ccco2)on1 C1(C(C)C)CN(C(c2ncoc2Br)=O)CCN1C(=O)CC1CCCC(=O)C1 CC1CCC(C(=O)CCC(=O)N2CCCC(C(N3CC=CC3CF)=O)C2)CC1 CCCCCC(O)C(=O)NCC1(C(=O)N=c2cc(Br)[nH][nH]2)Cc2ccccc2C1 C(=O)(C(C)c1ccsc1)N(C(CNC(C1(C(=O)OC)CC1)=O)C1CC1)C C1(CCC(=O)N2CCCC2)CCC(=O)N1.C1(CC(C)N)CCN(C(=O)CN)C1 c1(C(N2C(C)(CNC(C(CC=C)C)=O)CCC2)=O)ccc2nc(C)ccc2c1 c1(C(=O)NCC(C)NC(C2CCCC3(CC3)C2)=O)cc2c(o1)CCCNC2=O C1(C#N)(OC)CC(C(=O)NCC(O)CCNC(=O)C=CCn2cncn2)C1 C12(COC)CC(CNC(=O)CCN3CCCC3)(CN1C(=O)C(C)CSC)C2 c1(C(=O)NC2CCCC(N(C(c3ccc(CC)o3)=O)C)C2)cc(N)c(Cl)c(O)n1 C1(C(N2CCC3CN(C(C(=O)NC4CC4)=O)CC32)=O)Cc2ccc(F)cc2C1 c1(C(N(CCC(=O)NC(C)CC2CCC2)CC=C)=O)coc(COC)n1 N1(C(C(=O)NCC=C)C)CCC(NC(=O)Cc2cc(O)nc(O)n2)CC(C)(C)C1 C(=O)(C1CCc2cccc(F)c21)NCC(N(C(c1scc(C)c1)=O)C)C1CC1 c1(OC)ccc(-c2nc(C)cs2)cc1CNC1(c2cccc(Cl)n2)CC1 c1(C(N(CCNC(c2ccn(C(C)(C)C)n2)=O)CC)=O)cc(OC)c(C2CC2)nn1 C1(CNC(c2ccc(C)s2)=O)CC(C)N(C(=O)C=Cc2ccsc2C(F)(F)F)C1 c1(OCC(N2CCC(CNC(C(C)c3ccco3)=O)C2)=O)ccc(F)cc1Cl Cc1cc(C(=O)NC2(C(N3CC4CC=CC3C4)=O)CC2(C)C)nc(C)n1 c1(NC(CNC(CC(n2ccc(C)n2)C)=O)C2CC2)nc(Cl)nc2sccc12 N1(C(Cc2c(CC)cccc2)=O)CCC2(CC1)CN(c1nccc(C)n1)CCO2 c1(-n2c(-c3c(-c4c(OCC=C)cccc4)cn(C)n3)ncc2)c(C)cccc1C n1(Cc2ccccc2)nc(C2CCCCC2)nc1C1CCS1(=O)=O Cc1nc(C(F)(F)F)c(C(N2CCC(NC(=O)CC3CCOC3(C)C)C2)=O)s1 c1(CCNC(C2CCC(NCc3ccc(C)cc3O)C2)=O)c(Cl)cc(Br)cc1Cl c1(CNC2C(C(=O)Nc3cccc(CC)c3)C2)cccc(OC)c1Br C1(CNC(c2cc(=O)cc[nH]2)=O)CCCCN1C(c1cn(C(F)F)cn1)=O Cc1cc(CCNC(C2CCCN2C2CCCCC2)=O)ccc1Br c1(CC)ccc(CC(N2CC3C(CNC(=O)COC4CC(F)(F)C4)C3C2)=O)cc1 C1(NC(Cn2nnc(C)n2)=O)COC2(C1)CN(C(C1CCCC1C(=O)OC)=O)C2 N1(C(COC)=O)CCc2ccc(C(=O)NCC3CC(O)C(O)C3)nc2C1 N1(C(C=C(C)C)=O)CCCCCC(NC(C2CCCN2c2ccccc2)=O)C1 C1(CCOC)CN(C(c2cc(O)nc(Cl)c2)=O)CCN1C(=O)CC(O)C(C)C C(=O)(C1=NN(CCO)C(=O)CC1)NCCC1CC(NC(C(C2CC2)OC)=O)C1 C1(CC(=O)NC(CNC(c2ccn(CC(C)C)n2)=O)(C)CO)CC2CCC1O2 c1(CNC(C2COCC2Cn2cc(CCC(=O)NC)nn2)=O)cccc(CO)c1 C12(C(=O)NC3CC(NC(C(C)(C)NS(C)(=O)=O)=O)C3)CCCC1(C(N)=O)C2 c1(NCC(=O)NCC2N(C(CC(C)SC)=O)CC=C2)ccccc1[N+](=O)[O-] c1(CCC(N2CCC(CC(=O)NC(C)=O)CC2)=O)ccc(C(F)(F)F)c(F)c1C c1(C(=O)NCC(CCCC)NC(c2ccc(Cl)c(N)c2)=O)nnn2c1CCCC2 N(C(=NCC1(c2cccs2)CCCCC1)N1CCCC(C)(N(C)C)C1)C(CC)C Cc1cc(OCC(=O)N(CC(C)NC(C2CC(C)(F)C2)=O)C)ccc1Cl C1(COC)(NC(=O)Cc2cc(CC3CC3CF)no2)CCN(C(C)=O)CC1 C1(C2CCCCC2)(C(=O)NCC2CN(C(CCSCC(N)=O)=O)CC2O)CC1 Cc1cn2cc(CC(N3CC(CNC(=O)COC4CC4)C4(CC4)C3)=O)nc2s1 C1(C(=O)NC2CCN(C(C3(c4ncccc4F)CC3)=O)C2)C2CCC(F)(F)C12 N1(CC(=O)NCC(C)(C2CCC2)OC)CCN(C(C2(CO)CCCO2)=O)CC1 N1(C(c2c(C)snc2)=O)CCN(C(c2cccs2)=O)C(CC(F)F)C1 c1(C(N2CC(N(C)C(C3CC(c4ccccc4)O3)=O)C2)=O)c(Cl)cccc1Cl C1(C(N2CC(NC(C3(CC=C)CCOCC3)=O)C(O)C2)=O)CC2(CCC2)CO1 c1(C(=O)OC)cc(C)nnc1NCC1(F)CC(NC(=O)CN2CCS(=O)(=O)CC2)C1 c1(NC(C2(CC(C)C)CC2)=O)cn(C)nc1C(F)F CC1(F)CCC(C(=O)NC2C=CC(C(=O)NC3(C)CC(F)(F)C3)C2)CC1 N1(C(C(CCC)O)=O)C2CCC1(C1(C(=O)Nc3cnn(C)c3)CC1)CC2 c1(C(=O)NC(C)CC(C)NC(=O)Cc2cnsc2)cnc2c(c1)COCC2 C1(CC)CN(C(c2ncoc2C)=O)CCC1NC(=O)C(C)(C)c1nccs1 c1(C(=O)NCC(CO)NC(C(CC#C)C2CC2)=O)c(C)[nH]c2ccc(F)cc12 N1(Cc2c(OC)c(Cl)ccc2)CC2CCC1CN2C(c1nc(Cl)sc1Cl)=O c1(C(=O)NCCCN(CCCNC(c2scc(C)c2)=O)C)cccc2sncc12 C1(C)(NCCS(=O)(=O)NC(Cc2c(C)nccc2)=O)CCCN(S(C)(=O)=O)C1 c1(C(N(C(C)CNC(=O)CCC2CCCN2C)C)=O)ccc(S(=O)(=O)N(C)C)o1 C1(CCC)(NC(=O)C(N)=O)CCN(C(c2cc([N+](=O)[O-])sn2)=O)CC1 C1(C(N2CCC(N(C(c3ccc(SC(F)(F)F)o3)=O)CC)C2)=O)NC(=O)OC1(C)C c1(NC(C2N(C(c3c(N(C)C)cccc3)=O)CCC2O)=O)cc(O)ccc1Cl C(CCCCNC(=O)CCCc1ccc(C)s1)N(C(C(C)SCCCC)=O)CC c1(C(N(CCOCCN(CC)CC)C)=O)ccc(Nc2nnnn2C)c(F)c1F C1(CC(=O)N(C2C(NC(C(C)OCCC#C)=O)CCCC2)C)CN2CCC1CC2 N1(C(=O)CN2CC3CCC2C3)CCN(C(C2C=CCCCC2)=O)C2CCCC12 c1(OC)cc(C(=O)NC2CC(O)(CNC(C3CCCOC3)=O)C2)c(C)cc1O c1(-c2ccc(NC(Cc3ccc(C)s3)=O)cc2)cnc2n1CCCC2 c1(SC(C(=O)NCC(CC)NC(c2nocc2Br)=O)C)ccccn1 CCCCC(CN(C(=O)C(CC1CC1)NC(=O)C=C(C)C(C)(C)C)C)CC C(C(CC(F)(F)F)NC(=O)C(C1(C)CCC(=O)C1)=O)NC(C=CC(=O)N(C)C)=O C(=O)(CC(C)CC(=O)NCC1(O)CN(C(=O)CCCC2CCOCC2)C1)OC CCCCCC(CC)C(=O)N(CCCOCCN(C)C(c1ccc(C)cc1)=O)C C1(NC(c2scc(OC)c2)=O)CCCCC1CNC(c1c(C)cnn1C(C)C)=O C(=O)(C(C)C(C)O)N(CCOCCCNC(c1cc(C(C)C)no1)=O)C N1(CC)CCN(CC(N2CCC(NC(=O)C(CC(C)C)OC)CC2)=O)C(=O)C1=O CCC(CC(=O)N1CCC1CC1CC1)NC(c1ccn(C)c1C)=O C(=O)(C1=NOC(C)(C)C1)N1C(CNC(c2c(C)nc(F)cc2)=O)COCC1 c1(CC)cc(C(N2CCC(CC)C2C(N2CC(C(=O)OC)C2)=O)=O)c(C)o1 c1(C(=O)NCCC(CNC(=O)C2=CCSC2)O)nccc2c(Cl)cccc12 c1(C(=O)NCC(CO)OC)coc(CNC(=O)C(C)CO)c1 C1(C)(CNC(C(C2CCOCC2)OC)=O)CCCN1C(c1cccc(C2CC2)c1)=O C=CC(C)CN=C(NCC1CCCN1C)NC1CCOC(C2CCC2)C1 Cc1cn(C2CCOCC2)nc1C(=O)N(C(C)CNC(=O)CC1CC1C1CC1)C c1(C(N2CCC(CCOC)(NC(C3(Cl)CC3)=O)C2)=O)c(O)cccc1O c1(CC(=O)NCC2CC(F)CN2C(C2CC23CC3)=O)cnn2c1CCCC2 C1(CNC(c2cnc(CC)o2)=O)CCCCN(C(=O)C#CC2CC2)C1 c1(C(N)=O)ccc(C(=O)NCC2CC(O)(CNC(=O)C3=CCSC3)C2)cn1 Cc1cc(F)ccc1S(=O)(=O)NC1CN(C(C2(F)CC2)=O)CCC1F CCC(C)(CO)C(=O)N1CCOC(CC(=O)NC2CC3(CCCC3)C2)C1 C1(C#N)(C(=O)NCCCC(C)(C)NC(CCOC(C)C)=O)CC2CCC1C2 C12(C(=O)NCC(c3ccc(C)cc3)NC(C3CC(CF)C3)=O)CC(C)(C1)OC2C C(=O)(C(F)C(F)(F)F)N(C1CN(C(c2cc(COC)sc2)=O)C1)C Cc1cnsc1C(=O)NCC1(O)CC(C(=O)NC(C)CCc2cn[nH]c2)C1 N1(C(=O)OC(C)(C)C)CC2CC1CN2C(C1(S(C)(=O)=O)CC1)=O C1(CNC(c2cn(CCCC)nn2)=O)CN(C(C2CC(OC)C2)=O)CCO1 c1(C(=O)Nc2cccc(C3CCCCC3)c2)cc(Cl)c2ncccc2c1F C1(C(=O)OC)CCCC1NC(=O)N(C)Cc1ccnn1C C1=CC(=O)Oc2ccc1c(C)c2.c1(CC(=O)N(CCOC)C)cncc(F)c1 C1(OC)CC(CCNC(=O)Cc2ccoc2C)N(C(C2CC3CC3C2)=O)C1 N1(C(CC(n2ccc(C)n2)C)=O)CC(NC(c2cc(N)cc(F)c2)=O)C(C)(C)C1 C12(CNC(CC=C)CO)CCC1CNC2 C1(NC(=O)CO)CCN(C(=O)Cn2nc(C)cc2C(F)F)C(C)C1.C(C)=CC N1(C(C2(OC)CCC(C)CC2)=O)C2CCC1CN(C(=O)CSC(F)F)CC2 C(=O)(CCCCCCCNC(=O)OC(C)(C)C)N1CCC(OCC)C(C)(CC)C1 C1(CC)CN(C(=O)C(O)C2CCC2)CC1NC(=O)C(Cc1ccccc1)N(C)C C1(NC(CCCCCC=C)=O)CCCCC12CCN(C(=O)C(C)=C(C)C)C2 c1(C(=O)NCC2(NC(C(C)C3CCCO3)=O)CCOCC2)cc2[nH]ccc2s1 c1(OC)ccc(N)c(CC(N2CCC(NC(=O)COCC(C)C)C2)=O)c1 c1(C(N2CCC2C2CCC2)=O)ccc(CC2CCC2)cc1 C(CC(=O)NCc1ccc(O)nc1)(C(F)(F)F)NC(C(CCC)C#N)=O C1(CN(C)Cc2ccccc2)CN(CCl)CCO1.N1(C(=O)OC)CCC(CS(N)(=O)=O)C1 C1(C(N(CCCC)C)=O)CCN(C(=O)CCc2cncnc2)C(C)(C)C1 N1(CC(=O)NCCN(C(C2(C(=O)N(C)C)CC2)=O)CC)CCOCC1=O c1(OCCNC(CCc2ccc(OC)cc2)=O)ncc2ccnc-2[nH]1 CC(C)C(C)CCNC(=O)CC1CCN1C(=O)C(C)NC(C)(C)C C=C(Cl)C(C)(C)C(=O)N1CCN(C(c2cc(OCCOC)ccn2)=O)C(CF)C1 c1(N2CCC(CNC(CCc3cc(C)no3)=O)CC2)ncnc2scc(C)c12 N1(C(CCN(C(COCC(=O)NC)=O)C)=O)CC(C)CCC1C C1(CNC(C(C2CS(=O)(=O)C2)OC)=O)(NC(=O)Cc2nc[nH]n2)CCCCCC1 C=CCCCCC(C(=O)NC1CCOCC1)N(c1ccc(F)cc1)CCN(C)C C1(CC(=O)N(c2cccc(C)c2)C)CCCN(C(=O)CN2CCCCC2)CC1 C1(CNC(c2cnc(C)[nH]2)=O)CC(NC(=O)C(C)C2CCC2)C1(C)C O=C1NCC2(CCN(C(=O)CC3CCCN3C(C3CCc4nc[nH]c4C3)=O)CC2)O1 Cc1cc(Cl)c(C(N2CCCCC(Nc3cccc(NC(N)=O)c3)C2)=O)cc1N c1(C(=O)NC2CCN(C(CCCCOC)=O)C(C)C2)cc(C)sc1S(N)(=O)=O N1(C(C(C(=O)OC)C)=O)CCC(CNC(=O)COCCOCC(F)(F)F)(CO)CC1 N1(CC(N2C(CC(N3CCC(N(C)CC)C3)=O)CCC2)=O)CCCCC1C c1(CC(C(=O)NCCC2CCN(C(=O)Cc3cccnc3)C2)O)ccccc1Cl N1(C(c2ccnc(F)c2OC)C(=O)NCCOC)CCC2CN(C)CC2C1 C1(NC(CCC2C(C)(C)C2)=O)CC2CCCC(C1)N2C(=O)C=Cc1cccnc1 C1(C(=O)NCCCOCCNCCN(C(CN(C)CCO)=O)C)CCOC1 c1(C(=O)NC2CC(C)(NC(c3ccc(-c4cn[nH]c4)cc3)=O)C2)nccc(Cl)c1F Cn1nccc1C(F)=CC(=O)NC1(CCNC(C2(C(C)(F)F)CC2)=O)CC1 C#CC1(C(N2CC(O)(CC(C)C)C2)=O)CCN(C(=O)CC(CC)C2CC2)CC1 c1(-c2cc(C(N(CC(CC)NC(=O)C3=CCC3)C)=O)sn2)ccc(F)cc1 c1(C(C(N2CC(CNC(=O)C(=O)NC3CC3)CC(C)C2)=O)=O)occ2c1CCCC2 n1(CC)ccc(C(=O)NC2CCCCC2NC(c2occc2OC)=O)c1C c1(CC(=O)NCCN(C(=O)CCC2CC2(F)F)C)ccc(O)nc1 n1(CCN(C)C)cc(C#CCNC(=O)Cc2ccncc2)nn1 N1(C(c2c(CC)scc2)=O)CC(NC(C2(CC)CCCO2)=O)CC(O)C1 c1(C(N2CCS(=O)(=O)C(CCNC(C3(Cl)CC3)=O)C2)=O)nccn2c(Br)cnc12 c1(CN2CCC(C(=O)NCc3ccccc3C3CC3)CC2)ccc(O)c(F)c1 c1(C(=O)NC(c2ccccc2I)C2CCNCC2)cc(F)ccc1C(F)F C(=O)(CC1=CCCC1)N1CCC(N(C(C(C)NC(C)=O)=O)C)CC1 C12(C(=O)NCC3CC(C)N(C(=O)COC(F)(F)F)C3)CCC(C)(CC1)OC2(C)C C12(C(N3CC(NC(c4coc(C(F)(F)F)n4)=O)C3)=O)CCC(CC1)CO2 c1(C(=O)NCC2CCN(C(COC(C)=O)=O)C2(C)C)ccn2c(C)cnc2c1 CC(C)C(C(=O)NC1(CNC(=O)CCN2C(=O)CCC2=O)CCOC1)NC(N)=O c1(CC)ccc(NC2CCOCC2C(=O)OC)c(Br)c1 N1(C(CCOC)=O)CCCC(CCN2CCN(C(=O)CC(C)COC)CC2)C1 C1(C(N(CC(=O)N(C(C)CCO)C)C)=O)CC2CCC2C1 CC(C)(C)CCCCC(=O)NCC1(F)CCN(C(C2CC(C#N)C2)=O)C1 C1(C(N2CCN(C(CNC(CCCN=[N+]=[N-])=O)=O)CC2)=O)CCN2CCOCC12 N1(C(c2nc(C)cc(SC)n2)=O)CC2C(C(F)(F)F)CC2(N)C1.C(=O)O C12(CNC(c3cnc(C4CC4)s3)=O)CC(NC(c3ccco3)=O)(CO1)C2 c1(OCCCC)ccccc1C(c1nnnn1C1CCCC1)NC(C)C(CC)CC C(C(C)C(C)C)(C1CC1)N.c1(-c2cc(CC=C(C)C)on2)ccc(C)cc1 c1(OCCCOC)ccc(CN2CCCCC2C(=O)O)cc1 c1(N(C(C)CNC(=O)Cc2cccc(O)c2)C(C)=O)ccc(OCC(F)(F)F)cc1 C1(C(=O)NCC(CSC)(C)C)CC2CCC1N2C(C1CC2C=CC1O2)=O c1(C(N)=O)ccc(C(=O)NC23CC(CNC(C4CC4C4CC4)=O)(C2)C3)o1 C1(NC(C(C(C)C)SC)=O)C2CC1N(C(=O)CCc1cncc(Br)c1)C2C C(=O)(C(CC(F)F)NC(c1cnsn1)=O)NCC1(S(C)=O)CC1 C(=O)(CCC(C)OC)NCC(C1CCC1)NC(CNC(CC)=O)=O N=c1[nH]n(CC(=O)NC2(CNC(=O)C(F)n3ccnc3)CCC2)c(=O)s1 c1(C(N(C)CC2N(C(CC(C)SC)=O)CCCC2)=O)ccc(=O)n(C2CC2)c1 C(=O)(CCCCC(=O)N1CCCC1C(=O)N1OCC(C)O1)OC C12(CNC(C(CCOC)(C)C)=O)CCCCC1N(C(C1CC(SC)C1)=O)CC2 c1(CC)cc(OC)ccc1C(=O)NCCCNC(c1cnc(OC)s1)=O N1(C(COCC(C)C)=O)CCCC1C(C)NC(=O)CC1C=CCC1 C=C(C)CCC(=O)NC(C)(CNC(C1(CS(C)(=O)=O)CCOCC1)=O)CO C1(C2CCCN(C(c3nnc(C)cc3O)=O)C2)(NC(Cc2cnc(C)s2)=O)CC1 c1(OC)cc(C(=O)N(C(C)CCNC(=O)C(C)=C2CC2)C)c(Br)cc1C N1(C(CCNC(C2C(C)C2)=O)=O)CCCC(O)(CCNC(=O)C=CC2CCC2)C1 c1(C(N2CC(CNC(c3ncccc3Cl)=O)C3(C2)CC3)=O)cnn2cccnc12 C(=O)CCCC(=O)N1CCC(C(=O)NCc2scnc2C)C1C(C)C CC1CC(NC(C2COCCN2C(c2cc(C(N)=O)co2)=O)=O)C(=O)O1 C1(C(=O)NC2(CF)CCN(C(CCNS(C)(=O)=O)=O)C2)CCC(=C(F)F)CC1 C1(NC(N2C(C)CN(CCO)CC(C)C2)=O)Cc2c(O)cccc2N1C(C)(C)C CCCCC(C(=O)NCC(N1CCC2(CCC2)CC1CO)=O)C(C)C C(=O)(C(C(=O)OC(C)(C)C)OC)NCCCCSC.C12CCC1N(CC)C2=O N1(C(c2c(C)c(F)ccc2)=O)CC2=C(C1)CN(C(=O)C1=CCCN(C)C1)C2 N1(C(c2ccc(C)c(F)c2)=O)CC2C=CC1C(C(=O)NC1C=CCCCC1)C2 C(=O)(C1=CC(O)C(NC(C2(F)CCCC2)=O)C1)N1CC(C)C(F)(F)C1 C1(CC(=O)NCC(=Cc2ccco2)C)CCCCN(C(=O)OC(C)(C)C)CC1 N1(C(=O)CCOCC2CCCO2)CCCCC(C2CN(C(=O)C(O)C3CC3)C2)C1 c1(CN(CC(CC(=O)OCCCCCC)C)C=O)[nH]c2ccccc2c1C C1(NC(c2cc(OC)nn2C)=O)CC(F)(F)CC1NC(c1cc(C)c(C)o1)=O c1(CC(=O)NCC(CC)NC(c2ccsc2C)=O)c(C)ncnc1C N1(C(c2cc(C)ncn2)=O)C2CCC(C2)C1C(=O)NCC1(F)CC1 c1(C(=O)NC(C2OCCN(C(Cn3nnc(C)n3)=O)C2)C)c(C)ncn(C)c1=O C1(C(N2CCC(C(=O)OC)C2C)=O)C2CCN(C(c3nnn(C)c3N)=O)CC12 N1(CC(=O)NCCN(C(=O)CSc2ccnc(Cl)c2)CC2CC2)CCCNC1=O C1(C)(C(=O)NC23C(CN(C(Cc4n(C(C)C)ncc4)=O)C2)C3)CCCNS1(=O)=O c1(OC)ccc2c(c1)C(C(C)C)N(C(C1CC3CCCC3C1)=O)CC2 c1(C(=O)NC(CC)(CC)CCNC(=O)CC2CC2)ccc2c(c1)CC(C)O2 Cc1ccc(Cl)c(F)c1C(=O)NC1CCN(C(c2ccc(N)c(N)n2)=O)CC1F c1(C(=O)NC(COCC)C(=O)NC2COCC2N=[N+]=[N-])cc(F)ccc1O C1(COC)(NC(c2cccc(C3CCCOC3)c2)=O)CCN(C(C)=O)C1 C=CC(C(F)(F)F)NC(=O)C=CC1CCCN1C(c1oc(C)nc1CC)=O n1(CCC(=O)NCC2N(C(C(C)NC(COC)=O)=O)CC2)cc(Br)ccc1=O c1(C(=O)NCC2C(NC(c3ccc(CCC)[nH]3)=O)C2)cnn(CC)c1C C1(C(=O)NCC(c2cncnc2)C)CC2CCC(C1)N2C(=O)Cc1cnsc1 C1(CCC)(NC(=O)CC=CCc2ccccc2)CCCN(C(=O)C(C)(F)F)C1 c1(-c2cnc(OC)c(C)c2)cccc2c(C(=O)Nc3ccc(C#N)nc3)[nH]nc12 N1(C(=O)CCn2ccnn2)CCCN(C(=O)C=CC(F)(F)F)CC1c1ccccc1 CC1(C(=O)NCC2CC2NC(c2cc(Cl)c[nH]2)=O)CCC(F)(F)CC1 c1(C(=O)NC(CN(C(c2oc(C)c(Br)c2)=O)C)C)c[nH]c(=N)nc1O c1(CC)cc(CC(N2CCCC2CN(C(=O)C(C)=C2CC2)C)=O)n(C)n1 c1(C(N2CC(N(C(CC(C)OC)=O)C)C3(C2)CC3)=O)[nH]c2ccccc2c1C#N n1(C2CCN(C(=O)NC(C)(C)F)C2)c(O)nc2cccnc12 C1(CC(=O)N(CC(=O)NCC)C)CCC(NC(=O)Cn2cc(C)cn2)C1 C(=O)(C(CC(C)C)C(N)=O)NCC1CCN(C(Cc2c(C)nc(C)s2)=O)CC1O C(CN(C(=O)CCC1CCCCO1)C)(CO)(CO)NC(C=CC(=O)OCC)=O N1(C(c2nc(NC(=O)CCc3nccs3)sc2)=O)CCC2(CC1)CC(CO)C2 C(=O)(CCCCC(C)(C)C)NC(CC#C)C(=O)N1CCC(OCC=C)C1 c1(CC)c(C(N2CC(CNC(=O)CSC(C)(C)C)CC2C)=O)oc2ccccc12 C1(NC(COC)=O)CC(F)CN(C(c2c(Br)c(C(F)(F)F)nn2C)=O)C1 C1(NC(CCC(=C)Cl)=O)CC2CC1CN2C(=O)CC(=O)OC c1(OC)cc(Cl)c(NC(=O)C(N2CCC(c3ccccn3)CC2)=O)cc1OC N1(C(Cc2cnc(C)[nH]2)=O)CCC(NC(=O)Cc2cc[nH]n2)C1c1ccccc1 c1(N(C(=O)CNCS(=O)(=O)NCCC#N)CC)ccc(S(N)(=O)=O)cc1[N+](=O)[O-] N1(C(CCCC(C)(C)C)=O)CCCC(C2CC2NC(C2CC23CCSCC3)=O)C1 C1(C(N(CCCC(=O)NCCCOC=C)C)=O)CCC(C)(C)C1 C1(NC(c2ccnc(S)c2)=O)CCCC(CNC(=O)CCc2cncs2)C1 N1(CC)CCN(C(c2cccc(C(C3CC(F)CN3)=O)c2)=O)CC1=O N1(C(CCCCC#N)=O)CC(NC(C2CC2c2ccsc2)=O)C(N=[N+]=[N-])C1 O=S(=O)(c1ccc(NCc2cncc(Br)c2)c(Cl)c1)N1C2CCCC1CCSC2 c1(N2CC(Br)=C(C)CC2)nc2c(c(=NCCS(=O)(=O)C(F)F)[nH]1)CCC2 c1(CC)cscc1C(N1CCC(n2cc(C3CCOC3)nn2)C1)=O N1(CCCC(=O)NC(C)CCNC(C2CCS2(=O)=O)=O)C(=O)CN(C)C1=O c1(C(=O)NC2C(N=[N+]=[N-])CN(C(C3(F)CCC3)=O)C2)ccc2c(c1)C(=O)NCC2 CCC(CC(=O)NCC1C2CCC(C2)N1C(c1cc2c[nH]cnc-2n1)=O)C(F)F Cc1nc(NC2CC2)sc1C(=O)NCCC(C)CCNC(=O)C(C)(C)C N1(CC)CC(C(=O)N(C(C)CCNC(c2sccc2OC(F)F)=O)C)CC1=O N1(C(C(CCC)C)=O)CCN(C(=O)CCCc2ccc(Br)cc2)C(C(C)C)C1 C1(N(C(C2C(CC)CCCN2C(=O)CC2(O)CCOC2)=O)C)CCCC(C)(C)C1 C1(NC(C(c2cscn2)N(C)C)=O)CCC(NC(=O)C(c2ccccc2)F)C1 Cc1nscc1Cn1ccoc1=N.C(=O)(C(=O)Cc1ccccc1)N1CCCC1 c1(C(=O)NC2CCN(C(CSCC(=O)OC)=O)C2C)ccc(Cl)c(C)c1Cl C(C(C(C)C(C)C)NC(=O)C1=C(C)CCC1)NC(C(CCC)=CCC)=O C1(CNC(c2ncccc2Br)=O)CCCC(NC(c2ccnn2CC2CC2)=O)C1 N1(CC)N=C(C(=O)N2CCC(NC(C3CN(S(C)(=O)=O)C3)=O)CC2C)CCC1=O CN1CCN(C(C2CCN2C(C)(C)C)=O)C(CNC(c2cnc(N)c(O)c2)=O)C1 C1(CNC(c2c(C)con2)=O)CC2(C1)CN(C(c1nc(Cl)c(Cl)s1)=O)C2 C12(NC(c3cccc(N4CCCNC4=O)c3)=O)CC1CN(C(c1cscn1)=O)C2 Cn1nc(O)cc1C(=O)NC(C1(O)CCCCC1)(C)C.C12CC1C(=O)N2 N1(C(C)(C)C)CCOCC(CNC(C2CCC(F)CC2)=O)C1 c1(C(=O)NC2CCC(NC(c3c(CC)ocn3)=O)C2)sc(C(F)(F)F)nc1C C1(NC(C=C(CC)CC)=O)CC(NC(c2cc(-c3ccccn3)no2)=O)CC1O C1(C(=O)NCCNC(=O)CCCn2cncn2)CCn2nnnc2C1 C1(NC(C(COC)CC(C)C)=O)CCC2CN(S(=O)(=O)C(C)C)CCC2C1 C1(NC(CN(C)CC)=O)CCN(C(C2CCOC(=O)N2)=O)C1C(C)C N1(C(C(CCCC)F)=O)CCC2C(CCN2C(=O)CCC(C)SC)C1 c1(C(=O)OCCN2CCc3ccccc3C2)cccc2ccc(O)nc12 C=C(C)CC(C(=O)NCCCCCCCC)NC(C1COC(=O)N1)=O CCCCCC(O)C(C)C(=O)NCC1CCN1C(c1occc1C)=O C12(CNC(COCCC#C)=O)CC1CN(C(=O)C(C(C)C)n1cnnc1)C2 CC(CC(=O)N(CCC(C)NC(c1csc(C2CC2)c1)=O)C)C1CCCCC1 N1(C(C(C(C)C)NC(C)=O)=O)CCN(C(=O)CCOCC2CC2)C(C)C1 N1(C(c2ccc(CC)o2)=O)CCCC1C1CCCCN1C(=O)CCc1cnc[nH]1 c1(C(=O)NCC2CC(NC(CCC=CCC=C)=O)C2)cccc2ncccc12 N1(C(C(CC(C)C)O)=O)CC2(C=C(C(=O)NCCCC3(O)CCC3)CO2)C1 Cc1cc(C(=O)NCC2(O)CCN(C(=O)CCC3CCCOC3)CC2)cc(C)c1 N1(C(C2N(C(C(C)=CC=C)=O)CCC=C2)=O)CCC(F)(F)C(O)C1 C1(C(=O)NCCCCNC(c2cnc(OC)s2)=O)CCc2nn(C)cc2C1 Nc1cc(C(=O)NCCn2cnc(C(N3CCCC(F)(F)C3)=O)c2)cc(F)c1 C(=O)(N=S(C)(=O)C1CC(C(=O)O)C1)c1cccc(C)c1.N1CCC(O)CC1 C12(NC(C(c3c(C)nn(C)c3)C)=O)CCCC1CN(C(=O)CC1OCCCO1)C2 C(=O)(CCC(F)(F)Cn1cc(CC(C)C(N)=O)nn1)NC(C1CCCCC1C)C CCN=c1[nH]cc(C(N2CCC(F)(CNC(c3csnc3SC3CC3)=O)C2)=O)s1 CC(C)CCC(F)C(=O)NC(Cc1ccoc1)C(=O)NC(C)(C)C(=O)NO c1(OC)ccc(F)cc1C(N1CC2C(C1)N2C(=O)CCCc1ccc(O)cc1)=O C(C)(CNC(=O)CC1CCOC1C)(CNC(c1cc(C(C)(C)C)on1)=O)OC c1(OC)cc(C(=O)NC2CCN(C(=O)C(C)OC3CCCC3)CC2)cc(OC)n1 c1(C(N2CCC(N(C(C(C(C)C)OC)=O)C)C2)=O)ccn2ccnc2n1 c1(NC2(C(=O)NCC(=O)NC)CCC2)ccc2c(c1)CNC2=O.C(C1CC1)C1CC1 c1(C2CCN(C(C3(F)CN(C(c4cccc(O)c4)=O)C3)=O)C2)ccc(Br)c(Cl)c1 N#CC1(CC(N2CCOCC2CNC(C2C(Cl)(Cl)C23CC3)=O)=O)CCCCC1 c1(CCC)noc(CCCC(=O)NC(C)C(C)(C)NC(C2CC2CC)=O)n1 C(=O)(C1=CC2(CCOC2)C1)NCC(C(=O)NC(CC(=O)OC)C1CC1)CC1CC1 c1(C(=O)NC(C(CC)SC)=O)ccc(Nc2nc(C(=O)NC3CC3)cs2)nc1 CCCC(CNCC(=O)Nc1cc(C)cc(Br)c1)C(=O)Nc1ccccc1 C(CCCCC(F)(F)F)ONC(CCC1(NC(C)=O)CCC(=O)N1)=O CC1ON=C(C(=O)NC2COCCC2NC(c2cccnc2S)=O)C1C C1(OC(C2CNC(c3ccccc3)C2)=O)Cc2ccccc2C1=O Cc1ccc(F)cc1C(=O)NCC1CC(C)N(C(=O)Cc2cccc(C)c2O)C1 c1(CN(C2CCN(c3nc(SC)nc(=N)[nH]3)CC2)CC)ccc(C)cc1[N+](=O)[O-] C=Cc1ccc(C(N2CCC(CNC(c3cnn(C)c3C)=O)C23CC3)=O)cc1 C1(NC(C=C(COC)C)=O)COCCC1C(N1CC(COC(C)=O)C1)=O N1(C(CN(CCOCCOC)C)=O)CCN(C(C)=O)CC1CCOC N1(C(c2c(C(=O)OC)cccc2)=O)CCCN(C(=O)CCSCC(N)=O)CCC1 C1(C(=O)NC2CCN(C(CC3C(C)(C)C3(C)C)=O)CC2F)CCN2CCOCC12 Cc1nc(O)nc(C)c1CC(N1CC(NC(c2ccc(F)cc2)=O)C2CC12)=O C1(CC(=O)N(C)CC2C3CN(C(=O)C4=CCCC4)CC23)CCC12CCC2 c1(CC)ccccc1C(N1CCOCC1CCNC(=O)CC1CN(C)C1)=O c1(C(=O)NC(C(C)NC(C(C)Sc2ccccn2)=O)(C)C)ccc(C)nc1N c1(C(=O)NCC(CC(=O)NCc2scc(C)c2)C)ncc(F)cc1N c1(CC(N2CCN(C(CC(=C)C)=O)C(CCO)C2)=O)csc2nc(C)cn12 C1(C)(C(=O)NCC(CN(C(c2c(CCC)[nH]cc2)=O)C)C)CS(=O)(=O)C1 N1(C(C2CCCN(C(c3cc(CC)ncc3)=O)C2)=O)CCc2nc[nH]c2C1 N1(Cc2c(C)cc(C(F)(F)F)cc2)CC(C)CCOCC1C c1(C(=O)NC2C=CCN(C(Cc3cnc(C)s3)=O)C2)ccc2oc(S)nc2c1 Cc1cc(C(=O)NCC2CC3CCC2N3C(=O)CC(C)(C)C2CC2)nc(C)c1 C12(C(=O)NC3C(C)N(C(=O)CCCSc4ccccc4)CC3)CCCC1C2(F)F c1(CNC(C2(CC(=O)NCC(O)CO)CCC2)=O)cc(C(F)(F)F)ccc1O N1(CC(=O)N(C)CCN(C)C(c2ccccn2)=O)CCCCCCC1=O CC(CCC(C)(C)C)NC(=O)CN1CCN(C(C2COCCC2C)=O)CC1 CCC(C)C(O)C(C)C(=O)NCC(c1cccc(Cl)c1)NC(=O)C=CCO Cc1nc(Cl)ccc1C(=O)NC1CCN(C(=O)Cc2sccc2C)CC1C N1(C(C(C(C)C)SC)=O)CCC2(CCN(C(c3sc(CO)nc3C)=O)CC2)C1 N1(C(C(CCSC)NC(=O)CNC=O)=O)CCn2nccc2C1 C1(C(=O)NC2CC(NC(CSCC(N)=O)=O)C2)CCN(C2CCCCC2)C1 N1(C(C(C)(C)F)=O)CCC(F)(CNC(=O)C=Cc2cscn2)C1 CCCCC(O)C(C)C(=O)NC(CCC(=O)Nc1c(C)cccc1O)C(C)C c1(CCC(=O)NCC2(O)CN(C(C3CC3c3cccs3)=O)C2)cccc(O)c1 C=CCC(CNC(c1cnc(O)cc1C)=O)C(=O)N(C(C)CC(F)(F)F)C CN1CC(NC(=O)COCCNC(C2(F)CC=CC2)=O)CC12CCC2 N1(C(c2[nH]c(=N)sc2)=O)CCc2nc(CNC(=O)C(O)CC3CC3)sc2C1 N1(C(c2c(CNC(COC3(C#C)COC3)=O)ccs2)=O)CCC2(CC1)CC2CO O(C1CCOc2ccc(-c3ccccc3)cc21)C(C1C=CCNC1)=O n1(CC)nc(C(C)C)cc1C(=O)NCCCC(CO)NC(=O)CC(C)COC c1(C(=O)NC2CCCC(NC(CCSCCCC)=O)CC2)c(C)nc(O)nc1C CC1(O)CCC(C(N2CCOCC(NC(=O)Cc3csc(S)n3)C2)=O)CC1 C1(NC(C(CSC)O)=O)CC1C1CCN(C(C2(C#N)CCOCC2)=O)CC1 C(C(=O)NCc1cn(CC(=O)NC)nn1)(C(C)C)SCC.C1(C(N)=O)CC1 N1(C(CCCC#CC)=O)CCN(C(c2cc(CS(C)(=O)=O)on2)=O)CC(O)C1 Nc1c(F)c(F)cc(C(=O)NCCN2CCN(C(=O)C=CCO)CC2)c1Cl c1(OC)c(F)ccc(C(N2C3CCC2CN(C(=O)CC2CC2)C3)=O)c1F c1(CC(=O)NCc2nc(CNC(C(CCC)OC)=O)on2)n[nH]c2c1CCC2 N1(C(COC2CCN(C(c3ccc(C(C)C)o3)=O)C2)=O)CCC(C)CC1C Cc1cc(O)c(C(C)C)cc1C(=O)NCCCN(C(=O)COCCCC(C)C)C C(C)(C(C)C(=O)NCC1(C(=O)NC2C3CCC2CC3)CCCO1)OC Cc1n[nH]c(=NC(=O)C2CCCCN2C(C(CCO)C(C)(C)C)=O)s1 Cc1ccc(C=CC(N2CC(NC(c3cc(C4CC4)cs3)=O)CC2C)=O)c(C)c1 N1(C(C=CC)=O)CCC(CNC(c2cnnn2C)=O)C(C)C1 c1(OC)ccc(NC(C2C=CC(NC(C34CCCCC3C4)=O)C2)=O)cc1C c1(NC(C(=O)NC(c2nn[nH]n2)C)C)cn(C2CCCC2)nn1 Cc1cccc(CSC(C)C(=O)NCC(C)CNC(C2CCSC2)=O)c1 c1(OC)nc(Cl)cnc1C(=O)OC.c12cscc1C(=O)NCC1CN(C1)C2 c1(NC(CNS(NCC(=O)Nc2ccccc2)(=O)=O)=O)c(F)cc(Br)c(Br)c1F CC1(O)CCC(C(=O)NCC2CN(c3cncc(Cl)n3)CCO2)CC1 N1(C(c2cc(C)c(O)c(N)c2)=O)CC(NC(C2CC2C)=O)CC2(CCOCC2)C1 N1(C(C2C(OCC)C2)=O)CCC(C)C(CNC(=O)COc2cccc(CC)c2)C1 c1(N(C)Cc2cc[nH]n2)nc(=NC2CCCCC2C(C)(C)C)[nH]c2c1cnn2C c1(OC)ccc(C(=O)NCC23CC(C(=O)O)(CCO2)C3)c(N)c1 C1(CCNC(Cc2nc(=N)[nH][nH]2)=O)CN(C(c2ncccc2Cl)=O)CCCO1 C1(C)(CC)NC(=O)N(CC(N2CC(NC(=O)C(F)F)C2)=O)C1=O C1(C)(C(=O)NC(C(C)C)c2cccs2)CCCN(C(c2cscc2Cl)=O)C1 C1(C(=O)NC(CCCC)CNC(C2C3CCCC23)=O)CCC2(CC1)CC2 CCC(N=c1nc(N2CCCC(N3CCC3)C2)c2cccc(F)c2[nH]1)C1CCC1 c1(C(=O)NCCC(CNC(c2sccc2CO)=O)OC)ccc(C)cn1 C1(CNC(=O)CC(=O)Nc2nccs2)CN(C(c2n[nH]cc2Cl)=O)C2CC12 N1(C(=O)COCC2CCC2)CCN(C(C2(c3cccs3)CC2)=O)C(c2cn[nH]c2)C1 c1(C(=O)NC(c2ccc(Cl)cc2)c2ccccc2)cc(F)c(F)c(F)c1N c1(C(=O)NCCCN(C(=O)C(C)Cc2ccco2)C(C)C)cnc2c(c1)CCC2 Cc1oc2ncc(C(=O)NC(C)(CNC(c3cnc(Cl)[nH]3)=O)CO)c(=O)n2c1C N1(C(C(C)OCCC(C)C)=O)CCCCC(C(=O)NCc2ccc(O)nn2)C1 C1(C(N)=O)(CNC(C2CCN2Cc2ccccc2)=O)CN(S(=O)(=O)CC2CCC2)C1 c1(CC)nc(=NC(=O)NC(c2cc(OC)c(OC)cc2O)C)[nH]s1 N1(C(Cc2cn(CC)nc2)=O)CCCC(CC2(C(=O)N(C)C(C)C)CC2)C1 C1(C(N(CCC(=O)N(C)CC2CC2)CCCC)=O)CCC(C)=C(C)C1 CC1CCN(CC2(COCc3ccc(C(=O)N)cn3)CC2)CC1.C(CC1CC1)CC N1(C(c2sc(C)c(O)n2)=O)CCCC2CN(C(=O)CNC(C3CCC3)=O)CCC12 S(=O)(=O)(c1cccs1)NCC(=O)N(C)CC1CN(C(CSCCCC)=O)C1 Cc1ncc(Br)c(C(N2CCC(NC(=O)CC3(C)CCOCC3)C2(C)C)=O)n1 Cc1cccc2c1CN(C(C)C)C2.C12CCC(C1)n1cc(nn1)C(C)C(=O)N2 C1(C(C)NC(=O)Cc2cnsc2)CCN(C(c2nc(Cl)cs2)=O)C1 c1(C(N(CCN(C(C2C(C(=O)OC)C2)=O)C)C)=O)ccnn1C(CC)CC c1(OC)ncccc1C(=O)NCC1CC(CNC(=O)CSc2cc[nH]n2)C1 C=C(C)CC(C(=O)N(CC(C)C#N)C1CC1)NC(C1CC2C=CC1CC2)=O C1(NC(c2cn(C(C)C)nn2)=O)CC2CC(C1)N(C(c1cc[n+]([O-])cc1)=O)C2 c1(NCC2CC(NC(Cn3ccc(C)n3)=O)C2)c([N+](=O)[O-])c(C(F)(F)F)nn1C CCCC(C)(O)C(=O)N1CCN(C(c2cccc(C#N)c2)=O)C(C(F)F)C1 Cc1cc(Br)cc(N)c1C(=O)OC(=O)COC(C)(C)C.C1(=O)CCCN1C N#Cc1ncn(CCCCC(=O)NCC2(NC(C3CCCC3O)=O)CCOC2)n1 N1(C(CCC)=O)CC(C2CN(C(c3cnn(C=O)c3)=O)C2)C1.C(C)(C)(C)O C(C1CCCN1C)=CC(N1CCC(C(C(=O)N(C(CN(C(C)=O)C)C)C)(C)C)C1)=O c1(CNC(N(CCC(F)(F)F)CC)=O)nnc2c(Cl)cccn12 C(=O)(C#CC1CCOC1)NC(c1ccc(F)cc1)CNC(c1c(C)c[nH]n1)=O C=Cn1nccc1C(=O)NCc1cc(C(N2CC(c3nncs3)C2)=O)ccn1 CC(O)(Cc1ccccc1)C(=O)NCCCCNC(=O)COCC1CCCOC1 c1(NC2C(CC)CN(C(C3CCCN(C(N)=O)C3)=O)CC2)nc(C)nc(C)c1F C(=O)(C(F)(F)C(F)(F)C(F)F)NC1(CCNC(C2N(N=O)CCCC2)=O)CCC1 C(=O)(CC1=Cc2ccccc2C1)NCC1(CCNC(CC2CCC(C)(C)O2)=O)CC1 c1(C(=O)NCC2(NC(C(CCCC)F)=O)CCOC2)cc(C#N)ccc1C C1(C(=O)NC(C)C(c2ccccc2)O)CC(=O)N(c2ccccc2)C1 C12(C(=O)NC3C(CC(=O)N(CCN=[N+]=[N-])C)CCC3)CCC(CC1)CC2 c1(C(N2CC(C(=O)NCCCCC)C2)=O)c(-c2cc(F)nc(F)c2)cncc1F c1(-c2ccc(OC(C)C(=O)O)cc2)ccc(F)c(C=O)c1 C(c1ccc2occc2c1)=CC(=O)NC(c1onc(-c2c(C)ccs2)n1)C C12(C(=O)NCc3cc(C)on3)CCN(C(C3(CN(C)C)CCC3)=O)CC1C2 C1(NC(CCn2c(C(C)C)ncc2)=O)CC(F)CN(C(=O)CCC2CCCO2)C1 c1(C(N(CC(C)(C)NC(c2cc(C)nnc2)=O)C)=O)cc(F)ccc1F N1(C(CCc2n[nH]c(=N)s2)=O)CCN(C(=O)CNC=O)CC1C(F)F C(=O)(C1=NOC2(CCOC2)C1)NC1C=CCN(C(C(CC)SC)=O)C1 C(CS(=O)(=O)CC(=O)NC(C1CN(C(C2CCCC(=O)C2)=O)CCO1)C)OC c1(CCC(N2CCC(NC(c3cncnc3)=O)C2)=O)ccc(O)nc1 C1(C(C)NC(c2csc(CO)n2)=O)CN(C(C23CC(C#N)(C2)C3)=O)CCO1 C1(C)(CC)CC(NC(C2CCN2C(C2CCC(C)O2)=O)=O)CCO1 c1(C(C)=O)cccc(NS(=O)(=O)CCOCC(F)(F)Cl)c1F N1(C(c2cc(C)cc(C)n2)=O)Cc2ccccc2CC1CNC(C1CC1(Cl)Cl)=O C1(C(N(CCCO)C(=O)CC2C=NN(C)C2=O)=O)COCCC1NC(CCSC)=O c1(COC)cc(C(=O)NCCCCNC(=O)CC2C(C)C2(F)F)n[nH]1 C#CCC(C)(CC)C(=O)NCCC1CC(NC(C2CC3(C2)CC(C)C3)=O)C1 CC(C)P(=O)(CC(=O)N1CCC1CNC(=O)C(C)(C)CC(F)(F)F)C(C)C C1(C(=O)NC2(CO)CN(C(C3N(C=O)CCC3)=O)C2)CC12CCOCC2 c1(NC(C2C(NC(=O)C3=CCSC3)CCOC2)=O)cccc(Cl)c1O N1(C(c2cn(CC)nn2)C(=O)NCc2cccs2)CCCC(CC(N)=O)C1 c1(C(N2C3CN(C(C4C5COCC45)=O)CC2C3)=O)ccnc2c1OCO2 c1(C(=O)NC(C2CCCN(C(=O)COCC(F)F)C2)C)cc2c(ncn2C)s1 c1(C2C(C(=O)NC3CC(N(C(CC(=O)NCC#C)=O)C)C3)C2)ccccc1Cl N1(C(C2C(CC)C2)=O)CCC(C)(C)C(CNC(C2(C3CCC3)CC2)=O)C1 C1(CNC(C2CCCN(C(CC)=O)C2)=O)CN(C(c2cnsc2)=O)CC12CCC2 N1(C(COc2c(OCC)cccc2)=O)CCCC(C)(NC(=O)C(C)CC(N)=O)C1 N1(C(c2nnn(C)c2N)=O)CC(NC(C23COCC(C2)C3)=O)CC2(CCC2)C1 CC1C(NC(=O)Cc2ccc(Cl)cc2)CCN1C(C1(C#N)CC1)=O C1(C2CCCN(C(=O)C3=CCCC3C)C2)(NC(CC=C)=O)CC1 C1(C(=O)NC2CCC(NC(C3CC(CC)C3)=O)C2)COCCN1C c1(CC)c(OC)cccc1C(=O)NCC1CCCCN(C(=O)COC(C)(C)C)C1 C(C(C(C)(C)C)NC(=O)CCn1ncn(C)c1=O)NC(CC(=O)OC)=O CCCS(=O)(=O)C1CCCC1NC(=O)COc1ccc(CC(=O)OC)cc1 n1(CCN=C(NC(C=C)C)NCC2(O)CCC(F)(F)CC2)ccc2ccccc12 C1(C(N2CCC(CCC)C2)C(=O)NCc2cccs2)CCSC1(C)C c1(C(N2CC(O)(C(C)NC(=O)CCNC(N)=O)C2)=O)coc2c1C(=O)NCC2 N1(C(CN(CC)CC)=O)CCC(C(=O)CCSCN)CCC(F)C1.c1(O)cccc(Cl)c1 C(CC(C)C)(C(=O)NC1(c2nc[nH]n2)CC1)ONC(c1c(CC)ccs1)=O c1(C(N2CCC(CC=C)(NC(=O)Cc3nc(C4CC4)n[nH]3)C2)=O)c[nH]cc(C)c1=O Cc1cc(=O)n(C)nc1C(=O)NCCN(C(c1ccc(C2CC2C)o1)=O)C(C)C N1(C(Cc2onc(C)n2)=O)CC(NC(=O)Nc2ccc(F)c(F)c2)CC(F)C1 C1(C(N2C(CNC(c3c(C)coc3)=O)CCC2)=O)CCN(CC(C)C)CC1 C1(=O)CCC(F)(F)CN1.C(CC(C)(C)C(N)=O)n1cc(CN(CC(=O)O)C)nn1 c1(NC(CC)CNC(=O)C(CC)N(CCN(C)C)C(C)C)ccc2c(c1)CCC2 C1(C(=O)NCC2(F)CCN(C(C(C3CC3)SC)=O)CC2)Cc2cc(F)ccc2O1 S(=O)(=O)(c1cccnc1N1CCSCC1)NC(C)C1CC1 CCN=C(NCCCSCC)N1CCC(O)C1.Cc1nccn1CCCN1CCOCC1 CC(C)C(F)C(=O)N(CCNC(c1coc(C(N)=O)c1)=O)CCOCCO c1(CN=C(NCC2N(C)CC2)NCC2CCC2)csc(S(N)(=O)=O)c1 C1(O)(C(N(CC(C)NC(C(CC=C)C)=O)C)=O)CCCC(C)CC1 N1(C(CCC(C)OCC)=O)CCN(C(=O)CCSc2ccccc2F)CC1C Cc1ccc(Cl)c(F)c1C(=O)NCC12CC(C1)C(NC(=O)C=CCO)CO2 CC(CC(=O)NC(CC(=O)NC(CCO)C1CCC1)C1CC1)c1ccco1 CC1CCN(C(=O)C=CC2CCCN2C)C1C(=O)N(CCCO)CCO N1(CC)CC(C(=O)NC2(CO)CN(c3ccc(C#N)nc3)C2)CCC1=O C1(NC(CSCCCC)=O)CN(C(=O)COCc2ncnn2C)C(C)(CSC)C1 N1(C(C=CC=CC)=O)CCC(O)(C(C)NC(=O)C=CC2CCCCC2)C1 C(=O)(C(S(C)(=O)=O)C1CC1)NCCCC1N(C(C=C(CCC)C)=O)CCC1 C1(NC(C2C(C)CC2)=O)C(C(=O)NCCc2cnn(C)c2)C1(C)C c1(CC(=O)NC2(CCCNC(CNC(CCOC)=O)=O)CC2)c(C)ncnc1C C(N=c1ccn(CC)[nH]1)(c1nn(C)c(C)c1Cl)C1CCC1.N12CCN=NN=C1CC2.CC C1(CC(=O)NC(C2(CNC(c3cnc[nH]3)=O)CC2)C)C=CCCC1 C12(C(N3C(C(=O)Nc4ccc(Cl)cn4)CC3)=O)CCN(CC1)CC2 C(CN=c1cc(NCC2CC2)nc[nH]1)(C1CCCO1)NC(C)=O c1(C(=O)NC(C2CCCN(C(=O)C(F)(F)CC3CC3)C2)C)cccc2c1CCO2 C1(C(N2CCN(C(CC(CCC)O)=O)C(CO)C2)=O)CC2(CCCCC2)C1 N1(C(=O)NCCF)CCCC(C2CN(Cc3ccc([N+](=O)[O-])o3)C2)C1 C(=O)(C1=C(Cl)CCCC1)NC1CC(CNC(c2csc(C(F)(F)F)c2)=O)C1 C1(C(=O)NCC2N(C(c3n[nH]c(C)c3C)=O)CCOC2)C2CCC3C(C2)CC13 c1(C(=O)NC(C)CN(C(=O)CC2CCCN2C)C)ccc2c(O)nnc(O)c2c1 c1(NC(CCC2N(C(COc3cc(C)nn3C)=O)CCC2)=O)cc(F)c(Cl)cn1 C1(CC)CN(C(=O)C(C)(C)C(F)F)CCN1C(c1cc(CC)n(C(C)C)n1)=O C1(CNC(C(=O)C=O)=O)CNC(=O)CC12CCC2.n1(CCN)ccc(=O)c(Br)c1 N1(CC(=O)NCC(CC)NC(C2CC(O)CN2C(=O)NC)=O)C(=O)CCC1=O N1(C(CNC(=O)OCC=C)=O)CC(NC(c2ccc(=O)n(CC)c2)=O)C12CCC2 C(CC(=O)OCC)(C(F)F)N(c1ccccc1C)CCC C1(NC(c2[nH]nnc2-c2ccccc2)=O)CCCN(C(=O)CC2CC3CC3C2)C1 N1(C(=O)C(F)F)CCC(N=C2N=C(c3cccnc3)NNC(c3ccccc3)=N2)C1 C1(CNC(C2(NC(C)=O)CCC2)=O)CCN(C(C2CCCC2C(F)F)=O)C1 CCC(C)(C)C(O)C(=O)NC1CC(NC(c2coc(C3CCOCC3)n2)=O)C1 n1(CCC)nc2c(cc1=O)CN(C(c1cnn3c1CCC3)C(=O)NCC)CC2 c1(NC(CC2CCN(c3cc(OC)nc(OC)n3)C2)=O)cc(F)c(Br)cc1OC CC(C(CO)NC(=O)CCCS(N)(=O)=O)NC(=O)COC1CC(F)(F)C1 C1(C(=O)NC2(C3CN(C(=O)C4=CCSC4)C3)CC2)CCCC2(CCCCC2)C1 Cc1cncc(C(=O)NC2CC3CC(NC(c4cc[nH]n4)=O)C2C3)c1C CN1CCCC(Cn2cc(CC(=O)NC3CSC3(C)C)nn2)C1 c1(C(=O)N(C2COC3(CCNCC3)C2)Cc2ccco2)cccc2c1OCCC2 C(C(N=[N+]=[N-])C(=O)NCC12CC(CN1C(=O)CC1OCCC1C)C2)OCC CC1Cn2nccc2CN1C(c1ccc(CNC(C2CC2(F)Cl)=O)cc1)=O CCC(O)C(C)C(=O)NCC1(C)CCCN(C(=O)CC2CC2)C1 c1(C2C(NC(=O)C(C)CCSC)C2)ccccc1OCC1N(C(COC)=O)CC1 N1(C(c2ccc(C(C)C)nc2)=O)CCCC2CN(C(=O)CSC(C)C)CC12 n1(CC(=O)NC(C2(CNC(=O)CN3CCOCC3)CC2)C)nc(Cl)ccc1=O c1(C(C)NC(=O)C(=O)N(C)Cc2ccc(C#N)cc2)nc2ccccc2o1 c1(OC)c(C(=O)NCC2(CNC(C3COC(C)C3)=O)CC2)cc(Cl)cc1C N1(C(C2CCC3(CC2)CC3)=O)CCN(C(C2CC(O)C2)=O)CC1C1CCCC1 Cc1ccc(O)c(C(=O)NCCCC(O)C(=O)N2C(CO)CC2C)c1 C1(NC(CSCC=C)=O)COCCN(C(c2cc(C#N)on2)=O)C1 C1(C(=O)NC2C(NC(C3CCCS3)=O)CCCC2)Cc2ccncc2C1 CSC1=C(C(=O)N2CCCC(CCNC(C3(C#N)CCOC3)=O)C2)CCCC1 C1(C(=O)NCC2CN(C(c3cc(CCC)c(C)s3)=O)C2)CCC2C(CC1)C2(F)F c1(NC(=O)N(CCC(CCC)CCC)CCOC)c(Cl)oc2ccccc12 c1(-c2cccc(CC(c3ccccc3)(C)O)c2)ccc2ccn(CC=O)c2c1.NN=[N+]=[N-] C(=O)(CCCCC1CC1)NCC(c1ccccc1)N(C(c1nc(CC)sc1)=O)C CN1CCN(C(=O)C=C2CCN(C)C2)C(CNC(=O)CCN2CCC(F)C2)C1 c1(C(=O)NCC2CN(C(C(C(C)C)c3ccncc3)=O)C2)cc2c(s1)CCCC2 CC(C)CC(C(=O)NCCC1CC(=O)N(C)C1)ONC(C1CCCN1C1CC1)=O Cc1cccc2cc(C(=O)NC3CN(c4ncc(Br)c(O)n4)CC3(C)C)oc12 N1(C(c2ccc(Cl)cn2)C(=O)NC(C)(C)C)CCCc2oc(Br)cc2C1 N1(C(c2n(C)c(S)nc2)=O)CCN(C(=O)CN2CCOC2=O)CC1C1CC1 n1(CC2CN(C(c3cnccn3)=O)C2)ccc(Br)n1 c1(C(C)NC(C2CN(C(=O)C(C)Cc3cccnc3)C2)=O)cc(F)c(F)cc1F c1(C(=O)NC(C(C)(C)NC(c2cc(C(=O)OCC)no2)=O)C)ccc(Cl)c(Cl)c1 c1(C(=O)NCC2C(C(N(C3(C)CC3)CC)=O)CCO2)cc(=O)cc[nH]1 c1cn2c(n1)CCN(C(=O)C(C)(C)CN(C)C)CC2.C1(OCCC)CNC1 c1(C(=O)NC(CNC(=O)OC(C)(C)C)CO)noc(-c2ccccc2)c1Br CC1CCC(NC(=O)CN2CSCCSC2)CN1C(C1(C2CCC2)CC1)=O C1(CNC(CCOC(C)=O)=O)(NC(=O)CN2CCSCC2)Cc2ccccc2C1 N1(C(C2C(C#N)C2)=O)CC2CC(C1)C2NC(c1cc(Cl)ns1)=O CC(C)C(C(=O)N=c1cc(C(C)(C)C)o[nH]1)OC1CC1 N1(C(C2C(C)=CCS2)=O)CCC2(CC2C(=O)NCC(C)CC(C)O)C1 CCC(F)(F)CC(=O)N1CC(O)CC1CNC(c1ccc(C(C)C)s1)=O C1(NC(c2ccc(COC)o2)=O)CCC(C)N(C(c2cc3c(s2)CCC3)=O)C1 N1(C(c2cncc(OC)n2)=O)CCC(NC(c2ccc(C(C)(C)C)[nH]2)=O)C(C)C1 c1(CNC(=O)NC23COC(N2)C3)ccc(OC(F)F)c(O)c1 CCCCCCC(C)CC(=O)N1CCC(C(C)NC(c2ccc(F)cc2N)=O)C1 c1(C(=O)NC(C(C)NC(=O)CCC2CCC2)CO)ccc(C#N)cn1 C1(C(=O)OCC(c2ccccc2)OC)CCCN(c2nc(-c3cccs3)cs2)C1 C1(C(=O)NCc2c(CC)ocn2)C2CC2CN1C(c1cncc(OC)c1)=O C1(CC(=O)N(CCNC(=O)CC2CC3CC3C2)CC2CC2)(OC)CCCC1 c1(OC)ccccc1C(N1CCC2C(NC(c3cnc(C4CC4)s3)=O)C12)=O N1(C(C2CC(=C)C2)=O)CCC(CNC(C2CCCN2CC)=O)C1(C)C N1(C(CC2(C)CC2)=O)CCCC(C(=O)NCC2CC3(C2)CC3F)C1 c1(C(C(=O)NCC2(NC(=O)C(F)Cc3ccccc3)CCC2)O)ccc(Cl)cc1 N1(C(C(C)CC2CC2)=O)CC2(COC(CNC(=O)CCn3cncn3)C2)C1 c1(NC(C2N(c3nc(OC)c(C)cn3)CCNC2)=O)c([N+](=O)[O-])ccc(F)c1C N1(C(c2nc(CCC)sc2)=O)CCC2(NC(=O)CCc3nnc(S)n3C)CC2C1 N1(C(c2ccc(CNC(c3cnc(S)[nH]3)=O)o2)=O)CCN(c2cccc(Cl)n2)CC1 C(C)(CC(=O)NCCC(C1CC1)C1CC1)NC(C1C(C)CC1)=O C(C1CCC(C)CC1)=C(C)C(=O)NC1CCC1NC(=O)Cc1coc(C(F)F)n1 C1(C)(C(N2CC(CC=C)(NC(C(CC=C)OC)=O)C2)=O)CCC(=O)NC1 C1(CC(=O)NCCCCCN(C(=O)C(C)(C)CF)C)COCCN1C N1(CC(=O)NC(C(C)NC(CCCCC)=O)CO)CCc2sccc2C1 Cc1nc2cc(Cl)cc(C(=O)NC3CC3C(=O)NCC3CC34CC4)c2[nH]1 CC(N=c1nc(N2CC3C(C2)C3(C)C)c2c([nH]1)CCC2)c1ccncc1 N1(C(=O)CC2(Cl)CC2(F)F)CCC2C(C1)N(c1cccnc1)C2=O.C1(C)CC1.CO C#Cc1ccc(N(C(=O)COC(=O)CNc2cccc(F)c2F)C)cc1 c1(-c2ccc(C)cc2N(C)C)ccc2nnc(C(N3CCCC(C)(O)CC3)=O)n2c1 C1(O)(C(N(C2CN(C(=O)COCCCF)C3(CCC3)C2)C)=O)CCC(C)(C)CC1 Cc1cnn(C)c1CNC(=O)C(CCOC(=O)C(C1CCCCC1)=O)NCCO CC1(C)CC(CNC(C2CCOC2)=O)N(C(=O)COc2cncc(Cl)n2)C1 C(=O)(NNC(=O)NC1CC1)NC(c1nnnn1C)C CC(C)CCCC(=O)NCC1OCCC1C(=O)N(C(C)C)C(C)C c1(C(CN2CC(c3c(C)ncs3)(O)C2)=O)ccc2occc2c1 C(=O)(C(O)CC(C)C)NC1(CCC(=O)NCCCCCN(C)CC)CCCC1 C12(CNC(NCc3ncccn3)=NCC3CC3)CCCN(CC1)C2 c1(C(=O)NCC2(CNC(C3(CC)CC3)=O)CC2)cc(N)c(C)cc1C c1(OCC)ncc(C(N2CC(CCNC(c3c[nH]c(=N)c(C)c3)=O)C2)=O)cc1Cl C1(C(=O)NC2CCC(CCC(=O)N(CC(C(=O)OC)C)C)C2)NC(=O)CC1C C(=O)(C(=O)N=S(C)(C)=O)NCC1CC(Cc2cn(CC3(C)CCCC3)nn2)C1 Cc1cc(C(=O)NC2CC(NC(C3CS(=O)(=O)C3)=O)CC2O)cnc1O C1(CNC(C2(OC)CCC2)=O)CN(C(=O)COc2ccsc2)CCC1(F)F CCCC(CC)CCC(=O)NC(Cc1ccoc1)C(N1CCS(=O)C(C)C1)=O N1(C(C(CC#C)C)=O)CC2CCCC2(NC(c2cnn(CCO)c2CCC)=O)C1 O=C1CCC(CCNC(c2cccc(-c3ccc(O)nc3)c2)=O)C(=O)N1 c1(C(=O)NCC(C(=O)NCC(C(=O)NC)O)(C)C)c(C)cccc1O C(c1cccs1)=C(C)C(=O)NC1CCC1NC(=O)CC(C)F CC1(C)OC(C)(C)c2ccc(NC(=O)NCC3(CO)CC3(C)C)cc21 c1(C(=O)NCCC2(C(N(CCOC)C)=O)CC2)c(F)cncc1F c12cc(cc(F)c1)NC(=O)N2.N1(CC(=O)NC(C)(C)C)CCC(F)(F)CC1 CC1(C)CCC(CNC(c2cc3c([nH]2)CCOC3)=O)N(C(C2CNC(=O)N2)=O)C1 CS(=O)(=O)CCCC(=O)NCC1(CO)CCN(C(=O)CC2CC3CCC2C3)CC1 N1(C(c2cnc(CC)[nH]2)=O)C2CCC1C(CNC(C1(C(F)F)CCCCC1)=O)C2 C1(CC#C)(C(N2CCC(C)(CNC(C34CSC(C3)C4)=O)C2)=O)CC=CCC1 C1(c2n(CCC)nnn2)(NC2(c3cnn(C)c3C)CCC2)CCOCC1OC C(=O)(CC(O)CCC(C)CC)NC1COCCN(C(CSCCC)=O)C1 C1(C(=O)NC(CN(C)C)C(=O)NC2C(C)(C)C2(C)C)CCCC2(CC2)C1 N1(C(C2C(C)C2c2ccccc2)=O)CCCC(N(C)Cc2cnon2)C1 c1(O)cc(C#N)ccc1C(=O)NC(CCn1c(C)cc(C)n1)C.C(CO)S c1(OC2C(OC(=O)CCC3CCC(=O)N3)CC2)nc2ccccc2s1 N(C(=NCCC(C)(C)O)NC1CCN(C(=O)Nc2cccs2)CC1)C(CC)C N1(C(C2(C(CC)=O)CC2)=O)CCCC(CNC(C2(C(N)=O)CC2)=O)CC1 c1(CN(C(C2C(=C)C2)=O)CCNC(=O)C(O)Cc2cnc[nH]2)cccc(Cl)c1 CC(F)(CC1CCCC1)C(=O)N1CCC(C)(CNC(c2ccc(F)s2)=O)C1 CC(C)(COCCCCCCCC(=O)NC1CCCCC1O)C(=O)NC1CC1 CC1CC(C#N)(C(=O)NCC2CCOC2C(=O)NCCc2ccon2)C1 C(=O)(N1CCC(C(=O)N(C2CCSCC2)C)O1)C1(C)C(C)C1 C1(NC(CC)=O)C2CC3CN(C(=O)C(N4CC(=O)NC5CCCC45)=O)C1C3C2 C(=O)(C1=Cc2ccc(Cl)cc2OC1)N1CCC(N(C(=O)CCC(=O)NC)CC)C1 c1(N2CC(CC)NC(=O)C2)nc(CN2CCCC(N(C)C)C2)nc2c1COCC2 c1(C(=O)NCC2(CNC(C(CC)C(F)(F)F)=O)CCC2)cncc2ncn(C)c12 C1(NC(c2ccsc2Cl)=O)CCCC12CCN(C(=O)CSCc1ncc[nH]1)C2 N1(C(CC2CC(SC)C2)=O)CCCN(C(c2ncc(N)nc2C)=O)C(CO)C1 c1(C(C)=O)cccc(OCC(=O)NC2CCC2CC(=O)O)c1 C=CC(CCC)CC(=O)N1CCCN(C(=O)C=C(CCC)CCC)CC1 C(CN=c1nc2sccc2c(NCc2cnn3cccnc23)[nH]1)N(CCOC)C c1(C(N2CC(CNC(C(C)SCCCC)=O)N(C)CC2)=O)ccn2ncccc12 C12(NC(c3cccc(F)c3Cl)=O)CCCC1N(C(=O)C=CC1CC1)CCC2 c1(C(=O)NCC2C(CNC(CS(C)(=O)=O)=O)C2)n[nH]c2nccc(Cl)c12 C=CCC(CC(C)C)C(=O)NCC1CCN1C(c1cc([N+](=O)[O-])cnc1O)=O C1(C(=O)NC2CC(NC(c3cccc(CF)c3)=O)C2)CCn2nncc2C1 C(=O)(C(C)CC(C)C)N1CC2C(CNC(CC(OCC)OCC)=O)(C2)C1 n1(CCOC)cc(C(=O)N(C)CCNC(c2cn(C)cn2)=O)c(C2CC2)c1 N1(C(CN(C(=O)OC)C)=O)CCCC1COCC(=O)N(C1CC1)CC1CCCO1 N1(C(COC(C)=O)=O)CCCC(NC(c2cncc([N+](=O)[O-])c2)=O)C(F)C1 C1(C)(CC)CCC(C(N2CC(C)(NC(=O)CCN3C(=O)CCC3=O)C2)=O)O1 N1(C(C)NC2(C)CC2)CCC2CN(C(=O)OC(C)(C)C)CCC2C1 c1(CC)ccc(F)c(C(=O)NCC2CCCCCN2C(c2n[nH]cc2OC)=O)c1 N1(C(CN(C)C)=O)CCCC(C(C)(O)CNC(=O)CCNc2ccon2)C1 C#CC1CN(C(=O)C(CCOC)NC(=O)Cc2cccc(C)c2)CCO1 c1(C(N2CC3N(C(C(C)SC)=O)C(CC3)C2)=O)cnc2c(F)c(F)ccc2c1 Cc1cnc(NCC(C)N(C)C)c(S(=O)(=O)NC2CCCCC2(C)C)c1 c1(NC)ccc(C(=O)NCC(CC2CN(C(=O)C(C)SC(C)C)C2)(C)C)cc1F c1(C(=O)NC(C(C)(C)C)C(=O)NCCc2ccncc2)cccc2[nH]ncc12 N1(C(Cc2c(C)noc2C)=O)CCCC(O)(CNC(c2csc(C#N)c2)=O)C1 c1(CC)n[nH]cc1C(=O)N(CCC(=O)NCC(=O)NCCO)CC(C)C C1(NC(CC2ON=C(CC)C2)=O)CC2CC1CN2C(C1CCCC(=O)O1)=O N1(C(CC(C)(F)F)=O)CC2(CCC2)CCC1CNC(=O)CNC(C1CCC1)=O C1(F)(CNC(=O)CSc2ccc(Cl)cc2)CCCN(C(=O)CSC(F)(F)F)C1 c12n[nH]c3c1CN(CC3)C2.c1(-c2ccc(C(=O)OC(C)(C)C)s2)ncc(F)cn1 C1(CNC(C(C)(C)SC)=O)CC(NC(C2CCCC2O)=O)CCO1 N1(C(CCCCC)=O)CCN(C(=O)Cc2cncs2)C(c2ccccc2OC)C1 C12(CC=C)COC(C(F)(F)F)(C1)C2.C12CCCC(C1)N(C)C2 CC(C)CCC(C(=O)NCC(c1cnn(C)c1)O)NC(c1ccccn1)=O c1(OC)ccncc1CCNC(=O)NC1CCOC(C(C)C)C1 N1(C(CC)=O)CCC(C)(NC(=O)C(=CC2CCC(C)CC2)C)CC1 C1(NC(C(CN(C)C(c2cn(C)c(=O)n2C)=O)(C)C)=O)CC12CCOCC2 Cc1onc(Cl)c1C(N1CCN(C2CN(C(=O)CCCCCl)C2)CC1)=O c1(NC(C)=O)ccc(Cl)c(C(N2CCN(C(c3cc(Cl)ncn3)=O)C3CC23)=O)c1 N1(C(c2cnc(OC)nc2)=O)CC(C)C(NC(=O)CCN2CCOCC2)C(C)C1 Cc1cc(C(C(=O)NCc2ccc(C#N)s2)NC(c2ccnn2C)=O)ccc1Cl CC1C(NC(=O)CC2CCN(C)C2=O)CCN1C(=O)CCc1csnn1 Cc1nc(O)[nH]c1C(N1CCCC1(C)CNC(=O)C(O)Cc1ccccc1Cl)=O c1(CC(=O)NC(C(C)NC(C2CC2C(N)=O)=O)(C)C)cnc2c(=O)[nH]ccn12 C12C(C)CCCN1C(=O)C(OCC)OC(=O)C2.CCCC(C)(CC)NC(C)=O c1(C(=O)N(C(C)(C)C=CC(=O)NCCC2CCCCC2O)C(C)C)ncncc1Cl c1(C(=O)NC2C(NC(=O)C=Cc3cnccn3)CCCC2)nc2cnccc2s1 N1(CC)CC(CNC(=O)CCC2CC(NC(c3cc(C)no3)=O)C2)CC1=O N1(C(Cc2c(C)cco2)=O)CCC(C2CCN(C(c3cccc(C)c3F)=O)C2)C1 N1(C(C2CN(C(c3nc(=N)[nH]cc3)=O)CC2(F)F)=O)CC2CC3CC2C1C3 c1(OC)ccc(C(N2CCC(C)(CNC(C3(C)CCCC3C)=O)CC2)=O)c(Cl)c1 N1(C(CC2CN(C(CC3C(CC)CCC3)=O)C2)=O)CCOCC1CC(=O)NC c1(OC)ccc2c(c1)C(CCNC1CC1)=CC2.N(C)(CP(C)(C)=O)Cc1nnnn1C O=S(=O)(c1ccc2[nH]c(=NCCc3ccsc3)sc2c1)NCc1ncccn1 Cc1cc(C(N2CCCC(O)(CNC(=O)C=CS(C)=O)C2)=O)cnc1O c1(C(=O)NC2(CCCNC(C3C(C)(CC)C3)=O)CC2)nc(Cl)cs1 Cc1cccn2nc(C(N3CCC4(CCN(C(=O)CCCCCF)C4)C3)=O)cc12 C=CCC(C(=O)N(CCC)CC=C)C(C)C.C1(C2C(=O)N2)CCC(C(C)(C)C)CC1 c1(N2Cc3c(nc(C)s3)CC2)[nH]c(=NCC2CCSC2(C)C)nc2c1ncn2C C1(CNC(C=CC)=O)CCN(C(c2ccn(C3CCC3)n2)=O)C12CCC2 CC(C)CCC(O)C(=O)NC1CCCCC1NC(=O)Cn1cnc([N+](=O)[O-])n1 C1(C)(N(C)C)CCC(N=c2cc(NCC3CC=CCC3)nc(C(F)(F)F)[nH]2)CC1 c1(C(=O)NC(C(C2CCCCC2)NC(CCOC)=O)C)cnn(C)c1C(C)(F)F N1(CCN(C(CCCC(=O)NCCCCC)=O)C)CC(C2CN(CC)C2)C1.C(C)(C)(C)N C1(Cn2c(=O)ncn(CCC)c2=O)(OC)CCN(Cc2ccc(Cl)cc2)C1 N1(C(CC2C=NN(C)C2=O)=O)CC2(NC(c3n[nH]cc3Cl)=O)CCC1CC2 N1(C(C(C)Cn2cccn2)=O)CC2C(N(C)C(c3cn(C)nn3)=O)C2C1 C1(C(N2C(C(C)(C)NC(COCCOCC)=O)CCC2)=O)CC12CCOCC2 c1(C(N2CC3C(NC(CN(C4CCC4)C)=O)(C3)C2)=O)cncc2c1CCCC2 C(C(C)(C(C)C)NC(C1CCCOC1COC)=O)NC(COCCC=C)=O c1(CC(=O)NC(CNC(C2(C(=O)OC)C(=C)CC2)=O)C)c(C)noc1C c1(C2C(C(N(C(CCNC(CCC#C)=O)C)C)=O)C2)cc(Cl)ccc1Cl C1(c2nc(-c3ccccn3)no2)(NC(Cc2cc(C)ns2)=O)CCC(=O)NC1 C1(C(N2CC(NC(Cc3c(C)cc(O)cc3)=O)C2)=O)CCOC2(CCOCC2)C1 n1(CCC(N2CC(CNC(C(c3cccs3)N(C)C)=O)C2)=O)ncn(C)c1=O Cc1ccc(CC(=O)NC2(C)CC(NC(c3ccn(CC(F)F)n3)=O)C2)c(C)c1 C(CN(C(=O)Cc1cccn1C)C)(CO)(CO)NC(CC(C)n1cccn1)=O N1(C(C(C)OCCCC)=O)CCCC(N(C(=O)Cc2scnc2C)CC)C1 N1(C(c2cc(C)c(N)cn2)=O)CC(C2CN(C(=O)CC3CCCCC3(F)F)C2)C1 C1(CN(C(=O)NCc2n[nH]c(C)c2Br)C)CCCCC12OCCO2 N1(C(C=C(C)C2CCCCC2)=O)CC(NC(=O)Cc2ccoc2)CC12CCOC2 C(CC(C)C(=O)NCc1nocc1COC)=CCC.N12CCC=CC1C2=O Cn1nc(CNC(c2cnc[nH]2)=O)cc1C(=O)NCC1CCOC1=O c1(CN(C(C(C)OC(C)(C)C)=O)CCCNC(c2cncs2)=O)ccccc1 C12(C(=O)NCc3ccc(-c4cnc(C)nc4)cc3)CCC(N(C)C)(CC1)CC2 C(=O)(C1=C(c2ccccc2)SCCO1)N1CCC(NC(C=C(C)C)=O)C1C c1(C(C(=O)NCC(=C)C)N(C)CCN(CCC)CC)cnn(CC)c1C CC1(C(=O)NCc2nc(C(=O)NCC(O)C3CCC3)co2)CNC(=O)C1 C12(C(=O)NCCN(C(=O)C(C)C)CC)CCC(C)(C1)OC2.C1(=O)C(C(C)C)N1 N1(C(C(C)NC(c2cc(C#N)cn2C)=O)=O)CCn2c(C(F)(F)F)cnc2C1C C1(F)(CNC(c2nccc(N)c2)=O)CCN(C(c2cscc2F)=O)CC1 C1(NC(C2C(C)(C)CC2)=O)CCN(C(c2cc(O)nc(Br)c2)=O)C12CC2 CCCCC(F)C(=O)NC12CCC1CN(C(=O)C=CC(=O)NC1CC1)C2 c1(C(=O)NC(CNC(CC(CC)(C)C)=O)C)sc2ccncc2c1OCC C12(NC(=O)NCCN3CCC(NC(C(CC)F)=O)CC3)CCCC(C)(C1)OC2 c1(CN(C(=O)CCc2ccn(C)n2)C)cccc(CNC(C2CCC2CF)=O)c1 N1(C(c2ccc(OCCOC)nc2)C(=O)NC(C)(C)C)CC(=O)N(C)C(C)C1 c1(SCC(=O)NC(CCCNC(CCC(C)OCC)=O)C)ccc2c(c1)CCC2 c1(C(=O)NC(c2ccccc2)CNC(CC(CCC)O)=O)ccc2cnoc2c1 C(C(C(=O)NC(c1ncccn1)C)N(C)C)OC(CC(=O)NC(C)C)=O C1(CNC(CC2ON=C(C)C2)=O)(CO)CCN(C(=O)Cc2nccn2C)C1 c1(C(N2CCN(Cc3ccc(OC)c(Br)c3)C3C2C3)=O)ccn2cncc2c1 C1(C)(CC(=O)NCC(Cn2cc(C3(F)CCOCC3)nn2)OC)CCSCC1 CC(CC(C)(C)C)C(=O)N1CCCC(C)(NC(c2ccncc2)=O)C1 C12(C(N3CCC(CC#C)CC3)=O)CCCC1CCN2C(=O)CC(C)(O)C=C C1(NC(C(N2CCC(OCCCN)CC2)=O)=O)CCS(=O)(=O)CC1 c1(SC)cccc(C(=O)NC2(C)CCN(C(C3CC3C)=O)C2)c1Cl c1(C(=O)NCC(CNC(C(CC)n2cncn2)=O)(C)C)cc(Cl)ccc1OCC c1(OC)ccc(-c2cc(C(=O)NC(c3cc(Br)no3)C)n[nH]2)cc1F c1(NC(c2c(C)nccc2)C)nc2ccc(Cl)cc2c(=NC2CCCCC2F)[nH]1 c1(C(=O)NC(C2CCCCC2)CC)cc(Cl)cc(Cl)n1 CCCCC(CN=c1sc2cccnc2[nH]1)OC(C)=O c1(CN(C(=O)CN2CCCCCC2)CCNC(c2cn(C)nc2)=O)ccc(O)cn1 CC1CN(C(=O)CSc2nnnn2C)CC1CNC(=O)CN1CCCC1 C1(C(=O)NCCCN(C(C2N(C(C(C)C)=O)CCC2)=O)C)CCc2cnnn2C1 C1(C#C)(NC(CC2CN(C(COCCCC#C)=O)C(C)C2)=O)CC2CCCC12 c1(CC(N2CC(N(C(c3c(C)c[nH]n3)=O)C)C2)=O)c[nH]c2cccnc12 C1(NC(c2c(CNC(C(n3c(C)ncc3)C)=O)cc[nH]2)=O)CNC(=O)C(C)(C)C1 C1(CNC(c2nc(C)[nH]n2)=O)CCCCN1C(c1coc(Cl)n1)=O C(=O)(C(C)(C)CCCNC(c1cnn(C)n1)=O)N(C(CC#C)C)C C1(C(N2CCC(F)(CNC(COC(C)C)=O)C2)=O)CCc2ccccc2C1 C12=NC(C(F)(F)F)=CC(=NCC3(CCC3)N1)N2.C1(NC)(C)CC1.C(C)(C)O Cc1cccc(C)c1CNC(=O)C(F)(F)n1cc(C2(N(C)C)COC2)nn1 C1(C(=O)NCC(C)CNC(=O)C(c2ccccc2F)(C)C)CCc2cncn2C1 C#CC1(O)CCCN(C(C2(C3CC3)CN(C(C3CC3CCC=C)=O)C2)=O)C1 C1(CC(=O)OC)(CBr)CCN(CNc2cnc(Br)c(N)n2)CC1 C1(C)(NC(C23CN(C(C(CC(=O)OC)(C)C)=O)C(C2)CO3)=O)CC(C)(C)OC1=O N1(C(CN(C)C)=O)CCC2CCCN(C(c3ncc4[nH]cc(I)c4n3)=O)C2C1 C(CNC(=O)C1=CCCS1)(C(C)C(C)C)NC(c1c(CC)con1)=O c1(CN2CCN(C(c3cncc(Cl)c3)=O)CC2)cc(Cl)c(Cl)cc1O C1(CC)CCN(C(=O)CCCNC(c2cnn(CCOC)c2)=O)C1C CNS(=O)(=O)N1CCC(C(N2CCC(C(c3ccccc3)=O)C2)=O)CC1 Cc1cnc2n1C(C(=O)N1C3CCC1(CNC(=O)CCC1(C)CC1)CC3)CCC2 CCC(O)(CC)CCON(CC(O)Cc1ccccc1Br)C C1(C)(OC(C)C)CC(NCC(=O)NC(C)CF)C1(C)C c1(C(N2C(CCNC(CCN(CC)CC)=O)CC(OC)C2)=O)ccc(Cl)c(N)c1 C1(NC(C)=O)CCCN(C(C2CC=CC(CC(=O)N(C)C)C2)=O)C1 C1(N(C)C)(C(=O)NCCNC(=O)C(N2CCC(O)CC2)=O)CCCSC1 N1(C(CCOC)=O)C2CCC1CC(NC(c1nc3c(s1)COCC3)=O)C2 c1(C(=O)NCCN(C(=O)C(C)N(C)C)CCC)c(Br)nc2n1CCCC2 N1(C(C(CCCC)F)=O)CCC2CCN(C(=O)CS(=O)(=O)CCO)C2C1 N1(C(c2cc(N)c(N)nc2)=O)C2CCC1CC(NC(C1CCC=CCCC1)=O)C2 c1(C(=O)NCCC2CCCN(c3ncncc3I)CC2)ccc2[nH]ccc2n1 CC1(C)Cc2ccc(C(N3CCC3CNC(c3cc4cccnc4s3)=O)=O)cc2C1 N1(C(CN(CC(C)(C)C)C)=O)CC(C2CN(C(c3ccnc4cc[nH]c34)=O)C2)C1 c1(C(=O)NCC(CC)NC(C2(F)CCCCC2)=O)ccc2n[nH]cc2c1C Cc1cnc(CC(=O)NCCCN(C(=O)CCC2CCCOC2)C)s1 c1(C(=O)NC(C2CCCN2C(=O)CCc2cnc[nH]2)C)cccnc1-n1ccnn1 n1(CC)nc(C)c(C(=O)NCc2ccc(CNC(C3CN(C)C3)=O)c(F)c2)c1C C1(O)(CN(C(C(C)=C2CCC2)=O)C)CCN(C(=O)C(C)(O)C2CCC2)C1 N1(C(COc2cc(C)on2)=O)CCC2CCC(NC(C3CCC(C)(C)C3)=O)C1C2 c1(SC2CCCN(C(c3c(C)cco3)=O)C2)c(C)nn(C)c1C C(=O)(C1CCc2c[nH]nc21)N1CCCC(CNC(c2n(C)ncc2Cl)=O)C1 C=C(C)C1OCCCC1C(=O)NC(CNC(C1(CC(C)C)CCC1)=O)CCC C1(C(N2CC(COC)(NC(C3CCCOC3C)=O)C2)=O)C(C)CCC1C c1(C(=O)NCC(CC(C)C)(C)NC(=O)C(C)CC(N)=O)nsc2c(Cl)cccc12 C(CC(C)C(=O)NCCCCC(=O)NCc1ccccc1CO)=CC N1(C(C(C)Cc2ccc(F)cc2N)=O)CCC2CN(Cc3cncc(Cl)c3)CC12 C1(NC(Cn2ccc(C)n2)=O)CCN(C(=O)Cc2nnc(C)n2C)C1(C)C C(CCC(C)(C)C(=O)NC(C1CCN(C(c2ccc(C(F)F)s2)=O)C1)C)OC c1(OCC)cc(NC(C2CCC2)=O)cc(CNC(c2cc(=O)cc[nH]2)=O)c1 C(=O)(C(O)Cc1ccccc1)OCC(C)(C)Oc1ccccc1 N#Cc1c[nH]cnc1=NC1CC2CN(C(C34CCC(C3)OC4)=O)CC12 c1(C(N(CC(C)(C)CNC(C2CCC(C(N)=O)N2C)=O)C)=O)cnc2n1CCC2 N1(C(C2C(C)(C)C2)=O)CC2CC(N=C3Nc4ccccc4C=CN3C#N)CC1C2 CCC(CC(=O)NC1(C)CCN(C(=O)C(C(F)(F)F)OC(C)=O)C1)CC(C)C c1(C(N(C2CC3CCC(C2)N3C(C2CC23CC3)=O)C)=O)ccnc2ccccc12 c1(C(=O)NCC(CNC(C(CC=C)(C)C)=O)(C)C)cc(C#N)c(SC)nc1O C(=O)(CCCC(C)C)NCC(C1(O)CCN(C(c2c(C)nn(C)c2)=O)C1)C N1(C(c2cc(C)c(C)[nH]2)=O)CCCCC(C(=O)NC2CCC(N(C)C)C2)C1 C1(C(=O)NCC2(CNC(CC(C)N)=O)CCC2)(OC)CCCCCCC1 n1(CC)nncc1CNC(=O)C=CC(C)(C)NC(c1ccc(C)s1)=O N1(C(c2c(CC)cno2)=O)CC2CC1CN(C(=O)CN(S(C)(=O)=O)C)C2 CCC(C)C(=O)NC(COC(C)C)C(=O)NCC(C)(C)OCC1CC1 CCCCCC(C)CC(=O)N1CC(NC(c2cccc(=S)n2O)=O)C(C)C1 n1(CC(=C)C)nc(C2CCC2)nc1CCc1ncc(F)cn1 C(=O)(C1Cc2ccc(F)cc21)NC1(C)CC(NC(c2c(C)n(CCO)nc2)=O)C1 C1(C(C)NC(c2cnc(C)[nH]2)=O)CCN(C(c2scnc2C(C)(C)C)=O)CC1 c1(NC(C23CC(NC(C4CN(C)C(=O)CC4)=O)(C2)C3)=O)cccc(C#N)c1F C1(NC(c2n(C)nnc2)=O)C=CCC(C(=O)NCCCCCCO)C1 C1(NC(CC2CCCN(C(C3C(CC)N(C)CC3)=O)C2)=O)CCC2CCCC1O2 c1(CCCCCOC(C(C2CC(F)(F)C2)OC)=O)ccc(F)cc1 C1(NC(C=C(C)C(C)(C)C)=O)CC(CNC(=O)C=CI)C(O)C1 C1(CNC(CCCCSC)=O)CN(C(c2ccc(C)o2)=O)CCC12CCC2 C(C)(C)(C(=O)NCC1CCC(C(N)=O)O1)OC(C)=O.C12CCC1C(=O)N2 c1(CN(CC(C(=O)NC)C)C2CC2)ccc(Br)cc1OC C12CCN(CC1)C(=O)COC(C)(C)CN2C.C1(NC)CCCC1 N1(C(CCCCC=C)=O)CCC2(CCOCC2)C(NC(=O)C(CC)(CC)CO)C1 C1(C(C)C)CCCC1NC(C1(C2CCCN2C(=O)COC2CCCCC2)CC1)=O c1(CC(=O)NC(CC(C)NC(c2cn(CC=C)nc2)=O)C)ccc2c(c1)CCO2 c1(C(=O)NCC2(NC(C3CCCN(CC)C3)=O)CCOC2)cnc2n1CCS2 C=CCC(C)(C(F)F)NC(=O)CC(C(F)F)NC(c1cc(C(N)=O)co1)=O c1(C(=O)NC2C3CC(NC(c4c(CC)cno4)=O)CC32)cn2cccc(F)c2n1 C1(C(N2CCC(N(C(C=CC3N(C)CCC3)=O)C)CC2)=O)CCn2cncc2C1 c1(C(N(CCOC)CCNC(=O)CC2CN(C)C2)=O)ccc2oc(C)nc2c1 N1(C(c2cc(CCC)on2)=O)CCN(C(=O)CCc2cncc(OC)c2)C2CC12 N1(CC)CCC=C(c2cncnc2C(=O)NC(C)C(=O)NCC(C)C)C1 c1(CC(=O)N(CCN(C(c2cnc(S)[nH]2)=O)CC)CC)ccc2cccnc2c1 C1(C(=O)NCc2cn(CCNC(C=C(C)Cl)=O)nn2)CNC(=O)CC1C c1(C(=O)OC2CCN(C(=O)NC3OCC3(C)C)C2)ccccc1.CC1C(=O)N1 c1(-n2c(COCCOC)nnc2C(C)OC)nc2ccccc2[nH]1 N1(C(c2c(CC)nn(C)c2)C(=O)NC(C)C)CC2(C)CCC2(C)C1 Cc1nc2c(C(=O)NC3CCN(C(=O)Cn4ncnn4)C34CCC4)ccnc2[nH]1 N1(C(C2CCN(C)CC2)=O)CC2CCC1CN(C(=O)C(C)(C)CC#N)C2 c1(C(=O)NCC(=O)NCC(CC)NC(=O)C(F)(F)CC2CC2)ccc(F)cc1 c1(C(N2CC(F)(C(=O)Nc3cn(C(C)C)nc3)C2)=O)ccc(I)c(Br)c1 C1(NC(c2ncn(CC)c2)=O)C2CC1N(C(=O)CC(C)SC)C2C C1(C(N(CC)CC2CC2)=O)CN(C(c2noc(C)c2C)=O)CCC1(C)C c1(OC)cccc2c1OC(C(=O)NCCCCC1CN(C(C3CCOC3(C)C)=O)C1)C2 c1(C(N2CC(CNC(C(C(=C)C)(C)C)=O)C(C)C2)=O)ncc2ccccc2c1N c1(SC)cc(C(N2CC(C(C)NC(=O)CC3OCCCO3)C2)=O)ccc1F c1(C(N(CCN(C(CC2(C=C)CC2)=O)C)C)=O)cc2c(s1)CC(C)CC2C C12(C(=O)NCCCCCN(C(Cn3ccc(C)n3)=O)C)CC(C1)C(C(F)(F)F)O2 C1(C)(CNC(CC2CN(C(C)=O)C2)=O)CCN(C(=O)CC2CSCCO2)C1 C=CCC(C)(O)C(=O)N(CCCNC(=O)CCC(C)(F)F)CCO c1(OC)cc([N+](=O)[O-])ccc1NNC(=O)c1nn(CC(F)(F)F)c2ccccc12 CC(C)(C(=O)NCC1CCC(C(=O)NC(C2CCCCO2)(C)C)CC1)C(F)(F)F CCCC(C)(C)CC(=O)N1CCOC(C2(NC(=O)CC3COCC3(C)C)CC2)C1 c1(C(=O)NCC=CCNC(c2c(Cl)n[nH]c2C2CC2)=O)cc(F)cc(F)c1 c1(C(=O)NC(c2cn(CC3CCOC3)nn2)CCC)ncccn1 CCC(O)C(C)(C)C(=O)N(C)CC1(CNC(C2CCC(=O)OC2)=O)CC1 CC1(C)CCCC(CNC(=O)C2=NOC(CNC(=O)Cn3cccn3)C2)C1 c1(COC)ccc(C)c(NC(C2(NC(C3CCOC3)=O)CC2)=O)c1 Cc1ccc2nc(CNC(N3CCN(CC(C)P(C)(C)=O)C3CCC)=O)cn2c1 C1(CNC(C2CCC(CC)O2)=O)CC(O)CN1C(=O)COCc1nc[nH]n1 CC(C)C(CCCC(=O)O)NC(c1cc(C(F)F)[nH]n1)=O c1(C(N(C2CCN(C(C3CCOC3)=O)CC2)C)=O)c(F)cc(OC(F)F)cc1F C1(C(=O)NCc2cn(CC#C)nn2)CCN(C(=O)C=CCF)CCO1 c1(C(N(C(C)CNC(c2cc[nH]c2)=O)CC)=O)cccc2[nH]c(C)cc12 C1(c2c(O)cccc2)CCCN(N2CCC(c3nncs3)CC2)C1 C1(NC(C2C(C3(CC)CC3)C2)=O)CCOCC1NC(=O)CCSc1ccccc1 c1(C(N2CC(CN=c3ncc(Cl)c[nH]3)C3(COC3)C2)=O)ccc2scnc2c1 c1(C(N2C(CN(C(C(=O)NCC)=O)CC)CCC2)=O)cn(C)nc1Br C(=O)(C(C)C(C)NC(c1cc[nH]c1CCC)=O)NC(CCCC)C C1(NC(C2CCC(OC)C2)=O)COC2(CNC(=O)CCNC(=O)CO)CC1C2 N1(C(C(C=C)O)=O)CCc2c(CNC(C3CCOC3C3CC3)=O)cccc2C1 c1(C(=O)NC2(C)CCN(C(C3(Cl)C(C)(C)C3)=O)C2)coc2c1C(=O)NCCC2 C(=O)(CCCCCCCC)NC(CNC(C(CC=C)(C)O)=O)CC N1(C(c2c(N)ccc(OC)c2)=O)CC2CCCC(NC(=O)Cc3cnsc3)C2C1 C1(NC(C(C)=CC2CC2)=O)COC2(C1)CN(C(c1coc(Cl)n1)=O)C2 C(=O)(C1Cc2ccccc21)NC(C(=O)NCC(C(C)C)(C)O)CC1CCC1 C1(CC(=O)OCC)CCN(N2CCOCC2C(F)F)C1.C(C(F)(F)F)O c1(C(N(CCNC(CC(CCC)C)=O)CC2CC2)=O)cc(O)c2sccc2c1 C1(C(=O)NC(C(=O)N(C)Cc2nncs2)CO)CC2(CC2)CO1 CC(CNC(c1cnc(=N)[nH]c1)=O)C(F)C(=O)NC1CC1F c1(NC(C(CCCNC(c2scnc2Cl)=O)O)=O)cnc2[nH]cnc2c1 c1(C(=O)NC(CC)CN(C)C(C2(c3ccc(F)cc3)CCC2)=O)cc2c(s1)CCC2 C(=O)(CC(=O)NCC(c1ccccc1)CNC(C1CCC(F)C1)=O)NCC#C c1(C(=O)NC(CCNC(C(C=CCCC)O)=O)(C)C)cc(N(C)C)ccc1N N1(C(C=COCC)=O)CC2CCC1C1CN(C(c3occ(C)c3C)=O)CC21 N1(C(CS(C(C)C)(=O)=O)=O)C2CCC1C1CC1(NC(C1CC1F)=O)C2 CC1CC=C(C(=O)NCC(C)(C2CC2)NC(=O)C(C)OCCOCCO)CC1 CC(C)C(C(=O)N(C)CCN(C(=O)C(=O)NCCC(F)(F)F)C)NC(=O)CO c1(C(C)C)[nH]nc(C(N2CCC(NC(=O)CSc3ncccn3)C2)=O)c1Br Cc1conc1CC(=O)NC1CC(NC(=O)CCc2csc(Br)c2)C1 C12(CNC(c3cc(C)[nH]n3)=O)CN(C(C3(n4cccn4)CCC3)=O)CC(F)(C1)C2 CCCC(CCCNC(C1(C)CNC(=O)C1)=O)NC(=O)CCOCC(F)(F)F Cc1cccc2c1CN(C(=O)C(O)C1CN(C(=O)C(C)(F)F)C1)C2 C#Cc1cc(C(N2CCC(C)(CNC(C3CC4CCC3C4)=O)CC2)=O)ccc1C Cc1cc(=NC(=O)c2ncsc2NC(c2cc(Br)c(O)c(Br)c2)=O)[nH][nH]1 C(=O)(CCCCCC#N)NCCCCCC(=O)NC(C1CCCO1)CC N1(C(c2nc(OC)c(C)s2)=O)CC(NC(=O)CCc2cc(C)[nH]n2)C2CC2C1 C=CCC(CNC(=O)CC1CC1C1CC1)C(=O)NCCc1cocn1 C1(NC(C2(C(=O)NC)CC2)=O)CN(C(=O)C(C)SC)CC1c1ccnn1C c1(OCC(=O)NCC2CCC(NC(C3C(C)C3C)=O)C2)cccc(Cl)c1Cl C(=O)(CC(C)N(C)C)NC1C(C(=O)NC(C(=O)OCC)C2CC2)CC1 CP(C)(=O)c1c[nH]ccc1=NC(=O)Cc1c(F)cccc1Cl C1(CC#C)(C(=O)NCCCOC(F)(F)F)CCN(C(C2CNC(=O)C2)=O)C1 C1(NC(c2ccccc2F)C)Cc2ccccc2N(C(C2CCCC2C)=O)C1 c1(CC(=O)NC(C(CO)NC(c2c(CC)cco2)=O)C)ccc(OC(C)C)cc1 c1(OCC(=O)NCC(O)CNC(C2(C(F)(F)F)CC2)=O)ccccn1 N1(C(C(CC)(CC)CC)=O)CCC2(CCCCN(C(c3[nH]c(O)nc3C)=O)CC2)C1 Cc1ccc(C=CCC(N2CCC(NC(c3ccnnc3)=O)C(F)C2)=O)cc1 c1(C(N2CC3C(C(=O)NCC(C(C)(C)C)CO)(C3)C2)=O)cccc2c[nH]nc12 C1(NC(c2n(C)ncc2)=O)COC2(CCN(C(c3c(O)cccc3Cl)=O)C2)C1 Cc1nn(C)cc1C1=NOC(C(N2CCN(C(=O)CCF)CC2C(F)F)=O)C1 C12(CNC(c3ccc(Br)o3)=O)CCC(CC1NC(C1CCCS1)=O)C2 C(=O)(C(CCCC)NC(C1CCOCC1)=O)NC(CCC=C)C Cc1cc(Cl)cc(Cl)c1OCC(=O)NC(C)(C)C(C)NC(C1C=CCCC1)=O N1(C(CC2C(C)CCO2)=O)CCC(NC(=O)CO)C(F)C1 C1(n2cc(C(C)O)nn2)CC2CCC1(NC(=O)Cc1cc(Br)cs1)C2 N1(C(CCCCC#C)=O)CCC2(CC1)CC2CNC(=O)COCCCOCC=C n1(CCOC)cc(C(=O)NCC(C)CN(C(=O)CN(C)C(C)C)C)c(C)n1 n1(CC(=O)NC(C2CSC2)C)cc(CNC(=O)C(C)C2(O)CCC2)nn1 C(=O)(C(F)C(C)C)NCCC1CC(C(=O)NC(C=C)COC)C1 N1(C(C(C(C)C)N(C)C)=O)CCOCC2(COCCN2C(c2ccoc2)=O)C1 c1(C(N2CCC(C)(NC(C(CC)OCC)=O)C2)=O)nc(C)n(C)c1C C1(NC(c2cc(C)c(O)nn2)=O)CN(C(=O)CCC(F)(F)F)CC2(CCC2)C1 C#CC1C(C(=O)N(C)CCOCCNC(C2CCCOC2)=O)C1(C)C N1(c2snc(SC)n2)CCN(C(=O)CCc2c[nH]c3ccccc23)CC(O)C1 CC(C)CC(F)(F)C(=O)NCCN(C(=O)Cc1ccc(C(F)(F)F)cc1)C(C)C c1(NC(=O)NCCc2ccc(Cl)cc2F)c(F)ccc(Cl)c1F N1(C(CC(COC)(C)O)=O)CC2(CC(NC(=O)CC(C)SC)CO2)C1 CC1(C)CN(C(c2cccc[n+]2[O-])=O)C(CNC(C2CC(F)C(=O)N2)=O)CO1 c1(OC)ccc(Br)cc1C(=O)N(CC(C)NC(=O)C(n1cc(Cl)cn1)C)C C12(NC(C3N(C(CSCCCC)=O)CCC3)=O)CC1CN(C(=O)OC)C2 CC(C)(CNC(c1cc(CNC(C2CC2Cl)=O)cs1)=O)CC(F)F N1(C(c2cnc(C(C)C)[nH]2)=O)CC(NC(c2cnn(C(F)F)c2)=O)CCC1C C1(C(=O)NCC(C(C)C)NC(=O)C(C(C)C)C(C)C)CCc2cnn(C)c2C1 C1(NC(c2c(CCC)nco2)=O)CC(C)N(C(c2cnc(CC(C)(C)C)o2)=O)C1 C(=O)(C1CCCc2c1ncn2C)NC(CCNC(c1c(C)nns1)=O)(C)C CC1CNc2c(C(N3CC(C)(NC(=O)C(C4CC4)N(C)C)C3)=O)cnn2C1 c1(COC)cccc(C(=O)NC(C)CC(C)NC(=O)CCC(N)=O)c1C C(=O)(C(C)(O)C(F)(F)F)NC(C(C)(C)NC(CCC1C(C)C1)=O)C c12nocc1CCNC(=O)C2.CC(CNC(=O)C)NC=O.C(C)(C)(C)OC(N)=O CCCC(C(O)C(=O)NCCn1cnnc1)NC(C1CN(C)C(=O)N1)=O C1(NC(C(CC)CC2CCCC2)=O)CCCC12CN(C(c1cc(F)n(C)n1)=O)C2 C1(CNC(CCNC(C)=O)=O)CCC2(CC1)CCN(C(C1CC=CCO1)=O)CC2 c1(SCCC)cccc(C(N2CCC(F)(CNC(C3CCCCS3)=O)C2)=O)c1 C1(C(=O)NCC(C)(C)OCC(N2CCOC(C#N)C2)=O)CC(=O)NC(=O)C1 C(=O)(CCCCC(C)C)NC1CCC(c2nnc(C(CCCC)C(C)O)o2)CC1 C(C(C(C)(C)C)NC(C1(C)CC(C)(C)C1)=O)NC(c1cnc(C)[nH]1)=O Cc1csc2c(N3CC4CC(NC(=O)COCC5CCCCC5)C4C3)ncnc12 C#CCC(CC(F)F)C(=O)N1CCCC(C(N2CCC(F)(C#N)C2)=O)C1 CC1(C)CCCN(C(=O)CNS(C)(=O)=O)C1CNC(=O)CC1CSC1 c1(C(c2nnnn2C(C)(C)C)NCC(C)F)cnc2ccc(Cl)cn12 c1(CC(N2CC3CCN(C(c4ccco4)=O)C3C2)=O)cnc2c(=O)[nH]ccn12 CC(C)C(O)C(=O)N1CCCCC1C1CCNCC1 C(=O)(CCCC(=O)NN(CC(C)C(N)=O)C(C1CCC(OC)C1)=O)OCC CC(C)CC(=O)C(=O)NCC1(CN(C(=O)CC2CCOCC2)C)CC1 C1(C(=O)NC2(CF)CCN(C(=O)C=C(Cl)Cl)C2)CCc2nncn2C1 c1(NC2CC(CC(=O)NCCN3C(C)CCC3C)C2)c(F)cc(Br)cc1Br C1(CNC(C(=O)NCC)=O)CCC2(CCC2)C1NC(c1cccc(Cl)c1OC)=O c1(OC)ccc(C(=O)N(C2CCN(C(=O)C(F)(F)C(C)O)CC2)C)cc1C C1(C(=O)NCC2(CCNC(COCc3scc(C)n3)=O)CC2)CC(C)CC(=O)N1 c1(C(=O)NC(CC)CNC(c2csc(CC(F)(F)F)n2)=O)ccc(O)c(C)c1 c1(C(N(C(CNC(C2N(C(CCC)=O)CCC2)=O)C)C)=O)ccc(SCC)cc1 N1(C(CC2CCC(C)(C)C2)=O)CCCCC(NC(C2CC2F)=O)C1 N1(Cc2c(C)ccc(C)n2)CCC2C1CCCN2C(=O)Cc1ccc(Cl)cc1F c1(C(N2C(C)(C(=O)NCC3CN(C(C)=O)C3)CCC2)=O)ccc2cccnc2n1 C1(C)(COC)C=CC(NC(=O)C(CC2CNC2)Sc2cn(CC3CC3)nn2)C1 c1(C(=O)NC2CC(NC(c3cc(C)[nH]n3)=O)C2)n[nH]c(C(C)C)c1Br N1(C(CCC(=O)N(C(C)C)C)=O)CCC(NC(=O)CCC(C)N(C)C)C12CC2 N1(C(C)C(=O)NC2CC(CNC(c3coc(Br)c3)=O)C2)CCCCCC1 c1(C(=O)NCCCCNC(C2C(=C)CC2)=O)ccn(C2CCCCC2)n1 N1(C(CC2(C)CC2(Cl)Cl)=O)CC2(C1)CN(C(C1CCc3n[nH]cc3C1)=O)CCO2 C12(CNC(C(C)OCC=C)=O)CC1CN(C(C1CCOC1CC)=O)C2 C1(C(N(CCOc2c(C)cccc2)C)=O)COCCN(C(c2ccon2)=O)C1 C(=O)(C(C)(C)C(C)(C)O)NC(COC)CC(=O)NC(C)(CO)C(=O)OC C(=O)(CC(C(C)OC)NC(c1cc2occc2[nH]1)=O)N(C(CC)CO)C c1(C(=O)NCc2ccc(Br)c(Cl)c2)cccc2c1CCN(C(C1CCCC1)=O)C2 c1(C(N2CCC(CC(=O)NC)CC2)C(=O)NCCSC)ccc2c(n1)CCCC2 C1(C(=O)NCC(C)(C)CNC(c2cn(CC(F)F)cn2)=O)CC2CCC2C1 c1(C(N(C2CCN(C(C=CCC)=O)C2)CCC)=O)ccc(NC(C)=O)c(F)c1 c1(C(=O)NCC2CCC(NC(CCOCC)=O)CC2)cccc2c1OCO2 c1(NC(=O)CN2CCCC(CNC(C3CC3C3CC3)=O)C2)ccc(F)cc1 CCC(C)CC(C(=O)NCC(F)F)NC(=O)C1=CCCOC1 c1(C(N2CCCC(CC)(NC(C34CC(F)(C3)C4)=O)C2)=O)cccc2c1CC(=O)N2 C=C(Cl)C(C)(C)C(=O)Nc1cccc(NC(=O)CN2CC(C)CC(C)C2)c1 N1(C(C2CCN(C)CC2)=O)CCCC12CCCN(C(=O)C(C)(C)C(C)(F)F)C2 N1(CC)C(=O)CCC1C(=O)NC1COCCC1NC(=O)CSc1ccccc1F C1(CC(=O)NC(n2cc(C3CC3)cn2)C)CCN(C(=O)Cn2[nH]cnc2=N)C1 C1(CC)CN(C(=O)Cc2nn(C)cc2Cl)CCN1C(c1cnc(C(C)OC)s1)=O c1(C(=O)NC2(CF)CCN(C(c3sccc3F)=O)C2)cnc2ncccc2c1 c1(OC)cccn2c(=O)cc(C(=O)OCC(=O)OC(C)(C)C)nc12 N1(C(C=Cc2ncc(C)[nH]2)=O)CCC(CNC(=O)CC=C(Cl)Cl)C(C)C1 c1(CCO)ccc([N+](=O)[O-])nc1.c1(OCCOCCNC(=O)C=C2CC2)ccccc1 C1(COC)CN(C(c2scc(C)c2C)=O)CCN1C(C1CC1C)=O Cn1ccc(C(=O)NCC2(O)CC(NC(C3CCC3(F)F)=O)C2)n1 c1(C(=O)NCC2OCC(CNC(=O)C=C3CCC3)C2)sc([N+](=O)[O-])cc1Cl O=C(C(CO)c1cc[nH]n1)N1CC(CCO)(NC(C2(n3ccnn3)CC2)=O)C1 c1(CN2CC3CN(C(c4c(OC)nccc4)=O)CC32)ccc(Br)c(F)c1F c1(C(C)NC(c2cncnc2)=O)cccc(C2CCN(Cc3cnn(C)c3)CC2)c1 N1(C(C(=O)NCCCC(=O)OCC)C)CCC2NCCC2C1 C(=O)(C(C)CCCOC)N(CCN(C(CCSCC)=O)C)CCOC N1(C(c2nc(C)n(C)n2)=O)CC(C2CCCN(C(=O)C3=C(Cl)CCOC3)C2)C1 Cc1cc(S(=O)(=O)N2CCN(C(c3ccc(C)c(C#N)c3)=O)CC2)c(O)cc1Cl S(=O)(=O)(c1ccc(Br)nc1)N1C(C(=O)OC)(OC)CCC1 C1(C(N2CC(N(C(c3nccc(COC)c3)=O)C)C2)=O)CCOC2(CCCC2)C1 N1(C(C(C)Sc2nncn2C)=O)C2CCC1CC(NC(C1CCC(C)(C)OC1)=O)C2 c1(OCC)ccc(C(=O)NCc2ccsc2OC)c(OC)c1 N1(CC(=O)NC2C(CNC(CN(C3CCSC3)C)=O)COC2)CCCNC1=O CCC(CC)CCC(=O)N1CCC(CCNC(C2CCCC3(CCC3)O2)=O)CC1 CCC(CC(F)(F)F)C(=O)N1CCCCC(NC(c2cc3c(s2)CCC3)=O)C1 N1(C(Cc2cnc(C)s2)=O)CC(CNC(=O)COc2ccccc2)CC1(C)C N1(C(C=CC=CCC)=O)CCOC2(C1)CN(C(C1(C3CC3)CCCO1)=O)C2 C1(C)(C(N(CCC(C(C)C)NC(c2c(O)cccc2Cl)=O)C)=O)CCOC(C)C1 Cc1nc2ncc(C(=O)NC(C)CC(C)NC(C3CCC=CCCC3)=O)cc2o1 CP(C)(=O)CC(=O)NC1CCC(CC(N2CCCCC2C(F)F)=O)CC1 c1(C(=O)NCC(CNC(C#CC2(C)CC2)=O)CO)ccnc2cnnn12 C12(CNC(CN3C(C)CCC3C)=O)CC(CO1)N(C(=O)Cc1ccc(O)cc1)C2 CC1CC(C(=O)NCC2(NC(C3Cc4nncn4C3)=O)CC2)CC(C)(C)C1 N1(c2c(C)cnc(C)n2)CCC2CCC(NC(C3(O)CCCC3)=O)C1C2 Cc1nc2c(C(=O)NC3CCCC3NC(c3c[nH]c(=N)cc3C)=O)cccc2o1 CC1=C(C(=O)NC2CC2CNC(=O)C=Cc2ncccc2C)C(=O)OC1(C)C N1(C(COCCCC)=O)CCCC(O)(CC(=O)Nc2cc(Br)n(C)c2)C1 N1(C(c2ccc(I)cc2Br)C(=O)NC)CCN(Cc2ccccc2)CC1(C)C CC1CCCCN1CC(=O)NCC1CCCCC1NC(=O)COCCC(F)(F)F Nc1c(C(=O)Nc2cc(-c3ccccc3)cnc2O)cccc1C(F)(F)F n1(CC)nc(C(=O)NC(CNC(=O)CCNC(C2CCC2)=O)C(C)(C)C)cc1C C1(C(N(CCC(C)O)C)=O)CN(C(c2cscn2)=O)CC12CCC2 C#Cc1cccc(C(=O)NC(C)(C)CCNC(=O)C(S(C)(=O)=O)C2CC2)c1 c1(CC(=O)N(C2CCN(C(C(CC)n3ccnc3)=O)C2)C)cnn(C)c1C(F)F C(=O)(C1(C)NC(=O)c2ccccc21)NC(C)CCCNC(=O)C(Br)=C(C)C C(=O)(CCN(C(=O)Cc1ccco1)C(C)C)N(CCC)CC1CC1 N1(C(C#CC(=O)O)c2ccccc2)CCc2nnc(C(F)(F)F)n2CC1 C(C1(O)CCCc2ccccc21)NCC(N)Cc1cncnc1 n1(-c2cccc(C)c2)cc(S(=O)(=O)N2CCC2C(N2CCOCC2)=O)cn1 C1(OC(C(C)(C)Oc2ccc(CO)nc2)=O)CCOC(C)(C)C1 c1(CCC(=O)NCC(CNC(CC(=C)Br)=O)OC)ccc(OC)cc1 c1(C2(C(N3CC4C(NC(=O)C(F)C5CCC5)(CC4)C3)=O)CC2)ccc2c(c1)OCO2 c1(-c2cccc(C(=O)NC(c3nncn3C3CC3)C)c2)cc(=NC=O)[nH][nH]1 C(=O)(C(CC(F)F)NC(C1(N(C)C(c2nn(C)cc2Cl)=O)CCCC1)=O)OCC c1(-c2sc(C)c(C(=O)Nc3ccc(Br)c(C)n3)n2)cnc2ccoc2c1 n1(CC)nc(C)c(C(=O)NCC2(CCNC(=O)CCn3c(C)csc3=O)CC2)c1Cl C1(C(N2CC(C(N)=O)OCC2)=O)C2C(CN1C(c1cc[nH]c1)=O)C2(C)C c1(CC(=O)OCC(N2CC(OCC3CCC3)C2)=O)cncc(C(C)(C)C2CC2)c1 c1(C(N(C(CC)CNC(C2CCOC2C)=O)C2CC2)=O)nccc(N)c1Cl CC1(C)CN(C(C2COCCC2NC(c2csc(Cl)c2)=O)=O)CCO1 C(=O)(C1COc2ccc(F)cc21)N1CCC(NC(=O)C(F)=CCCF)C12CCC2 C1(NC(CC=CCC)=O)CC(O)CN(C(c2cscc2C(N)=O)=O)C1 C(C(=O)NCCc1cn(C(C)CCCCO)nn1)(C(=O)N(C)C)NC(C)=O.C1CN1 N1(c2ncc(C)cn2)CCCC2C1CCN2C(c1ccc2nc(O)sc2c1)=O N1(C(C2C=C(C)CS2)=O)CCCC(F)(CNC(=O)Cc2n[nH]c(C)n2)CC1 C1(O)(CNC(CC(CC)CC)=O)CCCN(C(=O)C#CC2(C)COC2)CC1 N1(C(C2N(C(C3CC(SC)C3)=O)CCOCC2)=O)CC(=O)NCC12CC2 C(=O)(C1CCCc2ccnn21)N1CCC(N(C(c2[nH]cc(CN(C)C)c2)=O)C)C1 N1(C(C)=O)CC(NC(N2CCN(C)C(c3cc(F)cc(F)c3)C2)=O)CC1(C)C C1(C(c2snc(C)c2N)NC(=O)NCc2cccc(C)c2)CCC(F)(F)CC1 C12CC(C1(C)C)NC2=O.C(C)(C(=O)NC(C)CCC1CCCC1)OC(C)=O N1(C(CS(CC)=O)=O)CCC2C(NC(C3(C)CC4CC4C3)=O)C2C1 C(=O)(C(C)(C)CNC(=O)C(CCC1CC1)NC(c1[nH]ccc1C)=O)NCC c1(C(N(C2CCN(C(=O)CCN3CCOC3=O)C2)CCC)=O)sccc1F Cc1c(ON2CCCCC2)cccc1C(=O)NC12CC(C(=O)NCCC#N)(C1)C2 c1(OC(C(N2CCC(NC(c3cnc(C)[nH]3)=O)CC2)=O)(C)C)ccc(F)c(F)c1 C1(NC(=O)CCc2cn[nH]c2)C2CC1CN(C(=O)C=Cc1ccccn1)C2 Cc1cc(C(=O)NC2CC(NC(=O)C3=CCCOC3)C2)cnc1C(F)(F)F c1(C(=O)NC2C(C)CCN(C(c3cncn(C)c3=O)=O)C2)cnc2nccn2c1 C(=O)(C#CC(C)(C)CNC(=O)CNC(N)=O)NCC1N(C)C(=O)OC1 CC1(OCC(=O)NC2(CCO)CCN(C(=O)CC34CC(C3)C4)C2)CCOCC1 C1(C(=O)NCCc2c(C(=O)NCCS(CC)(=O)=O)c[nH]n2)CC2CC(=O)C1O2 c1(C(=O)NCCC2N(C(=O)Cc3cncnc3O)CCCC2)ccccc1[N+](=O)[O-] Cc1ccc(Cl)c(C(=O)NCC2CCCC2NC(c2cnccc2Br)=O)c1 N1(C(c2ccc(N(C)C)cn2)=O)CCCCCC1C(=O)NCc1ccc(Cl)cc1 N1(C(CSc2cccc(C)c2)=O)CCC(CO)C(NC(=O)CC2C=CCC2)C1 Cc1ccc(C(C)(C)C(=O)NCC(C)NC(C2CCC(C)(C)CC2)=O)c(C)c1 C1(C(CN(CCO)Cc2cc(C)[nH]n2)=O)CCC(CC(=O)O)CC1 Cn1cc(C#N)cc1C(N1CC(NC(=O)CC(F)(F)F)C2(CC2)C1)=O CC1(F)CN(C(c2snc(Cl)c2Cl)=O)CCN(C(C2(O)CCC(F)(F)CC2)=O)C1 C1(C(=O)NCCCCNC(C(C)(C)NS(C)(=O)=O)=O)CC2COCCN2C1 Cc1ccc2cc(C(N3CC4(C3)CN(C(=O)C(F)=CCCF)C4)=O)ccc2c1 C1(CC(C)NC(=O)CCN2CCC2)CC2CCC(C1)N2C(=O)CCc1csc(=N)[nH]1 c1(CC)ccnc(C(=O)NCC2CCCN2C(=O)CNC(c2cnccn2)=O)c1 N1(CCNC(c2c(C)cc(C)s2)=O)CCCN(C(C2CCC(C(N)=O)O2)=O)CC1 C1(CNC(CCOCCOCC)=O)CCN(C(=O)CCS(C)(=O)=O)CC1F c1(C(=O)NC2CC(F)(CNC(C3(Cc4cnn[nH]4)CCC3)=O)C2)ccnc(Cl)c1F CC1=C(C(=O)NCCC(C)N(C)C(c2cn[nH]c2)=O)C(C)(C)CCC1 N1(C(C=CCOC)=O)C2CCC1C(CNC(=O)CC(c1ccc(F)c(F)c1)C)C2 N1(C(CC2(NC(C#CC(C)(C)O)=O)CC2)=O)CCCC2NC(=O)CC12 C1(C(N2CC(c3c(C)con3)C2)=O)CCC2CCC1N2C(=O)CC(C)(F)F c1(C(C(=O)OC(C)(C)C)Nc2nccc(-c3ccnn3C)n2)ccc(Cl)c(Cl)c1 c1(NCCCC(=O)NC2C(NC(CNC(=O)OC)=O)CC2)ccccc1OC CN1CCCCC1C1CC(CNC(=O)NC(c2cnnn2C)C2CC2)C(O)C1 c1(CNC(C(=O)NC(c2ccc(CN(C)C)cc2)C)=O)cc2c(Cl)nccc2o1 N1(C(C(CC2CCC2)OC)=O)C2CCC1CN(C(c1cc(C#N)cn1C)=O)C2 CC1(C)CC(C(=O)NCC2(O)CCC2)CN(C(c2ccc(C#N)s2)=O)C1 c1(C2(C(=O)NC(C3CN(C(CC(=O)NCC#C)=O)C3)C)CC2)ccc(F)cc1C C1(N(C(=O)COc2ccc(Cl)cn2)C)CC2CC1N(C(=O)C=C1CCSCC1)C2 N1(C(C2C(CC)C2(F)F)=O)CC2C(CN(C(=O)C(C)(C)C3CCC3)C)C2C1 c1(C(N2C(C(=O)NCc3ncccc3Cl)C=CC2)=O)ccc(O)c(F)c1 C(C)(CCN=c1cc(C)nc(N2CCCC(c3c[nH]nc3C)C2)[nH]1)OCC C(CN=c1[nH]c(=NC2CC(Cc3ccccn3)C2)[nH]c2c1COC2)SCCCC Cc1c(O)ccc(C(N2CCOCC2C(N2CCC(=O)C(C)C2)=O)=O)c1O C=CC(C)(O)CC(=O)NC(CCCOC)C(=O)NC(C1CC2(CCC2)C1)C C(C(COC)CC(=O)N1CCC(CN(C(=O)C=Cc2cncn2C)C)C1)OC c1(C(=O)NCC2CCOC2)cnn(CCNC(=O)C(F)C2CCCC2)c1 C1(CC#C)(C(=O)NC2CCCC2CNC(=O)CC2CC(N(C)C)C2)CCOCC1 Cc1cc(Cl)ccc1CC(N1CC(C)(NC(C2CCOC2C)=O)C1)=O CC(C)(C(=O)NCC#CC(=O)NCCCCCF)C(F)(F)F C(CC1CC1)(CC(=O)NC1CCCCC1O)NC(=O)CCc1csnn1 C1(C)(CNC(c2c(C)nn[nH]2)=O)CC(F)(F)CN1C(c1ccc2n[nH]cc2c1)=O N1(C(CC2(OC)CCC2)=O)CC2(CCC(NC(=O)CC3CCCC3C)CC2)C1 c1(C(N2C(C)COC(CO)C2)=O)cn2c(n1)CCN(Cc1ccc(Cl)s1)CC2 c1(CNC(C2(c3cccc(Br)c3)CCN(C)C2)=O)cnn2c1CCCC2 c1(C(N(CC2CCN(C(C=CCCC)=O)CC2)CC)=O)ccc([N+](=O)[O-])cc1 C(=O)(C(C)C(C)(F)F)N(CCC(C)NC(c1c(OCCC)cccn1)=O)C N1(CC)N=C(C(=O)N2CC(NC(=O)CSCc3cccs3)CC2C)CCC1=O C(=O)(C(O)CC(F)(F)F)NC1C(NC(CCCC(=O)N(CC)CC)=O)COCC1 c1(C(N2CCC(C)(NC(CC(CCC)C)=O)C2)=O)cc(F)c(F)c(F)c1F c1(C(C(=O)NCC(CC)NC(c2cccc(F)c2)=O)C)cccc2ccccc12 c1(C(N2CC(CC)N(C(=O)C=CCOC)CC2)=O)cnc2ccnn2c1C c1(CC(=O)NC)ccnc(NC(=O)Cc2scnc2C)c1 C(N=c1nc2c(ncn2C)c(NCc2cc(Br)ccc2F)[nH]1)C1N(CC)CCC1 CCCCC(CC)CC(=O)N1CCN(C(C2CC(C)(F)C2)=O)CC12CCC2 C(=O)(C1=Cc2ccccc2C1O)N1C(C2(NC(CCCN=[N+]=[N-])=O)CC2)CCC1 C12(C(=O)NCC(CNC(C3CC=CCC3C(=O)O)=O)O)CCN(CC1)C2 N1(C(=O)C(C2CCCCC2)O)CCCC2(CCN(C(C3CCOC3)=O)C2)C1 C12(C(N(CC(CC)NC(=O)Cc3coc(C4CCCC4)n3)C)=O)CCC(C1)C2 C1(CCC)CN(C(=O)CCC2CCC(=O)C2)CC1C(N1CC(CCC)C1)=O n1(C(C(=O)N(C(c2nn[nH]n2)CC)C(C)C)C)cnc2sccc2c1=O N1(C(C(C)OCCC#C)=O)CCOCC(NC(C2(C)CCC(=O)N2)=O)C1 C(=O)(CC(=O)N1CC(C(C(=O)NCC(F)Cl)OC)C1)NC C1(C(=O)NCC)C(C)C1C.C(=O)(CCOCC)N(C(C)CNC(C)=O)C(C)C C#CC1CCN(C(C2C(C)CN2C(=O)CC2CCCC(=O)N2)=O)CC1 C1(O)(CNC(CCC=CC)=O)CCN(C(=O)C2=CCC2)C1 c1(C(=O)NC(CNC(CC2(OC)CC2)=O)CC(C)C)nc(Cl)ccc1N N1(C(Cn2nc(C)oc2=O)=O)CC(N=[N+]=[N-])CC1C(=O)NCC1CC(C)C1 C1(CC(N2CCN(C(CNC=O)=O)CC(O)C2)=O)CCC2(CCOCC2)CO1 N1(C(CCOC)=O)CCCC1C1CCN(C(=O)C(C)OC2CCCCC2)C1 C12(NCCNC(CCCCNC(=O)OC(C)(C)C)=O)CCC(N)(CO1)C2 N1(C(C(CO)OC)=O)CC2CCCN(C(=O)CN3CCC3C)C2C1 C1(C(=O)NC2CCC(F)(CNC(c3nn(C)c(Cl)c3)=O)C2)CS(=O)(=O)CC(=O)N1 C(=O)(C1=CCCSC1)NCC1(OC)CCN(C(=O)Cc2cncnc2O)C1 c1(C(N2C(C)(CNC(C3(CC)CCCCC3)=O)CCC2)=O)cc(C)cc(Cl)c1N C1(NC(C(C)NC(C)=O)=O)CCCC(C(=O)Nc2ccc(CO)c(F)c2)CC1 Cc1ccc(C(N2CCC(CNC(c3ccc(C(F)(F)F)s3)=O)C2)=O)nc1 c1(SC(C)C)ccc(C(=O)OCC)cc1.C1(C=O)C=CCN(N(C)CS(C)=O)C1 C1(C(=O)NC2(C)CC(NC(CCC(C)(C)O)=O)C2)CC2CCC(C1)C2O C1(CCC(=O)NC2(C(C)N(C)C)CC2)CCN(C(=O)CC2CC(F)(F)C2)C1 C(CCC1CCC1)(C(=O)N1CCCC1)NC(=O)N(c1ccnc(Cl)c1)CC1CC1 CC(C)(C)CC(=O)N1CCN(C2CCN(C(C3(CCO)CC3)=O)CC2)CC1 c1(C(N2C(C)C3CC2C3NC(=O)CCc2ccn(C)n2)=O)ccc2n[nH]cc2n1 C(=O)(C1=CSCCO1)N(C1CCCN(C(c2c(C)ocn2)=O)C1)CCO C1(CC(N)=O)CCCCCN1C(=O)Cn1cc(CNC2CCOCC2)nn1 C1(NC(C2N(C(CCSC)=O)CC(F)C2)=O)CCCC2CCCCC12 C1(NC(c2c(C)ocn2)=O)CC2(C1)CC2C(=O)NC1CCCC1O C1(NC(CCN(C)CC)=O)CC1C1CCCN(C(C2(COC)COC2)=O)C1 c1(CN2CCC(O)(C(=O)NC3CCC(F)(F)C3)C2)c(Cl)ccnc1Br Cc1cc(CN2CC(F)(F)CC2C(N2CC(O)(c3cc[nH]n3)C2)=O)ccc1O c1(C(=O)NCC(C2CC2)NC(C(C=CC)O)=O)ncc(N)nc1C C1(NC(COCCCC#C)=O)CN(C(=O)CCC(=O)c2ccc(CC)cc2)C2CC12 C1(NC(CCc2ncc(C)[nH]2)=O)CCCCC12CCN(C(=O)C(Cl)=CCl)CC2 CC(=Cn1ccnn1)C(=O)NCCNC(C1CCC(=O)N1)=O c1(OC)cccc2c1CCC2=O.C(=O)(C(C)S(C)(=O)=O)N1c2cn(nn2)CC1 c1(-c2c(C)ccs2)ccc2cc(C(=O)Nc3cncnc3)sc2c1 c1(NC(CSCCC(=C)CO)=O)ccc([N+](=O)[O-])cc1[N+](=O)[O-] CC(CCN(CC(c1cccs1)C)C)CC(=O)O N1(C(=O)NCCc2cc(OC)c(O)cc2)CC2CN(C)CC2C1 N1(C(C(C)C2CC2)=O)CCN(C(=O)CCOC2CC2)CC(O)C1 Cc1nc(-c2cn(CC3CCCC3NC(C3CC34CC4)=O)nn2)ccc1F N1(C(CCC(C)(C)F)=O)CC2CCC(C1)C(NC(c1cc(Cl)no1)=O)C2 C12(NC(=O)CCc3cnc[nH]3)CC1CN(C(=O)COC1CCC1)C2 n1(CC)cc([N+](=O)[O-])c(C(=O)NC2CC3CC(NC(C4CC=CCC4)=O)C3C2)n1 CCCCCCCCC(=O)N1CSCC1C(N1CCCC(CO)(CO)C1)=O C1(C(N(CC(C)N(C(=O)Cc2ccno2)C)C)=O)CC(F)C(=O)N1 C1(C(C(=O)N(C(C)C(=O)[N+](C2CCN2CC(F)F)([O-])NC)CCC)C)CCC(=O)C1 Cc1c(C(=O)NC2COCCC2NC(c2c[nH]c(=O)cn2)=O)cnn1C(C)(C)C c1(CC=C)ccccc1C(=O)NC(C)CN(C(c1csnn1)=O)CC c1(C(=O)NCCNC(C2(C)N(C(C)=O)CCC2)=O)cc2cncn2c(O)n1 c1(C(N(C)CC2C(C(=O)OC)C2)=O)n[nH]c(O)n1.N12CC(C1)NC2=O Cc1cc(C)n2ncc(C(N3CCC(CF)(NC(c4cscc4C)=O)C3)=O)c2n1 c1(C(=O)NCC2CN(C(c3csc(C(F)(F)F)n3)=O)C2)cc(F)c2cn[nH]c2c1 C1(CNC(CN2CC(=O)N(C)C2=O)=O)CC2CCC1N(C(c1sccc1F)=O)C2 C1(NC(CCc2c(C)ncs2)=O)CC(O)CN(C(c2coc(C(C)C)n2)=O)C1 N1(C(CC(n2c(CC)ncc2)C)=O)CCCC12CCN(C(C1CCCO1)=O)CC2 C(=O)(C(O)CC(C)(C)C)NCCC(C)N(C)C(C1CC(CC(F)F)C1)=O C(N=c1cc(Cl)c(O)n[nH]1)C1C(N)CN(C(C(C)C)=O)C1.C(F)(F)F C1(NC(=O)Cc2cc[nH]n2)CC2CN(C(=O)Cc3cnsc3)CCN2C1=O c1(C(N2CCCC(C)(NC(C(CC(C)C)F)=O)C2)=O)cc(S(C)(=O)=O)co1 C12(NC(=O)C3=CCC3)CCCC1CN(C(c1cnc3[nH]cncc1-3)=O)C2 C(CCC(=O)NCCCCN(C(=O)C=CC(=O)OC(C)(C)C)C1CC1)C1C(C)C1 C1(C)(C(N(C2(C(N(CCCC)C3CC3)=O)CC2)C)=O)CC(C)=NO1 C1(NC(CCC(=O)OC)=O)CN(C(c2cnn(CCF)c2)=O)C2(CCCOC2)C1 C#Cc1ccc(C(=O)N(CCNC(=O)C(C)C2CCCO2)C(C)C)c(F)c1 C1(C(=O)OC)CCCCC1NC(=O)CC(C)NC(C1C2CC(=O)CC12)=O C1(C(CNC(C2CCS(=O)(=O)N2)=O)F)CCN(C(=O)C(CC2CC2)CC2CC2)CC1 N1(C(C(C2CC2)OC)=O)CC2CCC2(CCNC(c2cccn2C(C)C)=O)C1 C1(NC(=O)Cn2cc(CO)nn2)CCCC12CN(C(=O)C(CO)c1ccccc1)C2 N1(C(C(COC)OC)=O)CC2CCN(C(c3c[nH]nc3F)=O)CC2C1 CC1c2c[nH]nc2CCC1C(=O)NCC(O)CNC(C1CC(F)(F)C1)=O C(=O)(C(C)CC(C)(C)C)NCC1ON=C(C(=O)N(C)Cc2cc(C)ncc2)C1 c1(NC(C=Cc2cncc(C)c2)=O)nccc2[nH]cc(Br)c12 c1(CN2C(C(=O)Nc3cccc(C(=O)OC)n3)CC(F)C2)cc(F)c(Cl)c(Cl)c1 CC1(C#CC(=O)NC2CC(NC(=O)C(O)C(F)(F)c3ccccc3)C2)CC1 CC1CC2(CO)CC1(NC(C1CCN(c3ccncc3)C1)=O)C2 N1(C(C2CC(=O)OC2)=O)CCC(n2cc(CNC(=O)CCF)nn2)CC1 c1(OC)ccc(C(N2CC(NC(c3scnc3Cl)=O)CC2CO)=O)c(C)n1 CN1CCC(CCN(CC(=O)NC(=O)CC2CCC(=O)NC2)C2CC2)CC1 c1(C(=O)NC2(C)CCN(C(=O)CC3CCCCC3)C2)ccc(S(C)(=O)=O)s1 C1(C(C(=O)NC2CC(C)(NC(C)=O)C2)OC)CCC(F)(F)CC1 C(CCCCC(=O)NC1(C)CC(OC)CN1C(c1cc(C)n(C)c1C)=O)OCC N1(C(C(C(C)C)SCC)=O)CCC2C(NC(c3cc(C)nn3C)=O)CC12 C(=O)(CCC(=O)NN(C)C)NC1(n2cc(CC(C)(C)C)nn2)CN(C(=O)OC)C1 c1(CC)ccc(OC)cc1C(=O)NC1CCC1CNC(c1ccc(C)cc1N)=O c1(N2CCC(O)C(NC(c3c(OC)nccc3Cl)=O)C2)ncc([N+](=O)[O-])cc1I C(=O)(C1CCCc2ccnn21)NC1CCN(C(C(CC)SC)=O)CC1 c1(C(N2CC(C(N3CCCC(C(=O)OC)C3)=O)(CF)C2)=O)cccc2cc[nH]c12 N1(c2ccc(C)cc2C)N=C(C(=O)NC2CC(C)(C(=O)O)C2)CCC1=O n1(CC(=O)NCc2cnccc2Cl)ccc(=NCc2cc[nH]n2)nc1O C12(C(N3CC(NC(CC(c4ccc(Cl)cc4)N(C)C)=O)C3)=O)CC(C1)S(=O)(=O)C2 N1(C(C(C)CC2CCC2)=O)CCCC(C)(C(N2CC(CO)C3(CC3)C2)=O)C1 C1(N2CCC(COC(C(C)CNC=O)=O)C2)CCCCCC1.CC(F)(F)F C1(C(N(CCCCN(C(=O)CC(=O)Nc2ccccc2)C)C)=O)CCC=CO1 C1(CNC(C(CC)CC)=O)CN(C(C2(CCF)CC2)=O)CC2(CCC2)O1 C1(C(CNC(CC2(CC)CCC2)=O)C2CC2)CCN(C(=O)CNS(C)(=O)=O)CC1 N1(C(C2C(C)C2)=O)CCC2(CCCN(C(c3snc4ccccc34)=O)C2)CC1 N1(C(CNC(=O)C=CC(N2CC3C(CO)C3C2)=O)=O)CC2(CO)CCC1CC2 C(=O)(C=CS(=O)(=O)CC)N1CC(OCCNC(CC(CC)C)=O)C1 C1(N(C(=O)CCc2ccoc2)C)CCCC(CNC(=O)C(C)(C)C#N)C1 C1(CN(C(c2c(CC)noc2)=O)C)CCCCN1N1CCC(OC(C)C)C1.C=O C12(CNC(=O)CCn3ccnn3)CC(CNC(c3nc(C(F)F)cs3)=O)(CO1)C2 c1(CC(=O)NCC2CCCNCC2)cccc2sccc12 N(C(=NCCN(C)C1CC1)NCC(O)Cc1ccccc1)C(C)C.CC(C)C N1(C(c2n(C)nnc2-c2ccccc2)=O)CCC2(NC(=O)CC3CCC3)CC2C1 N#Cc1ccc(Cl)c(CNCCN2CCN(C(C3C4COCC34)=O)CC2)c1 C1(C)(CCS(C)(=O)=O)c2nnnn2CCS1.CC(CC(C)(C)OC)N1CCCC1 O(NC(=O)CCN(C(=O)C(c1ccnn1C)O)C(C)C)C(CC)CC c1(C=O)cc(C)ccc1C.c1(C(CC)(C)C)nnc(C=O)n1C.C1(=O)C(C)O1 C(c1cccc(F)c1F)=CC(N1CCC(NC(C(=O)N(C)C)=O)C(CO)C1)=O N1(C(=O)Cc2cnc(C(F)(F)F)s2)CCN(C(C2CC23CCCC3)=O)C(CF)C1 N1(C(C2OCCN(CC)C2)=O)CC2CC1CN(C(=O)CC1CCCO1)C2 N1(C(c2cccc(F)c2)C(=O)NCCCCCC)CCC2(COC(C(=O)OC)C2)C1 Cc1ccc2c(=NCC3C4CN(C(=O)CCOCC(F)(F)F)CC34)[nH]cnc2c1 C(=O)(C(C1COC1)NC(=O)CCN(CC(F)F)C)NCCC Cn1nnc2cccc(C(N3CCN(C(=O)C(O)C4CCC4)C(C4CC4)C3)=O)c12 c1(C(N2CCC(CN(C(C(CCC)OCC)=O)C)CC2)=O)cnc(OC)c(Cl)c1 C(CCCCCCC)NC(C(=O)N(CCC)C)=O.c12cc([nH]n1)COC2=O.OC C(=O)(C1CCCn2cnnc21)NC1CC(O)(CNC(c2c[nH]cc(C)c2=O)=O)C1 C1(C(N2C(CC(C)C)CC2)=O)N(C(c2cccc(F)c2N)=O)CC12CCCC2 c1(OC(C2COCCN(C(C3CC3(Cl)Cl)=O)C2)=O)ccc2c(c1)OCCO2 c1(C(N2CCCC(CNC(C(CCC#C)O)=O)C2)=O)cc(Cl)cc2ccncc12 c1(C(=O)NC2CC(CC(=O)N(CCCCO)C)C2)ccn(C)c1 C(=O)(C1=CCCCC1F)N1C2C(C(N(CC(F)(F)F)CC)=O)C(C2)C1 c1(C(C)C)ccc(C(N2CCC(F)(C(=O)NC(C)(C)CO)C2)=O)c(Cl)n1 C(=O)(C(C)(C)CNC(C1CCC(C(=O)Nc2ccncn2)C1)=O)NCC c1(CCC)cc(C(N2CCC(CCNC(c3ncccc3Cl)=O)C2)=O)ccn1 c1(CCNC(C2(C)CCC2C2CC2)=O)nnc2n1CCNC2 c1(C(=O)NC2(C)CC(NC(=O)Cc3ccco3)C2)ccccc1C(F)F CC1CCCC(N(C(=O)CN2CCN(Cc3nccs3)CC2)CC2CC2)C1 c1(C(=O)NC2C(NC(CSc3cccc(C)c3)=O)C2)ccc(C2CC2)nc1C c1(C(N2CCC(C)(NC(=O)CCCCC(N)=O)C2)=O)ccc2[nH]ccc(=O)c2c1 C(=O)(C1CCCc2ncc(C)n21)NC(C(CC)OCC1(F)CC(NC(N)=O)C1)=O C(CC1CC1)(C(O)C(N)=O)NC(C1(CN(C(c2ccc(SC)s2)=O)C)CC1)=O CC1CN(Cc2cccs2)CC1(c1nnnn1CCCF)NCCCCN(C)C c1(N2CCC(NCc3scc(CC)n3)C2)[nH]c(=NC2CC2CC)nc2c1cnn2C n1(CC(=O)NCCN(C(=O)C(C)(C(C)C)OC)CCC)cc(Cl)c(O)nc1=O N1(C(CN2CC(OC)C2)=O)CC(F)(F)CC1CCNC(=O)CC1(NC(C)=O)CC1 C#CCC(CC(=O)N1CCC2CC12)NC(C1COCC1(C)C)=O C1(C)(NC(C2(C(F)F)CC(=C)C2)=O)CCCN(C(C2(C)CCOC2)=O)C1 c1(CCC(=O)NC(CC)(C)CNC(=O)Cc2cc(C(C)C)no2)ccccc1C C1(NC(C2(C=C)CCOCC2)=O)CN(C(=O)CCCN=[N+]=[N-])C2(CCOC2)C1 c1(C(N2CC(N(C)C(C3(n4ccc(C5CC5)n4)CC3)=O)C2)=O)ccccn1 N1(C(C2SCC(=O)C2)=O)CCC2C(C(=O)NCCC(F)F)C2C1 c1(C(=O)NC2CCN(C(CC(C=C)C)=O)CC2(C)C)cc2c(s1)CCC(C)(C)C2 C1(C(=O)Nc2cnc(OCC)[nH]2)CCN(C(=O)Nc2ccc(F)c(C)c2)C(C)C1 N1(C(c2cccc(C)c2)=O)C(C(=O)O)CCC12CC2 C1(C(N(C2CCCN(C(=O)CC(C)(C)C#N)C2)CC)=O)Cc2c(C)cccc2O1 c1(OC)ccc(NC(C2CCCC(C(=O)O)CC2)=O)c2c1C(=O)NC2=O c1(C(C)CC)c(-n2nc(-c3cncnc3)nc2CCS(N)(=O)=O)cccc1Cl c1(C(N2CCCC2)=O)cc(C(CC(CO)NC(c2cccnc2)=O)=O)n[nH]1 CCCCCCN(CC(=O)NC1(F)CC(NC(=O)CC(C)n2cccc2)C1)C CC(C)(C(=O)NCC1(O)CC(NC(=O)CC#N)C1)N1CCCC1 c1(C(=O)NC2(CC(=O)NC3CCN(CC)C3)CC2)cccc(C#N)c1C N1(C(c2c(CNC(C=Cc3cccc(N)c3)=O)ocn2)=O)CCCC2(CC(O)C2)C1 C#Cc1ccc(C(=O)NC(C)(CNC(c2cccn3nncc23)=O)CO)cc1C Cc1[nH]cc(C(=O)NC2CC2NC(=O)Cc2c(Cl)cccc2Cl)c(=O)c1Cl C1(C(N(CC(C(C)C)C)C)=O)CN(C(c2cc(CO)[nH]n2)=O)CCC1(C)C C12(CC(N3CC(C(C)NC(CCCC#C)=O)OCC3)=O)CNC(=O)C(C1)C2 O=C(C1CCCc2ccnn21)NCC(C1CCN(C(C2CSCCS2)=O)CC1)O N1(C(c2cncc(N)n2)=O)CCCC(NC(=O)C(C2(O)CCCCC2)(F)F)CC1 N1(C(CN(C)C(c2ncccc2Br)=O)=O)CCCC2(CC2)C1 N1(C(C(CC)F)=O)CC2CC1(CNC(C1CC1c1cccc(OC)c1)=O)C2 C(=O)(C(CC)C(F)(F)F)NC1C(C)CN(C(c2cn3ccnc3s2)=O)C1 CC1(C)C(C(N2CCC(O)CC2)=O)CCN1C(=O)COCC(F)(F)F N1(C(C(COCC)C)=O)CCN(C(=O)CC2(C)CCCCC2)CC1CF c1(-c2cncc(C#CC)c2)cccc2sc(C(=O)Nc3cnc(C)c(C)c3)cc12 c1(OC)cccc(C(=O)NCC(C2CCC2)NC(c2cc(CO)n(C)n2)=O)c1C Cn1cncc1C(O)C(N1CCC(NC(C2CCC2)=O)C1)=O N1(C(c2c(NC)cccc2)=O)CCC(O)C(C(=O)NCC2CC(O)C2)C1 c1(C(=O)NCC2C3CN(C(C(COC)(C)O)=O)CC32)cc2c(cn1)NC(=O)CO2 c1(C(N2C(CC(N3CC(=C)C3)=O)COCC2)=O)cnc2ccc(Cl)cc2n1 c1(OC)c(C(=O)NCC(CO)NC(=O)CC(C)(F)F)csc1Cl C(C(C)(C)C(=O)NOCCCO)N(C)C(C1(CCN2CCCC2)CC1)=O O=C(C1CCc2scnc21)NCCC1CN(C(=O)CC2CCC=CCC2)CCO1 O=C(CC1=CCN(C(C2CC=CCC2)=O)CC1)N1CC=CC1 N#Cc1cc(C(N2CCC(CNC(=O)CC3CCC3(F)F)C2)=O)ccc1F CC(C)CC(C(=O)Nc1cc(Cl)cc(Cl)c1)NC(=O)C(c1ccc(C#N)cc1)O C1(CNC(c2c(C)scc2)=O)CCC2(CN(C(C3CCCC4(CCC4)O3)=O)C2)O1 C12(CNC(C=CCC)=O)CCC(CNc3cnc([N+](=O)[O-])cc3C)(CC1)OC2 c1(C(=O)NC2C(NC(C(C)OC3CCCC3)=O)CC2)csc(Cl)c1Cl c1(C(C(N2CCCC(C)(C(N(C3CC3)CC)=O)C2)=O)C)c[nH]c2ccccc12 C1(NC(Cc2cn(CC)nc2)=O)CCN(C(C2CCC2CC(C)C)=O)CC1 c1(C(=O)NC(C)CC(C)NC(c2cc(F)nc(F)c2)=O)ccnc2[nH]c(O)nc12 C1(NC(COc2c(CC)cccc2)=O)CCN(C(C2CCC(O)CC2)=O)C(C)C1 c1(C(=O)NC2C(CC)N(C(=O)CNS(=O)(=O)NC)CC2)nn(C)c(Cl)c1Cl N1(C(c2ccc(OCCO)nn2)=O)CC2CCCC2(NC(C2CC(F)(F)C2)=O)C1 C1(C(=O)NCCC)(NC(=O)CC2CCC3CC23)CCN(C)C1 C1(C(=O)NCCCN2CC(NC(c3cncc(C)c3)=O)C2)COCCC1(F)F c1(C(C)C)cc(C(N2CCC(C)(C(=O)NC3CCN(C)C3)C2)=O)ccn1 N1(C(C(CC#C)C)=O)CCCC(NC(=O)CN2CCS(=O)(=O)CC2)C1C c1(OC)cc(C(N2CC(CC=CC(=O)NCC(C)(C)CC3CC3)C2)=O)ncn1 C1(C(=O)NCCC(C(C)C)NC(C(CC)C)=O)CCc2cc(C)ccc2O1 c1(CC)nnc(CNC(=O)CC(C)NC(=O)CC(C)OC)s1 N1(CCN=C(NCC(C)OC)NCC(=O)NCCCl)C(=O)c2ccccc2C1=O c1(C(N2CCC(NC(Cc3nc(C)sc3)=O)CC2C)=O)cccc2c[nH]nc12 C1(O)(CNC(c2csc(O)n2)=O)CCCN(Cc2nc[nH]c2[N+](=O)[O-])C1 C1(C(C)(C)C)C(NC(=O)C=Cc2ccco2)CCN1C(c1ccc(C(F)F)o1)=O C(=O)(C(C)(C)CC(=O)N1CC(N(C(=O)Cc2cccc(Cl)n2)C)C1)OC c1(C(=O)NC2CC(CO)N(C(c3ccnc(C4CC4)n3)=O)C2)cn2c(n1)SCC2 C1(C(=O)NCC2(NC(c3cc(C)on3)=O)CCCCC2C)CCCCN(C)C1=O N1(C(c2ccn(C3CC3(F)F)n2)C(=O)NCC(=C)C)CCCC2(CC=CCC2)C1 Cc1nc2ncnn2cc1C(=O)NC1CCCN(C(=O)C2=CCCS2)CC1 N12CCC(C1)NC2=O.C=C(C)COCC(=O)NC(C)C1CC1 C(=O)(C1CC(O)c2ccccc21)NC(C)(C)CCNC(C1CC1C(C)(F)F)=O c1(C(=O)NC(C)C(F)NC(c2cc3n(n2)CCO3)=O)cc(-n2cccn2)ccn1 c1(CC)ncc(Br)c(C(=O)N(CCNC(C2CC2F)=O)CC2CC2)n1 C1(C(=O)NC2CN(C(CC)=O)C2)CCN(C(=O)C(CC)CCOC)CC1C C1(NC(C2CC(=C)C2)=O)CC2(C1)CC(C(N1CC(C(=O)NC)C1)=O)C2 N(C(=NCCC(O)C(F)(F)F)NC1CCOCC1)Cc1c(O)ccc(Cl)c1 C(CC(C)C(=O)N(C(CNC(=O)COCc1ccc(F)cc1)C1CC1)C)=CC C1(NC(=O)CCn2ccnc2)CC2(C1)CC2C(=O)NCCN1CC2CC2C1 CC1(C)CC(C(=O)NC2CC2NC(=O)C=C2CCC2)CNC1=O c1ccc(-n2[nH]nnc2=N)cc1.c1(S)coc(Br)n1 S(=O)(=O)(c1cccs1)N1CCC(CNC(=O)NC2CC(CC)C(O)C2)CC1 Fc1cccc2c1CCC2n1cc(-c2cc(Cl)ccc2Br)nn1 Cc1nc(=N)[nH]cc1C(=O)NCC(C)CNC(c1nnn(C)c1C(F)(F)F)=O C1(C(=O)NCCC2CCCN2C(C2(CN(C)C)CC2)=O)(OC)CC(C)C1 Cc1cc(CNC(=O)CCC2CCCN2C(=O)C(C)CC2CC2)n(C)n1 c1(OC)cc(C)c(CN2CC(NC(c3cncnc3)=O)C(F)(F)C2)cc1OC N1(C(c2n(C)ccc2)=O)CCC2(CCN(C(c3cc(Cl)c4c(c3)OCO4)=O)C2)C1 C1(NC(C2(CN(C)C)CC2)=O)CCC(NC(=O)C(C)(CC2CCC2)C2CCC2)CC1 c1(SC)nc(C)cc(=NCC(CC(C)C)NC(c2c(Cl)cnn2C)=O)[nH]1 CC(O)CCCCCC(=O)NCc1cn(C2CCN(C(C3(O)COC3)=O)C2)nn1 C1(C(=O)NCC2CC(O)CN2C(=O)CN2CC3CC3C2)Cc2nccn2C1 N1(C(c2ccc(C)s2)=O)CC2CC1CN2C(C1CCC(C(=O)OC)CC1)=O C(=O)(C1CNc2ccccc21)NC(C1N(C(c2cccc(CC)c2)=O)CCC1)C C#CCCCC(C)C(=O)N1CC(C)(C(=O)NC(c2ccccc2)CC)C1 C(=O)(C1=CCCN(C(=O)CC2C=CCC2)C1)NCC1CC[Si](C)(C)C1 C1(N(C(CCC)=O)C2CC2)CN(C(=O)CCCc2cccs2)CC1(C)C CC(C)CS(=O)(=O)CC(=O)N(CCCCNC(C12CC(C1)C(C)O2)=O)C c1(CC)cc(CC)[nH]c(=NCC(C)(C)CNC(c2nncs2)=O)n1 Cc1ccc(NC(=O)N(C(C)C)C)cc1S(C)(=O)=O.c1(C2CC2)ccccc1 C1(C(=O)NC(CN(C(c2cnn(CCN(C)C)c2)=O)CC)C)(CC)CCOCC1 CON1CC(C(N2CCC2C(N2CCCC2C2CCOC2)=O)=O)CC1=O Cc1cc(C(N2CCC(CF)(NC(c3ccncc3F)=O)C2)=O)cc2[nH]ccc12 C(=O)(C(O)C(C)(C)C)N1CC(NC(c2nccc(CC)c2)=O)C2(C1)CC2 C1(C(N2CC(OCCNC(=O)CCCC3CCC3)C2)=O)CCn2nncc2C1 CN1CCN(CC(=O)NCC(O)CNC(C2CC(=O)N(CC(F)(F)F)C2)=O)CC1=O c1(C(=O)Nc2cnn(C3CCCCC3)c2)ccc(OCC2CCCCO2)cc1 C1(C(=O)OC)CCC(C2CC2)N1C(N1CC2C(CSn3nc(C)oc3=O)C2C1)=O N1(C(c2cc(CC)oc2C)=O)CCCCCC(NC(C2(C)CCC2C(=O)OC)=O)C1 c1(C(N(C2CCCC2)CCCNC(CC(CC)C)=O)=O)cccc2c1CCCC2 C1(C#N)(C(=O)NC2C(C(=O)NCC=C(C)C)OCC2)CCCOC1 C(=O)(CCCF)N(C1CC(CCNC(C(C)NC(N)=O)=O)C1)CCO c1(N(C)C)ccc(C(N2CCC(O)(CNC(=O)CCc3nccn3C)C2)=O)nn1 C(CCc1ccccc1)(C(C)NC(=O)CNc1ccc(Cl)cc1)NC(CCC)=O c1(CC)cccc(C(=O)NC2CN(C(C3CC4CCC3C4)=O)C2)c1 c1(CC(=O)NCC2CC(O)(Cc3ccc(Cl)nc3)C2)cc(O)nnc1O C(C(C)(C)C(=O)N1CC(CC(C)(C)CNC(c2nc(=N)cc[nH]2)=O)C1)SC c1(CNC(c2ncn(C)c2)C(=O)OCc2ccccc2OC(F)F)ccccc1I C1(C(=O)NCC2(OC(C)C)CCC2)CC(C)N1C(C1CC(CC2CC2)C1)=O C1(CC(N2CCCC2C(C)NC(=O)C=CC2CCOC2)=O)(OCC)CCCCC1 Cc1nccc(=NCC2CN(C(=O)C(C)(C)CF)CCC2C)[nH]1 N1(C(CSC)=O)CC(NC(c2ncc(C(F)(F)F)nc2O)=O)CC12CCCCC2 C1(CCNC(c2c(C)nco2)=O)COCCN1C(C1COCCO1)=O c1(NC(c2n(CC=C)nnn2)C2CCC(=O)N2)cnc2ccnn2c1 c1(CC)cccc(CC)c1CC(=O)NC1CC(C)N(C(=O)Cc2ccnc(C)c2)C1 CCC(C)(CCC(C)C)C(=O)NCCOCCNC(=O)Cc1cnnn1C c1(OCC(=O)NCC(C)CNC(C2(Cl)CC2)=O)ccc(F)cc1F N1(C(C=CCCC)=O)CCC(C2(NC(c3cc(C)cc(O)c3)=O)CCC2)CC1 N1(C(C2N(C)C(=O)NC2)=O)CCC2(C1)CN(C(c1cc3ccsc3s1)=O)CCO2 N1(C(c2cnn(-c3ccccc3OC(F)(F)F)c2)=O)CC2CC2(O)C1 Cc1ncccc1C(=O)NCCC(O)C(=O)NC(C)COC(F)(F)F C#CC1(NC(c2cc(Cl)cnc2OCC=C)=O)CCCCC1 CC1(F)CCCCN(C(=O)C=C(Br)Br)C1 O=C1CC2C(C(=O)NCCC3(C(=O)NC4CC5C=CC4CC5)CC3)CC2O1 N1(C(C(CCC)N(C)C)=O)CCC2(C1)CN(C(=O)Cc1occc1C)CC(C)O2 C(c1ccccc1)=C(C(=O)NCC(CC=C)NC(=O)CC)C.C(=O)(C(CCC)N)N c1(CN(C(C(=O)NCC2CCCO2)c2ccoc2)C)cccc2ccccc12 C1(CC)CC1N=c1[nH]c(=NCc2ccn(C)n2)[nH]c2c(F)cccc12 C(=O)(C1=COc2ccccc2O1)N1CC2CCN(C(C3C(OC)CCC3)=O)C2C1 C1(C(=O)NC2CCN(C(C(C(C)C)(C)C)=O)C(C)C2)CN(S(=O)(=O)N(C)C)C1 C1(NC(c2cccc(C3(C)COCCO3)c2)=O)CCC2COC1O2 c1(OC)ccc(C(N2CC(NC(=O)Cn3nnc(=O)[nH]3)C(C)C2)=O)cc1O c1(CC(=O)NC2CC(O)(CNC(c3cnc(SC)s3)=O)C2)cncnc1O c1(C(C(=O)NC2C3CN(C(c4c(C)cc(C)o4)=O)CC32)C)c(C)nn(C)c1C C1(NC(=O)CCn2cc(Cl)cn2)CN(C(=O)CC(Cl)Cl)CCC1C(F)(F)F N1(C(C(CCC)N(C)C)=O)C2CCC1CC(C(=O)NCCCCCN=[N+]=[N-])C2 C=CC(C)N=c1[nH]c(=NCC2CCN(C3CC3)C2)[nH]c2c1CSC2 C1(O)(C(=O)NC(c2nc(C(=O)NC(c3cnn(C)c3)CO)co2)C)CC(CF)C1 c1(CC(=O)NCCC(CC)(C)NC(=O)CCc2cnoc2)cc(C)cc(C)c1 N1(C(c2cccc(C)c2)=O)CC(C)(C)CC1CNC(=O)Cc1cnc(C)[nH]1 N1(C(c2c(C)cccc2O)=O)CC2CCC(C1)N2C(C1CCC2(CCC2)CO1)=O c1(CC)oc(C)cc1C(=O)NCc1ccc(C(N2CCCC(CF)C2)=O)o1 C(CC(F)(F)F)N(C(CN(CCC#C)C(=O)C=C(C)CCC(=O)OC)CC)C S(=O)(=O)(c1ccc(Br)cc1NC1CC2C=CC1CC2)NC(CC)COC N1(C(c2c(CC)c(C)sc2)=O)CC(CO)C2(C1)CN(C(=O)CCNS(C)(=O)=O)C2 N1(C(CCC(=O)NCCC)=O)CC(CNC(=O)CNC(=O)C2CC2)OC(C)(C)C1 N1(C(C(CC)NC(=O)OC(C)(C)C)=O)CCC(CC)(NC(C2CC2F)=O)CC1 C(=O)(CC(C)(C)CC)N1CCC(C2N(C(C(=O)NCC)=O)CCC2)CC1 C(=O)(CS(C)(=O)=O)NC(CNC(c1nc(C)oc1)=O)CO c1(C(=O)NCC23OCC(NC(c4cnc(C)o4)=O)C(C2)C3)cn(C)c(=O)nc1O S(=O)(=O)(c1ccc(N2CCS(=O)C(C)(C)CC2)c(Br)c1)NC1C(OC)C(O)C1 Cc1c(C(N2CC(O)(C(C)CNC(C3CN(C)C(=O)N3)=O)C2)=O)ccn1C(C)C C1(O)(CN(C(C(COC)OC)=O)C)CCN(C(=O)Cc2cc[nH]c2)CC1 C(=O)(C#CC1CCOC1)NCCC1(C(=O)NCC2CN(CC)C(=O)O2)CCC1 c1(C(=O)NC2(CC(=O)N(C(C(=O)OC)CN(C)C)C(C)C)CCC2)ccc(C)nc1C CC1=C(C(=O)N2CC(CC(C)(C)CNC(=O)CC(C)CN(C)C)C2)COCC1 N1(C(=O)NC(c2cc(C)cc(Br)c2)C)c2ccccc2NC(=O)C1C C(C)(CC(C)N=c1[nH]nc(-c2ccon2)s1)NC(C(CCSC)O)=O N1(C(CN(C(C(C)C)=O)C)=O)CCC(C(C)CNC(C2CCCCN2C)=O)CC1 CC1CC(NC(=O)C=CC(N)=O)CCN1C(c1ccc(F)cc1Cl)=O c1(N(C)C)ccc(C(CNC(=O)Cn2cccn2)NC(c2ccn(C)n2)=O)cc1 C1(C(=O)NC2(C(C)(F)F)CC2)CCN(C(c2ccn(CCN(C)C)n2)=O)C12CC2 C1(NC(CN(C(C(C)(C)OCCCO)=O)C2CCCC2)=O)CCOC12CCOC2 c1(C(=O)NCC(C)N(C(=O)C(C)O)CC)c(C)[nH]c2ccc(OC)cc12 c1(-n2ncc(C)c2)cccc(C(N2CCN(C(=O)C3=CCOC3)CC2)=O)c1F C1(C(=O)NC(CC2CC2)C(=O)NCC2(C#N)CC2)(CC)CCNC1=O C1(N(C(CC=C)=O)C)CCN(C(c2csc(=NCC)[nH]2)=O)CC1C C1(C(=O)NC(C(C)NC(C2(C(C)(F)F)CCC2)=O)CO)COC(C)(C)CO1 C1(CNC(Cn2c(C)c(Br)cn2)=O)CC(C(C)(C)C)CCN1C(C1CCC1)=O C(=O)(C1CCc2nccn21)NC1C2N(C(c3c(O)ccc(C)c3)=O)C(CC2)C1 N1(C(C2N(CC)CCOC2)=O)Cc2[nH]nc(C(=O)N(C)Cc3ccns3)c2C1 C1(CCC)COCCN1C(=O)NCCc1csc(-c2cccs2)n1 C1(C(=O)NCCCCC2CCN(C(C(C)C3CCC3)=O)CC2)CNC(=O)CC1C C1(=CC(=O)NCC(C)N(C(C2CCC(C)CC2)=O)CC)CC2CCC(C1)N2C CCCCCCCCCC(=O)NCC1CCCCN(C(=O)Cc2conc2C)C1 C(CN=c1[nH]c2ccccc2s1)NC(c1cnc2ccccc2n1)=O c1(C(N2CC3CN(C(c4cnn(C)n4)=O)C3CC2)=O)ccc2c(c1)NC(=O)CN2 N1(C(c2ncncc2F)=O)CC2CCOC2(CNC(C2(O)CCSCC2)=O)C1 Cc1cc(C(N2CC(NC(c3c(C)cnn3C)=O)C(O)C2)=O)ncc1S(N)(=O)=O c1(NC(CC2(C)CN(C(C3CC(=O)NC(=O)N3)=O)C2)=O)ccccc1S(C)(=O)=O c1(C(N2CCCC(CN(C(Cn3c(C)ccn3)=O)C)C2)=O)cc2sccc2cn1 c1(OC)ccc(CC(=O)N(CCCNC(c2ccsn2)=O)C2CC2)c(C)c1 C=C(CNC(C1CC(C)(C)CN1C(c1ccncc1O)=O)=O)c1ccccc1 C1(NC(c2c(CC)occ2)=O)CCN(C(c2ccoc2C)=O)C(C)C1 C1(C(N2CCCC(N(C(C3N(C)CCCC3)=O)C)C2)=O)CC(=O)C12CCCC2 C1(C(=O)NCc2ccc(OC)nc2)CCCN1NC(=O)C1=NOC(C)(C)C1 c1(C(N(CC(C)NC(CCCC(=O)OC)=O)C)=O)c(Br)nc2n1CCOC2 N1(C(C(CC)n2cncn2)=O)CC(Nc2nnc(C)c(C)n2)CC2(CC2)C1 c1(C(=O)NC(CCCNC(=O)CC2CCCC23CC3)CO)cnc2ccc(F)cn12 C(=O)(CCCc1cccs1)N1CC(CN(C)C(C2(CO)CC2)=O)C1 Cc1nc(CC(C)C)c(C(=O)NCCCCNC(=O)C(C)Oc2ccc(O)cc2)s1 C1(CNC(CC=C)=O)CN(C(c2c[nH]cc2Br)=O)CCC12CCC2 N1(C(c2cc(OC)ncn2)=O)CCCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1 N1(C(C2C(NC(C(C(C)C)NC(C)=O)=O)CC=CC2)=O)CC2(CCOC2)C1 C1(N(C(C)=O)CCN(CC(C)O)C)CCCC1 c1(C(N(CC(CN(C(CCOCC)=O)C)O)C)=O)cc2ccccc2nn1 C(C)(C)(CCCCC(=O)N1CCC(NC(C2(CC3CCC3)CCC2)=O)CC1)OC N1(C(C(c2cnn(C)c2)OC)=O)C2CCC1CN(C(=O)C(C)CCN(C)C)CC2 C12(CNC(CC3(OC)CN(C(C4(CC=C)CCCC4)=O)C3)=O)CCN(CC1)CC2 N1(C(C2(C=C)CCC2)=O)CCCOC(CCNC(c2cc(SC)ccc2O)=O)C1 Cc1c(C(=O)NC23CC(C(=O)NCCCCC4CCOC4)(C2)C3)cccc1Br C(=O)(CCCNC(N)=O)NC(C(=O)NC(C)CCF)C1CCC1 N1(C(C(C2CN(C(C3C(C)(CC)C3)=O)C2)O)=O)CCC2(C=CCO2)C1 N1(C(CCOC)=O)CCCCC1C1CCN(C(=O)C(O)Cc2ccc(Cl)cc2)C1 c1(CN(C(c2c(OC)ncc(C(=O)O)c2)=O)C)cc(Br)cc(F)c1F Cc1cc(=O)n(C)nc1C(N1CCC(NC(=O)C(C(C)C)C(C)C)C(F)(F)CC1)=O c1(C(=O)NCC2CCN(C(C(CCOC)C)=O)C2)cc(Cl)cc(C)c1O c1(C(N2C3CCC2CC(CCCCc2c(C)con2)C3)=O)ncc2c(n1)CCOC2 Cc1cc(C=CC(=O)NC2CC2NC(c2nccn2C)=O)ccc1Br N1(C(c2cc(SC)oc2)=O)CCCC1(C)C(N1CCCC1(C)CO)=O N1(C(C2N(C)CCC2)=O)C2CCC1CC(NC(=O)CNC(c1cccnc1)=O)C2 c1(N2CC(C(C)NC(COc3cccc(C)c3)=O)C2)cc(C)nc2cnc(C)n12 N1(CC(=O)NC23CC2CN(C(c2cc(Br)n[nH]2)=O)C3)CCCS1(=O)=O C1(=O)C(SC)CCSC(C2CCCCC2)CN1.CCC(=O)OC.C1(=O)CN1 C1(NC(C2=C(C)OCCS2)=O)CCC2(CC1)CN(C(=O)CC1OCCO1)CCO2 c1(NC(C2(C)N(C(=O)NCC(=O)OC)CCC2)=O)ccccc1S(C)=O c1(C(=O)OC)cc(F)ccc1NC(C12CC(NC(=O)Cc3cnc(C)s3)(C1)C2)=O N1(C)CCN(C=O)CC1.C(=O)(C(C)C(C)NC(=O)OC(C)(C)C)OC c1(CCOC(C)=O)nc(=NC2CC3CCCC(C2)N3C(C2CC2F)=O)s[nH]1 CP(C)(=O)C(CC(=O)N1CC2(C1)CN(C(C1CCOCC1)=O)CCO2)C(F)(F)F c1(C(N2CCC(CCC(N3CCC(F)(F)C(F)C3)=O)C2)=O)cnn2cccnc12 CC1COCCC1N(C)C(C1(C)C=CCN1C(=O)Cc1cn[nH]c1)=O C1(NC(C2CN(CC)C(=O)C2)=O)CCCCN(C(C2CC3(CC3)C2)=O)C1 C1(c2nc(C3C(OC)COCC3)nn2CCN(C)C)Cc2nccnc2C1.C1(C)CC1 c1(C(N2CCC(O)(CCNC(=O)C3CC3)CC2)=O)c(C(F)(F)F)cccc1F c1(C(=O)NC(C)(C)CN2CCN(C(C3(C)CCCO3)=O)CC2)cc2ncccc2s1 N1(C(C(C)OCCOC)=O)CC(C)(C)CCC1CNC(c1nc(C)ccc1C)=O N1(C(C2N(C)C(=O)NC2)=O)CC(C2CCCCN(C(c3occc3Cl)=O)C2)C1 Cn1nc(CC(=O)NCCCC2CCCN2C(=O)Cc2csnn2)cc1Cl c1(C(N(C2CCN(C(C3CCC(F)CC3)=O)C2)C)=O)cc([N+](=O)[O-])cnc1N N1(C(c2c(CC)c(CO)ccc2)=O)CCC(CNC(=O)C(C)C)C(F)(F)C1 C(=O)(C1=NOC(C)(C)C1)NC1CCN(C(c2nc(C(C)C)sc2)=O)C(C)C1 C12(C(=O)NC)CC(C(F)(F)F)C1CN(C(=O)C(=O)NC(C1CC1CSC)C)C2 N1(C(C(F)OC)=O)CC(CNC(C2CCCOC2)=O)OC(C)(C)C1 C1(C(N2CCCC(CCC=C)C2)=O)CN(C(=O)CCc2ccc[nH]2)CC1(C)C N1(C(COCC(C)(C)C)=O)CCOCC1CNC(c1cnccc1C(F)(F)F)=O c1(C(=O)NCC2(CCNC(C3C(C)OCCC3)=O)CC2)cc2c(s1)CCCCC2 Cc1ccc(C(=O)NC2CCN(C(=O)CCn3ncn(C)c3=O)CC2)c(F)c1F N1(C(c2c(F)ccc(Br)c2F)=O)CCC2(CCC2N2CC(F)(F)C2C(=O)O)CC1 Cc1ccc(Cl)c(C(N2CCCCCC(NC(c3cc(O)ncn3)=O)C2)=O)c1O c1(CC(=O)NC(CC)(C)CCNC(C2CC3(CC3)C2)=O)ccc2ccccc2c1 C=CC1(NC(C2C3CN(C(C4CN(C5CCC5)C4)=O)CC23)=O)CCCC1 C(=O)(C1=Cc2cc(Cl)ccc2OC1)NC1CC(OCC(=O)NCc2ccsn2)C1 c1(C(=O)NCC2CCCN(C(CCCCC#C)=O)C2)c(O)cc(Cl)cc1Cl N1(C(C2CCC(N(C)C)CC2)=O)CC(NC(C2(F)CCOC2)=O)CC(F)C1 Cn1nc(CN(C=O)CCc2ccccc2F)c2ccccc12 Cc1nc(C2CC2)sc1CC(=O)N(CC(C)O)CCNC(C1CC2CC2C1)=O CC1=C(C)CC(C(N2CCOCC(NC(C3CCC(=O)O3)=O)C2)=O)CC1 c1(C(=O)Nc2c(CC)nsc2)c(CNC(c2c[nH]nc2CC)=O)cnn1C C(=O)(C1OCCc2ccccc21)N1CCN(CCNC(CC(CC)(C)C)=O)CC1 n1(CC(=O)NC2CCN(C(c3ccc(C)[nH]3)=O)C2C)ccc2ccccc12 Cc1cnc(C(N2CCN(C)C(CNC(=O)CSc3cccs3)C2)=O)c(C)c1 c1(C(=O)Nc2cc(O)nc(-c3ccccc3)n2)cc2n(c1)CCNC2 N1(C(C2CC(=C)C2)=O)CCN(C(C2(C)CCN(C(C)=O)CC2)=O)C(C2CCC2)C1 c1(OC)ccc(S(N)(=O)=O)cc1C(=O)NCCCCNC(=O)C(C)OCCN(C)C CC(CC1CCCO1)C(=O)NCCSCC(N1CCC1(C)CCO)=O N1(C(=O)C2CC2)CCCCC(F)(F)C1.C12(CCSC1)N(C)C2=O.C12(CCCC1)CCC(=O)N2 C1(NC(C(C)CN(C)C)=O)CCN(C(=O)CC2CCC(=O)NC2=O)CCC1CO C1(NC(=O)CC2CSC2)C2CC(NC(=O)CCNC(=O)Cc3cccs3)CC12 c1(C(=O)NCC(Cn2cc(C(C)O)nn2)OC)cc(C(F)(F)F)cc(F)c1 C(c1ccc(F)c(C)c1)=CC(=O)NCC1N(C(C(c2ccc(C)s2)C)=O)CCC1 N1(C(C2CCCC(OCC)C2)=O)CCCC(C2CN(C(=O)C3=C(C)OCC3)C2)C1 Cc1nnc(N(CCCNC(=O)CC(C)c2ccco2)C(C)C)o1 c1(C(=O)NC(C)C(F)(F)F)cc2c(s1)C1(CCN(Cc3ccccc3)CC1)OCC2 N1(C(CSc2c(C)ccc(C)c2)=O)CC2CC(NC(=O)C(C)(F)F)C(C2)C1 c1(N2CCC(C(C)NC(C(COC)(C)O)=O)C2)nc(C)ccc1C#N C(=O)(C(F)C(C)CNC(=O)Cc1c(C)cnn1C)N(C(C#C)C)CCCC N1(C(C(CC)(CO)OC)=O)CC(C(=O)NCCCOCC2CC2)CC(C)(C)C1 C1(NC(c2ccc(C(C)=O)c(F)c2)=O)CC2CC(C1)N(C(=O)CCC(C)O)C2 C(CCCCC(=O)NC(c1ncc(C)s1)C)N(C(C(C(C)C)SC)=O)C C1(CNC2(c3n(CC(=O)OC)nnn3)CSC(C(C)C)C2)CC(=O)N(C)C1 C1(NC(C2CC(C)C(C)CC2)=O)CN(Cc2cnc(Cl)cc2Cl)CC2(CCC2)C1 c1(OC)cc(Br)c(C(=O)NC2CN(Cc3cc4ccccc4o3)C2)cc1O C(=O)(C1=COCC1)NC(C1CN(C(c2csc(-c3cccc(Br)c3)n2)=O)C1)C CCC(=O)N1CC(OC(C(C)(C)O)C2CC2)CO1 c1(OCC)ccc(C(=O)NCC23CC2CN(C(=O)CCCF)C3)c2ccccc12 c1(C(N(CC(CNC(C=Cc2c(C)ccs2)=O)C)C)=O)c(F)ccc2ccoc12 CC1(C)CCC(CC(=O)NC2CCN(c3ncc(Br)cn3)C2)C1 c1(N)cc(F)cc(F)c1Cl.c1(SC)nccc(S)n1.N12CCCC1CCC2=O c1(OCCCN(CCC)C(C2CC23CCOC3)=O)ccc(F)cc1 C1(NC(C2(C)CC2Br)=O)CCCC2CN(C(=O)C(=O)Cc3ccccc3)CC12 C1(NC(C(C)NC(C)(C)C)=O)CC12CCN(C(=O)CS(N)(=O)=O)CC2 C12(NC(C(C)NC(CC)=O)=O)CCCC1(F)CN(C(c1c[nH]cc1CC)=O)C2 N1(C(CC=CCC)=O)CCCCC(CNC(=O)Cc2ccnc(Br)c2)C1 c1(CNC(=O)NCC2(C)CN(C)C(=O)C2)nc2ccccc2[nH]1 CCCC(C(=O)OC)C(=O)N1CCC=C(C(=O)Nc2cc(O)ccc2C)C1 C(CC1CCCCC1)(C(=O)NCCc1csc(C)n1)NC(CN(CCOC)C)=O c1(C(=O)NC2(CF)CCN(C(Cc3c(C)cnn3C)=O)C2)cc(S(C)(=O)=O)cs1 C12(NC(c3c(CCC)occ3)=O)CCC(CNC(c3scnc3CC)=O)(C1)OC2 Cc1cc(F)cc(C)c1C(N1CC(CNC(c2cn(CCO)nc2C)=O)C1)=O Cn1nnc2c(C(N3CCCC(NC(c4cc(N)cc(O)c4)=O)C3)=O)ccnc12 c1(OC)cc(OCc2nc(N(C)C)cc(C(F)F)n2)cc(SC(C)(C)C)c1 c1(C(=O)N)ccc(C(=O)N(C(C(=O)OC)C2CC2)CC2CC2)c(F)c1.C1(O)CC1 c1(CN(CCCNC(c2ccc(C)s2)=O)C(C)=O)ccc(F)cc1 [N-]=[N+]=NC1COCC1NC(=O)CNC(C1C(Cl)(Cl)C12CC2)=O c1(CNC(C2C(CNC(c3c(N)non3)=O)C2)=O)cnc(O)nc1O C1(CC(C)C)C(=O)N1.C(=O)(CC(=O)OC(C)(C)C)N(CC(=O)OC)CC C(=O)(C(O)CCS(C)=O)N(CCCN(C(=O)Cc1sccc1Cl)C)C N#Cc1cnc(N2CC(CN3CCN(C(c4ns[nH]c4=O)=O)CC3)C2)c(Br)c1 N1(C(c2c(F)cc(C)c(F)c2)=O)CCOC2(CCCN(C(C3CC(C)C3)=O)C2)C1 Cc1ccc(F)c(NC(=O)CCSC(F)(F)F)c1 c12cc(nn1C)CNC(=O)C1(CC1)CNC21CC1.Cn1cc(C=O)cn1.CO C1(NC(=O)NC(c2nc3c(s2)CCCC3)C)CCCCC12CCC2 c1(C(=O)NCC2C(NC(C3(C)CC(=C)C3)=O)C2)cc2ccccc2nc1C c1(C(=O)NC(C)CCCNC(c2csc(O)n2)=O)nnc(O)c2ccccc12 C(=O)(CC(F)(F)C(C)C)OCCCc1ccc(CC)cc1 N1(C(c2c(COC)cc[nH]2)=O)CCCC1C1CCCN1C(=O)CCCCl Cc1cn2c(n1)CCC(NC(=O)NCCn1ncnn1)C2 Cc1cnc(C(=O)NC(Cc2cn(Cc3ccccn3)nn2)CC(=O)O)c(C)c1 C12(CNC(=O)Cc3cnns3)CC(CCO1)N(C(c1ccc(O)cn1)=O)C2 N(C1CCc2ccccc21)C(C(C1(C)CC1)NC(C1C(C(C)(F)F)C1)=O)=O N1(C(Cc2ccc(OCC)nc2)=O)CCCC(C)C1CNC(=O)Cc1ccoc1C c1(C(N(C2CCN(C(C3(COC)CCCC3)=O)C2)C)=O)c[nH]c2cc(F)ccc12 Cn1cc(S(=O)(=O)N2CCC(C#N)(NC(c3ccc(Br)c(C#N)c3)=O)C2)cn1 N1(C(C(C=C)(C)C)=O)CCC2(CC1)CC(NC(=O)CC(C)C)C2 C1(NC(c2cn(C(C)C)nc2)=O)(CO)CCN(C(C2CC2C#N)=O)C1 c1(C(=O)NC(c2cccc(Cl)c2)CNC(C(CC)F)=O)oc(CC(C)C)nc1C N1(C(c2c(OC)nccc2)=O)CCC2C(CCCN2C(C2CCCOC2)=O)C1 C(=O)(N=c1[nH]n(C)cc1C(N)=O)NC1C(OC)CN(C(=O)OC(C)(C)C)C1 c1(C(=O)NC(CC(C)C)CNC(C2C3COCC23)=O)cccc(F)c1Br c1(C(=O)NC2C(CNC(C(CC#C)O)=O)C2)c(C)nc(CCNC2CCC2)nc1O S(=O)(=O)(c1c(C)cc(Cl)cc1Cl)NC1CCCC(CCCC)C1 Cc1noc2nc(C(=O)NCC3CCN(C(c4ccn(C)c4)=O)CC3)ccc12 N1(C(c2c(OC)cncn2)=O)CCC(C(=O)NC2(C)CC=CC2)C12CC2 C1(C(=O)NCC2CC(F)(CNC(C(CC=C)NC(C)=O)=O)C2)CCCC12CCC2 N1(C(c2ccc(CNC(C(CSC)O)=O)s2)=O)CCC(F)(F)CC1 C=CCCCC(C(=O)NC12CCCCC1C2)NC(=O)C(C)COC C1(C)(C(N(CCC)C2CC2)=O)CCN(C(=O)Cc2ccc(C)o2)C1 C1(CNC(CC(C)(F)F)=O)CN(C(=O)C(C)(C)CO)CC1(F)F C1(COCC)CN(C(c2cnc(-c3cccnc3)s2)=O)CC1(F)F c1(CC)nc(C)n(C)c1C(=O)NC1CC1NC(=O)CCP(C)(C)=O Cc1ccc(Br)c(NC(C2(C)CCCN2C(c2cc[nH]c2C)=O)=O)c1 C1(C)(C(=O)NC(C2(O)CN(C(C(c3ccc(C)cc3)=O)=O)C2)C)CCC(O)CC1 Cc1cccn2c(C(=O)NC(C3CCCN(C(C4CCCSS4)=O)C3)C)cnc12 C1(C(N(C(CNC(c2c(COC)ncs2)=O)C)C)=O)CCC(C(F)(F)F)CC1 C1(CCC)CN(C(c2n[nH]cc2C)=O)CC1C(=O)N(CC(Cl)Cl)C CC1(C)CC(CNC(=O)C(F)CC2CCCC2)N(C(=O)CCc2cnn[nH]2)C1 C1(NC(C2C(CC)CN(C(C3(OC)CCC(C)C3)=O)C2)=O)CCCCCC1F C1(C(=O)Nc2cc(C3CC3)ncn2)CC2C=CC1C2.CC12CCN1C2=O CCCC(O)CC(=O)NC1(CCNC(=O)C(C)(C2CC2)OC)CC1 O=C(C1=NOC2(CCC2)C1)NCCC1CSCCN1C(=O)C=Cc1ccc(F)cc1 C(=O)(C(CCSC)NC(=O)Cc1cccc(O)c1)NCC1(C(=O)OC)CCCO1 C1(C(=O)NC(C=C)CO)(NC(=O)CC(C)C2CC2)CC(F)C1 c1(CC)cccc(C(=O)NC2C3CN(C(C)C(=O)NCc4cccs4)CC23)c1 CC1(C)CN(C(c2sccc2Cl)=O)CCC1C(N1CCCCC1CCCO)=O N1(C(CCCCCNC(N)=O)=O)CCC2(CNC(C3CCCS3)=O)CCCCC12 C1(NC(Cc2c(C)cccc2F)=O)CCS(=O)(=O)C12CN(C(=O)C=CC(N)=O)C2 C1(CC)CCC(C(=O)N(C(C)C(=O)OC)C)O1.N1(C=O)CCCC1COC C(CN=c1nc(N2CCCC(n3nccn3)C2)c2ncccc2[nH]1)C1CC(F)(F)C1 c1(OC)ccc(C(=O)NCC#CCNC(c2cnccc2C)=O)cc1Cl c1(C(C(=O)NCCOCC(C)C)NC(C=CC(CC)C)=O)c(C)cccc1Br C1(NC(c2cn(CC)nn2)=O)CC1C1CCCN(C(=O)CCc2cc(Cl)cs2)C1 c1(N2CC(C)(NC(=O)C(C3CCCOC3)N3CCC3)C2)nccn2nnnc12 N1(C(CCCOCC)=O)CCC(N2CCCC2C(N2CCC(N(C)C)C2)=O)CC1 c1(C(=O)OCCC(C)C)ccc(C2CCCN(C(=O)CCc3ccc(Cl)s3)C2)cc1 n1(CC(=O)NCCC(C)N(C)C(c2snc(O)c2Cl)=O)c(O)nc2ccccc12 C1(CCC(N2CCC(CC3CC3)C2)=O)(NC(C2CC2[N+](=O)[O-])=O)CCCC1 C1(CS(N2C(C(C)(C)C)CCCC2)(=O)=O)CN(CC(F)F)c2ccccc2O1 CC(CCC(=O)NCC=CCNC(C1CCc2nccn2C1)=O)S(C)(=O)=O N12CCOC(C1)C2=O.C(C(C)S(C)(=O)=O)CNC(c1nc(CCC)oc1)=O c1(C(=O)NCC2(C)CCCN2C(=O)Cc2cnns2)cc(S(N)(=O)=O)co1 Cc1cn(C)nc1C(N1CCN(CC(=O)NC2(C(N)=O)CC2)CC1)=O N1(C(c2nc(C)sc2Br)=O)CCC(NC(=O)Cc2cc[nH]c2)CC1C C1(CC)CN(C(=O)CN(C)C(C)C)CCN1C(C1CC2CC2N1C(C)=O)=O Cc1c(C(=O)N(C)CCN(C(c2nn[nH]c2Cl)=O)C(C)C)nnn1C1CCOC1 c1(NC(C)CCNC(=O)CCC(=O)NCC(c2nccs2)=O)cc(F)ccc1F N1(C(CCC#CC)=O)CCCC(C2CCCN(C(=O)CCC3CC3(F)F)C2)C1 CCCCCCC(C)C(=O)N1CC(CNC(c2cc(COC)[nH]n2)=O)C(O)C1 C12(C(=O)NC(c3ncccn3)CC)COCC1CN(C(c1ccc(Cl)o1)=O)C2 c1(C(N2CC(F)(CNC(C3CC(=C)C3)=O)C2)=O)cc2cccc(Cl)c2nc1C C1(c2n(CCCCOC)nnn2)(NCCCC(F)F)CCCC(C)CC1 C1(NC(C2C(OC)(OC)CC2)=O)CC2CC1N(C(=O)CNC1CC3(C1)CC3F)C2 C1(NC(c2ccc(OC)nc2)=O)CCN(CCn2ccc(=O)cc2C)C(C)C1 C(=O)(C(C(C)(C)C)OC)N1CC(CNC(C2CCN(C(CC)=O)CC2)=O)OCC1 C(c1cncn1C)=CC(=O)N(C1CCCN(C(=O)C(F)C(C)C)C1)CC c1(NC(C2(OC)CCCO2)=O)ccc(OC)nc1.c12cn(nn1)CC(=O)C(=O)N(C)C2 N1(C(c2cnc(OCC)nc2)=O)CCCC(O)(CNC(c2nn(C)c(C)n2)=O)C1 O(C1CCCc2ccccc21)CC(=O)N(CCCN(C)C(C1(CO)COC1)=O)C c1(C(C(=O)NCC)SC)ccccc1CC.C1(=O)CN1C(C)=O CCCCCCCCCC(=O)NC1CCN(Cc2cccnc2OC)CC1O C(=O)(CCCC(=O)N(C)C)N1CC(CCOC)C1.C12CCC(CC1)CC(=O)N2 C1(NC(CC=C=C)=O)CC(C2CCN(C(=O)CCS(=O)(=O)c3ccccc3)C2)C1 C1(CC)CN(C(c2csc(Cl)c2)=O)CCC1NC(=O)CN(C)C(=O)OC(C)(C)C c1(C(=O)NCC(CCNC(CCCC=C)=O)O)cccc2[nH]nc(O)c12 CC(C)CC(=O)NCC(=O)N(CCC(C)(C)NC(=O)C(C)Oc1ccccc1)C C1(SCC(N2CC3(CCCC3)C2c2ccccc2)=O)CCC2(CCNCC2)CC1 c1(C(=O)NCC(C(C)C)(C)NC(=O)C(C)(O)C2CCC2)cc(C(F)F)ccc1F N1(C(C2(C)CC2(F)F)=O)CC(NC(C2(O)CCCCC2)=O)CC12CCCCCC2 Cc1cc(CC(=O)NC23CC(NC(=O)CSCCC(C)C)(C2)C3)cc(F)c1 N1(C(C=CC=CC)=O)CCC2(CC1)COC(CNC(C13CCC(CO1)C3)=O)C2 N12CC=C(C3(CCC3)NC(=O)C1c1ccns1)CC2.CCC(C)OC C(C)(C(C)(C)C(=O)NC1CCCC1)NC(C(C(C)C)=O)=O CC1=C(C)CC(C(=O)N(C)CC2(O)CN(C(c3ccc(Cl)o3)=O)C2)CC1 C1(C(N2CC(NC(c3cnc4ccoc4c3)=O)C(O)C2)=O)OCCOC12CCC2 C1(=CC(=O)NCC2C(NC(c3occ(C)c3C)=O)C2)CCOc2ccccc21 CCCC(C(=O)N(CC(C)(C)COC)C)OC=CCC(=O)N1CCCC1 C(CCF)(C(=O)NCCC(=O)NO)NC(CCc1n(C)ccn1)=O Cc1cc(CNC(=O)CNC(=O)CC2CC(=O)NC2=O)cc(C)n1 N1(C(CCC2(NC(C3N(C)C(=O)OC3)=O)CCCC2)=O)CCN(C)C2(CC2)C1 c1(CC(N2CCC(C)(CNC(C=CC(CC)C)=O)CC2)=O)cn(C)c2ccccc12 N1(C(CCCOC)=O)CCC2(CC1)CN(C(C1CCC3(CC3)C1)=O)CCO2 c1(C(=O)NCCCN(C(C(CC)n2cncn2)=O)CC)nn2c(c1C)CCCC2 C1(O)(CCNC(C2CC23CCC3)=O)CCN(C(=O)C(O)C2CCCC2)CC1 CC(C)(CC=CC(=O)NOCc1ccsc1)NC(C1CC12CC2)=O N1(C(C(C)N(C)C)=O)CCCC1CN(C(=O)CCc1cncs1)C C12(CC(=O)O)CN(Cc3nc4ccccc4[nH]3)CC(c3ccccc3)(C1)C2 C1(C(=O)NCC2C3CC(C(=O)OC)(C3)N2)CCOC(C)(CC)C1 C(=O)(C(=O)C(C)(C)C)NCC(CNC(C1(OC)CCOC1)=O)C CC12CCN(C(OC3COCc4cc(Br)ccc43)=O)CC1C2(Cl)Cl N1(C(CCC)=O)CCN(C(C2CCC2C#N)=O)CC(C)C1.c12ccc(cn1)[nH]2 C1(NC(CC=CCNC(C2N(C)CCOC2)=O)=O)Cc2ccccc2C1 C(=O)(C(CN(C)C)C(C)C)NCC1OCCN(C(c2ccn(CC(C)C)n2)=O)C1 Cc1cnc(C(=O)OC(C)(C)C)c(C)c1.C1(=O)CC(CCON(C)C(C2CC2)=O)O1 N1(C(C(COC)C)=O)CCCCC1C(=O)NCCC1CCC(C)CC1 Cc1cc2cccc(CNC3CCC4CCCCN34)c2[nH]1.N12CC3C(C3C1)C2=O C1(CC=C)(NC(=O)C(F)C(F)(F)F)CCCN(c2cc(C(F)F)ncn2)C1 c1(C(=O)NC2CN(C(c3c(OC)ncnc3)=O)CC(O)C2)ccnc2cc[nH]c12 Cc1ccc(OCc2cc(Br)cc(I)c2)c(-c2ccc(C(F)F)cc2)c1 c1(C(C)=O)cc(C(=O)NCC2CCCC2NC(C2CCSC2)=O)no1 C12(CNC(=O)C3CC3)CN(C(C3CC4(CCCC4)C3)=O)CC1(C(F)(F)F)C2 C1(NC(=O)CC2CCCC2)CC2CCC1N2C(c1cnn(CCF)c1)=O N1(C(C2CC(C)=C(C)CC2)=O)CC2CCN(C(=O)C=C3CCOCC3)C2C1 c1(C(=O)NCC(CNC(c2c(CC)ccs2)=O)O)ncc(C(C)(C)O)cn1 C1(NC(COC)=O)CCC2CN(C(C3(CSC)CCCCC3)=O)CC2C1 c1(OC)cccc(N2CCC(CNC(=O)CC3CCCCC(=O)N3)C2)c1[N+](=O)[O-] C1(CCNC(C(c2ccccc2Cl)C)=O)CSCCN1C(=O)CCOC1CC1 c1(C(N2CC(O)CC(NC(CC3CN(C)C3)=O)C2)=O)cc2c(cnn2C)nc1O C(=O)(CCCC(F)(F)F)NCC(CCC)C(=O)NCCCn1ccnn1 CC(F)(F)C(F)C(=O)N1CCCCC(CNC(C2CCCN2C2CC2)=O)C1 c1(CN2C3CN(C(COC(c4ccccn4)C)=O)C(C3)C2)c(F)ccc(O)c1F N1(C(CCCN(C)C)=O)Cc2cccn2CC(C(N2CCOC(C3CC3)C2)=O)C1 C(=O)(C(C)(C)CC#N)N(CC(=O)NC1CCC2(C(C)C)CC12)CC#C C1(N(C(C(CCC)SC)=O)C)CCN(C(c2ccc(CO)s2)=O)CC12CC2 c1(C(=O)NCC(CC=C)NC(C2OCCC2C)=O)csc2ccccc12 Cc1cncnc1C(=O)NCC1CC1CNC(=O)Cn1cccnc1=O c1(C(=O)NC2CCC3(C2)CN(C(c2sccc2F)=O)C3)c[nH]c2nccc(Cl)c12 C1(N(C(=O)CSc2cnsc2)C)CN(C(=O)Cc2nc[nH]n2)CC1O C(N=c1cc[nH]c(=NCCc2nc[nH]n2)[nH]1)C1C(C)(C2CC2)C1 c1(SC)cc(NC(C2CCN(C(N(C(CNC3CC3)=O)C)=O)CC2)=O)cnc1C N1(C(C(C=C)O)=O)CCC(N2CCC(CNC(=O)CC3CCS(=O)(=O)C3)C2)CC1 N1(C(c2c(C)ncc(Br)c2)C(=O)NC2(C)CC2)CCCC2(C1)CC2(F)F C(=O)(CS(=O)(=O)CCO)N(CC(CN(C(c1cc(OC)cc(Cl)c1)=O)C)O)C C(=O)(C(C)Cc1ccncc1)NC(CNC(COCCOCC#C)=O)CO N#CC1(NC(=O)Cc2cccnc2Cl)CCN(C(c2cnon2)=O)C1 C1(CNC(C2C3CCCCC23)=O)(NC(c2cccc(=O)o2)=O)CCC(F)(F)CC1 c1(NC(C(C2CN(C(=O)Cc3c[nH]nc3O)C2)OC)=O)cnn(C)c(=O)c1 c1(C(=O)NCC(C)(C(C)C)NC(C2(CCCC)CC2)=O)cc2c(cc1O)OCO2 N1(C(CC2CCN(C(c3ccn(C)n3)=O)C2)=O)CC2CCCC(O)C2C1 c1(C(=O)NC2CC3CN(C(C4C(C)(CC)C4)=O)C(C2)C3)ccc2ccn(C)c2c1 C1(C(N2CCCC(CCC(=O)NCC3(O)CCC3)C2)=O)C2CCCCCCC12 C(CO)(CCCCNC(c1cc(Cl)cnc1OC)=O)NC(CCC)=O N1(C(C2CCC(CC)O2)=O)CCCC(NC(C2(C)CCCCO2)=O)CC1 c1(C(=O)NCC(C)N(C)C(c2ccc(C3CC3)nc2)=O)cc(C2CC2)n(C)n1 C1(C(=O)NCC2CCN(C)C2)(NC(C(N2CCCC2)C)=O)CCSC1 c1(C(=O)NC2CCN(C(CCC#C)=O)CC2F)cccc2ncc(C)n12 c1(OC)nc(Cl)ccc1C(=O)N(C)CCNC(c1cc(-n2cnnc2)ccn1)=O C1(NC(C(N2CCC(N3CCC(N)CC3)CC2)C)=O)CCC(c2ccccc2)CC1 C1(C(=O)NCCc2cnc(NC(CCNC(=O)CO)=O)s2)CCS(=O)(=O)CC1 c1(CN2CCC(NC(=O)COc3cncc(Cl)n3)CC2)n[nH]c2ccc(Br)cc12 c1(CC(=O)NC2(CN(C(C(C)OCC)=O)C)CC2)cncc(O)c1 N1(C(=O)NC2COCC2F)CCC2CCCC2CC1 c1(NC(=O)NC2CC3CN(C(C(C)SC)=O)C2C3)c(F)ccc(OC(F)F)c1F c1(C(=O)NCC2C(C(=O)NC3(CC)CC3)C2)cc(O)n(C)n1 C1(NC(C(C=C)O)=O)CCCCC12CCCN(C(c1csc(Cl)c1)=O)C2 c1(CC(N2CCC(N(C(C(COC)(F)F)=O)C)C2)=O)c[nH]c2cccc(C)c12 C(=O)(C1=NN(C)C(=O)CC1)N(C)CC1CCCN(C(C23CCCN2CCC3)=O)C1 C(=O)(C#Cc1ccc2c(c1)OCO2)NC(CC)C(=O)NOCCC(C)C Cn1ncc(N)c1C(=O)NCC1(F)CC(NC(=O)CCC2CC2(C)C)C1 N1(C(CC2CCCN(C(c3n(CC)nnc3)=O)CC2)=O)CC2(CCC(=O)N2)C1 c1(OC)cc(NC(=O)C(C)(C2CC2)N(C(=O)C(C)n2ccnc2)C)ccc1O C(CO)(CCCNC(c1cnc(C(N)=O)s1)=O)NC(c1[nH]cc(C(C)(C)C)c1)=O C1(NC(C(Cc2ccc(C)cc2)C)=O)CCN(C(C2(CO)CCC2)=O)CC1CO c1(-n2cc(C(=O)NC3C(CNC(C4(CC)CCC4)=O)C3)nn2)cc(C)ccc1C c1(CN(C(CC)Cc2c(Cl)cccc2Cl)CC)cn(C)c(=O)c2cccnc12 C(=O)(C1=CC2CCCCCCC12)N(CCNC(CN=c1scc(C)[nH]1)=O)C CC(C)C#CC(=O)NC(C)(CNC(c1c[nH]nc1-c1ccccc1F)=O)C1CC1 N1(C(C=CC)=O)CC2CC(NC(=O)Cc3cccc(OCCOCC)c3)CC1C2 C1(C(=O)NCCC(CC)(C)O)N(C(=O)CCSC(C)C)CCCC1(C)C C(=O)(C(CCC)C(C)C)N1CCC(N(C(c2cc(CCC)c(F)cc2)=O)C)C1 CCC(C(=O)N1CC(OC)C(NC(C2CNC(=O)N2)=O)C1)C(C)(C)CC c1(-c2c(CNC(CC(C)NCCC(C)=O)=O)csn2)ccc(Cl)c(F)c1 c1(C(=O)NCC2CC(NC(C)=O)C2)ccc(C(=O)NCCO)cc1 C1(CC)CC(C(=O)NCCCc2ccc(OC(C)C)cc2)CCN1 CCCCCCC(C)C(=O)NCCCC(O)C(=O)NCCCCC(F)(F)F C1(NC(COc2c(C)cccc2)=O)CCN(C(=O)CN2CCOCC2)CC1C c1(-c2cc(C(=O)NC(c3ccc(O)cc3)C)c(F)nc2)cc2ccccc2o1 N1(C(C2(C(=O)OC)CC2)=O)CCN(N2CCOC(c3ccccc3F)C2)CC1 CCCCC(C)C(=O)N1CCC(NC(c2cn(C)nc2C2CCCCC2)=O)C1 C1(S(C)(=O)=O)(C(=O)NC(C)CN(C)C(C2CCCC(C3CC3)O2)=O)CCC1 CC(C)(C#N)CCC(=O)N1CCC2(CC1)CC2NC(=O)Cc1cncnc1 c1(C(N(CCn2cc(C(C)O)nn2)CC)=O)cnc(Cn2cc(Cl)cn2)s1 N1(C(=O)NC(CC2CCOCC2)CO)CCCC2(C1)C(O)CC2O C1(C(N2CC(C)(OCC(=O)NC(CC(C)(C)C)C)C2)=O)CCOC(C)(C)C1 c1(C(=O)NC(C)C=CC(=O)NCC2C3CCCCC23)cccc(=O)n1C N1(C(c2[nH]cc(C(C)=O)c2)=O)CC(NC(=O)C(C)c2ccsn2)C(C2CC2)C1 N1(CC(N2CC(C(C(=O)NC(C)C3CCC3)(C)C)(O)C2)=O)CCCCC1C c1(OC(C)=O)ccccc1C(C)CCNC(=O)CC1CN(C)C1 C12(NC(c3nn(C(F)F)cc3Cl)=O)CCC(C1)C(F)(F)C2 CN=c1cc(C(N2CC(NC(=O)CCCCc3cnc[nH]3)CC(C)C2)=O)cc[nH]1 O=C1NC(=O)C2(CN(C(C3CC4CNCC3C4)=O)C2)N1 c1(C(N2CCCC(C(=O)OCC)(CC)C2)=O)ccn2ncc(CC)c2n1 c1(OC)ccc(C(CNC(=O)C(C)(C)C)NC(=O)CCCn2ccnn2)cc1 Cc1ccc(C(=O)NCC2(F)CC(NC(c3occc3C)=O)C2)c(Cl)c1 c1(CCCNC(C2CCC(n3cc(CN(C)CC)nn3)C2)=O)cc(F)ccc1F c1(OC)cccc2c1C(C(=O)N1CCN(C)C(C)(C(=O)O)C1)CC2 N1(Cc2c(OC)c[nH]n2)CC2(CC(C(N3C(C)CCC3C)=O)C2)C1 c1(C(=O)NCC(CNC(C=CC(C)C)=O)O)ccc2c(c1)nc(O)n2C1CC1 C1(NC(C(C)OCCOC)=O)CCN(c2ncnc3[nH]ccc23)CC(O)C1 Cc1noc(C)c1CNC(=O)COC1CCN(C(c2ccc(=N)[nH]n2)=O)C1 c1(-c2nc(C3CC(C4CC4)C(CSNC(=O)OC(C)(C)C)C3)on2)ncc(Br)cc1F c1(N2C3CN(C(C4(COC)C=CCC4)=O)CC2CC3)ncnc2c(Br)cccc12 Cc1nc(CC(=O)NCC(C)(CO)NC(=O)Cc2ncoc2C)cs1 c12ncc(cn1)NC(=O)C1CC(C1)N(C)C2=O.C1(SC)CC(C)N(C)C1 c1(C(=O)NC(C(C)(C)C(=O)O)CO)csc2nc(-c3cccs3)nn12 N1(C(C(CCC)(C)C)=O)CCC(C)N(C(=O)C=Cc2cncs2)CC1 N1(C(Cn2nc(C)c(Cl)c2)=O)CCC(C)C(NC(c2cnn(CC(F)F)n2)=O)C1 c1(C(N2CCC(C)(CCNC(C(C)OCCC=C)=O)C2)=O)cc(CC)cnc1O C1(CSC2CCCC2)CCCC12CCN(C(=O)CNC(=O)Cn1cc(CO)nn1)C2 C(=O)(NN1CCCOC1=O)C1C(OC)(OC)CC1 C1(C(=O)NCC2(OCC)CN(C(=O)C(C)(C)C(=O)N(C)C)C2)CC2(CCOC2)C1 n1(CC)nnc2c1C(C(=O)NC1CC(O)C1)CN(C(C1(CC(=O)OC)CC1)=O)C2 C1(C(=O)NC(=O)Nc2cccc(Cl)c2)CN(C(=O)C(O)C2CC2)CCC1O C1(NC(=O)NC2CON(CC)C2=O)C2CCN(C(=O)CNC(=O)OC)CC12 N1(C(C(C)OCC(C)C)=O)CCC(CNC(=O)CS(N)(=O)=O)C(C)C1 C1(C)(NC(=O)NCC2N(C(CNC(C(C)(C)C)=O)=O)CC=C2)CCC(F)(F)CC1 CCCC(C(=O)NCCN1CCC(NC(=O)C(C)OCCC(C)C)CC1)N(C)C c1(C(=O)NCC(C2CCCC2)NC(C2C(OC)CCC2)=O)cc(C)nnc1O c1(C(N2CCC3(CCCN3)C2)=O)cccc(OC(F)(F)F)c1[N+](=O)[O-] N1(C(CC2CCC(=O)NC2)=O)CC(NC(C2Cc3cccnc3C2)=O)C2(CCC2)C1 C1(NC(c2ncc(F)cn2)=O)COC2CN(C(c3ccon3)=O)CC12 C1(NC(C(C2CN(C(C3CC(c4ccccc4)C3)=O)C2)OCC)=O)CCNC1=O N1(C(c2ccsc2OC)=O)CCN(C(c2nc(C)ccc2OCC)=O)C(C)C1 C(=O)(C(C)N(C1CCC1)C)N(C(C)CNC(=O)CC1CCCO1)CC c1(CNC2C(CCCC)CCCC2)cc(OC)c(OC)cc1O CC1=C(C(=O)NC(CCN(C)C)C(N2CC(=O)NC3(CC3)C2)=O)COCC1 C1(C(=O)NC(C2(CF)CC2)=O)COCC1NC(CC)=O.n1(CC)ccnc1 CC(C)(CNC(=O)COCCOC)CN(c1ccccc1)C(=O)CCSC(F)(F)F C1(Nc2snc(C)n2)CN(C(=O)C(C)(C)C2CC2)CCC1CO CC1(C)C(=O)N1S(C)(=O)=O.C1(C(=O)OCC(C)(C)C)CC(=C2CC2)C1 C(=O)(C(CC1CCCC1)NC(=O)CNc1cn[nH]c1)NCCNS(N)(=O)=O C1(C)CCCCC1.c1(C(=O)NCc2occ(CO)c2)csc(C2CC2)c1 c1(C(N2CCC(C)(O)CC2)=O)ccc2nccc(C3=CCNCC3)c2c1 C1(NC(CCC=CCC=C)=O)CC(C)CN(C(=O)CCc2ccccc2OC)C1 CCC(CC(=O)N1CC(CO)CC1CO)C(C)C C(CC(C(=O)N1CC(N(C(=O)CC2(C)OCCO2)C)C1)NC(C)=O)SC.COC C1(NC(CC(C(C)C)O)=O)CC2CCC1N(C(c1ccc(=N)[nH]n1)=O)C2 c1(C(c2ccccn2)N(CCC(C)OC)C)ccccc1 N1(C(CCCSC)=O)CC(F)CC1C(=O)NC(C(C)C)c1nc[nH]n1 N1(C(C2CC(c3ccccc3)(C)C2)=O)CCCC(C)(CNCc2nc(Cl)sc2Cl)C1 C1(NC(c2ncc(OCC)nc2)=O)CN(C(C2CCC(C)O2)=O)CC1C1CC1 CC1CN(C(c2cnn(C)c2C#N)=O)C(C)CN1C(c1cc2ccccc2s1)=O Cc1ccc(C(=O)NCC2CCN(Cc3ccc4c(c3)CC4)C2)c(I)c1 N1(C(C2C(C(C(=O)C(C)(C)CC(=O)OC)=O)C2)=O)CC(N)CC12CCC2.COC N1(C(c2cc(CC)nnc2C)=O)CC2CCCC2(NC(=O)CN2CCOCC2)C1 CCCCCCCCCCCC(=O)N1CC2(CC(C(=O)NCC3CC34CC4)C2)C1 C1(CNC(c2ccn(CCC)n2)=O)(NC(=O)CC2CCCCN2C)CCCCC1 N1(C(C2(COC(C)C)CC2)=O)CC(NC(c2cn[nH]c2)=O)C2CCCCC12 c1(C(=O)OC)ccc2sc(NC3CC(C)N(C(C4CC(C)OC(C)C4)=O)C3)nc2c1 C1(CNC(=O)NCCC2(c3ccccc3)CC2)CCCC23OCCC2CC13 c1(C(=O)NCCC2CCN(C(c3n(CC)ccc3)=O)C2)ncccc1C c1(C(c2n(CC)nnn2)NCCC2CCCO2)cc(Br)ccc1OC c1(CNC(c2cnc(NC(=O)OCC)s2)=O)cn(C)nc1C N1(C(C(CC(C)C)OC)=O)CC2CCCC2(NC(=O)CCC2CC(OC)C2)C1 C(CCS(C)(=O)=O)OCC.n12nnnc1C(c1cc(C)no1)NCC2 C(C(=O)N1CCCC1CCCNC(C1COCCN1CC)=O)(C(C)C)OCC N1(CC(N2CCOCC(NC(c3c(C)nsc3)=O)C2)=O)C(=O)C(=O)N(C)C1=O CC(c1ccccc1)=CC(=O)N(C(C)CNC(c1cnc(O)c(F)c1)=O)C C1(C2CCN(C(C3C(CCOC)C3)=O)C2)CCCCN1C(C1CC(C)C1)=O C12(C(=O)NC3(CNC(CN4C(C)CCC4C)=O)CCCC3)CCC(O)(CC1)CC2 C1(CNC(=O)Cn2cc(CN3CCC3c3cccnc3)nn2)CCC12CCC2 C12(NC(c3cc(CNC(c4ncn(C)c4)=O)no3)=O)CCN(CC1)C2 CC1CN(C(c2nn[nH]c2CC(F)(F)F)=O)CC1CNC(=O)C(=O)NCC(F)F C(=O)(C1CCCc2nc[nH]c21)N1C(C)CC(NC(C(CC)O)=O)C1 CCC(C)(CC)C(=O)NCC(c1ccccc1)N(C)C(c1n[nH]c2c1COC2)=O c1(C(=O)NC(C(C)NC(c2ccc(C)cc2O)=O)C)ccc2ncccc2n1 C1(C(N2CCC(NC(c3c(CC)oc(C)c3)=O)C2C2CC2)=O)CCCC(F)(F)CC1 N1(C(C2C(C)OC(=O)N2)=O)CC2C3CCC(C2C1)N(C(=O)C(F)=CC1CC1)C3 c1(C(C)NCC(=O)NC(CC)C)ccc(C)nc1 c1(C(N2CCN(CCN(C(=O)CC3CCOC3)C)CC2)=O)cc2[nH]ccc2s1 c1(C(N(C(C(N2C(CNC(C)=O)CCC2)=O)(C)C2CC2)C)=O)oc(C)cc1C C1(CNC(c2c(C)ncs2)=O)CCCCCN1C(c1ncn(C(C)(C)C)n1)=O C(=O)(C1Cc2ccccc21)N1CCN(C(c2c(F)ccc(OC)c2)=O)C2C1CC2 c1(C(N(C)CCNC(C2(C3CC3)CCC2)=O)=O)oc2ccccc2c1Cl C1(C2C(NC=O)C2)CCCN1C(=O)Cn1cnnn1.C(C(=O)NC)NC(=O)C1CC1 C1(NC(c2ccc(C(C)C)s2)=O)C2CCC1N(C(c1nc(Cl)cs1)=O)C2 N1(C(CC(CC)OC)=O)C2CCC1CC(N(C(=O)CCCC1CCCO1)C)C2 c1(OC)cc(F)c(NC(=O)CNC2CC3CN(c4nccnc4C#N)CC23)cn1 c1(C(=O)NS(Cc2ccc(OC)cc2)(=O)=O)cnc(Cl)c(Cl)c1 N1(C(CCCOC(C)C)=O)CCCC2(C1)CN(C(C1(C)CCN(C)C1=O)=O)CCO2 c1(C(N2CC3CCC2C(O)C3)C(=O)NCCCC)cc2ccnc(Cl)c2o1 C1(C2CCCN(C(c3cnc(Cl)c(Cl)c3)=O)C2)(C(=O)OC)CC1.C1C(CO)C1 Cn1nc(Br)c2ccc(COC(=O)CNC(=O)CNC3CCCCNC3)cc12 N1(CCC)CCCC1C(=O)NC1CC(O)C1CC(=O)NCCN1CC2CC2C1 C(CC(C)(C)C(=O)N1CCCC(CN(C)C(C2CCS(=O)(=O)N2C)=O)C1)OC c1(CCC(=O)NC2(CNC(COC(C)=O)=O)CC2)cccc(F)c1Cl C1(C(=O)NCC(C(=O)OCC)C)CN(C(c2cccc(C#N)c2)=O)CC1(F)F C12(NC(Cc3c(C)cccc3)=O)CCCC1N(C(=O)C=Cc1c[nH]cn1)CCC2 c1(OCC(=O)N(CC(C)NC(c2c(CC)c[nH]n2)=O)C)cccc(C(C)C)c1 C(N=c1[nH]c(=NCC(C)CN(C)C)[nH]c2c1COC2)c1cccc(COC)c1 C(N=c1[nH]c(=NCC2CC23CC3)[nH]c2c1CCC2)c1ncc(CC)s1 Nc1nc(Cl)ccc1C(N1CCOC(CNC(c2cc(C3CCC3)on2)=O)C1)=O c1(C(N2CC3(CC(CNC(C=C)=O)C3)C2)=O)ccc2c(c1)CCCN2 c1(C(=O)NC2COCCN(C(C(C)OC)=O)C2)nc2c(cc1Cl)OCCO2 c1(C(=O)NCCCCNC(C(C(=O)OC)(C)C)=O)cccc2c1OCCO2 C(=O)(C1=CCCOCC1)N1CCC(CNC(c2c(C)nc(C)s2)=O)C1c1ccco1 Cc1nnc2ccc(-c3cccc4[nH]c(C(N5CC(F)CC5C#N)=O)cc34)cn12 C(=O)(CCCCC(C)(C)C)NC(C(CO)NC(c1c(O)ccc(OC)c1)=O)C c1(C(=O)NCC2CN(C(C(CCC#C)O)=O)C2)cc2c(C)cc(OC)cc2[nH]1 C#Cc1ccc(C(=O)NC(CNC(C2(C#N)CC3(CC3)C2)=O)CC)cn1 C1(CN(C(C=CS(C)=O)=O)C2CC2)CCCN(C(=O)CCC(=O)c2cccs2)CC1 C(=O)(C(C)(C)CC(F)F)NCC1(C)C(C)CN(C(c2[nH]cc(CC)c2)=O)C1 C#CCC(C)(C)CNC(C12CC1CN(C(C1CC(N(C)C)C1)=O)C2)=O C1(CNC(c2ccc(C)nn2)=O)CC2(CCC2)CN1C(=O)C(=C1CCCCC1)F C1(C(N(CCCNC(=O)CC2COCCO2)C)=O)CCC(c2ccccc2)CC1 C(CC(CC)C(=O)NCCOCC(=O)N(C)CC1(C#N)CCC1)=CC C1(CC)CCN(C(=O)C(=O)Nc2cccc(OCc3cccnc3C)c2)CC1F c1ccc(N2CCCC(O)C2)cc1.CC(CC(=O)NCC1(NC=O)CC1)N(C)C c1(OCC)ccc(Cl)nc1C(=O)NC1CC1NC(=O)CC1CC=CC1 N1(C(C2(C(C)NC(c3cc(C#N)cn3C)=O)CC2)=O)CCCC2OCCC12 C(=O)(C(C)S(C)(=O)=O)N1CCN(CC(C)(C)NC(c2cccc(CC)n2)=O)CC1 C1(C2CCCC2)(C(=O)NCC2CCCN(C(C(C)NC(CC)=O)=O)C2)CCC1 N1(C(C2(F)CC2c2ccccc2)=O)CCC2CN(c3ncncc3I)CC2C1 C(=O)(Nn1cnnc1)c1cc(CCNC(c2ccn(CCC)n2)=O)on1 C#CCC(CC(=O)N(C)Cc1cccc(F)c1)NC(=O)C(C)C(C)C c1(C=O)cc(C)cc(N)c1.C(CC(O)C(=O)NCC1CCN1C(=O)CCC1CC1)SC c1(C(=O)OC)cc2c(s1)CN(CCC(C)P(C)(C)=O)CC2 c1(C(N2CCC(NC(c3cnc(C)o3)=O)CC2C)=O)cccc([N+](=O)[O-])c1N c1(C(N2CC(CC)C(NC(=O)C(C)(C)OC)CC2)=O)cc(F)c(Cl)cc1Cl N1(C(c2cc(CC)[nH]n2)=O)CCN(C(c2oc(C(C)C)nc2C)=O)CCC1C C=CC(C)(CC)C(=O)NCC(C)NC(=O)Cc1n[nH]c(=N)s1 C1(CC=C)(NC(=O)CCC=CBr)CCCN(C(c2ccccn2)=O)C1 C(C)(C(=O)N1CC(CCCCNC(=O)CCC2CC(C)C2)C1)N(C(C)=O)C S(=O)(=O)(c1ccc(-c2nc(-c3ccco3)nn2-c2cccc(F)c2)o1)N(C)C CS(=O)(=O)c1cccnc1NC1CCN(Cc2ccccc2)C1=O N1(Cc2oc3ccc(C(=O)OC)cc3n2)CCC2(CC1)CC(C(=O)O)=NO2 C1(C2CC2)(CNC(C=CC=CCC)=O)CCN(C(=O)C2=CCCCO2)C1 N1(Cc2c(C)ncs2)CC(C(=O)NCCC2NC(=O)NC2=O)CC(F)C1 CC(C)CC(C)(c1nnnn1C1(C)CC1)NCC(=Cc1cccnc1)F Cc1cn2cc(CC(N3CCC(O)(C(C)CNC(=O)C=C(Cl)Cl)C3)=O)nc2s1 CN1CCCC1C(=O)NCCC1CCCN1C(=O)Cc1cc[nH]c1 N1(C(C2C(C)CC2)=O)C2COCC1CC(NC(=O)CCc1ccccc1F)C2 c1(OCCC(=O)OC)cccc(NC(C)CC=C(C)C)c1 c1(C(N2CCCC(NC(C(C#C)(C)C)=O)C2)=O)ccc2c(=O)cc[nH]c2c1 c1(C(N2CCCC(N(C(C(C3CC3)OCC)=O)C)CC2)=O)ccc2c(c1)OCO2 CP(C)(=O)CC(=O)NCC1CN(C(=O)CCc2cncs2)C1 C(=O)(CN1C(=O)Cc2ccccc21)N1CC=CC(NC(C2CCC(F)C2)=O)C1 C1(CNC(C2CC(C#C)(O)C2)=O)C(C2CC2)CCN1C(=O)C1=CCCS1 C1(C(=O)NC(CN(C)C)(C)C)CCC2(CC2)N1C(c1cnccn1)=O N1(C(=O)N(CCCCCC)n2cc(C)cn2)CCOC(CC(F)(F)F)C1 C12(C(=O)NC3(c4onc(C)n4)CC3)CC(CO1)N(C(=O)CC1(CO)CC1)C2 N1(C(CCN(C(C(C)N2CCCC2)=O)C2CC2)=O)CC2(CCC(C)OC2)C1 CCCC(C(=O)NCCC1CCCN1C(c1snnc1C)=O)c1ccccc1 S(=O)(=O)(c1cccnc1NC1CCCC(P(C)(C)=O)C1)NCC(C)(C)COC(F)F C(=O)(C(C)(C)CC(F)(F)F)N1CCCC(CNC(C2N(C(C)C)CCCC2)=O)C1 c1(NC(=O)COc2ccsn2)ccc(CN(CC(=O)NCCOC)C)cc1 C1(CCC(=O)N(CC(=O)OC)CC=C)CCCN(C(=O)CC2(O)CCC2)C1.C(C)(=O)O C(=O)(CCC(=O)N1CCCC(NCCc2cn(Cc3ncon3)nn2)C1)N(C)C C=CC1(O)CN(C(c2n[nH]cc2CNC(=O)C(CO)OC)=O)C1 C(=O)(C(C)(C)CCNC(=O)C(F)C(C)(C)O)NCc1cc(C(C)C)n[nH]1 c1(C(=O)NCc2c(C(=O)OCC(=O)Cn3cncn3)cccn2)cc(F)cc(F)c1 Cc1oncc1C(=O)NC1CC(N(C(=O)Cn2ccc(-c3ccccc3)n2)C)C1 CCC(C)(CNC(=O)C#CC1(C(=O)OC)CCC1)C(=O)N(C)C(C)CC C(=O)(C1=CSCCO1)NC1C(OC)CN(C(c2ccc(OCC3CC3)cc2)=O)C1 c1(C(N(CCNC(C2(CC(C)C)CC2)=O)C(C)C)=O)cc2ccc(Cl)cc2o1 C=CC(C)(O)CC(=O)N1CCN(C(=O)CCc2ccc(F)c(F)c2)CC1CO N1(C(C2(Cn3ncc(C#N)c3)CC2)=O)CC(C2CN(C(C3C4CCCC34)=O)C2)C1 C1(NC(C2CCC(C)(C)OC2)=O)CCN(C(=O)CS(=O)(=O)NC2CC2)CC(O)C1 N1(C(C(C)=CC)=O)CCN(C(=O)COc2ccc(C)cc2)C(CCOC)C1 C1(NC(C=C(CC)C)=O)CC2CC1N(C(c1ccc(N(C)C)cc1)=O)C2 N1(C(C(C=C)O)=O)CCC(C2CC2NC(c2ccccc2CO)=O)CC1 c1(C(=O)NCCN(C(C2C(CCC)CCCC2)=O)C(C)C)ccncc1N=[N+]=[N-] CC(O)C(F)(F)C(=O)NCCC1CCCN1C(c1ns[nH]c1=O)=O c1(N2CCC(C)CC23CCC3)nc(N(CC(=O)NC2CC2)C)nc2cc[nH]c12 C1(C(=O)NCC(CCC)C)CN(C(=O)C(C)N2CC(C)C2)CC1(C)C C(=O)(C(C1=CCCCC1)N1CCC(F)(F)C(F)C1)Nc1cccc(OC)c1 CC(=O)CCCC(C)C(=O)N1CCC(C(=O)NCC2CC(C)C2)C(O)C1 C12(CSC)CC(CNC(CCNC(C(=O)C(C)NC(c3ccco3)=O)=O)=O)(CO1)C2 N1(C(Cc2ccc(OC)nc2)=O)CC2CC(NC(=O)C3=NOCC3)C2C1 c1(C(=O)NC2CC(NC(C3(C#N)CC(C)C3)=O)C2)nccc2ccn(C)c12 Cc1ccc(CC(=O)NC2(C)CCCN(C(=O)CC(C)CF)C2)c(Cl)c1 c1(OC)n[nH]cc1C(=O)NC1(C2CCCN2C(C2CCCN2C(C)=O)=O)CC1 CC(C)(CC#N)C(=O)NC1CC2(C1)CC(C(=O)NCCc1cnco1)C2 N1(C(C(CSC)C)=O)CCCC2(CNC(c3oc(C)nc3C)=O)CCCCC12 CCCCC(C(=O)NC1(C)CN(C(=O)CCN2CCOCC2)C1)N1CCCCC1 C1(CNC(c2cncc(Cl)c2)=O)(CO)CCCN(C(c2cncs2)=O)C1 c1(C(N(C)CC2(O)CN(C(c3n[nH]cc3Cl)=O)C2)=O)ccc2c[nH]nc2n1 N1(C(C)C(N2CCCCC2C(C)(C)CNC(=O)C=C2CC2)=O)CCP(C)(=O)CC1 c1(C(=O)OC(C)(C)C)ccc(C(=O)N(CCCN(C)C)C)o1.C12CC(C1)C(=O)N2 c1(NCC)ccc(Cl)cc1C(=O)N(CC(C)CNC(=O)C=Cc1cc[nH]n1)C CCC(F)(F)CN(C)C(C1CCC(CNC(=O)COc2ccn(C)n2)C1)=O C(=O)(C(CNC(C1(C)CCCC1)=O)C(C)C)NC1CC(C=C)C1 C1(O)(Cn2cc(CCN(CC)CC)nn2)CCCN(C(c2ccon2)=O)C1 c1(C(=O)NC2CN(C(C3CC(OC)C3)=O)C(C)(C)C2)c(F)ccc(Br)c1F C1(CC(NOCC=C)=O)C2CCC(C2)N1C(C1CC=CC1)=O.c1ccccn1 C(=O)(CCCC(=C)C)N(C1CCN(C(c2cccc(CCC)c2)=O)CC1)CC#C C1(C(=O)OC(C)(C)C)CN(C(C(C(C)C)N(S(C)(=O)=O)C(C)C)=O)CCC1(C)C C#Cc1ccc(C(=O)NCC2CCCCCN2C(=O)CN2CCCC2=O)cc1 C1(NC(C2CCC(C)(C)OC2)=O)CCC2CC1CN2C(c1cc(N)ccc1O)=O c1(COC(C2CC(C)(C(=O)OC)C2)=O)ccc(C)nc1 N1(C(c2cc(C)ns2)=O)CCC(CO)(CNC(=O)CCSC(F)(F)F)C1 N1(CCN(C)C(=O)Nc2ccc(C(F)(F)F)[nH]2)CCN(c2ccccc2F)CC1 CS(=O)(=O)C1(C(=O)NCC2CC(O)(CNC(=O)Cc3cscn3)C2)CCCC1 c1(C(=O)NCC2(NC(CNC(CC)=O)=O)CCCCCC2)cnc2cc(C)nn2c1 C(=O)(CCCC(=O)NC1CC1)N1C(CNC(c2cc(SC)oc2C)=O)CCCC1 C1(C(NC(c2ccncc2)=O)C2CC2)COCCN(C(N2CCCC2)=O)C1 c1(C(N(CC(=O)NC(C)CC2CCOC2)C)=O)cccc2[nH]ccc12 c1(CC(=O)OC)ccc(OC(=O)C(c2cc(Cl)ccc2F)C)c(Cl)c1 c1(C(=O)NCC(C(C)C)NC(=O)CC2CC2C2CC2)cc2cccn2c(O)n1 C1(CN(C(=O)CCc2cncs2)C)C2CN(C(=O)Cn3cc(Cl)cn3)CC12 N1(C(COCC#C)=O)CCC(C(=O)NCCCC(C)O)(C(C)C)C1 CCCCC(C(=O)N1CCC(NC(c2ccnc(Cl)c2)=O)C1C)N(C)C c1(NC(COC(C)C)C)nccc(N2CCC(C)(Cc3ccccc3)C2)n1 N1(c2cc(SC)ncn2)CCC2(CCCC2C(N2CCc3cccnc3C2)=O)C1 Cc1ncsc1CC(=O)NC1(C(N2CCC2CC2CC2)=O)CC(F)C1 c1(C(=O)NCc2ccccc2SC(F)(F)F)ccc(I)cc1Cl.C12CN(C1)C(=O)N2 C#Cc1ccc(C(N2CCOCC2CC(=O)NCCC2COC(C)(C)C2)=O)cn1 C1(CC(C)NC(=O)C(C)(C)C(C)O)CC2CCC(C1)N2C(=O)C1=CS(=O)CCC1 C(=O)(N=c1[nH][nH]c2c1CCCC2)C1(C)CN(Cc2cc(F)cc(C)c2O)C1 N1(CC(=O)NC(C(=O)NCCC2ON=C(C)C2)C2CC2)CCCCCC1 C1(C(N(CCC#C)CCOC)=O)CC(N=[N+]=[N-])CN1C(=O)C(CC)C1CC1 c1(OC)cc(C(=O)N(CC(C)NC(=O)CC2CCCCC2O)C)ccc1O CCC(F)(F)C(C)(C)C(=O)NC1(CCNC(c2cncc3nc[nH]c23)=O)CC1 C1(NC(c2c(C)cno2)=O)CCC2CN(c3ncncc3Cl)CC2C1 C12(NC(c3ccc(C(F)(F)F)nc3)=O)CCC(CN(C(C3CC=CCC3)=O)C1)C2 n1(C(C(=O)NC(C)CCF)C)cc(C(c2ccccc2)O)nn1 c1(C(=O)NCC2CN(C(=O)CC3OCCO3)CCO2)cc2[nH]ccc2s1 N1(C(c2c(CC)scn2)=O)CC(OC)CC(NC(=O)C(n2nc(C)cc2C)C)C1 c1(C(N(C)Cc2ccc(C(F)F)cc2Cl)=O)ncc2c(ncn2C)n1 C1(C(N)=O)(CNC(=O)CSC2CC2)CN(C(=O)CCc2cscn2)C1 CN(CC(=O)C1COC(C)(C)C1)N1CCC(C#N)CC1 C12(C(N(CCN(C(C(C)OC(C)(C)C)=O)C)C(C)C)=O)CC1COC2(C)C C1(O)(C(CNC(C(C)=C2CCCC2)=O)C)CCN(C(c2sccc2Cl)=O)C1 N1(C(C(C(C)(C)O)F)=O)CCC2CN(C(c3ccc4nncn4c3)=O)CC2C1 c1(OC(C)C)ccc(CN(C)C(C2CCN(CC3CCOC3)C2)=O)cc1 C1(NC(C2CCC(C)C2)=O)(CNC(C2CC(=O)CCO2)=O)CCOCC1 C1(NC(C(C)(C)C2CC2)=O)C2CC3C1C3C2C(=O)NCC1CN(CC2CC2)CCO1 O=C1C(Cc2cc[nH]n2)SCCN1.c1(CNC(=O)C(O)C2CCC2)cccnc1 N1(CCCOC(C)(C)C)CCC(CNS(=O)(=O)C(F)F)CC1 C1(CCC)CN(C(=O)C(F)=C(C)C)CCN1C(c1ccc(F)c(SC)c1)=O C(CC(C)(C)C(=O)NCCCN(C1CC1)Cc1ccco1)OC C1N=C2NC(=Nc3ccsc32)N2CC1C1(CC1)C2.CN1CCn2[nH]c(=N)nc2C1=O C1(F)(CNC(C2CNC(=O)N2)=O)CCCN(C(C2CC(=O)N(C3CC3)C2)=O)C1 N1(C(C2(Cl)C(C)(C)C2)=O)CC2C3CCC(C2C1)N(C(C1CCC2CC12)=O)C3 N1(C(C)=O)CC(O)CC1C(N1CC=CC1CNC(c1cnc(N(C)C)o1)=O)=O Cc1cc(C(F)F)cc(C(C(=O)NC(C)C(=O)NC)N(C)CCc2cncnc2)c1 C(c1ccccc1)=CC(CO)N(C(C1(CNCc2cccnc2)CC1)=O)C1CC1 C1(C(=O)NCC(CO)NC(C(Br)=C(C)C)=O)CNC(=O)CC1C CC1(C)COCCC1CC(N1CCN(C(C23CCCC2C3)=O)CC1)=O C(=O)(CCS(=O)(=O)c1ccc(OC)cc1)NCCCN(CCOC)C CC1CCN(C(=O)CCS(C)=O)C(C)C1NC(=O)CCCC1CC1C Cc1[nH]nc2c1CN(C(=O)CC1COCCN1Cc1cccc(F)c1Cl)CC2 c1(NC)cnncc1C(N1CC=CC1CNC(C1CC2(CCC2)C1)=O)=O C1(CC)CN(C(c2cc(C)nn2C)=O)CCC1Nc1nccc(C#N)n1 CCC1=C(C(=O)NCCCCC(=O)NCC(CC)n2cccn2)CCCO1 C1(CNC(C2C(COC)C2)=O)(CNC(=O)CSCC(N)=O)CCCO1 C1(C(=O)NC(C(=O)OC)C(C)O)C2CCCC2CN1C(=O)C(O)CN(C)C N1(C(COC2CCN(C)CC2)=O)CC2CC3CC2C1C3NC(C1CC1F)=O C1(C(N2C(CCNC(C(C)OCCOCC)=O)COCC2)=O)CC(C2CC2)=NO1 c1(C(N(C2CC(NC(=O)C(c3cnn(C)c3)O)C2)C)=O)cnn(C)c1C1CC1 CCC(C)C(C(=O)N(C)Cc1ccco1)N(C)C(c1ccncc1O)=O C12(C(N3C4(C(NOCCCC)=O)CC(C3)C4)=O)CCN(CC1)CC2 N1(C(CSCC=C)=O)CCC(C)(C)C(CNC(c2n[nH]c(C)c2C(F)(F)F)=O)C1 CCCCN=C(NCCN(C1CC1)Cc1cc(Cl)ccc1C)NC(C)C1CC1 Cc1cc(CNC2CC(Nc3ncnc4c3CCC4)C2)cc(C)c1O C12(CC(=O)NC34CC(CNC(C(C)OC)=O)(C3)C4)COC(C)(C1)C2 C1(NC(C(C=C)(C)O)=O)CC2CN(C(=O)C(CCC)NC(N)=O)CC12 N1(C(CCCCSC)=O)CCC2CN(C(C34CCCC3C4(F)F)=O)CC2C1 CN1CCCCC1C(c1cccs1)NC(C1CC2CC2N1C(c1cccnn1)=O)=O C(=O)(CCCCCC(C)(C)C)NCC1C(NC(C=CC(CC)C)=O)C1 N1(C(c2cc(OC)n[nH]2)=O)CCC2(CCCN(C(=O)CCC(F)(F)F)C2)C1 C1(c2n(CC)nnn2)(NCC2CC2(C)C)CC(C)OC(C)C1 C=C=CCCC(=O)NC1(C(N2CCN(C(c3c(C)cnn3C)=O)CC2)=O)CC1 C(C(C)C(C)C(=O)N(CCN(C)C(C1CC2(C1)CC(F)C2)=O)C(C)C)OC N=c1[nH]cncc1C(=O)NCCOC1CCN(C(c2cnc(C(F)F)s2)=O)C1 C1(NC(c2nc(Cl)c(Cl)s2)=O)CCSC12CN(c1ccc([N+](=O)[O-])cn1)C2 CC(C)(CC(=O)NC(C1CCN(CCCc2ccccc2)C1)=O)C(F)F O=C(CC(C(F)F)n1cc(Br)cn1)Nc1ncc(Cc2ccccn2)cc1F C12(CNC(CCC#C)=O)CC(CO1)N(C(C1CC1Br)=O)C2 c1(C(=O)NCC2N(C(C(CC)C(C)C)=O)CCCCC2)ccc2nnnn2c1 Cc1ccc(C(C)C)c(NC(C2CC2C(=O)NCc2ccncc2Cl)=O)c1 C1(C)(CNC(C(CCOCC)NC(c2cc(Cl)ns2)=O)=O)CC2CCC1C2 C(CN=c1[nH]cnc(Cl)c1C(C)=O)NC(c1cccc(CN(C)CC)c1)=O C(CCN(C)C(c1ccccc1SC1CC1)=O)(C(C)(C)C)NC(CCC#C)=O c1(CCCNC(COC(CNC(C2C(CC(C)C)C2)=O)(C)C)=O)nccn1C C(CCO)(C(F)F)N(C(C1(CNC(C2CCO2)=O)CC(=C)C1)=O)C c1(C(N2C(CNC(CC(C)(C)F)=O)CC(O)C2)=O)ccnc2ccsc12 c1(C(=O)NC(CCC=C)C)oc(CNC(=O)C#CC(C)C)cc1C C1(C=C)(CC(=O)NC(CC=C)CNC(=O)CNC(C2CCCC2)=O)CCOCC1 C(=O)(C(CCCc1ccccc1)N(CCC)CCc1ccccc1)NCCC C1(CCC)(NC(c2cnn(C)c2Cl)=O)CCN(C(=O)CC2CCOC2)CC1 C=CC(C)(O)C(=O)N1CCC(O)(CNC(=O)COc2ccc(SC)cc2)C1 N1(C(c2c(CC)nnc(C)c2)=O)CC2(C1)SCCC2NC(c1cc(C)ncn1)=O C1(NC(C2C(NC)CCC2)=O)CCC(NC(=O)CCOCCCOC)CC1 C12(C(=O)NCC3(F)CCN(C(C(CC=C)(C)C)=O)C3)CCC(N=[N+]=[N-])C1C2 N1(C(CC2C=NN(C)C2=O)=O)CCN(C(C2CC(=C3CCC3)C2)=O)CC(C)(C)C1 Cc1ccc(C(=O)NCC2(C)CCN(C(c3cc(C#N)on3)=O)CC2)c(F)c1Cl Cc1nnc2n1CCC(NC(CN(c1nnnn1CC(C)C)C)=O)C2 C(C(C)(C)C(=O)OC)(c1n(C(CC)(C)C)nnn1)NCC1CCC(=O)N1 N1(C(C(C)NC(CC)(C)C)=O)CCC(C2CCN(C(C3(COC)CC3)=O)CC2)C1 N1(c2cc(NCC3=CCCOC3)nc(COC(C)C)n2)CCC2(CCOC2)C1 C12(CNC(C(C(C)C)OC)=O)CCC(C1)N(C(=O)C=Cc1ccc(C)s1)C2 C1(CN(C(=O)CCc2ccccc2)CC)CCCN1C(=O)Cc1sccc1Cl C#CC1(C(=O)NC2CCC(CCC(=O)NCCCCCCOC)C2)CCCC1 N1(C(c2c(OC)cccn2)=O)C2CCC1C1CC1(NC(c1cncc(Cl)c1)=O)C2 C12CCC(=O)N(C1)C2.c1(SCC(=O)N(C2CCNOC2)C)ccc(Cl)cc1 C1(CC)CN(C(c2cc(C(F)F)nn2C)=O)CCC1NC(C1CNC(=O)N1C)=O CC(C(=O)NCCC1(C(=O)NC(C(N)=O)C(C)(C)C)CCC1)C(C)(C)C Cc1ccc(Cl)c(F)c1C(N1CCC(O)(CCNC(=O)CC(C)N(C)C)C1)=O c1(CC)nn[nH]c1C(=O)NCC1CC1NC(=O)Cc1ccnn1C N1(C(c2ncccn2)CC)CCC2(CC1)OCCC2NC(=O)C#CC(C)C C1(CC=C)CCCC1C(=O)NC1(CO)CN(C(=O)C(C)(C)N(S(C)(=O)=O)C)C1 C=CCC(C)(C)C(=O)NCCOCCNC(c1cc(OCC)cn1C)=O C1(C(F)F)(CNC(C=COCC)=O)CCN(C(=O)CN2CSCCSC2)C1 N1(C(C(C)c2cncs2)=O)CCN(CCSc2ccccc2O)CC1 c1(OC)ccncc1C(N1CC(N(n2ccc(C(F)(F)F)n2)C)C1)=O C1(C2(NC(COC(CC)C)=O)CC2)CCCN1C(=O)CC1CCOC1=O N1(C(C(=O)NC)=O)CCCC1CNC(=O)Cn1ccnc1C C1(C)(C(=O)NCCOCC(=C)C)CCCN(C(C2(OC)CCCOC2)=O)C1 c1(OC)ccc(C(=O)NC2CCCC2NC(c2n[nH]cc2C)=O)cc1 N1(CCC(N2CCCC(CNS(C)(=O)=O)C2)=O)Cc2ccccc2C1 O(NC(=O)C(C)(CO)NC(=O)CN1CCSCC1)CCC N1(C(c2ccc(C)c(F)c2)=O)CCC2(CCCN2Cc2ccc(F)c(Br)c2)CC1 CCC(C(=O)N(C1(C(=O)NC(c2nc[nH]n2)C)CCC1)C1CC1)OC c1(C(=O)OC(c2ncc(C)o2)C)[nH]c2ccc(Br)cc2c1F C1(C(=O)NCC2N(C(C(C(C)C)c3ccncc3)=O)CC2)CC2(CCC2)CO1 c1(C(=O)NC(C(=O)NCC(C2CC2)SC)CCC2CC2)cccc(C)c1O CC1CC2(CCO1)CC2C(N1CC(CNC(c2cccc(N)c2O)=O)CC1C)=O n1(CC(=O)NCC(CNC(C2CC(F)(CO)C2)=O)OC)ncccc1=O N1(C(c2cn(CCC)nc2)=O)CCN(C(=O)C(C)COC)C(CC(F)F)C1 c1(C(N(C2CCC(NC(=O)C=CC3CCC3)C2)C)=O)cnc(C(F)(F)F)c(F)c1 c1(C(=O)NCC(C(C)C)NC(=O)C=CSc2nc[nH]n2)ccn2ccnc2n1 C(CC(N)=O)(C(=O)NCc1ccncc1C)NC(CC1CC(=C)C1)=O Cc1ccc(C)c(NC(=O)CC2CN(C(=O)CCCOCCOC)CCC2C)c1 [N-]=[N+]=NCCCC(O)CC(=O)NCCCCC(=O)Nc1ccccc1 CCC(C)C(C(=O)NC1(C)CCSC1)NC(=O)C(=O)NCC N1(C(c2c(CC)onc2)=O)CCC(CC)C1CNC(=O)CSc1n[nH]c(O)n1 C(C)(C)(CCC(=O)N1CCC(C)(CNC(=O)Cn2cccn2)CC1)OC c1(NC(c2cn(C(C)C)nc2)C)ccc(S(=O)(=O)N2CC=C(Br)CC2)c(Br)c1 c1(-c2nc(C(CN3CC(C)O3)OC(F)F)on2)cccn2nnnc12 c1(C(=O)OCC)cnc(SC)nc1N1CCC(C(c2ccc(C)c(O)c2)=O)CC1 CC(C(F)(F)C(F)(F)F)NC(C1CCCC(O)C1)=O.C(C)(C)(C)OC(N(C1CC1)C)=O c1(CC)nc(=N)[nH]cc1C(=O)NCC(C1CC1)N(C)C(c1nc(O)sc1C)=O N1(C(CCCCC)=O)CCc2nc[nH]c2C12CCN(CC(C)C)C2 Cc1cc(F)cc(C)c1C(=O)N(C1CCN(C(=O)CCC(C)N(C)C)C1)C N1(C(c2ccc(CC)s2)=O)CCCC2(CCC(NC(C3CS(=O)(=O)C3)=O)C2)C1 C(CCCCCC(=O)NC1CC=C(C)CC1)NC(c1nc(CC)oc1C)=O C(=O)(C=CSc1cccs1)NCC1N(C(C=CCCC)=O)CC1 N1(C(CN(C(C)(CC2CC2)C2CC2)C)=O)CC=CC1C(=O)Nc1ccncc1 CCCCCCCOC(=O)C(c1ccc(O)cc1)OCC(F)(F)F C1(C(=O)CNCC(N2CCCCC2)=O)CN(C(C2C=CCCC2)=O)CCO1 N1(C(C(C)(C)OC(C)C)=O)CCC(n2cccn2)(NC(C2CCCO2)=O)CC1 c1(CC(=O)NCC2CCCN(C(C(C=CC)O)=O)C2)cc(Cl)ccc1Cl Cc1cc(C#N)cnc1CNC(C1CC=CCC1)C(N1CCC([N+](=O)[O-])CC1)=O c1(CC(N2CCC(CN(C(=O)C(CO)c3ccccc3)C)C2)=O)cccc(O)c1 Cc1cc(NC(=O)Nc2cc(C#N)nc(C3CC3)n2)cc(C)c1C c1(C(N2CCCC(NC(c3cc(OC)ns3)=O)C2C)=O)c(C)ccc(C)c1N O=C(CCCCCc1cccs1)NCC(CO)NC(=O)CCN1CCCS1(=O)=O C1(NC(C2C(C(C)C)(CC)C2)=O)C2CC(NC(=O)CCN3CCCCC3C)CC12 c1(C(N(CC(C)NC(C(COC)OC)=O)C)=O)cnn(C)c1CC(C)C c1(CC)cccc(C(N2CCC(CNC(=O)C(OC)OC)C2(C)C)=O)c1O C1(CNC(C2CCCC23CC3)=O)CC2CCC(C1)N2C(=O)Cn1ncccc1=O c1(OCC(=O)N(C2CCN(C(=O)COC3CCOCC3)C2)C)ccc(Br)cn1 C1(NC(COC(CNC(C(C)NC=O)=O)(C)C)=O)CCCCC1O CC(CC#N)C(=O)NNC(=O)C(C)(C)CCCCNC(=O)COCC1CCC1 Cc1ccc(C(=O)N(C)CC2CCCN(C(=O)CN(C)C3CC3)C2)cc1F C(CCC(C)(C)C(=O)N1CCC(C2CC2)CC1)NC(Cc1c(C)nccc1)=O Cc1ccc(C(=O)NC(C2CCCN(C(c3cc(Cl)sc3Cl)=O)C2)C)nc1C c1(C(=O)NCC2CCCN2C(=O)CCc2cnoc2)cc(Br)c(Cl)s1 c1(C(C)NC(C2(CSC)CCC2)=O)nccc(C)n1.C12(CC1)CC(=O)NC2 CCCCCCC(C)NC(=O)C(CC(F)F)N(C(=O)CN(C)CCC)C Cc1c(Br)cnc(NC(=O)Cc2ccc(NCc3cccnc3Cl)[nH]2)c1[N+](=O)[O-] C1(SC)CN(C(C2CC2c2ccncc2Cl)=O)CC1NC(c1cc(F)n[nH]1)=O N1(C(C(C)=C2CCCC2)=O)CCC(NC(=O)CCc2ccn(C)c2)CC1C N1(C(C(CC)OC)=O)CCCC1(C)C(=O)NC(CF)C(F)(F)F CCCCCCCC(=O)N(C)CC1CCCN1C(=O)C(S(C)(=O)=O)C1CC1 c1(CC)cccc(F)c1C(=O)NC1CCC1CNC(C1CCC1)=O S(=O)(=O)(c1cccnc1NCC1CC12CC2)NCCCS(C)=O c1(C(=O)NCCC(C(=O)Nc2cccc(CC)c2F)OC)cc2ccccc2[nH]1 C12(C(N3CCC(O)(CNC(C4CCCS4)=O)CC3)=O)CCC(C1)S(=O)(=O)CC2 c1(N2CCC(N(C)C(c3cn4c(n3)CCC4)=O)C2)ncnc2cccc(F)c12 CCC(C)(CCNC(=O)CN1CC(C)(C)C1)NC(c1ncccn1)=O C1(C(N)=O)CC2(CC(NC(=O)CC3CN(C(C4CCC4(C)C)=O)CCO3)C2)C1 C(=O)(N=c1[nH]n(C2CC2)cc1C#N)N1CCCC(N2C(C)COCC2)C1=O c1(NC(C(=C)CN(C)C)=O)c[nH]c2cc(Br)ccc12 C1(C(=O)NC2CC(N(C(CCCCC)=O)C)C2)CCC2(CCC2)OC1 C1(CC)C(NC(=O)C(C)Oc2cccc(F)c2)CCN1C(=O)CCOC1CCC1 c1(C(=O)Nc2n(CNC3C(C)(C)C3)ccc2)cccc(CO)c1 C1(C(=O)NCC(COCC)C)CC2C=CC1N(C(c1cnc(O)c(C)c1)=O)C2 N1(C(c2sc(C)c(O)n2)=O)CCC2CCN(C(=O)Cc3c(Cl)cnn3C)CC2C1 C=C(C)CCC1C(=O)N1.C1(C(=O)OC)(OC(C)(C)CC)CCNCC1 c1(C(=O)NC(c2ccc(-c3cccc(C(F)(F)F)c3)o2)C)ccsc1C#N N#Cc1ccc(CN2CCCCC2C(=O)NCC2CC2(F)F)o1 N1(C(CCOCCOC)=O)CC(C)N(C(=O)C(C)C(C)O)CC1C Cc1cc(C(=O)N(CCCCNC(C2C=CCC2)=O)C)c2ncccc2c1 c1(N(CC)CC)ncccc1S(=O)(=O)NCC(C)C.C1(N)CC2(C1)CC(F)(F)C2 N1(C(C(C)CF)=O)CC2CCN(C(c3ncccc3Cl)=O)CC(C2)C1 Cc1cc(F)ccc1CNC(C1(C)CCCC1(F)F)=O CC1CCOCCN1C(c1cnc(CNC(=O)C=Cc2ccsc2)nc1)=O C1(NC(c2coc(CO)c2)=O)CC(O)(CNC(c2cc(C3CC3)cs2)=O)C1 Cc1c(C(=O)NCC2CN(Cc3noc(C4CC4)n3)CCO2)sc2cc(F)ccc12 CC(CCCO)N=c1nc(N2CCN3CC(F)CC3C2)c2ncccc2[nH]1 C1(C(C)(C)C)CN(C(=O)C(C2CC(F)(F)C2)O)CCN1C(c1ccc(N)cn1)=O C=CCC(CC(F)F)C(=O)NC1CCC1CNC(c1cc(C)nn1CCC)=O N1(CC(C2CC2)OCC)CCCC(C)(CNC(c2cscc2C)=O)C1 N1(C(C2(CCNC(c3cn(CC)nn3)=O)CC2)=O)CC2(CC=CC2)C1 c1(C(=O)NCCCN(C(=O)C(O)C(C)(C)C)CC)ccc(OC(F)F)cc1F C1(NC(C(CC=C)NC(=O)OC(C)(C)C)=O)CCC12CN(C(=O)C1CC1)C2 C(=O)(C1=NNC(=O)C1)NC1CCC(CNC(C(Cc2c(C)cccc2)C)=O)CC1 c1(CC)nc(C)cc(=NCC2C3CN(C(c4cnn(CCO)c4C)=O)CC23)[nH]1 C(c1c[nH]c(=N)c(C)c1)=CC(=O)N(CCNC(C1(C(=O)OC)CC1C)=O)C c1(C(N2CC(C)(C)C(NC(=O)CC=C(Cl)Cl)CC2)=O)cc2cccc(Cl)c2[nH]1 C1(NC(CC2CCC(NC=O)CC2)=O)CC2CN(C(C3(C(F)F)CC3)=O)CC2C1 c1(SCC(=O)NCC2C(NC(c3c(C)cc(CC)o3)=O)CC2)cc(Cl)ccc1Cl C(=O)(CC(C)CN1CCCC1Cn1cc(-c2ccc(C(F)(F)F)s2)nn1)NC C1(CNC(c2cc(CC)on2)=O)CC2(CCOCC2)CN1C(C1CCNC1=O)=O N1(C(c2c(C)cco2)=O)CC2CCCC(N(C)C(c3cc[nH]c3C)=O)C2C1 N1(C(C2(CC#C)CC2)=O)CCC2(CC(NC(=O)C(c3ccc(Cl)c(F)c3)O)C2)C1 C1(NC(c2c(C)ncnc2)=O)CCCC12CN(C(=O)C(C)SC(F)(F)F)C2 C1(C)(CNC(C2C(CC)N(C(c3ncn(C(C)C)n3)=O)CC2)=O)CCC(=O)N1C N1(C(C(C)OCC=C)=O)CC(NC(c2csc(CCP(C)(C)=O)n2)=O)CC(F)C1 C1(C(C)C)CN(C(=O)CC(C2CC2)NC(c2cc(C)co2)=O)C1C(C)C c1(C(N2CC(COC)(NC(=O)Cn3nc(C)cc3C)C2)=O)cc2ccccn2c1 N1(C(CCC=C(C)C)=O)CC2(CCN(C(=O)Cn3ccc(C)n3)CC2)C1C(C)C C1(NC(CCC=C)=O)CCN(C(=O)C(C)Cc2cnn(C)c2)C12CCC2 N(S(=O)(=O)N1CCC(CC)CC1)C(C(CC=CC)C)=O C(C(C)(C)C(=O)N1CC2CC2(C(=O)NCC(O)(COC)CO)C1)OCC N1(C(c2oc(CC)c(C)c2)=O)CCOC2(C1)CN(C(C1COC(=O)N1)=O)C2 n1(CC)cc(NC(=O)C#CCNC(C2CC(=O)N2)=O)ccc1=O c1(NC(c2cc(CSC)no2)=O)ccc(F)c(O)c1.c12ccc(cn1)c(=O)[nH]2 N1(C(CCn2c(C)cc(C)n2)=O)CCC(NC(c2cc(Cl)on2)=O)C12CC2 C1(CC(=O)NCC(c2ccc(C(F)(F)F)cc2)NC(C(C)C)=O)CCS(=O)(=O)C1 Cc1cc(C)n(CCNC(=O)CC2CCOC2)n1.N12CC3C(C3C1)C2=O c1(C(N2CC(NC(CC3CC(=C)C3)=O)C(SC)C2)=O)c(C)cc(F)cc1Br N1(C(=O)C=CC2CCCO2)CCN(C(c2ccc(C(F)(F)F)[nH]2)=O)C2(CC2)C1 c1(C(=O)NC(CN(C(=O)CC2CCOC2)C)(C)C)cnc(S)nc1 C(CC1CC1)(CCCCCCCC)NC(C(C(=O)NCC(=C)C)C)=O c1(C(N2CCC(C)(CNC(c3cncc(Cl)c3Cl)=O)C2)=O)ccc(Cl)c(O)c1N c1(C(=O)NC(CN(C(C2(CC)CCCC2O)=O)C)(C)C)cc(C)cc(O)c1 Cc1cc(Cl)c(C(=O)NC2CCCN(C(=O)C(C)(C)C3CCOC3)CC2)cc1F C(=O)(CC(F)(F)C(C)C)N1CCC(NC(c2scc(C)c2)=O)C(C(C)C)C1 N1(C(CCC=C)=O)CC(C)CCC1CNC(c1ccc(C(F)(F)F)nc1N)=O CC1CN(C(c2c[nH]c(Br)c2)=O)CCC1NC(=O)COC1CC=CC1 Cc1ccc(C)c(C(N2CCN(C(=O)C(O)CCN(C)C)CC2CC2CC2)=O)n1 C1(NC(c2c(C)noc2)=O)C2CC(N(C(=O)C(C)c3ccsc3)C3CC3)CC12 CC1=NOC(=O)C1CCC(=O)NCCNC(c1cnc(C(C)(C)C)[nH]1)=O C1(C(N2CCC(CSC)C2)=O)CCCCN(C(c2c[nH]c(=N)o2)=O)C1 CC1CC(=O)NCCN1C(=O)CC(C)(C)N(C(=O)CCC1OCCO1)C Cc1cn2ccc(C(=O)NC3CC(F)CN(C(c4ccc(C)n4C)=O)C3)cc2n1 C(C(CC1CC1)C(=O)NOC1CCOCC1)NC(C1CCC(C)(C)C1)=O C1(CC)CCCC1C(=O)N(CCC(=O)NC(C)(CC)CC)CCO C1(C(F)(F)C(=O)NC(C)CNC(c2nnn(C)c2N)=O)(OC)CCCCC1 c1(C(N2CCC2C2CCCC2)C(=O)NCCCSC)nscc1C c1(C(=O)NCCOCCNC(C2(C)CC(C)OC(C)C2)=O)nc2ccccn2n1 c1(C(C)C(=O)NC2(CO)CCN(C(=O)C(=O)N(C)C)C2)cccc([N+](=O)[O-])c1 CC1=C(C(=O)NC2CCC(CNC(=O)CCC(C)OC(C)(C)C)CC2)CCC1 c1(C(=O)NCC2(O)CCN(C(C3(F)CCC3)=O)C2)nccc2c1NCCC2 C(=O)(C1=C(C)OCC1)NCC(CNC(C(CC)N1CCCC1=O)=O)CO c1(C(=O)NC2(C(=O)OC)CC(CO)C2)coc(CNC(C2CCC(=O)N2)=O)c1 C1(C)(C(N2CC(NC(Cc3ccc(C(C)C)cc3)=O)C(F)C2)=O)CCCS1(=O)=O c1(CS(C)(=O)=O)nnc(NC(C(=O)Cc2ccccc2)c2cccs2)s1 c1(CC2CC(N(C)C(=O)C3CC3)C2)ccccc1F.C1(=O)CCC2(CCC2)CO1 c1(C(=O)NC(C(=O)NC2CN(CCC)C2)CO)csc(C(C)OC)n1 N1(C(c2c(C)snc2)=O)CCc2ccccc2C1CNC(c1ncccc1F)=O CN1CCN(C)C(CNC(C2(NC(c3cnns3)=O)CC(CO)C2)=O)C1 C(=O)(CCCC(=O)NCC(O)CNCC(c1ccccc1F)OC)NC C1(NC(CCOC(C)C)=O)CC2CC(NC(=O)C(c3cccnc3)N(C)C)CC12 Cn1nc(O)cc1C(=O)NC(C)CCCCNC(=O)C(c1ccccc1)C1CC1 c1(N2CCC(CCOC)(NC(c3cc(Cl)on3)=O)C2)[nH]cnc2nc(Cl)cc1-2 N1(C(COCOC)=O)CCN(C(c2ccnc(C(C)(C)C)n2)=O)CC(C)(C)C1 Cc1cc(C#N)ccc1C(N1CC(C)N(C(c2nocc2C)=O)CC1C)=O C1(C(=O)NCc2c(C)nns2)CCC(C2CC2)N1C(c1cc(C(C)C)on1)=O C=CC(CCC)CC(=O)NC1CCCC12CN(C(c1c(C)cccc1O)=O)C2 C1(C(C)C)CCCC1C(=O)OC1CCC(OC(c2ccccc2)C)C1 N#Cc1cccc(C(N2CCC(C(=O)NCC3CC34CCOCC4)C2)=O)n1 N1(C(C(C(=O)NC(C)C)(C)C)=O)CCCC2(CC(NC(C3CC3CF)=O)C2)C1 N1(C(CC)=O)CC2(CC(C(N3CCC(O)CC34CC4)=O)CO2)C1 CC(CCc1cccs1)N=c1cc[nH]cc1S(=O)(=O)NCC1OCCCO1 N1(C(C(C)=C(C)C)=O)CCCC(F)(CNC(=O)CCCN=[N+]=[N-])CC1 N1(C(CC(C)(C)C#N)=O)CC2(C)CN(C(C3CCC3n3cccn3)=O)CC2(C)C1 C1(NC(C2C(C(=O)OC)C2)=O)CCCN(C(c2ncc(C)cc2F)=O)CC1 C1(C(NOCC2CC(=C)C2)=O)CC(NC(=O)CCCC#N)C1(C)C N1(C(CCCCCSC)=O)C2CCC1CN(C(c1cccnn1)=O)C2 N1(C(COCC(=C)C)=O)CCCC(N(C)C(c2cc(C(F)(F)F)n(C)n2)=O)CC1 c1(C(N2CC(NC(c3n[nH]c(C(F)(F)F)n3)=O)C2)=O)nc[nH]c2nccc1-2 c1(CN(CCNC(=O)C(Cc2cccc(Cl)c2)=NO)CC)ccc(F)c(F)c1 C=C(C)CC(C(=O)NCc1cnc(COC)o1)NC(C1CCCC1OC)=O C12(NC(CCCCSC)=O)COC(C1)C(NC(=O)COc1ccccc1C#N)C2 C(C(C)(C)CC(=O)NC(c1cncs1)CO)NC(C1(C)CC(C)C1)=O C(=O)(C(CNC(=O)C(=C1CCCCC1)F)C(C)(C)C)NCC(C(C)(C)C)OCC c1(C(N2CC(CC(C)NC(=O)C3=CCS(=O)(=O)C3)C2)=O)c[nH]c2nc(Cl)ccc12 C1(C(N2CCC(NC(c3ncc(CC)cn3)=O)C2C)=O)CC2COCC2C1 C=C(Br)CCC(=O)NCCC1(NC(c2ccc(CSC)o2)=O)CCCC1 C1(C(=O)NCCOCC)CCCN(C(=O)COCC(C)(C)C)CC1 CCC(N=c1[nH]c(=NCc2ccnc(C)n2)[nH]c2cc[nH]c12)C(C)C C1(NC(C(C=C)O)=O)CCCN(C(=O)CCC(=O)c2ccc(N)cc2)C1C Cc1[nH]c(C(F)(F)F)cc1C(=O)N(C(Cn1cncn1)CO)CC(F)F Cn1[nH]c(=NC(=O)c2c([N+](=O)[O-])ccc(-c3nn[nH]n3)c2Cl)c2c1CCOC2 C(=O)(CCNC(=O)C(C)N(C(=O)Cc1ccoc1)CCC)OCCC.C(C)=O C(=O)(C(CC(C)C)C(C)C)NC(C1CCN(C(C=CC(CC)=CC)=O)C1)(C)C N1(C(Cc2cc(C)nc(O)c2)=O)CCN(C(c2cc(CO)on2)=O)CC(C)C1 c1(C(=O)NC2CN(C(c3cc[nH]c3)=O)CC2F)cccc(C(F)(F)F)c1Cl N1(C(C(CSC)O)=O)CCC(C(N2CC(C#C)C2)=O)C(C)C1 n1(CC)cnc2c(NCCc3cn[nH]c3)[nH]c(=NC(C)C(C)COC)nc12 N1(C(CCN(C(C(CC)=CC)=O)CC)=O)CCCC1(C)CC C1(c2cn(C)nc2)CN(C(=O)C=CCO)CC1NC(C1CCCC1)=O Cc1ccc(C(=O)NC(C)(C)C(C)NC(c2cc(C)nc(O)n2)=O)c(F)c1 C1(NC(C(C2CCOC2)OC)=O)C(C)CCN(C(c2ncc(Cl)cc2Cl)=O)C1C C1(C)(NC(c2c(C)nc(CNC(c3cnnc(O)c3)=O)o2)=O)CCC(O)CC1 C1(CCC)CN(C(c2c[nH]nc2C(C)C)=O)CCN1C(=O)C(C)c1cc[nH]n1 c1(C(=O)NC2CC(C)N(C(=O)CCCN=[N+]=[N-])C2)ccc(=O)n(CC(F)(F)F)c1 Clc1cc2c(Br)ccnc2cc1CCCCc1ncc(Br)cc1N1CCC1 C1(NC(CC2(OC)CN(C(C3CS(=O)C3)=O)C2)=O)CN(C)CC1C C1(NC(c2c(CC)non2)=O)CC2(C1)CC(CNC(c1ccc(C)cc1O)=O)C2 C=CC(F)(F)C(=O)N(CC)CC1(O)CN(C(=O)CN(C)C2CC2)C1 CC(C)CC(O)CC(=O)NC(C(=O)N1CC(Cc2ccoc2)C1)C1CCC1 CC1c2c(F)cccc2CCN1Cc1cc2ccccc2nc1Br CCCC(C(=O)N(CCCSC)C1CC1)NC(=O)CC1CCCN1C(=O)OCC C1(CC(CO)(F)F)CCCN(N2CCC(c3cccc(O)c3F)CC2)C1 n1(CC)ccc(C(=O)NCC2(C(C)NC(=O)C(C)C(F)F)CC2)cc1=O Cc1ncncc1C(=O)NC(c1occc1C)(C)C.N1CCC(N2CC(O)C2)C1 c1(C(=O)NC2C(C)CCN(C(=O)CC3CCC(=O)O3)C2)ccn2ccnc2n1 N1(CC)CC(CNC(C2(NC(=O)COCCCOC)CC2(C)C)=O)CC1=O c1(NCCCC2COC(C)(C)O2)ccc(S(=O)(=O)NC(C2CCC2)=O)cc1F C#Cc1ccnc(C(=O)NC2(C(N3CCCC(F)CC3)=O)CCN(C)C2)c1 c1(N(C)C)ccc(C(N2C(C(N3CCC(O)(C(F)(F)F)C3)=O)CC3CC23)=O)cn1 c1(OC)cc(CNC(C2(CCNC(c3c[nH]nc3C)=O)CCC2)=O)n(C)n1 C=CC(CCC)CC(=O)N1CCC(C(=O)Nc2cccnc2OC)CC1C C1(CNC(c2cc(CC)oc2C)=O)CC2(CC2)CN1C(=O)Cc1cccc(Cl)c1 N(C(=NCSC)N1CCC(O)C1)Cc1c(OCC)cccc1OC CCC(COC)C(=O)Nc1nc(C(=O)N(CCCn2nc(C)cc2C)CCO)cs1 CCCC(O)C(=O)NCCC(C)NC(=O)C(COC(C)C)NC(C)=O.OCC c1(C(=O)NCC2CCN(C(COC3(C#C)COC3)=O)CC2)cccc(CC)c1C c1(C(C)(C)CNC(=O)NC2CC=C(C(=O)OCC)C2)cn2ccccc2n1 c1(C(=O)NC(CC)CN(C(=O)CCn2ccnn2)CC)conc1C1CCCO1 S(=O)(=O)(c1cccs1)N(CC(C)NCC1(O)CN(C(=O)CC2(C)CCC2)C1)C C1(C(=O)NCC2C(NC(=O)CN3CCC(O)CC3)C2)CN2CCCC2CO1 c1(NC(C2CN(S(CCOCC)(=O)=O)C2)=O)cnc(OC)nc1C C(CS(=O)(=O)CC(=O)N1CC=C(CNC(C2CCC(C)S2)=O)CC1)OC N1(C(C(C(C)(C)C)N(C)C)=O)CC(O)(C2(CNC(C3COC3)=O)CC2)C1 C#CCCCCCc1nc(-c2ccccc2)nn1C(C1CCCC1)C C(=O)(C(C)S(=O)(=O)C1CCOCC1)N1CC2(CC(NC(C(CC)(C)C)=O)C2)C1 C1(N(c2nonc2N)C(CC2C(C)(C)C2)=O)CCCN(C(C2CCCC2)=O)C1 C1([Si](C)(C)C)(CNC(CN(CCC)C(c2cncc(OC)n2)=O)=O)CC1 C1(C#N)(C(=O)NC2(CNC(C(CCOC)C)=O)CCOC2)CCOCC1 C1(CNC(c2ccc(CCC)cc2)=O)CN(C(C2CCOC2=O)=O)CCC1(C)C Cc1ccc(NC(=O)CCn2cc(C(N3CCN(C(C)C)CC3)=O)nn2)c(F)c1 CC1(C2CCCN(C(C(=O)NCCC3CC3)C3CCCC3)C2)CC1 O=S(=O)(c1ccc(C(=O)O)c(F)c1)NC1CCn2c(C3CC3)nnc2C1 N1(C(C(CC)C)=O)CCCC(C)(CNC(c2nc(C3CC3)ncc2Cl)=O)C1 c1(CC)cccc(C(N2CC3CCC3(NC(C3CC3C)=O)C2)=O)c1O C1(CNC(CCCCCSC)=O)CN(C(c2cnnc(C)c2)=O)CC2(CCC2)O1 c1(N2CC3CC(NC(C(CC)NC(C)=O)=O)CC3C2)nc2cc(F)ccc2o1 Cn1cc(C=CC(N2CCC(OCC(=O)NCCN3CCOC3=O)C2)=O)nn1 c1(SC)cc(C(=O)NCC2CCCN2C(=O)Cc2nc[nH]n2)c(C)o1 c1(CC(=O)NC2C(NC(C=C(C)c3cnn(C)c3)=O)C2)ccc2nc(O)[nH]c2c1 CCCC(C)C(=O)NCc1nc(CNC(=O)C(C)OCCOC)cs1 C1(C(=O)NOCCn2cnnn2)CN(C(=O)CC2CCSC2)CC12CCC2 c1(CC(=O)NC(CC)(CNC(C2CC2OC(C)(C)C)=O)CC)n[nH]c2ccccc12 c1(C(N=c2cc(C)n(C)[nH]2)=O)ccc2c(c1)CN(c1ncnc3sc(C)cc13)C2 N1(C(c2cnc(CC(C)C)[nH]2)=O)CC2CC1CCN2C(=O)CC1(CO)CC1 C(C(C)(O)CNC(C1CCN1C(C1CC(=O)C1)=O)=O)N(C)C C(=O)(C1CCCc2nncn21)NCC(CCNC(C=CC(=O)OCCCC)=O)O C12(NC(c3cn(CCC)nc3)=O)CCC(C(=O)OC(C)(C)C)(CC1)C2 c1(-c2cnc(CCC(=O)OC(C)=O)o2)ccc(C)cc1.C12(OC)CCC(C1)CO2 c1(C(=O)OC)c(F)c(NC(N2CCN(c3ccc(=N)[nH]n3)CC2)=O)cc(F)c1F c1(-n2cc(C3N(C(Cc4c(C)cccc4)=O)CCOC3)nn2)ccc(Cl)cc1F n1(CCC(=O)NC(C2CN(C(C(C(C)C)OC)=O)C2)C)ccc(O)nc1=O C#Cc1ccc(C(=O)NC(CNC(=O)CCCSC(C)(C)C)CCCC)cc1Cl c1(OC)cc(C(=O)NCCCN(C)C(c2cn(CC3CCOC3)nn2)=O)ccn1 CC1=C(C(=O)NCC2(CNC(C3(C)CC(F)(F)C3)=O)CCCC2)C(C)(C)CCC1 c1(C(=O)NCCN(C(=O)C=Cc2nc(C)c(C)[nH]2)CC)cnc(C(C)C)nc1C N1(C(CC2(OC)CN(C(c3c(CC)ocn3)=O)C2)=O)CC(C2CC2)(OC)C1 c1(CC(=O)NCCCN(C(=O)C(O)C(C)C)CCCOC)ccnc(Br)c1 N1(C(CC2CCC(=O)NC2)=O)CCN(C(=O)C(=O)Nc2ncc[nH]2)C(CC(F)F)C1 C1(C(=O)NCCC2CCCN(c3nc(Cl)ns3)C2)(OC)CS(=O)(=O)C1 c1(C(N2CCN(C(=O)Cc3csc4nccn34)CC2)=O)ccc2ccsc2c1 C#Cc1ccc(Br)c(C(=O)NC2CN(C(=O)C3=CC4CCC3C4)C2)c1 c1(CNC(=O)NC(C(=O)OCC)Cc2cscn2)cc(Cl)ccc1Cl n1(CC(=O)NCC2(F)CCC(NC(CCC#C)=O)C2)ccc(=O)c(O)c1C C1(C)(CNC(C(C=C)C)=O)CN(C(=O)CCc2ccccc2)CC1C N1(C(=O)Cc2cccs2)CCN(C(=O)COCCC2C=CCC2)C2(CCC2)C1 C1(C(=O)NC(C(=O)N(C(C2CCC2)C)CC)C)CCC(C(N)=O)C1 CC1C(N(C)C)CCN1C(=O)CCN(C(=O)C(C)(C)n1ccnn1)C1CC1 C1(CSCC)CCCN(C(C2CC(OC)CN2C(=O)Cc2[nH]cnc2C)=O)C1 C(CNC(=O)C(=O)C1CCCC1)(CC(=O)NCC1CC[Si](C)(C)C1)OC C12(CNC(=O)Cc3csc(NC=O)n3)CC1CN(C(=O)CCCc1nccs1)C2 C=C(C)CC(C)C(=O)NC1CCCCC1NC(=O)CCN(S(C)(=O)=O)C C1(NC(=O)CC2(c3ccon3)CCC2)CCOCC1C(=O)NCCC(F)F C1(CNC(c2cc(Cl)n[nH]2)=O)OCCC1C(=O)NCCCSC CC1CCc2[nH]c(=NCCCNC3CCOCC3)[nH]c(=NCCC3CC3)c2C1 Cc1cc(C(=O)NC(C2CCCN2C(=O)C(C)C2CCC2)C)nn1C(C)C c12cc(OC)cc-1c2CC(N1CCC(O)C(O)C1)=O.C(=O)(CC(C)OC)N1CC1.COOC C(CC(C)C(=O)NC(C)CCC(=O)N1CC(O)(c2nn[nH]n2)C1)OC c1(NC(C2CC(C(C)C)C2)=O)cc(CNC(=O)COC2(C)CCCC2)on1 C(=O)(CCCCC(F)(F)F)NC1(C)CCN(C(C2CCCCC2O)=O)C1 Cc1ccc(C(N2CCC(CNC(C3CCCC3)=O)C(C)C2)=O)c(C2CC2)c1 C(N=c1[nH]c(=NCc2ccc(F)c3[nH]ccc23)[nH]c2c1CSC2)C1CC(O)C1 N1(C(=O)NCC(=O)OC)CC2CC(N(c3cccc(OC)c3C)C)CC1C2 C1(N(C(C(C)CN2CCCCC2)=O)C2CCCC2CN)CCC(F)(F)CC1 C1(NC(C(C)c2cc[nH]n2)=O)CCC(NC(=O)CC=C(Cl)Cl)CC1 N1(Cc2c(C)cccc2Cl)CC2(CN(C(c3ccccc3Br)=O)CC2CO)C1 C1(C2CC2)(NC(CCC=C=C)=O)CCN(C(=O)C(CCC)C(C)C)C1 c1(C(CNC(=O)NC(c2ncc(C)s2)C)(C)O)ccc(F)c(C(F)(F)F)c1 C(=O)(C(C)CS(C)(=O)=O)NCC1[N+]([O-])(CC)CC1.N12CC(C(O)C1)C2=O C1(C#N)(C(N(C2CCCN(C(CCSCCCC)=O)C2)C)=O)CC12CCCC2 c1(CC(=O)NC(C)CCNC(=O)C(C)c2ccco2)ccc(C2CC2)cc1 c1(C(=O)NCCC(CCNC(C2C(C)OC(=O)N2)=O)C)ccc(S(N)(=O)=O)o1 c1(C(=O)NC2CCC(CNC(CCCNC(C)=O)=O)C2)cc2n(n1)CCO2 N1(C(C=CC(C)C)=O)CCC2(CC2C(=O)NC2CC3OC(=O)CC23)C1 C1(CCNC(CCNC(=O)NC)=O)COCCN1C(C1COC(=O)O1)=O C1(C)(C(=O)NC2CC(C)(CNC(C3CCCSC3)=O)C2)CCC(=O)C1 C#CC1(NC(=O)C(c2ccco2)NC(=O)C(c2ccnn2C)C)CCOC1 c1(C(N2C(CNC(c3ccc(C=C)cc3)=O)CC2)=O)cc(OC)c(OC)cc1C Cc1[nH]nc2c1CCC(C(=O)NC(C)CNC(=O)CNc1ccccn1)C2 CC1(CNC(c2ccc(CO)nc2)=O)CCC(NC(C2CC3(CCC3)C2)=O)C1 C1(NC(c2cc(C)sn2)=O)C=CCC(C(=O)NC(c2cn[nH]c2)C)C1 C=CC1(C(=O)NCCOC2CN(C(c3c[nH]nc3C3CC3)=O)C2)CCC1 C1(C)(NC(C2C(=C)CC2)=O)CCCN(C(=O)CC2C(=O)ON=C2C)C1 C=Cc1cncc(C(=O)NCCC(C)CCNC(=O)CCC(C)SC)c1 C(=O)(C(CNC(C1CN(C(C)=O)C1(C)C)=O)C(C)C)N1CCN(C(CC)C)CC1 C1(CNC(C(C)OCCCC)=O)CN(C(c2cc(Cl)cs2)=O)CCC1C c1(OC)ccc(C)nc1CC1CN(C(C2CC2CNC(=O)Cc2ccoc2)=O)C1 c1(-c2nc(C(C)OC)nn2CC23CCCC2C3)n[nH]c2c1CN(C(C)(C)C)C2 C1(CNC(C(CC)n2cncn2)=O)CCN(C(c2[nH]ncc2C#N)=O)CC1(F)F c1(CC(=O)NCC(C)CNC(c2csc(S(C)(=O)=O)c2)=O)cccc2occc12 Cc1ccc(C(=O)NCC(O)CCNC(=O)Cc2cnn(C)c2)nc1C Cn1c(C(=O)O)nnc1S.C1(=O)CC(C2CC2)NC(=O)CC2(CC2)CN1 N1(C(c2ccn(CCOC)n2)=O)CC(C)N(C(=O)COCP(C)(C)=O)CC1C C12(NC(CN(C(C)=O)C)=O)CCCN(C(C3=Cc4c(scc4)CC3)=O)CC1C2 CCCCC(CC(=O)NC(C)(C)CC1CCCC1)NC(c1coc(C(F)F)c1)=O C1(CNC(C2CCOC2)=O)CCCCN(C(=O)Cc2csc(Br)n2)C1 C(=O)(CN=c1cc[nH]cc1)NCC(N(C)C(C1CC2(CCC2)CO1)=O)C1CC1 O=C(CN=C(NCC1CCOC1)NC1(n2cc(Br)cn2)CC1)Nc1cccnc1 c1(C(N2CC3C(NC(CNCC)=O)C(C3)C2)=O)cnc2ccnn2c1.C(C)=O C1(CNC(C2N(S(CC)(=O)=O)CCC2)=O)CN(C(C2(n3cccn3)CC2)=O)CCO1 C(=O)(C1Cc2ccccc21)N1CC(C)C(NC(c2scc3c2OCCO3)=O)CC1 C(=O)(C(C)(O)C(C)(C)C)NCC(C)NC(c1ccn(CC(F)(F)F)c(=O)c1)=O CC1(C)CCCN(C(c2nsnc2O)=O)C1CNC(C12COC(CF)(C1)C2)=O CC1(C)CCC(n2cc(CSC3CC3)nn2)CN1C(C1CCN(C2CC2)C1=O)=O N1(C(C=CCC)=O)CCC2CC(NC(=O)CC(C)(C)CC)CCC2C1 C1(OCC(=O)NC(C)CC(C)NC(C2C3CCC23)=O)CCC(F)(F)CC1 C1(C(N(CCCNC(c2cc(COC)on2)=O)C)=O)OCCOC1(C)C C(=O)(C(C1=CCC2CC1C2(C)C)N(c1ccc(OC)cc1)C)NCC=C N1(C(c2cc(C)nc(O)c2)=O)CC2CCCC(Nc3cc(Cl)c(O)nn3)C2C1 n1(CC)nnc(C)c1C(=O)NCCOCCNC(C1(C)CC1(F)Cl)=O CCCC(C(=O)N1CC(Cc2cn(CC3CCCC3)nn2)C1)c1cccc(Cl)c1 N1(C(CC2(C)CCC2)=O)C2CCC1CN(C(C1C3COCC13)=O)C2 c1(C(=O)NC(C(C)NC(c2cc(C)nc(O)c2)=O)(C)C)coc2ccccc12 C(C(C)(C(C)C)NC(=O)C(C)Cc1cnco1)NC(C=C(COC)C)=O CC(CC(=O)NC1(CO)CN(C(c2ccn(C(C)(C)C)n2)=O)C1)S(C)(=O)=O N1(C(C(C)O)=O)CCC2(CC1)CCN(C(c1cccc3c1OCCN3C)=O)C2 C1(C)(C(N2CC(NC(c3c(C)nn(C)c3Cl)=O)C(C)CC2)=O)CCCCC1(F)F N1(C(C(=O)NC(CN(C)C)Cc2ccccc2)=O)C2CCC1CN(C)C(=O)C2 O=S(=O)(c1ccc(OC(F)(F)F)c(F)c1)NCc1cc2ccc(Cl)cc2s1 C(CCCN=c1[nH]c(Cl)ncc1Br)NC(N1CC(C)CC(C)C1)=O C1(CC)CN(C(=O)C(C)(F)F)CCN1S(=O)(=O)Cc1ccc(OC(F)(F)F)cc1 C1(NC(CSC)=O)CN(C(=O)C=Cc2ncc(C)[nH]2)CC1F C1(C#N)(CCCCCN(S(C)(=O)=O)C)CCNCC1.C(C)(C)(C)NC(=O)O C1(CCN(C)C(c2snc(Cl)c2Cl)=O)CCCCN1C(=O)CC1CCN(C)C1=O c1(CC)cccc(F)c1C(=O)NC(C1CCCN1C(C1CC=CC1)=O)C c1(C(=O)NC2C(NC(C(CC(C)C)C)=O)C2)cc(Cl)cc2ccncc12 c1(C(N2CCC(C)C2C(=O)NC2CC(=C3CC3)C2)=O)cc([N+](=O)[O-])c[nH]1 N1(C(C(=O)Nc2ccc(-n3cnnn3)cc2)=O)CC2CC3CC2C1C3O N1(C(CCCOC)=O)CC(NC(c2nc(Br)sc2C2CC2)=O)CC1C c1(NC(C2C(NC(c3cc(C)c(Br)cc3)=O)CCC2)=O)cnnc2ccccc12 C=CCC(C)(C)CCNC(=O)C(c1cccs1)NC(=O)CCOCC(C)(C)C Cc1ccc(N)cc1C(N1CCCC(CNC(C2CCCC(C)O2)=O)C1)=O C1(C(=O)NCC2C(NC(C3CC4(CSC4)C3)=O)COC2)CC(=O)C12CCCC2 c1(C(N2CCN(C(CC(=C)C)=O)CC2c2ncc[nH]2)=O)cccc2nc(O)oc12 C1(NC(CC2(C=C)CC2)=O)CCCN(C(=O)CCOc2cc(F)cc(F)c2)CC1 c1(C(N2CCCC(CC(=O)NC3(C#C)CCCCC3)C2)=O)cc(C)c(F)cc1C c1(C(=O)NCC(C2CN(C(c3n[nH]cc3Cl)=O)CCO2)(C)C)nnn2ccccc12 N1(CC(=O)NC2(NC(=O)C(=O)c3ccco3)CCC2)CCc2ccccc21 C1(C(N(CCCO)CC)=O)(CNC(=O)Cc2ccccc2O)CC12CCC2 N1(C(CCC#C)=O)CCC(C2CN(C(c3cncc4nc(O)[nH]c34)=O)C2)CC1 C1(COC)(CNC(=O)C(CO)N(C)C)CCCN1C(=O)CCNC(=O)C=CCl C1(C(=O)N(C)Cc2n[nH]c(C)n2)(CC)CCCN1C(c1nccs1)=O N1(C(CNC(CCC)=O)=O)CC=CC1(C)C(=O)N(C)CC1COCCO1 N1(CC(CN)C2CCC2)CCC(C2COCCO2)CC1 C1(O)(CN(C(CNC(=O)OC)=O)C)CCN(C(c2cnc(Br)s2)=O)CC1 c1(C(=O)NCC(CC)NC(=O)C(C)OCC2CC2)nc(C)c(C)s1 c1(OC)ccc(C(=O)NC2CCCC2CNC(C2CCC2(F)F)=O)cc1Br Cc1n[nH]c(C)c1C(=O)NC(C1CCN(C(=O)CNC(C2CCC2)=O)C1)C c1(OCCCC(=O)OC)cccc(Cn2cc(CNC(C3CCCS3)=O)nn2)c1 c1(CSC2(C(=O)NC(C(=O)NC)C3CCC3)CC2)cc(Br)cnc1O C1(CCn2cc(CC(=O)O)nn2)CCCN(C(C2CC23CC(F)(F)C3)=O)CC1 Cc1c(C2(C(=O)N(C3C4CN(Cc5ccccc5F)CC34)C)CC2)cccc1F C1(NC(c2ccnc(Cl)c2Cl)=O)CC2CN(C(C3CN4CCC3CC4)=O)CC2C1 c1(NC(C(=O)NC(c2nnc(C(F)(F)F)s2)C)C)nn(C)cc1Cl C1(C(N2CCC3(NC(c4ccc(F)o4)=O)CCCC23)=O)(OC)CCC(C)(C)CC1 c1(C(c2n(C(C(=O)OC(C)C)C)nnn2)NCC2CC2)ccc(F)c2occc12 C1(C(N2CCCN(C(C(CC)C)=O)CCC2)=O)COc2cccc(OC(C)=O)c2C1 c1(CNC(CC=C)=O)ccc(CNC(=O)CSS(C)(=O)=O)cc1 c1(C(=O)NCCCN(C)C(C2CC3(CC3)C2)=O)n[nH]c2c1CC(F)(F)CC2 n1(CC)nc(-c2cccc(Br)c2)nc1C1CC1(C)c1cccs1 C(CCC(C)C(=O)N1CCC(CNC(=O)CN2CCC(C)(O)C2)(OC)C1)OC N1(C(c2ccn(CC)n2)=O)CCC(C2CN(C(=O)Cc3cncc(F)c3)C2)CC1 C1(C(N2CC(CNC(CCN3CCN(C)C(=O)C3)=O)C2)=O)CCCC1S(C)(=O)=O n1(CC(=O)NC(C)CCNC(=O)CC2CCC2)nnc2ccccc12 O=C(CS(=O)(=O)CC1CCCO1)NCC(O)CCNC(c1ccoc1Cl)=O C1(C(N2CCOCC2C2CC2)=O)CCCC(CN2CCCC2)C1 Cn1cncc1C(O)C(=O)NCCC1(NC(=O)CCC2CC(F)(F)C2)CCCC1 Cc1cc(F)c(C(=O)NCCCC2CCCN2Cc2cnc(C(C)C)s2)cc1F C1(NC(C2N(C)C(=O)NC2)=O)CC2CCC1(NC(C1(F)CCCCC1)=O)C2 C1(N(C(=O)CC23COC(CF)(C2)C3)C)CN(C(c2csc(Cl)c2)=O)CC12CC2 N1(c2n(CCCOC)c(CS(=O)(=O)C(F)(F)F)nn2)CCc2ccccc21 c1(OCc2[nH]nc(SC)n2)c(C)nn(CC(F)F)c1C C1(NC(COCCOC)=O)CN(C(C23C4C5C6C4C2C6C35)=O)CCC1(C)C C(C)(N=c1[nH]c(NC2CSC2)nc2c1SCC2)c1nnc(C)s1 c1(C(C(=O)N(C2CCC(NC(=O)CC=CCO)CC2)C)CO)ccc(Cl)cc1 NC(=O)CCCCC(=O)N1CCC2CN(C(C3CCCN3C3CC3)=O)C2C1 c1(NC(C2(CC=C)CCN(C(=O)CCSCC(C)C)C2)=O)ccccc1[N+](=O)[O-] N1(C(CCC=C)=O)CC2(C1)CN(C(C1(c3ccsc3)CC1)=O)C2 C1(NC(C2CC(CC)OCC2)=O)CCCC2CN(C(C3(n4cnnn4)CC3)=O)CC12 c1(C(N(C(C(=O)N(CCC(=O)OCC)C)C)C)=O)n[nH]c(C)c1O N1(C(C2CC(C)=C(C)CC2)=O)CC(C2CCN(C(=O)C(F)(F)C3CC3)CC2)C1 c1(C(N(CC(CNC(C2CC(C)(CC)C2)=O)O)C)=O)cccc2c1OCC(=O)N2 C=C(C)CCC(=O)NC1CCCC1CNC(=O)CC12CCC(CC1)C2 C(=O)(C(CCC(N)=O)n1ccnn1)Oc1ccc(C)cc1.C1(=O)CCCO1 c1(CC(=O)N(CC(C)NC(c2nnc(S)n2C)=O)C)coc2cc(O)ccc12 C(=O)(CCC(F)(F)F)NC1CC(C(C)NC(=O)C2=NOCC2)C1 c1(CNC(N2CCC(CCC)C2)=O)ccccc1Cc1cn[nH]c1 N1(C(C2CC(CC)C2)=O)CCN(CCN(C)C)CC1.c12ccc(nc1)C(=O)NC2 c1(C2C(CC(=O)OC(=O)C(C)C)C2)cccc(C(=O)NCC(C2CC2)OC)c1 N1(C(CCOCCN(C)C)=O)CC2CN(C(C3(O)CCOC3)=O)CCC12 N1C(=O)c2ccccc2S1(=O)=O.CCC(C(=O)N1CC(O)C1)c1cccnc1 CC(F)CN=c1[nH]c(N2CCC(CN3CCCC3)C2)nc2c1CCCC2 C1(NC(C(C)(C)OCC)=O)CC2CC1N(C(=O)Cc1ccc(C(=O)NC)nc1)C2 Cc1c(C(N2CCC(OCCCNC(c3coc(Br)c3)=O)CC2)=O)cnn1C N1(C(COC(CC)C)=O)CCC(CF)(NC(=O)COCc2cccc(Cl)c2)C1 C=CC1(C(N2CC(OC)C(O)C2)=O)CCN(C(C2CCCO2)=O)C1 Cc1nc(CC(=O)NC(C)CNC(=O)CCCN(C)C)c(C)s1 c1(CC)cc(C(N2CCN(C(c3cnnn3C)=O)C3CC23)=O)cc(O)n1 c1(CC(=O)N(CC(=O)N(CCCOCC2CC2)CC)CC=C)cc(C)ns1 c1(C(CNC(c2c[nH]nc2C2CCC2)=O)NC(C(C)CF)=O)cccc(Cl)c1Cl c1(OC(C(C)C(C)NC(=O)N(C)C)=O)ccc2nncn2n1 Cc1c(C(=O)N(CC(C)O)CCNC(c2ccc(C#N)[nH]2)=O)nn2c1CCCC2 c1(C(=O)NCC2CC(NC(C(C)(C)C3CCOC3)=O)C2)ccc(N)c([N+](=O)[O-])c1 N(C(=NCCCCl)NC)N1C(C)CCCC1C.C1(S(C)(=O)=O)CCC1 N1(C(C(CC)CO)=O)CCOCC2(COCCN2C(c2ccc(O)nc2C)=O)C1 N1(CCC(C(=O)NC)NC(C2C(CCC)CCC2)=O)CC(=O)NC2(CC2)C1.OCC C1(C(=O)NCC2(N(C)C(c3[nH]cnc3C#N)=O)CC2)CC=CC(c2ccccc2)C1 N1(C(C(CSC)C)=O)CCC2(NC(c3ccc(C(F)F)nc3)=O)CC2C1 c1(CCNC(=O)NCc2snc(C(C)C)n2)ccc(F)c(C(F)(F)F)c1 c1(N(CCOC)C(=O)OC(C)C)ccccc1.c1(C2CS2)ccccc1 c1(C(N2CC(CNC(CC3(C(=C)F)CCC3)=O)(OCC)C2)=O)c(N)cccc1F Cc1cc(Cl)ccc1OCC(N1CCC(NC(C2CCC(O)C2)=O)C(O)C1)=O Cc1nc2ncnn2c(N(CC(C)NC(c2cnc(O)n2C)=O)C)c1C N1(CC(N2C(CNC(CCC(=C)Cl)=O)CC(OC)C2)=O)CCCCS1(=O)=O N1(C(CC(C)(C)C2CC2)=O)CCOCC(c2cn(-c3cccc(N)c3)nn2)C1 N1(C(COC(CC)C)=O)CCC(CNC(C2CCC(O)CC2)=O)C1(C)C C1(CC(C2CC2)NC(CN(C)CC)=O)CCCCN(C(C2CCCN2C=O)=O)C1 N1(CC(=O)NC(C)C(=O)NC2CC2)CCc2cc(CC(=O)O)ccc21 C1(C(CCCNC(C)=O)(C)C)CCCCN1C(=O)CN1CCS(=O)CC1 Cn1cc2ccc(CN3CC4(CC4C(=O)NCC4CNCCO4)C3)cc2n1 c1(C(=O)NC2CC(CCNC(C(C)N(C)C)=O)C2)c(F)c(F)cc(F)c1F C1(c2n(C(C)C)nnn2)(NCC2(C(C)(F)F)CC2)CCC(C#N)C1 C1(NC(c2cnc(CC)o2)=O)CCC2(CCN(C(=O)C(C)(F)F)C2)C1 C12(C(N3C(CNC(CCOCC)=O)C(CC)CC3)=O)CC3CC1C2C3(F)F CC(C)CC(C)(C)C(=O)N1CCCC(C(=O)NC2CCC(N(C)C)CC2)C1 N1(CC(=O)NCCC2CN(C(C(N)c3ccoc3)=O)C2)C(=O)CSC1=S C1(NC(C2(CCCC)CC2)=O)C2CCC1N(C(c1cc(C)n(C(C)C)c1C)=O)C2 c1(C(=O)NC2CCN(C(c3c(C)nn[nH]3)=O)C2)cc(Cl)ccc1OC(C)C C(=O)(C(C)(C)C1CCCN1C(C1CC(CF)C1)=O)N(C(C=C)C1CC1)C N1(C(C2N(C)CCC2)=O)CC2(CC2)CC1CC(=O)NCC1(CO)CC12CCC2 N1(C(CCc2onc(C)n2)=O)CC2CN(C(=O)Cc3cc(C(C)C)on3)CC2C1 N1(C(c2cnn(C)n2)=O)Cc2ccnn2CC(NC(c2cc(Cl)sc2Cl)=O)C1 c1(C(=O)NCCCC2CCN(C(=O)CC(F)(F)Cl)CC2)c(F)ccc(O)c1F N1(C(C=C(C)C(C)C)=O)CCCC(NC(=O)NCc2ccc(F)c(C)c2)C1C N1(C(CCC)=O)CC(C)C1C(=O)NC(C(F)(F)F)c1ccccc1 c1(CC)ccc(C)cc1C(N1CCC(O)C(NC(C2CC(C(F)(F)F)C2)=O)C1)=O c1(SCC(=O)N(C2CCN(C(C3CC3C3CCCO3)=O)C2)CC)cccc(C)c1 c1(CC)c(C(=O)NCC(O)CNC(C2(C)CCCNC2=O)=O)cccc1C c1(C(N2CC(NC(C3(SC)CC3)=O)C2)=O)ccc(F)c2ccncc12 C1(CNC(CCC(N)=O)=O)CCN(C(=O)CSCC(N)=O)CCC1(F)F Cc1cccc(F)c1C(N1CCC(NC(c2nccn2C)=O)C(F)C1)=O C1(CC(N)=O)CCCN(C(=O)Nc2ccc(Oc3ccc(Cl)cc3)cc2)CC1 C1(CC)CCN(C(c2coc(C)c2)=O)C(C(=O)NC(CO)CCC(C)C)C1 CCCC(C(=O)N1CCC(OCCNC(=O)C(C2CCCC2)C2CCC2)C1)OC Cc1nn2c(c1C(=O)NCC(C)N(C)Cc1c(F)ccc3occc13)CCCC2 C(=O)(C(CC)C(C)(C)CC)N1CCCC(F)(C(=O)NC(CCC=C)C)C1 c1(C(c2nnnn2CCOCC)NCCCC)cccc(Br)c1OC CC(C)CC(CNC(C1CC1C(C)C)=O)C(=O)NCCS(N)(=O)=O C1(CNC(c2c(SC)cccn2)=O)CN(C(c2nnsc2C)=O)CCC12CCC2 N1(CC(CO)NC(=O)NCCN(CC(=O)OC)C)CCC(C)CC1 C(=O)(C(C)CC(F)(F)F)NC1CCC(N(C)C(C2CC2c2cccs2)=O)CC1 C#CC1(C(=O)N(CCS(C)(=O)=O)C)CCN(C(=O)C(C=C)CC)CC1 CC1(CNC(C2(CO)CCCC2O)=O)CCN(C(C2C3COCC23)=O)CC1 c1(OC)ccc(-n2ccnc2SC2(C)CC(F)C2)cc1.N12CCN(CC1)C(=O)C2 CCCC(C(=O)N1CCC1C(=O)N(C)CC1CCCC1C)NC(N)=O N1(C(CN(C)S(N)(=O)=O)=O)C2CCC1CN(C(=O)C(C)(C)c1ccccc1)C2 Cc1ccc(C(N2CCC(O)C(C(N3CC(C)C3)=O)C2)=O)c(O)c1 CC1CCN(CC(N2CCC(N(C(=O)CCc3csnn3)C)C2)=O)CC1 CC1(C)CC(NC(=O)C(Cc2ccoc2)NC(C2CCS(=O)CC2)=O)C(C)(C)O1 C(=O)(CC1=CCCCC1)N1C(N)CC(C(C(=O)CCc2cncc(F)c2)=O)C1 CCCCCC(CNC(C1(C)CC1C(F)(F)F)=O)CO S(=O)(=O)(CCC(=O)N(C1CCCN(C(c2ccccn2)=O)CC1)C)NCCC C(=O)(C(F)(F)CC(Cc1ccccc1)OC(=O)NCCNC(C)=O)OCC CC1CCC(NC(=O)CN(c2ccncc2)C)CN1C(C1CCC2(CCC2)C1)=O N1(C(COCCC)=O)CC(N(C(=O)CN2C(=O)CCC2=O)C)C(C)(C)C1 c1(C(N2C(CNC(C(CCCCC)O)=O)COCC2)=O)cc(S(N)(=O)=O)oc1C C1(CC)CN(C(=O)Cn2cc(CO)nn2)CC1CNC(=O)CC1CCCC(C)O1 C(=O)(CCC(C)(F)F)N1CCC(CC)C1CNC(C1CC1(Cl)Cl)=O c1(C(=O)NCC2C(NC(C(CCC)O)=O)CC2)ncc([N+](=O)[O-])cc1C c1(OC)c(C(=O)NCC2CN(C(C3CC3(C)C(F)F)=O)CC2C)cccc1Cl c1(OC)cc(OC)[nH]c(=NCCNC(C2CCCN2CC(F)(F)F)=O)n1 Cc1cnn(CC(=O)NC2C3CCC2N(C(c2coc(C(F)F)c2)=O)C3)c(=O)c1 C(=O)(C(C(C)c1ccccc1)N(C(=O)Cc1ccccc1)CC(F)F)NC C1(NCC(C2(O)CCCCC2)C)CCC(=O)N(C)CC1 c1(NCC)cc(C(=O)NCCOCCNC(C2CC3(CCC3O)C2)=O)ccc1C c1(C(N(C)CC2CCN(C(C(C)SCCCC)=O)CC2)=O)cc(N)cc(C)c1F N1(CC(N2CCC(NC(c3cnnc(Cl)c3)=O)(CF)C2)=O)CCc2ccccc21 C(=O)(C(F)C(C)C(F)(F)F)N(C(C=CC)=O)CCNc1c(C)nn(CC(C)C)c1Cl C1(NC(c2cc(Br)c[nH]2)=O)COC2(C1)CN(CCCc1c(F)cccc1F)C2 Cc1nn(CCF)cc1NC(C1CCCC(NC(=O)CC2COCC(C)O2)C1)=O Cc1ccncc1C(=O)NC1C=CCN(C(C2(C)CCSCC2)=O)C1 Cc1ccc(-c2nc(C3CCCO3)nn2-c2ccc(Cl)cc2)cc1S(=O)(=O)N(C)C C1(CC)CN(C(c2csnn2)=O)CCN1C(=O)CC1(OCc2ccccc2)CC1 c1(OC)ccc(C(C)NCC(c2cc(Cl)cc(Cl)c2)CO)c(Cl)c1OC C(CC(C(=O)NCC1CCN(C(C2CCS(=O)(=O)N2)=O)CC1)NC=O)SC C1(CC)C(C(=O)NCC(CNC(c2c[nH]ccc2=N)=O)CO)CCN1C Cc1cc(=O)c(C(N2CCCC(N(C)C(C3CCN(C)C3=O)=O)C2)=O)c[nH]1 c1(C(N2CCC(C3CCCN3CCn3cc(Cl)cn3)C2)=O)ccccc1 C12(OC)CN(C1)C(=O)NC2.c1(CC(C)CO)ncccn1 c1(C(N2CC3C(NC(c4c(CC)nccc4)=O)(C3)C2)=O)cc2cc(C)ccc2s1 C(C(=O)NCCCOCCCNC(=O)C(C)(C)Cc1cnn[nH]1)(C(C)C)NC(C)=O C1(NC(Cc2nc(C)oc2)=O)CCN(C(c2cncc(Cl)c2Cl)=O)CC1O O=C1CCC(C(=O)NCC2(O)CN(C(=O)C=C3CCC3)C2)CN1 C#CC1C(C(N2CCC(N(C(=O)Cc3sc(S)nc3C)CCO)C2)=O)C1(C)C CCC(CC)C(C)C(=O)N1CC(OCC(=O)NC2CCCCC2C#N)C1 C1(CNC(C2(CC)CCCC2)=O)CCN(C(=O)Cn2cc(C#N)cn2)CC1(F)F c1(C(C(N2C(C=CC(=O)N(CC(=O)NC)C)CCC2)=O)C)ccc(O)cc1 CN=c1[nH]cc(C(=O)N(C(C)CCNC(C2CCCC3CC23)=O)C)s1 Cc1c(F)ccc(C(=O)NCC(O)CNC(=O)COc2ccsn2)c1C C=CCCCC(C(=O)N1CCOC(C#N)C1)NC(=O)Cc1ncccc1C N1(C(C(COC)O)=O)CC2(CNC(c3csc(O)n3)=O)CC1CO2 c1(Cc2c(NC(N(C(CF)CF)C)=O)cco2)ccc(C#N)cc1 N1(C(c2cc(C)nnc2)=O)Cc2occ(C(=O)N(C)CC3CCCC4CC34)c2C1 CN1CCC(C(=O)NCCCN(C)C(c2c[nH]ccc2=O)=O)CC1 C(=O)(CCN=C(NCc1ccc(-c2ccccc2)cc1)NC1CSC1(C)C)NC c1(C(=O)NCCCOC2CC(C(=O)N(CCN(C)C)C)C2)cc2n(n1)CCO2 c1(N(C)C)cccc(C(=O)N(C2CCCC2)CC(c2cccc(Br)c2)O)n1 CC1(NC(=O)C(c2ccccc2)=O)CC(NC(=O)CSC(F)(F)C(F)(F)F)C1 C(=O)(C1CCCc2cccnc21)NC(C)CNC(=O)C(O)CC(N)=O CCCCCC(O)C(=O)NCC1(CNC(=O)COC2(C)CCC2)CC1 CC(C)CC(C)C(=O)N1CCCC1C(C)(C)CNC(C1(C)CCCO1)=O CCCC(C)C(C)NC(=O)C(C)(C)NC(=O)CC(C)(C)C C=C(C)CCC(C)NC(c1cc(C)oc1C)c1nnnn1CCN1CCOCC1 C1(C(=O)NC(c2scc(C)n2)C)CC2CCCC2N1C(c1cc(F)cnc1O)=O Cn1nc(C(=O)NC(c2ccoc2C2CC2)=O)cc1C#N.C12CCC(C1)NC2C C(c1ccc(C2CC2)cc1)=C(C(=O)NC(CCO)c1ccco1)F N1(C(C=CC(=O)O)=O)CCC2(CC1)CN(C(=O)Cc1ccncc1)C2 Cc1ccc(SCc2ncncc2OCC(=O)Nc2ccnn2CC(C)C)cc1 c1(C(N2CC(O)(CNC(c3cccc(Cl)c3Cl)=O)C2)=O)c[nH]c2ccc(Br)cc12 Cc1ccc([N+](=O)[O-])c(C(N2CCC2CNC(C2OCCCO2)=O)=O)c1 C1(CNC(COC(CC)(C)C)=O)CN(C(C2(C)CC2C)=O)CCN1C c1(CC)ncc(C(=O)N(C2CCCCC2NC(c2cc(C(C)C)on2)=O)C)cn1 CC(CC(=O)NCC(C)(C)CC1CN(C(=O)CN2C(=O)CCC2=O)C1)C(C)(C)C C(=O)(C(C)CC(C)C)NCC(C1CC1)NC(c1ccc(OCCC)cc1)=O N1(C(=O)OC(C)(C)C)CCCC1(C)C(=O)NC1CC12CN(C(=O)CNC=O)C2 c1(C(=O)NCC2(COC)CN(C(=O)CC(C)(C)F)C2)cccc(S(C)=O)c1 N1(c2cc(C)nnc2O)CC(NC(c2cnc3[nH]cnc3c2)=O)CC(C)(C)C1 C1(C(=O)NCC2CC(OC)CN2C(=O)CSC(C)C)CCCC(C)(C)C1 N1(C(COCC=C)=O)CC(N(C)C(C2(c3cccc(F)c3)CCC2)=O)C(C)(C)C1 c1(NCc2cnc(SC)s2)cc(N2CCC(F)(CF)C2)nc(C)n1 N1(C(CCCNC(=O)OC)=O)CCC(CNC(C2CCCC2CF)=O)(OC)C1 C(=O)(C1=NN(C)C(=O)CC1)N1CCC(F)(C(=O)NC(c2ncccn2)C)C1 c1(OC)c(NC(=O)C(O)C2CN(C(C3CC4CCC4C3)=O)C2)c(C)nn1C C(N=c1nc(NCCCN2CCCC2)c2c([nH]1)CCC(C)C2)c1cn(CC)nn1 C1(NC(C2CN(C(C)C)C2)=O)CN(C(=O)CN(C)CCO)C2(CCOC2)C1 n1(CC)ccnc1C(=O)NCCOCC(=O)NCC1(C)CCCS1 Cc1n[nH]c(C)c1CCC(N1CCOC(C(=O)NCCCCCN(C)C)C1)=O c1(C(N2CC(CNC(c3cc(C4CC4)ccn3)=O)C2)=O)nc(F)ccc1Cl Cc1oc2c(F)c(F)c(F)c(F)c2c1C(=O)NCC(C(C)(C)C)N.C1(C(=O)[O-])CC1F C1(CC(=O)NCC(CCC)NC(=O)CC2(C#N)CC2)CCC(F)(F)C1 C1(CN(C(=O)C(CCN(C)C)NC(=O)OC(C)(C)C)C)CCC(F)(F)C1 C1(NC(C(CC)OC)=O)CC(CNC(C2(CC3CC3)CCCO2)=O)CC1O C1(CNC(c2cc(C)c(Br)cn2)=O)C2CCC1CN(C(=O)CCC(N)=O)C2 C(=O)(CC(C)(C(C)C)NC(=O)C(C)C)OCC.C1(=O)NCCO1 C1(NC(c2ccc3occc3c2)=O)CC12CCN(C(c1csnc1Br)=O)CC2 N1(C(=O)OC(C)(C)C)CCC(F)(F)C(Cc2cn(Cc3ccc(Br)cn3)nn2)C1 C(=O)(CC(C)(C1CCC1)C1CC1)NCC(CNC(c1c(SC)csc1)=O)(C)O C1(C2CN(C(c3ccc(F)c(O)c3)=O)C2)(NC(C2CC(C)OC2)=O)CC1 C=CCN=C(NCCc1ccc(COC)cc1)NC1CCOC1 C1(C)(CC)CC(NC(=O)CCn2nc(C)nc2C)CN1C(c1[nH]c(C)nc1C)=O C(CCCCN=[N+]=[N-])NC1CCN(C(CN(C(C(=O)NC)=O)C(C)C)=O)C1 c1(CNC(=O)CCC(CC)OC)nc(OCC)sc1NC(=O)CC1CC1.SC N1(C(c2ccc(OCCO)cc2)=O)CC2(C1)CN(C(=O)C(F)(F)C1CC1)C2 C(CNC(c1cc(Cl)c(Cl)n1C)=O)(CC(F)(F)F)NC(CC(COC)C)=O C1(C(=O)NCCCNC(C)=O)CC2(CC(NC(=O)C(C)n3cccn3)C2)C1 C(C1CCCN1C)=CC(=O)N(C)CC1(CNC(=O)C(=O)NC2CC2)CC1 N1(C(c2c(C)nc(=N)[nH]c2)=O)CCN(CCNC(=O)CC23CC(C2)C3)C2(CCC2)C1 C(=O)(CCCCCc1cccc(O)c1)N1CCC(NC(c2ccsc2)=O)(CF)C1 c1(C(N2CC3(C)CC2(CNC(=O)CCC(N)=O)C3)=O)cnn2cc[nH]c(=O)c12 CC(C)(F)CCC(=O)N1CCCCC(CNC(=O)C=Cc2cccc(O)c2)C1 Cc1cc(F)c(Br)cc1C(N1CC(C)N(C(C23COCC(C2)C3)=O)CC1C)=O C(=O)(C1=NOC2COCC12)N1CCCN(C(c2ccn(CCOC)n2)=O)CC1C c1(C(N(C)CC2CN(C(=O)CS(=O)(=O)NC3CC3)CCO2)=O)cc(N)cc(Cl)c1 C1(C(=O)NCCn2c(C)nnc2)CN(C(C2OC3CCC2C3)=O)CC1(C)C N1(CC(=O)N(C)CC2CN(C(=O)CCCc3cccs3)C2)CCCS1(=O)=O C(=O)(C(O)CC(F)(F)F)N(CCC)CCNC(=O)COCCN(C)C C=C=C(C)CC(=O)NC(CCSC)C(=O)N1CCCC1CCN(C)C Cn1ncc(C#N)c1C(=O)NC1CCCN(C(c2cc(N)ccc2F)=O)C1 N1(C(COc2cn(C)nc2)=O)CC(NC(=O)CC(F)(F)Br)C(O)C1 C=C(Br)CCC(=O)OCC(N1CCC(OCc2ccccc2)C1)=O C1(NC(=O)CC(O)c2ccccc2)CN(C(c2ccc(F)cc2)=O)CC1C(F)F CCCCC(O)C(=O)NCCN(C)C(C1Cc2ccccc2O1)=O CC1(O)CN(C(=O)C2=CCC(NC(c3ccoc3)=O)C2)CCC1O C(=O)(CCCCC(=O)NC1CCCC(CNC(=O)CCNC(N)=O)C1)N(C)C N1(C(CN(C(C(C)C)=O)C)=O)CCC(C(=O)NC2(C(F)(F)F)CCC2)C(O)C1 c1(C(=O)NC2(CCNC(=O)C(F)(F)F)CCC2)cnn(CC(F)F)n1 Cc1cccc2nc(N3CCC(C)(CNC(C4CCCCC4O)=O)CC3)oc12 C1(CC(=O)N(CCNC(Cn2cc(C(C)O)nn2)=O)C)CCCN(C)C1 N1(C(CNC(COC)=O)=O)CCC2CN(C(c3nc[nH]c3C(F)(F)F)=O)CC2C1 C(=O)(CC(C)P(C)(C)=O)NC1C=CCN(C(CC(=C)C)=O)C1 c1(C(=O)NC(CCCC)CNC(=O)CC2CCCN(C)C2)ccc(O)c(C)c1 Cc1ncc(N)cc1C(=O)NC(CCN(C(=O)CC1CC=CCN1C)C)C(C)C c1(CNC(C(CCC#C)O)=O)ccc2c(c1)CN(C(c1cnc(O)n1CC)=O)C2 C1(NC(c2nn(CC)c(C)c2)=O)CCCCN(C(C2C(C)C2(F)F)=O)C1 C(=O)(C(F)CCC(C)C)N(CCCCC(=O)NCCCC1(C)CC1)C c1(OC)ccc(C2CC2)cc1.C(CCC(=O)NCC)CNC(=O)C(CO)N(C)C c1(N2CCCC(NC(c3n(C)ncc3)=O)C(F)C2)ncnc2cnn(C)c12 C1(C(=O)NC(CC=C)CNC(=O)Cc2ccsn2)CC2OC(C)(C)OC2C1 N1(CC(C2C3CN(C4CCC5(C(=O)O)CC45)CC23)=O)CCN(C2CCCC2)CC1 N1(C(C(CCOC)C)=O)CC(C2(NC(=O)CCF)CC2)C1 c1(C(=O)NCCCN(C(C)C)C(c2ccc(C(F)F)o2)=O)c(Cl)ccnc1F c1(C(N(CC(C)NC(c2ccc(=O)n(C)n2)=O)CC)=O)snc2ccccc12 C1(C(=O)NCCC(=O)N(C)C2CC2)C2CC1N(C(c1cc[nH]c1)=O)C2 C(C)(C(=O)N(C)OC1CCCC1)NC(C(C)CN1CCOCC1)=O.C(C)(C)C C(=O)(C1CSc2ccccc21)NC1CCN(C(c2ccc(N)cn2)=O)CC1O C1(CNC(C2CN(C(CCOCCC)=O)C(CO)C2)=O)CC12CCOCC2 c1(OC)ccc(N(C(=O)Cc2noc(C3CCCO3)n2)Cc2ccc(F)cc2)cn1 CC1CC(NC(=O)CC2CCC2)CCN1C(=O)CN(c1ccccc1)c1cnco1 N1(CC2(NC(C(N)=O)=O)CN(C(=O)CC3CC=CCC3)C2)CCC(F)CC1 C#CC(CNC(=O)CNC(=O)CC1CN(C(c2ccoc2C(C)C)=O)C1)C(C)C CC(C)C(C)C(CNC(c1cnccn1)=O)NC(c1nc(C(C)(C)C)no1)=O c1(C(=O)NCC2(NC(C3CCC(=O)O3)=O)CCCC2)c(O)cc(Cl)cc1Cl C1(C(=O)NOCCC(C)O)CCN1.C(C(C)C)(C(C)C)CC.O CCCCCC(C)(CC)C(=O)N1CC2CC(NC(=O)C(C)(C)COC)CC2C1 C1(C(=O)NCC(CC=C)(C)C)N(C(c2[nH]ccc2COC)=O)CC12CCCC2 N1(C(Cc2c(C)non2)=O)CCC(N(C(=O)Cn2cnc(Br)n2)CCO)CC1 C1(CC=C)(C(N2CC(CO)C(O)C2)=O)CCN(C(=O)CCC2CC2)C1 c1(C(N2CCCC(C(C)NC(=O)C=Cc3cc[nH]c3)C2)=O)n[nH]c2c1CCCC2 N1(C(=O)COCc2ccco2)CCCC2CN(Cc3ncccc3F)CCC12 C12(C(ONC(C3(C)CC(NC(C4CCC4(F)F)=O)C3)=O)=O)C(=O)C3CCC1C2C3 c1(C(N2CC(O)(CCNC(CC3C(C)(C)CC3)=O)C2)=O)ccc(F)c2c1OCC2 N1(C(CC(=O)N(C)C)=O)CCC2(CCCC2CNC(=O)CC2CC2(Cl)Cl)CC1 CC(C)(F)CCC(=O)NC(C)(CNC(C12CC(F)(C1)C2)=O)Cn1cccn1 N1(C(=O)Nc2ccc(C)cn2)CC2CC(C1)N2C(C1(F)CCC1)=O c1(C(=O)OC)sc2ncc(Br)cc2c1NCCC(C(F)CO)OC N1(C(CC(=C)C)=O)CCC(C2CCOCC2)(CNC(=O)C=CC(C)CC)C1 C1(C(N2C3CN(C(c4coc(C5CC5)n4)=O)C(C3)C2)=O)CCS(=O)(=O)C12CCC2 N1(C(C2N(C(C)=O)CC(O)C2)=O)CC2CC(NC(=O)C#CC(C)(C)C)CC2C1 C(=O)(CCCn1cc(C(O)C(C)(C)C)nn1)NCCC(=C)C C1N=C2C=CC(=CN2)OCc2cccc1c2.c1cc(Cl)c(Cl)cc1F.C(=O)OC C1(C(=O)NC(CCNC(c2c(C)nc(CO)nc2)=O)C)CCOC2(CCC2)C1 C1(C(N2CCC(C)C2)=O)CCN(C(c2n[nH]cc2C(F)(F)F)=O)C2CCOC12 c1(CNC(=O)CC(O)CC2CC2)ncnc(C)c1OC.c12csc(n1)CNC2C C(C(CC1CCCC1)C(=O)NCC1CC(CF)C1)NC(CC=CC=C)=O C(=O)(C(C)(C)C1CCCO1)N(CC(=O)NC1(CN(C)C)CCC1)C1CC1 N1(C(C2CN(C)C2)=O)CC(C)CN(C(c2ccc(-c3ccncc3)o2)=O)CC1C C1(NC(c2cn(C3CCOC3)cn2)=O)(CC2CC2)CCSCC1 C1(C(C)C)CN(C(c2ccncc2)=O)CC1C(=O)NC(C)CN1CCOCC1 C1(C(=O)NCC2CC2CO)(CNC(COCCC(C)C)=O)CC(C)(C)C1 N1(C(C=CCOC)=O)CCCCC1C1(NC(c2c(C)n[nH]c2C)=O)CC1 CCCCCCC(CC)NC(=O)CC1(O)CCN(C(=O)CC(C)(C)C#N)C1 c1(SC2(C(N(C(C)CN(C)C(C3CC3C(F)F)=O)C)=O)CCC2)ccc(Cl)cc1 c1(C(N(CC(C)C)CCF)=O)cccc(Cn2cc(C3(F)CCOC3)nn2)c1 N1(C(C2(C3CCOCC3)CC2)=O)CCC(CNC(c2cnc(O)o2)=O)C(F)(F)C1 C(CC(=O)NCC1CCCS1)(C(C)C)NC(C1(C=C)CC1)=O C(=O)(CCCCCCS(N)(=O)=O)OCC1(C(=O)OCC)CCCC1 C(=O)(CC1=CCCCC1)NCC1CC1NC(C=C)=O.Cn1cc(N2CCC2)ccc1=O C1(NC(C2ON=C(C(C)C)C2)=O)CN(C(C2COC(=O)N2)=O)CC2(CC2)C1 C(=O)(CCC=CBr)N(CCOC)CCN(C(=O)C(F)n1ccnc1)CC CC(C)CCC(O)C(=O)N1CCOC(CCNC(=O)C(F)F)C1 Cc1ccc(N)cc1Br.C1(c2ccccc2)(C(c2nnnn2C)(F)F)CC1(F)F CC(O)CCC(=O)NCC1CC(C)N(C(=O)CCCCN(C)C)C1 c1(CC)cc(=NC2CN(C(c3cc(N(C)C)ccn3)=O)CC2C)[nH]c(Cl)n1 C1(CCC(=O)NC2(CNC(c3n(C(C)C)cnc3)=O)CCCC2)C(=O)NN=C1C C1(C=O)(CC)CC1(F)F.C(=O)(C(F)OC)NCCCN(OC(F)(F)F)CC N1(C(CC(C)C2CCCCC2)=O)CCC(CO)(NC(c2cscc2Cl)=O)C1 C1(NC(C(C2CC2)SC)=O)CCC(C(=O)NC2COCC2O)C1 c1(C(=O)NC(CN(C(CCCCC=CC)=O)CC)CC)cc(C)c([N+](=O)[O-])cn1 C1(CC)CC(C(=O)NC(C)(C)CN(C)C(c2oc(C)cc2C)=O)CCO1 c1(C(=O)NCCC2(O)CCN(C(C(C)CF)=O)C2)cnn2c1OCC(C)(C)C2 c1(C(=O)NC(C(C)NC(=O)COC2CCCCC2)(C)C)ccc2c(c1)NC(=O)CN2 C1(CC(=O)O)C(=O)NC1=O.c1(C(C)(C)C)ccc(CCC2CCOCC2)cc1 N1(C(c2cc(C)nn2C)=O)CCC(CO)(NC(C2C(C)C2(F)F)=O)CC1 C(c1cc(Cl)c2c(c1)OCO2)=CC(N1C(C(CC)O)CCC1)=O N1(C(CC(C)N(C)C)=O)CCCCC1CN(C)C(C1CCSCC1)=O CN1N=C(C(=O)NCC2CCC(NC(=O)CC3CC4(CC4)C3)C2)CCC1=O C=C=CC(C)C(=O)NC(c1ccccc1F)CNC(c1ccon1)=O c1(NC(C=C(CC)C)=O)cc(C(=O)N(CC)Cc2cccs2)cc(C)c1 c1(NC(CC(CCC)NC(C2CC(O)CN2C)=O)=O)ccc2c(c1)CCO2 C1(C(N(CCCCOC)C)=O)(CNC(=O)CCCN(C)C(C)=O)CCCO1 c1(C(=O)NC(C2CN(C(c3ncn(C)n3)=O)C2)C)ccc(C(F)(F)F)o1 c1(OCCNC(N2C(C)CC(C)C2)=O)ccc(Cl)c(F)c1 c1(C(N2CC(O)C(C)(C)C2)C(=O)NCCCSCC)ccc(F)cc1I O=C(C1c2ccccc2CN1Cc1cccnc1Br)Nc1ccccc1I N1(C(C2C(C)(C)CC2)=O)CCC2(CCC(CNC(=O)C3=NOCC3)O2)CC1 c1(C(=O)NCC2(C(C)NC(=O)CC3C=CCC3)CC2)ccnc(O)c1 Cc1c(Br)c(C(N2CC(NC(=O)CCc3nnc(S)n3C)C2)=O)nn1C C1(CNC(c2cc(Cl)c(Br)cn2)=O)CC1C1CCCC1 c1(C2CCN(C(C(=O)NCC3C(C)C3C)=O)C2)cc(F)cc(F)c1 c1(NC(CCOCCOC)=O)cccc(Cl)c1C.C1=CCNC1=O N1(C(c2cc(C(C)C)on2)=O)CCCC(NC(c2ccccc2)=O)C1C Cc1ccn(CC(N2CCCCC(NC(=O)CC(C)n3cccn3)C2)=O)c(=O)c1 N1(C(c2ccc(C#C)o2)=O)CCCC2CCN(C(=O)CC3(O)CCC3)CC12 CC1CCN(C(=O)OC(C)(C)C)C=C1C(=O)NC(C1CCC(O)C(O)CC1)=O C(=O)(C(C)(C)COC(C)(C)C)NCC(CNC(C1CC(F)C(=O)N1)=O)OC c1(CC)ccnc(C(=O)NC(CN(C)C)C(=O)N(C)CC2CC2(C)C)c1 Cc1cc(CC(=O)NC2(CCC(=O)NC3CNC(=O)O3)CCC2)no1 c1(C(=O)NCC(=O)NCCCN(C(C2CC2C(N)=O)=O)CC)ccc(C(C)C)cc1 CCC(CNC(=O)CC1CC(=O)NC1=O)N=c1[nH]c2cc(Br)ccc2o1 CC1CCOCCN1C(C1CCOCCN1C(=O)C(N1CCOCC1)C)=O c1(CC)oc(C)nc1C.C1C(C)(C)OCC(=O)N1.C12(CC1)C(=O)N2.C1CN1.CC N1(CC(=O)N(c2ccccc2O)C)Cc2c(Br)cccc2C1=O C1(CNC(c2nc(OCC)sn2)=O)CCCCC1Nc1ccccc1 Cc1cc(C(=O)NC2CCC(CNC(C3(C)CC(C#N)C3)=O)C2)c(C(F)(F)F)o1 C(CCCCC(=O)N1CCC(O)(C(=O)NC(C)C(C)(C)COC)CC1)OC C(CCCCC(=O)N1CCCCC1CN(C)C(C1CCCC(=O)CC1)=O)=CC Cc1ccc(S(=O)(=O)NCC(=O)NC23CCN(C(C4OCCO4)=O)CC2C3)cc1 n1(CCOC)nc(C)cc1CNc1ccc(-c2nc(C)cs2)nc1 O(N1CCC(CC(=O)NCC(C2CCC2)NC(C2(Cl)CC2(C)C)=O)CC1)CC C(=O)(C(N)C(C)CCC)C(=O)CCCCCN.C=CCC(C)N c1(N2C(CCNC(C3N(C)CC(C)(C)C3)=O)CCC2)ncc([N+](=O)[O-])cc1F c1(C(=O)NCC2(NC(C=C(C)C(C)C)=O)CCCCC2C)cn2cc(C)sc2n1 N1(C(=O)C2CCCc3ncnn32)CCCCCC(N=c2ncc3ccccc3[nH]2)C1 N(C(=NCCCC(=O)N(C)C)NCc1cc(Cl)cc(Br)c1)C(CC)CC C1(C(=O)NC(CC(=O)OC)C2CC2)CC2(C1)CN(C(C1CC(F)(F)C1)=O)C2 CC(C)(CS(N)(=O)=O)C(=O)N1CCC(CCNC(c2conc2C(F)(F)F)=O)C1 c1(NC2(C)CN(C(c3nccc(OC)c3OC)=O)C2)c(Cl)cc([N+](=O)[O-])cc1Cl Cc1ccnc(C)c1C(=O)NCC1CN(C(=O)COC(C)C)C(C)(C)C1 n1(CCC)cccc1C(=O)NC1CCCC1NC(=O)C(C)(C)N1CCCC1 c1(OC)c(C(=O)NC2CCCCC2NC(=O)CC(O)CC2CC2)nc(O)nc1O CC(O)(CC(=O)N(c1nc(CC(=O)NC)nc(=N)[nH]1)C1CCCNC1)CC(=O)O CC(C)CC(C(=O)N1CCOC(CCO)C1)NC(=O)C1=NNC(=O)C1 C1(CCNC(C(CC)OC)=O)CCCN(C(=O)Cc2nc[nH]n2)C1 C1(C(N(C(C2CCCC2)CNC(=O)CCCC(F)F)C)=O)CCCNS1(=O)=O N1(C(C2CN(CC(C)C)C(=O)C2)=O)CC2CCN(C(c3ccsc3)=O)CC12 Cc1ccc2c(c1)C(=O)N(CCCC(=O)Nc1cc(CC(C)C)[nH]n1)C2=O CC1(C(=O)NC2(C)CC=CC2)CCCN(C(C2CCCN2C(N)=O)=O)C1 C(=O)(CC1=CCOCC1)NCC(CNC(=O)C(O)CN1CCOCC1)OC c1(CC)cc(C(=O)NCc2ncc(C(=O)NCC3(C)CCC(=O)N3C)cn2)nn1C c1(OC)ccn2c(C(N3CCC3CNC(=O)CCC3CCCOC3)=O)cnc2c1 Cc1ccc(F)cc1C(=O)NCC1CN(C(c2csc(C3CCCO3)n2)=O)C1 C1(C(=O)NCC(CC)NC(=O)C(F)C(C)(F)F)CCC(=O)C(CC)C1 N1(C(c2c(C(=O)OC)coc2)=O)CCCC(CO)(NC(c2ccc(SC)o2)=O)C1 CCC(CNC(C1CCCSC1)=O)(CC)C(=O)N1CCC(C(C)(C)O)C1 C(=O)(CCC(=O)c1ccc(F)cc1)N1C(CNC(c2cnc(Cl)s2)=O)C=CC1 N1(C(=O)NC2CCC2)CCOC(C#N)C1.c12ccc(cc1)NC(=O)NC2C(=O)OC Cc1nc2cc(C(N3CCCC(NC(=O)C(Cl)=CCl)C(F)C3)=O)ccc2s1 N1(C(CC2C(C)CN(C(C34CC(F)(C3)C4)=O)C2)=O)CC2CSCC2C1 C(C(C)(CCO)N(C)Cc1n[nH]c(C2CC2)c1Cl)C(C)(C)C.C(=O)(C(=O)NC)NC N1(C(C2(SC)CC2)=O)CCC2CN(C(c3nnccc3C)=O)CC2CC1 C=C=CC(C)C(=O)NC(CC=CC)C(=O)NCC(=O)NC(C)CC.OC CCC(CC(=O)N(CCC(=O)N1CCC1CN(C)C)C)SC C#CCC(C)(CC)C(=O)N1CCC(CNC(c2cc(C)c(C)[nH]2)=O)CC1 Cc1cc(C(=O)NCCC(C)NC(c2cc(CO)[nH]n2)=O)on1 c1(C(C)NC(C2C(NC(C3(CC)CCOCC3)=O)C2)=O)ccc(Cl)cc1Cl C12CCCCCN1C(=O)NC(CC)CC(=O)O2.c1(OC(C)C)ncc(C)cc1F CCC(COC)C(=O)NCC(C1CC1)NC(c1cc(-c2ccccn2)c[nH]1)=O c1(CNC(=O)C(c2ccc(O)cc2)O)ccc(-c2cccc(Cl)c2)cn1 C(CC(O)C(=O)NC1CCCC(C(=O)NC2CC3CCC2O3)C1)SC CCC(C)C(C(=O)NCc1cc(C(=O)NC(C2CCCCC2)C)cs1)OC c1(C(=O)NC2CCC(C(N3CC(CC(=O)OC)C3)=O)C2)cccc(Br)c1F C1(C(=O)NCCN(C(=O)COc2cc(Cl)cc(Cl)c2)C)CCC2COCCC2C1 c1(C(C(=O)NCC(CC=C)NC(c2cccnc2O)=O)C)cc(F)cc(F)c1 c1(COCCC(=O)NCCC2CC2(Br)Br)ccccc1 O=C(CC1=NNC(=O)C1)NCC1CCC1CNC(=O)C(F)C(F)(F)F c1(CNC(C(c2ccccc2)NC(COCC)=O)=O)cc(=O)cc(C)[nH]1 c1(OC)c(C(C2CC23CC3(F)F)NCCCC(=O)Oc2ccccc2)cccc1Cl C(=O)(C1=CCCC1)N(CCCNC(c1cnc(-c2ccccc2)[nH]1)=O)C C(=O)(CCCCNC(C)(C)C)N1CC(c2cn(CCOC(=O)NCC)nn2)(O)C1 CC(C)(C)C(=O)C(=O)NC1COCCC1NC(c1csc(Cl)c1)=O C1(NC(n2ccccc2=O)=O)(CO)CCN(C(=O)COCC(F)F)CC1 c1(C(=O)OCC)ncc[nH]c1=NCC1CN(C(=O)NCC)C(C)(C)C1.C(C)(C)C C12=Nc3ccsc3C(=NCC(c3ccsc3)N1C)N2.C(C(C)(C)CC1CC1)OC N#Cc1ccc(C(N2CC3CC3(C(=O)Nc3cccc(Cl)c3Br)C2)=O)cc1F C1(NC(C(C)C)=O)CCC(NC(=O)N(c2ccccc2)C)C1.n12cc(nn1)C2 c1(C(=O)NCC(CNC(c2c(OC)cccc2F)=O)F)cc2n(n1)CCCC2=O C1(C(=O)NCCNC(CN(C(=O)CC=CCN)C)=O)CCC(O)CN1C n1(CC(C)C2CCC2)nc(-c2ccno2)nc1-c1ccc(-c2ccc(Cl)s2)nc1 c1(C(=O)NC2(CC)CCN(C(=O)CC(C)(C)C(F)F)CC2)cc2c[nH]cnc-2n1 c1(C(=O)NC(CC)(C)CCNC(C2CC2Cl)=O)cc(OC)ccc1OC Cc1cc(=NCC2CN3CCCCC3CO2)[nH]c(N2CCCC(C(C)C)C2)n1 C(C)(c1ccc(OC)cc1)=CC(=O)NC(CC)CN(C)C(C1CC2CCC1O2)=O C1(CC(=O)N(CC(C(=O)N(CCOCC)C)C)C)CCCCN1C CCCC(C)CCCC(=O)NCC(C)N(C)C(c1cnc(OC)cn1)=O N1(C(CCC2CCCN(C(c3noc(CC)c3C)=O)C2)=O)CCC(F)(F)C(O)C1 Cc1cc(C(=O)NC(C2(O)CN(C(c3cc(F)n(C)n3)=O)C2)C)nn1C(C)C CCCC(C)CC(C(=O)Nc1cccc([N+](=O)[O-])c1)N1CCC12CCC2 N12CCCC(C1)C(=O)NCCN(CCC)C(=O)C=CC2=O.C(C)(=O)NC1CC1 c1(CC(C)NCc2c(-c3cnn(CCN(C)C)c3)ncn2C)ccc(O)c(O)c1 C1(COC)CCC(c2nnnn2C(C)CC)(NC(C2CCCC2)C)CC1 N1(C(C2CC3(CC(OC)C3)C2)=O)CC2CC1CCC2NC(C1C2CC3C(C2)C13)=O Cc1cc(C(=O)NCC2CC(NC(C3CC(F)C3)=O)C2(C)C)cc(F)c1 c1(OC)ccc(C(=O)NCC2C=CCN2C(=O)CCc2ccc(C)nc2)nc1Cl C(=O)(C1=CC2(CCOC2)C1)N1CC2(OCC(NC(c3cn(C(C)C)nc3)=O)C2)C1 C1(C(N2C(C)(C)C(NC(=O)COCC3CCCC3)CC2)=O)CC2OC(=O)OC2C1 CCCC(C)(C)CNC(c1csc(-c2ccccc2)c1)c1nnnn1C C1(C(N2CC(C(C(=O)NCCCCO)OC)C2)=O)CC(=O)N(C)C1 Cc1nc(NC2CC(NC(=O)CSCC3CCCO3)C2)cc(C(F)(F)F)n1 N1(C(C2(NC(C(C)S(C)(=O)=O)=O)CCOCC2)=O)CCCC(C2CCC2)C1 C1(CCC)CN(C=O)CC1.C1(CC(=O)NCCN(CCC)CC)NC(=O)NC1=O c1(OC)cc(C(N2CCC(NC(c3cc(F)n[nH]3)=O)C(F)C2)=O)cnc1OC N1(CC(N2CCN(C(c3ccc(CC)s3)=O)CC2)=O)C(=O)CN(C)C1=O CC1(O)CCCN(C(C2COCCC2NC(C2(C#N)CC2)=O)=O)CC1 Cc1cc(C(=O)NC2(CCNC(=O)C#CC(C)C)CCCC2)ccn1 C1(C(N(CCn2cc(CC(COC)O)nn2)C)=O)CC2C=CC1C2 N1(C(c2[nH]cc(CC)c2)=O)CCN(C(C2(CC3CCC3)CC2)=O)CC1CC CC1(C)CC(NC(C)CC2=CCCC2)CCO1 C(CC1CCc2ccccc21)CCN1CCCC(C(N2CCC(OC)CC2)=O)C1 c1(CNC(NC(COCC)CC)=NCC2CC2)ccc(Cl)c(O)c1 c1(CNc2c(C(N3CCC(C#C)CC3)=O)n[nH]c2)c(Cl)ccc(C)c1F n1(SCC)c(C(N2CCCC2)=O)cnc1O.c1(-c2cn(C3CC3)nn2)cncc(F)c1 CN1CCCC(N(C)C(C2(F)CCN(C(C3CCCC3F)=O)C2)=O)C1 C(=O)(C(C)C(O)C(C)C)N(CC(=O)NCCN1CCCNC1=O)CCOC N1(CC)CC(CNC(=O)C(CN(C)C)NC(c2cc[nH]n2)=O)CC1=O CC1(C)CC(F)(F)CCC1C(=O)NC1CC(NC(C2Cc3ccccc3C2)=O)C1 C(C)(C)(C=CC(=O)NCCC(=O)CC1(CO)CCC1)SC.C(C)(C)(CC)O C1(C)(C(=O)NCC(CC(=O)OC)O)CC(O)CN1C(=O)CCC1(C)N=N1 C#Cc1ccc(Cl)c(NC(=O)CN2CCN(C(=O)COCC=C)C(C)C2)c1 C1(C(N(CC(C)NC(c2cc(C(C)C)[nH]n2)=O)C)=O)CC12CCCCC2 c1(CCC(=O)NCCOCCNC(=O)CSC2CCCO2)nc2ccccc2[nH]1 C(CC(C(=O)N1CCC(C(C)C)C1)NC(CC1=CCCOC1)=O)=CC CC(CC(=O)NCC1(N(C)C2CC2)CC1)NC(=O)CC1(C)CCOC1 CC1CN(C(c2snnc2-c2ccccc2)=O)CC(CCNC(=O)CCC2CC2)O1 CCCCN=C(NCC1=CCCCCC1)NCCOCC(C)(C)O C=CCC(CNCc1cnc(-c2cccnc2)s1)CC(C)C(C)(C)C c1(C(N2CC(NC(CC=C=C)=O)C(N=[N+]=[N-])C2)=O)cc2ccc(F)cc2o1 C1(C(=O)NC2C=CCC(C(=O)NC(C)Cn3cccn3)C2)(CC)CNC(=O)C1 C1(CC(=O)OC)COCCN1C(=O)C(c1ccco1)NC(=O)C=CC(C)C C1(C(=O)NCC(CNC(=O)C=Cc2ccsc2)CO)CCCC1C1CC1 c1(C2C(C(=O)NCC3CCN(C(c4ccc(COC)[nH]4)=O)C3)C2)ccccc1F c1(OC)c(CC(=O)NC2CC(C)(NC(=O)Cc3c[nH]nc3O)C2)cccc1Cl C1(CCNC(=O)CCc2cc[nH]n2)(OC)CN(C(c2csc(C)c2)=O)C1 C1(C(=O)NC(CCC)C(=O)N(C)C)(CC)CCN(C(=O)Cc2cn[nH]c2)CC1 N1(C(C(C)OC)=O)CC2CCOC2(CNC(=O)CC(C2CCC2)C2CCC2)C1 c1(CCC(=O)N(C2CC(NC(C(C(C)C)OC)=O)C2)C)cc(C)nc(C)c1 N1(C(C2CC(C)(C)OC2(C)C)=O)CCOC2(CCC(NC(=O)C=C(Cl)Cl)CC2)C1 C1(O)(C(=O)NCC(C2CCC2)NC(c2cc(C(F)(F)F)cs2)=O)CCSC1 c1(OC)ncc(Br)cc1C(C(=O)NCC1CCOC1)N(C)Cc1c(C)n[nH]c1C C(=O)(CCC(C)NC(c1ncncc1C)=O)NCC(COC)(C)O C(=O)(CN=c1cc[nH]cc1)NCC(CN(C(c1cc(C)c(O)nn1)=O)C)O c1(C(N(CCNC(=O)CCCSC(C)(C)C)CC)=O)cc(C)oc1C C(CC(C)C)(C(=O)NC(C1CCCN1C(c1oc(C)cc1C)=O)C)OC C1(CNC(c2ccc(C)nc2)=O)CN(C(=O)C=Cc2ccccc2)CCN1C C(=O)(C(C)C(O)C(C)C)NCC1(NC(c2cccc(C)c2Cl)=O)CCCCC1 CCC(CCCC(=O)N1CCC(CO)(COC)C1)NC(=O)CSCC(C)C N1(C(c2cn(CCOC)nn2)=O)CC(CC(=O)Nc2ccccc2Cl)CC1(C)C Cc1cc(C)c(C(=O)NC2CCN(C(c3nc(=O)cc(N)[nH]3)=O)C(C)C2)c(C)c1 c1(C(C(=O)NC(CN(C(=O)CCn2cccn2)CC)C)O)ccnn1C C1(CN(C(=O)CCC(C)N2CCOCC2)C)CCN(C(c2cncnc2)=O)CC1 N1(C(=O)Cc2cccs2)CCCC(C2CN(C(c3ccc4ncccn34)=O)C2)C1 C(=O)(C(CC)CCNc1ncc(NC)nc1)NCC1CC2C=CC1C2.C1(C2CC2)CC1 C1(NC(C2CC(C)(C)OCC2)=O)CN(C(C2CC(F)(F)C2)=O)CC(F)(F)C1 CC(C(F)(F)C(F)(F)F)=CC(N1CC(N(C(=O)CC2(CO)CCCCC2)C)C1)=O CCCCC(O)C(=O)NC(CC1CC1)CC(=O)NCc1ccc(C#N)o1 CC1CN(C(=O)CCNS(C)(=O)=O)CC2(CCN(C(C3(C)CC(F)(F)C3)=O)C2)O1 CC(C)(C(=O)NC1C2CN(C(=O)Cc3ccn(CC(F)(F)F)n3)CC12)C(F)F CCC(F)(F)C(=O)N1CCC(C(C)NC(C2CCSCC2)=O)C1 C(=O)(C(C(C)OC)NC(c1n[nH]c(C(C)CC)n1)=O)OCC C1(N(C(C(C2CCCC2)OCC)=O)C)CN(C(=O)Cc2ccccc2Cl)CC1O c1(OCC)ccc(Cn2nc(CC(C)(C)C)nc2C2CCOC2C)cc1 CC1(C)CN(C(C2CCOC2C2CC2)=O)CCC1C(=O)NC1CCCCCCC1 CCC(C(=O)NC(CN(C)C)C(=O)NCC1CCOC(C)(C)C1)C(C)C S(=O)(=O)(c1ccc(NCC(C)C#N)c2cnccc12)NC(C)CCC1CCCC1 C1(O)(CN(C(c2cc(CC)no2)=O)C)CCN(C(c2[nH]ccc2C)=O)C1 N1(C(C(C=C)c2ccccc2)=O)CC2CC1C2CNC(=O)C=CC1CCCCC1 N1(C(C2C(C)C2)=O)CC(CO)C2(C1)CN(C(c1ccccc1CN(C)C)=O)C2 C(C)(CCC(=O)NC1CCC(NC(=O)CSC2CCCCO2)CC1)SC N1(CC(c2ccc(Cl)c(Cl)c2)(CC)CO)CC(c2ccccc2)CCC1C c1(NC(C(CC)(C)CSc2nn[nH]n2)=O)ccc2cnn(C(F)F)c2c1 c1(C(=O)NC(C(C)C)C(=O)NC2(C)CCSC2)cc2ncccc2[nH]1 C1(NC(c2cc(CC)[nH]n2)=O)CCCN(C(c2conc2CC)=O)C1CC N1(C(c2cnc(CCC)s2)=O)CCCC12CCCN(C(c1ccc(C#N)[nH]1)=O)C2 C(=O)(C1CCc2c[nH]nc21)N1C(C(N(C(CC)CC)CC)=O)C=CCC1 Cc1cnc(C(=O)Nc2ccc(C(F)C(F)(F)F)cn2)c(C)c1 C(=O)(C1=NOC2(CCC2)C1)NCC1(CNC(C#CC(C)(C)C)=O)CC1(F)F c1(CC)nc(CCCNC(C2CC(O)(c3ccccn3)C2)=O)n[nH]1 N1(C(CSCCCC)=O)CC2CCOCC2(NC(=O)Cc2c(C)noc2Cl)C1 N1(C(c2ccc(C)cc2C)=O)CC2CCCCC2(NC(C2CC23CC(O)C3)=O)C1 C1(NC(=O)Cc2csnn2)CC2CN(C(=O)Cn3cnccc3=O)CCN2C1=O C(C)(C)(C(C)CC(=O)N1CC(N(C)C)C(C)C1)NC(c1c(C)scc1)=O C(=O)(CCC(=O)N1CCCC1)NCC(C)(CO)NC(Cc1c(CC)con1)=O N1(C(c2n[nH]c(C)c2Cl)=O)CCC2(C=C(C(=O)N3CC(OCC(N)=O)C3)C2)C1 Cc1cc(=NC(=O)C2=CCC(N(C3(C)CC3)C(=O)C3CC3)C2)[nH]n1C N1(C(C(C)(C)SC)=O)CCC(NC(c2c(C)cccc2Cl)=O)C(O)C1 c1(OC)ccc2c(c1)CCCC2N(C(=O)CC1(CN)CCOCC1)C(C(C)(C)C)=O c1(C(N(CC(CC)NC(=O)C(C)(C)F)CC)=O)cc(OC)c(Br)c(OC)c1 C=C(C)C1OCCC1C(=O)N(CCC(N1CCCC1CN=[N+]=[N-])=O)C(C)C c1(NC(Cc2ccc(C)cc2)=O)cc(Cl)ccc1C#N.C12CC(C1)CC(=O)N2.C(C)(C)N c1(NC)cccc(-n2cc(CNC(CCC(CC)(C(=O)OC)NCBr)=O)nn2)c1 Cc1sc(-c2nc[nH]n2)nc1C(=O)NC(C)CN(C)C(c1cc[nH]c1)=O c1(CC)nc(C)c(C(=O)NC2CCCC2(C)CNC(=O)C(C)SC)s1 C1(NC(C(CCSC)(C)C)=O)CC2CC(C1)CN(C(C1CC3(C1)CC(C)C3)=O)C2 N1(C(c2cn(CCC)nn2)C(=O)NCCOC)CCOCC1C1CCCO1 c1(C(N2C(COC)(CNC(=O)Cc3cc(C)no3)CCC2)=O)ccc(C#N)cn1 C1(C(=O)NCC(CNC(c2cnc(C)nc2)=O)OC)CCC(C(=O)N(C)C)CC1 Cc1cnccc1CNC(C1CCC(C2CC2)N1C(=O)CCc1cnccn1)=O C#Cc1c[nH]nc1C(=O)NC1CCN(C(=O)CCN2CCC(O)CC2)C1 C(=O)(C1=CCCCC1C)NCC(N1CC(CC)C(NC(=O)OC(C)(C)C)C1)=O c1(OC)cccc(CNC23CCC(C(=O)NCC4CNC(=O)C4)(CC2)C3)c1F N1(C(C(C)OCC(F)(F)F)=O)CCC(N(C(=O)C=Cc2ccsc2)CCO)C1 CCN=c1cc(C(N2CCC2CNC(c2nn(CC3CC3)cc2Cl)=O)=O)cc[nH]1 Cc1c(F)cc(C(N2CCOCC2CN(C)Cc2ccc(Br)cn2)=O)c(F)c1F N1(C(C2CN(C)C(=O)N2)=O)CCCC2CN(C(=O)CCc3nccs3)CCC12 C12(CCCCC1)C(=O)N(CC(=O)OC)C2.c1(C(=O)NC2CC2)cn(CCO)nn1 C(=O)(CCCCN(C1CCC1)C)NC(CC)CNC(C)=O.C1C(=O)N1 c1(OC)ncc(S(=O)(=O)NC(c2ccc(N3CCNC(=O)C3)cc2)=O)s1 C(=O)(CCC(=O)NC1CC(NC(=O)CCC(=O)c2cc(Br)cs2)C1)N(C)C C1(CNC(=O)C(C)(C2CC2)OC)(OC)CCCN(C(c2cc(=O)n(C)o2)=O)C1 C1(OC)(CNC(C2C(C)C2C)=O)CCN(C(c2nonc2C(C)C)=O)C1 C=CCCC(C(=O)NCC(C)(C)C=C)NC(=O)CCCOC N1(C(C(C)c2cc[nH]n2)=O)CCC(C2CN(C(=O)COC3CCOCC3)C2)CC1 N1(C(C2(C)CCC(O)CC2)=O)CC(NC(=O)CC2(O)CCOCC2)CC12CCC2 C1(CC(=O)NCC(C2CCC2)NC(C2OCCN(CC)C2)=O)CCS(=O)(=O)CC1 C1(C)(CC=CC(=O)N(C(C)C(=O)NCCN2CCCC2)C)CCCOC1 Cc1cc(C)n2nc(C(N3CC(CO)(NC(=O)CCCC(F)(F)F)C3)=O)cc2n1 N1(C(C(C)OCCCCCC)=O)CCC2CCC(C1)N2C(c1nnc(S)n1C)=O c1(C(N2CCC(O)(C(C)C)C2)=O)ccc2ccsc2c1.C12(CC1)C(=O)N2 CCC(F)(C(=O)OC)C(=O)N(CC(C)CNC(c1cc(C)c(C)cn1)=O)C C#CCC(C)(C(=O)NC1(CO)CC2(CCC2)C1)NC(=O)CCC(F)(F)F CC(C)S(=O)(=O)CC(=O)N1CCCC1C(=O)NCCCNC(=O)C(C1CC1)C1CC1 C1(O)(CN(C)C(C2COCOC2)=O)CN(C(=O)CCNC(C2CCC2)=O)C1 C1(C(N(C2CCCN(C(CC3CCC(C)CC3)=O)C2)C)=O)CC(S(C)(=O)=O)C1 C(N=c1[nH]c(=NCCc2cc[nH]n2)c2ncccc2[nH]1)C1CCCCC12CCC2 C1(NC(C2C(C3C(C)C3)C2)=O)C2CCC1CN(C(=O)Cc1cnn(C)c1)C2 c1(CC(=O)NCC(CC=C)N(C(CC=C)=O)CC)cc(Br)ccc1S(C)(=O)=O C1(C(N(C)C)=O)C=CCN1C(C1CCN(C(=O)CSC(C)(C)C)C1)=O c1(CC(=O)NCCCN(C(C=CC=CC)=O)CCO)cc(C(F)(F)F)n(C)n1 N1(C(=O)NCC(c2cccc(F)n2)C)CCc2cccc(Cl)c2C1C N1(C(C(COC)O)=O)CC(NC(C2(C3CCC3)CC2)=O)CC2(CCC2)C1 C1(C(C)C)N(C(=O)C(C)(F)F)CC12CCN(C(=O)CN1CC(=O)N(C)C1=O)CC2 c1(C(N2CCC(Cc3ccc(OC)cc3)C2)=O)cc(N)ccc1C Cc1nnsc1C(=O)NCCCOCCN(C)C(C1CCCN1C(C)C)=O c1(N(C2CC2)C2CC2)cc2c(N(CC(N)=O)CC(N)=O)c(c1)CCC2 c1(C(N(CCCNC(C(C)(C)OC)=O)C(C)C)=O)ccc2nc(C)c(=O)n(C)c2c1 C1(CNC(c2n(C(C)(C)C)nnn2)c2cn(CC3CC3)nn2)CC2(CC2)C(=O)O1 C1(NC(C2CCCCS2)=O)C2CCN(C(=O)Cn3cnc(C(F)(F)F)n3)C12 C1(CC)CN(C(=O)C(C)COC)CCC1NC(=O)Cc1conc1C C1(NC(C2OCCN(CC)C2)=O)CN(C(=O)CCOCC(C)(C)C)CC1C1CC1 c1(CC(N2CCC(NC(CCC(C)(F)F)=O)C2C2CC2)=O)n[nH]c2c1CCCC2 N1(C(CCC=CC)=O)CC(C(C)(C)C)CC(CNC(C2CC23CC(C)(C)C3)=O)C1 c1(CNC(C2(C)CC(=C)C2)=O)cccc(CN(C)C(C2CC2[N+](=O)[O-])=O)c1 C(=O)(C1=CCC(C)(C)CC1)NCc1occ(C(N2C(C(C)O)COCC2)=O)c1 c1(C(N2C3C(NC(COC)=O)CC(C3)C2)=O)cc2n(n1)CC(F)C2 C(=O)(C(=O)N=S(C)(C)=O)NC1CC(OC)CN(C(c2ccc3c(c2)NCC3)=O)C1 C12CC3(C1)CN(C3)C(=O)N(CC(C)(C)C)C2=O.c1(CC)ccc(Cl)c(Cl)c1 C(=O)(C(CC(C)(C)C)OC)N1CCC(N(CCC)C(C2CCC3CC2CO3)=O)C1 Cc1ccc(C=CC(=O)N(C2CCC(NC(C3(C)CCC3)=O)C2)C)cc1 c1(C(N2CC3CC(NC(CC(CCC)C)=O)C3C2)=O)ccc(Cl)c(F)c1F C12(CNC(C3C(C(C)(C)C)C3)=O)CCCC1N(C(c1cccc(F)c1Cl)=O)CC2 c1(CC)oc(C(=O)NCCC(C)N(C(=O)CC2CC3(CC3)CO2)C)cc1C C1(NC(Cc2c(Cl)cc(C)s2)=O)CC2CC(NC(C3(C)CCSCC3)=O)CC12 Cc1cc(=O)c(C(=O)NC2CN(C(=O)CCC3CCCCO3)CCC2F)cn1C CC1C(=O)N(CC(=O)NC2(CNC(c3csc(=N)[nH]3)=O)CCOC2)C(=O)C1C CC1CCC(C)N1CCNC(=O)Cn1cc(CNC(c2coc(Cl)n2)=O)nn1 Cc1cc(F)cc(C(=O)NCC2(F)CCN(C(=O)CN3CCCNC3=O)C2)c1N c1(CNC2C(CC=C)CCC2)cc2ccccc2s1 N1(C(=O)Nc2ccoc2I)CCN(c2ncccc2Cl)CC1 c1(COC)cc(C)n(-c2ccc(NC(=O)CC(C)c3cnn(C)c3)cc2)n1 N1(C(C(=O)NCc2ccc(Br)cc2)C2CCCC2)CCC(O)(C(Cl)(Cl)Cl)CC1 C(=O)(CCCCC(C)(C)OC)N(C1CCN(C(=O)CN2CCOC2=O)CC1)CC C#CCCCCC(=O)NC(CCN(C)C)C(=O)NCC1CCC(=O)O1 Cc1nc(CCC(=O)N2CCC2CNC(=O)C(C)(C)CN(C)C)oc1C C1(CNC(C2(C(C)C)CC2)=O)C=CCN1C(=O)C(C)CO Cc1cccn(CC(=O)NC2CCC(N(C(=O)C=CC3CC3)C)CC2)c1=O C1(C#N)(C(N2CC(O)(CNC(CCCc3cc(C)no3)=O)C2)=O)CCCCC1 C(C(C)(C)CC(C)O)NC(C1CC(O)(CNC(C=CC)=O)C1)=O C1(C(=O)O)CCCOCC1.C12CC(n3cc(CC4(O)CCC4)nn3)(C1)NC2=O C1(CNC(c2ccc(CC(C)C)s2)=O)CN(C(c2nnc(S)n2C)=O)CCC1C C1(NC(C(CC)COC)=O)CC2CCC(C1)N2C(=O)CN1CSCCSC1 C1(NC(=O)CCCSc2ccccc2F)CN(C(c2cccn2CO)=O)CC1F N1(C(CCC(=O)Nc2nccs2)=O)CC2(C1)CN(C(C1CCCCO1)=O)CCO2 Cc1cc(C2CCCN2C(=O)Nc2cccc(F)n2)cc(C)c1 C1(CC)CCCC12CCN(CC(=O)NC(C)CCCC(C)C)CC2 C1(NC(CN(CC(C)C)C)=O)CCN(C(=O)COCCO)C(C)C1 c1(CC(=O)NC(CCNC(c2c(C)nc(C)[nH]2)=O)C)ccccc1S(C)=O N1(C(C2=CCN(C(C(C)S(N)(=O)=O)=O)C2)=O)CC2(CCC2)OCC1C C12(CCN(C(C3CC(OC)C3)=O)C3CC3)CCC1CN(C(=O)C=CC(C)C)C2 N1(C(C2C(CC)C2)=O)CCCC2(CNC(=O)CCCc3nc(C)no3)CCCC12 C12(C(=O)NCC(c3ccccc3)NC(C(CC)OC)=O)CCC(O)(CC1)CC2 C1(NC(CCOCC)=O)CN(C(c2csc(=N)[nH]2)=O)CC1CC C1(NC(Cn2ccc(C)n2)=O)CC2CCC1CC2NC(c1nc[nH]c1C(F)(F)F)=O C12CCC3(CCC3)C1NC2=O.c1(CNC(c2nnn(C)n2)=O)ccc(Cl)c(Cl)c1 C1(C)(CC)CCC(NC(=NCCc2cccs2)NCC(F)(F)Cl)CC1 c1(CCNC(C2CCCC(NCc3ccc(F)cc3)C2)=O)ccc2c[nH]nc2c1 CC(C)C(CC1CCCC1)C(=O)NC(CCN(C(=O)C(C)N1CCC1)C)C(C)C c1(C(=O)NC(CNC(C2=CC(C)(C)C2)=O)C2CC2)cc(F)cc(Br)c1O C1(CC(=O)N(CC=C)CCC)CCN(C(C2(CC=C)CCCCC2)=O)CC1 N1(C(C(F)=CCC)=O)CC2C3CCC(C2C1)N(C(c1cc(Cl)c(O)cc1C)=O)C3 c1(C(=O)NCCCNC(Cn2c(C)c(Br)cn2)=O)cnc2[nH]ncc2c1 Cc1cc(C)c(C(N2CC(C(C)NC(c3ncccc3C)=O)C2)=O)o1 C(=O)(CC(C)(C)O)NC(C(=O)NC1C(C)CCC1)c1ccoc1 c1(NCC2(CO)C(C)(C)C2)ccc(S(=O)(=O)NCC(c2cccc(F)c2)O)cc1Cl C1(O)(C(C)NC(Cc2c(C)nc[nH]2)=O)CCN(C(c2ccc(CO)cn2)=O)C1 c1(C(=O)NC(C(=O)OC)(C)C(F)(F)F)cc(Br)c2nccnc2c1 CC1CC2CCC(C(=O)NCCN(C(=O)CCCN(C)C)C3CC3)CN2C1 c1(C(=O)NCC2CCCCN2C(c2cccs2)=O)cc(Br)ccc1O C1(CCOC)(C(N2CCC(N(C(C)=O)CC)C2)=O)CCCCC1.c1(C)nnc(C)s1 N1(C(C)=O)CCCC1C(=O)NCC(C)C(C)C.C12(CCC1)CCOC2=O N1(C(c2n[nH]c(C)c2C)=O)CC(C)(C)OCC1CNC(C1(S(C)(=O)=O)CCC1)=O C1(CC#C)(C(=O)NCCC2CCCC(C)C2)CCN(C(C2CCCCCC2)=O)C1 C(c1ncco1)=CC(=O)NC1C(NC(CC2(C(N)=O)CCC2)=O)CC1 C1(N(C(C2CCN(C)C2=O)=O)C)CCCN(C(c2cncn2C)=O)CC1 CC(CN(C(=O)C(c1ccn(C)c1)C)C)C(=O)NOCC1CCOC1 N1(C(C(C)C)=O)CCC(C(N2CCC(O)C(C)C2)=O)C(F)C1 Cc1ccnc(O)c1C(=O)NC1CCC1NC(C1(c2ccccc2)CC1)=O Cc1cc(C)c(C(=O)NCC2CCCN(C(c3cccc(C)c3N)=O)C2)c(C)n1 CC(CCN=c1cccc(S(=O)(=O)NCC2CC(S(C)(=O)=O)C2)[nH]1)S(C)=O C(C)(C)(CN(C(=O)Cn1cnnc1)CCN(C(=O)CN(CC(=O)NCCC(C)C)C)C)N N1(C(Cn2ccc(C(N)=O)n2)=O)CCCC(c2nnc(Br)s2)C1 c1(C(OC)OC)ccc(C(=O)NCC(C(C)(C)C)NC(=O)CCSC(C)=O)cc1 Cc1cc(C(C)C)ccc1C(N1CCC(NC(C2CC3(CSC3)C2)=O)C(C)C1)=O c1(NC(C)=O)cc(C(=O)NCC2CCCC(NC(c3cocn3)=O)C2)ccn1 c1(N(C)Cc2n[nH]c(C)n2)nc(=NC(C)c2nnnn2C)nc(N2CCCCC2)[nH]1 c1(NC(C(C(C)C)=O)=O)cccn2nnnc12 C1(C)(NC(C(C)SN2CCOC2=O)=O)CCCN(C(=O)C(Cl)=CCl)C1 C(CC)(CCC(=O)NCC1CC=CC1)NC(C(C)SCCCC)=O CP(C)(=O)c1ccccc1C(N1CC(CO)(NC(=O)CC2CC23CC3)C1)=O CC1(C2CCC2)CN(C(=O)C(C2(C)CC2)NC(=O)CC2CCCC23CC3)C1 S(=O)(=O)(c1cnccc1N(CC(c1ccc(C)s1)O)C)NCc1ncc(CC)s1 C(CCCCC(=O)N1CCOCC1CNC(C1(CN(C)C)CC1)=O)OC CCC(C)C(=O)C(=O)N1CC(OCCC(=O)NCC(C)(O)CC(C)C)C1 [N-]=[N+]=NC1(C(N2CCCC2(C)C2CC2)=O)CCN(C(=O)C#CC2CCC2)C1 CC1CC=C(C(=O)NC2(C3CC3)CCN(C(C3CC(C)(C)CCO3)=O)C2)CC1 C(CCNC(c1ccoc1Cl)=O)(C(C)C)NC(CC=CCC)=O S(=O)(=O)(c1cccc(CO)c1)NC12CC(NC(c3c(OC)cc(C)cc3)=O)(C1)C2 c1(OC)cc(C(=O)NCC2CCCC2NC(C23CCC2CC3)=O)ccn1 Cc1ccc(C=CC(=O)NCCC2CCN(Cc3ccn(C)c3)C2)cc1 c1(C(=O)NC(CC)CN(C(=O)CCC2CCCO2)C)ccn(C)c1C c1(C(=O)NCC(CNC(C(N2CCNC2=O)C)=O)(C)O)cn(C)[nH]c1=N C1(C(=O)NCC23CC(CNC(C4C(C)(C)C4)=O)(OC2)C3)CCc2nccn2CC1 N1(C(C(=O)NCCN2CC(C)C(C)C2)=O)CCC2(CC1)CN(C)CCO2 O=C(C(CO)C(F)(F)F)NCC1CCCCN(C(C2(C(F)F)CCCCC2)=O)C1 c1(CC(N2CCC(C(N(CC#N)CC#N)=O)CC2)=O)ccc2[nH]ccc2c1 C1(C(=O)NC(C)CN2CCOCC2)CSCCN1C(=O)Cc1cn[nH]c1 c1(C(C)C)conc1CC(=O)NC1CCC(NC(=O)C(C)C2CCCC2)C1 N1(C(COc2ccc(C)cc2)=O)CC2OCCN(C(c3coc(Cl)c3)=O)C2C1 c1(CC2NCCN(CC)C2)cc(OC(F)F)ccc1Cl c1(C(=O)NCC(CC=C)NC(=O)Cc2nnc(C)o2)cncc(S(C)(=O)=O)c1 N1(C(CCN2CCC(C)CC2)=O)CCC(C2CCN(C(C34CC(C)(C3)C4)=O)C2)C1 CC1(CC(N2CCC(O)(CNC(C3CCCN3C(N)=O)=O)C2)=O)CCS(=O)(=O)N1 Cc1nc(C(N2CCN(C3CCN(C(c4cnc(S)nc4)=O)C3)CC2)=O)cn1C C1(NC(COCCOCC#C)=O)CCCN(CCC2CCN(C)CC2)CC1 c1(C(=O)NCCC(=C)CNC(=O)COCCCF)cnc(Oc2ccccc2)cn1 c1(CC)c(C(N2CCCC(NC(=O)C=Cc3ccccn3)C2)=O)cccc1F C(=O)(CCC=CBr)N1C(CN(C(CC(=O)NCC#C)=O)CC)CCC1 C1(C(=O)NCCCSC)C2CCC(CC2(F)F)N1C(C1CCCC1C)=O N1(C(CCC(CC)NC(c2cc(Cl)ns2)=O)=O)CC2CCCC(N(C)C)C2C1 N1(C(CNC(CNC(C)=O)=O)=O)CCC2CN(C(C3CCC4CC4CC3)=O)C2C1 N1(c2nc(CC)nc(C)c2)CCC2(NC(c3nc(C)c(C)nc3C)=O)CCCC12 C1(CNC(=O)CSc2cccc[n+]2[O-])CC2CCC1N(C(c1cc[nH]n1)=O)C2 N1(C(c2c(NC)nccc2)=O)C(C)C2CC1C2NC(=O)COc1ccn(C)n1 O=C(C1=CCCCC1)NC12CC(C1)N(C(c1ccc(F)c(Br)c1)=O)C2 C12(Nc3cc(C)c(Cl)cc3)CCCC1CCN2C(=O)C(=O)NCCN(C)C c1(CNC(C2(CNC(=O)CCc3ccsc3)CCOCC2)=O)ccc(F)cc1O c1(C(N2CC(NC(C3(SC)CC3)=O)C3C(C2)C3)=O)c(C)cc([N+](=O)[O-])cc1C C(C(C(=O)N1CCC(O)(CNC(C23CCC(CC2)CC3)=O)C1)C(F)(F)F)OC C(=O)(C(CNC(c1cnn[nH]1)=O)C(C)(C)C)N(c1ccc(O)cc1)CC#C C12(C(=O)NCC3CN(C(c4ccc(Cl)o4)=O)CC3O)C3C4C1C1C2C3C41CO N1(C(C2CCSCC2)=O)CC(N=c2nc(Cl)c3c([nH]2)COC3)C2(CCC2)C1 c1(C(=O)NC(C(=O)OCC)C2CC2)cc(C(=O)O)cc(Br)c1 CC1(C)CC(C(=O)NC2CCC(NC(=O)CCc3cc[nH]n3)CC2)C1C(F)(F)F c1(C(N2CCC(C)C2CNC(c2ccnnc2Cl)=O)=O)ccc(F)cc1N N1(C(C2CC3CC2N(CCc2ccccc2)C3)=O)CCCC(C2CC2)CC1 CC1=C(C(=O)N2CCC(C)(C)C2CNC(c2cccc(C(C)C)c2)=O)CCCO1 c1(C(N2CC(OCCC(=O)N(C3CCSC3)C)C2)=O)csc2cncn12 c1(C(=O)NCC(C(N2CC(CC)OCC2)=O)O)cnn2c1OCC2 N1(C(COC)=O)CCC2CN(C(c3cccc(OCC=C(C)C)c3)=O)CCC2C1 N1(C(COCCC=C)=O)CC2CC(C(=O)NC(CCF)C(=O)OC)C(C2)C1 N1(C(c2cc(CC)sc2)=O)CC2CC(C(=O)N(CCO)CC)CC2C1 N1(C(=O)Cc2cn(Cc3ccc(Br)cc3)nn2)CC(O)C2(CCC2)C1 Cc1cc(C)c(C=CC(=O)NCC2CCCC2NC(=O)CSS(C)(=O)=O)c(C)c1 c1(C(=O)NC(CCNC(C2(C=C)CCC2)=O)C)cnc2cc(C)nn2c1 N1(C(C=C2CCC(C)C2)=O)CC2C(NC(c3ccc(CN(C)C)o3)=O)C2C1 C(=O)(CS(=O)c1cccc2nsnc12)NCC(C)NC(c1coc(C(F)F)n1)=O C=CCCC(C)(C)C(=O)NCC(C)CN(C(=O)CCCC(OC)OC)C N1(C(c2cnc(COC)s2)=O)CCC(C)C(CNC(c2cnn(CCO)c2)=O)C1 C(C)(CCCCNC(C1(CC2CC2)CC1)=O)NC(c1ccc(C(C)(C)C)[nH]1)=O C#Cc1cnc(C(=O)NCC(O)CCNS(=O)(=O)CCCC(=O)OC)c(C)c1 CCCCC#CC(C)(C)NC(c1ccc(C(=O)OC)[nH]1)=O C1(CNC(C2C3CC2N(C(=O)CC2CC4(CC4)C2)C3)=O)CC12CCOC2 c1(OC)ccn2ncc(C(N3CC(O)(CNC(=O)CC4C=CCCC4)C3)=O)c2c1 c1(N(C(=O)NC(c2ncc(C)[nH]2)CC)CC)cc(Cl)cc(Cl)c1Br CCCCC(F)(F)C(=O)NCC1(F)CC(CNC(c2ccnn2COC)=O)C1 c1(C(=O)NCC(C(C)C)NC(=O)C(F)(F)C(C)O)cc2cc(Cl)ncc2[nH]1 N1(CCCC(=O)NCCn2cc(C3CCC(OCCO)CC3)nn2)CCOCC1=O C1(=CCNC(CCc2scc(C)n2)=O)CCN(C(=O)Cc2occc2C)CC1 C1(C(=O)N(C(C(=O)NCCOCCOCC)C2CCCC2)C2CC2)CCC(F)(F)C1 c1(CC(C(=O)N(C2CN(C(COCC)=O)C2)CC)O)ccc(C(F)(F)F)cc1 c1(OCC(=O)NCC2N(C(C3CN(CC)C(=O)C3)=O)CC=C2)cc(C)cc(C)c1 c1(C(=O)NCC2CC(NC(C3C(OC)CCC3)=O)C2)ccc(Cl)c(O)c1 C(=O)(CS(=O)(=O)C1CC1)NCCCC1(CNC(C(C(C)O)C)=O)CC1 N1(C(C=C(C)C)=O)CC(CNC(=O)C(c2ccc(F)c(Cl)c2)(F)F)C2(CC2)C1 c1(C(N2CC(O)(CNC(C(C)C)=O)C2)=O)ccc(CNC(=O)C(C)O)cc1 c1(C(N2CCC(NC(=O)COC(CC)CC)C2)=O)cc(F)ccc1NC C(=O)(Nn1cccn1)c1ccc(NC(c2ccc(C#C)o2)=O)o1 C1(CNC(=O)CCCC2CC2)CC2(CC2)CN1C(=O)CCc1ccsc1 c1(SC)ccccc1C(=O)NC1CC2(C1)CC2NC(C1CCCCO1)=O N1(C(c2ncn(C(C)(C)C)c2)=O)CC2CCC1CN2C(c1cnn(C2CC2)n1)=O C(=O)(CC(C)CC(C)C)NC1C(SC)CN(C(c2ccc(C)nc2)=O)C1 c1(CC(=O)NC(CC)CN(C(C2CC2C(C)C)=O)CC)cncn1C1CC1 N1(C(C(C)(CO)NC(c2ccnc(C)n2)=O)=O)CCOC(C2CC2)CC1 N1(C(CSCCC#N)=O)CCN(C(c2nscc2Br)=O)CC1.C12CC1C2 N1(C(C2C(C(F)(F)F)CC(=O)N2)=O)CCCC(c2ccc(C(=O)NC)cc2)C1 CCCS(=O)(=O)CC(=O)N(C1CCCN(C(c2ccc(NC(C)=O)cc2)=O)C1)C c1(C2(NC(c3ocnc3CC3CC3)=O)CC2)ccc(Br)cn1 c1(-c2c(C(N(C)CC3COCCO3)=O)cccc2)cc(Cl)c(O)c(Cl)c1 N1(C(C(OCC)OCC)=O)CCCOC(CNC(C2(CCNC)CC2(F)F)=O)C1 Cc1[nH]nc(C(=O)N(C(C)C(=O)NCc2nnn(C)n2)C)c1C c1(C(C(N2CCC(OC)(CNC(=O)CNC(C)=O)C2)=O)(C)C)cccc(C#N)c1 c1(CN(C(C2(F)CN(C(=O)CNC(=O)OC(C)(C)C)C2)=O)CC)ccc(OC)nc1 C(=O)(C(F)(F)C(C)(C)O)NCC1C(CC)CN(C(=O)C(=O)NCC2CC2)CC1 C(=O)(C(C)(C)CCC(=O)NC1CCC(C)N(C(=O)COC(F)F)C1)OCC c1(C(=O)NCC(C)(CO)NC(CC(C)N(C)C)=O)cncc(OC(F)F)c1.C1CO1 Cc1ccc2c(c1)CC(C(=O)NCC(C1CC1)NC(c1sccc1C1CC1)=O)S2 C12(NC(C3N(C(c4cccc(CC(C)C)c4)=O)CC3)=O)CCCC1OCC2 c1(C(=O)NCC2C(NC(C3(N)CCC3)=O)C2)cocc1C.CCSCC C1(C)(C(=O)NC2CCC(N(C)C(c3ccnc(OC(F)F)c3)=O)C2)CCCCCC1 N1(CC(=O)NC(=O)NC)C(CNC(c2cn(CC(C)C)nn2)=O)CC2COCC12 C12(C(=O)OC)CCC(CN(C(=O)C(C(C)C)Nc3cccc(Cl)c3)C1)C2 CC(=O)CCCCC(=O)N1CCCC1CCC(N1CCC(O)C1(C)C)=O N1(C(c2cc(C)sc2C)=O)C2CCC1CN(C(C13CC(CN1C1CC1)C3)=O)C2 C(C(=O)Nc1ccccc1)(C(C)(C)C)NCc1nc(C#C)sc1 c1(OC)cccc(C(=O)NC2(CCNC(=O)CC(C)C3CCCO3)CCC2)c1 C=CC1(CC(=O)NC2CC(N(C)C(c3cnccc3C)=O)C2)CCCCC1 N1(C(C(C)n2ccnc2)=O)CC2COCC(C1)N2C(c1cc(Br)no1)=O N#CC1CCN(C(=O)C(N)c2cc[nH]n2)C1.c1(C2=CN2)ccc(N2CCCC2=O)cc1 CCC(CCCC(=O)N1CC2CC(C1)N(C)C2)NC(=O)C(F)n1ccnc1 C1(CNC(CN(C(C)C)C)=O)CC2(CCN(C(=O)CC3CCC4CC4C3)C2)CO1 c1(C(N2C3CCC2C(F)C(NC(=O)CC2CC2)C3)=O)ccnc2c(F)cccc12 c1(NC(C2CCN(N3CC(Cc4n[nH]c(C)c4C)C3)C2)=O)[nH]nc2ncccc12 C(CNC(=O)C(C)c1ccsc1)(C(=O)N(C1CC1)Cc1ncccn1)OC C1(C(N(CC(C)NC(c2ccc(CC=C(C)C)cc2)=O)C)=O)CC(S(C)(=O)=O)C1 N1(C(CC2N(C)CCOC2)=O)CCN(C(=O)CSC(F)(F)F)CC(CO)C1 c1(C(N2CCC(CN(C(C3C(COC)CC3)=O)C)CC2)=O)cncc2[nH]ccc12 CCCCCCCC(=O)N1CC(C(=O)NCCC2(OC)CCC2)C(C2CC2)C1 Cc1[nH]nc2ccc(C(N3CCOC(CNC(=O)CC4C=CCC4)C3)=O)c(Cl)c12 Cc1[nH]nc(C(C)C)c1NC(C1CCC1c1cccc(C(=O)O)c1)=O c1(C(C(=O)NCC(=C)C)N(C(CC2CC2)C(=O)OC)C)sccc1Br C=CCN=c1[nH]cc(C(N2CCC(O)C(NC(c3scc(C)c3Cl)=O)C2)=O)s1 CCCC(O)CC(=O)N(C1CCN(C(=O)C(CC)CCN(C)C)CC1)CCO c1(C(=O)NCC2(COC)CN(C(=O)CCCCc3ccccc3)C2)cc(C#N)no1 c1(C(=O)NCC2CN(C(c3ccc(OCCC)cc3)=O)CC2C)cccn(C)c1=O C(CCC(C)C)(C(=O)NC(C)CC1(O)CCC1)NC(C1CC(CC)C1)=O C(CCCCNC(=O)Cc1nnc(O)s1)N(C(C1(CC(C)C)COC1)=O)C c1(OC)cc(C(=O)NC2CCC2CNC(=O)C(C)Sc2ccccn2)on1 N1(CCC(=O)NC(CC)CNC(=O)CC(C)(C)C)c2ccccc2CCC1C N1(C(c2cc(C)nnc2C)C(=O)NC2COC2)CC(C)(C)CCC1C Cc1cnccc1C(C)C(=O)NC1CC(C)(NC(C2CCC(C)CC2)=O)C1 N(C(=NCCCCl)NC1CC12CC2(F)F)Cc1cccc(N(C)CC)c1 c1(SCC(=O)N(CC)CC2CCCC(C)C2)cc(Br)ccc1F C1(CNC(CN(CC#C)C(c2cc(C#N)cs2)=O)=O)COCC(=O)N1C N1(c2n(CCC=C)c(C3CCOC3)nn2)CCN(C2CCOCC2)C(=O)C1 N1(C(c2c(CC#N)cccc2)=O)CCCC(F)(CNC(=O)CN2CC3CC3C2)C1 N12CCc3nc(ncc3CC1)NC(CC(C)(C)C)C2=O.c1(C(=O)OC)cccs1 N1(C(c2ccc(CCC)[nH]2)=O)CCCC(O)(CNC(=O)Cc2cn(C)nc2C)C1 c1(NC(CN(C(CCC#C)=O)C2CC(C#N)C2)=O)cc(CO)cc(F)c1 c1(CNC2C(C(N=c3cc(C)n(C)[nH]3)=O)C2)ccc2cccc(O)c2n1 C1(NC(Cn2cc(C)c(C(F)(F)F)n2)=O)CN(C(C2CCC2(C)C)=O)CCC1C C(=O)CC1=CSC2=NCCN12.N#CCS(=O)(=O)NCCC1CCCNC1 Cc1cn2c(n1)CCC(C(=O)NCC(C(C)C(C)C)NC(=O)Cc1ccsn1)C2 CC(C)C(CNC(=O)C(C)OCC1CC1)NC(c1cc(Cl)cs1)=O Cc1cc2n[nH]cc2cc1C(=O)N(CC(C)O)CCNC(C1CS(=O)(=O)C1)=O c1(CN2CCN(CC(=O)Nc3cccc(OCOC)c3)CC2)ccc(O)c(O)c1O c1(C(N2CCC3CCN(C(C(=O)NC(C)C)=O)CC32)=O)cccc2nc(S)oc12 C1(OC)CC(CCNC(=O)Cc2csc(Cl)c2)N(C(=O)C(C)OCCC(C)C)C1 C(=O)(C1=NNC(=O)C1)N1CC(C(=O)NC2CCC(C(N)=O)C2)(SC)C1 c1(C(=O)NC2C(NC(Cc3c(C)nc[nH]3)=O)CCOC2)ccc(P(C)(C)=O)s1 c1(C(=O)NC23COC(CNC(C4CCCSC4)=O)(C2)C3)cc(F)c(F)cc1F N#Cc1ccncc1C(=O)NC(C(=O)NOCc1nc[nH]n1)c1cccs1 C1(CNC(c2snc(C)c2N)=O)CC2(C1)CN(C(C1(C)CCNC1=O)=O)C2 c1(SC(C(=O)NCC(C2CCC(C)CC2)(C)O)C)ccc(C#N)cc1 C(=O)(C(F)C(F)(F)F)Nc1cccc(C(=O)NCC2CCC(OC(F)(F)F)C2)c1F C1(C(=O)NCC(C)(C)CNC(=O)CC2CCOC2=O)(OC)CCS(=O)(=O)C1 C1(NC(CCSCCCC)=O)CC2CC1CN(C(c1ccc(COC)cc1)=O)C2 c1(OC)ccc(CNC(C2CC2NC(=O)CN2CCC(O)CC2)=O)c(OC)c1 CC1C(C)N(C(c2cc(C(F)(F)F)nn2C)=O)CCN1C(=O)CCCCC1CC1 C(=O)(C(CC(C)C)ONC(c1c[nH]c(C#N)c1C)=O)NC(COC)C C12(CC(=O)N(C3CCCC34CC4)C)CCC1CN(C(=O)C(C)(C)C1(O)CCC1)C2 c1(C(N(C)CC2CCCN2C(=O)C=CCO)=O)ccc2cc(Cl)ccc2c1 C1(N(C)C(C2(C)CC3(CCC3)C2)=O)CN(C(=O)Cn2[nH]cnc2=N)CC12CC2 C(CC(C)C)(C(=O)N1CCN(C(c2nc(C)n(C)c2C)=O)CC1C(F)F)OC C=CC(C)(O)C(=O)NN(C(=O)CCOC(C)C)C.C12CCC(CC1)CC2 O=C(C#CC1(C(F)(F)F)CC1)NCC1CC(NC(C2CCCCC2F)=O)C1 C(=O)(C1CCC(=O)c2cccn21)NC1CCCN(C(c2c(C)scc2)=O)C1 C(C)(C)(CCC(=O)NC(C)(C(=O)NCC1NC(=O)NC1=O)C1CCC1)OC N1(C(Cc2ccc(C)cc2)=O)C(CC(=O)NCC2CNC(=O)O2)C2CCCC12 C(CCCCC(=O)NCC1CC(C)N(C(=O)CN2CC(C)C2)C1)NC(C)=O C(=O)(CC(O)CC(C)(C)C)NC(CNC(c1n(CCC)ccc1)=O)(CC)CC c1(CC)cc(C(N2CCCC2CC(=O)NCC2(O)CN(C)C2)=O)c(C)o1 N1(C(c2nc(C(C)OC)sc2)=O)CCN(C(=O)C=C(C)Cl)CC1C(F)F c1(C(=O)NC2(CNC(C3(F)CCCC3)=O)CC2)n[nH]c2ccc(F)cc12 C1(CC)CN(C(=O)C(C(C)C)NC(c2ccn(C(C)C)n2)=O)CC1F c1(Nc2cn(C(C)C)nn2)ncccc1S(=O)(=O)N1CC(C)N(C)C(C)C1 N1(C(C2(COC)CCOCC2)=O)CCCC2(C1)CN(C(c1cnsc1C)=O)C2 C1(C)(CC)CC(NC(=O)CSCC(C)C)CN1C(c1cnsc1C)=O O=C(CCCCCn1cnnn1)NCC1(NC(c2ccc(Br)s2)=O)CC1 c1(OC)cc(CN2CCCC(C(=O)Nc3ccccn3)C2)c([N+](=O)[O-])cc1OC n1(CC(=O)NC(C2CN(C(C3CCC4CCC34)=O)C2)C)ccc(O)nc1=O c1(C(=O)OCc2sc(C)c(C(=O)N(C)C)n2)cn2c(n1)SCC2 C(=O)(CC(C)C(F)(F)F)NCCOC1CN(C(C2CCC(CCC)CC2)=O)C1 CCC(CNC(C1CC=CC(SC)C1)=O)C(=O)N(C)CCN(C)CCOC C1(Cn2c(NC(=O)NCc3n(CC)ncn3)ccn2)CCCN(C)C1 N1(C(COC(C)=O)=O)CC2COCC2(C(=O)NCC2CCCN2C)C1 c1(C(N2CCC(CN(C)CCC3NC(=O)NC3=O)CC2)=O)ccc2[nH]ccc2c1 c1(OC)cncc(C=CC(=O)NCCN(C(C2CNC(=O)CC2(C)C)=O)C2CC2)c1 C1(CC(=O)NC(C(C)NC(CSCC)=O)(C)C)CCCNC(=O)C1 Cc1cc(NC(c2cccc(NC(C3OCCC3C(=O)O)=O)c2)=O)ccc1Br c1(C(=O)NC(C(=O)NC2(c3cccs3)CC2)c2ccco2)cnc(O)c(F)c1 c1(OC(=O)CNC(=O)Cc2ccc(Cl)c(F)c2)scc2c1OCCO2 c1(C(C(=O)NC(C2CN(C(C(C#C)(C)C)=O)C2)C)C)ccc2ccccc2c1 C1(N(c2cncc(F)c2)C(=O)Cc2cc(Br)ccc2F)CCC2(CC1)CNC2 N(C1c2ccccc2OC1C(=O)O)CCn1cc(C(CO)O)nn1 C(=O)(CCCC(N)=O)NCC(CO)NC(c1ccc(CSC)cc1)=O N1(C(C(C2(O)CCCC2)NC(=O)CCCn2ccnc2)=O)CCOC2(CCC2)C1 C1(CNC(C2CC2F)=O)CCC2(CC1)CCN(C(c1c[nH]cc(Cl)c1=O)=O)CC2 N1(C(Cc2c(O)ccc(C)c2)=O)CCOC2CCN(C(=O)C(C)C(C)C)CC12 Cc1cc(=NCC23CC2CN(C(c2ccc4nsnc4c2)=O)C3)[nH]c(C2CC2)n1 N1(C(=O)CCC2(O)CCC2)CCC2CN(C(=O)COC3CCCC3)CCC2C1 C#CCC(CC#C)C(=O)NCC12CC(CNC(c3ccncc3F)=O)(CO1)C2 C=C(C)CC(C)C(=O)NC1CCC(C)(NC(=O)CNC(c2csc(=N)[nH]2)=O)CC1 CC(C(O)C(=O)NCCOC1(C)CCCC1)c1ccccc1 c1(NC(C2(NC(CN3CC(C)C3)=O)CCC2)=O)cnc2c(F)ccc(F)c2c1 C1(C(=O)Nc2cn(C(C)C)nc2)CCC2(CC1)CC(NCc1cc(O)n(C)n1)C2 c1(C(N2C(C(=O)Nc3nc(C)c(C#N)nc3)CC2)=O)cc(C)c2ccccc2n1 c1(C(=O)NC(C)C(CO)NC(=O)CN(C2CCSC2)C)nccc(Cl)c1O C1(NC(C(COCC)C)=O)CCC2CN(C(=O)CCOCCCOCC)CC12 Cn1cc(OCC(=O)NC2CCC(NC(=O)Cc3c[nH]nc3O)C2)cn1 Cc1nc(C(F)(F)F)cc(C(N2CC(NC(=O)C(=O)C3CCCC3)C2)=O)n1 C1(NC(c2c(CC)c(C)sc2)=O)CCCN(C(c2ccc(N(C)C)cn2)=O)C1C CC1(C)Cc2cc(C(=O)NC3CCCCN(C(=O)C(F)OC(F)(F)F)C3)sc2C1 c1(CC(=O)N(C2CCN(C(C=C3CCC(C)C3)=O)C2)C)ccc(C(N)=O)nc1 N1(C(C)=O)CCCCC1CC(N1CCC(C)(NC(c2nc[nH]c2C(C)(C)C)=O)C1)=O c1(C(=O)NCCC(C)(C)NC(=O)CC2CCCO2)ccc(Cl)c(C#N)c1 CC1c2cc(F)ccc2CCN1C(C1CCC1(C)C)C(=O)NC1CCOCC1 C12(CC)CC1CN(C(=O)C(C)N(C(=O)Cc1ncccc1C)C1CC1)C2 C1(NC(c2ccc(O)cc2)=O)C2CN(C(=O)CCn3cccc3)CC12 c1(OC)nc(C)ncc1C(=O)NC1(C2CN(C(C3COC(C)C3)=O)C2)CC1 CC(C)C(C)CC(=O)N1CC2CC(C(N3CCCCC(CO)C3)=O)(C2)C1 N1(C(c2ccc(C(C)(C)C)s2)=O)CC(O)CC1CNC(=O)CCC1NC(=O)NC1=O CCCC(C)(C)CC(=O)N1CCOCC(NC(C2CCC3(CCCC3)C2)=O)C1 N1(C(c2cnc(CC(C)C)[nH]2)=O)CC(CNC(C2CC(O)C2)=O)CC12CCC2 CC(C)C(O)CCN=c1[nH]c(=NC(C)C2CSC2)c2ncccc2[nH]1 CCC(C)(CCNC(c1ccsc1OCC)=O)NC(=O)CC1COC(COC)C1 C1(C(C(=O)NCC(CNC(C=CS(C)=O)=O)(C)C)(C)C)CCCCCCC1 C(=O)(C1=CCCCC1C)N(C)CC1N(C(c2cnc(CC(C)C)[nH]2)=O)CCC1 c1(C(=O)NC(CCOC)CNC(=O)C(C)(O)C(C)C)ccc2nn[nH]c2c1 n1(CC(=O)NCCCC2ON=C(C)C2)cc(NC(=O)C(C)N2CC(C)C2)c(C)n1 C(=O)(CC(C)CNC(=O)C(COC)N(C)C)NCC(=O)NCCCC c1(Cc2nc(C(C)OCCOC)n(C3CS(=O)(=O)C3)n2)cccc2cccnc12 CC1(C(=O)NCC(O)CCNC(c2cnc(N)nc2)=O)CC=CCC1 N1(C(C=CC=CC)=O)CC(C)(NC(=O)CC2CCCN2C(C)=O)C1 N1(C(c2ccc(C(N)=O)s2)=O)CCC2CN(C(c3cc4cscc4s3)=O)C2C1 C1(C)(CNC(C2CN(C(C)=O)CC2C)=O)CC2CCC1C2 N1(C(c2cc(C)n(C)c2)=O)CC(C)N(C(c2nnn(C(C)(C)C)n2)=O)CC1C Cn1cnc2cccc(C(N3CCCN(CCNC(C4CC45CC5)=O)CC3)=O)c12 C=C1CC(C)(C(=O)NC2CC(NC(=O)CC(C)SC)C2)C1 c1(CNC)ccccc1C(N1CC(c2ccsc2)CC1C)=O N1(C(c2c(C)nns2)=O)CCN(C(=O)Cc2ccco2)CC1CC(C)(C)C CC1CCOC(C(=O)NCCCN(C2CCCC2)C(c2cnn(C3CC3)c2)=O)C1 C(=O)(C(CCSC)NC(=O)CC1CCCC1)N.CCC(CN1CCCC1)OC c1(-c2ccc(CN3CCC(F)(CO)CC3)s2)ccc2occc2c1 C1(C(=O)NCC2(OCC)CC2)N(C(=O)C(O)CC(C)C)CC12CCCC2 c1(NCCC(=O)N(CCNC(C2CC2c2ccoc2)=O)CC)ccccn1 N1(C(c2n[nH]cc2I)=O)CCC2(CCCN2S(=O)(=O)c2c(Cl)cccc2Cl)CC1 Cn1ncc2c(O)cc(C(N3C4CCC3CN(C(=O)CC3CC3(Cl)Cl)C4)=O)cc12 C1(F)(CNC(c2cc(C)ncn2)=O)CCCN(C(=O)COC2CCCCC2)CC1 C1(C(=O)NCCCN(C(=O)C2=NOCC2)C(C)C)CC2CCCC(C1)C2 c1(C(N2CC(C)CC(NC(Cc3ccc(C)s3)=O)C2)=O)ccc2nc[nH]c2n1 C1(=O)CCCCCn2cc(nn2)CCCN1.c1(C(C(=O)OC)O)ccc(F)cc1 C1(CNC(COCCOC)=O)CN(C(c2cnc(C)nc2O)=O)CC12CC2 c1(OC)cc2[nH]c(C(=O)NC3CCOC4(CCC4)C3)cc2c(Cl)c1OC C(=O)(CC(C(C)C)OCC)NC(CC=C)CNC(C1CC(=O)N(CC(C)C)C1)=O C1(NC(=O)CCF)CCCC(NC(=O)CCn2cc[nH]c(=O)c2=O)CC1 N(C1CCc2c(F)cc(F)cc21)C(=O)NCc1cc2c(s1)CCC2 C1(O)(C(N2CCC(CN(C)CC3CCCO3)CC2)=O)CC2CCC1C2 n1(CCC)cc(Cl)c(C(=O)NCC2(C)CCC(NC(=O)CC(=O)N(C)C)C2)n1 C1(NC(c2nn(C)c(C3CC3)c2)=O)CCN(C(C2(CCF)CC2)=O)CC1CO C1(NC(c2c(CCC)nns2)=O)CC(O)CN(C(c2onc(C)c2C)=O)C1 c1(C(CC)=O)ccccc1NC(C)(CC)CCNC(=O)CCC(C)OC(C)=O C1(C(N(C)CC2(O)CN(C(C(C)OC3CCCCC3)=O)C2)=O)Cc2nccn2C1 c1(OC)c(C(F)(F)F)n[nH]c1Cc1noc(C2(C)CC2)n1 c1(CC(=O)NC2C(CNC(CC(CN(C)C)O)=O)CCCC2)cc(Cl)ccc1O N1(C(c2n(CC)ccn2)=O)CCC(C2CC(NC(=O)CN(C)C3CC3)C2)C1 C(C)(N=c1[nH]c(Cl)nc2[nH]ccc12)C1OCCN(C(C=CC(CC)=CC)=O)C1 C12CC(C)N1CCN(CCOCCO)C2=O.C(=O)(CSCC)NCC=C C1(NC(c2c(CC)occ2)=O)CN(C(=O)Cc2ncn(C)c2C)CC1F N1(C(CCC=CC)=O)CCCC2(C1)CN(C(c1cccc3nc(CO)[nH]c13)=O)C2 C(=O)(C1SCCc2ccccc21)NCCN(C1CCCCC1)C(C1CC(C)(C)C1)=O Cn1nc(C(=O)NC(Cn2cncn2)C(=O)NCCc2cccnc2)cc1C#N N1(C(CCc2cnn(C)n2)=O)CC2CCC(C1)N2C(c1ccc(C2CC2)s1)=O CCC(C)(COC)C(=O)N1CCCC(NC(=O)C=CCN2CCOCC2)CC1 C1(CNC(C=C(C)C)=O)COC(C)(C)CN1C(c1cc(C)c(C)c(F)c1)=O C=CCC(C(=O)NCC(CC(C)C)NC(c1cccc(C(F)F)c1)=O)OC N1(C(C=CCC)=O)CCC(C)C1CNC(C1(CCOC)CC1)=O C=CC(CC)CC(=O)NCc1ccoc1C(N1CCOC(C2(C)CC2)C1)=O FC1(F)CCC2(CC1)CC(NCc1cncc3ccccc13)CO2 C1(NC(c2cn(CCOC)nn2)=O)CC(NC(C2CCC3CCC2O3)=O)C12CCC2 C(=O)(C(CCC1CCC1)N1CCCCC1)NCCCSCC C1(C(N2CCC(C)(NC(c3cnn(CC)c3Br)=O)C2)=O)CC(C)(C)CN1C c1(C(=O)NCc2c(CN(C(C(CC=CC)C)=O)C)cccc2)cn2c(n1)CCC2 c1(CC(=O)NC2C(NC(c3c(CC)noc3C)=O)C2)ccc(OC)c(Br)c1 C1(N(c2cc(SC)ncn2)C)CC2CCC(C1)N2C(C1CCC(=O)N1)=O N1(C(c2cccnn2)=O)CCC(F)(C(N2CCC(O)(CO)C2)=O)CC1 N1(C(C(CCC)N(C)C)=O)CC(CNC(c2ccccc2COC)=O)C(C)(C)C1 C12(NC(CCCC)=O)CC1CN(C(C1CCCC1C(=O)OC)=O)C2 C(CN=c1[nH]nc(O)s1)CCN(C(=O)CCc1nccs1)C.C(CO)O C1(C)(CC)C=C(C(=O)N2CCOCC(NC(=O)CCC3CCCO3)C2)C1 N1(C(CC(COC)C)=O)CCC2(CC1)CC2CNC(=O)CCCCC(N)=O c1(C(=O)NC2CC(C)N(C(=O)Cc3cncn3C)CC2)cncc2n[nH]cc12 C1(C(=O)NCCCOC2CC(NC3CC4(CC4)CO3)C2)(OC)CCC(C)C1 C1(C(=O)NC(CC)CC(=O)OC)CCCCC1(C)NC(=O)C=CC(F)F C(C(C)(C)C(=O)NC1CNC(=O)C1)NC(CC(C)n1cccn1)=O C(=O)(CCCCC(C)(C)OC)N1CC2C(CNC(C(CCCC)F)=O)(CC2)C1.O C1(NC(C2CC3(CCO3)C2)=O)CC2(C1)CC(C(=O)NC1CCCC(O)C1)C2 c1(OC)cc(C(N2CCN(C3CN(C(C4(OC)CCC4)=O)C3)CC2)=O)ccn1 c1(C(=O)NC(C)C(C)C(=O)NCC2Cc3nccn3C2)c[nH]c2ncccc12 c1(C(=O)NC2(CCCNC(C3CCNC(=O)O3)=O)CC2)cnc2c(c1)COC2 c1(C(N(C(C)CNC(C23CC2C3)=O)C)=O)cc(N)ccc1Br C1(C(=O)NCCc2c(C)noc2C)CCN(C(=O)C(C)CCN(C)C)CC1O C(CCCC(C)(C)C(=O)NNC(=O)Cc1ccns1)NC(CC(C(C)C)C)=O CCC(C)(C)CCCC(=O)N1CC2CC2(CNC(=O)CCCc2nncn2C)C1 N1(C(c2cnn(C)c2Cl)=O)CC2OCC(C(N3CCC(C(C)(C)O)C3)=O)C2C1 N1(C(C2CC(CC3CC3)C2)=O)CC2(C(=O)NC3CCCC(O)CC3)CCC1CC2 c1(C(N2CCCN(C(=O)C(F)(F)C3(O)CCCC3)CC2)=O)ccnc2c1CCC2 C(=O)(C(CCC(N)=O)OC)N1CC(CCNC(C2C(C(=O)OCC)C2)=O)C1 C1(N(C(C)(C)C)C(=O)Nc2ccc(Cl)c(I)c2)COC2(CCNCC2)C1 C(=O)(C1CCCc2nc[nH]c21)NC1C2(CC(NC(C(CCC)C(=O)OC)=O)C2)C1 N1(C(C(C2CCCCC2)N(CC=CCl)C)=O)CC2COCC2(C(=O)O)C1 c1(C(=O)NCc2ccc(-c3ccc(Cl)cc3)cc2)c(I)ccc(Br)c1F c1(OC)cc(C(N2CC3CC2CC3NC(=O)CC2(OC)CCC2)=O)cnc1O C1(C(N2C(C#C)CC2)=O)CC12CCN(C(c1noc(C)c1C)=O)C2 N1(C(CSc2nn(C)c(C3CCCO3)c2)=O)CCN(C2CCOCC2)CC1(C)C n1(CC)nccc1CONC(C1C=CC(NC(C2CCC3CC23)=O)C1)=O c1(CN(CCCCCCNC(=O)C(=O)N2CCCC2)C)ccc(S(C)(=O)=O)o1 N1(c2nc(N(CC(CCC)C)C)nc3c2SCC3)CCN(C)c2ccc(Br)cc21 CCC(CCC(=O)NCCC(O)C(=O)OC)NC(=O)C(C1CCOCC1)C N1(C(c2c(CC)ccs2)=O)CCN(C(c2cc(C(F)F)cs2)=O)C(C)CC1C C(=O)(C(C)C(=O)N1CCCC1(C)C(N1CCN(C(C2CCCO2)=O)CC1)=O)OC C1(NC(C(COC(C)C)(C)C)=O)CCC(C)(C)N(C(=O)CN2CC3CC3C2)C1 C1(C(F)(F)F)(C(=O)NCC(CC)CNC(c2cncc(N)c2)=O)CC=CCO1 Cc1ccc2c(c1)C(CCc1nnnn1CCCC(C)(C)CS(C)(=O)=O)C(=O)N2 C(=O)(C#CC1(C)CC1)N(CC(C)N(C)C(c1csc(C2CC2)n1)=O)C C(CCCC(C)NC(=O)C(c1cnn(C)c1)C1CC1)NC(C(COC)C)=O Cc1ccc2c(C(=O)NCC(CC(C)C)NC(=O)Cc3ncc(C)s3)coc2c1 c1(C(N2CCC(C)C(CNC(c3cnc(S)nc3)=O)C2)=O)ccnc2c1CCC2 c1(NC(C(CCCOC)NC(=O)CC2CCCOC2)=O)cccc(N=[N+]=[N-])c1 C1(C(=O)NCC2N(C(CNC(c3c(C)onc3)=O)=O)CCC2C)CC(=O)N(OC)C1 n1(CC(=O)N(C2CCN(C(=O)C(CC)NC(C)=O)C2)CC#C)cc(Br)c(C)n1 CC1=C(C(=O)NCCC(C)NC(=O)Cc2sccc2Br)SCCO1 N1(C(C)=O)CCC2C(CCN2CC(c2cc(Br)ccc2Br)=O)C1 C1(C#CC(=O)NCC(CNC(c2cnc3ccnn3c2)=O)OC)(CC)COC1 N1(C(CCc2cc(C)[nH]n2)=O)CCC(C)(CNC(C2(C)CCCCC2C)=O)CC1 CC(C(=O)NCCCN(C(=O)CN1CCC(=O)NC1=O)CCO)C(C)C(C)(C)C CCCC(C)(O)C(=O)NCCCCCCNC(C1C2C3CCC(C3)C12)=O Cc1nc(C)c(CCC(N2CC(NC(=O)C(=O)NC3CC3)C3(CC3)C2)=O)c(O)n1 c1(OC)ccc(C(=O)N(CC(=O)NC2CCCCCC2F)C2CC2)cc1C c1(C(N(CC(C)NC(c2nn(C(CC)C)c(C)c2)=O)C)=O)c(C)nc2sccn12 c1(C(=O)NCC2CCCN2C(c2ccc(C(F)(F)F)s2)=O)cccc2oncc12 C(c1cnc(O)nc1O)=CC(=O)NCC1(NC(c2c(C)[nH]c(C#N)c2)=O)CCC1 C12(CNC(c3cncc(Cl)c3)=O)CCC(CC1)N2C(C1CC2(C1)CC(O)C2)=O c1(NC(C(C)OCC2(CN)CC3CCCC3C2)=O)cccc2ccccc12 N1(C(c2cc(N(C)C)ncc2)=O)CCC(C2(NC(C3CC3C#N)=O)CC2)C1 C1(NC(C(C)OC)=O)CC2(CCN(C(c3csc(-c4ccoc4)n3)=O)C2)C1 C1(C(=O)NCC(C=C)O)CCN(C(=O)C(C)OC)CC1 N1(C(c2cc(OC)ncc2)=O)CCCN(C(C2CCCCN2C)=O)CC1C c1(C(N2C(C(N3CCN(C=O)CC3)=O)C3CCC2C3)=O)cc2cc(F)ccc2o1 C1(NC(c2c(CC)n[nH]c2)=O)CC(NC(=O)C(CC)n2cncn2)C(O)C1 n1(CC(=O)NC2C(NC(C(C)NC(=O)NC3CC3)=O)C2)cc(Cl)cn1 C1(C(=O)NCCN(c2nc(C)[nH]c3nccc2-3)CCC)CCc2cnc(C)n2C1 c1(CC(=O)NC2C3CCN(C(C(C)c4cccs4)=O)C32)ccc2c[nH]nc2c1 C(=O)(CCCCC(=O)OC)N1C(CNC(c2c(CC)scc2)=O)CCC1 C12=CCN(CC1)CC2.c1(C(=O)NCc2nccs2)cnc(C(F)(F)F)s1 C1(NC(Cn2c(C)cnn2)=O)CN(C(=O)C(C)N2CCCC2)CC1C(F)(F)F c12c(cc(Cl)cc1-c1ccsc1)-c1nc(no1)C1CCN(CC1)CC2=O.CC(=O)NC c1(C(C(N2C(CO)CC(NC(CCCOC)=O)C2)=O)C)nc(F)ccc1Cl C1(C(=O)NC(c2ccccc2)C#C)CSCN1C(c1cnsc1C)=O n1(C(C)C)nccc1C(=O)NCCN(C(=O)C(O)Cc1cnn(C)c1)C1CC1 c1(C(=O)NCC2(N(C)C)CCCC2)ccc(NC(C2(C)CC=CCC2)=O)nn1 c1(C(=O)NCC2N(C(CC3C(C)C3)=O)CCC2)ccc(NS(C)(=O)=O)nc1 CCCCC(CC)C(=O)NCC1CCCN1C(c1ccc(O)c(N)n1)=O CC1(C)CN(C(c2cc(N)cc(F)c2)=O)C(CNC(C2CC2C2CCC2)=O)CO1 C1(NC(C)=O)C=CC(C(=O)NC2(C(=O)NCCn3cccn3)CC2)C1 CCC(C(=O)NC(C)C(C(=O)NCC(C)(COC)CO)C(C)C)C(C)(C)CC c1(C(N2C3CCC(NC(c4cc(CC)n(C)n4)=O)(C3)C2)=O)cc(S(N)(=O)=O)cs1 C(=O)(CC(CCCCCNCC1CCCC12CC2)C(F)(F)F)OCC C1(CC)(NC(=O)Cc2ccnc(OC)c2)CCN(C(c2ccccn2)=O)CC1 N1(C(c2cc(C)cc(O)c2)=O)CCN(C(=O)CCc2cnn(C)c2)CC(C)(C)C1 N1(C(C2CCC(OC)CC2)=O)CCOCC(NC(C23CCC(OC)C2C3)=O)C1 c12ccc(F)c(c1)S(=O)(=O)NC2=O.C1(CN(CC)CC)CC1C1CC1 c1(C(=O)NCCN(CCOC)C(C2CCC3CC23)=O)[nH]cnc1C N1(C(C(c2scc(C)n2)C)=O)CC(NC(=O)CCC23CCC(CC2)C3)C(C)C1 C(=O)(C1=CC(O)C(NC(c2scnc2CC)=O)C1)NC1C(C#C)CCC1 CC1CN(C(=O)C(C(C)O)N(C)C)CCC1CNC(c1cnco1)=O C(=O)(C(C)(C)C(=O)N(C)C)NCC12N(C(=O)C(C)(C)CF)CC(CC)(C1)C2 C1(NC(CC2CC(N(C)C)C2)=O)CC(O)CN(C(C23CCC(C2)C3(C)C)=O)C1 c1(CC(=O)NCC2N(C(Cc3nc(C)sc3)=O)CCC2)c(C)nn(C(F)F)c1C C(=O)(C(C)(C)CCNC(C1CCCN(CC)C1)=O)NC(CC)CC(C)O Cc1nnc2cc(N3CCC=C(CNC(c4cccc(F)c4F)=O)C3)ncn12 CCCC(C(=O)N1CCC(O)C(N(C)C(c2oc(CC)cc2C)=O)C1)C(C)C Cc1nc(N)cnc1C(=O)NCCCN(C)C(C1(C)CCCO1)=O C=CCC(CC(C)C)C(=O)NC(C(=O)NCC(F)(F)C1CC1)C(C)C N1(C(CN(CCNC(C2(CCC#C)OCCO2)=O)CC)=O)CC(C)OC(C)C1 Cc1nn(CC(=O)NC2CC(C(F)C(=O)NC(F)(F)F)C2)c(=O)o1 C1(CC)C(C(=O)NCc2cc(C)nn2C)CCCN1C(=O)C(O)CN(C)C C1(CCC(=O)NCC=CCNC(c2cc(Cl)ns2)=O)CCCCCC1 N1(C(CS(CC)=O)=O)CC2CN(C(c3cccnc3C3CC3)=O)CC2(C)C1 c1(C(=O)OC)ccn(CCNC(=O)CC2CCCN2C(=O)OC)n1 Cc1cc(NC(=O)C=CC2CC2)ncn1.C12CC(C1(C)C)C(=O)NC2 N1(C(CC(C)(C)OC)=O)CCN(S(=O)(=O)N2CC(C)OC(C)C2)CC1 C(=O)(C1=CNC2=NCCCC2=C1)N1CC(F)CC(NC(C2(CC(C)(C)C)CC2)=O)C1 c1(C(=O)NC(CC)CC(=O)NCC23CCC(CC2)C3)cccc(O)c1F C1(NC(CN(C(C)=O)C)=O)CC2CCC1(NC(=O)COCc1ccccc1C)C2 Cc1cc(O)cc(=O)n1CC(N1CC2(C1)SCCC2NC(=O)CC1C=CCC1)=O N1(C(C)=O)c2ccccc2CC1C(=O)NCC1([Si](C)(C)C)CCC1 C#CC1CC(NC(=O)C(C)CN(C(=O)CCC2CCCOC2)C)C1 N1(C(C(CC)n2ccnc2)=O)CC(O)CC1CNC(=O)C(C)(C)OCC(F)(F)F C1(C(=O)NC(CC)C(=O)NCC2CC3(CCO2)CC3)CC2(CCO1)CC2 c1(OC)ccccc1CCNC(=O)C(=O)NC(C1CCCO1)COC c1(C(=O)NCC2OCCN(C(c3onc(C)c3C)=O)C2)ccc2occ(C)c2c1 C1(C(=O)NCc2ccncc2F)CN(Cc2cc(F)cc(I)c2)CCC1(F)F C1(C(N(CCCNC(=O)CCC(=O)c2cccnc2)C)=O)CNC(=O)CC1(C)C c1(C(=O)NCCNC(C2(C)CC3(CC3)C(C(F)(F)F)CC2)=O)cccc2ccsc12 N1(C(C(C)(C)C)=O)CCCC(F)(CNC(C2CCC3(CCC3)C2)=O)CC1 C1(NC(C2C3CCOCC23)=O)CC2(C1)CN(C(=O)CCc1nnc(S)nc1O)C2 C1(C(=O)NCCCCNC(C(CC2CCCCC2)OC)=O)CCN(C)C1=O c12ncnc(c1C)N2CCCOCCOC.c1(C(CC)N)cccs1.C1(C)CCC1 c1(C(=O)NC(C2CN(C(C3OCCOC3(C)C)=O)C2)C)ccnc2[nH]nnc12 N1(C(C(CC#C)C)=O)CCN(C(c2cc(C)nc(C)n2)=O)CC1C Cn1c(-c2ccc(Cl)cc2)nnc1C1CCCCC1.C(C(C)CO)=[SH]C C1(NC(CC(=O)OCC)=O)CC2CN(C(=O)COCCO)CC2C1 c1(C(C)C)cc(=NC(C)C2COc3ccccc32)[nH]c(=N)[nH]1 C(=O)(C1=CCC(NC(=O)CC2CCCCCC2)C1)NC(c1ccsc1)C C1(C(=O)NC2C(C)NC(=O)CC2)CN(C(c2csc(C#N)c2)=O)CC(C)(C)C1 c1(-c2cn(C3CCN(C(CC4(C)CCC4)=O)C3)nn2)cncc(C(=O)O)n1 C(=O)(C1=CC2CCC(C1)C2)N1C(C)CC(CCNC(=O)C2CC2)C1 c1(CNC(C2C(C(N3CC(NC(N)=O)C3)=O)CCO2)=O)ccc[n+]([O-])c1 C1(C(=O)NCC2C=CC(NC(C3CCCC(N(C)C)C3)=O)C2)CN2CCCN1CC2 c1(C(N2C3C(NC(CCCCCC)=O)(CCC3)CC2)=O)ccc2c(c1)C(=O)NC2 CS(=O)(=O)C1CC(C(N2CCC2C(=O)Nc2cc(I)ccc2C(N)=O)=O)C1 C1(CNC(C(CC)CC)=O)CCCC2CN(C(=O)CC34CCC(CC3)C4(C)C)CC12 CC(CO)C(=O)NC(CNC(=O)CCOCC1CC1)CO C(=O)(N=c1[nH]oc2ncccc12)C1N(C(Cc2cn(C)nc2)=O)CC2(CC2)C1 C(CCO)(C(F)(F)F)NC(C1(N(C(C2COCC(C)O2)=O)C)CC1)=O c1(C(=O)NC2CCN(CCNC(=O)C=Cc3cocn3)CC2)cccc(F)c1F CCCC(CC)C(=O)NCc1cc(C(=O)NCC(CO)C2CCC2)cs1 C1(F)(C(=O)NCCC(C)(C)C)CCCN(C(C2(C)COC2)=O)C1 C1(C)(NC(CC(CC)(C)C)=O)CCCN(C(=O)C(C)Oc2ccc(Cl)cc2)C1 N1(C(C(F)OC)=O)CCC(CNC(c2cc(-c3ccccc3F)no2)=O)(OC)C1 Cc1ccc2[nH]c(C(N3CCCC(C)(NC(=O)CCC(C)O)C3)=O)cc(=O)c2c1 C(C)(C)(CCC(=O)NCCC(=O)NCC(C)C1CC1)NC(C)=O Cc1cc2c(C(N3CCC(CNC(=O)CCC(F)(F)F)C3(C)C)=O)cccc2o1 C1(C(c2occ(C(N(CC(=O)NCCC(C)(C)OC)C)=O)n2)=O)CCCN1C=O C1(NC(C2(C)CCN(C(C(C(C)C)F)=O)C2)=O)CCC2CCCC1O2 Cc1ccc2c(c1)C=C(C(=O)NCCCN(CCO)C(C1COC(C)C1)=O)CO2 Cn1c(C(=O)NCCOCC(=O)NC2CCN(C3CC3)C2)nnc1S C(C(C)C)(C(O)C(=O)N1CC2(C(N3CCCC(CCO)C3)=O)CC1CCO2)OC C1(NC(C2(CC)CC(F)(F)C2)=O)CC2(NC(=O)CCc3cccnc3)COC1C2 N1(C(CN(C(CC(=O)OCC)=O)C)=O)CCCC(OC)C1C O=C(C#CC1CCCOC1)NCC(=C1CN(C(C2CCS(=O)(=O)N2)=O)C1)F c1(C(N2CCC(CC)CC2)=O)cc(F)c(N(C(c2cnccn2)C)CC)c(Cl)c1 N1(C(CCSCC)=O)CCCC(C2CCN(C(c3ncn(C(C)C)n3)=O)C2)C1 c1(C(=O)NCCC(C)NC(c2ccn(CC(C)C)n2)=O)cnc2n1CCC(C)C2 N1(C(C=CCN(C)CC)=O)CC2CCC1CN2C(C12CCN(CC1)CC2)=O N1(C(C(CC)(C)C)=O)C2CCCC1CN(C(=O)CC1CN(C)C1)C2 C(=O)(C1CCc2ccccc21)N1CC2C(CC(=O)Nc3ccsc3O)(CC2)C1 N1(C(CCCOC)=O)C2CCC1CC(F)(CNC(=O)CC13CC(C1)C3)C2 c1(CNC(c2ccc(C)cc2)C(=O)O)ccc2cc(F)ccc2n1 c1(C(=O)NCCN(C(C(C(COC)C)C)=O)C)cncc(S(C)(=O)=O)c1 c12ccc(cc1Cl)[nH]c2=O.c1(Cc2nc(C)[nH]n2)ccccc1CS(N)(=O)=O N1(C(=O)CCN2CCC2)CCC2(CCCN2C(=O)Cc2nc[nH]n2)C1 C(CC(=O)N1CC(Nc2ncnc(=N)[nH]2)CC(C)(C)C1)(C(F)(F)F)OC C1(C(=O)NC2(CNC(c3c(C)nsc3N)=O)CC(CF)C2)CCCCNC1=O N1(C(c2cccc(SC)c2F)=O)CCCC2C1CCN2C(C1(F)CCC=C1F)=O CCC(O)C(C)(C)C(=O)N(CCCCNC(c1ncccn1)=O)C n1(CCCN(C(C(C2CCOCC2)C)=O)C2CC2)cc(C(C2CCCC2)C)nn1 C1(CNC(C2C(=C)CC2)=O)CCN(C(c2ccc(OC)c(N)n2)=O)C1(C)C c1(C(=O)NCCCNC(C(C)(C)c2ccsc2)=O)ccc2cccc(Cl)c2n1 C(c1cccnc1)=C(C)C(=O)NCCC1(O)CCN(C(c2scnc2C)=O)C1 Cc1nn(CC(=O)NC2CC3CC(NC(=O)CC(C)(C)F)C2C3)c(=O)n1C C1(CC(=O)NCC(CC)NC(=O)CSCCCc2ccccc2)COCCO1 c1(CC(=O)NCc2scc(CNC(c3c(C)cno3)=O)n2)cccnc1Cl c1(C(=O)NCC(CNC(C(C)OCCN(C)C)=O)(C)F)cccc(F)c1F c1(C(=O)NC(CNC(C(C(C)C)C)=O)CC(C)C)ccc2occc2n1 C1(C(N(C(C#C)C2CC2)C)=O)(NC(=O)CN(C)CCOC)CC1C c1(CNC(CC2CC(=C)C2)=O)cccc(CNC(C2COC(C)C2)=O)c1 CC1=C(C(=O)N2CCN(C(=O)C=C(Cl)Cl)CC(C)C2)CCC(C)(C)C1 c1(C(N(C2CCN(C(c3c(NC)cccc3)=O)C2)C)=O)cc(C2CC2)ccc1F C#CCC(CC(=O)N1CCC(C#N)(c2ccccc2)C1)NC(=O)NC CC1(C)CC(O)CCN(C(=O)CO)C1.C12(C)CCCN1C(=O)CO2 N1(C(Cc2cc(CC)on2)=O)CCC2(CCN(C(C3(OC)CC3(F)F)=O)C2)C1 CC(N)CCC(=O)NNC(=O)CC1(c2ccon2)CCC1 Cn1nccc(C(=O)NC2CCCN(C(C3(C)CC(C#N)C3)=O)CC2)c1=O C1(CNC(=O)CCSC(F)(F)F)CCCN1C(c1cc(F)c[nH]1)=O CC(C)(C)CC(O)C(=O)N1CCN(C(=O)COC(F)F)C(C2CC2)C1 c1(CC(=O)N(C(C)CCNC(C2CCCC23CCC3)=O)C)cccc2occc12 C1(C(=O)NCC=CC)CN(C(=O)Cc2scnc2C)CCN1C CCC(O)C(C)(C)C(=O)NCCN(CC(C)O)C(=O)C=C1CCCC1 c1(NC(C)=O)ccc(C)c(N(C)C)c1.C1(=O)C(CC(C)C)NC(=O)CC2CN1C2 N1(C(Cn2c(C)ncc2)=O)CCC2CN(c3nccc(C(N)=O)n3)CC2C1 N(C(=S)NNC(=O)CCc1csc(Br)c1)C(C)(C)C Cc1cc(C)nc(N2CCCC2(C)CNC(C2(Sc3ccccc3)CC2)=O)n1 c1(C(=O)NC(CC)CNC(CCC)=O)cccc2ncccc12 C12(C(=O)NCC(C(=O)NC)(C)C)CCN(C(=O)CC3CCCCC3)CCC1C2 C(C(O)CC(C)(C)C)NC(c1cc(CNC(CN(C(C)=O)C)=O)nn1C)=O C(=O)(CC1=CCCCC1)NC1(C2CN(C(CCCCC#N)=O)C2)CC1 C(=O)(C1=NOC2COCC12)NCC(C)CNC(=O)C1=Cc2ccccc2C1 C1(NC(C2=NOC(CC)C2)=O)CCC2(CCN(C(=O)C(C(C)C)C(C)C)C2)C1 N1(C(c2ccc(N(C)C)cc2F)=O)CCN(C(=O)CCCC2CC2)CC(C)(C)C1 N1(C(=O)OC(C)(C)C)CC(CC(=O)NCC2CCOCC23CCC3)OCC1(C)C C1(NC(C2=C(C)OCC2)=O)CC2CCC1N(C(=O)C(C1CCOCC1)F)C2 c1(C(=O)NCC2C(NC(CC(C)n3ccnc3)=O)C2)ccc2n1CCCC2 Cc1nc(C(=O)NCC2(NC(c3ccc(C4CCOC4)s3)=O)CC2)cs1 C1(C2CCN(C(c3n[nH]c(C)n3)=O)C2)(NC(C(Cn2ccc(C)n2)C)=O)CC1 C1(NC(CCSC)=O)CCN(C(c2ccn(CC3CC3)c2C)=O)CC1O N1(C(CC=CCC)=O)CCC(O)(CN(C(=O)C(O)C(C)CC)C)CC1 N1(C(C2(CC(C)C)CCNC2=O)=O)CCCC(NC(=O)CC2(C#N)CCC2)CC1 C1(NC(C2OCCN(CC)C2)=O)CC(C)CN(C(=O)CC2(CSC)CC2)C1 c1(C(N2CCC(C(N3CC(N(CC=C)C)C3)=O)(CC)C2)=O)ccc2nccn2c1 c1(C(N2CCOCC2C)C(=O)NCC=C)cn(C)c(=O)n(C)c1=O C(=O)(C(O)CCNC(=O)CC1(C)CC1)N(CC)CC1CCOCC1 C1(C(=O)NCC(C)(C2CC2)NC(C2(c3cccs3)CC2)=O)CCc2nncn2C1 C(=O)(C#CC1CC(F)(F)C1)NC(C1CCN(C(c2ccnn2CC#N)=O)C1)C CC(C)CCC(F)C(=O)N1CCC(CNC(=O)CCCC(C)C)C(C)C1 C(=O)(C(C)C(CC)CC)NCC(CC(=O)N(c1ccc(C)cc1)C)C1CC1 c1(N(CCC)C2CC2)ccc(Br)cc1.c1(C=O)ccc(C(N)=O)o1 CC1CCOC(C(=O)NC2(CF)CCN(C(c3nn[nH]c3C(F)(F)F)=O)C2)C1 C1(C(=O)NC(C)C(CO)NC(c2cocn2)=O)CCC12CCOCC2 CC(c1cccc(Cl)c1)=CC(=O)NC(C)CCCCNC(c1sccc1F)=O C1(C(=O)NC2(CO)CCN(C(c3n(CC)ccc3)=O)C2)Cc2cc(C)ccc2S1 c1(NCC2C(C)CCCN2C(=O)C=CCN(C)C)ncnc2sc([N+](=O)[O-])cc12 c1(NC(N2CC3(CN(C(c4cccc(F)c4)=O)C3)C2)=O)ccc(B(O)O)cc1 N1(C(c2cnc(N3CCC3)nc2)=O)CCC(NC(=O)CSSC)C(CO)C1.CO C1(CCNC(C=C(CCC)C)=O)CCN(C(=O)C=Cc2cocn2)C(C)C1 c1(CNC)cccc(-c2ncccc2C(=O)NC(C(F)(F)F)C2CC2)c1 C=C(C)C(C)(C)C(=O)NC1COCC1NC(=O)Cc1cn(CC(F)(F)F)nn1 C1(C(=O)NC2CN(C(C3(C(=O)NCC)CCC3)=O)C2)CC12CCSCC2 c1(C(=O)NCC(CC=C)NC(=O)CSC)nc(Cl)c(=O)[nH]c1N c1(-c2ccc(OCC(=O)O)cc2)ccc2ncc(C(N3CCC3)=O)c(Cl)c2c1 CC1(C)CCN(C(c2sccc2C#N)=O)CC1CNC(=O)C=CC1CCOCC1 C(=O)(CN=c1[nH]c(N2CCn3ncc(CC)c3C2)nc2c1CCCC2)NCC=C N1(C(C(=CC2CCCC2)C)=O)CCC(O)(C(C)CNC(C2CC(=C3CC3)C2)=O)C1 c1(C(NNC(N2CCN(C)C(=O)C2)=O)=O)ccc2c(c1)OCCO2 c1(N2CCC(NC(c3cn(CC)nn3)=O)C(F)C2)nc(Cl)nc(CC)c1C#N C1(C)(C(=O)N(CC23CC(CN)(OC2)C3)CC2CC2)CC2CCC1O2 c1(C(=O)NCC2(NC(C=C(CCC)CCC)=O)CCC2)ccnc2ncc(C)cc12 C(CN=c1[nH]c(Cl)ncc1C)c1c[nH]nn1.Cc1cc(C)n(-c2cccc(N)c2)n1 C1(CC)C(CC(=O)NC2CC(F)(CNC(=O)C(=O)NCCC(N)=O)C2)C1(F)F C1(NC(C(C)N(C(C)=O)C)=O)CCC(C(=O)Nc2cnncc2Cl)CC1 Cc1[nH]c(C(=O)NCC2CC2NC(C2(c3ccn(C)n3)CC2)=O)c(C)c1[N+](=O)[O-] C(=O)(C1=CCCCO1)N1CC2C(CNC(c3scc(C)c3)=O)C2C1 N1(C(COC(CNC(C(C(=O)OC)(F)F)=O)(C)C)=O)CC(C2=NOC(C)C2)C1 C(CCC(C)(C)NC(C1(NC(=O)CCCNC(N)=O)CSC1)=O)OC C1(NC(C(C)N2CCC2)=O)CC2(CCN(C(c3ccc4nsnc4c3)=O)CC2)C1 N1(C(CC(CC)(C)C)=O)C(C)CN(C(=O)C=Cc2ccccc2C#N)CC1C c1(C(N2CCCCC(NC(CC(=O)NCC3CC3)=O)C2)=O)c(F)ccc(Cl)c1F c1(-c2cc(C)cc(F)c2)csc(=Nc2cccc(Cl)n2)n1CCC#CBr C12(CNC(C(CC)n3nccc3C)=O)CC(CNC(=O)CN(C)C(N)=O)(CO1)C2 C(=O)(C(CCCNC(c1cc(CC)on1)=O)C1CC1)N1CC(C#CC)C1 c1(C(N(CCC(C)NC(C2C=CCC2)=O)C)=O)cccc2c1CCCC2 N1(C(c2[nH]nc(Br)c2-c2ccccc2)=O)CC2CC(NC(C3(O)CC3)=O)C1C2 C1(ONC(C2CC(CNC(Cc3c(C)cco3)=O)OC2)=O)C=CCCCC1 CC1=NN(C)C(=O)C1CC(=O)NCCC1COCCN1C(C1CC(C)(F)C1)=O S(=O)(=O)(c1cnc(NCCCCC)c(Cl)c1)NCCN1CCC(CO)C1 Cc1ncnc(O)c1C(=O)NCCOCCCNC(=O)C(C)OCC1CC1 c1(C(=O)NC2C(NC(C3C(CC)OCC3)=O)CCC2)cc2ccc(Cl)cc2o1 c1(OC)ccc(Cl)c(C(=O)NCC2C3CN(C(=O)C(C)(C)C(C)O)CC23)n1 CC1CC(C(=O)N2C(CCCNC(=O)Cc3sc(O)nc3O)CCC2)=NO1 n1(CCSC)nnnc1C(c1ccsc1C)NC1CC(C)(CC)C1 Cc1c[nH]c(C(=O)NC(C(=O)NC2(c3nc[nH]n3)CC2)C2CCC2)c1 CC(C)(C)C(O)C(=O)N1CCOCC1CNC(C1CNC(=O)N1C1CC1)=O C1(CC(=O)NC(CNC(C2(C=C)CCC2)=O)C2CCC2)(N(C)C)CCCCC1 CCC(O)C(C)C(=O)NC1CCC(CNC(C2OCCN(C)C2=O)=O)CC1 c1(C(=O)NCC2CCC(NC(c3n(C(C)C)ccn3)=O)C2)ccc(=O)oc1 c1(C(=O)NCC=CCNC(CC2C(C(=C)C)OCC2)=O)cccc2nn(C)cc12 c1(C(N2CC(CCNC(CC=C)=O)OCC2)=O)ccc2nnn(C(C)C)c2c1 n1(CC)cc(Cl)c(C(=O)NCC(C(C)(C)C)NC(c2[nH]nnc2C2CC2)=O)n1 C1(CCNC(C(COC)OC)=O)CN(C(=O)CNc2ncccc2O)CCCO1 C(=O)(C(C)(C)C(F)(F)F)N1CC(C(=O)NCCSCC)OC(C)C1 CCC(C)(CC)C(=O)NCC(c1ccccc1F)NC(c1cn(C)c(=O)n1C)=O Cc1c(CNC(C2CCCC(NC(c3cnc[nH]c3=N)=O)C2)=O)nnn1C N1(C(=O)NCc2c(C)c[nH]n2)CCN(C(=O)N(c2cn[nH]c2)C)CC1 CC1(C)CN(C(=O)COc2ccc(O)cc2)CC1C(=O)Nc1cncnc1 C1(CNC(C(C(C)C)N(C)C)=O)CC2(CCN(C(c3scnc3Cl)=O)C2)CO1 C(CCC(C)CC(=O)N1CC2CCC(CNC(C3(N(C)C)CC3)=O)(C2)C1)=C(C)C C1(CC)CCC(C(=O)NCCN(C(C2CC2c2ccccc2)=O)CC2CC2)CC1 Cc1cc(C(N2CCC(NC(C3CCCN(C)C3)=O)C2)=O)ccc1C#N C(C(=O)NC(C(=O)NC1(COC)CC1)C1CC1)(C(C)C)OC c1(C(N2C(CNC(C3(C)CC(C)(C)C3)=O)CCCC2)=O)c[nH]c(=N)c(C(=O)O)c1 CON(CC1CCCCCC1)C(=O)C(C1CCOC1)OC N1(C(CC2CC(C)C2)=O)CCC(C)(CNC(=O)COc2cc(F)ccc2F)CC1 C(C(CC(C)C)C(=O)NC(C1(O)CCN(C(c2oc(CO)cc2C)=O)C1)C)OC N1(C(COCC(C)(C)C)=O)CCC(C)(CNC(C2(C#N)CC3CC3C2)=O)CC1 C1(C(N(CC(C)(C)CNC(c2ccc(O)c(Cl)n2)=O)C)=O)CC2CCCCCCC12 C1(NCC2(O)CCN(C(=O)NCc3nncc(C)c3)CC2)Cc2ccccc2O1 C1(CN(C)C(C2CCOC2)=O)CCCCN1C(c1c(Br)nnn1C)=O C1(C(=O)NCC2(CNC(CC(=C)C)=O)CC2(F)F)NC(=O)OC1C N1(C(CCCNC(=O)OCC)=O)CC2(C1)CN(C(=O)C(Cl)=CCl)CC2CO C1(C(C)C)CCCC1C(=O)NCC1CC(NC(c2nc(C(C)(C)C)ns2)=O)C1 C(=O)(CC(C(F)(F)F)NC(C)C(=O)NC(C)=O)N1CC(C(N)=O)C(C2CC2)C1.CC Cc1cccc2c(CC(=O)NCCN(C(=O)C(C)Cc3ccncc3)C)c[nH]c12 c1(COC)nc(NCC2CC3CCC2N3C(=O)CC2COCCO2)cc(O)n1 N1(C(C2(CCC)CC2)=O)CCN(C(C2CCCCC(=O)N2)=O)C(C(F)F)C1 C1(NC(C2CCCC(C)CC2)=O)CC2CC(C1)CN(C(c1cc(N)ccn1)=O)C2 c1(C(=O)NCC(CNC(C)=O)OC)c2c(nn1C(C)(C)C)CCCC2 Cc1c[nH]c(=NCCCC(C)NC(=O)CCc2cccs2)nc1Cl C1(CC(=O)N(CC(CC)NC(=O)Cn2cccc2C(=O)OC)C)CCCC1C N1(Cc2cncc(C)n2)CCC(NC(=O)Cc2ccccc2)C(O)C1 C1(NC(C2=C(C)OCCS2)=O)CCC(N=c2ccc(C#N)n[nH]2)CC1 C1(O)(C(=O)NC(CCN(C(c2c(C)cccc2)=O)C)C(C)C)CCCC(C)CC1 C1(CN(C(=O)C(=O)Nc2ccc(C)cc2)C)CC(F)CN1C(C1CC=CCC1)=O C1CCCCC(=O)N1.C1(C(F)(F)F)(N)CCCC1.C1(C2CCC2)C(=O)N1C.CCO C(=O)(C(F)CCC(C)C)N1CCC(C(CO)NC(C(CC2CC2)OC)=O)CC1 C1(OC)CN(S(=O)(=O)Cc2ccon2)CCC1NC(=O)C(C)O c1(C(c2ccccc2)NC(C2CC3OCCC23)=O)ccc(Cl)cc1C(F)(F)F CN1CCCCC(C(N2CCC(O)(CCNC(C3C4CN(C)CC34)=O)CC2)=O)C1 S(=O)(=O)(c1ccc(NC2CCC(C)(C)CC2)cc1Br)N(CC)Cc1ccc(F)cn1 CC(C)(CS(N)(=O)=O)C(=O)NC1CC(CNC(C2OCCC2(C)C)=O)C1 C1(CNC(c2ccc(-c3cccc(Cl)c3)s2)=O)CCCN(C(C2C3CCC23)=O)C1 c1(OCC(N2CCC(NC(C(C)(C)O)=O)C(O)C2)=O)cccc2ccccc12 C(=O)(C1CCCn2cnnc21)N1CCC(C)(CNC(CCN(C(CC)CC)C)=O)C1 C#CCCC(O)C(=O)N1CCN(C(=O)C2=CCCC2)CC1c1cccc(OC)c1 N1(C(CCc2ccc(C)nc2)=O)CC2(CC2)CC1CNCc1cc(Cl)cc(Cl)c1 C12(C)CCC(C1)OC(=O)N2.CCC(F)(F)CNC(=O)OC(C)(C)C C1(C(=O)NCC2(CCC)CC2)CC2(CCN(C(=O)C(O)COC)C2)C1 Cc1c(C(=O)NC2CC2C2(NC(=O)OC(C)(C)C)CCC2)cnn1CC(F)F c1(C(=O)NCC2C(NC(C=Cc3cn(C)nn3)=O)C2)cc(F)cnc1O Cn1cc(C(=O)NCCCNC(c2ccccc2-c2cncnc2)=O)c(Cl)n1 C1(C(N(C(C(=O)OC)C2CC2)C)=O)CCN(C(C2CCC(C)C2)=O)C1 N1(C(C(CC)OC)=O)CC(CNC(c2csc(-c3cnccn3)n2)=O)CCC1C N1(C(CCC=C(C)C)=O)CCN(C(c2ccc(O)nc2C)=O)C(CC(F)F)C1 c1(NC2CN(C(CCC(=O)NCCCOC)=O)C(C)C2)ccc2nnnn2n1 c1(CNC(=O)Nc2cc(-c3ccnc(N4CCCC4)c3)ccn2)ccccc1Br C1(C(=O)Nc2cnc(C)nc2)CCC(C)(C)N(C(c2[nH]ccc2C)=O)C1 C1(C)(C(=O)NC2CC(C(C)O)C2)CCN(C(c2c[nH]ccc2=O)=O)C1 C1(CC)CN(CC)CCN1C(=O)CN1CCN(C(=O)NC(C)(C)C)CC1 C(=O)(C(CC(C)C)ONC(=O)Cn1ccnn1)NC(c1ncc(C)[nH]1)CC C(=O)(C(C)(C)CC=C)NC(CC#C)C(=O)N(C)Cc1c(C)cnn1C C12(CC(N3CC(CCO)(NC(c4cccc(SC)n4)=O)C3)=O)CCC(CC1)OC2 Cc1nc2ccccc2nc1C(=O)NC1CCC1NC(=O)C(c1cncnc1)C c1(OCC)ccc(CC(C)C(=O)NCCC(O)CNC(c2cnnn2C)=O)cc1 c1(COC)cc(NC2CCC(C)N(C(=O)C(F)CC3CCCC3)C2)nc(CC)n1 C12(NC(CSCC=C)=O)CCOCC1CN(C(c1cncc(C)n1)=O)C2 C1(OCC)CN(C(=O)NCC2CC(C(=O)O)C23CC3)CC1CO CN=c1nc(N2CCC(SC)C2)[nH]c(=NCCNC(=O)OC(C)(C)C)[nH]1 C1(C(=O)NCC2(C=C)CCC2)CCN(C(=O)COCCCC)C12CC2 Cc1ncc(N)cc1C(N1CCC(C(N2CC(OC(=O)N(C)C)C2)=O)CC1)=O N1(C(c2[nH]cc(C(C)=O)c2)=O)CC2(C1)CN(C(=O)Cc1cnco1)CC(C)(C)O2 CCC(CC)CCC(=O)N1CCC(CO)(NC(C2CN(C3CCC3)C2)=O)C1 c1(C(=O)NC(C)(CO)CS(C)(=O)=O)noc2c1CC(F)(F)CC2 C1(CCC(=O)NCC2(CC(C)C)CC2)CCC(NC(C2CCCCC2)=O)C1 CCN=c1[nH]c(C)c(C(N2CCN(C)CC2CNC(C2CC2COC)=O)=O)s1 N1(C(C(=O)Nc2cc(C)c(C)c(Cl)n2)=O)C2CCCC1CC(=O)NC2 c1(OC)ccc(C(N(CCOC)CC)=O)cc1.C1(N(CCCSC)C=O)CCC(C)O1 C1(CO)(NCCCn2cncn2)CC2CCC1CC2 N1(C(C)=O)CCCC(O)(CC(=O)NCC2CC2CNC(C2(F)CC=CC2)=O)C1 c1(C(C)(C)C)cccc(C(N2CCNC(c3ccccc3Cl)C2)=O)n1 C(=O)(C(C)(F)C(=O)N1CCC(C)(CNC(C2(CO)COC2)=O)C1)OCC N1(C(CC2C(CC)C2)=O)CCN(C(C)CNC(=O)C(C)(C)COC)CC1 C1(C(=O)NCCCN(C(c2cnc(OC)nc2)=O)C2CC2)CCCCC1(F)F c1(OC)ccc(C(=O)CCC(=O)NC2CCN(C(=O)CC3CC34CC4)C2C)cc1F C1(C(=O)NC(C2(O)CCN(C(c3[nH]nnc3C3CC3)=O)C2)C)CC2CCC1CC2 c1(C(N2CC3C(CNC(C(CCSC)(C)C)=O)(C3)C2)=O)ncc(Cl)c(N)c1Cl N(C(=NCC(C)N1CCCC(C)C1)NCC)C.CCC(C)(COC)C(F)F c1(C(=O)NCC23C(CN(C(C(CCCOC)C)=O)C2)CC3)c(C)ccc(Cl)c1N C(=O)(CS(=O)(=O)C1CC1)NCCC1N(C(C2CCC(C(=O)OC)O2)=O)CCOC1 C12CC(F)(F)CN1C(=O)CCSCC2.C1(C(=O)OCC)(OCC)CC1CC CC(CN(C)C)CCC(=O)NCCn1cc(C(=O)NCCS(C)(=N)=O)nn1 C#Cc1cn(C)nc1C(N1CCCC(NC(c2ccc(N)cc2Cl)=O)C1)=O C1(C(N(C2CN(C(CSCCC)=O)C2)C)=O)CCc2ccccc2O1 N1(C(c2cn(CCOC)nc2)=O)CCC(CF)(NC(=O)C(F)CC2CC2)C1 Cc1noc(C)c1C(C)C(=O)NCC1(F)CN(C(=O)C=CCF)C1.c1(Br)c(=O)n1 C1(C(=O)NC(CN(C(Cc2nc(C)[nH]n2)=O)C)(CO)CO)CN2CCCN1CC2 N1(C(c2cncc(SC)c2)=O)CC2CCC(C1)N(C(=O)COCC1CC1)C2 c1(C(=O)NC2CN(C(C=CCN(CC#C)C)=O)C2)n[nH]c2cc(Cl)ccc12 c1(OC)ccccc1C(C)C(=O)NCCN(C(=O)Cc1c(C)cnn1C)C1CC1 Cc1ncc2n1CCC(C(=O)NCC1CCN(C(=O)CCOC3CC3)C1(C)C)C2 C(CC(=O)NCC1(CCNC(=O)C(C)(C)c2cccnc2)CC1)(C(F)(F)F)OC n1(CC)ccnc1C(N1CCC1(C)CC(=O)NC(c1ccn(C)n1)C)=O NS(=O)(=O)c1sccc1C(C(=O)NCCO)NCC(c1ccccc1)O c1(C(N2CCC3CN(C(=O)COc4cccnc4)C3C2)=O)ccc2sncc2c1 C1(NCc2c(C(=O)OC)cno2)CC(C)N(C(=O)CNC(=O)C2CC2)C1 C1(C(N2CCC(F)(CNC(=O)C=CC3CCCO3)CC2)=O)CCC2CCCCN12 N1(C(c2cc(SCC)ncc2)=O)CCCC2CN(C(=O)CCC[N+](=O)[O-])CC12 CN1CCCC(CC(=O)NCC2(O)CCN(C(=O)CC3CCC(F)(F)C3)C2)C1 Cc1nscc1CNC(=O)CC1(CNC(=O)CC(C)N2CCCC2=O)CC1 c1(NC(=O)C=CCNC(=O)CSC(F)(F)F)cccc2c1CCO2 c1(CC)cc(C)[nH]c(=NCCC2CC(C)N(C(c3ccc(CC)o3)=O)C2)n1 c1(-c2nc(-c3c(O)cc(Cl)cc3F)on2)ccc2cnccc2n1 c1(OCCC)cccc(C(N2CC(NC(C3CCO3)=O)C(C)C2)=O)c1 c1(C(C)NC(=O)COC(c2snnc2C2CC2)=O)csc(-c2ccccc2)n1 C1(C(N(C2CCCN(C(c3cccc(=O)o3)=O)C2)C)=O)CC(C2CC2)C1 N1(C(C(C)NC(C)=O)=O)CCCN(C(c2csc(Cl)n2)=O)C(C)C1 C#Cc1ccc(C(=O)NCC(CC(C)C)NC(=O)C=Cc2cn[nH]c2)nc1 CC(C)C(C)(CNC(c1cccc(Cl)c1)=O)NC(C1CC2C=CC1C2)=O O(NC(=O)C(C)(C)CCNC(=O)CC1CCC(OC)CC1)CCC=C C1(NC(c2c(C)nc[nH]2)=O)(CNC(=O)C(F)(F)Sc2cnn(C)c2)CCCCC1 c1(C(N2CC(CNC(c3c(C)nc(C)o3)=O)OCCC2)=O)cc2c(s1)COCC2 c1(C(=O)NC(CN(C(C2OCCN(CC)C2)=O)CC)C)ccc(C)n(C)c1=O C1(N(C(=O)OC(C)(C)C)CCF)CCN(C(=O)CCC(C)(O)c2ccccc2)O1 S(=O)(=O)(c1cccnc1NC1CCC1(C)COC)N(C)CCOCCO c1(C(C)NC(=O)CC2CC2CNC(=O)COC2(C)CCC2)n[nH]c2c1CCC2 c1(N(S(CC)(=O)=O)CCN)ccccc1Cl.c1(C=O)cnc(Br)s1 N1(C(C2C(=C)C2)=O)CCOC(C(=O)NCC(F)Cl)CC1 C1(C(C)C)N(C(=O)OC(C)(C)C)CC12CCC2OC(c1cccc2nsnc12)=O n1(CCC(=O)NCCC2CCN(C(c3n(CC=C)ccc3)=O)C2)c(C)ccc1C C(=O)(C(=O)C(C)(C)C)NC1(CC=C)CCN(C(C2CCCC(O)C2)=O)C1 c1(C(=O)NCC2(NC(=O)Cc3ccc(Cl)cc3)CCOC2)csc2nccn12 N1(C(C2N(C(CCC)=O)CCC2)=O)CCC(NC(=O)C=Cc2nccs2)C(CO)C1 c1(C(=O)NCCCNC(CSCCOC)=O)sccc1C1CC1 c1(OC)cc2ncccc2cc1C(=O)NC1CCN(S(=O)(=O)c2ccccn2)C1 C(C(C)(C)CCNC(c1ccnc(C)c1)=O)NC(C(CC)OC1CCCCC1)=O N1(C(C(C(=O)OCC)F)=O)CCC(NC(c2oc(CO)cc2C)=O)CC(C)(C)C1 C1(NC(CC=CCC)=O)CCCC12CCN(C(c1nscc1C)=O)C2 c1(C2C(NC(=O)NCCNC(N(C(C#C)C3CCC3)C)=O)C2)cccnc1 C1(C(=O)NC2CC(C)(CNC(=O)CN3CCSCC3)C2)(CC)CC1(F)F c1(OC)ccc2nc(C)c(C(=O)NCC3CCCCN(C(C4CCCC4)=O)C3)n2n1 Cc1nn(C)c(N)c1C(N1CC=CC(C(=O)NCc2cncs2)C1)=O Cc1nnc(C(=O)NCC2CCN(C(=O)CNC(C3CCOCC3)=O)C2)s1 CC1CCCCC1NC(=O)NCCCCNC(c1cnc(OCCO)s1)=O C1(CC(=O)N(C)CC2CN(C(C3(N(C)C)CC3)=O)C2)CCCCN1C C1(N(C(C=C(COC)C)=O)CC2CC2)CCN(C(C2CCC(F)C2)=O)CC1 C#Cc1cccc(C(=O)NC2(CC(N3CCC(C)(COC)C3)=O)CCC2)c1 N1(C(c2n(CC)ncn2)=O)CCN(C(c2cc(OC)cs2)=O)CC12CCC2 CS(=O)(=O)CC(=O)NCC1CCN1C(c1csnc1Br)=O Cc1cnc(NC(c2cccc(F)c2F)C)c(S(=O)(=O)NC2(CCC(N)=O)CC2)c1 c1(C(N2CC3CN(C(c4cc(SC)ncc4)=O)C3C2)=O)cnc2ccc(C)cn12 C1(CNC(C=CSC)=O)CCC2CN(C(=O)C=Cc3cncn3C)CC12 N1(CC(=O)NCC2C(CNC(C3CC(OC)C3)=O)CCC2)CCCCC1=O C1(CNC(C2CC2(Cl)Cl)=O)CN(C(c2n[nH]cc2C2CC2)=O)CCO1 c1(N(C(=O)C(C2CCN(C(=O)Cc3ccc(C)o3)C2)F)C)cccc(F)c1F Cc1cccc(-c2ccc(NCc3cccc(C(F)(F)F)c3)nc2)c1F c1(NC(=O)NCCC(N2CCC(C(=O)NCC)C(C)C2)=O)ccc(OC)cc1C C1(NC(c2nccc(C#C)c2)=O)CC12CCN(C(C1CCOC(=O)CC1)=O)CC2 C1(NC(=O)NCc2cc(F)cc(Br)c2Cl)CCOC2(CCC2)C1 C1(C(N(C)Cc2ccccc2)=O)COCCC12CN(C(C1CNC(=O)N1)=O)C2 CN=c1cc(C(N2C3CCC2(OC)C3)=O)cc[nH]1 c1(C(=O)NC2(CNC(C(C)Oc3c(C)cccc3)=O)CC2)cc2n(c1)CCCC2 c1(OC)c(F)cc(NCc2cccc(C)c2OC(C)(C)C)cc1Br Cc1cc(C(=O)N(C)CCN(C(=O)CCN2CCC(C)CC2)C)oc1C c1(CCCCC)cc(NC(C2CCN(S(C)(=O)=O)C2)=O)ccc1OC C1(CCOC)CN(C(c2ccc(C)c(F)n2)=O)CCN1C(c1ccc(Cl)[nH]1)=O c1(C(N2CCCC(C(N(CC(c3nn[nH]n3)C)C)=O)C2)=O)cccc2c[nH]nc12 C=CCCCC(C(=O)NC1CC(=O)N(CC)C1)NC(=O)CCc1ccco1 Cc1coc(-c2ccccc2)c1C(=O)NCCCNC(=O)CCc1cc(Cl)no1 Cc1cc(CCC(=O)NC2CCC2NC(c2cccc(O)n2)=O)ccc1Cl c1(NCCC2CCC(NC(C3C(C(=O)OC)CCC3)=O)C2)cnn(C)c1C(C)C C(=O)(CCC(C)(F)F)NC(C)CNC(CSCC(=O)N(C1CCCC1)CC)=O c1(CC(=O)Nc2n(CC)ccc2)cccc(Br)c1.c12cn(nn1)CCCCCS2 C(=O)(CCS(=O)(=O)CC(C)C)OC.c12cc(n(C)c1)N(C)Cc1nnn(n1)C2.CC C(=O)(C1=C(C)OCCC1)NCCC1CC(C(=O)OCC)C1.C12(C)CC1NC2=O Cc1ccc(C(C)C(=O)NCC23CC(NC(=O)COc4cnn(C)c4)(C2)C3)o1 C1(C(N(CC(C)C)CCO)=O)C2CC3C(C2NC(C2CCCS2)=O)C13 C1(NC(C(N2CCCCC2)C)=O)CN(C(=O)C(O)CN2CCCC2)C2CCCC12 CC(C)CC(=O)NC1CCC(Cn2cc(Cn3cncn3)nn2)C1 c1(C(=O)OC)cc2n(c1C)CCN(CC(=O)N(C(C)C)CC1CCCO1)C2 Cc1cc(C(N2CC(C(=O)NCC3(C)CC(F)(F)C3)CC2(C)C)=O)ccc1C#N c1(C2C(C(=O)NCC3(F)CC(NC(C=C(C)C(C)(C)C)=O)C3)CC2)ccc(F)cc1 C1(C(=O)NC2(CNC(c3nn(CC)nc3C)=O)CC2)CCOC(=O)CC1 O=C(C1=NOC2(CCC2)C1)NC(CNC(=O)C(F)(F)c1ccncc1)C1CC1 C=C(C)CC(C(=O)NOCC(C)CC)NC(=O)CC1CC2CC2C1 C1(CNC(C2(C)CC=CC2)=O)C2CCCCC12 C1(NC(c2cnccc2C(F)(F)F)=O)C2CC(O)C1N(C(c1ccns1)=O)C2 N1(S(=O)(=O)CCC(F)(F)F)CCOC2(CCN(Cc3nc[nH]n3)CC2)C1 c1(CC)ccc(CC(=O)NC2CCC(N(C(=O)CN(C)C(=O)OC)C)CC2)cc1 C(=O)(CN=c1cc[nH]cc1)NC(CN(C)C)C(=O)NCCc1ncccn1 c1(C(=O)NCC(CNC(c2ccc(CC)cc2O)=O)CO)cc2cccnn2n1 C(=O)(C1=CCC2CCC1N2C(=O)CCc1nccs1)N1CC(C)OC(C)C1 c1(OC)ccc2[nH]c(=NC(C)CCC3CCC3)nc(N3CC=C(CO)CC3)c2c1 N1(C(C(CC)Sc2ccccc2)=O)CC(CNC(=O)C(C)NC(C)=O)C(C)(C)C1 C12(NC(CCOCC)=O)CCOC(NC(=O)CC(COC)COC)(C1)C2 C1(C(N2CCC(C)C2C(=O)NC2CC(O)C2O)=O)CCCC(C)(C)C1 c1(CN(C(=O)NC(C(F)(F)F)C2CCOC2)CC)cc(Cl)cc2nc(C)[nH]c12 C(N=c1cc(C2CC2)nco1)C1CCN(C(C=CCCC)=O)C1 C1(N(C(=O)Cc2cc(C3CC3)on2)C)C2CN(C(c3cc(Br)n(C)c3)=O)CC12 N1(C(c2occ(C)c2)=O)CCN(C)C(CNC(=O)C(F)CC2CCOC2)C1 CC1CC(CNC(=O)Cn2cnc(C#N)n2)CN1C(=O)Cn1ncccc1=O Cc1cnc(CNC(=O)NCCSCc2ccc(Cl)s2)cc1Br c1(C(N2CCC(NC(C=C)=O)C2)C(=O)NCC(=C)C)cscc1Oc1ccccc1 Cc1cnn(C)c1CC(=O)NCC(C(C)(C)C)NC(c1cc(Br)c[nH]1)=O C1(C(N(CC(C)C#N)C)=O)C=CCCN1Cc1cncs1 c1(C(N2CCC(N(C)C)C2)C(=O)NCCOC)cn(C)c2cc(Br)ccc12 C1(NC(CCC(C)SC)=O)CCN(C(c2sc(C)nc2C)=O)CCC1(F)F N1(N(c2nccc3occc23)Cc2c(C)nc(N(C)C)s2)CC2(C1)SCCC2CO CN1N=C(C(=O)NCC(O)CCNC(c2cc(C#N)n(C)n2)=O)CCC1=O Cc1ccc(C=CC(N2CCCC2CN(C)C(c2nc(C)ncc2Cl)=O)=O)cc1 C(CC(N)C(=O)N(CC(C)CN1CCOCC1)C)SC C(C)(CCC(=O)N1CC(C(=O)NC(c2nncn2C)C)(SC)C1)OC C1(OC)CC(C(=O)NC2CC2CNC(=O)CNC(C2CCCC2)=O)C1 C1(CCNC(CCCC=C)=O)CCCN(C(C2CSCC(=O)N2)=O)CC1 N1(C(C(C#N)=CC2CC2)=O)CC2C(CNC(=O)Cn3ccc(C4CC4)n3)C2C1 c1(C(CNC(=O)CC2CC(F)C2)NC(c2c(CC)c[nH]c2)=O)ccc(F)cc1F C1(C(=O)NCCCOCC(C)C)CCCC(NC(=O)CN=[N+]=[N-])CC1 N1(C(Cn2ncc(C)c2)=O)CCCC(C)(C)C1CNC(=O)C(C)c1cncs1 c12cc(ccn1)CNC2=O.C(CC)(C(=O)NCCC1(OC)CCC1)=CC=CC n1(CC)cc(C(=O)NCC(C2CC2)NC(=O)CCCNS(C)(=O)=O)cn1 c1(C(=O)NCC(CN(C(C=C2CCN(C)C2)=O)C)O)ccc([N+](=O)[O-])n1C C1(c2cc(CNC(=O)Cn3cncn3)on2)CCN(C(=O)C(F)CF)CC1 C1(C(=O)NCC2OCCN(C(c3ccc(C)cc3F)=O)C2)Cc2ccccc2CO1 C12CC3CC3N1C2=O.C1(C(N)=O)(C(=O)NCC2CC2C(F)(F)F)CC1 C1(C)(C(=O)NCCCOCCCNC(c2nc(C)sc2)=O)C(C)(C)C1(C)C c1(C(N2C(CNC(=O)C=CCF)CC2)=O)ccc(Cl)c(N2CCCC2)c1 Cc1cnc2cccc(C(=O)N(CCNC(=O)C3=NOC4(CCC4)C3)C(C)C)n12 C(=O)(C1CCOc2ccc(F)cc21)NC1CCN(C(CSC(C)(C)C)=O)C1(C)C N1(C(c2ccc(OC)s2)=O)CCCC(CNC(c2cnc(C3CC3)[nH]2)=O)C1 C(=O)(CCC(=O)NCCC1CCC(C(=O)Nn2nccn2)C1)OCC C(=O)(C1=CC2CC(C1)CC2O)N(C1CCN(C(c2cc3cccnc3[nH]2)=O)C1)C C(CC(=O)NCCN(C(c1cnoc1)=O)CC)SC.C12(CC1)C(=O)N2 C1(NC(CC2C(C)(C)C(O)C2)=O)COCCN(Cc2ccc(CO)c(F)c2)C1 C1(C(=O)NC(CCC)c2ccco2)CCN(C(C2(CO)CC(OC(C)=O)C2)=O)CC1 N1(C(COCc2cccc(C)c2)=O)CCN(C(=O)C(C)N(C)C(C)=O)C(CF)C1 C1CSc2ccccc2O1.N1(C=O)CCC(C2C(C(=O)NC3(COCC)CC3)C2)C1 S(=O)(=O)(c1ccc(O)cc1)NC1C(F)(F)CCN(Cc2n(C)cnc2)C1 C1(C2C(CCC(C)(C)C)n3nnnc32)CC2(COCCO2)C1.C(CC(C)CBr)OC Cc1cc(O)ccc1CC(=O)NC(C1CN(C(C2COCCC2(F)F)=O)C1)C CCCC(C(=O)NC(C)COc1cccc(Br)c1)c1ccccc1 C(=O)(CCCCN=[N+]=[N-])N1CCC(N(C)C(C2CC3(CCCO3)C2)=O)CC1 C(N=c1[nH]c2c(c(=NCC)[nH]1)COC2)C1CN(C)C1.S(=O)(=O)(c1ccccc1Cl)N c1(C(N2CC(CC(N3CCCC(C(=O)O)C3)=O)C2)=O)c[nH]ccc1=O c1(OC)nccc2c(C(=O)OCc3cc(Br)c(Br)o3)csc12 CCC(C)C(C(=O)NCC(C)CN(C(=O)CCCC1CCCO1)C)OC C1(C(=O)NC(CC(=O)NC)C)C(C)OCCN1C(=O)CC1CCCC2CC12 c1(CCNC(=O)COC2CC=CC2)ocnc1C1CC1.c12cn(nn1)CNC2=O c1(OC)c(C)nc[nH]c1=NCC1CCCC1NC(C1CC2(CCOCC2)CO1)=O C1(C(N(C2CN(C)C2)C)=O)CC(O)C(O)CC1CNC(C1CCCNC1=O)=O C1(CC(C2CCCCN2C(C2CC3(C2)CC3F)=O)C)CCN(C(C)C)C(C)C1 CN1CC(NC(=O)C=CCC2(NC(=O)CC3CCCC3)CCC2)C(C)(C)C1 CC(C)CCCN(C)C(C1CC1CN(C(=O)CCOCC(C)C)C1CC1)=O C(=O)(C(C)(C)CC(C)(C)C)NCC12CC(NC(c3c(Br)ccc(C)c3)=O)(C1)C2 c1(CNC(COC)=O)ccccc1CN(C(=O)C(c1cccc(C#N)c1)(C)C)CC N1(C(C(C)(C)C2CCOC2)=O)CCCC(CNC(c2cc(F)c[nH]2)=O)CC1 Cc1cc(F)cc(C)c1C(N1CCC(O)(CCNC(=O)CC(C)C)CC1)=O N1(C(C=CC(C)(C)C)=O)CCOCC1C(N1CCC(COC)C1)=O C1(C(N(CC(C)N(C)C(c2csc(C(F)F)c2)=O)C)=O)CC2(CCOC2)C1 c1(C(=O)NCC2CCN(C(=O)Cc3ccon3)C2)cccc(S(=O)(=O)CCO)c1 C(CC(N)=O)(C(=O)N1CCCC(F)CC1)NC(C1CC(=C)C1)=O c1(NC(C(C)C(C)O)=O)cc2c(ncn2C)[nH]1.C12(C)CCN1C2 Cc1ccc(C2CC2C(=O)NCCOC(C)(C)CNC(C2CCC(F)C2)=O)cn1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CN(C(C(C)Cc2cccnc2)=O)C(C)(C)C1 C(c1ccc(F)c(Cl)c1)=CC(=O)NCC1CC2CN(C(CC(CC)C)=O)CC21 c1(C(C)C)[nH][nH]c2ncnc(=NC(CCc3ccccc3)C(F)F)c1-2 Cc1[nH]c(=N)nc(O)c1CC(N1CC(NC(=O)CN2CCSCC2)C(C)(C)C1)=O C1(NC(C(CCC)=CCC)=O)CN(C(=O)CC2CCC(=O)N2C)CC12CCC2 C=C1CCN(C(=O)C(C(=O)OCC)OC)C(C(=O)NCC(C)CC2CCC2)C1 C1(C(N(C(C(C)C)C)C)=O)CN(C(c2cc(Cl)cn2C)=O)CCN1C C1(N(CC=C)C(C2CCOC2)=O)CC2CCC1CNC2 c1(Cc2ccc(C)s2)cc(F)ncc1C.c12ncccc1C(=O)OC2 Cc1cc(NC(c2csc(CNC(=O)C(C)(F)F)c2)=O)cc(CO)c1 C1(C(=O)NCC2(CC(=O)OC)CC2)(CC)CCN(C(=O)C(O)Cn2cncn2)CC1 C1(C(N2CC(C3N(C(c4c(CC)non4)=O)CCC3)(O)C2)=O)CCC(F)(F)CC1 c1(OC)ccc(C(N2CC(CNC(=O)CC3CC(F)C3)C2)=O)nc1Cl C1(C)(NC(N2CC(CCO)(NC(CC=C)=O)C2)=O)Oc2ccccc2NC1=O c1(NC2CC(F)(CNC(=O)CC3CCC4CC34)C2)cc(=O)n2ccccc2n1 C(=O)(C(F)(C(F)(F)F)C(F)(F)F)N1CCC(N(C)CCC2CC2)C2(C1)CC2 c1(C(=O)NCC(N(C(CCCOCCOC)=O)C)C2CC2)cccc(CCN(C)C)c1 C1(CC(C)NC(C(C)NC(COCCC)=O)=O)CCCC2CC12 n1(CC(C)NC(CC=C)=O)cc(CNC(c2ccc[nH]2)=O)nn1 Cc1c(CN2CCC(O)C2C(=O)Nc2cc(O)ccc2Cl)cccc1O C1(C(=O)NCc2ccnnc2O)(NC(CNC(=O)OCC=C)=O)CCN(C)C1 C(=O)(C(CCC(N)=O)N(C)C)N1CCN(C(c2c(C)oc(Cl)n2)=O)CC1CC1CC1 c1(CNC(c2nc(C(=O)Nc3ccsc3)sc2)=O)ccc2ccccc2n1 N1(C(c2ccc(OC)cn2)=O)CCN(C(C2CCC(N(C)C)CC2)=O)C(CO)C1 c1(CCC(=O)NCC2CC2CNC(=O)Cc2cnsc2)cccc(F)c1Br CC1CC(C)N(C(c2cn(C(C)(C)C)nn2)=O)CCN1C(=O)CO c1(SCC(N2CC(C(=O)OC)N(C)CC2)=O)cn2cc(C)ccc2n1 C1(C)(C(N(C)Cc2nncn2C)=O)CCCN1C(C1(n2cccc2)CC1)=O Cc1cc(Cl)ccc1C(=O)NCC#CCNC(c1ccncc1Br)=O Cc1nn2c(c1C(=O)N(C)CCNC(C1(C)CC1C)=O)CCCC2C CCC(C)C(O)CC(=O)N1CC(C(=O)NCC(=O)N(C)O)C(F)(F)C1 N1(C(CCCCCC=C)=O)CCC2CN(C(=O)CC(C)(C)COC)CCC2C1 N1(C(CONC(CN2CC(C)(OC)C2)=O)=O)CCC2C(CN(C)C)C2C1 Cc1ccc(C(=O)N(CC(C)CNC(C2CC3C=CC2C3)=O)C)nn1 C1(C(=O)NC2CCN(C(c3cc(CF)on3)=O)C2)CN2CCC1CC2 Cc1c(C(N2CC3CC(NC(=O)C4=CCOCC4)C2C3)=O)ccc2cncn12 c1(CC)ccc(C(C)C(=O)NC2CC(F)CN(C(=O)OC(C)(C)C)C2)cc1F C(N=C(NC1CCC1)N1CCCC(n2cncn2)C1)c1cc(C)cc(C)c1 C1(C(N(CCC(=O)N(CC)CC)CC=C)=O)CC12CCOC2 C12(CNC(C3(SC)CCC3)=O)CCCC1N(C(C1(C)CCN(C)C1=O)=O)CCC2 Cc1[nH]c(C(N2CCC(NC=O)C(O)C2)=O)c(C)c1C(=O)NC(C)(C)CF Cc1cc(C(N2CCCC2C2CCOC2)=O)ccc1O.N12CC(C1)OCC2=O N1(C(c2cnc(C)nc2)=O)CCC2(CC1)C(=O)NCC2C(=O)NC12CC(F)(C1)C2 C=CCC(C)(C(=O)N1CC(CNC(c2occc2Br)=O)C(C)C1)N(C)C N1(C(c2nc(OC)nc(O)c2)=O)CCN(C(c2cccc(N)c2O)=O)C(C)C1C c1(CS(C)(=O)=O)ccccc1NC(=O)NC(c1cccc(-c2cccc(Cl)c2)c1)=O C(=O)(C(C)C(CC)CC)N1CCCC(CN(C(c2cnc(CC)nc2C)=O)C)C1 C1(C(N(CCCOC(C)C)C)=O)CNC(=O)CN1C(c1ccsc1C#N)=O C(=O)(CCCC(=O)N1CCCC1c1nc(C(=O)Nc2cc[nH]n2)cs1)NCCC Cc1ccc(CCC(N2CC(NC(=O)C=Cc3cscn3)C3(CC3)C2)=O)cc1C c1(CNC(c2scnc2-c2ccc3ncnn3c2)=O)cccc([N+](=O)[O-])c1Br N1(C(c2cncc(OC)n2)=O)CCN(C(c2c(C)nn(C)c2N)=O)CC12CC2 C(=O)(CCS(=O)(=O)N(C)C)NCC(C)N(C(C1CC12CC2)=O)CC C1(CC)CC(O)CN1C(=O)C(F)=C(C)C1CC1 c12cc(C(N)=O)ccc1S2.N1(C(CCOC)=O)CC2CC1C2NC(C)=O C(=O)(C(CC(F)F)c1ccccc1)NC(C1CCCC1)CNC(C(C)C1CC1)=O C(CS(=O)(=O)CC(=O)NC1CCN(C(c2ccc(C)c(CSC)c2)=O)C1)OC c1(C(=O)OC)[nH]c(C)c(C(N2CC3CC(NC(c4cn[nH]c4)=O)C3C2)=O)c1C c12c(cccc1F)OC(C)C(=O)N1CC(C(O)C1)CNC2=O.C(C(C)C)OCC C12(C(=O)NCc3ncc(C)o3)CCC(CC1)N(C(c1cccnc1)=O)C2 c1(C(O)Cc2csc(Cc3ccccc3)n2)ccc(Cl)cc1.C12CCN1C2 Cc1oc(CO)cc1C(=O)NCC1CC(NC(c2ccn(CCF)n2)=O)C1(C)C C(=O)(CC(C)(C)CNC(=O)Cn1cccnc1=O)NC(C)(C)Cc1cccnc1 c1(OCC)ccc(NNC(=O)CCN(S(C)(=O)=O)C(C)(C)C)cc1 Cc1cc(NC(C2CC2C(C)C)=O)ccc1NC(C1(C)CCCO1)=O c1(C(N2CC3C(C2)N3C(C2(C(F)(F)F)CC2)=O)=O)ccc2nc(Cl)sc2c1 C1(CCOC)(C(=O)NC(C)CSc2ccc(CO)cc2Br)CCN(C(N)=O)CC1 N1(C(CCC=C=C)=O)CCCN(C(c2cccc3ccoc23)=O)C(C(C)C)C1 C12(NC(=O)COc3ccccc3)CC1CN(C(=O)CCSCC1CCCCO1)C2 c1(NC(C2(CCNC(CC3C(C)OCC3)=O)CCC2)=O)cncc(CN(C)C)c1 C#CC1(C(N2CCC(CC3CC3)C2)=O)CCN(C(=O)C(C)N(C)C)CC1 c1(C(=O)NC(CC(C)NC(=O)C(C2CCC2)C2CC2)C)cccc2c1ccn2C CC1(CNC(=O)NCc2ccccc2)CCN(C(C(F)(F)F)c2cccs2)CC1 C1(C(N(C)CCN(C)C(C2(C#N)CC2(C)C)=O)=O)CC(c2ccc(F)cc2)=NO1 CCC(CN(C)C)CC(=O)NCCC1(C)CCN(C(c2cc(C(C)C)on2)=O)C1 N1(C(c2nc(N(C)C)oc2)=O)CC2CC(NC(C3CC(CCO)C3)=O)C1C2 C(=O)(C1=Cc2ccccc2C1O)N1CC(NC(CC=C)=O)C2(C1)CC2 c1(CC(=O)NCCN(C(CC)C)Cc2cccs2)ccc(Cl)s1 n1(C(C)C)nccc1CNC(=O)CC1(N(C(=O)CC2CCCO2)C)CC1 c1(C(=O)NCCCC(=O)NC2CN(c3ccccn3)C2)ccc(F)cc1 N1(C(CCOCCCOC)=O)CC(C)(C)C1Cn1cc(-c2ncccc2Cl)nn1 CCC(CCCO)NC(=O)C(c1cn(C)nn1)NC(C1(C2(C)CC2)CC1)=O c1(C(N(CCCNC(CCOC)=O)C)=O)ccc(S(=O)(=O)N(C)C)o1 C1(C(=O)N(c2ccccc2)CCCC2CCCCC2)CCN(C(=O)C)CC1O C1(CNC(C(CC)n2cccn2)=O)CN(C(=O)C(C)n2cccn2)C2(CCC2)C1 c1(C(=O)NC(CC)(C)CNC(=O)CCc2cnco2)nc(C(C)C)oc1C C1(NC(C2CC(=O)N(CC(F)(F)F)C2)=O)CCC(C(N2CCSCC2)=O)CC1 C(=O)(C1=CCCSC1)NC(CCC)CNC(C1CCCCC1COC(C)(C)C)=O c1(C(N2CC3(CCN(C(C4(COC)CCC4)=O)C3)C2)=O)cnc2c(c1)nnn2C N1(C(c2ccc(OC)nn2)=O)C2CCC1C(CNC(C1COCCO1)=O)C2 N1(C(c2ccc(OC)s2)=O)CC(F)CC1C(N1CC2CC1CO2)=O C1(NC(C(C)(C)SC)=O)CCC(NC(=O)Cc2ncc(Cl)s2)CC1 C=C(CNC(C1CC(O)(CC(=O)OC)C1)=O)CCNC(=O)Cc1nocc1C N1(C(C2C(=C)C2)=O)CCCC12CCN(C(=O)CC1CC1)CC2 O=C(CS(=O)(=O)CCO)N1CCC(O)(CNC(C2Cc3cccnc3C2)=O)CC1 Cc1cc(C#N)ccc1C(=O)NCC1CC2CC1CN2C(c1ncccn1)=O c1(OC)coc(C(=O)NCCC2CN(C(C3CC3(F)F)=O)C2)cc1=O C(=O)(CC(C)C(=O)NC(C)C(C)C(=O)NCc1oc(C)nc1C)OC c1(CN(C2CCC(F)(F)C2)C)cccc(C(F)F)c1 C1(NC(c2c(C(C)C)ocn2)=O)CN(C(=O)C(C)(C)O)CC1n1cccn1 CC(F)(F)CCCC(=O)N1CCCN(CCNC(c2ccc(F)o2)=O)CC1 c1(C(=O)NCC2COCCN(C(CCCC)=O)C2)cnc2ncn(C)c2c1 C=CC(C)C(C)C(=O)N1CC2CC(NC(c3cn(C)nc3C)=O)C2C1 c1(C(N2CCCCC(NC(C(C)OCCN(C)C)=O)C2)=O)cncc2nnn(C)c12 CCC(C(=O)N1CC(c2sccc2C)C1)NC(=O)Cc1cccnc1 c1(NC(=O)Cc2cc(-c3cnc4[nH]ncc4c3)ccn2)cnc2ccc(Br)cn12 C1(N(C(=O)CC=C(Cl)Cl)C)CCCN(C(c2cccnc2C2CC2)=O)CC1 C(=O)(CCS(=O)(=O)N(C)C)NCc1nc(CNC(c2ccnnc2)=O)cc(O)n1 C1(C(=O)OCC2COCCO2)CCc2ccccc2S1 N1(C(CNC(C(F)=CC)=O)=O)CCC(N(C)C(c2ccc(SC)o2)=O)CC1 C1(CCC)CCN(C(=O)C(c2cnn(C)c2)NC(c2c[nH]cc2CC)=O)C1 c1(C(=O)NC(CNC(C(CC)(F)F)=O)C(C)(C)C)cccc2sncc12 c1(NC(C(C2CCCC2(C)C)NC=O)=O)ccc(O)cc1.C#CC(C)C1CC1 c1(SCC(=O)N(CCCNC(C(C)Cn2cccn2)=O)C)ccccc1O Cc1ccc2c(C(N3CCN(C(C4(C)CCOC45CC5(F)F)=O)CC3)=O)coc2c1 CC(C)CC(C(N)=O)NC(=O)NCc1cnn(C)c1F C1(C(c2cccs2)N(C)C(=O)OC(C)(C)C)CC2C=CC1N(C(C1CCC1)=O)C2 CC1(CNC(=O)C(c2ccc(F)cc2)F)CCCN1C(=O)CSc1ccccn1 C(CNC(=O)CNC(c1cccnc1)=O)(C(C)(C)C)NC(C(F)=CC)=O N1(CC(=C)C)CCCC(NC(=O)CCOC(C)(C)C)CC1 C1(C(=O)NC(C=C)C2CCC2)CCN(C(=O)C(N2CCOCC2)C)C1C CCC(C)(C)C(=O)C(=O)N1CCC2(CC2NC(c2ccc(CO)s2)=O)C1 c1(N(c2ccccn2)C)ccc(NC(=O)C(N2CCOC3CC23)=O)cc1 CN1CC2(CCN(C(C3(F)CCN(C(C4CC4C(C)(F)F)=O)CC3)=O)CC2)C1 c1(C(=O)NC(C)CC(C)NC(=O)C(N2CCSCC2)C)ccccc1[N+](=O)[O-] C1(C)(NC(C(N2CCN(C)CC2)C)=O)CCN(C(=O)C2=CCOC2)C1 N1(C(C2CN(C)C(=O)N2)=O)C2CCC(C2)C1CC(=O)NCCc1csnn1 c1(C(=O)NCC(CNC(COCCOC)=O)O)cc(O)nc(Cl)c1 N1(C(C2N(C(C)=O)CSC2)=O)CCOC2CN(C(=O)CN3CC(C)C3)CC12 CCS(=O)(=O)CC(=O)N1CCC(C(C)(C)C)(CNC(c2c[nH]cc(Cl)c2=O)=O)C1 c1(C(N2C(CNC(c3ccnc(C)n3)=O)CCC2)=O)cccc2cc[nH]c12 c1(CN(C(C)=O)CC2(F)CC(NC(=O)C=CC3CCCC3)C2)ccc(C)nc1 c1(C(N2CC(C)(C)CN(C(C3CC3F)=O)CC2)=O)cc(F)cc(S(C)(=O)=O)c1 CC(O)C(C)C(=O)Nc1cccc(CNC(c2cn(CCCF)nn2)=O)c1 c1(C(=O)NCCN(CC(C)O)C(c2ccc(N)c(N)n2)=O)ccc(F)c(Cl)c1F C1(CCCC)(C(=O)NC(CN(C(=O)C(C)C2CCOC2)CC)CC)CCC1 CC(CCCCC1CCC1)c1nc(-c2csc(C3CC3)n2)no1 Cc1ccc2c(C(=O)N(CCCCN(C)C(c3ccc(CO)s3)=O)C)csc2c1 Cc1ccc(OCC(=O)NC2CC(C)(NC(=O)C(c3ccccc3)C)C2)cc1C c1(C(=O)NC(C)C(C)NC(=O)CCc2nc[nH]n2)cc(-c2ccco2)no1 C1(CC(=O)Nn2cc(CO)nn2)CCCC1NCC1CSCCS1.c12ccc(o1)C2 C1(C(N(CC(C)NC(CCCC(C)C)=O)C)=O)CC2CC1CC2(F)F C1(CC(=O)NC(C(CN(C)OC)F)=O)(NC(C2CCC2(OC)OC)=O)CCCC1 S(=O)(=O)(c1ccc(Br)c(F)c1)N1CC(C)N(C(=O)Nc2ccc(F)cc2)CC1 CCC(C(=O)OC)C(=O)NCC1(CNC(=O)C(C)C2(O)CCC2)CCC1 c1(NC(=O)COC2CC(NC(=O)CN3CCCC3CO)C2)cnc2ccnn2c1 C(=O)(CC(O)C(Cl)(Cl)Cl)NCC1(F)CC(NC(C(C)C(C)(C)C)=O)C1 C(=O)(CCCCCOC)NC1(C(=O)NCC(C(=O)OCC)C)CSC1 c1(C(=O)NCC2C(Nc3cnc4n3CCC4)CC2O)ccn2nccc2n1 N1(C(C2C(C)C2C)=O)CC(CNC(=O)C(C)(C)CC2CC2)CC(C)(C)C1 C(=O)(C(CC(C)C)SC)NCC12CC(NC(Cc3c(OC)cccc3)=O)(C1)C2 CC1(C(=O)NCC2CCCN2C(C2(C)CNC(=O)C2)=O)CCNC(=O)C1 N1(C(C2CN(C(N)=O)C2)=O)CC(NC(=O)CCc2ncc[nH]2)CC12CCCOC2 N1(C(C(C)NC(N)=O)=O)CCN(C(=O)CCc2nnc(S)n2C)CC1CO C(C)(C)(CC(F)C(=O)N1CC(=O)N(C)C(=O)C1)NC(CCCCC#C)=O C(=O)(C1=CCCCCC1)NCC(C1(O)CCN(C(CN(C(C)C)C)=O)C1)C N1(C(c2c(CC)cccc2)=O)CC2CCC(C1)C(NC(C1CCCOC1)=O)C2 C(C)(CC(=O)OCc1cc(F)ccc1N1CCOCC1)(C(C)(C)C)N(C)C N1(Cc2nnc(CSC)s2)CCC(CC(N)=O)C2(CCOCC2)C1 CC(C)CCC(=O)NCCC(O)CNC(=O)C(C)(C)CN1CCOCC1 C(N=c1[nH]c2c(C)nn(C)c2c(O)n1)C1(Oc2cccc(C(=O)OC)c2)COC1 Cc1cccc(S(=O)(=O)C2CCN(C(c3cc(C(C)C)[nH]n3)=O)CC2)c1 c1(C(=O)NC2C(CNC(CCn3c(C)ncc3)=O)CC2)cc2n(n1)CC(O)CO2 c1(C(=O)NC(C2(O)CN(C(C3ON=C(CC)C3)=O)C2)C)c(F)cc(Cl)cc1F C1(NC(COC(C)=O)=O)CCOC(C(=O)NCC2(CC)CCCCO2)C1 C1(C(=O)NC(CC(=O)OCC)C)CCCCN(C(c2cncs2)=O)C1 N1(C(C2C(=O)NCC2)=O)CCN(C(=O)C=Cc2ccsc2)CC1 C1(CC#C)(C(=O)NCC(C2(O)CN(CCn3cnnc3)C2)(C)C)CCCC1 c1(C(N(CC(C)(C)NC(=O)CC2(C)CC2(Cl)Cl)C)=O)ccc(NC(N)=O)cc1F Cc1nnnn1CC(=O)N(CC(C)O)CCNC(=O)CN1CCCC1CO c1(-c2cn(CC3N(C(CNC(N)=O)=O)CC=C3)nn2)ccc(F)cc1F N1(C(=O)CC23COCC(C2)C3)CCC2(C1)CN(C(c1ccncc1C(F)F)=O)C2 N1(C(CCCC(=O)NCC)=O)CCC2(NC(=O)C=CS(C)(=O)=O)CCCC12 c1(C(=O)OC)cc(Br)c(F)cc1NC(=O)NC1C2CC1N(C(=O)CC(C)O)C2 Cc1cc(=O)oc(C)c1C(N1CCC(O)C(NC(c2ccncc2C(F)F)=O)C1)=O C1(C(N(C(C)CCNC(C2CCC=CCC2)=O)C)=O)CN2CCN1CC2 CCCC(C)(CCCn1cc(C(C)C(=O)NCC(=O)O)nn1)c1ccccc1 C1(C(N(CC(C)(C)OC)C)=O)CC2(CCC2)CN1C(c1cc(CO)c(C)o1)=O C1(NC(c2cnc(CO)s2)=O)COC2(CCCN(C(c3ccc(O)cn3)=O)C2)C1 CC(O)(CC(=O)N1CCCC1)C(F)(F)F.C12C3CN(CC13)C(=O)C13CC(C1)(C3)N2 O=C(CS(=O)(=O)NCCN1CCCC1)NC1C2CN(C(=O)CC3CCCC3)CC12 C(=O)(C(=O)C(C)(C)C)NC(C1(O)CN(C(COc2c(SCC)cccc2)=O)C1)=O c1(C(N2C(CCC)CN(C(=O)Cc3nccn3C)CC2)=O)c(C)nc(O)nc1C C1(NC(=O)NC)CCNC1=O.C(CC(=O)N(C)CCC1CN(C(=O)C(C)C)C1)OC CCCC(C)CCCC(=O)N(C1CCN(C(C2CCOCC2)=O)C1)CCO C1(C(=O)NCCCN(C(=O)C(C)CF)C(C)C)COc2c(F)cc(F)cc2C1 N1(C(c2ccc(C)cc2N)=O)CCC2(CC1)CN(C(c1ccc(C(N)=O)o1)=O)C2 c1(CC(=O)NCC2CC(NC(c3c(CC)[nH]cc3)=O)C2)cccc(C)c1C C1(C2CCCCC2)(C(=O)NC2(CC(=O)OC)CS(=O)(=O)C2)CC1(F)F c1(C(N(CCNC(=O)CCCNC(=O)C(C)(C)C)CC)=O)oc(SC)cc1C CCCCC(C)CCC(=O)OC.C1(C)(C)C(=O)N(C)C2CC(C2)OCC(=O)N1 N1(C(c2cc(SC)ncc2)=O)CCC(NC(c2cc(=O)n(C)o2)=O)C(F)C1 N1(C(CC(C(C)OC)NC(=O)CN2CC3CC3C2)=O)CCCC(C2(C)CC2)C1 N(C(=NCCNC(C1CC1)=O)NCc1ccc(Cl)c(F)c1)C1C(C)CCCC1 C(=O)(C(O)C(C)(C)C)NCC(CNC(C=Cc1ncc(C)[nH]1)=O)O N1(C(CC(CNC(C2COC(C)C2)=O)OC)=O)CC2CCC2(C)C1 N1(C(C2COCCN(C(=O)CCC3CCCO3)C2)=O)CC(O)C(O)C12CCC2 N(C(=NCCC(=O)N1CCC(Cc2ccccc2)C1)NC(C)C)C(CCC)CO N1(CC(=O)NC2C(CNC(C(C)C#N)=O)CCC2)C(=O)NC2(CCOCC2)C1=O C1(NC(CC2CCCC(C)(C)O2)=O)C2CC3CN(C(C4CCCCS4)=O)C1C3C2 Cc1cc(F)c(Br)cc1C(=O)NCC1CCCCN1C(c1ccoc1)=O c1(C(N2CCCC(NC(c3cnn(CCO)c3)=O)C2)=O)cc2cnccc2[nH]1 N1(C(C(COC)OC)=O)CCC(NC(c2cc(OC(F)F)cc(F)c2)=O)C(C)C1 N1(C(C(C)N(C)C)=O)CCC2(NC(c3ccc(C(F)(F)F)cc3)=O)CCCCC12 C1(C(N(CCCCC=C)CC)=O)CCCN(C(=O)CCCn2cccc2)C1 C1(F)(CNC(c2nccc(C)c2N)=O)CCCN(C(C2C3CC(=O)CC23)=O)CC1 N1(C(COCC(=O)NC)=O)CC(NC(c2cccc(C(F)F)n2)=O)CC1(C)C c1(CN(C(C)C)C(=O)Nc2cc3ccccc3o2)c[nH]c2c(Br)cccc12 N1(S(CCOC)(=O)=O)CCCC(C)(C(=O)NC2C3CCCCCC23)C1 Cc1cn(C)nc1C(=O)N(C)CCOCCC(=O)N(C1CCCC1F)CCO c1(OC)ccc(F)c(C(N2CC(F)(F)CC2CNC(=O)C(C)CC2CCC2)=O)n1 C1(C(=O)NC2(CO)CN(C(C(C(=O)OC)C)=O)C2)C2CCN(CC2)S1(=O)=O Cn1cc(C(=O)N(C)CCC2CCCCN2C(=O)C(F)=CCCF)cc1C(=O)NC C1(NC(=O)C#CCNC(c2cccc(C3CC3)c2)=O)C(O)C2CCOC12 c1(OC)ccc(C(C)NCC2CC2(C)C)c(OC(F)F)c1 CCCC(C(=O)N1CCN(C(=O)CS(N)(=O)=O)CC1CC(F)F)S(N)(=O)=O C1(CN(C)C(c2scnc2Cl)=O)CCCN(C(=O)C(F)n2ccnc2)C1 c1(-c2cccc(NC(CSCCC(=O)OC(C)(C)C)=O)c2)nnc2cnccn12 C1(C)(C(=O)NC(CC)CN(C(=O)C=CS(C)=O)CC)Cc2ccccc2C1 C(C)(CCC(=O)N(CCNC(c1c(-c2ccccn2)noc1C)=O)C1CC1)OC c1(CC)ccc(F)c(C(=O)NCC(CC)NC(=O)C(CC)N(C)C)c1 C(C)(C)(CCC(=O)NC(C1CC(NC(CCn2c(C)ncc2)=O)C1)=O)SCC c1(C(C)(C)C)nc(=N)[nH]c(=NCC2CCC3(CCC3)C2NC(c2n[nH]cc2Cl)=O)[nH]1 C1(CC#C)(C(=O)NC2CC(N(C)C(c3nnn(C(C)(C)C)n3)=O)C2)CCCOC1 c1(C(C(=O)NC2(CNC(CSCC)=O)CC2)C)ccc(OC)c(OC)c1 N1(C(C(=O)NCC2(F)CN(C(c3c(C)coc3)=O)C2)(C)C)CCN(C)CC1 Cn1cnnc1CCCNC(=O)CCC1CCN(C(C2CCC3CC23)=O)C1 C1(C(=O)NCCCC(C)(C)NC(C(CN(CC)CC)F)=O)CCn2nncc2C1 CC1c2ccccc2OC1NC(=O)NCCCCN(CCCN1CCC1)C c1(C(CNC(N2CCC(F)(CF)C2)=O)OC)cc(C#N)n(C)c1 Cc1cc(F)cc(C(N2C(CNC(c3ccncn3)=O)CC3COCC23)=O)c1N C(c1ccc(N(C)C)cc1)=C(C(=O)N(C1CN(C(=O)CSC2CC2)C1)C)C#N Cc1ncc(CNC(C2(NC(=O)C(C)C3CCOC3)CCSC2)=O)n1C C1(CNC(CCC#CC)=O)CC(NC(C2SCC=C2C)=O)C12CCC2 c1(OC)ccccc1C1CC1Nc1cnc(N2CCCCC2)cn1 C#CC1(C(N2CC(CNC(=O)CCC=C)C(C(F)(F)F)C2)=O)CC(=O)C1 c1(C(=O)NC2C(CNC(CC)=O)COC2)c(-c2ccccc2Cl)noc1C c1(C(N)=O)cn2ccc(-c3ccncc3)cc2n1.c12cccc(c1)NC(=O)C2 N1(C(Cc2cc(C)no2)=O)CCC(OC2CN(C(=O)CCn3ccnc3)C2)CC1 c1(C(N2CCC(NC(C(CCCC)CC)=O)C23CC3)=O)cc(C)nc2ccnn12 N1(c2n(C)ncc2[N+](=O)[O-])CC2CCC(C1)N2C(=O)Cn1cnnc1SC1CC1 C1(N(C(=O)C(N2CCCCC2)=O)C2CC2)CCCC12CC2.C(C(F)(F)F)NC=O C(=O)(C(CC(C)C)NC(C1CC1Cl)=O)NCc1ncc(C)n1C CCCCC(C)N=c1[nH]c(=NCCOCc2ccccc2)[nH]c2cc[nH]c12 CCC(C)(C)CC(=O)NC1CCN(C(c2c(C)ncn2O)=O)CC1F C(=O)(C1=COCCO1)N(C1CCCN(C(c2snnc2C2CC2)=O)C1)C C1(C(=O)OC)CCC(C(=O)NCC(O)CNC(=O)CC2CCCCC2O)CC1 CC#CCCCC(=O)NC1C=CCN(C(=O)CCn2cnccc2=O)C1 CC1=NOC(C(N2CCC(CC(=O)NC3CC3(C)C(F)F)C2)=O)C1 CCC(C)(C(=O)N1CC=CC(NC(=O)C(C)CO)C1)OC CC(C(F)C(=O)NCC#CCNC(c1cc(C2(C)COC2)no1)=O)C(F)(F)F CC(C)CC(CC(=O)NCC1CC(=O)NC(=O)C1)NC(C1(C2(O)CCC2)CC1)=O c12ccccc1C(=O)S2.C1(NC(=O)CC2(C)CCN2OC)COCC1OC N1(C(=O)CCC2CCCOC2)CC(CO)C2(C1)CN(C(=O)C1=CCCCC1)C2 Cc1cc(CC(N2CCC(CNC(c3cc(C(F)F)[nH]n3)=O)C2)=O)c(C)s1 c1(C(=O)NC(C2CCOC2=O)CC)ccc2nnnn2c1 N1(C(C2CC(C)C2)=O)CCC2(CCCCN(C(C34CCC(C)(CC3)OC4)=O)C2)C1 C1(CNC(CC(CCC)O)=O)CCC(C)(C)CN1C(=O)CC1(O)CCOCC1 c12c(C)n(C)n(c1=O)CC(=O)NC2=O.C(=O)(C1=CCC(C(=O)O)C1)OC(C)(C)C C#CCCCCN=C(NCC1CCOC1C=C)NC1CCOCC1 C(N=c1[nH]cncc1I)C(c1ccc(O)cc1)C(N1CCCC(C)(CO)C1)=O C(N=c1[nH]c2c(c(=NC3CC4CC5C(C4)C35)[nH]1)CCC2)c1c(C)scn1 c1(Cn2c(N(C)C)nnc2C(c2ccccc2F)C)cc2cc(F)ccc2[nH]1 N1(C(Cc2c(C)con2)=O)CCC(OCCNC(c2oc(C3CC3)nc2C)=O)CC1 CCC(C)(CCNC(=O)C(O)C(C)C)NC(C1CCCSC1)=O C1(C)(NC(C(n2cnc(C#N)n2)C)=O)CCCCC1C(=O)NCCc1cn[nH]c1 c1(C(N2CC(CCNC(C(C)CC(N)=O)=O)OCCC2)=O)cccc(C#N)c1F N1(C(c2ccns2)=O)CCC2CCCC12C(N1CCC2CCCC2C1)=O C1(CNC(c2c(C(C)C)nns2)=O)CC2(CC2)CN1C(=O)CC(O)C(C)C c1(NC(c2n(C)nnn2)c2ccc(CC3CCC3)s2)ccc2nscc2c1 c1(NC(C(C=CCCC)O)=O)ncc(C2CC2)cc1C.C12(CC1)CC(=O)N2C C=Cn1nccc1C(=O)NC1CCCC1NC(c1nocc1C(C)(C)C)=O C1(F)(C(=O)NC(CC)C(C)C)CCN(C(=O)CS(=O)(=O)NC)C1 C12(C(=O)NC3C(NC(c4ccc(CO)cc4)=O)COC3)CCC(CC1)OC2 c1(C(=O)NCC2C(NC(Cn3nnc(C(C)(C)C)n3)=O)C2)cccc(Cl)c1O c1(C(=O)NC(C(=O)NC(C)(C)C)(C)C)cccc(OCC(F)(F)F)c1 c1(C(N2CC(OCCNC(CC=CC)=O)C2)=O)cccc2nn[nH]c12 c1(-c2onc(-c3cccc(C)c3)n2)cc2scc(Cl)c2[nH]1 N1(C(C(C)(C)S(C)(=O)=O)=O)CCC2CN(C(C3CCSC3)=O)CC2CC1 C(=O)(C(C)CCC(C)(C)C)N1CC(CNC(CN(CC)CC)=O)OCC1 CCCCCCCCOCC(=O)NCC1CCCC1NC(c1cnc(S)n1C)=O C1(C2CCCO2)(C(=O)NCC(CNC(COc2cn(C)nc2)=O)O)CCCO1 N1(C(C(C)n2cncn2)=O)CCC(CO)(CNC(C2C3CNC(=O)C23)=O)CC1 C1(C)(CC)C=C(C(=O)NCCCN(C(=O)C(C)(O)C2CC2)C(C)C)C1 C1(C(=O)NCC(C)(F)F)(NC(c2cccnc2)=O)CCc2cc(Br)ccc2C1 Cc1noc(C)c1S(=O)(=O)NC(C)C(c1ccccc1)NC1(CBr)CCOCC1 c1(NC)c(C(=O)NCC2CC(NC(=O)CC(C)O)C2)cccc1N c1(NC(COCC2(C(=O)NC3CN(C(C)=O)C3)CC2)=O)ncc(C)o1 N1(C(C2(CC=C)COC2)=O)CC(C2CCCN(C(c3cc(C)ccc3F)=O)C2)C1 C12(CNC(CCCSC)=O)COC(CNC(C3CCC(C)(C)O3)=O)(C1)C2 C1(C)(C(N(C2CN(C(C(c3ccccc3)OC)=O)C2)C)=O)C=CCC1 Cc1nc(CO)ncc1C(=O)NC(C)CC(C)NC(=O)CCC(C)O C1(c2cn(CCCC)nn2)CCCCN1C(C1CN(C(=O)OC(C)(C)C)CCO1)=O CC1CCC(C(N2CC(NC(=O)Cn3cc(Cl)cn3)C3CC23)=O)CC1 N1(C(C2(C)CCN(C)C2)=O)CCCC(NC(c2cccc(CCO)c2)=O)CC1 c1(CC(N2CCN(C3CN(C(CCC=C(C)C)=O)C3)CC2)=O)cn2ccsc2n1 N1(C(CNC(CC)=O)=O)CCN(C(c2cncc(C(F)(F)F)c2)=O)C2CC12 c1(C(=O)NCC(C)NC(C2COCCC2c2ccccc2)=O)ccc(=O)n(C)n1 C1(CNC(=O)COC2CCCCCC2)CC2CN(C(C34CC(F)(C3)C4)=O)CC12 CCCC(F)(F)C(=O)N1CCOCC(C(=O)NC(C)Cc2nn[nH]n2)C1 C1(C(=O)NCC(CNC(c2nc(C)oc2C)=O)F)CC(C)OC(C)C1 N1(C(CC=C)=O)CCC(CF)(NC(=O)CSc2ccccc2C(F)(F)F)C1 C1(C(N(C)Cc2cscn2)=O)CC2(CCN1C(c1ncccc1Cl)=O)CC2 C1(CC)C(=O)NCCN1C(C1CCN(C(=O)Cn2ccnc2)C12CC2)=O c1(C(=O)NC(CC=C)C(=O)N(C)CC2(C)CCCO2)cncc(C=C)c1 c1(C(N2CCC(N3CCN(C(C(C)(C)C)=O)CC3)CC2)=O)cc(Cl)c(Cl)cc1F C1(CNC(C(C)NC(C2CCC2)=O)=O)CC2(C1)CN(C(c1ccoc1)=O)C2 c1(C(C(=O)NC(C(N2CC(OCC#C)C2)=O)C2CCCC2)F)ccccc1 c1(C(N(C)CC2N(C(C=CCCC)=O)CCOC2)=O)c(Br)ccc2c1OCO2 c1(C(=O)NC(C2CCN(C(CSC)=O)C2)C)cncc2nnn(C)c12 c1(CNC(C(=O)OCC)Cc2cccs2)c[nH]c2c(C)cccc12 O=C1CCc2cc(C(=O)N=c3ccn(C4CCOC4)[nH]3)cnc2N1 CC1CC(CNC(=O)CC=CCNC(C2CC3CCC(C2)C3)=O)CC(C)C1 C(N=c1[nH]c(=NC(C)c2nn(C)cc2Br)[nH]c2c1CSC2)c1ccc(C)c(F)c1 c1(CC)cc(C)nc(NCC2(C)CCC(NC(=O)Cc3ncc(F)cn3)CC2)n1 C(=O)(C(C)C(F)(F)F)NC1(CNC(CC2N(C(C)=O)CCOC2)=O)CCCCC1 C1(NC(c2c(C)nn(C)c2)=O)CCN(c2ccn3ccnc3n2)CC1(C)C Cc1ccc(C(=O)NC2CCN(C(C3(C)CCCCCC3)=O)C2C)cc1C N1(C(C=Cc2nc(C)sc2)=O)CCC(CNC(c2ccn(CC#N)n2)=O)CC1C c1(C(=O)NCCC(=C)CNC(c2ccc(C)o2)=O)cn(C)c(C)n1 N1(C(c2c(OC)c(C)sc2)=O)CC(C2CCCCN(C(=O)C(C)(C)SC)C2)C1 C1(CNC(C=C(CC)CC)=O)CCCC12CCN(C(c1nccn1CC)=O)CC2 N1(C(C(CC(N)=O)O)=O)CCC2CN(C(=O)CSC(F)(F)F)C2C1 C12(C(=O)NCC3(CN(C(C(CC)(C)O)=O)C)CC3)CCOC(C)(C1)C2 CCC(CC)(CO)C(=O)NC1CCC(O)CN(C(c2cnn(C)c2)=O)C1 C#CCCCC(C)C(=O)N1CC2CC(C(=O)NC(CCO)C(F)(F)F)C(C2)C1 c1(OC)cc(C(N)C(=O)NC(Cc2ccccn2)S(C)(=O)=O)ccc1Br C12(C(N(C)Cc3cnco3)=O)CC1CCN2C(=O)CCC1(N(C)C)CCCC1 c1(C(=O)NCC(CC=C)NC(C2CCN(C)C2)=O)ccccc1C(=O)NCCO N1(C(c2ccc(CNC(c3cc(OC)ns3)=O)nc2)=O)CCC(CO)C(C)C1 c1(NC(=O)Nc2ccc(C(N(C(C)C3CC3)C)=O)cc2)cc2cnccc2[nH]1 N1(CCOC(Cc2n(C)nnc2)=O)CCN(C(=O)CCNc2cccs2)CC1 N1(C(COc2cc(C)on2)=O)CCCN(C(c2ccnnc2)C2CCC2)CCC1 Cc1cc(C(=O)NC(C)(CNC(=O)C(O)Cn2cncn2)C2CC2)on1 Cc1cc(C)c(C(=O)NCCc2ocnc2CNC(=O)CC2(O)CCOC2)o1 N#Cc1cccc(CN2CCC(F)(C(N3CCC(O)C(O)C3)=O)C2)c1Cl c1(C(=O)NCC2CC(O)(CNC(C3CC3Cl)=O)C2)cc(Cl)ccc1Br c1(C(=O)NCCN(C(=O)CN(C)C(C)=O)CCC)cc2c(cc1N)OCO2 C1(NC(CCNC(c2ccccc2)=O)=O)CC2CN(C(=O)CCOC3COC3)CC12 CCC(CCCC(=O)NCC(=O)OC)NC(c1ccsn1)=O c1(N2CCC(C)(NC(C3C(C)C3)=O)C2)ncnc2cc(C3CC3)nn12 N1(c2ccnc(CC)n2)CCC(F)(F)C(CNC(c2ccoc2CC(N)=O)=O)C1 c1(C(C)=O)ccc(N)cc1.N12CCC(C1)OCCNC(=O)C1(CCC1)C2=O O=C(CC1=CCCC1)NC(Cc1ccccc1)CCNC(c1cncc(Cl)c1)=O c1(NC(C2CC(NC(c3c(C)cc(O)cc3C)=O)C2)=O)ncnc2ccccc12 CCC(C)C(=O)C(=O)NCC(O)CC(=O)N1CCN(CC)CC1 C=CCC(Cc1ccccc1)C(=O)NCCC(C)(C)NC(C1CCN1CC)=O CCC(C)(C)CC(=O)NCCCCNC(=O)C(C)OCCc1ccc(F)cc1 C(CCCCCNC(=O)C(F)(F)c1ccccc1)n1cc(CNS(CC)(=O)=O)nn1 CCC(C)(C)C(O)C(=O)NCC(C)CN(C(=O)Cc1ccc(C(N)=O)nc1)C c1(CN2CCN(CC(c3cccnc3)(C)C)CC2)cc(Cl)cc(Cl)c1 C1(C(=O)NC2CC(NC(c3nc(Cl)sc3C)=O)C2)(COC)CC=CCC1 C(=O)(C1Cc2ccccc21)N1CCC(C(=O)Nc2cc(C(=O)OC)n(C)c2)CC1C c1(NC(C2CN(C(c3scc(C)c3)=O)C2)=O)n[nH]c2ccc(Cl)cc12 Cc1nc[nH]c1CC(=O)NC(C)(CNC(c1ccoc1C1CC1)=O)CO Cc1cccc(CC(=O)NCC2CCN2C(=O)C(C)SC(C)C)c1Br c1(NC(=O)C(C)CC(C)C)cccc(C(=O)NC2C(NC(C)=O)CC2)c1C.C(=O)CO c1(CC)cccc(CC(=O)NC(C)C(C)NC(=O)Cc2nn(C)cc2Cl)c1 N1(C(CC)C(=O)NCC2CCCC2NC(=O)C(C)NC=O)CCOC(C(N)=O)C1 c1(Cc2nc(C)sc2)cn2cc(C(N3CCC(S(C)(=O)=O)C3)=O)ccc2n1 N1(Cc2c(CCC)cccc2)CC2(CN(C(=O)CCc3scnc3C)CCO2)C1 CN1CCOC(C(N2CCC(F)(CNC(C3(C(N)=O)CCCC3)=O)C2)=O)C1 C(=O)(CC(C)(C)CC(F)(F)F)NC1(C2CCN(C(COCC(=O)OC)=O)C2)CC1 N1(C(CCCN(C)C(C2CC3CCC2C3)=O)=O)CCC=C(F)C1 N1(C(Cn2c(C)nc3cc(O)ccc32)=O)CC2CC3(CCS3(=O)=O)C2C1 C1(O)(CN(C(C(COC)N(C)C)=O)C)CCN(C(C2(N(C)C)CCCC2)=O)C1 C(CCCCC(c1nnnn1CCCSc1ccco1)NCC1CC1)OCC C(=O)(C(C)(C)CC(=O)OC)N1C(CNC(CCNC(COC)=O)=O)CC(C)(C)C1 c1(OCC)cnc(C(=O)NC(C)C(C)NC(c2cc(C3CC3)ccn2)=O)c(Cl)c1 Cc1cc(C(N2CCC(C(=O)NC(CO)C3CC3)CC2)=O)ncn1 N1(C(c2c(C)csc2)=O)CCC(C)(CNC(=O)CCCc2cccc(Cl)n2)C1 C1(C)(C(N(CC(C)C)CC#C)=O)CC12CCN(C(C1(N)CCCC1C)=O)CC2 N1(C(CCCN(C)C)=O)CCC2(CC2)CC1C(=O)NCC1(C)C=CCCC1 C1(NC(c2c(OC)nsc2)=O)CCC2CCN(C(=O)CC3CC4(CC4)C3)C1C2 C1(C(N(C(c2cccc(Cl)c2)C)C2CC2)=O)CC2(C1)OCCO2 C1(NC(C2CC(N(C(=O)C(O)C3CC3)C)C2)=O)CN2CCCC1C2 C1(C(F)(F)C(=O)N2CCC(CN(C)C(c3ccoc3)=O)C2)(OC)CCCC1 C(CN(C(=O)CC12CCCC1C2)C)(CO)(CO)NC(C(C1CC1)OCC)=O CC1CC(C(=O)NCCCN2CCC2)CN(C(=O)C(O)c2ccco2)C1 N1(C(c2c(C)nn(C(C)C)c2)=O)CC(C2(NC(=O)C(CO)C(C)C)CC2)C1 C(=O)(C1OCCc2cc(O)ccc21)N1C2CC(NC(c3n[nH]cc3Cl)=O)C2CC1 Cn1cccc1C(N1CCC(CCNC(c2csnc2-c2ccccc2)=O)C1)=O C(=O)(C1=CCCOCC1)NCCC1(OC)CN(C(c2nc(C)ccc2F)=O)C1 C(=O)(CCCN=[N+]=[N-])N1C(CCC(=O)NC(C(N)=O)CO)CCC1 C1(C(=O)NCCCCCCCOC)CC2CCC(C1)N2C(C1CC(CC2CC2)C1)=O c1(C(N2C(C)C(C(=O)NCCN3CCCOCC3)CC2)=O)ccc2[nH]ccc2c1 CC1(C(=O)NC2CC(CCNC(=O)C(Br)=C(C)C)C2)CCCS1(=O)=O CCC(C)CCC(=O)Nc1c(Nc2ccc(OC)cc2)ncnc1C CCC(C)(O)C(=O)N(CCCCCCNC(c1nnn(C)c1C(F)(F)F)=O)C c1(OC)n[nH]cc1C(=O)NCC1(C(=O)NC(c2ncccn2)C)CC1 c1(OCC)ccc(C(=O)NCC(C2CCCC2)OC)nn1.C1(=O)CCC(C)N1 Cc1nccnc1C(N1CCOCC1c1cn(Cc2ccc(F)cn2)nn1)=O C(=O)(CCCCCN=[N+]=[N-])N1CCC(C(C(=O)NCCC2CC(CC)C2)(C)C)C1 N1(C(Cc2c(C)nc[nH]2)=O)CC2(CCNC(=O)CCc3ccncc3)CCC1C2 C1(CNC(CCCN(C)C)=O)(NC(C2CCCN2C)=O)CC(F)(F)C1 C1(CNC(c2n[nH]c3c2CCCCC3)=O)CCCC2(CN(C(=O)CCF)C2)O1 Cn1cnc2nc(NCCCCF)nc(N3CCCC(S(C)(=O)=O)C3)c12 N1(C(C2CCC(=C)CC2)=O)CCC2CN(C(C3CNC(=O)N3)=O)CCC12 c1(CNC(CNC=O)=O)ccc(C(=O)NCc2ccns2)nc1 C1(C(C)C)N(C(=O)C2CC2)CC12CCN(C(=O)C(F)(F)c1cscn1)CC2 c1(C(=O)NCC(C)N(C(C(C)OCC(C)C)=O)C)ccnc2ncnn12 C1(CNC(c2[nH]nnc2C2CC2)=O)CN(C(=O)CCC2CCC2)C2(CCC2)C1 n1(CC)cc(C#N)c(=NC(=O)c2n[nH]c3ccccc23)[nH]1.C12C=CCN1C2=O c1(C(=O)NC2CCC(C)N(Cc3ncnn3C)C2)nccc2[nH]ccc12 C(N=c1[nH]c(N2CCCC(C(C)(C)C)C2)nc2c1CSC2)c1n(C(C)C)ccn1 c1(C(=O)NCC(C)N(C(=O)CC2CC(C(N)=O)C2)CC)cc(C)oc1C C1(NC(C2C(CC)C2)=O)CN(C(c2csc(C(F)F)c2)=O)CC12CCOCC2 C1(C(=O)NCc2occ(C(=O)NCC(C)(O)C3CCC3)c2)C2CCC(=O)C12 CC(C(=O)NC1CCN(C(C2(O)CCCC2)=O)C1)C(C)(C)C c1(OCC)cc(C(C)NC(=O)C(C2CCOC2)OC(C)=O)sn1 c1(C(=O)NCC(CN(C)C(C2CCC2C(N)=O)=O)(C)C)cc(C(F)F)ccc1F Cc1ccc(CO)c(C(=O)NC2CCN(C(=O)Cc3nc(C)sc3C)CC2C)c1 c1(NC)ccc(C(=O)NC2CC(O)CN(C(c3csc(NC=O)n3)=O)C2)cc1F O=C(C#CC1CCCOC1)NC1(C2CN(C(C3CCCO3)=O)C2)CC1 C(c1ccc(C(F)F)o1)=CC(=O)NCCCN(C(C)C)C(c1cn(C)c(O)n1)=O CC1CC1(C(N1CC(CF)C1)=O)NC(=O)CC1CCOC1.C(=O)C1CC1 CCCCC(C(=O)NCC1(O)CCSC1)NC(=O)COC(C)C C(C(C(=O)N1CCCCC1CC1CC1)C(C)(C)C)NC(C(C)=CC1CC1)=O N1(C(c2ccnc(F)c2)C(=O)NCCC2CC2)CCC(C2=NOCC2)C1 c1(OC)ccc(F)c(C(=O)NCC2(F)CC(Nc3ncc(Br)cn3)C2)c1 C12(CCCO1)NC(=O)CCOC2.C(C(=O)N(C)CCO)SC C12(NC(CNC(=O)OC)=O)CCC(CNC(c3sc(C)cc3C)=O)(C1)OC2 c1(CN2C(C(=O)NC(c3ccc(I)cc3)C)CC(O)C2)cc([N+](=O)[O-])ccc1F C1(C(=O)NCC2(NC(CCNC(=O)NC)=O)CCOC2)OCCC1(C)C C12(NC(C3C(C)C3)=O)CC1CN(C(c1cc[nH]n1)=O)C2 CC1(C(N2C3CSCC2C3)=O)CCN(C(C2C3CCC(F)C23)=O)CC1 C12(CCN(C(=O)C=Cc3ncc[nH]3)CC1)C(=O)N2.c1(COC)csnc1Cl c1(C(=O)NC2CCC(COC)C2)cc(CNC(=O)C(O)C(C)C)nn1C c1(OC)ccc(CC(=O)NC(C)CC(C)NC(=O)C=C2CCCCC2(C)C)cc1O CCC(CC)CCC(=O)NC(C1CCN(C(c2ocnc2C(F)F)=O)C1)(C)C C1(C(=O)NC(CCN(C(c2cncc(C)n2)=O)C)C)CC2(CCOCC2)C1 C1(C(=O)NCC2COCCN(C(C(CCC)C(C)C)=O)C2)CNC(=O)CC12CCC2 c1(C(=O)NC23CN(C(C(=O)NC(C)C)=O)C(CC2)CC3)cnn2c1C(=O)NCC2 Cc1cc(C)c(CN2CCCN(c3nc(O)nc(O)n3)CC2)cn1 C1(NC(c2ccc(CSC)cc2)=O)CCCCN(C(C2CC(C)(C)CO2)=O)C1 C1(C(=O)NCCc2ncccc2F)C(C2CC2)CCN1C(=O)Cc1cncnc1 C1(CNC(c2c(CC)noc2)=O)CCN(C(=O)CNC=O)C1c1ccccc1 c1(CC)noc(C(=O)NC2CCC2NC(=O)Cn2[nH]cnc2=N)c1C Cc1conc1CC(=O)N(C(C)(C(=O)N(C)CCn1cnnc1)C1CC1)C CCCCC(C(=O)N1CCC(C(=O)NCC(CC)CC)C1(C)C)C(C)C Fc1ccccc1-c1cscc1CNc1nc(C2CCC2)no1 c1(C(=O)NC2(C(N=c3c(Br)cn(C)[nH]3)=O)CC2)c(Br)c2ccccc2n1C CCCC(C)(O)CC(=O)N1CCC(NC(=O)Cc2cc(C3CC3)nn2C)C1(C)C N1(N(CCOCC)C(C)C)CCCC(C(=O)OC)C1.c1(C=O)oc(C#N)cc1C N1(C(C2C(C(C)C)CCC2)=O)CCC(CNC(c2coc(Cl)c2)=O)CC1 c1(C(N(CC(CNC(CCC=CCC=C)=O)O)C)=O)cc(O)nc(CC)n1 C1(NC(c2c(C)ccc(C)n2)=O)CC12CCC(NC(c1nc(O)c(C)s1)=O)CC2 Cc1ccc(C(=O)NCC2CC2CNC(C2(C3CC3)CC=CC2)=O)c(C)n1 C(=O)(C(CNC(=O)C(C(C)O)NC(N)=O)C(C)(C)C)N1CCC(C)(NC(C)=O)C1 c1(C(N2C(C(C)NC(=O)COc3ccsn3)CC2)=O)cccc2c1OC(C)(C)C2 c1(C(N(CCOCCNC(Cc2c(C)cn(C)n2)=O)C)=O)ccc([N+](=O)[O-])o1 C1(CNC(CCC(C)c2ccccc2)=O)N(C(=O)Cc2cc[nH]n2)CCC1(C)C N1(C(C)=O)CS(=O)(=O)CC1C(=O)NC1CCC(C)N(C(=O)C(O)C2CCC2)C1 CC1=C(C#N)C2=NC3CC34CC(C4)NC(=O)C3(C(=N1)S2)CCCN(C)CC3 N1(C(C=C(CC)C)=O)CCN(C(C2CCC(=O)C2)=O)CC1c1cccc(Cl)c1 CC(c1ccccc1)=CC(=O)NCCC(=O)NCCCN1CCC1 N1(C(C(=O)Nc2c(C3CC3)cc(C)nn2)=O)CCn2c(C(C)C)nnc2C1C c1(NC(C2CCN(C(c3ccccc3Cl)=O)C2)C)ncc2ccnc-2[nH]1 C(=O)(C(CC(C)C)NC(=O)Cc1ccc(Br)c(C)c1)OCC=C C1(NC(c2cnn(CCC)c2C)=O)CCN(C(=O)CC2CCC3CC3C2)CC1F c1(C(=O)NCC(N2CCN(C(CC(C)OC)=O)CC2)C)cccc2c(C)n[nH]c12 C(=O)(CC(C)(C)C(F)(F)F)N1C(C)(CNC(C2(OC)CS(=O)(=O)C2)=O)CCC1 c1(CC(=O)N(C2CC(NC(c3n(SC)ccc3)=O)C2)C)cn(C)nc1C(N)=O c1(C(=O)NCc2occ(C(=O)NC(CN(C)C)CO)c2)[nH]ccc1C1CC1 C(=O)(C1Cc2ccccc21)NCC1CCC(C)CN1C(=O)Cc1cscn1 C(=O)(C1=C(Cl)CCOC1)N1CC(NC(CC2(CC)CCC2)=O)(COC)C1 c1(C(N2CC(OCCNC(c3ccn(CC)n3)=O)C2)=O)ncc(C)cc1OC N1(C(C(C)SCc2cccs2)=O)CCOCC1(C)c1cn(CCN(C)C)nn1 C1(C(C)C)N(C(=O)Cn2cc(-c3cc(N)n(C)n3)nn2)CCC1(C)C N1(C(C2(C)N(C)CCC2)=O)CCCC2(C1)CN(C(c1ccsc1C#N)=O)C2 c1(CC)ccc(C(=O)N(CC(O)CN(C(=O)CCc2csc(=N)[nH]2)C)C)c(C)n1 c1(C(N(C(c2cccnc2)C2CC2C(=O)OC)C2CC2)=O)n[nH]c(C)n1 c1(C(N2C3CC(CNC(=O)C=CCO)(OC3)C2)=O)ccc([N+](=O)[O-])nc1 N1(C(c2nc(C(N)=O)sc2)=O)CCC(NC(c2ccc(Cl)cc2Cl)=O)C(CO)C1 c1(OC)ccc2c(c1)CCC2Nc1ccc2nc(-c3ccncc3)[nH]c(=N)c2c1 CC1CCN(C(c2cnccc2Cl)=O)CC1NC(C1(C(F)(F)F)CCC1)=O C1(NC(CC(C)SC)=O)CCN(CCC2CC3CCC2C3)CC1 c1(C(=O)NCCC2N(C(C3N(C=O)CCC3)=O)CCSC2)ccc2nnnn2c1 N1(C(=O)CN(C)C(N)=O)CC=CC(OCCC(C2CC2)OCC)C1 c1(OCC)ccccc1OCCC(N1CC2CC2(NC(c2cnn(C)n2)=O)C1)=O N1(C(C(c2ccc(OC)cc2)=O)=O)CCN(C(C2CC(C)C2)=O)C2COCC12 N1(C(C2(C)CN(C(c3cc(C#N)ccc3F)=O)C2)=O)CCC2CCCC2C1 N1(C(CC2ON=C(CC)C2)=O)CCN(C(=O)C2=NOC(C(C)(C)C)C2)C2CCC12 C1(NC(=O)CCn2ccnn2)CC2CCC(C1)N2C(C1CC2CC1CO2)=O c1(CC)ccc(C(=O)N(C)CCN(C(C)C(=O)NC)C)o1 n1(C(CC)C)cc(C(C(=O)NC(C)C)N2CCC2C2CCOCC2)cn1 C1(CNC(CC2(C(F)(F)F)CC(=O)NC2)=O)CC2(CCOCC2)CO1 N1(C(C(CC=CC)C)=O)CC2CCC2(CNC(=O)COCCCF)C1 C1(C(=O)NCC(C)CN(C)C(C2COCCN2C)=O)CC(=O)NC(=O)N1 CC(C)CC(C)(CNC(C1CCCC(N(C)C)C1)=O)NC(=O)CSS(C)(=O)=O C=C=CCCC(=O)NC1CCOCC1C(=O)NCC1(C)CC(O)C1 CC1CCc2ncc(C(N3CC(NC(=O)CC(C(F)F)n4cccn4)C3)=O)n2C1 C1(OCCOCC(=O)NC2CCCCC2)CCCCN(C(=O)CSC(F)(F)F)C1 n1(CC(=O)NCC(CN(C)C(C2CCCCC(=O)N2)=O)O)ncc2ncccc12 C(c1ccc(=N)[nH]c1)=CC(=O)NCC1OCCN(C(c2c(C)ncn2C)=O)C1 N1(C(C2(CCOC)CC2)=O)CC(N(C(=O)Cc2cncnc2)C)C(C)(C)C1 c1(N(CCOC)CCNC(c2nnnn2CC(F)(F)F)=O)cnc2n1CCC2 C1(NC(C(C(C)C)NC(C)=O)=O)CCN(C(C2(C(F)(F)F)CCC2)=O)CC(C)(C)C1 CC1=NC(C(=O)NCC2CCCN2C(N)=O)CS1.C(=O)(CCC)N(C)C c1(C(N2CC(CC)(NC(=O)CCOCCC(C)(C)C)C2)=O)cccc2ccnn12 c1(C(=O)NCC2C(C)CN(C(C3COC(C)(C)C3)=O)C2)c(F)ccc(F)c1F C12(NC(CC3(OC)CC3)=O)CCN(C(c3ccn(C(C)C)c(=O)c3)=O)CCC1C2 C1(C2CC2)(C(=O)NC(C(C)NC(CCc2c(C)cccc2)=O)CO)CC=CC1 C(=O)(C1COc2ccc(Cl)cc21)N(CC(O)CNC(C1CC(C)(C)CCO1)=O)C CC(O)(C(=O)NCC1(NC(=O)Cc2nnc(-c3ccco3)o2)CC1)C(F)(F)F C(=O)(C1=CCC2CCC1N2C(=O)CCOCC(F)F)NCCc1c(C)nc[nH]1 C(CCCCCC(=O)N(CC(C)O)CCOC)NC(CCC(=C)Cl)=O CCCCCCC(C)C(=O)NC1CC2CC1N(C(c1ccc(C)nc1NC)=O)C2 N1(C(C(C)OCCC#C)=O)CCC2(C1)CN(C(c1cc(C(=O)OC)no1)=O)CCO2 C12(NC(C(C)CF)=O)CCCC1N(C(c1cc(-c3ccncc3)on1)=O)CC2 CCC(O)C(F)(F)C(=O)N1CCCOC(CCNC(=O)CN2C(=O)CCC2=O)C1 C1(C(=O)NC2CCN(CC(=O)NC(C)CCN3CCCC3)C2)(OC)CCOCC1 N1(C(CC(=O)OC)=O)CCCCC1CCNC(c1c(C)ccn1C)=O CCC(CC(F)(F)F)C(=O)N(C)CCN(C)C(c1ccc(SC)cc1OC)=O C1(C(N(CCCNC(C2(n3cccn3)CC2)=O)CCC)=O)CCN(C)C1CC CC(C)C(C(=O)NCC1CC1NC(=O)CCCc1ccncc1)NC(=O)N(C)C C1(NC(CN(CCC)C)=O)CCCC1CNC(=O)C(C)COC C(N=c1[nH]c2c(c(=NCCN3CCCOCC3)[nH]1)COC2)c1c(C)nc(F)cc1 C1(NC(c2c(C)csc2)=O)CCN(C(C2CCN2C)=O)C1c1ccccc1 C1(N(C(Cc2c(C)n[nH]c2)=O)C)CN(C(=O)CCC(=O)c2cccs2)CCC1C CC1(C)C(C(=O)NCC(c2ccccc2)C2CC2)CCN1C(c1cnns1)=O C1(Cn2c(-c3c(C)n(-c4ccccc4)nn3)nc(C3CC3)n2)CCCC(C)(C)C1 CN1CC2CCCC(C(=O)NC3(CO)CCOC(C)(C)C3)N2C1 c1(C(=O)NC2(CNC(C3=NNC(=O)CC3)=O)CCC2)cccc2ncccc12 c1(C(N2CCN(c3nnc(C)s3)CC2)=O)c(F)ccc(S(C)(=O)=O)c1F c1(C(=O)NCC(C)CN(C(=O)CC2CC3(CC3)C2)C)ccc2c(c1)COB2O CC1(C)CCC(O)(NC(=O)NC2(c3ccccc3)CC2)CC1 C1(C(=O)NCC=CCNC(C2(C(F)(F)F)CCO2)=O)CCC1(F)F C1(S(C)(=O)=O)(C(N2CCC(N(C(=O)C(C)(C)F)C)C2)=O)CCC1 C1(CCNC(c2cnc(OCC)s2)=O)CN(C(=O)CC2(C)CC2)CCS1(=O)=O C1(C(=O)NCC2CC(NC(C(CC=CCC)C)=O)C2)CCCC1C1CC1 C1(C(C)(C2CC2)CC)CC(C)(C)CN1C(=O)C=Cc1ccc(CSC)s1.C(=O)(C)O c1(C(N2CC3CCC(NC(C=CCC)=O)(C2)C3)=O)c(F)c(F)c(F)c(F)c1F C1(C(=O)NCCCN(C(C(C)OCCOCC)=O)C2CC2)COCCN1C C1(COC)CN(C(c2cnc(C#N)s2)=O)CCN1C(=O)Cc1cccnc1OC [N-]=[N+]=NC1CC(C(=O)NCC23CC(CN2C2CC2)C3)N(C(=O)CN2CC3CC3C2)C1 C1(CCOC)(NC(C2(O)COC2)=O)CCN(C(C2CC(C)(C(C)(C)C)C2)=O)CC1 N1(C(c2c(OC)n[nH]c2)=O)CC2(CCOCC2)CC1CNC(c1ncsc1C)=O Cc1cc(C(N2CC3CC3(CNC(=O)C=CC3CCCC3)C2)=O)c(N)cc1F Cc1cc(COC(C2(c3noc(C(F)F)n3)CCCCC2)=O)ccc1F C(CC(C)C(=O)NCC1CCN(C(C2CC3CCC2C3)=O)C1)=CC N1(C(C(=O)NCCCSC)C2CCCC2)CCC(F)(c2cccnc2)CC1 C1(COC)CN(C(=O)CN(C(=O)CC2(O)CCC2)C2CC2)C1(C)C C1(C(N2CC(C(=O)NC3COCC3C)(CC)C2)=O)CC2(C1)CC(O)C2 Cc1ccc(C)n1CC(=O)NC1(C)CN(C(=O)C(O)C(F)F)C1 N1(C(CC2(OC)CCC2)=O)CC(=O)NCC1C(N1CC2CCCCC12)=O C1(C(=O)NCCC(=O)NCC(=C)C)(CNC23CCC2C3)CCCN1C(=O)OCC C12(C(=O)NCC(CNC(c3cn(CC(C)C)nc3)=O)CO)C=CC(C1)OC2 C(c1cccnc1)=C(C)CNC1CCC(NC(C2C(C)C2C)=O)C1 C1(C(=O)NC2(COCC)CC2)CCC=CCC1.c12cncnc1C(=O)O2 c1(C(N2CC(COC)(CNC(C3CCN(C)C3)=O)C2)=O)cnc2sc(C)c(C)n12 Cc1nnc2n1CC(C(=O)N(C)CCNC(=O)COCP(C)(C)=O)C2 c1(C(=O)NCCN(C(c2cc(C#N)c(N)cn2)=O)CC)ccc(S(N)(=O)=O)cc1 N1(C(C(C)CC2CCCCC2)=O)CCN(C(=O)CSC2CC2)CC1CC1CC1 Cc1ccc(CN=C(NC2CCC2)NC2CCCC(C(F)(F)F)C2)cc1 C1(C(N2CCC(N(C(=O)CCC3CC3CC3CC3)C)C2)=O)CCC(F)(F)CC1 C1(C(=O)NC2(c3nn[nH]n3)CC2)C=CCC(NC(c2c(C(C)C)c[nH]n2)=O)C1 n1(CC)ccnc1C(=O)NCCCCCNC(=O)C(Cc1ccccc1)C1CC1 C=CCC(C)(CC)C(=O)N(C)CCOCCNC(=O)C(c1ccncc1Cl)C N12CCCCC1CC(=O)NO2.C1(NC(CC=C)=O)CC=CCC1 c1(C(N2CCC(C(=O)NCc3ccccc3F)C2)=O)ccc2ccsc2c1 C(=O)(C#CC1CCCCC1)NC(C(=O)OCC1CC(OCC)C1)CC(C)CC c1(CC)cc(C(N2CCN(C(=O)CSCCN(C)C)CC2COC)=O)ccc1C Cc1ccc(C(N2CCCC(N(C(=O)CCCC3CCC3)C)CC2)=O)cc1N C1(C(=O)NCC(C2CC2)NC(c2c(C)nc(COC)s2)=O)CNC(=O)CC1(C)C C(=O)(CCC(=O)C(C)(C)C)N(CC(=O)NC(C#C)CC1CC1)C1CCC1 c1(C(N2CCC(N(C(=O)CCN3CCCC3)CC)C2)=O)cc(F)cc2nn[nH]c12 Cc1noc(C)c1CC(=O)NCCOC1CN(C(c2cc(C3CC3)ccn2)=O)C1 C1(C(=O)NC2CC(CNC(C(CC)N(CC)CC)=O)C2)CC2OC1C1CC21 N1(C(=O)N(n2cccn2)C(c2cccc(F)c2)C2CC2)CCN(CCCO)CC1 c1(NC(c2ccccc2)CF)[nH]c(=NCCC2CC3(CCC3)C2)nc2scnc12 N1(C(c2c(C)nns2)=O)CCCCC1C1CCCN(CC2CCCCO2)C1 Cc1cccc2cccc(C(=O)NCC3(C)CCN(C(=O)C4=CCSC4)CC3)c12 C1(NC(C2C(C(C)C)OCC2)=O)CCCCCC1C(=O)N1CCCO1 c1(C(C)(C)C(N2CCN(C(c3ccc(S)cc3)=O)C3CC23)=O)ccc(C#N)nc1 C(c1nc2ccccc2o1)=CC(=O)NC(C(C)C)CNC(=O)C(CO)C(C)(C)C C1(C(=O)NCC2C(NC(CN3CC(CC)C3)=O)C2)CCN(C2CCCCC2)CC1 c1(C(N2CCC(C)(CCNC(C3N(C)C(=O)CC3)=O)C2)=O)ccc2ccoc2c1 c1(OC)cc(CCCN2CCCC(CO)CC2)cc(-c2ccccc2C)c1O N1(C(c2cn3ccsc3n2)=O)CCC2(CCCN2C(c2n[nH]cc2C2CC2)=O)C1 CC1C2CCC(C2)C1C(=O)NC1CC(n2cc(C3CCN(C)C3)nn2)C1 C1(C(N(CCNC(c2cnc(C)[nH]2)=O)C2CC2)=O)Cc2nn[nH]c2C(C)C1 C1(c2cc(C(=O)OCC=C)on2)CCN(C(=O)CCNC(C)=O)C1 N1(C(C(c2ccccc2F)OC)=O)CC2(CCN2C(=O)C(C)(C)C(N)=O)C1 N1(C(C2C(C)OCC2)=O)CCC(NC(c2ccc(C3(C)CCO3)cc2)=O)C1(C)C C1(C(=O)NC(c2nocc2C(=O)NCCS(C)(=N)=O)C)CC(=O)C1(C)C C(=O)(CCCC(C)(C)C)NC1C(CC)CN(C(c2ncoc2C2CC2)=O)CC1 c1(C(N2C(CNC(=O)Cn3ccnn3)CCC2)=O)ccc(-c2cn[nH]c2)cc1Cl C1(C(=O)NOCC2CC23CC3)(COC)C=CCN1C(=O)CC1(C)CCCCC1 C1(C(N(C)CC2N(C(CCC)=O)CCCC2)=O)Cc2cc(Cl)ccc2O1 C(=O)(C(C)C(C)S(C)(=O)=O)NCC1CC(C)N(c2ncc3c(n2)COC3)CC1 c1(COC)ncc(NC(=O)C(O)C2CN(C(=O)Cn3cnnc3)C2)cn1 C1(C(=O)NCCN(C2CCCCC2)C(c2c(OC)c[nH]n2)=O)(CF)CNC(=O)C1 C(=O)(CC(O)CNC(C12CC1CCN2C(=O)Cn1cncn1)=O)OC c1(-c2cc(C(N(C)CCNC(c3ccncc3)=O)=O)on2)ccc(Cl)cc1 CC1=NC(C)(CNC(=O)C(CCN(C)C)NC(c2ccn(C)c2C)=O)CS1 C1(CNC(CNC(=O)OC)=O)N(C(C2CCCN2C(C)=O)=O)CCCC1(C)C C12(CC)CC(CNC(C3(C(C)C)CCN(C(=O)OC(C)(C)C)C3)=O)(CO1)C2 C=C(Cl)CC(C(=O)N1CCC(C)(CC)C1)NC(c1nn(C)cc1C)=O c1(CCC)nccc(=NC(=O)C(c2ccccc2)Nc2cc3ccccc3[nH]2)[nH]1 N1(C(c2c(C)noc2)=O)CCN(C(C2CCS(=O)CC2)=O)C2(CC2)C1 O=C(C1=CC2C=CC(C1)C2)NC1(CF)CCN(C(=O)C(O)Cc2cnc[nH]2)C1 N1(C(C)=O)CCC2(COC)CN(C(c3cc(OC(F)F)ccc3C)=O)CC2C1 C(=O)(C(F)CC(C)(C)C)NC(CC#CC)C(=O)NCCC1CCCO1 C(C(CCO)NC(=O)CCC1(C)CN(C(=O)C(F)F)C1)N(C)C C(=O)(C(C)CN(C)C)NCC1CC(CNC(CN(C2CC2)CC)=O)C1 C1(C(C)(OC)OC)CCCCN1C(=O)N.c12[nH]c(nc1C)CNC2.C(C)(C)(C)O C12(NC(c3c(C)cc(F)s3)=O)CCN(C(c3coc(CO)c3)=O)CCC1C2 c1(OC)cnc(C(=O)NCCC2(OC)CN(C(c3ccc(C#N)o3)=O)C2)c(F)c1 CCCC(CC)CCC(=O)NC1CC(F)(CNC(C2(CC)CC2)=O)C1 c1(CNC(C2(CNC(=O)NCC)CC2)CCF)c[nH]c2cc(C)ccc12 Cc1cc(C(C)(C)C)oc1C(=O)NNC(=O)NCC1(C)CCOCC1 C1(CC(N2C(CN(C)C)CC2)=O)C2CN(C(=O)CCCOC3CCC3)CC12 c1(C(N2CCC(N(C(=O)Cc3csc(Cl)c3)C)C2)=O)cn(C2CC2)nc1C(F)(F)F C=CCCCC(=O)N(C1CCN(C(=O)CC(n2nc(C)cc2C)C)C1)C c1(C(=O)NCC(C)(CO)NC(C2CCN(C)C2)=O)ccncc1Br N(C1c2ccccc2CC1NC(c1cc2n(n1)CCC2)=O)C(CCC(C)(C)O)=O C12(CC)CC(C(=O)NCC(O)CNC(=O)C=Cc3ccn(C)c3)(CO1)C2 CC(C)C(C)(O)C(=O)NCCCN1CCC(NC(=O)CC2COCC2O)C1 Cc1ccc(S(=O)(=O)N(C)C)cc1C(=O)NC(C1CCCO1)CO CC(CCCNC(c1coc(C2CC2)n1)=O)NC(=O)CCn1cc(Cl)cn1 O(N1CCC(NCC(C(=O)OCC)C)CC1)Cc1csc(C#N)c1 CC1CN(C(C2CC(=O)N2)=O)CCCN1C(C1CCC(=O)N(C)C1)=O N1(C(C(=O)NC2CCCO2)C2CC2)CCC(N=c2nn[nH]n2C)C1.CO c1(CC(=O)N(C)CCN(C)C(c2ncn(C)n2)=O)c[nH]c2cccc(Cl)c12 N1(CCNC(=O)CCC2CCCO2)CCN(C(=O)CCOCC2CC2)CC1 CCCC(O)CC(=O)N(CCCCNC(=O)CC(C)F)C(C)C C(N=c1[nH]cc([N+](=O)[O-])c(O)n1)C1C(C)CN(C(=O)Cc2cncn2C)C1 C1(CNC(c2n(C)ccn2)=O)CCC(CNC(=O)Cc2csc(S)n2)CC1 c1(C(N2CC(C)(NC(C(c3n(C)cnc3)O)=O)C2)=O)ccc(F)c(F)c1 C1(CNC(=O)NCCC(=O)N(C2CCCCC2)C)OCCC1NC(=O)C(C)(C)C c1(-n2cc(CC(C)N(C(COC)=O)C3CCC3)nn2)ccc(S(C)(=O)=O)cc1C CC(C(=O)NCC1CC(F)(CNC(c2ccncc2C2CC2)=O)C1)C(F)F CC(C)C(C)(O)C(=O)N1CCCC(NC(=O)CCC(N)=O)C1C c1(C(=O)OCc2coc(Br)n2)cccc2ccc(O)nc12 C1(CNC(C(C)=C2CCC2)=O)CC2(CCN(C(=O)C=C3CCN(C)C3)C2)CO1 C(C(CNC(=O)CCCCc1cn(C(C)C(=O)O)nn1)C(C)C)OC N(C(=S)N1CCC(CO)C(F)C1)C(C)(C)C.C(N)=O c1(C(=O)OC)cnc(Cl)[nH]c1=NC(=O)c1n[nH]cc1-c1scc(C)c1C c1(CNC(C2CC(NC(=O)COCC(F)(F)F)C2)=O)c(F)cccc1F C1(CC(=O)NCCN(C(C2(CO)CC2(F)F)=O)C2CC2)CC2CCC1O2 CCC(C)C(C(=O)NC(C)C(N1CCCC1)=O)NC(c1nnc(S)n1C)=O C1(NC(CCn2c(CC)ncc2)=O)(CNC(=O)CO)CCCCC1C.C(C)(C)(C)N O=C(C1=CCS(=O)(=O)C1)NCC1CCCC(NC(=O)C2=C(Cl)CCOC2)C1 N1(C(C2=CCCN(C(C(C)OCC(C)C)=O)C2)=O)CCC2(CCN(C)C2)C1 c1(C(=O)NCC2C(C(=O)Nc3c(CC)nsc3)CCCC2)cccc(O)c1F C1(C(=O)NC(C(=O)OC)C2CCC2)CCN(C(=O)C2(C)CC(=O)N(C)C2)O1 c1(NCC2(OC)CCC2)ncc(C)cc1S(=O)(=O)NC(C1CCCC1)C1CC1 N1(CC)C(=O)CCC1C(=O)NCCNC(C1(Br)CC1(F)F)=O c1(C(N2CCC(NC(c3cc(C)ncc3)=O)C(F)C2)=O)ccc2cn(C)nc2c1 c1(C2(C)C(=O)N2)ccc(C(F)(F)F)cc1.C1(NC(CC)=O)CC(CF)C1 N1(C(C(C=C)OC)=O)CCC(C)(NC(c2cncnc2C)=O)C1 C1(COC)CN(C(C2(C(=O)OC)C=CCC2)=O)CCN1C(=O)C=CS(C)=O C(=O)(C(C)C(C)c1ccccc1Cl)NC(C1(O)CN(C(C2(C)CCC2)=O)C1)C c1(CC(N2CCC(CN(CC(=O)NC)C)CC2)=O)n[nH]c2ccccc12 c1(C(=O)N)cc2ncccn2n1.c1(COC)nc(NC2CC(CC)C2)cc(O)n1 N1(C(C(CCOC)OC)=O)CCC(C(N2CC(N3CCCC3)C2)=O)C12CC2 C1(CC)(OC)CN(C(=O)CCc2ccc(C(=O)OC)o2)C1 c1(C(=O)NCC2COCCN(C(C(C=C)(C)C)=O)C2)c(C)cc(Cl)cc1[N+](=O)[O-] c1(C(=O)NC(CNC(C2C(C(=O)OCC)C2)=O)C)cc(C)c(F)cc1Cl C1(C(CNC(c2cc(COC)no2)=O)(C)C)CCN(C(C2CC(=O)N2)=O)CC1 c1(C(=O)NC2(CNC(C3N(N=O)CCCC3)=O)CCOC2)ccc2[nH]ccc2c1 c1(CC)nc(C(N2CCCC(N(C)C(c3oc(Br)cc3C)=O)C2)=O)c(N)s1 N#Cc1ccc(C(=O)NCC2CCCCN2C(c2ccc(O)c(Cl)n2)=O)cc1 C1(c2onc(COC)n2)(C(=O)Oc2cccc(C#C)c2)CC2CCC1CC2 c1(C(=O)NC(CN(C(=O)CCc2cn[nH]c2)CC)C)cc2c(C)nn(C)c2s1 CCCCCCC(C)CC(=O)N1CC2(C1)CN(C(=O)C=CCn1cncn1)C2 C1(C(=O)NCC2(F)CCN(C(c3cccc(C)n3)=O)C2)Cc2nnsc2S1 Cc1ccc2oc(N3CC4CC(NC(=O)C(C)(C)N(C)C)CC(C4)C3)nc2c1 c1(OC)ccc(C(=O)NC2COCCC2NC(=O)Cc2ccno2)c2[nH]ncc12 C1(OCC)CC2CN(C(=O)CC3(N(C(=O)CC4CCCN4C)C)CC3)CC12 C(=O)(C1=CC(O)C(NC(C2CS(=O)C2)=O)C1)NCCN(C1CCCC1)C C1(NC(=O)CSc2cn[nH]c2)CCCN(C(=O)CNc2cncc(Cl)n2)C1CO C1(C(N2CCC3(CC(NC(CC=C)=O)C3)CC2)=O)CC12CCOc1ccccc12 N1(C(c2c(C)nc[nH]2)=O)CC2CCCCN2CC1CNC(=O)Cc1c[nH]nc1C n1(CCC)cc(C(=O)NCC(C)NC(c2cc(-c3ccccc3)c[nH]2)=O)c(C)n1 C1(NC(=O)CC(C)CF)CCC(F)(NC2(C3N(C(COCC)=O)CCC3)CC2)C1 N1(C(C2CN(CC)C(=O)N2)=O)CCC2CCN(C(c3cnc(C)nc3C)=O)CC12 c1(C(=O)NCCCN(C(C=C(CCC)C)=O)C(C)C)c(C(C)C)cccc1C CC1CN(Cc2cccnc2F)CC1Nc1ccccc1-n1cccc1 C1(N(c2ccccc2)C(CC=C)=O)CC(C2CCN(C(=O)CC(C)N(C)C(C)=O)C2)C1 CC1(C)CCCN(C(=O)Cc2c(F)cccc2Cl)C1CNC(=O)Cc1cc[nH]n1 c1(C(=O)NC2(CN(C)C)CCCCC2)cncc2n[nH]c(N)c12 C1(OC)CN(C(=O)CCCSC)CC1C(=O)NC1(NC(=O)CC2CC=CC2)CC1 C(=O)(CC(C)C(=O)N1CCC(C)(NC(=O)CSc2cccc[n+]2[O-])C1)OCC C1(N(C(=O)CC2CC3CC3C2)CC#C)CCN(C(C2CCCOCC2)=O)CC1 Cc1c(C(N2CCN(C(C3CN(C(N)=O)C3)=O)CC2C)=O)cncc1F c1(CC)cccc(C)c1C(=O)NCC12CC(NC(=O)C(C)CSC)(C1)C(C)O2 CC(CCC(=O)N(CCNC(=O)Cc1ccc(Br)nc1)C1CC1)N(C)C N1(C(CN2CCN(C)C(=O)C2)=O)CCC(C2(C)CC2)C1 C1(NC(C23OCC(C(C)C)(C2)C3)=O)CC2CN(C(C3CC34CCCC4)=O)CC2C1 c1(C(=O)OC)nc(Br)c[nH]c1=NC(=O)c1cc(-c2ccccn2)[nH]n1 c1(C(N(C2CC(NC(=O)COc3cccnc3)C2)C)=O)cnn(C)c1Cl c1(NC(C2C3CC2N(C(=O)CN2CCSCC2)C3)=O)cc(CO)ccn1 C(c1cccc(Br)c1)=CC(N1CCC(O)(C2(NC(=O)CCN3CCC3)CC2)C1)=O Cc1nc(Br)sc1-n1cc(CNC(=O)C(N2CCC(CC(F)F)C2)=O)nn1 Cc1nc(C(C)(C)C)sc1C(=O)NC1(C)CCN(C(=O)C=CC2CCCCC2)C1 N1(C(CCSC)=O)CC2CN(C(c3ccnc4c3CCC4)=O)CCC2(CO)C1 CON(C)C(=O)CCCCCNC(c1cc(Cl)ccc1C)=O n1(C(C)C)ncc(C(=O)N(C)CC2CCCN2C(=O)C=CC(C)(C)C)n1 N1(C(C2CC(CC)N(C(=O)Cc3cn(C)cn3)CC2)=O)CCN2CC(C)CC2C1 C(=O)(C1Cc2ccc(Cl)cc21)N(CC(C)N(C(=O)CSCc1ccncc1)C)C c1(CC(=O)NC(C(C)NC(C2C(CCC)CCC2)=O)C)cccc(C(F)F)c1 N1(C(C(C=C)(C)C)=O)CCC(NC(c2ccn3cccc3c2)=O)C2(CCC2)C1 N1(C(=O)CC2OCCO2)CC2(C(=O)NCC(O)C(F)(F)F)CC1CO2 N1(C(c2c(C)cco2)=O)CCCC(C(C)NC(c2cn(C(C)C)cn2)=O)C1 C1(NC(C(C)OCC#C)=O)CC(O)CN(C(=O)Cc2cc(Cl)ccc2Cl)C1 c1(C2CC(=O)O2)ccc(F)cc1F.c1(CCOC)ccc(CO)s1 c1(NC(C=C2CCN(C(c3ccc(C)[nH]3)=O)CC2)=O)cc2nncn2cn1 C1(CNC(=O)CSC2CC2)CN(C(=O)CC(C(F)F)n2ccnc2)C2(CCC2)C1 n1(CC)cc(CCNC(=O)C(Cn2cccn2)NC(=O)C(C2CC2)C2CC2)nn1 c1(C(C(=O)NCC2CCCO2)N(C(C#C)C)CCCC)ccsc1C CC(C)(CC=CCNC(c1cn(C(F)F)cn1)=O)NC(C1CCC1)=O c1(OC)ccc(C(N2CCOC(C(N3CCC(CCF)CC3)=O)C2)=O)cc1 c1(CN(C(c2cc(C(C)(C)C)ccn2)C(=O)NC2CCOC2)C)cccc(Cl)c1 CN1CC(NC(=O)C(CNC(c2cnco2)=O)CC2CCCC2)CC1(C)C C1(C(=O)N(CCN2CCN(c3ccnnc3)CC2)C2CC2)CC(C2CC2)=NO1 CC1(C)CC(NC(C2(CO)CCC2)=O)CCN(C(=O)Cc2nc(C3CC3)cs2)C1 C1(CCO)(NC(C2(CC)CCCO2)=O)CN(C(=O)C(C)NC(C)=O)C1 O=C1OC(C(=O)NC2(CNC(C3(O)CC3)=O)CC2)Cc2ccc(Br)cc21 c1(C(=O)NC2C(CNC(CCc3cnn(C)n3)=O)C2)cnc2cc[nH]c2c1 N1(C(CNC(=O)CC(F)(F)F)=O)CC2CN(C(=O)CC3=CCCC3)CC2C1.C1CO1 c1(C(=O)NC(C)CCCCNC(c2ccn(C3CCC3)n2)=O)cccc(Cl)c1F c1(N(CCOC)CCNC(C2CC2c2ccn(C)n2)=O)cc(OC)ncn1 C1(F)(CNC(c2c(C)snc2)=O)CCCN(C(=O)CCNS(C)(=O)=O)C1 CCCC(CCC)C(=O)NC(CC(=O)NCC1(CC)CCOC1)C1CC1 c1(CNC(C2COCCN2Cc2ccc([N+](=O)[O-])o2)=O)c(Cl)ccc(F)c1Cl c1(CC)cc(C(=O)N(CCCN(C(=O)COc2cccnc2Cl)C)C)ncn1 c1(C(C(=O)OCC)(F)F)n[nH]c(=NC(=O)N2CC3(C2)CN(C(C)=O)C3)s1 N1(C(c2c(C)cno2)=O)CCC(NC(C2CCN(C)CC2)=O)C(O)C1 c1(CN2CCC(N3CCC(NC(C#C)=O)C3)CC2)c(OC)cc(Br)cc1F C1(CC=C)(NC(=O)CC(C)(F)F)CCN(C(C2CC(C(F)(F)F)C2)=O)CC1 N12CCCC3(CC3C1)Nc1cc([nH]n1)C2=O.c1(C(C2(C)CCC2)=O)coc(C)c1 c1(OC)c(-c2cn(Cc3cncc(Cl)c3)nn2)cc(Cl)cc1Cl C12(NC(C(=O)NCC)=O)CCC(CN(C(=O)C(C)Oc3ccc(Cl)cc3)C1)C2 N1(C(C=CCC)=O)CC(CNC(c2c(C)ncnc2O)=O)C2(CCC2)C1 C1(OC)CCN(C(=O)CC(C)(C)n2cc(NC(c3cncs3)=O)nn2)CC1C C1(C(=O)NCCCCC2(C)N=N2)CCC2CN(C(c3ccoc3Cl)=O)CCC2C1 C1(C2CCC2)(CNC(C=CCN(C(C2(CCC)CC2)=O)C)=O)CC1 C1(NC(C=CCC)=O)CCN(C(c2ccc(C(F)(F)F)o2)=O)C(C2CC2)C1 c1(OC(C)CNC(=O)CC(C)(O)C2CC2)ccc(Cl)cc1 C(=O)(C#CC(C)(C)O)N1C(C)(Cn2cc(-c3ccc(C(C)C)s3)nn2)CCC1 c1(C(=O)NC(CC)CN(C(c2cccc[n+]2[O-])=O)CC)cccc2cccnc12 C1(OCC)(CNC(C)CC(=O)N2CCCCC2)CCSCC1.C(=O)OC C12CCCC1NC(=O)C2.C(=O)(CCN(C(=O)C(C)SC(C)C)C(C)C)OC C1(C(=O)OC)C(c2ccccc2)CCN1C(=O)CCC1CC1C1CC1 CC(N=c1[nH]c2c(c(=NCC3(C)CCC(=O)N3)[nH]1)CSC2)c1ccc(N(C)C)cc1 C1(NC(C2CCCOC2)=O)CC1C1CCCN(c2ncncc2I)C1 N1(C(C2(C)N(C)CCC2)=O)CC2CCC(C1)N2C(=O)COC(C)(C)C(F)(F)F c1(C(=O)NC2CC(NC(CCCc3onc(C)n3)=O)C2)cccc([N+](=O)[O-])c1Cl c1(C(=O)NCc2c(NCC)cccc2)cc[nH]c(=N)c1[N+](=O)[O-] C(=O)(C(=O)N=S(C)(C)=O)NC1CN(C(c2c(C)nc(C)s2)=O)C(C)(C)C1 c1(CC)cccc(CC)c1NC(N1CCCC(NC(=O)CC2CCOC2)C1)=O c1(C(=O)NCC(C2CCC2)NC(CNC(=O)OC)=O)cc(C)nc2ncnn12 N1(C(c2cc(CC)on2)=O)CCCC(N(C(C2CC(F)(F)C2)=O)CC2CC2)C1 CC1CCN(C(C2CCC3(CC3)N2C(c2n[nH]cc2Cl)=O)=O)CCS1 N1(C(c2cnc(=N)[nH]c2)=O)CC2CC(NC(=O)C3=CS(=O)CCC3)CC1C2 Cc1nccc(C(N2CCC(CO)C(c3ccccc3)C2)=O)c1C c1(C(N2CC(NC(CC3(C=C)CCCCC3)=O)C(C)C2)=O)c(N)cc(C)cc1F S(=O)(=O)(c1ccc(N(C)CCn2cccc2)c(Cl)c1)NCc1ncc(C)s1 O=C(CC(C(F)(F)F)NC(c1ccc(Cl)cc1)=O)NCc1cccnc1F c1(-n2cc(NC(=O)COC3CC(n4cc(C(=O)O)nn4)C3)nn2)ccc(Cl)cc1 C(=O)(C1=C(C)OCC1)N(C1CC(NC(C2(COC)CCC2)=O)C1)C c1(-c2nc(C(CCC)N(C)C)n(C3CCOC(C)C3)n2)nccn2cnnc12 N1(C(c2c(CC)cno2)=O)C(C)CC2CN(C(C3(OC)CCC3)=O)CC12 c1(C(=O)NC2C(CNC(c3cc(C4CC4)on3)=O)COC2)cc2ccccc2o1 CC1(C)C(C(=O)NC2(CCCC(=O)NCc3cc(=O)cc[nH]3)CCC2)C1(F)F N1(c2cccc(CN3CC(=O)NC3=O)n2)CC2CC1CN2C(C1(Br)CC1)=O N1(C(C(CC=C)CC)=O)CC2=C(C1)CN(C(=O)CN1CC(C)(C)C1)C2 c1(CNC(N(C(CSC)Cc2cnn(C)c2)CC)=O)nc2cccc(C)c2[nH]1 CC1(NC(C2CC2(C)Br)=O)CCN(C(C2CC(n3ccnn3)C2)=O)C1 CC1(C)CC(NC(=O)CCC2CCCN2C(C23CCC(C2)C3)=O)C(C)(C)O1 CC(C)(C)CC(F)C(=O)N1C2CC1CN(C(=O)C(C1CC1)C1CC1)C2 C1(C(=O)NC2(C)CN(C(c3c(OC)c(Cl)ncc3)=O)C2)CC12CCC1(CC1)CC2 c1(CC(N2CC(C)C(NC(c3coc(CO)c3)=O)C2)=O)cc(F)cc(Br)c1 C1(NC(c2cc(C)c(C)o2)=O)CC(F)CN(C(=O)CN2CCC(CO)CC2)C1 C1(NC(C(C2CCOCC2)OCC)=O)COCCN(C(C2CN(C)CCN2C)=O)C1 N1(C(C(CC)Oc2ccccc2C)=O)CC2(CC(NC(=O)CC=C)CO2)C1 C1(C)(C(=O)NC(C)C(=O)NCC(C)(O)C2(C)CC2)CC(=O)N(C)C1 C(=O)(C1=C(C)OCCC1)NC(CN(C(=O)CCC1CC(F)(F)C1)CC)C C1(C(N2C3C(NC(C(CCC)CC)=O)C(CC3)C2)=O)CCN(S(N)(=O)=O)CC1 N1(C(CNC(CC)=O)=O)CCCC1(C(N1CCC(C(C)O)CC1)=O)CC c1(NC(CC2(C)CCN(C(C3(CC)CCC3)=O)C2)=O)cc(OC)cc([N+](=O)[O-])c1 C(C)(C(=O)NC1CCC1NC(c1ccc(-c2ccncc2)s1)=O)(C1CC1)OC c1(C(=O)NCC2C(NC(CC(C)(C)O)=O)CCC2)coc2c1C(O)CCC2 C1(C2CCCN(C(c3ccc(C4CC4)nc3)=O)C2)(NC(CCCSC)=O)CC1 c1(C(N2CCC(F)(NS(CC)(=O)=O)C2)=O)c(Cl)cc(F)cc1Cl C#Cc1ccc(C(=O)N(C)CC2CCN(C(c3cc(CCO)on3)=O)CC2)cc1 NS(=O)(=O)c1cnc(C(=O)NCC2(n3ccnc3)CC2)nc1 C1(COC)CC(CNC(c2cc(=N)[nH]n2C)=O)N(C(=O)CCC(=O)N(C)C)C1 c1(C(N2C3C(NC(=O)CSC(F)(F)F)C(CC3)C2)=O)cccc2c1C1CCC2O1 Cc1c(C(=O)NCC(C)(C(C)C)NC(=O)C=Cc2cncn2C)noc1C1CC1 N1(C(c2c(C)scc2)=O)CCCC(CCNC(c2ccc(CC3CC3)cc2)=O)C1 C1(C(=O)NC(C#C)C)CCN(C(=O)C(COC)N(C)C)CC1 N(C(=NCC(C)(C)F)NC1CCOC1)CC(c1ccccn1)C N1(C(C(C)=C2CC2)=O)CCC(C(F)(F)F)C(NC(=O)C=CC2CC2)C1 c1(C(C)C)cc(CNC(c2ccc(C(F)(F)F)s2)C(=O)O)no1 CC(CC(=O)c1cccc(F)c1)C(=O)N1CC(CO)C(N)C1 N1(C(CCOCC(C)C)=O)CCOC(CCNC(c2ncncc2F)=O)C1 CCS(=O)(=O)CC(=O)NCc1ncccn1.c1(COC)nnn(C)c1C=O c1(C(=O)NC2CN(C(C(CC=C)C)=O)CC2O)sc2cccc(F)c2c1Cl c1(C(=O)NCC(C)(C)F)ccc2c(-c3cn(-c4cccc(F)n4)nn3)n[nH]c2c1 c1(C(N(CCCNC(c2sccc2F)=O)C(C)C)=O)ccc2n[nH]cc2c1Cl C12C(C)CCN1C(=O)CCN(C)CCNC2=O.C1(C(C)(F)F)(CCOCC)CC1 c1(C(N2CCC(CNC(c3c[nH]ccc3=O)=O)CC2)=O)cc(O)nc(C2CC2)n1 CCS(=O)(=O)CC(=O)N1CC2(CCN2C(c2ccn(C3CCOCC3)n2)=O)C1 CC1C(NC(=O)C(O)C2CC2)CCCN1C(c1cn(CC(N)=O)nn1)=O c1(NC(C(CNC(=O)OC(C)(C)C)C)=O)ccc(F)cc1F N(C1CCC(C)(C)c2ccccc21)Cc1ncc(C(=O)OC)cn1 c1(CC(=O)N(CCCNC(=O)C(N)=O)C)ccc2oc3ccccc3c2c1 C(CCC(C)C)(C(=O)NCCCCCOC)NC(CCCCCC)=O C1(C2(O)CN(C(C3CCC(F)(F)CC3(C)C)=O)C2)(CNC(C(C)O)=O)CC1 c1(C(N(C)CC2N(C(C(CC)C#N)=O)CC(F)C2)=O)cc(C(C)(F)F)ccc1C C1(c2ccc(OC)cc2)C(C(=O)NC2C(NC(C)=O)COCC2)CC(=O)N1C CC1CN(C(c2cc(C#N)cs2)=O)CC(c2cn(CC3(F)CCOC3)nn2)O1 c1(CC(=O)N(CCC(N)=O)CCC)noc(-c2cccc(C(=O)O)c2)c1C C(=O)(C1=NOC(C)C1C)NC1C(CC)N(C(c2ccc(C)c(C)c2)=O)CCC1 C(C(=O)NOCC(C)(C)O)(C(C)(C)C)NC(CC(COC)COC)=O C1(NC(=O)C=CC2CCC2)CN(C(=O)Cc2cn3ccsc3n2)CCC12CCC2 c1(C(N2CCC(C(C(=O)NC(CC)CCCO)(C)C)C2)=O)ccn2nccc2c1 CC1OC2CCC1(NC(c1cc(CNC(C3CCOCC3)=O)cs1)=O)C2 C=C1CC2CCC(C1)N2C(C1CCOC1CNC(=O)C(F)(F)COC)=O C1(C(N2CCC(CNC(c3cccc(C4CC4)c3)=O)CC2)=O)COC2COCC12 c1(CC(N2C(CNC(CCNC(C)=O)=O)C(C)CC2)=O)cccc(Br)c1Cl CC1(C(=O)NC2C=CC(CC(N3CC(F)(CO)C3)=O)C2)CCC(=O)NC1 c1(OC)cccc(F)c1C(=O)NC1C2CN(C(=O)CSc3nc[nH]n3)CC12 C#CCC(C)(C)C(=O)NCC(C)(C(C)C)NC(c1ccn(C)c(=O)c1)=O C12(C(=O)NC(C3CCCCN3C(=O)CC3CCCC3)C)CC(N=[N+]=[N-])C1C2 c1(CC)ccc(O)c(C(N2CCC(NC(C3CCCS(=O)(=O)N3)=O)C(CC)C2)=O)c1 Cn1cnc2c(NCCC(=O)N3CCCC3)[nH]c(=NCc3cnn(CCF)c3)nc12 C1(CC(=O)NC(CCOC)CO)CC(F)(F)CN1C(c1cc(C(N)=O)[nH]n1)=O N1(C(C2(C)COC2)=O)CCC2(CC1)C(NC(C1CCCC13CCC3)=O)CS2(=O)=O c1(C(=O)NCC(C)NC(C(c2ccc(N)cn2)C)=O)coc2c(F)cc(Cl)cc12 c1(OC)cnc(CNC(=O)C(Cc2cc[nH]n2)NC(=O)CC2CC(C)=NO2)nc1 c1(C(c2n(CCC)nnn2)NC2(n3cc(Br)cn3)CC2)ccc(Br)c(CC)c1 C1(C2(O)CN(C(c3n[nH]cc3Cl)=O)C2)(CNC(=O)COCC2(F)CC2)CC1 n1(CC)ccc(CC(=O)NC(C)C(=O)NCc2cn(C(C)CN(C)C)nn2)n1 Cc1cc(C(=O)NCCCOCCNC(c2conc2C(C)C)=O)cc(C)n1 C(=O)(NN1CCCC1C(N1CCC1CF)=O)c1c(C)snn1 C1(CNC(c2cnn[nH]2)=O)CN(C(=O)CCCc2ccncc2)C2CCCC2O1 C12CC(=NO1)C(=O)NC2.c1(CONC(C2CCC(CC)O2)=O)nnc(C)n1C N1(C(C2C(C)C2)=O)CCC(C2(NC(=O)CSc3ccc(F)cc3)CCC2)CC1 C12(CNC(c3n[nH]c(C)c3O)=O)CCC1CN(C(=O)CCC1CCOC1)C2 c1(C(N2CC(NC(c3oc(C)c(Br)c3)=O)C3(C2)CC3)=O)c[nH]c2c(C)cccc12 c1(COC)sc(C(=O)OCCC2(C#N)CCC2)nc1C c1(C(N)=O)ccc(F)c(CO)c1.C12CCN(C(=O)CN3CC=CC3)CC1C(=O)N2 C1(CC(=O)NCC(CO)NC(=O)CCc2ccco2)CCC(F)(F)CC1 c12ccc(cc1)s2.c1(C(CC)NC(=O)C(=O)NCC(C)N(C)C)ccccc1 c1(C(=O)NC2C(OC)CN(C(=O)CC(=O)NCC(F)(F)F)C2)cc(F)cnc1O CC1CCCC(CC(=O)NCC23CC2CN(C(c2cnnn2C)=O)C3)O1 n1(CC(=O)N(CC(C)NC(C2CCSC2)=O)C)ccc(O)nc1=O c1(CC)cnc(C(=O)NC2CN(C(=O)CCc3cncnc3)CC2C)nc1 c1(C(N2CCC(O)(C(=O)NC3C(C)(C)CC3)CC2)=O)ccc2scnc2c1 C1(C(=O)NCC(C2CC2)NC(c2ccnc(OC)n2)=O)CC2C(C1)C2(C)C n1(CC(N2CC(C)(NCc3cc(C(C)OC)n[nH]3)C2)=O)cc(-c2ccco2)nn1 N1(C(C2N(C=O)CCC2)=O)CC(NC(=O)Cn2nccn2)CC(F)C1 C1(NC(C(C)=CC)=O)CC12CCN(C(C1(COC)CCC1)=O)CC2 N1(C(c2c(OC)cc(C)cc2)=O)CCC2(CCN(C(=O)C3=CCCC3C)C2)C1 N1(C(C=C(C)C(C)(C)C)=O)CC(F)(F)CC1(C)CNC(C1(F)CCC1)=O c1(C(CN2CCN(CC)CC2c2nccn2C)=O)cc2c(F)ccc(Cl)c2[nH]1 CN1CC=C(CC(=O)N2CC(NC(=O)CCc3cccs3)CC23CCCC3)CC1 N1(C(C2CC(=C)C2)=O)CCC(OCCNC(C2CN(C)C2)=O)C1 C1(SCC)CC(c2nnnn2CCC2CC2)(NCCc2cccnc2)C1 c1(CC)ncnc(N2CC3CC2CN3C(c2cnc(OC)c(Br)c2)=O)c1F C(=O)(C1=CCCC1)NCC1CCC(NC(CCc2onc(CSC)n2)=O)C1 N1(C(=O)CN2CCCNC2=O)C2CCC1CN(C(C13CCC(CC1)CC3)=O)C2 Cc1cc(C(=O)NCCCCC(C)NC(C2CNC(=O)CC2C)=O)cnc1F CCC(C)(CNC(C1CN(C(C2C3CCCCC23)=O)CC1F)=O)C(N)=O c1(C(=O)NCC2CCCN(C(c3cc(C)c(C)nn3)=O)C2)n[nH]c2c1CCSC2 N1(C(COC(CC)CC)=O)CCOCC(NC(=O)CCc2ncc[nH]2)C1 C1(NC(CC=C)=O)CC(C)N(C(=O)COCC(=O)OCC)C1 C1(C(=O)NCC2CCCC(CNC(C(C)(C)CF)=O)C2)CCOCC1(C)C CN(C(=NCCF)NCCOc1ccc(Cl)c(Cl)c1)CC1OCCO1 c1(CC)oc(C(N2CCC(C(=O)OC)C2)C(=O)NC2CC2)cc1C(=O)OC C1(CC(=O)Nc2c(CC)nsc2)CC(C)(C)CN1C(=O)CCC1CCOC1 C(=O)(C#CC1CCOCC1)NC1CC(C)(NC(C(C)CC(F)F)=O)C1 c1(C(N2C(CCCNC(C3CNC(=O)N3)=O)CCC2)=O)coc2c(Cl)cccc12 Cc1cnc2c(C(=O)NC3CCC(NC(C4CC(C)(C)C4)=O)C3)c(Cl)ccc2c1 C1(C)(CNC(CN(C(c2c(C)ccs2)=O)CC2CC2)=O)CNC(=O)O1 C(=O)(CCCCN1C(=O)CCC1=O)N(CC(C)NC(C(C)=CC1CC1)=O)C C1(CN2C(C(=O)OC)CC3CC23)CCC2(CN(C(C)=O)C2)O1 c1(OC)cc(CN(c2nc3c(C)cccc3[nH]2)C)c(OC)c2ccccc12 C(C(CO)N=c1nc[nH]s1)NC(C(CC)C(C)C)=O N(C(=NCCOc1ccccc1F)NCC1CCCC1O)C(CC)CC1CCC1 Cc1cc(C(N2CCN(c3cc(=O)n(C)cn3)CC2)=O)c[nH]c1=N c1(C(=O)NC2(C(=O)NC3CCC3)CC2)ccc(N2CCCC2)cc1.CCS C1(OC)CC2CC(C(=O)NC3(CN(C(=O)C(F)(F)C4(O)CCCC4)C)CC3)CC12 CC1CN2CCN1C(C(=O)N(CC(O)CNC(=O)C(F)(F)C1CC1)C)C2 c1(C(=O)NC(C(C)(C)NC(C(CC)N2CCCC2=O)=O)C)nccc2[nH]ccc12 N1(C(C2N(C)CC(C)(C)C2)=O)CC(C)(CNC(c2cc(CO)[nH]n2)=O)CC1(C)C C=CCCCCC(=O)N1CCCC(F)(CNC(=O)C(C)C2CCCC2)C1 c1(NC(=O)OC(C)(C)C)ccc(Br)cc1F.CC1C2C1CNC(=O)N2 n1(CCCC)nc(C)c(C(N2CC3CC3(NC(c3cncnc3C)=O)C2)=O)c1Cl c1(C(c2nc(C(N3CCCC3c3ncco3)=O)[nH]n2)=O)cccc(Cl)c1 C(C(=O)NNC(=O)Nc1nc(C2CCCCC2)cs1)c1ccc(C)o1 n1(C(C)C)cc(C#N)c(=NC(=O)N2CCC(c3cccc(CO)c3)CC2)[nH]1 CC(CC1CCCO1)C(=O)NCC1CCN1C(=O)COCCF.C1(N)(CO)CCOC1 Cc1nn(C)c(Cl)c1C(N1CCC(N(C(=O)CC(=O)NC2CC2)CC2CC2)CC1)=O CC(C)CC(C)C(=O)N1CCCC1(C)CNC(=O)CC1OCCCC1(C)C C1(NC(c2c(CC)ocn2)=O)(CNC(c2cc(C)co2)=O)CCCCC1C C(C(=O)Nn1nnc2c1CCCC2)C1CN(C(c2cn(CCOC)nc2)=O)C1 C(C(C)(C(=O)NCC(C)(C)CN(C(=O)CC=C(Cl)Cl)C)OC)OC N1(C(CC(CC)O)=O)CC2(CCN(C(c3cnn(CCO)c3)=O)C2)C1 c1(CN2CCC(N(C(=O)Nc3c(C)c(O)ncc3)C)C2)cc2ccccc2[nH]1 c1(OC)cc(C(=O)NCC23CC2CN(C(=O)COC2CCOC2)C3)cc(F)c1F n1(C(C)C)cc(C(=O)NC2CCCCC2NC(=O)CCCNC(N)=O)ccc1=O c1(C(N(CC(CC)NC(C2CC2CC(C)C)=O)CC)=O)cn2ncnc2nc1C C1(CNC(C(C=CCCC)O)=O)CCC2(CCN(C(c3ocnc3C)=O)CC2)O1 C1(CC)CCC(C(=O)NCCNc2nccc(-n3nc(C)cc3C)n2)CC1 C1(CNC(C(C(C)O)N(C)C)=O)N(C(c2cc(=N)[nH]n2C)=O)CCCC1(C)C c1(CNC(C2N(C(C(C)Oc3ccccn3)=O)CC2)=O)ccccc1O N#Cc1ccc(F)c(C(N2CCC(NC(=O)C(F)n3cccn3)C(F)C2)=O)c1 N1(C(c2cccn(C)c2=O)=O)CC2(CCN(C(c3c(O)ccc(F)c3F)=O)C2)C1 c1(C(C)NC(C2(CNC(C(C)C)=O)CCC2)=O)cccnc1F CC1CN(C(=O)CC2CCCCN2C)CCN1C(=O)CNC(N)=O N1(C(COCc2cccc(OC)c2)=O)CCN(C(=O)CCCC(N)=O)C(C)C1C C1(CC(=O)N(C(C)CNC(=O)Cn2ccccc2=O)C)CC2CC(=O)C1C2 c1(OC(N(C)CC)=O)nc(C)cc(C)c1CNC1CC(O)(CSC)C1 c1(C(=O)NCC(CN(C(C(CCOC)C)=O)C)O)cc(C)c(C)c(S(N)(=O)=O)c1 c1(CC)ccnc(S(=O)(=O)N2CC(C)C(O)C(C)C2)c1 n1(CCC(C2CC2C(=O)OC)=O)cc(CNC(C2(CN)CC2)=O)nn1.CC CC1CCCCN(C(c2ccc(C(F)(F)F)c(-n3cncn3)c2)=O)C1 Cc1ccn(C(C)C(=O)NCc2occc2C(=O)N(C)CC2CCN(C)C2)n1 N1(C(=O)NC(C(C)C)c2ncc[nH]2)CC(NC(=O)CC(F)(F)F)CC2(CC2)C1 N1(C(CC(C)C2CC2)=O)CCC(C2CN(C(=O)CC3CCN(C)C3=O)C2)CC1 N1(C(CSCC=C)=O)CCn2c(c(CNC(c3cccc(OC)n3)=O)nc2C)C1 c1(C(=O)NC(CC)CNC(=O)CCc2cnc(CC)o2)ccc2ncccc2c1F Cc1ccc(C)n1CCC(=O)N1CC(OC2CCN(C(C3(CF)CC3)=O)CC2)C1 N#CC1(C(=O)N(CCn2ccnc2)CC2CC2)CC12CCCC2.n12cc(nn1)C2 C1(CCNC(CCCNC(C)=O)=O)CN(C(c2nonc2N)=O)CCCO1 Cc1cc(C(N2CCN(C(C3CCN(C)C3=O)=O)CC2c2cn[nH]c2)=O)c(C)n1C c1(OCC(N)=O)ccc(C(=O)NCC2CCN2c2cnc(F)cn2)cc1 Cc1c(F)cc(C(N2CCC2CNC(=O)CC2NC(=O)NC2=O)=O)cc1Br C(=O)(CCC(c1cccnc1)N(C)C)NC(C1CN(C(=O)COC(F)F)C1)C c1(COC)c(CO)cnn1C.N12CCOC(C1)C(=O)NC1CCC(C1)NC(=O)C2 n1(CC(C)C)cc(CC(=O)NCC(CO)NC(=O)C(F)C2CCC2)cn1 c1(CC(=O)NCCCCCNC(C2C3CCC2CC3)=O)ccc(Br)c(F)c1 C#CCCCCCC(=O)NC1CCC(O)CN(C(=O)C(CC)SC(F)(F)F)C1 C1(C(=O)NCCC(C)N(CCC)C)CC=CC(NC(C2CC23CCC3)=O)C1 N1(C(C(CC#C)(C)C)=O)CC2CC(C1)N(C(c1cc(SC)c(Br)cc1C)=O)C2 S(=O)(=O)(c1cc(C#N)ccc1Cl)N1CCN(c2ncnc3cc(C)[nH]c32)CC1 Cc1nc(C2(C(N3C(c4cc(C)no4)CCC3)=O)CC2)cs1.c1(C)occc1C(=O)O C1(C(N2CC(C3OCCN(C(CCNS(C)(=O)=O)=O)C3)C2)=O)CCCC(F)(F)C1 N1(CC2CCCN(c3c(OC)cccc3)C2)CCC(N=[N+]=[N-])(CO)C1 c1(C(=O)NCCC2CCC(NC(CCC(=O)NCCC)=O)C2)cc(F)cc(F)c1 C(=O)(C(C)CO)NCc1cn(CC(=O)N(CC(C)C)CCF)nn1 CCC(C)C1CC(=O)N2CCCC2C(C)(C)N1.C1(Cl)(N)CC1(F)F.C(N)=O C1(N(C(CN(c2ccccc2)C(C)=O)=O)C)C2CN(C(c3cnc(Cl)[nH]3)=O)CC12 C1(C)(CC)CCC(C(=O)NC2CN(C(c3[nH]c(C)cc3C)=O)C2)O1 C(=O)(C#CC1CCCO1)NCC(CNC(Cc1c(C)nn(C)c1C)=O)C C1(CC(=O)NCC2CC(OCC)C2)CN(C(c2ccnn2CCF)=O)CCO1 c1(C(N(CCC(C)NC(c2cnn(C)n2)=O)C)=O)ccc2nonc2c1 O=S1(=O)c2cnc(c(Cl)c2)N1.c1ccccc1.C(CCO)OCCCNCC1CSC1 N1(CC(=O)OC(C)=O)CCC(C(C)=O)C1.C(=O)(CC)N(CC)CC C1(NC(c2cc(C)no2)=O)CC2CCC1CN2C(=O)C(O)Cn1cncn1 c1(C(N2CCC(CCO)(CO)C2)C(=O)NCCCC)cccn2ccnc12 N1(C(C(CCNC(c2c(CC)n[nH]c2)=O)O)=O)CC(CO)CC(C)(C)C1 c1(CCC)nc2sc1CCNC(=O)N2.C1(CNC(C2CCCS2)=O)CCS(=O)(=O)C1 c1(C(=O)NCC2CCC(NC(=O)Cc3cccs3)CC2)cnc2n1CCCC2 C(=O)(C1=C(C)N(C)c2nnnn2C1C)N(CCCNC(=O)C(C)SC(C)C)CC c1(C(=O)NCC2CCN(C(C3(COC)CCC3)=O)C2)c(C)noc1C1CC1 C1(C)(NC(C(CCC)O)=O)CCCN(C(=O)C(CO)OC)C1 C(CO)(C(C)NC(=O)Cc1ccc(Cl)s1)NC(C1C(COC)C1)=O Cc1nc(CCC(=O)NC(C2CCCN2C(=O)CC(C)(F)F)(C)C)oc1C CS(=O)(=O)CC(=O)NCC(O)CNC(c1ccc(CC2CCC2)cc1)=O C1(CCC(=O)N(CC(C)(C)O)CC)CCCCN(C(=O)C(C)C(F)F)C1 c1(C(=O)NCCCNC(=O)CCc2ccccc2)n[nH]c2c1CC1CC21 C=CC(C)(O)CC(=O)N1CCOCC1C(=O)NC(C)C(=O)NCCC C1(CN(C(C(CNC(CCOCCOC)=O)C)=O)C)CCCCC1 c1(N2C(=O)CC(NC3(C)C(C)CCCC3)C2)ccc([N+](=O)[O-])cc1F C(=O)(C(C)(C)NC(=O)C(c1ccnn1C)C)NCCC(C)OC C12(CNC(CC(C)c3ccco3)=O)CC1CN(C(=O)CNC(=O)C1CC1)C2 C12(CNc3onc(C)n3)CCCCC1N(c1nnnn1-c1nn(C)cc1Br)CC2 c1(C(=O)NCC(C)N(C(c2onc(CC)n2)=O)C)ccc(F)cc1 C1(NC(COCC(=O)NC)=O)CC(CNC(C2CCCSC2)=O)C(O)C1 C12(C(=O)NCC3(C)N(C(c4cc(C(C)C)on4)=O)CCC3)CCOC1CCOC2 c1(C(=O)NCCN(CC(C)O)C(c2cc(F)ccc2Cl)=O)cccn2cnnc12 C(N=C(NCC1CCOC1)N1CCC(OCC(C)C)CC1)c1noc(C)c1C C1(C)(NC(C2CCCC(OC)C2)=O)CCN(C(=O)Cc2coc(C)n2)CC1 c1(C(N2CC(C)(CCC(=O)NC(C)C(F)F)C2)=O)cc2ncccc2[nH]1 C1(C(=O)NC(C2CCCN(C(c3ccn(C)c(=O)c3)=O)C2)C)CCCCC(=O)N1 N1(C(C=CCC)=O)CC(O)(C2(CNC(C34CCOC3CCOC4)=O)CC2)C1 c1(N(CCCC)C)ccc(C(C)NC(C2CC(=O)N(c3ccccc3)C2)=O)cc1 N1(C(C2CC3(CC(=C)C3)C2)=O)CCC(C2(NC(c3n[nH]c(CC)c3Cl)=O)CC2)C1 C1(C(=O)NC(C)C(C)C)(OC)CCN(C2CCCN(C)C2=O)CC1 C1(CNC(c2conc2CNC(C2CC3CC3C2)=O)=O)CC12CCCCC2 c1(CC(=O)N(C(CNC(c2c(CC)[nH]cc2)=O)C2CC2)C)ccc(C(C)=O)cc1 CCCCC(C(=O)NCCn1cc(C(N2CC(N3CCCCC3C)C2)=O)nn1)OC c1(C(N)=O)ccn(CCC(=O)NC2(CNC(=O)CC3(C(F)F)CC3)CCC2)n1 N1(C(c2c(C)c[nH]n2)=O)CCC(CO)C(NC(=O)CN2CC(C)C2)C1 CCC(CC)(C(N)=O)NC(=O)CC1CN(C(c2csnc2C)=O)CCC1C N1(C(=O)CSC(F)F)CCSCC1C(N1CCC(c2ncon2)C1)=O C(=O)(C(C)(C)CC(F)(F)F)NC(C(=O)NCC(CC)(CC)OC)C(C)(C)C C1(C(=O)NCCCNC(C2CC(=O)NC2)=O)COc2ccc3ccccc3c2C1 CC1(C)CC(NC(=O)CC2(O)CCCCC2)CN(C(c2cccc(Cl)c2F)=O)C1 c1(C(=O)NCC(CC)(C)NC(=O)COc2ccccc2F)cnn2ccncc12 C=C(C)C1OCCC1C(=O)NC(C)CNC(=O)CC1CC2CC2C1 Cc1cc(C#N)cnc1C(=O)NC(C1CCCCC1)CNC(c1csc(O)n1)=O CC1(CNC(C2CCC=CCCC2)=O)CCN(CC(=O)NC2CCCCO2)CC1 c1(CC)ccc(CN(C)C(N2CC(C)C2c2ccccc2)=O)cc1 N1(c2ccnc(C)n2)CCCC(C)(CNC(c2ccccc2F)=O)C1 N1(C(C=Cc2n(CC)ncc2)=O)CCCC(CCC)(NC(=O)Cc2cc[nH]c2)C1 C#Cc1ccc(C(=O)NC(C2CN(C(=O)CN(C)CC=C)CCO2)C)c(C)c1 c12cccc(c1)CNC(=O)CC2.C(C)(C(=O)NCC)COC(C)(C)C C1(CC)(NC(=O)C(C)(F)F)CCCN(C(=O)C(C)NC(=O)NC)C1 C1(NC(c2ccc(C(C)C)cc2O)=O)CCN(C(C2C(C)C2C)=O)C12CCC2 N1(OCC)CCC(C(=O)NCC(C2CCC2)NC(=O)C(C)Cc2ccncc2)C1 c1(-c2c(C(N(CC(O)CNC(C3CC(C)(F)C3)=O)C)=O)c[nH]c2)ccccc1F Cc1cncc(OCC(N2CCC2(C)CC(N2CC3CC2(CO)C3)=O)=O)n1 N1(C(CC(CC)O)=O)CCC2(CCCC2C(=O)Nc2ccc(C)c(C)n2)C1 N1(C(c2cnc(C)[nH]2)=O)CCCC2(CCCCC2NC(=O)Cn2ccccc2=O)C1 c1(NC(C2NCCN(C(CCC)=O)C2)=O)cc(C2CC2)nc(Cl)c1 c1(OC)ccc2nc(C)c(C(=O)NC3C4CN(C(=O)CCC5CC5)CC34)n2n1 C1(C(=O)NNC(=O)Nc2ncccn2)(NC2CC(C)C2)CCCCC1 C1(NC(C2(Cl)C(C)(C)C2)=O)CCCN(C(=O)COc2ccc(F)c(F)c2)CCC1 N1(C(CNC(C(C)N(C(C)=O)C)=O)=O)CC2C(OCC(N3CCOCC3)=O)C2C1 C(=O)(C(C)(C)C(=O)NCCN(CC(C)O)C(=O)COC1(C)CCCC1)NC c1(N(C)C(C2CCCN2Cc2ncccn2)=O)ccc(C(F)F)nc1 C=C(CNC(C1CC1COC)=O)CCNC(=O)C(=O)NN1CCOCC1 N1(C(C2CCC(CNC(C3(C=C)CCCCC3)=O)CC2)=O)CCCN(C)C(=O)C1 CC1CN(C(C2(n3cccn3)CC2)=O)C(C)CN1C(c1cc(O)cc(=O)o1)=O c1(N2C(CNC(c3scnc3C(F)(F)F)=O)CCC2)nc2ncc(Cl)cc2o1 CC1CCC(C(=O)NCCC(C)(C)NC(c2ccc(-c3ccco3)s2)=O)C1 N1(C(C2C(NC(c3ccc(Br)c(F)c3)=O)CCCC2)=O)CCn2ncnc2C1 C1(C(=O)NC2C3CN(C(CN(CC)CC)=O)CC32)CCc2nc[nH]c2C1 Cc1nc(N)cnc1C(=O)NCC1(O)CC(CNC(c2c(C)csc2Cl)=O)C1 c1(C(=O)NCC(C2CC2)N(C(=O)CC2CC2C2CCCC2)CC)cn(C2CCC2)nn1 c1(C(N(C)CCNC(c2ccncc2N(C)C)=O)=O)cncc(O)c1Cl C1(C#N)(C(=O)NC2CC(NC(c3ncn(CC)c3)=O)C2)CC2CCC1C2 c1(C(=O)NC2CC(CNC(c3cn(C)nc3)=O)C2(C)C)cccc(=S)n1O c1(C(=O)NC2C(NC(C(CC)N(C)C)=O)CCC2)cc(Cl)ccc1F N1(C(Cc2cnc(C)s2)=O)CC2(CC(C(=O)NOCCO)CO2)C1 c1(C(=O)NCC2CCN(C(COC)=O)CC2C)ccc2c(c1)C(=O)CCS2 CC(CCN(C)C)N=c1[nH]c2c(c(=NCC3CSCCS3)[nH]1)CSC2 N1(C(COc2cn(C)nc2)=O)CC(CNC(C23CC(F)(C2)C3)=O)N2CCC1C2 Cc1cc(C(F)(F)CNC(c2cc(C)n(CCN)c2C)=O)cc(C)c1 c1(-n2cc(CN(C(C(CCC)F)=O)C)nn2)ccc(OC)cc1OC C1(C(=O)OC2CCC(C#N)C2)CCC2(CC1)CC2(F)F C1(C(C)NC(C(C)OC)=O)C2CN(c3ncc(C(=O)OC)s3)CC12 CCCC(O)(CCC)CC(=O)N1CCOCC1CN(C)C(c1cnc(S)nc1)=O c1(CC)cccc2ccc(C(=O)N(c3c(C)cc(Br)cc3[N+](=O)[O-])CC)nc12 c1(OC)ncc(C(=O)NC(C)(C)CN(C)C(c2cnccc2Cl)=O)cc1C C=CCC(C(=O)N1CC(C(=O)NCC=Cc2ccccc2)C(F)C1)OC Cc1ccc(C(N2CCC(O)C2C(N2CCC(C)(F)CC2)=O)=O)c(O)c1 C(=O)(C(O)CC(N)=O)N1CC(CC)(NC(=O)CN2CCOC2=O)C1 N1(C(C2N(C)CCC2)=O)CC(F)(F)CC1C(=O)NCC1CC1CCC c1(C(=O)NCCC2CCN(C(=O)C(F)F)C2)nncc2ccccc12 N1(CC(=O)NC(C(C)NC(c2ccc(OCC)cc2)=O)CO)CCCNS1(=O)=O C#CCC(C)(C(=O)N(C(CCO)C(F)F)C)NC(c1[nH]cnc1C)=O C(=O)(C(CC)n1cncn1)NCCCN(C(CN(CCOC)C)=O)CCO C12(C(=O)NCC3(CCNC(c4c(C)nn(C)c4N)=O)CC3)CCCCC1C2(F)F n1(CC)nccc1C(N1CSCC1C(=O)Nc1cnn(CCO)c1)=O C1(CCC=C)(C(=O)NC(CC2CC2)COC)CN(C(c2cc(CCC)[nH]n2)=O)C1 C(=O)(C(CC(F)F)NC(c1nnn(C)c1N)=O)NCc1cncc(CC)c1 C=CC(CC)CC(=O)N(CCCN(C)C)CCNC(=O)C(c1cnn(C)c1)O CC(CCNC(=O)CC(=O)N1CCOCC1)C(F)(F)F.C12(CC(C)(C)C1)C(C)N2 N1(C(C2N(CC)CCOC2)=O)CCC2C(C(=O)NCC(O)(CC)CC)C2C1 c1(C(N2CC(CCNC(C3CC34CCC4)=O)(OC)C2)=O)ccc(F)c(Cl)c1F C1(CNC(C(N2C(C3CCC(N(C(C)=O)C)CC3)CCC2)=O)=O)CCC(=O)NC1 c1(OCC(=O)NCC(C2CCC2)NC(=O)C2=CCSC2)ccc(F)cc1Cl c1(CC(C)C(N2CC(C)N(C(=O)CCCC(C)(F)F)CC2)=O)cnn2ccncc12 c1(C(n2cc(CN(O)C(=O)N(C)C)nn2)CC)ccc(-n2ccnc2)cc1 Cc1cc(C(=O)NC(C2CCCN2C(=O)CCc2ccc(Cl)s2)C)c(C)o1 N1(C(C(C)OCCC(C)C)=O)CCC(C2CC2)(CNC(c2cnns2)=O)C1 N1(c2c(N)nc3ccccc3n2)CCC2(CC1)C(O)CC2O CC#CCCCC(=O)NC1CCC(C)N(C(c2ccc(C(C)(C)CC)cc2)=O)C1 N1(C(C(c2cccc(Cl)c2)CC)=O)CCC(CCOC)(NC(c2ccco2)=O)C1 C1(NC(CN(C)CC)=O)(COC)CCN(C(=O)C(C)Sc2ccncc2)C1 Cc1nc(C(N2CCC(NC(=O)CC3CC(C)C3)C(O)C2)=O)ccc1[N+](=O)[O-] C1(NC(C(C(=O)OC)OC)=O)CCCCCC1NC(c1c[nH]nc1C1CC1)=O c1(C(=O)NC(C2N(C(CCC(=O)OC)=O)CCC2)C)coc2cc(C)c(C)cc12 CP(C)(=O)c1ccc(C(N2CCCC23CCN(C(=O)CC2COCC2O)C3)=O)nc1 C1(C(=O)NCc2n(CC)ccn2)CCC(O)CN1C(C1CC2(CC2)CN1C)=O N1(C(Cc2cccc(OCC)c2)=O)CCC(C)N(C(C2CC3(CC3)CO2)=O)CC1 c1(N(C(C)=O)C)ccc(C(=O)NCC(C)NC(=O)CC(C)n2ccc(C)n2)cc1 CCS(=O)CC(=O)N(C)CC1CN(C(=O)COCc2ccn(C)n2)C1 Cc1c(C(N2CCN(CCO)CC2)=O)cccc1I.N12CCCCC1C2 c1(NC(c2cc(C)nn2C)=O)ncc(-c2ccc(F)nc2)cc1O c1(C(=O)NCC(CCNC(C2C(CCC)C2)=O)O)cc(C=CCOC)c(C)s1 c1(C(N2CC(C)CC(NC(c3c(C)nsc3)=O)C2)=O)cc(C)nc2[nH]nc(O)c12 C=CC1(C(=O)NCCN(C(=O)CSc2c(C)n[nH]c2C)CC(C)O)CCOCC1 N1(C(C2(OCC)CC2)=O)CC2(CCC(CNC(=O)CC(C)F)O2)C1 C1(NC(c2cnn(C)n2)=O)CCC(C(N2CCCC(CCCO)C2)=O)CC1 N1(C(c2ccc(OCC)cc2)C)CCC2(O)CCCCC2C1.c12noc(n1)SC2 N1(C(CCc2cccc(OC)c2)=O)CCN(C(=O)C(C)(C)C(=O)NC)CC(O)C1 c1(C(N2C3CC(NC(C4CCC(CC)CC4)=O)C2CC3)=O)cc2ncccc2o1 c1(C(=O)NCC2CCCCN(C(COCC=C)=O)C2)nccn2cc(C)nc12 C1(CNC(=O)C(N2CCCCC2C2(O)CCC2)=O)CCc2ccccc2C1 Cc1ccc(C(N2CCC(CS(N)(=O)=O)C2)=O)cc1-n1cccc1 c1(C(C(=O)NCC(C)N(C(=O)CCC2(O)CCC2)C)(C)O)ccc(Cl)cc1 CCCCS(=O)(=O)Cc1cn(C2CN(c3ccc(C(F)(F)F)cn3)C2)nn1 C1(NC(C2(COC)C=CCN2C(=O)C(C)=C(C)C)=O)CCCCCCC1 C(C(=O)NCCC1CCC(=O)N1)(C(C)C)NC(C(C)NC(COC)=O)=O C1(C#N)(C(N(C)CC2CCCN(C(C3CC(OC)C3)=O)C2)=O)CCOCC1 N1(C(C(CC)(C)C)=O)CCN(C(=O)Cc2cc(F)ccc2O)C(CF)C1 CC1CN(C(=O)Cc2ccc(F)cc2F)CCCN1C(C1(C)C=CCC1)=O C1(CNC(C(C)OCC2CC2)=O)CCC2(CN(C(=O)CC3=CCCCC3)C2)O1 C(C)(CC(=O)NCCc1nccn1C)NC(CC=C(C)C)=O C(=O)(CCCN(c1cccnc1)C)NC1CN(C(CCSCCC)=O)C1 N1(C(CC(CC)OC(C)C)=O)CCc2cc(C(C)=O)ccc2C1 CCCCCS(=O)(=O)CC(=O)NCC1CCC1NC(=O)Cc1ccco1 N1(C(C2(COC)COC2)=O)CC2(CC=CC2)C1C(C)C N1(C(C23CN(C(CCc4n(CC)ccn4)=O)C(C2)CO3)=O)CC(=O)NC(=O)C1C C1(CN(C(=O)CC2(C)CC2(F)F)C)CCC(NC(=O)C(=C2CCCCC2)F)CC1 c1(N2CCC(C)(COC)C2)nc(=NCC2(CCO)CC2)[nH]c2c1CCCC2 Cc1cc(CC(=O)NC2(C(=O)NOCC(C)(C)C)CCSC2)cc(F)c1 C(C(C)(C)CC(=O)NCC1COC(=O)N1)NC(C(C1CCCCC1)C)=O C(CN=C(NCc1nc(C(F)(F)F)cs1)NCC1CC12CC2)c1c(F)c(Cl)ccc1 Cc1ccc(C)c(CC(N2CCCCC(NC(c3sccc3C)=O)C2)=O)c1 N1(C(C2CCC(=O)N2)=O)CCCC(C2CCN(C(C3CCC(F)(F)C3)=O)CC2)C1 C1(NC(C(n2ncc(C)c2)C)=O)C2CC1CN(C(c1ccc(C(C)(C)C)s1)=O)C2 c1(C(N2CC(OC)C(NC(=O)CCNC(N)=O)C2)=O)cc2c(C)cccc2[nH]1 N#Cc1ccc(S(=O)(=O)NCCN2C3CCC2CC3)nc1 C1(C(=O)NCCCN(C(=O)CCc2cncc(O)c2)CC)CC(C)OC1=O C(=O)(C(C)(C)CC(=O)NCC1C(CC)CCN1C(=O)COCCN(C)C)OCC c1(NC(C(C)N(C)C(C2CC3(CCC3)CO2)=O)=O)cnc2[nH]cnc2c1 c1(C(c2n(CC=C)nnn2)NCC2CC23CCC3)c(F)ccc(C)c1F C1(CNC(C(C)NC(=O)NC)=O)CC(F)(F)CN1C(=O)C(O)CC1CCCC1 C#CC1(C(=O)N(C)Cc2cc(C)nn2C)CN(C(=O)CC2CCN(C)C2=O)C1 C1(C(=O)NCCNC(C2CCC(C(=O)OC)CC2)=O)CCCC2(CCC2)C1 C1(NC(c2cn(CCC=C)nn2)=O)C2CC1N(C(=O)Cc1csc(C(C)C)n1)C2 CN=c1cc(C(=O)N(C)CC2CCCCN2C(=O)CC(C)(C)F)cc[nH]1 C1(C(=O)NC2CCC(CCC(N3C(CC)CC(F)C3)=O)C2)CC(=O)NC(=O)C1 CCCCCC(F)C(=O)NCC1CC(OC)CN1C(c1cc2cccnc2o1)=O C=C1CCN(C(=O)CC(C)COC)C(C(=O)NCCN2CC=CC2)C1 c1(CC(C)C(=O)NCC#CCNC(C2(C)CCNC2=O)=O)ccc(F)c(F)c1 CCCC(CNC(=O)CC1CCSCC1)C(=O)NC1CCCC1N=[N+]=[N-] c1(OC)nccc(C)c1NC(=O)CC1CC(NC(=O)C(C)n2ccnc2)C1(C)C c1(CNC(Cc2cnc(C)s2)=O)ccc(C(=O)NCCC2(N(C)C)CCC2)nc1 C1(NC(CN(C(=O)Cc2cnoc2)C)=O)CCCC1(C)CO C(CC(CC)C(=O)NC1CC(OCC(N2CC3CCC3(C)C2)=O)C1)=CC Cc1ocnc1CCNC(C1CCCN1C(c1cc[nH]n1)=O)=O Cn1cnc(C=CC(N2CC(CNC(=O)NCc3ocnc3C(F)(F)F)C2)=O)c1 c1(OC)cccc(C(=O)NC2CCC(N(C(=O)CC3COCCN3C)C)C2)c1O c1(-c2c(OC)noc2C)ccc(F)c(C)c1-c1ccc(C(=O)NC2CC2)c(C)c1F C1(F)(CNC(CCSCC(N)=O)=O)CCN(C(=O)C(c2ccc(F)cc2)(C)O)C1 CC(CC(=O)N1CCCC1C(N1CCC2(CCC2)C1)=O)C(F)F C(CCN=c1[nH]c2c(cc1C#N)CN(C)CC2)NC(C(C)OCCOCC)=O C(C(=O)NCCn1cnc(CO)c1)(C(C)C)NC(C=CC(C)(C)SC)=O C1(CC)(NC(=O)C(C)CCOC)CCN(C(C2(C)CNC(=O)C2)=O)CC1 C12(NC(C)=O)COCCC1CN(C(=O)CCc1nnc(-c3ccsc3)o1)C2 c1(C(=O)NCc2nc(CNC(C=CCOC)=O)sc2)cccn2nccc12 C1(NC(=O)C=CCOCC(F)(F)F)C2CN(C(c3cscn3)=O)CC12 N1(C(CC2(C)N(C(C(CC=C)(C)C)=O)CC2)=O)CCC2(CC1)CSC2 C1(NC(C2CC(O)C2)=O)CN(C(c2cn3c(n2)CCCC3)=O)C2(CCC2)C1 CC(C)(C)C(C(=O)N1CCOCC1c1cccs1)C(F)(F)F C1(NC(C2CC(C)(C)N(C(=O)CCc3csnn3)C2)=O)CC2CCCCCC12 C(=O)(C(C)C(C)(C)C)NC12CC(NC(c3c(SC(C)C)cccc3)=O)(C1)C2 N1(C(CC)=O)Cc2nccn2CC(NC(c2c(C)cc(OC)cc2F)=O)C1 Cc1oc(Br)cc1C(=O)NC1COCC1CNC(C1CCCCCC1)=O Fc1ccc2c(c1F)CN(c1cc(NC3CC(CC(F)F)C3)ncn1)C2 C1(C(=O)NC2C(NC(=O)CCn3cncn3)CCC2)CC(=O)c2ccccc2C1 N1(C(c2cncc(C(C)C)c2)=O)CC2OCC(NC(=O)C3=CCC(C)CC3)C2C1 c1(C(N(CCNC(C(CCC)OC)=O)CCC)=O)ccc2c(=O)n(C)cnc2c1 c1(CC(=O)NC2CCN(C(C3(CC=C)CC3)=O)CC2C)ccc(OC)c(OC)c1 O=C(CC(O)CNC(C1(C(=O)C2CC2)CCC1)=O)N1CCC(OC2CC2)C1 c1(OC)ccc(C(C)CC(=O)NCCCC(C)(C)NC(=O)OC(C)(C)C)cc1 Cc1cc(-c2ccccn2)ncc1C(N1CCOC(CC2CCCCC2)C1)=O S(=O)(=O)(c1ccc(CC(N)=O)cc1)N1CCC(N(C)C(c2cc(Cl)n(C)n2)=O)C1 C1(C)(C(=O)NCC2(NC(CCn3ncc(C)c3)=O)CC2)CCCC1O Cn1cc(Cl)c(C(=O)NC(CC2CCCC2)C(=O)NCCc2ccoc2)n1 Cc1ccc(C(CNC(=O)CCc2cccc(C)n2)NC(=O)C#CC2CC2)cc1 N1(C=O)CCN(C(=O)Cc2coc(C(F)F)n2)CC1.C12CC1C2.CO Cc1nn(CC(C)C)c(C)c1CN1CCN(C(=O)CC(N)c2cscn2)CC1 C1(C2CCCN(C(C3(CC(F)F)CCC3)=O)C2)(NC(C(F)OC)=O)CC1 N1(C(C2(OC)CC(CO)C2)=O)CC2(CCC2NC(c2ccsc2SC)=O)C1 C1(NC(C2CCOC2C2CC2)=O)CN(C(C2(c3ccccc3)CC2)=O)CCC1F C1(S(N)(=O)=O)(C(=O)NCC2(C)CCC(NC(CC3(C(=C)F)CCC3)=O)C2)CCC1 CN(C)S(=O)(=O)N1CCC(CNS(=O)(=O)c2c(F)cccc2I)c2ccccc21 C1(NC(C2CN(S(C)(=O)=O)C2)=O)CC2CCC(C1)N2C(C1CCC2CC12)=O C1(CC(=O)NCCNC(CCC=C)=O)Cc2ccccc2C1=O N1(CCN(C(C2C(C)CNCC2)=O)CC2CC2)C(C)CCCC1C c1(C(C(C)NC(CSCC)=O)NC(c2ncsc2C)=O)ccc(C)cc1 c1(C(N2CCC(OCCNC(c3c(C)sc(O)n3)=O)C2)=O)cc2ccsc2[nH]1 N1(C(=O)CC(F)(F)F)CC2CC(C(N3CC4CCC(C3)O4)=O)C(C2)C1 C#CCC(C(=O)N1CC(CCO)C1)NC(=O)CCOCC1CC1 Cc1cc(O)c(F)cc1NC(C1CCN(C(=O)C(C)(O)CC(C)C)CCO1)=O c1(CNC(=O)NCCn2cnnn2)csc2ccc(F)cc12 C(CO)(CC(F)(F)F)NC(CC1(OC)CN(C(=O)Cc2cnc(C)s2)C1)=O C1(C(c2ccsc2)NC(N(CCOC)CC)=O)CC2C=CC1C2 C(=O)(C(C)(C)C(F)(F)F)N1CCC2C(C(=O)NCC(C)(C)SC)C2C1 c1(C(=O)NC(C(N2C(COC)C=CC2)=O)CC2CC2)ccc(C#N)cn1 c1(C(N2C(CNC(CC(C)(C)OC)=O)CC(C)(C)C2)=O)nnn2c1C(=O)NCC2 N1(S(CCCC)(=O)=O)CCc2ccc(NC(=O)CCCC(F)(F)F)cc2C1 Cc1noc(Cl)c1CCC(=O)NCCCC(C)NC(c1cnc(O)s1)=O C(CS(=O)(=O)N=S(C)(C)=O)NC(C(C)S(C)(=O)=O)c1nnnn1C1CCCC1 c1(C(C)C)nocc1C(=O)NC(Cc1cc[nH]n1)C(=O)NCCCc1nccs1 c1(C(N2CCN(C(CC(C)CF)=O)C(C3CCC3)C2)=O)nc2ccccn2c1F N1(C(C=C(C)CNC(=O)C(C2CCCCC2)F)=O)CCC2(CC=CCO2)C1 N1(C(CNC=O)=O)CC2(CC(NC(c3cn(CC4CC4)nn3)=O)CO2)C1.C1(C)CCC1 C=CC1(C(=O)NC2C(CCOC)CC2)CCN(C(=O)CS(=O)(=O)NC)C1 C1(C)(CNC(C(c2ccc(C)s2)C)=O)CCCC1NC(C1CCCCN1C)=O N1(C(C2N(C)C(=O)NC2)=O)C2CCC1CC(N(C)C(c1cccs1)=O)C2 N1(C(C(C)=C2CC2)=O)CCC(C2CCN(C(C3CN4CCCC3C4)=O)CC2)C1 c1(CC(=O)NCC2CN(C(=O)CC3CNC(=O)C3)CC2O)ncc[nH]c1=O N1(C(c2cc(COC)on2)=O)CCCC(CO)(NC(=O)CC(C)(C)CN(C)C)C1 Cc1nc(N2CCOCC(CNC(=O)C=Cc3cnn(C)c3)C2)cc(C#N)n1 N1(C(C)=O)CCN(CC(N2CCCC2CNC2CCC3(CC3)C2)=O)CC1 C1(C(N)=O)(CC)CCN(N2CCC(c3cc(O)nc(C(C)C)n3)CC2)C1 N1(C(CNC(=O)C(C)(C)CC)C2(CC)CC2)CCCC(C)(C(N)=O)C1 N1(C(c2c(NC)cccn2)=O)CCN(C)C(C)C1.C1(C(=O)N)C2CC3C(C2=O)C13 N1(C(COc2ccn(C)n2)=O)CC2(CCCN(C(=O)C(C)(C)n3ccnn3)C2)C1 C1(NC(C(CC)OCC)=O)CN(C(=O)Cc2cc(C)cs2)CCC12CCC2 C1(CNC(CSc2c(OC)cccc2)=O)CN(C(=O)C(C)(C)C(C)O)CCN1C c1(CCCC(N2C(CNC(C3SCCS3)=O)CC(OC)C2)=O)c(F)cccc1F C1(CNC(C2CC(O)(CNC(COc3cc(C)on3)=O)C2)=O)CC12CCOCC2 C1(C2(O)CCC2)(C(=O)NCC(CC(C)C)NC(C(CC)N2CCCC2=O)=O)CC1 Cc1cc(O)nc(C)c1C(=O)NC1CC2CC(NC(C34CC(F)(C3)C4)=O)CC12 CC1CC(NC(c2cn3ccc(C4CC4)cc3n2)=O)c2ncnn21 Nc1c(C(=O)NCC2CCN(C(=O)C(F)=CC3CC3)C2)cnc2ccnn12 C1(C(=O)NCc2ccc(CC)s2)N(C(=O)Cc2cccnc2)CCC1(C)C c1(C(C(=O)NCCCC)N(c2ccccc2OC)CC)cc(OC(F)F)cc(C)c1 C(=O)(C(C)CC(F)(F)F)N1CCC(OC2CCCN(C(c3csc(=N)[nH]3)C)CC2)C1 N(C(=NC)N1CCOCC1)S(CCNCC1(CC)CCOCC1)(=O)=O N1(C(c2cn(CCC)nn2)=O)CC2CCCC2(CNC(C2CC23CCC3)=O)C1 N1(c2ncnc(C)c2Br)CC2(CCCC2NC(C2CCC(F)(F)CC2)=O)C1 C(=O)(CCCCCN1CCOCC1)NCC(C)NC(C1CC1C1CCC1)=O C(CCCCCCC(=O)N(CC(C)O)CCNC(C1(C)CCNC1=O)=O)SC c1(CC(=O)NC(c2c(C)noc2C)C)ccc2c(c1)CCOC2 N1(C(c2nncc(CC)c2)=O)CC(O)CCC1C(=O)NCc1nc(N(C)C)no1 c1(OC)cc(C(=O)NCC(F)CNC(=O)Cc2cc(C)ns2)cc(Cl)c1OC c1(C(N(C(C)CNC(c2cc(CCO)on2)=O)C)=O)ccnc(CC2CC2)c1 c1(OC)ncc(C(=O)NC(CO)C(C)NC(c2cc(CC(C)C)c[nH]2)=O)cn1 S(=O)(=O)(c1ccc(-c2ccc(Cl)c(Cl)c2)cc1)NCC(CC)N(C)C CCCC(C(=O)OC)C(=O)NC1CC(C(=O)NCC(C)C2CC2)C1(C)C C#Cc1nc(NC(=O)COC2CC(NC(=O)C(n3nccc3C)C)C2)cs1 c1(C(=O)NCC(N(C(c2c(C)noc2C)=O)C)C2CC2)c(F)c(C)cc(N)c1F c1(C(N(CCCCCCNC(C2CC(SC)C2)=O)C)=O)ccc(C#N)cc1O CC1CN(C(=O)Cc2ccncc2Cl)CC(C)CN1C(c1cscc1F)=O C(N=c1[nH]c2cc(F)ccc2o1)C1(C)CN(C(C(CC)SC)=O)C1.C1CCCCC1 C1(C(=O)NC(C2CCCC2)CNC(Cc2nc(COC)sc2)=O)CCC2CC1CO2 N1(C(c2nc(OC)c(C)s2)=O)CCCC1C1CCCCN1C(=O)Cc1cnc[nH]1 n1(CCC(=O)N(C)Cc2ccc(F)cc2[N+](=O)[O-])cnc2c(N)ncnc12 c1(C(=O)NCC2CN(C(c3cc(C(CC)C)no3)=O)C2)ccccc1CN(C)C c1(C(=O)NCC2(CNC(CC3COCC(C)(C)O3)=O)CC2)cc2cccnc2[nH]1 Cc1cc(C(=O)N(CCCN(C)CCOCCN(C)C)C)c(C)o1 N1(C(CC=CC=C)=O)CCN(C(=O)COCCOC)CC1c1cccc(F)c1 c1(NCCCC(C)O)ccc(S(=O)(=O)NC2CCCC=C2Br)cc1Cl C1(C(=O)NCC2(C)CCN(C(Cc3c(C)ccnc3)=O)C2)CC2COCC(C1)C2 C(CC(=O)NCC(O)CN(C)C(C1CC1C(F)(F)F)=O)SC Cc1cc(O)cc(=O)n1CC(=O)NCC(C1CC1)N(C)C(C1(C)CCCCO1)=O C12(NC(C3(C)CN(C(c4ccccc4NC(N)=O)=O)C3)=O)OCCCC1C2(F)F c1(C(C(=O)NC2CC(C(=O)OC)C2)N(C)C(C2CC2)C2CC2)ccccc1C C1(CC(N2CCC(NC(CC(CC)O)=O)CC2)=O)CCC(=O)NC1=O Cc1cncc(C(=O)NCC23CC(NC(=O)CC4CCCC(C)C4)(CO2)C3)c1Cl c1(OC)ccc(C(=O)NC(C2CN(C(C3(F)CCOC3)=O)CCO2)C)cc1F N1(C(c2cc(C)[nH]n2)=O)CC2(CCN2C(C2CCCN2Cc2ccccn2)=O)C1 C1(CC(=O)NCC(C)CNC(=O)CNc2cccs2)OCCC1(C)C Cn1nc(O)cc1NC(C1CC(NCc2c[nH]ccc2=N)C1)=O CC1CC(C(=O)NCCCc2cn(C)cn2)N(C(c2ccco2)=O)C1 C12(C(=O)NCC(c3ncc[nH]3)C)CCC(CC1NC(=O)Cc1ccn(C)c1)C2 S(=O)(=O)(c1ccc(NCc2cn(-c3nccs3)nn2)c(F)c1)NC(CC(=O)NC)C Cc1nnc2n1CCC(C(=O)N(CCCCNC(=O)CC1(O)CCOC1)C)C2 CC1(C2CCCN(C(C3CCCCCN3C(=O)CCC3CCC(=O)C3)=O)C2)CC1 C1(C)(NC(C2N(CCC)C(=O)CC2)=O)CCCN(C(=O)CN2CCCC2)C1 CC(O)(CC(=O)NC1(CNC(=O)C(=Cc2cscn2)F)CCOCC1)C1CC1 c1(C(=O)NCC(C)NC(c2c(C)ncn2C)=O)ccc(-c2cccs2)cc1F c1(C(=O)NCC2(CCNC(C(C=C)O)=O)CC2)coc2cc(C(C)C)ccc12 Cc1cc(C)c(C(N2CCN(C(c3cc4n(n3)CC(F)C4)=O)CC2C)=O)c(C)c1 CCCCC(O)C(C)C(=O)N1C(C(=O)NC(c2ccco2)C)CCC12CC2 c1(CC)[nH]c(Cc2ccccc2N)cc1C(=O)N(C)CC1CC1.C1(CC(=O)O)CC1 c1(CCC(N2CC(C(C(=O)NCC(C)N(C)C)C)C2)=O)cn(C)cn1 c1(C(N2CC(N(C(c3ccn(CCCC)n3)=O)C)C(O)C2)=O)cc(O)ccc1Cl C1(NC(C2N(C(C(C(=O)OCC)OC)=O)CCOCC2)=O)CCCCC1N=[N+]=[N-] C1(NC(CN(C)C2CC2)=O)C=CC(NC(=O)CCCc2cnn[nH]2)C1 c1(C(N2C3CC(CNC(=O)Cc4cc[nH]n4)(OC3)C2)=O)cc(F)c(Cl)cc1Cl C(N=c1[nH]c(=NCc2csc(Br)c2)c2ccccc2[nH]1)C1CCCC(C)(C)CC1 c1(NCc2nc(C(C)(C)C)sc2)nccc(=NCc2cccc(N)c2)[nH]1 c1(C(N2CCC(C(C)NC(c3nc(C)[nH]n3)=O)C2)=O)cc(Br)c(C)cc1F C(CCCC(=O)NC(C1CCC1)C1CC1)NC(C(C)n1cccc1)=O S(=O)(=O)(c1ccc(NCCCc2ccc(Cl)s2)c(C#N)c1)N(C(C)CO)C C(=O)(CCCCC(C)(C)OC)NC1C(CNC(CC(=O)NCC#C)=O)CC1 CCCCC(O)C(C)C(=O)NC(CC=CC)C(=O)N1CC(C(C)CC)C1 n1(CC=C)cc(C(=O)N(CCCN(C)C(c2ccoc2C)=O)C)cn1 C1(CNC(c2c(C)noc2)=O)CN(C(=O)Cc2cnn(C(C)C)c2)C(C)(C)C1 Cc1sncc1C(N1CCC1(C)C(N1CC(OCC(C)C)C1)=O)=O Cc1ccc(C(=O)NCC(C)(C)CNC(c2ccnnc2NC2CCC2)=O)n1C C1(N(C(=O)COCc2ncc[nH]c2=O)CCF)CCC2(CC2)C1.c12cnn(c1)C2 Cc1c(Cl)ccc(C(=O)NCC2CN(C(c3cc(C(C)C)cnc3O)=O)C2)c1N C(=O)(CCN=c1[nH]c(N2CCCC(C3CCC3)C2)nc(=N)[nH]1)NCC(C)C C(C)(C)(CC(=O)NCCC1(C)CC1)N(C(C(C)C)=O)C.C1CC(=O)N1 Cc1cc(Cl)c(C(=O)Nc2c(C)noc2-c2cnn(C)c2)s1 C1(NC(=O)COc2cncc(Cl)n2)CCCCC12CCCN(C(c1ccoc1)=O)C2 N1(C(C2C(C=C)C2)=O)CCC2(CC1)CN(C(=O)CCc1ccncc1)CC(C)O2 C(=O)(CCC(C)COCCO)N1C(C(=O)NOCCOC)(CC)C=CC1 C1(C(N2CC(C=C)(O)C2)=O)CC2(CCN1C(=O)C(c1cnn(C)c1)=O)CC2 c1(NC(=O)NCC23CCC(C)(OC2)C3)c(F)ccc2occc12 c1(C(=O)NC(CCCNC(C2CCN(C(C)=O)C2)=O)C)cc(C#N)n(C)n1 c1(CC(=O)NCCC2(SCC)CN(C(C3C(OC)CC3)=O)C2)cnccc1C C1(NC(c2cnc(OC)s2)=O)CN(C(C2(NC(N)=O)CC2)=O)CCC1O C1(C)(CCNC(c2c(C(C)C)n[nH]c2)=O)CCN(C(C2CCC2)=O)C1 C#CCCCCCCC(=O)N(C)CCNC(c1c(C)sc(C)c1C#N)=O N1(C(CC(C)OC)=O)CCC(CCNC(c2[nH]ccc2C)=O)CC1C C(=O)(CCCSC1CC1)NCC#C.C12(CC1)C(=O)N2.C12CC1C(=O)NC2=O c1(CC(=O)N(CCC(C)C)C(=O)CC2CCN2CCO)ccc2n[nH]cc2c1 C1(NC(=O)CC(F)(F)F)CCCCCC1.C12CC(C)(C1)NC(=O)C(C)NC2=O c1(C(=O)NC2CC(CC)C2)ccc(C(=O)Nc2cn(C)nn2)cc1.C1(OC)CC1COC c1(C(=O)NCC2CN(C(c3cc(C)sn3)=O)C3C2C3)cc(Cl)cc(Cl)c1 C1(CCC)(NC(=O)C=C2CCC2)CCCN(C(=O)CC2(C)CCOCC2)C1 c1(C(C)=O)ccc(C(=O)NC(C)CCCNC(=O)C=CC2CC2)o1 N1(C(C=CC(C)N)=O)CCC2(CC(O)c3ccccc3O2)C1 c1(OC)ccc(COC(=O)C(Cc2ccc(C)cc2)NC(=O)OC(C)(C)C)nc1 C1(C(N(CCCCO)CC)=O)C2CN(C(=O)NC(C)C(=O)N(C)CC)CC12.C(C)=O c1(C(=O)NC(CN(C(C(C)OCCOC)=O)C)(C)C)ccc(SC(C)(C)C)cn1 N1(C(CCOCCN(C)C)=O)C2CCC1CC(NC(=O)C1=CCCOCC1)C2 c1(OC)ccc(CNC23CC(C(N4CC(O)C4)=O)(C2)C3)cc1 CSC1=C(C(=O)NCC2CCCC2NC(=O)C(n2cc(Cl)cn2)C)CCCC1 CC(O)(C(=O)NCC1CCCN(C(c2ccc(Cl)c(I)c2)=O)C1)C(F)(F)F C1(CC)CC(NCCNC(=O)CCc2c(C)c[nH]c2C)CCO1 c1(C(N2CCOC(C(=O)N(C)C)C2)C(=O)NCCC)cc(Br)c(Br)o1 N1(C(C(C)C2CCCC2)=O)CC(NC(=O)CC2CCN(C)CC2)CC(C)(C)C1 c12ncccc1C(=O)NC2C1CC1.c1(SC(=O)NC(C)C)ccc(Cl)cc1 CC1=C(C(=O)N2CC(CCNC(=O)CSCCN(C)C)C2)S(=O)(=O)CCO1 c1(SCC2CC2)ccc2c(c1)CCN2C1CC1.N1(C=O)CCNC(=O)C1CC(=O)O N1(C(c2cc(P(C)(C)=O)ncc2)=O)CC2(CC(O)C(O)CO2)C1 C1(NC(c2cc(C3CCC3)n[nH]2)=O)CCC2CC1CN2C(=O)CC(C1CC1)C1CC1 C1(C(=O)NCCNC(C2N(C(=O)OCC)CSC2)=O)CN2CCN1C(C)C2 C1(C(N(c2nccs2)CC(=O)OCC)=O)CCOC(c2ccc(F)cc2)C1 c1(OCC(N)=O)ccc(C(N2CCC(c3cn(-c4ccnc(Br)c4)nn3)C2)=O)cc1 N1(C(CCSC)=O)CC(NC(=O)C(C2CCCCC2)O)CC2(CCOCC2)C1 c1(C(N(C(CNC(c2nc(CC)sc2)=O)C2CC2)C)=O)cnc2ncnn2c1O C1(CNC(CNC(=O)OC)=O)CC2(CCN(C(=O)Cc3ccsn3)CC2)C1 c1(OC)ccc(C)c(C(=O)NC2CCCCC2N(C(=O)C(F)C(C)(C)O)C)c1 CCC(CC)(CCNC(c1cnnc(C)c1)=O)NC(C1CC1(C)Br)=O C1(CCC)CN(C(=O)COC2(C)CCOCC2)CCN1C(c1cccc(F)c1)=O C1(C(=O)NC(C)CCNC(=O)C=C(Cl)Cl)CC2(CCCCC2)CO1 CC1Cc2c(F)cc(Br)cc2C1NC(C1CCCC(F)(F)C1)=O N1(C(CSc2ccc(C)cc2)=O)CCCC(C)(NC(=O)CCc2nc(=N)[nH][nH]2)C1 CCC(CO)(C(=O)N1CCC(C)(CCNC(C23CCC(OC)C2C3)=O)C1)OC C1(NC)CCCCC1NC(=O)C(=O)NC1(c2ccc(Br)cc2)CCCC1 CC1(C)C(c2ccccc2F)CCN1C(=O)NCCc1cccc(C(F)F)c1 N1(C(c2scc(C(=O)OC)c2)=O)CCOC2CN(C(=O)CCCC(C)=O)CC12 c1(CCN=C(NC(CC)C)NCc2ccc(F)cc2C)ccc2c(c1)ncn2C c1(C(=O)NCC(C)NC(c2cc(C(C)(C)C)ccn2)=O)cc(F)ccc1C(F)F N1(C(C2(CN(C)C)CC2)=O)CCN(C(c2cccc(F)c2)=O)C(C2CC2)C1 CP(C)(=O)C1CC1.c1(C(=O)NCc2ccoc2)snc(N2CCCC2)c1Cl c1(C(=O)NCC(C)N(C(c2nc(C)ccc2C)=O)CC)cc2cccc(C)c2[nH]1 c1(NC(Cc2c(C)noc2)=O)ccc(C2CCC(=O)N2)cc1 N#Cc1nc(Cl)ccc1NC(=O)CC1CC(CNS(=O)(=O)CC2CCC2)C1 CC(C)C(C#N)C(=O)NC1CC(N2CCN(C(c3ccc(C(N)=O)s3)=O)CC2)C1 C1(CCNC(C2(CC)CCCC2)=O)CCCN(C(=O)C=CC=C(C)C)CC1 C(N=c1ccnc(NCc2ccc(-n3c(C)ccc3C)cc2)[nH]1)C1(SC)CCC1 C1(NC(C2C(OCC)CC2)=O)CC2CC1N(C(C13CC(C1)C3)=O)C2 N1(C(CSCCC)=O)CCN(C(c2cc(C)sc2NC)=O)C(C2CC2)C1 N(C1CCc2c(F)cccc21)CC(N1CCc2sccc2C1)=O CCC(CCC(=O)NOCCCF)NC(c1sccc1C)=O C(C)(CN=c1nc2c(cnn2C)c(NCC2(F)CCC2)[nH]1)OCC=C C1(C(=O)NC(CCC)CCC)CN(C(=O)C2=C(C)OCC2)C(C)(C)C1 c1(CNc2cncc(C(=O)NCc3cnn(C)c3Cl)c2)ccc(I)c(F)c1F N1(C(CC=C=C)=O)CC2(CCN(C(C3Cc4ccccc4S3(=O)=O)=O)CC2)C1 C1(C#N)(NC(c2ccc(C)s2)=O)CCN(Cc2ccc(Cl)nc2F)C1 N1(C(C2C(C#C)C2(C)C)=O)CCN(C(c2cc(F)n(C)n2)=O)CC1CCO C#CCC(C)(C)C(=O)NCCC1(C(=O)NCCN2CCOCC2C)CC1 c1(CN(C(=O)CC(C2CC2)NC(C2(C)CCCS2)=O)CC)ccncc1 N1(C(C2(CCNC(Cc3nc(C)[nH]n3)=O)CC2)=O)CCCC(C)C1 N1(Cc2ccc(OCC=C)cc2)CCC2C(CCCN2C(=O)C(C)N2CC(C)C2)C1 c1(SC(=O)NCC2CCN(C(C)=O)CC2)c(C)nn(-c2ccc(Cl)cc2)c1C Nc1cc(F)c(Cl)cc1C(N1CC(O)(C(Cl)(Cl)Cl)C1)=O C=C(Cl)CC(C(=O)NC(C(O)CO)C1CC1)NC(=O)C(c1ccn(C)n1)C N1(C(c2cc(C)c(Cl)s2)=O)CCCC(C)(NC(=O)CCC2C(=O)ON=C2C)C1 C12(NC(C3CC(C(=O)OC)C3)=O)CCCC1N(C(=O)C=C1CCSCC1)CCC2 c1(C(=O)NC2C(CNC(C(CC#C)C)=O)CCC2)n[nH]c2c(C)cccc12 c1(NC(C2CC(=C)CN2C(=O)C=Cc2ccc(O)cc2)=O)cnc(C#N)c(C#N)c1 C1(OC)COCCC1CC(=O)NCCCCCNC(c1oc(C)nc1C)=O N1(C(Cc2ccc(C)c(Cl)c2)=O)CC2CC1CCN2C(C1CS(=O)(=O)C1)=O c1(-c2n(C)nc(C3CCCO3)n2)cc(=O)sc2c1CCCC2 Cc1cc(C(N2CC(CCNC(c3ccn(C(C)(C)C)n3)=O)C(C)C2)=O)[nH]c1C N1(C(c2nccc(CC)c2)=O)CCCC1C1CCCCN1C(=O)CC(F)F CCC(CCC(=O)N(CCN=[N+]=[N-])C)NC(=O)C#CC1CC1 C1(CC(=O)NCC2(C(C)NC(=O)CN3CC4CC4C3)CC2)CC2(CCC2)CO1 C12(NC(c3c(C)ccs3)=O)CCC1CN(C(=O)CCOc1cccc(CO)c1)C2 C1(CC(=O)N(C2CN(C(C=C(C)C(F)F)=O)CC2(C)C)C)Cc2ccccc2O1 N1(C(c2nc(C)oc2)=O)CCCN(C(C2CCCCNC2=O)=O)CC1 c1(NC(C(CN(C(CC(CCC)C)=O)C)C)=O)ccc(F)cc1C c1(C(N2CCC(NC(C3C(OCC)C3C)=O)(CF)C2)=O)ccnc2ccsc12 C(=O)(CCC(O)C(C)(C)C)NC(C)CN(C(=O)Cn1cc(C(F)F)cn1)C c1(CNC(C2(COC)CCOC2)=O)cccnc1CNC(=O)C(C)=CC(C)(C)C C1(C(=O)Nc2scnc2C2CC2)CCN(C(=O)C(F)F)C1c1ccccc1 N1(C(C=CCN(C)CC)=O)CC=CC1(C)C(=O)NC(c1scnc1C)C C1(C(=O)NCC(=C)CC)CN(C(=O)CCc2cc(C)nn2C)CCN1C N1(C(C(CC)(C)O)=O)CC2CCC1C(NC(c1csc(O)n1)=O)C2 C1(C)(C(=O)NC(c2ccc(Cl)cc2)CC)CCCN(C(C2CC(O)CCN2)=O)C1 C1(NC(c2n(CC)cc(Cl)c2)=O)CC2CCC(C1)N2C(=O)C=CC1CCOCC1 c1(-n2c(NCCc3cnc(C)s3)ccn2)cncnc1O C(=O)(NNC(=O)C12CC3CC1C2C3)c1ncc(C)s1 C(=O)(CC(C(C)C)c1ccccc1)NC(CNC(C(C)OCCOC)=O)(C)C Cc1cc(C(=O)NC2CCC(N(C)C(c3c(C)ncnc3C)=O)CC2)ccc1N C(=O)(C(C)CC(C)(F)F)N1CC(C)CC(NC(Cc2cccc(COC)c2)=O)C1 c1(CSCC(=O)N(CC(C)NC(C=CCCC)=O)CC)ccco1 N1(C(C2CCC(=C)CC2)=O)CCN(C)CC1C(N1CCC(C)C1(C)C)=O c1(C(CNC(=O)CSC2CC2)NC(C2N(CC)CCC2)=O)ccc(F)cc1 c1(OC)cc(OC)cc(CC(=O)NC2CC(CNC(=O)C(C)n3cnnn3)C2)c1 CC(CS(C)=O)N=c1nc(N2CCC3(CCC3)CC2)c2c([nH]1)CCCC2 c1(N2CCC(S(CC)(=O)=O)C2)nc2ccsc2c(=NCCC(C)N2CCCC2)[nH]1 Cc1cc(C(N2CC3(CNC(=O)CC4CC(F)(F)C4)CC2CO3)=O)ncc1N C(=O)(C1=CCCCCC1)NC1C(C)CN(C(=O)C(c2ccc(Cl)cc2)CO)C1 C1(C(=O)NC2C3CN(C(c4cccc(N)c4)=O)CC32)CC12CCSCC2 C(C(C)C(=O)NCCN(CCCN(C)C)C(=O)Cc1n[nH]c(C)n1)OC N1(C(C2CCC(=C)CC2)=O)CC(NC(C2(C)CCOCC2)=O)C(C2CC2)C1 C#CCCN=C(NCCCc1cccnc1)NC(c1cccc(Cl)c1)C S(=O)(=O)(c1cccc(NCC2CC3(C2)CN(C(=O)OC(C)(C)C)C3)c1)N(C)C CC(O)C(N)C(=O)N(CCCO)C(c1cc(C2CC2)nn1C)=O O(N(C)C(=O)CNC(=O)C(F)CC1CN(C(c2cc[nH]n2)=O)C1)CC C1(C(NOCC=C)=O)CCC(NC(=O)C(C)OCC(C)C)CC1 c1(-c2cn(CC=C)nn2)nc(-c2cccc(Cl)n2)nn1CC(N)=O N1(CCNC(Cc2cc(C)[nH]n2)=O)CCN(C(c2[nH]nnc2C)=O)CC1 COC1CC(NCCC2C(=O)Nc3ccccc32)c2ccccc21 C1(OC)(CF)CN(C(C2(CNC(=O)C(C)CC3CCC3)C=CCC2)=O)C1 N1(C(C2(C#C)CCCCC2)=O)CC2CCC1C(CNC(=O)C(C)CC(F)(F)F)C2 C1(C(=O)NCC2ON=C(C)C2)CC(=O)CN1C(C1CS(=O)C1)=O N1(C(c2c(C)nc(C(C)C)s2)=O)CC(CNC(=O)CCOC2COC2)C(C)(C)C1 C(C1=CCN(C(c2cc(N)ccc2C)=O)CC1)NC(CCNC(C)=O)=O c1(C(=O)NC2C(C(=O)Nc3c(OC)cccc3O)C2)c(Br)ccc(OC)c1F c1(NC(=O)NC2C(CC)C2)ccc2c(c1)C(=O)N(C)C2=O Cc1cccc2c(C(N3CCC(CNC(C4(O)CC4(C)C)=O)C3)=O)coc12 N1(C(C(C)NC(C=C)=O)=O)CCC2(CC1)CC2(C)C(N1CC(O)C(N=[N+]=[N-])C1)=O C(=O)(C(CO)C(F)(F)F)NCC1OCCC(NC(c2cncc(COC)c2)=O)C1 c1(C(=O)NC(C2CCCCN2)C)cc2occc2s1 c1(N(C(=O)Cn2nnc(C)n2)CC)cccc(OC(F)F)n1 C1(C)(N2CC2=O)C(C)(C)C1(C)C.N1(C(CC=C)=O)CCCC1C1CCOC1 c1(C(N)=O)cccc(CNC2CCOC(c3cccc(F)c3)C2)n1 C1(C(=O)NCCCCC#C)COCCN(C(c2ccc(F)cc2)C)C1 c1(CC=C)cccc(S(=O)(=O)NC2CCNC(C(=O)OC)C2)c1 c1(C(=O)NC(CCCOC)C(=O)NC2CC=CCC2C)cc2ccccn2c1 C1(CNC(CCOCC(C)C)=O)CC(C)(C)CCC1NC(=O)CC1CCOCC1 c1(OC)ccc(F)c(C(N2CCC(NC(=O)C(F)C(F)(F)F)C2C2CC2)=O)c1 c1(NC(C2N(C(C3C(C(N)=O)CCCC3)=O)CC2)=O)cc(Cl)c(Cl)c(Cl)c1 C#CC1CN(C(=O)CCc2ccn(C)n2)CCN1C(=O)CCc1cc(C)on1 C(=O)(C1=C(Cl)CCC1)NCCCN1CCC(CO)C1.C12(CC(C(F)F)C1)C(=O)N2 c1(OC)cccc2c(C)c[nH]c12.C12CC3CCC1N3CC(=O)NCC2.C1(N)CCC1 Cc1ccc(C(=O)NC(C)CN(C(=O)CC2CCC(C)CO2)C)c(F)c1F C(=O)(C(CCC(N)=O)n1cc(CO)nn1)N1CCC(NCc2ccc(OC)s2)CC1 CC(N=C(NCC(F)F)NCC1CCC(CC2CCCC2)CC1)C1CC1 C=Cc1cncc(C(=O)NC2(C)CCCN(C(=O)Cc3ccc(OC)cc3)C2)c1 CC(C)(C)CC(O)CNC(=O)CC1(C)CCN1C(c1cc(O)cs1)=O C12(C(=O)OC)CCCCC1N(C(=O)Cn1ccc(=O)cc1)CC2 C1(C(N(CCCNC(CC2N(CC)CCC2)=O)CCO)=O)CC12CCOC2 c1(C(=O)NCC(C2CC2)NC(CN(C(C)=O)C)=O)cc(=O)c2ccc(O)cc2o1 C1(NC(CCSCC(C)C)=O)CCN(C(C2CSC2)=O)C1C1CC1 c1(NC(Cc2cc(CC)no2)=O)ccc(C)cc1Cl c1(C(N2CC(C)C(CNC(=O)Cc3nnc(O)s3)C2)=O)csc2ccc(F)cc12 c1(CC(=O)NC23CCN(C(c4cnc(OC)s4)=O)CC2C3)cnc2ncccn12 c1(C(N2CCC(CCNC(=O)C3=CCSC3)CC2)=O)cnc2c(c1)OCC(=O)N2 c1(N(C)C)ccc(NC(C2(CNC(=O)CC3(C)CC3(F)Cl)CC2)=O)c(Cl)c1 c1(CC)c(C(N2CCCC(CC(=O)NCC3(C(C)C)CCCO3)C2)=O)nnn1C C1(C(=O)NC2CCC(O)C2)C2CCCC1CN(C(=O)Cn1cc([N+](=O)[O-])cn1)C2 n1(C(=O)OCc2ccc(NC)c(F)c2)ccc2c(Br)cccc12 Cc1cc(C(=O)NCC2(O)CCCN(C(=O)Cn3cc(CO)nn3)C2)ncc1F C1(N(C(CCOCCOC)=O)C2CCCC2)CCN(CCCN(C)C)C1 C1(NC(CC)=O)CC(C)CN(C(c2csc(-c3csc(C)n3)c2)=O)C1 C1(CNC(c2cc(C(C)C)no2)=O)C(O)C(O)CN1C(C1(CO)CCCCO1)=O c1(C(=O)NC2(CNC(C(CSC)OC)=O)CCOCC2)cc(C)nc(O)c1 c1(C(=O)NCC2C(NC(C(=O)NCCC(N)=O)=O)CCCC2)cccc2c1CCN2 N1(CC)CC(C(=O)NC2CC3CC(NC(C4CCC(=O)N4C)=O)C3C2)CCC1=O C(=O)(C=CS(F)(F)(F)(F)F)NCC1(O)CCN(C(c2cccc(C(C)C)n2)=O)C1 C1(CNC(C2(C)CC(C)=C(C)CC2)=O)CC(N=c2[nH]nc(C(F)(F)F)s2)C1 C1(NC(C2CCCCS2)=O)CCSC12CN(C(C1CCC(CO)CC1)=O)C2 C1(NC(c2cc(C)cc(O)n2)=O)CCN(C(C2CC2c2cnc[nH]2)=O)CC12CCC2 N#CC1(C(=O)NC2CCCCN(C(=O)CC3COC4CC3C4)C2)CCCC(=O)C1 C(C1(O)COCc2ccccc21)NC(c1cc(N2CCCCC2)cc(C)c1)=O N1(C(C2(SC)CCC2)=O)CCOCC1C(N1CCSC(C(=O)O)C1)=O n1(CC(C(C)C)OCC)nc(C(F)(F)F)c(C(F)(F)F)c1C(=O)O N1(C(=O)C2=NOC(C3CC3)C2)CCC2(CCN(Cc3cc4ncccc4[nH]3)C2)C1 C(=O)(C1CCCc2nc[nH]c21)NC1CC(C)(C)CN(C(c2csc(S)n2)=O)C1 C1(C(=O)OC)CCC(NC(N2CCC2C(N)=O)=O)C1 C(=O)(CC1COc2ccccc21)NC1CC(NC(C2CC(=O)NC2)=O)C1 c1(C(=O)NC(C2CCCN(Cc3cscn3)C2)C)cccc(F)c1F C1(C(=O)NC(CNC(C2CC3C(C)(C)C3C2)=O)(C)CO)CCn2nnnc2C1 CC1(C#CC(=O)NCC(O)CC(=O)N2CC=CC2C(=O)NC)COC1 N1(C(c2c(CC)nn(C)c2)=O)CC(NC(C2CCOC(=O)N2)=O)CC12CCCC2 C1(CC#C)(C(N2CCC(CCS)C2)=O)CCCC1.C(=O)(C)NCC(=O)OC(C)(C)C C1(C(=O)NCC(c2ccccc2)CNC(=O)Cc2cccs2)C(Cl)(Cl)C12CC2 C=CCN=C(NCC(C)(C(C)C)OC)NC1(OC(C)C)CCOC1 CCCCCCCCCCC(=O)N1CC2(CNC(=O)CN(C)CC)CCC1CC2 C(=O)(CC1=NN(C)C(=O)C1)NCC(C(=O)NCC(CC)CC(C)C)OC C1(F)(CNC(CC(=O)NCC#C)=O)COCCN(C(=O)Cc2ccoc2)C1 C(=O)(N1CC2COCC2O1)C1(C(F)(F)F)CCC(=O)CC1 N1(C(c2c(NC)snc2C)=O)CC2CCN(C(=O)CC3CCCCN3C)C2C1 C=CC(CC(=O)N(C)CCOCCN(C)C(C)=O)c1ccccc1 C(=O)(C1=CCCSC1)Nc1nc(C(=O)OCC)c(C2CC2)s1 c1(C(=O)NCCCC(=O)NC2(CC)CCC2)cc(OC2CC2)cc(O)c1 c1(SC)ccc(NC(=O)N(C)Cc2c(O)cccc2F)cc1SC Cc1ccc(CCNC(C2CC(=O)CN2C(C2CC(C)N(C)C2)=O)=O)cc1 C1(CCNC(c2cc(-c3ccco3)on2)=O)CN(C(=O)COC(F)F)CCO1 C(CCCC(=O)NC(c1ccccc1)C(=O)NCC1(C)C=CCCC1)OC FCCCN=C(NCc1ccccc1N1CCCCC1)NCCN1CCCCCC1 C(=O)(C(F)(F)CCn1ccnn1)N1CCN(C(CCCOC(C)=O)=O)CC1 c1(C(N2CCN(C(COCc3n(C)ncc3)=O)CC2)=O)ccc(S(N)(=O)=O)o1 c1(C(=O)NCCC2(NC(=O)CCOC3CC3)CC2)cn(C2CC2)nn1 CC(C)S(=O)(=O)CC(=O)NCC1CCN1C(=O)CN(c1ccc(Cl)cn1)C C(C)(C(C)C(=O)NC(C1CCC1)C1CC1)NC(c1c(CC)ocn1)=O N1(C(C2N(C(C(CC(C)C)N(C)C)=O)CC2)=O)CCOCC(C)(C)C1 C1(CNC(C=CCC2(NC(CC(=O)OC)=O)CCC2)=O)CC12CCOC2 C(C(CC(C)C)OC)NC(C(COCC)NC(=O)C(C)OCOC)=O C#Cc1ccc(C(=O)N(C2CCN(C(c3cc(C)c(Cl)s3)=O)CC2C)C)c(C)c1 C12CCCCN1C(c1nccs1)C(=O)NC2=O.CC(C)C.C1CCS1 c1(CC)ccccc1-n1cc(C(O)CC(=O)Nc2cn(C3CCC3)nn2)nn1 c1(CC(c2ccc(O)cc2)(COC)NC2CCS(=O)(=O)C2)ccc(F)c(F)c1 c1(CC(=O)NCC2CC(CCNC(=O)Cc3ccco3)C2)cncc(Br)c1 C(=O)(C(F)(F)CC)NC(C1CCCCC1)C(C)NC(C1COCC1C(N)=O)=O C1(C)(C(N2CC(C)(C)C(NC(=O)Cc3cccnc3)C2)=O)CCCCCNC1=O CC(C(=O)NCC1CCCCC1NC(=O)CCC(C)(C)O)C(F)(F)F CC(CC(=O)NC(C(=O)N(C)CC1CC(F)(F)C1)C1CCCO1)C1CC1 N1CCCN(C(c2cncn2C)=O)CC1.C(=O)(C(C)CN)OCC c1(C(=O)NC2C(NC(C(CC)C(F)(F)F)=O)C2)cc2ccccc2cc1Cl C1(NC(C2CCC(=O)N2)=O)CCC(n2cc(-c3ccc(CCO)cc3)nn2)CC1 c1(CC(=O)NCC2(NC(=O)CC3CCC4CC34)CCC2)ccc(OC(F)F)c(F)c1 c1(CN(CC#C)C(=O)NCCCN2CCOCC2)ccc(SC)nc1 n1(CC(=O)NC2C(CNC(CS(CC)=O)=O)CC2)ccc2nc(O)nc(O)c12 c1(CC(N2CC(C)(NC(C3CCC(CC)O3)=O)C2)=O)cc(F)ccc1Br Cc1ccc(F)cc1C(F)(F)C(=O)NCC(C1CC1)NC(C1CCCC(C)C1)=O OCCCCCCCCOc1cc(-c2ccccc2F)cc(F)c1 C1(C(=O)NC(C=C)C)CC2CCC(C1)N2C(=O)CN(C)C1CC1 c1(NC(C(C(C)NC(c2c(CC)ncnc2)=O)C)=O)ccc(O)c(C)c1 C1(CNC(=O)OCC)CN(C(=O)CC2(C(F)(F)F)CC2)CCO1 c1(C(N2CC3C(NC(C4CCC5(CCC5)O4)=O)C(C3)C2)=O)occ2c1CCCC2 CC(O)C(C)(C)C(=O)N1CCCC2(CNC(=O)CCC(F)(F)F)CC12 C(=O)(CS(=O)(=O)C(C)C)N1CCC(OC2CCN(C(C=CC(CC)C)=O)C2)CC1 C1(C(=O)NCCC2(C(=O)NC(C=C)C(F)(F)F)CC2)CC2(CCO1)CC2 c1(C(C=O)C)ccccc1.C(C(=O)NOCCCC1CC1)OCC CCC(CC)C(C(=O)N1CC2CC2C1C(=O)Nc1cccc(O)c1)OC c1(CN(C(C(CC)OC)=O)CC(=O)NC)cc2ccccn2n1 c1(C(N2CCN(CCCC3CCCO3)CC2)=O)ccc(SC)cc1Br.CO C(=O)(CCCC(C)=O)NCC1C(C(=O)NC(CC=C)CC)CCC1 c1(CN2CC3CC(CN(S(CC#N)(=O)=O)C3)C2)c[nH]c2c([N+](=O)[O-])cccc12 C(C(=O)NNC(=O)CNCCCCC(C)=O)c1ccc(OC)cc1 C12(NC(=O)CCc3ccccc3Cl)CCC(CN=c3[nH]cncc3Cl)(CC1)OC2 C1(NC(=O)COCC2CC2)COCC1NC(=O)CSC(F)(F)F N1(CC=CCNC(C2COC(=O)O2)=O)CCN(C(=O)C(F)=CC2CC2)CC1 C1(C(=O)NC2CCCC(NC(C(CSC)(C)C)=O)C2)Cc2nncn2C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NCC(C1CCOC1)NC(C(C)OC1CCCC1)=O C1(C(N2CC(CC)N(C(c3ccc(F)cc3)=O)CC2)=O)CCc2nn(C)cc2C1 Cc1c[nH]cc(C(N2CCOC(CN(C)C(C3(C)CC(=O)N(C)C3)=O)C2)=O)c1=O Cc1nc(Cl)cc(=NCC(C)NC(=O)C(F)(F)C(F)F)[nH]1 N1(C(C(CC=CC)C)=O)CC(NC(c2cnn(C(C)C)c2)=O)CC12CCC2 C1(CC)CCC(C(=O)NC(C(=O)N2CC(OC)C2)c2cccs2)O1 N1(C(c2ccc(Cl)o2)=O)CCC2(CCC(NC(C3(CO)CCC3)=O)C2)CC1 C1(C)(CNc2c(C(=O)OC)cccn2)CCN(C(=O)CC2CCCO2)CC1 c1(OC)nc(Nc2nc(-c3ccco3)oc2C)c2cc(C(C)C)sc2n1 c1(NC(c2c(NCc3cncc(C)n3)nc(Cl)cc2)=O)cc(Br)c(F)cc1F CC1(C)CCCN(c2ccc(-c3cccc(Cl)c3)nn2)C1 CC(C)(CC(=O)N(c1ccc(Cl)nc1)c1ccc(Br)cc1)C(=O)O N1(C(C2(C=C)CCN(C(=O)C=C3CCC(C)CC3)C2)=O)CCC2=C(CCCC2)C1 N1(C(C(C)(C)NC(=O)OC)=O)CCOC2(C1)CN(C(=O)CC(C)(C)C1CC1)C2 c1(C(C2(C)CC2)C)nc(-c2cc(I)nn2C)n(C(c2ccccc2)C2CC2)n1 c1(C(=O)NCCCN(C(=O)CCOCCN(C)C)CCC)c(C)nsc1N C1(CC(=O)NCC(N2CCC2c2ccco2)=O)C(NC)CC1O.c1csc(F)c1 CN1CCN(C(C2CCN2C(c2ccns2)=O)=O)CCC1=O CC(C)C(C(=O)NCCCN(C(=O)CCc1nccs1)CCO)NS(N)(=O)=O N1(C(c2cc(C(C)=O)[nH]n2)=O)CC(C(=O)NCC(C)(C)CCl)OC(C)C1 N1(C(c2n(C=C)ncc2)=O)CCC2CN(C(c3ccccc3SC)=O)CC2C1 C(=O)(C(N)CCC(C)(F)F)NCc1cccc(CCN(C)C)c1 C1(CCNC(C(C)OCc2cn(CC3CC3)nn2)=O)OCCC1(C)C Cc1nc(C(=O)NC2CCC(C)(CNC(C3NC(=O)OC3C)=O)CC2)cc(O)n1 c1(OC)cc(F)ccc1C(c1cn(CC(=O)NC2CC2)nn1)N1CCOC1=O N1(C(C23CC(NC(=O)OCC(CC(C)(C)C)CO)(C2)C3)=O)CCC2(CCCC2)C1 C1(OC)CC2CC1CN(C(C1(CNC(=O)C(C)N(C)C(C)=O)CCCCC1)=O)C2 CCCCC(C(=O)NCc1cc(C(N2CC3C=CCC(C3)C2)=O)ccn1)C(C)C c1(COC)cc(C(N2CCC(O)(CN(C)C(c3csnc3C)=O)C2)=O)ccc1F CC(C)(C)C#CC(=O)NCc1ncoc1CCNC(=O)C(C1CC1)C1CC1 C#CCC(C)C(=O)NC1CCN(C(c2cn(-c3cnn(C)c3)cn2)=O)C1C C(CC(=O)N1CC(O)(c2cn(-c3ccsc3CO)nn2)C1)(c1cccs1)NC c1(C(=O)NCc2cn(CC(C)Nc3ccccn3)nn2)ccc(C(C)(F)F)cc1 C(=O)(C1=NOC2(CCC2)C1)NC(C1CCN(C(C(C)C)=O)C1)C c1(C(C(F)(F)F)N(C(N2C(C(=O)O)CCCC2)=O)CCF)cc(Cl)cc(Cl)c1 C1(NC(CC2(C)CC2)=O)CCCCN(C(=O)CCC2(C#N)CCC2)C1 Cc1ccc(=O)n(CC(=O)NC2CC3CC2N(C(C2CCS(=O)(=O)C2)=O)C3)c1 Cc1nn(C)c(C(=O)NC2CCCCN(C(C3C=CCCC3)=O)C2)c1Cl c1(C(=O)NC2CN(C(CC3(OCC)CC3)=O)C2)cc(C)n(C(C)CC)n1 CN1CC(O)(CNC(=O)C(O)C2CN(C(c3ccccc3)=O)C2)C1 N1(C(CCc2n(C)ccc2)=O)CC(C(=O)NCc2ccccc2)C2(CCC2)C1 n1(C(C)(C)C)cc(C(=O)C(=O)NCCNC(=O)Cc2n[nH]c(O)n2)cn1 c1(NCc2ccc(NC(c3cc(=O)c(OC)co3)=O)cc2)cc(F)c(Br)cc1Cl C(=O)(CC(C)CF)NC(CCNC(c1c(COC)ccs1)=O)C C1(C(C)OC)CCN(C(=O)C(C)N(S(C)(=O)=O)CCO)CC1 Cc1nc(C)c(C(=O)N(C(C)CCNC(C2CCOC3(CCC3)C2)=O)C)c(C)n1 C=CCCCCC(=O)N1CC(N(C2(F)CC=CC2)C(C2CCCC2)=O)C1 C1(CC(=O)NCC(CCOC)NC(c2cc(OCC)cs2)=O)CCC(C)C1 c1(C(=O)NC2CCC(NC(c3scc(C)c3)=O)C2)cnc(Cl)cc1Cl C1(CNC(CCN(CC)Cc2cccc(Cl)c2)=O)CC2(CO1)CN(C(C)=O)C2 C(=O)(C1=CCC(C)(C)CC1)NC1CCN(C(C(C)Cc2cnco2)=O)CC1F C1(C(=O)NC(CC)COC)CCCN(C(=O)CSCC(F)F)C1 CC(CNC(c1ccc(C2CC2)s1)=O)(CO)NC(=O)C(c1ccccc1)=O Cn1c(C(N2CCC(n3cc(-c4ccc(=N)[nH]c4)nn3)C2)=O)cnc1Br c1(C(=O)NC(CC)CN(C(=O)CC(C)SC)C)cc(Br)cn1C(C)C N1(C(C(n2cc(Cl)cn2)C)=O)CC2(CCCC(CNC(c3ccoc3)=O)O2)C1 C1(C)(SC)NC(=O)C2=C1N(c1ccccc1Cl)C(=S)NC2c1[nH]nc2cnccc12 C1(C#N)(C(=O)NC(CC)CNC(=O)C2=C(C)OCCC2)CCS(=O)(=O)CC1 CC1CC(=O)NC(C(=O)NCCCN(CCO)C(C2CCCC3(CC3)C2)=O)C1 c1(C(N2CCC(N(C(=O)CC3CCC4(CCC4)O3)C)C2)=O)c(N)cccc1[N+](=O)[O-] N1(C(c2ccn(CC)n2)C(=O)NCCOCC)CCOc2ccc(Cl)cc2C1 c1(C(=O)Nc2ccccc2OCC2CC2)cnn2cccnc12 N1(CC(=O)NCC2(OC)CN(C(=O)C(C)c3ccsc3)C2)CCC(O)CC1 C1(NC(CCCCCC)=O)CCN(C(c2nccc(Cl)c2C)=O)CC(C)(C)C1 c1(C(c2nnnn2C)Nc2c(OC)c(F)c(C)cc2)cccc([N+](=O)[O-])c1C N1(C(C2COC2CO)=O)CCC(N2CCOC2=O)CC1 c1(CC(=O)NC(C(=O)N(C2CC(OC)C2)C)CC2CCC2)ccc(C)cc1 c1(CN2CC3CN(C(c4cccs4)=O)CC32)ccc(F)c(O)c1F C1(O)(C(=O)NCC(C2CC(NC(c3nc(Cl)cs3)=O)C2)C)CCCCCC1 C(=O)(CCC(C(C)C)NC(c1ccc(C#N)[nH]1)=O)N(CC(C(C)C)OC)C c1(C(c2ccco2)(CC)NCC(CSC)OC)nnnn1C1CCCC1 C1(C(=O)NCCc2n(C)ncn2)CC(NC(C2CC(O)C2)=O)C1(C)C C(=O)(C(O)(C(F)(F)F)c1ccccc1)N(CCN(C(=O)COC(F)F)C)C c1(OC)ccc(CC(=O)NCC2(O)CCN(C(=O)C3=CCCC3C)CC2)cc1F c1(NCc2cc(C)n(C)n2)[nH]c(=NC2CCC(N(C)C)CC2)nc2c1cnn2C N1(C(CC=CCC)=O)CC(NC(C23COCC2C3)=O)C(C2CC2)C1 Cc1nc2cccc(C(N3CC4CCCC4(CNC(C4CC(C)C4)=O)C3)=O)n2n1 C1(NC2CN(C(CC3C(C(N)=O)COC3)=O)C2)CC(NC(N)=O)C12CCC2 C(c1cccn1C)=C(C(=O)NCC1(O)CC(NC(C2CC(CC)(CC)C2)=O)C1)F N1(C(C2N(C(C)=O)CSC2)=O)CCCC(C2CCN(C(=O)Cc3cnoc3)C2)C1 [N-]=[N+]=NC1(C(N2CC(O)(CCNC(c3ccoc3Cl)=O)C2)=O)CC1 CCC(F)(F)CC(=O)N.C(CCSC)(C(=O)N1CCCCC1CC(N)=O)CCO C1(C(=O)Nc2ccc(C3CCN(C(C4C(C)C4)=O)CC3)cc2)CC2CCCC2C1 C1(C(C)NC(=O)C=CS(C)=O)CCN(C(C2(CCF)CC2)=O)CC1 c1(NC2CC3(CCN(C(CCNS(C)(=O)=O)=O)CC3)C2)nc(O)c2ccccc2n1 N1(C(CCCOCC)=O)CC(CCNC(C2(N3CCOCC3)CC2)=O)OC(C)C1 C=Cc1cncc(C(N2CC(O)CC2C(=O)N(CCC)C2CC2)=O)c1 c1(C(c2nnnn2C2CCC2)NCc2cc(C)on2)nc2ccccc2[nH]1 N1(C(CN(CCSC)C)=O)CCN(C(=O)CSc2ncccn2)C2CCCC12 N1(C(c2c(C)c[nH]n2)=O)CC2CCC(C1)C2NC(=O)CSc1cccc(Br)c1 c1(C(N2CCC(CCOC)(NC(CCC#C)=O)C2)=O)c(SC)nc(O)nc1C n1(CC(=O)NCCN(C(CC(CC)OC)=O)CCCN(C)C)c(C)cc(O)cc1=O CCC(C)(C)C(O)C(=O)NC1CCC(C)N(C(=O)Cc2ccnn2C)C1 C1(CNC(C(CC)(C)C)=O)CCCCN(C(=O)Cc2ccccc2C)CC1 c1(NCc2cn(C(COCC)C(=O)N(C)C3CC3)nn2)cncc(C#N)c1 N1(C(CC2CCN(C)C2)=O)CCOC2(CCN(C(c3cc(O)ccc3O)=O)C2)C1 C(=O)(C1=CCCSC1)NCCC1(NC(c2c(C(=O)OC)c[nH]n2)=O)CCCC1 C(N=C(NC1CCOCC1)N1CC2C(C(F)F)C2C1)c1n(C(C)(C)C)ncn1 C(=O)(CC(C)(C)CC(=O)NCC(O)CNC(c1ccsc1C)=O)OC Cc1c(NC(=O)Nc2nccs2)cnn1CC1CCCO1 N1(C(C(C)OC)=O)CCC(F)(C(=O)NOC2(C)CC(O)C2)C1.O(C(F)(F)F)CCN CCC(C(=O)NCCN(CC(C)O)C(C1(CF)CC1)=O)n1ccc(C2CC2)n1 CC1(NC(C2CCCS(=O)(=O)C2)=O)CCCN(C(=O)C(C2CC2)C2CC2)C1 N1(C(C(CC)(C)O)=O)CCC(C(=O)Nc2sccc2C(N)=O)C(O)C1 C1(N(C(CCSCCCC)=O)CC)CCCN(C(c2cc(C(C)C)on2)=O)C1 c1(OC)ccc2c(c1)OC(NC(C1CCC(C)(C)C1)=O)C2 C12(CNC(c3nc(COC)oc3)=O)CC(CO1)N(C(C1CCCC(C)(C)O1)=O)C2 CC1(CCNCC2(C)COC2)NC(=O)NC1=O N1(C(C(C)(C)CO)=O)CCC2(CCCC2CNC(=O)C(=Cc2c[nH]cn2)F)CC1 c1(COC)ncsc1C(=O)NCCCC1CCCN1C(=O)CCC1CCOC1 N1(C(C2(C(=O)OCC)CCCC2)=O)C2CCC1C(NC(=O)CC(C)(C)C)C2 CS(=O)(=O)c1ccc(Br)cc1C(N1CCCC(c2n[nH]c(S(C)(=O)=O)n2)C1)=O C(CCCC(=O)NCC1(CO)CN(C(=O)Cc2sccc2C)C1)OCC C1(NC(c2cccc(C(N)=O)n2)=O)CN(C(C2C=CCS2)=O)CCC1CO N1(C(CNC(CCOCC#C)=O)=O)CCN(C2CC2C(F)(F)F)CC1 N1(C(COC(CC)C)=O)CCC(CC=O)(OC)C1.C(=O)(C(O)Cc1[nH]cnc1C)NC c1(C(C)=O)ccc(C(=O)NCC(O)CC(=O)NCC2CC(F)(F)CO2)nn1 C(CCCC(C)C)N(C(C(C)N(C(=O)C(O)Cn1cncn1)C1CC1)=O)C1CC1 N1(C(c2c(C)[nH]c(=N)s2)=O)CC=C(CCNC(=O)CC(C)C(F)F)CC1 c1(OC)c(C)cc(C(=O)NC(C)CNC(=O)CC2C(C)(C)C2(C)C)cc1C c1(C(=O)NCCCN(CCCN(C)C)C(C2(C)CC2F)=O)ccc(CO)cc1 CC(C)CS(=O)CC(=O)NCC(C)(CC(C)C)NC(c1ccc([N+](=O)[O-])o1)=O c1(C(C(=O)NCCOC)N(C(C)CC(C)C)CCC#N)sc(C)cc1C N1(C(c2cc(SC)oc2)=O)CC2CC(NC(=O)Cn3ncn(C)c3=O)C2C1 CC1(C)CCN(C(=O)CC2CC(NC(C3CCC3)=O)C2(C)C)C1 c1(OCC)cccc(C=CC(N2CCCC2c2ccc3cc[nH]c3c2)=O)c1OC c1(C(C(=O)NCC2(CC(=O)NC3CC(O)CC3O)CC2)O)cccc(Cl)c1 N1(CC(=O)NCCNc2nnc(C)n2C)CC2CCC(C1)N2c1ccccc1 C1(C(=O)NCC(C)NC(c2cnc(-c3ccccn3)s2)=O)CCCC12CCOCC2 C1(C(N2CC(n3cc(-c4cncc(Cl)c4)nn3)C(O)C2)=O)CCS(=O)(=O)N1 C1(C)(CCC(=O)NCCOCCCNC(C(C)c2ccsc2)=O)CC1(F)F c1(C(=O)NCCN(C(=O)C(CC)NC(N)=O)CCC)ccc2nsnc2c1 N1(C(C(CN(C)C)(C)C)=O)CCC2CC2(NC(c2cccn3nnnc23)=O)CC1 N1(C(CC=C)=O)CCCCC(NC(=O)C(c2cccnc2)C)C1 CC(C)C(C(=O)N1CCN(C(C2(C(F)(F)F)CC3CCC2C3)=O)CC1C)C(C)C N1(C(C2C3CCCOC23)C(=O)NC(CC)C)CCCOCC1C N1(C(CSCCC)=O)CC2C3CCC(C(CN)C3)C2C1.C(=O)(C(C)(C)C)C(=O)CSC c1(C(C(=O)NC(CC)C)N(CCCOC)CCOC)cccc2ncccc12 C1(CCOC)(NC(C2CSCC(=O)N2)=O)CCN(C(C2CC(Cl)(Cl)C2)=O)C1 Cc1ncn(C)c(=O)c1C(N1CC2CC2(NC(=O)COCCCF)C1)=O C1(NC(CCOC(C)=O)=O)CN(C(c2cn(C3CCCC3O)nn2)=O)CC1C C=C1CC2CCCC(C1)N2C(=O)C(C)(CSC)NC(c1nnc(S)n1C)=O C=CCC(C)(CNC(=O)C=C(C)CNC(C1CCOC1C1CC1)=O)CO C(CC1=CCN(C(=O)C(C)CF)CC1)NC(c1c(CC)nc[nH]1)=O C12(NC(=O)CC3CC(NC(c4cccc(CO)c4)=O)C3)CCCC1OCC2 C1(CNC(CC=C)=O)CC2CCC1N2C(=O)Cc1n[nH]cc1Br c1(C(N(CCN(C(c2[nH]nnc2C)=O)CC)CC)=O)cc2cnccc2[nH]1 O=C(CCn1ccc(I)n1)NNc1ccc(Br)nn1 c1(C(=O)NCCNC(C2CC(CC)(CC)C2)=O)ccn2[nH]c(=N)nc2c1 C(=O)(C(C)C(C)c1ccncc1C(F)(F)F)NC1CN(C(c2nnc(C)s2)=O)C1 C1(NC(c2c(C)nncc2)=O)CCCC12CCN(C(C1CCC(CO)CC1)=O)C2 Cc1ncc([N+](=O)[O-])n1CC(N1CC(NC(c2nc(=O)n(C)[nH]2)=O)C(C)C1)=O N1(C(C(C(CC)(C)C)O)=O)CCCC2(CCN(C(=O)C=Cc3cn(C)nn3)C2)C1 C(C1=NOC2CC12)(c1nnnn1-c1cccc(C#N)c1)CCNc1nc(C)[nH]n1 c1(CCSC(C)CC(N)=O)nc2ccccc2n1CC(F)F C#Cc1cn(C)nc1C(=O)NCC1CC(NC(=O)C(F)CC2CCC2)C1 N1(C(CNC(=O)OCC=C)=O)CC=CC(NC(c2ncccc2C)=O)C1 C(CC(C)C)(C(=O)N1CC(NC(c2cnns2)=O)CC(F)C1)NC(C)=O c1(OC)cncc(C(=O)N(C2CCC(NC(c3cc(N)ccc3C)=O)C2)C)c1C C1(C(=O)NC2(CNC(c3ccc(C(C)=O)nn3)=O)CC2)CC2CCC(C1)C2 c1(C(C)(C)C)cccc(C(N2CCC(O)(CNC(C3(C)CC(F)(F)C3)=O)C2)=O)n1 C12(C(C(=O)O)NC(=O)CCc3nc(-c4nc[nH]n4)no3)CCC(CC1)C2 Cc1ccncc1C(=O)NCCn1cnc(C(=O)NCCc2cnco2)c1 Cc1coc(C=CC(N2CCC(NC(=O)Cc3ccncc3)C2C)=O)n1 C1(C2(O)CCN(C)CC2)(C(=O)NCCC(C)CCNC(=O)C(F)=CC2CC2)CC1 c1(C(=O)NC(C(C)C)CNC(C23CC2CCC3(F)F)=O)ccc(O)c([N+](=O)[O-])c1 C1(NC(c2cccc(CC)n2)=O)CN(C(C2CC23CC3)=O)CC1N=[N+]=[N-] C1(C(N(C(C)CNC(c2c(F)ccc(C)c2F)=O)CC)=O)CCc2nn[nH]c2C1 c1(C(=O)NC2CC(C(=O)Nc3cnc(Br)nc3)C2)cccc2c1OC(F)(F)O2 c1(C(=O)NCC(c2ccccc2)CC)occ2c1CCC2 Cc1c(C(N2CCCN(C(c3ccc(=N)[nH]n3)=O)CC2)=O)[nH]c2cc(Cl)ccc12 N1(C(C(CCC2CCC2)NC(c2cccc(CC)n2)=O)=O)CCC2(CCSC2)C1 C1(N(C(C)(C=O)C2(N)CCC2)C(=O)C=CCCC(C)C)CCC(C2CC2)C1.CO C(=O)(C(C)(O)CC(F)(F)F)N1C(CNC(CCN(C)CC)=O)CC1 N1(C(C(CCC)N2CCCS2(=O)=O)=O)CC2C(=O)N(C3CC3)C(=O)C2C1 N1(C(C=C(CC)C)=O)CC2CC(C1)N(C(c1ccnc(-c3cc[nH]n3)c1)=O)C2 c1(C(=O)NC2C(OCC)CN(C(C(CC)NC(N)=O)=O)C2)sc2nn[nH]c2c1C C(=O)(C(F)(F)C(F)(F)C(F)(F)F)N1CCC(O)(CNC(=O)CCCCC(F)F)C1 N1(C(C(C)(C)c2cccs2)=O)CC2CC2(NC(c2c(Cl)n[nH]c2C2CC2)=O)C1 C1(C(=O)N(C)CCOCCCNC(=O)Cc2ncoc2C)(CC)CCC(O)CC1 C(=O)(C(C(C)O)N(C)C)N1CC(CCNC(=O)CSC(F)(F)F)(OC)C1 CC(C)C(C)CC(=O)N(CC(=O)Nc1cnn(C(C)(C)C)c1)C N1(C(c2cc(CNC(CCC#C)=O)sc2)=O)CC2COC(=O)C2C1 N1(C(c2c(CC)nnc(C)c2)=O)CCN(C(c2ncccc2C)=O)C2CCC12 c1(OC2N(C(=O)OC)CSC2)cccn(CC(N2CCCCC2)=O)c1=O c1(NCc2c(CC)cccc2)nccc(=NCc2nnc(-c3ccccc3)n2C)[nH]1 N1(C(C(CC#CC)NC(=O)Cc2ncccc2F)=O)CC2(CCCCC2)C1 c1(CC)nc(C)oc1C(=O)NCc1ccc(CCNC(=O)Cn2cnnc2)cc1 C1(C(=O)NCCCOCC#C)CCN(C(C2CC=CCC2)=O)C1 N1(C(C(=Cc2cccs2)C)=O)CC(NC(=O)Cc2cnc(C)cc2C)CC(C)C1 n1(CC)ccnc1C(C)NC(=O)C(C1CCN(C(C2(CC)CCC2)=O)C1)C N1(C(Cc2c(C)ncnc2C)=O)CCCC1C1CCCN1C(=O)CCOC1CC1 c1(CNCC(=O)NC(c2ccc(F)cc2)C(=O)OC)ccc(C#N)cc1F N1(c2cc(C)c(C(=O)N(S(C)(=O)=O)C3CC3)cc2)CCCC(C)(C(F)(F)F)CC1 C1(NC(Cc2c(C)cc(F)cc2)=O)CC2CC(C1)N(CCCc1ccncc1)C2 c1(C(N(C(c2ccccc2)CNC(c2c(C)onc2)=O)C)=O)cc(O)ncc1Br C(C)(C(C)CC(C)C)(c1n(CCCOC)nnn1)Nc1ccc(F)cc1SC N1(C(CCC(=O)OC)=O)CCN(C(=O)CC2CCCS2(=O)=O)C(C2CCCC2)C1 c12nn(cc1C)S(=O)(=O)C(=O)CN2C(C1C(OC(C)=O)CCOC1)=O.C(C)(C)(C)O C(C(O)C(=O)N)NCCN(C(=O)CS)CCOCCO.c1(N(C)C)nccn1C CN1N=C(C(=O)NC2CC(C(=O)NC(=O)C=Cc3cc[nH]n3)CC2O)CCC1=O C#CC1(C(N2CCC2C(C)O)=O)CN(C(C2CCCCC2)=O)C1 N1(C(C2CC(C)=C(C)CC2)=O)CCC2(CCCC2NC(=O)CC(C)C)CC1 C1(C(N(C(CCC)C)C)=O)CC(=O)N(NC(C(=O)NC)C2CC(CCC3CC3)C2)C1 C(C1=CCN(C(=O)CC2CCCN2C(c2ccns2)=O)CC1)OC C1(NC(C(CC)(C)O)=O)CN(C(=O)CCn2cnc3ccccc23)C2(CCC2)C1 N1(C(C(C#C)(C)C)=O)CCC(CC)(NC(c2ncccc2CC)=O)CC1 C1(CNC(c2ncn(C)c2)=O)CC2(CC2)CN1C(=O)CC(=O)NC1CC1 N1(c2cc(C)c(C#N)cn2)CCC2(CN(C(=O)Cc3ccnn3C)CC(C)O2)C1 Cc1ccc(C(c2cccc(C(N3CCC4(CC3)CC4)=O)c2)=O)c(Br)n1 C1(NC(CCC=CC)=O)CCN(C(=O)CCn2cccnc2=O)C(C)C1 N1(CC(=O)NCCN(CCC)C(c2ccc(COC)[nH]2)=O)CCCC1C C#CCC(CC(=O)N(CCCC(C)(F)F)C)NC(C12CC(C)(CCO1)C2)=O C1(C(=O)NCCN(C(C(F)=CCC)=O)CC2CC2)CC2(C1)CC(F)C2 CC(C)(C)C(O)C(=O)NCC1(NC(c2cc(C(C)(F)F)on2)=O)CCCCCC1 N12CCC(O)CC1CC(=O)NOCC2=O.C(C(=O)OC)(OCC)OCC C(=O)(CCC(=O)NC1CCCC1)NCCCN(CCC)C(c1ccsn1)=O C1(NC(c2ccc(SC)o2)=O)CCC2(CC1)CN(C(=O)CC(C)N(C)C)CCO2 c1(C(N2CCC3C(NC(C4N(C=O)CCC4)=O)C32)=O)c(F)cc(Cl)cc1F c1(OC)cc(C(N2CC3C(C(=O)NCCn4cccnc4=O)C3C2)=O)ncn1 C1(c2nc(-c3ccc(F)c(NC(C)C)c3)no2)(OC)CCC(C)(C)C1 CCC(CC(=O)NC(CC1CC1)C(N1CCN(C(C)(C)C)CC1)=O)CC(C)C C(=O)(N(CCC(=O)N(C(C)C(C)C)Cc1ccco1)OC)c1ncc(OC)nc1 N1(C(C2(COC)C=CCC2)=O)CC2CCC(C1)C2NC(c1cnc(C(C)C)o1)=O c1(CC(=O)NC2CC(CNC(C(C)C3CC3)=O)C2)ccc2c(c1)CCCS2(=O)=O C(CCNC(c1nc(C)c(C)s1)=O)(C(=O)N(CC(c1nn[nH]n1)C)C)OC C1(CCCNC(c2c(SC)scc2)=O)CCCCN1C(=O)CC1COCCO1 N1(C(COCC(C)C)=O)CCN(C(=O)CC(O)CCc2ccccc2)C(CO)C1 Cc1cccc(C(C)NCC2CCCCN2C2CCCC2)c1 N1(CC(N2CC(C(C(=O)N(CCC(=O)OC)CC)O)C2)=O)CCC(C)CC1 Cc1cc(Br)ccc1C(=O)NC1CCCCN(CC(C)O)C1 Cc1ccnc(OC(=O)CC2(CS(C)(=O)=O)CC2)c1.C1CO1 C(=O)(C(CC(F)F)NC(N)=O)NCc1cn(-c2n(C)ncc2Br)nn1 c1(CC(=O)NCC=CC(=O)NC(CC)(C)C)csc(C)c1 c1(C(=O)NC(C(C)NC(C2CN3CCN2CC3)=O)CO)[nH]nc2ncnc(O)c12 c1(C(N(C)CC2(O)CCN(C(c3c(C)con3)=O)CC2)=O)cccc2sncc12 Cc1cnn(CC(=O)NC2(CC(=O)N(C(C)C)CC3CC3C)CCCC2)c1 c1(NS(C(C)C)(=O)=O)ccc(C(=O)NC2CC(NC(C3(CF)CC3)=O)C2)cc1.C(N)=O c1(C(=O)OC)ccc(C(=O)NCC(O)CN(C(=O)CC(=O)NC(C)C)C)nc1 C1(N(C(=O)CN(C2CC2)CC)CC)CCCN(C(=O)C(CO)c2ccccc2)C1 C(=O)(C1=CC2(CCOC2)C1)N1CCC2(CC(C(=O)NCC3C(=O)NCC3)C2)C1 CC(CC(=O)N1CCC2(CC2)CC1C(=O)NCCN(S(C)(=O)=O)CCO)C(C)(C)C C=CCC(CNC(=O)C=CC1CCC1)C(=O)NC1(CC=C)CC1 C=CC(C)(C)CC(=O)NCCN(C)C(=O)OC(C)(C)C N1(C(C2(C(=O)OC)COC2)=O)CC(NC(C2CC(=C3CCC3)C2)=O)CC(F)C1 Cc1cc(C(N2CC3CC3(NC(=O)CC3CC=CC3)C2)=O)nnc1O CC1CCC(C(N2CSCC2C(=O)NC(CCO)C2CCC2)=O)CC1 CC(CCCCNC(C1(C)CC=CC1)=O)NC(C1CC(=O)N(O)C1)=O N1(C(C2CC(OC(C)(C)C)C2)=O)CCC=C(C(=O)NC23CCCCC2C3)C1 c1(OCC)cc(C)ccc1C(=O)N(C)CC1COCCN1c1nc(Cl)c(C#N)s1 C12(NC(C(C)S)=O)CC1CN(C(c1csc(-c3ccncc3)n1)=O)C2 Cc1cc(C2CC2)ncc1C(=O)NCC1CC1NC(c1cc(C(N)=O)cs1)=O C1(CC(=O)N(C)C)CC2(CCN(CC(=O)NC3(O)CC3)CC2)CO1 c1(NC(=O)Nc2nc(CC(C)C)sc2)ccccc1-c1noc(-c2ccco2)n1 c1(C(=O)NCC2(C)N(C(CC(C)SC)=O)CCC2)cc2c(ncn2C)[nH]1 CCCC1C(O)C(=O)N1C.C1(C(=O)NCC(F)F)(CCOCCO)CCC1 C1(C(=O)NCC2C(C#N)CC2)CN(C(=O)CCN=[N+]=[N-])CC1C(F)F CC1(C(=O)NCC(=O)NCC(=O)NC2(CC(F)F)CC2)CCC(=O)C1.C(N)(=O)N C(C(=O)NC1CC(NC(=O)Nc2cnn(C)c2)C1)(C(C)C)CC.C12(C)CCCN1C2 C(=O)(C1c2ccccc2-c2ccccc21)NC1CC(NC(CC(=O)NCC)=O)C1 C=CC(C)CC(=O)NC(C12CCC(CC1)C2)CNC(C1CC(=O)N(C)C1)=O N1(CC(=O)NCC(c2ccccc2F)Oc2ccccc2)C(=O)NC2(CC2)C1=O N1(C(c2c(C)csc2)=O)CCOCC(C(=O)N(CC(C)(C)CN(C)C)C)C1 C(CS(C)(=O)=O)(C(=O)O)Cn1c(CNC2(C)CC3(CC3)C2)nnc1N1CCCC1 c1(N(C)CCOCCNC(=O)CC2(C)CCCC2)ncnc2c1nnn2C C(=O)(CC(O)CC(C)(C)C)N(CC(C)(C)CNC(C1(C)CC(C)(C)C1)=O)C C1(NC(c2cn3ccsc3n2)=O)CN(C(=O)CN2CC3CCC2C3)CCC1O C(=O)(CCCC(=O)NCC)NC1(C(N2CC(=O)NCC2C)=O)CCSC1 N1(C(C2(CNC(CC3CC(SC)C3)=O)CC3(CC3)C2)=O)CC2(CCC2O)C1 C(CNC(=O)CC1CC(SC)C1)(C(C)(C)C)NC(C1CC(C)(CC)C1)=O N#CC1(O)CC(C(N2CCCCC2CNC(C2CC23CC3)=O)=O)C1 C1(C(=O)NC(C(C)SC)C)CC2(CCC2)CN1C(=O)C(C)NC=O.C(C)C c1(OC)cc(C)c(-c2cccc(CN3CC(C)OC(C)C3)n2)c(C)c1 C=CCCCC(=O)N(CCC(C(C)C)NC(c1ccn(C2CCC2)n1)=O)C c1(OC)nc(C)cc(=NC2CC(NC(=O)CCc3cc[nH]n3)C(O)C2)[nH]1 C1(CC(C(=O)NCC(=C)C)N2CCC(CN(C)C)C2)CCCCC1C(C)C O=S1(=O)CCCC(n2nc(-c3cccnc3)nc2-c2cc(C3CC3)no2)C1 CC1CCN(C(=O)CCc2cn(C)cn2)C1C(=O)Nc1cnn(C)c1C(N)=O c1(N2c3ncc(s3)C(=O)N3CCC2C3)nc2ccc(F)cc2o1.CC(F)(F)C1CC1 C1(CNC(=NCCOCC=C)NCC(c2nccs2)C)CCCCC1(C)C c1(C(=O)NCC2CCCC2NC(c2cnn(CCC(F)(F)F)c2)=O)ccc(O)nc1 C(CCNC(=O)N(CCCN(C)C)CCCN)OC C(=O)(C(O)(CN(C)C)C(F)(F)F)NCC(CNC(c1cc(C)oc1C)=O)(C)C N1(C(C2OCCN(C)C2=O)=O)CC2C3CCC(C2C1)N(c1nnc(C(N)=O)s1)C3 c1(C(=O)NCC2N(C(CN(C)CC)=O)CCN(C)C2)nccn2ccnc12 c1(C(N(CC(=O)NC2CCS(=O)(=O)C2)C)=O)cnn2c1OCC(F)C2 C(=O)(C(F)(F)CF)NCC1(N(C(CC2(C)CC2F)=O)Cc2ccccc2)CCCC1 N1(C(C(CCC)OC)=O)CC(NC(=O)C=Cc2ccsc2)C2(CC2)C1 C1(=CC(=O)NCCC(C)NC(=O)C2=CCCSC2)CCCCCC1(F)F c1(NC(C(CCC)NC(=O)C=CC(C)(C)SC)=O)cnn2c1OCCC2 c1(C(=O)NCC(CN(C(c2cc(OCC)no2)=O)C)(C)C)n[nH]c2c1CCC2 C(=O)(C1=C(C)OCC1)NCCCN(C(C(c1ccc(CC)cc1)(C)C)=O)CCO C(=O)(C1=CCCC1(C)C)NC1CCCN(C(c2c(C)nc(C(C)(C)C)nc2)=O)C1 C#CC1(O)CC(C(N2CC(C(O)C(=O)NCc3cc(CC)no3)C2)=O)C1 c1(C(=O)O)ncc(OCC)c(OCC)n1.c1(C(=O)OCC)ccc(O)nn1 CC(C)CC(CN(C)C)C(=O)NC(c1ccccc1)CNC(=O)Cc1ccoc1 c1(C(=O)OC(C2CCCCC2)C(=O)NC2CSCCS2)cc2c(cn1)OCCO2 N1(C(CSC2CN(C(COCCC)=O)C2)=O)CCC(CC2CC2)C1 C1(C(=O)NCCC(COC)O)(CNC(=O)C=C(C)C(C)C)CCCCO1 CC(C)C(F)(CNC(C1CCCN1C)=O)C(=O)NC1CCC=CCC1 C(=O)(CCC(C)(C)O)N(CCCN(C(=O)C(C1CCCCCCC1)O)C)C C(=O)(C(C)=CCNC(=O)COC1(C)CCC1)N(CCCCC)C C(=O)(CCCCCC#N)N1CCC(C(NOCC(C)(C)O)=O)(CO)C1 c1(C(=O)NC(CNC(CC(CC)C)=O)C2CCC2)cc([N+](=O)[O-])c2nsnc2c1 Cc1cn2c(=O)c(C(N3CC(CNC(=O)C(=O)N(C)C)CC3C)=O)cnc2s1 CC(O)(CC(=O)NC1CCCCN(C(c2ccc(C#N)cc2)=O)C1)CC(=O)O c1(C(=O)NCc2n(CCOC)c(S)nn2)cc2c(Br)cccc2[nH]1 c1(OCC)cc(CNC(=O)Cc2ccccc2I)ccc1OC.C12(CC1)C(=O)N2 C1(CNC(c2cccc(NC(C3CCCNC3)=O)c2)=O)Cc2cccc(Br)c2C1 c1(C(=O)NC(C2CN(C(C3(C)CC(F)C3)=O)CCO2)C)cc2n(n1)CCC2 C(=O)(C(CCOCCO)NC(c1ccc(O)nn1)=O)N1CC(C)(N(C)C)C1 c1(C(CC)C)nc(N(C2CCCN(C(C3CCCC3C)=O)C2)C)cc(C)n1 N1(CC)CCN(CC(c2cn(CC3CCO3)nn2)C2CCCC2)CC1 C(=O)(N1CC(C)(O)CO1)C1CC(NC(C(COC)(C)OC)=O)C1 C1(CC=C)(NC(C2CC=CCC2)=O)CN(C(=O)CNC(C2CCCC2)=O)C1 c1(C(N2C(C(C)(C)NC(C(C=C)O)=O)CCC2)=O)ncc2ccccc2c1O c1(C(=O)NCCCCN(C)C(c2cccnc2CO)=O)ccc(O)c(Br)c1 Cc1nn(C)c(Cl)c1C(=O)NCC(C(C)C)NC(c1cn(C(C)(C)C)nn1)=O C#CCC(C(=O)NCCC1CN(C(c2cnc(S)[nH]2)=O)CCO1)C1CC1 C12(CNC(CCC(C)NC(=O)CC3CCC34CCC4)=O)CC(C)(CCO1)C2 N1(C(c2cc(CC(C)C)nn2C)=O)CCN(C(=O)C=Cc2cscn2)C(CO)C1 N1(CCC(N2CC(C)C(NC(=O)COCC3CCCC3)C2)=O)CCP(C)(=O)CC1 C1(CNC(C2(C)CC2)=O)C2CCC(C2)N1C(c1csc(NC(N)=O)n1)=O C(CC(C(=O)N1CC(CNC(=O)CCC2(C#N)CCC2)C(C)C1)OC)OC Cc1ccc(CC(C)C(=O)O)s1.O1NC(=O)NC(=O)C1 Cc1cc(NC(C23CCC(NC(C4CC5CC(=O)C4C5)=O)(CC2)C3)=O)cnc1C C1(C(=O)NCC2(C(=O)OC)CCCO2)(OC)CCSC1 C1(C(=O)NC(CC)CNC(c2cnnn2C(F)(F)F)=O)CNC(=O)CC12CCC2 C(=O)(C1=COCCC1)NCCCCC(C)NC(C1C(C(=O)OC)C1)=O S(=O)(=O)(c1ccc2ncsc2c1)NC(C1(CNCc2ccc(C)c(Br)c2)CC1)=O N1(C(C2CCCCC2COC)C(=O)NC)CCN(c2ccccc2)C2CC12 c1(OCC)cncc(C(=O)N(C)CC2CCCC(NC(=O)CCOC)C2)c1 N1(S(CC)(=O)=O)CCCCC1C(N1CCCC(CNC(c2ccn(C)c2)=O)C1)=O Cc1ccc(-c2noc(CC(=O)NC3CC(NC(=O)CC4CCCO4)C3)n2)cc1 N1(S(c2cccc(C(C3c4cccc(N)c4CC3)=O)c2)(=O)=O)CCCC2(CCC(=O)N2)C1 C12C3CCC(C3)N1C(=O)C2.c1(C(=O)NCCCCCN(C)C)cccc(F)c1F C1(C(=O)NC(COC)C(=O)OC)CCN(C(c2conc2C)=O)C12CC2 c1(C(C(=O)NCC(CNC(C(C)c2ccon2)=O)O)=O)ccc(O)cc1 C=CCC(C(=O)NCC(C)(C1CC1)NC(=O)C(C)Oc1cccnc1)NC(C)=O C(CCCCC(=O)NC(C(F)(F)F)C1CCCC1)NC(C1N(CC)CCOC1)=O C1(NC(c2ccc(C)s2)c2nnnn2C)CC(=O)N(c2ccccc2)C1 C(CCCCC(=O)N1CC(C)(C)CC1CNC(C1(F)CCCOC1)=O)N(C)C c1(SCCC(N2C(CNC(C3(CC=C)CC3)=O)CC2)=O)ccccn1 c1(C(=O)NCC(CC=C)NC(=O)C(N2CCOCC2)(C)C)ccc(CO)c(F)c1 c1(NC2CCCC3CN(C(=O)OC(C)(C)C)CC32)nc[nH]c2ncc(C(=O)O)c1-2 CC1CC(NC(=O)C(F)(F)c2ccccn2)CN1C(=O)CN1CCC(C)(C)C1 Cc1nc(=N)[nH]c(=NCC(C)CNC(=O)CC23CCC(CC2)OC3)[nH]1 C=CCC(F)(F)C(=O)NCC1(CNC(=O)CCSCC(C)C)CC12CCC2 N1(C(CC2(C#N)CC2)=O)CCC2(NC(c3ccc(CCN(C)C)cc3)=O)CC2C1 c1(C(=O)NCC(C(O)C2CC2)C2CC2)cc([N+](=O)[O-])c(O)cc1N N1(C(C(C)OCCC=C)=O)C(CNC(=O)COCC2CCCO2)CC2CCCC12 C1(CC)(CC2CCOC2)CCCN1C(=O)NCC(F)F c1(C(C(=O)NCC2CC(NC(c3nc(CCC)sc3)=O)C2)O)ccc(Cl)c(Cl)c1 c1(C(N(CC(C)NC(C2(C3CC3)CC=CC2)=O)CC)=O)ccc2c(c1)NC(=O)C2 N1(CC(=O)N(C(C)C)CCN(C(=O)Cc2cccs2)C)CCC(C)(O)C1 N1(C(C(CC)SC)=O)CC(C(=O)NCCS(C)(=N)=O)CCC1C c1(C(N2CCC(OCCNC(=O)CCc3csnn3)C2)=O)cc(F)cc([N+](=O)[O-])c1 CC(C)C1=NOC(C)(C(=O)NC2CCCC(NC(=O)Cc3cnoc3)C2)C1 C1(C)(C(N2CC(C)(C)C(CNc3ncnc4[nH]cnc34)C2)=O)Cc2ccccc2N1 C12(C(N(C)CC3CC3(C)C)=O)CCC(NC(=O)Cc3cccnc3O)(CC1)C2 C=C(C)C1OCCC1C(=O)NCCCCC(N1CCN(C)CC1C)=O c1(C(=O)NCC2(C)CCCN2C(C2CCCC23CC3)=O)nc[nH]c2ncnc1-2 CC1CC(NC(=O)CSC2CCC2)CN(C(=O)CNC(c2ccccn2)=O)C1 C=CC(C)N=c1nc(N2CCC(c3nc4c(s3)CCC4)CC2)c2c([nH]1)CCC2 C12(NC(C#CC(C)(C)C)=O)CCCC1N(CC(O)COc1ccc(F)cc1)CCC2 Cn1cc(C=CC(=O)NCC2(NC(c3nn(C)cc3Cl)=O)CCOC2)cn1 N1(C(c2onc(C)c2C)=O)CC(NC(=O)CC2(C)CC2(Cl)Cl)CC2(CCC2)C1 CS(=O)(=O)c1ccc(Cl)c(S(=O)(=O)N2CCCCC2c2ncon2)c1 N1(C(c2n(C)ccn2)=O)CCCN(C(c2cc(C(F)(F)F)ns2)=O)CC1 C1(NC(c2cc(C)ncc2)=O)CCN(C(C2CC2C2CC2)=O)C12CCC2 C1(C(N2CC(CN(C(C=CCOC)=O)C)C2)=O)C(c2ccccc2)C1(F)F C1(Cn2cc(CCN(C)CC)nn2)CCCN(C(=O)CCCC2CC2C)C1 C(CS(=O)(=O)NCC(=O)NCCC(CCNC(C(C)OCCNCCO)=O)C)OC c1(CCC)ccc(C(N2CC3CC3(CNC(=O)C(C)C(C)(F)F)C2)=O)cc1N c1(OC)cc(C(=O)NCC(C2CCCCC2)NC(=O)CC(C)F)cc(OC)c1O C=C(C)C1CN(C(C23CC(C)(CN2C(c2cc(C#N)n(C)n2)=O)C3)=O)CCO1 C(=O)(CC(C)CC(=O)NC1CCC12CN(C(c1ccn(CC(F)F)n1)=O)C2)OC c1(CC)cc(-c2ccc(C(N3CC(F)CC3C(=O)OC)=O)nn2)ccc1F C1(CC(=O)NC2CC3CN(C(C4(O)CCSC4)=O)CC23)CCCC2(CCC2)O1 C1(O)(CNC(c2c(OCC)ccs2)=O)CCCN(C(c2scnc2C)=O)CC1 C(=O)(C(C)(C)F)NCCN(CC(C)O)C(c1scnc1C(C)(C)C)=O C(=O)(C1CCc2cc(F)ccc21)N1CCC(F)(CNC(C2C(=O)NCC2)=O)CC1 C12(C(N3C(CNC(C4C(=C)CC4)=O)CC3)=O)CCC(CC(C)(C)C)(CC1)CC2 c1(CC(=O)NCCCOCCNC(C2CSCCS2)=O)noc2cc(F)ccc12 c1(C(CC)NC(C(Cc2cc[nH]n2)NC(CC=C=C)=O)=O)ccccc1F C(CC(N)=O)(C(=O)NC1CCN(CC2CC2)C1)NC(C1(C#N)CCCC1)=O CCC(C)CC(=O)NC1CC1NC(C1CC1c1ccncc1Cl)=O C1(C(=O)NC2CC(C)N(C(C3CC(C(=O)OC)C3)=O)C2)CCC(C2CCCO2)O1 c1(OC)ccccc1NC(c1cn(C2CN(C(=O)COCC(F)F)C2)nn1)=O c1(OC)cc(C)cc(C(=O)NC2CC(NC(c3cc(O)nc(C)c3)=O)C2)c1C C12(O)CCCN(C1)C(=O)CC(=O)NC2.C1(C(=O)Nc2nccs2)CCOC(=O)N1 n12ncc3c1C(NCCC2)CCC3.N1(CC)CCCC(c2ccc(C(C)C)cc2)C1 CC(C(=O)NCCC1(O)CN(C(C2CC(=O)N(c3cn[nH]c3)C2)=O)C1)S(N)(=O)=O C12(NC(c3c(C)n[nH]c3)=O)CCCN(C(=O)Cc3ccccc3[N+](=O)[O-])CC1C2 C1(C2CC2)(C(=O)NCC2CCC(=C)CC2)CN(C(=O)CC(C)n2cccn2)C1 C1(F)(CNC(CN(C(=O)CC2CC2)C)=O)CCC1 C1(NC(=O)CC2CCC=CCC2)CCC2CN(C(=O)Nc3ccc(F)cc3)CC12 C#Cc1cccc(C(N2CCCC(CN(C(=O)CC3CCCO3)C)C2)=O)c1Cl N1(C(C(CC=C)C)=O)CCOCC(CNC(=O)CCc2cc(C)n(C)n2)C1 C(=O)(C(F)(F)C1CC1)N(CCCN(C)C)CCNC(C1CC(F)(CO)C1)=O C(=O)(CCCC#N)N1CC(CC(CNC(C(C)Sc2ccccn2)=O)(C)C)C1 c1(C(N(C2CN(C(CNC(CCC)=O)=O)CC2O)C)=O)ccn2c(C)cnc2c1 c1(N(C2CNCC(F)(F)C2)C(c2c(O)cccc2Cl)=O)ncc2[nH]ccc2n1 N1(CC(=O)N(C(C2CC2Cl)=O)CC)CC(=O)Nc2ccccc21 C1(NC(C2CC(C)CC(C)C2)=O)CCC2CN(C(C3CC3F)=O)CC2C1 CC(C)C(C)(O)C(=O)NCc1ccc(CNC(C2Cc3nncn3C2)=O)cc1F c1(C(=O)NCC(C)N(C(=O)C(Cl)=CCl)C)ccnc(N2CCC(C)C2)c1 CCCC(C(O)C(=O)NC1(C(=O)NC)CCC1)NC(c1coc(CC)n1)=O.CCF Cc1ccc(CC(N2CCC(N(CCO)C(C3(C)C=CCC3)=O)C2)=O)c(Br)c1 Cc1ccc(CC(=O)NCC2CN(C(=O)CC3COC(=O)C3)CCO2)c(Cl)c1 N1(C(CCc2c(C)n(C)nc2)=O)CCC(NC(=O)C(=O)NCC2CC2)CC(O)C1 C(=O)(N1CC(O)CO1)C1CCC(N(C(c2c(CC)ccs2)=O)C)CC1 N1(C(C(CCC)C=O)=O)CCC(N)CC(C)(C)C1.C(=O)(CC)NCC N1(C(C(COC)(C)OC)=O)CCC2(CC2)CC1C(=O)NCCC1CCCCCC1 N1(C(C(C(C)(C)C)O)=O)CC2CCN(C(=O)C3CCc4ccccc43)CC2C1 n1(CCC)cc(Cl)c(C(N2CCCC2CN(C)CC)=O)n1 C1(C(=O)NC2(CCC=C)CCN(C(=O)CC3CC3)CC2)CCCCC(F)(F)C1 CCC(O)CC(=O)NCCCOCCC(=O)Nc1cccc(Cl)n1 Cc1cc(O)ncc1C(=O)NCC1CC(NC(C2CCCN2C)=O)C1 C1(C)(C(=O)NC(C2CN(C(=O)CC(c3cccs3)N(C)C)C2)C)CC(C#N)C1 C(c1cnccn1)=CC(=O)NC1CC(CCC(=O)N(CC#CC)CC#C)C1 c1(C(N2CC(CC(=O)NC(C#N)C(N)=O)C2)=O)c(F)cc(Br)cc1Cl C1(CNC(=O)C(F)n2ccnc2)C2CC1N(C(C1CCC13CCC3)=O)C2 N1(C(C(CCC)C)=O)CCC(C2CCOCC2)(CNC(c2ccc(C)s2)=O)C1 C1(CNC(C2C(C)C2C)=O)CCCCC1NC(c1ccn(CCN(C)C)n1)=O c1(CC)ccc(C(=O)NCCC(C)NC(C2(N3CCOCC3)CC2)=O)o1 C1(C(=O)NC(C(=O)N(CC=C)CC)CO)CC12CCOCC2 c1(CNC(C2(CC)COC2)=O)ncncc1C(N1CC(F)(CO)C1)=O c1(SC(c2ccccc2)CCC)c(N=[N+]=[N-])cnnc1O c1(N(C(C)=O)CCN(C(C)CC2CCOCC2)CCN(C)C)ccccc1F C(C(CC)(CC)NC(=O)CC1CCC(=O)NC1)NC(C(CC)C1CCC(=O)N1)=O c1(CNC(C(C2CN(C(C(C=C)C)=O)C2)O)=O)cccc(C(=C)C)c1 C(CC(=O)NCCN1CCOCC1)(C(F)(F)F)NC(c1cn(C)nc1)=O c12nc(c3ccsc3n1)NC1(C3CN2C3)CC1.C1(OCCC)CCNCC1 C1(C(=O)NCC2(O)CCN(C(Cn3c(C)ccn3)=O)C2)CN2CCN1CC2C CC(CC(N)=O)C(=O)NCC1CCCN(C(=O)CC2CC3CCC2C3)CC1 C1(C(N2C(CN(C(C3CC(C)C3)=O)C3CC3)CCC2)=O)CC2(CSC2)C1 N(C(=NCc1ccc(N2CCOC(C)C2)cc1)NCC1CNC(=O)O1)C(CC)C c1(-c2ccc(CNC(c3cccc(NS(C)(=O)=O)c3)=O)nc2)cc(F)ncc1O N1(C(CC(C)C(F)F)=O)CC2CCCC(C1)N2C(C1NC(=O)CC1C)=O c1(C(N2CC(NC(=O)CC3CCCO3)CC(C)C2)=O)ccn2nnnc2c1 C(=O)(CC(C)(C)CNC(C1CN2CCC1CC2)=O)NCc1ccc(C)o1 c1(CNC(C2(CNC(=O)OC(C)(C)C)CC2)=O)cn(Cc2csnn2)nn1.C1CCCO1 C(=O)(C(C)C(F)(F)F)N(C1CCN(C(=O)CN(c2ccccc2)C)C1)CC C1(CNC(C23C(CN(C(c4nc(N(C)C)oc4)=O)C2)C3)=O)CN(C)C(=O)CCO1 C12(NC(c3cc(C(C)C)[nH]n3)=O)CC1CN(C(c1ncncc1Cl)=O)C2 C(=O)(C(CNC(C1CCCCS1)=O)N(C)C)NC1(C(C)C)CC1 CN1CCCC(C)(C(=O)NCC(C)(C)NC(c2coc(CC3CC3)n2)=O)C1 CC1CCC(C(=O)NC(C2CCCN2C(c2ccnn2CCF)=O)(C)C)O1 N1(c2ccnc(NS(C)(=O)=O)n2)CC(Cc2ccc(F)c(Cl)c2)CC(C)C1 C1(=O)C(Cn2cncn2)N1.C1(C(N(C(CSC)C)C)=O)CCN1CC.C(C)(C)(C)O Cc1ccncc1C1C(=O)N1.C1(CN(CCNc2cc[nH]n2)C(C)C)CCOC1 c1(C(=O)NCC2C(CN(C)C)C2)cccc(CNC(=O)COC(C)(C)C(F)(F)F)c1 C(=O)(C1=CCOCC1)NCC(c1ccccc1)NC(C(C)n1cnnn1)=O N1(C(C)=O)CCC(C=O)C1.c1(CC(=O)NCCCOCCNC)cn(C)nn1 CC(C)C(C)CC(=O)N1CCC(C(C)C(=O)NCC2=NOCC2)CC1 c1(CC(=O)NC(C)CN(C(=O)CC2CC(C)(C)C2)C2CC2)cccc(C(F)F)c1 C(CNC(=O)CSCC1CCCO1)(CC(F)(F)F)NC(=O)CC1CC1 Nc1cc(C(=O)N(C2CCN(C(=O)CC(F)(F)F)C2)CCO)cc(O)c1Cl C1(NC(CSCC#C)=O)CCN(C(c2csc(C(=O)NCC3CC3)n2)=O)CC12CCC2 c1(C(C)(C)C)ccc(Cl)cc1C(N1CC(C(N)=O)(CNC(=O)Cc2cnoc2)C1)=O n1(CC)nc(C(=O)N(CC(C)O)CCNC(=O)C(O)c2cnc[nH]2)c(C)n1 C#Cc1cnc(C(=O)NCC2CC2NC(c2ncoc2-c2cccs2)=O)c(C)c1 C12(NC(c3coc(CSC)c3)=O)CCC(CC1)N(C(C1(O)CC3CCC1C3)=O)C2 c1(CC(=O)NCC2C(NC(=O)CCc3nncs3)CC2)ccn(C(F)F)n1 n1(CC)ncc2c(NC(CNC(=O)CS(=O)(=O)C3CC3)C(C)C(C)C)ncnc12 N1(C(c2c(C)nn(C)c2F)=O)CCCC2(C1)CN(C(C1CNC(=O)N1C)=O)C2 C(=O)(C1=C(Cl)CCOC1)NC(CNC(c1nc(C)n(C)n1)=O)(C)C1CCC1 Cc1cc(Cl)c(NC(c2nc(C(=O)N(CC(O)C(F)(F)F)CCO)cs2)=O)cc1C C1(C(=O)OC)(C(N2CC3CC(NC(C4CSCC(=O)N4)=O)C3C2)=O)CCS(=O)(=O)C1 Cc1cc(=NC2CCc3nc(C)sc3C2)[nH]c(NC(c2cn(C)cn2)C)n1 C(=O)(C1=CCOC1)NC1C(NC(Cc2nc(C(C)(C)C)sc2)=O)CC1 c1(C(N2CCN(C(c3c(Cl)cc(C)s3)=O)CC2C)=O)cnc(C)c([N+](=O)[O-])c1 c1(C(N2CCC(NC(C3CC(=O)N(O)C3)=O)C(F)C2)=O)cc2c(s1)COCC2 NC1CC12CCN(C(c1ccc(C3(C(F)(F)F)CC3)cc1)=O)CC2 S(=O)(=O)(c1ccccc1CCC#N)NCc1c(C)cc(F)cc1 CC(C)CC(O)C(C)C(=O)N1CCC(NC(c2ccc(CO)s2)=O)C1C(C)(C)C N1(C(C2CCCC(C(=O)OC)C2)=O)C2CCC1CC(=O)NC2 C123CCC(CC1)(C2)C(=O)N3.C1(C(=O)NC(c2nn[nH]n2)(C)C)CC1C#N CC1(C)C(CNC(c2ccc(SC(F)F)cc2)=O)CCN1C(c1ccon1)=O C(=O)(C1SCCc2ccccc21)C(C(=O)N(CCC)C)=O.N(C)C C1(CNC(C2C(CC)C2)=O)CCN(C(=O)CCC(=O)c2ccccn2)C12CC2 N1(C(C(C(C)C)O)=O)CCC2(CCOCC2)C(NC(=O)CC2CC3CCC2O3)C1 C#CCC(C(=O)NCCC(O)CNC(c1cnccc1C)=O)C1CC1 S(=O)(=O)(c1cccnc1NC(C1CCC1)C)NCC1(C(C)C)CC1 N1(C(C(C=C)OC)=O)C(C(=O)N(C)CC2(CO)CCC2)CCC1C c1(C(=O)NC2C(CNC(C(C)c3cc[nH]n3)=O)COC2)cc2ncccc2o1 S(=O)(=O)(c1ccnc(F)c1C)N(S(NC1CC(OCC)C1)(=O)=O)C C(CCCC(CO)NC(=O)C(C)c1cc[nH]n1)NC(c1cccc(OCC)c1)=O Cc1cccn(CC(=O)NC2(C)CCN(C(C3CC(C)(F)C3)=O)C2)c1=O C(=O)(C1=CCC(NC(C2(CC(C)=O)CC2)=O)C1)NC(CC)CSC c1(C(=O)NCCOCCCNC(C(=O)NCCOC)=O)cccc([N+](=O)[O-])c1Cl S(=O)(=O)(c1cccc(F)c1)N1CCC2(C(NC(c3ccc(C)cc3C)=O)C2)CC1 CCC(C)(CC)C(=O)N1CCN(C2CCN(C(=O)CC3CCC(=O)N3C)C2)CC1 CCCCC(=O)NC1CCN(C(C23CSC(C2)C3)=O)C1 Cc1csc2c1CN(N1CC(c3nnc(CO)n3C)C1)C2 CCCN=C(NCCC(O)(CC)CC)N1CCCC(OC)C1.C1C=CCO1 c1(C(N(CCCNC(C2CC(C3CCC3)C2)=O)C)=O)ccc(S(N)(=O)=O)cc1F n1(CC)cc(Br)c(CC(=O)NCC(C)(C)Cn2cc(C(C)(C)CO)nn2)n1 c1(C(=O)OC)cc(=NCC(C)SC)nc(-c2ccccn2)[nH]1 C1(C(C)NC(C23CC(C#N)(C2)C3)=O)CCCN(C(=O)Cn2cnnc2)C1 C1(NC23CC(NC(c4c(N(C)C)c(F)ncc4)=O)(C2)C3)CCCN1S(=N)(=O)N(C)C C1(CC)CC(O)CCN1C(=O)CCCC(C)NC(=O)CC1CCCC(=O)N1 CC1(C)CC(NC(c2ccccc2O)=O)CN(C(c2nc(=N)cc[nH]2)=O)C1 c1(NC(Cc2c(-c3c(CC)scc3)cccc2)=O)c(OC)cccc1O C1(NC(c2ncc(OC)nc2)=O)CCC2CN(C(=O)Cc3n[nH]c(C)n3)CC2C1 N1(C(C(C)SCC)=O)CC(C(=O)NC(c2ncc[nH]2)C)C2(CC2)C1 c1(C(=O)NCC2CC(NC(CC3CN(C(C)C)C3)=O)C2)cc2cccnn2n1 c1(C(=O)Nc2c(CC)c[nH]c2)cc(F)ccc1CNC(c1ncoc1C1CC1)=O Cc1csc2ncc(C(N3CC(CNC(C4(C)CCCCC4)=O)CCC3C)=O)n12 c1(CC(N2CCC(c3ccc(F)cc3)CC2)=O)cnc2ccccn12 N12CC3CC(C1)C3NC(=O)C(C)CN(C)c1ccc(cc1)C2=O.COOC N1(c2nccc(OC)n2)CC=C(CNC(=O)CN2CC(=O)N(C)C2=O)CC1 C(C1=CCN(C(C2CC2(C)C)=O)CC1)NC(C(C)(C)NC(=O)NCC)=O CC1C(C(=O)NCC2(F)CC(NC(=O)C(C#N)C3CC3)C2)C1(F)F Cc1cc(CC(=O)N(CC(C)NC(c2c(Cl)csc2C)=O)C)cc(C)c1 C(=O)(CS(=O)(=O)CCO)N(C1CCCN(C(=O)CCc2cncs2)C1)CC c1(C(N2CCC(N(C(=O)CCc3cccnc3)CC)C2)=O)ccc(N)c(F)c1F C1(C(=O)NC(C)(CNC(=O)CC2CC2C(F)(F)F)C2CC2)(NC(C)=O)CCCC1.CN c1(CC(C)C)ncc(C(=O)NC(CO)C(C)NC(c2ccc(C3CC3)o2)=O)s1 c1(OC)cc2c(cc1C(=O)NC1CC1NC(c1ccccc1S(C)=O)=O)CCC2 C1(CNC(CCOCCCOC)=O)CCN(C(=O)C(N2CCSCC2)C)C1 C1(C)(CNC(C(F)=CC)=O)CCC(NC(=O)C=Cc2nccs2)CC1 C(CN=C(NCC1CC2CCC1CC2)N1CCC(NS(=O)(C)=O)C1)SC c1(SC)ccc(C(=O)N(CC(C)N(C)C(C2CCN(C)C2=O)=O)C)c(Cl)c1 N1(C(C2N(C(C3CC4(C3)CC(O)C4)=O)CC=C2)=O)CCC(O)C(F)(F)C1 C1(C(=O)NCCC(CC)(C)O)CCC2(CC2)N1C(c1oncc1CC)=O C1(O)(NC(=O)NCC(O)(COC(C)(C)C)CO)CCCN(Cc2n(C)c(Cl)cn2)C1 c1(C(N2CC(C)(CNC(COCC)=O)C(C)C2)=O)cccc2c1NC(=O)CC2 N1(C(C(C)Cn2ccnc2)=O)CCCC(C)(NC(C2CCCC(C)(C)O2)=O)C1 C1(NC(c2cn(C)nc2C(F)F)=O)CC2CCC1C(NC(=O)Cc1cn[nH]c1)C2 c1(C(=O)NCCSCC(=O)N(CC(=C)C)CC)snnc1C c1(C(c2cn(CC3CN(C(=O)C4=CCCC4)CCO3)nn2)C)cc(F)cc(Cl)c1 C1(C(C)NC(C2C(OCC)C2)=O)CCN(C(C2CCN(C(C)(C)C)CC2)=O)CC1 C1(N(C)C)(CNC(C(C2CCCN(C(=O)Cc3cnoc3)C2)C)=O)CCOCC1 N1(C(C2N(C)CC2)=O)CCC(C)(C)C(C(=O)NCC2CCCNC2=O)C1 CN1CCCC(C)(CC2(C3CC3)CCC2)C1.C1C(n2cc(C3CC3)nn2)C(=O)N1 CCCCC(CC)CC(=O)N1CC(F)CC1CC(N1CCN(C2CC2)C(C)C1)=O N1(C(CS(C(C)(C)C)(=O)=O)=O)CCC2(CC1)CCN(C(c1cc(=O)cco1)=O)C2 c1(C(=O)NC2CC(NC(c3c(C)onc3Cl)=O)C2)cc2ccccc2oc1=O CC1CCCC=C1C(=O)N1CC2CCC(N(C)C(c3cc(F)ccc3Cl)=O)C2C1 C1(NC(C(=O)NC(CC(N)=O)C2CC2)=O)CCC2(CC1)CC2CO C1(NC(CCOC(C)C)=O)CC(C2CCCN(C(=O)C=CC3CCOCC3)C2)C1 N1(C(C(C)O)=O)CC(NC(c2cnn(C(C)(C)C)c2)=O)C(c2ccnn2C)C1 C1(NC(C(C)OC(C)=O)=O)CN(C(=O)CCC2(C)CC2)CC1n1ccnn1 C=CCCCCC(=O)N1CC(OC)CC1CNC(c1cc(O)n(C)n1)=O C1(C(C)NC(=O)CCc2ccncn2)CCN(C(=O)CS(N)(=O)=O)CC1 c1(C(=O)NCCNC(C(C)NC(CC)=O)=O)cnn(C)c1 c1(C(N2C(C)CC(NC(C3(O)CCSC3)=O)C2)=O)ccc2nonc2c1 N1(C(CCC)=O)CCCCC1C(=O)N(CC(C)(C)CNC1(c2cccs2)CC1)C N1(C(c2cnn(C(C)C)c2N)=O)CCN(C(=O)Cc2ccc(Cl)s2)CC(O)C1 c1(C(=O)NC(CNC(C=C(C)C)=O)CC(F)(F)F)cc([N+](=O)[O-])ccc1Br CC1CN(C(=O)Cn2ccnc2)CC(C(=O)NCC2(CO)CCCCC2)O1 C(C(C)C(F)C(=O)N1CC(C)(C#N)C1)NC(CC1CC(SC)C1)=O c1(C(=O)NC(CNC(c2c(C)nncc2)=O)CO)cccc2c1COCC2 C=CCC(C)C(=O)NC1CCN(C(c2cc(C3CCCC3)n(C)n2)=O)C1 C12(C(=O)Nc3n(CC)nnc3)CCC(C(N3CCC(O)C3)=O)(CC1)CC2 C1(C(=O)NCCC(C)NC(C2CC3(CCOCC3)C2)=O)CCCCC(F)(F)C1 N1(C(C2CC(CN(C)C)C2)=O)CC2(CCN2C(=O)Cc2cc[nH]n2)C1 C1(C(=O)NC(CC)(CC)C(C)C)CC(C)(C)CCN1C(=O)CC(O)CN(C)C Cc1cn(C(C)C)cc1C(=O)NC(C)CCCNC(c1cc(C)on1)=O c1(NC(CC(CNC(c2c(CC)n(C)nn2)=O)O)=O)cnc2ccccc2c1 C12(CNC(=O)Cc3cncnc3)CC1CN2C(c1ccc(C2CCC2)cc1)=O Cc1nc(C(=O)NCC(C)(CC(C)C)NC(c2nc(C)oc2C)=O)cc(O)n1 C1(C(=O)NC(c2nc[nH]n2)C)CC2C=CC1N(C(C13C(=O)C4CC1C3C4)=O)C2 S(=O)(=O)(c1cccc2c1OCCO2)N1C(C)C(=O)NC(=O)C1 C1(C(N2CCCC2c2cnn(C)c2)C(=O)NC(C)C2CC2)CC2C(C1)C2(F)F c1(C(N2CCCC(O)C2)=O)cncc2[nH]ccc12.C1(N(C=O)CC)C2CC3C(C2)C13 C1(C(N2CC(CCNC(c3c(C)ncs3)=O)OCC2)=O)COCC(=O)N1C(C)C CC1C(NC(=O)CC2NC(=O)NC2=O)CCCN1C(=O)Cn1ccnn1 N1(C(C2(N(C)C)CCCC2)=O)CCC2OCCN(C(c3cc(O)n(C)n3)=O)C2C1 Cc1cc(-c2ccc(CNC(c3ncn(C(C)C)n3)=O)nc2)cnc1C#N c1(C(=O)NCC(=C2CN(C(c3c(C)nn(C)c3)=O)C2)F)cc(Cl)ccc1F C1(F)(C(N(C)Cc2ccc(CO)cc2)=O)CCCN(C(C2COCCN2C)=O)C1 C(CCCCCNC(c1ccc(C2CCOC2)s1)=O)NC(C1(CC#C)CCC1)=O CCCS(=O)(=O)c1ccccc1C(=O)NCC1COCCN1C(=O)CC1CSC1 CC1(C(=O)NC2CC(NC(c3cccnc3O)=O)C2)CCC2CC2C1 C(CC(N)=O)(C(=O)NC(CC(F)F)C(C)C)NC(C(CC)OC)=O N1(C(c2cc(CC(C)C)on2)=O)CC(C2(NC(=O)Cn3cnc(C#N)n3)CC2)C1 c1(CNC(CC2C(NC(C(C)OCCC#C)=O)C2)=O)ncc(CC)[nH]1 c1(OC)c(Cl)cc(C(=O)NCC2CC(F)(F)CN2C(C2CNC(=O)C2)=O)cc1Cl C1(C(N(CCCN(C(C(C)NC(N)=O)=O)C)C)=O)CC1C1CCCC1 C(=O)(CCC(C)(F)F)NCC1N(C(C(C)NC(=O)C=Cc2cn[nH]c2)=O)CCC1C N1(C(CN(CC(C)(C)C)C)=O)CCCC(CC(=O)NCCCOCC2CC2)CC1 C1(C(=O)NCC2CN(C(C(CCOC)O)=O)C2)CN(C(C)C)c2ccccc2O1 c1(N(CCN(C(C)C)C(c2ccc3cc[nH]c3n2)=O)C)nc2cc(Br)cnc2s1 C1(CC(=O)NCCN(C(CC=C(C)C)=O)C(C)C)CCN(C)C1 c1(CCC)cc(CN2C(C(=O)NCC(=O)OC(C)(C)C)CC2)nn1C c1(NC2(CNC(c3[nH]cc(CC)c3)=O)CC2)cc(CC)nc(C)n1 CC(O)C(N)C(=O)NCC1(CO)CC2CC2C1 c1(C(C)=O)cc(C(=O)NCC(C)(C)CNC(=O)CCOCC(F)F)cnc1C c1(CS(=O)(=O)NCC(c2cccnc2F)(C)C)cc2c(s1)CCCC2 C1(C(N2CCC(CS(=O)(=O)NC)C2)=O)CC(=O)N(C)C1c1cccs1 n1(CC(=O)NCCN(C(=O)C(C2CCC2)N(C)C)C(C)C)cnc([N+](=O)[O-])n1 C(CCN(C)C(C12COCC(C1)OC2)=O)(C(C)(C)C)NC(c1c(C)n(C)cc1)=O c1(C(=O)NC2CCC(CNC(=O)C(c3cccc(F)c3)O)C2)cc(O)ccc1Cl c1(NC(c2c(NC(C3C(C)C3)=O)c[nH]n2)=O)ccc(F)c(Cl)c1F n1(CC(=O)NC2CN(C(C3C(C)=CCC=C3)=O)CC2F)nc2ccccn2c1=O N1(C(C(CC2CCC2)OC)=O)CCC(CNC(C2(C(F)(F)F)CC2)=O)C1(C)C C1(C(=O)N(CC(C)SC)C)(COC)CCN(C(=O)C=CC2CCOC2)CC1 N1(C(c2c(C)cccc2F)=O)CC2CCCC(Nc3ncnc4ccsc34)C2C1 N1(C(C(C)(C)OC)=O)CCC(O)(CCN(C(=O)COc2ccon2)C2CC2)C1 Cc1cc(-c2nc(C3CCOCC3)nn2C2CCSCC2)ccc1C1CCOC1 C(=O)(CCCCCC(C)O)NC(c1ccc(-c2c(C)cc(O)cc2)cc1)CC(=O)O C1(NC(C(C(C2CC2)OCC)N2CCC(C(=O)OC)C2)=O)CCC(F)(F)CC1 N1(C(C2(C)CC2(F)F)=O)CC2CC2(NC(c2ccc(C#N)[nH]2)=O)C1 C12(NC(=O)C3CC3)CCCC1N(C(=O)Cc1ccoc1)CC2 CCC(C)C(O)C(=O)N1CCC(N(C(c2cc(F)ccc2SC)=O)CC)CC1 c1(OC)ccc(F)c(CN2CCCC(NC(C3CC3C)=O)C2)c1 Cc1cc(C)c(C(CO)NC(=O)CCc2cc3ccccc3[nH]2)c(C)c1 Cc1cn2cc(C(N3CCC4CN(C(=O)CCCC(C)C)CC4C3)=O)ccc2n1 Cc1ccc(CC(=O)NCC2(NC(=O)CCC(N)=O)CCCCC2C)c(Br)c1 N1(C(C2(SC)CC2)=O)CCC(CNC(=O)CCCSCC(C)C)C(C2CC2)C1 c1(C(=O)NCC2(CN(C)C(c3cccnc3)=O)CC2)[nH]nc2c1CCC2(C)C C#Cc1ccnc(C(N2CCCC(C(C)C(N3CCC(C)(OCC)C3)=O)C2)=O)c1 C(=O)(C(C)CC(C)(F)F)NC(c1ccc(OC)cc1)CNC(C(COC)(F)F)=O CCC(O)C(F)(F)C(=O)NC1CCCC(NC(=O)C(c2cccnc2)O)C1 N1(C(c2cccc(CC)c2)=O)CCN(C(=O)C(F)CC2CCCC2)CC1COC C1(CCNC(C=Cc2c(C)ccs2)=O)CC(F)(F)CN1C(=O)CC1C=CCC1 CCCCCC(O)CC(=O)NCCC1CC(NC(c2cc(C3CC3)n(C)n2)=O)C1 c1(C(=O)NC2COCCN(C(=O)OC(C)(C)C)C2)cc(O)nc2ccccc12 CC(C)C(F)(F)CC(=O)NCC1(CNC(C2(C)CC3CC3C2)=O)CCC1 N1(c2ccc(S(=O)(=O)NCC3CN(C)C(=O)C3)cn2)CC2CS(=O)(=O)CC2(C#N)C1 C1(CC(=O)NCC2N(C(c3c(C)cccn3)=O)CCCC2)CCCC(C)(C)CC1 C1(CNC(C(CCC)O)=O)CCN(C(=O)CC(C)(C)C)C1(C)C C(C)(C(C(=O)NCC1(CCCF)CC1)C(C)C)NC(C(CC(C)C)=O)=O C1(CNC(c2cc(CC)[nH]n2)=O)CCN(C(c2c(C)cnn2C)=O)CC1C Cc1cc(C(=O)NCCCOCCNC(c2ccoc2C)=O)c(C)n1NC(N)=O c1(OC)ccc2c(CC(N3CCCC(N(C(=O)C(C)CF)C)C3)=O)coc2c1C CC(C)(O)C#CC(=O)NCC1(C(C)(C)C)CCN(C(C2CN3CCN2CC3)=O)C1 C=CCCC(C(=O)N=c1ccn(CCNC(=O)C(O)C(F)(F)F)[nH]1)NC(C)=O C#CCCCCC(=O)NC1(CCNC(=O)CN(C)CC)CCCC1 N1(C(CSCC=C)=O)CCC(O)(CCNC(=O)C(C)Sc2ccccn2)C1 C1(C)(OC)CCCN(C(=O)CC2CN(C(=O)CCc3ncccc3C)CCO2)C1 c1(CC(N2CCCC(NC(C3C(=C)C3C(=O)OC)=O)C2)=O)cc(F)ccc1O c1(C(N2CC(OC3CN(C(CC4(C)CC4)=O)C3)C2)=O)ccc(-n2cccc2)cc1 C(CCCC(=O)NC1CCCC1NC(C1(N2CCOCC2=O)CC1)=O)NC(=O)OC C1(CCNC(c2cc(C)n(CCO)n2)=O)CCCN(C(=O)C=CCO)CC1 Cc1ccc(C(N2CC(NC(=O)Cc3ccnn3C)C3CC23)=O)cn1 C#Cc1ccc(C(=O)N(C)CCOCCNC(=O)C(C)(C)C#CC)c(C)c1 C(=O)(CC(CC(C)C)NC(C1CCCC(CF)C1)=O)NC(C#C)C c1(C(=O)NC2CN(C(C3C4CC4C4CC34)=O)C2)c[nH]c2cccc(Br)c12 C1(F)(CNC(COCCCC)=O)CCN(C(c2n[nH]c(C)c2O)=O)C1 c1(OCC)cc(Br)c(C)nc1NC(C1CC1NC(=O)Cn1cc(Br)cn1)=O N1(c2nc(C)nc(=N)[nH]2)CCC(C)(C)C(CNC(=O)CC2CC(C)OC2C)C1 c1(C(=O)NCC2C(NC(C3CN(C(=O)NC)C3)=O)C2)cnn(CCOC)c1 C(=O)(C(F)C(C)C(F)(F)F)NCCCOCCN(C(C=CCCC(C)C)=O)C c1(N2CCC(CC)(NC(=O)CC3(O)CCCC3)CC2)ncc2c(C)cccc2n1 N1(C(C2CCC(CC)CC2)=O)C2CCC(C2)C1CNC(C1CC12CCC2)=O N1(C(c2c(C)nsc2)=O)CC(CNC(c2ccc(CO)nc2)=O)OC2(CCC2)C1 Cn1cc(C#CCNC(=O)CCN(CCCO)C(C2CCC3(CC3)C2)=O)cn1 N1(C(C(C)=C2CCCC2)=O)CCCCCCC1C(=O)NC(c1ccoc1)C CCC(C)(CO)C(=O)NCC(CNC(c1csc(N2CCCCC2)n1)=O)OC N1(C(=O)CCc2ccc(F)c(F)c2)CCN(C(=O)COC2CC=CC2)CC(O)C1 c1(C(N2C(C(N3CCC(OC)C3)=O)CC3CC32)=O)cn(CC#N)c2ccccc12 Cc1cn2ccnc(C(N3CC(NC(c4ccoc4)=O)C4(CC4)C3)=O)c2n1 N1(C(COCCOC)=O)CCC(C)C1CNC(=O)Oc1ccccc1Br Cc1noc(C(C)C)c1C(N1CCC(C)(NC(=O)C(C)c2ccco2)C1)=O C(=O)(C1=NOC(C)(C)C1)NCC(C(C)C)NC(c1cc(Cl)ncc1Cl)=O CCC(CNC(C1CN(C(C2CCC=CCC2)=O)CC1F)=O)(CC)OC c1(C(=O)NC2(CNC(C3CCS3(=O)=O)=O)CCSC2)ccnc(CO)c1 c1(CC(=O)NCC2CN(C(c3c(C)csc3Cl)=O)CC(C)C2)cnc2ncccn12 c1(C(=O)NCC2(C)OCCN(C(C(F)=CC)=O)C2)ccc2c(c1)CCN2C C#CCC(O)C(=O)N(C(CNC(c1cc(C(N)=O)co1)=O)C1CC1)C N1(C(c2c(C(C)C)c[nH]c2)=O)CCC(F)C(NC(=O)C(C)C#N)C1 n1(C2(C(C)NC(C(C)N(C(COCC)=O)C3CC3)=O)CC2)nccn1 CS(=O)(=O)c1cccc(Cl)c1C(=O)NC1CC(O)CN(C(=O)Cc2cnns2)C1 c1(C(=O)NCC2CN(C(=O)C3=CCCC3)CCO2)cc(Br)nc(Br)c1 C1(C)(CN2CCN(C(c3c(C)nc(C(F)(F)F)o3)=O)CC2)CCC(=O)NC1 Cc1cccc(-n2cc(C3CCN(C(C)CC(C)(C)O)CC3)nn2)c1F Cc1sc2ncc(C(=O)NC(C)CCCCNC(=O)CC3CCC(=O)N3)n2c1C C(=O)(C(CO)C(F)(F)F)OCC(=O)Nc1c(CC)nccc1C c1(C(=O)NCC2COCCN(C(c3cccc(C)n3)=O)C2)cc2c(s1)COCC2 CC(C)C(CNC(=O)CC1CCC(C)CO1)C(=O)Nc1cnccc1C1CC1 N1(C(C(CO)OC)=O)CC2(CCN(C(=O)CCC(C)CN(C)C)C2)C1 C1CCC(=O)N1.N1(C(C2CO2)=O)CC=CCC1.C=C1CC(CC(=C)C)C1 Cc1nc(CCNC(=O)CC2CCCC2NC(=O)C(O)CN(C)C)cs1 C1(NC(C2CC3(CSC3)C2)=O)CN(C(c2cc(O)cs2)=O)Cc2ccnn2C1 Cc1cc(N2CC(N(CC(O)CN(C)C)C)C2)n2ncnc2n1 N1(CCCCNC(C(C)NC23CC(F)(C2)C3)=O)CCc2sccc2C1 C1(CNC(C(CC)N2CCCC2=O)=O)CCN(C(c2cc(C)on2)=O)CC1CC N1(C(c2ccn(CC)n2)=O)CCC(C(F)(F)F)C(NC(C2CC2C#N)=O)C1 c1(OCC)c(F)c(C(N2CCN(C(=O)C(C)C(C)CC)CC(O)C2)=O)cc(F)c1F c1(CC(=O)NCC(C)N(C(C2(CC)CC2)=O)C)cc(F)ccc1F c1(C(=O)NCC(C)N(C(C(C)OCCC#C)=O)C)ccc(C(C)(C)C)nc1 C1(NC(CSC(C)C)=O)CCCC1C(N1CCC1C1CCCC1)=O c1(C(=O)Nc2ccccc2)cccc(CN(CC(=O)NC2CCCO2)C)c1 C1(CNC(C=C)=O)CCC(F)(CNC(=O)C(C)(C)CCOC)CC1 c1(CC(=O)N(C)CC2CCN(C(CC(C(C)C)O)=O)C2)ccc2nsnc2c1 C1(N(C(c2ccc(OC)o2)=O)C)CCCN(C(=O)C(C(C)OC)N(C)C)C1 C(CC(C)C)(C(=O)N(CCC)CC)NC(CCCOCC=C)=O N1(C(c2c(C)n(C)cc2)=O)CCCC(NC(=O)CSc2n[nH]c(O)n2)C1C c1(OC)c(C(N2CCC(C(C)C(=O)N(C(C)CC(C)C)C)C2)=O)cnn1C c1(NC(=O)NCc2nc3n(c2)CC(C)CC3)ccc2c(c1)CCCS2(=O)=O CN1CC(=O)N(CC(N2CC3C(CNC(c4cc5sccc5s4)=O)C3C2)=O)C1=O C1(N(C)C(C2C(Cl)(Cl)C23CC3)=O)CN(C(=O)CCS(N)(=O)=O)CCC1CC1CC1 C1(NC(C2(C=C)CNC2)=O)CC2OCCCC12 C(=O)(C(C)(C)C(=O)NC1CCN(C(c2cnc(S)nc2)=O)CC1C)NC CCCCCC(O)C(C)C(=O)N1CCCN(C(=O)CC(F)(CC)C2CC2)CC1 Cc1cnc2c(CN3CCN(CC(=O)Nc4ccc(F)cn4)CC3)cnn2c1 c1(C(=O)NC2CCC(CNC(C(CCOC)(C)C)=O)C2)coc2cc(O)ccc12 N1(C(C(CC#C)C2CC2)=O)CC2CCC2(CC(=O)NC2CC(OC(C)C)C2)C1 C1(N(C(C(F)OC)=O)C)CC2CC1N(C(c1ccoc1C1CC1)=O)C2 C=CCC(C)(C)CC(=O)N1C2CCC(C2)C1CNC(=O)COC(C)CC C=CCC(CC=C)C(=O)NC1CCCN(C(C2CCOC(CCC)C2)=O)C1C Cc1ccc(CN(C(C2CCOC(C)C2)C(=O)NCCC#N)CC2CC2)nc1 C1(CCC)CN(C(=O)C2CC2C2CCC(C)(C)CO2)CCN1C(=O)Cn1cnnn1 C1(C)(NC)CCN(C(=O)C(C)(C2CC2)N(C(=O)CCc2cccn2C)C)CC1 C(=O)(C(C)C(F)(F)F)NC1CN(C(CC(OCC)OCC)=O)CC1C C1(NC(c2ccc(CN(C)C)[nH]2)=O)CC2(C1)CN(C(c1cnn(C)c1Br)=O)C2 C(N=C(NCCOCCOC)N1CCN(CC)C(C)C1)c1ccc(C(=O)OCC)cc1 C1(CCCC)CCCN(C(=O)CNC(=O)NCC2CCCC2(F)F)C1 N#CCCCC(=O)N1CCCCC1CC(=O)NCC1(C(N)=O)CC1 C(C(C(=O)NCc1ccon1)C(C)(C)C)NC(CC(C)CN(C)C)=O C1(C)(C(=O)NCC(CO)NC(C2(C)N(C(CCC)=O)CCC2)=O)CCCCCC1 c1(NCC2CCN(C(C(CCC)NC(N)=O)=O)C2)cc2nc(CCC)nn2cn1 c1(C(N2CCC(C(C)NC(c3cnc(OC)nc3)=O)C2)=O)cccc2c1NCC2 CC1(CNC(C2CC2C(N)=O)=O)CCN(C(=O)NCC2CC=CCC2)C1 C1(NC(CC2(COC)CC2)=O)CCN(C(c2ncsc2Br)=O)C(C)C1 C1(NC(CC(CC)C2CCC2)=O)CC(C(=O)N2CCCC2(C)C2CCC2)=CC1O Cn1cc([N+](=O)[O-])c(OCC(=O)N(C2CC2)C(c2ccccc2)C2CC2)n1 c1(C(N(CC(N2CCC(Cc3nnc(C(C)=O)s3)C2)=O)C)=O)ccc(Br)cc1F C1(C(=O)NC2CC(F)(CNC(c3c(CC)n(C)nc3)=O)C2)CC12CCCCC2 CCCCC(CNC(c1cnn(C)c1)=O)NC(c1cccc(CC(F)(F)F)c1)=O C1(C(N(C(COC)C)C)=O)CCCC1CNC(C12COCC1C2)=O c1(CC(C(=O)O)NC(c2c(C)noc2N)=O)c[nH]c2cc(F)ccc12 c1(C(=O)NC2C(CNC(C(C)NC(C)=O)=O)CC2)ccc(C2CC2)nc1O C1(C(=O)NCC2CC(O)CN2C(c2cscc2Br)=O)CC12CCCCC2 Cc1c[nH]nc1C(=O)NCCC1(CCO)CC1.n12cc(nn1)C2.c1(O)ccccc1 N1(C(C2(COC)CCOCC2)=O)C2CCC1CC(NC(C1CCS(=O)(=O)N1)=O)C2 C(c1cnc(O)nc1O)=CC(=O)NC(CNC(CCC=C(C)C)=O)CC(C)C C1(N(C(CCC#C)=O)CCF)CCCN(C(=O)CC(=O)NCCCCCC)C1 c12ncc(C)cc1S(=O)(=O)NCC(C1CCCCC1)Cc1ccccc1CN2.OC Cn1nc(O)cc1C(N1CC(F)CC1CNC(c1cnnc(Cl)c1)=O)=O c1(NC(C2CCS2(=O)=O)=O)cc(C(=O)NC(CN(C)CC2CC2)C2CCC2)ccn1 CC1OC(C)C(C(=O)NCC2COCCN(C(c3c[nH]ccc3=O)=O)C2)C1C C1(C(=O)NCC2([Si](C)(C)C)CC2)CN(C(C2CCCS2)=O)C2(CCC2)C1 CC1CCCC1(C)C(N1CC2CC1C2NC(c1c(Br)noc1C1CC1)=O)=O CC(C)(C)CCCC(=O)N1CC2CC1C2NC(=O)CC1COCC(C)(C)O1 N1(S(CC)(=O)=O)CCCC1C(N1CCC1NC(=O)CN(C)C(C)C)=O c1(-c2nc(C)sc2)ccc(CCNC(=O)NCC2CCC(=O)N2)cc1 C1(C(N(CCO)CC)=O)CCCCC1n1cc(C2CC3CCC2C3)nn1 C(N=c1ccc2nnnn2[nH]1)C1(C)CC1Br.C12(CCC1)NC(=O)C2 n1(CC)cc(C(N2CCCC2C(=O)OC(C)(C)C)=O)c(C2(CC)CCOCC2)n1 c1(C(c2nnnn2C(C)(C)C)CCCN)cccc(N(C)C)n1.CN(C)C(N)=O N1(C(C2CC(N(C)C)C2)=O)CC2CCC(C1)N2C(C12CCN(CC1)C2)=O C12(NC(c3cc(CO)[nH]n3)=O)CCCC1N(C(c1cc(=O)cc(Cl)[nH]1)=O)CCC2 C1(NC(C(C=CC)O)=O)CCC(O)CN(C(=O)CCOc2cc(F)ccc2F)C1 C=CC(C)(C)CC(=O)N1CCCC1C1(C(=O)N(C(C)C(C)CO)C2CC2)CC1 c1(C(=O)NCCN(C(=O)C=Cc2ccc(Cl)s2)C)cncn(C)c1=O c1(C(C)C)scnc1C(=O)NC1CCCC1CNC(=O)CC(C)N(C)C C(=O)(C#CC1CCOC1)NCC(C)C(C)(C)C(=O)NCC1=NOC2(CCC2)C1 Cc1c(Cl)ccnc1C(=O)N(CCN(C)Cc1ccc(C#N)cc1)C(C)C C1(C(N2CC(NC(CSC)=O)C(CC3CC3)C2)=O)C(F)(F)C12CCC2 C1(CNC(c2c(CC)c[nH]n2)=O)CC(C(=O)Nc2cnc(OC(C)C)nc2)=NO1 CCC(CC(F)(F)F)C(=O)N(C1CCC(NC(=O)C2=C(Cl)CCOC2)CC1)C c1(OC)cccc(NC(=O)CC2CCN(C(=O)C(C)Cn3cccn3)CC2)c1 c1(NC(c2nc(C)c(Br)s2)c2nnnn2C2CCC2)ncc(F)cc1Cl N1(C(c2ccn(C)n2)=O)CCN(C(=O)CSc2ncccn2)C(C#N)C1 c1(CC(=O)NC2CC(C)(CC)N(C(C3(SC)CC3)=O)C2)ccc(Cl)c([N+](=O)[O-])c1 CCC(C)(C)CC(=O)N1CCC(c2nnnn2C)(C(=O)NCCSC)CC1 Cc1cccc(-n2nnnc2SCC(=O)Nc2ccn(C3CCCC3)n2)c1 c1(NC(=O)Cc2ccno2)nc2c(s1)CC(Nc1cccc(C#N)c1)CC2 c1(OC)cnc(C(=O)NCC2C3CC2N(C(=O)C(C(C)C)SC(F)(F)F)C3)nc1 c1(OC)ccc(CC(N2CCCC2CCNC(=O)C(C2CCC2)OC)=O)s1 N1(C(C2CCN(C(C)C)C2)=O)CCCCC1(C)CO Cc1cc(-c2cn(CCNC(C3CCC(CCC(C)C)C3)=O)nn2)cnc1C C1(CC)CN(C(c2ccc(OC(C)=O)c(F)c2)=O)CCN1C(c1occc1Br)=O C(=O)(C1=CC2CCC(C1)C2)N(C1(C(N(C2C(C)COCC2)C)=O)CC1)C c1(CC)cc(C(N2CC(NC(=O)CCc3cc(C)on3)CCC2C)=O)cc(O)n1 c1(-n2c(CCCC#C)nc(CCC(C)C)n2)ccc(F)cc1F N1(C(CSCCC#N)=O)CC2CC(C(=O)NC(CCO)C(F)F)(C2)C1 N1(C(C(C)=CC)=O)CC2CCC1C(NC(=O)C=CC1CCCC1)C2 C=C(Br)CN=c1[nH]c(N2CCC(CO)C(C)C2)nc2c1CCC2 c1(C(=O)NC(C2(O)CN(C(c3c(CC)nco3)=O)C2)C)cc2cc(F)ccc2s1 C12(CNC(c3c(C)[nH]cc3)=O)CC(CCO1)N(C(c1cc(Cl)ccn1)=O)C2 c1(C(=O)NCCC(C)NC(=O)CCCCc2ccc(F)cc2)ccc(N)c(F)c1 c1(C(=O)NCC(CCNC(c2nn(CC)c(C)c2)=O)O)cn2cc(Cl)cnc2n1 c1(C(=O)NC2CCN(c3nc(Cl)ncc3Br)C2)cc2cn[nH]c2cn1 N1(CC(C)C)CCC(C(=O)NCCCCN(C)C(c2cc[nH]n2)=O)CC1 N1(C(CCOC)=O)CCC(C(N2CCOC(C#N)C2)=O)C12CC2 C12(C(=O)NCC3=CCN(C(c4c(C)cccc4O)=O)CC3)CC=CCN1CCC2 C1(C(N2CCC(O)(CNC(c3ccc(OC)nn3)=O)C2)=O)CCCCC(F)(F)C1 C12(C(=O)NC(CC)CN(C(=O)Cc3ccc(F)cc3)C)CCN(C1)S(=O)(=O)C2 C1(NC(=O)C(c2ccccc2)O)CCN(C(=O)CCc2cncnc2)C12CCC2 C=CCC(CC)C(=O)NCC(CC(F)(F)F)NC(c1cnc(N)c(N)c1)=O C=C(Cl)C(C)(C)C(=O)N(CC(C)(C)NC(=O)CC1CCC1C)C C(CC)(CC)(CCNC(=O)CC1CCCN1C)NC(C(CC)COC)=O c1(C(N2CC(CC(N3CCC(O)(C(N)=O)C3)=O)C2)=O)cc2ncccc2[nH]1 c1(C(N(CCOC)CCNC(C2CC23CC(F)(F)C3)=O)=O)ccc(C)c(Cl)c1F C(C(=O)N1CC=CC1)(C(C)(C)C)NC(C1(SC)CC1)=O N1(C(c2cccc(C)c2N)=O)CCC2(CC1)COC(c1ccccc1)C2 CC1(C)CN(C(C2CCOC2)=O)CC(CNC(C2(C(F)F)CCC2)=O)O1 C=CC1(NC(c2csc(Cl)n2)c2nnnn2C2COC2)CCOCC1 N1(C(C)C)CC2CC1CN2C(=O)C(C(C)(C)O)NC(=O)CNC(C1CC1C)=O c1(C(N(C2CN(C(c3cn(C(C)(C)C)nn3)=O)C2)C)=O)ccc(C(N)=O)nc1 CC(CCCC(=O)NC(c1cccs1)C)NC(=O)CCS(N)(=O)=O C1(NC(C(C(C)C)F)=O)CC2CC(NC(=O)CN3CCCCC3)C1C2 N1(CC(=O)N(CCCCCNC(C(C2CC2)SC)=O)C)C(=O)C(C)C(C)C1=O C12(OC)CCC(C(=O)OCC(=O)N(C3CC(O)C(F)C3)c3ccccn3)(CC1)C2 C1(C(N(C2(C#C)CC2)C)=O)CCN(C(=O)CC2(N(C)C)CC2)CC1(C)C c1(NCC(C(C)C)NC(c2ccc(C)s2)=O)ccnc(-n2ccnc2)n1.C1CC1 C(=O)(C(F)C(C)C(F)(F)F)NC(CC(C)NC(C(C(C)C)F)=O)C c1(OC)ncc(-c2n[nH]c(CNC(=O)C(=O)NCCN)n2)cn1 CCC(CC(=O)N(CCC(=O)NC(COC)CCO)CCCO)C(C)(C)C C(CCN1CCN(CC(N)=O)CC1)(C(C)C)OC.C(=O)(C1CC1)O C(c1c(F)cccc1F)=CC(=O)NCC1C(C)CCN1C(=O)C(=O)NC1CC1 c1(C(=O)NCCCN(C(=O)C(C)CN(C)C)CC)cccnc1OC(F)F CCC(C)(O)C(=O)NCCCN(C(=O)C(C)(C)N1CCCCC1)C1CCCC1 c1(C(=O)NCC2(O)CN(C(C(CO)OC)=O)C2)cc(F)ccc1-n1cccn1 Cc1c(C=CC(=O)NC(CNC(C2OCCC2(C)C)=O)C(C)C(C)C)cnn1C C(C(=O)NCC1(O)CCCN(C(=O)CC(C)(F)F)C1)(C(C)(C)C)SC C(=O)(C1=C(C)OCCS1)NCCC(C)N(C(=O)CC1CC(N(C)C)C1)CCC Cc1ncnc(O)c1C(=O)NC(CNC(=O)CC1C=CCCC1)C(C)C CCC(C)C(CC(=O)NC(C(F)F)C(C)(C)C)NC(c1sccc1C)=O c1(CNC(=O)NC(C)CCC(F)F)c(Cl)ccnc1Br C(CC(O)CNC(C1CC1CF)=O)NC(c1ccc(-c2ccco2)o1)=O C1(NC(c2n(CCC)ncc2)=O)CCCCC1CNC(=O)C(C)(C)c1ccsc1 n1(CC)nc(C(=O)NCc2csc(C(=O)NCC(O)CN(C)C)c2)c(C)n1 Cc1ccc(C(=O)NCCC2CN(C(=O)CCCC3CC3)CCO2)cc1C N1(C(C(C2(O)CCC2)NC(=O)CC(C2CC2)C2CC2)=O)CCCOCC1 C=CC(C)C(C)C(=O)NCCOCCNC(c1cnc(CC2CC2)s1)=O CC1(C(=O)NCC(CNC(c2nccc3nn[nH]c23)=O)CO)CC(C2CC2)=NO1 C(=O)(C1=CCCOCC1)NC1C(CC(C)(C)C)CN(C(C2CC(O)C2)=O)C1 c1(C(=O)NC2C(NC(C(Cn3ccc(C)n3)C)=O)CC2)cncnc1C(C)(C)C C1(C(C)C)CCC(C)CC1NCC(=O)NCC1CCCN1C(c1cscc1Cl)=O C1(CNC(C(C)(C)NC(Cc2ccc(C)s2)=O)=O)CCOCC1(C)C c1(C(N2CCC(N(C)C)C2(C)C)C(=O)NC(CC)C)cccc2cnccc12 C12(C(N3CCCCC(NC(C(C)N(C(C)=O)C)=O)C3)=O)CCC(CO)(CC1)CC2 c1(C(=O)NC2(CNC(c3cncc(OC)c3)=O)CC2)ccnc(O)c1Br C12(NC(CCC(C)OC)=O)CCOC(CNC(C3CCC(C)(O)CC3)=O)(C1)C2 C(=O)(C1=NN(C)C(=O)CC1)NCCN(C(C(CC)NC(N)=O)=O)CC(C)O Cc1ccc(CC(=O)NCC2CCCN(Cc3ncc(Br)s3)C2)cc1 CCC(C(=O)NCC(O)C(=O)NCc1csnn1)SC CC1CC(C(=O)NCC2CCCN2C(=O)COC2CCCC(C)C2)CC(C)(C)C1 C(C)(C)(CC(=O)NCc1cc(C(N2CCC(CO)CC2)=O)ccn1)SC C1(CNC(C2(CC=C)COC2)=O)N(C(=O)C(C)Oc2cccnc2)CCC1(C)C C(=O)(C(C)(C)C(C)(F)F)NCC1N(C(c2c(C)cc(CC)o2)=O)CC1 n1(CCC=C)c(N2CC(C)(C(N)=O)C2)nnc1-c1ccc(C(F)(F)F)cc1 Cc1nn(C)c(C(F)F)c1C(=O)NCC1CCCN(C(=O)Cn2nccn2)CC1 N1(C(c2ccc(CCC)s2)=O)CC(CO)C2(C1)CN(C(=O)C(C)NC(C)(C)C)C2 N1(C(c2c(CC)scc2)=O)CCCC(O)(CCNC(=O)C(CO)N(C)C)C1 C1(NC(c2scc3c2OCCO3)=O)CC2CCC(C1)N2C(C1(CO)CCCO1)=O c1(C(N(CC(CNC(CCc2cncc(C)c2)=O)C)C)=O)cccc2ccsc12 Cc1ccc(C(C(=O)NC2CC2)N(C2CCCC(N3CCCC3)C2)C)nn1 C1(C(=O)NCC(C)NC(=O)OC)CCN(C(c2cc(O)nc(O)n2)=O)C12CC2 N1(C(C2(C#N)CCCO2)=O)CC=C(CNC(c2cnn3c2CCC3)=O)CC1 C(=O)(C(F)(F)C(F)(F)OC(F)(F)F)N1CC(C)C(C)(NC(=O)CC2(C)CC2)C1 C1(CC)C(NC(c2ccoc2)=O)CCCN1C(=O)C(C)n1cccn1 N1(C(C=CCOCCOC)=O)CCC(CNC(c2cncc(CO)n2)=O)C(C)C1 C(=O)(C(F)C(C)CNC(=O)CN1CCOC1=O)NCCCOC C(=O)(CC(O)CC(C)(C)C)N1CCC(C(=O)NCC2CC(OCC)C2)C1(C)C C1(NC(C(CC2CC2)NC(C2C(CCC)CCC2)=O)=O)C=CC(C)(C)CC1 N1(C(c2cn(C(C)C)nn2)=O)CC=C(CC(=O)NCC2CCOC2C)CC1 c1(OC)cncc(CCC(=O)NC2CCC(NC(C3CCOC(=O)N3)=O)C2)c1 C1(CNC(C2(C)C(C)(C)C2(C)C)=O)CN(C(=O)Cn2ncnn2)C2(CCC2)C1 C1(NC(c2cc(C)no2)=O)CC2CN(C(=O)Nc3cc(Cl)cc(Cl)c3)CC2C1 C1(NC(=O)CN(C(N2CCCC2)=O)C2CC2)CCCN(C(C2CCC3(CC3)C2)=O)C1 c1(-c2cc(C)c(O)nc2)nc(C2Cc3ccccc32)nn1-c1ccc(Cl)cc1Cl C12CCCCC13CCC3NC2.C1(C(=O)O)CCCCC1c1nc(S)n[nH]1 C1C(C(C)C)C(=O)N1.C(C1=CCCN(C)C1)Oc1ccc(-n2cc(SC)nn2)cc1 N1(C(CC)=O)CC(OCC(=O)NCC(CO)SC)C1.C(CO)O C#CC1C(C(=O)NCC(CCCC)NC(c2nc(C)c(C)s2)=O)C1(C)C c1(CC(CNC(c2cccc(CC(C)(C)C)c2)=O)CO)cccc(Cl)c1Cl c12[nH]nc(c1Cl)C(=O)N1CC(C)(C1)NC2=O.c1(CC)nc(-c2nc[nH]n2)sc1C c1(C(=O)NCC2CCCC2NCCNC(CNC(C)=O)=O)cccc(C(N)=O)c1 C(=O)(C(C(C)C)NC(c1ccc(OC)cc1)=O)NCCN(C(C(COCC)C)=O)C C1(NC(C(C)OCC(C)C)=O)CCN(C(C2(c3ccccc3)CCCC2)=O)CC1 c1(C(=O)NC2(CNC(C(C=C)(C)O)=O)CCCCC2)cnc2[nH]nc(O)c2c1 N1(C(Cc2nc(=N)[nH][nH]2)=O)CCC2(CCCN(C(C34CCCC(CO3)C4)=O)C2)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N(CC(=O)NCCc1ccon1)CCOC Cc1ccc(C(=O)CCC(=O)NC2CCC2NC(=O)C=Cc2ccoc2)cc1C c1(CC)cc(C(N2CC3CC3(NC(c3cn(C)cc3C)=O)C2)=O)ncn1 C1(C(N(C2CCCN(C(c3c(C)oc(C)c3C)=O)C2)C)=O)CN(C)CCN(C)C1 C1(CS(=O)(=O)NCC(c2ccccc2)C)CCC2(CCOCC2)CO1 n1(C(C)(C)C)ccc(=NC(=O)C(=O)NCC2CSC2)[nH]1 Cc1nnsc1C(=O)NCC(C1CC1)N(C)C(c1cn(C(C)C)nn1)=O C(=O)(C(C)(C)CF)NCc1c(C(=O)NC(c2ccncc2)C)nco1 N1(C(C23C(CN(C(c4ccc(NC)cn4)=O)C2)CC3)=O)CCCC2(CCCO2)C1 N1(C(C2ON=C(C)C2)=O)CC=CC(NC(C2CCN(CC(C)C)C2)=O)C1 CS(=O)(=O)C1CCCC1C(=O)NCC1CN(C(c2cn[nH]c2)=O)CC1O c1(CCCC)ccc(C(F)F)cc1.c12cn(nn1)C(C)C(=O)N(CC)C2 CN=c1cc(C(=O)NCCSCC(=O)NCC(C)(C)C(F)F)cc[nH]1 c1(CN(C)CN2CC(NC(C3CC4CCC3C4)=O)CC2=O)cccc(F)c1 N1(C(C2CC(C)C2)=O)CC2CCC(NC(c3ncc[nH]3)=O)CC2C1 C12CCC3CN(CCC3C1)C(=O)Cn1cc2nn1.C(=O)(CCCC(C)(C)O)OC c1(C(=O)NCC2N(C(CN(CCC)C)=O)CCCC2C)sc2cccnc2c1Cl Cc1ccc(C(N2CC=CC2(C)C(=O)N(C)CC2COCCO2)=O)nc1 C1(C)(CC)CCCN(C(c2ccnc(NC(=O)CC3CC4(CCC4)C3)n2)=O)CC1 c1(C(N2CCC(NC(c3c(C)n(C)cc3)=O)C2)=O)cc2ccccc2c(=O)n1C c1(C(=O)NC(C)CNC(c2ccc(C(F)(F)F)cn2)=O)cc2cc(Cl)cnc2o1 C(=O)(CC(C)(C)O)N(C1CCN(C(C2CC23CC3)=O)C1)CC#C C(=O)(CC(C=C)CCC)NCCCC(=O)NC(CC=C)CNC(=O)CC(C)C(C)C CC(C)CC(C(=O)N1CC=CC1(C)C(N1CCC(C)C(C)(C)C1)=O)C(N)=O N1(C(C(CCC)=CCC)=O)CC2CCCC2(NC(=O)Cn2ncc(Cl)c2C)C1 C1(C(=O)NCC(C(C)C)NC(=O)CCC23CCC(CC2)C3)CC2(CCCC2)CO1 C(CCCCCCCO)NC(CC1N(C(Cc2c(C)cccc2)=O)CCCC1)=O C1(N(C)C(c2cc(C3CC3)no2)=O)CCC(NC(C2CCCCC2F)=O)CC1 C1(C(=O)NC2C(C)CN(C(=O)CC3CCCOCC3)CC2)CN2CCN1C(C)C2 Cc1ncc(CN(C(c2snnc2C)C(=O)NCC2CCCO2)C)[nH]1 c1(C(=O)NCC2CCN(C(C3CC(=C)C3)=O)C2(C)C)oc2c(Cl)cccc2c1C CNS(=O)(=O)N1CCC(C(=O)NCC(C)NC(=O)C(C)CSC(F)(F)F)CC1 c1(OC)ccc(Cl)c(C(N2CC(OC)CC(NC(=O)C3=CCSC3)C2)=O)n1 c1(C(N(CC(C)NC(c2cc(CCCCC)[nH]n2)=O)C)=O)ccc2sncc2c1 C(C(C)(CC(C)C)NC(=O)C(CC)C1CCCCC1)NC(CC(CC)OC)=O C1(S)CCCCC1C(=O)O.C(c1ccccc1)=CC(=O)N(C(C)CCO)CCC c1(C(=O)N(C)C)cccnc1NC1C(CNC(c2cnc(C(=O)OC)s2)=O)C1 C12(C(=O)NCC(C3CC=CC3)O)CCC(CC1NC(c1ccncc1F)=O)C2 O=C(C1SCCc2sccc21)NCCNC(c1cnc(Cc2ccccc2)[nH]1)=O c1(C(=O)NC2CCC2)ccc(OC(c2ccccc2)C2CC2)cc1 C1(CC(=O)NC(C#C)C2CC2)CC(NC(=O)C(C)C2(O)CCC2)C1 c1(C(N2CC(CC(C)NC(C=CC(C)(C)SC)=O)C2)=O)cncc(CO)c1 C(=O)(C(Cc1cc[nH]n1)NC(C1CCN(C)C1)=O)NCCN(CCC)CC C=CCCC(C(=O)NCc1ncccc1F)NC(=O)CC(C)SC c1(N2CCN(C(C3CC=C(C)CC3)=O)CC2)ccn2nccc2n1 C1(NC(CCCC)=O)CC2CCC(C1)N2C(c1c(C2CCC2)cnn1C)=O Cc1cncn1C=CC(=O)NCC1CCCC1NC(=O)C(n1nccc1C)C N1(C(c2c(OCC)cccc2)=O)C2CCCC1CN(C(C1CC3C=CC1C3)=O)C2 Cc1nnc(O)c(C(N2CCCC(NC(=O)CCc3cccs3)C(F)C2)=O)c1C N1(C(CSCC(C)=O)=O)CC2COCCC2(NC(c2cnc3ncccn23)=O)C1 C(=O)(CCCC(=O)OC)NC(c1cn(C)nn1)C(=O)NC1CCCC(CC)C1 N1(C(C)=O)CC2CC2(C(=O)NC2(C)CC(NC(=O)CSCc3ncc[nH]3)C2)C1 C1(C(=O)NCCCCNC(C(C2CCCCCC2)(C)C)=O)OCC2CCCCC12 C1(C(C)NC(C2(F)CCC2)=O)CCCN1C(C1CCC(=O)N1)=O c1(C(=O)NC2CCC(CNC(C(CCN(C)C)O)=O)CC2)cccc2cncn12 N1(C(C(CC)N(C)C)=O)CC2CCC2(NC(=O)C=Cc2nccn2CC)C1 N1(C(c2ccc(C)cn2)=O)CCCC2(NC(=O)CCc3ccncn3)CC2C1 Cc1nc(NC(=O)C(n2cc(-c3cnn(CC(=O)O)c3)nn2)C)oc1C c1(C(=O)OC)ccc(CC(=O)NC2CCC(NC(=O)Cc3cnoc3)CC2)cn1 N1(c2cc(NC(C)CC(N)=O)nc(COC)n2)CCN2C(=O)C(=O)NCC2C1 c1(C(=O)OC)csc(CCNC(=O)Cn2cc(C3CC3C3CCCO3)nn2)n1 c1(C(N2C(CNC(C=Cc3c(C)ccnc3)=O)C=CC2)=O)cncc2c1CCC2 C(=O)(C(F)(F)CO)N1C(C2(O)CN(C(C3(COC)C=CCC3)=O)C2)CCC1 N1(C(c2cc(C#N)cs2)C(=O)NCCCSC)CCCCCC1c1cccnc1 Cc1cccc(Cl)c1CC(=O)N(C)CCN(C)C(c1coc(C(C)C)n1)=O CC1C(NC(=O)CC2C=CCCC2)CCCN1C(c1nccc(N)c1Cl)=O C1(CCNC(C2(C(=O)OC)CC2)=O)CCN(Cc2cc(Cl)ccc2Cl)CC1(F)F c1(C(=O)NC(C(=O)NC2C(C3C(C)C3)C2)CC2CCC2)cccc([N+](=O)[O-])c1 C1(=CC(=O)NC2CC(C(=O)OC)CC2O)CCCCC1(C)C C1(NC(NOCCN(C(CC)=O)C)=O)CCN(C(=O)COCC(F)F)C1 c1(C(=O)NC(CN(C)C(c2cc3sccc3[nH]2)=O)(C)C)cc(Cl)ccc1C(F)F CCCC(C(=O)NCCOC1CC(NC(=O)Cn2cncn2)C1)NC(N)=O.C(C)O c1(C(=O)NC23C(CN(C(c4c(CC)ccc(C)c4)=O)C2)C3)cnc([N+](=O)[O-])n1C c1(C(N2C(CN(C(c3c(C)nns3)=O)C3CC3)CCC2)=O)ccc(F)c(C)c1N c1(C(=O)OC(C#C)CC2CCOCC2)nn(C)c2c(Br)cncc12 c1(C(=O)NCCC2(NC(C(C)c3cc[nH]n3)=O)CCC2)cnc2c(c1)ncn2C c1(C(=O)NCC2CC(NC(C(COC)O)=O)C2)oc2ccccc2c1OC C1(CNC(C(CC)c2ccccc2)=O)CCCC1N=c1nc[nH]s1 C1(C(N)=O)CN(C(C2CCCN2C(N)=O)=O)CCN1CCCC1CC1 c1(NC(C2(C)CCN(C(C(=C)F)=O)C2)=O)ccc(C)cc1C O=C(CC(=O)NC1CC1)NCCC(O)CNC(=O)CC1COCC1O c1(CC(N2C(CNC(C=Cc3scc(C)n3)=O)CCC2)=O)cccc2nonc12 C(c1cccc(F)c1)=C(C(=O)NC1C2CCN(C(C3COC(=O)N3)=O)C12)F c1(C(=O)NC2CCN(C(C(CCSC)N(C)C)=O)C2C(C)C)ncc(F)cc1C C(C(CC1CC1)C(=O)N1CCC(F)(CO)C1)N.c12ncccc1c(=O)c2=O N1(C(C(c2ccccc2)C)=O)CCCC(C(C)(C)C(=O)NCCS(C)(=O)=O)C1 c1(SCC(=O)NC2CCCCC2NC(c2c(Cl)n[nH]c2C2CC2)=O)ccc(F)cc1 C12(NC(=O)CNC(N3CCCC3)=O)CC(CNC(C3SCCS3)=O)(C1)C2 Cc1ccc(=N)[nH]c1C(=O)NC(C1(O)CN(C(C2CC3(CC(=O)N3)C2)=O)C1)C C1(C(=O)NCc2onc(C)n2)CCN(C(=O)CCCn2ccnc2)CC1 C1(CNC(c2ccc(C)s2)=O)CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CCC12CCC2 N1(C(CSCC)=O)CCCC2C(CCCN2C(c2cn(C(C)C)nc2Br)=O)C1 C1(C(=O)NC2(CC)CCC2)C(CNC(c2cncn2C(C)C)=O)C1(C)C n1(CC)cc(C(N2CC3C(COC(CC4CCN(C5CC5)CC4)=O)C3C2)=O)c(C)n1 C1(CC=C)(NC(c2ncn(C)n2)=O)CN(C(=O)CCN(C2CCCC2)C)C1 N1(CC(=O)NC(=O)NCC)CC2CCC(C(=O)OC)C2C1 Cc1cc(C(=O)NC2C(ON)COC2)nc(Cl)c1 c12ccc3sc(c(C)c3c1)C(N(C1CC1C)C)C2=O.c1(OC)ccccc1 C=CC(C)(CC)C(=O)N1CCCC(CN2CCN(C(c3csc(C)n3)=O)CC2)C1 C1(NC(c2cnc(CCC)s2)=O)CC2CCC(C1C)N2C(c1ccc(N)cc1)=O c1(CC)cnc(CC(=O)NCCC2(NC(c3cccnc3)=O)CCC2)[nH]1 N1(C(C(CC)(C)COC)=O)CC2CC(C)N(C(c3cccc4ccoc34)=O)C2C1 Cc1cnc(N2CC(NC(=O)CCSc3ccccc3)CC2C)nc1S(C)(=O)=O Cc1csc(CCC(=O)NC(C)CC2CN(C(c3cn(C)nn3)=O)C2)n1 C1(C(=O)NCC(CNC(=O)C=CC2CCC2)O)C2CC3C(C2=O)C13 c1(C2(C)CC2)ccc(C(=O)NCC2(F)CCN(C(C3(O)COC3)=O)C2)cc1 N1(C(CN(C(c2ccnc(C)c2C)=O)C)=O)CCn2ncc(C)c2C1 C1(N(C(C)C)Cc2ccccc2)CCCN(C(=O)CC2CCNC2=O)C1 N1(C(c2nc(C(C)C)oc2)=O)CC(NC(c2cc(CF)on2)=O)CCC1C N1(C(C2(C)CC(=C)C2)=O)CC2CN(C(=O)Cn3nnnc3C3CC3)CCC2(CO)C1 Cn1cc2ncc(C(=O)NCC3CC(NC(c4cnc(=N)[nH]c4)=O)C3)cc2n1 C(=O)(C1=CCN(C(c2ccnnc2C)=O)CC1)NC(c1ccc(C)nc1)C c12cncc(c1)NC(=O)C(=O)C2=O.C12CC(C1)O2.CCCCOCC(C)N c1(OC)ccc(C(N2CCCCC2CCCCNC(=O)Cc2cn[nH]c2)=O)c(F)n1 C1(C(=O)NCc2cccc(C(=O)Nc3cc(Br)nc(Br)c3)c2)CCCCC1(F)F N1(C(CC(C)=C(C)C)=O)CCC2(CCCN(C(C3CC4CC3CO4)=O)C2)C1 N(C1CCNC(=O)c2[nH]ccc21)C(C)C[Si](C)(C)C C#Cc1ccnc(C(=O)NC2CC3CC2N(C(c2cc(C)oc2CC)=O)C3)c1 C(C(C(C)(C)C)NC(c1cc(F)n[nH]1)=O)NC(C1CCC(C)O1)=O N1(C(CC(C)(C)N(C(C(CC)N(C)C)=O)C)=O)CC(O)(C2CC2)C1 N1(C(C2CCCC(=O)N2)=O)CCC2(CCCC2NC(=O)CC2CCNC2=O)CC1 C1(C(=O)NCCC(=C)CNC(C2(CC(F)F)CCC2)=O)CCCC1C1CC1 C1(C(N2CCC(C(N3C(CC)CC3)=O)(CO)C2)=O)CCCCC(=O)N1 C1(C#CC(=O)N2CCCC(NC(c3sccc3OC)=O)C2)(CC)COC1 O=S1(=O)NCc2cccc(NCCc3cc(O)ncn3)c21 C1(CNC(Cc2cccc(OCC)c2)=O)CCCN(C(c2ncoc2C)=O)CC1 c1(OC)ccc(C)cc1C(=O)NC(C1(O)CN(C(c2cc(C)nc(O)c2)=O)C1)C c1(C(N(CCC(C(C)(C)C)NC(C2C(C(=O)OC)C2)=O)C)=O)c(C)ccc(Cl)c1O Cc1cccc(NC(=O)C(C)SCCNC(=O)Cc2ccnn2C)c1 N#CC1CCN(C(c2ccccc2C2CCC2)=O)C1 C1(NC(C=CCOC)=O)CN(C(C2CCCCC(=O)N2)=O)Cc2nccn2C1 c1(C(c2nnnn2C2COC2)NC(C(C)N(C)C)C(N)=O)ccc(Br)c(F)c1F c1(C(NOCC(=O)NC2CCCCC2F)=O)occ2c1CCC2 C(=O)(CCS(C)=O)NC1(C(=O)NCC(CCOC)NC(C)=O)CC1 C(C(C)(C)CNC(=O)C(F)C1CCOC1)N(C(C=CCC)=O)C C(=O)(CCCCCCS(N)(=O)=O)NC1C(CNC(C#CC2(C)CC2)=O)CCC1 O=C1CCSc2ccc(C(=O)NCC3CCCN(CCCO)C3)cc2N1 C(=O)(CC(C)(C)CC(F)F)N(CCOCCCNC(C(CC=CC)CC)=O)C.C(C)=O N1(C(CNC(C)=O)=O)CCCCCC1C(=O)NC(c1ncccc1C)C C(=O)(C1=NOC(C(C)(C)C)C1)N(C)CC1CN(C(=O)C(C)(C)CC2CC2)CC1O C#CCC(C(=O)NCCN1CCC(O)C1)NC(=O)Cn1cnc(C#N)n1 N1(C(C(C)(C)CF)=O)CC2CCC1C(CNC(c1snc(Cl)c1Cl)=O)C2 c1(C2C(C)C2)sccc1C(N1CC(CNC(c2ccc(C3CC3)o2)=O)C1)=O C1(NC(C(C(C)O)(F)F)=O)CC2CC(NC(=O)Cc3cnc[nH]3)CC2C1 C1(C(=O)NC2C(CNC(c3ccn4c3CCCC4)=O)C2)CN2CCCN1CC2 N1(C(c2c(C)c(N)cnc2)=O)CCn2nc(CNC(=O)C(F)=CC3CC3)cc2C1 N1(C(c2cc(C)n(C)n2)=O)CC2(C1)C(NC(=O)C#CC1CCCC1)CCS2(=O)=O N1(C(CC(CC)(F)F)=O)CCC(C2CCOCC2)(CNC(c2cnc(S)[nH]2)=O)C1 N1(C(c2c(CC)nn[nH]2)=O)CCOCC(CNC(C2(C)CCCOC2)=O)C1 c1(NCCNCCNC(COC)=O)cc(N2CCC(c3ccno3)C2)ncn1 c1(OC)ccc2c(=NCC(C)SC)[nH]c(=NC(C)Cc3ccc(C)s3)[nH]c2c1 CCCCCCN1CCC(CC(=O)N(CC(C2CC(C)(C)C2)O)CC)C1 c1(C(=O)NC2C(CO)CCN(C(CSCC)=O)C2)cc(F)c(C)cc1Cl C(=O)(CCC(F)(F)C(F)(F)F)NCC(C)NC(c1c(C)ccnc1)=O c1(CNC(c2cc(C)nn2C)=O)cc(Cl)c2c(c1)OCCO2 C1(NCC(O)Cn2cc(C=O)cn2)C2Cc3ccc(Br)cc3C12 c1(C(=O)NC2C(OC)CN(C(=O)C(F)OC)C2)ccc(Cl)c(F)c1N C1(CNC(COCCCC)=O)(CO)CCN(C(=O)CC(C)(C)OC(C)=O)C1 CCS(=O)(=O)c1cccc(C(N2CCC2CN(C)CC2CC23CCOC3)=O)c1 C1(CNC(CCCNC(C)=O)=O)C(C)CCN1C(=O)CNC(=O)CCc1ccccc1 CC(C)(CN=c1nc(N2CCC(F)C2)c2c([nH]1)CSC2)N1CCCC1 C(=O)(CCCC(C)(C)C#N)NCC1(C(N(CC(C)SC)C)=O)CCC1 Cc1nc(N2CC3CCN(C(c4ccsc4)=O)C3C2)c2sccc2n1 c1(C(N2C3(CNC(C(C)C4CCC4)=O)CCC2CC3)=O)c[nH]c2cc(F)ccc12 c12ncc(cn1)[nH]c2=O.c1(C(=O)OC)coc(C(=O)NC2CCCC2CF)c1 CC1CCC=C1C(=O)N1CC(F)CC1CNC(=O)CCC1CCCC1 C1(F)(CNC(COCC(C)(C)C)=O)COCCN(C(C2CCCOC2)=O)C1 c1(OC(C)C)cccc(C(c2nnnn2C)NCC23CCCN(CC2)C3)c1F C(c1ccc(C)nc1)=CC(=O)NC(CCNC(c1c(OC)cc(C)s1)=O)(C)C N1(C(CC2ON=C(CC)C2)=O)CC(=O)CC1C(=O)NCC1CC2(CC2)CO1 C(C(=O)c1ncc2n1CCCN(CC)CC1CCCCN1C2=O)(C(C)(C)C)SC C(C(=O)NCc1ocnc1C(=O)NCC1CC(C)(O)C1)(C(C)(C)C)OC c1(C(=O)NCCCCCCN(C(CC(=O)NCC#C)=O)C)ccc(F)c(F)c1N c1(C(=O)NC2CCN(C(=O)CO)C23CC3)cc2sc(Br)cc2[nH]1 C(=O)(C1Cc2ccccc21)NC1CC(C)N(C(=O)CCOCCN(C)C)CC1 c1(CCC(=O)NC(C(C)(C)NC(CNC(=O)OC)=O)C)c(C)noc1Cl C(=O)(C(C)C(C)O)N1CC(CC)(NC(C2(CC(C)C)CCCC2)=O)C1 c1(C(=O)NC(C(=O)NCCC#C)C2CC2)cccc(C#C)c1 c1(C(=O)NCC(CC)NC(C2CC2(C(C)C)CC)=O)cc(OC)nc(F)c1 C(CC(C(=O)N=c1ccn(C2(C)CC2)[nH]1)NC(c1ccc(CF)cc1)=O)OC c1(CCC(N2C3CC(NC(c4nn(C)c(O)c4)=O)(C3)C2)=O)cccc(F)c1Cl c1(Sc2c(CC)cccc2)nc(C)cc(Oc2ccccc2F)n1 N1(C(=O)NC2CCCN(c3nn[nH]n3)C2)CCC(O)(C2CC2)CC1 C12(C(=O)NC3CCC(=O)NC3)CC(CO1)N(C(=O)Cc1ccccc1F)C2 Cc1ccc(C(N2CC(C)CCC2CNC(c2nc(C)c(C)s2)=O)=O)cc1C Cc1cc(C(N2CC(c3c(F)cccc3Cl)(O)C2)=O)c(N)c([N+](=O)[O-])c1 C(CC(C)(C)C(=O)Nc1ccc2c(c1)CC2)NC(C(CC)NC(C)=O)=O C(=O)(C(O)CCCc1ccccc1)NC(c1ccnn1C)COC C1(C(N2C(CN(C(c3c(C)noc3)=O)C)CCC2)=O)NC(=O)CC1C(F)(F)F c1(C(N2C(C(C)NC(=O)C(=Cc3c[nH]cn3)F)CCC2)=O)cc2n(c1)CCOC2 C1(C(N2C(CNC(c3ccc(C(F)(F)F)cn3)=O)CC2)=O)COCCOC1 Cc1c(NC(C2CN(C(c3cn(C)nc3C(F)F)=O)C2)=O)ccc(C#N)c1F c1(CCNC(C2CC(N(C)CC3C(C)C3)C2)=O)cccc(Cl)c1Cl N1(C(CCc2cc(C)[nH]n2)=O)C2CCC(C(=O)NCCCN(C)C(C)C)C1CC2 C1(NC=O)C2CCCCC12.CC1(C)C(C(N2C(C(=O)O)CCC2)=O)C1CO C(=O)(CCC(=O)C(C)(C)C)N1CCC(N(C)C(C2CC3(CCC3O)C2)=O)(CO)C1 c1(OC)cc(CC(=O)N(CCNC(=O)C=Cc2cocn2)C2CC2)ccc1C CC1(C)CCCC(O)(NC(=O)NC2(CC3(C)OCCO3)CC2)C1 c1(N2CC(CCC)OCC2)nc2ccsc2c(=NCC2CCCS2)[nH]1 C12(CNC(C(C)(C)OC)=O)CN(C(c3ccc(C(C)(C)C)cc3)=O)CC1CCO2 C12CC3(CC(C3)NC1=O)C2.N1(C(c2ccc(C)o2)=O)CCOC(CO)C1 Cc1c(Br)cc(C(=O)NC(C)Cn2cc(CC(C(=O)O)C3CC3)nn2)c(=O)n1C N1(C(C23N(C(CCCC)=O)CCC2C3)=O)CCN(C)CC1CCO CCC(CNC(C1CC(C)=NO1)=O)(CC)NC(=O)C(C)SC(F)(F)F C1(NC(CCN(CC)CC)=O)C2CCC1N(C(c1cc3sccc3[nH]1)=O)C2 C(=O)(C1=CC2CCC(C1)C2)N(CCCNC(C1C2(CC(OCC)C2)C1)=O)CCO c1(C(N(CCNC(C2C(=C)C2)=O)CCOC)=O)cnc(P(C)(C)=O)cn1 c1(OC)ccc(C(=O)NC(C)C(C(C)C)NC(c2ccc(C(C)C)nc2)=O)cn1 CC1=NN(C)C(=O)C1CC(=O)NC(C)Cn1cc(C2CCC(C)(C)CC2)nn1 c1(C2(O)COC2)cccc(NCc2ccc(C3CCCC3)cc2)c1 c1(CCC(=O)NCCCCC(C)NC(c2nonc2N)=O)ccc2[nH]ccc2c1 N1(C(C2(CC=C)CN(C(C3CCCCN3C)=O)C2)=O)CC(C)CCCC1C C1(C(N2C(C)C(C)N(C(c3c[nH]c(=O)cn3)=O)CC2)=O)CC2(C1)CC1(CCC1)C2 C(CC(O)C(=O)N1CCC(NC(=O)C=Cc2cn(C)nn2)C1C(C)C)SC N1(C(C2C(C)OCC2)=O)CCCCC(NCc2cnc(-c3ccccc3)o2)C1 C12(NC(=O)Cn3cccc3)CN(C(=O)Cc3cc(C(F)F)no3)CC1CS(=O)(=O)C2 n1(CCC(=O)NCC(CC=C)NC(c2ccns2)=O)nc(O)c2ccccc12 C(C(C)C(C)C)N(C(CN(C(CN(C1CC1)CC)=O)C1CC1)=O)C C1(c2ccc(OC)cc2)C(NC(=O)C(C)(C)CO)CC(=O)N1C1CC1.C1(C)C(=O)N1 C(=O)(CCC(C(C)C)NC(=O)CC1(CSC)CC1)NC(COC)(C)C(N)=O C(c1cocn1)=CC(=O)NCCCCC1CN(C(C2(C3CCCO3)CC2)=O)C1 CCCCCC(O)CC(=O)NC(C1CC(NC(C2(CC(C)C)CC2)=O)C1)C N1(C(C(Br)=C(C)C)=O)CC(C)CN(C(C2CCN(C)C(=O)C2)=O)CC1C c1(CC(=O)NCC(C(C)(C)C)NC(CCCOCCOC)=O)ccc(Cl)c(C)c1 c1(C(N2C(CNC(C3CC3C(F)F)=O)CCC2)=O)cc2n(n1)CC(F)C2 CCCCCCC(=O)NC1CN(C(=O)CC23CCCN2CCC3)C(C)(C)C1 C1(NC(C2CC(C)C2)=O)CCCCN(Cc2ccc(Cl)nc2)C1 C1(NC(c2[nH]cc(CNC(CCC=CCC=C)=O)c2)=O)CCOC1C=C C1(CNC(CCOCC#C)=O)CN(C(c2cc3c(ccn3C)[nH]2)=O)CCC1(F)F C=C(C)C1OCCCC1C(=O)NCC1CC(NC(c2ccc(C)c(C)c2Cl)=O)C1 N1(C(C2N(C(N)=O)CCC2)=O)CC2CCC1C(NC(=O)CCc1ccoc1)C2 C1(C(=O)NC2CCCCN(C(C(N3CCNC3=O)C)=O)C2)C2CCC(C2)C1(C)C N1(C(c2ccc(C)o2)=O)CCC(C)C1CNC(C1(N2CCOCC2)CCC1)=O C=CCCCCC(=O)NC1CC(NC(=O)C=Cc2ccccc2)C12CCC2 N1(C(CCCNC(CC(C2CC2)OC)=O)=O)CC(C(N)=O)CC(C)C1.C(=O)N C1(NC(C2(C(=O)NCC)CCCC2)=O)CC(C)N(C(=O)CCC(C)OC)C1 C1(NC(=O)CSCC2CCCO2)CC2CCC(C1)N2C(c1coc(Br)c1)=O CC1COC(C(=O)N(C2(CC(=O)N(C)Cc3nccn3C)CC2)C)C1 C(=O)(CCC(C)N(C)C)NC1(CC)CN(C(=O)C=Cc2scnc2C)C1 N1(C(C(CC)CC)=O)CCCC(CCNC(C2CC3C=CC2CC3)=O)CC1 C1(C(N(CCCNC(c2cncc(OC)c2)=O)C)=O)CCc2nc(=N)[nH]cc2C1 c1(C(=O)OCC)cccnc1C(=O)NC1CC(CCNC(=O)Cc2conc2C)C1 N1(C(COCC(C)C)=O)CCCC(C)C1CNC(=O)CCCc1ccc(F)cc1 C1(C(=O)NCCn2c(CC)ncc2)CCN(C(=O)COCC(C)C)C12CC2 Cc1ccc(C#N)cc1C(N1CC(C(N2CC3CC2CC3CF)=O)C(CO)C1)=O c1(C(=O)NCC(C2(NC3CCC3(C)C)CCCC2)OC)cccc(C)c1C#N C1(C(N2CCC=C(F)C2)C(=O)NC)CC(C)(C)OC(C)(C)C1 c1(C(N2CCC(CCF)C2)=O)cc2c(Br)c(Cl)ccc2s1 C1(NC(CCCC(C)NC(c2cc(C(N)=O)[nH]n2)=O)=O)CC12CCCCCC2 C1(c2nnnn2Cc2nnn(C)n2)(NCc2c(C)nns2)CCN(C)CC1C C(=O)(CC(C)(C)CC(C)=O)NC1(C(=O)NC2C(C)(C(=O)OC)C2)CCCCC1C c1(CCCC(=O)Nc2c(C(=O)OC)cnn2C2CCCCO2)cc(Br)ccc1Br N1(c2nccc(OC)n2)CCC(NC(=O)CC2CCCOC2)C(C)(C)C1 C(=O)(CC(CCCC)NC(c1ncccc1N)=O)NC(CCC)C N1(C(c2ccc(C)c(O)n2)=O)CCCN(C(C2CCCOC2)=O)CCC1 CCCCCCC(C)C(=O)NC1CCCC1C(=O)NCc1cccc(CO)n1 CCC(C)CCCC(=O)NCC1(O)CCCN(C(=O)CCCNS(C)(=O)=O)CC1 CCCCC(CC)CCC(=O)NCC1CN(C(=O)C(n2cc(Cl)cn2)C)CC1O c1(C(N2CCC(COC)(NC(c3cc(C(N)=O)sn3)=O)C2)=O)ccn2c1CCCC2 N1(C(c2c(CC)c[nH]c2)=O)CCCC1(C)C(N1CC2C=CC2C1)=O C1(CNC(C(CC=C)OC)=O)CCCCCN1C(=O)C(COC(C)C)OC n1(CC)nc(-c2cn(C(C)CC(=O)N3CCOCC3)nn2)cc1C CCCC(=O)NNC(=O)NC1CCN(C(C)=O)CC1 c1(NC(C2(C)CC(NC(C(C=CC)O)=O)C2)=O)ccnc(SC)c1 N1(CC)CCCC(COC(=O)CCC2CCCN2C(=O)COc2cccnc2)C1 N1(C(C2CC3CCC2C3)C(=O)NC)CCCc2n[nH]cc2C1 C1(C(=O)Nc2cc(C(F)(F)F)ccn2)CN(c2ncc(I)cn2)CC(F)(F)C1 N1(C(CC(=O)OCC)=O)CCCC(CCNC(C2(C(F)F)CCCC2)=O)C1 Cc1n[nH]cc1C(C(=O)C(C)C)N(CCN(C)C)CC1CCCO1.N c1(N2CCC(C(C)NC(=O)CC(C)(C)N(C)C)CC2)ncnc2ccsc12 C1(C(N(C2CCN(C(C3(CCC)CCC3)=O)C2)CC)=O)CCC2(CCC2)O1 C1(C)(NC(C2C(C)(C)NC(=O)C2)=O)CCCN(C(=O)CCC(=O)NCC2CC2)C1 N1(C(c2c(C)occ2)=O)CCC(CCCCCNC(=O)COC2CCOC2)CC1 CCCC(C(=O)NCC(C(=O)N(CCN=[N+]=[N-])C)OC)C(C)C C=C(C)CC(C(=O)NC1(CC(=O)NC(c2ccns2)C)CCCC1)OC C(=O)(CCCCCC(C)C)NC1C(OC)CN(C(c2sccc2C#N)=O)C1 CCCCC(CC(=O)N1CCOC(CCO)C1)NC(=O)CC1COCCCO1 N1(C(CCC#C)=O)CCC(CCC)(COC)C1.C1(=O)CCC2CC(C2)N1 N1(C(C(C)O)=O)CC(NC(c2ccc(N3CCOC3=O)cc2)=O)CC12CCCC2 C1(C(=O)O)CN(C(c2ccccc2)=O)CC12CN(CC1CCCCO1)C2 c1(OC)ccc(I)cc1CN1CCN(C(C2(S(N)(=O)=O)CC2)=O)C(C)C1 C1(C(=O)NCC2CCOC2)CCN(C(C2C3CC4C(C3=O)C24)=O)C12CCC2 c1(N(C)C)ccc2[nH]c(=O)cnc2c1.C12CCN(C(C(C)C)C1)C(=O)NC2 C1(CNC(C2C(C)C2(F)F)=O)CC2(CC2)CN1c1nnc(C(F)F)s1 c1(C(N2C(CCNC(C(CC(=C)C)C)=O)COCC2)=O)cc2cccc(O)c2[nH]1 C#CCCCC(C)C(=O)NC1(CCC(N2CC(OC)CC2CO)=O)CCCC1 N1(C(C(C)NC(CC)(C)C)=O)CC(CCO)(NC(=O)C(C)NCCCN(C)C)C1 c1(C(=O)OC)cc(Nc2ccc(-n3ccnc3C)nc2)c([N+](=O)[O-])c(Br)c1 CC1CC(C(=O)NC2(CNC(=O)CCc3ccc(Cl)cc3)CCCCC2)CCO1 C(=O)(C(C)(C)C(O)CC)N.c1(CC(=O)NCC(CC)OCCS)nnn(C(C)(C)C)n1 CCCCCC(C)c1noc(C(F)(F)C2COC2)n1 Cc1ccc(C(N2CC3C(C2)N3C(=O)C(C)NC=O)=O)c(I)c1 C(=O)(C1=CCC2CCC1N2C(C1OC2CCC1C2)=O)NC1(C=C)CCCC1 c1(C(c2nnnn2CC)NCc2c(C(=O)OCC)nco2)c(Cl)cccc1Cl CC1(C)OC2(CNC(=O)C=Cc3cccc(Cl)c3)CC1(NC(=O)CS(N)(=O)=O)C2 C(=O)(C(C)C1=CCCC1)NC(C1CCN(C(c2c(O)ccc(OC)c2)=O)CC1)C CCCC(C(=O)N(CC(O)CNC(c1cc(CN(C)C)on1)=O)C)c1ccccc1 C(C(CO)N=c1[nH]c2cccc(F)c2o1)NC(C1CCCC2(CC2)C1)=O C(C(C(C)(C)C)NC(c1nc(O)c(C)s1)=O)NC(Cn1ncc(C(=O)OC)c1)=O C(=O)(CC1OCc2cc(Cl)ccc21)N1CCC(O)(CC(N2CC(F)C2)=O)CC1 N1(Cc2c(C)cc(C)[nH]2)CC2CC1CN2C(c1ccc(Sc2cccc(Cl)c2)o1)=O c1(C(=O)NCC2C(NC(C3CCN(C(C)=O)C3)=O)CCC2)ccc(F)c(Cl)c1N C12(NC(C(C(C)C)SCC)=O)CC(CO)(C1)OC21CN(C(=O)COCC(C)C)C1 c1(CN2CC(NC(c3ccccc3OC(F)(F)F)=O)C2)ccc(F)cc1Cl c1(C(=O)NC(C)CCNC(=O)CNC(=O)CC(F)(F)F)cnc2c(c1)COCC2 Cc1cccc(C(C)(C)C(N2CC(NC(=O)Cc3nc(C)c(C)[nH]3)CC2C)=O)c1 c1(CC(=O)NC23CC(NC(C4(OCC)CCCC4)=O)(C2)C3)ccc(Cl)c(F)c1 N1(C(c2c(C)nco2)=O)CCN(C(c2cc3c(s2)CCC3)=O)C2CCCCC12 C=C(F)C1(CC(N2CC(F)(CNC(=O)C(C)Oc3ccc(F)nc3)C2)=O)CCC1 c1(CCC)ccccc1C(=O)NC(C)CCNC(=O)CCC1CCOCC1 C1(C2CCN(C(c3ccc(F)nc3F)=O)C2)(NC(=O)C(=Cc2c[nH]cn2)F)CC1 Cc1ccccc1Cn1ccnc1C(c1nnnn1C1CC1)NCCCOC C1(NC(=O)CCc2cscn2)CCOC(C(N2CCSCC2CO)=O)C1 c1(C(N2CCN(c3cc(F)ccc3O)CC2)=O)ccc2ccccc2n1 C1(C(C)C#N)CCN(C(c2cn(CCC3(N(C)C)COC(C)C3)nn2)=O)CC1 C(=O)(C(C)C(O)C(C)C)N1CCN(C(c2c(C)c(SC3CC3)ccc2)=O)CC1 c1(OC)ccc(C(N2CCN(CC(N)=O)C(=O)C2)C(=O)NC(C)C)c(OC)c1 N1(C(c2csc3c2CCCC3)=O)CC(Nc2cc(F)ncn2)CC12CCCC2 Cc1cc(C(=O)N(C)CC2CCN(C(=O)COC3CC3)CC2C)cc(C)c1C c1(C(=O)NC2(C)CCN(c3nnc(CCOC)s3)C2)n[nH]c2c1COC2 c1(OC)cnc(Cl)[nH]c1=NCCC1CCN(C(c2cn(C(C)(C)C)nn2)=O)C1 N1(CC(C)(C)NC(C2C(=C)C2C(=O)N)=O)CCC(C(N)=O)CC1.c1(C)csc(=N)[nH]1 C(=O)(C(=O)C(C)(C)C)N1C(CN(C)C(c2cccnc2F)=O)CCC1 c1(C(=O)NC2CN(C(C(C(C)O)NC(N)=O)=O)C2)cc2cccc(F)c2o1 C(CCCCCNC(=O)COCCC1CCCCC1)NC(CC1(C)CCCC1)=O C1(C(=O)NC(C)CCCOC(F)(F)F)C2CN(C(c3cccnc3N(C)C)=O)CC12 CC1(C)CN(c2ncnc(=N)[nH]2)CC(CNC(c2noc3c2CCCC3)=O)O1 C(=O)(C1=CCN(C(C2(COCC)CCCCC2)=O)CC1)C(=O)Cc1cc[nH]c1 C1(NC(C(CN(C)C)NC(C(C=C)C)=O)=O)CCc2nncn2C1 C1(C(C(=O)N(C(CC)CNC(=O)CCn2ccnn2)C)C)CCC(=O)N1 c1(CCC)n[nH]c(=NCC2CCN(C(=O)CC(C)(C)N(C)C)C2)s1 c1(C(=O)OC)ccc(NC(c2c[nH]nc2C2CCN(C(=O)C(N)=O)C2)=O)s1 S(=O)(=O)(C(F)(F)F)NCCC(=O)N(CC(O)CNC(C1CC=CC1)=O)C C1(C(=O)NCc2onc(C)n2)CN(C(C2CC(N(C)C)C2)=O)CCN1C c1(CC)nnc2n1CCCC2C(=O)N1CCCC(N(C)C(C2OCCO2)=O)CC1 c1(CC(N2C(CCC(=O)NC(C)(C)C(N)=O)CCC2)=O)cccc(F)c1F N1(C(C=CC=CCC)=O)CC23CCCC2(C1)CN(C(c1cc(O)cc(O)n1)=O)C3 N1(C(CCN(CCCCC)CC)=O)CC(CNC(=O)CSCCC)CC1(C)C C1(N(C(C(C)SC(F)(F)F)=O)C)CCCCC1N(C(=O)C=Cc1cocn1)C CC1CN(C(C2CCC(n3cccc3)CC2)=O)CC1NC(C1(CO)CCCO1)=O C#CCC(CC(=O)N(CCC#C)C)NC(C1CCCC1O)=O c1(C(N2C(CCNC(C3(C)CC(=C)C3)=O)CCCC2)=O)cc(C)cc(F)c1 c1(C(c2nnnn2CCN2CCOCC2)NC(c2nncn2C)C)nn(C)cc1Br C1(C(C#C)C)CCN(C(c2ccncc2)C(=O)NC(C)CC)C1 C1(COC)(NC(=O)CCc2ccc(=N)[nH]c2)CCN(C(c2c[nH]c(=N)s2)=O)CC1 N1(C(CC=CC)=O)CC(NC(=O)Cc2c(Cl)cnn2C)C(O)C1 C(CC)(CC(=O)Nc1csc(C)c1)N(C(CCOCC#C)=O)C C1(NC(C2C(C)CC(=O)N2)=O)CCC2CN(C(=O)CCn3cnc(=N)[nH]3)CC2C1 n1(CC(=O)NC2C(CC)CN(C(C3CC(Cl)(Cl)C3)=O)CC2)nnc2c1CCCC2 C(=O)(CCCS(N)(=O)=O)N1CCN(C(=O)NC2C(C)(CC)C2)CC1 C12(NC(Cn3ncc(C)c3)=O)CCCC1CN(C(c1cccc3[nH]ccc13)=O)C2 N1(C(c2ccn(C)c2)=O)CC2(CCCC2)C1C(=O)NC1CCCCCC1CO N1(C(CCC#C)=O)CCC2(CC1)CC(C)N(C(c1ccc(OC)c(SC)c1)=O)C2 c1(-n2cc(C(=O)NCC3OCC(CNC(CC=C)=O)C3)nn2)ccc(Cl)cc1Cl N1(C(C2CN(CC)C(=O)C2)=O)C2CCC1CN(C(=O)C(F)(F)C(C)O)CC2 C=CC1(NC(=O)CC2CC(NC(C3CC(C)(C(=O)OC)C3)=O)C2)CCCC1 c1(OC)cc(F)ccc1C(N1CC2CC2(C(=O)Nc2ccc(N(C)C)cc2)C1)=O Cc1c(C(N2CCC23CCNC3)=O)cc(Br)cc1Br C(=O)(C1=CCC2(COC2)OC1)N(C)CC1CCCN(C(c2csc(=N)[nH]2)=O)C1 c1(CC)[nH]ccc1C(=O)NCC(C)CNC(=O)CC(C)NC(c1ccco1)=O c1(C(=O)NCC2C(NC(=O)C=Cc3cccs3)CC2)cnc(CC2CC2)nc1O c1(CC2CCN(C(c3nc(C)c(C)s3)=O)C2)ccc([N+](=O)[O-])c(C)c1 C1(CNC(C(COC)(C)C)=O)COCCN1C(=O)CC1COC2CC1C2 C(CC(C)CCNC(C1CC2C=CC1C2)=O)NC(c1cc(CC)no1)=O CC(C)(C)C(CCO)CN=c1[nH]c(N2CCOC(C#N)C2)nc2c1COC2 c1(-c2cn(C34CC(NC)(C3)C4)nn2)cc(C)c(Cl)c(C)c1.c1(CC(=O)N)ccccc1I Cc1cccc(CC(=O)NC(C2CN(C(=O)C(O)C3CC3)C2)C)c1C Cc1cc(C(=O)N(C)CC2CCN(C(=O)C(C3CCOCC3)O)C2)nn1C(C)C c1(C(N2CC3C(CCNC(C(CC)SC)=O)(CC3)C2)=O)c(F)ccc2c1OCC2 C=CC1CN(C(=O)CC2CCN(C(=O)CSCC)CC2)CC1O C1(NC(=O)CCc2ccsc2)CCCN(C(=O)CCCn2ccnc2)C1 c1(NC(C2CC2(F)F)=O)cc(F)cc(F)c1.N12CCCC1C1(CC1)N(C)CC2=O CC1CN(C(c2ccnnc2S)=O)CCC1NC(=O)CCSC(F)(F)F N1(C(CC(CC)SC)=O)CC(C(=O)NCc2ccnc(C#N)c2)CC(C)(C)C1 CCC(C)CCn1cc(CCNC(C2CCC3CC23)=O)nn1 CC(c1ccc(F)cc1F)=CC(N1CCC(O)(C(=O)OC(C)(C)C)C1)=O C1(CNC(c2c(C)cccn2)=O)CCC2(CN(Cc3cc(F)c(Br)cc3F)C2)O1 C12(NC(c3cccc(C4CCC45CCC5)c3)=O)CC3CC(C1)CC(Cl)(C3)C2 N1(C(c2ncc(C)cn2)=O)CCCCC1C1CCCN1C(C1CC(F)(CO)C1)=O N1(C(C(C)N(C(C)=O)C)=O)CCC2CN(C(c3ncc(Cl)cn3)=O)CCC12 C(=O)(C(C)(C)CCCNC(C1COCOC1)=O)N(c1c(OC)ccnc1)C c1(C(N2CC(C(C(=O)NC(C)CC(C)C)OC)C2)=O)c[nH]ccc1=O c1(CCN2C(C)CN(S(=O)(=O)CCBr)CC2)cn(C)c2cc(F)ccc12 CCC(Cc1ccccc1)C(=O)NCC(O)CNC(c1cc(C(=O)OC)c[nH]1)=O C1(C(=O)NC2CC(F)C2)CCS(=O)CC1.C12CCC1C(=O)NC2 c1(C(=O)NC(C2CCCN(C(=O)CCNS(C)(=O)=O)C2)C)cc2ccccc2o1 CC(=O)C(CC(C)C)OC(C1(C2CC2)CN(C(C2CCC(O)CC2)=O)C1)=O C1(C(=O)N(CC(O)CN(c2nnc(Cc3cc[nH]n3)s2)C)C)(COC)CCCC1 Cc1nonc1CNC(C1(CCNC(=O)C(O)CC2CCCC2)CCCC1)=O C1(CNC(COCCCC)=O)CCN(Cc2cnc(CC(C)C)s2)C1 C(=O)(C(C)(O)CCc1ccccc1)NC(CNC(c1c(C)ncnc1)=O)CC(C)C Cc1ccc(S(=O)(=O)N2CC3CN(C(c4cc(C)c(I)c(C)c4)=O)CC3C2)cc1Cl C1(NC(=O)CCCC2CC2)CN(C(C2(C3CCC3)CC2(F)F)=O)CC2(CC2)C1 C1(OC)CCCN(C(c2sccc2CNC(=O)C(F)OC(F)(F)F)=O)C1 c1(C(=O)NCC2N(C(=O)CCCC3CCCCC3)CCC2)cc2ccncc2[nH]1 CCCC(C)(CC)C(=O)NCC1(C(=O)OC(=O)CC2OCCC2C)CCOCC1 C(C(=O)N(C(C)CC)CCO)OC(C)C Nc1c(C(=O)NCC2CCCN(C(=O)CCC(F)F)C2)cnn1-c1ccccc1 N1(Cc2c(-c3cc(OC)c(Cl)cc3)cnn2C)CCC2CCCN(C)C2C1 C1(CC)C(NC(=O)C2=NNC(=O)C2)CCCN1C(=O)CC1CCCCC1O c1(C(=O)NC2(CCOC)CCN(C(=O)C(C)C3CC3)C2)ccc2[nH]c(=N)sc2c1 Cn1nc(O)cc1C(N1C(CC(=O)NCc2ccc(I)cc2)CCC1)=O N1(C(CC(C=C)(C)C)=O)CCC(C2CCN(C(c3ccc(CO)nc3)=O)C2)C1 c1(C(C)=O)sc2ccccc2c1C(=O)NC(C(=O)O)c1cnsc1 c1(CC)nc(C)[nH]c1C(=O)NCc1cn(CC(C)NC(C2CC3CC3C2)=O)nn1 N1(C(CC2CC(C)(C)C2)=O)CC2C(CC(=O)NOCC34CCC(CC3)C4)C2C1 N1(C(C=C(C)C)=O)CCN(C(=O)Cc2csc(=N)[nH]2)C(c2cc(F)ccc2F)C1 C1(O)(CCNC(=O)CC2OCCO2)CCN(C(=O)CCSc2ccc(Cl)cc2)C1 C#Cc1cccc(C(=O)NC(C)CCCNC(=O)C(C)CC(C)C)c1Cl c1(CC(N2CC(N(C(C(C)OC)=O)C)C(O)CC2)=O)ccccc1S(C)(=O)=O C1(NC(C(C)=CC2CC2)=O)CCCC12CN(C(c1ccc(F)c(C)c1)=O)C2 C(=O)(CC1=CCN(C(c2cnnn2C)=O)CC1)Nc1cccc(C)c1C c1(N(CCC(C)N(C(=O)CC)C)C(CC2(C(=C)F)CCC2)=O)cnn(C)c1C#N c1(C(C)C(=O)NCC(C)(C)NC(c2ccsc2Cl)=O)ccc(F)cc1F c1(C(N2CCC(C(C)(C)NC(=O)C(N)=O)C2)=O)ccc(C2=CCOCC2)cc1 C(C)(CC(=O)NCC1CCN1C(=O)CCNC(c1cccs1)=O)=C(C)C c1(OC)ccc2c(=O)c(SC)cn(CC(N3CCC(c4ccnn4C)C3)=O)c2c1 C1(C(=O)NCC2CCC(CNC(C(CC)(C)C#N)=O)CC2)CN(CP(C)(C)=O)C1 CC1(C)CN(C(c2cnco2)=O)C(CNC(c2cnc(O)s2)=O)CO1 CCCCC(CNC(C1CCCN1C1CCCCC1)=O)NC(c1ccccc1)=O c1(OCC(=O)NC(CC2CN(C(C3(CC)CC3)=O)C2)C)cc(C)c(Cl)c(C)c1 C1(NC(C(C)OCC2CCCCO2)=O)CCCN(C(C2CC=CCC2)=O)C1 c1(CNC2CC(NC(c3cccnc3O)=O)C2)ccc(Br)c(F)c1F C1(C(=O)NC2(CC#C)CCCCC2)CCCCCCN1C(C1CCCOC1)=O C1(C(N(CC(C)OC)C)=O)CCN(C(=O)OC(C)(C)C)CC1C C(=O)(C(CC1(C#N)CC1)N1CCCC1)NC(C1C(C(C)(C)C)CC1)=O C1(NC(C2(O)CC2)=O)CCC2CN(c3cc(O)nc(O)n3)CC2C1 c1(CC)cccc(C)c1C(C(=O)NC1CCCC1)N(CCC(=O)OC(C)C)C C(C(C)(C)C)SC.C(C)(C)(C)ON.C1(=O)NCCO1 CC(C)(F)C(C)(F)C(=O)NC1CCC(CNC(c2ocnc2C(F)(F)F)=O)CC1 c1(NC(C)CC#N)[nH]c(=NC(C)c2cccnc2C(F)(F)F)nc2c1cnn2C C(CN=C(NCc1cnc(C2CC2)[nH]1)N1CCC(C2CCOCC2)C1)OCC=C c1(C(=O)NC(C)CCCNC(=O)COCC2CCCO2)cccc2c1OCC2 N1(C(C=CC(=O)N(C)C)=O)C2CCC1C(CNC(C1CCCOCC1)=O)C2 c1(SCC2NCCN(C(c3ncc(C(=O)OC)cn3)=O)C2)cc(F)ccc1C C1(C(=O)NCC2(OC)CC(C)C2)(NC(c2cc(C)ns2)=O)CCN(C)C1 C1(NC(C(CSC)O)=O)CCC2CN(C(=O)CN=S(C)(C)=O)CC12 c1(C(N(C)CCNC(c2cc(O)n(C)n2)=O)=O)[nH]cc2c1CCS2(=O)=O CCC(C)(C)CCCNC(=O)CC(C1CC1)NC(c1cc(O)cc(F)c1)=O C1(NC(C(CSC)c2ccccc2)=O)CCN(C(=O)CCC(C)(C)C)C(C)C1 Cc1nn(C)cc1CCC(=O)NCCC1CN(C(c2csc(C)c2C)=O)CC1O C1(COC)(NC(=O)CN2CCC2C)CCN(C(c2ccc(N)cc2F)=O)CC1 Cc1c[nH]cc(C(=O)NC(C2CCCCC2)C(C)NC(c2nnn(C)n2)=O)c1=O c1(NC(c2ccc(CNC(c3ccncc3O)=O)cc2)C)cc(F)ncc1Br S(=O)(=O)(c1ccc(F)c(F)c1F)N(C(=O)Cn1ncc2ncccc12)CC(F)F C1(C(N(C(CC)CC)CC)=O)CCCN(C(=O)CCC2CCOC2)C1 Cc1cccc(C(O)C(=O)NCCC2CCN(C(C3CC3C)=O)CC2)c1F N1(C(=O)NC(=O)N(C2CC2)Cc2cccnc2)CCOC(C2CC2)C1 C(C1C(C(N2C3CCC2C(CNC(c2coc(Cl)n2)=O)C3)=O)C1(C)C)=C(C)C C1(NC(C(CCC)NC(c2cnccc2OC)=O)=O)CC(=O)N(C)C1=O C1(C(=O)NCC2CCCC(C(=O)NCC=C(CCC)C)C2)CC12CCCCC2 Cc1cc(C)c(NC(=O)CC2CC(C3CCC3)C2)cc1Cl N1(C(COCCOCC#C)=O)CCCC1CNC(c1coc(C)c1)=O CC1(C)OC(=O)CC1C(N1CCOC(CC(=O)NCC2C3CCCC23)C1)=O CC1C(NC(c2ccoc2Br)=O)C(C)CCN1C(c1cc(C2CC2)nn1C)=O C1(N(C(c2ccc(OCC)cc2)=O)C)CN(C(=O)COCCF)CCC1O N1(C(C(C=C)C)=O)CCN(C(c2cncc(C(F)(F)F)n2)=O)CC12CCC2 c1(C(=O)NC2C(NC(C(COC)C)=O)CCC2)cccc2nc(OCC3CC3)oc12 c1(COC(=O)CC2CCC3CC23)cccc2c1OCCC2 N1(C(c2nncc(C)c2)=O)CCCCC(NC(=O)CCc2ccsc2)C1 C1(=O)C2=NN(C(=O)CC2)C1C#C.C1(C(=O)OC)CCC(CCCC)CC1 N1(C(c2cc(C)cc(F)c2)=O)CCC2(CCCC2NC(=O)C=C2CCCC2)CC1 C12(NC(C(C)(C)O)=O)CCOCC1CN(C(=O)CS(=O)(=O)C(C)(C)C)C2 c1(CNC(CCSCCCC)=O)ccc(C(=O)NCC2CC3C=CC2C3)cc1 c1(N(CCC)C)ccc(C(=O)NCC(C)NC(c2c[nH]nc2C2CCC2)=O)cc1 c1(CC)cc(C)nc(C)n1.C1(NCO)CC2(Cc3ccccc3)CN1C2 C1(O)(CCNC(c2cncc(COC)c2)=O)CCCN(C(=O)CCS(C)=O)C1 c1(C(=O)OC)cc2ccccc2[nH]c1=NC(CNC(c1cnsc1C)=O)CO CCC(CC(=O)NC1CCC1NC(=O)C(C)NC=O)C(C)C CC(c1ccc(F)cc1F)=CC(=O)NC1CC1NC(=O)CC1CCC(C)(C)C1 C(=O)(C1=NN(C)C(=O)CC1)NC(CN(C(C1Cc2ccccc2C1)=O)CC)C CC1(C)C(C)(C(=O)NC2CCC(NC(=O)CCOc3cccnc3)CC2)C1(C)C c1(COC(C(C)CNC(=O)C=CC2C(C)C2(Cl)Cl)=O)ccc(Cl)cc1 c1(OC)cncc(C(=O)NCC2CC2CC(=O)NCCN2CCNC2=O)n1 C1(CN2CCC(NC(COC)=O)C2)OCCC1C(=O)OC(=O)Cc1ccccc1 C(=O)(C1=CCN(C(=O)C(CC)CC(C)C)CC1)Nc1cn(CCOC)nc1 C=C1CCC(C(N2C(CNC(=O)CC(c3ccc(C)cc3)C)CC3CC23)=O)CC1 C(=O)(C1=CC(C)(CC)C1)NC(CCCC)CNC(c1cccnc1C)=O C=Cc1ccc(C(=O)N(CCC(C)NC(c2ccc(COC)[nH]2)=O)C)cc1 CC(CC(=O)N1CC(CNC(c2cnn(C(F)F)c2)=O)C(F)(F)C1)C(F)(F)F c1(CNCC23C(CN(c4c(C)cncn4)C2)C3)c(Cl)cccc1I C1(CC)CN(C(c2ccoc2C2CC2)=O)CCN1C(=O)C(C)SC(C)C CC1C(NC(=O)C(N2C(C)CCC2C)C)CC2CCC1N2C(c1ccccc1)=O C(=O)(C1=C2CCCN=C2NN1)NCC(CCCC)NC(C(C)=CC)=O C1(C(=O)NC(COC)C(=O)NC2CC2(C)C)C2(CC2)C12CC2 N1(C(CC2(C#N)CC2)=O)C2CCC(C(N3CCn4cnnc4C3)=O)C1CC2 c1(OC)cc(C(=O)NC2CCC2NC(C2CC(C)=NO2)=O)cc(F)n1 c1(C(=O)NC2CN(C(C3(COC)CCOC3)=O)C2)cc(Cl)cc(C)c1N C1(C)(C(N2C(CNC(c3cnc(C(C)C)[nH]3)=O)CC2)=O)CCC(F)(F)CC1 c1(N2CC3CC(NC(=O)C(F)n4cccn4)C3C2)cc(=O)n2cc(Cl)ccc2n1 O=S(=O)(c1ccc(Br)cc1NCC1CC2CC2C1)NCc1cccc(C(F)F)c1 C#Cc1ccc(CCC(=O)N2CC(NC(=O)CC(C)(C)C#N)C2)cc1 c1(C(N2CC(N(C)C(C34CC(C3)C(C)(C)O4)=O)C(O)C2)=O)ccn2nnnc2c1 Cc1ccc(-c2cccnc2S(C)=O)cc1-n1cccc1 C(=O)(CC1=NNC(=O)C1)N1CC(CNC(Cn2ncc(C)c2)=O)C(n2ccnn2)C1 N1(C(N(C)C)=O)CCCN(C(=O)NC2CCC(F)CC2)CC1 c1(C(=O)NC2CCC(OCC)CC2)ccc2[nH]c(C)cc(=O)c2c1 C1(C(=O)NCc2cc(C(N3CC(CN=[N+]=[N-])OCC3)=O)no2)CCCC(F)(F)C1 O=C(C#CCNC(=O)C=CC1CC1)NC1CC(F)(F)C1 C(=O)(C(C)(C)F)NC(CN(C(c1csc(CC(F)F)n1)=O)CC)C C1(C(C)C)CCCCN1C(c1ccc(CNC(c2cccs2)=O)o1)=O N1(C(C(C)NC)=O)CCC12CCN(S(=O)(=O)CC1CCC1)CC2 C1(CC(=O)NCC(c2ccccc2)NC(C2C(C)C2)=O)CCN(C2CC2)C1=O C#CCCCC(=O)N(C)CCC1CCN(C(=O)COC2CCCC(C)C2)CC1 N1(C(c2cnc(CC)[nH]2)=O)CC(CNC(c2cc(C(C)C)n(C)n2)=O)CCC1C C(=O)(C(C#N)C(C)(C)C)N(CC(C)NC(=O)C1=CC2C=CC1C2)C c1(C(=O)NC2C(NC(CCN(C(CC)CC)C)=O)C2)cc(C)c(O)c(C)c1 C1(NC(CC2N(C(C)C)CCC2)=O)(CO)CCCN(C(c2cnsc2)=O)C1 N1(C(CC2(N(C)C)COC2)=O)CCOCC(NC(=O)Cn2ncn(C)c2=O)C1 C(N=c1[nH]cncc1I)C1CC(NCc2c(C(=O)OC)cccc2)C1 c1(C(N2CC3(CN(C(CCC=C)=O)C3)OCC2)=O)ccc2c3c(cccc13)CC2 N1(C(N2CCC(C(=O)Nc3ccc(CC)nc3)(CC)C2)=O)Cc2ccccc2C1 S(=O)(=O)(c1ccc2nc(O)[nH]c2c1)N1CC2CN(C(CC(CC)C)=O)CC2C1 CCC(CC)(CCNC(=O)C(C)OCC(C)C)NC(=O)CC1CCC(=O)N1C C1(n2cc(C3(C)CCCN3C(c3cc(C#N)c[nH]3)=O)nn2)CCc2c[nH]nc2C1 c1(OCC(=O)NC2CC2CNC(=O)C(O)CC2CC2)ccc(Cl)cc1Cl c1(OCC(=O)NCC(=O)NC(C2CC2)C)c(C)cc(Cl)cc1Cl.CCCN C12CCC(CC1)C(=O)N(C(C)C)CCN(C)C2.c1(CC)oncc1C(=O)NC c1(OC)ccc(C(=O)NC2CCC2NC(c2ccnn2C2CCOCC2)=O)cn1 CC1CC(C(=O)NCC2CCN(C(c3ccc[nH]3)=O)C2)CN1c1ccccc1 C1(O)(CNC(C2(CC)CCC2)=O)CCN(C(=O)CC2CCCC(=O)N2)C1 N(C1COc2ccccc21)C(C1C2(CCN(C(c3ccc(O)nc3)=O)CC2)C1)=O N1(C(C(C(C)(C)C)O)=O)Cc2ccc(CNC(=O)CSCC(N)=O)cc2C1 Cc1cc(CCC(=O)NC(C)C(C)NC(c2nnsc2C(F)F)=O)no1 CC(C)CC(C(=O)NC(C)(C)CC(N1CCCC(C)(C)C1C)=O)C(N)=O c1(NC(C(N2CC(C)(C(F)(F)F)C2)=O)=O)nnc2n1CCCCC2 c1(NC(=O)Nc2cccc(CS(=O)(=O)NCCC)c2)c(Cl)nn(C)c1Cl Cc1c(C(c2nnnn2C)Nc2ccc(Br)c(C(C)O)c2)cnc2ncnn12 C1(CC)CC(C(N2CCC2C2CCCC2)C(=O)NC2CCCCC2)CC1O C1(C(=O)OCC2(F)COC2)CC(C)(C(C)C)CCO1 S(=O)(=O)(c1cc(F)cc(Cl)c1)NC(c1nccc(OC)c1OC)=O C(C(COC)CC(=O)NCCCC1CN(C(=O)CC2CN(C)C2)CCO1)OC c1(N2CCC(=C)C2)nc(=NCc2sccc2Br)[nH]c2ncn(CC)c12 c1(CC2N(C(c3c(NCC)[nH]nn3)C)CCOC2)ccccc1F C1(C(=O)NC2(CCC(N3C(CN(C)C)CCC3)=O)CCC2)COCCC1C c1(OC)ccc(NC2CN3CC2CC3=O)cc1.c1(C(=O)NC(C)C)cccs1 C1(C(=O)NCC(C)N(C)C(c2cccs2)=O)CC2CSCC(C1)C2(F)F C(=O)(CCCOC(=O)CO)NC1CC(NC(C(C)C2CCCC2)=O)C1.CC(C)(C)C n1(CC)nnc(C(=O)NC(C)(CO)C(=O)NCC2(C(N)=O)CC2)c1C O=[N+]([O-])c1cc(NCc2ccccc2-c2nc[nH]n2)c2c(c1)OCCO2 C(=O)(C1=C(C)OCCS1)NCC(CCCC)NC(C12CCCN1CCC2)=O C1(C(c2n(CCCSC)nnn2)NCCC2CC(C)C2)CC2CCC1CC2 c1(NCc2c(CC)nco2)cc(NC(c2cnn(C)c2)C)ncn1 C(c1cncnc1O)=CC(=O)NCCC(C)(C)NC(C1N(C)C(=O)NC1)=O N1(C(c2c(C)csc2)=O)CC2(CC(CC(=O)NOc3ccc(Br)cc3)C2)C1 C(CC1CC1)(C(=O)NC1CC(CCC(=O)NC(C)CN2CCCC2=O)C1)OC N1(OC)CC2CCCCCC2(C#N)C1.c12cc(C#N)ccc1[nH]c(=O)[nH]2 c1(N(CC(C)CO)C)nc(N2CCCC(F)C2)c2c(n1)CCC2 C1(C)(C(N2CC(C(C)NC(=O)Cn3nnc(=N)[nH]3)C2)=O)CCCC1O c1(C(=O)NC2CCC(F)(CNC(CCCCNC=O)=O)C2)cc(Cl)cnc1O C1(NC(CCc2onc(C)n2)=O)CC2CN(C(c3ccc(C(C)C)o3)=O)CC12 C(=O)(N=c1ccn(C(F)F)[nH]1)C1CCN(Cc2ccc(C(=O)OC)cc2)C1=O c1(C(=O)NCC2CCN(C(CCSC)=O)C2)ccc2nccc(C)c2c1 C=Cn1nccc1C(=O)NC1(CNC(c2ccnn2C2CC2)=O)CCCCC1 C1(NC(C2(C(N)=O)CC2)=O)CCCCN(C(c2c[nH]nc2C(F)(F)F)=O)C1 c1(C(N2CC(OCCNC(c3cc(OC)no3)=O)C2)=O)cc(Cl)c(Cl)n1C C1(C(N2C(N(CCO)CC)CCC2)=O)CC(O)CCN1C(c1[nH]cc(C)c1C)=O C(=O)(C1=CC2(CCOC2)C1)N1CCN(C(c2cccc3c2CCC3)=O)C(CF)C1 C1(C)(C(=O)NCCC(N2CCN(C)CC2)C)CCCN(CCC2CCCCC2)C1 c1(C(=O)OC)ccnc(N2CCOC(C(C)NC(c3ncoc3C)=O)C2)n1 N#CC1CN(C(=O)C(CNC(C2(N3CCOCC3)CCC2)=O)OC)CC12CCC2 C12(COC)CC(CNC(=O)Cc3nocc3C)(CN1C(=O)C1=CC(C)(CC)C1)C2 c1(C(N2CCC(N(C(C3CC4=C(N3)CCC4)=O)CC)C2)=O)ncc([N+](=O)[O-])n1C c1(C(=O)NCC(C)(CO)NC(C2CCN(C)C2=O)=O)ccc2nonc2c1 Cc1cn2c(C(=O)NCC=CCNC(C3CCC(=O)N3)=O)cnc2s1 C1(C2CCN(C(C=CC)=O)CC2)NC(=O)CCC1NC(=O)C=C1CCC1 C1(=CC(=O)NCCN(C(C23CCCCC2C3)=O)CC)CCN(C)CC1 C1(NC(C(c2n(C)nnc2)(F)F)=O)(CO)CCCN(C(C2CSCC(=O)N2)=O)C1 C1(C(N2C(C(N(CCN=[N+]=[N-])C)=O)C=CCC2)=O)CC2CCC(C1)C2 C1(C(C)NC(C=CCOC)=O)CCC(NC(=O)C(COC(C)(C)C)N(C)C)C1 c1(C(C)NC(CC)CNC(=O)OC(C)(C)C)cncnc1 C1(NC(CCNC(=O)NC)=O)COCCN(C(c2sncc2Br)=O)C1 c1(C(=O)NCC(CC)NC(C23CCC(OC)C2C3)=O)c(F)ccc(Cl)c1[N+](=O)[O-] CCCC(C(=O)OC)C(=O)N1CC(C(O)C(=O)NCC2CC=CCC2)C1 N1(C(CCc2cc(C)n(C)n2)=O)CC2(NC(=O)Cc3ccncn3)CCC1CC2 N1(C(c2c(CC)ncs2)=O)CCC2(CC2NC(=O)Cc2nc[nH]n2)C1 c1(OC)ccccc1SCC(=O)NCC1CC(NC(=O)CCc2ncc[nH]2)C1 C1(C(=O)NC(C)C(C)n2cccn2)CC2(CC2)CN1C(=O)CC1CCOCC1 N1(C(c2c(C)ccc(F)c2)=O)CCCC2(CCN2S(=O)(=O)C(C)C#N)C1 CC1CN(CCc2cccc(F)c2)CCC1NC(=O)Cc1ncc(Cl)s1 C(=O)(C1CCc2cc(O)cc(=O)n21)NC(C)C(c1ccc(O)cc1)=O C1(NC(=O)C2=Cc3cccnc3C2)C2Cc3c(Br)cccc3C12 N1(C(C(C)(CCF)NC(C=C(CC)CC)=O)=O)CC2(CNC(=O)N2C)C1 c1(OC)ccc(CN2CCC(NC(=O)C(C)Cc3ccccn3)CC2)cc1Cl C1(O)(CCNC(CN2C(C)CC2)=O)CCCN(C(c2cccn2C2CCC2)=O)C1 S(=O)(=O)(c1ccc(NCc2ncnn2C)c(Br)c1)NCC1CC(C)C1 N1(C(CCN(C(CCC)C)C)=O)CCC(O)(CNC(c2oc(C)cc2C)=O)CC1 CC(F)(F)C(F)C(=O)NC1CCOCC1C(=O)NCCC1(OC)CCC1 N1(C(=O)NCCOc2ccccc2F)CCC2(CNC(=O)N2)C1 c1(CC)cc(C(=O)NC2(CC)CCN(C(c3ccoc3Cl)=O)CC2)ccc1F N1(C(C2C(CC)OCC2)=O)CCC(CC(N2CCCCC2CN(C)C)=O)CC1 C1(C(C(=O)NC(CC)C(=O)OC)(C)C)CCCN(C(=O)C(n2nccc2C)C)C1 c1(C(=O)OC2CC(C(=O)OC)(COC)C2CO)cc(C#N)ccc1F CC1(C)CC(C(=O)NCC2(F)CC2)CN(C(=O)CN2CCC(F)CC2)C1 N1(C(C(C)(C)c2cnsc2)=O)CCN(C(c2nc(O)[nH]c(=O)n2)=O)C2(CCC2)C1 Cc1c(N)ccc(C(=O)NCCC(C)NC(C2(C)CC=CCC2)=O)c1Cl C12(CNC(C=CC)=O)CCCC1CCN2C(c1cc(-c2ccccn2)[nH]n1)=O N1(C(CC(C)CN2CCCC2)=O)CCCC(COCc2ccccc2)C1 C1(C(N(C2CCN(C(c3cscc3OC)=O)C2)CC)=O)COC2CCCCC12 C1(NC(C2CCOC2)=O)CCN(C(=O)Cc2cn3ccsc3n2)CC1O c1(C(N2C(C)CC(NC(C3(O)CC3)=O)C2)=O)cc2cc(Br)cn2cn1 Cn1cc(C2=CCCN(C(c3cc(Br)c4c(c3)nnn4C)=O)C2)cn1 N1(CC)C2CCC1CN(C(=O)CC(C)(C)N(C)C(c1cc(C)cc(O)c1)=O)C2 c1(C(=O)NCC2CCC(NC(CC3(C)CC3F)=O)CC2)onc2c1CCCC2 N1(C(C)=O)CCC2(NC(=O)C(O)(C3CC3)C3CC3)CC2C1 CCCCC(CNC(=O)C(C)(C)c1cnc[nH]1)NC(=O)Cc1nnc(O)s1 CCC(C)C(C(=O)N(CCCNC(=O)C=Cc1ccco1)CC)OC c1(OCC#C)ncccc1C(=O)NCCC(C(C)C)NC(=O)Cc1cnco1 c1(C(c2n(C(C)C)nnn2)NCC2CC23CCC3)ccc(C#N)cn1 C(=O)(C(C)(O)CCC)N1CC(NC(c2c(CC)c(C)sc2)=O)C1 C(=O)(CCCCCCSC)N(CCC(C(C)(C)C)NC(C(CCC)OC)=O)C N1(C(C=CC=CCC)=O)CCCC(NC(=O)C=CC2CCOCC2)CC1 CCC(O)C(C)C(=O)NCC(O)CNC(C1CCN(CC(C)C)C1)=O CCCCC(C(=O)NC1(C)C(=O)N1)C(C)C.c1(OC(C)C)ccc(S(C)(=O)=O)cc1 C1(NC(=O)C=CC2CCCO2)CCCC12CN(C(C1(C(F)F)CCCC1)=O)C2 c1(OC)cccc(NC(C2(NC(=O)C(=CC3CCCC3)C)CCCCC2)=O)c1 N1(C(C(C)C2CCCO2)=O)CC(C)N(C(=O)CSCc2ccccc2)CC1C C(=O)(CCN(OC)C(=O)C(C)CCC(C)(C)C)N(C1CN(CC)CC1C)C1CC1 C1(O)(CC(=O)NCC(CCNC(C2CCOCC2C)=O)OC)CCCCCC1 C1(C(=O)N)CCN(C(=O)CC2CCCSC2)CC1F.Cn1cnnc1C(C)(C)C c1(C(=O)NCCN(CCC)C(C2CC3(C2)CC(C)C3)=O)cc(Br)ccc1F c1(OCC)ccc(Cl)c(C(=O)NC(CNC(c2cncc(F)c2)=O)C2CCC2)n1 C=CC1(C(N2CCC(COC)C2)=O)CCN(C(=O)CC2(O)CCCC2)CC1 N1(C(c2c(COC)scc2)=O)CCN(C(C2CC3(CC3)CN2C)=O)C(C(F)F)C1 C1(c2c(SC)cccc2F)CS(=O)(=O)CC1C(=O)NCCNC(=O)C1=CSCS1 N(C1COc2ccccc21)C(C12N(C(COCCCC#C)=O)CCC1CCC2)=O c1(OCC#C)ccc(NC(c2cc(C#N)cs2)c2nnnn2C2CCC2)c(C)c1 Cc1cc(C(N2CCC(NC(=O)C3=CCCO3)C2(C)C)=O)ccc1-n1cccn1 Cc1ccc(C(N2CC(NC(=O)Cc3cccc(O)c3)C2)=O)cc1NS(C)(=O)=O N1(C(CCCc2cc(C)no2)=O)CC(NC(C2CN(S(C)(=O)=O)C2)=O)C2CC12 C1(NC(CCn2c(C)ncc2)=O)C(C)CN(C(=O)C=Cc2cccs2)CC1C C1(c2ccccc2)(NC(CC(=C)I)=O)CCN(C(c2ccncc2)=O)C1 C1(NC(c2ccc(C)s2)=O)CC2CCC1(CNC(c1csc(O)n1)=O)C2 C#CC1(C(N2CC(=O)NCC2CC)=O)CCN(C(=O)CC(C=C)CC)CC1 C(=O)(C1CCCc2ncnn21)N1C(CN(C)C(c2nncs2)=O)CCC1 C(=O)(C1=CCC(C)CC1)NCCC(C(=O)N(C)Cc1c[nH]nc1C)OC CC1(NC(=O)C=CCBr)CN(C(=O)C(O)CF)C1 c1(CN(C(=O)CCC2CC(NC(C3(N(C)C)CCC3)=O)C2)C)ccncc1 N1(C(C(C)(C)C2CC2)=O)CC2COCCC2(NC(C2CCc3cnnn3C2)=O)C1 C1(C(N(C(C)C)CCN(C)C(c2nn(C)cc2N)=O)=O)CCN(C)C(=O)C1 N1(C(C(CC)C#N)=O)CCCC(CO)(NC(=O)CCc2cc(C)n(C)n2)C1 C1(CC=C)(C(=O)NCC2(Cl)CC2(F)F)CCN(C(c2cc(OC)cnn2)=O)C1 c1(OCC)ncc(C(N2CCC(N(C)C(c3cc(OCC)n[nH]3)=O)C2)=O)cn1 N1(C(C2CNC(=O)N2)=O)CC2CCCC(NC(C3(C4CC4)CCCO3)=O)C2C1 c1(C(=O)NCC2C(C)CN(C(=O)C(O)C(C)(C)C)CC2)cc(S(N)(=O)=O)c(Cl)o1 CC1(C)CCN(C(=O)CCS(N)(=O)=O)CC1NC(C1CCN(C(N)=O)CC1)=O c1(C(N2CCC(NC(=O)C(=Cc3c[nH]cn3)F)C23CC3)=O)cc2ccccn2n1 CC1(C(=O)NC2COCC2NC(c2[nH]ccc2C2CC2)=O)CC2CCC(C1)S2 N1(C(C2=C(C)OCCC2)=O)CCOC2(CCCN(C(C34CCC(CC3)O4)=O)C2)C1 C1(NC(C=C(CCC)C)=O)CCCCC12CCN(C(c1cnco1)=O)C2 N1(C(CC(CCC)C2CC2)=O)CC2CC(CNC(=O)C(C#N)C(C)C)CC1C2 Cc1ccnc2sc(C(=O)NC3CC(NC(=O)CS(=O)(=O)C(C)C)C3)c(C)c12 C1(NC(c2ccc(C)s2)=O)CN(C(c2cccs2)=O)CC1c1ccnn1C c1(OC)cccc(C(N2CCCC(CO)(NC(C3CC3CF)=O)C2)=O)c1O Cc1nc(O)nc(C)c1C(=O)NC1(CNC(C2OC3CCC2CC3)=O)CCOC1 C1(NC(C(CN(C)C)N(C)C)=O)CCCCCC1C(N1CC2(C1)CN(C)C2)=O C1(C(N2CC(CNC(c3c(OC)csc3)=O)OCC2)=O)CC(C2CCC2)C1 C12(C(=O)NC(c3cc(C)no3)C)CCCC1CCN2C(=O)Cn1cc(CO)nn1 C(CC)(CCC(=O)N1CCC(CCC)(CO)C1)NC(C(C=C)CC)=O C(CN=c1[nH]nc(Sc2ccccn2)s1)NC(C(COC(C)C)(F)F)=O c1(C(=O)NC(C)C(C)NC(=O)CC2(C#N)CCCCC2)ccc2n[nH]cc2n1 c1(CC(=O)NC(C(=O)N(C)CCC2CC2)C2CCC2)ccccc1 c1(CC)cncc(C(=O)N(C2CCCN(C(=O)CC3(OC)CCC3)C2)CCO)n1 Cc1cc(NC(=O)C(C)(C)C#N)ccc1NC(c1ccccc1SC(F)(F)F)=O c1(CCC)cc(C(N2CCC(CC=C)(NC(c3sccc3C)=O)C2)=O)sc1C CCC(C)(C)C(=O)NC(C1CCOC1)CNC(c1ccn(C)c1C1CCC1)=O c1(C(N2CC(F)CC(NC(C=C(C)C)=O)C2)=O)ccc2cccnc2c1 C1(O)(CC(=O)NC(C)C(C)NC(C2CCC(=O)NC2)=O)CCCOC1 n1(CC(=O)NC2(C3N(C(c4nc(CCC)sc4)=O)CCC3)CC2)ncn(C)c1=O N1(C(c2ccc(CCC)cc2)=O)CCCCCC(NC(C2CC(O)CN2C)=O)C1 C1(NC(CC2CC(=C)C2)=O)CCN(C(=O)Cc2n[nH]c(C)n2)C1C(C)C CCC(C)CCC(=O)NC(C1CCCCC1)CNC(c1cnc(O)s1)=O OS(=O)(=O)CCCCCO.CN1CC(OC)CC1 c1(C(CN(C(C(CN(C(C)=O)C)(C)C)=O)c2ccccc2)O)ccc(Cl)cc1F C(=O)(CN=S(C)(C)=O)N1CC(OC)C(NC(=O)C(F)(F)C(F)F)C1 C1(CCOC)(NC(c2ncc(C)cn2)=O)CCN(C(c2oc(C)nc2C)=O)C1 C12(C(=O)NCCCCC(C)NC(C3C(OCC)C3)=O)CCC(O)(CC1)CC2 C1(NC(C(CCC)=CCC)=O)CN(C(c2ccc(C)o2)=O)CCC1CO N1(C(c2nc(CC)oc2C)=O)C2CCC(C2)C1C(=O)NCc1cccnc1 N1(C(c2ccc(C)cc2)=O)CCC2(CCCC2NC(=O)C=CCO)C1 C1(C(=O)NCC2CCC(NC(c3c(C)cc(O)nc3)=O)C2)CC(F)(F)CCC1(C)C c1(OCC)ccc(C(=O)NCC2(C)CCCN2C(=O)CCP(C)(C)=O)cc1OC C1(C(N2C(CNC(c3cnc(OC)nc3C)=O)CC2)=O)CC2CC1CC2(F)F N1(C(C(C)OCC)=O)CC(CNC(=O)CC2CCCCC2)CC12CCC2 c1(C(=O)NCC2(NC(=O)C(Cl)=CCl)CC3CCC2C3)ccn2ccccc12 C1(NC(C=CC(=O)OCCCC)=O)CC2CCC(C1)N2C(c1ccc(SC)o1)=O C=CCCCC(=O)NCC1(F)CCC(CNC(=O)Cc2cc(C)ccn2)C1 C1(C)(CC)CCC(C(N2CCC(F)(C(N3CCC(F)(CF)C3)=O)C2)=O)O1 n1(CC)nccc1C(C)NC(=O)CCC1(NC(c2cncnc2)=O)CCCC1 C#CCCC(O)C(=O)N1CC(NC(=O)C(C2CC2)SC)C1 N1(C(C2(CC(=O)NC)CCC2)=O)CC2CCN(C(=O)C3=NOCC3)CC2C1 N1(C(C(C2CN(C(C3OCCCC3(C)C)=O)C2)OC)=O)CCCC(N=[N+]=[N-])C1 C12(C(=O)NC(CCC)C(F)(F)F)CCCC1CN(C(=O)C(C1CCC1)OCC)C2 C1(CNC(COCCC(C)C)=O)CCN(C(c2cnc(S)n2C)=O)CC1(F)F C(=O)(C1=C(Cl)CCC1)N1C(CCNC(=O)C(C)(C)c2ccc(Cl)s2)CC(OC)C1 C(C(CC(=O)Nn1cccn1)C1CC1)NC(CC(=O)OC(C)(C)C)=O c1(CNC(CC)=O)ccc(CNC(c2ccc(C)cc2C(C)(C)C)=O)cc1F c1(C(=O)OC)cc(C)ccc1C(N1CCOC(C2CC(C(=O)O)(OC)C2)C1)=O n1(C(C(=O)N(CCC(=O)NC(C#C)C2CC2)C(C)C)C)ccc(C)n1 C(CO)(C1CCc2ccccc21)N(c1c(C)cccn1)CC(=O)OC(C)(C)C c1(NC(=O)N(C(C)(C)C)C)ccc(CN(C)C)cc1Cl.CC1CO1 N1(c2cccc(C(N(CCC(C)NC(C(CC)C)=O)C)=O)c2)C(=O)CCCC1=O N1(C(CN2CCC(C)(C)C2)=O)CCCC2CN(C(=O)CC3CCOC3)CCC12 C1(CC(=O)NC(C=C)C(F)(F)F)CCCN(C(=O)Cc2cn(C)cn2)CC1 C(CCCC(CO)NC(C12CC(C)(C1)C2)=O)NC(c1c(Cl)cn(CC)n1)=O C(=O)(C(C)(C)C1=CCSCC1)N(C(CCNC(C(CCC)C)=O)C)C C1(NC(C2(CC(=O)OC)CC2)=O)CC(NC(C2CCN(C)CC2)=O)C12CCC2 C1(CCC(=O)OCC)CCCN1N1CCC(Cc2ccccc2)C1.C1CO1 C(C1CN(C(c2[nH]nnc2C2CC2)=O)CC1C(=O)NCc1ccc(OC)o1)=CC CCCCC(C(=O)NC(C(=O)NC1(CO)CCC1)C1CCC1)C(C)C C1(CNC(C(C)Cn2cccn2)=O)CCN(C(c2ccn(C3CC3)n2)=O)CC1 C12(CCOC)CCN(CC1)C2=O.c1(CNC(=O)Cc2cnoc2)cc(Cl)ccn1 C=C=CC(C)C(=O)N(C(CNC(=O)Cc1csc(=N)[nH]1)C1CC1)C c1(C(N2C(CNC(c3cccnn3)=O)CC(OC)C2)=O)coc2c(F)cccc12 C1(NC(=O)OC(C)(C)C)CC(NC(=O)Cn2cccc2)C12CCC2 N1(C(c2cc(C)cc(O)n2)=O)CCC2CCCC12CNC(C1CCC(C)CC1)=O n1(CC(=O)NCC23CC(CN2C(c2ccc(CO)o2)=O)C3)nnc2ccccc12 C1(C(N2CC3CC(Nc4ncnc(C(F)(F)F)n4)C2C3)=O)CCCC(F)(F)C1 CC(C)C(C(C)NC(=O)COC1CCC1)NC(c1nc(Cl)cs1)=O c1(OC)ccc(C)c(C(=O)NCC(O)CNC(c2nn(C)cc2Br)=O)c1N c1(C(=O)N(CCCc2ncnn2C2CC2)C2CC2)ccccc1S(=O)(=O)NCC1CCC1 c1(C(=O)NC2CCN(C(Cn3c(C)nnn3)=O)CC2C)cc2n(c1)CCCC2 C=CCC(C)(C)CC(=O)N(C1CN(C(c2ccc(C#N)c(O)c2)=O)CCC1C)C C1(CNC(c2c(C)ccc(C)c2)=O)CCC2(CCC2)C1NC(c1sccc1C)=O c1(CCC)ccc(-c2ccc(C(N(C)Cc3noc(CC)n3)=O)s2)cc1 C1(C(N(CCCNC(C=CSC)=O)C2CC2)=O)CCc2nn[nH]c2C1 Cc1cccc(C)c1NC(=O)CN1CCN(C(C2CCCCO2)=O)CC1 CC(C(=O)NCCC1(NC(=O)Cn2ncnn2)CC1)OC(C)(C)C N1(C(C=C(C)C)=O)CCOC(C)C1C(=O)NCc1cc(C)c(C)s1 CC1CC(CC(=O)NCCS(N)(=O)=O)CN1C(=O)C=Cc1cncs1 CCC(CC)(C(=O)NC(C1CCCN(C(=O)Cc2noc(CSC)n2)C1)C)OC c1(C(=O)NC2C=CC(CNC(C3(C)ON=C(C)C3)=O)C2)sc(Cl)c(Cl)c1C N1(C(CC(C)F)=O)CCN(C(C2NC(=O)OC2(C)C)=O)C(c2ccc(F)cc2)C1 C(=O)(CCCCC(C)C)NC1C(SC)CN(C(=O)COc2cncc(C)n2)C1 CCCS(=O)(=O)C(C)C(=O)NCCCCC(C)NC(=O)C(C)(C)C1CC1 N1(C(c2c(C)nc(-c3cccc(OC(F)(F)F)c3)[nH]2)=O)CCC2OC(=O)OC2C1 CC1=C(C(=O)NC2CCC23CN(C(=O)C(F)CC2CCC2)C3)CCCC1 C(=O)(C(C(=O)NCCNC(=O)C(N1CCCCCC1)C)c1ccccc1)OCC C1(NC(c2ccc(Cn3ccnn3)o2)=O)CN(C(=O)C2=NOCC2)C2(CCOC2)C1 C=CC(C)CC(=O)NC(C1CCCN(C(=O)C(C2CCC(=O)CC2)F)C1)C C1(C(=O)NC2CC(NC(C(C(C)C)NC(C)=O)=O)C2)CCS(=O)(=O)C1(C)C c1(OC)cccc(F)c1CC(N1CC(CNC(c2cnc(C)o2)=O)CC1C)=O C1(C(N(CCOCC)CC)=O)CCN(C(C2(C)COCCO2)=O)C1(C)C C1(NC(c2nccc(CC)c2)=O)CC2(CCCN(C(C3CCC(C)O3)=O)C2)C1 C1(C(=O)NCCC2(COC)CC2)(NC(C2CCCCS2)=O)CCSC1 c1(OC(C)C)ncccc1C(=O)NC1CC(CCNC(C2CCCC(C)C2)=O)C1 C(=O)(C(C)(C)C(C)(F)F)N1C(CCC(N2CC(C=C)C2)=O)CCC1 C1(O)(CC(=O)N(C2CCN(C(=O)COCP(C)(C)=O)C2)CC)CCOC1 CC(=O)CCCCC(=O)NC(C)(C)CC(=O)Nc1c(C)cc(C)cc1C n1(CC)cnc(CCNC(=O)Cn2cc(CNC(c3coc(C)c3)=O)nn2)c1 C1(COC(=O)NC2CC=CCC2)CCCCN1C(=O)CCC(F)F Cc1c(-n2cc(CN(C)C)nn2)cccc1Br.N1(C(C(C)=O)=O)CCC(O)C(OC)C1 CCCC(O)CC(=O)NC1CCCCC1NC(C1(F)CCCC1)=O C1(NC(C(C)NC(=O)NC)=O)CCC(C)N(C(c2cnc(C)nc2COC)=O)C1 C1(COC(c2ccc(CSC)cc2)=O)CNC(=O)CC2(CCC2)O1 c1(C(N2CC(NC(C(CCCC)NC(N)=O)=O)C(C)C2)=O)cn2nc(C)sc2n1 N1(C(C23CC(C(=O)OC)(C2)C3)=O)C2COCC1CC(NC(=O)C(C1CC1)SC)C2 c1(N(C(=O)Cn2cc(CC3CCCC3=O)nn2)C)nccnc1Cl Cc1noc(C)c1C=CC(N1CC(N(C)C(c2ccsc2C)=O)C(O)C1)=O C(=O)(C(C)CC(=O)NC1CCCC1C(N1CCN(CC2CC2)CC1)=O)OC c1(C(N2CCCC2c2ccccc2Br)C(=O)NCCCC)ccc(C(F)(F)F)cn1 C(=O)(C(C)(C)CC1CC1)NCC(COC)NC(=O)CC(C)C1CCCO1 N1(C(C(=O)NCCOC)CSC2CC2)CCN(C2CCOC2)C(=O)C1 C(=O)(C(C(C)(C)C)N1C(=O)CCC1=O)OC.c12cn(nn1)CC(C)NC(=O)C21CC1 c1(C(N(C(CCNC(c2n(C(C)C)cnc2)=O)C)C)=O)ccn2nccc2n1 C=C(Cl)CC(C(=O)NCCN(CCCF)C)NC(c1cccc(O)c1Cl)=O C1(=CC(=O)NC2CC(CCC(=O)N(CC(O)CO)C3CC3)C2)CCOCC1 CC(C)(CCCNC(C1(F)CC=CCC1)=O)NC(=O)CC1CCOCC1 c1(C(N(CCCNC(C2(C)ON=C(C)C2)=O)CCO)=O)nnc(O)nc1O c1(NC(Cn2c(C(C)C)ncc2)=O)ccc([N+](=O)[O-])cn1 C1(OC)CCC2(C(=O)NC(C3CCOC3)CNC(=O)Cc3ccoc3C)CC12 c1(C(N2C(CNC(CC3(Cl)C(C)(C)C3)=O)CCC2)=O)cccc2c1CCC2=O C1(C(=O)NCC2C(NC(c3c(N(C)C)cc(F)cc3)=O)C2)CCc2ccnn2C1 CC(C)CC(O)C(=O)NCCCN1CCC(NC(=O)Cc2cnns2)C1 c1(C(=O)NC(CN(C)C)C(=O)N2CCC2C2CCCOC2)ncn2c1CCC2 C(=O)(C(CC)CC(C)C)N(C1(CC(=O)NC(C(=O)N(CCC)CC)CC)CC1)C c1(OC)csc(COC(=O)C(=O)OCc2ccncc2)n1 O=C(C#CC1CCCCO1)N1CCC(CNC(=O)Cc2cnccn2)C12CC2 c1(CNC(C2C(NC(CC3(C(C)(F)F)CC3)=O)COC2)=O)nc2cccnc2s1 C1(OC)CC(CO)N(C(=O)CCN(CCO)C(c2cc(CO)oc2C)=O)C1 c1(CC)cc2c(NC3CC4CN(C(=O)CCCC5CCC5)CC34)ncnc2s1 N1(C(c2ccc(OC)nn2)=O)CCC(CC(=O)NCCC(C)(C)C)C1(C)C C1(NC(C(CC)(CC)CO)=O)C(C)(C)CN(C(=O)CCN(C)C(C)=O)CC1(C)C C(C(C)(C)CN(C(C1C=CCC1)=O)CC)N(C(=O)C=CCN1CCCC1)CC N1(C(c2ncc(Cc3ccccc3C)s2)C(=O)NCCOC)CCC2(CC1)CC2 c1(OC)ccc(C(O)CN2CCC(Nc3ccc(CN)cc3)C2)cc1Br N1(C(CC2(C)CC2)=O)CC2CCCCN2CC1CNC(=O)C=CBr c1(NC2(c3n(CC)nnn3)CCC(c3ccccc3)C2)ccc2c(c1)C(=O)NCC2 n1(CCOC)cc(-c2ccc(C(=O)NCCCCCO)s2)c(C(F)(F)F)n1 C1(C(N(CC(CC)NC(c2occc2C)=O)C)=O)CC12C(=O)Nc1ccccc12 C(=O)(C1=CCC(C)CC1)NCC(CNC(c1c(Br)sc(C)c1C)=O)O c1(CNC(=O)NC(C)C)cccc(C(N2CCC(N3CC(C)(C)C3)C2)=O)c1 C#CCC(C)(C(=O)NCc1cn(CC)nn1)NC(=O)Cc1ccnc(O)c1 c1(C(C)C)cccc(CC(=O)NCCCNC(C2(C3CCCO3)CCCC2)=O)c1 CCCCC(CC)CCC(C)Nc1nccc(N)n1 CC1CCC(C(=O)NCC2=CCCOC2)N(C(c2cn(C3CC3)cn2)=O)C1 N1(C(C(C(CC)C)O)=O)CCC2(CCN(C(=O)CSCc3ccccc3F)C2)C1 C1(C(=O)NCc2cc(C)c(C)o2)CCN(C(C2(C)CC(=O)N(C)C2)=O)C(C)(C)C1 c1(CNC(=O)CSC2CC2)ncoc1C1CN(C(=O)CCOC2CC2)C1 C(=O)(C=NOC)N(CC(CC)NC(C1CCCN1c1cnccn1)=O)C N1(C(c2c(OC)cnnc2)=O)CCC(N(C)C(c2n[nH]cc2[N+](=O)[O-])=O)C(C)C1 N1(C(CCC2C(C)C2)=O)CC(CNC(=O)CCc2cncs2)C(F)(CO)C1 C1(CC)CN(C(C2(O)CCSCC2)=O)CCC1NC(c1cc(F)ccc1O)=O O(N(C)C(=O)COC1(C)CN(C(=O)CCc2ccnn2C)C1)CC(=O)OC C(=O)(C(C(C)C)OC)NCCN(CCOC)C(C1(CO)CCCC1)C.C1(=O)CN1 N1(C(CC(C)OC)=O)CCC(C)(CNC(C2(c3cccs3)CCCCC2)=O)C1 Cc1ccc(O)c(CNC(=O)Nc2ccc(OC3CCOC3)cc2)c1 C(=O)(C(F)CC(C)C)NC(C1CCOC1)CNC(c1c(CC)onc1C)=O CCCCC(C)CCC(=O)NC(COCC)C(=O)Nc1cscc1C CC1CCCN(C(c2cscn2)=O)C1CNC(C1CCCN1C1CCCCC1)=O C1(CC)C(NC(c2cnc(OC)s2)=O)CCN1C(c1ccnnc1)=O C1(NC(C(CC)=CCCC)=O)CN(C(C2(CN(C)C)CC2)=O)CCC1O N1(C(C2N(C(C)=O)CCC2)=O)CC(NC(=O)CCC(N)=O)Cc2ccccc21 CCCC(C)(CCC)C(=O)NCCc1cnc(CNC(=O)C(C(C)O)N(C)C)s1 c1(C(N(C(C)CNC(=O)C(C)(C)N(C)C)C)=O)ccc(F)cn1 S(=O)(=O)(c1cccc2ccccc12)NC(c1cc(OCC)ncc1)C CCCC(C)CCCCNC(=O)N(C)C(c1ccc(Cl)c(Cl)c1)C Cc1ccnc(NCCN2CCSCC2)n1 C=CC1CNCC1NC(C1C2CC1N(C(=O)COCC(=C)C)C2)=O C1(C(N(C23CC(C4CCCN4C(=O)NC(C)(C)C)(C2)C3)C)=O)C2CCCC12 N1(C(CN(C(=O)CCn2cncn2)CCC)=O)CCOC(CN=[N+]=[N-])C1 c1(C(N2C(CNC(C3C(C(=O)OC)CCCC3)=O)CCC2)=O)cccc(O)c1F N1(CC2CN(CC)C2)CCC(NC(=NCc2ccnn2C)NCC(C)(F)F)CC1 N1(C(CCCc2nc(C)sc2)=O)CC(NC(=O)Cc2ccsc2Cl)C2CC12 C=CCC(CC(=O)N1CCCC(COC)C1)NC(c1cc(C)c(N)cn1)=O C1(C(=O)NCCCNC(=O)OC)CCCN(C(C23CCCC2C3)=O)CC1 Cc1ccc(CC(=O)NC(C2CCN(C(C3CC3c3cnn(C)c3)=O)C2)C)cn1 C(CS(=O)(=O)NCC(=O)N(CCCNC(=O)Cc1nccn1C)CCO)OCC c1(C(=O)NCC=CCNC(c2n(C)ccc2)=O)cc2c(nc1O)CC(C)(C)CC2 C1(C(=O)NC(CC(=O)NCc2onc(C(C)C)n2)(C)C)CC(=O)NC(C)C1 N1(C(C(CCC)n2cccc2)=O)CCCC(C2(NC(=O)CCn3ccnn3)CC2)C1 C12(CCCC1C)C(=O)N2.c1(CC2CN(C(=O)OC(C)(C)C)C2)[nH]nnc1C1CC1 Cc1ccn2c(N(CC(N3CCSC4(CCC4)C3)=O)CC(C)C)cnc2c1 N1(C(c2cc(C)ns2)=O)CC(CCNC(=O)CCC(C)(C)F)OC(C)C1 N1(C(C2(CC=C)CCC2)=O)CCC2(CCC2)C(CNC(=O)CCCC(N)=O)C1 C1(CC)(NC(=O)C=CC2CCCCCC2)CCN(C(c2nnsc2SC)=O)CC1 CC1CN(C(c2cncc(Cl)c2)=O)CCC1NC(C1(O)CCOC1)=O N1(C(C2CC(n3cc(C(CC)OC)nn3)C2)=O)CC(O)CC1CN(C)C1CC1 c1(C(=O)NCC2CCC(C)O2)ccc(C(=O)OC(C)(C)C)cc1.C1CCN1C C1(C(=O)NCCN(C(=O)C(O)CC(C)C)CCC)CC2C=CC1CC2 c1(NC(N2CC(C3OCCN(C(C(C)C)=O)C3)C2)=O)ccc(N)c(Cl)c1 c1(CCNC(c2ccc3c(c2)C(C)CCC3)=O)cccc2c1OC(C)(C)C2 Cc1cccc(C(=O)NCC2(CC(N3CC[Si](C)(C)CC3)=O)CC2)c1N c1(CNC2CC(C(=O)NC(CO)C(F)(F)F)C2)ncc(Cl)cc1F c1(C(=O)NC(CNC(CC(CC)OC)=O)(C)C2CC2)cc(OC)cc([N+](=O)[O-])c1 C=CCCC(F)(F)C(=O)NCCC1CCCN(C(C2(C#N)CCCC2)=O)C1 C1(C(=O)NCCN(C(=O)CCCCc2ccc(F)cc2)CC)CCC(F)(F)CC1 C1(NC(CCCOCCC)=O)CCCCN(C(c2cnc(CCC)s2)=O)CC1 C=CCC(CC=C)C(=O)NCC1(F)CCN(C(C2CC2C(C)C)=O)C1 c1(CNC(CCN(C(=O)CC2CC3CCC2C3)CC=C)=O)cnc(O)c(F)c1 CCCCC(C(=O)NCC(C)(O)CNC(C1CC(OC(C)=O)C1)=O)N(C)C c1(NC(C2C(C(=O)OC)C2)=O)ccc(C(=O)NC2CC2c2cnc(C)[nH]2)c(C)c1 CC(C)(C)CC(=O)N1CCC(CNC(=O)C(C)(C)CC2CCC2)C1 N#Cc1cc(C(=O)Nc2cccc(-c3cccc(C(=O)O)c3)c2O)ccc1O C(=O)(C(C)(C)CCCF)N1CC2(CN(C(c3c(C)c(N)cnc3)=O)C2)C1C(C)C C1(C(N(CCCNC(C2CCN(OC)CC2)=O)CCC)=O)CCCC(C)CC1 C1(C(=O)NCC(c2ccccc2)CNC(CCCCC)=O)OCCN(C)C1=O C1(CCC)COCCC1N=c1ccc(Br)c(S(=O)(=O)N2CCC(C)(C)C2)[nH]1 N1(CCC(=O)NCC2CC(NC(C(C3CCCOC3)OC)=O)C2)CCN(C)CC1 c1(N(C)C)ccc(N)c(C(N2CCC(O)C(NC(C3CCCS3(=O)=O)=O)C2)=O)c1 Cc1cc(C(=O)NCCN(C)CC2CN(C(=O)C(C)(C)S(C)(=O)=O)C2)n(C)n1 C1(C(=O)NC2(C(=O)NC3C(CCC)CCC3)CSC2)CC2C=CC1O2 c1(C(N(CCCNC(C(C)SC)=O)C(C)C)=O)cc(OC)c(OC)c(OC)c1N c1(C(=O)NCc2ccc(Cl)nc2)ccc2occc2c1.C12(CCC1)C(C)NC2=O C#Cc1cnc(C(=O)NCCCNC(=O)CC2CCC(C3CC3)CC2)c(C)c1 CC(C)CC(O)CNCC(c1ccccc1)c1nc[nH]n1 c1(CNC(c2cc(N3CCCC3)ccn2)=O)ncc(C(=O)NOCC2CCCO2)cn1 C(C(C)(C)C(=O)N1CC(N(C)C)C1)N(C)C.C1(=O)C(C2CC2)N1C c1(C2C(C)C2)c(CSc2cccc(-c3cn(C(C)C)nn3)c2)cnn1C N1(C(CC23C(CN(C(CSCC)=O)C2)CC3)=O)Cc2ccncc2C1 C1(NC(C(N2C(C)COCC2)=O)=O)CN=C2N=CNN2C1 C1(C#N)(C(N2CC(C(N3CCC(CCOC)C3)=O)OCC2)=O)CC(F)(F)C1 c1(C(N2CC3C(CNC(c4c(SC)cccc4)=O)C3C2)=O)cccc(Cl)c1N c1(N2CCC(NC(c3cccc(SC)c3)=O)C(F)C2)ncnc2[nH]cc(C#N)c12 c1(C(=O)NCC2(NC(CC3(C)CC3F)=O)CCCCC2)cc(S(C)(=O)=O)co1 N1(C(C2C3CCCCC23)C(=O)NC(CC)C)CCc2c(cnn2CCNCC)C1 C=C(C)CC(C(=O)NCC1CCCC12CC2)NC(=O)CCc1cn[nH]c1 N1(C(C2(CC(=O)OCC)CC2)=O)CCC(NC(=O)C(C)CC2CC2)C1 c1(C(=O)NC2C(CNC(C(CCSC)O)=O)CC2)nc[nH]c2nccc1-2 C=CCC(CC(C)C)C(=O)N1CCC(CF)(NC(=O)C(CO)NC(=O)C(C)C)C1 c1(CC)cnc(C(=O)NCc2noc(C)c2CSC)cn1 N1(C(c2cc(C)on2)=O)CC(C(N2CC(O)CC2(C)C)=O)CC(F)C1 C1(CN(C(=O)CCOC)CC)CCN(c2nnnn2C(C)COC)CC1 C1(C)(CC)C=C(C(=O)NCc2csc(C(=O)N(c3ccccc3)CC)c2)C1 C1(C)(CO)C(=O)N1.C(CC=O)N(C(=O)CN(CC)CC)CC#C.NC C1(c2cn(CC(C)C)nn2)CCC(C(=O)NC(C)CC(=O)O)CC1 C1(C(=O)NC2CCC(NC(CC(=O)NCC)=O)C2)CC(=O)NC2CCCCC12 c1(OC)nc(C)ncc1C(N1CC(NC(=O)CN2CC(=O)NC2=O)CC1C)=O CCCCCC(CC)C(=O)NCC(CO)NC(c1ccc(S(C)(=O)=O)cc1C)=O c1(CSCC(=O)NC(C)CCNC(=O)CC2CC3CC3C2)ccc(C#N)cc1 CC1CN(C)CCC1N(C(=O)C=CCNC(C1CCCSC1C)=O)C C(=O)(CCCCCCCCCO)NC1C(C)N(C(=O)CCn2cccn2)CCC1 C1(NC(C=C(CC)CC)=O)CCS(=O)(=O)C12CN(C(c1cc(C)c(Cl)cc1C)=O)C2 C1(F)(C(=O)NCCN(C(C2(CCC)CCNC2=O)=O)CC)CCCN(C)C1 c1(COC)ccc(C(c2nnnn2C2CCOC2)NCc2cc(Cl)sc2Cl)cc1 C(c1ccc(F)cc1)=C(C(N1CCC(C(C)NC(=O)CN2CCCCC2=O)C1)=O)C#N C1(CNC(C2(NC(N)=O)CC2)=O)CN(C(=O)C(F)C2CCCC2)CCO1 CC1CN2CCN1C(C(N1CC3(CC(NC(C4CCN(C)C(=O)C4)=O)C3)C1)=O)C2 c1(CNC(C(C)SC)=O)cnn2c1CN(C(=O)CCc1cscn1)CC2 N1(C(c2n(C(CC)CC)ncc2)=O)CC(C2CN(C(C3CC(O)C3(C)C)=O)C2)C1 CC1CCN(C(C2(C)C=CCN2C(=O)CCc2ncnn2C)=O)CC1(C)C Cc1ccc(F)cc1C(N1CCCCC(CNC(=O)C(C)N2CC(C)C2)C1)=O C=C1CCC(C(N2CCOC(CNC(c3ccncc3Br)=O)C2)=O)CC1 CC1CC(C)(C(N2CCC(F)(CNC(c3ccco3)=O)CC2)=O)CCO1 C1(C(=O)NCC(COC)NC(c2cccnc2)=O)CCCCN1S(C)(=O)=O N1(C(CC2(OC)CC2)=O)CCOC(CNC(=O)CC2(C)OCCO2)C1 C1(NC(c2cc(C)c(C)o2)=O)CC(F)CN(C(=O)C(C(C)O)N(C)C)C1 Cc1cn2c(n1)C(C)CC(C(=O)NCC1CCCN1C(c1cn(C)nc1Cl)=O)C2 N1(C(CN(CCC)C)=O)CC2CC2C1.c1(N(C(=O)CC)C)nnc(C2CC2)o1 Cc1sc(Cl)nc1C(=O)NCCOCCNC(C12CCN(CC1)C2)=O O=C(N=c1cnc(Cl)c[nH]1)c1ccc(NCc2c(Cl)nc3sccn23)cc1 CC(C)(C)C1=NOC(C)(C(N2CC3CCC3(CNC(C3CNC(=O)C3)=O)C2)=O)C1 C1(C(=O)OC)CN(C(C2C3C2CC3)=O)CC1OC.C1C(O)C(=O)O1 C1(CC)CN(C(=O)Cc2ccc(Cl)s2)CCC1NC(C1CC(SC)C1)=O Cn1c(NC(=O)COS(C)(=O)=O)nc2ccc(F)cc12 n1(CC(=C)C)nnnc1C(c1ccnn1CC)NC(c1ccc(Cl)s1)C c1(C(=O)NC2(CO)CCN(C(=O)CCc3cnco3)C2)ccc2c(c1)COC2 C1(NC(=O)C(F)(F)C2CCCCC2)CCC2(CCN(C(C3CC(F)C3)=O)CC2)C1 CC(C)(CO)CC(=O)NC1CCN1CC(=O)Nc1cc(Cl)cnc1O c1(N(C2CCC2)CCNC(c2cnsc2)=O)ncnc2cc(C3CC3)nn12 Cc1c(C(N2C3CN(C(c4n[nH]cc4I)=O)CC23)=O)ccnc1Cl Cc1ccc(C2CN(C(=O)CCn3cc(C(n4cc(Cl)cn4)(C)C)nn3)C2)c(Cl)n1 c1(C(N2CCC(CNC(C3N(C)CCC3)=O)C2)=O)ccccc1CCC(F)(F)F CCC(CC(=O)NC12CCC(CC1)N(C(c1sc(CO)nc1C)=O)C2)C(F)F CC(C)CC(CNC(=O)CN1CCCNC1=O)NC(C1CCN1S(C)(=O)=O)=O Cc1nc(C(C)C)ncc1C(=O)NCC1CC(C)(C)CN1C(=O)C(F)C(C)C CC(C)CCCOCC(N1CCCC1c1cn(C2COCC2O)nn1)=O C1(N(C(C(C)CF)=O)C)CC2CCC(C1)N2C(=O)CCNC(c1cnccn1)=O Cc1cccc(-c2cn(C(C)C(=O)Nc3csc(CNC(=O)CC(C)(O)CO)n3)nn2)c1 C1(CNC(C2C(CC)CCC2)=O)CC(F)CN1C(=O)CNC(c1ccoc1)=O N1(C(CCCC#C)=O)CC(C(C)(C)C)CC(CNC(=O)C(F)(F)C(O)C2CC2)C1 CCC(CC(=O)NCC1CC(NC(c2cccn3ccnc23)=O)C(O)C1)C(F)F C(=O)(C1=CCCOC1)N1CC(CCCCNC(C2CC3(C2)CC3(F)F)=O)C1 C#Cc1ccc(NC(N2CCC(NC(C3(CC(=O)OC)CCC3)=O)C2)=O)c(C)c1 Cn1nccc1C=CC(N1CCCC1CCCNC(C1C=CCC1)=O)=O N#Cc1cc(Cl)c(C(=O)NC2(C3CN(C(=O)C(O)Cn4cncn4)C3)CC2)s1 CCCC(F)(F)C(=O)NC(C)C(=O)NCCCc1cn(CC)nn1 c1(C(N(C2CCN(C(C3CC(=O)N(C)C3)=O)CC2)CC#C)=O)cc(C)c(Cl)cc1C c1(C(C(=O)NC(C)CN(C(=O)CSC(F)F)C)C)c(F)cccc1F C1(C(N2CC(=CCC)C2)=O)CC=CC(NC(C2CC2(C)COC)=O)C1 CN1CCCC1(C)C1CCN(C(=O)C(=O)NCCC2CN(c3ccccn3)C2)C1 C1(C(N2CC(C(C)NC(=O)CC3(O)CCCN(C)C3)C2)=O)(OCC)CCS(=O)(=O)C1 C(c1ccccc1F)=CC(=O)NC1CC(C)(NC(=O)C(Cl)=CCl)C1 C(C)(C)(CC(=O)N1CCOCC1CNC(c1ccn(C2CC2)c1C)=O)OC N1(C(C2OCCC(NC(=O)CN3CCCCC3)C2)=O)CCC2C(O)CC12 CN1CCC(C(=O)NC2CC(N(C)C(c3csc(CC(F)(F)F)n3)=O)C2)CC1=O c1(NC(C2CC(F)(CF)C2)=O)ccc(F)c(-n2cc(-c3ccccc3)nn2)c1 c1(COC)nc2n(n1)CCCC2NC(=O)NC1CCSC(C)C1 C#CCC(C)(C)C(=O)NCC1(C)CCN(C(=O)CCC(C)(C)O)CC1 c1(C(N2CCC(C(C)(C)NC(C=CCCC=C(C)C)=O)C2)=O)ccc[n+]([O-])c1 N1(C(c2c(N)non2)=O)CC(CNC(=O)CC(F)(F)F)C(O)C1 C1(C(N(C(CNC(c2ccc(C)cc2F)=O)C)C)=O)CC(C2CCCC2)C1 c1(C(=O)NC2(CC=C)CN(C(C3CCCC3O)=O)C2)cccc(CNS(C)(=O)=O)c1 C1(CC(N2C(C(=O)NC(c3ccc(C)s3)C)CC2)=O)CCCC2CC12 c1(CN2CCC(NC(c3sccc3F)=O)C(F)C2)cnc2ccccc2c1 N1(C(c2cc(C(C)(C)C)n[nH]2)=O)CC2CCN(C(C3CCOCC3)=O)CC2C1 CC(CC(=O)N1CCC(C)(C)C1CNC(c1cnn(C)c1Cl)=O)C(F)F C1(C#N)(C(=O)NCC(c2ccccc2)NC(C(N2CCSCC2)C)=O)CC2CC2C1 C1(C(N2CCCC(CCC=C)C2)=O)CCC(C)(C)N(C(C23CCC(CC2)C3)=O)C1 N1(C(Cc2c(C)nsc2)=O)CCC2(CC1)CC2C(N1CCCC(C(C)C)C1)=O N1(C(C2(C=C)CCC2)=O)CCCC(CCC)(NC(c2cnn(C(C)(C)C)c2)=O)C1 N1(C(C2C=C(C)CS2)=O)Cc2n[nH]cc2C1C(=O)N1CC2CCC2C1 C1(C)(CN(CC(C)C)C(=O)NC2CCSC2C)CCCCC1 C1(C(=O)NCCN(C)C)CCCC1NC(c1conc1CNC(N)=O)=O N1(C(c2cc(CNC(c3c(CC)cns3)=O)ncc2)=O)CCc2nn(C)cc2C1 C1(C(N2CCC(N(C(=O)C=C(C)C(F)F)C)C2)=O)CCC(C)(C)CO1 c1(CCNC(N2CC3(CCC(=O)NC3)C2)=O)c[nH]c2cc(Br)cc(F)c12 c1(C(C(C)C)NC(N2CCc3cccc(Br)c3C2)=O)cccc(N=S(C)(C)=O)c1 c1(CC)nccn1C(C)CC(=O)N(CCC(C)NC(C1(C(C)C)CC1)=O)C c1(CC(=O)NCCOCCNC(CC2CC(=C)C2)=O)nc(C)c(C)s1 Cn1nccc1C=CC(N1CCC(CNC(=O)CC2(n3cncn3)CC2)CC1)=O C1(C(=O)NC(C(=O)COC2CC2)CNC(=O)Cn2ccc(C3CC3)n2)CCCOC1 C12(OC(C(C)(CF)CCl)=O)CN(C(=O)OC(=O)OC(C)(C)C)CC1(C(F)(F)F)C2 Cc1cc(C(N2CC3C(CN(C)C(c4ccnn4C4CC4)=O)C3C2)=O)cc(C)n1 C1(C(C(=O)N(C)C)N(C)Cc2cc(C)c(C)s2)Cc2ccccc2C1 c1(CN(CCC(N2CC(Cc3c(C)ccs3)C2)=O)C)ccc(F)c(F)c1 C1(CCNC(c2n(CCOC)ccn2)=O)CN(C(=O)CC2CCCC2)CC1C CCC(C)CC(=O)NC1CCCC1CC(=O)NC1(C(=O)OC)CC(F)(F)C1 Cc1sc(Cl)nc1C(=O)NCCCOCCCNC(C1(C2CCC2)CC1)=O C1(NC(c2cc(C3CC3)no2)=O)CN(C(c2cc(Cl)no2)=O)C2CC12 N1(CC2CCCC(C)O2)C(=O)CCN(C(c2cccc(F)c2Cl)C)C1=O.C1(C)CC1 C1(CC=C)(NC(c2c[nH]ccc2=N)=O)CCN(C(C2(CC)CCCCC2)=O)C1 c1(C(=O)NC2CC(NC(C(c3ccc(Br)cc3)C)=O)C2)cnc(O)n1C Cc1c(-n2nnnc2C(C)C(=O)Oc2cccc(F)c2)cccc1Cl c1(OCC)cc(CN2CCOC(CC(=O)NC3(c4ccsc4)CC3)C2)c(Br)cn1 C1(C(=O)NC(C2CCN(C(C3COC3)=O)CC2)C(C)C)CCC(C)(C)OC1 c1(N2CCCCC(CSC)C2)ccc(S(=O)(=O)NC2CC=CC2)cn1 N1(C(CSCc2nc(C)[nH]n2)=O)CCSCC1CCNC(=O)CC(F)F CCCCC(CNC(=O)C(CC1CC1)OC)NC(C1CCN(CC(F)F)CC1)=O c1(OC)nscc1C(N1CCC1C(=O)NCCOc1ccccn1)=O c1(Oc2ncc(Cl)cc2CN(CCOC)NCC)ccc(Br)cc1[N+](=O)[O-] Cc1nc(O)ccc1C(N1CCC(C(C)NC(=O)C(c2cncn2C)O)C1)=O N1(C(C2(C)CC2)=O)CC2CCC2(CC(N2CCOCC2CC2CC2)=O)C1 CC1(C)CC=C(C(=O)NC2CC3(C2)CC3C(=O)NCC2(O)CC(O)C2)CC1 c1(SC)ccccc1CC(=O)NC(C)(CNC(C1CCNC(=O)C1)=O)C(C)C C1CCN(C(=O)C)CC1.n1(CC=O)nnnc1C.CC Cn1ncc(C(=O)NC2CC(NC(C3CCC3(C)C)=O)C2)c1-n1cccc1 N1(C(COCC(C)C)=O)CCCC(C)C1CNC(=O)CCn1cc[nH]c(=O)c1=O Cc1ccc(C(=O)N(CC(O)CNC(=O)C=CCn2cncn2)C)c(C)c1 c1(OC)ncccc1C(=O)NCCC(O)C(=O)NC1CCC2CC12 CCC(CC)C(C)C(=O)NCC(N1CCN(C(=O)C(C#N)=CC2CC2)CC1)C1CC1 c1(C(=O)NCCC2OCCN(C(CC=C(C)C)=O)C2)ccc(C)cc1O C(=O)(CCCC(C)(C)C)N1CCC(CCNC(C(CCCNC(C)=O)C)=O)C1 C1(C2CC2)(NC(CC=C)=O)CCN(C(=O)CC2CCCC(C)(C)C2)C1 CN1CCOC(C(N2C(C(=O)NCCCS(C)(=O)=O)CC3CC23)=O)C1 C1(C(N2CCCC(CCNC(c3c(OC)c[nH]n3)=O)C2)=O)CC2CCC(C1)O2 C1(=O)CCCC2(CC2)N1.C1(C(NOCC(=O)OC)=O)CC=CCC1 C(=O)(C(C(C)(C)C)C1CC1)N1CCC(N(C(c2cc(OCC)n[nH]2)=O)CCO)C1 C(=O)(CC1=CCCC1)NC(C(c1ccccc1OC)NC(C=CC=CCC)=O)C C1(C)(C(=O)NCC(CC=C)CO)CC(C(C)C)=NO1 N1(C(C=NOC)=O)CCC2CC2(NC(c2ccc(-n3cc(Br)cn3)cc2)=O)CC1 c1(CN2C(C3CCN(C(C4CN(S(CC)(=O)=O)C4)=O)C3)CCC2)nccc(C)n1 C(=O)(C(COC)CC)N(CCCNC(C1(CC=C)CC1)=O)C(C)C c1(C(N(C(C)C)CCn2cccn2)=O)ccc(S(=O)(=O)NCC2=CCCOC2)cc1 N1(C(C2C(C)OCC2)=O)CCC(CNC(c2cccc(C3(C)CC3)c2)=O)C1(C)C C1(C(=O)NCC2CN(C(C(Cc3c(C)nc[nH]3)O)=O)C2)CCc2ncccc2C1 C1(OC)CN2CCCC2(C(=O)NCCC2CCCN(C(=O)C(C)(C)C3CC3)C2)C1 c1(OC)cc(C(C)NCC2CCCCC23CC3)cc([N+](=O)[O-])c1 N1(C(c2c(CC)n(CC)nn2)=O)CCC2CN(C(=O)CNS(=O)(=O)C3CC3)C2C1 N1(C(CC(C)O)=O)CCC2CN(C(c3cn(C)c(=O)nc3O)=O)CCC12 N1(C(C2(CC)COC2)=O)CCC(CF)(NC(=O)C=C2CCCC2)C1 C1(C(N2C(C=C)(c3cn(CCCC)nn3)COCC2)=O)CCCC(C)(C)CC1 C1(COCC#C)COCCN1C.C(CCC(=O)NCC1CC1CNC=O)O Cc1ccc(F)cc1C(N1CCC(O)(CNC(c2cnc(Cl)[nH]2)=O)C1)=O n1(CC(=O)NC2C3CC2CN(C(=O)CCc2nccs2)C3)nc2c(n1)CCCC2 N1(C(CCn2ncc(C)c2)=O)CCC2CCC(NC(C3CC=CCO3)=O)C12 C(CCCCC(=O)NC1CCCCC1CNC(C1CC(O)C1)=O)N(C)C Cc1cc(C(N2CCC(NC(c3cccc(Cl)c3)=O)C2(C)C)=O)c(C)c(C)c1 c1(C(=O)NC2C(NC(CCOCC#C)=O)CC2)ccc(C(C)C)nc1O Cc1cc(C)nc(CC(=O)NCC(O)CNC(=O)CC(c2c(C)noc2C)C)n1 Cc1ccccc1-c1nnn(CC(=O)Oc2ccsc2)n1 Cc1cc(C#N)c[nH]c1=NC1CN(C(=O)Cc2cccc(F)c2)C1 C1(NC(CCCC(=O)NCC(C)(C)N(C)C)=O)CCc2c(nnn2C)C1 N1(C(C=Cc2n(C)ncc2)=O)CCC2(CC1)CC2C(=O)NC1CCCCCC1F C12(C(=O)NCC3(O)CCN(C(=O)CC4(O)CCC4)CC3)CCC(CO)(CC1)CC2 CC(C(=O)NC1CC(CNC(C2(C#N)CCOCC2)=O)CC1O)S(N)(=O)=O c1(CC)ccc(C(=O)NCC2CCCCC2NC(=O)C(F)(F)C2CC2)cc1F C1(NC(C23C(CN(C(C4CC(OCC)C4)=O)C2)CC3)=O)CC(CO)C12CCC2 C(C(C(=O)N1CCCCC1CC(N)=O)C(C)C)NC(C=C(CC)CC)=O C1(C)C(=O)N1.C(CC1CC1)(CO)NC(COCCCC)=O N12CC(CC1=O)C(=O)NC2.C1(C)(N(C)C)CC(NC(=O)CCC2CC2CC2CC2)C1 C(=O)(C(C)(COC)CC)N1CCC(N(CCC)C(C2CC2c2ccnn2C)=O)C1 Cc1cc(C2(NC(C3CC(NC(c4cn(CCOC)cn4)=O)C3)=O)CCC2)no1 CC1CN(C(c2ccc(O)c(OC(F)(F)F)c2)=O)CCN1C(=O)C(O)C(C)(C)C C1(CCC)CN(C(=O)CN(CC(=O)OC)C)CC1C(=O)NCC1CC1F c1(C(c2n(CC)ncn2)=O)ccc(Cl)cc1.C(=O)(CCC1CCCO1)N c1(CC(=O)N(CC(CNC(CN(C)CC)=O)C)C)cnn(C)c1C c1(C(N2CCOCC(CNC(CCC#C)=O)C2)=O)ccc(S(=O)(=O)C(C)C)cc1 c1(C(=O)NC(C(C)C)CNC(C2(F)CC2C)=O)ccc(=O)n(CCF)n1 c1(C(N2C(CN(C(C(C)=C3CCC3)=O)C)CCC2)=O)cc(Br)nn1C N1(C(C(COCC)NC(=O)CCCC(=O)N(C)C)=O)CCCC(O)(C2CC2)C1 c1(CC(=O)NC2CC(C)(NC(Cc3n(C)ccn3)=O)C2)cccc2nsnc12 C1(C(=O)NC(CC)C(C)(F)F)CN(C(c2sccc2CO)=O)CC(C)(C)C1 C1(NC(c2c(C)nc(Cc3nncs3)s2)=O)CC2CCC1N(C(=O)C(C)(C)F)C2 CCC(CC)(CO)C(=O)N1CCC(NC(C2CCOCC23CCC3)=O)CC1 C(=O)(C(C(C)O)NC(C1CCCCC1O)=O)NCCC(=O)OCC C1(CN2CC(NC(C3CCOCC3CO)=O)C2)Cc2ccccc2CCO1 C1(CN(C)C(C2CCN2C)=O)CCCN1C(=O)C=CC1(C)COC1 N1(C(c2c(CC#N)ccs2)=O)CCCCC1C1CCN(C(C2(O)CCC2)=O)C1 C1(C(=O)NC2CCC(C(N3CCC(O)(CC)C3)=O)C2)(CC)CCNC1=O C1(C2CCCN(C(c3c[nH]ccc3=O)=O)C2)(NC(c2c(F)ccnc2F)=O)CC1 CCC(C)(CCC(C)C)C(=O)NCCC1(NC(=O)C(F)C2CCC2)CCCC1 C1(C(C)(C)NC(C(c2ccn(C)n2)C)=O)CCN(C(=O)CO)C1 c1(CNC(C2CC(NCc3ccc(C)c(Br)c3)C2)=O)n[nH]c2c1CCCC2 C(CCNC(=O)C=Cc1cccnc1)(C(=O)NC1CC1C(C)C)OC C1(C(=O)NCC2(NC(C(C)N(C)C)=O)CC2)CCCN1CC1CCCO1 CC1(CCNC(C2CCC(NC(c3cccc(O)n3)=O)C2)=O)CCOCC1 N#Cc1c(N2CC(CNC(c3cnc(S)n3C3CC3)=O)C2)nnc2c1CCCC2 c1(C(N2CCCC(NC(c3cn(CC=C)nc3)=O)C2C)=O)nccn2nccc12 c1(C(=O)NCCC(C(=O)NCc2cc(C)ns2)OC)c[nH]c2cccnc12 c1(C(=O)NC(CNC(CCN(C)CC)=O)(C)CO)cc(C)n(C)n1 c1(C(=O)NC(C)CN(C(=O)COc2cncc(Cl)n2)C)c(Cl)oc2ccccc12 C1(C(=O)NC2(CC#C)CCCCC2)CCN(C(c2cc(=O)cc(C)[nH]2)=O)CCO1 N1(C(C(CC#C)C)=O)CCCC2CN(C(=O)CCS(C)=O)CC12 c1(C(CCOC(=O)C2CC2)NCC=C(C)C)ccc(O)cc1 C(CC1CCOCC1)(C(=O)N1CC(C#N)C1)NC(C(C)N(CC)CC)=O N1(C(c2c(N)cn(C)n2)=O)CCC2(CCCN(C(=O)C(F)CC3CCC3)C2)C1 c1(C(=O)NC2CCC(CNC(C=CS(C)=O)=O)CC2)cccc2nc[nH]c12 c1(C(=O)NCC2(OC)CCN(C(c3csc(C)c3C)=O)C2)cnccc1C#N N1(c2ncnc(C)c2F)CCCC(C)(C)C1CNC(=O)CCc1ccn(C)n1 Cc1ccccc1COCC(=O)NCC1(NC(=O)CCC(C)C2CC2)CC1 C1(C(N(C2C3CN(C(c4cncn4C)=O)CC23)C)=O)CN2CCN1CC2 Clc1ccc2c(c1)CN(c1nccc(N3CCC(OCCF)C3)n1)CCN2 C(=O)(C(C)(C)C(F)(F)F)NC1CCN(C(c2cc(CCCCC)on2)=O)C1C C(=O)(C(COC)N(C)C)NC(C1CCOC1=O)C(=O)N(CC#C)CC1CC1 C(=O)(C1CC(=O)c2ccccc21)NC1C(SC)CN(C(=O)Cn2ncnn2)C1 c1(NC(N2C(CC(=O)NCCOC)C(=O)NCC2)=O)cncc2ccc(F)cc12 N1(C(C(CCC(N)=O)n2cc(CCN(C)CC)nn2)=O)Cc2cccc(C)c2C1 N1(CCC(=O)N(CCCN2CCCC2=O)CCOC)CCP(C)(=O)CC1.C(CSC)N N1(C(=O)NCC)CCN(CCOCC)CC1.C1(c2nnnn2CC)(NCC)CCC(C)S1 C#Cc1cncc(C(N2CCC(NC(c3cnccn3)=O)C2C)=O)c1 Cn1cnn(CCC(=O)NCCOCCNC(c2conc2C(F)(F)F)=O)c1=O C1(C(=O)NC2C(C)CN(C(c3cc(Cl)c(Br)s3)=O)C2)CCc2ccccc2O1 C1(NC(c2sccc2SC(F)F)=O)CC2CC(C1)N(C(=O)C=CC(F)(F)F)C2 CCC(CC(C)C)C(=O)N(CCNC(c1ccnc2cc[nH]c12)=O)C1CC1 C(=O)(CCC(C)(C)F)NCC(C)CC(=O)N1CCOC(CCF)C1 C1(CNC(c2c(C)nc(C)s2)=O)C2CCC(C2)N1C(=O)CNC(=O)CN(C)C CC(CC(=O)N1CC(CNC(C2(CC(F)F)CC2)=O)OC(C)(C)C1)CC(F)(F)F CS(=O)(=O)c1ccc2c(c1)CN(C(=O)C=C1CCSCC1)CC2 C1(COC(C2CC(=O)N(c3ccccc3Br)C2)=O)CCc2ccccc2C1 CCC(C)(O)C(=O)NC(C)CCCNC(=O)C(F)(F)Cc1ccc(Br)cc1 c1(C(N(C)Cc2nn(C)c(C3CC3)n2)=O)cnc(O)c(Br)c1 N1(C(CCSCCC)=O)CCS(=O)(=O)C(CCNC(c2cnn[nH]2)=O)C1 C(CCC(C)C)(C(=O)N1CCC12CCC2)NC(C1ON=C(CC)C1)=O C1(C(N(C(C)CCNC(=O)OC(C)(C)C)C)=O)CC(c2cnn(C)c2)=NO1 N1(C(C2C(OC(C)=O)C2)=O)CCC(C(C)NC(=O)Cn2nnc(=N)[nH]2)CC1 C1(CNC(c2c(CC)nn[nH]2)=O)CCC(C)N(C(c2cc(C(F)F)ncn2)=O)C1 C1(CC)CCN(C(=O)CC(O)CN(C)C)C(C(=O)NCC=Cc2ccoc2)C1 c1(SCC2(C(=O)NC3CCCN(C(c4nnc(C)s4)=O)C3)CC2)cc(F)ccc1C C(C)(C(N=c1ccnc[nH]1)C(C)C)NC(CCn1c(C)cc(C)n1)=O N1(C(c2ccsn2)=O)CCC(n2cccn2)(CNC(C23CSC(C2)C3)=O)CC1 C1(CN(C(C2(CCOC)CC2)=O)CC)CCN(C(C2CC(F)C(=O)N2)=O)CC1 N1(C(C2(CC=C)CCCC2)=O)CCN(C(C2CC23CCC3)=O)CC1 Cc1nc2ccccn2c1C(=O)NCCC1(NC(c2cccc(=S)n2O)=O)CC1 c1(C(N2CC(O)C(F)C2)=O)ncccc1NC(=O)CC1CCNC(=O)C1 CCC(C)(C(=O)NCC(C)CNC(=O)CCNC(N)=O)C(N)=O CCC(C)CC(C(=O)N(C)CC1(C#N)CC1)NC(=O)C(=O)NCC(F)F C(=O)(CCCCCF)NC(C1CCN(C(=O)C(C)(O)c2cscn2)C1)C c1(OC)cc(C(=O)NCCC2CC(NC(C3CCCO3)=O)C2)c2ccccc2n1 N1(C(c2n(CC)ccc2)=O)CCC(C(=O)NC2CCCC2CN(C)C)C(C)(C)C1 C1(C(=O)NCC2C(NC(c3c(CC)noc3)=O)COC2)CN(C)CCC1O N1(C(Cc2cc(C)on2)=O)CCC(NC(=O)C(=O)N(C)C)C(CO)C1.C1C(=O)N1 C(=O)(C1=CCN(C(=O)C#CC2CCOC2)CC1)N1CCC(CN(C)C)C1 c1(C(=O)OC)cc(S(=O)(=O)NCC2CC2)c(F)cc1Br Cn1cc(C(=O)OCc2ccc(C#N)[nH]2)c(C2CC2)n1 N1(C(c2cc(C)cc(C)c2N)=O)CCN(C(=O)Cc2cscn2)CC(C)(F)C1 Cc1cn2nc(C(N3CC(C(C)NC(C4CCCC4)=O)C3)=O)cc2c(=O)[nH]1 N1(C(C(C)OCCC#C)=O)CC(NC(c2cccc(C)c2Cl)=O)CC12CCC2 C(=O)(CC(C(F)(F)F)c1ccon1)NCC1N(C(c2cc(C)[nH]n2)=O)CC=C1 c1(C(=O)NC2(C)CN(C(CN(C3CC(C)(C)C3)C)=O)C2)cc(C2CC2)ccn1 C12(NC(C3(OC)CCSC3)=O)CC(CNc3ccnc(SC)n3)(C1)OC2C CC(C)(C)C(O)C(=O)N1CCCC(CNC(C2CCCC2O)=O)CC1 c1(SCC(=O)N(C2CCC(NC(=O)CCc3ccco3)C2)C)ccccc1Cl C1(C(N2CCOC(C3CCC3)C2)=O)(NC(CN(C2CCC2)C)=O)CCC(C)(C)C1 Cc1ccc(CN(C(c2ncc(Br)s2)C(=O)NCC2CC2)C)s1 c1(C(=O)NCCNC(C2C(CC)CCN2C(C)=O)=O)nc(C)c(C)[nH]c1=O Cc1sc2ccccc2c1C(N1CC2CC(NC(=O)CC3CCC3(C)C)C1C2)=O c1(C(=O)NCCCCNC(C2C(C(C)C)(CC)C2)=O)ccc(OC)c(F)c1F c1(C(C)C)cc(N2CC(NC(=O)C(C)OCc3ccncc3)CC2C)nc(Cl)n1 N1(C(C(CO)NC(c2ccc(O)cn2)=O)=O)CC2CCC(O)CC2C1 c1(OC)ccc(C(C)NC(=O)NCC2(C(=O)OC(C)(C)C)COC2)nc1 c1(CC(=O)N(CCCNC(C2N(OCC)CCOC2)=O)CC)cnc2ncccn12 c1(OC)nc(C)ccc1C(=O)NC(C1CCCN(Cc2c(C)noc2Cl)C1)C C1(NC(c2cn(CC(C)C)nn2)=O)CCC(C)(CNC(=O)COCC(F)F)C1 C1(C(N(C2CCN(C(C(CC=CC)C)=O)CC2)CC)=O)CCc2ncccc2C1 C(=O)(C1CCC(=O)c2ccccc21)N(CCNC(c1cccc(=S)n1O)=O)CC c1(C(=O)NCC(N2CC3CNC(=O)C3C2)=O)c(F)ccc(I)c1Br C(=O)(C(C)C(C)(C)C)N1CC(NC(c2cc(C(=O)OC)[nH]c2)=O)C(C)C1 c12cc(Br)c(nc1C)N(CC)CCNC2=O.C(=O)(CNC(=O)NC)N c1(CC(=O)OC)ccccc1NCC(c1cc[nH]n1)OC c1(SC)ccc(C)c(C(N2CC(CNC(=O)C(C)SC(F)(F)F)C(C)C2)=O)c1 c1(SCC)cc(C(=O)NCCn2cc(CNC(=O)C(C)C3CC3)nn2)on1 CCC(C)(C(=O)O)NC(=O)C(F)CC1CC1 C(=O)(CCCN(C)C(C)C)NOCC(C)(C)C.C12(CCC1)C(=O)N(CCC)CCCC2.N.O N1(C(CSCC#C)=O)CCCN(C(c2ccc(Cl)nc2OC)=O)C(C(C)C)C1 C1(CC)CN(C(=O)COCCF)CCN1C(=O)CCc1cn(C)nn1 c1(C(N2C(CNC(c3c(C)nc(CC)o3)=O)CC2)=O)cc(OC)cc(Cl)c1OC c1(CC(N2CCC(NC(C(C)SC)=O)C2C2CC2)=O)cc(Cl)cnc1C n1(CC)ccc(CNC(c2ccoc2CNC(=O)C=CC2CCC2)=O)n1 c1(C(=O)NC2C(CC)C2)sc(C2CCCC2)nc1C(F)(F)F.C12CC(C1)C(=O)N2 c1(CNC(C2COCCC2NC(=O)CCC2CCOCC2)=O)cccnc1F C1(CNC(C2OCCN(C(C)=O)C2)=O)CC2CCC(C1)N2C(=O)C=CS(C)=O N1(C(CC(=O)NCC)=O)CCC(NC(=O)CCC23CCC(CC2)C3)C(CC)C1 c1(Cn2cc(C(C)Nc3cc(OC)cc(C)n3)nn2)cccc2c1OCCO2 c1(C(=O)NC2C(NC(=O)C3=CCCS3)COCC2)cc2c(s1)COCC2 c1(C(=O)NC2C3CC(NC(C(C=C)OC)=O)CC32)ccc(S(C)=O)cc1 C=CCC(C(=O)NCC1CC(C(=O)NC(C)CS(C)(=O)=O)C1)OC C(CC1CCC1)(C(=O)NC1(CNC(c2cc(CO)on2)=O)CC1)OC C1(C(=O)NC2C(NC(c3c(OC)n[nH]c3)=O)COCC2)CC(F)(F)CS1(=O)=O c1(C(C)(C)C(=O)Nc2ncc(CCN3CCCC3)s2)cccc(N=S(C)(C)=O)c1 C(=O)(C(C(C)(C)C)n1ccnn1)N(CCOC)CCNC(=O)C=CC(=O)NC Cc1ccc2[nH]cc(CN=C(NCc3ncnn3C)NC3CCCC3)c2c1 C1(C(=O)NCCN(C(=O)Cc2cnccn2)CC2CC2)Cc2ccccc2CO1 N1(C(c2ncn(CC)n2)=O)CC(O)CC1CNC(c1coc(C(C)C)n1)=O c1(C(=O)NC2(CCCNC(C(CC)O)=O)CC2)cn2cc(C)nc2s1 N1(C(C2OCCOC2C)=O)CCCCC1C1CC1=O.n1(CCCNCC)cncn1 N1(C(CCC)=O)CC2OCC(NC(c3sc(N4C=NC=CC=C4)nc3C)=O)C2C1 N1(C(C(C)(C(C)C)OC)=O)CCC2(C1)CN(C(C1(N=[N+]=[N-])CC1)=O)CC(C)O2 N1(CC(COC)O)CC2CCC(NC(c3n[nH]c4c3CCCCC4)=O)CC2C1 C(C1CCN(C(=O)CC2C=CCCC2)CC1)=CC(=O)NC1CC(CSC)C1 C(N=c1nc(CC(F)(F)F)[nH]s1)C1CCCN(C(C(CC)N(C(N)=O)CC)=O)C1 c1(SC)ccc(CC(=O)NCC2CC2NC(C2CCC2)=O)cc1 c1(NCC2CC(NC(c3cnc(C)nc3O)=O)C2)ncnn2c(Br)ccc12 CCCC(C)(C(=O)OCC)NC(c1ccccc1)=O.C1(=O)CCCO1 c1(C(N2CC(NC(CC(CC)C3CC3)=O)C(F)C2)=O)cccc(C#N)c1 c1(C(=O)NC2(CC)CN(C(COCC)=O)C2)c(C(C)(C)C)nc2n1CCCC2 c1(NC2CC3(C(NC(CSCc4cccc(C)c4)=O)C3)C2)cccc2c1CCC2 c1(C(=O)OC)ccc(C(F)(F)F)c(O)n1.C12CC(C1)C(=O)NC1CC1CNC(=O)C2 c1(C(=O)NCCCNC(CCNC(=O)OCC)=O)ccc(S(=O)(=O)CF)cc1 N1(C(=O)Cn2cnc(C(F)(F)F)n2)CCCC2(C1)CN(C(c1ccncn1)=O)C2 CC1(C(=O)NC2CC(CNC(=O)C(c3cccs3)C3CC3)C2)CC1(Cl)Cl C(N=c1nc(N2CC(C)(C)OC(C)(C)C2)cc(C)[nH]1)c1ccn(CCC)n1 C(=O)(CCCC(CC)NC(=O)C(O)C1CCC1)NCCCOCC=C C12(NC(Cc3cnc(C)s3)=O)CCCC1N(Cc1ncc3ccccn13)CC2 C1(NC(=O)C(F)(F)c2cncs2)CCC2CCN(C(c3cnsn3)=O)C1C2 n1(CCC#C)c(N(CCO)CC2CCC2)nnc1C1CCC1 CCC(C(F)(F)F)NC(=O)C(CCOC)NC(=O)CC1CC2C=CC1C2 C(=O)(CC(C)(C)C(F)F)NCC(C(=O)N(C)CCN1CCCC1)O C1(C(N(CC)CC2CCCC2O)=O)C(CNC(=O)C(=O)NC2CC2)C1(C)C CCC(C)(CCNC(=O)Cn1cnnc1)NC(C1CCCOC1C)=O N1(C(c2cccc(C3CC3(F)F)c2)=O)CC2(CCN2C(=O)CSc2cccs2)C1 C1(NC(c2cc(C3CC3)no2)=O)CS(=O)(=O)CC1NC(c1cc(Cl)cnn1)=O Cc1occc1CC(=O)NC(C)(C)C1(NC(=O)Cn2cc(C3CC3)nn2)CC1 CC1CCCCC1(C)n1cc(CCC2CN(C(c3cc([N+](=O)[O-])n[nH]3)=O)C2)nn1 c1(CC)nc(N2CC(COC)(NC(C3(C(N)=O)CC3)=O)C2)c2ccsc2n1 CC(C)(C)C(=O)NCCC1CN(C(=O)CCc2ccccc2)C1.c12nc(cs1)C2 C1(CCNC(c2cnc(COC)s2)=O)CC2CCC(C1)N2C(C1CC=CCC1)=O C(=O)(CC(C(F)(F)F)OC)N1CC(CC)(NC(c2ccn(C(C)C)n2)=O)C1 c1(CC(N2C(CC3CCC3)CC2)=O)ccnn1C(=O)NCC1(CC)CCC1 c1(C(=O)NC(CC)CNC(c2cnc(C(C)(C)C)s2)=O)cc(Cl)c(F)c(Cl)c1 CCCCCCCCCCC(=O)N1CCC(NC(C23CCCCC2C3)=O)C1(C)C c1(C(=O)NC2C3CN(C(C(CCCOC)C)=O)C2CC3)ccc2c(c1)NC(=O)C2 C#CCC(C)(C(=O)NCC(O)C=C)NC(=O)CNC(=O)NC1CC1C C1(C(=O)NCCCCC#CC)N(C(=O)COC2CCOCC2)CC12CCCC2 CC(CCN(C)C)C(=O)N(C(C)CN(C(=O)COC(F)(F)F)C)C C1(c2ccc(F)cc2)(NC(=O)CCOC2CC2)CCN(C(C2CC2F)=O)CC1 c1(C(=O)NCC=CCNC(c2cc(C(C)C)on2)=O)oc(Br)nc1C(F)F C12(N(C(C(=O)NCC)=O)CC(F)F)CC1CN(C(c1cn(C3CC3)nn1)=O)C2 C1(C(=O)NCC(CN(C)C(C2C3(CC3)C23CC3)=O)(C)C)C2CCC(C2)S1(=O)=O C1(CCNC(C2CCC(=O)N2)=O)CC(F)(F)CN1C(=O)CSC1CC1 c1(C(=O)NC2CN(C(c3c(C)nnn3C)=O)CC2O)coc(S(N)(=O)=O)c1 Cc1ccc(CCCCC(=O)NC2CCC2NC(=O)Cn2nc(C)nc2C)cc1 C#Cc1ccc(Cl)c(N(CCC#N)C(=O)NCC(=O)Nc2cccs2)c1 C1(CNC(c2ncc[nH]2)=O)C=CCN1C(=O)CCCc1cc[nH]n1 O=C(N=c1[nH][nH]cc1C(N1C2CCC1CC2)=O)c1ccc(C2CC2)cc1F c1(C2(CC(C3CC3)Oc3cccc(CC)c3)CC2)ccc(Cl)cc1Cl Cc1cc(C(N2CCC(NC(C3CCOC3C)=O)C(C)(C)C2)=O)cc(N)c1O c1(C(c2nnnn2C2CC(NCC)C2)NC(C2CCCCO2)CC)sccc1Cl N1(C(C(C2CCC2)NC(CC2C(C)=NNC2=O)=O)=O)CC2(C1)CC(C)(O)C2 CC1CN(C)CC(C(N2CCCC2C2(NC(C3COC(C)(C)CO3)=O)CC2)=O)O1 C1(C(CC)C)CCCN1C(=O)C=CCN(C(=O)CSc1nc[nH]n1)C C(=O)(C(C(C)(C)C)N(C)C)N1CCC(NC(c2c(Cl)nc(N(C)C)s2)=O)C1C1CC1 C12CC(C)(C)CN1C2=O.C(C)(C)(CCNC)NC(COCCC=C)=O c1(C(=O)NC(C)(CNC(=O)C(F)(F)C(O)C2CC2)C2CC2)ccc2ncnn2c1 CC1(C)CNC(=O)C1NC(=O)CC1CCCCN1C(=O)CC1CSC1 c1(C(=O)O)cc(CN2CC3(CC3)CC2C(N2CCOCC2CO)=O)ccc1O C1(NC(C(CC)c2ccccc2)=O)CC(C)N(C(C2CC(=O)N(C)C2)=O)C1 CC(CC(=O)NC(C)(C(=O)N(C)CCc1ccccc1)C1CCC1)C1CCCO1 C1(NC(CC2C(C)(C)C(O)C2)=O)CN(C(c2cc(Cl)ccc2F)=O)CC1C#N c1(C(=O)NCC(C)NC(C(CC=CC)C)=O)ccc(N)cc1Br n1(CC)ccc(C(=O)NCC2CC3CCC2N3C(=O)CC2CSCCS2)cc1=O C12(C(=O)NCC(CN(C(C3CCC(=C)CC3)=O)C)C)CCC(CC1)OC2 c1(N(c2cnc(C(=O)NC3(COC)COC3)nc2)C)cc(C#N)ncn1 C(=O)(CC(F)(F)C(F)(F)F)NCC12OCC(NC(CSCC#C)=O)C(C1)C2 Cc1cc2c(C)n1C1C(N(C)C(C3(CO)CC3)=O)CCN(C1)C2=O.C1(CF)CC1 CN1CCN(C(c2ncnn2C)C(=O)NCC2CCCO2)C(c2nn[nH]n2)C1 C(=O)(C1=CCC(C)CC1)N1CCCC(C)(NC(c2nncc(CCC)c2)=O)C1 c1(NCc2c(Br)ccc(C)c2)ccc(S(=O)(=O)NCCCCF)cc1Br CN(C)S(=O)(=O)N1CC(C(=O)NCCNC(C2CCCC(O)C2)=O)C1 C1(CC(=O)NCC2CCN(C(c3nc(CC)[nH]n3)=O)CC2C)CC2(CCCC2)CO1 C1(NC(Cn2cc(C(C)=O)nn2)=O)CCCC(NC(C2CC(=O)N(O)C2)=O)C1 C1(CCN(CCOCCN(C(C)=O)C)C)CC2CCC1C2.c12nccc(n1)NC2 C1(NC(CNC(C)=O)=O)CCN(C(=O)C(c2ccccc2F)C)C1C N1(CC)CCCCC1C(=O)NCC=CCNC(=O)C(F)CC1CCCC1 C1(CNC(CC(=O)NCC)=O)CC(COC)CN1C(C1CC12CCC2)=O C(=O)(C(CO)C(C)(C)C)NC(COC(C)C)C(=O)NCC1CC1 C(=O)(C(F)(F)c1nccs1)N(C1CN(C(C2CCN2C2CCCC2)=O)C1)C c1(C(=O)NC(CNC(C2C(C(=O)NCC#C)C2)=O)(C)C2CCC2)cc(C#N)on1 Cc1nc(C(N2CCC(C(C)(C)NC(C3CCCC3C)=O)C2)=O)c2ccccn12 N1(C(C(CN(C)C)(C)C)=O)CC2CC(NC(c3cnn4c3NCCC4)=O)CC2C1 c1(OC)cc(C(=O)N(CCCN(C)C(C2(C)CC2F)=O)C)ccc1Cl c1(OC)ccc(C(C2C(C#C)(C(=O)NC(C)CNC(=O)CC3CC3)C2)=O)c(C)c1 CC(N=c1cc(NCC(C)CN(C)C)nc(C(F)(F)F)[nH]1)c1nccn1C O(P(C)(=O)CCOC)C(C1C(=O)CC1C(F)(F)F)=O c1(-n2cc(C3(NC)CCN(C(=O)C(C)OC)C3)nn2)cc(F)c(F)cc1Cl C=CCC(CC(C)C)C(=O)N1CCCN(C(c2cnncc2C)=O)CC1C c1(CC2N(C(NC3CCc4ccccc43)=O)CCOC2)c[nH]c2ccc(F)cc12 C12(C(=O)NC(CCNC(C=CCC)=O)(C)C)CCCN(C1)S(=O)(=O)C2 C1(CNC(C2N(CCC)CCC2)=O)CN(C(c2ccncc2Cl)=O)CC1(F)F CC1(C(N2CCC(C#N)(CNC(=O)OC(C)(C)C)CC2)=O)CCCNC1=O Cc1cc(C(=O)N(CCCOCCN(C(=O)CC(C)(C)F)C)C)ncc1C(F)F C1(C(N2CCC(OC)(CNC(=O)Cc3cn[nH]c3)C2)=O)CCCCC12CCC2 c1(C(=O)NCCCCNC(c2cc(C3CC3)ns2)=O)cc(Cl)ccc1Cl c1(C(N2C(C(N3CC4CC4C3)=O)CC(C)C2)=O)cn2cccc(Br)c2n1 N1(C(CCCOCC(=C)C)=O)CCC(CC(=O)N(C(C)CO)C2CC2)C1(C)C c1(SC(CC)C(=O)NC(C)(C)C)cc(C(=O)O)cc(C(F)(F)F)c1 N1(C(c2c(CCC)n[nH]c2)=O)CCC2(CC1)COC(CNC(=O)CSC(C)C)C2 C(CCCC(CO)NC(C1CC12CC2)=O)NC(c1c(CC)nc(C)s1)=O C1(CCCNC(=O)C=CCF)CCCCN1C(C1CC(n2cnnc2)C1)=O c1(-c2n(N(CC)C)ccn2)cc(C)nc(N2CC(CO)(CO)C2)n1 Cn1ccc2[nH]c(C(=O)N(CCCNC(C3CC3F)=O)C)cc12 N1(C(C(C)N(C(=O)CCNC(=O)COC)CCC)=O)CCn2ccnc21 C1(NC(CC2(C)CCC2)=O)CCCCC1NC(=O)C=Cc1cc[nH]c1 Cc1cc(C)cc(S(=O)(=O)NC2CCCN(Cc3cncc(Cl)c3)C2)c1 Cc1ccc(C2CC2C(=O)NC2CCCN(C(C3C4(CC4)C34CC4)=O)CC2)c(Cl)n1 CCCCCCC(C)(C)C(=O)N(C)CCOCCO.C12CCN1CC(=O)NC2 C1(C(=O)NC2CCN(C(C)=O)C2)CCCCC1CNC(=O)CSCC(C)C C(=O)(C1=CNC2=NCCC2=C1)NC1CC(C)CN(C(c2ccc(CO)s2)=O)C1 c1(CCC(=O)C2CC2)nc(NCC2CC2NC(=O)CCOC2CC2)no1 C12(CCCCC1)C(=O)N2.C1(F)(CN(C)C)CC(NC(c2cc(Br)co2)=O)C1 c1(OC)cc(C(F)(F)F)ccc1CNC(=O)NCc1cc(O)cc(O)c1 C(=O)(CC1=CCN(C)CC1)NC1CC2(CN(C(c3ccc(OC)nc3)=O)C2)OC1 n1(CC(=O)NCCN(C(=O)CCC(=O)OC)CCOC)nc(C(F)(F)F)cc1C N1(C(C(C)OCCC=C)=O)C2CCC1C(NC(C1CCC(CC)CC1)=O)C2 N1(C(CC2C3CN(C(C(C(CC)O)C)=O)CC32)=O)CC(C)OC2(CCC2)C1 c1(C(N(C)CCOCCNC(C2CCCSC2)=O)=O)ccnc2c1ncn2C C(CN=c1[nH]c(=NCCCC(=O)NC)c2ccccc2[nH]1)SCCNC(CC)=O c1(NC(C2C(C(=O)Nc3c(C(=O)OC)cccc3O)C2)=O)cc(C)cc2[nH]ncc12 c1(OC)cc(C(=O)NC(c2ccccc2)CNC(C2C=CCC2)=O)n(C)n1 CC(CCC(=O)NCc1cn[nH]c1)NC(=O)C(O)CN1CCCC1 C1(C(C)N(C(C2CC3CC3C2)=O)CCO)CCCN(C(=O)CCN(S(C)(=O)=O)C)C1 C1(CN=c2nc(SC)[nH]s2)CC2CCCC(C1)N2C(C1(CO)CC(C)(C)C1)=O Cc1nnc2c(C(=O)NCCC(F)(F)CC(=O)O)cccn12 c1(CNC(=O)Nc2ccc(C(C)O)cc2)ncc([N+](=O)[O-])o1 N1(C(C2C(CC)N(C(c3ncn(C)n3)=O)CC2)=O)CC(C)C(C)C1C CS(=N)(=O)C1CC(NC(=O)C(O)C2(N)CC2)C1 c1(C(C)C)nnc(C=CC(=O)NC2C=CCN(C(C3CC4CCC3O4)=O)C2)o1 S1(=O)(=O)c2ccc(nc2)N1C.Cc1cccc(CNC2CCC3CC23)c1 C1(OC)CN(C(c2cccc(C#N)c2)=O)CCC1NC(=O)CC1CCC(C)(C)C1 C1(C)(C(N(C2CCN(c3nnnn3C)CC2)C)=O)CCCC1(F)F C1(C(=O)NCC2CCCC23CC3)CC2CCC(C1)N2C(=O)C1=C(Cl)CCCC1 CC(CC(N)=O)C(=O)N1CC(C)C1C(=O)NCCC1CCC(C)(C)C1 c1(C(=O)NC(CCNC(C2C(C#C)C2(C)C)=O)C)cc2c(nc1O)CCCC2=O C(CCCCC(=O)NC1CCOC1=O)N(C(=O)CC1CC(=O)NC1=O)C N1(C(C(CC=C)C)=O)CCCCC12CC(NC(c1cc[nH]c(=N)c1)=O)C2 c1(C(=O)NC2COCCN(C(C(c3nc(C)sc3)=O)=O)C2)ccc(N)c(C)c1C c1(CC(C)C(N2CC(NC(=O)CN(C)C)C(CC3CC3)C2)=O)ccc(F)cc1F C(=O)(C1CCCc2nc[nH]c21)NCC(CNC(c1cc(OC)ncc1)=O)F c1(CC)nc2n(n1)CC(C(=O)NC)CC2.N12CC(C1)C(OC)C2=O c1(OCC(N2CCC(O)(C3(C(=O)NCC4CCC4)CC3)C2)=O)cccc(Cl)c1Cl C1(O)(Nc2cccc(CCC)c2)CCN(c2ncc(C)c(OC)n2)CC1 C1(NC(C(CC)NC(N)=O)=O)CC2CCC1CN(C(c1ccc(F)c(NC)c1)=O)C2 C12(CCCC1)c1cn(nn1)CCCNC2=O.C(C(N)=O)N(C)C c1(C(N2CCN(C(C3CN(C(C)=O)C3)=O)C(CF)C2)=O)ccc2c(n1)CCOC2 c1(N2CC(CCCCC(C=C(CC)CC)=O)C2)nc(C)ccc1C#N.N c1(C(=O)NCCC2CN(C(CCCC)=O)C2)ccc(F)c(C(C)(C)C)c1 Cn1nnc2c1CCN(CC13OCC(C(=O)NC4CCC5(CCC5)O4)(C1)C3)C2 N1(C(=O)CC2CC2(Cl)Cl)CCN(CCNC(C2(O)CCC2)=O)CC1 c1(C(N2C(CCC)CN(C(=O)C(CC)OC)CC2)=O)c(N)cccc1[N+](=O)[O-] c1(OC)cccc(Br)c1CN1CCC(OC(c2cnn(C(C)C)c2C)=O)CC1 N1(C(C2(C(=O)OC)CC2C)=O)CC2(COC(CNC(c3ccc(O)nc3)=O)C2)C1 Cn1nccc1C=CC(=O)NCC1CCN1C(C1CCC2CC12)=O Cc1nc(C2CCOC2)sc1C(=O)NC(C1CCN(C(=O)C(=O)NC2CC2)C1)C C(c1c(C)coc1C)=CC(=O)NC(CC)CN(C(=O)C=Cc1csc(C)n1)C C1(CC)CC(O)CN1C(c1cc(C2CC2)on1)C(=O)NCCc1ccccc1Br N1(C(N2C(C)Cc3cnccc32)=O)c2ccccc2C(NC2CC2)C1(C)C N1(C(COCC)=O)CC(C2CCCN(C(c3coc4c(F)cc(F)cc34)=O)C2)C1 c1(C(=O)NCCCN(C(c2noc(CC)c2C)=O)C)cc2ncccc2o1 C(=O)(CC(CN)C(F)F)NCC(C(=O)OCC)CN C1(NC(c2cccs2)=O)CCN(C(=O)C(c2cccc(Cl)c2)(F)F)CCC1CO N1(C(C=COCC)=O)CC2CC1CN(C(c1nc(-c3nc[nH]n3)sc1C)=O)C2 C(=O)(CCC(CC)NC(CCOCC=C)Cc1ccccc1)OC(C)(C)C CC(C)C(C)(O)C(=O)NC1CC(C(F)F)(NC(C2CC3CCC(C2)O3)=O)C1 N1(C(C2(C)C(C)(C)C2)=O)CC2(C=C(C(=O)NC3CCCC4(C3)N=N4)CO2)C1 C(=O)(CS(C)(=O)=O)NCC(C(C)C)NC(C(C)NC(=O)NC)=O CC1CN(C(=O)C(=O)N(C)C)CC(C)N1C(=O)COC1CCC1 C(=O)(CCCC(=O)N(C)C)NCCC1CCC(NC(CCC(=O)N(CC)CC)=O)C1 c1(C(=O)NC(CCNC(c2n(C(C)C)ccn2)=O)(C)C)cc(F)c(CO)c(F)c1 N1(CC)CCC(N=c2[nH]c(N3CCC(CC)C(C)C3)nc3c2COC3)CC1 N1(C(C(C)Sc2ccccc2Cl)=O)CCC(NC(c2ccn(C)c2)=O)C(C)(C)C1 Cn1nnnc1CCCN.N1(C(=O)NC)CCC(CCCn2ccnn2)C1 C=CCC(C)(C)CC(=O)NC1C=CC(CC(=O)Nc2cc(C)cc(C#N)c2)C1 C1(C(C(=O)N(CC(=O)NC(C2C(C(=O)OC)C2)C)CC2CC2)F)CCCCC1 C1(C(c2n(CCC(=O)OCC)nnn2)NCC2(CO)CC2)CCCOCC1 c1(CN2CCC(CNC(c3cccc(N(C)C)c3)=O)C2)ccc(C#N)cc1 C1(CC(=O)NC(CNC(c2c(COC)scc2)=O)C(C)(C)C)CCCNC(=O)C1 C(=O)(CC(O)C(C)(C)C)NC1(COC)CCCN(C(c2coc(Br)n2)=O)C1 C1(CNC(c2cnc(C(C)OC)s2)=O)(NC(c2cc(C#N)c[nH]2)=O)CCOCC1 c1(N(CCC(=O)NC2(C(=O)OC(C)(C)C)C(C(C)C)C2)C2CCCC2)cccnc1 C1(CC)CCC(=O)N1Cc1ccc(CNS(C)(=O)=O)cc1Cl c1(C(=O)NCCCNC(Cc2nc(C(C)OC)sc2)=O)cc(C)cc(F)c1 c1(SC)cccc(C(=O)NCCCOCCNC(c2cc(Cl)ccn2)=O)c1 C=C(C)C(CC(=O)NCC1CCC1NC(c1cn(C(C)(C)C)nc1CC)=O)OC C1(N(C(CCNC(C)=O)=O)C)CC2CCC(C1)N2C(C12CS(=O)(=O)C(C)(C1)C2)=O C1(NC(CC(CC)C)=O)COC2CN(C(=O)CSCC(N)=O)CC12 CC1CCC(NC(c2cc(N)cc(O)n2)=O)CN1C(=O)CCC(N)=O c1(CC(=O)N(CCNC(C(C2CCCCC2)OC)=O)C)ccc2ccccc2c1 C1(C(C)NC(C(c2ccccc2)C)=O)CCCN1C(c1cn(C2CCC2)nn1)=O C(=O)(C1=CC2CC=CCC12)NCCCCN(C(=O)C(c1cccc(F)c1)(F)F)C N1(c2ccnc(NC3CCN(CC(C)(C)C)CC3)n2)C2CCC1C(=O)NC2 Cc1ccc(C(=O)NC2CCCC2(C)CNC(c2ncncc2Cl)=O)c(N)c1F c1(C(=O)Nc2nc(-c3cc(Br)cs3)cs2)cc(O)c2occc2c1 Oc1nnc(-c2nc(-c3ccccc3Br)nn2CC2CCOC2)c(O)n1 c1(NC(c2nnnn2C2CCCCCC2)C2(CS(N)(=O)=O)CC2)ccc(O)c(Cl)c1 C1(C(=O)NCCC(=O)NCC)COCC1NC(C1(Cl)CC1(F)F)=O C1(CC(N2CCC(CC=C)(NC(C3CCCCC3)=O)C2)=O)SC2=NCCN2C1=O CCC(C(=O)NC1(C)CC(NC(C2(c3ccnc(Cl)c3)CC2)=O)C1)C(C)(C)CC C1(C(C(N2CC(C(CC)=O)C2)=O)C)CCCN(C(=O)CC2CC(=O)C2)C1 N#Cc1ccc(COC2CCCN(CC(F)(F)F)C2)cc1 N1(C(C2CCC(=O)N2)=O)CC2CCCC2(C(=O)NCCOC2CCCCC2)C1 c1(C(N2C3CC(CNC(c4cc(C)on4)=O)C(C3)C2)=O)cccc2c1OCC(=O)N2 N1(C(=O)Cc2c[nH]ccc2=O)CCCCC(C2CCCN2)C1 c1(C(N2CCCC(N(C(c3cc(SCC)ncc3)=O)C)C2)=O)ccc(N)c(Cl)c1 C12(NC(c3c(C)c(Br)ccc3)=O)CCCC1N(C(=O)CCC(C)(F)F)CC2 C(C(O)C(C)(C)C)NC(CN(CC(C)C)C(c1n(CCC)ccc1)=O)=O C1(C(N2CC(C(=O)NCCC=CC=C)(SC)C2)=O)CCC(C)(C)OC1 CC1CCC(OCC(=O)Nc2cccnc2OC(F)(F)F)CC1 CCC(CC)CCCn1nc(C2CCCC2)nc1CN(c1ccccc1)C N1(C(c2scc(C)c2)=O)CCN(C(C2CC(C)CC(C)C2)=O)CC(C)C1 C(=O)(CCC(CC)OC)NC(CCC)CNC(=O)CC1CC(C(F)F)C1 N1(C(c2n[nH]c(C)c2O)=O)CC2CCCC2(C(N2CCC(CCO)CC2)=O)C1 C1(O)(C(=O)NC2CC(O)C2)CCN(C(c2cc(C(F)(F)F)no2)=O)C1 c1(OC)ccccc1C(CNC(C1CCC(O)CC1)=O)NC(=O)CCCOC CC1(C)CCc2cccc(C(=O)NCC3CCN(C(C4(CO)CCOC4)=O)C3)c2O1 N1(C(C(C)CC2CC2)=O)CCCC(N(CCO)C(c2cnc(O)o2)=O)C1 c1(OC)cccc(C(C)=CC(N2CCC2CNC(C2CC2C2CCCO2)=O)=O)c1 C(C)(C(C)(c1nnnn1C)NCC1(CC(=O)OC)CC1)OC C1(NC(CCN(CC=C)C(C2CNC(=O)O2)=O)=O)CC2CCC(C1)C2 Cc1ccc(C(=O)NCC2(O)CCCN(C(C3(C#N)CCCOC3)=O)C2)c(C)n1 c1(CC)cccc(CC(=O)NCCCOCCOCCNC(=O)CC(C)O)c1 C1(C(=O)NCC=CCNC(CC)=O)CCc2nnc(C)n2C1 C#Cc1ccc(C(N2CC3C(CNC(c4cscc4COC)=O)C3C2)=O)cn1 C=C(CNC(C1(CNC(c2cnccc2C)=O)CC=CC1)=O)C1CCOCC1 c1(CC(=O)NCC(CCCC)NC(C2(C)COC(=O)OC2)=O)cc(C)ccc1C N1(C(C(C)OC)=O)CC2=C(C1)CN(C(c1ccc(-c3cccnc3)s1)=O)C2 N(C(=NCCN1CC=C(C)CC1)NCCNC1CCCCC1)CC(CC)(C)OC c1(OCC)ccc(OC2(CC(=O)NC(=O)NC3(OC)CC(F)(F)C3)CCC2)cc1 C1(CC)CCCCN1C(=O)C(c1cnn(C)c1)NC(=O)C(C)C1CCC1 C1(C(=O)NCCCCCCNC(c2c(OC)nccc2)=O)OCC2CCCC1C2 CC(C)CC(CO)NC(=O)NC1CCCC(NC(=O)CC2CCC2)C1 C(CN=c1c(Br)c[nH]cc1[N+](=O)[O-])C1C(C)CCCN1C(c1ccco1)=O c1(C(=O)NCCN(CCC)C(C2C=C2C)=O)cc(F)cc2cccnc12 C(=O)(CC(=O)NCC1CC(NC(=O)CC(C)n2ccnc2)C1)OC C1(NCCN2CCC(CN(C=O)CC)CC2)COc2ccccc2O1 C1(CC)CCN(C(=O)CN2CCC(OC)C2)C(C(N2CCCN(CC)CC2)=O)C1 c1(C(=O)NCc2cccc(C(=O)NCC(C)(C)C(N)=O)n2)ccc2cncn2c1 c12ccnn1C1CN(C1)C2=O.N1(C(C2CCCCC2)C(=O)OCC)CCCCC1 c1(Cn2cc(CC34C(CN(C(=O)CSC(F)F)C3)CC4)nn2)ccc2nc[nH]c2c1 N1(C(C2CCOCC2)=O)CC2(C1)CC2(F)F N1(C(c2c(C)nc[nH]2)=O)CC(NCc2ccc(Br)cc2C(=O)O)CC(C)C1 C1(N(C(C=CCCC(C)C)=O)C)CCC(NC(C2CCOC2=O)=O)CC1 C1(C(=O)OCc2c(C)cc(C)s2)CC2CCCCCCC12 Cn1nc(CC(N2CCN(C(=O)Cc3csc(Cl)c3)C3CC23)=O)c2ccccc12 N1(C(c2ccc(=NC)[nH]c2)=O)CCC2CC1CN(C(=O)CCC(N)=O)C2 C12(C(N3C(CCNC(CCN(C)CCO)=O)COCC3)=O)CCC(C)(C1)OC2 C(c1cn(C)nn1)=C(C(N1CCC(N(C(=O)C(CO)OC)CC#C)C1)=O)F CON(CCC(=O)N1CCC2CC12C)C(=O)C1CCC(O)C1 N1(C(Cc2ccc(C)nc2)=O)CC2CCCC2(NC(=O)CC(C)N(C)C)C1 CC1CC(=O)NC(C(=O)N(CCCNC(C2(C)CCCNC2=O)=O)C)C1 N1(C(C(C(C)C)NC(C)(C)C)=O)C2CCC1C(C(=O)Nc1scnc1C(F)F)C2 c1(C(N(CC(C)C(=O)NC2CCC(=O)NC2)C)=O)ccc(O)cc1 CCCCCCC(F)C(=O)N1CC2CCCC1(CNC(c1cnnn1CC)=O)C2 C(C)(C)(CCCNC(C1CC=CCN1C(=O)C(C)CSC)=O)OC C1(CCNC(c2cnc(CC(C)(C)C)s2)=O)CCN(C(c2cc(F)cs2)=O)CC1 C1(NC(c2ccc(-c3ccco3)[nH]2)=O)C=CCN(C(c2ccccc2C2CC2)=O)C1 c1(C(=O)NC2C(OC)CN(C(=O)Cc3ccon3)C2)cc(O)nc(C)n1 N1(C(C2CN(C(N(C)C)=O)C2)=O)CC(CNC(=O)CC2(C)CC2)OC(C)(C)C1 C(=O)(C(C)S(=O)(=O)C1CCOCC1)NC1CN(C(CCC(C)SC)=O)CC1C C(=O)(C1=CC2(CCN(C(=O)CN)C2)C1)Nc1scc(CCCCCCC)n1 Cc1ccc(=NCCC(=O)N2CC(CN(C(=O)C(CO)C(C)(C)C)C)C2)[nH]c1 C1(C(N2CC(CC)OCC2)=O)CCCCCN1C(c1c[nH]nc1C)=O c1(C(=O)NCC(N(C)C(C2CC3CCC(C2)C3)=O)C2CC2)ccn2c1CCCC2 C(=O)(C1CCc2cccc(F)c21)NCC1N(C)CCN(C(CC(CC)(F)F)=O)C1 C1(NC(CN2CC(CC)C2)=O)CCCCCN(C(c2[nH]cc3c2CCC3)=O)C1 N#Cc1cc(F)c(C(=O)NC2CN(Cc3ccc(I)o3)CC2O)c(F)c1 c1(OC)cccc2c(C(=O)NCCOC3CN(C(C4CNC(=O)C4)=O)C3)n[nH]c12 O=S(=O)(c1c(Cl)cc(Br)cc1Cl)N1CCCC1c1nc2ccccc2[nH]1 C(=O)(C1CCc2ccc(Cl)nc21)N1CCCC(C)(NC(C2CC(OC)C2)=O)C1 c1(C(N2CC3C(CNC(c4ccc(Cl)s4)=O)(C3)C2)=O)nc2ccccc2[nH]1 c1(-c2nc(-c3c(C)cc(C(=O)OC)s3)on2)c(F)ccc(C)c1F c1(OC)cc(CC(N2CCC(C(C)NC(=O)Cc3cn[nH]c3)C2)=O)ccc1Cl C(c1cccc(Cl)c1Cl)=CC(=O)NCc1nc(-c2cccc(OC)c2)oc1 C(C(C)(C(=O)NCC1CCCC(CO)C1)NC(C1CCC(F)(F)C1)=O)SC C1(CNC(C(C)C2CCCC2)=O)CN(C(c2cc(N)cc(O)c2)=O)CCCO1 Cn1nc(-c2cn(C3CN(C(C4(CCCC(O)CO)CC4)=O)C3)nn2)cc1N c1(C(N2CC(C)CC(NC(C(C)OCCC#C)=O)C2)=O)ccc2sc(C)nc2c1 CS(=O)(=O)c1ccc(C(N2CCCC(C(=O)NCC(N3CCNCC3)=O)C2)=O)o1 n1(CC(N2C(CN(C(CC3C(C)C3(F)F)=O)C3CC3)CCC2)=O)cccnc1=O c1(C(=O)NCC(CNC(=O)CCn2cncn2)F)ccc(C2CC2)o1 N1(c2n(CC(=C)C)c(-c3ccc(C)cc3)nn2)CC2CC1CN(C)C2 C(=O)(C(C)C(=O)NC1CC(NC(=O)C#CC(=O)N(C)C)C(O)C1)OC c1(C(N2C(C(C)NC(C3CC4CC4CC3C)=O)CCC2)=O)n[nH]c2c1CCCC2 C(=O)(C(C)(C)n1cnc(C)c1)NC(CN(C(C(C1CCCC1)OC)=O)C)C CCC(C)(CCNC(=O)CCc1cncn1C)NC(c1cc(C)n(C(C)C)n1)=O S(=O)(=O)(c1ccc(C#N)c(NCCCS(C)(=O)=O)c1)NCCC(C1CC(F)(F)C1)C c1(C(=O)NC)ccc(CC(Cl)=CCl)s1.O=C1CCSCCCOCC2(CC2)CN1 c1(C(N2CC(SC)C(NC(=O)C(C)(C)C(C)C)C2)=O)ccc(C#N)cc1C c1(CSCC(=O)NC(c2cncc(O)c2Cl)=O)nc2ccccc2s1.C12CC1C2 c1(C(C(=O)NCCSC)NC(=O)CC2CC=CC2)cccc(C(F)(F)F)c1 C1(C)(CC(N2CC(F)(CC)C2)=O)CCN(C(=O)CCOC2CC2)C1 C1(NC(=O)COCC(F)F)COC2(CCCN(C(c3c(O)cccc3Cl)=O)C2)C1 Nc1c(C(=O)NCC2N(C(c3cnc(S)[nH]3)=O)C3(CCC3)C2)ccc(Cl)c1O S(=O)(=O)(c1ccc2oc(=O)c3ccccc3c2c1)NC1C=CC(OC)C1(C)C c1(NCC2(CC(C)C)CCC2)ccnc(N2CC3C(Br)C3C2)n1 c1(C(N(C(=O)OC(C)(C)C)C)C)nccn1C.C1(C(C)N)CC1O c1(N(C(=O)CN2CCCC2CNC(=O)CC2(C)CC2)C)ccc(CC(N)=O)cc1 C(C(CC1CCCC1)C(=O)NC1CC(=O)N(CC2CC2)C1)NC(C=CC)=O N1(C(C(C)=C(CC)C)=O)CCCC1CN(C(c1n[nH]cc1C1CC1)=O)CC C(=O)(CS(=O)(=O)C1CC1)N(C(C)CNC(C1CCN(Cc2ccccc2)C1)=O)C C1(NC(CC2(C=C)CCC2)=O)CC(NC(=O)CCSCC(N)=O)C12CCC2 C(=O)(CCC(CF)CF)NC1CN(C(Cn2c(C)ncc2)=O)CC(C)C1 c1ccc(SCc2nc(NC(c3onc(C(C)OCCC)n3)=O)sn2)nc1 c1(C(N(CC(C)(C)NC(=O)CP(C)(C)=O)C)=O)ccc(O)nc1Cl CCC(C#N)C(=O)N(CC)CC1CCN(C(C2CN(C3CCOC3)C2)=O)CC1 N1(C(C(C(C)C)C)=O)CCC(NC(=O)C=CCF)C(CO)CC1 C(=O)(C(F)(F)CC(C)C)N(CCN(C(c1ccc(F)c(N)c1)=O)CC)CC C1(C(N(C(C)C)CCN(C2(C)CCOCC2)C)=O)CCc2nccn2CC1 c1(C(N2CC(F)(CNC(c3c(CC)cco3)=O)C2)=O)cc2c(C)c(C)ccc2[nH]1 Cc1nn2cccnc2c1CNC(=O)CCC(C)(F)F.c12ccccc1CNC2 C(=O)(C(F)CC(C)(C)NC(=O)C(CO)C(F)(F)F)N(C)CC1(O)CCCC1 N1(C(C(CC#C)C2CC2)=O)CCC(NC(c2ncsc2C)=O)CC(C)(C)C1 CCC(C)(O)C(=O)NC1CCCCC1NC(C1(O)CCCCC1)=O Cc1ccc(N2CC(NC(=O)CC3COCCN3C(c3cscn3)=O)CC2=O)cc1 C1(NC(CN(CCOC)C)=O)CN(C(=O)CC2CCCCO2)CC1CO N1(Cc2c(C)n[nH]c2)CCC(O)(C(=O)NCCCc2cccs2)CC1 S(=O)(=O)(c1cccc(N2CCC(O)C2)n1)NCc1ccc(OC(C2CCC2)C)nc1 N1(C(=O)Cn2nnc(C3CC3)n2)CCOC2(CCN(C(c3nncs3)=O)CC2)C1 C(=O)(CCC(=O)NN(C)C)N1C(C(=O)NC2CC(=C)C2)C=CCC1 C#CC1CCCCN1C(=O)C(c1cccs1)NC(=O)C=CC(F)F C1(NC(=O)N(C2CC(c3ccon3)C2)CCN2CCCC2)CCOC1 CCC(F)(F)C(=O)NC(C1CN(C(C2CN(C3COC3)C2)=O)C1)C Nc1ccc(C(=O)NC2CCN(C(=O)CCc3nnc(C4CC4)o3)C2)c(Br)c1 CCCC(C(=O)NC1CCC(NC(C2(CC(C)C)CC2)=O)CC1)C(C)C N1(C(c2cc(OC)n[nH]2)=O)CC2C3CCC(C2C1)N(C(C1CCCC(O)C1)=O)C3 C(C(F)(C(=O)N(C(C)C)CC1CCC1)C(C)C)NC(c1c(OC)nn(C)c1)=O c1(C(N2CC(C(=O)N)(CCO)C2)=O)ccc(CO)nc1.C1(OCC)CC1C C1(OC)CC2(C1)CC(NC(C1CCC(NC(c3cc(C)c(CO)o3)=O)C1)=O)C2 C1(NC(c2ccc(C(=O)NC)nc2)=O)CC(C)CN(C(=O)C2=CCCCC2)C1 CC1CC(NC(=O)CC2C=CCC2)CN(C(=O)COc2ccc(O)cc2)C1 C(=O)(C1=C(Cl)CCC1)N1CCC(OCCNC(c2cnc(C(C)OC)s2)=O)C1 C1(C2(C(=O)NCCCN(C)C)CC2)CCCN1C(C1(C2CC2)CC1)=O.C(N)(=O)N C1(C(N(CC#C)CCOC)=O)CCN(C(C2CC2F)=O)C1C C1(C(=O)NCCC(=C)CNC(=O)CCn2ccccc2=O)CC(=O)NC(CC)C1 c1(C(=O)NC(CC(=O)NC(CC=C)(C)C)C2CC2)ccc2c[nH]nc2c1 n1(CCN(C)C)cc(C(=O)NCC2(NC(=O)CCCn3cccn3)CCC2)cn1 C1(C(=O)OC)CN(C(=O)CC2(OC)CCC2)CCO1.c1(OCCN)ccc(Cl)cc1 C1(C(=O)NCC=CCNC(C2(C)CCC3CC3C2)=O)CCn2ncnc2C1 N1(CC#CC)CCN(C(=O)CC2CN(C(C3CCOC3C3CC3)=O)CC2C)CC1 C1(N(CC(C)C)C(C2CC=CCC2)=O)CCN(C(=O)C(C)N2CCCC2)CC1 C(=O)(CS(=O)c1ccc(Cl)cc1)NC1(C)CN(C(Cc2cn(CC)nn2)=O)C1 C1(C(=O)NCC(C2CCC2)OCC)C=CCCN1C(=O)CNC(C)=O C(=O)(C(C)CC(C)CC)N1CC(NC(c2cnc(CC)[nH]2)=O)(COC)C1 c1(C(CNC(=O)COCC2CC2)CNC(c2coc(Cl)c2)=O)ccccc1 c1(C(N(C)CCNC(c2csc(Cl)c2)=O)=O)cccc(C2CNC(=O)C2)c1 c1(OCC(N2CC(NC(CC)=O)C(C)C2)=O)ccc(Cl)c(F)c1 CCC(C#N)(CC)C(=O)NCC(C)C(N1CCC(SC)CC1)=O C(=O)(CCCCCC(C)C)N1CCC(C(=O)NCC(C)(C2CC2)OC)C12CC2 C1(CNC(=O)CC2CCCCC23CC3)CC2(C1)CN(C(=O)CCCn1ccnn1)C2 C(CCC(=O)NC1COC(=O)C1)N(C(=O)C(C1CC1)C1CC1)C Cc1nc2ccc(C(N3CC(NC(C4CC5(CC5)C4)=O)CC(O)C3)=O)cc2[nH]1 c1(C(N2C(CO)CC(NC(c3ccc(CC)[nH]3)=O)C2)=O)cnc2n1C(C)CCC2 C#Cc1cnc(C(N2CCN(C(c3cc(C)co3)=O)C(CC)C2)=O)c(C)c1 C(=O)(C1=COCCC1)NC(C)CCCCNC(=O)C(O)c1ccsc1 C(=O)(CC(C)C(F)(F)F)NCC1(NC(COC(CC)C)=O)CCC1 C(C)(C(=O)NCCC1CC(C(=O)NCC(O)CN(C)C)C1)OCCC#C CC1CC(OC(=O)COc2cccc(Cl)c2)CN(C(=O)CCCOC(N)=O)C1 C(CCC(C(=O)N(Cc1ccco1)OC)NC(=O)CCN(C)CCO)OC Cc1ccc([N+](=O)[O-])c(C(N2CC(NC(c3ccc(N)c(Cl)n3)=O)CC2C)=O)c1 C1(CN(C(CCCOC(C)=O)=O)C)CC(F)CN1C(C1CCNC1=O)=O N1(C(C(C)C)=O)CC2(CCOCC2)CC1CNC(c1ccn2ncccc12)=O CC1C(NC(=O)CC(C)C2CCCO2)CCN1C(c1ccc(Cl)nn1)=O N#Cc1ccc(Cc2cn(CC(=O)NCC3CC(C(N)=O)=NO3)nn2)cc1F N1(C(C2CC(CC)(CC)C2)=O)C2CC1CN(C(C1CC(S(C)(=O)=O)C1)=O)C2 c1(C(N2CCC(O)(CCNC(C(C)(C)C)=O)CC2)=O)coc2c(F)cc(Cl)cc12 C1(NC(C(C)O)=O)CN(C(c2cccnc2)=O)CC12CC2 c1(C(=O)NC2CC(CC(=O)NC(C(=O)NC)(C)C)C2)cc(S(N)(=O)=O)ccc1O C1(C(N2CC3CC3C2)=O)CSCCN1S(=O)(=O)Cc1ccc(Cl)cc1 CC(C)C(C(=O)NCCCOCCCNC(c1ncoc1-c1ccco1)=O)N(C)C C1(CNC(CNC(=O)OC)=O)CC2COCC2N1C(C1CC2(C1)CC2F)=O Cc1noc(C(N2CC(F)(C(N3CC(CCN(C)C)C3)=O)C2)=O)n1 Cc1c(C(N2CCCC2CN(C(C2(C)CCOC2)=O)C2CC2)=O)cnn1C1CC1 C12(CNC(CCCN(CCC)CC)=O)CN(C(C3C(C)C3(F)F)=O)CC1CCO2 N1(C(CC(F)(F)F)=O)CC2C(C1)C2(C)C.c1(-c2cn(CCCC)nc2)cccc(N)n1 Cc1cccc(C(=O)NC2CC=C(C(=O)N3CCC(N4CCC4)C3)C2)c1N C1(N(C)C(C2CS(=O)(=O)C2)=O)CCN(C(=O)CC2(C(F)F)CC2)CC1 c1(C(N2CCSC3CCC23)C(=O)NC(CC)C)cnc2c(F)c(F)ccc2c1 C(=O)(C(C)C(F)(F)F)NC(COCC)C(=O)NCCc1ccnn1C C(C)(CCC(=O)NCC1CC2(CC2)C1)NC(CN(CCC)C)=O c1(OC)cc(C(=O)OCCC(C)CO)cnc1-c1ccc(F)cn1 Cc1cc2c[nH]nc2c(C(N2CC(NC(C3CCCOCC3)=O)C2)=O)c1N c1(C(=O)NC2C(CNC(c3ccc(C(N)=O)cc3)=O)CC2)cncc2ccsc12 C1(C)(C(N2CCC(NC(C(COC)C)=O)C(O)C2)=O)CCC(C)(C)CC1 N1(C(c2c(CC)con2)=O)CC(CNC(c2cc(Cl)ncc2OC)=O)CC(C)C1 c1(NCC2CCCN(C(C(C=C)NC(=O)OC(C)(C)C)=O)C2)cc(Cl)ncc1Br C(=O)(N=c1cc(C2CC2)[nH][nH]1)C1N(Cc2c(NC=O)ccc(F)c2)CCNC1 C1(C(=O)Nc2cccc(CC)c2)CC2CN(C(c3cc(CCO)on3)=O)CC2C1 C1(C(N2C(CN(C(=O)C(F)=C(C)C)CC)CCC2)=O)C(F)(F)C12CCC2 n1(CCOC)ccc2c(C(=O)NCCCn3ccnc3)cccc12 Cc1cc(C(=O)N(C2CCCCC2)CCNC(C2CC23CCC3)=O)ns1 C1(C(N(c2ncc(C)s2)C)=O)CCC(C)(C)CC1.C12CCC(CC1)N2 N1(Cc2n(CC)ccn2)CCC2C(CCCN2c2ncc(F)cn2)C1 C1(OC)(CNC(c2cc(C)cnc2C)=O)CCN(C(c2c(C)csc2Cl)=O)CC1 C12CC(CC(CC=C)O1)OC(=O)C13CCCC21C3.O(CC)CC C(=O)(C(CNC(=O)C(F)CC1CN(C(=O)COC)C1)OC)OC.C(C(F)F)S N1(C(C#C)=O)CCOCC(C(=O)Nc2cccc(SCCN3CCOCC3)n2)C1 C(C)(C)(CC(=O)NCC(N1CCOCC1)C)N(C(C1C(C(C)C)CCO1)=O)C O=C(C1=CCSC1)NCCC1CCCCN1C(c1cc(C2CCOC2)[nH]n1)=O c1(CC)cc(Sc2cccc(C)c2)ccc1CC(C(=O)O)n1ccnc1 Cc1ccc(C(N2CC(CNC(=O)C(C3CCC(=O)N3)C)C2)=O)c2c1NCCC2 Cc1cc(Cl)c(C(N2CCCC(CCNC(=O)C=Cc3cn(C)cn3)C2)=O)cn1 CCC(CC)(CO)C(=O)N1CCN(C(c2cc(C(N)=O)c[nH]2)=O)C2(CC2)C1 N1(C(C2CCN(C(c3c(C)nc(C)s3)=O)CC2O)=O)CCn2nc(CO)cc2C1 CC(C)CS(=O)(=O)CCC(=O)N1CCCC2(NC(c3coc4c3COC4)=O)CC2C1 N1(C(CCCC#C)=O)CC2CC(C(N3CC(C=C)(CF)C3)=O)CC2C1 c1(C(N(C2CCCN(C(C(N3CC(C)C3)C)=O)C2)C)=O)cnc2[nH]c(O)nc2c1 C(CC(=O)N1CC(NC(c2ccn(C(C)(C)C)n2)=O)C(C)(C)C1)(C(N)=O)NC(C)=O c1(CN(C(C2CCN(CCCc3ccccc3)C2)=O)CC)csc(C(C)C)n1 C1(C(=O)NCC2CCN(C(c3c(C)cn(C)c3)=O)CC2)COCC(C)(C)O1 N1(C(Cc2cc(C)no2)=O)CCCC1(C)CNC(=O)CC1CC(N(C)C)C1 c1(C(N(CC(CC)NC(=O)Cc2nocc2C)C)=O)conc1C C=CCCC(C)(C)C(=O)NCc1ccnc(C(=O)NCc2ccc(Cl)nc2)c1 N1(C(C(C)(C(C)C)OC)=O)CCC2(CCCCC2NC(=O)Cn2cccn2)CC1 Cc1cccn2cc(C(N3CCN(C(=O)COC4CCCOC4)CC3)=O)nc12 n1(CC(=O)N(CC(C)NC(c2cc(CC)oc2C)=O)CC)cc([N+](=O)[O-])cn1 C1(C(C)(C)C)CCCC(C(=O)NCC2CCN(C(=O)CCNC(=O)CO)C2)C1 CS(=O)(=O)c1cncc(-c2cnc3[nH]cc(C(N4CC(F)(F)C4)=O)c3c2)c1 C=CCCCCCCCC(=O)NC1CC(NC(c2ccnc(C)c2C)=O)C1 C1(NC(c2cc3n(n2)CCO3)=O)CC1C1CCCN(C(C2(O)CCC2)=O)C1 c1(CC(CNC(C2(O)CCCC2)=O)NC(C(N2CCOCC2)C)=O)ccccc1 Cc1cn2nc(C(=O)N(CC(C)CNC(=O)C(C)c3ccco3)C)cc(C)c2n1 c1(C(N(C(C)CNC(=O)Cc2cc(C3CC3)on2)C)=O)nccn2ccnc12 c1(C(=O)NCC2C(NC(c3nc(C)sc3)=O)C2)nc(C)n(-c2nc[nH]n2)n1 Cc1cccc2[nH]cc(C(=O)NC3CC(F)CN(C(C4CC4C)=O)C3)c12 N1(C(C2C(C=C)C2)=O)CC(NC(c2cccc(-c3ccc[nH]3)c2)=O)C(C)C1 c1(C(N2CC=CC(NC(c3nnn4c3COCC4)=O)C2)=O)ccc2nnnn2c1 CCC(CC(=O)N(C1CN(C(C2CNC(=O)CC2C(F)(F)F)=O)C1)C)C(C)C Cc1cc(F)cc(C(=O)NC(C)(CNC(=O)C(=Cc2c[nH]cn2)F)C2CC2)c1N C(=O)(C(CCC(N)=O)NS(C)(=O)=O)NCCNC(c1n(CN(C)C)ncc1)=O C=C(Cl)CC(C(=O)NC(C1CCCC1)CC)NC(=O)C=Cc1ccoc1 N12CCC=CC1C2.C(=O)(O)NCCN(CC)CC c1(C(=O)NC2CCN(C(C3C(C)C3)=O)C2)cc(C(F)(F)F)c(Cl)cn1 C1(NC(c2cc(Cl)ns2)=O)CCCCC1NC(c1ccoc1C(F)(F)F)=O c1(CCC(N2CC(C)N(C(=O)C(CO)NC(N)=O)CC2)=O)nc2ccccc2o1 C=C1CC(C(=O)NCC(C)(C)C2CCC2)(CCCC#N)C1.C1(=O)CN1 N1(C(CCC#C)=O)CCN(C(C23CCC(c4ccccc4)(CC2)C3)=O)CC1CC C1(C)(C(=O)OC(C2CC2C(C)C)=O)CCCCO1.C12(CC1)CN2.C(=O)N(C)CC c1(C(N(C2CCN(C(c3c(SC)scc3)=O)C2)C)=O)cccc(F)c1 c1(C(=O)NC2CN(C(C3CC4(CSC4)C3)=O)CC2C(F)F)cc(=O)cc(Cl)[nH]1 c1(C(=O)NC2(CNC(C(CC)(C)C(N)=O)=O)CCCC2)ccc2c(c1)CCN2C CN1CC(C(=O)NCC2CCN(C(=O)COCC3CCC3)C2(C)C)CCC1=O S(=O)(=O)(c1ccc(NCC2(C)CSC2)c(Br)c1)NCC1C(C)OCC1 C(CCCCC(=O)N1CCC(C)(NC(C)=O)C1)NC(C1(OC)CC1)=O N1(C(Cn2nc(C)oc2=O)=O)C2CCCC1CC(NC(=O)C1=NNC(=O)CC1)C2 CC1CCC(CNC(=O)C=CCO)CN1C(c1cc(N(C)C)cc(Br)c1)=O Cc1ncc(C(=O)NC(C(=O)NCc2nnc(C)o2)C2CCCC2)c(C)n1 N1(CC(=O)NC2CC3(C(C(N(C4CCCCC4)C)=O)C3)C2)CCC2(C1)CN(C)C2 CC1CCC(NS(=O)(=O)CC(=O)N(C)CCN(C(=O)CC2CCOC2)C(C)C)CC1 Cc1sc2ccccc2c1CNC(=O)Nc1ccc(=O)n2c1CCC2 Cc1cc(C)c(C(N2CC(NC(=O)COC3COC3)CC(O)C2)=O)c(N)c1 c1(OCC)ccc(S(=O)(=O)N2CC3(CC3C(N3CCCOC(C)C3)=O)C2)c(F)c1 N1(C(C(CC#C)C)=O)CCCC(NC(c2cncc(Cl)c2)=O)CC1 c1(OCC)cc(C(=O)NCC2(CN=c3[nH]nc(C)s3)CCCC2)ccc1[N+](=O)[O-] C12(NC(=O)NCCC(N3CCCCCC3)C)CC(NC(=O)OC(C)(C)C)(CO1)C2 N1(C(c2c(Cl)cn(CCC)n2)=O)CC2CC(NC(=O)Cc3csc(C)n3)C1C2 c1(N(CCC)CCC)ccc(C(=O)OC)cc1.C1(NC(=O)CO)(CCCCF)CCOC1 c1(C(=O)NCCOC2CN(C(C)=O)C2)cccc2ccsc12.N12CCCC1C2=O Cc1cc(N(C)C(=O)NCc2cn(CCN3CCOCC3)nn2)no1 N1(C(c2nccc(C)c2F)=O)CC2(C1)CN(C(C1CC1C)=O)CC(C)(C)O2 Cc1cccc(CC(=O)NCCN(C(=O)C(c2nc(C)cs2)C)CC(C)O)c1 Cc1c(CC(=O)NCC(CC2CC2)C(=O)N2CCC(C(F)(F)F)C2)ncn1C C1(CC)CC(CNC(=O)CCSCc2ccccc2)N(C(=O)C2=CCOC2)C1 c1(OC)cc(C(=O)NCC2CN(C(c3cnco3)=O)CC2C)cc(Cl)c1 Cc1ccc(NC(C2CC(O)CN2C(=O)CC23CCCC2C3)=O)cc1OC C(C(C)CC(F)(F)F)NC(CC1CN(C(C(C=C)OC)=O)CC1C)=O CCC(O)C(C)(C)C(=O)NCC(C)(C)NC(c1ccccc1-c1ccccc1)=O N1(C(c2c(OC)ccnc2)=O)CC2CC(CNC(=O)Cc3cnn(C)c3)C2C1 C12(NC(C3CC=CCO3)=O)CCCN(C(c3coc(Br)c3)=O)CC1C2 C1(CC(=O)NCC2(CNC(CC(CC)OC)=O)CCCCC2)CC2(CCC2)CO1 c1(CC(C)NC(c2cnc(COC)s2)=O)ccc(CNC(=O)CC(C)(C)O)cc1 c1(C2C(F)(C(=O)NC3C(NC(c4cnco4)=O)C3)C2)ccccc1 C(CC(C)C)(C(=O)NC1CN(C(=O)C=Cc2cnccc2C)CC1C)NC(C)=O C1(NC(C23OCC(CC)(C2)C3)=O)CC(C)CN(C(=O)C(c2ccc(Cl)cc2)C)C1 C(=O)(C(C)(C)C(F)(F)F)NCC1(NC(c2ncc(C(=O)OC)cn2)=O)CC1 C(=O)(C(CNC(C1(NC(C2C=C(C)CS2)=O)CC1(C)C)=O)OC)OC N1(c2ccc(C(=O)OC)nn2)CCCC2(COCC(=O)N2)C1 C1(CNC(C=CC)=O)CCCC1NC(=O)C(C)(C)c1cscn1 Cc1cc(O)ncc1C(=O)NC1CN(C(C2CC2C)=O)CCC1CO C1(N=[N+]=[N-])(C(=O)NCC(N2CCC(C(=O)OC)CC2)=O)CCNCC1 C#CCC(CC(F)F)C(=O)N1CCC(OCC(=O)NC2CCOC2)C1 C=CCC(C)(CC)C(=O)N1CCCC(CN(C(=O)CCCc2cccnc2)C)C1 c1(C(N2CCC(F)(CNC(CC(C)F)=O)C2)=O)cc(Cl)cc(Cl)c1 C1(C(N2CC(N(CC=C)C)C2)=O)(OC(C)=O)CCN(C(=O)CCN=[N+]=[N-])C1 c1(C(=O)NCC2C(C)CN(C(=O)CN3CCC(C)(O)C3)C2)ccc(C#N)c(O)c1 N1(C(c2cc(C)cc(Cl)c2)=O)CC2OCC(NC(=O)CS(=O)(=O)CC3CCC3)C2C1 C(=O)(C#CC1(C)CCCO1)N(CCC(C)NC(=O)C1CCc2c[nH]nc21)C N1(C(C2C3(CCN(C(CCCOC)=O)C3)C2)=O)CC(C)(C2CCC2)C1 N1(CC(=O)N(c2ccc3ncccc3c2)CC)C(=O)NC2(CCCC2(C)C)C1=O C(COCC)(C(=O)NC1CSC1)NC(C(C)=CCC)=O C(N=c1nc(N2CCC(C(F)F)C2)c2c([nH]1)CCC2)c1cc(C(C)C)on1 Cc1c(C(=O)Nc2cn(C)nc2OCC(F)(F)F)oc2c1ccc1ccccc21 c1(C(=O)NCCC2CN(C(c3c(C)nc(O)[nH]3)=O)C2)ccc([N+](=O)[O-])s1 N1(C(C2CC(=C)C2)=O)CCCC1C(C)NC(=O)C(C1CCOCC1)F c1(C(=O)NCCN(C(C(CSC)C)=O)CCOCCO)nc(C(F)(F)F)oc1C c1(C(N2CCN(C(CC(C(C)C)O)=O)CC2)=O)cnc2onc(C(C)(C)C)c2c1 c1(C(C)C)cc(C(=O)NCCCNC(C2CC23CC3)=O)n[nH]1 Cc1ncc([N+](=O)[O-])cc1C(=O)NCCNc1ccc(C#N)cc1 C(=O)(CCC=CC(C)C)N1CC(CCCCNC(CSCCCC)=O)C1 N1(C2CCN(C(C(C)(C)N3CCCC3)=O)C2)CCN(C(c2cc[nH]n2)=O)CC1 n1(C(C)C)ncc(Cl)c1C(=O)NC1CC2(C1)CC2NC(=O)CCc1ncc[nH]1 c1(C(=O)NC2CN(C(C3C(C)OC(=O)N3)=O)C2)ccc(N)cc1F C(CCCCC(=O)N1CC(O)CC1C(=O)NC(c1cnn(C)c1)C)OC Cn1cc(C#N)cc1C(N1CC2CC1C2CNC(c1csc(Cl)n1)=O)=O C1(NC(c2n(CC)ncc2Cl)=O)CCCN(C(C2CC23CC(C)(C)C3)=O)CC1 c1(C(=O)NC2(C)CCN(C(c3ccc(C(C)=O)o3)=O)C2)cncc2cccnc12 C1(C(=O)OCC)CCCCC1CNC(C1CC1Cl)=O.C1C(O)CN1 Cc1nc(O)nc(C)c1CC(=O)NCC1CC1NC(c1ccc2scnc2c1)=O c1(SCC2(OC(=O)C=C(C)Cl)CN(CC)C2)ccc(C)cc1Cl N1(C(CC2(C=C)CN(C(c3nscc3C)=O)C2)=O)CC2NC(=O)OC2C1 CN1CCC(C)(C(N2CCCC2CNC(c2cc(N)cnc2Cl)=O)=O)CC1 N1(CC(C)(C)N(c2cnn(C)c2)CC)CCCOC(CC)C1 C1(C(C)C)CN(C(=O)C(CCC2CC2)NC(C2CC(F)C(=O)N2)=O)CCO1 C(=O)(CC(C)(C(F)F)N(C)C)NC1(C)CCN(C(c2cnc(OC)c(C)n2)=O)C1 C1(F)(CNC(C(COC)OC)=O)CCN(C(=O)CCCCc2cnn[nH]2)CC1 c1(C(=O)NCC2C(NC(C3(SC)CC3)=O)CCCC2)cc(F)cc(N)c1N CC1=C(C)CC(C)(C(=O)NCCC(C)NC(c2cc(Br)sn2)=O)CC1 c1(CN2C(C(N3CCC(C(F)(F)F)C3)=O)CSCC2)cc(Br)cc(F)c1F CC(O)C(C)(C)NC(=O)C(C1CCN(C(=O)C(F)C2CCCC2)C1)F C(=O)(C(C)(C)NS(C)(=O)=O)NCCC(=C)CNC(C1C(COC)C1(F)F)=O N1(C(CC2CC(OC)C2(C)C)=O)CC2CCC(C1)N2C(=O)C(C)(C)N1CCCC1 C1(C(N2CCC(c3ccccc3)C(F)(F)C2)=O)CC2CCC(C1)C2(F)F CC(C)CC(Cn1cc(C(C)CC2CCC2)nn1)NC(C1(C(F)(F)F)CC1)=O C1(CNC(CC(CC)C2CC2)=O)CC12CCN(C(=O)C(C)NC(=O)C(C)(C)C)CC2 C1(CNC(CCCCC(=O)NCC)=O)CC12CCN(C(C1CC3CC3C1)=O)CC2 C12(NC(c3cnn4c3CCC4)=O)CCCC1CN(C(c1cc(Cl)ncn1)=O)C2 c1(C(=O)NCCC2CN(C(C3CCC(O)C3)=O)C2)cc(Cl)c2c(c1)OCCCO2 C1(NC(C(C)(C)S(C)(=O)=O)c2n(CCC)nnn2)CC2(CCCCC2)C1 c1(C(C(C)C)NC(=O)NCC2(C(=O)OCC)CC=CC2)ccc(C)cn1 c1(C(N(CC(CNC(C(c2ccccc2)SC)=O)O)C)=O)cccc2c1CCO2 N1(C(C(C)NC(=O)OC)=O)CCC2CCN(C(c3ccc(C(N)=O)o3)=O)C2C1 N1(C(=O)NCC(C(F)(F)F)N2CCC2)CCOCC12CCC(CO)CC2 C(=O)(C1=CC2C=CC(C1)C2)NCCCOCCNC(C(C(CC)CC)C)=O Cc1cc(C(=O)NC(C)(CNC(C2CCCC2(C)C)=O)CO)nn1C(C)(C)C N1(C(CC=CC=C)=O)CCN(C(=O)Cc2c[nH]nc2O)C(C(F)F)C1 c1(C(N2CCC(NC(C3CCCC4CC34)=O)C2)=O)ccc(Br)c(Cl)c1 C(N(C)N1CCC2(CCC(COCCO)CC2)C1)c1c(C(=O)OC)n[nH]c1 c1(C(=O)NCC2(CNC(=O)Cn3cnccc3=O)CCCC2)cc(Cl)ncc1Cl c1(C(N2CCC(CCNC(C3N(C)C(=O)NC3)=O)C2)=O)cc(Cl)ccc1C(N)=O Cc1noc(C(F)F)c1C(N1CCC1CNC(=O)C=CCn1cncn1)=O n1(CC(=O)NC2(CNC(c3sc(CC)c(C)c3)=O)CCOC2)cc(C)ccc1=O c1(NC(C(=O)N(C(C)CN(C)C)CC)=O)cc(Cl)cnc1O C(=O)(C1=CC2CCCC12)N1CCCCC(NC(COc2cc(C)c(Cl)cc2)=O)C1 C#CCC(C)C(=O)N1CCCC1C(C)NC(c1cnn(C(C)C)c1Br)=O C(=O)(C(O)CCN(C)C)NC(C)CC(=O)NCC12CCC(CC1)C2 CC(C)(C)C(O)C(=O)N1CC=CC(NC(=O)CCC2CCOC2)C1 CCCC(C)(C)CC(=O)NC.C12CC3(C1)CC3C(=O)N(C)CC(C)(C)O2 n1(CC)ccc(C(=O)NC2CCC(CNC(=O)C(F)C3CCOC3)CC2)c1C C1(C(=O)NCC(C)N(C(c2ccc(CO)cn2)=O)CC)CCc2nc[nH]c2C1 c1(C(=O)NC2CCN(C(=O)C(C)(C)F)C2)ccc(CC)cc1F C1(C(=O)NCCCCNC(C2CCCC(C(F)(F)F)O2)=O)(CC)CNC(=O)C1 N1(C(C2C(C)(CC)C2)=O)CCCC(N(C)C(c2ccc(O)c(C)c2)=O)CC1 C=CC(C)(C)CC(=O)N1CCC(N(CC(=O)NCCCCCF)C)C1 CC1CC(C)(C)CCC1NC(=O)CCC1(C)CN(C(c2cc(Cl)no2)=O)C1 C(CCC(C)C)(C(=O)NCC1(C)CC(F)(F)C1)NC(C1(C)CC(=C)C1)=O c1(C(C(=O)N(CC(C)CNC(c2cn(C)c(O)n2)=O)C)(F)F)cccc(F)c1F N1(CC(=O)NC(c2ncccc2F)C)CCN(c2ccc(Cl)nn2)CC1 N1(C(c2cc(CC)n(C)n2)=O)CCN(C)C(CNC(=O)C=CCN2CCCC2)C1 CC1CCCn2cc(-c3nc(COc4cccnc4)nn3-c3ccnnc3)nc21 N1(C(C2(COC(C)C)CC2)=O)CCCC(F)(CNC(=O)CC2SC(=N)NC2=O)C1 Nc1ccc2oc(C(N3CCC(CNC(c4cnc5n4CCC5)=O)C3)=O)cc2c1 C12(CC(N3CCC(C=C)C3)=O)CCC1CN(C(c1c(CC)cnn1C)=O)C2 CCCC(C)(CC)C(=O)NC1COCC1CNC(=O)C=CCO C(C)(C)(CC(F)C(=O)NCc1n[nH]c2c1CCC2)NC(CCNC(=O)NC)=O C1(C)(C(=O)NCC2(C)CC(C)C2)C=CCN1C(C1CCCC1F)=O C1(N(C(=O)CC2CCOC2)C)CCCN(C(C2(C)CC2(Cl)Cl)=O)CC1 C(=O)(C1CCc2cc(F)ccc21)C(C1CC(O)C1)=O.C1(CN)CCCCCN1C=O CC(=O)CCN=C(NCC1(CO)CCCOC1)NCC(c1cccc(Cl)c1)(C)O CC1CCCC1(C(=O)NCCc1cn[nH]c1)NC(=O)CCC(C)N(C)C C(=O)(C(O)C(C)CC)NCCC1(NC(CNC(COC)=O)=O)CCCC1 C(C(COC)C(=O)NCC(C1CCCN1C(=O)C(=O)NCC(F)F)(C)C)OC C1(NC(Cc2ccc(C)s2)=O)CCC(C)N(C(c2sc(C)cc2C)=O)C1 N1(C(c2cc(-c3cccs3)cs2)C(=O)NC(CC)C)CCC(C)C2(CCC2)C1 C1(NC(=O)C(Cc2cc[nH]n2)NC(C2CCSC2)=O)CC(C2CC2)C1 C(CN=C(NCC1CCCN(S(C)(=O)=O)C1)NC(C)C1CC1)c1c(C)cn(C)n1 C1(C#N)(CNC(c2n(CCOCC)nnn2)C(=Cc2ccco2)C)CCOCC1 c1(C(N(CCCNC(=O)C(F)CC2CC2)C2CC2)=O)nccn2nccc12 C1(NC(CN(C)CCO)=O)CCC(N(C(=O)Cn2nnc(C3CC3)n2)C)C1 CC1=Cc2ccccc2C1CC(=O)N1CCOCC1CNC(C1CCC(=O)O1)=O c1(CC)cn2c(C(=O)NC(C)C(C(C)C)NC(C3COCCO3)=O)cccc2n1 C1(C(=O)NCC(CN(C(c2ccnc(C)c2C)=O)C)(C)C)CCC2(CCOC2)O1 CC1(C)CCN(C(=O)Cc2cccnc2O)CC1CNC(c1cccc(=O)o1)=O Cc1cc2c(C(=O)NCC3(F)CC(NC(c4cc[nH]c(=N)c4)=O)C3)cccc2o1 C(C)(CC(C)(C)CO)NC(CC1C2CN(C(c3ccnc(C)n3)=O)CC21)=O c1(NC(CCC2CCN(C(CN(CCOC)C)=O)C2)=O)cc(O)ccc1F C1(C(N(C)CCOCCO)=O)CCCC12CCN(C(=O)Nc1cscn1)C2 C=CCC(C(=O)NCC(C)(C1CC1)OC)NC(=O)C=CC(C)(C)C Cc1[nH]nc2cc(C(N3CC(O)C(O)C3CNC(c3ccn(C)n3)=O)=O)ccc12 CC1CN2CCC1C2=O.C(CCS(=O)(=O)N(C)C)NC(=O)CC1CC1(C)C C=CCCC(CC(C)C)C(=O)N1CCN(C(=O)CC2(C#N)CC2)CC1CO N1(C(c2n(CC)c(O)nc2)=O)CCN(C(c2ccc(N)cc2F)=O)C2CC12 c1(OCCC(=O)NC(c2ccccn2)CNC(=O)Cc2cnns2)ccccc1 C(=O)(CCC(C)(C)C(=O)N1C2CCC1CN(C(=O)CC1(O)CC1)CC2)OC N1(C(C(F)=CC)=O)CCC(n2cccn2)(CNC(=O)CC2(N(C)C)CCCC2)C1 c1(C(=O)NC2CN(C(C)=O)CC2c2ccccc2F)nc(C)c(C)nc1C c1(CC(c2n(CC)nnn2)NCCNc2ccc(Cl)cc2Cl)cc2ccccc2o1 c1(C(N2CCC(NC(c3onc(C)c3C)=O)C2)=O)ccc(P(C)(C)=O)cc1 CC(=O)CCN=C(NCc1cc2ccccc2o1)N1CCS(=O)(=O)CC1 c1(C2C(C(=O)N(CCCNC(=O)C(F)=CCF)CC3CCCO3)C2)ccccc1 C(CCCC(c1nnnn1CCC1(C)CC1)NCc1ccno1)OC CC(C(CO)NC(=O)Cn1ccc(=N)[nH]1)NC(=O)CC1(n2cncn2)CC1 CC1(C)CN(CCCC(CC2CC(NCC(=O)NCC(CC3CC3)CO)C2)=O)C1 CC(C)C(CC(=O)N1CC2CCCC2(NC(C2CN3CCC2CC3)=O)C1)C(C)C CN(C)NC(=O)CCC(=O)NCC1CCN1C(C1CCS1(=O)=O)=O Cc1nc2n(n1)CCN(C(=O)C(C(C)C)NC(=O)C1=C(Cl)CCOC1)C2 C(=O)(C(C)C(O)CC)N(CCN(C)CC)C1CC1.c12ccc(cc1)-c1noc(n1)C2 c1(C(=O)NCCN(C(=O)CC(C)C)CCOCC)cc(C)cc(Br)c1O N1(C(C=Cc2ccc(CC)cc2)=O)CCCC2(NC(=O)CS(=O)(=O)NC)CC2C1 N1(C(c2csc(C(F)F)n2)C(=O)NCCC2CC2)CCN(c2cncnc2)CC1 C12(C(N3C(CNC(C(C(C)C)C)=O)COCC3)=O)C3CC(CC13)C2(F)F C#CCCCC(=O)N1CCC(CCOC)(NC(=O)C(CO)OC)C1 C1(C(=O)NCc2cccc(NC(=O)CCC(C)SC)c2)(CC)CC(C)(C)C1 C(C(CNC(C1(OC)CCCC1)=O)CO)NC(CC=CCC)=O C12(NC(COCCCC#C)=O)CCN(C(=O)CS(=O)C(F)(F)F)CC1C2 O=C(C1CCCn2cnnc21)NCCCCCNC(C1OCCOC12CCC2)=O c1(OC)cncc(C(=O)NC2CCC(CCNC(c3nccn3C)=O)C2)c1 C(C1=CCN(C(c2snc(Cl)c2Cl)=O)CC1)NC(c1cc(C2CC2)ccn1)=O N1(C(C=CSC)=O)CCN(C(C23COC(CF)(C2)C3)=O)C(C)C1 CC1CN(C(=O)CCc2csc(=N)[nH]2)CCN1C(=O)C#CC1CCC1 c1(C(=O)NCCS(C)(=O)=O)n[nH]c2c1CN(C(c1cc[nH]n1)=O)C2 CC1(C(N2CCC(C)(CCNC(=O)Cn3nccn3)C2)=O)CCCOC1 Cc1cccc2cc(C(N3CCCCC3CN(C)C(C3(N(C)C)CC3)=O)=O)cnc12 C(CC)(CC(=O)N1CC=CC1COC)NC(CC=CC=C)=O N1(C(Cn2ccc(C)n2)=O)CCC(CNC(=O)CCc2cc(C)nn2C)C(O)C1 CCC(CCCC(=O)N1CCC(CO)C(C)C1)NC(=O)CCP(C)(C)=O CC1CCC(C)(C(N2CC(NC(=O)C=CC3CCCO3)C(C)C2)=O)C1(C)C c1(C(=O)OC(C)(C)C)csc(CC=CC)n1.C(CC(C)SC)N(C(C)=O)CC C(CC)(c1ccccc1)=CC(=O)NC(CC#C)C(=O)NCCC(C)N1CCC1 c1(C(=O)NC2C(NC(CCOCCCOC)=O)CCOC2)cc2sc(Cl)cc2[nH]1 c1(NCC(C(CC)C)O)ccc(S(=O)(=O)NCc2c(C)cc(C)cc2C)cc1Br c1(CC)cc(Cl)ccc1C(=O)OC(CN(C)C)C(F)(F)F c1(OCCN(C)C(C2CCCCN2C(=O)C=Cc2ccoc2)=O)ccc(F)cc1 N1(C(C2C(C=C)C2)=O)CCN(C(=O)C(C)(C)n2ccnn2)CC1CCC C1(CNC(c2ccccc2OC(F)(F)F)C)CCCC2(CCC2)O1 N1(CC=C)CCN(C(CNC(c2cscc2C)C(=O)NC2CC2)C(=O)OC)CC1 C1(OC)CC(CNC(C2CC2F)=O)N(C(=O)C(C)CSC(F)(F)F)C1 C1(C(=O)NCC2CC(O)CN2C(=O)Cc2ccsc2Cl)CCC=CCCC1 c1(C(=O)NC(CCN(C(c2c(C)cco2)=O)C)C(C)C)cccc(Cl)c1F c1(C(C)OC)nc(-c2cc(C(C)(F)F)cs2)n(-c2ccc(F)nc2)n1 CC1CCC(CNC(C2(N(C)C)CC2)=O)CN1C(=O)CCCn1c(O)nnc1O c1(C(N2C(CNC(C(C#C)(C)C)=O)CC(C)(C)C2)=O)cc(C)cc(Cl)c1N CCC(CC)C(C)ONC(C1COCCN1OC(C1CN(C)C(=O)N1)=O)=O c1(C(=O)NC(CSCC)C(=O)Nc2ccccc2)cnc(O)c(C)c1 N1(C(C2(COC)COC2)=O)CCCCC1C(=O)Nc1cccc(C)n1 Cc1c(C(=O)NC(CNC(C2CC2C2CCCC2)=O)(CO)CO)sc2nccn12 S(=O)(=O)(c1ccccc1F)N1CCN(CC(=O)N)CC1.N1(C(C(C)O)=O)CCCC1CN N1(CCNC(=O)NC(C(C)C)c2cccs2)C(=O)NC2(CCc3ccccc32)C1=O CC(C)CC(C(=O)N1CCC(C(C)NC(c2cc([N+](=O)[O-])c[nH]2)=O)CC1)C(N)=O Cc1oc(C#N)cc1C(=O)NCCCOC1CCN(C(=O)CC(C)CF)CC1 c1(CN(C(C(=O)NCC(CC)O)=O)C(C)C2CC2)ccc(N2CCCC2=O)cc1 CC#CCCCC(=O)N1CCC(CC(N)=O)(NC(C2CC3(CCC3O)C2)=O)CC1 c1(SC)cc(C(N2CCC(C(C)NC(=O)CCC(N)=O)C2)=O)c(C)o1 C1(C(N2CCN(C(C3OCC(C)(C)C3)=O)CC2)=O)CC2CCC(C1)O2 C1(OCC)CCN(C)C(C)CNC1=O.C1(C(CC)CC)CC(SC)C1 c1(NC)cc(C(N2CCC2CNC(C2CC(C)=NO2)=O)=O)cc(C2CC2)c1 CC1OC2CCC1(NC(=O)CC1CC(F)CN1C(=O)C(C)NC=O)C2 C1(NC(c2c(C)oc(C(C)C)c2)=O)CN(C(=O)CSc2cnn(C)c2)C(C)(C)C1 N1(C(c2nnn(CC)c2C)=O)CCC(CNC(c2cccc(=O)o2)=O)C(C)C1 c1(NCC(c2ccc(C(C)C)cc2)O)cnc2ccc(F)cc2n1 C1(NC(C(=O)NCCOCCCC)=O)CCCCCN1C(=O)CNC(C)=O N1(C(CCCn2c(C)ncc2)=O)CC2CN(S(=O)(=O)C(Cl)(Cl)Cl)C2C1 C(=O)(C(CC1CC1)NC(=O)C(n1nccc1C)C)NCC1CC(CSC)C1 N1(C(c2ccc(C)c(I)c2)=O)CCC(C)N(C(C2CCCCS2)=O)CC1 c1(OCC(=O)NCCC2(O)CN(C(=O)C(F)C3CC3)C2)ccc2c(c1)CCCC2 C(CNC(C1(N=[N+]=[N-])CC1)=O)(CC(C)C)NC(C(C)NC(C)=O)=O C1(C#N)(C(N(C(C)CCNC(c2c[nH]nc2C(C)(C)C)=O)C)=O)CCCOC1 C1(OCC)CC(C(N2CCOCC2CC)=O)(OC)C1(C)C N1(C(C2C(OCC)C2)=O)CC(C)CN(C(=O)C=C2CCOCC2)C(C)C1 C12(CC)CC(CO)(C1)OC21CN(C(=O)CC(=O)NC)C1.C1(=O)C=CCN1 c1(C(N2CCC(NC(CC3CCC(C)(C)C3)=O)(CF)C2)=O)nnc(O)nc1O C1(C(=O)NCC(C)NC(=O)CC2CN3CCN2CC3)CN2CCCC1CC2 Cc1cc(C)c(C=CC(=O)NC2CCC(NC(=O)CC3CS(=O)(=O)C3)C2)cc1C N1(C(C2(CNC(c3ccccc3F)=O)CC(=C)C2)=O)CC2(CCNC2=O)C1 CC1(C)CCC(C(=O)NCC(C)(C2CC2)NC(=O)Cc2ccncc2Cl)C1 N1(C(c2cnc(CC)o2)=O)CC(F)CC1CNC(c1ccn(C2CC2)n1)=O C(=O)(C(C)(C)C(F)c1ccccc1)NCC(C)CN(C(=O)CCc1nc[nH]n1)C C1(C(=O)NCCNC(c2ccoc2)=O)C=CCN1C(=O)CCCn1ccnn1 C(=O)(N1OC2CCC1CC2)c1nc(C(C)NC(=O)CCCCCF)oc1 c1(C(=O)NC(C)C(CO)NC(=O)Cc2ccccc2F)nnn2c1C(=O)NCC2 CC#CC1CCN(C(c2cnc(OC)nc2)C(=O)NC(C)CC)C1 Cc1ncc(Cl)c(C(=O)NCC2CCN(C(c3cc4[nH]ccc4s3)=O)CC2C)n1 C1(CNC(CP(C)(C)=O)=O)CN(C(C2CC(=O)NC(=O)C2)=O)C2CCN1C2 C1(C(=O)NCC2N(C(CNC(C)=O)=O)CC(C)(C)CC2)CCc2ccccc2O1 C1(NC(c2c(C)n[nH]c2)=O)CCN(C(c2[nH]nnc2C2CC2)=O)C(C2CC2)C1 C1CCC(C)NC(=O)COC2(CC2)C(=O)N1.c1(COC(C)C)n[nH]c(O)n1 C1(C)CC(=O)N(C)C1.C1(CCC(=O)NCC)CCCCN(C(=O)CSCCOC)C1 Cc1[nH]c(C(N2CC(NC(=O)CC3CC(=O)NC3=O)C(C)C2)=O)c(C)c1C c1(OC)noc(C2CC2)c1C(=O)N(C1CC(NC(c2cc(C(N)=O)co2)=O)C1)C C(=O)(CCCCC(=O)NC1CC(C)(CNC(C2CC=CCC2)=O)C1)OC CC1OCCCC1C(N1CC(CC(C)(C)CNC(c2sccc2Cl)=O)C1)=O C(CCC(=O)NC(C1CCCC1)CNC(C1(CNC)C=CCC1)=O)OCC=C.C1CC1 Cc1ccc(C)c(C(=O)NCC(C2CC2)NC(=O)C(C(C)C)NC(N)=O)c1 c1(NC2CCN(C(Cc3c(C)cccn3)=O)C2)ncnc2sc3ccccc3c12 N1(C(c2c(C(C)(C)C)ncs2)=O)CCN(C(c2ccc(Cl)c(F)c2)=O)C2CCC12 Cc1noc(C2CC(C(=O)NC(C)CN(C(=O)C(C)n3ccnn3)C)C2)n1 c1(-c2c(CC)cccc2)cc(C(=O)NCCCC)nc(C(F)(F)F)n1 C(=O)(C(C(C)N(C)C)c1ccccc1)NC(C)CSC.C1(=O)CN1C(C)(C)C.CO Cc1cc(N)c(C(N2CCC(NC(C3(C(F)(F)F)CCC3)=O)C(O)C2)=O)c(F)c1 N1(CC(COC)(F)F)CCC(=O)N(CC(C)(C)C(c2ccccc2)OC)C1=O CC1CN(C(=O)Cn2ccc(C(F)(F)F)n2)CC1NC(C1(C(F)F)CCCO1)=O N1(CC(=O)NC2C(C)CCOC2)C(=O)NC2(CCCC(C)(C)C2)C1=O c1(C(=O)NCc2occ(C(=O)COC)n2)ccc(CN)cn1.C(C)(C)(C)OCC c1(C(N2C(C(=O)NCc3ccnc(Cl)c3F)COCC2)=O)ccc(Cl)c(Cl)c1Cl N1(CCC(C)(C)C)CCCC(C2CCCN(C(=O)OCC(C)C)C2)C1 C1(CNC(c2c(CC)c[nH]c2)=O)CC2CC1CN2C(=O)CCc1ccc(N)cn1 c1(OC)cccnc1C(=O)NCCC1CCC(NC(=O)Cc2cnsc2)C1 C1(C(=O)NCCCCCCO)COc2cc(Br)ccc2O1 c1cc2c(s1)CCC(NC1C3CC3C3CC13)C2 n1(CCN(C)CC2CC2(C)C)cc2ccccc2n1 CC(C)(C)C(C(=O)NCc1conc1C(=O)O)NC(C1CNC(=O)C1)=O c1(C(=O)NC(CNC(Cn2nnc(C)n2)=O)CC(F)(F)F)ccc2nc[nH]c2c1 CC(C)CCC(=O)C(=O)NC1CC2(C1)CC2C(N1CCC(O)C(C)C1)=O O=S(=O)(c1ccc(N2CCCC(CCF)C2)c(Br)c1)NC1CCN(CCO)C1 c1(C(=O)NCC(CC)NC(=O)C(O)C2CC2)ccc(O)c(C(C)=O)c1 C(CCC(=O)NC(c1ncccn1)C)NC(C=CC=CCC)=O C1(CN(C(=O)Cn2ccccc2=O)C)COCCN1C(c1csnn1)=O CC1(C)CCCC1C(=O)NCC(C)(C1CC1)NC(c1ccon1)=O CC(CN(C)C)CC(=O)N1CC(C2CN(C(=O)C(C3(O)CCOCC3)O)CCO2)C1 C=Cc1ccc(C(=O)NCC2CN(C(c3cc4scnc4[nH]3)=O)C2)cc1 N=c1cc(C(N2CCCC2c2c(F)cccc2Cl)=O)c(F)c[nH]1 C12(C(=O)NC(COC)CO)CCC(CC1)N(C(C1C=CCC1)=O)C2 C(=O)(CC(C)C(=O)N1CCC(C)(CNC(=O)CCOCC(F)F)C1)OCC CC(C)C(CNC(=O)COCCc1ccc(Cl)s1)NC(=O)C(C)CC1CCCC1 CCC(C)C(C(=O)NC1COCC1O)NC(=O)CCN1CCCCC1 c1(CC)nncn1NC(=O)C(CNC=O)NC(C1C2(CC2)C12CC2)=O CC(C)C(F)(F)CC(=O)N(CCCCN(C)C(c1ccc(SC(F)(F)F)o1)=O)C c1(C(N2C(CNC(C3OCCN(C)C3=O)=O)CCCC2)=O)coc(S(N)(=O)=O)c1 c1(C(=O)OCCOC23CC2COC32CCC2)cc2c(Br)ccc(Br)c2[nH]1 c1(C(=O)NC2C=CCN(C(C(CC)C#N)=O)C2)cc(Cl)ccc1O N1(C(C2(CCC)CC2)=O)CC(NC(c2c[nH]ccc2=O)=O)C(S(C)(=O)=O)C1 CCC(C)(O)C(=O)NCC(C1CC1)NC(=O)Cc1nncn1C(C)C C1(C(=O)NC2(C(F)(F)F)CC3CCC2C3)CCC12CCOCC2 C1(NC(C(OC)OC)=O)C2CC3C(C2)C13C(N1CCC(F)(CF)C1)=O C(CN=c1[nH]c(-c2ccccc2)ncc1C(=O)OC)C1CN(C(CC=CC=C)=O)C1 c1(C(=O)NC2C=CCN(C(CSCC(=O)OC)=O)C2)ccc(F)c(F)c1F N1(C(CNC(C)=O)=O)CCC(=CCNC(C2CCCC2CC(C)(C)C)=O)CC1 c1(CN2C(C(=O)Nc3cc(F)ccc3Cl)CC(=C)C2)ccc2cc[nH]c2c1 C1(CC(=O)NCC(C2CC2)NC(=O)C=CCn2cncn2)CC(O)C12CCC2 C1(NC(c2nc(C)n(C)c2)=O)CCCCN(C(C2OCC3CCCC23)=O)C1 c1(C(C(C(c2cccs2)NC(=O)CNCC(F)(F)F)=O)=O)csc(CN)n1 N1(C(c2nc(CC)sc2)=O)CCC(CN(C(=O)CNC(=O)CC(C)(C)C)C)CC1 N1(C(CC(CCCC)O)=O)C2CCCC1CC(NC(c1ccc(F)cc1O)=O)C2 C#CC1(C(N2CC(N(C)C)C(CNC(C3CC3F)=O)C2)=O)CCCC1 CC1CC(=O)NCC1C(=O)N(C1CN(C(c2cc(C(C)C)sn2)=O)C1)C C1(NC(CCC#CC)=O)C2CC1CN(C(=O)C=CCn1cncn1)C2 c1(CC(=O)NC(CNC(C=C(C)C(C)(C)C)=O)C(C)(C)C)ccc(Br)c(Cl)c1 C(=O)(C(O)CC[S+](C)C)N(C1CCCN(C(C=C(CC)C)=O)C1)C CCCCC(O)CC(=O)NC1(C)CCCCC1C(N1CC(O)(CCO)C1)=O CC1(C)Cc2[nH]nc(C(N3CCC(NC(=O)C4=CC(O)CCC4)C(F)C3)=O)c2C1 N1(C(C2C(C)CCC2)=O)CC2(CCC(NC(=O)CC3CCOCC3)CC2)C1 C#Cc1cnn(C)c1C(=O)NCCCOCCCNC(c1ccc(=O)n(C)n1)=O C=CCC(CC(=O)N1CCC1c1cn(CC(C)(C)CC(C)O)nn1)SC.C(C)(C)C C1(C(N2CC(O)(CNC(C(C)(C)N3CCCC3)=O)C2)=O)CCCCN1CC(F)F C(c1ccc(F)c(OC)c1)=CC(N1C(CNC(C(C)=CC)=O)CC(O)C1)=O N1(C(C(CCC)F)=O)CC(NC(=O)Cc2ccc(O)cc2Cl)CC12CCCC2 C1(NC(C(C)Cn2cccn2)=O)C2CC1N(C(=O)Cc1ccccc1C(F)(F)F)C2 c1(C(N(c2ncc(C(C)=O)o2)C)=O)ccc2c(c1)C(=O)CCC2 C1(C(C)C)C(=O)NCCN1C(C1(C)CCN(C(=O)CN2CCOCC2=O)C1)=O C1(CC(=O)NCCCCC2CC2)C2CN(C(C3CC3[N+](=O)[O-])=O)CC12 C1(C(N2C(CN(C(COCCC(C)C)=O)C)CCC2)=O)CCN(C)C(=O)C1 N1(C(CS(CC)(=O)=O)=O)CC2(CCCC2)C1C(=O)NC1CC2CCC1O2 c1(C2(C(=O)NCCCNC(C(=O)NC)=O)CC2)ncc(C)o1 c1(CN2CCC(C(=O)NCC3CN(C)C3)C2)cc(Br)ccc1O N1(C(CC(COC)(C)C)=O)CC(C2CN(C(C3CC3C)=O)C2)C1 N1(C(COCCC=C(C)C)=O)CCCCC1C1CCCN(C(=O)CO)C1 c1(CC(N2C(C)C(NC(=O)CCN3CCC3)CC2)=O)cc(F)ccc1F C1(NC(Cc2cnc(C)s2)=O)CC12CC(NC(=O)C(O)C(C)C)C2 C(=O)(C(CC(C)C)c1ccc(Cl)cc1)NC(CC)CNC(=O)CCc1cccn1C c1(OCC(=O)N(C2CCN(C(c3n[nH]cc3C3CCC3)=O)C2)C)ccccc1 C1(CNC(C2CCC=CCC2)=O)CCCCN(C(C2CC2C2CC2)=O)C1 CCC(C(=O)NC1CC(C(=O)NC(CC)CCC(=O)OC)C1)C(C)(C)CC C(CN=C(NCC1COCC1O)NC1CCC(=O)NC1)NS(C)(=O)=O c1(CC)ccnc(C(=O)NC(C2CCCN2C(=O)Cc2sc(C)nc2C)C)c1 C1(CCNC(c2c(C)scn2)=O)CN(C(C2CC3(C2)OCCO3)=O)CCCO1 C(=O)(CCCN(C)N=O)N1C2(CNC(CCN3C(C)CCCC3)=O)CC(C1)C2 c1(C(=O)NC2(C)CCN(c3snc(SC)n3)C2)nc(C2CC2)ncc1Cl C(N=c1[nH]c(=NC)[nH]c(=NCC2CCCC(CC)CC2)[nH]1)C1C(=C)C1 c1(CC)c(N2CCC(CNC(c3ccc(C(C)=O)c(C)c3)=O)C2)ncnc1Cl c1(C(N(C2CCCN(C(C3(C#C)CC3)=O)CC2)C)=O)nc(C)[nH]c2nccc1-2 c1(C(=O)NCC2CCCCN(C(C(C)CF)=O)C2)cc2cccc(Br)n2c1 c1(CC(=O)NCC2N(C(C(CC=C)CC)=O)CC(O)C2)cccc([N+](=O)[O-])c1 c1(COC)ncc(C(=O)NCC(CO)NC(c2nnc(C)s2)=O)c(O)n1 C12(NC(CCc3cccc(OC)c3)=O)CCN(C(C3CCCCC3)=O)CCC1C2 NS(=O)(=O)C1CCc2ccccc2C1NCc1cc(Br)ccn1 N#Cc1cncc(C(=O)NC(C(=O)O)C(F)(F)F)c1 C(=O)(C1CCCc2nc[nH]c21)N(C1C(N(C(c2c(C)snn2)=O)C)CCCC1)C C1(C(=O)Nc2ccccc2Cl)CN(C(=O)C=CCOc2ccccc2)CC1O c1(C(=O)NC2CCC(N(C)C(c3cc(F)c[nH]3)=O)CC2)cc(O)c2sccc2c1 C(CC(=O)N1CC=C(CO)CC1)(C(C)(C)C)NC(C1C(C)(C)C1(F)F)=O Cc1nc(NC(C2CSC2)C)cc(=NCc2ccc(OCC(N)=O)nc2)[nH]1 CN=c1[nH]c(C(N2CCC(NC(=O)C(c3cncn3C)N(C)C)C2)=O)cs1 Cc1ccnnc1C(=O)NC1CCCC(CN(C(=O)CC(C)(F)F)C)C1 c1(-c2n(C)ncn2)ccc(Cl)cc1C(=O)OCc1ccc(-c2ccno2)cc1 C1(CNC(CC2(NC(c3cc(CCC)nn3C)=O)CCC2)=O)CCOC(C)(C)C1 C1(C(=O)NC(C)CNC(=O)C(c2ccccc2)C)COC2(CO)CC1C2 n1(CCC)nc(C)c(C(=O)NC(C2(CNC(C3COC(=O)N3)=O)CC2)C)c1C C1(C2(NC(C=CC(C)=O)=O)CC2)CCCCN1C(=O)CCn1cc(Cl)cn1 CC1CC(C(N2CCOC(C)(CNC(c3ncccc3CO)=O)C2)=O)CCN1C N1(C(c2nc(C(C)OC)oc2)=O)CCN(C(=O)CSc2cnn(C)c2)CCC1C c1(OC)cc(Cl)cc2[nH]c(NCC(=O)NC(c3ccc(F)cc3)C)cc12 c1(C(N2CCC(NC(C(C=C)(F)F)=O)CC2)=O)cc(C)c(C)c(F)c1 C=CCC(F)(F)C(=O)NCC1CC(NC(=O)C(CCF)NC(=O)OC(C)(C)C)C1 N1(S(CCOC)(=O)=O)CCN2CCNCC2C1 O=C(CCCCNC(c1cc(C2CCC2)[nH]n1)=O)NCC1CCOC1=O c1(NC(C2C(C)CCN(C(=O)C=CCOCCO)C2)=O)ccc(Cl)c(C#N)c1 c12ccc(C)cc1S(=O)(=O)N1CC(CCC1C)O2.C(CN=[N+]=[N-])OC C(=O)(C(C#N)C(C)(C)C)NC(CC#C)CC(=O)NCCC1CC(F)(F)C1 C1(C(=O)NCCC2(NC(CN3CC(CC)C3)=O)CCC2)CCOC(C)C1 N1(C(CNC(CC(C)(C)C)=O)=O)CCCC(C)(CNC(=O)COC2CCOC2)C1 C(CC(C(=O)N(C1CC1)CC1CCCN1C(c1ccn(C)n1)=O)N(C)C)N(C)C N1(Cc2cncc(-c3ccc(C(=O)OC)cc3)c2)CC2CC(F)CC2C1 Cc1cc(N)cnc1C(N1CCC(C(O)CNC(=O)C(C(C)C)NC=O)CC1)=O c1(C(N2C(C)CC(CNC(c3c(Cl)ncc(C)c3)=O)C2)=O)ccc(S(C)=O)cc1 C1(CC(=O)N(C(CC)C)CC2CCNCC2)Cc2ccccc2C1 N1(C(c2nccc(CNC(C3C(C)(C)C3(F)F)=O)c2)=O)CCCC(O)CC1 C1(NC(C2CCC2)=O)CCCN(C(=O)CSc2ccc(OC3CCC3)cc2)CC1 C1(NC(=O)CCF)CN(C(c2cccc3ccoc23)=O)C2(CCCOC2)C1 CC1NC(=O)CCC1CNC(C1CC2(CC2)CN1C(c1cncn1C)=O)=O C12=CC=C(C=C1)C2.Cc1ccsc1N1CCC(OCC(F)F)C1 C=CC(C(=O)N1CC(O)(CNC(C2CC(F)C2)=O)C1)OC S(=O)(=O)(c1cccc(C(N2CCCC2C(C)(C)O)=O)c1)NC(C(C)C)C1CC1 c1(NC(=O)NC(c2ncc(C(C)(C)C)o2)C)ccc(N2CCOCC2)nc1 N1(C(C2(C#C)CC(=O)C2)=O)CCC(C)C(CC(=O)NCCN2CCOCC2=O)C1 c1(C(N2C(C(=O)NCC(C)CCO)CCC2)=O)cccc(-n2ccnc2)c1 c1(C(C(N2CCC(CNC(c3c(CC)cncc3)=O)C2)=O)O)cccc(C)c1F Cn1c(C(=O)NCC(C2CCCC2)NC(=O)COC2CCOC2)ccc1[N+](=O)[O-] c1(C(C)(C)C(=O)NCCCNC(c2ccn(CC(F)F)n2)=O)c(F)cccc1F c1(C(=O)O)cnc[nH]c1=Nc1ccc(C2(O)CC2)nc1 C1(n2ccnc2CN2CCCC2c2cccc(C(=O)O)c2)(CC#C)CC=CCC1 c1(CNC(C2CC(NC(COC)=O)C2)=O)ccnc(O)n1.C1(C)CC1 Cc1sc2cncn2c1C(=O)NCC(=O)NCc1ccc(C(F)F)o1 c1(CN(c2ccc(F)cn2)C(N2CCC(O)CC2)=O)ccc2sc3ccccc3c2c1 C1(OCC(=O)N(C2CCC2)C)CCC(NC(=O)CCc2c[nH]c(=N)[nH]2)CC1 c1(NC(C2CCN(Cc3ccc4ncoc4c3)CC2O)=O)cc(Cl)cc(Cl)c1Cl C1(NC(=O)CN2CC=CC2)CCCCN(C(C2(Cc3ccccn3)CC2)=O)C1 C(=O)(C1=CCCC1C)NC1C(OC)CN(C(=O)Cc2nocc2C(C)C)C1 c1(Cc2ncc(C(N(CC)CC3CCN(C4CCNC4)C3)=O)s2)ccccc1F N1(C(C2CC(C)(C)O2)=O)CCC2(CC2C(=O)Nc2ccnc(C3CC3)n2)C1 N1(C(c2cnc(N3CCN(C)CC3)nc2)=O)CC=C(CNC(=O)C2=CCC2)CC1 N1(C(CCCC)=O)CC2CCCC1C2CNC(c1ccc(-n2cnnn2)cc1)=O CC(C)CCCCC(=O)N(C1CCCC1)CC1CCCO1 C(CCCCNC(C1CCC(=O)N1)=O)N(C(CCOC(C)C)=O)C C1(NC(Cc2scc(C)c2)=O)CC2(C1)CC2NC(c1nc(C2CC2)oc1C)=O CCCN=c1[nH]c(N2CCCC(C(C)(C)C)C2)nc2cccnc12 c1(C(N(C2CN(C(=O)CCC3CCOC3)C2)C)=O)ccc2c(c1)NC(=O)C2 C(=O)(C(C)(C)CC(C)(C)C)N1CC(C(N(CC(CC)(C)OC)C)=O)C(C(C)C)C1 C1(CN(C)S(N)(=O)=O)CCC2(CCC2)C1CNC(=O)C1CC1.C1(=O)CN1.C(N)=O c1(C(N(CCCCNC(C2(C(F)(F)F)CCC2)=O)C)=O)cc2cccc(F)c2s1 c1(C(N2CCCC(N(C(C(C)O)=O)CCO)CC2)=O)ccc(P(C)(C)=O)s1 C(C)(C)(CCCNC(C1CC(n2cnnc2)C1)=O)NC(C1CCC(OC)C1)=O c1(C(=O)NCC(C(C)C)NC(C2(CCC)CCC2)=O)cccc2c1nc(O)n2C c1(Oc2ccccc2)nc(F)ccc1Br.O=C1CC(c2cccs2)N1 N1(C(C2(OC)CC(C)C2)=O)CC(C(=O)NCCn2ccnn2)C(C)C1 CC1(CNC(=O)CCC2(NC(=O)C(N)=O)CCC2)CC1(F)F Cc1cccc2c1OC(C(=O)NCCCCCCNC(C1(C(C)C)COC1)=O)C2 N1(C(c2c(C)sc(O)n2)=O)CCC(F)C(NC(c2cc3sccc3s2)=O)C1 Cc1ccc(F)cc1C(N1CC2CC1C2NC(C1CC2CC2CC1C)=O)=O N1(C(CCCC(C)C)=O)CCN(C(c2cnc3n2CCCC3)=O)CC(C)(F)C1 N1(C(C=Cc2cn(C)nc2)=O)CCN(C(c2csc3nccn23)=O)C2(CCC2)C1 Cc1cc(C(=O)NC2(CNC(=O)CCCC3CCOCC3)CCC2)no1 CC1COC(C(=O)NC2(C)CC(NC(=O)CSc3n[nH]c(O)n3)C2)C1 C(CC(=O)NCCNC(=O)CC1(NC(C)=O)CC1)(OCC)OCC C1(C(N2CC(C)(CNC(C3(C(=O)OCC)CCC3)=O)C2)=O)CC12CCOCC2 C1(NC(=O)C(c2ccc(F)cc2)F)CCC12CN(C(=O)CC1COCCOC1)C2 N1(C(C(C)N(C)C)=O)CCC(NC(C2C=CCCC2)=O)C12CCC2 c1(C(N(C)CC2CCCC(NC(=O)Cn3cncn3)C2)=O)c[nH]nc1S(N)(=O)=O c1(C(=O)NCCCN2CCN(c3nc(C4CC4)ns3)CC2)nc2c(o1)CCCC2 C=C(C)CC1C(=O)N1.C1(=CC(=O)NCC=C)CCN(C(C2CC2(F)Cl)=O)CC1 C#Cc1ccc(NC(=O)NCC(c2ccc(OC(F)(F)F)cc2)(F)F)c(C)c1 CC(CNC(=O)CNC(=O)C(CO)OC)C(C)(F)F.c1ccccc1 CC(C)(F)C(=O)NCCOC1CCN(C(=O)CN2CCOC2=O)C1 Cc1cc(C(N2CCOC(C(C)(C)O)C2)=O)ccc1Br.N12CCC(O)(CC1)C2=O C1(NC(C(CC)(C)O)=O)CC2CCC1CC2NC(=O)CC1COC(C)(C)CO1 N1(C(N)=O)CCCCC1C(N1CCC(NC(c2ccno2)=O)C1)=O C1(NC(C2(CC#C)CCC2)=O)CC2CC(C1)N(Cc1ccc(F)cc1)C2 N1(c2ncc(C)cn2)CC23CCCC2(CN(C(=O)Cc2csc(C)n2)C3)C1 N1(C(CCCOCCC)=O)CCN(C(C2CCCC(=O)N2)=O)C(CC(F)F)C1 c1(C(N(CCC(=O)NCC2(CC#C)CCCC2)C)=O)ncccc1O C(CN=C(NCCC(=O)C(C)(C)C)N1CCC(c2cccc(Cl)c2)C1)C(C)O.OC C1(NC(c2cnc(C)o2)=O)CCC12CN(C(=O)COCc1ccccn1)C2 c1(C(N(C(=O)CC2=CCNCC2)c2ccc(CC)cc2)=O)cc2scc(Cl)c2[nH]1 c1(C(=O)NCC2C3CN(C(C(CCC)C#N)=O)C2C3)cccc2c1OCCO2 C1(N(C)C)CN(C(C(=O)NCc2ccc(F)cc2)C2CCOC2)CC1C1CC1 C1(CC(=O)N(CCOCCOC)C)CC(C)(C)CN1C(=O)CCN1CCCCC1 c1(C(N(C2CCN(C(c3c(C)nc(C(C)C)s3)=O)CC2)C)=O)c(O)cccc1O CN1CC(C)(C(=O)N(CCCNC(C2C3CCC(C3)C2(C)C)=O)CCO)CCC1=O C1(NC(c2cccc(SCC)c2)=O)CCN(C(=O)CCc2ncc[nH]2)C(C2CC2)C1 N1(Cc2cccc(CCC)c2)Cc2c(C(=O)O)ccc(F)c2C1 CC(O)C(C(=O)N=S(C)(=O)c1cnn(C)c1)NC(c1ccco1)=O C#CCCC(O)C(=O)NCC(CNC(c1occ2c1CCC2)=O)C(F)(F)F N1(C(C2(c3nc(C)c(C4CCC(C)(C)OC4)o3)CC2)=O)CCC(C)(C)C1C N1(CC(C)(N)C2CCCC2)CCCN(N2CCOCC2)CC1 C1(NC(C2(OC)CC2)=O)CC(C)N(C(c2conc2C)=O)C1 C1(C)(CS(=O)(=O)NC)CCCN(C(=O)NCCC(CO)NCc2ccccc2)C1 C1(C(N2CCN(Cc3ccncc3O)C(CO)C2)=O)CCCC(F)(F)CC1 c1(C(=O)NCC2(C(F)F)CCN(C(C(C)(C)OC)=O)C2)c(F)ccc2[nH]ccc12 N1(C(Cc2nnc(C)s2)=O)CCCOC(CNC(=O)C(=O)N(C)C)C1 N1(C(CC(CNC(C2CCC(CO)CC2)=O)OC)=O)CC(O)CC(O)C1 C(=O)(CC(F)(F)C(F)F)N1CCC(CN(C)C(c2c[nH]cc2C2CC2)=O)C1 C(=O)(N=c1ccn(Cc2ccccc2)[nH]1)C1CCCC(CC)CC1 N(S(=O)(=O)N1CCNC(C)(C)C1)C(c1cc(C(=O)OC)c(F)cc1)=O N1(C(C=CCC)=O)CC(OC)C(CNC(=O)C2=COCC2)C1 C12CCN(CC1)C(=O)C1(CCOC1)CC1C(C1)C(=O)N2C.C(C)(C)(C)C1CC1 C1(NC(C(C(C)C)NC(C(CC2CCC2)OC)=O)=O)CCCCC12CC2 Cc1cc(C(=O)NC2CN(C(=O)CC3CCS(=O)(=O)C3)C2)c(N)c(Cl)n1 N1(C(c2c(C)scc2)=O)CC=C(C(=O)NOCC2OC(=O)CC2(C)C)C1 c1(CC)ccc(-c2nc(C)c(NC(c3sccc3-c3ccc(F)cc3)=O)s2)cc1 Cc1c(C)n(C)c2ccc(C(=O)NC3CCCC3NC(C3CCCSC3)=O)cc12 c1(-c2cc(CN(C)Cc3cn(-c4ccnc(C(=O)O)n4)nn3)no2)cccc(C)c1 C1(NC(C(c2ccnn2C)C)=O)C=CCN(C(=O)COC(F)(F)F)C1 Cc1cc(C(=O)NCCC2CSCCN2C(C2CCCSC2)=O)ncc1F c1(N2C3CN(C(CC(C)n4ccnc4)=O)C(CC3)C2)ncc2cccnc2n1 C1(CCONC(CC2OCCN(C(C3(C)COCCO3)=O)C2)=O)CC2CCC(C1)C2 C(=O)(C#CC1CCCCC1)NCC1(F)CCCN(C(C(CC(=O)OC)C)=O)C1 CC1(C)CCC(C(=O)NCc2cc[nH]n2)CN1C(C1CCCN1C=O)=O Cc1ncn(C)c(=O)c1C(=O)NCCCC(CO)NC(c1c[nH]c(=N)o1)=O CC(CCC(=O)N=c1cc(C2CC2)n(C)[nH]1)NC(=O)C(C)(C)C#N CC(C(=O)N1CCC(F)(CNC(C2CCCC3(CC3)C2)=O)CC1)S(C)(=O)=O C(c1c(Cl)cccc1Cl)=C(C)C(=O)NCC(C)NC(=O)CCP(C)(C)=O C(=O)(C(C#N)C(C)C)N1CC(C)C(C(=O)NCCn2cccnc2=O)C1 Cc1ccc(-c2cncc(C(=O)NC3CC(CNC(C4OCCO4)=O)C3)c2)cc1 C(C(C)(C)CC(=O)N1CCN(C)CC1CNC(=O)Cc1cccnc1F)N(C)C C(=O)(CC1=CCCC1)NCCC(=C)CNC(=O)CC1CCCC(C2CC2)O1 c1(C(=O)NC2C(CNC(c3c(C)occ3)=O)COC2)cnc2c(C)cccc2c1 N1(C(=O)NC(c2cn(C)nc2)CO)CC(Cn2cccn2)Cc2ccccc21 C(=O)(C(CNC(=O)CCc1nc(=N)[nH][nH]1)C(C)C)NCC(CC)C#N c1(C(=O)NCC2(C)CCCC2NC(c2c[nH]c(C#N)c2)=O)cccc2oncc12 C1(NC(C2(OC)CC2)=O)CCCC(CNC(c2nocc2C)=O)C1 c1(OC)ccc2nc(N3CCC(CO)C3)[nH]c(=NCCC(C)(C)C)c2c1 Cc1cn(CC(N2CC(CNC(=O)C(C)(C)C)C(C)C2)=O)c(=O)nc1O N(C(=NCCCF)N1CCC(CNC(=O)C(C)(C)C)C1)Cc1cc(C)cc(C)c1 C1(CC(=O)N(CCCCO)C)CCCN1C(c1nocc1Cl)=O c1(CC)cccnc1C(N1CC(C(=O)OC)C(c2ccc(OC)cc2)C1)=O N1(C(C2COCCN2c2ncccn2)=O)CCC2(CCC(c3ccccc3)CC2)C1 CC1CC(C(N2CCC(N3CCN(Cc4ccnn4C)CC3)C2)=O)CCO1 Cc1ccc(C(=O)O)cc1CN1CC2(CC(N3CCC(C(=O)N)C(O)C3)C2)C1 C12(C(=O)NC3CCN(C(C4CCC(C)O4)=O)CC3)CC=CC(C1)OC2 N1(C(CN(C)CCO)=O)CCC(NC(c2coc(C(F)F)n2)=O)C(F)(F)CC1 c1(C(C(=O)NCc2c(OC)nccc2)NC(=O)COSC2CC2)ccc(F)c(C)c1 c1(CCC)cccc(CS(N2CC3C(NC(=O)COC)C3C2)(=O)=O)c1 c1(C(=O)NCC(CNC(=O)CSC2CC2)CO)cc(Cl)cc2c1NCCC2 CCC(CC)C(=O)N1CCCCC1c1cn(-c2cnn(C)c2)nn1 c1(OC)cc(NC(=O)C(c2cccc(C(=O)O)c2)(C)C)c(Cl)cn1 c1(CNC(CC2N(C)CCCC2)=O)c(I)ccnc1O C1(F)(C(N(CC(CC)O)C)=O)CCCN(C(=O)COC(C)(C)C)C1 c1(NC(=O)NCCCCOC)ccc2c(c1)S(=O)(=O)N(c1nccs1)C2=O C1(C(=O)OCC)CCCCN1C(C1(N(C)C(c2c[nH]nc2SCC)=O)CC1)=O C1(OC)C(C(F)(F)F)C2CCCC1N2C(c1cccc(C=CC(=O)OC)c1)=O C1(C(N2CCC(CNC(c3ccc(C(C)C)cc3)=O)C2)=O)CC(C)(C)CN1C c1(C(=O)NCC2COCCN(C(c3c(C)cc(Br)cn3)=O)C2)cc2ccccn2n1 N1(C(=O)COCC(F)F)CCN(C(=O)COc2ccccc2Cl)C(CCO)C1 C(C(=O)NCC1(C(=O)Nc2csnc2C)CC=CC1)(C(C)(C)C)OC Cc1csc(C2CCCN2C(c2ncoc2C2CC2)=O)n1 c1(C(N2C3CC(NC(C(C)n4ccnc4)=O)C3CC2)=O)noc2c1CCCCC2 c1(C(=O)NC(CN(C(C2(OC)CC(C)C2)=O)C)(C)C)ccc2cc(C)ccc2n1 O(NC(=O)C(F)C(C)CNC(c1cc(CC)on1)=O)CCC(=C)C C1(NC(C2N(C(CC3CC(=C)C3)=O)C(C3CC3)CC2)=O)CCCC(O)C1O N1(C(=O)CN2CC=CC2)CC2CCC(C(=O)NC3(C(F)(F)F)CC3)(C2)C1 c1(NC(C2(F)CN(C(c3sc(C)c(O)n3)=O)C2)=O)ccc2c(c1)CCC2 CC(C)CC(C(=O)NCC(=O)N(C)O)NC(c1cc(Cl)c[nH]1)=O c1(C(=O)NC(C(C)NC(C2(C)CS(=O)(=O)C2)=O)CO)ccc2c(c1)CC(C)(C)O2 N1(CC)CCN(Cc2ccc(C)nc2O)CC1.c1(C(=O)OCC)ccc(N(C)C)cc1 c1(CN(C)Cc2ccc(C)s2)nc2cc([N+](=O)[O-])ccc2o1 C(=O)(C(C)(C)C(=O)OC)NC1C(NC(CC(=C)C)=O)C1 c1(C(=O)NC23CC(NC(c4cnc(OC)s4)=O)(C2)C3)cc(F)cc2cnccc12 C(=O)(C(C)(C)CCCNC(C1CN2CCN1CC2)=O)NCC(CSC)(C)O C1(NC(C(C)=CC)=O)C2CC(NC(=O)COC)CC12 CCCCCCC(CC)C(=O)N1CCC1(C)C(=O)Nc1cncc(C(=O)OC)c1 N1(C(c2ccc(OC)cc2)=O)CCC2(NC(=O)C(C)n3ccnn3)CCCC12 N1(C(C2C(CC)C2)=O)CC(CN(C)C(c2cc(F)sc2Br)=O)C2(CC2)C1 CCC(CO)CCNC(=O)COC1CCN(C(=O)CCCCC)C1 C1(CC(=O)NCC2CCN(CC)CC2)OCC2CCN(C(C3CCC(=O)N3)=O)CC12 CC1CC(NC(C2(c3ccncc3)CC2)=O)CCN1C(C12CCC(C1)C2)=O C(CCN=C(NCc1cc(C)on1)NCC1(n2cccc2)CC1)SC C(=O)(C(CNC(=O)C(C)COC)(CC)CC)NCc1ncc(OC)nc1 C1(C(N(CC(CNC(c2c(C)cncc2C)=O)O)C)=O)CCCCN(C)C1=O C1(NC(CC2(C=C)CCC2)=O)COCCN(C(=O)C(CC)=CC)C1 O=C(CC(F)(F)F)NC1CCCCN1C(=O)CCNC(=O)C=CCl N1(C(C2C(CC(=O)O)C(O)C2)=O)CCCCC(n2cc(C(=O)O)nn2)C1 C(C)(CCC(=O)NC(C(=O)N1CCC(O)(CO)C1)C(C)OC)SC c1(CN(C(=O)NCC(N2CCC(C)CC2)C(C)C)C2CC2)ccc(Cl)nc1O N1(C(CC(c2ccccc2F)C)=O)CCC(O)(CNC(=O)CSC(F)(F)F)CC1 CC1CCCCC1(C)C(=O)NC1CCC1CNC(c1cncc(F)c1)=O C1(OC)CN(C)C(C)(C(=O)NCC2(F)CN(C(c3cccc(N)n3)=O)C2)C1 N#Cc1ccc(O)c(C(=O)NCC(c2cncc(Br)c2)NC(C2(O)CC2)=O)c1 C(C)(C)(CCCN=c1ccc(Br)c(S(=O)(=O)NC(CO)C2(C)CC2)[nH]1)OC N1(C(C(CC=C)CC)=O)C2CC=C(C(=O)N3CC(CO)OC(C)C3)C1CC2 c1(C(N(CCC(C(C)C)NC(c2occ(C)c2)=O)C)=O)ccc2c(c1N)CCC2 N1(C(C(=O)NCc2cccc(C(F)(F)CF)c2)=O)CC2CC1C(O)(C(F)(F)F)C2 CN1CCN(C(=O)CN2CC(=O)NC2=O)CC1C(=O)CCOCCCN=[N+]=[N-] c1(NC2CCN(C(CNC(c3n(C)ncc3)=O)=O)CC2)cccc2c1OCC2 C1(C(=O)NCC(COC)(C)C)CCN(C(=O)CCOC(C)=O)CC1C c1(C(N2CC3C(CNC(COC(C)=O)=O)(C3)C2)=O)cc2ccccc2o1 c1(OC)nn(C)cc1C(=O)NCCCC(=O)N1CCC1C(C)C CC1CCC(CO)(NC(=O)C(C)NC(C2CC3CCC3C2)=O)C1 C12(C(=O)NCC(CC)NC(c3ccnc4ncnn34)=O)C3CCC(CC13)C2(F)F C1(C(=O)OCC)COCCN1C(=O)Cc1cc(Br)cs1.C12CC(F)CN1C2=O C1(NC(c2cnc[nH]2)=O)CCCN(C(=O)Nc2cccc(F)c2)C1 C#CCCC(O)C(=O)NC1CC(F)CN(C(c2ccccc2NC(=O)NC)=O)C1 CC(C)CC(O)C(=O)NCCC1CSCCN1C(=O)CCCc1ccncc1 C(CC(C)CCNC(=O)C(F)=C(C)C)NC(CSCCC)=O c1(N(CC(C(=O)OC)C)C(c2nnn(C)c2N)=O)ccc(F)cc1 CCCCC(O)CC(=O)NC1CC(NC(=O)C(F)Oc2ccc(Cl)c(F)c2)C1 C=C(Cl)CCC(=O)NCC(C1(O)CCN(C(=O)C=Cc2cn[nH]c2)C1)C C1(NC(CSCC(=O)OC)=O)CC2CC(C1)N(C(=O)CC1CC3(CCC3)CO1)C2 N1(C(C2N(C(C)=O)CCC2)=O)CC=C(CCNC(=O)CCCn2ccnn2)CC1 CCCCC(C(=O)N1C2CCC1(CNC(=O)CC(O)CCC)CC2)NC(N)=O N1(C(=O)CCCCc2ccc(F)cc2)CCN(C(c2cnns2)=O)C(CF)C1 C1(C(N(C2CCN(C)CC2)C)=O)CCC(C)(C)N(c2cccnn2)C1 C1(NC(C2(CC#C)CCC2)=O)CCN(C(=O)C=CCSC(F)(F)F)C(C2CC2)C1 CCC(N=c1[nH]c(=NCCCC2CC2(Cl)Cl)c2cc(Cl)ccc2[nH]1)C(C)C Cc1cn(-c2ccccc2)nc1C(=O)N(C(C)CCNC(C1CC(C)(C)O1)=O)C CC1CCCCCCN1C(=O)C=CC1CCCN1C(=O)C(C1CC1)C1CC1.C1(C=O)CC1 C1(CC(=O)OC)CC(O)CN1C(c1ccc(SC)o1)=O.c1(N)sccc1Cl C1(NC(C(CC)=CC)=O)CN(C(C2CCC(OCCCC)CC2)=O)CCC1(C)C c1(C(N2C(C(=O)NC(c3nc(C)sc3)C)CCC2)=O)cc(C2CC2)ccn1 N1(C(C)=O)CCN(C(=O)CCc2cncs2)C(COC)C1 N1(C(C2C3CCC2(c2cncs2)C3)=O)CCN(C(=O)Cn2cccc2)C(CO)C1 c1(N(C)C)nc2ccc(C(=O)NC3CN(C(C4CC5(CC5)C4)=O)CC3C)cc2o1 C(=O)(C1=CCCN(C(=O)Cn2ncccc2=O)C1)Nc1c(C)nn(C)c1 c1(OC)ccc(C(=O)NCCCNC(C2COC3(CCC3)C2)=O)c(OC)n1 c1(C(=O)NC(C2N(C(COC)=O)CCC2)C)cccc2c1OC(C)C2 c1(C(=O)Nc2cccc(Cl)c2CO)c(F)ccc(Br)c1Cl C(=O)(C1=NNC(=O)C1)NC1C=CCN(C(C(c2cccc(C)c2)F)=O)C1 c1(NC(C2CN(C(c3cnnc(Cl)c3)=O)CCN2)=O)cnc2cc(Br)ccc2c1 Cc1nsc(C(N2CCC2CNC(=O)CC2CC2C)=O)c1N C1(C(N2CC(N(C(c3cc(SC)c(C)o3)=O)C)C(F)C2)=O)CCCCNC1=O CC1(C)CCC(NC(=O)CCn2cc(-c3ccc(Cl)cc3Cl)nn2)CO1 N1(C(C(C)OC)=O)C2CCC1C(CNC(c1ncoc1-c1cccc(F)c1)=O)C2 C1(N(C(C(C)OCC=C)=O)C)CCCCC1NC(c1ccc(-c2cccs2)[nH]1)=O C1(OC)CCN(C(C2(C)CCN(C(c3ccc(O)cc3)=O)C2)=O)CC1 c1(C(=O)NC2C(CO)CCN(C(CN(C)CCO)=O)C2)cc2cc(Cl)ccc2o1 CC(C(=O)NC1CC2CCC(C1)N2C(c1cc2sccc2[nH]1)=O)C1=CCCC1 C=CCC(C)C(=O)NC(CNC(c1cc(C(C)C)ns1)=O)CC=C c1(-n2cc(C(CC#N)NC(C3CC3)=O)nn2)ccc(Cc2ccccc2)cc1 C(c1ccc(C)c(C)c1)=CC(=O)NCC(CC=C)NC(c1nn(CC)nc1C)=O N1(C(CC(C=C)C)=O)CC2(C)CC1(C(=O)NC1CCC(F)CC1)C2 Cc1cn2cccnc2c1C(=O)NCC=CCNC(=O)C(C)(C)CF c1(C(C(=O)NC(C)CNC(=O)C=CCOCc2ccon2)O)cccnc1 CN1CCCCC1C(=O)NC(C)(CNC(=O)C=CC1CCOC1)C1CCC1 C(C(CC(C)C)C(=O)N1CC(F)(F)CCC1C)NC(c1cn(CC)nn1)=O N1(C(C(CC2CC2)OC)=O)CC(NC(c2c[nH]c3ncccc23)=O)C2(CCC2)C1 c1(OCC)cc(C(=O)NCC(C)N(C(=O)CC(C2CC2)C2CC2)CC)ccc1C CCC(CNC(C1(C)CC=CCO1)=O)(CC)NC(=O)C(C)(C)CNC(C)=O N1(CC(C(C)(C)C)CO)CCCC2(C)CCCC12 c1(C(=O)NCCOC2CCN(C(C=CC(CC)C)=O)C2)oc(C)nc1C c1(C(CNC(C(C)NC(=O)C(F)(F)F)=O)O)cccc(Cl)c1N c1(C(CNC(C(CC)Cc2cccc(C)c2)=O)=O)ccc(C(=O)OC)c(O)c1 c1(OCC(=O)NCC(CNC(CN(C)CCO)=O)CO)ccc(C(N)=O)cc1 C1(C(=O)NC2CC=CC2)(CNC(c2ccnn2CCF)=O)CCCO1 C12(C(N3CC(NC(=O)CN4CCOCC4=O)C(O)C3)=O)CCC(F)(CNC1=O)C2 N1(C(C2N(C(CC)=O)CSC2)=O)CC(NC(c2ccc(C3CC3)s2)=O)C2(CC2)C1 C1(c2nc(CC(C)NC(=O)OC(C)(C)C)[nH]n2)CCN(c2ncccn2)CC1 c1(C(=O)NC(CC)CN(C(=O)CC2CC2)C)c(-c2ccccc2)nc2sc(C)cn12 C1(CNC(C(C)N2CCC2)=O)CN(C(c2ccnc(F)c2Cl)=O)CC(C)(C)O1 C(c1cc2ccccc2n1C)=CC(=O)N(C1CN(Cc2ccccc2)CC1(C)C)C O=C1CCOCC(C(=O)N(CCOCc2cccs2)Cc2ccco2)C1 C1(C(N2CCC(COC(C)=O)C2)=O)CC1C1CN(C(=O)Cc2nocc2C)C1 c1(C(N(CCCNC(CC(C)SC)=O)CCO)=O)ccc2ccncc2n1 CC(CC(=O)NCC1C2CN(C(c3cc(C(N)=O)ccn3)=O)CC12)C(C)(C)C n1(CC)nc(C)cc1C(N1CC2CC1(C(=O)N(C1CCCC1C)C)C2)=O c1(C(=O)NC2C(C)CN(C(=O)Cn3nc(Cl)ccc3=O)C2)nc(O)nc(O)c1N C1(C2N(C(Cn3cc(C4N(C)CCC4)nn3)=O)CCC2)(C(F)(F)F)CCCCC1 c1(C(N(CC(CNC(c2c(C)csc2)=O)C)C)=O)c(F)c(C)cc(N)c1F Cc1cccc(C=CC(=O)NCC2CC2CNC(c2nccnc2C(N)=O)=O)c1 c1(C(=O)NC(C)CN(C(=O)CCCNC(=O)C(C)(C)C)C)ccncc1F Cc1ccc(OCC(N2CC(F)(CNC(=O)Cc3cnoc3)C2)=O)c(Br)c1 C(C1=CCN(C(=O)CN2C(=O)CNC2=O)CC1)NC(=O)CC1C=CCC1 C(=O)(CC(CCCC)NC(C1CCCN(C)C1)=O)NCCCCC#CC N1(C(C(C)(C)c2ccncc2)=O)CCCC2(C1)CN(C(=O)C(F)F)CCO2 CC1(C)CCN(C(c2cccc3ccsc23)=O)CC1NC(C12CCC(C1)C2)=O C1(C2CCCN(C(c3ccc(=N)[nH]n3)=O)C2)(NC(CCCC(C)C)=O)CC1 c1(C(N(CC(CC)NC(=O)CC2CCC(=O)N2CC)C)=O)ncnc2sccc12 CC1(C#CC(=O)NC2CC(NC(c3ccc(C(F)(F)F)c(Cl)c3)=O)C2)CC1 c1(C(=O)NCC2CC(C)N(C(=O)Cc3cnccn3)C2)ccn(CCO)c(=O)c1 C(CCCCCNC(N(C)Cc1scc(SC)n1)=O)NC(=O)OC(C)(C)C N1(C(Cc2cnc(C)s2)=O)CCN(C(=O)C=CC(C)(C)C)CC1 C1(c2cn(CCC3C(=O)N=C(C)S3)nn2)CC(C)(C)CN1C(=O)Cc1ccc(C)o1 c1(CNC(C(=O)NCc2cccc(OC)c2)=O)cc2ccccc2s1 CN1C(=O)CCC1(C)CNC(=O)Cc1csc(C2CCCNC2)n1 C1(N(C)C)CN(C(=O)COc2ccsc2)C(C)(C)C1.C12CCOC1CNC2=O N1(C(CNC(c2cccnc2)=O)=O)CC(NC(C2C(F)(F)C23CC3)=O)C(CO)C1 c1(OC)cccc(C(=O)NCC(C2CC2)N(C(=O)CCC(=O)N(C)C)C)c1 N1(C(CCCCCSC)=O)CC(NC(=O)C=Cc2ccc(O)cc2)CC12CCC2 C1(CC)(CC)CN(C(C2CC(Cc3ccc(F)c(F)c3)C2)=O)CCS1 C1(NC(C2(CC)CC2)=O)CN(CC(=O)Nc2cncc(Cl)n2)CC2(CCOCC2)C1 C(CCCOC)(C(=O)NCc1cccc(Cl)n1)NC(CC(=O)NCC#C)=O C1(C2(O)CCC2)(SCCCCC(=O)NC2CC(C(=O)NC3CC3)C2)CC1 N1(Cc2onc(C(=O)OC)n2)CCCC1C(C)NC(=O)NC(F)(F)C(F)(F)F C1(NC(CC2(OC)CC2)=O)CC2CCC1CC2NC(C1CCCC(F)C1)=O c1(C(N2CCCC(CNC(C(CC#C)C)=O)C2)=O)n[nH]c2ccc(F)cc12 CC(O)C(C(=O)N1CCCCC1c1cn(C(C23CC(CO2)C3)C)nn1)N(C)C Cc1cc(C)nc(N(C2CCN(Cc3cc(O)ccc3Cl)CC2)C)n1 C1(CNC(c2c(C)cno2)=O)CC(C)N(C(=O)COc2ccc(C(C)C)cc2)C1 c1(C(=O)NC2C(NC(C(C3CCOCC3)OCC)=O)C2)cccc(OC2CC2)n1 CP(C)(=O)C(CC(=O)N1CCOCC1c1cccs1)C(F)(F)F C1(C(=O)NC(CNC(CCCNC(=O)OC)=O)C)CCCCC(=O)N1 N1(C(C=CC2N(C(C(CCC)C#N)=O)CCC2)=O)CCCC2(CCC2)C1 C(C1=NOC2CN(C(C3(F)CCCC3)=O)CC12)NC(c1cccc(CO)c1)=O c1(C(=O)NC(C(C)NC(Cc2cncc(C)c2)=O)C)coc2c(F)cc(Cl)cc12 N1(C(C=C(COCC)C)=O)CC(OC)CC1CNC(=O)CCc1cn[nH]c1 c1(C(N2CCC(CNC(C=C3CCN(C)C3)=O)C2)=O)ccc2cc(Cl)ccc2n1 Cc1[nH]ccc1C=CC(=O)NC1COCC1C(=O)NCC1CC1c1ccccc1F C1(C(=O)NCC2CCC(C)(O)C2)CCCCCCN1C(c1ccc(CO)o1)=O N1(C(c2cc(COC)no2)=O)CC(CNC(c2c[nH]nc2OC)=O)C(O)C1 C1(C)(C(=O)Nc2c(C)cc(NC(C3CS(=O)(=O)C3)=O)cc2)CCOC12CC2(F)F c1(C(N(C(CN(C(CC(C)OC)=O)C)C)C)=O)[nH]cc(C(C)=O)c1C C1(NC(C(CC)OCC)=O)CC(F)CN(C(=O)C(C)(C)n2ccc(C)n2)C1 Cc1cc(C(=O)N(CCCN(C(C2CC2F)=O)C(C)C)Cc2ccccc2)sc1C c1(C(c2n(C)nnn2)NCc2c[nH]c(=N)nc2O)ccc(Br)cc1F N1(C(c2ccc(OC)nn2)=O)CC2(CCCN(C(c3csc(C(N)=O)n3)=O)C2)C1 C#Cc1cccc(C(C)NC2CC(C(=O)Nc3cnc(C)c(C)c3)C2)c1 C(=O)(C1=C(Cl)CCOC1)N1CC(NC(C(C)(C)SC)=O)C(C(F)F)C1 C(CC(=O)N1CCCC1C(C)NC(c1ccc(CO)cc1)=O)(C(N)=O)NC(C)=O C(=O)(C(C)(C)C(F)(F)F)NC(C1(O)CN(C(=O)CS(=O)(=O)NC2CC2)C1)C C(=O)(C#CC1CCOC1)NCC1C(C)CN(C(=O)C2=NOC(C(C)(C)C)C2)C1 CCC(C)(CO)C(=O)N1CCCC1C(N1CCC(COC(C)=O)C1)=O C1(C(N(CCOC)CCNC(c2csc(Cl)c2)=O)=O)CCC12CCC2 C1(C(N(CCOCCCNC(c2cnc(C(C)O)s2)=O)C)=O)OCCN(C)C1=O N1(C(CCOCCC)=O)CCN(CC2CN(C(=O)CCCF)C2)CC1 c1(CCC(=O)NC(COC)CNC(c2ncsc2C)=O)ccc(F)nc1 c1(C(N2CC3CN(Cc4ccc(C(=O)O)o4)CC32)=O)ccc(F)c(F)c1Cl c1(C(N2C(CC(=O)Nc3cc(C)ncc3)COCC2)=O)ccc(C#N)cc1 N1(C(C=Cc2ncc(C)[nH]2)=O)CCCC2CN(CC(O)CC(F)(F)F)CC12 N1(CC(=O)NCC(CCOC)O)CCN(C(=O)C(C)O)CC1 c1(C(N(C(C)C)CCN(C)C(C2CC23CC3)=O)=O)nccc2[nH]ccc12 c1(C(C(=O)NCCCc2cccs2)N(CC(C)(C)CO)CC)sc(F)cc1Cl N1(C(c2cc(SC)no2)=O)CCN(CC(CNC(=O)CSC)OC)CC1 CC(C)CC(CO)N(C)C(c1cc(CNC(C2CNC(=O)N2)=O)ccn1)=O N1(C(C(COC)N(C)C(c2cc(Cl)cn2C)=O)=O)CCN(C2CC2)CC1 N1(CC(=O)N(CCCCCC)C(C)C)CCC(C)C(Cn2cc(C)cn2)C1 N1(C(Cc2nc(COCC)sc2)=O)CCN(C(=O)Cc2c(C)noc2C)CC1C C1(NC(C(C)CN(C)C)=O)CCCCN(C(=O)COCc2ccc(F)cc2)CC1 CCC(CC)CCCC(=O)NCC(C)N(C(C1COCCN1C=O)=O)CC c1(SC)cccc(-c2cccnc2C(=O)Nc2cnn(CCO)c2)c1 c1(N(C)C)ccc(C=CC(=O)Nc2nnc(C3CC3)o2)cc1.C12(O)CN(C1)C2 N1(C(C(c2ccccc2)C)=O)CC=C(CNC(C2CC2c2cccs2)=O)CC1 C1(C(=O)NC2CCCN(C(CCCC(C)O)=O)C2)CSC2(C)CCC(=O)N12 C(C(CC(C)C)NC(=O)CC1CN(C)C1)NC(COC(CC)(C)C)=O N1(C(c2cc(C#C)c(C)cc2)=O)CCCC12CCN(C(=O)CCc1cc[nH]n1)C2 c1(N(C(=O)CC2CN(C(c3ccsc3C(F)(F)F)=O)CCO2)C)ccccc1C#N c1(C(N(C2CCN(C(=O)C(O)CCS(C)=O)CC2)C)=O)nnn2c1CSCC2 c1(C(=O)NC2CC(C(=O)NCCN(CCOC)C)C2)cncnc1C C(=O)(N1OC2C=CC1CC2)C1OCCC(NC(c2nc(CC)oc2)=O)C1 c1(C(C)Sc2ccc(-c3ncnc(C(F)(F)F)c3F)cc2)ccnc(C2CCC2)c1F N1(C(CC=C)=O)CCN(C(C2CC2F)=O)CC1c1cccc(F)c1 CCS(=O)c1ccccc1C(=O)NCCC1(C)CCN(C(C2C3COCC23)=O)C1 C1(NC(c2c(C)n[nH]c2C)=O)CCN(C(c2cnc(C3CC3)[nH]2)=O)C12CC2 N1(C(CCOCCOC)=O)CC(C)(NC(=O)CN(C2CCOC2)C2CC2)C1 c1(C(=O)NC2(CNC(C(CC)C)=O)CC3CCC2CC3)cc2cccc(Cl)c2o1 C1(CNC(C(CC=C)CC)=O)CC2CCC1N(C(=O)C(C)C1CC1)C2 c1(NC(C(=O)N(C2CCCCC2)CC(=O)NC2(C)CCCC2)=O)ccc(F)cc1 N1(C(c2cc(C)c(O)nn2)=O)CC(NC(=O)C(C)c2ccsn2)CC2(CC2)C1 c1(C(N2CC(C)C(CNC(=O)CSC(C)(C)C)C2)=O)cc2c(ncn2C)s1 c1(C(N2CCC3CN(C(C4C(C)C4)=O)CC32)=O)nccc2cccnc12 C1(C(N(C(C)C(=O)OC)CCC)=O)CC2CCC(C1)N2Cc1cnc(C)nc1O N1(C(=O)NCCc2ccc(C)c(F)c2)CCc2cc(F)cc(Cl)c2C1 C1(NC(C2(NC(C)=O)CC2)=O)CN(C(=O)CCc2ccc(Cl)nc2)CC1O C1(C(=O)NC(C2C(=C)C2)=O)CCCCN1CCNC1CCCN1S(=O)(=O)CC CC1CC2(CC2)CN1Cc1cc(C(F)(F)F)ccc1-c1scnc1S C#CCCC(O)C(=O)NCCN(c1cc(C(=O)OC)nc(C)n1)C1CCCC1 C1(NC(c2cnc(C)n2C)=O)COC2(C1)CN(C(C1CCCN1C1CC1)=O)C2 CC1(CNC(c2csc(C(F)F)c2)=O)CC(NC(C2(C3CC3)CC2)=O)C1 C1(O)(C(C(=O)N(CC(C)NC(C(C)n2cccn2)=O)C)(F)F)CCCCC1 n1(CC)nnc(C)c1CNC(=O)COCCNC(=O)CC1CCCC1NC(C)=O C(N=c1[nH]c(=NCC2(C3CC3)CC2)c2ccccc2[nH]1)c1nc(N(C)C)sc1 c1(CC#N)ccc(C(=O)NCCCN(C(=O)Cc2ccccc2)C2CC2)cc1 O=C1OCc2cc(C(=O)NC3CN(C(c4ccc([N+](=O)[O-])cc4O)=O)C3)ccc21 C(=O)(C(C)C(F)(F)F)NCC(CCCC)NC(=O)COc1cccc(C)c1 C1(CC=C)(C(N2CCOC(CCF)C2)=O)CCCN1C(C1C(C)C1C)=O CON(CCC(=O)N(CC(F)(F)Cl)C)C(=O)CC1CCCNC1=O Cc1cc(Cl)cc(C(=O)NC(CNC(C2CC(C(C)C)=NO2)=O)C(C)(C)C)c1N C1(CCNC(CC2(C=C)CCC2)=O)CN(C(C2CCC(=O)C2)=O)CCO1 c1(NC2(CO)CCCN(C(C(CSC)(C)C)=O)C2)ncnc2sc([N+](=O)[O-])cc12 Cc1ncnc(C)c1OCC(=O)NCCC(C)N(C)C(C1NC(=O)OC1(C)C)=O N1(C(C(C)=C(CC)C)=O)CCC(CO)(CNC(c2ccc(CCSC)cc2)=O)C1 c1(C2N3CCC(C3)NC2=O)nc(C)c(C2CC2)s1.CCCOC c1(OC)ncnc(C)c1C(=O)NC1CC(CNC(=O)COc2cncc(Cl)n2)C1 c1(C(=O)NCC2CC(NC(C3C(C)OC(C)C3)=O)C2)cc(N)cc2c1OCCO2 N1(C(C)C)CCC(CC(=O)NC(C)C(C2CC2)NC(=O)C(c2ccccc2)=O)CC1 C1(O)(C(C)NC(c2c(CC)cno2)=O)CCN(C(c2ocnc2C(F)F)=O)CC1 c1(C(=O)NCCC2N(C(C34CC(C)C3C4)=O)CCCC2)c(Cl)nc2ccccn12 N1(C(C2(OC)CCCOC2)=O)CC2CCC(C1)N2C(c1snc(C)c1N)=O c1(C(N(C)CCOCCCNC(=O)C(C)(C)C)=O)ccnc2[nH]cnc12 c1(C(=O)NC2CN(C(c3c(C)nccn3)=O)C(C)C2)cncc2nc[nH]c12 c1(CN(C=O)Cc2nc(C(=O)OCC)sc2)cccc(COCC)c1 C(=O)(CCC(=O)NCCCC(C)NC(=O)C(C)N(S(C)(=O)=O)C)NCCC c1(N(C(c2cn(CCC)nc2)C(=O)NC(C)CC)C)sc(C)cc1C C1(CNC(C2CCN(C)CC2)=O)(NC(c2cnn[nH]2)=O)CCC(F)(F)CC1 C(=O)(C1=CS(=O)CCC1)N1CC(C)C1.C(C(=O)Nc1ccccc1)(C(C)C)SC N1(CCC)CCC(C(N2CCCC(NC(=O)CC3C(C)C3(F)F)C2)=O)CC1 C(N=c1nnc(CO)c(C(=O)OC)c(O)n1)c1c(OC)ccc(Cl)c1F c1(C(N2CCN(C(c3nnc(C)s3)=O)CC2CF)=O)c[nH]c(=O)c2ccnn12 N12CCC(C3CC3NC(=O)C3C(C3)C1=O)CC2.C1(CC#C)(C(=O)OC)CCC1 C(=O)(C1=CCCOCC1)N1CCC(CC=C)(C(=O)NCc2cncn2CCC)C1 C1(NC(C(C2CC2)OCC)=O)CC1C1CCCN(C(=O)C2=CCCCC2)C1 c1(NC(C2C3CN(C(c4c(C)nc[nH]4)=O)C2C3)=O)cc(C#N)cnc1C C1(NC(=O)Cc2ccc(F)nc2)CCC2(CCN(CCCCO)CC2)C1 c1(NC(C(CC)Br)=O)ccc(C2CCCN(C(c3n[nH]cc3Cl)=O)C2)cc1 CS(C)(=O)=NC(=O)C(=O)NC1C=CCN(C(C2(C3CCCO3)CC2)=O)C1 O=C1CCC(N2CC(C(=O)NC(CNC(=O)CSc3nc[nH]n3)C3CC3)C2)CC1 C1(C(=O)NC2(CCC(=O)N(CCCN(CC)CC)C)CCC2)OCCOC1C N1(C(c2c(CC)scc2)=O)CCC(CNC(c2scc(C)c2OC)=O)(SC)CC1 n1(CC(N2CC(c3c(CNC(C=C(C)C(F)F)=O)nco3)C2)=O)cnnc1O c1(C(=O)NC(CN(C(C=C(C)C(C)(C)C)=O)C)(C)C)cc(C)c(Br)c(Cl)c1 c1(NC(N2CC(OCCOC)CC2(C)C)=O)nc2ccccc2nc1C C1(C(=O)NCC(c2ncncc2Cl)=O)CSc2ccccc2O1 c1(OCCC(=O)NC2C(NC(C(C)OC)=O)C2)ccccc1Sc1ccccc1 c1(OC)ccc(CN2CCCC(CC(=O)NC3CCOCC3)C2)cc1[N+](=O)[O-] c1(N(C(=O)CCc2ccccc2C)C)ccc(C)cc1NCC C1(C)(CC(N2C(C)(CCC)CC2)=O)CCN(C(c2cc(C)no2)=O)C1 n1(CC(=O)NCC2(CCNC(C3CC4C(C3)C4(F)F)=O)CC2)cnc2ccccc12 C(C)(CNC(=O)C(C)=C(C)C)(CNC(=O)CCC1(C)CC1(F)F)OC C1(CNC(CC2CC(SC)C2)=O)CC2(CC2)CN1C(c1cc(O)ccc1C)=O N1(Cc2c(C)nn(C)c2)CCCC(NC(c2ccc(Cl)c(Cl)c2)=O)CC1 O=C(CCC[N+](=O)[O-])N1CCN(C2CCCN(C(C3CCCCCO3)=O)C2)CC1 c1(C(N2CC(CCNC(CSS(C)(=O)=O)=O)C2)=O)cnc(O)s1 c1(NC(C2C(NC(c3nscc3Br)=O)C2)=O)nc(Cl)ccc1C(N)=O C1(O)(C(C)NC(CNC(CC)=O)=O)CCN(C(=O)C(C)(C)C2CC2)C1 c1(C(=O)NCC(C2CCCCC2)C)ccc(NS(=O)(=O)CCBr)cc1Cl C(=O)(N=c1[nH]c2sccc2s1)C1CC2(CC(NC(c3nccc(C(=O)O)n3)=O)C2)C1 Cc1cccc2cc(C(=O)NCCC(C)NC(C3(C(C)C)CCCO3)=O)oc12 CC1CCCN(C(=O)COC2CCCOC2)C1CNC(c1n[nH]cc1Cl)=O c1(C(N2CCC(C)(NC(Cc3c(C)noc3)=O)C2)=O)ccc2nonc2c1 CC(C)(CC(=O)NC(COCCN1CCCCC1)C(=O)Nn1cnnc1)C1CC1 N1(C(C2CC(C)CN(C(=O)C(C3CC3)C3CC3)C2)=O)C2CCC1CC(F)C2 C=Cc1cc(C(=O)Nc2ncsc2-c2ccc(Br)cc2)cc(-c2nn[nH]n2)c1 CC1(CNC(c2ccc[n+]([O-])c2)=O)CN(C(C2CN(C3CCC3)C2)=O)CCO1 N1(C(C(CN(CC)CC)F)=O)CCC(F)(CNC(=O)C2=CCOC2)CC1 C(=O)(C1=NOC2(CCC2)C1)NC1C2(CN(C(CCn3ncc(C)c3)=O)C2)SCC1 N1(C(C2C(C)C2)=O)CCCC(CNC(=O)Cc2cc(Cl)n(C)n2)C1 C1(NC(C(c2c(C)noc2Cl)C)=O)CN(C(C2(C(F)F)CC2)=O)CC1S(C)(=O)=O C1(F)(C(=O)NCC(C(C)C)(C)NC(=O)CC2CCC(C)(C)CO2)C(C)(C)C1(C)C N1(C(c2c(C)nco2)=O)CCC2CCCC12CNC(c1cc(C)n(C)c1)=O N1(C(CCOCC(C)C)=O)CC(NC(=O)C(C)(C)CN2CCN(C)CC2)C(C)C1 N1(C(C)=O)CC2CC2(C(N2CC(NC(=O)CSCCSc3n[nH]c(O)n3)C2)=O)C1 N1(C(c2cc(C)c(Cl)s2)=O)CCOC2(CCCN(C(=O)C=Cc3ccsc3)C2)C1 c1(OC)ccccc1CC(=O)NC12CC(C(=O)NC3CCC(n4ccnc4)C3)(C1)C2 C1(C(=O)NC2CCC(OC)C2)CC2CC2N1Cc1cnn(Cc2ccccc2)c1 CCC(C)C(C)C(=O)NCC1(C(=O)NCC23CC(F)(C2)C3)CCCO1 C1(C(=O)NC2(CC(C)C)CC2)CCC(C)(CNC(=O)CCCC2CCCCC2)C1 C1(C2CCN(C(c3cccc4sccc34)=O)C2)(NC(CC=CC=C)=O)CC1 C(=O)(CC(C(F)(F)F)OC)NC(CCCC)CNC(=O)C(F)=C(C)C C=CCC(C)C(=O)NC1CC(C(C)NC(C2CCCC2(C)C)=O)C1 C1(N(C)C)(NC(CC2CC(c3ccccc3)(NC(CSC)=O)C2)=O)CCCSC1 C(=O)C1=C(C#N)CCC1.C(=O)(C(C)CN(C)C(C)=O)OCC(COC)O c1(C(=O)NCCN(C(C)C)CC)cnn(C)c1O CN1C(=O)C(=O)N(CC(=O)NCCOCCNC(=O)C(=O)NC(=O)C2CC2)C1=O CCC(C)(C(=O)NCCC1CCN(C(c2ccc(Br)o2)=O)C1)C(N)=O C1(NC(C(C(=O)OCC)OC)=O)CCC2(CC1)CC2NC(=O)CNC=O CCCC(O)CC(=O)NCCCN(C(=O)CCCc1cnccn1)C1CCCC1 c1(NC(N2CCCC2c2cccnc2F)=O)cc(F)cc(Br)c1Cl C1(NC(C(C=CCCC)O)=O)CCCN(C(=O)CC2(OC)COC2)CCC1 C(=O)(C(CC)NC=O)N.C(C(=O)NCCCNC(C)C)N(CCOCC)C C1(CN(C)C(c2cc(C(F)(F)F)cs2)=O)CCCN1C(=O)CC1CCC1 C1(CNC(c2c(COC)n(C)nc2)=O)CCN(C(=O)CNC(=O)OC)CC1O N1(C(c2cc(OC)nn2C)=O)CCn2cnnc2C1.N12CCOC(C1)CC2=O CON(CCC(=O)NC1CC(=O)N(C)C1=O)C(=O)C1=NOC(C)C1 c1(CCNC(N2C(c3nc(C)c(C)s3)CCC2)=O)cc(F)cc(F)c1F C1(C(=O)O)(NC(C2CCCN(c3nccs3)C2)=O)CC2CCC1C2 C1(CC)CN(C(=O)C=CBr)CC1NC(=O)C(c1cnn(C)c1)O C1(NC(c2csc(O)n2)=O)CCCC(NC(c2n[nH]c(O)n2)=O)CC1 C=Cn1nccc1C(=O)NCC(c1cccc(OC)c1)NC(c1cc(C)sc1N)=O C(=O)(CCC(C)(C)C#N)NCC1(CNC(c2ccc(CC)cc2C)=O)CC1(F)F N1(C(C(C=CC)O)=O)CCCC(C2CN(C(=O)Cn3cc(Br)c(C)n3)C2)C1 Cc1cc(C(=O)NCCN(C(=O)C2=CCCC2C)C2CC2)c2[nH]cnc2c1 C1(NC(C2CC2c2ccc(-n3cccn3)cc2Cl)=O)CCCC(C(F)(F)F)CC1 c1(C(=O)NCCCCC(C)NC(c2cc(Cl)nnc2O)=O)ccc(F)c(F)c1F C1(CN(C(c2ccn(CC(F)(F)F)n2)=O)CC)CCN(C(c2cc(O)cs2)=O)C1 N1(C(C(CCCC)C)=O)CC(C)(C)C(NC(=O)C(C(C)C)C(C)C)C(C)(C)C1 N1(C(C2C(C=C)C2)=O)CCN(C(=O)Cn2nccc2C)C(c2nccn2C)C1 CC1CN(C)CC1NC(C1(CCO)CN(C(=O)Cc2nnc(S)n2C)C1)=O CC(=O)CCCCC(=O)N1CC2CC1(C(N1CC3C(C1)C3(C)C)=O)C2 N1(C(=O)C=CCO)CCC(Nc2nc3cccnc3s2)C2(CCC2)C1 C(=O)(C#CC1(C)CCCO1)N1CC(CCOC)N(C(=O)C=CC(C)(C)C)CC1 Cc1cn2c(C(=O)NCCCCCCNC(C3C(F)(F)C34CCC4)=O)cnc2s1 N12CCC(O)C(C1)CN2C.C1(C)(C=O)C=CCC1.C1(C=O)CC(n2cnnc2)C1 c1(COC)c(C(=O)NCCNC(c2nc[nH]c2C(C)(C)C)=O)nn[nH]1.C(C)(C)C c1(C(=O)NCCOCCNC(C(CC)O)=O)cc(OC)c(OC)c([N+](=O)[O-])c1 CN1CCCC(C)(CNC(C2CCC(C3CC3)N2C(=O)Cn2ncnn2)=O)C1 c1(C(N(CCCNC(CCOCC#C)=O)CC)=O)cc(CC(C)C)on1 c1(CN(C(=O)C=CC(C)(C)SC2C(C)C2)C)c[nH]c2ccccc12 c1(C(=O)NC2C(NC(CN(C)C)=O)CC2)cc(Cl)c(F)cc1O C(C(=O)N1CC(C)(C(F)C(=O)NC2CC(=O)N(CC)C2)C1)(C(C)C)OCC.CC C(CC(C(=O)N1CCC1C(=O)OC)NC(=O)CC(C)(C)C)OC N1(C(CSCC#C)=O)C2CC1CN(C(c1ccoc1Br)=O)C2 C12(NC(=O)CN3C(=O)CNC3=O)CCN(C(c3ccncc3C(F)F)=O)CCC1C2 CC(C)CCN=C(NCC(C1CC1)N(C)C)N1CCC(CC(C)C)CC1 N1(C(C2C(C(C)NC(c3ccc[nH]3)=O)C2)=O)CC2CC3CC2C1C3 N1(C(C(C(C)C)O)=O)CCC2CN(C(=O)Cc3cc(Br)cs3)CC2C1 C1(C)(C(N(C)Cc2cncs2)=O)CCCN1C(c1cc[nH]c(=N)n1)=O c1(CCC(=O)NCCOCCNC(C2C(C)CCCC2)=O)cccc([N+](=O)[O-])c1 c1(C(N2CC3C(CNC(C4CC4F)=O)(C3)C2)=O)cccc(F)c1C1CC1 C(=O)(CC1=CCCC1)NC(CCN(C(c1[nH]nc(OC)c1Cl)=O)C)C C1(CCC)CCN(C(=NCc2cccs2)NC(C)COC)C1 c1(CN2CC(CC(=O)Nc3cc(OC)ncc3)C2)cccc2c1OCCCO2 Cc1ccc(C(=O)N(c2ccccc2)Cc2ccccc2F)c(O)n1 c1(CNC(C(C2CC2)OCC)=O)cc(C(=O)NC2CCC2O)co1 c1(C(N2CC3C(CNC(c4ccncn4)=O)(C3)C2)=O)cc(F)cc(F)c1Br c1(OC)cccc(C(=O)NCC(C2CCCCC2)NC(=O)C=CC2CCOC2)c1N CC(CN(C)C)CC(=O)NC1CN(C(=O)C(N)=O)CC1c1ccccc1 N1(C(c2c(CC)cccc2)=O)CCOCC(NC(C2(C)CCNC(=O)C2)=O)C1 c1(NC(C2C(NC(c3ccc(C(N)=O)o3)=O)C2)=O)cc(OC(F)(F)F)ccc1C N1(C(CC(COC)(C)C)=O)CCCCC1C1CCCN1C(C1CCOC1)=O Cc1ccc(C(=O)CCC(=O)N2CC3C(C(C)NC(=O)CCC(C)C)C3C2)cc1 Cc1nn(C)c(C)c1CC(N1CCCC1CN(C(=O)Cc1cnc[nH]1)C)=O c1(C(=O)NCC2C(CNC(CCC=CC)=O)C2)cccc([N+](=O)[O-])c1NC C1(OC)CC2(C(=O)N(CCC(C)NC(c3cccn3C(C)C)=O)C)CC12 c1(CC)ccccc1NC(C12CC(NC(=O)COc3cncc(C)n3)(CO1)C2)=O C1(C#N)(C(N2CC(CNC(C(C=C)(C)O)=O)C(N(C)C)C2)=O)CCC(=O)CC1 N(C)(S(=O)(=O)N(C)C)CC(=O)N(C)CC1CN(C(C(C2CC(F)(F)C2)OC)=O)C1 C1(C(N(C(CNC(CCCCOC)=O)C)C)=O)CCS(=O)(=O)CC1 c1(C(=O)NC23CC(NC(Cn4nnc(=N)[nH]4)=O)(C2)C3)cccc(Cl)c1Br Cc1ccc(C(C)(C)C(=O)NC2CC(CNC(C3CCCS3)=O)CC2O)cc1 C(=O)(C(C)CC(C)C)N1CCC(C(CNC(CCN(CCCCC)C)=O)C)CC1 Cc1ccc(CNC(=O)C(=O)NCc2ccc(O)cc2F)c(F)c1F C1(CC=C)(NC(c2cccc(N)n2)=O)CCCN(C(=O)C(CC)c2ccccc2)C1 C(CCCS(C)(=O)=O)NC(C1CC(n2cc(-c3cnc(C)s3)nn2)C1)=O CC(C)C(CNC(c1cccn1Cc1ccccn1)=O)NC(=O)CC(C)F c1(C(N2C(C)(CC)CC(NC(=O)C#CC3CC3)C2)=O)c[nH]c2ccc(F)cc12 C1(C(=O)Nc2ncc(C(=O)OC)[nH]2)C2CC1N(C(C1CC13CCC3)=O)C2 C1(C(N2CCSC(C)C2C)=O)CCCN1NC(=O)CSC1CCOCC1 C(N=C(NCC(F)F)N1CCOC(C2CCC2)C1)c1ccc(N(C)C)cc1 c1(C(N(CC(=O)NCC2CC2C(F)(F)F)CCC)=O)cncc(CC)c1 C(=O)(C(CO)C(C)(C)C)NC(C)(C)C(=O)NC1CC2CCC(C1)S2 N1(C(CC2(CNC(c3ccnnc3)=O)CCC2)=O)CC2CCC(CO)(C2)C1 c1(COC(CCOC(CC)C)=O)cccc(C)c1.C1(C)CN(C)CC(=O)N1 C#Cc1c[nH]nc1C(=O)NC1CCCN(C(C2(C)CC2c2ccccc2)=O)C1 C1(NC(C2CC23CCC3)=O)CCC2(CC1)CCN(c1nc(Cl)nc3ccsc13)C2 Nc1c(C(N2CC(CNC(=O)CC3CC(F)(F)C3)C2)=O)cnn1CC(F)(F)F N1(C(c2cccc(C#C)c2)=O)CCC(NC(C2CCC3CC3C2)=O)C2(CCC2)C1 N1(C(C2C(=C)CC2)=O)CCC(N(C(=O)CCN2CCCCC2=O)CC2CC2)CC1 N#CC1CCCCC1NC(C1C2CC1N(C(=O)CCCNC(N)=O)C2)=O C1(O)(N(C(=O)C(=O)NCC(F)(F)F)C)CCN(C(=O)CC(F)(F)F)C1 N1(c2c(C)cncn2)CC2CC(NC(=O)Cc3ccc(S(C)=O)cc3)CC2C1 N1(C(CC2(C)CC2)=O)CCN(C(c2ccnn2C)=O)C(CCO)C1 Cc1ccc(OC(=O)CCC2CCC(C3CC3)O2)c(I)n1 c1(NC(=O)NCCC(CCNC(C2CN(C(C)=O)C2)=O)C)ccccc1S(C)=O Cc1ccc2c(c1)CC(C(=O)NCC1(O)CN(C(=O)CC3(C)CCCO3)C1)S2 C1(CNC(C(n2c(C)ccn2)C)=O)CC(F)(F)CN1C(c1cccc(F)c1N)=O N1(C(C2(C#N)C(C)C2)=O)CCCN(C(C2(Oc3c(F)cccc3F)CC2)=O)CCC1 c1(C(N2CC(C(C)NC(C=CSC)=O)OCC2)=O)cc(F)c(C)cc1Cl c1(CC(=O)NC(C)CN(C)C(c2cncnc2)=O)ccc2c(c1)CC2 C1(NC(c2cc3occc3s2)=O)COCCN(C(c2ccc(Cl)nc2O)=O)C1 N1(C(c2cc(CCC)on2)=O)CC2(CC(CNC(C3CCCCC3O)=O)C2)C1 c1(NC(C2CCN(C(=O)CCc3cncnc3)CC2O)=O)nc(Cl)cnc1Br C1(O)(CNC(=O)Cc2cc(C3CC3)on2)CCCN(C(C2CC3CC3C2)=O)C1 c1(CN(C)C(=O)NC2CC(F)CN2Cc2ccccc2)ccc(Cl)c(F)c1 C12(NC(c3c(CC)nc[nH]3)=O)CC(CNC(=O)C(C)OC(C)(C)C)(C1)OC2C CCC(CC(=O)NCCCC(=O)Nc1ccc(O)cc1)C(C)C c1(C(=O)NCCNC(C(=O)N(C)C)=O)ccc(O)c2ncccc12 Cn1cnc2c(NCc3nccn3C(F)F)nc(N3CCn4c(cnc4Br)C3)nc12 C1(C(=O)OCC)OCCNCC1N(c1ccnc(F)c1)C(c1cocn1)=O S(=O)(=O)(c1c[nH]ccc1=NC1CC2CC2C1)NCC(COCC)(C)C c1(C(=O)O)ccc(F)c(Cl)c1.C1(N)C2CN(C(C3CC4CC3C4)=O)CC12 CC(CCC(=O)N(C)Cc1ccnn1C)NC(=O)COC(C)(C)C C(=O)(CC(C)(C)C(C)(F)F)NCCC1CCCN(C(c2[nH]c(=NCC)sc2)=O)C1 C1(C(=O)NCC2(C(N)=O)CN(C(CCC(=O)OC)=O)C2)CCN(S(N)(=O)=O)CC1 Cc1nc(C)n(O)c1C(=O)NCC1CCCN1C(c1cccc(CN(C)C)c1)=O C1(NC(C(=Cc2ccccn2)C)=O)CCN(C(c2cnn[nH]2)=O)C12CCC2 N1(C(c2c[nH]c(=NC)s2)=O)CC(C(=O)NC2(C)CC3(CC3)C2)CC12CCC2 C(=O)(CC(C)C(F)(F)F)N1CC(C)(O)C1.C(CN(C(=O)CSC)C)(C(C)C)OC CC(C)C(O)C(=O)NCC1CN(C(C2(C)CC2(Cl)Cl)=O)C1 C12(C(=O)NCC3N(C(C4NC(=O)C(F)C4)=O)CC4(CC4)C3)CC3CC(CC(C3)C1)C2 c1(C(=O)NC2CCCN(C(C(c3c(C)n[nH]c3C)C)=O)C2)cc2n(n1)CCO2 Cc1cc(=O)c(C(=O)NC2CCC(NC(c3occc3Br)=O)C2)c[nH]1 C(=O)(C(C)C1=CCCC1)N(C(C)CN1CCOC(=O)C1)CCO CC1CN(C(=O)Cc2cc(Br)ccc2F)CCN1C(c1cccc(=O)o1)=O C1(CC)CN(C(c2cncc(C(C)C)c2)=O)CCN1C(C1CCCC1C1CC1)=O N1(C(C2C3N(C(COC4(C#C)COC4)=O)C(CC3)C2)=O)CC2(C1)CC(C)(F)C2 Cc1cn2ccnc(C(=O)NCC3CCN(C(=O)C4=CCCCC4C)CC3)c2n1 c1(C(c2nnnn2CCCC)NC(C(=O)NCCOC)=O)nc2ccccc2s1.S Cc1sc(Br)nc1-c1cn(-c2cccc(C(=O)NC(C)C(F)F)c2)nn1 N1(C(C(C)=C2CC2)=O)CCCC1C=CC(=O)NCCCCC1CC1C N1(C(=O)OC)CCC(N(C)N2CCN(c3nc(C4CCCCC4)no3)CC2)C1 C1(C(=O)NC2CCCN(C(c3ccc(=N)[nH]c3Cl)=O)C2)CCc2cncn2C1 C1(NC(C(CCSC)O)=O)CC2CC(NC(c3sc(C)cc3Cl)=O)CC12 C=CC1CCCCN1C(C1(CNC(c2ccco2)=O)CCCCC1)=O C1(C(=O)NC2(C(=O)Nc3cccc(C4CC4)c3)C(C)(C)C2)CCCC(=O)C1 C1(C(=O)NCC(CC)NC(=O)CN(C(=O)COC)C)CCCC(F)C1 Cn1nc(C(=O)NCC(F)CNC(c2ocnc2C(F)(F)F)=O)cc1Br C1(NC(CN(c2ccccc2)C(C)=O)=O)CN(C(=O)CCc2cnco2)C2(CCC2)C1 c1(C(=O)NC(CCNC(c2cc(CC)nn2C)=O)CO)ccc2ncccc2n1 N1(C(CCC(C)N(C)C)=O)CCN(C(c2ccc(C(F)F)o2)=O)C(C)C1 C(=O)(C(F)C(=O)N(C(C)C(=O)NCCCn1cc(C)cn1)C)OCC CCCC(O)CC(=O)N1CCN(C2CCN(C(=O)CCN3CCCCC3)C2)CC1 Cc1sc(Br)nc1NC(c1ccc(Cl)cc1)c1nnnn1CCC1CC1 N1(C(CN(C)C(c2ccsc2)=O)=O)CCC2(NC(C3CCOC3)=O)CCCCC12 C1(N(C(c2c(C(C)(C)C)noc2)=O)C2CC2)CCCN(C(=O)CC23CCCC2C3)C1 CC1CN2CC1(C)C2=O.C1(C(=O)NCc2ccc(Cl)nc2)CC2CC(=O)C1O2 c1(C(=O)NC(c2cn(CC3CCCO3)nn2)CCC)cccc2c1C(=O)NC2=O CC(C)(CCCC(=O)NC1CC(=O)NC(=O)C1)NC(c1cccnc1S)=O C1(C)(C(=O)NC(C2CN(C(c3ccc(CN(C)C)s3)=O)CCO2)C)CCC(F)(F)C1 c1(C(N2C3CCN(C(=O)OCCOC(C(=C)C)=O)C3CC2)=O)cccc(S(=O)(=O)F)c1 C(CC(C(=O)N(C)CC1CCCCC1)NC(=O)Cc1ccc(O)cn1)OCC C(CC(=O)NC1CCCC(NC(C2=CC=C2Cl)=O)C1)(C(N)=O)NC(C)=O c1(C(C)NC(c2ncccc2-c2ccc(F)s2)=O)ccccc1C#N C(=O)(CCCCCCCO)Nc1cccc(C(=O)OC)c1.c12cn(nn1)CCS2 CCCC(C)(O)C(=O)NCC1CC(OC)CN1C(c1cc[nH]c1C1CC1)=O C(=O)(C(C)(C)CS(C)(=O)=O)NCCN(C(c1cc2nnn(C)c2s1)=O)C(C)C c1(C(N(C(C)CCNC(=O)Cc2ccsn2)C)=O)coc2c1NC(=O)CCC2 c1(OC)cc(C(=O)NC2CC(CO)N(C(=O)C=CCN(C)C)C2)n(C)n1 Cc1cnc(N(CC(C)CO)C)c(S(=O)(=O)NCCc2nccn2C)c1 C12(NC(C(C)(C)C)=O)CC1CN(C(=O)C(C)(C)Oc1ccccc1)C2 c1(C(N2CC(O)(CCNC(CCCCC#C)=O)C2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 C1(C2CCN(Cc3cc(C(F)(F)F)nc(Cl)n3)CC2)(NC(C2CN(C)C2)=O)CC1 C(=O)(C1=CNC2=NCCC2=C1)NC(C1CCCN1C(=O)CC1COCCO1)C c1(C(=O)NCC(CC)(CC)NC(C2CCCS2)=O)c(Cl)cncc1Cl CCC(F)(F)CC(=O)N1CC(F)CC1C(=O)NC(c1nc(C)no1)CO N1(C(c2cn(CCC(c3ccc(C)cc3)(C)C)nn2)C2CC2)CC(=O)NC(=O)C1 Cc1ccc(OCC(=O)NCCC2CC(NC(c3cc(Br)[nH]n3)=O)C2)cc1 c1(CC)cc(NC(=O)C(c2cccs2)NC(C2CCC3(CC3)C2)=O)ccc1C C12(C(N3CC(O)(CN(C)C(c4cnn(C)c4C4CC4)=O)C3)=O)CCC(CC1)CC2 C1(C(=O)NCCCCNC(C2(C)CC(F)C2)=O)CCc2ncnn2C1 C(=O)(C1=C(Cl)CCCC1)N1CC(CC)N(C(C2CCCC2)=O)CC1 N1(CC2CCN(C(=O)OCC)C2)CC(=O)N(CCCCC2(C)CSCCO2)C1=O N1(C(c2cccc(C(C)C)c2)=O)CCC12CN(C(=O)Cc1ccnn1C)C2 Cc1cc(NC(c2cc(Br)sc2C)=O)ccc1NC(C1CCCO1)=O C1(NC(CCC=CC(C)C)=O)CC=C(C(=O)NC(C)(C)C(F)F)C1 c1(C(N(CCCNC(C(C)OCC)=O)CC2CCCC2)=O)cc(C)ccc1F N1(C(COC(C)=O)=O)CC(C)(NC(=O)CCc2cnccn2)C1 c1(OC2CCC(NC(=O)C)C2)cc(Oc2ccsc2)ccn1.CC(F)(F)C1(C)CC1 c1(NC(C(N2C(C)(C)CC(N)C2)=O)=O)cc(F)cc2cccnc12 Cc1cc2c[nH]nc2cc1C(=O)NC1CN(C(c2c(F)ccc3ccoc23)=O)C1 c1(C(=O)NCC(CNC(C(C(=C)C)(C)C)=O)F)cc2ccc(SC)cc2[nH]1 C1(C(=O)NC(CC(C)NC(c2cccc3nccn23)=O)C)CN2CCN1CC2C Cc1ncc(CNC(=O)C(c2nn[nH]n2)C2CC2CO)cc1Cl N=c1[nH][nH]cc1C(=O)N(C1(C(=O)NC(C(N)=O)C2CCCC2)CCC1)C1CC1 N1(C(CN(C)CCO)=O)CCCC1CCN(c1ccccc1)C(c1cccn1C)=O c1(C(N(CC2OCCN(C(C=CCN(C)CC)=O)C2)C)=O)cc(O)cc(=O)o1 c1(CC)[nH]nc(Cl)c1C(=O)NCCCN(C)Cc1scnc1C1CCCC1 c1(C(=O)NC2(CO)CC2)ccc(F)c(N2CCC2)c1 C(=O)(C1=NOC2COCC12)NCC(C)NC(c1c(C)c(F)cc(Br)c1)=O N1(C(C)C)CCC(Nc2cccc(CCN3CC(N4CCOC4=O)C3)n2)CC1 C1(NC(c2ccn(C)n2)=O)CN(C(=O)Cc2ccc(F)cc2F)CC2CCCC12 Cc1cnn(C)c1C(=O)NCC1(N(C(c2[nH]cnc2C#N)=O)CC)CCCCC1 C(C(C)C(F)C(=O)NOCC1(C)CCCC1)NC(C(C(CC)C)N(C)C)=O c1(OC)cc(C(N2CC3CC(CNC(c4ccns4)=O)C3C2)=O)cnc1C Cc1ccc(C(=O)NCC(C)NC(c2ccc(C(C)C)cc2)=O)cc1F c1(C(=O)OC)cccc(C(N2CCCN(C(=O)CCN3CCC3)CC2)=O)c1O N1(C(C(CC2CN(C(C3CC(=C)C3)=O)C2)F)=O)CCCC(C)(C)C1C N1(C(C2(CC)CC2)=O)CC2CC(NC(c3ccnn3C3CCC3)=O)C(C2)C1 Cc1sc2ncc(C(=O)NCC3(CNC(C4CCC5C4C5(F)F)=O)CC3)n2c1C C1(N(C(C2C(C=C)C2)=O)CCC)CCCN(C(c2ccccc2SC(C)C)=O)C1 C1(CC)CCN(C(c2ccc(C3CC3)o2)=O)C1C(=O)NCCc1noc(C)n1 c1(C(=O)Nc2cc(COC)no2)[nH]c2cc(-c3ccccc3OC)ccc2c1C CCC(C(F)(F)F)NC(C1CCC1CNC(c1snc(C)c1N)=O)=O C(=O)(C1=CCCCC1C)NC(C(=O)NC(c1c(C)nccn1)C)C C1(NC(C2C(CC)C2)=O)CCSC12CN(C(c1ccn(C(C)C)n1)=O)C2 C1(N(C(=O)Cn2cc(Cl)cn2)CC2(C)CNC2)C2Cc3ccccc3C12 CC1CCCCN1CC(N1CC(O)CC1C(=O)N(C)Cc1cnccn1)=O C1(C#N)(C(N(CCC(C(C)C)NC(CCC(=O)NCCC)=O)C)=O)CC12CCC2 C(C1(O)CCCc2ccccc21)NC(C1(CCc2ccccc2)CC1)=O C1(CNC(C2(CC)CC2)=O)C2CN(C(=O)C(c3cccc(OC)c3)(C)C)CC12 c1(C(N2C(CCNC(CCCC=C)=O)CC(OC)C2)=O)cc2c(C)cccc2o1 C(=O)(CS(N)(=O)=O)NCC1N(C(C(N(c2ccccc2)CC)C2CC2)=O)CC=C1 N1(C(CC(C=C)CC)=O)CCC2CN(C(c3ccc(C(F)(F)F)nc3)=O)CCC12 C(c1ccc(C)c(Cl)c1)=CC(=O)NCC1CCCN(C(C(CCC)(C)O)=O)C1 CC1(C)CCc2cc(Br)ccc2N1C(=O)CC1COC(C(F)(F)F)CN1 c1(C(=O)NCC2CCCC(NC(=O)CCSC(F)(F)F)C2)ccc2snnc2c1 c1(NC(c2cc(COC)no2)c2nnnn2CCCSC)ccc[n+]([O-])c1 Cn1nc(C(N2CCCC2C(=O)N(CCO)Cc2ccccc2)=O)c(Br)c1Cl CCC(CO)C(=O)NC1CCN(C(=O)Cc2ccc(OCCN(C)C)nc2)CC1 c1(C(=O)NC2CN(C(c3n[nH]c(C4CC4)c3Cl)=O)C2)cc2c(cc1O)OCO2 C1(C(=O)NCC2(C=C)CCC2)CN(C(C2(CSc3ccccc3)CC2)=O)CCO1 c1(N2C(C)CC(NC(c3n(C(CC)C)ncc3)=O)C2)nc(C)nc(Cl)c1C C1(CC(=O)NC)CN(C(C2(CC(F)F)CC2)=O)CCN1C(=O)C(C)S(C)(=O)=O c1(C(N2C(CC(N3CC=CC3CF)=O)C3CCCC32)=O)ccc2c[nH]nc2c1 C#CC1(O)CCN(C(C2C3CC4C(C3NC(c3cc[nH]c3)=O)C24)=O)CC1 Cn1ncc2cc(C(N3CCC4CN(C(C5SCCS5)=O)C4C3)=O)sc12 CCC(C)C(O)CC(=O)N1CCCC(C)(C(=O)NC2CC3(CCC3)C2)C1 c1(C(=O)NCC2CC(NC(C(CC#C)C)=O)C2)c(Cl)ccc([N+](=O)[O-])c1Cl CCC(CC(=O)N(CCC(N1CC2(CCC2)CC1CO)=O)CCO)CC(C)C C=CCC(C(=O)NC12CC1CN(C(=O)COCC1CCC1)C2)c1ccccc1 c1(C(=O)OC)ccc(C(=O)NC2CCCC2NC(C2(C3(C)CC3)CC2)=O)c(C)c1 C1(C(N2C3CC(NC(COCCC=C)=O)CC2CC3)=O)CN(S(=O)(=O)N(C)C)C1 N1(C(=O)C=CCO)CCCC1CNC(=O)C(c1ccccc1)O C1(N(C(CCC=C=C)=O)C)CN(C(c2cc(CO)oc2C)=O)CC12CC2 c1(CC)c[nH]nc1C(=O)NOC(C)(C)C(=O)NC1CC1NCCO N=c1nc(N2CCCC(F)(F)CC2)[nH]c(=NCCNC2CC2)[nH]1 N1(C(C2CC(CCC)C2)=O)CC(F)CC1CC(=O)NC(c1ccoc1)C c1(OC)ccc(CN2CCC(C(C)OC)C2)cc1-c1cccc(C(C)(C)C)c1 N1(C(C2C(c3n(C)ccn3)C2)=O)CC2(CCN2C(C2CC23CC3)=O)C1 Cc1cncc(C(N2CCN(C(C3CC4(CCC4O)C3)=O)C(C)C2)=O)c1Cl N1(C(C2COCCN(C(c3nncc(OC)c3)=O)C2)=O)CCC(C2(C)CC2)C1 C1(C(N2CC(COC)(NC(C3(C4CC4)CC3)=O)C2)=O)Cc2ccccc2S1 Cc1ccnc(NC(=O)C(=O)NC2COCCC2C)c1 c1(C(C(=O)NCCN(C(=O)Cc2cccs2)C(C)C)C2CCCC2)cnn(C)c1 Cc1cc(C(=O)NC2CCC(C)N(C(=O)CCc3cn(C)cn3)C2)c(F)cc1F S(=O)(=O)(c1cc(C)cnc1NC1CCSC12CCC2)NCC(CC)CC(C)C c1(NC(C2CCCC(NC(=O)CC3CCCC3O)C2)=O)ccc(O)c(F)c1 CCC(C(=O)NC(C)(C)COCCCNC(C1CC1CN(C)C)=O)C(C)C O=C(CC1CC(=O)Nc2ccccc21)NCC#CCNC(C12COCC1C2)=O C1(C)(NC(c2n(CC)ccc2)=O)CCN(C(=O)CC(C)n2ccc(C)n2)CC1.CCOC Cc1ncnc(C)c1NC(C1CCCN1C(=O)C(C)n1cccn1)=O N1(C(C(CCCC)F)=O)C2CC=C(C(=O)NOC3CCC(O)C3O)C1CC2 c1(C(N2C(C)CC(NC(C34CCN(CC3)C4)=O)C2)=O)ccc2c(c1)OCO2 Cc1ccc2c(c1)SC(C(N1CCCC(N(C(=O)C3=C(Cl)CCC3)C)CC1)=O)C2 C(CC(O)C(=O)NC1CN(C(=O)C(C)OCc2ccc(C)cc2)C1)SC C1(CC(C)NC(c2cnn(C3CC3)c2)=O)CCCCN1C(c1cc(CF)on1)=O N1(C(CCc2n(C)ncn2)=O)CCN2CC(C(=O)Nc3ccccc3)CC2C1 c1(CC(=O)NCCN(C(=O)C(C)(C)NC(=O)OC)CCC)c(F)cncc1Cl Cc1nc2ccc(C(=O)NCC(C)(O)CNC(C3CCOC3C)=O)cc2o1 C(C)(C)(CCCC(=O)NC1(C(=O)N(C)C)CC1)NC(c1scc(C)c1)=O c1(C(C)C)cnn(C)c1C(=O)NC1CN(C(=O)COC2(C)CCOCC2)CC1O Cc1ccc(C(N2CCC(F)(C(=O)Nc3cnc(C)c(Br)c3)C2)=O)cc1O c1(C(N(C2CCCN(C(C(C)C)=O)C2)C)=O)nnc(O)cc1O CCC(CC)C(=O)N1CCC(C(N2CC(c3noc(C)n3)C2)=O)(COC)C1 C1(NC(C2(CC=C)COC2)=O)CCOC(CNC(=O)CC2(O)CCC2)C1 c1(CC)nn(C)cc1C(=O)NC1CC(F)(CNC(c2cccc(OC)c2)=O)C1 c1(CC)[nH]nc(C(=O)NC(CNC(=O)CC2COCCN2C)C(C)C)c1[N+](=O)[O-] c1(CC)c(C(=O)NCCCCCN(C(=O)C(C)O)C)cnn1C(C)(C)C CC(C(=O)NCC1CCN(C(=O)C=Cc2ccc(O)cc2)C1)C(C)(F)F N(C(=NCC1CC1)NCC1CC(=C2CC2)C1)CCc1n(C)ncc1 C1(C(N2C(COC)(CNC(=O)CN3CCCC3=O)CCC2)=O)Cc2nncn2C1 c1(CN2C(C)CCC(NC(c3cnc(C)[nH]3)=O)C2)cccc2ncccc12 N1(C(C(CC)CC)=O)CCC(C2CCN(C(C3(N(C)C)CC3)=O)C2)CC1 c1(OCC)ccc(C)nc1C(=O)NCc1ccoc1C(=O)Nc1ccccc1C C#Cc1cnc(=NCCCCC(C)NC(=O)COc2cc(CC)on2)[nH]c1 C(=O)(C(O)CC[S+](C)C)NCC1C(NC(c2cccc(NC(C)=O)c2)=O)C1 C1(C)(CNC(C2C(C(C)(C)O)C2)=O)CCN(C(C2CCCCO2)=O)C1 C(=O)(CCCCC(N)=O)N1CCC2(NC(CCC(=O)NCCC)=O)C(C1)C2 Cc1cn(C)cc1C(=O)NCCC(C)(C)NC(=O)Cc1ccncc1Cl C(=O)(CC(O)CCOC)N(CCCNC(=O)C(c1ncccc1C)(F)F)CC c1(C(=O)NC2CCCCC2CNC(C2(CO)CCCC2)=O)ccc2c(c1)CCO2 C=C(F)C1(CC(N2CC(C(O)C(=O)NCC3(C)CC(O)C3)C2)=O)CCC1 N1(C(C=CC)=O)CCCC2CN(C(=O)CC(C)(C)OC)CCC12 C1(C(=O)NC(c2cn(C)nn2)CC)CN(C(=O)C(=O)NCCOC)CC(C)(C)C1 c1(CC)nc(=N)[nH]cc1C(=O)NC1CC12CC(NC(=O)Cn1cccnc1=O)C2 c1(OC(C)=O)ccc(C(N2CC(c3cn(C4CC4)nn3)C2)=O)cc1C#N c1(C(=O)NC2CC(CCNC(C3C(C)CN(C)C3)=O)C2)ccnc2ncccc12 C1(C2CCN(C(c3ccn(CCF)n3)=O)C2)(NC(C(CC)OCC)=O)CC1 N1(C(C2C(COC)C2)=O)CCC1CNC(=O)Cc1cnsc1 CCC(CC(=O)N1CCCC1(C)C(=O)Nc1ccc2nccn2c1)CC(C)C N1(C(C(=O)NCC)=O)CCC(CO)(CNC(C2CCN(C)C2C)=O)C1 C12(CNC(C3=CC(C)(C)C3)=O)CC(NC(=O)CCCCN(C)C)(C1)C1(CCC1)O2 C(=O)(CCCC(F)(F)F)NC(C(=O)NC(c1cncs1)C)C1(O)CCC1 C1(CCNC(COC2CC(NC(c3n(C)ccc3)=O)C2)=O)CCOC1(C)C C1(NC(C2(C)CCN(C(C)=O)C2)=O)CCCN(C(=O)C2=CC(C)(C)C2)CC1 Cc1ccc(C(C)C(N2CCCC2CC(=O)NCCCO)=O)cc1 c1(C(=O)NC(CC#C)C(=O)NCCN2CCCNC2=O)cnc(O)cc1C c1(C(=O)NC(C(C)NC(C=CCCC=C(C)C)=O)C)cc(C(F)(F)F)cc(Cl)c1 CC1CCCN(C(=O)CCC2(C)CN(C(C3CCC4CCC34)=O)C2)C1 C(=O)(C(C)(CO)OC)NCCCN(C(=O)C(=Cc1cnn(C)c1)C)CC N1(C(C(CCSC)O)=O)C2CCCC1CN(C(=O)CC=Cc1ccccc1)C2 C1(NC(C(C)(C)CF)=O)C(CN=c2[nH]nco2)CCC12CCC2 CC1CCCCC1(C)C(N1CC(c2ccccc2)(NC(=O)CNS(C)(=O)=O)C1)=O C1(NC(CN(C(C)C)C)=O)CCC(NC(C2CC(Cc3ccccc3)C2)=O)C1 c1(CNC(C23C(CN(C(C(CC)N(CC)CC)=O)C2)C3)=O)c[nH]c2ccccc12 N1(C(CCOC(C)C)=O)C2CCCC1CC(NC(C1CC3C=CC1O3)=O)C2 N1(C(C2(COC)CCCN(C(=O)CC(C)(C)C)C2)=O)CCC(SC(C)(C)C)C1 c1(C(=O)NC(CNC(CC(CCC)C)=O)C(C)C)cc2c(cn1)OCCC2 c1(OC)ccc(C(=O)NCCCCNC(c2ccnc(OC3CC3)c2)=O)c(F)n1 C1(C(CNC(c2cnn(C(F)F)c2)=O)O)CCN(C(C2C3CCCCC23)=O)CC1 C(=O)(C1CCOc2ccc(F)cc21)N(C1CCN(C(=O)CS(C)(=O)=O)C1)C c1(CCN=C(NC2C(C=C)C2)NCCc2cn(C)cn2)c(C)[nH]c2ccccc12 Cc1c(Br)noc1C(=O)NCC1(NC(=O)C(F)(F)c2cnn(C)c2)CC1 Cc1c(F)ccc(C(=O)NC(C)CNC(=O)CCS(N)(=O)=O)c1N N1(C(CSc2n(C)nnn2)=O)CCN(C(C2CCCCC23CCC3)=O)CC(O)C1 N1(C(C(=O)NCC)=O)CC(C(N2CCC(NC(C)=O)C2C(C)C)=O)C2(CCC2)C1 C1(C(=O)NCC2(O)CC(C(N(C3CCCC3)CC=C)=O)C2)CC2CCC1C2 C(=O)(CS(=O)(=O)C1CC1)N1CC2C(N(C(c3cc(C)c(F)cc3)=O)C)C2C1 Cn1ncc(C(N2CC(NC(=O)Cc3csc(S)n3)C(F)C2)=O)c1[N+](=O)[O-] c1(C(=O)NC2C(CNC(Cc3cc(C)on3)=O)CC2)ccc2c(c1)OCC2 CCC(C)(C)CCCC(=O)N1CC(O)CC1C(N1CC(c2nc(C)no2)C1)=O C1(C(N(CCNC(c2ccnn2CCC(F)(F)F)=O)CC)=O)CCC(=O)N1CC C1(C(=O)NC(CNC(c2ccn(C(C)C)n2)=O)C2CCC2)CC(O)CN1C Cc1cncc(CC(=O)NCC2(NC(=O)CSC3CC3)CCOC2)c1 c1(C(=O)NCC2N(C(C(C)SCC)=O)CC(OC)C2)ccc(C)cc1CC C1(NC(c2n(C)cnc2)=O)CC2(C1)CC(CNC(=O)C=CSC(C)(C)C)C2 CCC(C)(C(=O)N1CCC(CO)(CNC(c2ncncc2OC)=O)C1)C(N)=O C(C(C)(C)CN=[N+]=[N-])NC(c1c(CCNC(c2ccc(CC)o2)=O)n[nH]c1)=O Cn1[nH]c(=NC(=O)C2CCn3nccc3C2)c2ccncc12 C(=O)(C1=CS(=O)CCC1)NCCN(CC(C)O)C(c1cc(F)ccc1N)=O N1(C(=O)C=Cc2cnccn2)CCC2(CC1)CN(C(C1CCNC1=O)=O)C2 C1(CC(=O)NCCCCCNC(c2c(CCC)occ2)=O)CCC(=O)N1C C1(C(N2CC(CCC)N(C(=O)CNC=O)CC2)=O)Cc2ccncc2N1 N1(C(C(CC(C)C)F)=O)CCc2sccc2C1CNC(=O)Cc1ccnn1C S(=O)(=O)(c1ccc2[nH]c(=NCC(C)OC)ccc2c1)NCC(COCC)O Cn1ncc(NCc2ncc(Cc3nnnn3C)[nH]2)c1C(N)=O C1(C(=O)NCc2ncc(C)o2)CC(F)CCN1C(=O)Cn1cncn1 C(CCN(C)C)(C(=O)N1CCCC1CO)N(C(C(C)N1CCCC1)=O)C CCCC(C(=O)N(CC(C)C(N1CC(O)CC1CC)=O)C)NC(N)=O CS(=O)(=O)c1ccc(CN2CC3C(NC(c4ccc(Br)c(Cl)n4)=O)C3C2)cc1 CC1CN(C(=O)CC2CCC(F)(F)CC2)CCC1NC(=O)C(C)(C)C1CC1 C1(CC#N)CN(Cc2c(C)cccc2F)CCN1C(=O)Nc1cccc(C)c1Br CC(C(=O)N1CC(O)(C(C)(C)CNC(C23CSCC2C3)=O)C1)C(C)S(C)(=O)=O c1(C(N(CC(C)CNC(=O)CCCN2CCCC2)C)=O)cnc2[nH]cnc2c1 c1(OCC(N2CCC(F)(CNC(C(C)SCCCC)=O)C2)=O)ccc(Cl)c(C)c1 c1(N2CC(C)C(O)CC2)nc(=NCc2cc[nH]c(=N)c2)[nH]c2c1SCC2 CC(C)(F)C(C)(F)CNC(C1(C)CCN(C(=O)C2=CCCCO2)C1)=O C1(C(=O)NCc2ccncc2)CC12CN(c1ncc(Br)cn1)C2 C(=O)(CCCC(C)(C)C)NCC1C(NC(C2(COC)CCC(=O)N2)=O)C1 Cc1cnc2c(C(N3CCCC3CNC(=O)Cc3ccns3)=O)cccc2n1 Cc1ccc2oc(=NC3CN(C(C4CCN(CC(C)C)C4)=O)CC3C)[nH]c2c1 C12(NC(CCCC)=O)CCC(CNC(C3CCC34CCC4)=O)(CC1)C2 C1(NC(C2CC23CCOC3)=O)CN(C(c2cc(Cl)nc(Cl)c2)=O)C2CCCCC12 C1(NC(Cc2c(SC)cccc2)=O)CN(C(=O)CCOCC(F)F)CCC1(C)C C12(CNC(c3cccc(C)c3)=O)CC(C1)C(NC(=O)C(c1cncn1C)O)CO2 c1(C(N2C(CNC(c3n(CC)cc(Cl)c3)=O)CCC2)=O)ccc(C)c(OC)c1 c1(C(CC(=O)N2CC(Cc3nn[nH]n3)C2)N(C)C)ccccc1F N1(CC)CCOC(C(N2CCC(C(C)(C)CNC(=O)CC(C)F)CC2)=O)C1 C1(C)(NC(C=NOC)=O)CCCCC1C(N1CC2CCC(C1)O2)=O c1(C(=O)NC(CN2CCN(C(C=C(CC)C)=O)CC2)C)ccc(Cl)cc1O N1(C(CCCC)=O)CC(CO)C2(C1)CN(C(=O)C(C1CC1)C1CC1)C2 c1(C(=O)NCCC=CC)cc(C(=O)OC)cs1 c1(OC)cc(CC(N2CC(CNC(=O)COc3cnn(C)c3)C(O)C2)=O)ccn1 N1(C(C(CC)C)=O)CCC(NC(c2ccnc(Br)c2N)=O)CC1C c1(OC)ccc2c(C(N3CCC(C)(NC(c4cc(C)co4)=O)C3)=O)n[nH]c2c1 N1(C(C2(CC=C)CC2)=O)CCCC(NC(c2c(C)cc(C)oc2=O)=O)CCC1 C1(C(=O)NCC=CC(=O)NCC2CN(C3CCC3)C2)CCCCC1F C(c1ccc(SC(F)F)cc1)=CC(=O)NC1C2CC1N(C(c1cscn1)=O)C2 C(=O)(CC(C)C(C)(C)C)N(CC(=O)NCCSC)CCOC c12cc(ccn1)NC(=O)CC1CCN(C1)C2=O.C12(CN(C)C1)OC2.CCC.OC c1(C2(C(=O)NC(CNC(CC3(OC)CCC3)=O)C)CC2)nncn1C C1(NC(C(CC)c2ccccc2)=O)CCN(C(=O)CC2CC(F)(F)C2)C12CCC2 C1(C)(CNC(CC(C=C)C)=O)CCCN(C(=O)COC)C1 N1(C(c2c(C)csc2)=O)CCC(C)(CNC(C2CC23CCCC3)=O)C1 CCC(CC)C(F)C(=O)NCC(C(=O)N1CCC(C(=O)NC)C1)C(C)(C)C C(c1ccc(Cl)cc1Cl)=CC(=O)NCC(C1CCOC1)NC(C1CCOC1)=O C1(C(=O)N2C3(CC3)CC2)CCN(C(=O)C2CC2)O1.C1(CC2CC2)CC1 N1(c2ccc(S(=O)(=O)N(C)CC3(CC)CCCC3)cn2)CCC2CCNCC2C1 CC1CCN(C(=O)CC2(O)CCC2)C(C(=O)NCC(C)(O)C(F)F)C1 c1(C(=O)NCC(C)(O)CNC(=O)Cc2cnc[nH]2)ccc(-n2cnnc2)cc1 c1(N2C(=O)C3C(C3)C2)ccc([N+](=O)[O-])c(O)c1.CC1(C)CC1 C(=O)(CC(C)(C)O)N1CCC(C(C)NC(c2c(CC(=O)OCC)scc2)=O)C1 CC1CN(C(=O)Cc2sccc2Cl)CC(C)C1NC(=O)CCc1cncs1 C(=O)(C1=NN(CCO)C(=O)CC1)N(C1CC(NC(CC(=C)C)=O)C1)C N1(C(C2(CSC)CC2)=O)CCCCCC(NC(=O)C(F)(F)CN(C)C)C1 C(=O)(C1=CCCN(C(=O)CC(=O)NC2CCC(C(F)(F)F)CC2)C1)OCC Cc1ccc(S(=O)(=O)N(C2C3CCC2C(C)N3)CC(C)C)cc1C(F)(F)F c1(C(=O)NCC(CNC(c2ccc(OC)s2)=O)O)sc(C)cc1Cl c1(NCC)cc(Cl)ccc1C(=O)NC1CCN(C(=O)CC2CC3(CC3)CO2)C1 c1(CC(=O)NCC(CC(C)C)NC(C2CC2C(C)O)=O)ccc2ocnc2c1 CC(C)(F)CCC(=O)NC(C)(C(=O)NCC1CCCCS1)C1CCC1 CC(C)(C)CC(C)(C)C(=O)N1CC2C(C(=O)NC3CN4CCC3(F)CC4)C2C1 Cn1cncc1C(O)C(=O)NCCC1(NC(c2ccc[nH]2)=O)CCC1 C1(C(C)NC(C2C3CC4C(C3)C24)=O)CCN(C(c2ccnn2C2CC2)=O)CC1 N1(C(c2onc(C)c2C)=O)CC2CCC(CNC(=O)C=Cc3ccoc3)C2C1 N1(C(C2(CCC)CC2)=O)CCN(C)C(C(=O)N(C2CC(CO)C2)C)C1 C1(C(=O)NCC(C)N(C(CN(CCC)C)=O)C)CC(OC(C)(C)C)C1 C=C(C)CC(C(=O)NC1CCCC1CC(=O)NCC1CC12CCCC2)OC Cc1cc(C#N)cnc1C(N1CCC(C)C(CC(N2CCC(OC(C)C)C2)=O)C1)=O c1(C(=O)OCC=C(F)F)cncc(F)c1I N1(C(C=CCN(C)C)=O)CCC(NC(c2ccc(OCF)nn2)=O)C(O)C1 CCC(C)(C)C(O)C(=O)N1CC(N(C(=O)C(C)Cc2cnc[nH]2)CCO)C1 C(=O)(CCCC(C)(F)F)N(C(C)C)CCN(C(=O)CCc1cncnc1)C c1(C(=O)NC2C(NC(C(C)n3cncn3)=O)CCCC2)c[nH]c2ccc(F)cc12 C1(NC(C2C(C)=C2)=O)CC2CCC(C1C)N2C(=O)C(F)(F)c1ccccc1 N1(c2ccc(C(N3CCC(c4c(C)ccnc4)C3)=O)cc2)CC(C)(C)OC1=O C1(NC(CN2CCP(C)(=O)CC2)=O)CCCCCN(C(C2CCC(F)(F)C2)=O)C1 N1(CCNC(C(CCC)C)=O)CCN(C(c2cnc(Cl)cc2N)=O)CC1 C1(CNC(COCC(=C)C)=O)CN(C(c2ccnnc2O)=O)C2COCC2O1 C1(C)CCCN(C(=O)C(C)OCCC=C)C1.C1C(=O)N(N(C)C)CCO1.CC c1(C(N(C(C(=O)NCC(COCC)C)C2CC2)C)=O)ccnc(C)n1 c1(CC)ccc(F)c(C(=O)NCC(CNC(C2(CC)CCCO2)=O)OC)c1 C1(NC(C(C)CSC(F)(F)F)=O)CN(C(C2CCC2)=O)C(C)(C)C1 n1(CC)cc([N+](=O)[O-])c(=NC2CC(NC(=O)CCCc3nccs3)C2)[nH]1 CC(C)C(CNC(C1(CCF)CCC1)=O)NC(=O)Cc1cccn1C C=CCCCCCN=c1cc[nH]cc1S(=O)(=O)N1CCCC(O)C12CCC2 N1(C(COCC)=O)CC(CNC(C2CCN(CC(C)(C)O)CC2)=O)C(C)C1 c1(C(N2C(CC(N3CC(O)C(O)C3)=O)CC(F)C2)=O)ccc(Cl)nc1Cl c1(C(C(=O)N(CC(C)NC(=O)CC2CSCCS2)CCOC)=O)ccc(C)cc1.CC N(C1CCc2c1cnn2CC)C1CCCN(C(C(C(CC)CC)O)=O)C1 c1(C(C)NC(=O)COC(C)(C)C)nocc1C(N1CCC1CN(C)C)=O C=CCC(CC(=O)NCC(C)O)NC(C1(C)CCN(C)CC1)=O CCC(CC(=O)N1CC(N2CCC2)C1)NC(C1(Br)CC12CCC2)=O c1(C(N(C2C3CN(C(C(C(C)C)OC)=O)CC32)C)=O)cc2c(o1)CCCC2 Cc1cc(C)c(CC(C)NC(=O)N(C)C)c(C)c1.C1C(O)CN1CCO C(=O)(Nn1cnnc1)c1c(C)nn(CC(O)CNc2nn(C)cc2Br)c1 n1(C2N(C(CNC(CSC)=O)=O)CCC2)cc(C=Cc2cccs2)nn1 C1(NC(C2(n3cc(CSC4C=CCCC4)nn3)CC2)=O)CCOC(c2cccs2)C1 c1(-c2cn(CCC(=O)N(C(c3ccc(C)cc3)C)C)nn2)cccc(F)c1C#N C1(C(=O)NCC(C)(C)OCCC2CC2)CCCN1N=O.C12(CC1)C(=O)N2 Cc1oc(C(=O)NCCn2cc(CNC(=O)Cc3ccns3)nn2)cc1CO C#CC1CCCC(NC(C2(N(C)C(c3nncn3C)=O)CC2)=O)C1 N1(C(C2CC(C)(CC)C2)=O)CC(NC(=O)C(C2(OC(C)=O)CCCC2)(C)C)C(C)C1 C=CCC(C)(C)CNC(=O)CNC(=O)CNC(=O)CS(C)(=O)=O c1(C(N2C(C3(NC(CNC=O)=O)CC3)CCCC2)=O)cccc2cnnn12 c1(CC)ccc(C(=O)N(C(C)C(=O)N2CC(N3CC(C)(O)C3)C2)C2CC2)cn1 C(=O)(CP(C)(C)=O)N1CCCC(CN(C(CC2(CC=C)CCCC2)=O)C)C1 C1(CCOCC)CN(C(=O)C(N2CC3CC(C)C3C2)=O)CCCO1 C1(CC(N2C(C(C)NC(C3(c4c(C)c[nH]n4)CC3)=O)CCC2)=O)CCCCC1O c1(C(=O)NCC2(NC(C3C(C#C)C3)=O)CCCCC2)ccc2nccnc2c1 CC1CCCC1(C(=O)N(C)CCc1cnn(C)c1)NC(=O)CN(C)C c1(C(N(C)CC2(O)CN(C(=O)CCC3CCCN3C)C2)=O)ccc(CO)nc1 C(=O)(C(C)CCCC(C)=O)NCC1C(NC(CCC(CC)OC)=O)CCC1 N#Cc1ccc2ncnc(N3CCn4c(C(F)(F)F)nnc4C3)c2c1 c1(C(=O)NC2CCC(CNC(C3CC=CCO3)=O)C2)noc2cc(Cl)ccc12 C1(NC(c2c(C)n[nH]c2)=O)CC(CNC(=O)C=Cc2ccco2)C(O)C1 N1(C(CC(c2nccn2C)NC(C2CC(C)(CC)C2)=O)=O)CC(O)CC1COC n1(CC)c(=O)cc(Cl)n(CC(N2CC(OC(C)(C)C)C(c3ccccc3)C2)=O)c1=O c1(C(N2CC3C(C(=O)Nc4ccc(I)cc4F)C3C2)=O)cc(C(F)(F)F)ncc1Br CN1CCN(C2CCN(C(C3CCN(C(c4ccsc4)=O)C3)=O)CC2)C1=O c1(N2CC(OCCCOCCOC)C2)cc(Cl)nc(C2CCC2)n1 CC1(C(=O)NCC(C2CC2)NC(=O)CCCC(F)F)CCC(=O)NC1 N1(C(C(C)=C(C)C)=O)CCC(NC(=O)C(C)(F)F)C(CO)CC1 N1(C(C2C(C)(C)C2(F)F)=O)CCN(C(=O)Cc2ccon2)C(C2CCC2)C1 c1(NC(CCOC)CO)cc(N2CCC(NC(=O)OC(C)(C)C)C2)nc(C)n1 N1(C(CC=CC)=O)CCC=CC1C(=O)N(C)Cc1nc(C)no1 Cc1nc([N+](=O)[O-])cn1CC(=O)NCC1(F)CCN(C2CCSC2)CC1 c1(NC(CC)=O)ccc(O)c(C(=O)NCCC(CC(=O)NC2CC2COC)C)c1 C(=O)(N1OC2CCC1CC2)C1(CC=C)CN(C(=O)CCCC#N)C1 C#CCC(C)(C)C(=O)NC(C1CCN(C(C2C(C(F)(F)F)C2[N+](=O)[O-])=O)CC1)C N1(C(C2CC(=O)OC2)=O)CCC(CCNC(c2coc(C(F)F)n2)=O)C(F)(F)C1 N1(C(C(CC)NC(c2cnc(C)o2)=O)=O)CC(=O)N(C)C2CC12 c1(C(=O)NC2CC(NC(c3ccc(C(C)=O)nc3)=O)C2)ccc(OC)nc1OC Cc1cc(C23NCC(=O)NC(CC)(CC2)CCCNC3=O)no1 C(=O)(CCCC(=O)N1CCC(CN(C(=O)C(C(C)C)c2cccnc2)C)C1)NC Cc1cccc(C(F)C(=O)NC(CNC(c2scnc2C)=O)CO)c1 C1(CCNC(c2c[nH]nc2Cl)=O)CSCCN1C(c1cccc(CC2CC2)c1)=O O=C1CN(C(=O)COc2cccnc2)C(C(=O)NC(C2CCOC2)CO)CN1 CCC(C)C(C)C(=O)N1CCCC1CN(C)C(C1CC(=O)C1(C)C)=O C(=O)(C(C)(C)CC(C)(C)C)NCC(C)NC(=O)C#CC(C)(C)C c1(CN(C)C(C2CN(C(=O)CCS(C)=O)C2)=O)ccc(N2CCCC2)nc1 N1(CCC2C(CNC(=O)NC(c3ccco3)c3ccco3)CCO2)CCCOCC1 Nc1ccc(Cl)cc1C(=O)NC1CC(NC(c2ccc(Br)cc2F)=O)C1 c1(C(=O)NCCN(CCC)C(C2(CO)CCCC2)=O)cc(C)cc(Br)c1 C#CCC(CC(=O)NC1(C)CCCC1(F)F)NC(=O)CP(C)(C)=O C(=O)(C(F)CCC(C)C)N1CC(NC(c2c(C)cc(C#N)s2)=O)C(C)C1 Cc1cc(CC(=O)NCCNC(=O)CC2CCN(CC(F)(F)F)CC2)cc(F)c1 C1(C2CCN(C(C3CCC(=O)N3C)=O)C2)(NC(CCN(C(CCC)C)C)=O)CC1 CC12CSCC1CN(C(C1CCC(CNC(c3ccccn3)=O)O1)=O)C2 c1(C(=O)NCCC2CC(F)(F)CN2C(c2ccccn2)=O)cccc2c1NCC2 N1(C(=O)CCn2cncn2)CC2CC1CN2Cc1ccn(-c2ccccc2)n1 Cc1nsc(C(=O)OC(C)CCC(=O)O)c1I CN(S(=O)(=O)N1CC(O)C(O)C1)C(c1cccc(CO)c1)=O C(=O)(CS(=O)(=O)CCC(F)(F)F)NCCC1CCC(NC(C2(C)CC2)=O)C1 C1(C(=O)NC(C)CNC(c2csc(O)n2)=O)OCCC2CCCCCC12 C(=O)(CC(C)(C)CNC(=O)C(C)C1CCOC1)Nc1cccc(CSC)c1 C1(CNC(CS(=O)(=O)NC)=O)CC2CC1CN2C(C1CCN(C(N)=O)CC1)=O c1(C(N(CC(CC)NC(=O)CCn2nc(C)nc2C)C)=O)ccc(O)c(F)c1 C1(C(=O)NC2CCN(C(CN(C)C(=O)C3CC3)=O)C2)CCC2CC2CC1 c1(C(=O)NC(CNC(CC(CC(C)C)O)=O)(C)C)cc(Br)c2n[nH]cc2c1 C1(C(=O)NC(C)CC2(O)CCC2)C=CCN(C(=O)C=Cc2ccncc2)C1 c1(C(=O)NCC2(NC(CCN3CCN(C)CC3)=O)CC2)cnc2sccn12 CN1CCCC(C(=O)N(C2CN(C(=O)CCCn3ccnn3)C2)C)C1 C(=O)(C(CC)C(C)(C)CC)N1CC(C=C)(CC(=O)NC(c2cnccn2)CC)C1 C1(CC)CN(C(=O)Cc2cccnc2Cl)CCC1NC(c1nc(C)no1)=O c1(C(=O)OCC)cnc(NC(=O)C)cn1.c1(CC(=O)NCCOC)cc(C)on1 c1(CCC(c2nc(C(=O)OCC)on2)N)cccc(Br)c1 C12(CC)CN(C(C3(Cl)CC3(C)C)=O)C(CNC(=O)CC3CCCC(=O)N3)(C1)C2 N1(C(C(C)S(N)(=O)=O)=O)CC(NC(=O)C(C2CC2)C2CC2)CC2(CC2)C1 c1(C(N(C)Cc2cn(CC3CCOC3)nn2)=O)n[nH]c2c1CSCC2 Cc1cnc(Br)cc1NC1CCN(CC2CCCC2)CC1 c1(CC(N2C(CCNC(CC(C)CF)=O)CCCC2)=O)c[nH]c2cc(F)ccc12 C1(C(=O)NC2CC(NC(CN3C(C)C(C)C3)=O)C2)CCc2cnnn2C1 C(C(C(=O)NCC1CC1NC(=O)CCc1n[nH]c(=N)s1)OC)OC c1(CC)cnc2[nH]cnc(NCC(C)(C3CC3)NC(=O)CC3COCCO3)c1-2 N1(C(C(COCC)C)=O)C2CCC1CN(C(=O)C(C)(C)C(F)F)C2 CC1OCCOC1C(=O)NCC(C)(C)CN(C(=O)CCc1ccccc1F)C c1(C(=O)NCCCCCCNC(c2ccc(O)c(F)c2)=O)c(F)cncc1Cl Cn1cc(CC(N2CCC(CNC(=O)C=CC(C)(C)C)C2)=O)cn1 N1(C(C(CCC)C)=O)CCOC(C(=O)Nc2cncnc2O)CC1 C(N=c1cc[nH]cc1[N+](=O)[O-])C1OCC(CNC(COC(C)(C)C)=O)C1 n1(CC(N2CCC(CNC(c3c(Br)cn(C)n3)=O)C2)=O)cccc(N)c1=O c1(OCC)ccc(C=CC(=O)NC2CN(C(C3(C)CC(C#N)C3)=O)CC2C)cc1 c1(C(=O)NCC2CC(C)N(C(C3CC3(F)F)=O)CC2)snc2ccccc12 C(CC(=O)NC(CO)CO)N(C(=O)COC(C)(C)C)C(C)C c1(C(N2CC(C)N(C(=O)CS(=O)(=O)NC3CC3)CC2)=O)cccc([N+](=O)[O-])c1N C=CC(C)CC(=O)NC(CNC(c1ccc(Cn2ccnc2)o1)=O)CO C#CC1(O)CCN(C(C)C(N2CCCC2(C)CNC(=O)CC2CCNC2=O)=O)CC1 Cc1cc2cc(C(=O)NC(C)CCCNS(C)(=O)=O)[nH]c2cc1Cl Cc1c(F)ccc2c(=O)c(C(=O)NC3CCCC34CN(C(=O)CCF)C4)c[nH]c12 Cc1cccc2c1C(NC(N1CC3CCC3C1)=O)CCC2 Cc1nc(C)c(C(=O)NCc2ccc(C(=O)NC3CCCN(C)C3)s2)o1 c1(CC)c(C(=O)N(C)CCNC(=O)CSC(C)C)cnn1-c1ccccc1CC CN1C(=O)CCC1CC(=O)NC1CC2C(NC(c3cnc[nH]c3=N)=O)C2C1 C123CCCC1N(CC2)C(=O)C(C)NC3=O.CC(C(=O)NC1CCCC1)c1cccs1 N1(C(C(CC(=O)OC)NC(C)=O)=O)CCCC2(NC(=O)C(C)(O)COC)CC2C1 n1(C(C)C)ccnc1C(=O)NC1CCC(CNC(c2cnc(C3CCC3)o2)=O)C1 C#CCCC(O)C(=O)N1CC(NC(=O)C(C)=C(C)C)C(C)C1 c1(OCC)cccc(NCC(=O)NCC(CO)NC(=O)CC(C)c2ccco2)c1 Cc1ccc(NC(c2ccnn2C)=O)c(-n2cc(-c3ccncc3)nn2)c1 C1(NCC(Cc2c(OC)ccc(C)c2)CO)Cc2ccccc2OC1C1CC1 CC1(C)COCC2(CCN(C(C3CC(=O)C3(C)C)=O)CC2)O1 c1(N2C(C)(CNC(C(CCCOC)C)=O)CCC2)ccn2nccc2n1 c1(C(=O)NC(C2CC2CNC(C2CC2c2ccco2)=O)C)nccc(C#N)n1 N(C1c2ccccc2CC1NC(=O)CCCCCO)C(C1CN(C)C(=O)N1)=O C1(NC(C(F)OC)=O)CCCCC12CCN(C(=O)CC(=O)OC(C)(C)C)CC2 C(=O)(C1=CS(=O)CCC1)NC1CC2CC(NC(c3ccc(CN(C)C)o3)=O)CC21 c1(CC)nc(C)ccc1NC(=O)NCc1ccc(C)c(OC(F)F)c1 c1(NCc2cn(C3C(F)(F)CCCC3)nn2)cnc2cnccn12 C1(CC(N2CC(NC(c3cnnn3C3CC3)=O)C2)=O)CCC=CCC1 N1(C(Cn2nc(C)c(Cl)c2)=O)CC(C)CCC1CNC(=O)CC1COC(C)(C)C1 N1(C(c2ccc(SC)cc2)C(=O)NCC)CCc2[nH]nc(C3CC3)c2C1 C1(O)(CN(C(C(C2CCCC2)OC)=O)C)CCN(C(=O)C=C2CCN(C)C2)C1 c1(C(=O)NC(C(=O)N(C)CC2CC(=C)C2)c2ccoc2)ccc(C)nc1O C1(C)(C(=O)NCC2C(NC(C(C(C)C)O)=O)CCC2)CCN(C)CC1 Cc1c(Cl)c(C(=O)NCC23CC2CN(C(C2CCCCC2O)=O)C3)nn1C c1(C(=O)NC2CC(NC(C(C)CC3CCCCC3)=O)C2)cccn2[nH]c(=N)nc12 C1(NC(N(CCN(CC(C(C)c2ccccc2)O)C)C)=O)CCC2(CCC2)CC1 Cc1ccc(C(=O)NC23CC(NC(=O)C(c4cc(F)cc(F)c4)C)(C2)C3)c(O)n1 N1(C(C2(C3CCCO3)CCC2)=O)CCSCC1CCNC(C1CS(=O)(=O)C1)=O C=CC(C)(CCOC)C(=O)NCC(C)(CNC(=O)Cc1ccsc1)OC CC1C(C(=O)NCC(CC2CC2)C(N2CCCN(C)CC2C)=O)=NOC1C C1(CNC(c2n(CC)ccn2)=O)CN(C(C2CCCC2O)=O)CCC1(C)C C1(C(N2C(CN(C(=O)C(C3CC3)C3CC3)C)COCC2)=O)CC2CCCC(C1)C2 CC(CNC(C1CC(=O)C1)=O)C(=O)NC(c1nc(=O)o[nH]1)C C(=O)(C#CC1CCCCO1)NC1(CO)CN(C(C(C)Cc2ccc(F)cc2)=O)C1 C1(CC)CCN(C(C2CC(O)C(F)C2)=O)C1C(=O)N(C)Cc1ncco1 c12ccc([N+](=O)[O-])cc1C(=O)O2.CCCCCCCC1CC1 C1(NC(=O)C2CC2)CC2CN(C(c3sccc3-n3cnnn3)=O)CC12 N1(C(=O)CCN2CCC2)CCC(C2OCCC2NC(=O)CSCC(F)F)CC1 c1(C(N(C(C)CN(C(=O)C(C)C(F)(F)F)C)C)=O)cc2c(Cl)cc(Cl)cc2[nH]1 C(c1ccc(OC)c(F)c1)=CC(=O)NCC(CC=C)NC(=O)C(C)C(CC)CC c1(NC(C(CC=CC)NC(c2occc2C2CC2)=O)=O)cc(C)cnc1C c1(OC)cccc2c(C(=O)NC(CNC(=O)C(C)SC)CC(C)C)n[nH]c12 C1(CCOC2CN(C(C3CN(C(N)=O)C3)=O)C2)CSCN1NC(C1CCC1)=O N1(C(C2N(C)CCC2)=O)CCC2(CCCN2C(c2ccc(C(C)(F)F)nc2)=O)C1 N1(C(c2cn(C)nn2)=O)CC(NC(=O)C#CC2(C)CCCO2)C(S(C)(=O)=O)C1 CCC(C)(CO)CN=c1[nH]c(=N)[nH]c(=NCc2nc(-c3ccccc3C)cs2)[nH]1 Cc1c(C(=O)NCC(O)CNC(C2C3(CC3)C23CC3)=O)ccc(Br)c1F C1(C(N(CCN(C)C)C)=O)C2CN(c3ccnc(C(=O)O)n3)CC12 C(=O)(C1=CCCCCC1)N1CC(C)C(CNC(=O)Cn2cnc3ccccc23)C1 C1(O)(CN(C(c2nc(COC)sc2)=O)C)CCCN(C(C2(C(F)(F)F)CC2)=O)C1 C12(CNC(CCn3c(C)nc(C)n3)=O)CCC1CCN2C(c1ccc(O)nc1)=O CC1=C(C(=O)NCC(C2CCCN(C(=O)CCc3cnn[nH]3)C2)(C)O)SCCO1 Cc1sc(C(N2CCC(N(C(=O)C(C)n3ccnn3)C)CC2)=O)nc1Br c1(C(N2CCOCC2C(=O)OC(C)C)C(=O)NCCOC)cc(Cl)c(OC)cc1Cl c1(CC(C)C)cc(F)ccc1CCNC(=O)NCCC1COC(C)(C)C1 CCCCC(CC)C(=O)NCC1(COC)CCCN1C(=O)C(C)(C)S(C)(=O)=O c1(C(N(CCNC(CCC2C(C)C2)=O)C)=O)cc2cc(F)ccc2s1 N1(C(C2CCC=CCC2)=O)CCCC1(C)CNC(C1(c2ccccn2)CC1)=O N1(C(C2C(C=C)CC2)=O)CCCCC(NC(c2cc(O)n(CC)n2)=O)C1 N1(C(CCCCSC)=O)CC(NC(c2sc(C3CC3)nc2C)=O)C2(CCOCC2)C1 C1(CC)CN(C(=O)C(C)(C)CSC)CC1C(c1ccc(Cn2ccnc2)cc1)=O c1(C(N2C(C(CNC(C(C)SC)=O)(C)C)CCC2)=O)cc2ccc(OC)cc2o1 C1(C(N2CCC(NC(C=CC=CC)=O)C2C)=O)CCC(C)C(C)C1 C1(C(=O)NCC(C)NC(CC(=O)NCC#C)=O)CC1C1CCCC1 C(=O)(C(C)(C)C(C)C)NCC1CC(NC(Cc2c(C)nsc2)=O)C1 C1(NC(C2N(C(COC(C)(C)C)=O)C3(CC2)CC3)=O)CCOC12CCOCC2 N1(C(C(CC)OC)=O)CC(NC(C2C(OCC)C2C)=O)CC(F)C1 C1(C(=O)NC2C(CNC(Cc3cc(C(C)C)no3)=O)COC2)OCCN(C)C1=O c1(C=O)ccc([N+](=O)[O-])n1C.C1(CNCC)CCCCN1C(=O)CCCOC C1(CC)CN(C(c2ccncn2)C(=O)NCc2ccccn2)CC(C)S1=O C1(CCNC(C2(CC#C)CCCO2)=O)CCN(C(=O)Cc2ccc(C)s2)C(C)C1 C(C(=O)N1CC=C(C)CC1)(C(C)(C)C)NC(C(CC=C)C)=O N1(C(CC2(CC)CC2)=O)CCN(CC(C)NC(C2CCC(CC)CC2)=O)CC1 N1(C(c2n(C)nc(CNC(C3(C)CC3(C)C)=O)c2)=O)CCCC12CCOCC2 c1(-n2cc(C(COCc3ccccc3)OC)nn2)ccc(C(N)=O)cc1 C1(C(=O)NCC(C(=O)NC)O)CC2CCC(C1)N2C(=O)COC(C)C C1(c2cccs2)(C(=O)NC(C)CN(C(=O)CCc2ccccn2)C)CCOCC1 c1(CC)onc(C(N2CC(C(=O)NCCC(C)C(=O)OC)(COC)C2)=O)c1C c1(C2(CC)CCCC2)ccc(F)cc1.C1C(C)NC(=O)C2CC2C(=O)N1CC C(=O)(C(F)(F)CC(C)C)NCC(CC)NC(=O)C(C)n1ccnc1 C1(NC(c2ncccc2C2CC2)=O)CCCCCC1NC(C1CCCC1CF)=O C1(O)(CNC)CCCCCC1.C12CN(CCO1)C2=O.C1(=O)C(O)CCC1=O N1(C(CN(C2CC2)CC)=O)CCC(C)(NC(=O)C(c2ccccc2)C)CC1 C1(C(N2CC(OC(C)=O)C2)=O)C2CC3C(C2NC(=O)C(C)CC2CC2)C13 C(=O)(C(O)C(F)(F)F)N1CC(C(Cn2cc(C3(C)CCOC3)nn2)=O)C(O)C1 c1(C(NNC(c2c(SCC(C)C)cccc2)=O)=O)cccc2c1OC(C)(C)C2 C#Cc1cc(NC(=O)CC(CC)c2ccccc2)cc(C(=O)NC(C)(C)C)c1 N1(C(Cc2cc(C)nn2C)=O)CCC(C2CC2)C1C(N1CCC(OCCF)C1)=O N1(CC)CCCC1CC(=O)NC1(C)CC(NC(C2CC2C(C)(F)F)=O)C1 c1(CC)ccc(F)c(C(=O)NC2CCN(C(=O)C=CCOC)C(C)C2)c1F Fc1cc(NCc2cc(-c3ccccc3)cc(Cl)n2)c2ncccc2c1 N1(C(CCCC=C)=O)CCC2(CC1)CN(C(c1scnc1C)=O)CCO2 C=CCCC(=O)NCc1ccc(C(=O)NCCCF)s1 C12(C#CC(=O)NC1)COC2.C(=O)(CCCC(C)=O)N1C(C)CC(CC)C1 c1(NC(C2C(C)C2C)=O)ccc2[nH]c(C(N)=O)cc2c1 N1(C(CC(CC)C2CC2)=O)CCCC12CCN(C(C1COC3COCC13)=O)C2 c1(OCC(=O)NC(C(C)NC(c2c(C)noc2Cl)=O)C(C)C)nc(O)nc(O)n1 N1(CC(=O)N(CCCNC(C2(C3CC3)CCCO2)=O)C)CCC(=O)NC1=O c1(C(=O)NC(C2CCN(C(c3c(CC)c[nH]n3)=O)C2)C)ccc(S(C)(=O)=O)o1 C1(=O)C2=NOC(C2)CN1.C(C(CO)NC(C1CCO1)=O)SCC CCCC(C(=O)NCC1CC2(CCC2)C1)NC(=O)CN1CC2CC2C1 c1(CN2CC(C)N(C(=O)Cn3cccn3)CCC2)c2c(nn1C)CCOC2 c1(C(n2cc(C(=O)OC)nn2)C)ccc(N)cc1C(N1CCC(CC)CC1)=O C1(NC(c2c(OC)cns2)=O)CC2CN(C(c3onc4c3CCCC4)=O)CC2C1 C1(C(N2CCCC(CCNC(C3(CC)CCC3)=O)C2)=O)C2CCC(F)(F)C12 C12CCN(CC1(F)F)OCCNC(=O)C2.c1(Cn2cncn2)c(Cl)ccnc1Br c1(NC2COCCN(Cc3c(C#N)c(F)ccc3)C2)ccn2ncc(Br)c2n1 C1(NC(CC(C)C(F)F)=O)CN(C(c2cc(C#N)cs2)=O)CC1C1CC1 C12(C(=O)NC3(CCNC(CCn4ccc(C)n4)=O)CC3)CCCC1CC(=O)C2 CCC(C(=O)N(CC(C)(C)NC(c1cnoc1C)=O)C)Sc1ccccc1 C(=O)(C(C)(O)C(C)C)NC(c1cccc(OC)c1)CNC(CC(COC)C)=O CC(C)(C)CC(C)(C)C(=O)NC1C2CCC1N(C(=O)C(O)C(F)(F)F)C2 C(=O)(C1=CS(=O)CCC1)N(C)CC1CCN(C(CCCn2c(C)cc(C)n2)=O)C1 N1(C(C(C2CCCC2)OC)=O)CCCC(CO)(CNC(c2ccc(O)nc2)=O)C1 c1(C(=O)NC2CN(C(C(C(C)C)C(C)C)=O)CC2O)cc2c(F)c(F)ccc2s1 C(=O)(C1CCCc2sc(=N)[nH]c21)NC1CCCN(C(C(C)(C)c2cccs2)=O)C1 c1(OC)ccccc1NC(=O)C(N1CC(O)(CN(C)C(C2C3CCCC23)=O)C1)=O N1(C(CCC(C)=O)=O)CC2CC(C(=O)NCCCC3CC3)CC2C1 C(=O)(CCCSC)NC(C(=O)NC(COC)COC)C1CCCO1 n1(CC)ncc(Cl)c1C(N1CCCC1(C)CNC(C1COCC1OC)=O)=O c1(CNC(C)COc2ccccc2)cnc(Cl)cc1Br c1(CNC(=O)CN(CCO)C(c2ccccc2CO)=O)cc(Cl)ccc1F C1(C(N(CCNC(C2CCS(=O)(=O)C2)=O)CC)=O)Cc2ccccc2N1C(C)=O Cc1c(C=CC(=O)NCC2CCN(C(=O)C(O)Cn3cncn3)CC2)cnn1C C#CCC(C(=O)N1CC[Si](C)(C)C1)NC(c1ccc(F)cc1)=O C1(C(N2CC3C(NC(CC4C(=O)NC(=O)N4)=O)C3C2)=O)C2C=CC(C2)C1CO C(CN=c1[nH]c2c(c(=NC3CCN4CCC3C4)[nH]1)CCCC2)N1C(=O)C=NC=CN=N1 c1(N(C)Cc2ccsc2)nc(=NCC2CCN3CCC2C3)[nH]c2c1SCC2 C(=O)(C1CC(=O)Nc2ccccc21)N1CC(NC(C2(OC)CCOCC2)=O)C1 CCC(C(=O)NC1CCN(C(c2ccc(F)c(O)c2)=O)CC1F)C(C)C N1(C(c2c(C)nns2)=O)CCC2(NC(=O)C(C)SCc3ccccc3)CCCC12 C(=O)(CS(=O)(=O)C(C)C)NC(CC)CN(C(C1CC2CCC(C1)O2)=O)CC C1(NC(CCCC=C=C)=O)C(C)CN(C(=O)C=CCOC)CC1C c1(CCN(C2CCSCC2)C)ccc(C(=O)O)cc1 Cc1nn(CC(=O)NCC2CCCC2NC(=O)C=Cc2ccsc2)c(=O)o1 C1(O)(C(=O)NC(CCC)CNC(=O)C(O)CN(C)C)CCN(CC)C1 C1(CNC(C2CC(OCC)C2)=O)CN(C(=O)C#CC2CCCOC2)CCC1(C)C N1(C(C(CC)NC(C)=O)=O)CCN(CC(N2CC(Cn3ccnn3)C2)=O)CC1 c1(C(=O)NC2CC(CS(C)(=O)=O)C2)cccc(S(=O)(=O)CF)c1 CC(C)(C)C(CNC(C1CC12CC2(F)F)=O)C(=O)NCc1cccc2[nH]ncc12 CN1CCN(C(=O)CN2CCN(C(=O)C=CC3CCCCC3)CC2)C(CO)C1 C(=O)(C1OCCc2ccccc21)NCCN(C)C(c1nnc(O)cc1O)=O n1(CC)nc(C)cc1C(=O)NCCC1CCN(C(C23CCCC2C3)=O)CC1 c1(SCCOC)ccccc1C(=O)OC1(C(=O)OC)CC(C)(OC)C1 C1(C(N2CC(OCCNC(=O)C3CC3)C2)=O)CC(=O)N(CC(F)(F)F)C1.C1CCC1 CC(CC=Cc1ccccc1)C(=O)NC1CCC1C(C)C C(C(C)C(=O)NC(c1ccccc1)CNC(c1cnn(-c2ccccc2)c1)=O)OC c1(C(=O)NCC2C(C(=O)NC(c3cncc(F)c3)C)CCC2)cc(Cl)n(C)n1 C=C1CCC(CNC(=O)CC(CC)N(C(=O)CCC2CCCO2)C)CC1 c1(C(=O)NC2(C3CCN(C(Cn4ccc(C)n4)=O)CC3)CC2)occ2c1CCC2 N1(C(C2(C#N)CCCC2)=O)CCOC(C(N2CCOCC2C(F)F)=O)CC1 C(=O)(CS(=O)(=O)c1ccccc1Cl)N1CCC2(CC(NC(COC(C)C)=O)C2)C1 n1(CC(=O)NC(C(C)NC(=O)C(C)c2ccsn2)(C)C)ncc2cccnc12 CC(C)C(C(=O)NCC1(CCNC(=O)CC2COCCN2C)CC1)NS(C)(=O)=O C(=O)(C(C)N(C(=O)CCSC(F)(F)F)C)N(CCOCC#C)C N1(C(C(CCC)C(C)C)=O)CC2CCCN(C(c3ccn(CCF)n3)=O)C2C1 c1(C(=O)NC2CCN(C(c3c(N)cccc3)=O)CC2CO)nc[nH]c2ncnc1-2 C1(C(N(CC(C)NC(C2CC(=O)CS2)=O)C)=O)CCC(F)(F)C1 N1(C(CCCCONC(=O)NC(CC)(CC)CC)(C)C)CCSC(C)(C)C1 Cc1ccc(CNC(=O)CN2CC(C)CCC2C)c(C)c1.C(=O)(C1CC1)O C12(NC(c3cc(Cl)c[nH]3)=O)CCCC1CN(C(C1Cc3cscc3C1)=O)C2 C(C(CC1CC1)C(=O)N(C1CCSCC1)C)NC(C=CC(C)C)=O Cc1cc(C(=O)NCCOCC(N2CCCC2(C)C(C)C)=O)[nH]c1C c1(CC)c(C(N2CC(NC(=O)CN3CCOCC3)CC(C)C2)=O)cnc2ncnn12 Cc1cnsc1C(=O)NC(CC1CCOCC1)C(=O)NCc1cnco1 c1(C(N(CCNC(C2=CC(C)CC2)=O)C2CC2)=O)cc2c(F)c(F)c(F)cc2[nH]1 CC(CC(C)(C)C)C(=O)NC1CC(CNC(c2cccn2CC#N)=O)C1 c1(C(=O)NC(CC(C)NC(c2c(C)ncs2)=O)C)cc2ccccc2nc1O c1(C(N2CCCN(C(C3(C)CC3(F)F)=O)CC2)=O)nnn2ccccc12 CC1(N=c2[nH]nc(C(F)F)o2)CCC(NC(=O)N=c2cc[nH]cc2)CC1 C1(C)(CNC(C2CN(CC)C(=O)C2)=O)CCCN(C(C2CCC(C)CC2)=O)C1 N1(C(c2c(CC)cns2)=O)CC2ON=C(CNC(=O)Cn3cncn3)C2C1 c12cccc(n1)C(=O)NCCC1(CC1)N2.CCC(CC)=CCOC C1(C(N2CCC(C(C)NC(=O)CSc3cn[nH]c3)CC2)=O)CCC(=O)CC1C N1(C(CC(C)SC)=O)CC2(CCN(Cc3cn4ccccc4n3)CC2)CC1C C1(CCN2C(Nc3ccccc3)CCCC2)(OC)CCN(CCC=CCl)CC1 N1(C(c2cnc(C)c(N)c2)=O)CCOC2(CCCN(C(=O)C(O)CC(C)C)C2)C1 c1(OCC)ncc(F)c(N2CC3CC(C2)N3Cc2nccn2C)n1 N1(C(c2cc(OCC)n[nH]2)=O)CCCCC(NC(c2cc(C(C)(C)C)n[nH]2)=O)C1 Cc1cnc(C(=O)NC2(C)CC(NC(=O)CCC3CCCC(O)C3)C2)cn1 c1(C(=O)NC2CC3(C(C(=O)NCc4ccc(OC)nn4)C3)C2)c(C)oc(C)c1C CCCC(O)CC(=O)NCC1COCCN(C(=O)C(C(C)O)N(C)C)C1 c1(C(=O)NCc2c(CC)nn(C)c2)nc(=NCCN(C)C)[nH]c2c1CCCC2 c1(NC(N2C(C(c3n(C)ncc3)=O)CC3CC23)=O)c(Cl)cc(C#N)cc1Cl c1(C(=O)NCCOCCN(C)C(C2CC2C(F)(F)F)=O)cccn(O)c1=O Cc1cc(NC(c2ccc(F)c(Br)c2)c2nccn2C)cc([N+](=O)[O-])c1 C(C(=O)N1CC(C(C)C)=NO1)n1cc(C(N2CCCC(CCCO)C2)CC)nn1 c1(C(n2c(-c3nc(C4CCC4)cs3)nc(C(CC)O)n2)C)ccc(C#N)cc1F c1(CC(=O)NC2CC(OCC(=O)N(C)CC34CCCC3C4)C2)cc(F)ccc1F C1(C(N(CC)Cc2ccoc2)=O)CC(C)(C)CN1C(=O)Cn1cccn1 C1(C(=O)NC(C)Cc2ccccn2)CN(C(c2c(C#N)ncn2C)=O)CC12CC2 N1(C(C(CC)F)=O)CCC2(NC(C3C(c4ccccc4)C3[N+](=O)[O-])=O)CCCC12 C1(NC(C2N(C(CC)=O)CCCC2)=O)CC12CCN(C(=O)CC(C)C(C)C)CC2 c1(C(N2CC(CNC(C(CC)OCC)=O)OCCC2)=O)cc2ccc(C)cc2[nH]1 c1(C(=O)OC)ncccc1NC(N1CCCC(Cn2cc(C(C)(C)C)nn2)C1)=O CC1CN(C(=O)CCCCCF)CC(CCNC(c2cc(C3(C)CC3)on2)=O)O1 Cc1ccc(F)c(OCC(=O)N(C(CNC(C2CC3CC3C2)=O)C2CC2)C)c1 c1(C(=O)NCCN(CCC)C(C2COCC2C(F)(F)F)=O)ncoc1C1CCCO1 C1(CC(=O)NC2C(NC(CCN(CC)CC)=O)CCOC2)CCCC(C)(C)O1 N1(C(c2ccc(CCC)s2)=O)CCC2CCN(C(c3nccc(C)n3)=O)CC2C1 c1(C(C)=O)cc(Br)ccc1NC(C1CC(F)CN(Cc2ccnc(F)c2)C1)=O c1(C(=O)NC(=O)C)c(F)cccc1F.CC1(CO)CCC(NC(=O)CN2CC3CC3C2)C1 S(=O)(=O)(CC(C)(C)CNCCC1CC1)NC(C1CN(C(=O)OC(C)(C)C)CC1O)=O C1(NC(C(c2cccnc2)NC(C(C)C)=O)=O)CC2CC1C(O)C2O C(=O)(C1CNC(=O)c2ccnn21)NCC1N(C(CC2CC(OC)C2)=O)CCCC1 Cc1ccc(CCC(N2CCCC2CCC(=O)NC(CC2CC2)CO)=O)cc1Br C(C(CNC(=O)CCOC)OC)NC(COCCCC)=O c1(C(N(C2CCN(C(C3(C#N)CCC3)=O)C2)CC)=O)cc(F)c[nH]1 c1(N2C(C(=O)OC(C)=O)CC(O)C2)cc(NC)c(N(C)C)nn1 CC1=NS(=O)(=O)NC=C1C(=O)N1CCOCC(NC(=O)CS(=O)(=O)CCOC)C1 c1(C(N2CCCN(C(c3c(CC)c[nH]c3)=O)CC2)=O)cnc(C(C)(C)C)nc1O C(=O)(CC1=NN(C)C(=O)C1)NC1CCCCCN(C(c2c(C(=O)OC)coc2)=O)C1 c1(C(=O)NCC2(F)CC(CNC(CC3(C=C)CC3)=O)C2)nc(C2CC2)oc1C c1(CCCC(N2CCC(CN(C(=O)CCN(C)C)C)C2)=O)csc2ccccc12 c1(OCC(=O)NCC2CC(CNC(C(C)NC(CC)=O)=O)C2)ccc(CO)cc1 C1(C)(NC(CCCN(C(=O)OC)C)=O)CCN(C(=O)C(C(C)C)N(C)C)C1 c1(C(=O)NC(C)C(C)NC(=O)CSC2CCCC2)cn(Cc2ccccn2)nn1 N1(C(C(CCCNC(CC(=C=C)C)=O)O)=O)CCn2c(cnc2C)C1 C1(NC(c2ccc(COC)o2)=O)C=CCC(C(=O)Nc2cnn(CCF)c2)C1 N1(C(CC(C)(C)OC)=O)C2CCCC1CC(NC(c1csc(Cl)c1)=O)C2 N1(CCOC)CCN(C(=O)C(CCC2CC2)NC(=O)Cn2cnnc2)CC1 C1(NC(c2cc(C(C)(C)C)sc2)=O)CCCC(NC(C2COCCO2)=O)C1 C1(NC(C(C2CCC2)NC(c2ccc(C(N)=O)[nH]2)=O)=O)CC(F)(F)C1 C1(N(C)C)CCN(C(=O)C(C2(C(N)=O)CCCCC2)(F)F)C1.c1ccccc1 CC(CNC(=O)C(C)n1cncn1)C(=O)Nc1ccncn1 CC(=O)CCCC(=O)N1CCC(C)C1C(=O)NCc1ccccc1C#N C1(C(N)=O)CN(C(=O)Nc2ccnc(F)c2)CCN1 c1(CC(=O)NC(C(C)C)CNC(=O)CC2CCCSC2)ccc2cccnc2c1 N(C)(C1CCCc2cccnc21)C(=O)NC(c1ccc(C(F)(F)F)cc1)C(C)C CC1OC(C)C(C(=O)OCC(=O)Cc2ccc(CN)cc2)C1C C1(C)(C(N(CCCNC(CCc2onc(C(C)C)n2)=O)C2CC2)=O)CC(O)CN1C c1(C(=O)OC)nccnc1NC1CN(C(C2CC2Br)=O)C1 c1(C(N(CCCNC(=O)C=Cc2nccs2)C2CC2)=O)ccnc2c1CC(=O)N2 c1(C(=O)NCCNC(CC(c2ccc(C)cc2)(C)C)=O)c(C)ccc2nonc12 c1(OCCCC(=O)N(C2CCN(C(c3ccccn3)=O)C2)CC)ccccc1F c1(C(=O)NC2CC(CNC(=O)C(O)c3ccco3)C2)cnc2c(c1)CCOC2 N1(C(C(C)=C(CC)C)=O)CC(NC(=O)Cc2cccc(Br)c2)C(O)C1 CC(C(C)(C)O)N(C)C(C1CCN(C(=O)C=CC2CCOC2)C1)=O c1(CC(N2CC(C)C(C(F)(F)F)C2)=O)ccc(Br)cc1Br c1(C(N2CC(CC)C(c3ccccc3)C2)=O)cc2cccc(C)n2n1 C(=O)(CCCCC(N)=O)NC(C(=O)NCC1CCC(CC)O1)(C)CSC C1(C(=O)OC)C2CC2CN1C(C1CC(C)(NC(=O)C(O)C2CCC2)C1)=O c1(C(=O)NC(C)Cc2ccccn2)cccc(Cl)c1C1(O)COC1 N1(C(COCC(C)C)=O)CCC2CN(C(=O)C(C)C(F)(F)C(F)F)CCC12 CC1(C)CCN(C(=O)CCCc2ccsc2)C(C(=O)NCC2CCC(=O)NC2)C1 c1(C(=O)NCC2C(C)CCN(C(=O)Cn3nccn3)C2)cccc2c1nnn2C C(CCCCCC(=O)Nn1ccnn1)NC(C(CC)SC)=O c1(OC)ccc(F)c(C(=O)NCC2COCCN2C(=O)CN2CCS(=O)CC2)n1 C1(C(=O)NCc2n(CC)cnc2)CC(F)(F)CN1C(=O)C(=O)NOC CCC(CCCC(=O)NCC(O)CC(C)C)NC(C1C2CCC(F)C12)=O C(=O)(C1=NOC2(CCOC2)C1)N1CC2CC(C)C2C1.C1(=O)CN1C c1(C(=O)NC23CCN(C(c4n(CC)ccn4)=O)CC2C3)cccn2ccnc12 c1(NC2(C)CCN(C(=O)NC(c3c(C)n[nH]c3C)C)C2)cc(N)c(C)cc1Br c1(C(C(=O)NC2(CC(=O)OCC)CC2)NC(CCSCC)=O)c(C)cccc1Br C1(NC(=O)C2=CCCCO2)CN(C(c2ccc(Cl)nc2Cl)=O)CC2(CCC2)C1 c1(C(=O)NC(CN(C(C(CC)C#N)=O)C)C)cc2cc(C)cc(C)c2[nH]1 C1(CNC(CCc2c(C)ncs2)=O)CCCCN(C(c2coc(C#N)c2)=O)C1 C(=O)(C(CCC)NC(c1ocnc1CCC)=O)N(CC#C)CCF C(C(N)=O)(C(C)(C)C)NC(c1c(C)n(-c2ccccn2)nn1)=O C1(CNC(C2(CC)CC2)=O)CN(C(=O)C(N)=O)CCC12CCOC2 C=CCC(C)(O)C(=O)N1CC(F)(C(=O)NCCCCCOC)C1 c1(C(=O)NCC(CO)NC(CC2C(C)(C)C2(C)C)=O)cnc2nc(Cl)ccc2c1 C1(SC)COCC1NC(=O)CC1CCN(C(=O)C=CC(C)C)C1 NC(=O)CCC(C(=O)NC(C1CCCO1)C1CC1)n1cc(Cc2cncnc2)nn1 C1(NC(C2CCC(F)(F)C2)=O)CCN(C(=O)CN2CC3CC3C2)C12CC2 c1(C(=O)NCC2CC(NC(C(C)NC3CCOC3)=O)C2)cc(C2CCCC2)[nH]n1 N1(C(c2c(CC)cc[nH]2)=O)CC=C(C(C)(C)C(=O)NOCC2CCCO2)C1 C1(NC(C(CSC)O)=O)CN(C(c2cccc(-c3cccnc3)c2)=O)CC1F C1(O)(COCC)CCCN(C(=O)C(C(C)(C)C)n2cc(-c3cc(OC)no3)nn2)C1 c1(CNC(CCC)=O)cn(CC2CCCN2C(c2ccnn2CC)=O)nn1 N1(CC)CCN(CC(=O)NC2(CF)CCN(C(C3CC4CCC4C3)=O)C2)CC1 Cc1cc(F)c(CC(=O)NC(C)CNC(C23CC2COC3(C)C)=O)cc1F c1(C(=O)NC(C(C)C)CNC(=O)CCCCCNC(N)=O)cccc2nn(C)cc12 C1(C(=O)O)CCN(C(C2CCN(S(=O)(=O)CC3CC3Cl)CC2)=O)CC1 N1(Cc2c(C)ncs2)CCC2CN(C(=O)CCc3cccc(Br)c3)CCC12 CCC(CC)C(F)C(=O)NC1CCN(C(=O)Cn2cc(C(C)O)nn2)C1 c1(C(N(CCNC(=O)C(c2ccccc2OC)O)CC)=O)ccnc2[nH]ncc12 C(=O)(N(CCC(=O)NC1C2C=CC(C2)C1CO)OC)c1c(CC)c[nH]c1 C(C(=O)C1CCOc2ccccc21)OC(Cn1nc(C)c(Cl)c1)=O C#Cc1ccc(CNC(=O)C(C)CN(C)C(C2OCCC2(C)C)=O)cn1 CCCN=C(NCc1cc(OC)ccc1F)N1CCC(C2CCCCO2)C1 C(=O)(C1CNc2ccccc21)OC.CC12CN(CC(=O)N1)C2 C=CC(C)(C)C(=O)NCC1CC(F)(CNC(=O)CNC(=O)OC)C1 C12(C)CCN(N3CCC(CC3)N(C)OC(=O)N1C)C2.c1(SCC)ccccc1 C1(CC(N2CC(C(=O)NC)OCC2)=O)CN(C(=O)CCC(C)=O)C(C)(C)C1 c1(C(N2C(CNC(Cc3ccc(C#C)cc3)=O)C=CC2)=O)cc(F)c(F)cc1F C1(NC(CC(C(C)C)NC(=O)CC2CC=CCC2)=O)CC2COCC(C1)C2 c1(OC)ncc(CNC(C2CCN(Cc3ccsc3)CC2)=O)cc1Cl C1(N(C(C2N(C)CCC2)=O)C)CC2CCC(C1)N2C(=O)CNC(=O)CN(C)C n1(C(C)C)cc(Br)c(C(=O)N(C)CCNC(C2CC3C=CC2C3)=O)n1 c1(C(C)C)cccc(C(N2CCC(NC(=O)CCc3cnoc3)C(F)C2)=O)c1N C1(NC(c2c(C)coc2C)=O)COC2(C1)CN(C(C1CC3CC(=O)C1O3)=O)C2 Cc1nc(C)c(C(=O)NC2CC(C)(C(=O)NCCOCC(C)(C)O)C2)s1 Cc1c(NCc2cccc(C(C)C)n2)nc[nH]c1=NCC1(C2CCC2)CCC1 C1(O)(COC)CCN(C(CC2C(C)(C)C2(C)C)C(=O)NCCOCC2CC2)C1 C1(CNC(c2cn(CCC)nc2)c2nnnn2C(C)C)CCC2(CC2)C1 C=CC1OCCCC1C(=O)N(C)CCNC(=O)Cc1ccnnc1O C(=O)(C1=CNS(=O)(=O)N=C1C)NCC1(F)CC(CNC(CC=CC)=O)C1 c1(OC)c(C(=O)Nc2ccc(CNC(C)C(=O)O)cn2)cccc1C c1(C(=O)NCC2C(C)CN(C(=O)C(C)CF)C2)cc(S(=O)(=O)N(C)C)c[nH]1 C(=O)(C(C)(C(F)F)c1ccccc1)N1CCC(N(C)C(c2csc(=N)[nH]2)=O)CC1 C12CN(CCC1(F)F)C2=O.C12(NC(C3C(C(=O)OC)C=C3)=O)CC(SC)(C1)C2 CC(C)C(O)C(F)(F)C(=O)NC1CCC(N(C(=O)C(F)C(C)C(F)(F)F)C)CC1 C1(C2CCN(C(C3CC4CCCC4C3)=O)CC2)(NC(CSCC(N)=O)=O)CC1 c1(C(N2CC3CN(Cc4cnn(C5CC5)c4)C3C2)=O)cc(Br)cc([N+](=O)[O-])c1F C1(C(=O)NC(CN(C(=O)CNCCNC(N)=O)CC)C)CC1C1(C)COC1 C1(NC(C(C=C=C)C)=O)CCN(C(=O)Cn2ncc3ncccc23)CC12CCC2 C1(C)(COC)CC(NC(c2ncc(C(F)F)s2)=O)CN1C(c1nnn(C)n1)=O CC1CCCC(O)(C(=O)NCC23CC(CO2)N(C(c2c[nH]ccc2=O)=O)C3)CC1 c1(C(=O)NCC2(CNC(=O)CC3CCC(=O)O3)CCOC2)ccc(C(F)F)nc1 C(CCCCC(=O)OCc1ccccc1)NC(=NC)NCc1cc(O)nc(O)n1 c1(C(C)CC(=O)NC2CCC2CNC(c2nccn2C)=O)ccc(F)cc1F CCC(C=O)CC.C(=O)(CC(=O)OC(C)(C)C)N(CC(C)NC(=O)COC)CC C1(C(N2CCC(C)C2CNC(C2CCCN2C=O)=O)=O)CCc2nnc(O)n2C1 c1(OC)ccc(F)c(N)c1C(=O)NC12CC1CN(C(=O)C#CC1CCOC1)C2 Clc1cc(Br)c(CNC(c2nnnn2CC2CC2)C2CC23CCC3)s1 c1(C(=O)NCC)ccc(NC(c2scnc2Cl)C)cc1Cl c1(COCC(=O)NCC(C(=O)NC2(C(=O)OC)CSC2)O)ccnc(O)c1 C1C(C)C(=O)N1CC.C(=O)(CCCc1nccs1)NCC(=O)OCC c1(C(N2C(CNC(CCCC(C)=O)=O)COCC2)=O)cn(C)c(=O)nc1O N1(C(c2cnn(C)c2)C)CCc2c(C(N)=O)cccc2C1 N1(C(C2CC(C#C)(O)C2)=O)CCC2(CC1)CC(C)N(C(c1coc(CC)n1)=O)C2 c1(N2CCC(OCC)(CF)C2)ncnc2scc(Br)c12.C12CC1C(=O)N2 Cc1cc(CNC(=O)C(=O)NCCCC2CCCN2C(N)=O)c(C)o1 c1(C(C)CC(=O)NCC(CO)NC(C2SCCS2)=O)c[nH]c2ccccc12 c1(CN2CCC(NC(c3ccc(O)cn3)=O)CC2)cc(F)c(O)c(Br)c1 C(C1=CCN(C(C2(CC(F)(F)F)CC2)=O)CC1)NC(=O)Cc1ccccn1 N1(c2nnc(-c3nn(C)c4c3CCC4)n2CCC#N)CC2CCCC(C1)C(=O)N2 C1(C)(C(=O)NC2CCC(NC(C3C(C)(O)CCC3)=O)CC2)CCCCNC1=O c1(C(C)C)c(C(=O)NCC2C=CCN2C(=O)CN2CC=CC2)cnc2ncnn12 O=S(=O)(c1ccc(N2CCC(CO)C2)cc1Br)NCCN1CCCCC1 c1(C(=O)NCCN(C(=O)CC2CCC(C)(C)O2)CC)c(N)sc(C)c1C n1(CC)cc(C(N2CC(NC(c3occc3C)=O)CC2C)=O)c(C(C)C)n1 N1(C(CC(C)CNC(=O)CCOCC(F)F)=O)CC2(CCC1CO)CC2 Cc1cc(=O)ccn1CC(=O)NC1CCC(N(C)C(c2cc(C(F)F)no2)=O)C1 c1(NC(C(=O)NC(C)CC2CCC2)=O)ccc2cn(C(C)C3CC3)nc2c1 N1(C(c2c(C)ocn2)=O)CC(CC(=O)NC2CCCC2(F)F)CC1(C)C CCC1c2ccc(OC)c(OC)c2CCN1C(=O)C1=CCSC1N c1(C(N2CC3C(NC(CP(C)(C)=O)=O)(CCC3)C2)=O)ccc2c(c1)CCC2=O Cc1cc(C(=O)NCCC2CC(NC(=O)COCCN(C)C)C2)ccc1Cl CCCCC(C)(F)C(=O)NC(CNC(=O)C(C)Sc1ccc(F)cc1)C(C)C N1(C(C(COC)(C)OC)=O)CC2(CC(NC(c3cc(Cl)ccc3N)=O)C2)C1 N1(CC)C(=O)CCC1C(=O)NC1(CO)CN(C(c2ccn(CCOC)n2)=O)C1 Cc1cc(F)ccc1S(=O)(=O)N1C2CCC1CN(C(c1cccc(CO)c1)=O)C2 C=C(Cl)CC(C(=O)NCC(C)(O)CCCC)NC(=O)Cc1cnns1 c1(OC)cc([N+](=O)[O-])ccc1C(N1CC(NC(C2CC3C=CC2O3)=O)C(C)C1)=O C1(CNC(c2c(CC(C)C)onc2)=O)CCC2(CCC2)C1NC(C1CCOC1)=O c1(C(N(C(C(=O)NC2CCC(C)CC2)C)C2CC2)=O)c[nH]c2cccnc12 c1(C(=O)NCCC2CN(C(C3CCCC3)=O)C2)nccc(F)c1Cl C1(NC(CSC(C)C)=O)CCOC(C(=O)NCC2CC2c2ccno2)C1 c1(C2C(C)(NC(N(CC(C)O)CCF)=O)C2)ccc(F)cc1F C(=O)(CCCC(=O)NCCOCCCN(C)C(C1CC2CCC1CC2)=O)N(C)C C12(C(N(c3nc(C)no3)C(CN3CC(F)(CC)C3)=O)=O)CC(CO1)N(CC)C2 C1(C(N2CCC3(CCCO3)C2C)C(=O)NCCCC)CC2OC(C)(C)OC2C1 C(=O)(C1SCCc2sccc21)N(C)CC1CCCN(C(C2(C(F)F)CC2)=O)C1 C=CC1CN(C(C2CC3C=CC2CC3)=O)CC1NC(=O)COCCCCC c1(CC(=O)NCC(C2CCN(C(=O)Cn3cccc3)CC2)C)ccc(F)nc1 C(=O)(C(CCNC)N(CCC(N)=O)C)NCCOC C1(C)(NC(c2cnc(CC)o2)=O)CCCN(C(=O)CCc2cnco2)C1 C(=O)(C(C(F)(F)F)C(F)(F)F)NC1CCCC(NC(=O)Cc2cccnc2)C1 c1(OC)ccc(S(=O)(=O)N2CCN(Cc3csc(C)n3)CC2)c2cccnc12 C1(C(N(C(C)CNC(=O)CCC(N)=O)C)=O)CCC(=O)C(C)C1 N1(C(c2cn(CC(N)=O)nn2)=O)CC(C2CN(C(=O)CC3(O)CCC3)C2)C1 N1(C(C(CC=C)C(C)C)=O)CCOC2CN(C(=O)CCOCC3CCC3)CC12 c1(NC(C2CN(C(c3c(NC)nsn3)=O)CC(F)C2)=O)c(O)cccc1C#N N1(C(C=CC(C)NC(=O)CCC(N2CCC2)C)=O)CCC(CCO)CC1 C(C(C)(C)CC(=O)N(C1CC1)Cc1ncccn1)OC.C12(CCC1)C(=O)N2 c1(CC(=O)NC2(CF)CCN(Cc3nc(C)oc3)C2)c[nH]c2c(C)cccc12 C1(C(=O)NCC(c2nccs2)C)CC2CCCC2N1C(=O)C1=COCCC1 CCC(F)(F)CCn1nc(-c2cc(SC(C)C)ccn2)nc1C1CCC(=C2CC2)CC1 c1(CCCC(N2C(C)CC(NC(=O)CC=CCN(C)C)C2)=O)ccc(Cl)c(Cl)c1 C1(C(=O)NC(CC)(C)CC)CCC2(CC2)N1C(=O)Cc1cccc(O)c1 c1(CC(C(=O)NCCC)C2CCCCC2)ccnc2ccc(OC)cc12 c1(SC)cc(C(=O)NC(C)(CNC(=O)C(C)OCCC(C)C)C2CCC2)ccc1F Cc1nc(O)ccc1C(N1CCC(F)(CNC(c2cn(C)c(=O)n2C)=O)C1)=O C1(NC(CN2CCC(C)C2)=O)CN(C(C2(C(F)(F)F)CC(O)C2)=O)CC1CO c1(C(=O)NC(C2CCN(C(C(CC)=CC)=O)C2)C)nccc2ccncc12 C1(C(N2CCC23CN(C(c2c[nH]c(Br)c2)=O)C3)=O)(OC)CC2(CCC2)C1 C12(COC)CC(CNC(=O)CCOC)(CN1C(=O)CCN1C(=O)CCC1=O)C2 C1(CC(=O)N(C2CCN(C(=O)C(C)NC=O)C2)CCC)CCCOCC1 CC1CN2CCN1C(C(=O)NC1CCC(CNC(=O)C(C)(C)CO)C1)C2 C12(CNC(c3c(C)sc(Cl)n3)=O)CCCCC1CN(C(=O)C(F)(F)C(C)O)C2 C12(C(=O)NCCN(C(c3cn(C4CCOC4)nn3)=O)CC)CCC(CC1)C2(C)C c1(C(N2CC3CN(C(c4cnc(N(C)C)o4)=O)CC32)=O)c(F)cc(Br)cc1Cl N1(C(CN2CCC(OC)C2)=O)C2CCC(C2)C1C(=O)NC(c1ncn(C)n1)C c1(NC(N(C2CC3CNC2C3)CC(F)(F)F)=O)ccc(C#N)cc1.CS CCC(CC)CCCNC(=O)C(Cn1cncn1)OC N1(C(C(C)O)=O)CCC(CO)(CNC(=O)C(C)C2CCC2)CC1 c1(N(C)C)ncc2c(n1)CCC(CNC(=O)NC1CC(N3CCCC3)C1)C2 C(CCC1CC1)(C(=O)N(C)Cc1cccc(C)c1)NC(C=CC(CC)C)=O Cc1nnc2n1CCCC2C(=O)NCC1CCN1C(=O)C=Cc1ccc(C#N)cc1 CC(C)(C)C(C(=O)NCC(C1CCC1)NCC1(O)CCSCC1)NC(S(C)(=O)=O)=O C1(C(=O)NC2CCCN(C(CC3C(CC)C3)=O)C2)CCCCCN1C C1(S(C)(=O)=O)(C(N(OC)CC2C(Cc3ccccc3F)C2(F)F)=O)CCC1 Cc1[nH]nc2cc(C(=O)NCC(C3CC3)NC(C3CC3(C)C)=O)ccc12 c1(OC)cccc([N+](=O)[O-])c1C(N1CCC(NC(=O)C(C)(F)C(C)(C)F)C1)=O c1(C(=O)NC(CCCCNC(c2cc(CC)nn2C)=O)C)ccn2c1CSCC2 C(C1CCCCC1)=CC(=O)N(C1C2CN(C(C3CCOC(=O)C3)=O)CC12)C N1(C(c2c(=N)[nH]cnc2)=O)CC2(C1)C(NC(c1ccsc1)=O)CCS2(=O)=O N12CCN1C(CC(F)(F)F)C2.N1(CC(=O)N)CCCCCC1.C(CC(F)(F)F)CC N1(C(c2c(CC)ocn2)=O)CCC(N=[N+]=[N-])(C(=O)NC(C)C2=CCCC2)C1 N1(C(C)=O)CCC(OCCNC(C2(CS(C)(=O)=O)CC2)=O)CC1.C1SCCCS1 c1(CN2CC(C(F)(F)F)CC(C)C2)ccc2ncccc2c1 N1(C(=O)OCC)CCC(c2ncc(C(=O)NC(C)CO)s2)CC1 C(C(C)(O)CCCC)NC(C=CC(C)(C)NC(=O)CS(=O)(=O)NC)=O CCCC(C)(C)C(=O)N(CC(=O)N(C)Cc1cn(C)nn1)C C(c1ccccc1Br)=CC(N1CCN(CCNC(C(C)(C)OC)=O)CC1)=O N1(C(C2CC23CCOC3)=O)CC23CCCC2(C1)CN(C)C3.Cc1nsc(N)c1Br C(CC(C)C)(C(=O)NC1CC(CNC(C2CNC(=O)O2)=O)C1)NC(C)=O C1(C(=O)NC2CC(CCNC(=O)Cc3ccns3)C2)CC2CCC1O2 c1(NC(=O)CC2CCCO2)cc(Cl)c(O)c(Cl)c1 CCCCCCCCC(=O)NC1CCCCN(C(=O)CCCCC(C)CC)C1 Cc1ccc(=O)n(CC(=O)NCC2CCC(NC(=O)CCCC(N)=O)C2)c1 c1(OC)c(C(N2CCCC(O)(CNC(=O)Cc3cncnc3)C2)=O)ccc(F)c1F C(=O)(C1=COCCC1)N1C(CCNC(=O)C=C2CCC2)CSCC1 c1(CC)ncc(Cl)c(C(N2CC3CCC3(NC(=O)C(C)C(C)C)C2)=O)n1 C1(NC(CCN(C(c2nc(N(C)C)oc2)=O)CCO)=O)CC(C(N)=O)C2CC12 N1(C(C2C(CC)CCCC2)=O)CCC(C)CC1CNC(c1nc(O)c(C)s1)=O c1(OC)ccc2c(=NC(C)N3CC=CCC3)[nH]c(-c3ccccn3)nc2c1 Cc1nccc(CC(=O)NC2(CCNC(C3CCO3)=O)CCC2)n1 C(=O)(C(C)(C)CCNC(=O)CC1CCSC1)NC(c1c(C)nccn1)C Cc1cc(NC(=O)Cn2cc(-c3ncnn3C)nn2)ccc1Cl.C12CC(C1)OC2 C1(C(C)C)CN(C(=O)CC2CC3CCC2N3C(c2ccc(CO)s2)=O)CC(=O)N1 C(=O)(C(C)(C)CC(F)F)NC1C(CC)CN(C(c2cnoc2C2CC2)=O)C1 C#Cc1ccc(C(N2CCC2CNC(c2ccc(=O)n(C)n2)=O)=O)cc1C c1(C(=O)NC2C(F)CCN(C(CC3(COC)CC3)=O)C2)cnc2c(n1)CCCC2 N1(C(C(CC)C)=O)CC(C)N(C(=O)CNC(=O)NC)CC1C c1(NC(C(=O)NC(C)Cc2ccnn2C)=O)cccc2c1OCC2 O=C(CC(C(F)F)NC(C12CC(F)(C1)C2)=O)Nn1ccnn1 c1(C(N2C(C(=O)NCC(c3cccs3)C)CC2)=O)cn(C)cn1 C1(CNC(=NCCCC)NCCc2ccc(C)c(C)c2)CC2CCCCN2C1 c1(-n2cc(C3CN(C(=O)C(F)OC(F)(F)F)C3)nn2)ccc(F)cc1Br.O=C C1(NC(CCSC)=O)CCOCC1C(=O)NC(=O)Cc1cnsc1 N12CCCCC1CNC(=O)C2=O.c1(C(=O)OCC)cnc(C2CCOC2)s1 C1(C(=O)NCCN(C(c2c(C)c[nH]n2)=O)CC2CC2)CCCN(CC(F)(F)F)C1 C1(CC)(NC(=O)C(C)CC(N)=O)CCCN(C(=O)C=C(C)CN2CCOCC2)C1 c1(CC)cnc(OC)c(N2CCC(C3OCCO3)C2)c1 C(=O)(CCCCC(F)F)N1C(C)CN(C(c2cc(C(C)(F)F)ccn2)=O)CC1 C1(CC)(CC)CC(NC(C2CC(C)(C)CN2C)=O)CN1C(=O)Cc1cn(C)nn1 N1(C(c2scnc2Cl)=O)CC2=C(C1)CN(C(c1cnc(C(F)F)cn1)=O)C2 C(CC(=O)N1CC(C#N)(CCF)C1)(C(F)(F)F)NC(C1(C)N(C)CCC1)=O N1(C(CC(CC)(C)C)=O)CC2CC1CCC2NC(c1ccc(OC)c(N)c1)=O C(=O)(CCCCCCCS(C)(=O)=O)NCCC(=C)CNC(C1CC1(C)OCC)=O c1(C(=O)NC(c2ccc(C)cc2)CNC(CCC#C)=O)cc(C)ncc1Br c1(C(=O)NCC2(F)CC(NC(CN3CCC(C)(O)C3)=O)C2)ccc2c(c1)NCC2 C(=O)(C(CNC(=O)CCC1CC1(C)C)CC1CC1)N(C(CSC)C)C C12CCN(CC1)C(=O)C2C1CCC(C)O1.Cc1cnn(CCN2CCCCC2)c1 N1(C(=O)NCC2CCC2)CCOC2CN(C3CC(c4ccc(F)cc4F)C3)CC12 c1(-n2ncc(C(=O)NC3CC(N(C(CCN(C)CC)=O)C)C3)c2)ccccc1F C1(NC(=O)CN2C(=O)CCC2=O)CCC2(CC1)CN(C(c1cnsc1)=O)CCO2 N1(C(C(C)=C(C)C)=O)C2CC1CN(C(c1ccccc1Cl)=O)C2 n1(CCCCO)nc(CCOc2ccccc2)nc1-c1ccc(F)cc1 C1(C(=O)NCCc2c(C(=O)N)c[nH]n2)C(C)(C)C1(F)F.C(C(CO)C)OC(C)=O N1(C(C(C2CC2)SC)=O)CCC(C(=O)NCc2cc(C)cc(F)c2)CC1(C)C C1(CC(=O)NCCCOCCN(C(C2(CC)CCC2)=O)C)CCn2cncc2C1 Cn1c(C(=O)NC(CO)CCCNC(c2cc(O)cs2)=O)cc2sccc12 N1(CC2(C)CC2c2ccc(F)cc2)CC(c2ccc(Br)cc2)CCC1=O C1(C(=O)Nc2cccc(CF)c2)Cc2ccccc2C(=O)O1 CCCC(C(=O)N1CCCCC1CNC(C1(CC(C)C)CCCC1)=O)NC(C)=O c1(N(c2c(OCC)cccn2)C(C2C3COCC23)=O)c(C#N)cnc2ccnn12 CN1CC(O)CC1C(=O)NC1CCC(C)(CNC(=O)Cc2cncnc2)C1 c1(C(N2CC3(CN(C(c4ccc(C(C)=O)cn4)=O)C3)C2)=O)cc(C)ccc1[N+](=O)[O-] C1(NC(=O)NC(C2CC3C=CC2C3)C)C2CC3CC1CC(O)(C3)C2 Fc1cc(F)c2[nH]c(=NCc3cc(Cl)cc(Cl)c3)oc2c1 C(=O)(CCCC(C)(C)C)N1C(CC(=O)NCC2(OCC)CCC2)CCCC1 CC1=C(C(=O)N2CCC(C)(CC(=O)NCCC(C)C(C)C)C2)COCC1 C(=O)(C1=CCCSC1)OC(C(c1cccc(C)c1)N(C(C)=O)CCC1CCCC1)=O n1(CCCNC(C2(C)N(C(c3scc(C)c3C)=O)CC2)=O)cnc2ccccc12 CC(C(=O)NCCC1(C(=O)NCCC2CC=CC2)CCCC1)S(C)(=O)=O c1(OC)ccc(=NCC2CC(NC(c3cc(C#N)on3)=O)C2)[nH]c1OC C1(CC)(NC(=O)CC2(C)CC2)CCCN(C(C2CCC2c2ccc(F)cc2)=O)C1 C(=O)(CCC(F)(F)C(F)F)N1CCC(C(=O)NCCNC(=O)Cn2cccc2)CC1 c1(NC(=O)C(=O)NCC2(C)ON=C(C)C2)ccc(SCC(F)F)cc1C c1(OCC)ccc(C(=O)NC(C2CN(C(=O)C(C(C)C)NC=O)C2)C)cc1 C(C(C)NC(C1(C(=O)CN(C(CC(C)C)=O)C(C)C2CC2)CC1)=O)OCC C1(NC(c2ccc(C)nc2)=O)CCN(C(=O)Cn2c(C)csc2=O)CC1F N1(C(C(C)NC(C(C)C)=O)=O)CC2CS(=O)(=O)CC2(NC(=O)C=C2CCC2)C1 C=CCCCC(C)(C)C(=O)NC(CC1CC1)CC(N1CCCC2(C1)N=N2)=O CCCCC(O)C(C)C(=O)N1CCCC(C(C)C(=O)N(CC(C)(C)CN(C)C)C)C1 CON1CCC(CC(=O)N(CCNC(C2COCCN2C)=O)C2CC2)CC1 CC(C)CCC(F)C(=O)NC1(C(N2CC(c3nc(=O)o[nH]3)C2)=O)CCOCC1 C#CCCCCCCC(=O)N1CCC(C)(NC(c2ccc([N+](=O)[O-])c(Br)c2)=O)C1 C(C)(C(=O)NC1CCC1CNC(=O)CCC1CCCC1)(C1CC1)NC(C)=O c1(C(N2C(CNC(C(C)CF)=O)C(C)CCC2)=O)ccc2ncccc2n1 C1(NC(C2CCN(C3CC3)CC2)=O)COC2(C1)CN(C(c1n[nH]cc1Br)=O)C2 C(=O)(CC(C)C1CC1)NCC(C)N(C)C(c1csc(-c2ccsc2)n1)=O c1(C(=O)NC2CC3N(C(C(CC)(C)O)=O)C(CC3)C2)ccc2c(C)[nH]nc2c1 CC1(NC(C2CN3CCC2CC3)=O)CCN(C(c2ncncc2Cl)=O)CC1 c1(COC)cc(C(=O)Nc2nc(-c3ccc(Cl)s3)cs2)n[nH]1 CCC(C)(O)C(=O)NCCCC(C)NC(=O)CNc1cccnc1 N1(C(C2CCN(C(C(CC)CCOC)=O)C2C)=O)CCOC2C(O)CC12 Cc1cc[nH]c1C(N1CCC(CC2CCCCC2)C1)C(=O)NCSc1ccccc1 C1(O)(CN(C(=O)C(F)C2CCC2)C)CCCN(C(c2cccnc2S)=O)C1 N1(C(c2c(N)c3c(cn2)CCC3)=O)CCN2CCN(C(c3cnsc3)=O)CC2C1 c1(C(N(C(CNC(COCCCC)=O)C)CCSC)=O)cnn(CC(C)C)c1C CC1=C(C)CC(C(=O)N(C2CN(C(c3cnn(C(C)C)c3C)=O)CC2O)C)CC1 C1(CNC2CC(OCC(=O)OC)C2)CCN(C(C2CC=CCO2)=O)C1 C#CCC(C)(C(=O)NCCC(C)C(C)C)NC(c1cc(C#N)oc1C)=O Cc1ccc(C(=O)NC(c2ccc(F)cc2)CNC(C23CC(F)C2C3)=O)cn1 N1(C(CCC(=O)NCCC)C(=O)OC)CCC2=C(CCC(=O)N2)C1 Cc1cccc2cc(C(=O)NC3C4CC3N(C(c3ccc(=O)n(C)c3)=O)C4)[nH]c12 N1(C(CCOC(C)C)=O)CC(NC(C2CCNC2=O)=O)C(C(F)(F)F)C1 C1(CCNC(C(COC)O)=O)CCCCN1C(c1csc(C(N)=O)n1)=O C1(NC(CN(C)C)=O)CN(C(c2cnn3cccc(Cl)c23)=O)C2(CCOCC2)C1 Cc1c(C(=O)NC(C2CN(C(C3(N=[N+]=[N-])CC3)=O)C2)C)cc(C2CCCC2)n1C C1(C(=O)NC(C2CCN(C(c3ccc(=N)[nH]n3)=O)CC2)C)CCCOCC1 C(C(N)=O)(C(N)=O)NC(c1c(CNC(CC)=O)ocn1)=O C(c1ccncn1)=CC.c12n[nH]cc1C13CC(C1)(C3)C(=O)NC21CC1 N1(C(c2c(CC)csc2)=O)CCCC(C)C1CNC(=O)Cn1cc(Br)c(=N)[nH]1 C1(N(C(COCCC=C)=O)CC)CN(C(=O)Cc2cnnn2C)C2(CCOC2)C1 C#CC1CCCCN(C(=O)NC2CCOC2c2cnn(CCOC)c2)C1 CCCCS(=O)(=O)CC(=O)NC1CCCN(C(=O)CC2CC2(C)C)C1 C12(CNC(c3nc(C(C)C)sc3)=O)CC1CN(C(C1(C)CC(C#N)C1)=O)C2 c1(OCC)ccc(C(=O)NC2CC(C(=O)OC)C3C2C3)cc1O c1(NC(C)=O)cccc(NC(C2C3CN(CCOCc4cc(O)n[nH]4)CC23)=O)c1 c1(C(N2CC(C(C)NC(C3CC(C(F)(F)F)C3)=O)OCC2)=O)ccc(F)cc1Cl c1(OC)nccc(C(=O)NCCCCNC(=O)CC2CCCC(C)C2)n1 N1(CCCCCC)CCCN(C(C2CCN2C)=O)CC1.C(C(=O)N)=CC=CCC c1(C(=O)NCCCN(C(=O)Cc2cnccn2)C)cnc(P(C)(C)=O)cn1 C1(C(N(C(C)C(=O)NCC2(C3(O)CCC3)CC2)C2CC2)=O)CC2(CCCCC2)C1 C(C(C)(C)CS(C)(=O)=O)N(C(C(C)CN(C)C)=O)C1CC1 C1(C(=O)NC(C2(CNC(=O)CCC(C)(C)C)CC2)C)C(O)C(=O)N(C)C1C C1(C2CC2)(C(N(CCCCCO)C)=O)CN(C(C2CC2(F)Cl)=O)C1 CC(CN(C)C)C(=O)NCC(O)CNC(c1ncoc1-c1cccs1)=O N1(C(CNC(c2ncc(NC)nc2)=O)=O)CC(C)CC(C)C1 C1(NC(c2occc2Cl)=O)COC2(C1)CN(C(=O)CCc1cccc(F)c1)C2 N1(C(C2ON=C(C)C2)=O)CCCC(NC(C2CCC(O)C2)=O)C1C C1(CCNC(CC(=O)NCC#C)=O)CC(F)(F)CN1C(=O)CCOCC(C)(C)C N1(C(C(C2CC2)OCC)=O)CCN(C(c2ccc(Cl)c(Cl)c2)=O)CC1C(F)F C(C(O)CC(=O)NCC1CN(C(c2ccnc(C(C)(C)C)n2)=O)CC1O)N(C)C C1(NC(COC(C)=O)=O)CCCCCC1C(=O)NC(C)(C)CCF C(=O)(C(C(C)C)n1cnnc1)NCC(=O)NC1CC(C#C)C1 N1(C(CSCCC)=O)CC2CN(C(=O)C3=NOC4(CCC4)C3)CCC2(CO)C1 C1(c2cn(C(C)C)nn2)CN(C(=O)COc2ccc(F)cc2F)CCN1C C#CC(CC(C)(C)C)NC(C12CC1CCN2C(=O)C(O)C(C)(C)C)=O C1(C(N(CCCCN(C(CC(C)C2CC2)=O)C)C)=O)CCCC(=O)CC1 S(=O)(=O)(c1ccc(N2CCC(OCCN(C)C)C2)c(F)c1)Nc1c(C)cncn1 Cc1cccc(C(=O)NC2C3CC2N(C(C2CCCCN2C2CCCC2)=O)C3)c1 CCCCCC(O)C(=O)NC1CCN(C(C2(C(N3CCCC3)=O)CC2)=O)C1 c1(C(N2CCCC(N(C(C(CC)N(C)C)=O)C)C2)=O)nc(Cl)ccc1OC(C)C N1(C(CN(CCC)C(C)C)=O)CCc2ccsc2C1C c12cc(F)ccc1N2.n1(CCOC)ccc(C(=O)N)n1.c12cnc(s1)[nH]c2=O.OC CC1CCCC(C)N1C(C1CSCCN1C(=O)CCCOC(C)(C)C)=O C=C(C)CC(C(=O)Nc1cnn(C)c1CC)NC(=O)C=C(CCC)CCC C1(n2cc(C3CCN(C(=O)CC45CCCC4C5)C3)nn2)CCC(F)(F)CC1 C1(NC(CNS(NC)(=O)=O)=O)CCC(C)(NC(C2CC3CCC(C2)O3)=O)CC1 CCN=c1[nH]cc(C(N2CC(O)CC2CNC(c2ccsc2NC)=O)=O)s1 c1(C(=O)NCCN(C(=O)CSC(F)(F)F)CC)ccc(Sc2n[nH]c(C)n2)cc1 C(CC(C)(C)C(=O)N1CCC(CN(C(=O)CCCCO)C)C1)OC c1(NC(=O)NC2C(C)CN(C)CC2)nc2c(cc1C#N)CCC2 N1(C(Cn2c(C)cc(=O)cc2)=O)CCC2(CC(NC(c3cnco3)=O)CO2)C1 C1(CC=C)(NC(=O)C(F)=C(C)C2CC2)CCCN(C(=O)C(C)COC)C1 N1(C(Cc2nc(C)on2)=O)CCCC2(CCCN2C(c2csc(C)c2N)=O)C1 CCC(C)CCCC(=O)N1CSCC1C(=O)NCCCOCCCO c1(C(N2CC3CCCC3(C(c3ccon3)=O)C2)=O)ccc2cccc(C(=O)O)c2n1 N12CCC(C1)C(C)CSC1CC(C1)C(=O)NCC2=O.C#CCOCCOCC=C c1(CC)ccccc1OCCC(=O)NC12CC1CN(C(N1CCOCC1=O)=O)C2 c1(C(=O)NC(C2CC2C(N2CC(F)CC(F)C2)=O)C)cnccc1C#N C(=O)(N(CCC(=O)OC)OC)C1C(C(=C)C)OCC1.C12(CCC1)CCN2 C1(NC(c2c(CC)nn[nH]2)=O)CC2CCC1CN2C(c1ccc(Cl)s1)=O N1(C(C(c2ccccc2)OC(C)=O)=O)CCCCC(NC(=O)C2=NOCC2)C1 C#Cc1cc(C(N2CCOC(C(C)NC(=O)C=CCC)C2)=O)cc(N)c1 c1(CC(=O)N(CC(=O)NC(C)(C)C)C(C)C)cccc2ccccc12.C1CN1 C(=O)(C1=CCCOC1)N(C(C(=O)NCC=CCCC)CC)C c1(CCCC(N2CCN(CC(=O)N(CCSC)CC)CC2)=O)c(F)cccc1F C1(C(=O)NCCCCCCNC(=O)C(F)c2ccco2)CC2CCC(C1)C2 C(=O)(CCCCCCNC(c1cccc(C)c1C#N)=O)NCC(CC)(CC)CO CC(O)(CC(=O)NCCC1CN(C(c2cc(CCCO)on2)=O)CCO1)C1CC1 C(=O)(C(CNC(=O)C(O)Cn1cncn1)N(C)C)NC(c1cc(Br)no1)C N1(C(CC(CC)(F)F)=O)CCC2(CC2)CC1C(=O)NCCn1nc(C)nc1C CC1CCCC(C)N(C(c2ccc(CNC(=O)CSCC(N)=O)cn2)=O)C1 c1(C(=O)NCCC(C)NC(Cc2ccc(C)c(O)c2)=O)cc2ccc(O)nc2s1 C1(C(=O)NC(CCC)(C)C)(CNC(=O)CC2CC3CCC2C3)CCCCC1 N1(C(CCOC(C)C)=O)CC(Nc2cnccc2CN(C)C)C2(CC2)C1 C1(CC)(NC(c2cc(C)[nH]n2)=O)CCN(C(=O)CCC(=O)c2ccncc2)CC1 c1(N2CCN(CCC)C(=O)C(=O)N2)cc2c(cn1)C(=O)CCC2.CC.CC C1(NC(c2c(C)ncs2)=O)CCN(C(C2CC2(C)C)=O)C12CCC2 c1(C(=O)NCC(CC=C)NC(=O)CC(C)n2ccnc2)c(Br)cnn1C c1(C(=O)NCCC2CC(NC(C3(c4ccsc4)CC3)=O)C2)cccn2nccc12 C(C(C)CC(=O)N(CCCNC(=O)Cc1n[nH]cc1Br)CCO)OC C1(CNC(C(C=C)O)=O)CCCCN(C(c2c[nH]c(=NC)o2)=O)CC1 C(=O)(C(C#N)C(C)(C)C)NC(C)C(CO)NC(c1ccc(SC(F)(F)F)cc1)=O C1(N(C)CCO)CCCN(C(=O)NC(c2ccccn2)C(=O)NCCN)C1 N1(C(COCCCC)=O)CCN(C(=O)C(=Cc2ccco2)C)CC1CCOC N1(C(CC(CC)C2CCC2)=O)CCN(C(c2ccncc2)=O)CC1c1ncc[nH]1 C1(C(=O)NCCC(CNC(c2c[nH]nc2C2CC2)=O)O)CC2(CCCC2)CO1 C1(CC=C)(NC(C2CCCN(C)C2)=O)CCCN(C(=O)CC2CCC(C)C2)C1 c1(C(=O)NC2(C)CN(C(C(C(C)C)n3cnnn3)=O)C2)cn2c(n1)CCC2 C1(C(C(=O)NCC2(C(=O)OC)CC2)C)CCCCN1C(C)=O.C1CC1NC=O Cc1ccc(CC(C)C(=O)NC2CCN(C(c3ccc(OC(F)F)s3)=O)C2)cc1 N1(C(CC2N(CC)CC2)=O)CC2CCCC(N(C)C(=O)C3CC3)C2C1.C1(=O)CN1 C1(C(N)=O)CCN(C(C2CC2CNC(=O)CCCF)=O)C1 c12c[nH]c3c(cccc13)[nH]2.c1(C(=O)NCCN(CCOC)C)ccnc(Cl)c1 CCS(=O)(=O)C=CC(=O)N1CCCC1C1CCN(C(c2ccc(CC)c(O)c2)=O)C1 CCCC(C)CS(=O)(=O)N(CC(C1CCCCC1)O)C c1(C(=O)NC2CCN(Cc3cc(OC)nc(C)n3)CC2O)cc(F)c(Cl)cc1I C12(NC(CCCc3c(C)ccs3)=O)CCOC(CNC(c3cnco3)=O)(C1)C2 C=Cn1nncc1S(=O)(=O)Oc1ncc(F)c(C)n1 C(=O)(CCC(CC)c1ccccc1)NC(CC)CNC(c1nc(C)[nH]c1OC)=O C(c1cnc(OC)nc1)=CC(=O)NC(CCN(C(CC(CC)C1CCC1)=O)C)C c1(CNC(C2CCN2C(C2(F)CC2(Cl)Cl)=O)=O)cccc(-c2ccoc2)c1 C(=O)(CC(=O)NC(CNC(c1sccc1C(F)F)=O)C1CC1)OC C(=O)(C(O)CCc1ccccc1)NC1CC(n2cc(CC(C)(F)F)nn2)C1 c1(C(=O)NCC2CCCN(C(=O)C(F)C3CC3)C2)nccc(Cl)c1O CC1CN(C(=O)CC2CCC2)CCN(C(=O)CC2CC(=O)NC2=O)C1 c1(C(=O)OC)cc(OCC(=O)Nc2nc(CC(F)(F)F)cs2)ccc1F C(N=c1cc[nH]c(C#N)n1)C1CCCN(C(CC(C)OC)=O)C1 C(=O)(N1CC(n2cc(C3(CCO)CC3)nn2)CO1)c1cc(COC)no1 N1(C(C(CCC)F)=O)CCC2CCN(C(c3nc(Cl)cs3)=O)CC12 c1(CNC(C2CC(O)(CNC(C(C)NC(CC)=O)=O)C2)=O)cncc(F)c1 C(N=c1[nH]c(N2CCOC(c3ccco3)C2)nc2c1COC2)C1C(C)(C)NC(=O)O1 c1(CC(C)C(=O)NCC2CCCC2NC(=O)CN2CCCCC2)ccccc1F c1(C(=O)OC(C)(C)C)sccc1NS(C)(=O)=O.C12(CC=CC1)NC(=O)NC2 N1(C(C(C(C)C)Sc2ccccc2)=O)CCCC(O)(C(N)=O)C1 CCC(CO)(C(=O)NCCC1CCN(C(c2ccn(CO)c2C)=O)C(C)C1)OC N1(C(c2cc(C)n(C)c2)=O)CCN(C(c2ccc3nccn3n2)=O)C2(CCC2)C1 C1(NC(Cc2c(C)cc(C)s2)=O)CCN(C(C2CCC(C)(C)CO2)=O)C12CCC2 CC(C)CCCCCC(=O)NCC(C(=O)NCC1(O)CC(C)(C)C1)N(C)C CC1(C)CC(C)(CNC(c2cnc(Cl)[nH]2)=O)CN1C(c1ccnnc1O)=O N1(C(c2c[nH]c(=NC)s2)=O)CCC(C)(C)CC1C(=O)NC(C1CCCC1)CO C(CC(O)(CC)CC)SC(C=CC(N1CCN(CC(=O)NCCC)CC1)=O)(C)C c1(C(=O)NCCCC(C)NC(C2C(C)C2C)=O)ccc(O)cc1Cl C(=O)(CS(=O)(=O)C1CC1)N1C(CC(=O)NC)CN(C(=O)C(OC)OC)CC1 C1(C(N(CC(C(=O)NCc2nnc(C)s2)C)C)=O)CC2COCC2C1 CC(C)(CCCNC(=O)CNc1ccccn1)C(=O)NCC1(O)CCOC1 C(=O)(C1CNC(=O)c2ccccc21)NC(CCCC)CNC(c1nccn1C)=O Cc1cccc(SCC(=O)NC(C)(C)CNC(c2cnn(C3CC3(F)F)c2)=O)c1 N1(CC(=O)NCC2CC(CNC(c3c[nH]c(=N)s3)=O)OC2)CCCCC(O)C1=O c1(CNC(=O)NCc2c(OC)cc(Br)cc2)cnn2c1CN(C)CC2 c1(SC)cc(C(N2CC=CC2CNC(=O)C(c2cncnc2)C)=O)c(Cl)cc1Cl N1(C(CC(C)C2CC2)=O)CCC(NC(C2(C)CC(C)(C)C2)=O)C1C(C)(C)C c1(SCC)ccccc1C(N1CCOC(CCNC(C2(F)CC2)=O)C1)=O C(=O)(C1=NN2CC(C)CN=C2N1)NC1CCC(CNC(c2c(C)cco2)=O)CC1 c1(C(N2CCCC(c3onc(C)n3)C2)C(=O)NCC2CC2)cc(Cl)cc(Cl)n1 C1(NC(C=C(CC)C)=O)CC2CC(C1)N(C(=O)Cc1c(F)cc(OC)cc1Cl)C2 C(C#CCCO)NC(=O)CCNC(=O)CCc1cscn1 N1(C(C2CCCC2O)=O)CCN(C(=O)CC2CC2(Cl)Cl)C(c2ncc[nH]2)C1 C(=O)(CCCS(N)(=O)=O)N1CC(NC(C=CC=CC)=O)C(c2ccccc2F)C1 C(=O)(C(C#N)C(C)(C)C)NC(C(=O)NCC(C)Cn1cccn1)n1cccn1 N1(C(C2(C(C)C)CNC(=O)C2)=O)CC2(CCN(Cc3cscn3)CC2)C1 C1(SC)CN(C(c2csc(C(C)(C)C)n2)=O)CC1NC(=O)C(C(C)C)OC N1(C(C(CC)OCC)=O)CCC(C2CC2)C1C(N1CCC12CC(O)(CO)C2)=O C(CC(C(C)(C)C)NC(=O)CN1CCSCC1)N(C(C(c1ccc(Cl)s1)C)=O)C c1(-c2nn(CC3CCCC(CC)CC3)c(C3CC3)n2)ccc2ncccc2c1 C1(CNC(Cc2c(C)con2)=O)CCC2CN(C(c3ccc(N)c(F)c3)=O)CC12 O=C1NCC2CN(C(=O)NCCc3ccc(Br)c(F)c3)CCC2N1 c1(C(=O)NCCC2N(C(CCC)=O)CCCC2)cc(F)cc2cc[nH]c12 CC1(NC(c2ccsc2-c2ccncc2)=O)CCN(C(C2CC23CCC3)=O)C1 CCC(C)(C)C(=O)NCCCCCN(C(=O)CC(C)(C)c1ccccc1)C N1(C(C(CCSC)OC)=O)CC(CNC(=O)COCC(C)C)CC12CCC2 c1(C(C)=O)cnc(N2CCCC2C(N2CCC(C3CCCNC3)CC2)=O)c(C)c1 CCCCC(CC)CC(=O)N(C1CCN(C(c2nn(C)c(N)c2C)=O)CC1)CC Cn1cc(NC(=O)CCC(N)=O)cc1C(N1CCC(CSc2ccc(F)cc2)C1)=O CCC(CC)C(F)C(=O)N1CCC(F)(C(=O)N(CC(F)F)C2CCC2)C1 c1(C(=O)NC2CCC(C)N(C(=O)CCC3CCCC3)C2)ccc(P(C)(C)=O)s1 C1(N2CC(CCC)C2)CCC2(CC1)CCN(C(=O)NC1CC1(F)F)CC2 Cc1cnc(C(=O)NC2CC(F)CN(C(C3CCOC3C(F)(F)F)=O)C2)c(F)c1 C12(NC(c3c(Cl)sc(Cl)c3Cl)=O)CCCC1(F)CNC2 C(=O)(C(N)CCC(=O)C(C)C)NC(c1c(OCC)cccc1)CC(C)C CN1N=C(CC(=O)N2CCC3(CCCN3c3nccn4nnnc34)C2)CC1=O c1(C(=O)NC(CC(=O)O)c2cccs2)cnc2[nH]nnc2c1 C1(CNC(Cc2cn(C)nc2)=O)CCCC(Cn2cc(C3COCC3O)nn2)C1 N1(C(CC(C)C2CCCCC2)=O)CC2(NC(c3cc(Br)c[nH]3)=O)CC1C2 c1(C(=O)NC(CN(C(C(C)OCC=C)=O)C)C)c(Cl)csc1Cl N1(C(C(C=CC)O)=O)CC2CCCC(C1)N2C(=O)C(C1CC(F)(F)C1)O C1(C(=O)NC2C(CNC(c3ccn4ccsc34)=O)CC2)CC2(C1)CC(O)C2 CCC(CC(=O)N(CCCNC(c1ccnc(OC)n1)=O)CCCO)C1CCC1 c1(CC(=O)NCCN(C2CCCC2)C(C2CC23CCC3)=O)cn2ccsc2n1 c1(C(N2C(C(N3CC(SC)C3)=O)C(O)CC2)=O)ccc(Cl)c(C#N)c1 CC1C(N(C)C)CCN1C(=O)CCCCN(C)C(C1CCC(=O)NC1)=O C(=O)(C1=C(CC)CCCC1)NC(CCC)CCCNC(c1ccc(N)c(F)c1)=O CCC(C)CC(=O)NCC(c1ccccc1)C1CCC1 C1(CNC(CSc2ncc(C)o2)=O)CC(F)CN1C(c1ccc(Cl)s1)=O C(C1=CCN(C(C2CCN2CC)=O)CC1)NC(C1CC(SC)C1)=O C12(C(N(CCNC(c3cnc4[nH]ccc4c3)=O)CC)=O)C3C4C1C1C2C3C41C#N C1(CNC(=O)CCOC2CC2)CC2CN(C(c3cccnc3O)=O)CC12 c1(C(C)=O)cc(NC2CCN(C(C3CC(=O)N(O)C3)=O)CC2)ccc1[N+](=O)[O-] N1(C(C(c2cccc(C)c2)CN)=O)CC(C)NCC1C C1(OC)CC2(C1)CN(C(C1CCCN(S(=O)(=O)CC3CC3)CC1)=O)C2 N1(C(CSC)=O)CCCC1(C)C(N1CCC(CC2(O)CCC2)CC1)=O C=CCCCCCCC(=O)N(C(C)CNC(C1CCCN(C(=O)OC)C1)=O)CC N1(C(C(=O)NC(C2CC2c2cccc(F)c2)C)=O)CC(F)(F)CC1c1ccccc1 CCCC(O)CC(=O)N1CCC(C(C)NC(=O)C(N2C(C)CCC2C)C)C1 N1(C(c2c(CC)n(CCO)nc2)=O)CCOC2(CCN(c3ncc(I)cn3)C2)C1 C(C1CCCC1)=C(C)C(N1CCC(C(F)C(=O)N(CCC(C)(C)O)C)C1)=O C1(NC(c2cnc(C)s2)=O)CCCC2CN(C(=O)CCc3cc(C)sc3C)CC12 N1(CC(=O)NCCCN(C(C)C)Cc2c(C)nc[nH]2)CCOCC1=O c1(C(N(C2CC(C(N3CCC3(C)CCO)=O)C2)C)=O)nncn1C c1(SC)nccc(=NC(=O)c2cncc(CNC(C3(C#N)CCC3)=O)c2)[nH]1 S(=O)(=O)(c1cc(C#N)ccc1F)N1CCC(C)(C(N2CCC(C)CC2)=O)C1 c1(-c2ccc(NC(c3ccc(C)c(F)c3)=O)cn2)csc2ccncc12 c1(C(N2CCCN(C(=O)C=CC3CCCO3)C(CO)C2)=O)c(Cl)ccc2c1OCO2 C1(C(N(CCCC=C)C)=O)CCN(C(=O)CCCC2CC2C)C1 CCC(C(=O)NCCN(C)C(C1CC1C(=O)OC)=O)SC C1(NC(CCCC)=O)C2CC1N(C(c1cc(C(C)C)sn1)=O)C2 C1(O)(CNC(Cc2c(C)n(C)cn2)=O)CCN(C(=O)C(C)(C)C(C)C2CC2)CC1 c1(C(=O)NC2CCC(CNC(C=CS(C)=O)=O)C2)ccc2c(c1)CCCC(=O)N2 C1(NC(CCCc2nnc(C)n2C)=O)CCOC2(CCOC2)C1 N1(C(CC(=C=C)C)=O)CC(C(N2CC(OC(=N)O)C2)=O)C2(CC2)C1 Cc1cc(C(=O)NCCn2cc(CNC(c3cnsn3)=O)nn2)ccc1O CC1SCCCC1C(=O)NC1COCCC1C(=O)NCC1(CCN=[N+]=[N-])CC1 C12(NC(c3c(C)onc3-c3cccs3)=O)CCOCC1CN(C(=O)CC(C)C)C2 c1(CN(CC(C(=O)OC)CN)C)nc2cc(O)ccc2o1 C(=O)(C1=NNC(=O)CC1)NCC1OCCN(C(C(C(C)C)N2CCCCC2)=O)C1 C1(C(=O)NC(c2ccco2)C)(CN(C(C(CC)C)=O)C)CC12CCC2 CCCC(O)(CCC)CC(=O)N(CC(CC)NC(=O)CC1CCC(=O)NC1)C O=C(N1CC(O)CCO1)C1CC2CCC(C1)N2C(C1CC(O)C1)=O C1(NC(=O)CN2CCCNS2(=O)=O)CCCC12CN(C(c1ccnnc1O)=O)C2 N1(C(c2ncc(CC)nc2)=O)CC2CCN(C(=O)C(C)CCOC)C2C1 c1(N(CCCCC=C)C)nc2cccnc2c(=NCC(C)C(Cl)(Cl)Cl)[nH]1 CC(CC(=O)NCC(CO)NC(=O)C=Cc1cnn(C(C)(C)C)c1)C(F)F c1(OC)nn(C)cc1C(=O)NC(C)C(C)C(=O)N1CC(OC)C(C(N)=O)C1 N1(C(C2CCC(=C)CC2)=O)CC(C)(C(=O)NC2CC(=O)N(OC)C2)CC1(C)C C(=O)(C#CC1CCCCO1)NC(C)CNC(c1ccc(N)c(O)c1)=O C1(CNC(c2c(SC)cccc2)=O)CC12CCN(C(=O)Cn1nnc(C)n1)CC2 CN1C(=O)NCC12CN(C(=O)C(O)CNC(=O)C=CC1CC1)C2 Cc1ccc(F)c(NC(C2(CNC(c3cnn(CCF)c3)=O)CCCC2)=O)c1 C(=O)(C(CC1CCC1)N1CC(CCc2cnccn2)C1)NC(C)C N1(C(c2n[nH]c(C)c2Cl)=O)CC2CCC(NC(C3CCN3C(C)(C)C)=O)CC2C1 c1(C(=O)NCC2N(C(CCCC=C)=O)CC(O)C2)cc2ccccc2oc1=O C1(CNC(c2c(CC)ncs2)=O)N(C(=O)CC2CCOC2(C)C)CCCC1(C)C C1(CC(=O)N(C2CCCN(C(c3ccn(C(F)(F)F)n3)=O)C2)C)CCCN(C)C1 C1(CC=C)(C(=O)N(CCC(=O)NC)CC2CC2)CCN(C(=O)C(O)CN(C)C)C1 C1(CNC(c2c(CC)[nH]c(=N)s2)=O)CN(C(c2cc(COC)cs2)=O)CC12CC2 C(C(C)(C)CC(=O)N1CCCC1CN(C(c1cncc(OC)c1)=O)C1CC1)OC Cc1cc(Br)ncc1CNC(=O)C(=O)NC1CCCC1(F)F [N-]=[N+]=NCCCCCCCS(=O)(=O)NC(C1CN(c2nncs2)C1)=O C(CCSC)(C(=O)N1CC(F)CC1CO)NC(C(CC)=CCCC)=O N1(C(c2ccc(Cl)cn2)=O)CCC2CCN(c3nc4cc(Br)ccc4o3)CC2C1 C#CCC(O)C(=O)NCCN(C(C1(NC(=O)OC(C)(C)C)CCOC1)=O)C1CC1 c1(OC)cccc(S(=O)(=O)N2CCC(C(C)Nc3ncc(F)cn3)CC2)c1 c1(C(C)(C)C)nsc(N)c1C(=O)NCC1CCC(NC(=O)C2=CCC2)CC1 N1(C(c2c(CC)occ2)=O)CCCC1C=CC(=O)N(C1(C)CC1)C c1(C(N2CC(CN(C(c3c(C)nc[nH]3)=O)C)C2)=O)c(C)nc(=N)[nH]c1C c1(C(=O)NC(C(C)NC(=O)Cn2ccc(C(F)F)n2)C)c(F)ccc(C#N)c1F C1(C)(C(=O)NC2(C)CC(C(=O)NCCCCOC(C)C)C2)CC=CCC1 N1(C(C(C)NC(COC)=O)=O)CC2CCC1C(C(=O)Nc1cccc3c1COC3)C2 C1(CNC(c2ccc(COC)o2)=O)(CO)CCCN1C(=O)C(F)C1CCOC1 c1(C(N2C(CNC(C(C)CC3CCCC3)=O)CC2)=O)ncsc1S(N)(=O)=O C1(C(C)NC(c2n(CC)cnn2)=O)CN(C(=O)Cc2ccnc(F)c2)CCO1 c1(C(N2CC(C)(NC(c3c(OC)c(=O)cco3)=O)C2)=O)ccc([N+](=O)[O-])cc1O N1(C(=O)COCCCF)CCN(C(c2cncs2)=O)C(c2cc(F)cc(F)c2)C1 c1(C(=O)NCC(CO)NC(c2c(SC)n(C)nc2)=O)nc(C)n2ccccc12 C1(CNC(C2C(C)(C)C2)=O)CC12CCN(C(=O)CNC(=O)C1CC1)CC2 C(C(c1nnnn1-c1nnc(C)n1C)Nc1ccccc1)(C(C)C)OC C12(C(=O)NC(CNC(C(CCCC)F)=O)(C)C3CC3)C(=O)C3CCC1C2C3 C(=O)(CC(O)C(N)=O)N.c1(OC)ccccc1CN(C(c1ccc(S)o1)=O)C1CC1 CC1(C)CN(C(=O)C2=CCOCC2)CC1NC(=O)CCC(=O)c1ccc(F)cc1 CCCCC(O)CC(=O)N(CC(CO)(CO)NC(C1OCCC1(C)C)=O)C C=C1C(NC(c2nn(C)c(Cl)c2COC)=O)CC2CC1C2(C)C C1(CNC(CNC(CN(C)C)=O)=O)CCCCN1C(c1csnc1Cl)=O N1(C(CCc2n(C)cnn2)=O)CCC2CN(C(c3ccsc3Br)=O)C2C1 N1(C(C(c2cccc(Cl)c2F)(C)C)=O)C2CCC1C(CNC(C1(F)CC1)=O)C2 C12CCCC(C1)C(=O)N2.c1(C(=O)NC(c2nc(=O)o[nH]2)C)ccc(CO)o1.C(N)=O C(=O)(C(C)C(C)(F)F)NC1(CF)CCN(C(c2cnc(C(C)C)s2)=O)C1 CC1=C(C)CC(C(=O)NC2(CNC(C3CC(C)(C)O3)=O)CCCCC2)CC1 c1(NC(CCCN(C2CCC2)C)=O)ccc(F)cc1Cl N1(C(CC2CC(C)C2)=O)CCC2(CCOC2)C(CNC(C2CNC(=O)CC2C)=O)C1 C(=O)(C1=CCCN(C(=O)CCOCC(F)F)C1)NC(CC(=O)OC)C1CC1 C1(C(N2CCCC(OCC=C)C2)=O)CN(C(=O)C=CCF)CCC1(C)C c1(C(N(C(C)CNC(C2CC(O)C2)=O)C)=O)csc2ccc(F)cc12 C1(OCC)(CNC(=O)C(C)OC2CCCC2)CN(C(=O)Cn2cc(CC)cn2)C1 CC1CCC(F)(F)CN1C(C1(CCNC(=O)CCP(C)(C)=O)CCC1)=O C(=O)(CCc1cnoc1)N(C(C)C(=O)NCC(C)(C1CC1)OC)CC C1(NC(C=CCCC)=O)COC2(C1)CN(C(=O)CCC(=O)OC)C2 C1(OC)CCN(CCC23CN(C2)CC(=O)N3)CC1.C(C)(C(=O)NCCCC)=CC C1(CNC(C2CCCO2)=O)CCN(C(c2cc(-c3ccccn3)n[nH]2)=O)C1 C1(CCN(C)C)(NC(=O)COCCNC(=O)CCc2cn[nH]c2)CCC1 S(=O)(=O)(c1c[nH]ccc1=NCCn1ccnn1)N(CCC(C)O)C C(CCCCCNC(=O)C(C1CCCOC1)OC)NC(c1cnc(OC)s1)=O c1(C(N2CC(CNC(C(C(C)(C)C)SC)=O)OCC2)=O)cc([N+](=O)[O-])cnc1O c1(CC(=O)NC2(CN(C(CC=C)=O)C)CC2)ccc(Br)cc1OC c1(N2CCN(C(CC3CCC(=O)NC3)=O)CC23CC3)ncnc2c(Br)csc12 c1(CC)nn(C)cc1C(N1CCC(CO)(NC(=O)CC2CC(OC)C2)C1)=O N1(C(c2c(OC)nc(C)cc2)=O)CC2CCC1CC2NC(C1COCC(C)O1)=O CC1CC(NC(=O)CSCC(c2ccccc2)=O)CN1C(C1CC2(CC2)C1)=O c1(CC)oc(C(=O)N(CCCNC(C2CC(CC3CC3)C2)=O)CC)cc1C N=c1nc(C(=O)N(CC(=O)Nc2ccc(-c3cnc[nH]3)cc2)C2CC2)cc[nH]1 S(=O)(=O)(c1ccc(N2CCC(c3ccc(C)s3)C2)c(Cl)c1)N(CC(CC)C)C C1(N(C)C)(C(=O)NCCCOCCO)CCCC1.C1(CC(=O)NCCS)C=CCC1 C1(C(N2CC=CC2C(=O)N(CC(O)COC)C)=O)(CC)CCNC1=O n1(CC)cnc2nc(=NCCSC)[nH]c(NCCC(C3CCCCC3)O)c12 CCCCC(=O)NC(C)(C)CN(C(=O)Cc1cnn(C(C)C)c1)C N1(Cc2ncc(C)s2)CCC(O)C(C(=O)Nc2ccc(CO)s2)C1 Cc1ccc2[nH]c(C)c(CNC(=O)NCCC(F)(F)C(F)F)c2c1 c1(CCC(NNC(=O)OC(=O)CC2CCC2)=O)ccnc2ccccc12 N1(C(CCc2n(C)ncc2)=O)CC2(C)CN(C(=O)CC3(O)CCC3)CC2(C)C1 C1(CNC(c2c(CC)onc2)=O)CN(C(=O)CC2CCS(=O)(=O)C2)CCC1(F)F C(=O)(CCC(F)(F)C(F)F)N1CC(CNC(c2ccc(C)c(C)c2O)=O)C(O)C1 c1(NC(CC2CCN(C)C2=O)=O)cccc(C#N)c1.C123CC(C1)N(C2)C3=O CCC(CC)C(C)C(=O)N(CCCN(C)C)CCNC(=O)CC1CCS(=O)(=O)C1 N1(C(CCCN(C(c2n(C(C)C)ncc2)=O)C)=O)CCCC12CCOCC2 C12(NC(c3cc(C)cc(C)c3)=O)CCC(CNC(c3ccoc3Cl)=O)(CC1)OC2 N1(C(=O)C=NOC2CCCCO2)CCC(Nc2cc(F)c(O)c(F)c2)C2(CC2)C1 c1(OC)ccc(COC(C2CCN(C)C2)=O)cc1C c1(C(=O)Nc2c(Cl)c(C)n(C)n2)n[nH]c2c1CN(C(=O)C=CC(C)C)CC2 N1(C(c2c[nH]c(=N)s2)=O)CC2OCC(NC(c3ccc(O)nc3)=O)C2C1 C1(CNC(CCC#N)=O)(CNC(=O)CCc2cnco2)CCCCC1 C1(CC(=O)NCC(C2CN(C(C3(C(N)=O)CC3)=O)C2)F)(N(C)C)CCC1 O=C1COCC2(CN(C(=O)N(C3CC3)Cc3cccc(N4CC=CC4)c3)C2)N1 Cc1cncc(=NNC(=O)NCC2CCN(C)C3(CC3)C2)[nH]1 c1(C(=O)OC)cc(C(=O)NC23CCC(NC(=O)CCCC(N)=O)(CC2)C3)cc(Cl)c1 Cc1c[nH]c(C(=O)N(C(C)(C(=O)NCC(O)CNC(N)=O)C2CC2)C)c1 N1(C(C#CCNC(C2(C=C)CCCC2)=O)=O)CC2CCC1C(O)C2O CC1CN(C(=O)CN(CCCN(C)C)C)CC(N(CC(F)(F)F)C(=O)O)O1.CCO c1(C(=O)NC2CC(N(C(C3CC(C)=C(C)CC3)=O)C)C2)c(F)ccc(Cl)c1F C(N=c1[nH]cnc2c1COC2)C1N(C(C2C(C)CC(=O)NC2)=O)CCC1 C=CC(C)(C)CC(=O)NC1(C)CCN(C(C2CCC(=O)NC2)=O)C1 C(=O)(CCc1csnn1)NC1(CN(C(=O)C(F)OC(F)(F)F)C)CC1 c1(C2C(C(=O)OC)=CCCC2)cc(C)[nH]c(=NCC(COC)C(F)(F)F)n1 c1(NC(C(C(C)C)OCC)=O)c(F)ccc(Cl)c1Cl.c12nccnc1[nH]c(=O)[nH]2 C#CCC(CC(=O)NCCC1CC(OC)C1)NC(c1cc(F)cnc1O)=O C1(NC(COC2C(CC)CCCC2)=O)CC(C)CN(C(c2[nH]cc(C)c2C)=O)C1 c1(C(=O)O)cnn2cccnc12.c12ccc(cc1)C(=O)NC(CC=C)CO2 c1(C(C(=O)NCC2CCCCC2CC(F)(F)F)O)ccc(F)cc1F C1(CNC(CN(CCC)C)=O)CN(C(c2sc(CCC)nc2C)=O)CCC1C Cc1nnc(O)c(C(=O)NC2CC(CNC(=O)CCC3(C)N=N3)C2)c1C c1(C(=O)NCCC2CCCN(C(c3coc(Br)c3)=O)C2)cc2cnccc2[nH]1 O=C(N=c1ccc(-c2ccccc2)n[nH]1)c1csc(N2CCCC2)n1 C=CC(C)(O)CC(=O)NC(C)(C)CC=CC(=O)Nc1cnn(CCF)c1 N1(C(C(C)C(C)(F)F)=O)CC(C)(C)CCC1CNC(c1ccc(C(F)(F)F)[nH]1)=O c1(OC)ccccc1C(=O)NCC(C)(O)CNC(c1snnc1C1CCC1)=O N1(C(=O)C(O)C2CCC2)CCC(C2CCCN(C(c3ccc(O)cc3O)=O)C2)C1 C1(NC(C2CCC3CC23)=O)CCC(F)(CNC(C2(n3cccn3)CCCC2)=O)C1 C1(C(C)(C)C)C(=O)N1.c1(CC)nc(N(C)C)sc1Cc1ccccc1 Cc1nn(CC(N2CC(CNC(=O)Cc3cnc(C4CC4)[nH]3)C2)=O)cc1Br N1(C(C(CSCC)NC(=O)CC2CCC(C)CC2)=O)CC(O)C(C)(C)C1 Cc1cccnc1CCC(N1CCOC(CN(C(=O)C=Cc2cc[nH]n2)C)C1)=O c1(OCCCOC)ccc(C(N2CCC(NC(C3(C)CS(=O)(=O)C3)=O)C2)=O)cc1 C1(CN(C(C(C=C)O)=O)CC)CCN(C(C2C=C(C)CS2)=O)CC1 CCC(C)C1c2nnnn2CCN1.c1(C(N2CC(SCC)C2)=O)ccc(Cl)o1 C1(C(=O)NC(C)CC(N)=O)CCC2CCC1N2C(c1cc2ccccn2n1)=O N1(C(C(CC)C2CCC2)=O)CCC(C(F)F)(CNC(=O)C=CC(C)C)C1 N1(C(C2C(C)(C)OC(=O)C2)=O)CCN(C(C2(CC3CCC3)CC2)=O)CC(C)(F)C1 Cc1cc(C(N2CC3CC3(CNC(c3nnsc3C)=O)C2)=O)nc(C)n1 Cc1nc(Br)oc1C(=O)NCC1CN(C(=O)C(c2ccccc2)C)CC1C Cc1cc(NC(=O)C(=O)Nc2ccccc2-c2ccco2)cc(F)c1 O=C(C1=Cc2ccccc2C1O)NCC1(NC(C23CC2CCC3(F)F)=O)CCC1 N1(C(CC(CC)OC)=O)CC(C2CCCCN(C(c3cc(C)no3)=O)C2)C1 Cc1nc(CCNC(C)(CCCO)c2nnnn2CC2CC2)sc1CC1CCOC1 Cc1c[nH]c2ncc(C(N3CC(NC(C4CC4(C)CCN(C)C)=O)C3)=O)cc12 N1(C(COCC(C)C)=O)CCC(NC(c2ccn3ncccc23)=O)C(F)(F)CC1 N1(C(C2(CC)CC2)=O)CCC2CCN(C(=O)C(C(C)(C)C)c3ccccc3)CC12 N1(C(c2c(C)cncc2C)=O)C2CCC1CN(C(C1(C)CC1Br)=O)C2 C(=O)(N=c1ccn(C2CCCC(=O)N2)[nH]1)NCCOC.C1(=O)C=CC(C)N1 C(=O)(C(CNC(=O)CC(=O)OCC)C(C)C)NCC(F)=CC c1(C(=O)NC2CC(NC(C3(CC)CCOC3)=O)C2)cc(C(C)C)cc(F)c1 N12CC3CN(C3C1)C(=O)NCC2=O.c1(CCC(=O)OC)cc(C(F)(F)F)no1 c1(NC(C(=O)NCC2CC(F)(F)C2O)=O)cnc(S)n1-c1ccccc1 C1(C(=O)OCC)(C(C)C)CCN(C(=O)C2=CCCO2)C1 Cc1cc(Br)cc(C(N2CC(CNC(=O)C(C)(C)C)C3CC23)=O)c1N C(=O)(CCC(C)(C)C#N)NCC1C(NC(c2c(C)cnnc2O)=O)CC1 C1(OC)CN(C(C2CC(=O)CC(=O)N2)=O)CCC1NC(=O)COC1CC1 CCC(C)C(C(=O)N1CCOC(CC)CC1)N(C)C.N12CCC(OC)(C1)C2=O C1(C(=O)NC(CC(C)NC(C2(COC)CC2)=O)C)CCC2(CC1)CC(O)C2 N1(C(c2cn(C)c(=O)cc2)=O)CCC(C2(NC(=O)Cc3cncnc3)CC2)C1 C1(C)(C=O)CN(N2C(COC)CC(O)C2)CCO1.C1(C(C=O)C)CCCCC1 c1(C(C)NC(c2c(COC)noc2)c2nnnn2C2CCCCC2)ccc(Cl)cc1 c1(C(N(CC(=O)NCC(C)COCC)CCC)=O)ccc(C)o1 c1(OC)ccc(C(=O)C(=O)NC2CCCC2NC(C23CC(C)C2C3)=O)cc1 c1(SC)cc(C)c(C(N2CCC(NC(=O)C(C(C)C)NC(C)=O)C2C)=O)s1 c1(C(=O)NC(Cn2cc(C3(C(=O)OCC)CCCO3)nn2)C)cccc(C#N)c1 C(CCC(c1nnnn1CC1CC1)NCCn1nnc(C)n1)OCC=C c1(OC)c(F)cc(C(N2CC(O)CC2C(=O)Nc2nnco2)=O)cc1F C(CC(C)NC(=O)COC)NC(C)=O.C(CC(C)C)OCCOCC(=C)C CN1CCOCC1CC(=O)NC1(CNC(=O)CCCC#N)CC1 C1(NC(c2cc(C)n(C(C)C)c2)=O)COC2(C1)CN(C(C13COC(CO)(C1)C3)=O)C2 c1(CC)cc(OC)ccc1C(=O)N(CCCNC(c1csc(C(C)C)n1)=O)C N1(C(c2c(OCCC)cccc2)=O)CCC(C)(NC(=O)CC(C)C2CC2)CC1 Cc1nc(-c2nc[nH]n2)sc1C(=O)N(C)CCNC(C1CC(C)CO1)=O CCCC(O)C(=O)N(C1CN(C(c2ccc(S)cc2)=O)CC1O)C CC1CC(CNC(=O)CN2CCCNC2=O)CN1C(=O)CCCNC(N)=O c1(C(N2CC(CC(N3CC([N+](=O)[O-])C3)=O)OCC2)=O)cccc(F)c1F C1(C(=O)NCc2c(C(N(C)Cc3c(CC)noc3)=O)scc2)CCCC(=O)C1 N1CCCN(CCCCNC(=O)CC2(O)CC2)CC1.C1(CC=O)CCCCC1 C(=O)(C(C#N)C(C)C)N1CC2C(CN(C(C=C(CCC)C)=O)C)C2C1 C1(C)(CNC(C(C)OCCOCC)=O)CN(C(=O)CCN=[N+]=[N-])CCO1 N1(C(c2ccc(NC)nc2)=O)CCC2CCCC12C(=O)NCCN(C)OC N1(C(C(CC(F)F)N(C(=O)Cn2ncccc2=O)C)=O)CC(C#N)C2(CCC2)C1 c1(C(N2C(C(C)(C)NC(C(C)CO)=O)CCC2)=O)ccn2ccnc2n1 C1(NC(=O)C2=CCSC2)CC(F)(F)CC1NC(c1csc(Br)n1)=O N1(C(c2c(C)ncn2C)=O)CCCC2CN(C(C3OCCO3)=O)CC12 c1(NC(=O)CC2CCCCO2)cnc(CNC(=O)C(O)C2CCC2)nc1 N1(C(CC(=O)NCC)=O)CC(CN(C(=O)C(CCOC)OC)CC)CC2(CC2)C1 N1(C(CSc2n(C)nnn2)=O)CCCC(N(C(C23CC4CC2C3C4)=O)C2CC2)CC1 Cc1cnn(C)c1CC(N1CCN(C(=O)CC2(C)CC(F)(F)C2)CC1)=O C(=O)(C(C)(CO)NC(=O)C(C)O)NCc1cc(C(C)C)n[nH]1.C1CC1 C(=O)(C1CCCc2ccccc21)NCC1(CNC(C(CC)CC(F)F)=O)CCC1 c1(N(C)Cc2nc(=N)[nH][nH]2)nc2cc[nH]c2c(=NCCCOC2CCCC2)[nH]1 C#CC1(NC(C2CN(C(C3(C(C)C)CC3)=O)CC2C)=O)CC2CCCC12 N1(C(C(=O)NCC)=O)CCCC12CCC(NC(C1CCCC1)=O)CC2 C1(NC(C2CCC(CNC(C(C(C)C)SC)=O)CC2)=O)CCCCC1C#N C1(CNC(CP(C)(C)=O)=O)CN(C(=O)C=Cc2ccccc2)CC1(F)F CCC(C)C(O)C(C)C(=O)NC1CCC(CCC(N2CC3CC2CN3C)=O)C1 N=c1nc(C(=O)NC(Cc2ccccc2)C(=O)O)cc[nH]1 c1(C(=O)NC(C(C)C)C(C)NC(C2(C)C(C)(C)C2(C)C)=O)cccc2occc12 C1(C)(C(N(C(CC)CNCC)C)=O)CC1(F)F c1(OCC(C)C)ccc(C(=O)NC(CNC(C2CCOC(=O)N2)=O)C(C)C)cc1 c1(CC(N2CC(C)OC(CCNC(c3c[nH]nc3F)=O)C2)=O)cccc2ccoc12 N1(C(Cc2nc(C)sc2C)=O)CCC2CN(C(=O)CC3CCCOC3)CCC12 CC(C)C(C(=O)N1CCOC(CCNC(C2C=CCC2)=O)C1)C(C)C c1(CC(N2CCC(C(=O)NCCC3CC(C)C3)C2)=O)ccccc1C#N C12(CNC(C3C(=O)NCC3)=O)CCCC1CN(C(=O)Cc1c(F)cccc1F)C2 CN1CC2CCC1C(CNC(=O)CCOC1CN(C(=O)C(C)(C)N=[N+]=[N-])C1)C2 N1(C(C2CCC(=O)NC2)=O)CCC2(CCC2CNC(c2csc(Cl)c2)=O)CC1 Cc1nc(C(N2CCCC2C2(C(=O)NC3CCCSCC3)CC2)=O)c(C)o1 c1(C(N2CC(C(N)=O)C2)=O)ccc2c(n1)CN(C(C1CCNC1)=O)CC2 c1(C(N(CC(C)(C)CN)CC)=O)ccc(C(C)C)c(C)c1 C(C(N=[N+]=[N-])C(=O)N1CC2CC1(C(=O)NCC(c1nccs1)C)C2)OCC N12CC(O)CC1Cc1cn(nn1)CCSCC2=O.Cn1ccnc1-c1ccccc1 N1(C(C(C(=O)OCC)(C)C)=O)CC2(NC(C3CCCS(=O)(=O)C3)=O)CCC1CC2 c1(CNC(C2(F)CCN(C(Cc3c(C)cc(C)s3)=O)C2)=O)cccc(C#N)n1 n1(CCNC(=O)C=CC2CC2)ccc(C(=O)NCCc2cccnc2)c1 c1(C(N2CCN(C(C(C(C)C)OC)=O)CC2C)=O)n[nH]c2cc(C(=O)OC)ccc12 c1(C(N2CCC(F)(CNC(c3c(C)ocn3)=O)C2)=O)ncnc(O)c1Br c1(C(N2CCC(NC(C(CC=C)(C)C)=O)C2C2CC2)=O)cnc2cc(C)[nH]c2c1 c1(C(N2CCC(NC(CCSC)=O)CC2C2CC2)=O)cc2cn[nH]c2cn1 Cc1ncc(Br)cc1C(=O)NCC(O)CNC(=O)CC1CC1 c1(C(N2CCC(NC(c3c(C)onc3C3CC3)=O)C2)=O)c[nH]cc(Br)c1=N C1(C(=O)NCC2CC(CNC(CCC(C)OCC)=O)C2)CC2CC(=O)C1O2 C1(C(=O)NCC(CC)OC)CCCCCCN1C(=O)CC1(OCC)CCC1 c1(C(=O)NCC2C(NC(CC(CN(C)C)O)=O)CCC2)cc(F)cc(Cl)c1N N1(C(CCC(=O)NC)C)CCOCC(c2cn(-c3ccc(C)cc3)nn2)C1 Cc1cc(C(N2CC(CNC(C3CCc4cnnn4C3)=O)C2)=O)c(N)cc1F c1(CN=C(NC(C)C)NC2CCN(CS(C)(=O)=O)C2)cccc2c1COC2 c1(C(=O)NCC(C)(C2CC2)NC(C(CN(C)C)N(C)C)=O)cccc(CC#N)c1 C1(NC(c2n(CCCC)ncc2)=O)CCN(C(C2CCCCN2C)=O)CC1O CCCC(C)C(C)NC(=O)C(C)(C)CN(C)C(c1ccsc1Cl)=O c1(C(=O)OC)cncc(NC(c2ccccc2Oc2cnccc2SC)=O)n1 n1(CSCC)nnnc1C(c1cncn1CCC1CC1)NC1(C)CCCC1 C1(CNC(C2C(C)(C)CO2)=O)CC(F)CN1C(=O)CSC1CCS(=O)(=O)C1 C#Cc1ccc(C(=O)NC2(C(=O)NCC3CN(C4CC4)C3)CC2C)nc1 C12CCN(CC1)C(=O)CC2F.C1(CNC(C(F)=CCC)=O)(OC)CCSC1 N1(C(C(CC)C#N)=O)CCC2(C)C(C1)C2(F)F N1(C(c2c(C)cc(Br)cn2)=O)CCC2(C1)CN(C(=O)C(C)(C)CF)C2 N1(C(CC2N(C)CC=CC2)=O)CCC2CN(C(=O)CCc3cc[nH]n3)CC2C1 c1(SCC(N2CCC(CCNC(CCc3n(C)ccn3)=O)C2)=O)ccc(F)cc1 C1(CNC(C(CCC)NC(C)=O)=O)CN(C(=O)CSC(F)F)CCCO1 N1(C(C2CC2)=O)C2CCC1CC(C(N1CCCC(F)(F)CC1)=O)C2.CC1CC2(CC2)C1 c1(C(N2C(CO)CC(NC(C=CS(C)=O)=O)C2)=O)nccc2cc[nH]c12 C(C(=O)OC(C)(C)CC)(C(C)(C)C)N(C)C(=O)NCC1(c2ccsc2)CC1 C1(C#N)(C(=O)NC2C(C)CN(C(=O)C=C(Cl)Cl)C2)CC12CCCC2 c1(OC)cc(C2CCCN(C(=O)Nc3cccc(F)c3)C2)cc(F)c1 C(=O)(C(=O)N=c1ccn(CC2CCCO2)[nH]1)N1CCC(CN(C)C(N)=O)C1 C=CC1CCN1C(=O)CC(C)N(C(=O)CSCC(N)=O)C CC(C1OCCc2ccccc21)NC(=NCCF)NCCn1cnc2c1CCCC2 Cc1cccc(C(=O)NC2CC(N(C)Cc3ccc(OCF)nc3)C2)n1 c1(Nc2cccc(N3CC(NC(C)=O)C3)c2)nc(OC(C)C)c2ccccc2n1 C12(C(N3CC(CCNC(C4CCC(C)(C)O4)=O)C3)=O)CCCN(CC1)C2 N1(C(c2n(C)nc(SCC)c2Cl)=O)CCC12CCN(C(=O)C(C)CBr)CC2 CCC(C(=O)N(C(C)CCO)C)N(C)C(C1CCO1)=O N1(C(Cc2ccc(C)c(C)c2)=O)CC(NC(C2(C)CC2(F)F)=O)CC12CCC2 C=CCC(C(=O)N1CC(C(=O)NCC2(CC)CC2(F)F)C1)NC(C)=O N(C(=NCCC(C)=O)NCC1(OC)CCOC1)CCC1(COC)CCC1 C12(NC(C3C(C)CCCC3)=O)CCCC1N(C(=O)Cc1cccc(F)c1)CC2 Cc1cc(C(=O)NC(C)CCNC(c2cnns2)=O)c2c(c1)CCO2 c1(NC(C(=O)NCC(C)(C)NC(c2cc(SC)oc2C)=O)=O)cccc(Br)c1O N1(C(c2cc(OC)nn2C)=O)CCCCC(CNC(c2cnc(=N)[nH]c2)=O)C1 CC1OC2(C(N3CC(C)(NC(C4CCCN4Cc4ccsc4)=O)C3)=O)CCC1C2 n1(CCC(=O)NC(CC)CNC(c2c(C)cnn2C)=O)cc(C#N)c(O)nc1=O C1(NC(c2cnn(CC)c2C2CC2)=O)CN(C(=O)C(C)(C)C#N)CC12CC2 Cc1csc(C=CC(=O)NC2CC(NC(c3ccc(Br)cc3)=O)C2)n1 c1(CC(=O)N(CC(C)NC(C(C)SC)=O)C2CC2)ccc(-n2cccc2)cc1 c1(C(N2CCN(C(CCCOC)=O)CC2C)=O)cc2occc2n1C c1(COC)cncc(C(=O)NCCC2(NC(=O)C#CC(C)C)CC2)c1 N1(C(CN)=O)CC(C2CCN(C(=O)CC(Cl)Cl)CC2)C1 N1(C(=O)Cc2ccc(C(F)(F)F)c(Cl)c2)CCN2CCc3ccccc3C2C1 C1(NC(c2nccc(C)n2)=O)CCCN(C(=O)C(c2cncnc2)C)CC1 C=CCC(CC(C)C)C(=O)NCCN(C(C1CC1OC)=O)Cc1ccc(Cl)nc1 C(=O)(C1=CC2(CCOC2)C1)N(CC(C)NC(=O)C(c1ccccc1C)(C)C)CC C(=O)(CCC(=O)NC(C)CC(=O)NC(N1CC=C(C)CC1)C)NC c1(Cn2c(C(N(CC(CNC(C(CC)C)=O)C)C)=O)ccn2)ccccc1C c1(C(C)C)nc(CC(N2CC(O)(CNC(=O)C(F)c3ccco3)C2)=O)cs1 C=C=CCCC(=O)NCCCOCCOCCNC(c1ccnn1CC(F)F)=O C1(NC(c2c(CC)nco2)=O)CC(OC)CN(C(=O)C(C)(C)OC)C1 c1(C(c2n(CCC)nnn2)NCc2conc2C2CCCC2)cc(Cl)ccc1F c1(OC)cc(C(=O)NC2COCCC2NC(=O)Cc2noc(C(C)C)n2)cc(C)c1 c1(C(COC)NC(=O)NCCN2CC=CC2)cc2ccccc2o1 C1(NC(C(C=C)OC)=O)CCCC(C(=O)NCc2nc(O)ccc2C)CC1 c1(C(=O)NC(C(=O)N(CC(C(=O)NC)C)C)C)ccccc1C C1(C2(O)CN(C(=O)OC(C)(C)C)C2)(NCCN2CCN(C(CC)C)CC2)CC1 N1(C(C2C(c3n(C)ccn3)C2)=O)CCCCC(NC(C2C=CCCC2)=O)C1 N1(C(CN(C(=O)OCC)C)=O)CCCC2(CNC(C3OCCC3C)=O)CCCC12 S(=O)(=O)(CCC(=O)NCC(c1ccc(C)cc1)NC(=O)C(C)C1CC1)N(C)CC CCCCC(O)C(C)C(=O)NCC(C)CN(C)C(c1cccnc1OCCO)=O c1(C(=O)NC2(CO)CCN(C(C34C(C)OC(CC3)C4)=O)C2)ccc2nn[nH]c2c1 Cc1ccn2cc(C(=O)NC(C)CC3CN(C(C4CC(Cl)(Cl)C4)=O)C3)nc2c1 N1(CC(=O)NCC(=O)NC(c2cnn[nH]2)C)CCCCC1C c1(N2CC(C)C(NC(c3cncnc3C3CC3)=O)CC2)ncc(Br)cc1[N+](=O)[O-] C#CCCCCCCC(=O)NC1CC(O)CN(C(c2cc(C#N)cn2C)=O)C1 N(C1CCCc2cn(-c3ccccc3)nc21)C(c1c(C)sc(C(F)(F)F)n1)=O N1(C(C(C)N2CCC2)=O)CC(NC(=O)CCc2ccsc2)CC12CCC2 CC1(C)CN(C(C2CNC(=O)N2)=O)CC(CNC(c2ccc(F)c(C#N)c2)=O)O1 c1(C(=O)NCCC(C)NC(C(C)(C)OC)=O)ccc2c(c1)C(C)(C)CO2 c1(C(=O)NCC2C(NC(C(C)(C)CC3CC3)=O)C2)cc2cccnn2c1 C=CC(C)(O)CC(=O)NCCCOCCN(C)C(C1CC(=O)N(CCCC)C1)=O C12(NC(=O)COCc3cccc(Cl)c3)CC1CN(C(=O)CSCC(F)F)C2 c1(CC(=O)NC(CNC(C(C)OC)=O)CCOC)cccc2cn[nH]c12 c1(CSC(C)COC(F)F)nc2ccc(F)cc2n1Cc1ccccc1 c1(N2CCC(C)C(NC(c3ccc(SC)o3)=O)C2C)cc2nnc(C)n2cn1 c1(C(=O)NC2CN(C(C(COCC)C)=O)C2)cc2cncn2c(O)n1 C1(C(N2CCC(COC)(NC(c3nccnc3N)=O)C2)=O)CC(S(C)(=O)=O)C1 c1(CCC)sc(C(N2CC(CCNC(C3CC3C)=O)C2)=O)cc1Br C1(C(=O)NC(C(=O)N(CCSC)C)CC2CCC2)CCCC(C)C1 CCC(CCC(=O)NCC(=O)NC1CCOCC1)NC(=O)C(COC)OCC CC(N=c1cccc(Br)[nH]1)C1CN(Cc2ccccc2)CCO1 O=C(CCCC(F)F)NCCOCCCNC(C1(F)CCOC1)=O N1(C(C2CCC(CN(C)C)O2)=O)CC2CCC2(CNC(c2ccc(F)cn2)=O)C1 CC(C)(Cl)C(=O)NCC12CC(NC(c3coc(C4CC4)n3)=O)(C1)C2 C1(C(N2C(C(N(C)CCn3ccnc3)=O)C=CC2)=O)CN2CCCC1C2 C1(CNC(C2N(C)C(=O)NC2)=O)(NC(c2cccc(Cl)c2)=O)CC2CCC1CC2 C1(OCC(N2CCC(CNC(C3(CC)CC(F)(F)C3)=O)C2)=O)CCC(F)(F)CC1 N1(C(C=C)=O)CC2(CCC2)CC1CNC(c1csc2nnsc12)=O N1(C(c2ccc(=NC)[nH]c2)=O)CCC(C(=O)N2CCCCC(C)(F)C2)=C(F)C1 N1(C(C(C)=CC)=O)CC(C)(C)CCC1CNC(=O)C(=O)NCCC(N)=O C1(C(=O)NC2CC(CCNC(C(C)N(C)C)=O)C2)CCN(C2CC2)C1=O C1(C(N(C)CCNC(C2CC3(CSC3)C2)=O)=O)CC2(CC2)CN1C CS(=O)(=O)C1CCN(C(C2CCCC2)=O)CC1.C12OCC3CCN(CC13)C(=O)C2 CC1CN(C(c2nnc(S)n2C)=O)CCC1NC(c1coc2c1CSC2)=O C1(CCC(=O)NC(C(=O)OC)C2CCOC2)CCN(C(CC)C(=O)O)C1 c1(C(=O)NCC2(O)CN(C(C3CC(=O)N(C(C)C)C3)=O)C2)cncc2c1CCCC2 c1(C(C)C)cncc(C(N2CCC(O)(CNC(c3cc(C(F)F)[nH]n3)=O)C2)=O)c1 C1(NC(c2cncnc2)=O)CCCC(NC(C2(Cl)CC3CCC2O3)=O)CC1 C=C(CNC(=O)Cc1csc(C(C)(C)C)n1)CCNC(C1(O)CC(CF)C1)=O N1(c2nc(C)c(C)s2)CCN(CNC(c2ccc(C(C)C)s2)=O)C(=O)C1 c1(OCC(C)(C)NC(=O)CCC2CCCN2C(=O)CC2(O)CCC2)cccc(Cl)c1 N1(C(CCC=C)=O)CCCCC1c1n[nH]cc1C(=O)Nc1ccsc1C N1(C(c2cc(C)n(C)n2)=O)CCC(C(=O)NCC(O)C(C)O)C12CC2 C1(NC(=O)CC2CCCC2(F)F)(CO)CCCN(C(=O)CCCC2CCCC2)C1 CC(O)C(C)(C)CNC(=O)CC(CNC(c1coc(CO)c1)=O)C1CCC1 c1(-n2cc(C(=O)NC(C)C(CO)NC(=O)C(F)F)nn2)cccc(CO)c1 c1(SCC)cc([N+](=O)[O-])cc(OCC)c1O.C12CN(CC(C)O1)CC1(CC1)C(=O)N2 c1(CC)cc(C(=O)NCC2CCC(NC(c3nnc(C)cc3O)=O)C2)cc(Cl)c1 N1(c2ccc(OCC)cn2)CCC(C(N2CCC23CCC3)=O)(OCC)CC1 c1(-c2cn(C(CNC(C3C(C(CC)=O)C3)=O)C)nn2)cc(C)nn1C CC(CCOC)C(=O)N(c1ccccc1-c1nn[nH]n1)CC1CCOCC1 CC(CC1CC1)C(=O)NC1CCC1CNC(c1cnc(O)o1)=O N1(C(C(CC)SC)=O)CCCCC(CC(N2CCC2CSC2CCCC2)=O)C1 c1(C(=O)NC2(C(=O)NC(C(=O)NC)CC(C)C)CCCC2)c[nH]c2cnccc12 C1(C(=O)NCC=C=C)CN(C(=O)C(CC)OCC)CC1C n1(CC(=O)NCC(CCOC)NC(C2(CO)CCC2)=O)nc(C)cc1C(F)F Cc1ccc(C(=O)NC(C2(O)CCN(C(C3CCS(=O)(=O)C3)=O)C2)C)n1C C(c1cncc(O)c1)=CC(N1CCC(O)(C(C)NC(c2cc(Cl)cnn2)=O)C1)=O N1(C(c2c(C)ccs2)=O)CCOCCC1C(=O)NCC1(O)CCC(C)C1 c1(CCC(=O)NCC2COCC2NC(C2CC23CCC3)=O)cccc(Br)c1 C(=O)(C(C)C(C)OC)N1CC(NC(C2(NC(=O)OCC)CC2)=O)C1 Cc1ccc(C(=O)NCC(O)CNC(C2CC(C3CC3)=NO2)=O)c2c1CCC2 c1(OC)cc(OC)c(C(=O)NCCNC(c2[nH]cc(C(=O)OC)c2C)=O)cn1 C=C(C)CCCC(=O)NC1CCC(N(C(=O)Cc2cccc(OC)c2F)C)C1 C=Cc1ccc(C(c2nnnn2C2COC2)Nc2cc(C)cc(F)c2)cc1 CC(C)C(C(C)C)NC(=O)CC(CC1CC1)NC(c1coc(CO)c1)=O c1(NC(=O)Cn2cc(C3(OC(F)F)COC3)nn2)nncc2ccccc12 CCCC(C(=O)NCC12CC1CN(C(=O)COCC=Cc1cccnc1)C2)C(C)C C(C)(N=c1[nH]c(N(CCCNC(C)=O)C)nc(=N)[nH]1)c1nc(CCC)sc1 c1(C(=O)NC2C(NC(=O)CCCCc3cccc(O)c3)C2)cc(F)ccc1F c1(NC(C2CC(NC(C3CC3(F)F)=O)C2)=O)ncc2c(Br)cccc2n1 C1(C(NOCCC(=C)C)=O)CC(NC(C2CC(CCC)C2)=O)CCO1 c1(-c2cn(CC(CCNC(C(C)(C)O)=O)F)nn2)cccc(-c2ccco2)c1 C(CN=c1[nH]cnc(=N)[nH]1)C1CCN(C(Cc2n(C)nnc2)=O)CC1 C(=O)(CCCC(=O)N1CC(C)CCC1C(=O)NCc1ccc(F)cc1F)OCC N1(C(=O)COCC2CCCCC2)CCN(C(c2cccc(F)c2O)=O)C2(CC2)C1 N1(C(CNC(C)=O)=O)CC2(CC(CNC(=O)CCc3cnc(C)o3)C2)C1 C12(NC(CC(CC)C)=O)CCCC1N(C(c1ccnc(Cl)c1N)=O)CC2 c1(OC)ccc(O)c(C(N2CCN(C(=O)Cc3cnc(C)s3)CC2CCO)=O)c1 C(=O)(C1CCCn2c(Br)cnc21)N1CC(NC(C(C)=C2CC2)=O)C(O)C1 C1(CCNC(CC2CC(OC)C2)=O)CCCN(C(c2cc(OC)ns2)=O)CC1 Cc1ccc2c(n1)CCN(C(c1cc(C3CC3)on1)C(=O)NC1CC(F)(F)C1)C2 N1(C(CC(CC)C)=O)CCC2CCN(C(=O)C(C)(C)c3cccnc3)CC2C1 C1(OC)CN(C(C2CC(F)C(=O)N2)=O)C(C)(CNC(=O)CCc2cc(Cl)no2)C1 S(=O)(=O)(c1cccc2cccnc12)N1CCC(NC(=O)CC2COCCO2)C1 C1(CNC(c2cc(C)[nH]n2)=O)COCC2(CCN(C(C3SCCS3)=O)C2)O1 C1(CC)CN(C(c2ccc(C(=O)CF)cc2)=O)CC1NC(=O)C(C)CSC C(=O)(C1=CC(C)(C)C1)N1CC(CCNC(c2ccc(C(C)C)cc2)=O)C(C)C1 C(c1cccc(N)c1)=CC(=O)NCCC1CCC(NC(c2c(CC)cno2)=O)C1 Cc1cncc(CCC(=O)NCC(C)(C2CC2)NC(c2cnsn2)=O)c1 c1(C(c2n(C(CC)(C)C)nnn2)NCCCSC(F)F)cncc(C)n1 Cc1ccc(F)cc1C(=O)NC1CCCC1CNC(C1CCC(N=[N+]=[N-])C1)=O c1(C(N2CCCC(NC)C2)=O)cnc(O)nc1O.C1(OC)CC2N(C1)C2 N1(C(C(CC=CC)C)=O)CC(C(N2CCCC2CNC(N)=O)=O)C(F)(F)C1 C=Cc1ccc(C(=O)NC(C)CCCNC(c2cc(OC)cs2)=O)cc1 Cc1ccc2oc(=NC(C)C3CN(C(=O)C(C)CCN(C)C)CCO3)[nH]c2c1 c1(OC)ncc(C(=O)NCC2(O)CN(C(C3CCC(N(C)C)CC3)=O)C2)cc1F c1(SCc2[nH]nc(NC(CCc3nccc(C)c3)=O)n2)cc(N)ccc1Cl C(=O)(C(CC(C)C)n1nnnc1C(C)C)NC1(CF)COC1.c1(OC)ccc(Cl)cc1 N1(C(C2CCC2)=O)CCN(C(=O)CC(C(F)F)c2ccccc2F)C(CO)C1 C1(NC(COC2(C)CCC2)=O)CCC2CC1CN2C(=O)CC1CN2CCC1CC2 C(CCC(=O)N1CC(COCC)C1)NC(=O)OCC.C1(=O)C(C)N1 C(=O)(CCCCCC(=O)OC)NCCC(CNC(CCC#CC)=O)O c1(C(=O)NCC(=O)NCCCn2cccn2)cc(CO)on1 C(=O)(C(C)(F)C(C)(C)F)NC1CCC(NC(c2ccnc(OC(C)C)c2F)=O)C1 C12(CO)CC(CO)(CCO1)C2.C1(CC(C)(C)NC(=O)C(=O)N)CCCCC1 CC(C)CC(C(=O)NCC(C)C)NC(=O)C1CC1.C1(N)CCN(C(=O)C(C)OC)C1 N(C(=NCCCF)NC1CCc2sc(Cl)cc21)C(c1cc(Cl)sc1Cl)C(C)C N1(C(CC2(CC=C)CCCC2)=O)CCC(CNC(=O)Cc2cc(C)on2)CC1C c1(-c2c(CNC(c3ccc(N4CCCCCC4)nc3)=O)c[nH]n2)cccc(Cl)c1 CCS(=O)CC(=O)N1CCC(C)(C(=O)NOCCCCF)C1 N1(C(C(C)NC(N)=O)=O)CCC(CNC(=O)CCc2nc(C(C)C)no2)C1(C)C C(=O)(C1=CCCCNCC1)N1CCC(N2CCC(NC(C)C)CC2)CC1 c1(COC(C)C(=O)NCc2ccc(C(C)(C)C)cc2)cccc(Br)c1 CC1CCN(CC(=O)NC(Cc2cc[nH]n2)C(=O)NCCN(C)C)CC1 C=C(C)CC(C)C(=O)N1CCN(C(C2(SCC)CC2)=O)CC1c1cccc(Cl)c1 C1(NC(C2(OC)CCCC2)=O)CCN(C(C2CCCN2C(C)=O)=O)C1C(C)C C1(CC)C(C(=O)NCC(C)(C)n2ccnc2)CCN1C(=O)CCC1(C)CC1 c1(C(=O)NC2(C)CC(NC(C3C4CCC3(c3cnco3)C4)=O)C2)cc(Cl)ccn1 C1(CNC(CCCC#C)=O)CC2(CCN(C(c3csc(=NC4CC4)[nH]3)=O)CC2)C1 N(C(=NCCc1ccc(Cl)cc1Cl)NC(C)C)CCc1ccc(SC)cc1 c1(NC2CC3CN(C(C4(F)CCOCC4)=O)CC32)ncc2c(n1)COC2 c1(C(=O)NC(CNC(c2ccoc2)=O)C2CCC2)c[nH]c2ccncc2c1=O Cc1ccc(C(N2CCN(Cc3c(C)noc3C)C3CC23)=O)c(I)c1 c1(C(N2C(CC(=O)NCC(=O)OCCCC)CCCC2)=O)cc(OC)ccc1C C1(CNC(CCC(C)SC)=O)N(C(=O)C(CO)N(C)C)CCC1(C)C C12(C(N(CCNC(c3cnoc3C3CC3)=O)CC)=O)CCCC1CC(F)(F)CC2 C1(NC(C2(C)CC2)=O)C2CC3C1C3C2C(=O)NCCC12CC(CO1)C2 C1(C(=O)NC(C2CCN(C(C3(C#C)CCC3)=O)CC2)C)(CC)CCCCO1 CC1(C)CC(NC(=O)C=CCNC(C2CC2(C)C(F)F)=O)C1 C1(NC(C(CC=C)CNC(C2(C(=O)CC)CC2)=O)=O)CC(C)CC(C)(C)C1 C1(CNC(c2ccc(CSC)o2)=O)CN(C(C2(C(F)F)CC2)=O)CC12CC2 N1(C(c2nn(CC)nc2C)=O)CC2=C(C1)CN(C(=O)CC1CCC(C)CC1)C2 c1(C(=O)NC2(CNC(c3c(OC)c(F)ncc3)=O)CC2)cc(F)c(F)cc1F C12(C(N3CCC(=CCNC(c4cocn4)=O)CC3)=O)CC1CCC2(F)F C1(C(N(CCNC(CCCCC(=O)NCCC)=O)CC)=O)CCCC2CCCN12 Cc1ccc(CC(N2CC3(CC3)CC2CNC(c2cn[nH]c2)=O)=O)cc1F C12(CNC(c3n(CC)cnn3)=O)CCCC1N(C(=O)CNC(C)=O)CCC2 c1(N2CCN(C(CNC(c3c(CC)[nH]nc3Cl)=O)=O)CC2)ccn2nccc2n1 N1(C(CSCC(C)C)=O)CC2(C1)C(NC(=O)C(C)CC(F)F)CCS2(=O)=O N1(C(c2ccnn2CC2CC2)C(=O)NCCC2(C)CC2)CCOC2CCC12 CN1CCC(C)(CNC(C2CC2CNC(=O)CCc2cncn2C)=O)C1 N1(CC)CCOC(C(=O)NC2CC(CNC(c3ccnn3C)=O)C(O)C2)C1 N1(C(C2(c3ccc(C)cc3)CCCCC2)=O)CCCC(NC(=O)C2CC2)C1C C1(N(C(C(CC)=CC)=O)CC)CCN(C(c2c[nH]nc2-c2ccc(C)o2)=O)CC1 C1(CC(N2C(CN(C(c3cc(OC)cnn3)=O)CC)CCC2)=O)COC(C)(C)C1 N1(C(CCC(=O)OCC)=O)CCCN(C(=O)C(C)(C)NC(c2ccccc2)=O)CC1 Cc1cc(F)cc(C(N2CC3CC2CN(C(=O)CCC2CC2(C)C)C3)=O)c1N C1(OCC)CN(C(=O)Cc2cc[nH]n2)CC1CNC(c1cc(Br)no1)=O N1(C(=O)CCCCCOc2ccc(Cl)cc2)CCC2CN(c3ccccc3)CC12 C1(O)(C(C)NC(C(C)(CO)OC)=O)CCN(C(c2ncn(C(C)(C)C)n2)=O)CC1 C(CO)(C(=O)NCCCC1(C)CC1)NC(C1C(C)(CC)C1)=O c1(C(N(CC(C)NC(c2ccc(F)c(F)c2)=O)CC)=O)noc2cc(Cl)ccc12 C1(C(N(C)Cc2cncs2)=O)(CC2CC2)CCC1 C1(NC(C2(C(=O)NC)CC2)=O)CC(NC(=O)CS(C)(=O)=O)CC1O C1(NC(C2N(C)C(=O)CC2)=O)CCCCC1N=c1[nH]nc(-c2ccccc2)o1 c1(N2C(C)(CNC(=O)C3=CCC3)CC(F)(F)C2)ncnc2ccc([N+](=O)[O-])cc12 O=C(CCC(=O)Nc1ccccc1)NCC(CNC(=O)CNC(C1(O)CCC1)=O)F C(=O)(C1SCCc2sccc21)N(CCNC(c1ccnc2ncccc12)=O)CC CC#CC1CN(C(C2CN(C(C3(COC)CC=CC3)=O)CCO2)=O)C1 C1(C(N2CCCC(CC=C)C2)=O)CC2(CCN1C(C1CCNC1=O)=O)CC2 c1(CC)c(N2CCN(C(=O)C(C)NCS(C)(=O)=O)C(C)C2)nc(C)nc1Cl C(=O)(C1CNC(=O)c2ccccc21)NC(CC)CNC(=O)CSC(CC)CC CC1CCCN(C(=O)C=C2CCC2)C1CCNC(c1cccc(C(F)F)c1)=O C1(C(=O)NCCCCCNC(c2cc(C(C)C)no2)=O)CCSCN1C CCCCCS(=O)(=O)CC(=O)N1CCC(N(C(=O)CCn2cnccc2=O)C)C1 C12(NC(CC(CC)(F)F)=O)CCCC1CN(C(=O)Cc1cccc(O)c1OC)C2 Cc1noc(CCNC(=O)CC2CCCN2C(=O)CN2CCOCC2)n1 C(=O)(CCC(=O)N1CC2CC2(CNC(C2(C(C)(F)F)CCC2)=O)C1)NCCC c1(CCC)sc(C(N2CCC(CCNC(=O)CCc3ccon3)C2)=O)cc1CC C(=O)(CC(C)CNC(C1CCN(C(=O)CCC2CC2C)C1)=O)NC C(=O)CC(C)CC1CCC1.C1(CCO)(CNC(C(OC)OC)=O)CN(C)C1 c1(C(=O)NCCN(C(=O)CCc2ccn(C)n2)CC)cc(F)cc(S(N)(=O)=O)c1 C#Cc1ccc(CC(=O)NC2CC(C(F)F)(NC(C3(C)CCOC(C)C3)=O)C2)cc1 Nc1cc(C(=O)NCCOC2CCN(C(C3CC4COCC4C3)=O)C2)ncc1Cl CC1(C)CCCC(C)(NC(C2CCN2C(=O)CC2CCCC23CC3)=O)C1 c1(C(N2CCOCC2)C2CC2)nn2c(c1NC(=O)NCC(COC)F)CCC2 c1(C(=O)NC(C(C)C)(C)CNC(=O)CC2C(C)(C)C2(C)C)cnc2ncccn12 N1(C(c2cccc(C)c2)=O)CCC2C(CCCN2C(=O)Cn2ccc(C)n2)C1 CCC(C)C(=O)C(=O)N1CCC(CC)C1C(=O)NC(C)(C)CCF CC(N=c1[nH]c(=NCC2CC(=C3CC3)C2)[nH]c2cc[nH]c12)c1nc(Cl)ccc1Cl C(=O)(CCCCCCNC(=O)C(C)(O)C1CC1)N(C)CC1CCN(C)C1 c1(CC)ncccc1C(N1CCC(CCNC(=O)CSc2nncn2C)C1)=O CCCC(C(=O)NC(CNC(C1CC(=O)N(c2ccc(F)cc2)C1)=O)CO)OC C1(C(=O)NC(C(CC)C)CO)CCCCC1(C)NC(c1ccc(O)cn1)=O C1(C(N(C(C)CNC(c2cn(-c3ccccc3)nn2)=O)C)=O)CCS(=O)(=O)C1 C1(NC(c2c(N)cc(C)c(F)c2)=O)CN(C(C2CS(=O)(=O)C2)=O)C2(CCOC2)C1 C(C(=O)N(CC(=O)N(C)C1CC1)C)(C(C)(C)C)NC(C(CC)SC)=O Cc1cc(N)n2ncc(C(=O)N(C)CC3(O)CCCN(C(=O)C(F)F)C3)c2n1 c1(OC)ccc(NC(=O)Nc2ccc(OCC(O)CNC(C)C)nc2)c(F)c1 N#CC1CN(C(=O)CCC=Cc2cccs2)CC1NC(=O)C1=COCC1 Cc1ccc(C)c(CN2CCN(Cc3cc(C)c(C#N)o3)CC2)c1O C1(C(=O)NC(CSC)(C)C)CCCCC1CNC(=O)Cn1nc(C)nc1C C(=O)(NNc1cccc(C(C)(C)C)c1)c1c(CCC)nccn1 C(=O)(CCC(=O)c1ccccc1N)N(C)CC1(NC(C(C)SC)=O)CC1 OCCCCCC(c1nnnn1Cc1ccccc1)NCc1cc(Cl)ccc1F C1(CNC(CN(C(C(C)C2(O)CCC2)=O)C2CC2)=O)CC2OC1C1CC21 C1(NC(c2n(C)nc(Br)c2)=O)CN(C(=O)C=CC2CC2)Cc2nccn2C1 N1(C(C(CCSC)NC(N)=O)=O)CC2CCC1CN2C(C1CC1F)=O CCCS(=O)(=O)CC(=O)NCC(C)(C)CN(C(=O)Cc1nnn(C(C)(C)C)n1)C c1(C(N(CC(C)N(C(C2C(OCC)C2)=O)C)C)=O)ccnc(N(C)C)c1 CCC(C)C(CC(=O)NCC1CCOC1)NC(=O)C(CC(C)(C)C)OC CC1OC(C)(C)OC1(C)C(=O)NCCNC(=O)CSCc1cccs1 c1(C(=O)NC2(CN(C(=O)CC3CC4(CC4)CO3)C)CC2)cn(C)c(=O)n1C Cc1cc(C(=O)NCCCCN(C)C(C2(O)CC(CF)C2)=O)ncc1Cl C1(CCN(C(=O)CC(C)(C)F)C)CCCCN1C(=O)C=Cc1cc[nH]n1 N1(C(c2n(CCC)nc(C)c2)=O)CC(OC)CC(NC(=O)CCC2CC2C)C1 c1(C(N2CCN(C(C3(CC#C)CCC3)=O)CC2CC)=O)cccc2oc(=N)[nH]c12 C(=O)(C1CCCc2n[nH]cc21)NC1CC(O)CCN(C(C2CN(C)C2)=O)C1 CCC(CC(=O)NCc1cccc(O)n1)SC.N12CC(C)(C1)CCC2=O n1(CCC)nc(C(C)OC)nc1-c1cc(Br)c(Cl)s1 CC1CCC(CC(N2CC3CC(NC(=O)CCc4cccnc4)C3C2)=O)CC1C C1(NCCCNC(CC)=O)CCCN1NC(=O)c1ccc(C)nc1 c1(C(=O)NCCCN(C)C(c2ccc3nn[nH]c3c2)=O)ccnc2c1ccn2C c1(OC)cccc2sc(C(N3CC(CNC(=O)C(C)CF)CC(C)(C)C3)=O)cc12 c12nc(C)c(o1)C(=O)NC2.N1(CCC)CCCC1CC(=O)NC1CN(C(C)=O)C1 N1(C2CCN(C(c3c(C)cc(NC(=O)NC4CC4)s3)=O)CC2)CC(C)OC(C)C1 c1(OC)cc(C(CC(N)=O)NC2(c3nnnn3C)CCCC2)c(C)cc1C CCC(CCCC(=O)NC)OC.C1(C(=O)NC)(CCCOCCF)CC=CC1 CC1CN(C(c2c[nH]c(Br)c2)=O)CC1NC(C1COCCN1C)=O c1(C(=O)NC2(CNC(C3CC4CCC4C3)=O)CC2)cc2cc(Br)cn2cn1 C=C(C(=O)NCC1CN(C(=O)Cc2ccc(C)c(O)c2)CCC1O)C(F)(F)F C1(CC(=O)NC(C(=O)NCC)C)C2CCCC2N1C(=O)C=Cc1cc[nH]c1 C1(CC(=O)NCCn2c(C)ncc2)Cc2ccccc2CN1C(=O)CNC(C)C CC(C)CCCC(C)C(=O)NCCCN(C)C(C1(c2ccncc2)CC1)=O C1(C(=O)NCCC(CCNC(COC(C)=O)=O)C)CC(C)(C)CN1C n1(C2(C(=O)NC(CN(C(C(C)N(C(C)=O)C)=O)C)C)CC2)ncc(Br)n1 C1(C)(NC(Cc2c(CNC(C(C)OC)=O)nco2)=O)CCCCCC1 Cn1nc(C(F)(F)F)c(I)c1CNC(C1CCCC1c1ccc(Br)cn1)=O c1(C(=O)NCC(C(=O)NC2CCC2)N(C)C)ccc(O)cn1 c1(CC(=O)N(C(C)CNC(C23CC(F)(CO2)C3)=O)C)nnc2n1CCC2 c1(C(=O)NCCC2CC(NC(CCS(C)=O)=O)C2)cccc2nsnc12 C(=O)(C1=CC2(CN(C(C3(C)CCCC3O)=O)C2)OC1)NCCOCC#C C1(OC)(CNC(c2nnnn2C(C)(C)C)c2csnn2)CCCC1 c1(C(N2CCC(n3ncc(C)c3)CC2)=O)oc2ccccc2c(=O)c1C C1(CCNC(=O)CCCc2ccccc2)CN(C(C2CCCOC2)=O)CCCO1 C1(C(N(C(C)CNC(c2cnc3n2CCCC3)=O)CC)=O)CN(CP(C)(C)=O)C1 c1(N2CCC(NC(CCC=C)=O)C(F)C2)nc(C(C)C)ccc1C#N N1(C(CN(CCC)C(c2cccc(=O)o2)=O)=O)CCOC(C(N)=O)C1 C1(CC(=O)NCC(C)CNC(C2CS(=O)(=O)C2)=O)CC2C=CC1CC2 N1(C(c2nc(OC)nc(O)c2)=O)CC(NC(c2sc(F)cc2C)=O)CC2(CC2)C1 C1(C(N2C(C)CC2C(=O)NCC2(C(N)=O)CC2)=O)CCC2(CCC2)C1 c1(C(=O)NCCCC2OCCN(C(C(CC=CC)C)=O)C2)cc([N+](=O)[O-])oc1C c1(OC)ccc2c(C(=O)NCC3C(C)CCN3C(c3cc[nH]n3)=O)ccnc2c1 N1(C(c2c(N)ccc(C(F)(F)F)c2)=O)CC2CC1CCC2NC(=O)Cc1cnoc1 c1(OC)cc(=NC(=O)N2CCCC(CNc3ccccc3)C2)[nH]n1C N1(C(C2(C=C)CCN(C(=O)CCC3CC(OC)C3)C2)=O)CCn2nc(C)nc2C1 c1(C(N2CCC(C)(CNC(C(C=C)O)=O)C2)=O)ccc(OC)cc1OCC(F)F N(C(=NCCc1cccs1)NCC1CCN1CC)CC(N(OCC)C)=O N1(C(c2n(CC#C)ccc2)=O)CC(CNC(C2CC2Br)=O)OC2COCC12 N1(C(c2cc(CC)no2)=O)CCC(C(=O)NCC2C(=O)NN=C2C)C(O)C1 C(C)(C(CC(=O)N1CCSC2CCC12)NC(c1cc(O)nc(C)n1)=O)OC C1(C(=O)NCC2(NC(c3cc(C)n(C)n3)=O)CC2)CCN2CCOCC12 c1(C(N2CCN(C(c3c(C)nsc3)=O)C(C)C2C)=O)ccc2nc(CO)[nH]c2c1 N1(C(c2cnn(C(C)C)c2F)C(=O)NC)C2CCC1CC1(C2)N=N1 C1(O)(C(N2CC(OC)(CNC(=O)Cn3cc(C(C)=O)nn3)C2)=O)CCOC1(C)C Cc1nc(Cl)ccc1Cc1noc(CC2CN(C3CC3)C(=O)O2)n1 C(CO)(C(C)N=c1[nH]c(N2CCN(CC)C(C)(C)C2)nc2c1CCCCC2)SC N1(C(CC=C)=O)CCC(NC(=O)CC2CN3CCN2CC3)C(CC)C1 C(=O)(C(C)(C)CN(C)C(C1CC(C)(O)C1)=O)N1CCC(OC)C1 c1(C(=O)NC(CCN(C)C(c2ccns2)=O)c2cccs2)nc(=O)n(C)[nH]1 C(=O)(C(O)CCNC(C1CC(C)N1C(C1CC=CC1)=O)=O)OC c1(CNC(CN(C(C=C(C)c2ccco2)=O)C2CCC2)=O)ccn(C)c(=O)c1 C1(CCN(C)C(C2CC2c2cnc[nH]2)=O)CCN(C(C2(O)CCCC2)=O)CC1 c1(CC)cccc2[nH]c(C(=O)NCCCCC(C)NC(=O)COC(C)C)cc12 C1(C)(C(=O)NCC2(F)CCN(C(C3CCC(=C)CC3)=O)C2)CCCNC1=O N1(C(C(CC)C(C)C)=O)CC2=C(C1)CN(C(=O)Cc1ccc(Cl)cc1C)C2 C1(NC(C2C(CC(C)C)C2)=O)CC(C)(NC(=O)CC(C)n2cccn2)C1 c1(N2C3C(C(=O)Nc4ncc(C)s4)C(C3)C2)ncc2cccc(O)c2n1 c1(C(=O)NC2C3CN(C(C4(COC)CCCC4)=O)CC32)ccc(=O)n(CCF)n1 c1(C(=O)NC2C(NC(c3ccc(CSCCC)o3)=O)CCC2)cc(N)ccc1Cl N1(CCNC(C2C(C)C2)=O)CCCN(C(c2cn(C)nc2-c2cccnc2)=O)CC1 C1(C(C(=O)NC(C)CCNC(c2cc(Cl)n(C)n2)=O)C)CCC(C)(C)CC1 CC(C)(C)CC(C(=O)NC1CC2CC2C1)NC(=O)CC1CCCO1 C1(CCNC(CC(C)OC)=O)CCN(C(C2(C)CC2C(C)C)=O)CC1 N1(C(C(C)OCCC(C)C)=O)CCCC(CNC(=O)CC(C)(C)C2CCCC2)C1 c1(C(=O)NCC(C)(C(C)C)NC(CCC#C)=O)nc(O)nc(O)c1F C1(=O)C(CC(C)C)ONC(=O)CCOC23CC2CN1C3.CC.OC C12(C(=O)NC3CC(F)(CNC(Cc4cccc(OC)n4)=O)C3)CCCN1CCC2 c1(C(N2CC(O)(CCNC(CC3(C=C)CCC3)=O)C2)=O)cc(O)ccc1OCC C1(CN(C(=O)C(N2CCOCC2)=O)CC2CCN(C)C2)COCCN1C N#CC1(C(=O)NCCC2CCCCN2C(=O)C2=NNC(=O)C2)CC2CCC1CC2 C1(C(N2CCC(CCNC(c3coc(CO)c3)=O)C2)=O)Cc2ccccc2CO1 c1(C(=O)NC(C(=O)Nc2ccc(-c3ccco3)nc2O)=O)cc(Cl)c([N+](=O)[O-])[nH]1 N1(C(C2OCCC(C)(C)C2)=O)CCC2(C=C(C(=O)NC3CCN(CCF)C3)C2)C1 C1(NC(COCC#C)=O)CCC(C)(NC(c2ccccc2OCCC)=O)CC1 c1(C(=O)NCC(CNC(c2c(C(C)C)ccs2)=O)OC)cncc(C2CC2)c1 c1(OC)cc(C(N2C3CCC(C3)C2C(=O)NCCC(C)C(=C)C)=O)ccc1[N+](=O)[O-] c1(C(=O)NCC23N(C(C(C(COC)C)C)=O)CC(C2)C3)cnc2ncccn12 N1(C(C2CC(=C3CC3)C2)=O)CC(C2CC2C(=O)NCC2(SC3CCC3)CC2)C1 Cc1cc(F)cc2[nH]c(NC(=O)NC34CC(CNC(=O)OC(C)(C)C)(CO3)C4)cc12 c1(CCC(=O)N(CCN(C(CCNC(=O)NC)=O)C)C)ccc(F)cc1F C1(C(=O)Nc2c(CC)nn(C)c2)COC2(C1)CN(C(=O)CC1C(C)(C)C1(C)C)C2 Cc1cc(C(=O)NC(c2cn(C)nn2)C(N2CCC(O)C2)=O)ns1 C1(C(=O)NCC2CCC(CNC(C3(CC)COC3)=O)C2)Cc2cncn2C(=O)N1 Cc1ccn(C(C)C(=O)NCCCN(CCCNC(=O)CC2CCCO2)C)n1 C(=O)(C1CCCc2scnc21)NC(C1CCCCC1)CNC(c1cnn(CC)n1)=O C(C)(CC(=O)NC)CCN1CCOCC1.c1(C2C(=O)N2C2CCOC2)cn(C)nn1.CS c1(C(=O)NC(C)CN(C)C(C2C(C)(C)C2(C)C)=O)cc(N)c(Cl)cn1 N1(C(CC(COC)(C)O)=O)CC2(C1)SCCC2NC(=O)CN1C(=O)CNC1=O C12(OC)CCC(NC(C3CC(C(=O)NCc4ccncc4Cl)(CC)C3)=O)(CC1)C2 C12(C(N3CCCC(C=C)C3)=O)COCC1CN(C(=O)CSCC(N)=O)C2 C1(CNC(=O)C=C2CCC2)CCCN(C(=O)Cc2ccc(F)nc2)CC1 C(C(C(C)C(C)C)NC(=O)CSc1n[nH]c(C)n1)NC(c1nccc(NC)c1)=O c1(NC(N2C(CCCC)CCC2)=O)cc(C#N)cnn1 C1(NC(C=CC(C)NC(c2nc(C)n(C)c2)=O)=O)CCCCCC1C C1(NC(CCOCCN(C)C)=O)CC1C1CCCN(C(C2(C3CC3)CC2)=O)C1 C1(C(=O)NCCNC(C2CCCN(CC)C2)=O)CCc2nncn2CC1 Cc1ccccc1NNC(=O)C(C)Cc1nc(C2CCCCCN2)no1 CCS(=O)(=O)C1CCN(C(=O)CCc2nnc(-c3ccccn3)o2)C1 C(CN=c1[nH]c(=N)[nH]c(=NCC(c2ccco2)C2CCCC2)[nH]1)SC(C)C N1(C(C(C2CN(C(C3(OC)CCCC3)=O)C2)O)=O)CC(C)CCCC1C C(=O)(C1=NOC(CNC(c2coc(C(F)F)c2)=O)C1)NC(C(=O)OCC)C C12(C(=O)NCC3(O)CN(C(c4c(COC)cccc4)=O)C3)CC1CCC2(F)F C1(C(C)C)CN(C(c2cnc(O)o2)=O)CC1C(=O)NC(C)CCO C1(C(=O)NCC(=C)CC)CC2(CCN1C(c1cnco1)=O)CC2 c1(C(=O)NC2CCC(CCNC(c3ccc(CC)o3)=O)C2)ncc(C)cn1 c1(CC(CNC(C2CC2CF)=O)N(C)C(C2(C)COC2)=O)ccccc1 c1(CN(CC(=O)NCCC(C)N(C)C(C2CC=CCO2)=O)C)ccccc1 C1(CC(=O)NCCC2(C)CC2)(OC)CN(C(c2occ(C(=O)OC)n2)C)C1 N1(C(CCC(C)O)=O)CCC(CNC(=O)COC2CCCCC2C)C1(C)C c1ccccc1.C1(C(N(CCN(C(C2(CCC)CC2)=O)C)SC)=O)CC(CF)C1 C1(CC)CN(C(=O)C(=O)Nc2cc(C)ccc2N(C)C)CC2(CCCOC2)O1 N1(C(C2CCC(CC)CC2)=O)CC(C(=O)NC(C)(CO)C(C)C)CCC1(C)C c1(C(N(C(CNC(C2(CO)CC(F)(F)C2)=O)C2CC2)C)=O)cccc2sccc12 CCCCCC(=O)NCCC(O)C(=O)NCC1(CSC)CC1 c1(C(=O)NCCCCNC(c2ccc(F)c(F)c2F)=O)ccc2nc[nH]c2n1 C1(CNC(CC2(C=C)CC2)=O)CN(C(c2ncc(OC)nc2OC)=O)CC1(F)F C1(NC(c2ccc(F)o2)=O)(CO)CCCN(C(=O)CCc2cncs2)C1 c1(OC)ccc(C)c(C(=O)NC2CN(C(=O)C(C)(C)C(=O)N(C)C)CC23CC3)c1 Cc1cccc(C(O)C(C)NC(c2cccc(C)n2)c2nnnn2C(C)C)c1 c1(C(=O)NC2CCN(C(CCn3ncc(C)c3)=O)CC2C)ccn2c1CCCC2 CCCC(CC(C)C)C(=O)NCCN(C(=O)CC(C)(C)C(F)(F)F)C1CC1 N1(C(CCN(C)C)=O)CC2(CCC(C(=O)NCc3ncccc3F)O2)C1 c1(C(=O)NCC2(F)CC(COC)C2)ccncc1NC(C)=O.C12CC1C(=O)N2 c1(N(C(CCC)C2CCCC2)C(c2ccc(CSCCOC)o2)=O)cccc(C)c1 C1(C2C(N)CN2)CCCN(S(=O)(=O)C(F)F)C1 N1(C(c2c(CC)con2)=O)CCCCC(NC(=O)C(C)N(S(C)(=O)=O)C)C1 c1(CC)c(C(N2CCC2CNC(=O)CCc2ccnc(Cl)c2)=O)cnn1C Cc1[nH]nc(C(N2CC3CC2C3CNC(C2CCCC2)=O)=O)c1Cl c1(CN2CC3C(C(=O)NCc4nn[nH]n4)C3C2)c(F)cc(I)cc1F c1(OC)cc(C)c(Cc2cn(C3CC(NC(C4(C#N)CCCO4)=O)C3)nn2)c(C)c1 c1(C(=O)NC(C2CCCC2)CNC(c2c(CC)nco2)=O)cnc(C)nc1OC N1(C(C(C)SC(F)(F)F)=O)CC2CC3CC2C1C3NC(c1cc(C(N)=O)c[nH]1)=O c1(C(N2CC(C)(CC(=O)Nc3ccc(F)c(CO)c3)C2)=O)cc(F)c(O)c(F)c1 C12(C(=O)NCC3CC(OCc4nccc(OC)n4)C3)CC3CC(C(=O)N1)C2C3 N1(C(CN(CCC#C)C)=O)CC(NC(=O)CSc2nccn2C)C(C(F)F)C1 O=C(C#CC1CCCC1)NC1CC2CC(NC(c3cc4ccncc4[nH]3)=O)CC21 N1(C(c2c(OC)nsc2)=O)CCCN(C(c2coc(C(F)(F)F)c2)=O)C(CO)C1 N1(C(CC2CC(=C)C2)=O)CCC(OC)(NC(=O)CC(F)(F)F)C1 Cc1cc(Cl)ccc1CNC(=O)CC1CCCN(C(=O)C(C)n2cccc2)CC1 c1(CC)cccc(C(CCC)NC(=O)CC2CN(Cc3cc(Cl)cn3C)C2)c1O c1(NC)cnc(Cl)cc1C(N1CCN(C(=O)C(O)Cc2ccccn2)CC1)=O N1(C(c2cc(C)ns2)=O)CCC=C(CNC(C23CCC(O)C2CC3)=O)C1 N1(C(CC(C)O)=O)CC2(C1)CN(C(=O)Cc1ccc(F)cc1C(F)(F)F)CCO2 c1(C(=O)NCC2(O)CN(Cc3cc(C(=O)OC)sc3)C2)nc(O)sc1C C12(C(=O)NC(C#C)(C)C)CCC(CC1NC(=O)COC)C2 CC1=C(C)CC(C(=O)NCCC2COCCN2C(=O)CN2CCCCC2)CC1 C1(C(=O)O)CCCC(N=c2ccc3c([nH]2)CCCCCC3)CC1 C12(NC(CC3C(CNC(C(C)C4CCCC4)=O)C3)=O)CCCN(CCC1)C2 c1(NC(C(=O)NC(CN(C(C)=O)CC)C)=O)ccc(Sc2ccc(I)cc2)cc1 c1(-c2cn(CC(CNC(C)=O)(F)F)nn2)ccc(NC(=O)CC(F)(F)F)c(F)c1 C(=O)(CCC(=O)NCCN(C)C(C1(C)CC=CCC1)=O)NC(C)=O C1(N(C(=O)C(C)(C)NC(=O)Cc2ccc(Cl)s2)C)COC(C)(C)C1 c1(C(N2CC3CCC(C2)N3c2ccncn2)=O)ccc([N+](=O)[O-])nc1 N1(C(CN(CC)CC)=O)CCC(F)(F)C(CNC(c2cc3cnccc3o2)=O)C1 C1(C)(NC(=O)OC(C)(C)C)CCCCC1CC.C=CC1C(=O)OCC(=O)N1 C(=O)(C(C)C(F)(F)F)N1CCCC(CCC(=O)NCCc2cn(CC)nc2)C1 CCC(CC(=O)NC1(CCNC(=O)C(C)(C)CF)CCCC1)C1CCC1 c1(C(N(CCN(C(c2cc(CC)sn2)=O)C)C(C)C)=O)ccnc2ccsc12 N1(C(C(C)C(F)F)=O)CCC(NC(=O)C=Cc2ccncn2)C12CCC2 N1(C(C2(C#N)C(C)(C)C2)=O)CCC(C2(NC(=O)C(F)C(C)(C)O)CCC2)CC1 c1(C(=O)NCC2OCCN(C(C3(COC)CCCCC3)=O)C2)nccc(Cl)c1C c1(C(=O)NCCS(CC)=O)cnc(CNC(C2(C)CCCCC2)=O)nc1 CCCCS(=O)(=O)CC(=O)NC1CN(C(C2CN3CCN2CC3)=O)CC1C C=CCCCC(C(=O)N(C(C)CSC)C)NC(c1cnc(C)nc1)=O c1(C(=O)NCC(C(=O)N(C)CC2(COC)CCC2)OC)c(C)cccc1O c1(OCC)cc(C(N2CCC(CF)(NC(c3cc(Cl)no3)=O)C2)=O)cc(Cl)c1O C1(NC(c2c(C)noc2)=O)COC2(CCN(C(=O)Cc3cccc(Cl)n3)C2)C1 C(CS(C)(=O)=O)N(C)C(C1C=CCN1C(=O)Cn1cc(CO)nn1)=O C1(NC(c2ccc(Cl)nn2)=O)COC2(C1)CN(C(C1C(F)(F)C13CCC3)=O)C2 C1(CCC(=O)N(C2CCCOC2)C)CCCN(C(c2cnn(CCO)c2)=O)C1 C(N=c1cc(C2CC2)nc[nH]1)c1c(CNC(CC2ON=C(CC)C2)=O)cccc1 c1(NC(C(C2CCN(C(=O)CSc3ncccn3)C2)C)=O)cccc(O)n1 C1(NC(Cc2nc(C)sc2)=O)(CNC(=O)C(c2cnn(C)c2)C)CCCCCC1 N1(C(c2cc(OC)ncn2)=O)CCC(NC(=O)CC2CCNC(=O)C2)C(F)C1 c1(C(=O)NC2COCCN(C(c3c(CC)ocn3)=O)C2)ccc2nncn2c1 c1(C(=O)NCC(C2CCC2)NC(c2c(C)cns2)=O)cnc2n1CCCC2C N(C1CCCOc2ccc(Br)cc21)(C(N1CCS(=O)CC1)=O)Cc1c(CC)n[nH]c1 C(=O)(CCCC(C)NC(c1ccncc1N)=O)NCC(C(=O)OC)C CC1CN(C(C2CC=CCO2)=O)CC(C)N(C(c2ccc3c(n2)NCC3)=O)C1 C(CC(C)C(=O)NCCCCCN(C)C(C1COCCN1C)=O)OC N1(C(C2CN(C(=O)CN(c3cnn(C)c3)C)C2)=O)CC2CC(SC)C1C2 Cc1cc(C)c(C(=O)NCC2CCN(C(c3ccnn3CC#N)=O)C2)cc1C N1(CC)CCC(C(=O)NC2(C)CN(C(=O)Cc3ccccc3O)C2)CC1 C1(C(CC(=O)NC2(CNOCC3CCC3)CC2)=O)CCC(=O)N2CCCCC12 C1(O)(C(C)NC(C(CCC)O)=O)CCN(C(c2cnn(C)c2)=O)CC1 N1(C(CCC)C)CC(C(N2CC(O)(C(C)NC(C3CNC(=O)C3)=O)C2)=O)CC1=O Cc1csnc1C(=O)NC(C)CCN(C)C(C1CCCCS1)=O CC#CC1CCN(C=O)CC1.C1(CC=O)CCC(C)CO1.C12CCN1N1CC2C1 C(C(=O)NCCOCCNC(C1CC(SC(C)(C)C)C1)=O)(c1cccs1)SC CCCCC(O)C(=O)NCC1CN(C(C2CN(C)C(=O)N2)=O)CCCO1 c1(C(N2CC(C(N3CCOC4(CC4)C3)=O)C(F)C2)=O)nccc2cc[nH]c12 c1(CC(C)C)cc(=NCC2CCCN(C(=O)C(C)OCC3CC3)C2)[nH]cn1 c1(CN2C(C(=O)N=c3ccn(CCO)[nH]3)CCC2)ccc(Br)cc1[N+](=O)[O-] C=CC(C)(C)C(=O)N1CCC(CCC(=O)NCC2COC(=O)N2)CC1 C12(C)CCC(C1(C)C)NC2=O.c1(CC(CC(=O)OCC)N)ccc(Cl)c(F)c1 c1(C(=O)NCCn2ccnn2)csc(Cc2ccco2)n1 c1(CC2C(NC(C3(C(C)NC(c4c(C)[nH]cc4)=O)CC3)=O)C2)ccccc1F C1(C2C(=O)N2)Cc2ccccc2C1.c1(C2N(CC)CC2)ccc(Cl)cc1 N1(CCN2C(CSCC)CCCC2)CCN(c2ccccc2)C(C)C1=O c1(C(N2C(COC)CN(C(c3ccsc3)=O)CC2)=O)cn2nc(C)sc2n1 CN1CCN(C(=O)C(F)C2CC(NC(c3cnc(=N)[nH]c3)=O)C2)CC12CC2 C12(CNC(c3n[nH]cc3Br)=O)CCC(C1)N(C(=O)CCC1CCCC1)C2 c1(OCC(C)(C#N)C2CCOC2)cc(Br)ccc1F N1(C(C(C(C)C)SC)=O)CCN(C(=O)C(C)(C)F)CC1CF.C1C(=O)N1 C1(NC(C(CC)=CCCC)=O)CCSC12CN(C(C1CCCN1S(C)(=O)=O)=O)C2 N1(C(c2cc(CC(C)C)on2)=O)CC(N(C)C(c2cc(=O)n(C)o2)=O)C2(CC2)C1 CC(CCCNC(C1(F)CCOC1)=O)N(C(=O)CCN(C)CCO)C1CC1 N1(CC(=O)NC(C(=O)NCC(=O)OCC=C)C2(O)CCC2)CCNC(=O)C1 C12(NC(Cn3nc(C)n(C)c3=O)=O)CCCC1N(c1nccc(C#N)n1)CC2 c1(C(=O)NCC23N(C(C(C#C)(C)C)=O)CC(C2)C3)ccc(OC(C)C)c(Cl)c1 c1(C(C)C)cccc(C(=O)NC2CCC(CCNC(C34CCC(CC3)O4)=O)C2)c1 c1(C(=O)NC2(C)CN(C(C3CC34CCOC4)=O)C2)nnn2c1C(=O)NCC2 c1(CC)ccc(C(=O)NC2(CF)CCN(c3nc(SC)ns3)C2)cc1 c1(N(C(CCSC)C(=O)N2CCCC2)C(=O)C=Cc2ccco2)ccc(O)nc1C C1(CNC(CCn2c(C)ncc2)=O)CN(C(=O)C(C)C(C)(C)C)CC1(F)F Cc1ccc(C(=O)NCC2(O)CN(C(c3c[nH]nc3OC(C)C)=O)C2)c(N)c1Cl C(=O)(C(CCC1CC1)NC(c1cc(C(F)F)[nH]n1)=O)NCCc1cc(C)on1 C1(NC(C2C(OCC)CC2)=O)CC2(CC(OC3CC3)C2)C1 CCC(CCC(=O)N(C1CCCN1C(=O)C(C)=C(C)C)C)NC(=O)OC c1(C(N(CCCNC(CCCOC(C)=O)=O)C)=O)ccc(N2CCOC2=O)cc1 C(=O)(CC(C)(C)C1CC1)N1CCC(NC(=O)COCC2(C)CC2)C1 c1(NC(C2CC(NCc3c(CBr)nn(C)c3O)C2)=O)c([N+](=O)[O-])ccc(Cl)c1Cl c1(SC)ccc(Cl)c(C(=O)NC2CN(C(c3cccc(C)c3O)=O)CC2O)c1 C(=O)(C#CC1CCCOC1)N1CCCN(C(C2(F)CCCCC2)=O)CC1CO c1(CN2CCC(N(C(c3ncc(C)nc3)=O)C)C2)ncccc1[N+](=O)[O-] c1(C(=O)NC(CC(C)NC(CCC2CC2)=O)C)cc(C)ccc1N1CCCC1.CCS N(C(=NCCCCl)NCC12CCCC1C2)CCSc1cc(C)c(Br)cc1 c1(CC(C(=O)NC2CC(C(C)(C)C)C2)NC(COC)=O)ccccc1Br C(CCNCC(F)(F)F)(N=c1cc(C(=O)OC)n(C)[nH]1)OC C1(CC)=CC(C)(N)C(C(=O)Nc2nc(C(F)(F)F)cn2C)=C1 C1(NC(c2ccsn2)=O)CCN(C(C2(F)CCCC2)=O)CC1F C(=O)(C1CCc2cccc(O)c21)N1CCCC(N(C(CNC(=O)OC)=O)C)C1 C=C(Cl)CCC(=O)N1CCC1CNC(C1(N(C)C)CC1)=O C1(C(CO)NC(C2(SC)CC2)=O)CCN(C(c2cncn2C(F)(F)F)=O)CC1 c1(C(N(CCNC(=O)CCN2CCC(O)CC2)CC2CC2)=O)cc(F)cnc1O C1(CNC(c2nccc(CC)c2)=O)CCN(C(c2sc(C)cc2C)=O)C12CCC2 c1(C(=O)NC2CC(C(F)C(=O)NCc3cnccn3)C2)ccc2cc[nH]c2n1 c1(CC(=O)N(C2CN(C(C3(CCF)CCC3)=O)C2)C)ccc(C(F)(F)F)cc1 N1(C(C2CC(C)NC(=O)C2)=O)CCN(C(=O)Cc2c(F)cccc2F)CC(O)C1 c1(C(=O)NC2CC(NC(C(c3ccc(C)cc3)O)=O)C2)ccc(I)c(F)c1F Cc1c[nH]c(C(C)(C)C)c1SC1CC(N2C(NC(=O)OC(C)(C)C)CCCC2)C1 N1(c2c(C)c(N3CCCC(CC(C)C)C3)ncn2)CC(C)S(=O)(=O)C(C)C1 CCC(CCCC(=O)NCCOC1CCOC1)NC(c1cnc2ccccn12)=O C(c1ccc(F)cc1Cl)=CC(=O)Nc1ncc(F)s1.C12CN(C1)C2=O N1(C(C2CCN(C)C2)=O)CCC(C2(NC(C3OCCOC3(C)C)=O)CCC2)CC1 c1(C(=O)NC2(CC)CC2)cccn2cnnc12.C123CCC(CO1)(C2)C(=O)N(C)C3 C(CC(=O)N1CC2CC1C(F)(F)C2)(C(F)(F)F)NC(C(CCCC)C)=O C12(OC(C(COC)(C)OC)=O)CCC1CN(C(c1cc(N)ccc1F)=O)C2.C(C)O c1(CC(=O)N(C2CCCCC2N(C)C(C2CC3C=CC2O3)=O)C)sc(O)nc1O N1(C(CCC)=O)CC2CC1CCN2C(=O)COCc1cccnc1 C12(NC(c3ccc(C)nc3)=O)CCC1CN(C(C1CCC(C3CC3)C1)=O)C2 C12(C(=O)NC(C3CCN(C(=O)Cc4cccnc4)CC3)(C)C)CCN(CC1)C2 c1(C(=O)NCC2C(CNC(c3sc(C)c(C)c3C)=O)C2)cc(O)cc([N+](=O)[O-])c1 N1(C(CC(C=C)(C)C)=O)CCC2(C1)CN(C(C1CCCCS1)=O)CCO2 c1(C(N2CC3CCCC(C2)N3C(c2cnns2)=O)=O)c(F)cccc1[N+](=O)[O-] c1(C(=O)NCC=CCNC(C(=O)NCC)=O)cn(C2CN(CC)C2)nn1 Cc1ccccc1-c1csc(C(C)(CCCO)N2CCSCC2)n1 Cc1cc(C(=O)N(C)CCOCCCN(C)C(c2cc(F)n(C)n2)=O)cn1C Cc1c(C(=O)NCC2CC2NC(C2(Cl)CC23CCC3)=O)cncc1Br CC1C(NC(=O)CC2CSCCS2)CCN1C(c1c[nH]c(=O)cn1)=O c1(C(C)NCC=C)ccc(-c2cnc(O)[nH]2)c(F)c1F C1(CC)CCC(C)CN1C(=O)C(C)CN(C(=O)CC1(C#N)CC1)C CC1(C)C=C(C(=O)NCC2(C)CCCN2C(=O)Cc2cc(Br)cnc2F)C1 N1(C(c2csc(C)n2)C(=O)NCC(=O)OC)CCCC(CC(C)C)(CO)C1 c1(CC(=O)NC(CNC(C(CC)NC(C)=O)=O)COC)ccc(O)c(OC)c1 C1(C(N(CCN(C(=O)CC2CCCCN2C)C(C)C)C)=O)CC2CCC(C1)C2 Cc1cnccc1C=CC(N1CC(O)(CCNC(=O)C(n2cc(C)cn2)C)C1)=O Fc1ccc2c(CNC3(c4cncc(Br)c4)CCC3)n[nH]c2c1F CC(C)C(C(=O)OC(C)(C)C)NCCCC1CCCCN1Cc1cnccn1 C1(C#N)(SC)CN(C(=O)CC(CNC(C2CC(CF)C2)=O)C2CCC2)C1 CCCCC(O)C(=O)NC1C=CCCC1C(=O)NC1CC2CC2C1 CCC(CC)(C(=O)NC1C=CC(C(=O)NCC(O)CCC2CC2)C1)OC C1(NC(C(N2C(C(C)(C)OC)CCC2)c2nocc2C)=O)CCC(F)(F)CC1 Nc1cccc(C(=O)NCC2(NC(=O)CCCc3cnn[nH]3)CCCCC2)c1 C(=O)(C(CCF)NC(=O)C(C)CSC)NC(CCC)C1CCCC1 CCCCC(O)C(=O)NCCOC1CN(C(c2cncnc2C)=O)C1 N1(C(c2cnn(C3CCOCC3)c2)=O)CCN(C(C2SCCS2)=O)C(CF)C1 c1(CCCC)n[nH]c(=NCC2CCCC2NC(=O)CCOCCOC)s1 Cc1cccc(C(N2CCC(N(C(=O)C(Cc3cccc(Cl)c3)=NO)C)C2)=O)n1 C1(NC(C2(c3ncc(F)cn3)CC2)=O)CN(C(=O)C(O)C(F)F)CCC12CCC2 C12(CCOCC1)C(=O)N2.c1(COCCSCC2CCC2)cn(C(F)F)nn1 c1(OC)ccccc1C(N1CCCC1CN(C(=O)Cc1ccnc(C)c1)C1CC1)=O N1(CC)CCCC(N(CC(C)(C)CC(c2ccccc2)C)C(=O)NC(C)(C)C)C1 c1(C(C)(C)C)ccc(C(=O)NCC(O)CCNC(=O)CC2CCOC2=O)cn1 N1(C(CC(=C)Br)=O)CCN(C(=O)C2=COCC2)C(c2cn[nH]c2)C1 c1(C(=O)NCCCC2(NC(C3(C(=O)NC4CC4)CC3)=O)CC2)cc2cccnn2n1 N1(C(Cn2c(C)cnc2)=O)CC2=C(C1)CN(C(c1ccsc1C(F)F)=O)C2 C(CCC(C(=O)NC1(c2ncsn2)CC1)NC(C1CCC(O)CN1C)=O)OC c1(OCCCC(=O)N(C(C)C2CC2)CCC2CCCNC2)ccccc1F c1(C(=O)NCC(CC)NC(=O)C(c2cccc(C)c2)(C)C)cc2n(c1)CCC2 Cc1cc(C(=O)N(C2CCCN(C(C3(C)CCCCO3)=O)C2)C)nn1C N1(C(=O)C(O)Cc2ccccc2)CCC2(CC1)OCC1CC21 N1(C(CCOC(C)=O)=O)CCC(CCN(C(=O)Cc2cc(Cl)n(C)n2)C)CC1 N1(C(c2c(CC)nns2)=O)CC(NC(c2ocnc2CC)=O)CC1(C)COC CCCCCC(C)(CC)C(=O)N(C(C)CNC(=O)CN1CCCC1=O)CC c1(C(N2CC3COCC3C2)=O)cc2c(-c3cccc4ccoc34)cccc2[nH]1 C1(C(N(C2CC2)CC2N(C(c3n[nH]c(C)c3N)=O)CCC2)=O)CCCCC1(C)C c1(NC(C2CC(F)CN(c3ncnc4sccc34)C2)=O)c(F)c(F)c(Br)c(F)c1F c1(NC(c2ccn(CCC)n2)c2nnnn2C2CCC2)c(F)cc(Cl)cc1Br c1(C(N2CC(CC(CNC(CCC3C(C)C3)=O)(C)C)C2)=O)c(Cl)cncc1Cl c12cn(C)nc1NC2=O.C1(NCC)CCN(C(C2CC(O)(COC)C2)=O)C1 N1(c2c(C)cc(CC)cc2C)CCC2(CCCN(C(C)=O)C2)C1 c1(NC(C)=O)ncc(S(=O)(=O)N2CCOC(C(=O)NCC34CC(C3)C4)C2)s1 CCCC(C(=O)NCC1CCCN(C(c2cnccc2COC)=O)C1)OCC CC1(C)CCC(C#N)N1C(=O)CC(Cc1ccccc1)n1cnnn1.C1CO1 C1(C(=O)NCCCCN(C(CC2CC(=C)C2)=O)C)CCCCO1 CC(C)CC(Cc1ccccc1)C(=O)NC(Cc1cncn1C)C(=O)O c1(C(N(C(CC)C2CC2)C)=O)conc1C(C)NC(=O)CCCSC1CCC1 N1(C(C2CC(CC)C2)=O)CCN(C(=O)C(CC)CCOC)CC1C C(CCCC(=O)NC1COCCC1NC(=O)COCCc1cccs1)SC Cc1cc(N2CCC(C(=O)NOC(C)C)CC2)nc(N(C)CP(C)(C)=O)n1 C(=O)(C1CCCn2cnnc21)NC(C)CCNC(c1c[nH]cc1C1CC1)=O C=CCC(F)(F)C(=O)N1CC(n2cc(C(N3CCCC3)C3CC3)nn2)C(O)C1 N1(C(COC(C)(C)C)=O)CCC2(CC1)CN(C(=O)CCC1NC(=O)NC1=O)C2 N1(C(C2CC(=C)C2)=O)CC(NC(C2(CC(F)F)CC2)=O)CC(F)C1 N1(C(C2C(C(=O)OC)CCC2)=O)CC2CN(C(c3ccsc3Cl)=O)CC2C1 N1(C(c2c(N(C(C)C)C)cccc2)=O)CCN(C(=O)CC2CC2)C(CCN(C)C)C1 c1(OC)ccncc1C(=O)NC1CC(C)N(C(c2sccc2CO)=O)C1 c1(OC)c(F)ccc2[nH]c(C(=O)NCCN(C(=O)C(C)O)C)cc12 Cc1cc(C(=O)NCC2CCN(C(=O)CN(C)C)C2)cnc1O c1(COC)cccc(C(=O)N(C)CC2CCN(C(=O)C(C)N3CCC3)C2)n1 O=C(N=c1ccnc2[nH][nH]cc1-2)C1CC(F)CN1Cc1ncnc2sc(Br)cc12 c1(C(C)C(=O)NC2CN(C(=O)C=CC3CCOC3)CC2C)c(F)cccc1F C1(N=[N+]=[N-])(C(N2C(C#C)CCC2)=O)CCN(C(c2ccc(CC)nc2)=O)C1 C12(C(N(C)CC3(O)CCN(C(c4cn(CCC)nn4)=O)C3)=O)CCCC(C1)OC2 C(C)(C)(CC(F)C(=O)NC(CO)C1(C)CC1)NC(C(C)n1ccnn1)=O C(=O)(C1=CCCCC1C)NC1(C(=O)Nc2nc(C)nc(O)c2)CCC1 n1(Cc2cn(CCOCCNC(CCn3ccc(C)n3)=O)nn2)cccnc1=O C(=O)(CC(C)(C)C)NCC(CN(C(Cc1nc(CC)sc1)=O)C)C Cc1[nH]nc2c1CCC(C(N1CC3COCC(C1)C3NC(=O)C1=CCCC1)=O)C2 CCC(CCC(=O)NC(COC)CCO)NC(=O)C(C)CSC N1(C(C(CO)OC)=O)CC(=O)CC1C(=O)NC(CCO)C1CCC1 N1(C(c2cccc(C#C)n2)C(=O)NCC)CCC2(CC1)CC(N(C)C)CO2 N1(C(C2CC(CC)(CC)C2)=O)CC2CCCC2(NC(=O)Cc2csc(Cl)n2)C1 C#CC1(O)CCN(C(=NCC2C(C)(C)C2(F)F)NCC(F)F)C1 c1(C(=O)NCC(CC(C)C)NC(c2occ(C)c2)=O)ccc(Cl)c2occc12 C(=O)(C1=CCCCC1)NCC(N1C(CNC(=O)Cn2cncn2)CCC1)=O C1(CNC(C(CC)COC)=O)CC2(CC(NC(=O)Cc3cccc(Cl)c3Cl)C2)C1 C1(C(N2CC(C(=O)NCCC3CCCCC3O)(SC)C2)=O)CC12CCCCC2 C#CC1(C(=O)NC(C)C(C(C)C)NC(c2coc(N(C)C)n2)=O)CCCC1 c1(CNC(CC2(OC)CC2)=O)cnn2c1CN(C(=O)CC1(OC)CCCC1)CC2 C=C(C)C1CN(C(C2C3CCC(C3)N2C(=O)CC2(NC(C)=O)CC2)=O)CCO1 C(=O)(C1=CCCC1)NC(C)Cn1cc(CNC(=O)C(F)CC2CCCC2)nn1 C1(NCc2ccc(OC(F)(F)F)cc2Cl)CCCCC12CCCC2 C(=O)(CC(C)C(C)C(C)C)N1CC2CC(Nc3cc(CCC)nc(Cl)n3)C2C1 c1(NC(C(=O)Nc2nc(COC)nc(O)c2)=O)cc(NC(C)=O)cc(C)c1 c1(NC2CCN(C(C3CCCO3)=O)C2)ccc([N+](=O)[O-])c2cccnc12 c1(C(N2CCC(C)(NC(C(C(CC)C)O)=O)CC2)=O)c(OC)cc(OC)cc1N N#Cc1ccc2[nH]cc(C(=O)NC3CCN(C(=O)CC4CCCC(=O)N4)C3)c2c1 c1(C(N2CCCC(CCNC(CCCC)=O)CC2)=O)cnc2nccnc2c1 O=C(C1CCCn2cnnc21)NCC1CCCN1C(=O)CCCOC1CCOCC1 c1(C(N2CC(N(C)C(C3CCCCN3C)=O)C2)=O)cc2c(s1)CCSC2 N1(C(Cn2ncc(C)c2)=O)CC2CCC(C(N3CC4C(C(N)=O)C4C3)=O)(C2)C1 C1(CNC(C=C(CC)C)=O)CCCCCN1C(=O)C(C)Oc1ccccn1 Cc1cc(C)c(C(N2CC3CC3(NC(=O)CCC3CC(C)(C)CO3)C2)=O)cc1N c1(NC(C(CCCOC)NC(=O)Cc2cncn2C)=O)cccc(C#N)c1C C1(C(=O)NCC2CC(C)(C)OCC2)CCN(C(=O)CCCC2CCC2)C(C)(C)C1 C1(C(=O)NC(C)CCCNC(=O)C#CCN(C)C)COCC(C)O1 c1(CN2C(C3CCN(C(CC(C=C)C)=O)C3)CCCC2)cnc2ccc(F)cc2c1 c1(OC)ccc(C(=O)NC2CCN(C(c3cn(C4CC4)cn3)=O)C2)c2sccc12 c1(CNc2cc(NCC3N(CC)CCCC3)ncn2)cc(F)c(Cl)cc1C CCC1=NOC(CC(N2CCC(CCNC(c3nc[nH]c3C(C)(C)C)=O)C2)=O)C1 C(c1nc(C)cs1)=CC(=O)NC(CNC(c1c(CC)c[nH]n1)=O)(C)CO C1(NC(=O)Cc2ccsn2)CCCN(C(=O)CCc2cccc(Cl)c2)CC1F C(=O)(C(C)C(O)C(C)C)N1CCC(CC(C)NC(C23CCCN2CCC3)=O)CC1 Cc1sc2cc(F)ccc2c1CNCc1ccccc1I N1(C(COCCCC)=O)C2CCC1CN(C(=O)CC(C)(O)CCC)C2 c1(C(N2CC(NC(C3=C(SC)CCCC3)=O)C2)=O)cccc2c1ccn2C Cc1cc(=NC2CCn3ncnc3C2)[nH]c(=NCCSCCCO)[nH]1 Cc1c(C(=O)NCC2CCCCN2C(C2CC2C(=O)NCCO)=O)cnn1C c1(CC(C)C)ccc(C=CC(N2CCN(C)CC2CNC(c2cnc[nH]2)=O)=O)cc1 C1(CNC(C(C)OCCOCC)=O)CCCN(C(=O)CNC=O)C1 CC(C)CC(O)C(=O)N1CC(CO)CC(C)C1.N12CCCCC1(C)C(=O)NOCC2 c1(OC)ccnc(C(=O)NCC2(O)CN(C(C3(c4cc[nH]n4)CCC3)=O)C2)c1C C(=O)(CCC(=C)C)NCCCOCCCNC(C1C(CC#C)CCO1)=O O(NC(=O)C(C)(C1CCC1)NC(=O)C=C1CCOCC1)CCN(C)C C1(C(=O)NCCN(CCC)C(c2cc3scnc3[nH]2)=O)CCCC1S(C)(=O)=O C1(N(C(CN(C)CC)=O)C)CCCCN(C(C2CCC(C(F)(F)F)CC2)=O)C1 c1(C(=O)NCC(C)(CO)NC(c2cc(C)ns2)=O)cc(S(C)(=O)=O)c(C)o1 C(=O)(C1=CC2CCC1C2)NC1(C)CN(C(c2c(C)[nH]c(C#N)c2)=O)C1 c1(C(=O)NCCOCCNC(C2CC2F)=O)ccnc(CO)c1 N1(C(c2c(C)n(CCO)cc2)=O)CCCN(C(=O)COCC(F)(F)F)CC1 N(C1CCc2cc(F)ccc21)c1nnc(CCCC)n1Cc1cccs1 C(=O)(C#CC1CCOCC1)N1CCCC(O)(CNC(c2n(C)ccc2)=O)C1 C1(CNC(Cn2nc(C)c(Cl)c2)=O)CC2(CCN(C(C3(F)CCOC3)=O)CC2)C1 C1(NC(=O)NC2CC(Nc3cccc(F)c3)C2)CCCN(C(C)=O)C1.C(N)=O c1(C(=O)NC(C)CN(C)C(c2csnn2)=O)ccc(C(F)(F)F)cc1C(F)F C1(NC(=O)C=Cc2cccc(O)c2)CCN(C(=O)C(O)C2CCC2)C12CCC2 C(CC(=O)NCC(C)C(C)C)(CC(C)C)NC(c1ccc(C)c(C)c1)=O N1(C(C2CCC(C)S2)=O)CCCC2(C1)CN(C(c1cncc(F)c1)=O)C2 N1(C(c2c(CC)cncc2)=O)CC(C)C(NC(c2cn[nH]c2)=O)C(C)C1 CC(CCCNC(c1cn(Cc2ncccn2)nn1)=O)NC(c1csc(Cl)c1)=O C12(C(=O)OC)CCCC1(C(=O)NCC1CC1)C2.c12coc(n1)CNC2=O.C(=O)CF C1(C)(C(=O)NCCOC(C)=O)CCCN(C(C2CC23CNC3)=O)C1 c1(CC(=O)NC2CCC(F)(CNC(CCc3cn(C)nc3)=O)C2)ccc(F)c(F)c1 c1(OCC)cncc(C(N2CCC(CC(=O)N(C)Cc3ccccc3)C2)=O)c1 C(=O)(CCCC(=O)NCC(C(C)C)NC(C1NC(=O)OC1C)=O)OCC c1(N(CCCC)CCCC)cc(-c2cccn2C)cc(C#N)c1 C1(C(N2C(CN(C(C)=O)C)CCC2)=O)Cn2c(C)nnc2CN1C C1(C)(N(C)CCNC(C2(C(=O)O)CC=CCC2)=O)CCCCC1 C12(CNC(COCCCOC)=O)CCC1CN(C(=O)CNC(=O)CCCCO)C2 c1(C(=O)NCCOCCNC(C2(C)CC2(F)F)=O)ccc(Br)cc1O c1(CC(=O)NCC2CCCCN(C(=O)COCC3CC3)C2)c(Cl)cccc1Br Cc1cc(Cl)c(C(N2CCC(C)(CNC(=O)Cn3ccsc3=N)C2)=O)s1 c1(C(=O)NC(CC(C)C)C(=O)NCCCCC(F)(F)F)c[nH]c2cccnc12 c1(-c2c(-c3cc(-c4n(CCCCC=C)ccn4)n[nH]3)csn2)ccc(OC)cc1 O=C(Cn1cc(-c2ccccn2)nn1)NNC(=O)c1coc(C2CC2)n1 c1(CC)ccc(C(=O)NCC(=C)CCNC(=O)C(O)Cn2cncn2)cc1CC c1(OCC)ccc(OC(C)C(N2CCC(NCc3nc(CO)cs3)CC2)=O)cc1 N1(C(C23N(C(COCC)=O)CCC2C3)=O)CCC(C#N)(OCC)C1 c1(C(=O)NCC(C2CCCC2)NC(C2CC2C2CC2)=O)ccnc2cc[nH]c12 C1(CC)(CC)CC(NC(C2(C(=O)NC)CC2)=O)CN1C(=O)C(C)SC1CC1 Cc1cc(C(N2CCCC(C(=O)NCCOCCON)C2)=O)cc(C)c1Br CN(NC(=O)C(C)(C)CC1CC(=O)NC1)C1CC1 c1(N(CC#CC)NC2CCNCC2)ncnc2cc[nH]c12.c1(C)c(C)cccc1Br C(=O)(CC1=CCCC1)N1CCC(C2N(C(C(C)OCC#C)=O)CC2)CC1 c1(CCn2cc(C(=O)NC(C)C3CC3)nn2)ccc(OCC2CCCO2)c(F)c1 c1(C(=O)NC(C)C(C)NC(c2onc3ccccc23)=O)cc2nc[nH]c2cc1N C1(CNC(CC=C(C)C)=O)CN(C(=O)CCOCC2CCCC2)CCC12CCC2 CC1CCCCC1(CNC(c1cnc(C(C)(C)C)nc1)=O)NC(=O)C=C(Cl)Cl C1(OCC)C(C(N2CC(C(C)NC(=O)Cc3ccoc3)C2)=O)C1C O(NC(=O)Cn1ccnc1)CC(=O)NC(COC)COC Cc1ccc(NC(=O)C(N2CCN(C(=O)C(C)(F)F)C3CC23)=O)c(Br)c1 CC1(C(N2CC3CC3(CNC(c3ccnnc3O)=O)C2)=O)CCNC1=O c1(C(C)NC(N(C)CC)=O)noc(Cc2conc2C(F)(F)F)n1 c1(-n2c(-c3n(CCC)nc(C)c3)nc(-c3cnn(CC)c3)n2)cccc(Cl)c1C N1(C(C(C)=CC)=O)CC=C(CCNC(=O)C(C)C(C)O)CC1 N1(C(c2cnc(OCC)s2)=O)CC=CC(NC(=O)C=Cc2cccs2)C1 N1(C(COC(CC)(C)C)=O)CC2CC(NC(=O)CC3CN4CCC3CC4)C2C1 c1(OCC)c(CNC(Cc2cccs2)CO)cc(C)cc1Cl c1(C(N2CCN(CC(=O)NCC(CC)N(C)C)CC2)=O)cccc([N+](=O)[O-])c1OC C(C)(C(C(=O)N1CC(CC(F)(F)F)C1)NC(=O)C=CC(F)(F)F)OC N1(CC(N2C(C3(NC(c4c(C)cno4)=O)CC3)CCC2)=O)CCC(CO)CC1 CCCCC(CNC(=O)CCc1ccccc1OC)NC(C1CC(C)OC1C)=O CCCC(CCc1ccccc1)C(=O)N(CCNC(=O)C=CC=C(C)C)C(C)C C12(C(=O)NC3(CC)CC3)CCCCC1CS(=O)(=O)C2.C12(CC1)C(=O)NC2 C1(CC)CC(C)CN(C(C2CCOC2CNC(c2ccsn2)=O)=O)C1 C(c1cccc2cccnc12)=CC(N1CC(NC(C2C(CCC)C2)=O)C(C)C1)=O N1(C(Cc2cccc(C3CC3)c2)=O)CCN(C(=O)CSCCCC)C(C)CC1C C#CCC(C(=O)NCC(C)(C)CNC(=O)C(CC)c1ccccc1)C1CC1 c1(-c2c(C(=O)NC(C(=O)OC)C)ccnc2)ccc(F)cc1C(=O)O CCC([O-])C(C)(F)F.N1C(NC(C)CCC(C)(C)C)=NCCC2(CC2(C)C)C1 N1(C(C2(SC)CC2)=O)CC(C2CCCN(C(C3CCC4(C3)CC4(F)F)=O)C2)C1 C1C(CC(C)C)C(=O)N1.c1(C(CF)N)ccc(C)cc1.n1(CCCC)nnnc1CC Cc1cc(C(=O)NCC2COCCN2C(c2cc(C(C)C)sn2)=O)sc1Cl N1(C(C2CCC(OC)CC2)=O)CC2CC1CC2NC(c1csnc1C1CC1)=O CCCCC(CCCC)NC(C1(C)CC(O)CN1C(=O)C=C(Cl)Cl)=O N1(C(C(C(C)C)C)=O)CC2(CC(NC(c3cccc(O)c3Cl)=O)CO2)C1 C1(C(=O)NC(CNC(Cc2cccc(NC(C)=O)c2)=O)CO)CCCS(=O)(=O)C1 N1(C(CCCC#C)=O)CCN(C)CC1CNC(C1COC(=O)N1)=O C1(CN(CC(=O)Nc2ccc(OC)cc2C)C)CCc2ccccc2O1 Cc1ccc(NC(=O)NC2CC(=O)N(CC3CCC3)C2)cc1I C1(NC(C2C(C(C)OC)C2)=O)CC2(C(=O)N(C34CC(C3)C4)C)COC1C2 C(=O)(CC(C)(C)C(=O)OC)NC(C1CCCC1)CNC(C(C)=C(CC)C)=O N#Cc1c(N(C2CC3CC2CN3)C(=O)Cc2ccc(F)cc2Br)cc(Br)cc1F C1(CC(N)=O)CCN1C(=O)C(=O)NCCOCCCC(=O)OC(C)(C)C N1(C(C2(C)N(C(c3cncc(C)n3)=O)CC=C2)=O)CCC(O)C(C)(C)C1 Cc1cc(Cl)c(C(=O)NC(Cc2cn(-c3ccc(Cl)cn3)nn2)CC(=O)O)s1 n1(CC)cccc1C(N(CC(=O)NCC(C)C)CCc1cn(C)cn1)=O c1(CC(N2CC(NC(C(F)(F)C3(OC)CCC3)=O)C2)=O)ccc(F)cc1Br C1(C)(NC(C2C(COC)(COC)C2)=O)CCCN(C(c2cccc(N)c2F)=O)C1 C1(C(N2CCN(CCOCC)CC2)=O)CC(=O)N(C)C1c1cnn(C)c1 C12(C(=O)NC(C)CCCCNC(=O)C(C)(C)C3CCCCO3)CC3CC1C2C3O n1(CC(=O)NCC(C)=CC(N2CCC(CC(C)(C)C)C2)=O)ncccc1=O Cc1nn(C)c(C)c1C(=O)NC1CCCC1C(=O)Nc1nnc(C(C)C)s1 C1(NC(C(C=C)(F)F)=O)CCN(C(c2ccnn2CCCC)=O)CC1C(N)=O N1(C(c2ccc(CC)c(N)c2)=O)CC(C)CN(C(C2(O)CCCCC2)=O)CC1C C(=O)(C#CC(C)(C)CNC(C1CCC2(CC1)CC2)=O)N(C)CC1(CF)CCC1 C(CC(C)(C)C(=O)NCCCOCC(=O)NC(C(O)CO)C1CC1)OC C1(C(N2CCC(C(=O)N(C)C)C2)=O)CC(F)CN(C(c2ccc3c(c2)CC3)=O)C1 C(C(C(F)(F)F)N1CCN(C(C2CCC2(C)C)=O)CC1)NC(C(CC)=CC)=O c1(CC(N2C(CCC(N3CCCC(C(=O)OC)C3)=O)CCC2)=O)cc(Br)ccc1Cl N1(CC)CC2CCC(CN(c3ccc(Cc4cccc(F)c4)s3)C)C2C1 c1(N2CCC(COC)C2)nc(=NC(C)(COC)COC)[nH]c2c(C)nn(C)c12 N1(C(C(C)(F)F)=O)CC2CCC1C1CN(C(=O)CN=c3ccc(C#N)c[nH]3)CC21 N1(C(CC)=O)CCOC2(CCC(C(=O)NS(=O)(=O)C)CC2)C1 C=CCC(CNC(=O)C(C(C)C)SC)C(=O)NCCN(C(C)C)C(C)C C(=O)(CC1COCc2ccccc21)N(CC(C)N(C)C(c1cc(Cl)c[nH]1)=O)C Nc1nonc1C(=O)NCC1(CCNC(C2CC=CCO2)=O)CC1 C(C(COC(=O)C(C)(C)C)C(F)(F)F)OCCOC(C)=O.c1(C(=O)O)nc(O)sc1C C(=O)(C1CCc2ccccc21)Nc1n(-c2ccc(C)cc2)c2c(n1)cccc2 c1(C(C)NC2CC3CC3C2)cccc(N=[N+]=[N-])c1 Cc1ccc(CO)cc1NC(=O)C(=O)NCCOc1cnn(C2CCCCC2)c1 c1(NC(C2(CCC=C)CC2)=O)cc(N2CCN(C(c3ccno3)=O)CC2)ccn1 N1(C(c2n(C=C)nnc2)=O)CCCCCCC1C(=O)NC(c1cn(C)nn1)C N1(C(CCn2cc(-c3ccc(N)c(Cl)c3)nn2)=O)CCN2C(=O)OCC2C1 Cc1nc2cc(Cl)cc(C(N3CCCC(C)(CNC(=O)C=CC4CC4)C3)=O)c2[nH]1 C(CC(C)C(=O)NCC1CCCN1C(=O)CN1C(=O)CCC1=O)=CCC Cc1cccc2c1OC(C(N1CCC3CN(C(c4nc(Cl)cs4)=O)CCC13)=O)C2 N1(C(C=C2CCC(C)CC2)=O)C2CCC1CN(C(c1cc(C(N)=O)[nH]n1)=O)CC2 c1(C(=O)NC(C(C(C)C)C)CNC(c2cnc[nH]2)=O)cc(S(C)(=O)=O)ccc1O Fc1ccc(-c2ccc(Nc3cc(Br)cnc3F)cn2)c(F)c1 C(c1c(C)nn(C)c1Cl)=CC(=O)NC1CC(NC(C2(CSC)CCC2)=O)C1 CCCC(C)CC(=O)N1CC(C2(NC(=O)C(c3nc(C)cs3)C)CC2)C1 c1(OC)ccc(C=CC(=O)NCC(CNC(=O)C2=CCCC2C)OC)cc1O N1(C(CC(CC)C)=O)CCCC(C)(C(=O)N(C)Cc2cc[nH]n2)C1 O=C1CC(CC(=O)N2CCOC(CCNC(C3CCCC4CC34)=O)C2)=NN1 C12(C(N3CC4N(C(c5ncn(C)c5)=O)C(CC4)C3)=O)CCCN1S(=O)(=O)CC2 C1(NC(C2CC2(Cl)Cl)=O)COCCN(C(C2CC3(CCC3)CO2)=O)C1 N1(NC(C2CCN(C(C3C(C(=O)OC)C3)=O)CC2O)=O)CCN2C(=O)NCC2C1 C#CCC(O)C(=O)N(C(C)CCNC(c1ccc(-n2[nH]c(O)nc2=O)cc1)=O)C C1(CNC(C2CCN(CC)C2)=O)CN(C(c2ccnc(S)c2)=O)CC12CC2 C1(C2(N)CCC2)(C(=O)NCC(CC#N)(F)F)CC1 CC1CCCN(C(=O)C(C2CCN(C(c3ccc(C4CC4)o3)=O)C2)F)C1 CCCC(C(=O)N(CC(C)NC(C12CCCN(CC1)C2)=O)C)S(N)(=O)=O N1(C(C(CC)n2ccnc2)=O)CC(CNC(=O)CCc2ncc[nH]2)CC1(C)C C1(C(N2CCOCC(NC(c3cccc(C)c3C)=O)C2)=O)CCCC2CCCN12 C#CC(CC)(CC)NC(C1CC1CNC(=O)CC1CCC(C)CO1)=O C1(O)(CN(C)C(C2(C)CC2C(F)(F)F)=O)CCN(C(c2ccn(C)c2)=O)CC1 CC1(C)CN(C(C2CCC(=O)N2)=O)CCC1C(=O)NC1CCCCC1 CCC(CC)(CCC(=O)N1CCC1COC1CCCCN1)[N+](=O)[O-] c1(C(N2C(CNC(C3CCOCC3)=O)CC(OC)C2)=O)cnn2c1OCC2 c1(N2CCCC(CNC(C(CCC)(C)O)=O)CC2)ncnc2[nH]c([N+](=O)[O-])cc12 N1(C(C=CC(C)NC(=O)CN2CCCC2)=O)CCC(O)CC1C N1(C(c2nc(C)oc2C)=O)CCC(C2(NC(=O)CC3(C)CC3)CC2)CC1 c1(CN(C)C(=O)NCC2C(C)(C)C2(F)F)c(Br)c(C(F)(F)F)nn1C Fc1cc(CNc2cc(C(F)(F)F)ccc2F)c2ncoc2c1 n1(C(C(=O)N(CC(=O)N(CCCOC)C)CCC)C)nc(C)cc1C N1(CC)OCC(NC(=O)CC2CC(NC(=O)NC(C)(C)C)C2(C)C)C1=O c1(C(N2CCCC(O)(CNC(CCNC(C)=O)=O)C2)=O)ccc(O)c(C)c1C CN(C)NC(=O)CCC(=O)N1CCC1(C)CC(=O)NOCC1(C)CCC1 C1(Nc2ccc(CC)s2)CCCN(C(=O)C(=O)N(C)C)C1C(=O)OC c1(CC)cc(C(N2C3CCC(C3)C2CNC(=O)C(C)CO)=O)cc(N)c1 CCC(CC)CCC(=O)NCC1CN(C(c2ccc(O)c(CO)c2)=O)CC1C c1(CC)cn2c(n1)CCC(C(N1CCN(C(c3cc(C4CC4)cs3)=O)CC1)=O)C2 C1(CCNC(C2CC(C)=C(C)CC2)=O)CC(N=c2nc(C(C)C)[nH]s2)C1 N1(C(C2C(OC)C2)=O)C2CCC1CN(C(C1CN3CCCC3CO1)=O)C2 C1(C(N(CC(=O)NC2CC2)CC2CSCCO2)=O)(CO)CCCCO1 C(=O)(CCCC(=O)N(C)C)NC1CCC(CNC(c2cc(C)oc2C)=O)CC1 Cc1cc(C(=O)N(C)CC2CC(F)CN2C(=O)CC2CCC(=O)N2C)cnc1O C1(C(=O)NC(COC)(C)C(N)=O)CCC2(CC2)N1C(=O)Cc1cc[nH]n1 CN1CCCC(C(N2CC(O)CC2C(=O)NCc2nncn2C)=O)C1 N1(C(c2cc(CC)sn2)=O)CC2CCC1CN(C(=O)C(C1CC(F)(F)C1)=O)C2 C(CCSC)(C(C(=O)NCCCF)N1CCCCC1C1CCCC1)OC C1(NC(C(C2CCCC2)OCC)=O)(CNC(=O)CN(C(=O)COC)C)CCOC1 C1(NC(c2ccnc(-c3cc[nH]n3)c2)=O)CCCCN(C(C2CCCC(F)C2)=O)C1 c1(C(=O)NCC2N(CC(C)C)CCCC2)cc(Br)cc2c1OCCC2=O Cc1cc(N2CCC2CNC(c2nc(C(F)(F)F)sc2C)=O)ncn1 c1(OC)nc(-c2cncnc2)ccc1C(=O)N(CC(O)C(C)C)C C1(NC(C=CCCC)=O)(CF)CCN(C(c2ccc(SCCC)nc2)=O)C1 C1(NC(c2ccc(NC(c3cc4n(n3)CCC4)=O)nc2)=O)CCCCC1(F)F C(=O)(C(C)C(C)NC(=O)C(C)OCCN(C)C)NC(CC#C)C Cc1cccc(C(N2CC(NC(c3cccc(-c4ccco4)c3)=O)C(F)C2)=O)c1 C1(C)(CNC(CCC#CC)=O)COCCN(C(c2cnc(N(C)C)nc2)=O)C1 c12ccc(cc1)CC(=O)NCC(C)CS2.c1(C(=O)NCC)cnccc1C C(CCC(=O)N(C1CCCCC1)CCNC(=O)C(C)c1cc[nH]n1)SC C1(OC)COCCC1NC(=O)CCN(C(c1cc(C(C)(C)C)on1)=O)C1CC1 c1(C(N2CC(NC(c3c(C)c(Cl)cnc3)=O)C(F)CC2)=O)nccc2occc12 C12(NC(C(C)C#N)=O)CCCC1CN(C(c1ccc(OCC(F)F)cc1)=O)C2 c1(C(N2CCC(O)(CNC(C(CCC#C)O)=O)C2)=O)ncnc2ccsc12 CCC(CCC(=O)N1CC(O)C(O)C1CC)NC(c1cn(C(C)C)nc1C)=O c1(C(N(C)CCNC(c2nonc2N)=O)=O)cncc2ccccc12 C1(NC(=O)COCCCF)CCN(C(=O)Cc2ccco2)C1c1ccccc1 Cc1cc(N(c2ccccc2)CC(=O)NC2CC3(CCOC3)C2)cc(C)c1Cl CC1CC(NC(C2CCCN2C)=O)CN(C(c2cn(C3COC3)nn2)=O)C1 C1(CN2CC(C3CCCN3)C2)CCCOCC1.CC(CC1CCCCC1)C(=O)NC C(=O)(C(F)C(=O)N(C1CCCC1)CCCNC(c1cncc(F)n1)=O)OCC c1(CC)c(N2CCC(CNC(=O)CS(=O)CC)C2)nc(C)nc1Cl CC1CN(C(c2cscc2F)=O)CC(C)N1C(c1c(N)sc2c1CCC2)=O C(C(C)(CC(=O)N(C)CCN(C(=O)Cc1cnns1)C)C(F)(F)F)N(C)C c1(-c2nc(CN(C(=O)NC(C)Cc3nc[nH]n3)CC)on2)ccc(C)cc1 C1(NC(c2ccc(C)n2C)=O)CN(C(=O)C(F)(F)c2cnn(C)c2)CC12CC2 C12(OC)CCC1CN(C(=O)CCCCNC(=O)CCCCN(C)C)C2 Cc1cnc(C(=O)N(CC(C)NC(=O)C(Cc2ccccc2)C2CC2)C)c(F)c1 CCN=C(NCc1cc(C(F)(F)F)no1)N1CCC2(CCCCN2C2CC2)C1 C1(CNC(C(CC)OC)=O)COCCN1C(c1csc(N2CCOCC2=O)n1)=O C1(CNC(CCc2ccc(N)cn2)=O)CCCN(C(C23CC4CC2C3C4)=O)CC1 CCC(C)C(C)C(=O)NCCC1CCN(C(=O)Cc2cncn2C)CC1 c1(SCC)cc(=NC(=O)c2sc(NC(C3(F)CCCCC3(F)F)=O)nc2Cl)[nH][nH]1 c1(C(=O)NCCC2CN(C(CN(C(C)=O)C)=O)CC(C)O2)ccn2cnnc2c1 C=CCCCCCCCC(=O)N1CCC(NC(=O)CCn2cccc2)CC1C c1(CNCc2cc(OC)ns2)cc2ccc(F)cc2nc1Cl Cc1cc(Br)ccc1-c1noc(NC(=O)NCC2(CC3CCC3)CC2)n1 C1(NC(c2c(C)n(C)cn2)=O)CCC2(CC1)CN(C(C1CNC(=O)N1)=O)CCO2 CC1(NC(C2C(C(F)F)C2(C)C)=O)CC(NC(=O)CSCC2CCCO2)C1 c1(C(=O)NC2CC3(C(NC(=O)COC4CC=CC4)C3)C2)cccc2[nH]cc(Cl)c12 C1(C(CC2CC2)(C)C)CCCN(C(=O)Cc2ccn(C(C)C(=O)N)n2)C1.C1CC1 C1(C(N2CCCCC2c2cn(CCCF)nn2)=O)C(Cl)(Cl)C12CC2 CC1(C)COC(CCC(=O)NCC2(NC(=O)CCCc3ccc(F)cc3)CC2)C1 N1(C(C(CCCC)CC)=O)CCC2(CCCCN(C(c3cnnc(O)c3)=O)C2)C1 C=Cc1ccc(CNC(C2N(C(=O)CC34CCCC3C4)CCC2(C)C)=O)cc1 c1(CNC(C(C)NC(c2ccoc2)=O)=O)ccc(C(=O)Nc2ccsc2)nc1 C1(NC(C2CC(C(=O)OC)C2)=O)C=CCCC1C(=O)N(CC(C)(F)F)C c1(C(N2CCCC3(NC(CCCCC)=O)C(C2)C3)=O)cc(O)nc2ccccc12 c1(C(=O)NC(C)CNC(=O)CN(C)C(=O)OC(C)(C)C)ccnc2[nH]c(O)nc12 C1(CNC(C2(COC(C(C)(C)C)=O)CC2)=O)OCC2CCC1C2 C1(C(C)(C)C)C(=O)NCCN1C(=O)C(C)(C)C1CCN(C(=O)CC2C=CCCC2)C1 Cc1cc(OCC(=O)NC2CCC2CNC(C2(C#N)CCCCC2)=O)ccc1Cl c1(NC(CSCC)C)ncc(S(=O)(=O)N2CCCC3(CCCCC3)C2)cc1Cl N1(C(C(C)C(F)F)=O)CC2(CC(C(=O)NCc3ccccc3C#N)CO2)C1 C(CCc1nn[nH]n1)(C(=O)O)NC(c1ccc(C2CCOC2)cc1)=O C1(CNC(C=CC)=O)CCCCN1C(c1cc(-c2cccc(Cl)c2)ns1)=O C12(CNC(c3cc(C)n(C)c3)=O)CC(CCO1)N(C(=O)CC1(CO)CC1)C2 C1(C(=O)NC2CC3(C(C(=O)NC4CN(CC)C4)C3)C2)C2CCCCCC12 c1(N(C(CCN2C(=O)OCC2)C2CCCC2)C2CC2)ccc2c(c1)CCC2 O=C(C#CC1CCOC1)NCC1(O)CC(NC(C2Cc3nccn3C2)=O)C1 CON1CCC(C(=O)NC(C)CCNC(C23CCCCC2C3)=O)CC1 C(=O)(C(S(C)(=O)=O)C1CCC1)NCC(CC)(CC)NC(=O)CCCc1ccsc1 c1(NC(C2N(Cc3c(C)cncc3)CCCC2)=O)ccc(Br)c(Cl)c1F c1(CNC(c2ccc3nnsc3c2)=O)cccc2ccnn12 N#Cc1ccc(=NCCCN=C(N)NC2CC(C(N)=O)C2)[nH]c1 c1(OCC(=O)Nc2nnc(C3CCCO3)o2)ccc(Cl)c2cccnc12 N1(C(C2CC(=O)NCC2)=O)CC2CCN(C(c3cc(Br)cnc3Br)=O)C2C1 C(=O)(C1CCc2ccccc21)NC12CC(NC(Cc3cccc(C#N)c3)=O)(C1)C2 N1(C(C2CCCN(CCC)C2)=O)CCCN(C(=O)CCc2cnn[nH]2)CC1CO c1(C(=O)NC(C(C)NC(c2cnc(OCC)nc2)=O)C)cc(N)cc(O)c1C c1(C(=O)OC)cc([N+](=O)[O-])ccc1OCC(F)C(F)(F)F N(C(=NCc1ccc(Br)cc1F)N(C)Cc1ccnn1CCC)C(C=C)C C1(CNC(CC=C)=O)CN(C(c2nc(CC(F)(F)F)sc2C)=O)CC1C C=CC1CN(C(=O)CC2CN(C(=O)C(C)(C)OCC)CC2C)CC1O c1(NC(C)CN2CCCCC2)cccc(C(=O)N(CCCO)C2CCC2)c1 C1(NC(COCCCC#C)=O)CC2CCC1CN2C(=O)C(c1ccc(C)o1)C N1(C(c2nccc(C3(C)CC3)n2)=O)CC2CN(c3ccc(Cl)cc3)CC2C1 c1(CN2CCC(CNC(c3cccc(Cl)c3O)=O)C2)cccc2ccncc12 N1(C(=O)C=Cc2cocn2)CC=C(C(=O)N2CCC23CC(O)C3)C1 C1(O)(C(C)NC(CC2CC(=C)C2)=O)CCN(C(=O)CC2CC(=O)NC2=O)C1 N1(C(C(c2ccccc2F)OC)=O)CCOCC(CNC(=O)C(C)(C)CCF)C1 c12ccnc(c1)N2.C1(C(C)(C)C)CCCN1C(=O)C(C)OCCc1ccccc1 C(c1cc(OC)cc(C)c1)=CC(=O)NCC(CC)NC(CN(C)CCOCC)=O c1(Oc2ncc[nH]2)cccc(NC(=O)CCSc2cccnc2)c1.CC1C(=O)O1 C(=O)(CC(C)(C)C(F)F)NC(C(=O)NC(c1c(C)nc(C)[nH]1)C)c1cccs1 C(=O)(C(CN=[N+]=[N-])NC(=O)CCc1cc(OC)no1)N1CC(COC)(CO)C1 c1(C(N2CCCSCC2)=O)ccc(-c2ccccc2)c2c1OCO2 C1(NC(Cc2cc(C)sc2C)=O)CC(F)CN(C(c2ccc(C(C)O)cc2)=O)C1 c1(C(=O)NC(CNC(c2ccc(SCC)nc2)=O)(C)CO)cccc(C)c1F c1(OC)cc(CCNC(C2CC(F)CN(C(=O)C(C3CC3)SC)C2)=O)ccc1C c1(C(=O)OC)ccc(C)nc1Oc1ccccc1.C12COCCN1CCNC2=O c1(C(=O)NCCCC(O)C(=O)N2CC3CC3C3CC23)cnn2ccc(Cl)c(F)c12 CCCC(CC(C)C)C(=O)NCc1ccc(Cl)o1 Cc1cc(C(N2CC(NC(=O)CC3CC(F)C3)CC23CCC3)=O)c(N)c(Cl)c1 Cc1nn(CC(N2CCOC(c3ncc[nH]3)C2)=O)cc1Br C12(NC(CS(=O)(=O)N(CC)CC)=O)CCCN(C(=O)C(CO)NC(N)=O)CC1C2 C1(NC(CCSCC)=O)CCN(C(=O)CCCc2cccnc2)CC1F C1(C(=O)NC(C(=O)NC2CC(C(=O)OC)C2)c2cccs2)CC(=O)CCO1 C1(N(CC(=O)NC)C)CCN(C(c2cccc(N3CCNC3=O)c2)=O)CC1 c1(NC(C(n2cc(CN(C)C)nn2)(C)C)=O)ccc2c(c1)OCO2 CC(C)C(CC(=O)NCC1CC(C)(C)CN1C(=O)C=Cc1cn(C)cn1)C(C)C N1(C(C2C(C)(CC)C2)=O)CC(NC(=O)CCn2cnnn2)C(c2ccc(F)cc2)C1 C1(C(=O)NC2CCC(NC(c3ccc(C)n3C)=O)CC2)CNc2ccccc2O1 N1(C(COCC(=O)NC)=O)CC2COCC2(C(=O)Nc2nn(C)cc2Cl)C1 C1(C(C)C)C(NC(c2occc2C2CC2)=O)CCN1C(c1ccn(C2CC2)n1)=O C1(C#N)(C(N(CCCNC(=O)CC(C)c2ccncc2)CC)=O)CCCC1 N(C1=COCCC1)C(C1C2CN(S(=O)(=O)Cc3ccc(O)cc3)CC12)=O C1(NC(COC(CC)CC)=O)CCCN(C(c2csc(C)c2C)=O)CC1 N1(C(c2c(CC)[nH]nc2Cl)=O)CCC2(CCCC2NC(=O)C=CCN(C)CC)C1 c1(OCC(=O)NC2(CC)CCN(C(=O)C(C)c3cc[nH]n3)C2)ccc(F)c(F)c1 C1(NC(c2nc(C)oc2C)=O)CC2CCC1(NC(=O)CC1(C)OCCO1)C2 N1(C(c2cc(CC)oc2C)=O)CCC(N(C(=O)CCc2ccoc2)C)C(C)C1 C12(NC(C3CC(=O)NC3)=O)CC1CN(C(=O)Cc1cccc(OC(F)(F)F)c1)C2 CC1=CCC(C)(C(=O)NCC2C3CCCC2N(C(C2C4CCC(=O)C24)=O)C3)CC1 C1(C(=O)NC(C)C(C)NC(=O)C(C)(C)CC2CCC2)CCC(C(N)=O)CC1 N1(C(c2c(C)onc2SC(F)(F)F)=O)CC2(CCCCN2C(=O)CCN(C)C)C1 O=CN1CCN(C(=O)CC2CCN(C(=O)Nc3cc(Cl)cc(Cl)c3)C2)CC1 CCC(O)CCNC(C1(CCNC(=O)C(C2CCOCC2)C)CCC1)=O N1(C(C2(OC)CCOCC2)=O)CC(NC(=O)CC2(CS(C)(=O)=O)CC2)CCC(O)C1 C1(C(=O)NCCCCCN(C(c2ncn(C(C)C)n2)=O)C)CCC2C(C1)C2(F)F c1(OC)ccc(CN2CC(NC(N3CCN(C(=O)N(C)C)CC3)=O)C2)c(F)c1 N1(c2scc(C)n2)CCCC(C(=O)NCCNC23COCC(C2)C3)CC1 C(=O)(C1=NNC(=O)C1)NCC#CC(=O)NC1(CC(=O)OC)CCC1 C1(NCc2ccc(C)cc2)CCN(C(c2cncn(C)c2=O)=O)CC1O c1(NC(C2C(CNC(CC=C=C)=O)CCC2)=O)ccc(C)cc1CC(=O)OC C(=O)(CCCC(C)(F)F)N1C(CC)CN(C(c2cn(CCO)nc2C)=O)CC1 C1(C(=O)NCC2CCC(O)C2)CCN(C(c2ccc(Cl)c(I)c2)=O)C2CCOC12 c1(C(C#C)NC(CCN(C(=O)C=CC(C)CC)CC=C)=O)ccccc1 C1(=O)C(CC(C)C)CN1.CCCC(C)(C)N(C(=O)CC1C=CC(SC)C1)C1CC1 N1(C(c2cnn(C)c2C)C(=O)NC2CC(C(=O)OC)C2)CCC(S(=O)(=O)C(C)C)C1 C1(NC(C2CC=C(C)CC2)=O)CC2CC1N(C(c1cc(Cl)ccc1O)=O)C2 C1(CCOC)(NC(=O)CCC2CCCCC2)CCN(C(=O)CC2C=CCC2)C1 C(=O)(CC(C)C(=O)N1CC(CNC(c2cc(F)ccc2C)=O)C1)OC N1(Cc2cn(CC(=O)NCC(COC)(C)COC)nn2)CCOC2(CCCC2)C1 C1(N(C(c2ccc(COC)cc2)C(=O)NCCCC)C)CCCC(C)(C)C1 Cc1ccc(-c2cccc(CO)c2O)c2nc(NC(c3cccc(Cl)c3)C)cn12 C(C(C)(CC(C)C)NC(C1OCCN(C(c2ncc(F)cc2C)=O)C1)=O)OCC N1(C(C(C(=O)NC(C(CC)(C)F)=O)(C)C)=O)CC(CO)C(C)(C)C1 N1(C(C2C(C)(NC(c3c(CC)nn[nH]3)=O)CCCC2)=O)CCCC(C2(C)CC2)C1 N1(C(C(C)NC(c2ccoc2)=O)=O)CCC2C(C1)CN2C(=O)CCC1(C)CC1 CC(C)C(F)(F)CC(=O)N(C)CCC1CCN(C(c2cnc3n2CCS3)=O)CC1 C=CCCCCCCC(=O)OC.C1CCCN(C(=O)C(C)C2(O)CCC2)C1 C12(C(=O)NCCN(C(C(C(C)(F)F)F)=O)C3CC3)CC3CC1C2C3(F)F N1(C(CCC(CC)C)=O)CCn2ncc(CN(C(=O)CC3COC(=O)C3)C)c2C1 c1(SCCn2cc(C(=O)OC)nn2)ccc(NC(N2CCCCC2C)=O)cc1 N1(CCCc2cccs2)CCN(CC(=O)OCc2onc(CCCC)n2)CC1 C1(C(=O)NCc2c(C(=O)NCCCC(C)O)[nH]cc2)CN2CCC1C2 N1(C(CC(C)N(C)C(c2occ3c2CCC3)=O)=O)CCSCC(C)C1 N1(N(S(=O)(=O)Cc2ccc(COC)o2)CC)CC2CN(c3nccc(Br)n3)CC12 C1(CNC(CC(C)c2cccnc2)=O)CC(O)CN1C(=O)Cc1cccnc1 C(=O)(C(CCC1CCC1)NC(C1CC(=C2CC2)C1)=O)N(C1CC(=C)C1)C c1(C(C(=O)NC2C(NC(C3(C#C)CCC3)=O)CCC2)(F)F)ccccc1F c1(C(=O)NCCC2CCC(NC(CCOC)=O)C2)cc(N(C)C)cc(C#N)c1 n1(C)cc(CO)nn1.c1(C(CN2C(C(C(=O)N)F)CCC2)=O)occc1C(C)C c1(C(N2C(CNC(C(CC#C)O)=O)C=CC2)=O)c(-n2cnnn2)sc(C)c1C Cc1cc(S(N)(=O)=O)cc(C(=O)NC(C)C(C)NC(=O)CN2CCCCC2)c1C CCC(C)CCCCC(=O)NC1CCN(C(c2cc(Br)ccc2Cl)=O)C1 c1(OC)nn(C)cc1C(=O)NCC1CC(F)CN1C(c1nc(=N)cc[nH]1)=O CC(C)CC(C(=O)N1CC2(CCC2)CC1C(=O)N(C)CC1CC1)C(N)=O C1(CNC(=O)CC(F)F)CN(C(C2COCCC2(F)F)=O)CC12CCC2 C1(C(C(N2CCC(C)C2)=O)(C)C)CCCN(C(C2C3CN(C)CC23)C2CC2)C1 Cc1ccc(=N)[nH]c1C(N1CCC(C)(CNC(C2CC23CC(O)C3)=O)C1)=O CCC(CC)(CC)C(=O)N1CC2CC1C2NC(=O)Cn1ccc(C)n1 N1(C(=O)OC(C)(C)C)CCC(C(N2CCN(CC(O)C3CC3)CC2)=O)(C(F)F)C1 c1(C(N(CC)Cc2cccnc2)=O)n[nH]c2c1CCC(N)C2 C1(C(=O)NCC(C)CC2CC2)CCC=CC1NC(=O)CC1CCCC(=O)C1 C(=O)(CC(C)(C)C(=O)N1CC(CC(C)NC(=O)C=CBr)C1)OC c1(OC)ccc2[nH]c(C)c(C(=O)NC3CC(NC(C45CC(F)(C4)C5)=O)C3)c2c1 C1(NC(c2cc(C(C)C)c(Br)cc2)=O)CC12CCN(C(C1CCCOC1)=O)CC2 CC1CCC(CC(=O)NCC2(NC(=O)COCCCC(C)C)CCC2)CC1 C(CC(=O)NC1CCCC(NC(=O)CNc2nccs2)C1)(C1=CCCC1)OCC CC(CC(=O)N1CCC(N(C)C(c2ccc(C(N)=O)[nH]2)=O)C1)C(C)(C)C c1(C(=O)NC(C2CCC(C)CC2)C(=O)O)cccc(C#N)c1F c1(C(N(CCNC(C=CC(C)(C)SC)=O)CC2CCCO2)=O)cn2cccnc2n1 CCCC(C(O)C(=O)N1CC(C(=O)NCC)C1)NC(=O)Cc1csc(C)c1 C(=O)(C(C#N)C(C)C)N1CCC(NC(c2c(C)cco2)=O)(CF)C1 C1(NC(c2ccc(Br)nc2)=O)CCN(C(C2(c3ccccc3)CCC2)=O)CC1O C1(CNC(=O)Cc2csnn2)CN(C(=O)Cc2ccccc2F)CCC12CCOC2 c1(N(CC#C)CC)nnc(Cc2cc[nH]c2)n1CCC(=O)NCc1cccnc1C N1(C(C(Cn2ccc(C)n2)C)=O)CC(C)CN(C(=O)C(C)CC2CCC2)CC1C c1(C(=O)NCC2(O)CCN(C(C(CCC)OC)=O)C2)c(F)ccc(Br)c1N c1(OC)cc(F)c(F)cc1NCc1cc(O)cc(Br)c1 C(c1cccc(CO)c1)=CC(=O)NC1CN(C(Cc2c(C)nsc2)=O)C2C1C2 C1(C(=O)NCC2(O)CCN(C(Cn3c(C)nnn3)=O)CC2)CCc2nnnn2C1 c1(C(C)=O)csc(C(=O)N(Cc2cn(C(C)(C)C)nn2)CC2(F)CCOC2)c1 C(=O)(C1=COCCC1)NC1CN(C(C2(CC#C)CCCO2)=O)CC1CCC C1(NC(C(N(C(CCC(=C)Cl)=O)C)C2CC2)=O)CCOC(C)(CC)C1 Nc1nc(Cl)ccc1C(N1CCOCC1CCNC(c1cccc(Cl)c1)=O)=O CC1CCc2[nH]c(C(=O)NCC3(O)CN(C(C4CC5C(C4)C5(C)C)=O)C3)cc2C1 c1(OC)cc(C)c(CC(=O)NC2CCCC2CNC(=O)C(F)(F)COC)c(C)c1 c1(CNC2CCC(C)(C)CC2C(N2CCNC(=O)C2)=O)ccc2ccccc2c1 c1(N2CCCC(O)CC2)nc(N2CCOCC3(CCC3)C2)c2ccsc2n1 Cc1c(C(N2CCC(F)(C(=O)NCC3COCC3(C)C)C2)=O)cccc1F Cc1cnc(C(N2CC3CC3(CNC(=O)C(C)CC(N)=O)C2)=O)c(F)c1 C(=O)(C1=C(Cl)CCC1)N(C)CC1OCCN(C(c2c(C)noc2C)=O)C1 c1(C(=O)NCC2(C)CCN(C(Cc3nnc(C)o3)=O)C2)ccc(F)cc1Br c1(C(c2nnnn2C)NCCCNC(C)=O)c2c(nn1C)CCCC2 C1(CNC(CCC#C)=O)CCC2(CCN(C(=O)C(F)C(F)(F)F)CC2)CO1 c1(C(N2CC(NC(CCCN(C(C)=O)C)=O)C(C)C2)=O)cc2occc2s1 C12(C(=O)NC3C(NC(=O)C4=COCC4)CS(=O)(=O)C3)CCC(O)(CC1)CC2 c1(C(=O)NCCN(C2CCCC2)C(c2ccc(CC)o2)=O)cc([N+](=O)[O-])n[nH]1 c1(C(N2CC(CNC(CSc3n(C)nnn3)=O)C3C2C3)=O)nc2c(s1)COCC2 c1(COC(c2c(C)sc(O)n2)=O)ccc(S(C)(=O)=O)cc1 CC(CNC(=O)CC1(C#N)CC1)C(F)C(=O)Nc1cncc(C2CC2)c1 N1(C(C2CC(OC)C2)=O)CCC(C)(C(=O)NCC(C)CC(C)C)CC1 c1(OCC)ccc2c3[nH]c(cc13)CC(=O)NNC2=O.c1(OC)ccccc1Cl C1(NC(CC=CC(C)(C)C)=O)CCCC(NC(C2CC(F)(CO)C2)=O)C1 C1(NC(c2cn(CCC)nc2)=O)CCCC(NC(c2cc(C#N)on2)=O)C1 c1(C(N(C2CC(NC(C3CC4(CC4)CO3)=O)C2)C)=O)cc2sccc2n1C C(C)(CCC(=O)NC1CC2(C1)CC2NC(C1(N)CCCC1)=O)SC C12(C(=O)NC(CC(C)C)CNC(=O)Cc3cnco3)CC3CC(C(=O)N1)C2C3 Cn1ccc(=O)c(C(=O)NC2CCC(CNC(C3CC4(CCC4)C3)=O)CC2)c1 c1(C(C)(C)C(=O)NCCn2cc(CC(CO)C3CC3)nn2)ccccc1Cl c1(C(N2C3(CNC(C(C)(C)OCC)=O)CC(C2)C3)=O)cc(C)nc(Cl)c1N N1(C(CN(C(C)=O)C)=O)CC(CNC(=O)CN2CC(C)C2)C2(CCC2)C1 C(C(C)CC(=O)NC1CC(F)(CNC(c2coc(-c3ccccc3)n2)=O)C1)OC C1(C2CCCN(C(=O)C=C3CCC3)C2)(NC(Cc2ncc(C)s2)=O)CC1 C1(NC(C2CCN(CCC)CC2)=O)CC2CN(C(c3cc4ccsc4[nH]3)=O)CC12 N1(C(C2CC(OCC)C2)=O)CC2(CCC2)CC1CNC(=O)C1=C(C)OCC1 C1(C(=O)NOC(C)C)CCCCCC1N=c1cc(NCCC)nc(C(C)C)[nH]1 Cc1ccc(C(N2CCC(C)(CNC(C34CCCCC3C4)=O)CC2)=O)c(O)c1 c1(C(N)=O)ccc(CC(N2CCC(C)(NC(C3COCC34CCC4)=O)C2)=O)cc1 c1(C(N2CC(NC(c3ccn(CCCC)n3)=O)C(O)C2)=O)cc2ncccc2[nH]1 CC1CN(C(=O)CCC2NC(=O)NC2=O)CC(C)N(C(=O)Cc2cnoc2)C1 C1(C(N2C(CC=C)(C(=O)NCC(CC)CC)CCC2)=O)CC2CCCC2C1 CC(C)(CC(F)C(=O)N1CC(=O)NC(=O)C1)NC(=O)CSCC(F)F C1(CC(N2CC3(CCN(C(C4C(C)C4)=O)C3)C2)=O)CCC2(CC1)OCCO2 C1(C(=O)OCC)CC(N)CCOC1.N12CCC(CC1)SC(c1ccccc1)C2=O c1(C(=O)NC(C2CN(C(c3cnc(O)c(F)c3)=O)CCO2)C)cc2cscc2s1 C=CCC(C(=O)NCC1(CNC(C2(C)CC=CCC2)=O)CCC1)c1ccccc1 C1(c2nnnn2CC2CC2)(NC2(CC(C)C)CC2)CCOC(P(C)(C)=O)C1 O=C(Nn1ccnn1)C(F)C1C2CCCC2N1C(=O)Cn1ccccc1=O CC1Oc2cc(F)ccc2C1Nc1nc2ccsc2c(=NCC2(N(C)C)CCC2)[nH]1 Cc1cc(Cl)cc(C(=O)N(CC(O)CNC(=O)CC2CCCC2)C)c1O C12(CNC(c3ccc(CCC)s3)=O)CC(NC(C3CCCC3O)=O)(C1)C(C)O2 C1(CC(=O)NCCC(C)NC(c2ccc(C(C)(C)C)cn2)=O)OCCOC1(C)C N1(C(C2C(=O)OCC2)=O)CCCC(N(C(=O)CCn2cccn2)CC2CC2)C1 N1(C(CC(=O)NCC#C)=O)CCN(C(=O)C=CC2CCCN2C)CC12CC2 c1(C(=O)OCC)ocnc1-c1cn(C(C)C(=O)NCC(N)=O)nn1 N1(C(c2ccsc2C)C(=O)NCCSC)CC(CO)C2(CC2)C1 Cc1ccc2nsnc2c1C(=O)NCC12CC1CN(C(c1cnncc1O)=O)C2 Cc1ccccc1CC(=O)N(CCCCC(=O)NCC(O)CCC1CC1)C FCCN=C(NCc1ccc(-n2cc(Cl)cn2)cc1)Nc1ccncc1 C1(OC)CC(CNC(C2CN(C3COC3)C2)=O)N(C(=O)Cn2nc(C)cc2C)C1 CCCC(C(=O)NC1(CNC(=O)CN2CCCC2CO)CCC1)N(C)C Clc1ccc(C2=CCC(C3CC3)CC2)c(NCCOc2ncccn2)n1 Cc1cc(F)ccc1CC1CCCC(NC(=O)NC2(c3cccc(F)c3)CC2)C1 C(=O)(C(C)N=[N+]=[N-])NCC(C(C)C)NC(c1cc(CC(C)C)c[nH]1)=O C1(CCNC(CNC(=O)NC)=O)CCN(C(=O)C(C2(N(C)C)CCCC2)C)C1 C1(C(C(=O)NC(C2CCCC2)C#C)C)CCN(C(=O)Cc2cncn2C)C1 CN1CC=C(CC(=O)N2CC3CCN(C(=O)CN4CCCCCC4)CC3C2)CC1 c1(CC)ccc(C(=O)NCC2(C)CCC(NC(=O)CSCCN(C)C)C2)nc1 c1(OC)cccc(N(C(=O)C(C)CNC(=O)Cc2ccoc2)C)c1 c1(CN2CCC(N(C(=O)C(CO)c3ccccc3)C)CC2)cc2cnccc2[nH]1 C1(CC)CN(C(=O)CCSCC(N)=O)CCN1C(C1CC2CC2C1)=O C=CCCCC(C)(C)C(=O)N1CCC(C(N2CCOC3COCC23)=O)C1 CC(C)(O)C(F)(F)C(=O)N1CC2CC(NC(c3csc(Cl)c3Cl)=O)CC2C1 C1(CNC(C)=O)CN(C(C2CC(=O)N(CCc3ccc(F)cc3)C2)=O)CCCO1 c1(NC)ccc2cc1OCCNC2=O.C1(C(=O)OC)CCCN(C(=O)CO)CC1 C1(O)(CNC(=O)C(F)C2CC2)CCCN(C(c2ccc(OC(F)F)nc2)=O)C1 N1(c2c(C)c(Cl)ncn2)CCCC2C(NC(c3ccc(C(F)(F)F)cc3Cl)=O)C12 C1(C(=O)NCc2cnns2)(CNC(C2C(=C)C2)=O)CC=CC1 Cc1ccncc1C(=O)NC(c1nocc1C(=O)NC1(C(C)(F)F)CCC1)C C(c1ccc([N+](=O)[O-])s1)=CC(=O)N(CCCCNC(C(COC)(C)OC)=O)C C1(NC(C2CCC(=C)CC2)=O)CC2CCC(C1C)N2C(c1csc(=NC2CC2)[nH]1)=O CCC(C(=O)N1CCC(CNC(C2CC(F)(CO)C2)=O)C1)NC(c1ccco1)=O C=C(C)C1OCCC1CNC(=O)C(Cn1cccn1)NC(=O)C=CCOC C(=O)(CCCC(C)(C)C#N)NC1(C)CCN(C(c2c(C)nc(COC)s2)=O)CC1 N1(C(C2CN(C)C(=O)N2)=O)CC2(C)CN(C(C3CCC(C)CC3)=O)CC2(C)C1 Cc1ccc(Cl)c(O)c1C(N1CCC(C(C)NC(c2cc(Cl)cs2)=O)CC1)=O C1(C(=O)NCCC(CC)C)CCN(C(c2ncccn2)=O)C12CCC2 Cc1ccccc1Oc1ccc(C(N2CC(CS(C)(=O)=O)C2)=O)cc1 N1(C(C2CCC(CC)O2)=O)CCOC(CNC(c2nccn2CCCSC)=O)C1 N1(C(C(C)SC(C)C)=O)CCC2(C1)CN(C(c1ccccc1CC(F)(F)F)=O)C2 CC1CN(C(=O)Cc2ccccc2)CCC1CNC(c1csc(CO)n1)=O C1(NC(COCCOCC#C)=O)CN(C(=O)C(C)(C)c2cccs2)CC1C CC1(NC(=O)CO)CC(c2nn[nH]n2)(C(=O)O)C1.c1(S)cccc(Cl)c1 Cc1cccc2c1ccn2CC(N1CCN(C(=O)C(C)O)C(C(C)C)C1)=O C1(F)(CNC(C2(NC(N)=O)CC2)=O)CC2CCC(C1)N2C(c1ccnn1CCF)=O c1(CC(=O)NC2CN(Cc3cncc(F)c3)CC2O)ccc(Br)cc1Br N1(C(CCCCOC)=O)CC(CNC(c2cnn(C)c2C(C)C)=O)C(F)(CO)C1 CCCCC(C(=O)NC1(CCOC)CC1)NC(=O)Cc1c(C)cccc1C N1(C(C)C(=O)N(C2CN(C(=O)CN(c3cnc(S)[nH]3)C)C2)C)CCCC(O)C1 C(CCC(N)=O)(C(=O)NCCSC1COCC1O)NC(=O)OC(C)(C)C C(=O)(C1=CC2CCC(C1)C2)NC1C(CC)CN(C(=O)CCc2nc(O)n[nH]2)CC1 O=C1CN(C(c2cc(O)cs2)=O)C(C(N2CCC(CCO)C2)=O)C1 Cn1ccnc1C1CC1C(N1CC(O)(CCNC(C2CCC(=O)O2)=O)C1)=O C=C=CCN=c1nc2ncn(CC)c2c(NCC(=O)NCC2CC2)[nH]1 NC(=O)CCCC(=O)NC1CCN(C(C23CCN(CC2)C3)=O)C1 N1(C(C2CCN(CC)C2)=O)CC(CNC(c2cnc(=N)[nH]c2)=O)C2(CCC2)C1 c1(C(CNC(=NC)NCc2cc(-c3ccc(F)cc3)n[nH]2)(F)F)ccc(F)cc1 N1(C(C=CC(=O)OC)=O)CCC(F)(CNC(C2CCCN(C(C)=O)C2)=O)C1 c1(C(=O)OC(c2cn(C3CCCCC3)nn2)C)[nH]nc(C(N)=O)c1-c1ccccc1 C(=O)(C#CC1CCOCC1)NC1CC(CNC(c2c(C)cc(O)nn2)=O)OCC1 c1(CC(=O)N(C(C)CCNC(=O)CC2CC(CF)C2)C)cc(O)nc(C2CC2)n1 C1(C(=O)OC)CC(=O)N(c2cn(CC3CN3Cc3ccc(F)cc3)nn2)C1(F)F C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CCC2(N(C(CC(C)SC)=O)CCC2)C1 C(=O)(C(CNC(=O)CNC(=O)N)CC(C)C)N1CCCN(CC=C)CC1.CC C(=O)(C(CNC(=O)C(c1n[nH]c(C)n1)C)CC1CC1)N(CC(C1CC1)OC)C c1(C(=O)NC(CC(N2CCC(C#C)C2)=O)(C)C)ncn2c1CCC2 CCCCCC(O)CC(=O)N1CC2(CCCN(C(=O)CC(C)C(F)F)C2)C1 Cc1cc(NC(C2(NC(c3cn(C)c(C)n3)=O)CCOCC2)=O)cc(Cl)c1 C1(C(C)NC(c2cc(OC)no2)=O)CCCCN1C(=O)COCC1CCOC1 C(=O)(C1CCc2nnc(C)n21)NCC(CC)NC(c1cc(CCC)on1)=O C1(NC(c2[nH]cc(CC)c2)=O)CCN(C(=O)C(F)=C(C)C)C(C)C1 N1(C(c2c(CC)onc2C)=O)CC2CC1CC2CNC(c1ccns1)=O Cc1cccc(C#N)c1S(=O)(=O)NCCCn1cc(Cl)c2cccnc12 C1(NC(C(CC)OCC)=O)C2CN(C(=O)CC(C)(C)c3cccs3)CC12 c1(OCC(=O)NCCCNC(CC=CCCCCC)=O)ccc(C(N)=O)cc1 c1(C(N(CC(C)(C)CNC(=O)COC2CC=CC2)C)=O)cccc(F)c1F Cc1cccc(C(=O)NC(CNC(c2cccc(-n3cccn3)n2)=O)CO)c1 C(CCC(C)C(=O)OC(C)C)OC.C12CCN(CC1)CC2(C)C CCC(C(=O)NC1(CN(C(=O)C(c2ccc(Cl)s2)C)CC)CCC1)NC(C)=O c1(C(N(C(C)CNC(C2CC(N(C)C)C2)=O)C)=O)cnc(Cl)c(N)c1 C1(NC(C(C)N(C)C)=O)CC12CCN(C(c1cc(C#N)ccc1F)=O)CC2 Cc1ccn2ncc(C(=O)NC3CCCC(NC(c4cnc(O)s4)=O)C3)c2n1 CC(C)C(C(C)NC(=O)CCCn1ccnn1)NC(=O)CCc1ncccn1 c1(SCC)cccc(C(N2CCC(C)(NC(C3CCCC3)=O)C2)=O)c1 c1(C(N2CCC(NC(C3C=CCC3)=O)C(O)C2)=O)cc2ccccc2oc1=O CC#CCC1C(=O)N1.c1(C(C)NC(C2(OC(C)=O)CC2)=O)ccncn1 c1(CN(C)C)ccccc1C(=O)NCC1CC1CNC(c1ccsc1)=O C1(C(N2CCN(C(C(=O)NC(C)C)C)CC2)=O)CC(C(=O)O)CCN1C C1(NC(C2C(C(=O)OC)CCC2)=O)CCN(C(=O)CC(C)(C)O)C1C N1(C(CCC(=O)NC)=O)CC2(C1)OC1(C)CC2(NC(=O)CC2(C(F)(F)F)CC2)C1 CN1CCCC(CC(=O)N(C)CC2CCCN(C(=O)CC3(C)N=N3)C2)C1 Cn1cc(Cl)cc1C(=O)NC1CC(NC(c2cc(O)ncn2)=O)C(O)C1 CCCCCC(O)C(=O)NCC1(OC)CN(C(C2CC3(CCC3)CO2)=O)C1 C1(CNC(C(C)C2CCCC2)=O)CCCCC1NC(=O)CC1CCSC1 C12(NC(C(C(C)C)OCC)=O)CCCC1(F)CN(C(=O)C=C1CCOCC1)C2 c1(C(=O)NCC(CCOC)NC(C2CCCN2C=O)=O)sc(OC)nc1Cl C=CCC(C)(C)C(=O)NC1CCN(C(c2ccn(C3CC3(F)F)n2)=O)CC1F N1(CC2(Cl)C(C)(C)C2)CC2CS(=O)(=O)CC2C1 C1(C(=O)NC2(CCOC)CCCC2)CC=CCC1NC(=O)Cc1ccc(O)nc1 C(=O)(CC(O)(CCC)CCC)NC1CC2CN(C(CC(CCC)O)=O)CC1C2 C12(CNC(C3ON=C(CC)C3)=O)CCCC(CN1C(=O)CSC(F)F)C2 CC1(C(N2CCC(CC3CCC3)C2)=O)CN(C(=O)C(F)F)C1 c1(N2CCC(NC(C)C)CC2)nccc2sccc12 C1(C(C(=O)NC2(C)CC2)N(C(c2ccccc2)C(=O)NC)C)CCCCC1(C)C c1(OC)ccc(C(=O)N(C2CN(C(C3(n4cccn4)CCOCC3)=O)C2)C)cc1 CCCC(C)(O)CC(=O)N1CCCC1C(C)NC(c1cc2ccncc2o1)=O c1(C(N2C(CCNC(C(CC)C)=O)COCC2)=O)c[nH]c(C)c(Cl)c1=O N1(C(COC(C)=O)=O)CC(N(C)C)CC1C.C1C(=O)N1CCC C1(NC(c2ccncc2Cl)=O)CCC2(CC1)CC2NC(c1ccc(=O)oc1)=O C1(CNCC2C(C(=O)OCCOC)CCCC2)CCc2nnnn2CC1 c1(C(=O)NC(C(C(C)C)NC(CCCCCSC)=O)C)c(C)ncn(C)c1=O c1(C(=O)NC2(CNC(C(CC)(C)C(F)F)=O)CCC2)ccc2nnc(O)n2c1 C(=O)(C(C)C(C)(F)F)NCC1(CCNC(CCCc2nc(C(C)C)on2)=O)CC1 Cc1ccc(-c2nc(CC(N3CC(C(C)NC(C4CC4Cl)=O)C3)=O)cs2)cc1 CC(C)(C(=O)NCC1CCCC1C(=O)NC1CC2CC2C1)c1cnsc1 C1(C(N2CC(N3CCCC3)C2)=O)(CNC(C(CC)O)=O)CCCCC1 c1(OCCCC(=O)NC2CC(F)(CNC(CN(C)CC)=O)C2)ccccc1Cl C(=O)(CC(O)CCCCC)N1C(C#C)CN(C(=O)C=CC(C)C)CC1 Cc1cnn2cc(C(=O)NCCC(C)CCNC(c3ccc(=O)oc3)=O)cnc12 N1(C(c2n[nH]c(O)n2)=O)CC=CC(C(N2CCN(C3CCC3)CC2)=O)C1 C1(C(=O)NC2CC(OC)C2(C)C)CC(F)(F)CN1C(=O)CCNS(C)(=O)=O S(=O)(=O)(c1ccc(NCC(C)(C)C(C)O)c(Br)c1)NCCCC(C)C C1(NC(c2cc(CC)on2)=O)CN(C(=O)CCOC2CCOC2)C2CCCCC12 C=CCC(CNC(=O)Cc1c[nH]nc1O)C(=O)NCC1CC(C)(CC)C1 Cc1ccc(CNC2CCC(NC(c3cc(C)ccc3F)=O)C2)c(O)c1 N1(C(C(CCN(C)C)N(C)C)=O)CCCC(F)(CNC(c2cc(O)ncn2)=O)C1 C#CCCCCCC(=O)NCC1CCN(C(c2n[nH]c(C)n2)=O)CCC1(F)F N1(C(C(C)SC)=O)CC2CCN(C(c3oc4ccccc4c3C)=O)CC(C2)C1 N1(C(C(C)SCC)=O)CCCCC(C(=O)NCCCN2CCCC2C)C1 c1(OC)ccnc(-c2nnc(N3CC(C)(C)C3c3ccco3)n2C)n1 CCCCC(CN1CCCC(C#N)C1)CC N1(C(C(C)CO)=O)CC(C(=O)NC2CC(CO)(CO)C2)C2(CCC2)C1 C1(C(N(CC)CC2CCCN(C(=O)CCC(=O)C3CC3)C2)=O)CN(C)CCN1C c1(C(=O)NC2CC(CNC(C3C(C)(C)CO3)=O)C2)ccc(CC2CC2)cc1 CCC(C)CC(C(=O)N1CCCCC1C(C)C)Nc1cc2ccccc2o1 C1(NC(C(C=CC)O)=O)CN(C(c2ccnc3ccnn23)=O)CCC12CCC2 C1(C(C)NC(=O)C(F)C(C)C)CC(C(C)(C)C)CN(C(=O)Cc2cnccn2)C1 Cc1cc(C)c(C(=O)NC(C2CN(C(c3c(C)cnn3C)=O)C2)C)c(O)n1 C1(NC(C(C)c2ccco2)=O)CN(C(c2ccc(N(C)C)nc2)=O)CC1N=[N+]=[N-] C#CC1CCC(NC(C2CCN(C(=O)C=Cc3ccccc3)CC2)=O)C1 c1(SCCC)ccc(C(=O)NC2CN(C(C3CCC3)=O)CC2O)cc1 c1(N2CCS(=O)(=O)CC2)cccc(S(=O)(=O)NC2CCSC2)n1 C1(CNC(CC2(C=C)CC2)=O)CCN(C(=O)Cc2cc(COC)nn2C)CC1 Cc1nn(C)c(C(=O)N(C)CCN(C(=O)CCCCNC(=O)C2CC2)C)c1Cl c1(CC)cc(N(C(CCNC(=O)C=Cc2ccco2)C(C)C)C)nc(C)n1 c1(C(N(C2CCCN(C(c3nnn(C)c3C)=O)C2)CC)=O)cc(Br)c(C)o1 C12CN(CCCO1)C(C1CC1)C(=O)NC2.c1(C(=O)OC)cc(C(N)=O)co1 c1(C(C)C)cnn(C)c1C(=O)NCc1scc(CCN2CCOCC2)n1 N1(C(c2c(CC)nccc2)=O)C2CC1CN(C(c1cnccc1C(F)(F)F)=O)C2 C1(c2nc(NC(=O)OC(C)(C)C)nn2-c2ccc(Br)nc2)CCC2CCCCN12 CCC(C)CC(=O)C(=O)N1CCC(C(=O)N(CCCF)CC)C1 Cc1nn(CC(N2CCCCC(N(C(=O)CCCCC#N)C)C2)=O)c(=O)n1C N1(C(C(CCC)OC)=O)CCC(NC(c2[nH]c(C3CC3)nc2C)=O)C(O)C1 c1(C(N(CCC(=O)OC(C)(C)C)CC)=O)ncccc1OC.C(C)(C(=O)N)N(CC=C)I c1(C(=O)OCc2nc3ccccc3[nH]2)cccc2ccc(Br)cc12 CCCC(CCC)C(=O)N1CC2C=CC1C(C(N1CC(CC(=O)OC)C1)=O)C2 N1(C(C(C)SC)=O)CCC(O)(CNC(=O)CCC2CCCOC2)C1 C(CCC(=O)NN1CC(c2cn(CC3(c4ccccc4)CCCC3)nn2)C1)C1C(C)C1 N1(C(C(C(C)C)SC)=O)CC2CCN(C(c3cccc4nc[nH]c34)=O)CC2C1 N1(C(C(C)Cc2ccccc2Br)=O)CCC2C(CCN2Cc2ccc(Cl)cc2)C1 C1(C(=O)NC(C)Cc2cn[nH]c2)CCN(C(c2cnn3c2OCC3)=O)C12CC2 c1(C(=O)NCC(CN(C(=O)CCC(F)(F)F)C)O)cccc2nc[nH]c12 C(c1ccc(C(F)F)o1)=CC(N1CCC(CN(C(c2c(C)cns2)=O)C)C1)=O C#Cc1ccc(NC2CCN(CSCCNC(=O)OC(C)(C)C)CC2C)cc1 Cc1c(F)ccc(C(=O)NCC2CN(C)CCN2C(=O)CSC2CC2)c1C c1(NC(C(C(CNC(c2c(C)ccnc2C)=O)C)F)=O)cnc(C)nc1C C(C)(C(C(=O)N1CCCC1CCNC(C1CC=CCC1)=O)N(C)C)OC CC(c1ccsc1)=CC(=O)NCC1COCC1NC(C1CCCCO1)=O Cc1nc2cc(C(=O)NCCC(C)(C)NC(C3CC(O)C3)=O)ccc2o1 c1(COC)nc(N2CCC(=CCNC(C3CCCOC3)=O)CC2)cc(Cl)n1 C1(NC(C2C(C(C)C)OCC2)=O)(CO)CCCN(C(=O)COCCCF)C1 Cc1c(CC(N2CCOC(CCNC(c3cncs3)=O)C2)=O)cnn1C CC1(C)C2CCC1(C(N1CCC(CCCNC(=O)CCc3ncc[nH]3)CC1)=O)C2 N1(C(C=CC(C)(C)OCC)=O)CCC(CO)(NC(=O)C=Cc2ccncc2)C1 N1(C(c2c(C)non2)=O)CCOC(C)(CC(=O)NCC2CC3(C2)CC(O)C3)C1 C=CCC(F)(F)C(=O)N1CC(CNC(C2CC2C(=O)OC)=O)(OC)C1 CCC(CC(=O)N1C(C(=O)N(C)CCNC(C)=O)CC2CC12)C(F)F C(=O)(CC(C(F)(F)F)NC(=O)CN1CCC(=O)NC1=O)N1C(C(=O)NC)CC(O)C1 N1(C(c2c(C)nns2)=O)CC(CO)C2(C1)CN(C(C1CCCN1C(C)C)=O)C2 Cc1cc(OCC(=O)NC(C)C(C)NC(c2c[nH]c3ncccc23)=O)ccc1Cl C1(C(=O)NCC2(C(C)C)CC2)CN(C(c2cncc(C3CC3)c2)=O)C(C)(C)C1 N1(C(CC2(OC)CC2)=O)CCC(C(=O)NCCCC2C=NNC2=O)CC1C C(C(C)(O)C(=O)N(CCCNC(=O)C(C)n1cncn1)CCO)OC N1(C(c2n(C=C)nnc2)=O)CC(F)(F)CC1C(=O)NCCN=[N+]=[N-] Cc1nc2ccc(C(=O)NCc3cn(CC4C(C)C4(F)F)nn3)cc2nc1C C(=O)(C(C(C)(C)C)NC(=O)C(CCSC)NC(c1cc(C(N)=O)c[nH]1)=O)NC C12CCN(CC1)C(=O)NC(C(C)C)CNC(=O)N2.c1(C(=O)N(C)C)cccnc1 Cc1cncc(C(=O)N(CC(=O)NCC2CCCC(CO)C2)C(C)C)n1 C1(OC)(OC)CCC(F)(F)CC1NC(=O)C(CN)CN CC(N=c1nc(-c2ccccc2)[nH]s1)C(c1ccccc1)C(C1CC1C)=O C1(O)(C(=O)NC2C(CNC(C3C(OC)CCC3)=O)CC2)CCCCC1 c1(N)ccc2nccn2n1.C(=O)(CCOCCNC(C1(N(C)C)CC1)=O)N.O N1(CCN(CCC)CCOCc2cccc(F)c2Cl)CC(C)OC(C)C1 c1(NC(C(CNC(C=CC(CC)C)=O)CC2CC2)=O)cccc(O)c1F C1(CCC)(NC(=O)CC2(C)CC2)CCN(C(=O)C#CC2CC2)CC1 c1(CNC(C2COC(=O)O2)=O)ccccc1CNC(C1(F)C2CCCC12)=O C(=O)(C(C)(C)NC(C1CCOC1C1CC1)=O)NC(C(=O)NC)C1CC1 c1(C(N2CC(O)(CCNC(C(=O)OCC)=O)C2)=O)cc(COC(C)(C)C)nn1C c1(C(C)NC(=O)C(C2CC=CCC2)NC(c2ncccn2)=O)c[nH]ccc1=O [N-]=[N+]=NC1(C(=O)NCCCOC(F)(F)F)CCN(C(=O)CCC2CCC2)C1 CC1(C)CCC=C1C(=O)N1CC(CCNC(c2cc(C(F)F)[nH]n2)=O)C1 c1(C(N(CC(=O)N(CCCCCCC)C)CC2CC2)=O)cc(O)cc(=O)o1 C=Cn1nccc1C(=O)NCCCCC1CCCN(C(=O)CN(S(C)(=O)=O)C)C1 C1(CN(C)C(C2CCC(F)(F)C2)=O)C2CN(C(c3cccc(CO)n3)=O)CC12 C1(NC(c2cc(C)cc(Cl)n2)=O)CCN(C(c2c(C)ncn2C)=O)CC12CCC2 c1(CC)nn(C)c(C(=O)NCC2CCN(c3nccc(C(N)=O)n3)C2(C)C)c1Cl CC1CCN(C(C2CC3(CC3)C2)=O)CCN1C(=O)CCCCCc1cccs1 N1(C(c2c(N)c(F)cc(F)c2)=O)CC2CCN(C(=O)C=CC(F)(F)F)CC2C1 c1(CC)cc(C(=O)N(CCCNC(C2CCCCC(=O)N2)=O)C2CC2)c(C)nn1 C#CC1CN(C(=O)CSc2ccccc2O)CCN1C(=O)C(C)CC1CCC1 Cn1ccc2c(C(N3CCCC(C(=O)NCCc4ccsc4)CC3)=O)cccc12 C1(C#N)(OC)CC(C(=O)NC(CO)C(C)NC(C2C=CCC2)=O)C1 C(=O)(C1CCc2ccc(C)cc21)N1C2(CCN(C(CCCOCC)=O)C2)CCC1 C1(N(C(CCC=C)=O)CCF)CCCN(C(c2nc(Cl)c(Cl)s2)=O)C1 c1(NC(N2CCC(C(C)(O)C(F)(F)F)CC2)=O)c(O)ccc(F)c1Br N1(C(c2cc(C)on2)=O)CC2C3CCC(C2C1)N(CC(O)CC1CCCCC1)C3 c1(NCC(CC)CO)[nH]c(=NCc2cccc(Br)n2)nc2c1ncn2C Cc1cccc(NC(C)C(=O)Nc2ccsc2C(=O)NCC(F)F)c1 C1(NC(c2ccc(C3CC3)o2)=O)CCCN(C(=O)CCC2CC2(F)F)C1 C1(NC(C2CCN(C(C3CCC(F)(F)C3)=O)C2)=O)CC2CC3C(C2)C13 Cc1cc(NC(c2coc(Br)n2)c2nnnn2CC2CCCO2)ccc1O C1(C(=O)NC2CCC(CO)C2)CC2CCC1N2C(c1n[nH]c2c1COC2)=O C1(C(N2C(CNC(c3c[nH]nc3C3CCCO3)=O)CC2)=O)CCc2c[nH]nc2C1 C1(NC(c2n(CCCSCC)nnn2)c2cnoc2)(C)COCC1(C)C Nc1cc(O)cc(C(N2CCC3CCC(NC(c4cccc(F)n4)=O)C23)=O)c1Cl C1(c2ccccc2)(NC(=O)Cc2cc[nH]n2)CCN(C(=O)C(F)=C2CCCC2)C1 C=C=C(C)CC(=O)N1CCC(CCCNC(=O)CC2CCC(=O)N2CC)CC1 Cc1cc(C#N)c(O)nc1C(=O)NCC1CN(C(c2cn3ncccc3n2)=O)C1 c1(C(=O)NCC(C)NC(C2(CC3CC3)CC2)=O)ccncn1 c1(C(N2CCCC(CNC(C(CO)NC(N)=O)=O)C2)=O)ccc(F)c(CO)c1 CN1C(=O)CCCC1C(N1CCN(CCNC(c2cc3n(n2)CCC3)=O)CC1)=O C1(NC(CN(C(=O)OC)C)=O)CCCCC1NC(c1oc(C(F)F)cc1C)=O CCCCCC(C(C)(C)C)NC(=O)NC1CCCC(CO)C1 Cc1ccc2nc(C)cc(C(N3CCC(NC(=O)C(C)CN(C)C)C3)=O)c2c1 N1(c2c(C)c(NCc3nc(Cl)cs3)ncn2)C2CCC1CN(C)C2 C(CC=O)ON.N1(CC(=O)N(C(=O)Cc2ccco2)C)CCCC1 N1(C(C2C(C(=O)OC)C2)=O)CCC2(CC1)CCN(C(=O)CCc1ccoc1)CC2 c1(NC(=O)OCC)c(C)cc(C)nc1OC.C1(N2C(O)C2=O)CC2CC1CN2 n1(CC)nnc(C(=O)NC(CC(N2CCC(CC3CC3)CC2)=O)C2CC2)c1C C(C(C)C)(C(O)C(=O)N(C(C)C(=O)NCC(c1ccc(F)cn1)O)CC)OC CC(CO)N(C(=O)CC1(C(=O)NCCC2CC2C)CC1)C N1(C(c2cnc(CC)[nH]2)=O)CCC(NC(c2cc(C3CC3)nn2C)=O)C(C)C1 c1(C(N2CCn3c(C)cnc3C2)=O)ccc2nc(C)c(C)nc2c1 N1(CC(C2CCOC2)OCC)C(=O)CN(CCc2ccccc2)C1=O C(N=c1ccnc(NCCc2ncccc2C)[nH]1)C1(C=C)CCCCC1 N#CC1(C(N2CC3(C2)CN(C(c2ncc(Cl)cc2F)=O)C3)=O)CCCOC1 C1(C(=O)NCCOCCN(C(=O)CCc2nncs2)C)CCC2CC2CC1 c1(NC(N2Cc3c(ccc(SC)c3)C2)=O)ccnc2c1ccn2C C(=O)(C(F)C(=O)NOCC(=O)NC1CCCCCC1)OCC CCC(C)C(C)C(=O)N(CC(CO)(CO)NC(=O)C=C1CCN(C)CC1)C N1(C(c2nc(CCC)oc2)=O)CCC(CNC(=O)C(C2CCC(=O)N2C)C)CC1 C(CNC(=O)C(C)SC)(CC(=O)NCC1(CO)CCCC1)OC c1(OCC(=O)NCCCC(C)NC(C2CC(NC)C2)=O)ccccc1[N+](=O)[O-] c1(CC)nc[nH]c1C(=O)NC1CCN(C(C2CCCC2C(N)=O)=O)C1 C12(C(=O)NCCN(CCC#C)C)CCC(CC1NC(=O)C(CC)SCCOC)C2 C(CC(C)(C)C(=O)N1CCCC(NC(N)=O)C1)SC.C12CCCCN1C2=O N1(C(c2c(C)c(F)cnc2)=O)CC(NC(C23CCC(C2)C3)=O)C2(CCC2)C1 C1(C(N(CCCCC(=O)NC(C)(C(N)=O)C2CC2)C)=O)CCC(C#N)CC1 c1(C(C)=O)cccc(NCC(C)(C)Cn2cc(NC(c3cnccn3)=O)nn2)c1 C=C=CC(C)C(=O)N1CCCC1CN(C(c1ccc(CNC(C)=O)o1)=O)CC c1(C(=O)NCC2(C)CCN(C(C3COCCO3)=O)CC2)ccc(S(N)(=O)=O)o1 O=C1Cc2cc(NC(CC3CCN(C(c4cccnc4Cl)=O)C3)=O)ccc2N1 c1(OC)ncc(C(=O)NCCCCCn2cc(C(C)(C)O)nn2)cn1 C1(NC(Cc2n(C)ncc2)=O)CCN(C(=O)CCCC2CCCC2)C12CCC2 C(CC(=O)NOCCCCC1CC1)(C(F)F)NC(COCC(N)=O)=O c1(OCC=CC(=O)NCCN(C(=O)CN2CCN(C)CC2)CC)ccncc1Cl.NCC c1(CCC(=O)NCC23OCCC(NC(CCSC)=O)(C2)C3)c(O)nc(=N)[nH]c1C N1(C(C2C(COC)C2)=O)CC2CCC(C1)N2C(c1cc(C2CCOC2)[nH]n1)=O C(=O)(N=c1[nH][nH]c2cc(Cl)ncc12)C1C(NC(C(C)SC)=O)COC1 Cc1cc(CNC(=O)CC2(NC(=O)CCCCC(C)C)CCC2)cc(C#N)c1 c1(N(CC(C)NC(c2cc(OC)c(Cl)cc2)=O)C)cc2nncn2cn1 C(=O)(C1=CS(=O)(=O)CCC1)NC(c1ccc(C)cc1)CNC(=O)Cn1ncnn1 C(C(=O)N=c1ccn(CCO)[nH]1)(C(C)(C)O)NC(c1c(C)nc(O)s1)=O C1(C(N2CCN(CC#C)C(=O)C2)=O)N(C(=O)CC2OCCC2C)CC12CCCC2 C1(CN(CCCNC(=O)Cn2cnnn2)CC)CCCCC1C(F)(F)F C(=O)(C1CCc2ccccc21)NC1(C)CCCN(C(c2oc(C)c(CO)c2)=O)C1 N1(CC(=O)NCCC2CC(NC(C34COCC3C4)=O)C2)CCCOC1=O c1(-c2cccc(C(NOC)=O)c2F)ccc2c(c1)CCN(C(=O)CCCCBr)C2 C1(C(=O)OC)CCCN1S(=O)(=O)NCc1nnc(C2CCCCC2)[nH]1 c1(N2CC(C)C(NC(c3nc(O)sc3C)=O)C2)nccc(C#N)c1[N+](=O)[O-] Cc1csc(CC(=O)N(C(Cc2cccnc2)C(=O)O)Cc2ccccc2)n1 C1(NC(C(=O)OC)=O)CCN(C)C2(CCC2)C1.C1(CC)CN2CCC1(C(F)(F)F)CC2 Cc1ccc(=O)n(CC(N2CCCC(NC(=O)C(S(C)(=O)=O)C3CC3)CC2)=O)n1 Cc1oc(Br)cc1C(N1CC(NC(=O)C(O)Cn2cncn2)CC(F)C1)=O c1(OC2(C(=O)NC(C(C)NC(=O)Cn3ccc(C(F)F)n3)C)CC2)ccc(Cl)cc1 c1(OCC)nc(Cl)ccc1C(=O)N(C)CCNC(c1cc(CC)ccc1C)=O CC(C)C(C#N)C(=O)N1CC(c2cccs2)(NC(=O)C(Cc2cnc[nH]2)C(C)C)C1 c1(COC)c(C(=O)NC2(c3ccc(C)cc3)CCOCC2)csc1C N1(C(c2cnc(COC)[nH]c2=N)=O)CCN(C(=O)CC2CC(F)(F)C2)CC12CC2 C1(C(=O)C(C2CCN(C3CCSCC3)CC2)=O)CCCC(N2CCC2)CC1 N1(C(c2cc(CC)n(C)n2)=O)CCCN(C(C2CC3CCCCCC23)=O)C(C)C1 c1(OC)cccc(CN2CCC(NC(=O)C(C)(C)C3CC3)C2)c1Cl c1(OC)cccc(C(=O)NCC2CCCN2C(=O)CC(C)NC(N)=O)n1 N1(C(C(CNC(C=CC(C)(C)C)=O)CC2CC2)=O)CCOCC2(CCC2)C1 N(C(=NCCCSc1ccc(F)c(OC)c1)N1CCS(=O)(=O)C(C)(C)C1)C(CC)C c1(OC(C(=O)NCCN(CCC)CCCC(F)(F)C(F)F)C)ccccc1Cl C(=O)(CC(F)(F)F)N(CC(C)CNC(c1cnc(C(C)(C)CF)o1)=O)C c1(C(C)(C)C)nc(N2CC(C(N)=O)C(C(N)=O)C2)c2cncc(Br)c2n1 N1(C(C(C)C#N)=O)CCC2(CCCCN(C(c3cnc4n3CCS4)=O)C2)C1 Cc1sc2ccc(Cl)cc2c1C(=O)NCC1CC1NC(c1ccc(C(C)C)[nH]1)=O c1(C(=O)NC(C)CNC(=O)C2CC2)[nH]ccc1CC1C2COCC12 C(=O)(C(O)C(F)(F)F)N(CC(C)C(=O)N1CCC1C)C N1(C(CCN(CCCCC)C)=O)CC2(CCN(C(C3NC(=O)C4CCC34)=O)C2)C1 N1(C(c2c(OC)scc2)=O)CCCN(CCNC(C2CC(C)C2C(F)(F)F)=O)CC1 c1(C(=O)NC2CC3CN(C(CCCC#C)=O)CC2C3)c([N+](=O)[O-])c(C)nn1C N1(C(c2cc(CC)ncc2)=O)CCN(C(=O)C(C)P(C)(C)=O)CC1CC(C)(C)C n1(CC(N2CC(OCCNC(CN(C(C)=O)C)=O)C2)=O)ncc(O)nc1=O C1(C)(C(=O)NCCCOC=C)CCCN(C(=O)Cc2ccccc2C#N)C1 N1(C(c2c(NCc3cccc(CC(=O)O)c3)ccs2)=O)CCc2ccccc2CC1 C(=O)(CC1=CCN(C)CC1)N(CCNC(C1OCCCO1)=O)CC C12(NC(c3[nH]cc(CC)c3)=O)CC(C1)N(C(C1CC(CC)C1)=O)C2 Cn1nc(C(=O)NCC(C2CCOC2)NC(c2cnnn2C)=O)c2c1CCSC2 Cc1cc(F)c(C(=O)NC2CCN(C(=O)CN(C)C(C)C)C2C)cc1F CC1CC2(CCN(C(=O)Cc3cnns3)CC2)CN1C(=O)C(O)C1CC1 C1(CNC(=O)C=CC2CCOC2)CC2COCC2N1C(c1ccc(O)nc1Cl)=O c1(C(=O)OC)ccc2nc(NC(=O)Nc3cncn3-c3ccccc3)sc2c1 C1(C(N2CC(CNC(c3[nH]nc(C(N)=O)c3Br)=O)C2)=O)CC2CSCC(C1)C2 N1(C(C2CCC(C)O2)=O)CCCCC1CCNC(=O)C=CC1CCC1 C(=O)(C(C)CNC(c1cocc1C)=O)NC(COCC)C Cc1nc(O)nc(O)c1CC(=O)NCCCC1(N(C(=O)CC2(C)CCCC2)C(C)C)CC1 C12(NC(c3c(C)cc(=O)oc3C)=O)CC(C)(C1)OC21CCN(C(=O)C(C)C)CC1 c1(C(N2CCN(C(C3CC(CC)C3)=O)CC2C)=O)cc2c(s1)CCOC2 C1(CC#C)(C(N2CCCCC2C)=O)CCN(C(=O)Cc2ccc[nH]2)C1 n1(CC(=O)NCC2N(C(COC(CC)C)=O)CCCC2C)cnc2ccccc12 N1(C(c2scc(C(C)=O)c2)=O)CC2(C1)CN(C(C1CCCNC1=O)=O)C2 C(=O)(CCCCC(N)=O)NCc1scc(CNC(c2cc(C)n(CC)c2C)=O)n1 Cc1cc(CN2CCCC(C(N3CCCC34CC4)=O)CC2)ccc1F C(CC1=CCN(Cc2cc3sccc3s2)CC1)NC(=O)C(C1CCOCC1)O N1(C(C(C)OCC=C)=O)CCCC(CO)(NC(c2ccc(F)cc2F)=O)C1 c1(C(=O)NC2C(NC(C3(COC)C=CCC3)=O)COCC2)cc(C#N)ccc1O CN1CC2(C)CN(C(=O)C(C3CCNCC3)F)CC2(C)C1 c1(C(N(CC(CC)NC(C2(COCC)CC2)=O)C)=O)cnc(COC)n1C Cc1cc(NC(=O)CC2C3CN(C(=O)CC4(C)CCOC4)CC23)cc(O)c1 n1(CC(=O)N(CCC(=O)NCC2CCCC(F)C2)CC#C)nc(C)ccc1=O c1(C(N2C(C)(C(=O)NC)CCC2)C(=O)NC2(C)CC2)cccc2nsnc12 C1(NC(c2cc(OC)nn2C)=O)CCCN(C(c2cc(CO)nnc2C)=O)C1C CC1CC(C)N(C(c2cnco2)=O)CCN1C(c1cc2nccc(Cl)c2s1)=O C(N=C(NC)N1CCC(OC)C1)C1(S(C)=O)CCC1.N1(C2CCC2)CCCC1 C(=O)(C(CO)C1CC1)N(CCNC(C(C)C)=O)C C1(NC(C2(CC#C)CCOC2)=O)CC2C1CCN2C(=O)Cn1nc(C)ccc1=O c1(C(N2CC(CCNC(c3cnc(C(=O)OCC)s3)=O)C2)=O)c(Cl)nn(C)c1Cl CC1CC(=O)NCC1C(=O)NC1(C)CCC(NC(=O)C(c2ccccc2)=O)CC1 CCCC(CC)CCC(=O)NCC1CC(NC(=O)C2=C(C)CC2)CCO1 C1(NC(C2C(NC(C3(CC=C)CC=CC3)=O)CC2)=O)CCC(C)(C)CC1 N1(C(Cc2c(C)n[nH]c2C)=O)CC2CCCC2(NC(=O)COCC(C)C)C1 C1(CCC)CCN(C(=NCC(C)(C)CC)NCCOCC2CC2)C1 n1(CC(=O)NC(C(C)C)C(C)NC(=O)CCc2cccs2)cc(F)ccc1=O C(C(CC(F)(F)F)NC(=O)C(C(C)(C)C)C1CCC1)NC(CC=C)=O c1(C(N2CCC(C(=O)OC)(COC)C2)=O)ccc(=O)n(C2CCCC2)c1 C1(CN(C(CC(C)c2ccco2)=O)C)COCCN1C(=O)Cc1cncs1 CCC(CC)(C(=O)N1CC2CC1C2NC(C1(C)CCCCCC1)=O)OC C1(C(=O)NCC2N(C)CCC2)CC(O)CN1C(=O)CC1CC2(CC2)C1 c1(N2CCCC(OC)C2=O)cc(NC(C(CC)C)=O)cc(C(=O)OC)c1Cl c1(NC(C(=O)NC(C(=O)NCC(C)C)C)=O)cccc2c1CNC2=O C1(C(CC)(C)C)CCC(C(=O)NCC2CCCCN2C(c2scnc2C)=O)CC1 CCC(C)C(=O)NC(C)CC1CN(C(=O)C=C2CCC(C)C2)C1 CCC(C)CCCC(=O)N1C2CCC1C(C(=O)NCc1nc(C)c(C)[nH]1)C2 c1(CNC(C2(F)CN(C(CCc3cnc(C)s3)=O)C2)=O)ccc2[nH]ccc2c1 c1(C(COC)(C)O)cn(CCCC(=O)NCc2nc(C(=O)O)co2)nn1 C1(NC(C(F)=CC)=O)(COC)CCN(C(=O)Cn2cnnc2O)CC1 C12(C(N3CCC(N(CCC)C(c4coc(Cl)n4)=O)C3)=O)CC(CO)(C1)OC2(C)C Cc1cccc2ccc(C(=O)N(CC(C)NC(=O)C(Cl)=CCl)C)nc12 c1(C(=O)OC(CC)C(=O)OC(c2cnc(C)s2)C)cc(C)ccc1NCC c1(-c2nc(N(CC#C)CC)sc2)ccccc1F.C(F)(F)F c1(C(=O)O)ccc(N)c(Cl)c1.C1(CN(CCCN(C)C)C(=O)CS)CCCC1 N1(C(C(=O)OC)=O)CC2CC2(C(=O)NC(CC(=O)NC)C)C1 C=Cc1cnn(C)c1C(N1CCCC(CNC(=O)C(C)(CO)OC)C1)=O c1(C(=O)OC)cccc(C(=O)NC2CC(C)(NC(c3ccncc3C)=O)C2)c1OC C1(C(=O)NCC(CN(C(C(CCCCC)O)=O)C)C)CC(c2ccccn2)=NO1 c1(NCCNC(CC)=O)nccc(=NC(CCCO)c2ccccc2)[nH]1 CC(C)(C)C(C#N)C(=O)NC1(C(=O)NC2CS(=O)C2)CC1 C=CCCC(CC(C)C)C(=O)NCC(CC(C)C)NC(=O)C(=O)Cc1ccsc1 C12(CNC(C(C=C)(C)C)=O)COCCN1C(=O)CN(C(c1nonc1N)=O)C2 N1(C(c2ccn(COC)n2)=O)CCC2(CC2NC(=O)CCN(S(C)(=O)=O)C)C1 Cc1noc(C)c1C(=O)NCC=CCC1(O)CC(C(N2CC2)=O)C1 C(=O)(C1=CCCN(C(C(=O)NC2CC2)C(C)CC)C1)OC NC(=O)CC(C(=O)NCCC1CCCC1O)NC(=O)C1=CCSC1 N1(CC)CCCCC1C(=O)NC(C)(CNC(c1c(C2CC2)noc1C)=O)CSC Cc1ccc(I)c(C(=O)NCC2CCN(Cc3ncsc3C)C2)c1 C(CC(=O)NNCc1cn(C2CCOC2)nn1)NC(=O)OC(C)(C)C C1(CNC(C(C)C)=O)C(C2CC2)CCN1C(c1cncn1C)=O CCCCC(CC)C(=O)N1CC(F)(C(=O)NC(C2CSC2)C)C1 C12(NC(Cn3ncc(C)c3)=O)CCCC(CN(C(=O)CCc3ncc[nH]3)C1)C2 c1(C(CC)C(=O)NC2CCC2NC(=O)CCc2nncs2)cc(F)c(F)c(F)c1 CC(CCCCNC(=O)CC1(O)CCC1)NC(c1cnn(C)c1C(F)(F)F)=O C(=O)(CC(O)CC(C)C)N1C(COC)(CNC(=O)C(C)(C)C2CCC2)CCC1 CCCCCCC(=O)N1CCC(CF)(NC(C2CCN(CC)C2)=O)C1 c12ccc(cn1)C(=O)NC2.C1(O)(CNC(C2CCC(CC)C2)=O)CCCCC1.C1(C)CC1 Cc1nc(=N)[nH]c(C)c1C(=O)NCC1(O)CN(C(C23CCCN(CCC2)C3)=O)C1 N1(C(C(=C(C)C2CC2)F)=O)CCN(C(=O)CNC(c2cscn2)=O)CC1C(C)C C1(NC(CC=CC)=O)CN(C(=O)C(CC)C2CCC(=O)N2)CC1(C)C Cc1ncc(NCc2nnn(C)c2C(F)(F)F)cc1C(N)=O C#Cc1ccc(CC(=O)NC(CNC(=O)Cc2ccco2)C(C)C(C)C)cc1 c1(C(=O)NCCC(C)CCNC(C2(C)CCC(=O)C2)=O)nnc(O)nc1O CC(C)C(F)(F)CC(=O)N1CCN(C(C2CC2(C)C)=O)C(CN(C)C)C1 N1(C(c2c(CCC)nco2)=O)C2CCC(C(=O)Nc3ccc(CO)cc3)C1CC2 O(N1C(=O)c2ccccc2C1=O)CC(N1C(CCC)CC1)=O C1(CNC(C(C)(F)F)=O)CCC2(CCN(C(C3CC(C)(O)C3)=O)CC2)CO1 N1(C(c2cc(C)c(C)s2)=O)CC(NC(c2ccn(C(C)C)n2)=O)CC(F)C1 C1(CC)C(C(=O)NCc2cc(OC)n(C)n2)CCCN1C(=O)CN1CCSCC1 C=C(C)C(O)CC(=O)N1CCN(C(=O)C=CC(c2cccnc2)=O)C(CCC)C1 CON(CCC(=O)NC(C)CC(C)(C)OC)C(=O)C1C2CCC(F)(F)C12 c1(C(=O)NC2C(NC(CC(CC)(F)F)=O)CC2)cc2ccc(F)cc2nc1C Cc1c(C(N2CCCC2CNC(C2(F)CCC2)=O)=O)cnn1-c1cccc(F)c1 c1(C(=O)NC(CC)(C)CNC(=O)C(C(C)O)N(C)C)ccc(=NC)[nH]c1 c1(NC(C(=O)NC(CNC(CC2N(C(C)C)CCC2)=O)(C)C)=O)ccc(Cl)cc1 c1(CNC(C2(C3CCCO3)CCC2)=O)cccc(Br)c1F CCCCC(O)C(=O)N1CCCC1C1(C(=O)NCCC(C)(C)O)CC1 N1(C(C2CCC(=O)C2)=O)CCC(C2CC(NC(C3CCCCC(=O)N3)=O)C2)CC1 c1(CC(=O)NCC(C)(C)CNC(c2cn(C(C)(C)C)nn2)=O)ccc(O)nc1 C(CCCC(=O)NCCC1(O)CCN(C(C2C=CCCC2)=O)C1)OC(C)C c1(C(=O)NCC2(C(=O)NCC(=C)F)CCC2)cc(Cl)c(N)cc1F c1(C(N2CCCC(O)(CNC(C(C)OCC)=O)C2)=O)cnc2c(c1)COC2 N1(C(C2CC2C2N(C(Cn3c(C)ncc3)=O)CCC2)=O)C2CCC1CN(C)C2 CCC(C)(CO)C(=O)N1CCN(C(c2ccc(C)c(Cl)c2)=O)C(C(C)C)C1 N1(C(=O)CCCc2nccs2)Cc2ccccc2C(c2cccs2)C1 c1(C(=O)NC2C(CNC(C(C)(C)COCC(F)F)=O)C2)c(F)cc(C#N)cc1F Cc1cnc(-c2cn(CC3CN(C(=O)C(c4ccc(Cl)cc4)C)C3)nn2)nc1 CN1CCN(C(c2cncnc2)=O)C(CNC(c2csc(C(N)=O)n2)=O)C1 c1(CC(=O)NC2CCN(C(COCCC)=O)C2CC)ccc(C)cc1Cl c1(OC)n[nH]cc1C(=O)NC(CO)C(=O)N(C1CC1)Cc1ccoc1 CC(C)C(C(=O)NCC1CCCCC1NC(c1ccc(Cl)nn1)=O)n1cnnc1 c1(OC)cc(C(=O)NC2CN(C(=O)CNC(=O)NC3CC3)CCC2O)cnc1F C1(C(=O)NC2CC(CNC(C3N(S(C)(=O)=O)CC3)=O)C2)CCS(=O)(=O)C1(C)C C1(NC(CCCC)=O)CCN(C(=O)CC2(N(C)C)COC2)C(C)C1 C1(NC(C=CCOC)=O)COC(C)(C)CN1C(=O)C(=O)NCCOCC(F)(F)F CN(CCNC(C1CCCCC1)=O)N1CC(c2nncs2)C1 C(=O)(C(C)(C)CC(=O)NCC(C(N1CC(C2(C)CC2)C1)=O)N(C)C)N(C)C C=CCCCCCCCNC(c1ccc(O)c(Br)c1)=O C1(CNC(C(CCO)N(C)C)=O)CCCCN(C(=O)C(N)=O)C1 CCCCC(C(=O)NCC1CC(NC(C2CSCN2C(C)=O)=O)C1)C(C)C C(=O)(C1Cc2ccccc21)NCCC(C)NC(c1cc2c(ncn2C)s1)=O C(=O)(C1=CS(=O)(=O)CCC1)NCCC1N(C(C2(C)COC2)=O)CCSC1 c1(C(=O)NCCCN(C(=O)CCCCC2CC2)C)cc(C#N)cn1C c1(OC)cc(F)c(C(=O)NC2CCN(C(c3cc(O)ccc3Cl)=O)CC2)c(F)c1 N1(C(CSCCOC)=O)CCOCC(C(=O)N(CC(C)(C)COC)C)C1 C1(SCC)CCC(C(N2CC(C(C)NC(C3(F)CCOC3)=O)C2)=O)CC1 C1(OCC(=O)NCC2CC2CNC(=O)CN2CC3CC3C2)CCCCCC1 c1(CN(C(=O)NCC(c2cccc(Cl)c2)(CC)O)C)ccc(CC(=O)OC)cc1 Cc1ccc(C(=O)NCCN(C)C(c2ccc(C3CC3C)o2)=O)c(C)n1 C(=O)(CC(C)C(F)F)NCCC(=C)CNC(=O)COc1cccc(C(C)(C)C)c1 CCC(CC)(CC)C(=O)NC1CNCC1(C)c1nc(-c2ccc(F)cc2)no1 N1(C(C2C=CCN(C(c3n(CC#C)ccc3)=O)C2)=O)CCOC(C)C1C C(=O)(C(C)(CO)OC)N(CCN(C(=O)Cc1cn(CC)nn1)CC)CC C(N=c1[nH]c(=NCCC2(C)CCCO2)[nH]c2c1CSC2)C1(C)CSCCO1 c1(C(=O)NC2C(NC(C(CC)SC)=O)CCCC2)c(N)cccc1[N+](=O)[O-] c1(OC)cc(OC)cc(CNC2(c3nnnn3C)CCCCC2CC#N)c1 N1(C(C2(CC)CCC2)=O)CCOCC(NC(c2cccc(CO)n2)=O)C1 c1(C(c2nnnn2CC2CCOCC2)NCCOCCO)cnccn1 C1(C(=O)NCCN(CCC)C(c2cccn2C)=O)CCCC1S(C)(=O)=O CCS(=O)(=O)C=CC(=O)N1CC2(CCN(C(=O)Cc3cc(Cl)ccc3Cl)C2)C1 c1(C(=O)NC2CC(F)(CNC(C(C)N(C)C)=O)C2)cnc2c(cnn2C)c1 Cc1ccc(F)c(S(=O)(=O)SCCNC(=O)NC23CC(C)(C2)OC32CCC2)c1 c1(C(=O)NC2CC(F)(CNC(C(C)C3CCOC3)=O)C2)ccc(=N)[nH]c1Cl CC(C(=O)NC(C1CCCCC1)CNC(=O)COc1cccc(Cl)c1)C(F)(F)F C(=O)(C1=CC2CCCCCC12)NC(CNC(c1c(C)c(F)c(F)cc1)=O)(C)C C1(C)(NC(CC2CC(=C)C2)=O)CCCCC1C(=O)N(CC(F)F)C1CCC1 C1(C(=O)NC(c2cccnc2)C(=O)NCCC2(C)CCCC2)CC1C1CCCC1 N1(C(C2C3C(NC(C(C)c4ccco4)=O)C4C(C3)C42)=O)CCC2(CCSC2)C1 Cc1cc(C(N2CCOCC2CN(C)C(c2ccc(F)cn2)=O)=O)c(N)cc1F C1(C(=O)NC2(COC)CC2)CCN(C(c2ccccn2)=O)C1C(C)C C1(NC(c2c(C)csn2)=O)CCC2CCN(C(c3cnc(CC(C)(C)C)o3)=O)C12 Cc1cc(CC(=O)N(C)CCOCCN(C(=O)CCF)C(C)C)cs1 c1(C(=O)NC(NCC(C)(C)CC2CCC(C(=O)OC)CC2)=O)cccc(Cl)c1Cl c1(C(N(C(c2nnn(C)n2)=O)C2CC2)=O)cc(Cl)ccn1.C12CCN(C1)C2 N1(C(Cn2cc(CNC(C(C3CC3)OC)=O)nn2)=O)CC(CO)CC1(C)C N1(C(CC(=C)Cl)=O)C(CC(N2CC(N3CCC3)C2)=O)C2CCCC12 CC1CCC(Cl)=C(C(=O)NCCNC(c2cccc([N+](=O)[O-])c2O)=O)C1 C(=O)(C1=NOC2(CCC2)C1)NC1(COC)CCN(C(c2ccsc2C)=O)C1 CN1C(=O)CCCc2occ(C(=O)N(C)Cc3cn(-c4ccnc(F)c4)nn3)c21 c1(CC)nc(C)ncc1C(=O)NCC1CC1NC(c1ccc(OC)nc1Cl)=O c1(C(N2CC(OC)(CNC(=O)CC3CC3(Cl)Cl)C2)=O)cccc2[nH]ccc12 CC(CC(C)(F)F)C(=O)N1CC2CC(O)C1C2NC(c1ccn(CCN(C)C)n1)=O Cc1ccc(O)c(C(N2CCC(N(C)C(C3CCOC3C(C)C)=O)C2)=O)n1 C1(NC(c2n[nH]cc2I)=O)CCN(C=CC(=O)Oc2ccc(OC)cc2)CC1 Cc1ccc(CCC(=O)N(CC(C)N(C(=O)CC2(C(F)F)CC2)C)C)s1 c1(C(C)C)ccccc1C(N1CC(NC(c2nnn(C)n2)=O)CC1C)=O N1(C(COCCCCC)=O)CC2CC1CCC2NC(C1CC2(CSC2)C1)=O C1(C(=O)NCC=CCNC(C2C(C(C)C)OCC2)=O)CCC(=O)N(CC(F)(F)F)C1 C1(C)(NC(c2c(C)ncnc2)=O)CCCN(C(=O)CC(c2cccc(F)c2)C)C1 C1(CC(=O)NCCOc2cccc(Br)n2)CCc2sccc2C1=O C1(NC(C=CCNC(CCc2n(C)ncc2)=O)=O)CCCCCC1O C(=O)(C#CC1(CC)COC1)N1CC2C(C(=O)NCc3ccc(SC)o3)(C2)C1 C1(F)(C(N2CC(NC(C(C(CC)O)C)=O)C3(C2)CC3)=O)CCC(F)(F)CC1 N1(C(C#CC2(C)CC2)=O)CCN2C(=O)C(NC(c3cnccn3)=O)CC2C1 C12(CCNC(c3cc(C)on3)=O)CCC1CN(C(=O)C=C(C1CC1)C1CC1)C2 c1(C(N(C2CCCC(NC(c3ccccc3CC#N)=O)C2)C)=O)cnc(=N)[nH]c1 CN1C(=O)CC(C(N2CCCN(C(=O)CC(C)(F)F)CC2)=O)C1c1nccn1C C(=O)(C(C)(O)C(C)C)NC1CC(CCC(=O)Nc2ccc(OCC=C)cc2)C1 N1(C(C(C)(C)C2CCCCO2)=O)CCC(NC(C23CSC(C2)C3)=O)C(C)(C)C1 S(=O)(=O)(c1cc(Br)c(C(=O)NOCc2ccc(C)cc2)cc1Br)NC(C)=O C1CC12CCC2.CC(C(C)NC(=O)COC1CC(NC(=O)CN(C)C)C1)n1cccn1 C(=O)(CC(CCC)NC(=O)CCCCCF)N1CC(OCC#C)C1 C1(OC)CCCC(C(N2CCC(C(=O)N(C)Cc3n[nH]c(C)n3)C2)=O)C1 N1(C(CSCCC)=O)CCC(NC(C2CC3(CC3)CO2)=O)CC1c1ccccc1 C1(C)(C(N(CCCO)CCC)=O)CCCN(C(c2ccc(F)s2)=O)C1 c1(C(CNC(C)CN2CCOCC2)N(C)C)ccc(Cl)cc1 C=CC1(CC(=O)N(C2CCCC(NC(=O)CC3CCC3)C2)C)CCCCC1 Cc1sc(C)c(S(N)(=O)=O)c1NC(N1CC(N2CCOCC2)CC1C)=O C1(C(=O)NCCCN(C(=O)CCC2CC(F)(CO)C2)C(C)C)CCC(C)C1 c1cc2ncc(CNC3CCCCC3c3ccccc3)cn2n1 c1(OC)ccc(C(=O)NCC2CN(C(C3(C#N)CC(=O)C3)=O)CC2O)c(F)c1F C(=O)(C(C(C)C)NC1CCC(NC(=O)Cn2cnnn2)C1)NCc1snc(C)n1 C1(CC)CCCCC1OCC(=O)NCC1CCC(NC(c2sncc2Br)=O)C1 C(=O)(CC(C(C)OC)NC(C1CC2C=CC1O2)=O)NCC(C#C)OC C(CN=[N+]=[N-])(C(=O)NCCCc1ncn(C)n1)NC(c1c[nH]c(=NC)s1)=O C1(N)CCOC12CCOC2.N#Cc1nccnc1N1CCN(c2ccccn2)CC1 c1(CC(N2CCC(CC(=O)NCc3cccc(Cl)n3)C2)=O)cc(F)cc(Br)c1 C(CCN(C)C(C1(P(C)(C)=O)CC1)=O)(C(C)(C)C)NC(C1C(C)CCO1)=O C1(C(N(C(CCCC(=O)OC)=O)CC(C)N(C)C)=O)CCn2cnnc2C1 C1(NC(C2CN(CC(C)C)C2)=O)CCN(C(=O)CCP(C)(C)=O)CC1(C)C C#CCC(C)(C)C(=O)NC1CC(C)CN(C(=O)CCCc2ccc(F)cc2)C1 c1(CC)ccc(C2C(=O)N2)o1.N1(C)CCC1(C)C(=O)OC.C(C)(C(=O)OC)OC C(=O)(CC(N)Cc1ccc(Br)cc1)N(CC)Cc1ccc(Cl)s1 C(=O)(C1=CCC1)NC1(CCCCNC(C(C)c2cccs2)=O)CC1.CC(O)C1CC1 C1(N(C(=O)CC2CCC(C(F)(F)F)O2)CC#C)CCN(C(C2(F)CCC2)=O)CC1 C1(N(C(CC=CCNC(C2N(CC)CCCC2)=O)=O)C)CCCCC1(C)C CCCC(C(=O)OC(C)(C)C)OC.c1(C2C(=O)O2)ccc(F)cc1 CCCC(F)C(=O)NCCC1(NC(C2CCCN(CCC)C2)=O)CCC1 c1(CC(=O)NCC2CN(C(CC(C)c3cccs3)=O)CC2O)cc(F)ccc1O n1(CC)ccc(CC(=O)NC2CCCC2NC(=O)Cn2cc(CO)nn2)n1 C(c1ccccc1[N+](=O)[O-])=CCNC(C1CC(O)C1n1cccn1)=O C(C1COCc2ccccc21)NC(C1CC(n2cc(CC(C(C)C)O)nn2)C1)=O c1(CC2(C(CC)=O)CC2)ncnn1C.N1(C=O)CC(NC(CCOCCOC)=O)C1 c1(C(N(CC(CN(C(CCCC(C)=O)=O)C)O)C)=O)cc2c(F)ccc(F)c2[nH]1 C(=O)(C(CC)C(=O)N(CCCOCCNC(=O)CCc1ncc(C)[nH]1)C)OCC NC(=O)CCCNC(C1(CC(C2CC23CCC3)=O)CCCO1)=O C1(=O)NNC(=O)NCCCOCCS1.c1(-c2[nH]c(=N)sc2)cccc(OC(F)F)c1 CC1(C)CCC(CC(=O)NC2(CNC(C3CCSC3)=O)CCCC2)CC1 C1(C(=O)N(CCCC(C)O)C)(CC)CCCN(C(=O)C=CCF)C1 c1(C(N(C)CC2(O)CCN(C(C(C)SC(C)C)=O)C2)=O)ccc2c(c1)CCO2 c1(NC(=O)NC(c2ccn(C)c(=O)c2)C)cc(O)nc(OCC(F)(F)F)n1 CC1(CN=c2[nH]nc(C3CC3)o2)CCCN(C(=O)Cc2cncnc2)C1 S(=O)(=O)(c1cc(F)ccc1N1CCCN(C)CC1)N1C(c2cccc(C)c2)CCC1 c1(OC)ccnc(C(=O)NCCN(C(=O)CCSC(F)(F)F)C)c1OC N1(C(CC(CC)C)=O)CCC2(CC1)CN(C(c1nc(Br)c[nH]1)=O)CCO2 C12CCN(CC1F)C2=O.c1(CNC(C2CC(=C3CC3)C2)=O)cnn(CCF)c1 c1(-c2cn(Cc3nccc(OC)c3)nn2)ncc(C#N)cc1C S(=O)(=O)(c1csc(C(=O)NC2CCCC2CNC(c2cc(OC)ns2)=O)c1)NC Cc1cc(C(F)F)n(CC(=O)NCC2COC(CNC(=O)C(F)(F)C3CC3)C2)n1 c1(C(=O)NC2(CNC(CCCOCC=C)=O)CC2)ccc(Br)c(N)c1 C1(C)(C(=O)NC(CNC(C(C2CCCC2)OCC)=O)CC)CCOCC1 CC(CCCNC(C1CC(CCO)C1)=O)NC(=O)Cn1nnc(-c2cccs2)n1 CC1(C(=O)NCC2CCC(NC(=O)C(F)(F)CC3CC3)C2)CC2CC2C1 n1(CC(=O)NCC2CC2CC(N2CCOC(CN3CCC3)C2)=O)cccnc1=O C(=O)(CC1=NNC(=O)C1)NC1CCCN(C(c2nc(CC)oc2)=O)C1C CCC(C)C(O)C(C)C(=O)N1CC(F)CC1CNC(c1coc(C)c1)=O C12(C(=O)NCC)CCC(NC(=O)C3=C(C)OCCC3)(CC1)CC2 C1(C(=O)NCc2occ(C(N(C3(COC)CCC3)C)=O)c2)CC2CCC(C1)O2 N1(C(=O)Cc2cc[nH]n2)CCC2CN(C(c3sccc3-n3cnnn3)=O)CC2C1 c1(C(CC(=O)NC2CC2NC(=O)CN(CCNC(N)=O)C)=O)ccccc1Cl c1(C(N2C(CNC(C=C(C)c3cccs3)=O)CCCC2)=O)ccc(=O)n(C(C)C)c1 N1(C(CCCC)=O)CCN(CC(=O)NCC(F)OCF)CC1 c1(C(C)C)ccoc1C(=O)NC(C)CC(C)NC(C1CC(CC2CC2)C1)=O c1(C(=O)NCC(CO)NC(CCc2ccc(C)s2)=O)ccc2sccc2c1 C=CCS(=O)(=O)CCNCc1cnc(OC)cc1F C(=O)(C(C(C)O)NC(C1(C)CCOCC1)=O)N1C(CCC)CCC1 C1(C(N(CCCNC(C(C)N(C2CCCC2)C)=O)C2CC2)=O)COCC(C)(C)O1 CC1(C)CCC(C(=O)O)(NC(C2C3CCN(CC4CCCCC4)CC23)=O)C1 N(C1CCCn2c(C)nnc21)C(c1cc(C)n(-c2cccnc2)c1C)=O N1(C(C(CCC)S(N)(=O)=O)=O)CCC2CC(NC(=O)CCCCSC)CCC2C1 c1(OC)ccc2c(c1)OCC(C(=O)NC(C)(CNC(=O)CC(F)F)C(C)C)=C2 c1(OC)ccc2c(=NC(C)c3cc[nH]n3)[nH]c(=NCC(C)(C)C(F)(F)F)[nH]c2c1 N1(C(c2cc(C3(C)CC3)on2)=O)CCC2(NC(C3CCC=CCC3)=O)CC2C1 C(C)(C)(CCCC(=O)NCc1c(C)cnn1C)NC(CCC=CCC=C)=O c1(CC)cc(=NC(=O)Nc2cc3nc(Cl)ccc3o2)[nH]n1C C(C1CCCC1)=C(C)C(=O)NC1CCC(C(=O)NCCCc2ncnn2C)C1 C1(C#CC(=O)NCCCOCCN(C)C(C2(C)CCCN2C)=O)(CC)COC1 CCC(COC)(CC)C(=O)NCCC1=CCN(C(c2snnc2C)=O)CC1 C1(C)(CNC(COCC)=O)CC(F)(F)CN1C(c1cc(C)cc(Br)c1O)=O C1(CNC(C23CC2CNC3)=O)CC(O)(Cn2cccn2)C1 Cc1nc(CC(C)C)oc1C(N1CC(NC(=O)CCCn2ccnc2)C(O)C1)=O CC1CC=C(C(=O)N2CCCC2C2(O)CN(C(C3(F)CCC3)=O)C2)CC1 Cn1cc(C(=O)CNC(=O)C(F)(F)c2nccn2C)cn1 c1(C(=O)OCC)cccc(C#CCNC(CCO)C(C)(C)C)c1 C12(CC(=O)NCC(C)(O)CNC(c3ccc(F)s3)=O)CCC(CC1)C2 c1(CC)ncc(C(C(=O)NCCCC2CC2)N(C)C2CC2)cn1 CC(C)CCCC(C)C(=O)NC1(C(=O)NCCCCCC2CC2)CCC(C)(C)C1 CC1(C)CC(=O)NC1CNC(c1c[nH]nc1CNC(C1CC2(CCO1)CC2)=O)=O C(CCNC(C1COC1)=O)(C(C)C)NC(C(C)(C)N(C)C)=O C=CC(C)(C)CC(=O)NCC(c1ccc(C)cc1)NC(=O)COCC(=O)NC Cc1cc(C(=O)NC(C2CCCCC2)CNC(=O)C(C)OC2COC2)cs1 C(=O)(N=c1[nH][nH]c2c1CN(C(c1ccc(Br)cc1)=O)C2)c1ccc(C#C)cc1 CN=c1nc(N2CCC(COC)C2)[nH]c(=NCc2ccc(CSC)cc2F)[nH]1 C1(C(=O)NC(CC=O)=O)CCC2(CCC2)C1NC(C1CCCC1)=O.C1(NCCO)CC1 CC1CC2CN(C(c3ccc(C4CC4)s3)=O)CC2N1C(c1ccc(CO)cc1)=O Cc1cccc(C(=O)NC(C)(C)CCN(C)C(C2CCC(C(N)=O)N2C)=O)c1Cl CCC(CC)CCC(=O)N1CCC(O)(CCNC(C2(CC)CC2)=O)CC1 Cn1c(C(N2CC(C(=O)NCC3CC3[N+](=O)[O-])CC2(C)C)=O)cccc1=O C1(C(F)(F)F)(C(=O)NCC(C)N(C(=O)CCC2CC2(C)C)C)CCO1 CCCCCCC(C)C(=O)NCCCCCCNC(c1ccc([N+](=O)[O-])[nH]1)=O N1(C(CN(C2CCC2)C)=O)CC(C(F)(F)F)CC1C(=O)NC.c1(C2(C(Cl)(Cl)C)CC2)ccno1 C1(CNC(Cc2ccn(C)c2)=O)(CO)CC12CCN(C(C1CC(F)C1)=O)CC2 N1(C(c2c(SC)cccc2)=O)CC(NC(=O)CC2(C)CCCO2)C2(CCC2)C1 n1(CC)ccnc1C(=O)NCc1cc(C(C)C)n[nH]1 N1(C(c2cc(OC)nc(OC)c2)=O)CCN(C(=O)C#CC(C)(C)C)CC(C)(F)C1 C(CCCCC(=O)NCCc1csc(C)n1)NC(C1(CCOCC)CCC1)=O c1(CN(CC(=O)NCC(C)(C)CNC(=O)COC(F)F)C)ccc(C)cc1.CO C=Cc1ccc(C(N2CC(NC(C3CC34CCOCC4)=O)CC(F)C2)=O)cc1 C1(CC(=O)NCC2(NC(C3COCCO3)=O)CCC2)CCCC(F)(F)C1 C1(NC(c2c(CC)cc(Cl)cc2)=O)CCN(C(=O)CSC2CCOC2=O)C1(C)C C#CCC(C(=O)N1CC(F)(F)C1C1CC1)NC(=O)CCC1CCCOC1 O=C(C=C(Cl)Cl)NC1CC(F)(CNC(c2cnn[nH]2)=O)C1 C1(CC)(OC)CCN(C(=O)NC(C2CC2)C)C1 CCC(C(=O)NCC1CCN1C(c1sccc1C(C)(C)C)=O)Oc1ccccc1 C(C(O)C(=O)NC1CC(O)C1CC(=O)NCCc1c[nH]nc1C)=CC C1(CNC(NC(C)CN2CCCC2)=NCC2CC3(CC3)C2)COC2(CCCCC2)O1 Cc1cc(C)c(NC(C2(F)CCN(C(=O)CC(=O)NS(C)(=O)=O)CC2)=O)c(C)c1 N1(C(c2c(C)noc2)=O)CCCC(C)C1CNC(c1coc(O)n1)=O c1(C(=O)NCC(C)(C)CNC(C2SC3C=CC2C3)=O)ccc([N+](=O)[O-])nc1 Cc1cc(C(=O)NCCCNC(=O)C2=NOC(C(C)(C)C)C2)ncc1F C1(NC(C2N(CC)C(=O)CC2)=O)CC(O)CN(C(=O)CCN2CCN(C)CC2)C1 c1(C(N2CC(C(=O)NCc3n(C)ccn3)C(F)CC2)=O)cc2c(cn1)OCCC2 C(=O)(CCCCCN(C)C(C1CC2CCC1CC2)=O)NCC(c1nccs1)C CC#CCC(C)N=c1[nH]c(=NCC2CCS(=O)(=O)C2)[nH]c2cc(OC)ccc12 C1(CC)CN(C(C2CCCS2)=O)CCN1C(c1cncc(-c2ccco2)c1)=O C(=O)(C(CC(C)C)NC(=O)Cc1c(C)cnn1C)NCC(=O)NCCOCC C1(CN2C3C(C(=O)NC4CC(C(N5CCCC5)=O)C4)C(C3)C2)CC1C1CCCC1 c1(C(=O)NCCN(C(=O)CSCC(C)C)CC)cnc2n1CCS2 C1(CC(=O)NC(C#C)(C)C)CCN(C(=O)C=CCN(C)CC)C1(C)C C1(C(C)CNC(c2cnccn2)=O)CCN(C(C2NC(=O)C3CC23)=O)CC1 C#CCCCCC(=O)NC1(CNC(C23CC2COC3(C)C)=O)CCCCC1 Cn1cc(Cl)cc1C(=O)NC1(C)CC(NC(C2(CC3CC3)CCCO2)=O)C1 c1(C(=O)NCC2(O)CC(NC(C(CC#C)C3CC3)=O)C2)ccn(CC)c(=O)c1 c1(CNC(CCCC(C)NC(c2csc(Cl)c2)=O)=O)ccc(C)c(C#N)c1 c1(CNC(C(CNC(C2CC3CC(=O)C2C3)=O)CC2CC2)=O)cc(F)cc(F)c1 c1(NC(=O)CCOC2CC(CNC(C(CCC)O)=O)C2)cccc(Cl)c1Cl O=C(NNC(=O)c1cccc(C(F)(F)F)c1)c1cccc(NS(=O)(=O)C2CC2)c1 C1(C(=O)NCCCCN(C)C(c2cccn2C)=O)CCC1(F)F N(C1CCc2c(F)cccc21)C(=O)NCCC1(OC)CCC1 Cc1c(N)ccc(C(=O)N(C)CCN(C(=O)C(C)N2CCC2)C(C)C)c1C CCCC(CC)CCC(=O)NC(C)(CNC(=O)Cn1cncn1)CC Cc1ccc2c(c1)C(=O)NCC2NC(=O)NC1CCOC(c2cccnc2)C1 C1(N(C(=O)CN(c2ccon2)CC)CCC)CCN(C(c2ccccc2)=O)C1 N1(C(c2c(C)nc(C)n2O)=O)CC2CCCC2(CNC(C2CCS(=O)(=O)C2)=O)C1 N1(C(c2c(CNC(C(C3CCC(=O)N3)C)=O)occ2)=O)CCC2CCCC12 CCCCC(C(=O)N(C)Cc1cc(=O)cc[nH]1)NC(C1CCC(=O)C1)=O CCC(C(=O)NCC(O)CSC)c1ccco1.C1CO1.C(C#N)O Cc1cc(C)n(CCCC(=O)NCc2ccc(C(C)NC(=O)CC(C)O)cc2)n1 c1(C(CNC(C2(CC=C)CC=CC2)=O)NC(=O)CCC2CCCC2)ccc(F)cc1 c1(CC(CCC)NC(=O)NC(c2cncnc2)C)ccc(F)cc1F c1(C(=O)NCC(C(N2C(C(=O)NC)CC(C)C2)=O)N(C)C)c(C)[nH]c(C)c1C c1(C(N2C(CC(=O)NCC3(OC)CCCOC3)CC2)=O)cc[nH]c2nccc1-2 c1(CNC2(CC(=O)Nc3ccc(CN)c(Cl)c3)CCC2)ccc(F)c2ccccc12 c1(NC(C2N(C(c3c(C)ncnc3)=O)CC(F)C2)=O)ncc([N+](=O)[O-])cc1F N1(C(CCC=CC)=O)CC(NC(=O)Cc2cc(Cl)ccc2O)CC12CCC2 CC1CC(NC(=O)C=Cc2ccsc2)CN1C(c1cc(Br)no1)=O c1(C(=O)NC2C(NC(CS(CCOC)(=O)=O)=O)CCC2)ccc2sc(C)nc2c1 N1(C(C(C)S(C)(=O)=O)=O)CC2CCCN(C(c3ncsc3S(N)(=O)=O)=O)C2C1 C(=O)(CC(CC)C(C)(C)C)N1CC(N(C(=O)CNc2cccc(F)c2)CC)C1 c1(C(=O)NC2CC(Nc3ccnc(Cl)n3)C2)cc2c(nc1O)CCCC2 CC12CN(C(C3(Br)CC3)=O)CC1(C)CN(C(c1cnn[nH]1)=O)C2 CC(C)(O)C(C(=O)N(C1CCCN1)Cc1ccccc1)NC(=O)OC(C1CCC1)=O N#Cc1ccc(CN2CC(C(=O)Nc3ccsc3CO)CC(F)C2)c([N+](=O)[O-])c1 CC(CC(F)F)C(=O)N1CCC(CN(C(=O)CCCC2CCCC2)C)C1 C(=O)(C(C)(C)C(F)(F)F)NC1CC(C(C)NC(=O)CCOCCN(C)C)C1 CCC(CN(C)C)CC(=O)N1CCN(C(=O)Cc2nc[nH]n2)C(C2CC2)C1 c1(C(N2C(CC)CC(NC(C3CC3F)=O)C2)=O)cc(CC(C)C)nc(O)c1 c1(NC(c2cc3cnccc3[nH]2)=O)cc(C(F)(F)F)cc(Cl)c1F.N12C3CN1CC23 c1(OC)cnc(N2CCN(C3CCN(c4ncccn4)CC3)CC2)nc1 N1(C(C2C(CC)OCC2)=O)CC(CC(=O)NCc2ccsc2)CC1(C)C C(C(C)(O)CC(=O)NC1CCC1NC(=O)C=CCN(C)Cc1ccccc1)OC c1(C(N2CC(CNC(CC3C=NN(C)C3=O)=O)C2)=O)c[nH]c2nc(F)ccc12 c1(C(C(=O)NC(C(=O)OC)C)N(C)Cc2cscc2Br)ncc(Cl)n1C Cc1csc(C(C(C)C)NC(C2(CSC3CC(C)(C)C3)CCCO2)=O)n1 CC1CCCN(C(C2(C(N)=O)CC2)=O)C1CNC(=O)CC=CC(C)(C)C c1(C(=O)NCCC2CCN(C(C3(COC)CC3)=O)C2)cc2sccc2n1C N=c1[nH]c(C(=O)NCc2cc(C(=O)NC3(CCF)CCC3)n[nH]2)cs1 C1(C(=O)NC(C2(C(=O)NC3CC4CCC3O4)CC2)C)CC2(C1)CC21CC1 N1(C(C(CC)SC)=O)CCC2CN(C(=O)Cn3cc(C#N)cn3)CC12 c1(C(=O)NC2(CC(N3CCC(O)CC3)=O)CCC2)c[nH]c2ccccc12 Cc1cc(CNC(=O)C(C)CC2CC2)oc1C(=O)N(C)Cc1csnc1C c1(CC)noc(C)c1C(=O)NCC1CCC(NC(CC2C(CC3CC3)C2)=O)CC1 c1(CC)c(N(CCNC(=O)Cc2ccc(C)cc2)CC)nc(C)nc1Cl c1(C(N2CC(NC(c3n(CC)nc(C)c3)=O)C(F)CC2)=O)[nH]nc2cnccc12 Cc1cc(C(N2CCOCC2CN(C)C(c2csc(C(N)=O)n2)=O)=O)cc(C)n1 c1(C(=O)OC)ccncc1S(=O)(=O)N1CC(C)N(Cc2cccs2)C(C)C1 C12(NC(C(c3ccc(Cl)s3)C)=O)CCC(CNC(=O)C(O)C3CC3)(CC1)OC2 C(=O)(C1=CCCCC1)N(C(C)C(=O)NCCOC(F)F)C1CC1 c1(C(C)C)cccc(CNC(=O)NCCSc2cnn(C)c2O)c1 CCCCC(CC(=O)NC1CN(C)CC1(C)C)NC(=O)C(CSC)OC N1(C(C2C(C(=O)OC)C2)=O)CCCC(C(N2CC(n3ccnn3)C2)=O)C1C C(=O)(CCCn1cccn1)N(C1CCC(NC(=O)Cc2csnn2)C1)C Cc1[nH]nc(C(=O)N(CCNC(C2(C#N)CC2(C)C)=O)CC2CC2)c1[N+](=O)[O-] C(C)(C(=O)N(CCNC(C1(C2CC2)CC1)=O)C(C)C)(C(C)C)NC(C)=O N1(C(c2c(C)onc2)=O)CCC2(CCOCC2)C(NC(=O)CC2CCC3CC23)C1 C1(CCO)CCCCC1N=c1[nH]c(=NCc2cccc3ccsc23)[nH]c2c1CSC2 c1(C(=O)NC2CCCC(N(C(C3CC(O)(CC#C)C3)=O)C)C2)cc(Cl)cnc1C Cc1nc(C(N2CCC(OCC(=O)NCc3cccs3)C2)=O)cs1 CN1CCC(C)(C(=O)NC2CC(CNC(c3ccc(CO)o3)=O)C2)C1=O c1(C(C(=O)N(C(Cc2nnc(C)o2)=O)C2CC2)O)cccc2c1OCC2 C1(C(=O)NCC(CC=C)NC(c2cccn2CC)=O)(CC2CCC2)CCCCC1 N1(c2n(C(C)C)nnn2)CCC2(CCN(C(=O)Cc3cn4c(n3)CCCC4)C2)C1 C1(C(=O)NCCCOCCCNC(C(=Cc2cccs2)C)=O)CCCCNC1=O C(C(C)(CC(C)C)NC(C1CC2CCC(C1)S2)=O)NC(C1(CC)COC1)=O c1(C(=O)NCC(c2nc(C(F)(F)F)cs2)C)nc(-c2ccccc2)ncc1F C1(C2CC2)(CNC(CCc2cn(C)nn2)=O)CCN(C(=O)C2=CCCSC2)C1 S(=O)(=O)(c1ccc(NCCOCCO)c(C#N)c1)NC1CCC(=C)CC1 c1(CC)cccc(F)c1C(N1CC2CC2(CNC(C2(O)CCC(C)(C)C2)=O)C1)=O C1(C)(CNC(C2(C(F)F)CC(=C)C2)=O)CCCN(C(c2cnc(N)cn2)=O)C1 N1(C(c2ccn(C)n2)=O)CCC(C)(CNC(c2cnn(Cc3nccs3)c2)=O)C1 N(C(=NCCN1CCOC(C)C1)NC(C)C)C(Cn1ncc(C)c1)C.N1CCOCC1 N1(C(CSC(C)=O)=O)CC2OCCN(C(=O)C=CCCC(C)=O)C2C1 CCCC(C#N)C(=O)N(C(C)CNC(=O)CSc1ccccc1OC)C C=CCC(CC=C)C(=O)NC1(C(=O)NCCNC(N)=O)CCOCC1 C(C(C)(C(=O)NCC1CCCC1(C)CO)NC(=O)CNc1cccnc1)SC C1(NC(C(C(C)C)=O)=O)CC(C)CN(C(c2cnn(CCF)c2)=O)C1 C1(C(N2CC(NC(=O)C(F)(F)F)C(NC(=O)C=CCOC)C2)=O)(CC)CCNC1=O c1(NC(C)=O)cnccc1C(=O)NCCCC(C)(C)NC(=O)CC1CN(C(C)C)C1 C1(NC(CC(CCC)(C)O)=O)CC1C1CCCN(C(c2nn(C)c(C)c2N)=O)C1 Nc1c(C(=O)NCC2CC(CNC(=O)Cc3cnc[nH]3)CO2)cc(Cl)[nH]1 N1(CC)CCCCC1C(N1CCN(CC2CN(C(=O)C3CC3)CCO2)CC1)=O N1(C(C(c2cncn2C)N(C)C)=O)CC(C2CN(C(c3cccnn3)=O)C2)C1 Cc1nc(C(C)C)oc1C(=O)NCC1C(C)CCN1C(C1CCC=CO1)=O C1(CCC)(COC)CCCN1C(C1CCN(C(c2c[nH]c(C)c2)=O)C1)=O N1(C(CCC=CC)=O)CCC2(CC1)CN(C(=O)C(c1ccncc1C)C)C2 c1(C(C(=O)NCC(CNC(c2nc(CCC)sc2)=O)(C)O)C)c(C)noc1C CCC(C)(F)C(=O)NC1CCC1CNC(c1cccc(CSC)c1)=O Cc1cc(Cl)cc(NC(C2CC3CC3N2Cc2ccn(CCF)n2)=O)c1I Cc1cc(F)cc(C(=O)NCC2CCN(C(c3ccncn3)=O)CC2)c1C C#CCC(C)(CC)C(=O)NCC12CC(CN1C(=O)Cn1cc(C(=O)OC)nn1)C2 C1(C(=O)NC(c2noc(C)n2)CC)(NC(=O)COCCCC(C)(C)C)CC(O)C1 Cn1c(C(=O)NC2C3CC2N(C(=O)CSc2ccccc2)C3)cc2sccc12 C(=O)(CC1=CCCCC1)NC1CC(C)N(C(=O)CCc2ccc(F)c(F)c2)C1 N1(C(c2c(NC(C)=O)cnc(Cl)c2)=O)CCC(NC(=O)CSCC(F)(F)F)C(O)C1 CC12CC(C(=O)NCC3(CNC(=O)CCCC#N)CC34CCC4)C(CO1)C2 N1(C(C(CC)=CCCC)=O)CCC=CC1C(=O)NCC1CCN(C2CC2)C1 N1(CC)CCCC1CC(=O)NC1COCC1NC(c1cc(Br)n[nH]1)=O c1(CNC(C(=O)N(c2cccnc2)CC)=O)cccc(N2CCCCC2)c1 C(=O)(CC(C)(C)NC(=O)CCc1ccn(C)c1)NC(C(C)C)CN(C)C Cn1cc([N+](=O)[O-])c(C(N2CC(NC(=O)CCc3nccs3)CC(O)C2)=O)n1 n1(CCOC)nc(C(=O)NCC2CCC(C)CN2C(=O)C2=C(C)OCC2)ccc1=O C1(CNC(=O)CCc2ccoc2)CCN(C(=O)Cc2cccc(F)c2O)CC1O c1(C(N(C(CCNC(CSCC(C)C)=O)C)C)=O)ccc(-c2cccs2)cc1F N(C(=NCC(=C)C1CCOCC1)N1CCC(S(C)(=O)=O)C1)C(C=C)C c1(C(=O)NC2(C)CCN(C(C3CC4CCC4C3)=O)C2)cc2c[nH]cnc-2n1 N1(C(c2ccon2)=O)CC2(CCN(C(c3cc4c[nH]cnc-4n3)=O)CC2)C1 C1(=O)CC(F)(F)CN1.N1(CCOCC)CCN(C(=O)OC(C)(C)C)CC1 C12CC(F)CN1C2C1CC(C)C1.C(C(=O)OC)NC(=O)NC CCCCC(CN=c1nc(C(=O)OC)[nH]s1)NC(c1cc(C)n(C(C)C2CC2)n1)=O Cc1ccc2c(c1)CCCC2N(C)Cc1cc(OC(C)(C)C)ns1 c1(CC)c(C(N2CC(C)(NC(c3ccnn3CC)=O)C2)=O)cnc2ncnn12 c1(-c2c(C)nn(C)c2C)ccc2nc(C(=O)N(c3cccnc3CO)CCO)[nH]c2c1 N1(C(C(C)(CO)OC)=O)CCC(NC(C23CCCC2CCC3)=O)CC(O)C1 C1(CNC(C(N2C(CC(=O)OC)CC2)C)=O)CC2C=CC1O2 C(=O)(C(CCCC)N(C)C)NCC(C(=O)NCC(=C)F)(C)C c1(C2(C)CC2Nc2cc(F)nc(F)c2)ccc(F)cc1Cl C(=O)(C1CCCc2c1[nH]c1ccc(Br)cc21)NC1(C(=O)OC)C2CC3CC(C2)CC1C3 C(=O)(C1SCCc2sccc21)NC1C(NC(c2cc(CCC)on2)=O)CC1 CC1(C)CC(C(=O)NC(c2nc[nH]n2)C2(CO)CCC2)=NO1 C1(CC(=O)NCC(CC)NC(C23CCCN2CCC3)=O)CC(C)(C)C(=O)N1 N1(C(C=CCN(C)CC)=O)CC2(C1)SCCC2NC(c1[nH]cnc1C)=O Cc1oc(S(C)(=O)=O)cc1C(N1CCC2CCN(C(c3cnc(S)[nH]3)=O)CC12)=O CCC(CC)(C(=O)N1CC2CC(NC(=O)CC3NC(=O)NC3=O)CC2C1)C(C)C C=CCN=C(NCc1ccc(C#N)cc1)NCc1cn(C(C)C)c(=O)nc1O c1(C(=O)NC(C(C)NC(c2ccc(C)cc2O)=O)CO)ccn2c(C)cnc2c1 CN1C(=O)CCCC1C(N1CC(CC(=O)NCC(CO)C2CC2)C2(CC2)C1)=O O=C(CCCCC1CC1)NCCC1CCN(Cc2cnco2)CC1 N1(C(C2(NC(C)=O)CCCC2)=O)CCC(COC)(NC(=O)CCC(C)(C)F)CC1 N1(C(C(CCC)NC(c2ccc(C)c(C)n2)=O)=O)CCOC2C(O)CC12 N1(C(Cn2ncc(C#C)c2)=O)CC(NC(=O)C(C)(C)OCC)CC(O)C1 Cc1cc(C(N2CCC(C(C)NC(=O)CCCc3cncs3)C2)=O)nc(O)c1 Cn1nc([N+](=O)[O-])cc1C(N1CCCC1C(C)(C)NC(C1CC2C=CC1O2)=O)=O C1(CNC(C=COCC)=O)CN(C(c2ccc(NC(C)=O)s2)=O)C2CC12 c1(C(=O)NCC2N(C(CC3ON=C(C)C3)=O)CC(F)C2)ccccc1S(C)(=O)=O N1(C(c2n[nH]c(C3CC3)n2)=O)CCN(C(C2CN3CCN2CC3)=O)C2(CCC2)C1 C1(NCC(C2CCCC2)N)CC2(C1)CC(N)C2 C(O)CC(C(=O)N1CCC(O)(C(N)=O)C1)NC(=O)CC1C(C)(C)C1(C)C c1(C(N2C(CNC(C(c3ccc(Cl)cc3)C)=O)CC2)=O)cnc(=NCCF)[nH]c1 c1(C(C(=O)NCC(CNC(C(=O)NCC)=O)(C)O)O)ccc(F)cc1C c1(Cc2nc(C(=O)NC3CC(NC(C)=O)C3(C)C)sc2)n[nH]c2c1CCC2 N1(C(C(=O)N(C(C)(C)C)C)=O)CCCC2C(NC(=O)C=C3CCCC3)C(C)(C)C12 c1(C(=O)NCC2CCCN2Cc2nc[nH]n2)ccnc(-c2ccccc2)n1 c1(C(N(C(CNC(C2N(CC#C)CCC2)=O)C)C)=O)ncnc2sccc12 N1(C(C2(C)CN(C(C(n3c(C)ncc3)C)=O)C2)=O)CCC2(C=CCO2)CC1 c1(OCC(=O)N(CCO)Cc2cccc(O)c2)ccc(Br)cc1Cl c1(C(N2CC(CC)C(c3cn(CCOC(C)=O)nn3)C2)=O)cc(C#N)ccc1F CS(=O)(=O)CCCSC.C(CF)(CF)S CC#CCC(C(=O)NCC1NC(=O)NC1=O)NC(=O)Cc1ccc(C#N)cc1 C1(C(=O)OC)CCCC(C(=O)NC2(C)CCN(C(=O)CSC(F)(F)F)C2)C1 c1(C(=O)NC(C2CCCCN2C(=O)CCOCC2CC2)C)cncc2sccc12 N1(C(CN(C)C2CC2)=O)CCC2CCCN(C(=O)CC3CCOCC3)C2C1 C#CCC(C)(C(=O)N1CCOC(CC(C)C)C1)NC(c1cnn(C)c1)=O Cc1nn(C)c(C)c1CC(N1CC(CC(C)NC(=O)C(=Cc2cnc[nH]2)F)C1)=O c1(C(=O)NCC2(O)CN(C(C3CCCC3C(F)F)=O)C2)c(F)ccc2[nH]ccc12 CN1CCN(C(=O)CC2CC2)C(CNC(C2CC(=O)NC(c3ccccc3)C2)=O)C1 N12CC3(CC(C3)CNC(=O)CC(C3CC3)C1=O)C2.c1(OOC)ccc(F)cc1Cl.O C1(C(=O)NC2(CNC(Cc3cn(C)nc3)=O)CCOC2)CN2CCC1CC2 c1(OC(CC(=O)OC(c2ccc(OC)cc2)C)C2=CCCC2)nc(Cl)cn2ccnc12 Cc1csc(Cl)c1C(N1CC(NC(=O)C(C(C)C)c2ccn(C)n2)C(O)C1)=O C(=O)(C(C)(O)C(F)(F)F)N(CCCNC(C1CCN(C2CC2)C1=O)=O)CC N1(C(C(C(C)O)C)=O)C2CCC1CC(NC(C1CC3C(C1)C3(F)F)=O)C2 N1(CC)CC=CCC12CC(C(=O)NCCNc1ccc(F)c3c1CCC3)CCC2 c1(C(N2CCOC(C3CC3)C2)C(=O)NCCCOC)ccc(C#N)s1 C(=O)(CCCCC(=O)N1CCC(C(C)CNC(=O)Cc2cc(C)[nH]n2)CC1)OC c1(C(=O)NCC2C(NC(c3occ(C)c3)=O)CCC2)sc(F)cc1Br C1(CNC(C(C2CCOCC2)C)=O)CC2CCC1N2C(=O)C=Cc1ccoc1 c1(NC(C2N(C(CCOCC=C)=O)C(C)CC2)=O)ccc(F)c(C(F)(F)F)c1F C=CCCCC(C)(C)CNC(=O)CCCCNC(=O)CN1CCOCC1 C(CN=c1[nH]c2c(c(=NC3CCOC(C(C)C)C3)[nH]1)COC2)SC(C)C C1(C(N(CC2=CCCOC2)C)=O)CN(C(C2(C)SCCCS2)=O)CC1C c1(NC(N2CCCC2)=O)ccc(Nc2ccccc2CC(F)(F)F)cc1 N1(C(C(CC#C)CC#C)=O)CC2CCCCC2(CNC(c2ncoc2CC)=O)C1 CC1CN(C(c2cc[nH]c2C2CCCC2)=O)CC1CNC(=O)COC1CC1 c1(C(=O)NC(C)(C)CCC2CC2)oc2ccccc2c1CO C1(CNC(C(C(CC)O)C)=O)CN(C(c2[nH]nnc2C)=O)CCC12CCOCC2 Cc1cc(C#N)cnc1C(N1CC(NC(C2CCCC(=O)N2)=O)CC1C)=O C1(COC)CCN(N2CCC(c3cccc(F)c3C)C2)C1 C(=O)(C1=COCCO1)N1CCN(c2c(C(C)NC(C(C=C)O)=O)cccn2)CC1 C1(n2cc(-c3cn(CCOC)nc3)nn2)Cc2ccccc2C1O.C1C(=O)O1 S(=O)(=O)(c1ccc(Cl)cc1)N1C(C(=O)Nc2c(C(C)C)ccc(F)c2)CC(O)C1 Cc1ccc(C(=O)NC2CC(C(=O)Nc3cccnc3C(F)(F)F)C2)c(O)c1 N1(C(C(C)N(C(C(C)OCCOC)=O)C)=O)CCCC(C)(C)C1C Cc1cc(F)c(NC(=O)C(=O)NC(C)CCNC(=O)NC(C)C)c(F)c1 C12(CNC(CC(=O)NCC)=O)CCCCC1N(C(c1ncccc1Cl)=O)CCC2 N1(C(=O)Nc2ccc(C(C)(C)C)cn2)CC2(CC2C#N)C1 c1(C(=O)NC2C(NC(C3(C#C)CCC3)=O)CC2)ccc(F)c(OC(F)(F)F)c1 CC1CCC(C)(C=CC(=O)NCC2(O)CN(C(=O)Cc3cccnc3N)C2)C1(C)C C(C(C)(C)CC(=O)NC1C2CC1N(C(c1cnn(CCO)c1C)=O)C2C)OC C(=O)(C(C(C)(C)C)OC)NCCC1(O)CCN(C(c2c(OCC)nccc2)=O)C1 N12CCN(C)CC1NC(=O)c1c(cncc1)C2=O.c1(CNC(C)C)c[nH]nc1Cl c1(C(=O)NCCC2CCN(C(C3COCC(C)O3)=O)CC2)ccc(Cl)c(F)c1F c1(NC(C(CC)(C)CNC(=O)CC2CNC(=O)O2)=O)ccc2nc[nH]c2c1 C12(CC(N3C(C)CC(CNC(=O)Cn4cccn4)C3)=O)CCC(CN(C)C)(CC1)C2 c1(C(=O)NCC(C(C)(C)C)NC(c2cn(C3COC3)nn2)=O)ccc(Cl)nc1N c1(C(N(C2CCN(C(=O)Cc3nccs3)C2)C)=O)cccnc1OCCO c1(CC)nc(C)[nH]c1C(=O)NCCC1CCN(C(c2cc(C3CC3)on2)=O)C1 C(C)(N=c1[nH]c(=N)c2occc2[nH]1)c1cnc(C)s1 CN1CCN(C(=O)CCc2nc(=N)[nH][nH]2)CC1.C(=O)(C=CC(=O)N(C)C)NCCOC c1(CC)ccc(C(=O)N(C)CC2(C(=O)NC3(c4ccn(C)n4)CC3)CC2)cc1F C(=O)(C(C(C)(C)O)NC(c1n[nH]cc1C)=O)NC1(CCCC)CC1 C(=O)(CCC(C)(C)OC)NCC(CC=C)NC(c1cnc(CC(C)C)[nH]1)=O N1(C(C(CC)F)=O)CCC(CNC(=O)C=Cc2ccncn2)C(F)(F)CC1 N1(C(c2onc(CC)n2)=O)CCC2(C1)CN(C(C1(CC)CCCC1)=O)C2 CCCS(=O)(=O)C(C)C(=O)NCC(C)NC(c1cccnc1F)=O Cn1ncc(C(=O)NCCCOCCCNC(=O)CCC2CCCOC2)n1 C(c1cccc(Br)c1)=CCN(C1CCCCO1)C(C1COCCN(C(=O)CO)C1)=O CC1CCCCC1NC(=O)C(N1CCOC(CCN)C1)=O C12(O)CCN(C1)C(=O)C(C)c1ccsc1C(=O)NC2.c1(OC)ccccc1OC.CO C1(C(=O)NCC=CCNC(C23CC(O)C2C3)=O)C2CCC1(c1cscn1)C2 c1(C(N(CCCNC(c2cc(=O)cc(Cl)[nH]2)=O)C)=O)ccc2c(=O)ccoc2c1 CC1CCN(C(c2cn(C(C)(C)C)nn2)=O)CCN1C(C1CCCCC(=O)C1)=O c1(NC2CCN(C(C(C)C(F)F)=O)C2)ncnc2cccnc12 N1(C(c2nc(C)oc2)=O)CC(C(=O)NCC2CCCS2)C(F)C1 CC1(CNC(C2(C(F)(F)F)CC2)=O)CN(C(C2CC(O)C2)=O)CCO1 c1(CC)c[nH]c(=NCC2(C)CCN(C(=O)C(Cc3cccs3)NC(C)=O)C2)cn1 N1(C(C(CC(=O)OC)C)=O)CCC2CN(C(c3cn(CCO)nn3)=O)C2C1 CC(=O)CCCCC(=O)N1CCC2(CC(C(=O)NCC=CC(C)(C)C)C2)C1 c1(C(=O)NC2CCC(NC(c3c(C)nc(F)cc3)=O)C2)ccc2ccccc2c1 C1(C(=O)NCC#CCNC(C2CC3(CCCC3)CO2)=O)Cc2ccc(F)cc2O1 c1(C(N(C)CC2COCCN2C(C2C(C)C2C)=O)=O)ccc(F)c(C(F)(F)F)c1 C1(NC(CC(C)OCC)=O)C=CCN(C(=O)C(c2ccc(Cl)cc2)CO)C1 C1(N=[N+]=[N-])(NC(CC(C)CN(C)C)=O)CCN(C(C2CN3CCN2CC3)=O)C1 c1(C(=O)NC2C(CNC(CCc3nnc(C)o3)=O)C2)ccc2occc2c1 N1(C(C(CC)n2ccnc2)=O)CCC(C(C)CNC(=O)Cc2ccoc2)CC1 N1(CC(N2C(CCNC(=O)C=CC3CCCC3)CCCC2)=O)CCS(=O)(=O)CC1 C1(C(N2CCC(C(=O)Nc3ccc(Cl)cc3)(CF)C2)=O)COc2ccccc2O1 N1(C(CC(=O)NCC(F)(F)F)=O)CCC2CN(C(=O)C(F)(F)CO)CC2C1 N1(C)CC2CC(F)(F)CCC2(C(=O)OC)C1.C1(C(OCC)OC)CCOC1 Brc1ccc2oc(-c3nc(Cn4cncn4)nn3CCc3cccnc3)cc2c1 N1(C(=O)CC2CCC=CCC2)CCN(C(=O)CCCC(F)(F)F)C2CCCCC12 C1(CNC(C23CCCCC2C3)=O)(CO)CCCN(C(=O)C=C2CCC2)C1 N1(C(C2(CC#C)CCCO2)=O)CCC2(CC1)CC(NC(c1cccnc1O)=O)C2 n1(CC(=O)NC(CNC(C=CCC)=O)C(C)C(C)C)cc(C#N)c(O)nc1=O c1(OC)ccc(S(=O)(=O)N2CCC(NCC3CCC4(CC3)OCCO4)C2)cc1 C1(NC(C2C(C(N)=O)C2)=O)COC2(C1)CN(C(c1c[nH]c(=S)cn1)=O)C2 N1(C(c2cc(C)sn2)CC)CCN(c2nccc(N3CCCC3)n2)CC1C NS(=O)(=O)c1ccc(C(N2CC3(CCCN3C(C3(O)CC3)=O)C2)=O)s1 Cn1ccn2ncc(CNC(C3CC4(CC4)CN3C(=O)OC(C)(C)C)=O)c12 C12(NC(CC=C)=O)CCCC1N(C(=O)CCCOc1ccc(C(N)=O)cc1)CC2 c1(C(=O)NCC2N(C(C=C3CCC(C)C3)=O)CC2)cnn2c1CCCC2 C1(C(=O)NCC(CNC(c2ccnnc2C)=O)OC)CCC=CCCC1 c1(C(N2C(CCOC)CN(C(=O)CC3CC3(C)C)CC2)=O)cc(S(C)(=O)=O)co1 c1(C(=O)NCC(C)(C2CC2)NC(c2c(OC)nn(C)c2)=O)c(Cl)ccc(C)c1N N1(C(C2CC(=C)C2)=O)CCCC2(NC(=O)CC3CCC34CCC4)CCCC12 Cc1cc([N+](=O)[O-])cnc1NC(C1CC(F)CN(C(=O)CSC(F)F)C1)=O C(=O)(C#CC1CCCC1)NCC(C(N1CCCC(C)(C)C1)=O)C1(O)CCC1 C(=O)(C(CCCNC(c1ccccc1)=O)N1C(CO)CCC1C)NCCOC N1(C(C(C(=O)OC)C)=O)C(C(=O)Nc2cnn(C(C)C)c2)C2CC(F)C1C2 c1(NC(C2CCCN2C(=O)Cn2cncn2)=O)ccc(O)c(CO)c1 N12CCC(C(C)C1)C2.Cc1cnccc1OCC(=O)OCC(=O)Oc1cnccn1 c1(CN(C2CCCN(CCO)CC2)c2ncc(F)cn2)ccc2nc[nH]c2c1 C1(OC)CN(C(c2cc(Cl)cc3c2OCC3)=O)CC2(CCC2)C1 c1(C(=O)NC(CC(C)C)(C)C)cc(S(=O)(=O)Nc2ccc(Cl)cc2)ccc1O C1(NC(C(C)NC=O)=O)CC2CN(C(=O)Cc3cc(Cl)cc(Br)c3)CC2C1 c1(-c2nccc(CC)c2)cc([N+](=O)[O-])ccc1C(=O)NCc1cccs1 c1(C(N2CC(NC(C(C)NS(C)(=O)=O)=O)C(F)CC2)=O)ccc2ccn(C)c2c1 c1(OC)ccc(-c2nc(C(=O)NC(c3ccc(Cl)cc3)C(C)(C)C)cs2)cc1 N1(C(c2cnc(OC)s2)=O)CC(C2(NC(=O)Cc3ccncc3Cl)CC2)C1 C1(NC(c2n(CCC)nnn2)(C2CCCCC2)C)CCc2cnc(C)n2C1 Nc1ccc(C(=O)NCC2CN(C(C3CCC(N=[N+]=[N-])C3)=O)CCCO2)nc1N N1(C(C23CC(C(F)F)(CO2)C3)=O)CCOc2c(Br)cc(F)cc2C1 C1(C(=O)NCC(CC(C)C)NC(c2cc(Cl)c(Cl)s2)=O)CCc2nc(O)[nH]c2C1 CC1(C)COCCN1CC(N1CCOCC1c1noc(C(F)(F)F)n1)=O C1(C(N2CC(NC(C(C)=C3CCC3)=O)C2)=O)CC(c2cccnc2)=NO1 C1(C)(COC)CCCN(C(C2CC(F)CN2C(C2C3CCC(F)C23)=O)=O)C1 Cc1nc(CC(=O)NC2(c3csc(C4COCC4c4nn[nH]n4)n3)CCC2)co1 C(=O)(C1=CCCCCC1)NC1CN(C(c2cc(CCC)oc2C)=O)C(CO)C1 C1(C(=O)NCCCCN(C(CCC(=O)NCC)=O)C)CNC(=O)CC12CCOC2 Cc1ccc(F)c(C(=O)NC2CCCCC2NC(=O)CC(C)(C)C2CC2)c1F C1(C)(C)C(=O)N1.C1(CC(=O)NC2CC2C)CCCN1C(=O)C=C(C)C.C(C)(=O)NCC C(=O)(C(CC(C)C)N(C)C(c1ncncc1OC)=O)NC(COC)CCO c1(C(=O)NC2C(C)N(c3nnc(C(N)=O)s3)CCC2C)cnc2c(c1)ncn2C C1(C2N(C(C3(F)CC3)=O)CCC2)CCN(C(C2(c3ccncc3)CC2)=O)CC1 C1(C(N2CC(C(C)NC(=O)COCCC(C)C)C2)=O)C2CCC3(COC(=O)C13)O2 C(=O)(C(C)(C#N)CC)N(CCN(CCN)CC)CCOC.C1(=O)CN1 C(C)(CC1CCC1)(CN=c1cc(NCc2sc(C)cc2Br)nc(C)[nH]1)OC C(=O)(C(C(C1CCC1)OC)N(CCC(N)=O)C)NCCNCC Cc1ccc(NC(=O)C(C)N(C(=O)C(=O)N(C)C)C(C)C)c(F)c1F N1(C(CCSC)=O)CCN(C(c2ccc(C(F)(F)F)nc2)=O)CC1C#N N1(C(c2c(CC)nccc2)=O)CC(C(=O)NCc2ccc(O)nn2)CC(C)(C)C1 c1(OC(c2cc(C)ncc2C)=O)cc(C)n(C)c(=O)c1 C1(Cn2cc(CCNC=O)nn2)CN2CCCC2CO1 c1(CC(=O)NCC2CC(NC(C(CC)N(C)C)=O)C2)cc2ccccc2nc1O c1(C(=O)NC2C(CNC(c3cnoc3-c3ccco3)=O)C2)nccn2nccc12 C1(C(=O)NCCNC(N2CC(OC)C2)=O)Cc2ccccc2C1(C)C C(CCCCO)N(C(c1ccn(CCNC(C2C=CCC2)=O)c1)=O)CCO C1(O)(C(C)NC(=O)CC2CCCC2)CN(C(=O)Cn2cccn2)C1 C1(C(=O)NCC(C)CNC(=O)C(c2cccc(F)c2)O)CCC12CCC2 C1(NC(C=CC)=O)C2CCC1N(C(C1(NS(CC)(=O)=O)CCCCCC1)=O)C2 n1(CC)c(C(=O)NC2(C(=O)NC3CCOC3(C)C)CCN(C)C2)cnc1O N1(C(c2c(OC)noc2C)=O)CCC2(C1)CN(C(C1CCC3(CC3)C1)=O)CCO2 c1(NC(c2cc(CCCC)oc2C)c2nnnn2C(C)C)ccc(C(N)=O)c(C)c1 c1(C(c2nnnn2CCOCC)NCC(=C)CC)cccc(F)n1 c1(C(=O)NC2CN(C(c3c(COC)cc[nH]3)=O)C(C)CC2)c(C)cc(C)nc1O CON1CCC(C(=O)NCCCCCNC(C2(S(C)(=O)=O)CC2)=O)CC1 C1(NC(CN(C(=O)C(CC2CCCC2)NC(N)=O)CC(C)C)=O)CCCCO1 C12(C(N3C(COC)CCC3)=O)CC(C)(CN1C(=O)C(C1CCCCC1)C)C2 C1(NC(C2(COC)CC2)=O)(CO)CCN(C(=O)C)CC1.c1(N(C)C)ccccc1 C#CCC(C)(C)C(=O)N1CCN(C(=O)CCC2(CC(C)(C)C)CC2)CC1 N1(C(C(CC)C#N)=O)CCC(O)(C(C)NC(=O)C(=O)NC(C)C)CC1 C1(NC(C2C(C)=C2)=O)CN(C(c2cnn(C(C)(C)C)c2C)=O)CC2(CCC2)C1 C12(CCC1)C(=O)NCC(OCC(C)C)CNC2=O.C(CSC)=CC c1(CC)[nH]nc(Cl)c1C(=O)NCCC1(NC(=O)C(CO)c2ccccc2)CC1 N1(C(c2cc(C)sc2)=O)CCC(C(C)(O)CNC(=O)CCc2nccn2C)CC1 c1(C(=O)NCCN(CC(C)O)C(=O)CC2CCCOCC2)nnc(O)cc1O C(=O)(C1=CSCCO1)NC(C)CCNC(C12COC(CCO1)C2)=O C(CCC1CCC1)(C(=O)N1CC2(CCC2)C1)NC(CCc1ccc(C)o1)=O N1(C(c2cn(CC)nc2)=O)CCC(NC(N2CCCC(C)C2)=O)C(C)C1 C1(C(=O)NC2CC(CNC(C(C)P(C)(C)=O)=O)C2)CCN(S(N)(=O)=O)CC1 c1(C(=O)NC2(C)CC(NC(C3C(C=C)C3)=O)C2)cccc([N+](=O)[O-])c1C CN1CCOC(C(N2CCCC(O)(CNC(c3nn[nH]c3Cl)=O)C2)=O)C1=O C(=O)(C1=CCCC1C)N(CCNC(c1ccc(CN(C)C)o1)=O)CC CC#CCCCC(C)(c1nnnn1CCCOC)NCC12CCC(CC1)C2 C1(C(=O)NCC(N(C)C(C2(n3cccn3)CC2)=O)C2CC2)CC2CCC2C1 C1(C(=O)NC(c2ncc(C)s2)C)(NC(c2c(C)noc2C)=O)CCN(C)C1 CCC(C(=O)OC)C(=O)N1CCC(C(N2CCC(OC)CC2)=O)(CC2CC2)C1 c1(CN(C(c2nc(CC)sc2)C(=O)NCC(F)F)C(C)C)cnc(OC)c(C)c1 C(=O)(CC(F)(F)F)N1CC(C(=O)NCc2nccn2C2CC2)(CC)C1 c1(SCCC)cccc(C(=O)NCC(CC)NC(c2cc(CC)on2)=O)c1 c1(C(=O)NCCC(C)NC(c2cccc(NCC#C)c2)=O)ccc(C)cc1F c1(CNC2C(C(=O)Nc3c(C)cncc3)CCC2)ccc(Br)nc1Br C12(NC(c3cc(Cl)cs3)=O)COCCC1CN(C(c1cc3n(c1)CCC3)=O)C2 N1(C(C(C=CCCC)O)=O)CC(NC(c2cc(C(N)=O)no2)=O)Cc2ccccc21 Cc1cc(Cl)c(C(=O)N(CC(O)CNC(=O)C=CC2CCOC2)C)cc1N Cc1cc(=O)n(C)nc1C(N1CCC(C2(NC(c3cccc[n+]3[O-])=O)CC2)C1)=O CC(=O)CCCC(=O)NCC1(F)CN(C(c2cccc(SCCC#N)c2)=O)C1 C#Cc1ccc(CNC(C2CCCCCN2C(c2nnc(CC)o2)=O)=O)cc1 C12(CNC(C(COC)C)=O)COCCN1C(=O)CN(C(=O)C=CC1CCC1)C2 c1(C(=O)NC2C(NC(COCC(=O)NC)=O)CC2)csc(=NC2CC2)[nH]1 c1(C(C)NC(c2cnc[nH]2)=O)ccc2c(c1)CN(C(C1C(C)(C)C1(C)C)=O)C2 c1(-n2c(-c3cc(C)n(C4CCOCC4)n3)nc(C(C)O)n2)ccc(Cl)c(I)c1 N1(C(C(C=C)c2ccccc2)=O)CCCC(C2CN(C(=O)C(C#N)CC)C2)C1 C1(CCC)(C(=O)N(CCCNC(=O)Cc2cncc(C)c2)C)CCNC1=O C=C(C)CC(C(=O)N1CC(O)(C(F)(F)F)C1)NC(=O)C(C)c1cccs1 N1(C(C(C(C)O)C)=O)CCCC(C2CN(C(c3ccc(C4CC4)nn3)=O)C2)C1 C1(C)(NC(CCCc2nc(C)sc2)=O)CCN(C(C2CC2c2cccnc2)=O)C1 C1(C(=O)NCC2(O)CC2CO)CCCN(C(C2COCOC2)=O)CC1 CC(C(CO)NC(c1cnc(-c2cnccn2)s1)=O)NC(C1CC(C)(C)O1)=O c1(C(CC)OC)cn(C(C)C)nn1.c1(CCC2CC2)ccc(C(=O)NCCC2CC2(F)F)o1 N1(C(CCCC=C)=O)CCN(C(c2cc(CCC)n(C)n2)=O)C2CCCC12 C(C(C(C)C)NC(=O)CNCCCC(C)C)(c1ccccc1)NC(CC=CC)=O C1(NC(C(C)C2CC2)=O)CCOC12CCN(C(c1ccc(C(F)F)cn1)=O)CC2 c1(C(N(C(c2ccccc2)(C)C)C)=O)ccc(CNC(c2ccco2)=O)cc1 C1(C(=O)NC2CC(C)N(C(=O)CC3(C)CCCCC3)CC2)CCc2nnnn2C1 C1(NC(CC(=O)NC(C)O)=O)C2CC3C(C2)C13C(N1CCNC(=O)C1)=O c1(OC)ccc(CC(N2CC(CCO)OC(C)C2)=O)c(OC)c1 Cc1cc(C(=O)CN2CCOC(CCS)CC2)cc(C)c1.C(=O)(C(C)C(C)C)N CC1CN(C(=O)CCC2CC(F)(F)C2)CC(CCNC(=O)C2=COCC2)O1 C(=O)(C(C)(C)C(C)(F)F)N1CC(C)C(NC(=O)C(C#N)C(C)(C)C)C1 N1(C(C(c2ccccc2F)OC)=O)CCC(CO)(NC(c2cnoc2C)=O)CC1 C1(COC)(NC(=O)CC=C(Cl)Cl)CCCN(C(=O)C(C)(C)Nc2ccccn2)C1 N1(C(CCc2cccc(C)c2)=O)CC(NC(C2CCC3(CC3)C2)=O)C2CC2C1 c1(C(=O)NC2CCN(C(CSCC#C)=O)C2C)ccc(-n2nc(C)cc2C)nc1 c1(C(=O)NC2CC(C)C2)cc(C2CC2)ncn1.c1(C(C)C)cc(NC=O)on1 C(CC1CCC1)(C(=O)NCC1=CCCC1)NC(=O)Cn1cnnn1 C(=O)(C(C)(C)CCCF)N1CCCC(CC=C)(NC(=O)C(C)OC)C1 c1(C(N(C)CC2CCN(C(=O)CC(O)CN(C)C)C2)=O)cc2c(ccn2C)[nH]1 c1(OCC(=O)NC(Cc2onc(C(C)C)n2)C)ccc(Cl)cc1Cl C1(NC(Cc2c(C)ocn2)=O)CCC(F)(CNC(=O)C(C)(O)C2CCOCC2)C1 C1(NC(CC(C)Oc2ccc(F)cc2)=O)CC2CN(C(c3cn[nH]c3)=O)CC2C1 C1(O)(CC#N)CCCN(CCC2CCCC(=O)C2)C1 c1(C(=O)NC(C(C)NC(=O)CC2CCC(=O)NC2)CO)ccc(Cl)c(C(F)F)c1 N1(C(CN(C(C)=O)C)=O)CCOCC1CCNC(c1cc(O)n(C)n1)=O C#CCS(=O)(=O)CCNC(=O)Nc1cccc(C(=O)OC)c1 N1(C(CC=CCC)=O)CCN(C(C2(F)CCOC2)=O)CC1c1ccc(F)c(F)c1 N1(C(CC2(CNC(C3(O)CCSCC3)=O)CC2)=O)CC(O)C(O)C1 CC(C)(C)C(=O)NCC(=O)NCCC(=O)NCC1CCN1C(=O)C(F)=CCCF C(N=c1[nH]ccc(C#N)c1[N+](=O)[O-])C1(C)CCCN(C(=O)CC2CC(F)(F)C2)C1 Cc1ncc(C=CC(=O)N(CCCNC(C23CC(C)C2C3)=O)C(C)C)s1 CC(C)C(C(=O)N1CC2CC1(CNC(C1CCC1)=O)C2)NC(N)=O Cc1ncc(Cl)c(C(N2CCC(C)(CCNC(=O)Cc3cc(C)ns3)C2)=O)n1 CCCC(CO)NC(c1coc(CNC(C2(CCC)CCC2)=O)n1)=O c1(NCC2(CC)CCOCC2)ccncc1S(=O)(=O)NCCC(C)(C)OC c1(C(N2CCC(NC(CC=C=C)=O)(CO)C2)=O)cc(S(C)(=O)=O)oc1C Cc1cn(-c2ccccc2Br)nc1C(=O)NOCC(N1CCCC1)=O.OC(F)(F)F N1(C(C(C=C)O)=O)CC2(COC(CNC(c3cnc(C)nc3C)=O)C2)C1 Cc1cccc(CC(=O)N(C(C)CNC(C23CCC(CO2)C3)=O)C)c1F c1(OC)cc(C(=O)NCC2CC2NC(=O)Cn2nnnc2C)ccc1OC(F)F C1(NC(CN(C(Cc2nc(C)sc2)=O)CCCO)=O)CC1C1CCC1 c1(CC)cc(C(=O)NC2CCCC2CNC(=O)COC(F)(F)F)ccc1F N1(C(CCN(C(=O)C2=C(Cl)CCC2)CC=C)=O)CCN2C(=O)CCC2C1 c1(C(=O)NCC23C(CN(C(c4cccc(OC)n4)=O)C2)C3)cnc2[nH]nnc2c1 C(=O)(CC(C)(C)C)N(CC(C)(C)CNC(c1cc(C)co1)=O)CC c1(C(=O)NC(CN(C(c2ccc(CO)cn2)=O)CC)C)c(SCC)cccc1F CC(F)(CNC(c1cc(Cl)n[nH]1)=O)CNC(C1CC1C(N)=O)=O CC(CO)C(=O)NC1(C2CCCN2C(=O)Cc2ccn(-c3ccncc3)n2)CC1 c1(C(N(CC(C)NC(c2cccc(C#N)c2)=O)C)=O)cc(O)nc2c1CCCC2 N1(C(CSCC=C)=O)CC2CC(C(N3CC4CCC3C(O)C4)=O)C(C2)C1 c1(C(=O)NCC(C(C)C)NC(C2CCCC2CF)=O)ccncc1Cl c1(COC)ccc(C(=O)NC2CCC(N(C)C(c3coc(C(C)=O)c3)=O)C2)o1 CC1(C)CN(C(c2cc(C(C)(C)C)on2)=O)C(CNC(=O)CC2CC=CC2)CO1 c1(C(=O)NC(COCC)CO)coc(CNC(=O)C(C)OC2CC2)n1 C12(NC(=O)Cc3ccnc(F)c3)CCCC1N(C(c1ns[nH]c1=O)=O)CCC2 c1(C(N2CCC(NC(C=C(C)C)=O)CC2C2CC2)=O)[nH]c2ccccc2c1Br c1(OC)ccc(C(=O)CN2CCCC2C(N2CCCC(O)C2)=O)cc1 C(=O)(C(CCC1CC1)NC(=O)Cn1cnc(=N)[nH]1)NC1(CO)CC(C)C1 N1(C(c2c(CCC)n[nH]c2)=O)C(C(=O)NCC2CCN(CC)C2)C2CC(O)C1C2 C(=O)(CC1=CCCCC1)NCC1CC(OC)CN1C(C1CCC(=O)C1)=O CC1CN(C(=O)CCSc2ccc(Cl)cc2)CCCN1C(=O)CCCN(C)C CCC(CO)CCNC(=O)CN1CCC(NC(=O)OC)C1.C12(CC1(F)F)CN2 C1(C)(C(C)NC(=O)CCn2cc(CO)nn2)COc2ccccc2O1 C1(NC(C(CNC(CCNC(=O)NC)=O)CC2CC2)=O)CC12CCCCC2.C(C)(=O)O Cc1ccc(O)c(CC(=O)NCC2CCN(C(=O)CCF)CC2)c1 C1(C(=O)NCC(C)CN(C)C(c2ncncc2C#N)=O)CC2(CCC2)CO1 N1(C(C2(OC)CCCCC2)=O)CC2CCC(C1)N2C(=O)CCc1cnc[nH]1 C1(C(=O)NC(C)CCCNC(c2nnc(S)n2C)=O)(CC)CCC(O)CC1 Cc1cc(NC(=O)NCC2CCN(CCO)CC2)ccn1.C(C(C)(C)C=O)N C1(C(=O)NC(CC(C)C)CN(C)C)CCCCN(C(c2cc(C#N)cn2C)=O)C1 C1(C(c2nnnn2C2CCOC2)NCCCSCC=C)C2(CCC2)C12CCC2 C1(C(=O)OC)CCN(C(c2ccc(CNC(c3ccc(Cl)o3)=O)nc2)=O)C1C c1(CC(=O)NCC(CNC(c2cc(C)sn2)=O)O)ccccc1CC#N N1(C(CC(C(=O)OC)(C)C)=O)CC2CCCC1CN(C(c1csc(CO)n1)=O)C2 C(=O)(CCCCC(C)=O)N1CCC(CC=C)(NC(C2CCCC2(C)C)=O)C1 N1(C(c2sc(C)c(C)c2C)=O)CC2(C1)CN(C(=O)C1=COCCC1)CCO2 C1(C(=O)NCCC(C)NC(c2cc(C)nnc2)=O)CCC2(CC1)NC(=O)NC2=O C1(CC=C)(C(N2CC(O)(C(C)(C)CNC(=O)Cn3nnc(=N)[nH]3)C2)=O)CC=CC1 c1(OCC(N2CCCC(c3nc4ccccc4o3)C2)=O)csc2cc(Cl)cnc12 C1(C(N(CC=C)CCO)=O)CN(C(=O)C(C)(C)CCC)CCN1C C12(C(=O)NC(C(C(=O)OC)C)C)CCC(CNC(=O)CC3COCCO3)(CC1)CC2 c1(-c2c(OC)ccnc2)cccc2c1CN(Cc1c[nH]c3ncccc13)CC2 c1(OCC(=O)NC2CCC(C(=O)NCC3CC(O)C3)CC2)cccc(F)n1 N1(C(CC(C)CF)=O)CC2CCCC2(CNC(c2ncn(C)n2)=O)C1 c1(COC)n[nH]c2c1CN(C(=O)Nc1ccc(C)c(F)c1)CC2 C1(C(=O)NC2CCNC2=O)(NC(c2coc(CO)c2)=O)CCCCC1 CC(C)CC(CNC(C1(CNC(c2nccn2C)=O)CC12CCC2)=O)CO C12CCCC1NC(=O)C2.C1(NC(C2CC2Cl)=O)COCC1N.C(C)OC c1(C(=O)NC(C2CCN(C(=O)CC(O)C3CC3)CC2)C)cc2ccccc2n1C N1(C(CCN(CCCCC)C)=O)CCCC(CCNC(c2cnccn2)=O)CC1 C1(C(C)NC(Cc2nc(C)[nH]n2)=O)CCN(C(=O)CC2CC2(Cl)Cl)CC1 N1(C(C(C)=CC2CC2)=O)C2CCC1CN(C(=O)CC(C)(C)C(=O)OC)C2 C1(C(C)(C)C)(CNC(C(CC)F)=O)CCN(C(C2(CSC)CCC2)=O)C1 N1(C(C2(F)CC2)=O)CC(NC(C(C)Oc2ccccc2)=O)CC12CCCCCC2 C1(NC(=O)COC(F)F)CCC(CNC(c2cnn(CC)c2)=O)C1.c1(C)nc[nH]n1 CC1(C(N2CCN(C(c3cc(C(N)=O)[nH]n3)=O)CC2)=O)CCC12CCC2 c1(OC)ccc(C)nc1C(N1CCSCC1CCNC(=O)CCc1cscn1)=O n1(CC(=O)NCC(C2CCC2)NC(C(C)C2CC2)=O)ccc([N+](=O)[O-])n1 C(=O)(CCC1C(=O)Nc2ccccc21)NC1C(C)N(C(c2cnccn2)=O)CC1 C(=O)(C(F)CCC(C)(C)C)NC(C(=O)NC(C=C)CO)(C)CSC Cc1coc(C(C)C)c1C(=O)NCCC1CCCCN1C(=O)C(F)OC(F)(F)F C(=O)(C1=NNC(=O)CC1)N1CC(C#N)(CNC(C2=C(C)CCC2)=O)C1 c1(C(=O)NC(CC)CN(C(C2C=CCC2)=O)CC)c(Br)c(C)nn1C c1(CC(=O)NCC2(NC(C3(C)COC(=O)N3)=O)CCCC2)ccc2sccc2c1 C1(CC#C)(C(=O)NC2C=CC(CNC(=O)Cc3ccc[nH]3)C2)CCOC1 c1(C(=O)NCCNC(c2ccc(CN(CC=C)C)cc2)=O)cc(C)cc(Cl)c1 c1(C(=O)NC2(COC)CCCN(C(=O)C(C)(C)F)C2)ccn2c(C)cc(C)nc12 n1(CC)nc(C)cc1C(N1CC2CC1C2C(=O)NCC(C)(CO)OC)=O Cn1nc(C(=O)NC2CC(F)(CNC(C3CC34CCC4)=O)C2)cc1C(N)=O N1(C(C(CC)(C)C)=O)CCC(C2(NC(c3cnc4sccc4c3)=O)CC2)C1 c1(C(=O)NCC(=O)NCCC2CCCO2)ccnc(OC)n1 C1(CCNC(C2OCCC2C(C)C)=O)(OC)CN(C=O)C1.C1(N)CC1C=C(C)C N1(C(C2(C)CCC(=O)NC2)=O)CC23CCCC2(C1)CN(C(=O)Cn1cnnn1)C3 N1(C(CCOCCCNC(=O)CC2CC3(CC3)C2)=O)CC12CCCCC2 Cc1cn2nc(C(N3CC(NC(=O)CCC(F)(F)F)C4(CC4)C3)=O)cc(C)c2n1 c1(NCc2cc(OC)nn2C)[nH]c(=NC(CCO)C(F)F)nc2c1ncn2C C1(CNC(C2CC=CC(n3cc(CSC)nn3)C2)=O)CN(C)CC(C)O1 O(NC(=O)C(CCOC)NC(c1cncc(OC)c1)=O)CC1CC(=C)C1 c1(-c2nc(CC)oc2)nc(C2CC2C)nn1CCc1cccs1 C1(CNC(CCSCCC)=O)CC(O)CN1C(=O)CC(C)(C1CCC1)NC(C)=O C1(C2CCCCC2)(C(=O)NC2C(NC(CN(S(C)(=O)=O)C)=O)CS(=O)(=O)C2)CC1 CCCCC(CC(=O)N(CC1=CCCOC1)C)NC(=O)C(C)c1cccs1 Cc1noc(CC(N2CC(CNC(=O)CC3(CS(C)(=O)=O)CC3)(CC3CC3)C2)=O)n1 C(=O)(C(C)CS(C)(=O)=O)Nn1cc(C(N(CCN(C(C)C)C2CC2)C)=O)cn1 c1(C(=O)NCC(O)CNC(c2cnc(-c3ccco3)s2)=O)cccc(C2CC2)c1 c1(C(=O)NC2CC3C(NC(=O)CCC4CC(F)(F)C4)C3C2)ccc2ccnn2c1 CC(C)C(C(=O)NC(C)CF)NC(=O)CN1CCCNC1=O C1(NC(C23CC(COC)(OC2)C3)=O)CN(C(=O)C(F)(F)C2CC2)CCC1C C1(CC(=O)N(CCNC(C2N(C(C)=O)CCC2)=O)C(C)C)CCC(=O)N1C Cc1ccnnc1C(=O)N(C(C)CN(C)C(c1ccc(C2CC2C)[nH]1)=O)C C=CCCCC(C(=O)NCC1NC(=O)NC1=O)NC(=O)C(F)C(C)(C)O N1(C(CNC(CC(C)C)=O)=O)CC2C(CC(=O)NC(C)Cc3nccn3C)C2C1 c1(NC(CCN(CC#C)C(C2CCC(=O)N(C)C2)=O)=O)cncc(C#C)c1 c1(OC)cnc(F)c(C(N2CCCCC(NC(C34CCCC3OCC4)=O)C2)=O)c1 c1(C(=O)NC(C(C(C)C)NC(=O)Cc2cc[nH]n2)C)cc(Cl)cc2cccnc12 C1(C(N(CC(=O)OC(C)C)C(c2ncn(C)n2)=O)=O)CCC(=O)N(C)C1 c1(C(=O)NCC2CCN(C(C(COC)(F)F)=O)CC2)cc(F)cc2cccnc12 C1(C(=O)N(CCN2CCCC2)Cc2cc(F)cc(C#N)c2)CN(CCl)CCC1(F)F c1(C(N2CC3C(C(=O)NCc4ccccc4)C3C2)=O)cc([N+](=O)[O-])sn1 c1(C(N(CCCCNC(C2C3(CC(OCC)C3)C2)=O)C)=O)occ2c1CCCC2 C1(CNC(=O)CN2CCCCC2)CCCC2(CN(C(C3CCCC3(F)F)=O)C2)O1 C1(C(CNC(c2cc(CCC)on2)=O)C)CCN(C(c2cnccc2C)=O)CC1 C(=O)(C1=C(Cl)CCOC1)N1C(CNC(C2CN3CCC2CC3)=O)CC(O)C1 Cc1oc(S(N)(=O)=O)cc1C(N1CCC(F)C(CO)C1)=O c1(C(=O)NC(CN(c2cc(C(=O)OCC)ncn2)C)C)ccc([N+](=O)[O-])c(C)n1 c1(-c2c(-c3n(-c4ncc(C)s4)ccn3)csc2)ccc2ncsc2c1 N1(C(=O)C=Cc2cccs2)CC2CCC(C1)N(C(C1CC1c1ccccn1)=O)C2 CN1N=CC(CC(=O)NCC2(F)CCN(C(c3c[nH]nc3Cl)=O)C2)C1=O N1(CC(=O)NCCC(C)(C)NC(c2c(SC)scc2)=O)CCCCCCC1=O C1(CN(C(=O)NCC)C(C2CCOC2)C)CCCC1(C)OC C1(C(=O)NCC2N(C(c3c(C)snn3)=O)CCC2)CC12CC(F)(F)C2 Cc1cc(C)c(C(=O)N(C2CC(NC(=O)COCCCF)C2)C)cn1 CCC(C)C(CC(=O)NCc1ccc(Cl)nc1)NC(c1cccc(CO)c1)=O c1(C(=O)OC)ccc(NC(C23CC2CN(C(=O)CS(C)(=O)=O)C3)=O)cc1O Cc1cc(N)cnc1C(N1CCOC(C(N2CCC(C)(C(C)C)CC2)=O)CC1)=O c1(-c2ccc(C(=O)NC3(CNC(c4csc(O)n4)=O)CC3)o2)cc(F)ccc1F C1(COC)(NC(=O)C(C2CCC2)OC)CCN(C(c2cn(C3CC3)nc2C)=O)CC1 c1(C(=O)NCCCC(C)NC(c2csc(Cl)n2)=O)[nH]ncc1C#N C1(C(=O)NCC2N(C(C(C)CC(N)=O)=O)CC2)CN2CCCN1CC2 c1(C(=O)NCc2ccc(C(F)F)nc2)ccc(N2CCCC2=O)cc1 c1(C(=O)NCCNC(C(CC)C2CCOCC2)=O)cnc2c(c1)c(O)nc(=O)n2C C#Cc1ccc(F)c(C(=O)NCCCNC(c2cc(Cl)c(C)cc2OC)=O)c1 c1(C(=O)NC2CCC(C(=O)NCC3CCN(CCC)CC3)C2)ccc(F)cc1C C1(CNC(C(C)(C)C2CCCCC2)=O)CCCCN1C(=O)Cc1ccc(O)cc1 c1(C(=O)NCCCCNC(C(C(C)O)N(C)C)=O)c[nH]c2ccc(F)cc2c1=O c1(C(=O)NCCCC2(NC(C)=O)CC2)cc(C#N)oc1C C(C(=O)NOCCC(=O)N(C)C)(c1ccco1)NC(C(CC)N(C)C)=O Cc1cc(C#N)c(O)nc1C(=O)N(C1CN(C(=O)CC2CC(O)C2(C)C)C1)C c1(C(=O)NCC(CNC(Cc2c(CC)con2)=O)CO)ccc2n[nH]cc2c1Cl c1(C(=O)NCCN(CCOC)C(c2cn(C)nn2)=O)cccc(OC)c1 C(=O)(C(C#N)C(C)C)N1CC(CNC(c2cc(C)on2)=O)C(O)C1 CCCCC(O)C(C)C(=O)NCCOC(C)(C)CNC(C12CCC(C1)OC2)=O c1(OC)c(C(=O)NC2CC2c2cccs2)cnn1-c1ccccc1 C1(NC(C2CCC(CC)O2)=O)CCCCN(C(=O)Cc2nc[nH]n2)C1 c1(C(N2CCN(C(C(CCC)OC)=O)C(C)C2C)=O)ccn2c1CS(=O)(=O)CC2 C1(CN(C(C2C=CCCC2)=O)CC)CCN(C(C2C(C)C2C)=O)CC1 c1(C(=O)N(CC(=C2CCCCC2)F)Cc2ccccc2)cc2occc2s1 C=C(C)CCC(=O)N1CC2CC2(NC(=O)CCc2ccc(N(C)C)cc2)C1 C1(C(=O)NCC2CC(OC)C2)(CC)CCCN1C(=O)Cc1c[nH]nc1O c1(C(N(C)CC2CCN(C(=O)CCN(C)C)C2)=O)cccc(-c2nnco2)c1 C12(C(=O)NCC(CC)NC(c3ccc(=N)[nH]c3Cl)=O)COCC1C2(F)F C1(N(C)C(c2cncn2C)=O)CCN(C(C2(C)C=CCCC2)=O)CC1 c1(C(N2CCC(N(C(=O)Cc3cn(CC)cn3)CC)C2)=O)cncnc1C1CC1 N1(C(CC(=O)NCC#C)=O)CCCC(NC(C2CC2(F)F)=O)C(F)C1 c1(C(=O)OCC)cccc2nc(N(C3CCC4CNCC34)C)[nH]c12 N1(C(CCSC)=O)CC2(C1)SCCC2NC(c1nnc(S)n1C)=O n1(C(C)C)cnc2c(NCc3nc(Br)cs3)nc(N3CCC4C(C3)C4(F)F)nc12 c1(C(N2CC(NC(C=C(C)Cl)=O)C(C(F)(F)F)C2)=O)cncc(N)c1C C1(=CC(=O)NCC(C)OC)CCN(C(=O)CCC2CC2(C)C)CC1 c1(-n2c(Cc3nnn(C(C)(C)C)n3)nc(CCOC(C)=O)n2)ccc(Br)c(F)c1 C1(C(=O)NCc2ncc(C)nc2)CN(C(=O)C(C)(C)F)CC1(F)F c1(C(=O)NC(CNC(C(COCC)(C)C)=O)(C)C)ccc(C)c(C)n1 CC1(C)COCCC1C(=O)NC1(C)CC(C(=O)NCC2(CO)CCCO2)C1 C1(C2CC2)(NC(c2cc(Cl)ccn2)c2n(CCCC)nnn2)CCOC1 c1(C(N2C(C(N(CCOC)C)=O)C3CCC2C3)=O)cc(Cl)cc(Cl)c1O C1(N2CC(C)NC(C)C2)CCN(C(=O)Cc2ccc(Br)cc2Cl)CCC1C CCCCCC(O)C(C)C(=O)N1CC(O)(CNC(C2CCSC2)=O)C1 N1(C(C2(COC)CCCO2)=O)CCCN(C(=O)CCCC(=O)NC(C)C)CCC1 c1(CCC(=O)NCC2CC(C)(NC(C(C)SC)=O)C2)cccc(F)c1Br c1(C(CNC(=O)C=CBr)NC(C(CSC)OC)=O)ccccc1F C=CCCCC(C)NC(=O)CC1CCCCC1NC(C1CCC1C#N)=O c1(OCC(=O)NCCN(CCOC)C(c2cccs2)=O)ccc(F)nc1 Cn1ccc2c(C(N3CC(NC(=O)CSC4CC4)C(F)C3)=O)ncnc12 Cc1nc(C(C)NC(=O)C(C2CCC2)NC(C2CC2(F)Cl)=O)n[nH]1 Cn1c(SCCC(=O)NCCCOCCNC(=O)C(N)=O)nc2ccccc12 Cc1occc(=O)c1OCC(=O)NC1CCC(C)N(C(C2CC2F)=O)C1 c1(C(C(=O)N(CC(C)NC(C2OCCCO2)=O)C)O)cc(F)cc(F)c1 C=CCC(CNC(=O)C(CC(=C)C)NC(=O)CC1CCC(=O)NC1)CC(C)C c1(C(=O)NC(c2cc(C)cc(F)c2)CO)ccccc1S(=O)(=O)C(F)F CCC(C)CCCCC(=O)NC(CC1CC1)CC(=O)N(C1CCCC1)CC(C)C N1(C(C(CCC)(C)C)=O)CCC2(CCCC2C(=O)Nc2n[nH]c(C(F)(F)F)n2)C1 CC1CCC(NC(=O)COCCOCCO)CN1C(c1cc(O)nc(O)n1)=O C1(CNC(C2(CO)CC(C)(C)C2)=O)CC2CCC1N2C(=O)CC1C=CCC1 C(c1cccc(O)c1)=CC(N1CC(C(N)=O)(CNC(c2cnc(CC)s2)=O)C1)=O C(=O)(C1=CCCOCC1)N1CCCC(CC=C)(C(=O)NC2CC(C(N)=O)C2)C1 C(=O)(C(C)(C(C)C)NC(C)=O)N(CCC)CCNC(C1CC1C#N)=O C(=O)(CCCC(=O)N1Cc2c[nH]nc2C1)N(C(C1CCCCC1)CO)C c1(CNC(C(c2cnn(C)c2)C)=O)c(Br)ccc2ccccc12 C1(C(CC)O)CCC(NC(=O)NC2C3CN(C(C)(C)C)CC23)CC1 N1(C(c2ccc(C(C)(C)C)o2)C(=O)N(C)C)CCC(F)(F)C(CO)C1.C1C(=O)N1 C(=O)(C(C)(C)CCCC(=O)NC(CNC(c1cc(F)ccc1F)=O)C1CC1)OC N1(C(C)=O)CCOC(C(N2CC(CO)(NC(=O)C(C)CN(C)C)C2)=O)C1 c1(C(=O)NC2C(C=C)CN(C(=O)CCNS(=O)(=O)CC)C2)cc2ccccn2c1 c1(NC(N(CCNC(=O)C(C(C)C)OC)CC)=O)cn2cc(Cl)ccc2n1 C1(CNC(CCCCN(C)C(C2CCC(C(N)=O)C2)=O)=O)OC(=O)NC1(C)C CC1C(NC(C23COC(CCO2)C3)=O)CC2CCC1N2C(C1(F)CCC1)=O c1(NC(=O)NC(COC(=O)CC=C(Cl)Cl)=O)cc(Cl)cc(Cl)c1F Cc1cc(NC(=O)C(=O)NC2CC3CC(CO)CC23)cc2cccnc12 Cc1nn(C)c(C)c1C(=O)NCC1(NC(=O)CCc2cncc(O)c2)CCC1 N1(S(CCOC)(=O)=O)CCCC(NC(C2(CC(F)(F)F)CCCOC2)=O)C1 N1(C(c2cc(C)oc2)=O)CCC(F)(CNC(C2(CO)COC2)=O)CC1 c1(C(=O)NC2C3CN(C(C4CCN(C(C)=O)C4)=O)CC2C3)ccc(C)c(C)c1O N1(C(c2c(OC)c(=O)cco2)=O)CC2CC(O)C1C2NC(C1CC2(CCC2)C1)=O c1(-c2scc(CC(=O)NC3(C)CC(CN=[N+]=[N-])C3)n2)ccc(F)cc1 N(C1CCCc2occc21)C(CCN(C(=O)C(C)OCCN(C)C)CC#C)=O c1(C(N(C2CCN(C(C3CCC3(F)F)=O)C2)C)=O)ccc(N)c(N)n1 Cc1cc([N+](=O)[O-])cnc1C(=O)NC1CCN(C(=O)C=CCF)C1 c1(C(=O)NC(CCN(C(C(CCOC)C)=O)C)C(C)C)[nH]nc2c1CCC2(C)C CC1(C)C=C(C(=O)NCC(O)CC(=O)NCCc2cccnc2O)C1 C1(CNC(C(=O)NCC)=O)CCC(NC(c2csc(C(C)(C)C)n2)=O)CC1 c1(N(C)CC2CCCCC2O)nc2c(c(=NCC3(C)CCCO3)[nH]1)COCC2 c1(CC)cccnc1C(=O)N.C1(C(C)C2=CC=C2)CCN(C(=O)CN(C)S(N)(=O)=O)C1 N1(C(CNC(C)=O)=O)CCCCC(NC(c2cc(F)cc(Cl)c2)=O)C1 C=CCC(C)(C)CC(=O)N(CC(C)NC(c1ccc(OC)c(Cl)c1)=O)CC c1(C(=O)NCC(CNC(=O)C(F)(F)CO)CO)ncc(Cl)cc1F N1(C(CC(C)O)=O)CCC2C(C(=O)NCc3ncc[nH]3)C2C1 c1(C(=O)NC2CC(NC(CS(CC)=O)=O)C2)cc(O)nc(OC)n1 C(CC(C)C)(C(=O)NCc1cnc(C)s1)NC(CC=C)=O C1(C(N2CC(CNC(C(n3ncc(C)c3)C)=O)C2)=O)OCC2CCCC1C2 CC1(NC(=O)CCOC2CCCC2)CCN(C(C23CCC2C3)=O)CC1 N1(C(C(C)OCCC=C)=O)CC2(CCC2)CC1CNC(=O)Cn1ncnn1 N1(C(C=Cc2c(C)ncs2)=O)CC2CN(C(=O)CC3CN(C)C3)CCC2(CO)C1 C(=O)(C1=CCc2ccccc21)NCC1CC2CCC1N2C(c1c(C)cno1)=O C(C)(C)(CCC(=O)NC1CCSC1)NC(c1cccc(CC)c1)=O c1(C(N(CCC(C)NC(CC(=O)NCC)=O)C)=O)ccc2ccn(C)c2c1 C(CC(=O)NC1(CO)CCCN(C(=O)C(C)N(C)C)C1)(C(N)=O)NC(C)=O C(CC(=O)NCCc1nncs1)(C(F)(F)F)NC(CC=C)=O c1(OC)cccc2scc(CN(C(=O)C(=O)NCCOC3(C)CS(=O)(=O)C3)C)c12 CC1CN(C(=O)Cc2ccon2)CC1NC(c1coc(Cn2cccn2)c1)=O Cc1cc(N)c(C(=O)N(C)CCOCCCNC(=O)CCc2cnc[nH]2)c(F)c1 c1(NCC=C(C)C)[nH]c(=NCC2CCOC(C)C2)nc2c1cnn2C N1(C(CN(CCC)C)=O)CCN(CC(C)NC(c2cnc(CC(C)C)[nH]2)=O)CC1 c1(C(N2CC3(CC(CC(=O)NOCC4CCCC4)C3)C2)=O)cc2ccccc2o1 C(N=c1[nH]nc(C(F)(F)F)s1)C1CN(C(C=C(C)C)=O)C(C)C1 c1(C(=O)NCCN(CCC)C)cc(C(C)C)cnc1O.N12CC3CC3(C1)C2=O C(C(=O)NC12CC1CN(C(c1csc(C)c1)=O)C2)(C(F)(F)F)OC(C)=O c1(N2C(C3(NC(c4c(C)n[nH]c4C)=O)CC3)CCC2)nccc(S(C)(=O)=O)n1 C=CC(C)(C)CC(=O)N(C1CCCCC1N(C(=O)CC1CCCC(=O)N1)C)C C(N=c1cc[nH]c(=NCCC2CCC(S(C)(=O)=O)CC2)[nH]1)c1cn(C)nc1CO N1(C(c2c(CC)nns2)=O)CCOC(CCC(=O)N(CC(F)(F)F)CC)C1 N1(C(CS(C)(=O)=O)=O)CCC(O)(CNC(c2ccnc(CO)c2)=O)CC1 C1(C2CCCN(C(=O)Cn3nnc(C)n3)C2)(NC(CC2CC(OCC)C2)=O)CC1 CC1(NC(=O)C(O)CCn2cncn2)CCCC1(F)F.C12(CC1)CC(=O)N2 N1(C(c2nc(C)oc2C)=O)CC2CCCC2(NC(C2C=C(C)CS2)=O)C1 c1(C(N(CCCN(C)C(C2(C)CCNC2=O)=O)C)=O)ccc(N)c2ccccc12 C(CCCCCCCO)=CC(=O)NCCCCCNC(c1cn2c(n1)SCC2)=O Cc1cccc(C(N2CCC3C(NC(c4ccn(C5CCCC5)n4)=O)C23)=O)c1F c1(C(=O)NCCN2CCC(NC(C(CC)(C)O)=O)CC2)ccc2ncnn2c1 C1(C(=O)NC(CC)CC(=O)NC2CC(C)(C(N)=O)C2)CCN(C)C(=O)C1 N1(C(C2(C)C=CCCC2)=O)CC2(NC(=O)C3=CCCCO3)CCC1C2 c1(C(=O)Nc2c(OC)ccc(C#N)c2)c[nH]ccc1=Nc1ccccc1 c1(C(N(CCCN(C(C(C)n2cccn2)=O)C)C)=O)cc2cc(F)ccc2cn1 N1(C(C(C)OCCOCC)=O)C(C(N2CCC(N(C)CC)C2)=O)CCC12CC2 N1(C(C2CCCN2CC(F)(F)F)=O)CCC(F)(F)C(CNC(C23CCC(C2)C3)=O)C1 C(CCCOC)(C(=O)NCCc1cccc(O)n1)NC(C(C=C)(C)C)=O c1(C(=O)NC(C2CCOC2)CNC(=O)CC2CCCCC2)coc2c1CS(=O)(=O)C2 CCC(CO)(C(=O)N1CCC(C(N2CCC(C)(OC)CC2)=O)C(C)C1)OC CC1(C)CC=C(C(=O)NCCC2(O)CCN(C(c3ccc4c(c3)CC4)=O)C2)CC1 C(c1cnc(O)nc1O)=CC(N1CC2(CCN2C(=O)Cc2cccs2)C1)=O c1(SCC(N2CC(CNC(C=NOC)=O)OCC2)=O)c(C)cccc1C c1(CNC(CCCC(=O)OC)OC)cnc2n1NCCC2 N1(C(C2C(C=C)CC2)=O)CC(CNC(c2cccnc2OCC)=O)CC(C)(C)C1 c1(C(N2CCC(N(C(C3SCCC3C)=O)CC)CC2)=O)cc(F)cc2c1CCC2 CC(C)CC(F)(F)C(=O)N1CC2CCCC2(NC(=O)CC2CCC(C)(C)CC2)C1 N1(C(CCNC(c2ccco2)=O)=O)CCCOCC1CNC(=O)CC(F)(F)F C1(CCN(CCCNC(CC(C(=O)OC)(C)C)=O)C)CNC(=O)CC12CCOC2 CCC(C(=O)NCC(CC)NC(c1nc(C(C)C)ncc1Cl)=O)C(C)(C)CC CC1CCOCC1C(=O)NCC(CO)NC(c1ccsc1)=O c1(CC)cncc(C(=O)NCC2(NC(c3cc(C)c(CC)s3)=O)CCOC2)c1 c1(CN(C(C2C(CC)OCC2)=O)C)cccc(CNC(=O)CC2(C)CC2(Cl)Cl)c1 c1(C(=O)NC(CCC)C(=O)N2CC(N(C)CCO)C2)ccc2c(c1)CCC2 N(C1CCCc2ccccc21)C(Cc1cc(OC)cc(SC)c1Cl)=O C(C)(C(C)(C)C(=O)NCC(O)CC1CCC1)NC(CCC#CC)=O C1(N(C(=O)CCc2cncnc2)C)CN(C(=O)Cn2ccccc2=O)CC1F N1(CCOC)CCN(C(C)CNC(c2ccc(I)s2)=O)CC1 N1(C(Cc2c(OCC)cccc2Cl)=O)CC2(CCN(C(=O)CS(C)(=O)=O)CC2)C1 C(N=c1ccnc(C)[nH]1)C1CCCCN(C(C(C)NS(CC)(=O)=O)=O)C1 c1(NCC2(CC#C)CC2)cccc(-n2ccc(C)n2)c1 C1(CNC(Cc2ccc(C)o2)=O)CN(C(c2ccn(CC(C)C)n2)=O)CC1(C)C C1(NC(CSCCOC)=O)CCN(C(c2cnc(O)n2C)=O)C(C2CC2)C1 C1(NC(c2ccns2)=O)CCSC12CN(C(=O)C(F)(F)c1nccs1)C2 c1(NC)cc(C(=O)NCC2CC3(CC(NC(=O)C(C)(C)OC)C3)C2)cc(Cl)n1 N1(C(c2n(CC)ccc2)=O)CC2(CNC(C3(C#N)CCCCC3)=O)CCC1CC2 C(=O)(C1=CCCCC1C)N(CCNC(C1(C)CC(=C)C1)=O)CCC CC1CCc2c(C(N3CCC(Cn4cc(C(C)(C)CC5CC5)nn4)C3)=O)csc2C1 Cc1cccc(Cl)c1C(N1CCCC(CNC(C2CC2c2ccccc2)=O)C1)=O C1(C(N2CC=CC(NC(C3(OC)CCCCC3)=O)C2)=O)CCN(C2CC2)S1(=O)=O C1(COC)(NC(=O)CC(C)(C)O)CCN(C(c2ccnc(C(F)(F)F)n2)=O)CC1 CC1(C(=O)NCC(N)=O)CC12CCN(C(c1ccc(C#N)cc1)=O)CC2 c1(C(=O)NCC(C2CC2)NC(C2C(CC(C)C)C2)=O)c[nH]c2cnc(Cl)cc12 C1(C2CCN(C(=O)CC3CCCC(F)(F)C3)C2)(NC(=O)CC2CC3(CC3)C2)CC1 CCCCC(=O)C(=O)N1CCCC1CCC(=O)NCc1cccc(CC)c1 C1(C(N2CC(NC(c3ccc(C4CC4)o3)=O)C3(C2)CC3)=O)Cc2ccccc2S1 c1(C(N2CCC(c3cnn(C)c3)C2)C(=O)NC(C)C)ccc(CO)o1 CC(CCc1ccccc1)C(C(=O)Nc1ccccc1)N(C1CCCCC1)C N#Cc1cnc(C(N2CC3CC3(C(N)=O)C2)=O)c(Cl)c1 C1(CC)CCCCC1NC(=O)Cc1csc(COC)n1 C=CCCCCCCCC(=O)N(CC(O)CN(C)C(c1ccc([N+](=O)[O-])[nH]1)=O)C C(C(=O)N1CCC(NC(c2cc(Br)c(C)o2)=O)C1C)(C(F)(F)F)OC(C)=O C1(C)(C(=O)NC(CC=C)(C)C)CCCN(Cc2nc(C3(S(N)(=O)=O)CC3)no2)C1 C1(C(=O)NC(C2(O)CCC2)(C)C)CC(NC(c2nocc2Cl)=O)CCO1 C12(NC(c3c(CC)n[nH]c3)=O)CCC1CN(C(C1(C)CCC(C)CC1)=O)C2 C1(C(=O)NCC2CCN(C(C(CC)C#N)=O)CC2)CCc2nnc(O)n2C1 C1(NC(C=NOC)=O)COCCN(C(=O)C(c2cncn2C)=O)C1 c1(CNC(=NC)NCC(C)(C)CCCO)cccc(S(N)(=O)=O)c1 N1(C(C(c2cn(C)nn2)NC(=O)Cc2cnc(S)nc2)=O)CC(F)(F)C1C1CC1 CC1OCCN(C(=O)CN2CCOCC2)C1C(=O)NC(COCCNC)C c1(C(=O)NC2C3N(C(CCCCC=C)=O)C(CC3)C2)cnc2nccn2c1 C1(CC)CCC(C(=O)NCC(CNC(c2[nH]ccc2COC)=O)OC)O1 Cc1ccc(C(N2CCCCC2C(C)NC(C23CCC2CC3)=O)=O)cc1O C(=O)(C(F)(F)C(C)(C)O)N1CCCC(C)(NC(C=CC(C)N(C)C)=O)C1 C#Cc1cn(C)nc1C(=O)NCc1ccc(CNC(=O)C(C)CS(C)=O)cc1F N1(C(=O)C(F)CC2CCC2)CCC2CN(C(C3(F)CCC3)=O)CC2C1 c1(C(N2CCC(C(N(C3CCN(C)C3)CCC)=O)C2)=O)cccnc1Br C(=O)(CC(=O)NCC(C1CCCC1)NC(=O)CN1CCCC1C)NCC#C CC1C(NC(c2cc(C#N)on2)=O)CCCN1C(=O)COc1ccc(Cl)c(Cl)c1 Cc1cc(C(N2CC=CCC2CNC(C2(CO)CC(C)(C)C2)=O)=O)sc1C N1(C(CN(C)C(c2cscn2)=O)=O)CC(NC(c2cccc(Cl)n2)=O)CC(O)C1 C(=O)(C1=CCCC1C)NC(CN(C(C1(c2cccnc2Cl)CC1)=O)CC)C N(C)(C[Si](C)(C)C)Cc1ccoc1C(=O)OC.C1CC(=O)NCCO1 C1C(C)CC(=O)N1.Cc1nn[nH]c1C(=O)NCC(O)COC(C)C c1(C(N(C(CNC(COCCCC)=O)CC)CC)=O)cnc2c(c1)nc(O)n2C Cc1ccncc1C=CC(N1CC(F)(F)CC1CNC(C1CC1C(C)(F)F)=O)=O C(=O)(CCS(N)(=O)=O)NCc1n(C)nnc1C(=O)Nc1c[nH]nc1C(F)(F)F CCC(C)C(=O)OCC1CC(NCC(N2CC=CC2C(=O)OC(C)(C)C)=O)C1 C(=O)(C1Cc2ccc(F)cc21)N(CC(C)(C)NC(c1ccc(O)cc1)=O)C C(=O)(C#CC1CCCCO1)N(CC(C)O)CCNC(=O)CCC1CCOCC1 N1(C(CNC(=O)OC)=O)CCC(O)C(NC(=O)CC2CCOCC2(C)C)C1 c1(C(N(CC(CNC(c2c(CC)cno2)=O)O)C)=O)nccc2ccn(C)c12 S(=O)(=O)(c1cnc(NC(c2ccc3c(c2)CCO3)C)cc1C)NCCCCCC N1(C(c2nncn2CC)C(=O)NC(CC)C)CC(CO)OCC1C CCCC(C(=O)NCc1ocnc1C(=O)NCCc1scnc1C)N(C)C Cc1cc(C(=O)NCC2(CNC(C3CCS(=O)(=O)N3)=O)CCC2)ccc1C(F)F N1(C(c2c(C)onc2)=O)CCN(C(=O)C(=O)N(C)C)C(CCO)C1 N1(C(C(C)NC=O)=O)CCC(CNC(=O)CN2CCNC(=O)C2)C12CC2 N(C(=NCCCCCCC1CCOCC1)NC1C(F)(F)C12CC2)C1C(C)C1C CS(=O)C1CCC(NC(=O)NCC2CCC(OC(F)(F)F)CC2)C1 C1(CNC(c2nc(CCOC)oc2)=O)CN(C(C2CC3CC3C2)=O)CC1C(C)C C1(C(N2CC(C3CN(C(C(CC=C)(C)C)=O)C3)C2)=O)Cc2cc(Cl)ccc2O1 c1(NCC(C2CC2)SC)nccc(=NCCCc2ccc(O)nc2)[nH]1 N1(C(c2cc(COC)no2)=O)CCOC(CN(C(=O)C(C)CCOC)C)C1 c1(OC)cc(I)c(C(N2CC(C(=O)Nc3c(Cl)ccnc3Br)C2)=O)cc1OC N1(C(COCCOC)=O)CC(CNC(=O)CCCCCNC(C)=O)CCC1C CC(C)(CN=c1[nH]c(=NC2CC(F)(F)C2)[nH]c2ccsc12)c1ccccc1Br C=CCC(C)(C)C(=O)NC1CC2CC1N(C(=O)CCc1cccnc1C(F)(F)F)C2 C12(CNC(C3CC(NC(Cc4n(C)ccc4)=O)C3)=O)CCN(CC1)CC2 n1(C(CC)C)cc(C2CC(C(N3CCCC3C(=O)OC)=O)(NC3CC(O)C3)C2)cn1 c1(C(=O)NCC#Cc2cccc(F)c2)nc2ccccc2c2ncccc12 N1(C(CC2CCCN(C(C3(C#N)CCC3)=O)C2)=O)CCCC(C2CCC2)C1 C(=O)(C1CCCc2scnc21)Nc1cc2[nH]nc(C(C)(C)C)c2cc1 c1(CC)nc(C)n(C)c1C(=O)NCC(C)(C(C)C)NC(=O)Cc1cncnc1 N1(C(C2C(CNC(C(C=CCCC)O)=O)CC2)=O)CC(CO)C(O)C1 CCCCC(C(=O)NC1CN(C(=O)COCC2CCCC2)C2(CCC2)C1)C(C)C C1(C(=O)NCC(CC)(C)NC(c2cc(C3CC3)[nH]n2)=O)CCC(=O)N(C)C1 c1(Cc2cccc(COC)c2)ccc(C)c(C(N2CCCC2C(=O)NCSC)=O)c1 CC1=C(C(=O)N(CCCNC(c2cnn(C)c2F)=O)C2CC2)SCCO1 c1(N2CCN(C(=O)Nc3ccc(Cc4cncs4)s3)CC2)cncc2nnnn12 CC1NC(=O)CCC1NC(=O)CC1CCCCN1C(=O)CC1CNC(=O)O1 c1(C(N2C(C3CCN(C(C(F)=CC)=O)C3)CCC2)=O)ccc2ncnn2n1 c1(CC)ccc(C(N2CC(NC(c3cncc(N(C)C)c3)=O)CC2C)=O)cc1N C(C)(C)(C(=O)NCC1(CO)CCC1)C1(C)N=N1.C1(C(C=O)F)CCOCC1 C1(C(N(C2(CC(=O)NC3C(SC)COC3)CC2)C)=O)CC(C)CCO1 O=C(C1=CS(=O)CCC1)NC1CN(C(=O)COCc2nc[nH]n2)CC1C(F)(F)F Cc1cc(NC(C2CC2C(N2CCCN(C(CC(C)C)=O)CC2)=O)=O)nc(C)c1 C=CC1CN(C(C2CC3(CCC3OC)C2)=O)CC1NC(c1ccc(CO)nc1)=O CCC(C)CCCC(=O)N1CCOCC1CC(=O)NC1(c2cccs2)CC1 CC1CN(C(C2C3C4CCC(C4)C23)=O)CC(C(N2CCC(C3CC3)C2)=O)O1 C1(O)(CNC(C(C)OCCC#C)=O)CCN(C(c2cc(CCC)n(C)n2)=O)C1 C(=O)(C#CC1CCCCC1)NCC1CC(C)N(C(=O)Cc2csc(C3CC3)n2)C1 CC(C)CC(C(=O)NC(CO)C(C)NC(c1c2c(nn1C)CCC2)=O)C(N)=O N1(C(CC(=O)NCC)=O)CC(CNC(c2coc(Cl)n2)=O)C2CC12 C1(C2CCCCC2)(C(N2CCCC(CNC(=O)CCC3CC3)C2)=O)CCCCC1 c1(C(N(CC(C)CNC(C2CC2F)=O)C)=O)ccoc1NC(=O)OC(C)(C)C C1(C2CC2)(NC(C(CCC)O)=O)CCN(C(=O)Cc2cnc3n2CCCC3C)C1 c1(C(=O)NC(C(C)C)C(C)NC(c2cnsn2)=O)ccc2c(c1)S(=O)(=O)NC2 Cc1cnc(C(N2CC(NC(=O)CN3CCS(=O)CC3)CC2CO)=O)cc1C#N c1(C(=O)NC(CNC(c2ccc(CC)nc2)=O)C)ccc(F)c(C(F)F)c1 c1(C(N2C(CNC(CCCOC)=O)CC2)=O)ccnc(-n2cncn2)c1 O=C1CC(=O)NC(C(=O)NCc2ccoc2C(=O)NCC2CC2C2CCC2)C1 CCCCCCCCC(C)C(=O)OCC.C12C(C1(F)F)NC2=O C1(C(N(CC(CO)(CO)NC(C2C=CCS2)=O)C)=O)C2CCCCCC12 c1(C2C(C(N3CC(NC(C=CCN(C)CC)=O)C(OC)C3)=O)C2)cccc(C#N)c1 CC1CCC(=CC(=O)NC2CCCC2NC(=O)CC2COCC2O)C1 N1(C(c2c(N)nccn2)=O)CC=C(CCNC(c2csc(Cl)c2Cl)=O)CC1 C(=O)(CC(C)(C)C)NC(C)C(=O)N(C(C)CNC(c1cc[nH]c(=N)n1)=O)C C(=O)(C(C)C(C)(C)C)N1CC(NC(c2cc(CCC)c(C)s2)=O)C(CC)C1 C1(CC(=O)NC2CCC2NC(c2cc(Cl)cs2)=O)CCCCC1O c1(C(C(C)NC(=O)Cn2cnnn2)NC(C2C(CCC)C2)=O)ccccc1 CS(C)(=O)=NCC(=O)NCC1OCCC1C(=O)NCCc1ccncc1F C1(C(=O)OCc2ccc(Br)c(C(F)(F)F)n2)(CO)CCC(F)(F)CC1 CC(C)C(CNC(c1cn(C2CCOC2)nn1)=O)NC(C1(C)CCCO1)=O Cc1cn(C(C)C)cc1C(=O)NCC(O)CCNC(=O)CCc1ccn(C)c1 C(CCCCCCCCCO)NC(=O)Nc1cc2ccc(O)nc2s1 N1(C(CC=CCC)=O)Cc2[nH][nH]c(=NC(=O)c3ccc(O)cc3)c2C1 C1(C(N(C)CC2CCN(C(=O)Cc3cccnc3)C2)=O)CCC2(CCCC2)CC1 c1(C(=O)NCC2C(CNC(=O)COC3CC=CC3)C2)cc2c(Cl)nccc2o1 Cc1ncc(C(N2CCC(CNC(C3CC34CCC4)=O)C23CC3)=O)cc1N C1(CC(=O)NC(CC)CN(C(=O)CN(C)C2CC2)C)OCCOC1(C)C Cc1ccn(C(C)CNC(c2cc(CNC(=O)Cn3cnnc3)cs2)=O)n1 C1(C(=O)NC2C(CNC(c3ccnc(C)c3C)=O)COC2)CC2CCCC(C1)C2 C1(C(N2C(CCC#C)CCC2)=O)(NC(=O)C=CC(C)(C)SC)CCCC1C c1(C(=O)NC(C)CN(C)C(C2CCOC2c2ccccc2)=O)ccn2ccsc12 Cn1ccn2cc(C(N3CCC(C)(CNC(C4C5CCCC45)=O)C3)=O)nc2c1=O CCCCC(O)C(=O)NCc1ccc(CNC(=O)Cc2cccnc2Cl)c(F)c1 C(=O)(C1=CCCCC1C)N1CC(CC=C)(C(=O)NCC2CC(CO)CO2)C1 Cc1oc(C2CC2)nc1C(N1CCCC1C1CCCN(C(=O)CSCC2CC2)C1)=O c1(CNCC2(C(=O)OC)CNCCC2)c(Cl)c(COC)nn1C N1(C(C=C(CC)CC)=O)CCN(C(C2(CF)CC3(CCC3)C2)=O)C(C2CC2)C1.C(=O)OC C12(CNC(C(C)(C)O)=O)CCC1CN(C(=O)CCN1CCCCC1=O)C2 C1(CCNC(C(c2ccccc2)C)=O)CN(C(=O)C2=CCSC2)CCS1(=O)=O C(CCC(O)C(=O)NC1CC2CC2C1)NC(CN1CC(C)(OC)C1)=O CCCCC(C(=O)N1CC(N(C(=O)CN2CCS(=O)CC2)C)C1)C(C)C Cc1cccc(C(N2CCC(O)(C(=O)N(C)C)C2)=O)c1N CC1CN(Cc2cccc(Br)c2O)CCCN1C(c1ccc(F)c(Cl)c1F)=O N1(C(CC2(C(=O)OCC)CCC2)=O)CCOC2C(C(F)(F)F)C12 Cc1cnc(Cl)[nH]c1=NCC1CCC2(CCC2)C1NC(c1ccc(Cl)nn1)=O C(CC(C(C)C)NC(c1ccc(C)nn1)=O)N(C(Cc1nc(CC)sc1)=O)C c1(C(=O)NC2C(NC(C(c3c(C)ccc(F)c3)(F)F)=O)C2)ccc2nsnc2c1 N1(C(C2C(C)(C(=O)N(CCCO)CC)C2)=O)CCN(c2ccc(CC)cn2)CC1 n1(CCC(=O)N(C2CCC(NC(=O)CC3CC=CC3)C2)C)ccnc1O N12CCCC(CC1)C2=O.C(CC(COC)NC(=O)CSC)OC.C(=O)(C(C)C)NC C(C)(CC(F)(F)C(F)(F)Br)(c1n(CC)nnn1)NCc1ccc(C(C)(C)O)cc1 c1(CNC(C(C(C)C)NCCCC2CCCO2)=O)cc(S(=O)(=O)N(C)C)c[nH]1 N1(C(C)=O)CCC2(C1)CN(C(c1csc(C3CC3)n1)=O)CC(C)O2 n1(CCOC)nc(C(=O)NCC(O)Cn2cccn2)ccc1=O O=C(C(C1=NOC2CC12)N1CCN(C2CCC2)CC1)NCc1ccoc1 c1(C(CC)C)nc(-c2nc(-c3cnn(C)c3)cs2)n(CC(C)(C)C)n1 N1(C(c2cc(CC)[nH]n2)=O)CC(NC(c2ccc(OC3CC3)cc2)=O)CC1C CC1CC(C)N(C(=O)CCCCCc2ccccc2)CCN1C(c1cncs1)=O c1(C(N2CCCC(C(C)NC(=O)C(c3cccs3)N(C)C)C2)=O)cncc(F)c1C c1(CCC)cc(C(=O)NC2CN(C(C3(C4CCCO4)CC3)=O)CC2C)ccc1F C1(CNC(=O)CSc2n[nH]c(O)n2)CN(C(C2(O)CCOCC2)=O)CC2(CCC2)O1 c1(NCCCCCSC)cc(Br)ccc1S(=O)(=O)N1CC2CC1CS2(=O)=O N1(C(CSCC2C(=O)OCC2)=O)CC2(C1)CN(C(c1cccc(CCO)c1)=O)C2 Cc1cnc(NCc2ncccc2C)c(S(=O)(=O)NCC2CCC(O)C2)c1 c1(C(=O)NCCCOCCNC(C2CCN(OC)CC2)=O)ncc2n1CCCC2 c1(C(=O)NC(C2(OC)CCC2)C)c[nH]nc1CNC(c1cc[nH]n1)=O Cn1nc([N+](=O)[O-])cc1C(=O)NC1CCC(CNC(C2(C#N)CCCCC2)=O)C1 c1(N(C(c2cncc(-c3cnc(NC)nc3)n2)=O)CC2CC2)cc(O)nc(=N)[nH]1 C(C(C)CC(=O)NCc1cncnc1O)NC(C=CCN(C)CC)=O CC1CCN(C(C2(C)CC(=O)C2)=O)CC1N(C)C(c1cncn(C)c1=O)=O C1(CN(C(c2ccc(OC)o2)=O)C)CN(C(=O)CCC(C)(C)F)CC12CC2 c1(C(N2CCC(N(CC(C)O)C)CC2)C(=O)NCCSC)csc(C#N)c1 N1(C(c2n(CCC)ncc2)=O)CCC(NC(=O)Cc2nocc2C)C1C c1(NC(c2nnnn2CCCF)(CC)C2CC2)ccc(OC(F)F)cc1C(C)C C1(N(C)C)(C(=O)NCC2CC(NC(C3(c4ccno4)CCC3)=O)C2)CC(CO)C1 N#Cc1ccc(C(N2CCC=CC2C(=O)NOCC2CCOC2)=O)cc1 N(C(=NCC(C)c1nccs1)NCc1ccc(F)cc1)C(CC)C N1(CC)CC(C(N2CCC2CNC(c2cccc(O)c2Cl)=O)=O)CCC1=O CC(C)(CNCCCC1CC1(F)F)C(N)=O C12=NNC(=NC(=O)N1)C=C2.C1(N(CC)CC)CCCN(CCS(N)(=O)=O)C1 c1(C(N(C2CCN(C(=O)C#CC3(C(F)(F)F)CC3)C2)CC)=O)cc2ccccc2s1 c1(C(=O)NCC(CCCC)NC(C2(F)CC2)=O)cc(F)c(F)cc1NC(C)=O c1(C(=O)NCC2CCC(NC(CCCCC)=O)CC2)ncc2c(F)cccn12 N1(C(CC(CC)SC)=O)CCN(C(c2cc(C)cc(Cl)c2)=O)CC1C1CCC1 N1(C(C=Cc2nc(C)sc2)=O)CC(CNC(c2coc(CO)c2)=O)CC(C)(C)C1 C1(C)(CNC(=O)NC2(CC)CCCC2)CCCN1C c1(CNC(C(CSC)O)=O)nc(C)c(C(=O)NCC2(C)CCCC2O)o1 C1(NC(c2ccnc(C3CCCC3)n2)=O)C=CCN(C(C2(C(F)(F)F)CCC2)=O)C1 c1(C(=O)NCCNC(CC(C(C)C)O)=O)cc(Cl)c(O)c(Cl)c1 Cc1ccncc1C(=O)NCC1CCCN1C(c1cccnc1N)=O C(=O)(C(Cc1ccccc1)N1CCCCC1)N(C(C1(C(F)(F)F)CC(F)C1)=O)CCO N1(C(CC2C(C)(C)C2)=O)CC(NC(=O)Cc2ccc(C(F)(F)F)nc2)C(O)C1 c1(CN2CC(CC(=O)NCc3cc(F)cc(Cl)c3)C2)cn2cc(Cl)ccc2n1 c1(CCn2cc(C3COC(C)(C)O3)nn2)ccc(Br)cc1Cl C(=O)(C1=CC2(CN(C(c3csc(C)c3)=O)C2)OC1)N1CC(C(=O)OC)C1 C1(C)CCN(C(=O)NCCNC(C2(C)CC2)=O)C1.C(c1cccs1)=NC(=O)OC(C)(C)C N1(C(c2c(CC)non2)=O)CCC(NC(c2nc(Cl)sc2C)=O)CC1C N1(C(c2c(OC)csc2)=O)CC2CCC1CN2C(=O)CC1CC1C C1(C)CCCCN1C(=O)COCCCC(C)C.Cc1nnc(CCNC(COC)=O)s1 c1(C(N2C(CC)CN(C(=O)Cc3csc(C)n3)CC2)=O)cn2ncnc2nc1C Cc1nc(C(C)C)sc1C(N1CCC(C)C1CNC(=O)C(F)(F)C1CCCC1)=O C1(C(=O)NCC2CC(NC(C34CC(C(=O)OC)(C3)C4)=O)C2)CCCC1S(C)(=O)=O c1(OC)ccc(C2CC2C(=O)NCCCC(C)NC(C2(CO)CC=CC2)=O)cc1 C1(CCC)(NC(c2cc(C)nc(C)c2)=O)CCN(C(=O)C=C2CCC2)CC1 C(=O)(CC(C)P(C)(C)=O)NCC(C)N(C(CCN(C)CC)=O)C C12(C3CCN(CC3)CC(=O)N1)CC2.c1(NC(CN(C)C2CC2)=O)ccccc1F C1(CCOC)(NC(C2C(C)(C)C2(C)C)=O)CCN(C(=O)C(O)C(F)F)C1 c1(N(CCCNC(=O)C(C)C2CCCC2)C(C)=O)cc2nncn2cn1 Cc1cnn2cc(C(=O)N(CCNC(=O)C=Cc3ccccc3)C(C)C)cnc12 CCC(F)(F)CC(=O)NC(C)Cc1ccc(CNC(C2(C)CCCCO2)=O)cc1 N1(C(C2C(OC)CCC2)=O)CC(CNC(=O)C=C(C)C(C)(C)C)C(C)(C)C1 C(C(COC)CC(=O)C12C(C1(F)F)C(=O)N(C(C)C)CCNCCC2)OC Cc1nc(O)nc(C)c1CC(N1CC(CNC(=O)C(C)CC(F)F)C(C)(C)C1)=O C(CNC(c1c(Br)noc1C1CC1)=O)(C(C)(C)C)NC(C1C(=C)C1)=O CC1=C(C)C(C(N2CCC(C3CCCCN3C(=O)Cc3ccno3)CC2)=O)CC1 C(=O)(N=c1[nH]n(C)cc1I)c1cccc(C(CC)O)c1 CC(CC(=O)NC1CC2CCC(C1)N2C(C12CCCCC1C2(F)F)=O)C(C)(C)C Cc1ccnc(C(N2CCCC(CNC(c3csc(-c4cn[nH]c4)c3)=O)C2)=O)c1 C1(NC(CC(=C)C)=O)COCCC1C(=O)NC1N(C=O)CCC1.SCC c1(C(N2C(C(=O)NC(c3onc(C)n3)C)CC(F)C2)=O)cncc(F)c1C N1(C(CCOCC)=O)CCC(C(F)(F)F)C(NC(c2ncccc2C)=O)C1 C(CCCC(=O)NC1CCC(NC(C2CC(C)(C)C2)=O)C1)OCC c1(C(N2C3CN(Cc4cc(OC)cc(Br)c4)CC32)=O)cccc2ccncc12 C(=O)(CC(C)C(C)(C)NC(c1ccc(CO)cn1)=O)NCc1n(CC)c(C)nc1 N1(CC)CCC(N=c2[nH]c3cc(C)ccc3c(=NCC3(C)CCCC3(F)F)[nH]2)C1 C1(C(=O)NCC2(NC(c3c(C)cccn3)=O)CCCCC2)NC(=O)OC1(C)C C#CC(C(C)(C)C)NC(=O)C(c1ccccc1)NC(=O)C(C)N(C)C(C)=O C(=O)(C1=NOC2(CCC2)C1)N(C)CC1CN(C(=O)CCc2ccsc2)CCO1 C12(CNC(C(N)=O)=O)CC(C1)C(NC(=O)CN1CC3C=CC1C3)CO2 C#CCCCC(C)C(=O)NCCCOCCN(C)C(C1CN(C(=O)C2CC2)C1)=O C1(CNC(c2c(C)nc[nH]2)=O)CCCCN(C(C2(c3ccccc3)CC2)=O)C1 C1(C(N2CCC(NC(C34OCC(C)(C3)C4)=O)CC2)=O)CCC2(CC1)CC2(F)F c1(C(N2CCCC(N(C(c3cnn[nH]3)=O)CC)C2)=O)c(C(F)(F)F)ncn1O N1(C(c2cc(CNC(=O)C=C(C3CC3)C3CC3)oc2)=O)CC2COCC2(C)C1 N1CCC(O)C(F)(F)C1.C(C(=O)NCC)(C(=O)CC)NC(=O)OCC Cc1cccc(C(=O)NC2CCCC2C(=O)NC(c2cnn[nH]2)C)c1O CC(=O)C(C)CC(C)C(=O)N(CCC(=O)Nc1ccc(C)cc1C)C CC(C)CC(F)(F)C(=O)NCC1CC12CN(C(=O)OC(C)(C)C)C2 c1(C(N2CCC(C)(NC(C3N(C(C)C)CCC3)=O)C2)=O)ncn2cc(Cl)ccc12 CCC(C(=O)N(CC(=O)Nc1cccc2[nH]ncc12)C(C)C)C(F)(F)F c1(C(=O)NC(C)CCNC(C2CCCN2C(N)=O)=O)ccc2[nH]c(=N)oc2c1 CN1C(=O)CSC1=CC(=O)NCC1(CO)CCN(C(=O)C(Cl)=CCl)CC1 C1(N(CCCNC(=O)OC(C)(C)C)CC)CC2(C(F)(F)F)COC1C2 c1(C(N2CC(C)(F)C2)C(=O)NCCCSC)ccc(-c2cccnc2)cc1 c1(C(=O)NCC(C2CC2)Nc2ccnc(C3CC3)n2)cc2occc2s1 S(=O)(=O)(c1cc(C(F)(F)F)ccc1Cl)NC(C)C(=O)N(C)CC1CCCCNC1 CC(CC(F)F)C(=O)N(C1CCCCC1N(C(=O)CC1(C)CCC1)C)C N1(C(CC(C)(C)OC)=O)CC(NC(c2cnc(O)cc2C(F)(F)F)=O)CC(O)C1 C1(CC)CN(C(=O)CC(C)(C)OC)CCC1NC(=O)CC1CN(C(C)C)C1 C1(CC)CCC(C(=O)NCC(C2CCCCC2)NC(=O)CC(C)c2ccco2)O1 C(C(=O)N1CCCO1)NC(=O)CC(CC1CC1)NC(C1CC2(CCO1)CC2)=O Cc1nc(N2CCC(CNC(C3(C)CC(O)CN3C)=O)CC2)cc(C(F)(F)F)n1 C1(C(N2CC(CNC(C3(COC)CC3)=O)(COC)C2)=O)CNC(=O)CC1C.C1(C)CC1 C1(CCC)(NC(=O)CCN(C(=O)CCc2cn[nH]c2)C2CC2)CCNC1=O N1(C(CCN(C(c2nccnc2C)=O)CC)=O)CC2(CCC2O)C1 N1(C(CS(=O)(=O)NC(C)(C)C)=O)CCC2C1CCCN2S(=O)(=O)c1nccs1 N1(C(COCc2ncc(C)o2)=O)CCCN(C(C2CCC3(CCC3)C2)=O)CCC1 N1(C(C(C)OCCOC)=O)CC(CCNC(C2(C(C)(F)F)CC2)=O)(OC)C1 C(=O)(C(C)C(F)(F)F)NC(CCNC(CN(CCOC)C)=O)C C1(C(=O)NCCN(C(C#CC(C)C)=O)C2CCCCC2)CCCS(=O)(=O)C1 C(CCC(N)=O)(C(=O)C(C(C(C)O)(F)F)=O)n1cc(C2SCCN(N(C)C)C2)nn1 N1(n2cc(C3(O)CN(C(Cn4nnc(C)n4)=O)C3)nn2)CCN(C)CC1C c1(OC)cccc2c1CN(C(c1ccc(Cl)cc1C(F)(F)F)=O)CC2 C1(C(N(CC(C)O)CCNC(c2nn[nH]c2Cl)=O)=O)CC(C)CC(=O)N1 CCCC(C(=O)N(C)CC1CCCCN1C(=O)Cc1cncn1C)C(C)C c1(C(=O)NC(CC)CNC(=O)CC(C2CC2)C2CC2)noc(CC)c1C c1(CC(=O)NC(CCNC(C(C)C23CC(C2)C3)=O)C(C)C)ccc(Cl)cc1 C1(NC(Cc2ccc(SC)cc2)=O)CN(C(=O)CN2CCCNC2=O)CCC1C c12ccc(O)cc1CCNC2=O.N1(CC)CCC(O)(CC)CC1 N1(C(c2cc3sccc3[nH]2)=O)CC2CN(C(c3n(C)ccn3)=O)CC12 CCCC(C#N)C(=O)N1CCCC(CCNC(=O)CCc2ccc(F)cc2Cl)C1 N1(C(CSCCCC)=O)CC=CC1CNC(=O)C(n1cc(Br)cn1)C C1(C)(C(N(CCCN(C(c2cc(OC)n[nH]2)=O)C)C)=O)CCC(=O)N1 n1(CCC)ccc(C(=O)NCC2CCN2C(=O)C(CC)NC(N)=O)n1 N1(C(CC)=O)CSCC1C(=O)N(CC(CC)NC(c1cc(C(F)(F)F)no1)=O)CC N1(C(=O)OC(C)(C)C)Cc2ccccc2C1C(=O)Nc1c(C)cc(O)nc1C C1(CNC(C(CC)(C)N(C)C)=O)(CO)CCN(C(=O)CC(=O)NC)CC1 N1(C(CNC(C(CC)CC)=O)=O)CCN(C(C2CC(=O)N(C)C2)=O)C2CCC12 N1(CC(N(CC)CC)C2CC2)CCCC(C(=O)OC(C)(C)C)CC1 BrC12CC3CC(CC1C3)C2CN1CCC1C1CCOCC1 Cc1ccc2oc(C(=O)NCC3(C)CCN(C(C45CCC(CO4)C5)=O)C3)cc2c1 C(CCN=C(NCc1csc(C(C)(C)C)n1)NC1CCS(=O)(=O)C1)=C(C)C c1(C(N(CC(C)N(C(CCSCC(C)C)=O)C)C)=O)cccc2ccsc12 CC(Cc1cnccn1)N=c1ccn2ncc(S(=O)(=O)NC3CS(=O)(=O)C3)c2[nH]1 c1(C(=O)OC)cc(Br)c(C(C)OC(c2nc(NCC(C)OC)on2)C)o1 C1(NC(CC2N(C)C(=O)CC2)=O)CC2CC1N(C(c1occc1Cl)=O)C2 C1(C(C)(C)C)CCN(c2nnc(-c3cncc(O)c3)n2C)CC1 c1(C(=O)NC2(CNC(C3C(C)(C)C3)=O)CCOC2)cc2c(o1)CCCNC2=O CCC(C)C(=O)NCC1CCN(C(=O)C(C)OCCC(C)C)C1 C1(NC(c2c(C)[nH]cc2)=O)CN(C(c2c(C(C)C)cnn2C)=O)C2CCCCC12 C(C(C(C)C(C)C)NC(c1cnnc(C2CC2)c1)=O)NC(Cc1ccc(C)s1)=O N1(C(C(CC)CNC(=O)C(C)CC2CCC2)=O)CCC2C(C(N)=O)C2C1 N1(C(CC2CCCN(C)C2)=O)CC2(C1)CN(C(c1nocc1C1CC1)=O)C2 c1(OCC)ncccc1C(=O)NCCC1CCC1NC(=O)CCC(=O)N(C)C.OCC C1(O)(C(C)NC(C2CCC(=O)O2)=O)CCN(C(c2csc3nccn23)=O)CC1 C1(NC(c2c(CC)n(CC)nc2)=O)C(C)CCN(C(=O)C(C)c2ccsc2)C1C c1(N2CCCC(C)(NC(C(C(C)(C)C)O)=O)C2)c(F)cccc1[N+](=O)[O-] N1(C(C2(OCC)CC2)=O)CCC(O)C(N(C(=O)CCC(C)CN(C)C)C)C1 N1(C(C(N2CCOCC2)=O)=O)CC2CC1CN2CCC(=O)O N1(C(C(C2CCN(C)CC2)(F)F)=O)CC2CC1CCC2NC(c1csc(S)n1)=O C1(C(=O)NCc2nn(C)c(=O)o2)CC(N=[N+]=[N-])CN1C(=O)COCCCF c1(C(=O)OCC)n[nH]c(=NC2CC(NC(=O)Cc3ccc(C)cc3)C2)s1 C1(NC(C(C2N(C(=O)OC(C)(C)C)CCC2)O)=O)(CO)Cc2ccc(Cl)cc2C1 c1(NC(C(N2CCC(C(CC)CC)CC2)c2nscc2Br)=O)ccc(C)c(C#N)c1 N1(C(C(C)OC)=O)CC2CCN(C(c3c(C(F)(F)F)nn(C)c3C)=O)CC2C1 N1(C(C(C(C)C)O)=O)CC(F)(F)CC1CNC(c1c(Cl)ccnc1F)=O c1(C2CCN(N(c3cc(C)no3)C)CC2)cc(OC)cc(OC)c1Cl.CC C1CCC(C)NC(COC(C)C(F)F)C(=O)N1.C(=O)(OC)OC c1(CN2CCCCC(NC(C3CCc4nn[nH]c4C3)=O)C2)ccc2[nH]ccc2n1 N1(C(C(CC)COC)=O)C2CCC1CC(O)(CNC(c1cn(C)nc1CC)=O)C2 C1(NC(=O)CNC(c2ccc(F)cc2)=O)C=CCCN1C(=O)C(O)CN1CCCC1 C1(NC(c2c(OC)cccc2)=O)CCN(C(=O)Cc2ccc(Br)nc2)CC1(C)C C1(C(NOCC=C)=O)C(CC)CCCN1C(=O)CC1CCCC1 C(=O)(CC(C(F)F)NC(=O)CCC1CC1C)N(CCC#C)CCOC N1(C(C2CCC(C)(CC)O2)=O)CCN(C(C2CN3CCC2CC3)=O)CC1CCO N1(C(Cc2cc(C)n(C)n2)=O)CCCC2C1CCCN2C(=O)CSCCC#N N1(C(C(OCC)OC)=O)CC2(C(=O)N(CCCCOC)C)CC1CO2 C1(C)(CNC(c2ccc(C)o2)=O)CCC(NC(c2csc(-c3ccco3)n2)=O)C1 C12(C(N(CCN(C(=O)CC3Cc4ccccc4O3)C)C)=O)CCOC1CCOC2 C(=O)(C(C(=O)N(C(C)C(=O)N(CCC(F)(F)F)CCO)CC)OC)OC c1(C(=O)NC(CC(=O)N(C)CC2CC(F)C2)(C)C)cnc2[nH]cncc1-2 C1(C(N(CCOCCN(C(c2cc(CC)[nH]n2)=O)C)C)=O)CCCC2(CC2)C1 N1(C(C2N(CC)CCC2)=O)CC2CCCC(C1)N2C(=O)COC(C)=O Cc1nnccc1C(=O)NC(CNC(C1(CC(C)C)CCC1)=O)C(C)C C(C(=O)N1CCN(CCCNC(C2CCC=CCC2)=O)CC1)(C(C)C)NC(C)=O c1(C(=O)NCC2N(C(C(CC)OC)=O)CCC2(C)C)ccc(S(N)(=O)=O)nc1 C1(C(N(CCNC(c2c(O)cc(O)cc2O)=O)C2CC2)=O)CCCCC(F)(F)C1 c1(C(N2CC(NC(c3cc(C(C)C)[nH]n3)=O)C(O)C2)=O)ncnc2c1CCCC2 N1(C(CC2C(=O)NC(=O)N2)=O)CCN(C(=O)Cc2ccns2)C2(CCC2)C1 Cc1cccc(-c2cn(Cc3csc(C)c3)nn2)n1 c1(C(=O)OC)ccc(=NCCc2ncco2)[nH]c1NC(c1cccc(C(C)=O)c1)=O c1(C(C(=O)NC(C)C(CO)NC(=O)CC2CN(C)C2)(C)C)cc(F)cc(C#N)c1 C1(NC(C(CC=CC)C)=O)CCOC2(CCN(C(=O)COCC(=O)NC)CC2)C1 C=CC(C)(O)CC(=O)NC1CN(C(c2ccc(C)c(N)c2)=O)CC1C c1(C(=O)NC2CCOC(c3ccccc3)C2)ccc2c(c1)C1CCCC2N1 C1(NC(C2C(C=C)C2)=O)CN(C(=O)CCc2ccnc(OC(C)=O)c2)CC1F C1(C(=O)NC(C(C)C)CNC(c2ccccc2F)=O)CC2CCC(C1)O2 C(C(C(C)C(C)C)NC(c1c(Cl)nsc1Cl)=O)NC(Cc1ccc(C)cc1)=O C(=O)(CC(C)CCCCCC)N1C(CCNC(C=CCCC)=O)CC(OC)C1 C1(NC(C(C)n2cccn2)=O)CC1C1CCCN(C(=O)C2=CCCOCC2)C1 C(=O)(C1=NNC(=O)C1)N1CCCC(CNC(C(c2ccc(C)cc2)C)=O)C1 C1(O)(C(N2CCCC(O)(CNC(c3cc(OC)n[nH]3)=O)C2)=O)CCC(C)(C)CC1 Cc1nc2[nH]n(C)c(=O)c2c(C)c1CCOC(=O)COC(F)F C1(CC(=O)NCCCN(C(c2c(C)nc(C3CC3)[nH]2)=O)C)CN2CCN1CC2 Cc1coc(C2CC2)c1C(=O)NCC1CCCN1C(=O)CC1CCCO1 N=C1NC(=O)C(CC(=O)NCC2(NC(=O)Cn3cnc(C(F)(F)F)n3)CC2)S1 N1(C(c2c(CC)nn[nH]2)=O)CCC2CCC(C1)N2C(C1CCCN(C(C)C)C1)=O c1(CNC(C(=O)N(C)C(c2ccccc2)c2ccccc2)=O)cscc1Cl c1(C(N2CC(CCO)(NC(c3ccc(CC)cn3)=O)C2)=O)ccc2cncn2c1 C(=O)(C(C1=CCC(CC)CC1)c1nnnn1C1CC(F)(F)C1)NC1(C)CC1 c1(N2CCCC(NC(C(=O)NC)=O)C2C)ncnc2c1ncn2CCC(C)(C)CO c1(N2CCC(CC=C)(NC(C3CC4C=CC3C4)=O)C2)cnc2ccccc2n1 Cc1ccc(S(=O)(=O)N2CCC3(CC(NC(=O)C(C)CBr)C3)C2)cc1Br C1(C(=O)NC2CC(NC(c3c(N)cccc3Cl)=O)C2)CCc2nnc(O)n2C1 C(=O)(C(F)S(=O)(=O)c1ccccc1Br)N1CC(C)(C)OC(C)(C(F)(F)F)C1 C1(NC(C(CC=C)CC=C)=O)CC1C1CCCN(C(c2occc2C)=O)C1 S(=O)(=O)(c1cnc(NC2CCC(=O)NC2C)cc1C)NC(CCC)CCC C1(N(C(COCCOCC)=O)C)CCN(C(c2ccn(C3CCOCC3)n2)=O)C1 C1(CNC(c2cc3c(s2)CCC3)=O)CCN(C(=O)Cc2cncnc2)C12CCC2 C(=O)(C#CC1CCCC1)NCCOC1CCN(C(Cc2n(C)c(S)nn2)=O)C1 Cc1cccc(C(N2CC(C(=O)Nc3ccn(C)n3)C(F)C2)=O)n1 c1(C(N2CC(NC(c3c(C)nccn3)=O)C(C)CC2)=O)cccn2[nH]c(=N)nc12 Cc1ccc(CNC(=O)CCCCCNC(c2ccnn2CCN(C)C)=O)cc1O C1(NC(C(CSC)C)=O)CCN(C(c2ccc(CC#N)cc2F)=O)C12CC2 C1(CC=C)(NC(c2cccc(C3(C#N)CC3)c2)=O)CCN(C(=O)C=C(Cl)Cl)C1 C1(C(=O)NCC(C(C)C)NC(C2(C(C)(C)C)CCCC2)=O)CC(=O)N(C)C(=O)N1 c1(C(=O)NCC2(OC)CCOC2)ccnc(CNC(C2CCC(CO)CC2)=O)c1 C1(C(=O)Nc2n(C)nnc2)CC2(CC2)CN1C(c1cc(C(C)C)ccc1O)=O CC1=CCC(C)(C(N2CCCC(F)(CNC(c3cc(C)cnc3C)=O)C2)=O)CC1 C1(CNC(c2cscc2F)=O)CC2(CC2)CN1C(=O)Cn1cccn1 C1(CCNC(C2(CSC)CCC2)=O)CN(C(=O)CCC2CC2(C)C)CCO1 C1(NC(COC2(C#C)COC2)=O)CC2CC1N(C(=O)CC=C)C2 N1(Cc2cnc(C)s2)CCC(C2CCCN(C(c3cnc(C(C)C)nc3O)=O)C2)C1 N1(C(CSCCC(C)C)=O)CCN(C(=O)CCN2CCC2)C(C(F)F)C1 C(=O)(CCP(C)(C)=O)N1CC(C(C)NC(C(CCC)OCC)=O)OCC1 C#Cc1cncc(C(=O)NC2(C)CN(C(c3sc(C(C)OC)nc3C)=O)C2)c1 Cc1nn(C)c(=O)c(C(N2CCC(CNC(C3CCC4CC34)=O)C(C)C2)=O)c1C C1(C(N2C(C(=O)NC(CC=C)C3CC3)C=CC2)=O)CCC=CCCC1 CC1CCCC(C(=O)NCC23CC(CN2C(=O)C(C2(O)CCCC2)F)C3)CC1 N1(C(=O)Nc2ccc(OC)cc2)CCN(C(C2CCC(=O)N2C)=O)C(C)C1 c1(C(=O)NCCN(C(C2CCCCC2C)=O)CC)cnc2n1CCC2 C12(C(=O)NCC3CCN(CCc4cccc(C)c4)C3)CCC(C)(C(=O)O1)C2(C)C CC1(C(N2CC(C3(NC(c4ccc(N)c(F)n4)=O)CC3)C2)=O)CCCCNC1=O c1(C(N2C(C)(C)COC(C(=O)O)C2)=O)cnc2ccc(F)cc2c1 N1(C(c2c(OC)ccnc2)=O)CC(CNC(c2cccc(OC)n2)=O)CC(C)C1 CCC(C)(CC)C(=O)NC1CCC1NC(C1CC1c1ccccc1)=O C1(NC(=O)NC2(NC(=O)OC(C)(C)C)CC(O)C2)CCCCN1C c1(C(C(C)(C)C)NCC(c2cccnc2)(C)O)cccc(Cl)c1 N1(C(C2(OC)CCOC2)=O)CCN(C(C2(n3cc(Cl)cn3)CC2)=O)C2(CCC2)C1 C1(CC(N)=O)(NC(CCC#C)=O)CCCN(C(c2ccnc(SC)c2)=O)C1 C(CC(C(=O)NCCCC1CCCN1C(=O)Cn1cncn1)OC)OC C1(NC(c2cc(CC)c(C)s2)=O)CN(C(=O)C(C)CC(C)(C)C)CCC12CCC2 C1(CCNC(CC=C)=O)CN(C(=O)Cc2cc(C)ccc2C(C)=O)CCCO1 CC1(C#CC(=O)NC2(C3CN(C(=O)C(c4ccccc4)F)C3)CC2)CC1 c1(C(=O)NCCN(CCC)C(C23CCCC2(C(N)=O)C3)=O)ccc([N+](=O)[O-])cc1 c1(C2(C(N3CC(NC(C4(F)CCCC4)=O)C3)=O)CC2)ccc([N+](=O)[O-])cc1 C(=O)(C(C)CC(F)(F)F)NC1CC(CCNC(c2cc(CC)ncn2)=O)C1 c1(C(N2CC(C(=O)NC(CCCC)CO)OCC2)=O)ccc(F)nc1C c1(CNCC2(C)CCCC2)ncccc1S(=O)(=O)NC1CC(C)(C)OC1 C(CCNC(c1ccc(F)n1C)=O)(C(=O)NC(C(C)(C)O)C1CC1)OC C1(CC)CC(C)CN(C(C2COCCC2NC(=O)C(C)OCCC(C)C)=O)C1 c1(-c2n(CC=C)c(N3CCOC4CC34)nn2)ncc(S(C)(=O)=O)cn1 c1(C(C)C)cc(C(=O)NC2CC(C)(NC(=O)COCC(F)(F)F)C2)cc(O)n1 N1(C(C(CCOC)C)=O)CCC(CNC(c2ccsc2C)=O)C(O)C1 C1(C(N2CC(=CC)C2)=O)CCC2CCC1N2C(C1SCCS1)=O N1(C(c2ccc(C#C)nc2)=O)CC2CCN(C(C3CC3F)=O)C2C1 C=CCCCC(C(=O)NC)NC(=O)CCC(C)(C)NCc1noc(CCC)n1 c1(C(=O)NC(CC)(CNC(=O)Cc2c[nH]nc2O)CC)cc2ccncc2[nH]1 C1(C2CC2)(OC)CN(C(C2(C)CCCN2C(c2ccoc2)=O)=O)C1 N1(C(C(CC)n2ccnc2)=O)CCN(C2CCCN(C(C3(SC)CCCC3)=O)C2)CC1 N1(C(C(C)C)C)CCCC(C(N2CCCC(c3cccc(C(=O)O)c3)C2)=O)CC1 N1(CC(=O)NC(CCCNC(C2ON=C(CC)C2)=O)C)C(=O)CC(C)(C)C1=O n1(CC(=O)NC(C2CC(NC(C(C)=C3CC3)=O)C2)C)cnnc1O C(=O)(C1=NN(CCO)C(=O)CC1)C(=O)C1=CCCOC1.C1(N)CC2(C1)CC(C)C2 c1(OC)cc(C(N2CC(CNC(=O)Cc3ccc(Cl)c(Cl)c3)C2)=O)cc(C)n1 C=C(C)CC(=O)NCCOCCNC(CCCc1nc(C)no1)=O c1(C(N(C2CCC(NC(c3cc(C)[nH]n3)=O)C2)C)=O)sc2ccc(F)cc2c1C C1(NC(c2nc(C)sc2)=O)CCN(C(=O)CC2CCCC(C)(C)C2)CC1F N1(C(c2n[nH]c(C3CC3)n2)C(=O)NC)C2CCC1c1ccccc12 N1(CC)CCN(C(c2nccc3ncncc23)=O)c2ccccc2C1 C1(CNC(c2nc(C)[nH]n2)=O)CCC2(CN(C(C3CCCS3(=O)=O)=O)C2)O1 C(=O)(CC(C)C(C)C)N1CCC(OC)(CNC(c2cccc(Cl)c2)=O)C1 C(c1c(Cl)cccc1Cl)=CC(=O)NCCC1(O)CN(C(Cc2ncc(C)o2)=O)C1 c1(C(=O)NC2(C3CCCN3C(=O)CCNn3cncn3)CC2)ccccn1 c1(C(=O)NC(C2N(C(c3cnc(C(C)C)[nH]3)=O)CCC2)C)nn(C)cc1[N+](=O)[O-] C12(C(=O)NCC(C(C)C)(C)C)COCC(c3ccc(Br)cc3)(C1)C2 CC1CCCC1(C)C(=O)NCCC1CCCN1C(c1cc(=O)n(C)o1)=O C1(CC(N2CCCC(C3N(C(C(N)=O)=O)CCCC3)C2)=O)CCC2(CCC2)CO1 c1(C(=O)NCC(C)(CO)NC(=O)C=Cc2ccco2)ccc(C#N)cn1 C1(CNC(C(C)(C2CC2)OC)=O)CCC(C)CN1C(=O)CCc1ccoc1 CC1(NC(C2CN(c3cccs3)C2)=O)CCC(NC(=O)CCCN2CCCC2)CC1 C1(c2cn(CCN3CCOCC3)nn2)(NC(c2cc(C)[nH]n2)=O)CCCOC1 c1(CC2NC(=O)N(CCc3cccc(OC)c3)C2=O)cc2c(s1)CCOC2 Cc1nc(=N)[nH]cc1C(=O)NC(C1CCCC1)CNC(=O)C1=CCCSC1 c1(C(N(C(CNC(C(CCSC)OC)=O)C)C)=O)ccc(C(=O)OC)cc1C#N C1(C(=O)NCc2cccc(C)c2)(NC(CCCNC(C)=O)=O)CCCC1C N1(C(C2C(NC(c3cc(C)sc3C)=O)CCC2)=O)CC2CC(C)C2C1 c1(C2C(NC(N3CCCC(CN(C)C)C3)=O)CCCO2)ccc2ccoc2c1 c1(CC(N2CCC(N(C(CC(=C=C)C)=O)C)CC2)=O)ccc(CNC=O)c(C)c1.C(C)=C C1(NC(C2C(C=C)CC2)=O)CCC(N(C)C(c2ccc(C(C)C)nc2)=O)CC1 C12CN(CC13CCC3)C2=O.C12(CNC(C3N(C)CCCC3)=O)CCC(CC1)OC2 C(C(C)(CC(C)C)NC(c1cc(OC)ncn1)=O)NC(C(CC=C)OC)=O C1(C(=O)NCC2(CC)CCCO2)CC(C)(C)CCN1C(c1cccc(F)c1N)=O Cc1ccccc1C=CC(=O)NCCC(C)N(C)C(C1CC(C)(F)C1)=O c1(C(=O)NC2CCC(CNC(C3(C=C)CCOCC3)=O)C2)cnn2c1NCCC2 c1(NC(C2CCCN(Cc3cccc(Cl)n3)C2)=O)ccc2oc(O)nc2c1 N1(C(c2cc(C)oc2C)=O)CC2(CC2)CC1C(=O)NC12CC1COC2(C)C c1(C(N(CCC)CCNC(C2CC2CF)=O)=O)cccc2nc(C(F)(F)F)sc12 C12(C(=O)NC3CCN(CCC)C3)COCC1CN(C(=O)Cc1nocc1C)C2 N1(C(CC(=C=C)C)=O)CC2CCCC2(NC(c2cccc(Cl)c2Br)=O)C1 c1(OC)c(C(N2CCC(C)(CCNC(c3ccc(=N)[nH]c3)=O)C2)=O)c(C)nn1C c1(C(N(C(C)CCNC(c2cn(C(C)(C)C)cn2)=O)C)=O)cccc(CF)c1 c1(OCC)ccc(C(N)CC(=O)NC(C)CN2CCOCC2)cc1 C(=O)(C(F)C(F)(F)F)NC(CC1CN(C(c2c(SCCC)cccc2)=O)CC1)C N1(C(Cn2c(C)ncc2)=O)CC2CCN(S(=O)(=O)C(F)(F)F)CC2C1 C1(NC(CS(=O)(=O)NC)=O)CCCN(C(c2cn3ccsc3n2)=O)C1C Cc1cc(Oc2cnc(=NCc3ccccc3)[nH]c2)cc(C)c1O C1(C(NCC2CCCN2C(=O)Cc2sc(SC)nc2C)=O)CCN(C)S1(=O)=O.CC S(=O)(=O)(c1ccc([N+](=O)[O-])cc1)N.C1(OC)CC(c2ccc(Cl)cc2)N(CCC#N)C1 C(C1SCCc2ccccc21)NC(N(c1ccc(F)c(F)c1)CC(C)C)=O C(C(CC(C)C)C(=O)NCc1csc(N(C)C)c1)NC(C1CCN(CC)CC1)=O c1(C(=O)NCC(CN(C(c2c(C)c(C(F)(F)F)n[nH]2)=O)C)O)ccc(Cl)nc1O c1(C(N2CCCCC(NC(c3c(C)noc3C)=O)C2)=O)cc2n(n1)C(C)CCC2 c1(NC(C2C(C(=O)NC(C(=O)OC)OC)C2)=O)sccc1S(N)(=O)=O C(C1c2ccsc2CCN1C(=O)C(O)Cn1cncn1)NC(c1cc(O)cs1)=O c1(C(=O)NC2CN(C(c3c(C)n[nH]c3)=O)CC(O)C2)[nH]c2ccccc2c1Cl c1(C(=O)NC(C)Cc2nc[nH]n2)ccc(CNC(c2ccc[nH]2)=O)nc1 Cc1c(C(=O)NC(C)CN(C(=O)C(F)F)C2CC2)cnn1C1CCCC1 CC(CNC(c1snc(Cl)c1Cl)=O)CN=c1[nH]c2cc(F)cc(F)c2o1 C(CC(C)C(=O)NCCCC(C)(C)NC(=O)C(C)NC=O)OC c1(CC(N2CC3CN(C(c4n(CC)ncc4)=O)C3C2)=O)ccc2ccccc2c1 Cc1cnc(Cl)c(S(=O)(=O)N2CCC(C3(C(=O)N=c4[nH]oc(C)c4C)CC3)CC2)c1 c1(NCC(=O)NCCOCC)c(C(=O)O)nc(O)c2ccccc12 Cc1cccn2cc(C(N3CCCN(C(=O)Cc4csc(=N)[nH]4)CC3C)=O)nc12 C1(C(N(CC(=O)NC(C)Cc2cn[nH]c2)CC#C)=O)CCC(=O)NC1 C(Cc1ccc(Cl)cc1)(CCC(F)(F)F)NC(C(C)NC(C)=O)=O C1(C)(C(C)C)CCC(NC(=O)OC(C)(C)C)C1.C1CCC(=O)O1 C1(N(C(=O)COC)C(c2ccc(OCCC)cc2)C)C(C)OCC12CCNCC2 N1(CCC(C)C)CC2(CCN(C(C3(C)CC3(F)Cl)=O)CC2)CNC1=O C1(COC)CC(CNC(=O)CCC2CCCN2C)N(C(c2ccc(C#N)o2)=O)C1 C1(CC)CN(C(c2c(C)nn(C(C)C)c2C)=O)CCC1NC(=O)C(C)(C)C c1(C(=O)NCC2N(C(CC=C)=O)CC(F)(F)C2)cc2c(nc1O)CCC(CC)C2 C(=O)(CCC(CC)NC(=O)CCc1cncc(O)c1)NC1(COC)CC=CC1 c1(NC(C(COC)OC)=O)cccc(C(=O)NCCN(C)C)c1 c1(C(=O)NC2(CF)CCN(C(c3c(C)ccn3C)=O)C2)n[nH]c2c1CC(C)CC2 Cc1cc(C(N2CCC(CO)(CNC(C3(O)CCOC3)=O)CC2)=O)cc(C)n1 C1(CNC(C(CCN(C)C)O)=O)CN(C(c2ccc(C3CC3)s2)=O)CC(C)(C)C1 Cc1sc(C(N2CCC(C)(NC(=O)C(CC#N)c3ccccc3)C2)=O)nc1O CCC(C)(O)C(=O)NOCC(=O)NCCc1ccc(C)c(C)c1 C(=O)(C(O)CC[S+](C)C)NC(C1(O)CCN(C(C=CCCC)=O)CC1)C CC1CCN(C(C2(CC3CC3)CC2)=O)CC1CNC(C1(F)CCC1)=O C1(CC)CN(C(C2(C)C(C)(C)C2(C)C)=O)CCC1CNC(C1(C)CC=CCC1)=O C(=O)(C(C)(O)C(F)(F)F)N1CC(OC)C(NC(c2ccc(P(C)(C)=O)o2)=O)C1 N1(C(C=Cc2c(C)coc2C)=O)CC(NC(=O)CCC2CCCO2)CC(F)(F)C1 N1(C(c2c(C)nc(O)s2)=O)CCC2(CC(C(N3CCC(CO)C(C)C3)=O)C2)C1 c1(C(=O)NCCCCNC(CC(C=C)CC)=O)cc(N)c(Br)c(F)c1 C1(NC(C2(C)CCCN(C(C3CCC(C(N)=O)C3)=O)C2)=O)CCCCCCC1O C=CCC(C(=O)NC1CN(C(c2ncncc2Br)=O)CC1O)C(C)C c1(C(N(C(C)CNC(=O)CCCc2cncs2)C)=O)cc2ncccn2n1 CC1CC=C(C(=O)NCC(O)CCNC(c2cccc(Cl)c2N)=O)CC1 C(C(C)(O)CC(=O)NCCCCN(C(=O)C=C(C)CN1CCOCC1)C)OC c1(C(N(CCOCCN(C)C(c2nc(Cl)cs2)=O)C)=O)cnn2c1OCC(F)C2 C1(C2CC2)(CNC(c2cnc(F)c(Cl)c2)=O)CCN(C(C2CCCOC2)=O)C1 c1(C(=O)NCCCC(C)NC(c2cc(O)ccc2Cl)=O)ccc(Cl)cc1O N1(C(c2cncc(N3CCC(C)CC3)c2)=O)CC2CC1CN(C(=O)C1=CCC1)C2 N1(C(C(C)C2CCC2)=O)CCC(CNC(C2CC2C(F)F)=O)C12CCC2 S(=O)(=O)(c1cccnc1NCc1ccc2nn[nH]c2c1)NC(C=C)C1CC1 CCCC(C(=O)NCCC1CCCN(Cc2cn(CC(C)C)nn2)C1)C(C)C c1(OC)ccc(C(C)Nc2nc(-c3cncs3)n[nH]2)cc1[N+](=O)[O-] c1(N2CCC(NC(c3ccc(OCC)cc3)=O)C2)ncnc2c1oc1ccccc21 c1(COC)ccccc1C(=O)NC(C(=O)N(C)Cc1csc(C)n1)C1CC1 C(=O)(C1CCC(=O)c2ccccc21)N1C(CNC(=O)CSCC(F)(F)F)CCC1 c1(OC)cnnc(C(=O)NC(C)CC2CN(C(C3CC(C)N(C)C3)=O)C2)c1 C(=O)(C1=CC2CCCCCCC12)N1CCN(C(c2ncc(CC)nc2)=O)C(C)C1 C1(CNC(c2ccc([N+](=O)[O-])[nH]2)=O)CN(C(c2cc[nH]c2)=O)CCC12CCOC2 C(=O)(C1CS(=O)(=O)c2ccccc21)NCC(C)CNC(c1cc(Cl)ncc1O)=O N1(C(C(CCCOC)C)=O)CCC(C2CC2)C1CNC(=O)Cc1cccs1 c1(CC(=O)NCC)ccc(C(N)=O)cc1.C1(N2CC=CC2)CCC(OC)CC1 c1(N2C(C)CC(C(=O)Nc3cnc4n3CCOC4)C2)cc(Cl)nc(S(C)(=O)=O)n1 N#CC1(C2CC2)CCN(CC(=O)Nc2ccccc2N2CCOC2=O)C1 C(C(C)(C)C(=O)N1CC(NC(=O)C(c2ccccn2)O)C(C)C1)NC(C)=O C(=O)(C(CC(C)C)CC(C)C)N1CCCC(CN(C(C2(SC)CCC2)=O)C)C1 c1(SC)ccccc1CC(=O)N(C1CN(C(C2OCCC2(C)C)=O)CC1F)C N1(C(c2ccc(O)cc2)=O)CCC(NC(C2(n3ccnn3)CC2)=O)C(O)C1 N1(C(CCC(=O)NCCCOC)=O)CC2CC(C1)CN(C(C1CCN(C)C1)=O)C2 N1(C(c2cc(OC)ncc2)=O)CCC(C2CCN(C(=O)C=NOC)CC2)C1 CC1CCCN(C(=O)Cc2nc(=N)[nH][nH]2)C1CNC(=O)Cn1ccc([N+](=O)[O-])n1 N1(C(c2c(C)scn2)=O)Cc2c([nH][nH]c2=NC(=O)c2cncc(F)c2)C1(C)C CCC(C#N)C(=O)N1CC(NC(c2ccc(-c3ncc[nH]3)nc2)=O)C(O)C1 c1(C(F)(F)F)ccc(F)c(Cl)c1.CC1CNC(=O)C2CC2CN1 CCCCC(O)C(C)C(=O)N1CCC(C)(C)C1CC(N1CCC(CCCO)C1)=O c1(C(=O)NCCC2N(C(CCCC#CC)=O)CCC2)[nH]cc2c(=O)n(C)ccc12 c1(C(=O)NC(C)C(C)(C)NC(=O)CNC(=O)CN(C)C)ccnc2ccnn12 C#Cc1cccc(C(N2CC(F)(CNC(c3cc4n(c3)CCCC4)=O)C2)=O)c1Cl c1(C(=O)NC(CCOC)CNC(=O)CC(C)CN(C)C)cc2ccccc2cc1O N1(C(C2N(CC)C(=O)CC2)=O)CCC(C2CC2)(NC(=O)CCNC(=O)C=CCl)C1 CCC(O)C(F)(F)C(=O)N1CCC(CN(C(=O)Cc2cnccn2)C)C1 c1(COC(C(C(C)C)OC)=O)c(C(F)F)cccc1F C1(NC(CCCCSC)=O)CC2(C1)CN(C(=O)C(C)Sc1nnnn1C1CC1)C2 Cc1nn(C)c(C)c1CCC(=O)NCC(O)CCNC(C1(N(C)C)CC1)=O c1(C(N2CCC(N(C3CC(SC)C3)CCNCC)CC2)=O)cc(C)nc(C(F)(F)F)n1 c1(C(C)NCC(=O)OCCc2c(C#C)cccc2)cc(Br)cc(Br)c1O c1(C(N(C)Cc2ccc(CNC(C3CC34CC4)=O)cc2)=O)cc(O)cnc1Cl N1(Cc2ccc(C(=O)OC)[nH]2)CCN(CCC(=O)N(C)CC2CCC2)CC1 CCC(C)C(=O)NCCC(=O)N(CCN(C(=O)C(C1CC1)OC)C)C C(C(C)(C)C)(C(F)(F)F)NC(N(C)CC1(CC2CC2)CCC1)=O C1(C(=O)N)CCC(OC)C1.CCC(CC)=CC(=O)NCCNCC#C C(=O)(CCC(CF)CF)NC1(C)CC(C(=O)NC2CCCC(N(C)C)C2)C1 CN1CCOC(C(=O)NCc2ccnc(C(=O)NCC(C)(C)N(C)C)c2)C1 CCC(C(=O)N(CCOC)C1CC1)C(C)C.c1(CC=O)ccccc1 c1(C(=O)NC2C(NC(=O)Cc3cnccn3)CC2)c[nH]c(=O)c2ccnn12 CCC(C(=O)NC1COCC1C(=O)NCC1CCCC12CC2)C(C)C c1(OC)ccc(Cl)c(C(N2CCC3CC2CN3C(=O)COC(F)(F)F)=O)c1F N1(C(C(c2c(OC)cccc2)=O)=O)CCCC(N=c2cnc3ccccc3[nH]2)C1 CCCCC(C)(F)C(=O)NC1CCN(C(c2cc(C#N)c[nH]2)=O)CC1 c1(OC)cnc(N2CCC(C(=O)OC(C)(C)C)CC2)nc1.N1(C(C)=O)CCC(O)CC1 CC1CC(NC(C2(C3CCC3)CC2)=O)CN(C(=O)CSc2nncn2C(C)C)C1 N1(C(C2(C)CC(=O)C2)=O)CC2(CC(C(=O)NCc3ccc(O)nn3)CO2)C1 C1(CC(NOCC(C)(C)C)=O)CCCN(C(C2CCCSC2)=O)C1 C12CC3CC3N1C2=O.c1(C(C)NC(=O)CCCN(C)C)ccccc1F c1(C(=O)NCC2CC(CCn3cc(-c4ccncc4)nn3)C2)cccc(CCF)c1 CC1CCC(CO)N(C(=O)C(Cc2cc(Br)no2)COC(C(C)(C)C)=O)C1 N1(C(Cn2c(C)nnn2)=O)CCC(CC(=O)NC2C=CCCC2)C1(C)C N1(C(C(=O)NCCCC)=O)CCNC(=O)C1.C1(C(C)C)COC1=O C1(C(N2CCCC(C(=O)NC(COC)(C)C)C2)=O)CCC2C=CCC1O2 C1(NC(C(C)N(C(C)=O)C)=O)CCOCC1NC(c1cnon1)=O c1(CN(C)CC2CCCN(C(=O)C3=NNC(=O)CC3)CC2)cnc2[nH]ccc2c1 C(=O)(C(COC(C)C)NC(=O)Cc1cnc(C)[nH]1)N(CC#C)C(C)C c1(C(=O)Nc2cc(CO)cc(OC)n2)ccc2c(c1)CCN2.C1(C)CN1 c1(NC(=O)NCc2ccsc2)ncc(C(=O)NCC(CO)C2CC2)s1 CC1(C)COC(C(=O)NCC2C=CCN2C(C2CC(=O)CCO2)=O)CO1 c1(OC)ccc2c(c1)C1=NC(=NC(C)C(c3ccco3)N1)N2.C(CN(C)C)SC C(=O)(C(F)C(C)(F)F)N(CC(C)N(C(C(N1CCOC1=O)C)=O)C)C CC(CC1CC1)C(=O)N1CCCC1C(C)NC(=O)Cn1cnc(CCN(C)C)n1 c1(C(=O)NC2(COC)CN(C(C3(C)CC3F)=O)C2)[nH]c2ccc(F)cc2c1C c1(NC(CC(C)C)=O)cccc(NCC(=O)NC2CCCN2C(=O)C2CC2)c1 C1(OC)(OC)CCS(=O)(=O)CC1NC(N1CCC(F)(N(C)C)CC1)=O c1(Nc2cnc(OC)nc2)c(C)cccc1[N+](=O)[O-].n12c(COC)nnc1CCC2 C1(CN(CCCN2CCCC2=O)C)CCC2(CCC2)CO1 c1(C(=O)NC(C)(CNC(=O)C2CC2)C2CC2)cnc(O)cc1C(F)(F)F C(=O)(C(O)C(C)(C)C)NCC(C)(C1CCC1)NC(c1cc(COC)on1)=O C(=O)(CC1=CCCC1)N1C(C(C)(C)NC(c2csc(CO)n2)=O)CCC1 C(C(=O)N1CC(O)CO1)SCC(=O)NCCCC1CC=CC1 C(=O)(CN=c1cc(NCC(C)CCC(C)(C)C)nc[nH]1)N1CC(SC)C1 C(=O)(CCCCC(=O)Nc1c[nH]nc1C(=O)NCCc1ccncc1)OC C1(C(=O)NC(CN(C(COC(CC)C)=O)C)(CO)CO)CN2CCCN1CC2 C(=O)(CCCC(F)(F)F)NC1CCC(CC(=O)Nc2ccc(C)c(CO)c2)C1 C(C(C)CC=O)OCCOC(C)=O.C1(C(C=O)OC)COCC1C(F)(F)F Cn1ncc(C(=O)NC2COCC2Cn2cncn2)c1C(N)=O CC1(Nc2cccc(NC(C34CCC(C(=O)O)C3C4)=O)c2)CCN(C(N)=O)CC1 C(=O)(C=C1SCC(=O)N1C)NC1CCC(CCNC(C(C)CC2CCCC2)=O)C1 O=C(C(O)C(F)(F)c1ccccc1)OC1CNC1=O C1(COC)(CNC(=NCC2CC2)NCC(Cl)C(F)(F)F)CC12CCC2 c1(C(C)NC(=O)CONC(C2CCC(=O)N2)=O)ccc(F)nc1 c1(CC(C(=O)NCC(CN(C(COCC(=O)NC)=O)C)(C)C)C)ccccc1C S(=O)(=O)(c1ccc(NCC2CSCCS2)cc1Br)N(CC(CC)C)C CCS(=O)(=O)c1ccc(F)c(C(=O)NC(C)(CNC(=O)C(O)P(C)(C)=O)CO)c1 c1(C(=O)NC(c2cccc(Cl)c2)CNC(C(CC)NC(N)=O)=O)cncc(C)c1 C(CCCCCNC(C12CSCC1C2)=O)NC(=O)Cc1ccc(Cl)cc1 C1(CC(=O)NCC2(COC)CN(C(c3cc(CO)[nH]n3)=O)C2)CCCCN1C c1(OC)ccc(OCC(CN(C[Si](C)(C)C)c2ccccc2)O)c(C)c1 Cc1ccc(C(=O)N(CC(=O)NCc2ccn(C)n2)C2CC2)o1 C(=O)(C1CCc2c[nH]nc21)N1CC(C2(NC(C34CCC(O)(CC3)CC4)=O)CC2)C1 Cc1cnn(C)c1CC(=O)N(C1CCCN(C(C2(C#N)CCCO2)=O)C1)C N1(C(c2cc(OC)no2)=O)CCC2CN(C(=O)C(C)Cc3ccco3)CC12 N1(C(C(CCC)C)=O)CCN(C(=O)CN2CCC(F)(F)C2)CC1c1nccn1C CC12CCC(CC(=O)NC3C4CC(NC(=O)CC=CC(C)(C)C)CC34)(CO1)C2 c1(NC(C2CN(C(C)=O)C2)=O)ccc(C)c(NC(=O)CCC2OCCO2)c1 C1(C(N2CCCC2CN(C)C(c2csc3nnsc23)=O)=O)(OC)CCCCCC1 CCCC(C(=O)NCCC1(C(=O)N(CC(C)(C)CC)C(C)C)CCC1)NC(N)=O C(CCO)(C(C)(C)C)NC(C1C(CCC)CN(C(C2CCCN(CC)C2)=O)C1)=O C#CC1CN(C(C2CCC(C)(CC)O2)=O)CCN1C(=O)CCc1cnc[nH]1 N1(C(CNC(C2C(=C)C2)=O)=O)CC(N(C(=O)Cn2cccn2)C)C1 C#CC1(NC(=O)CCN(C(C2CCC(C)(C)C2)=O)CC2CC2)CCCOC1 C1(CC)C(C(N2CC(CO)C2(C)C)=O)CCN1C(c1cc[nH]c(=N)c1)=O CCS(=O)(=O)C=CC(=O)NC1CCCC1CNC(c1cccc2sncc12)=O c1(C(=O)NC2CCN(C(CC(=C=C)C)=O)CC2O)ccc([N+](=O)[O-])cc1F n1(CC)cc(C(N2CC(CC(C)NC(C3CC3F)=O)C2)=O)c2ccccc12 c1(C(=O)NC2CCCN(C(C3(C(C)(C)C)CCCC3)=O)C2)occ2c1CCC2 CC(C(=O)NC(C(=O)NC1CNC(=O)C1(C)C)C(C)(C)O)C(C)(C)C C(=O)(C1=CC2(CCOC2)C1)NC(CNC(CC(COC)(C)C)=O)C(C)C C1(NC(Cc2c(C)scc2)=O)C2CC3C(C2)C13C(N1CC(=O)NCC1C)=O C1(NC(C2CC3(CCOC3)C2)=O)CN(C(C2CC3CC3C2)=O)Cc2nccn2C1 N1(C(c2ncc(C)o2)C(=O)NCC)CCC2C(O)CCCC2C1 C1(NC(Cc2c(OC)nccc2)=O)CCN(Cc2cc3occc3s2)CC1C C(C#C)(CNC(=O)C1CC1)NC(COCC#C)=O.C1C(=O)NCCCO1 c1(OC)ccc2c(C(=O)NCC3CCN(C(C4CCCO4)=O)CC3C)c[nH]c2c1 n1(CC(=O)N(c2ccccc2)C2CC2)cnc2sccc2c1=O.C1CC2CC12 C1(C(=O)NCC2(CNC(C3CC4C=CC3O4)=O)CC2)CCC2(CCC2)CO1 C(=O)(C1=CC(C)CC1)NC1C(OCC)CN(C(c2c(C(=O)OC)cnn2C)=O)C1 C1(C(=O)NCC(C=C)O)CCC(CNC(=O)COC2CCOCC2)CC1 c1(C(=O)NC(C)CCC(=O)NC(C)CC(C)(C)O)ccc(C)cc1 N1(C(c2c(OC)ccc(O)c2)=O)CCCN(C(C2(CCO)CC2)=O)CCC1 C(=O)(CC(C)P(C)(C)=O)NC1(CNC(C(COC(C)=O)(F)F)=O)CCOCC1 C(=O)(C(C(F)(F)C1CC1)C1(O)CCC1)N1CC(CNC(CC(C)c2ccco2)=O)C1 N1(C(C=CSC)=O)CC(C)CN(C(=O)CC2(O)CCCN(C)C2)C(C)C1 c1(OCC(=O)NCC2(COC)CN(C(=O)CCC3CCCC3)C2)ccccc1Cl Cc1noc(Cl)c1CCC(=O)NC1CCC(NC(C2CCOC2)=O)C1 C(CCC(=O)N1CCCC1C1CCOC1)NC(C1CC(OC)C1)=O N1(C(CC(C=C)(C)O)=O)CC=C(C(=O)NCC(C)(O)C(=O)OC)CC1 N1(C(C2CN(C(C(C=C)OC)=O)CC2C(C)C)=O)CC(C)OC(C)C1 C(=O)(C1CCOc2ccccc21)N1C(CNC(=O)CCc2cccc(O)n2)CC1 Cc1nc(CC(N2CC(NC(=O)CCc3cccn3C)C(C)C2)=O)[nH]c1C C(C(C)C)(C(O)C(=O)NC(N1CCC(C)C1C)=O)OC.c1cc(OC)n(C)n1 Cc1cc(=O)n(CC(=O)N(C)CCNC(=O)C(CCO)N(C)C)c2ccccc12 N1(C(CCc2cc(C)on2)=O)CCC(NC(=O)Cn2cc(C(F)F)cn2)C(F)C1 N1(C(CS(=O)(=O)NC)=O)CCC(CNC(=O)C(CC(C)C)OC)(OC)CC1 C1(N(CC=CC(=O)NC2CC2)CC)(C(N2CC(C)(OC)C2)=O)CCCO1 c1(C(C)C)ncc(C(=O)N(C2CC(NC(=O)COCCN(C)C)C2)C)[nH]1 CCC(CC1CCCCC1)C(=O)NCCC1CC(NC(=O)CSCCC#N)C1 N(C(=NCCC(C)N1CCOCC1)NC1CCc2nnnn2CC1)CCOC CCCC(C(=O)NC1CC(C)N(C(=O)C(C)c2ccsc2)C1)NC(N)=O c1(C(C)N(C(=O)C(N2CCC(N(CC(N)=O)C)CC2)=O)C)cccc(Cl)c1 C1(NC(C2(C)CC2F)=O)CC2CC(C1)CN(C(c1cc(OC(C)(C)C)ncc1)=O)C2 C(N=c1[nH]c(Cl)ncc1[N+](=O)[O-])C1(C)CCN(C(c2cnc(C3CC3)o2)=O)CC1 Cc1ncc(C(N2CC(O)(CCNC(c3nncn3C3CC3)=O)C2)=O)c(C)n1 Cc1ccccc1C(C)CC(=O)N(C)C.C12(CC1(F)F)C(=O)NC2 N1(C(c2cc(C)nc(O)n2)=O)CC(C)(C)OCC1CNC(c1c(C)csc1Cl)=O c1(C2(C(N3CCC(F)(NC(C4CNCCO4)=O)C3)=O)CC2)ccc(F)cc1Cl C(=O)(CS(=O)(=O)C(C)(C)C)NC(CNC(CC1C(C)CCO1)=O)C1CCC1 N1(C(C(C(C)NC(CCCCC=C)=O)C)=O)CCC(O)C12CCCC2 C12CCN(C1)C(=O)NC(C)CN(C)C(=O)N2.c1(C(=O)OC(C)(C)C)cnn(C)c1 c1(C(=O)NC(C(=O)NCCOC(CC)(C)C)CC2CCCC2)ncn(C)c1C C1(NC(c2nn(C)c(Br)c2)=O)CCCCN(C(c2ccc(O)cn2)=O)C1 N1(C(C(CC)C#N)=O)CC2=C(C1)CN(C(c1cnn(C(C3CCCC3)C3CC3)c1)=O)C2 c1(N2C(=O)CC(C(=O)NCCCN(C(=O)Cn3ccnn3)C)C2)cc(F)ccc1F c1(C(N(C(C)C)CC)=O)cc(Cl)n[nH]1.C=C(C)C(=O)NC(=O)OC(C)(C)C C(CC(=O)NCCOC1CN(C(C2CC2(c2ccccc2)F)=O)C1)(C(F)(F)F)OC c1(C(=O)NC2C(Cn3cc(C(C(C)C)O)nn3)CCC2)ccc([N+](=O)[O-])cc1 C1(NC(C(C)=CC)=O)CCN(C(C2CC(=O)N(CC(F)(F)F)C2)=O)CCC1CO N1(C(CN(C2CC2)CC)=O)CCC2CN(C(c3coc(S(=O)(=O)NC)c3)=O)C2C1 C1(C(=O)NCC2CC2)CC2CC2N1C(c1ns[nH]c1=O)=O C1(O)(CC=C)CCCC1NC(C1CCCN(C(=O)Nc2ccccn2)C1)=O N1(C(c2ccc(C#N)cc2)=O)CCC2CCCC12CNC(C1CC2(CC2)C1)=O C(N=c1[nH]c2c(c(=NC3CN(C4CC4)C3)[nH]1)CCCC2)c1cc(Cl)c(C)c(Cl)c1 C1(CNC(C2CCC(N(C)C)C2)=O)(NC(=O)CC2(C)CC2)CCC(C)(C)CC1 C(=O)(CCCC(=O)CC)NCc1c(C(N2CCC(C=C)(O)C2)=O)occ1 N1(C(C2(CC#C)CC2)=O)CC(NC(C2CC23CCSCC3)=O)CC(F)(F)C1 c1(C(=O)NCCCNC(=O)CSCc2ccncc2)c[nH]c2nccc(Cl)c12 CC1(C)CN(C(=O)CNC(=O)CC2(C#N)CC2)CCC1NC(=O)Cc1cccnc1 CN1CC(C(=O)NC(CC2CC2)C(=O)NCCc2ccco2)CCC1=O C(=O)(C#CC1CCC1)NCC1C(NC(C(c2c(C)n(C)nc2)O)=O)CCCC1 C(N=c1nc(C)c([N+](=O)[O-])c[nH]1)C1CCN(C(C=COCC)=O)CC1C c12ccc(cc1)CNC2=O.C1(C(=O)CN(CC)CC)CC(C)C1.c1(N)cnns1 CCC(C)C(C)CCNC(=O)CC1CCCN(C(c2cccn2C)=O)C1 C(=O)(N1CC2COCC2O1)C1CCC2CN(C(C3CC3(F)F)=O)CC21 c1(C)ccc2cc(C(=O)NC3(C)CC(NC(C=C(CC)CC)=O)C3)[nH]c2c1.C(C)(=O)O c1(C(N2CCC(C(N3CC(OC(=O)NC)C3)=O)C2C)=O)c(Cl)c(C)nn1C c1(-c2cc(C)c(F)c(C)c2)ccc(S(=O)(=O)NCCc2ccsc2)cc1C C1(C(N2CC(C)(NC(=O)C(F)CC3CC3)C2)=O)CCCC(C#N)C1 C1(NC(Cc2cn(CC)nc2)=O)CC2CC(NC(=O)Cc3csnc3C)CC12 CC1COCCC1NC(C12CC1CCN2C(c1cnco1)=O)=O CN1N=C(C(=O)NC2CCOCC2C(N2CCC(C(C)(C)C)C2)=O)CCC1=O C(=O)(C1=CCC(C)(C)CC1)NCCC1N(C(C(C(=O)OCC)C2CC2)=O)CCC1 c1(OC)cc(OC)c(C(N2CCCC(C(=O)NC(C)CC(C)C)CC2)=O)c(Br)c1 Cc1cc(N(CC(N2CC3CNC3C2)=O)C(c2cc3sccc3s2)=O)cc(C)c1 O=C(C1=CCS(=O)(=O)C1)N1CC(CNC(C2CC(F)(CO)C2)=O)C2CC12 C1(C(=O)OC(C)(C)C)CC12CN(C(=O)NCCCCCCSC)C2 Cc1nc(C(F)(F)F)cc(=NC(CNC(c2c[nH]nc2C(F)F)=O)C(C)C(C)C)[nH]1 C(CC(C(C)C)NC(=O)Cn1cnccc1=O)N(C(c1cnc(C(C)=O)s1)=O)C Cc1ccc2[nH]cc(CC(N3CCCC3(C)CNC(c3cnoc3)=O)=O)c2c1 c1(OCC=C)ccc(C(=O)NC(C)(C)C(C)NC(=O)CCCCN(C)C)cc1 c1(C(N2CC(NC(c3cccc(CC)c3)=O)C(C#N)C2)=O)ccc(Cl)c(C)c1Cl N1(C(Cc2nc(C)[nH]n2)=O)CCC(CNC(C2CC(=C3CCC3)C2)=O)C(O)C1 N1(C(C2C(C)C2)=O)CCC(N(C)C(C2(CCc3ccccc3)CC2)=O)C1 CC(C(C)(C)NC(C12CC(CC(F)F)(C1)C2)=O)NC(C1CCOC1=O)=O C1(C)(C(=O)NCc2cc(C)ncc2)CCCN(CC(=O)C2CC2c2ccccc2)C1 N1(C(Cn2ccc(C)n2)=O)CCC(C)N(C(=O)C(C)Oc2ccccc2)CC1 CC(CC(F)F)C(=O)N1CCC1C1CCCCC1.C12CC(F)(C1)CNC2=O C(=O)(CS(=O)(=O)C1CCCC1)N(C(C)CCNC(=O)CCc1ccon1)C c1(CCNC(=O)NC2CCN(c3ccccc3)C2)c(F)cc(F)cc1F c1(C(=O)NC(Cn2cc(CCCC=C)nn2)C)cc(C)sc1S(N)(=O)=O O=C1CC(=O)NC(C(N2CC=CC2C(=O)NCc2conc2C2CC2)=O)C1 c1(OC)cc(C(=O)NCC(C)NC(c2csc(C#N)c2)=O)cc(Cl)n1 C1(C(=O)NC(CNC(C(C)N(CC(F)(F)F)S(C)(=O)=O)=O)(C)C)CC2(CCC2)CO1 c1(CC)oc(C(=O)NC(c2ccccc2-n2cccn2)C)cc1C c1(C(N2CC(NC(C3CC(SC)C3)=O)C(CO)CC2)=O)cc([N+](=O)[O-])nn1C c1(CC(C)C)ncc(C(=O)NC2CC2NC(c2cncn2C(C)C)=O)s1 CCCC(C(=O)NC(C)CN(C(=O)CSCC(F)(F)F)CC)N(C)C c1(C(=O)NCC(CC=C)NC(=O)C(C)C2CCC2)cc(C)nc2c1c(C)nn2C N1(C(=O)CCn2cncn2)CCC2(CCCN(C(C34CCCC3C4)=O)C2)C1 C1(C(NNC(=O)NCCCCN2CCCCC2)=O)CCC2C(C1)C2(F)F C#CC1CC(NC(C2C=CC(NC(C3(N(C)C)CCC3)=O)C2)=O)C1 CCCC(C(=O)NC1(CCC)CCCC1)NC(=O)CSCC c1(-c2cc(C(=O)NC3CC(NC(CC4N(C)CCC4)=O)C3)on2)ccccc1F N1(C(C(CC=C)NC(C)=O)=O)CC(NC(=O)CC(C)O)C2(CC2)C1 N1(C(c2c(C)nsc2)=O)CC2(C1)CN(C(c1ncc([N+](=O)[O-])cc1F)=O)CCO2 C(=O)(C1=C(C)OCCS1(=O)=O)N1CC(CCNC(C(C(CC)C)OC)=O)OCC1 N1(C(COCC=C)=O)CCCC1(C)C(=O)Nc1ccc[n+]([O-])c1 C1(CNC(C2CC3(CCC3)C2)=O)C(C2CC2)CCN1C(c1csc(C(F)F)n1)=O C(C)(CCCN=c1[nH]cc([N+](=O)[O-])cc1Br)NC(Cc1c(C)ccc(F)c1)=O Cc1cc(C(=O)NCCCOCCNC(=O)CC(C)F)ncc1N C1(CO)CCC1C(F)(F)F.C1CC=CCSC1 Cc1nc(N2CCCC(CC(=O)Nc3ccns3)C2)sc1C(CN(C)C)=O Cc1cc(O)ncc1C(=O)NOC1CCNC1=O.C(=O)(CC1(C)CC1)N c1(CNC2CCC(NC(=O)CCN3C(=O)C=CC3=O)C2)cccc(Br)c1O C1(CCN(C(C(C)OCCOCC)=O)C)CCCN(C=O)CC1.C(C)(C)(C)NC(=O)O N1(Cc2cc(OC)cc(F)c2)CCC2(CCS(=N)(=O)CC2)C1 C=CC(C)(C)CC(=O)N1CC2CCC1(CNC(C1CCCN1CC)=O)C2 C1(NC(CS(CC)=O)=O)CCC2(CC1)CCCN(C(=O)C#CC1(C)COC1)C2 C1(NC(CSCCNC(c2c(C)cc(F)s2)=O)=O)CN2CCC1(C)CC2 c1(C(=O)NCC2(C(N)=O)CN(c3cnsn3)C2)cc2cc(Cl)ccc2[nH]1 c1(CC)sc(C(=O)N(CC(O)CN(C(=O)C(O)C(F)F)C)C)cc1C C1(CC=C)(C(c2ccc(N)cc2)=O)CCN(C(=O)CC)C1.C1(C=O)CC1(C)Br CC1(C)CN(C(=O)CCN2CCCC2)CC1NC(=O)CC1C=CCC1 c1(OC(C)C(=O)NC2CC(NC(=O)CC3COC(C)(C)C3)C2)cccc(F)c1 C1(CNC(C(c2n(C)cnc2)O)=O)COCCN(C(c2ccc(CF)cc2)=O)C1 N1(C(c2c(C)c[nH]n2)=O)CCC2(COCC(CNC(c3cscc3Cl)=O)O2)C1 N1(CCNC(CC2C(C)CCC2)=O)CCN(C(c2cn(C)[nH]c2=N)=O)CC1 C=CCCCCC(=O)NCC1CCN1C(c1cnc(C(N)=O)s1)=O N1(C(C2(F)CCN(C(c3c(OC)ccc(Cl)c3)=O)C2)=O)CCc2cccnc2C1 c1(NC(C2CN(C(CCCOC)=O)CC23CC3)=O)cccn2ncnc12 CC(CC(=O)N1CCC(C(=O)NCCc2ccncn2)C1)C1CC1 c1(CC(=O)NC2CC(NC(C=C(CC)CC)=O)C2)c[nH]c2nc(F)ccc12 C1(CN(c2cc(OC)ncn2)C2CCC(N)CC2)Cc2ccccc2C1 c1(NC(=O)NCC(c2cccc(OC)c2)(F)F)cc(C)c(F)cc1Cl O(NC(=O)C(C)(C)CCNC(=O)C(F)C1CCOC1)CC(C(C)C)O C=C1CC2(C1)CC(C(=O)NCC1(O)CCN(C(C3(C(F)(F)CC)CC3)=O)C1)C2 C1(F)(C(N(CCNC(c2n[nH]c(C)c2C)=O)C2CC2)=O)CCN(C)CC1 Cc1cc(C=CC(N2CC3CN(C(=O)C=CC(F)(F)F)CC3C2)=O)ccc1F c1(N(CC=C)C(C)C)nnc(SC)n1-c1cc[nH]n1.c1(S)ccccc1 c1(C(N2CCC(C)OC(C)C2)=O)coc2c1N(C)C(=O)CCC2 NS(=O)(=O)c1ccc(C(=O)NCCC2CCCN(C(C3(CF)CCC3)=O)C2)cc1 C1(C(N(CC(CNC(C2C=C(C)CS2)=O)O)C)=O)CCCC(C)(C)C1 CC(CC(N)=O)C(=O)NCCCC1(CNC(C2CC2C(N)=O)=O)CCCC1 N1(C(C(CN(C)C)(C)C)=O)CC2(NC(c3ccc(F)s3)=O)CCCC2(F)C1 c1(C(=O)NC2C(NC(COc3cccc(C)c3)=O)CC2)cc2n(n1)CCC2 N1(C(C2CCC(NC(c3nnc(O)nc3O)=O)C2)=O)CCC2(CCCOC2)C1 C(=O)(C(F)CC(C)C)N(CCOCCN(C(C(n1c(C)ncc1)C)=O)C)C C1(C(N(C(C#C)C)C)=O)C=CCN(C(=O)CCc2cccnc2)C1 Cc1ccccc1C(N1CC(NC(=O)Cc2ccccc2C(F)(F)F)C(O)C1)=O C(=O)(CC(C(F)(F)F)OC)N1C(COC)CN(C(c2cocn2)=O)CC1 C(CCCCCCCO)=CC(=O)NC(C(C)C)C(C)NC(=O)C(C)(C)c1cscn1 c1(C(N(C(CC)C(=O)N2CCCC2CC)C)=O)ccnc(C)n1 C1(NC(C(COC)(F)F)=O)CC2CC1N(C(=O)C(C)OCCc1ccccc1)C2 C1(C(N2C(CC(C)C)CC2)=O)CCCC(NC(c2c[nH]cc2C(C)C)=O)CC1 C(C)(CO)(C(C)(C)O)NC(CC(CNC(CC1ON=C(CC)C1)=O)C)=O C1(OCC(=O)NC2C(NC(c3c(C)snc3)=O)CC2)CCC(F)(F)CC1 c1(C(C(=O)N(CCN(C(C)C)C(C2CCCS2(=O)=O)=O)C)C)cccc(Cl)c1 N1(C(c2nnn(C)n2)=O)CCCC2(C1)CN(C(=O)CCCC1CCCO1)C2 C(=O)(CC(O)CC(C)C)NCC1C(C(N2CC(C(C)O)C2)=O)CC1 C1(CNC(c2ccc(CCC)[nH]2)=O)CC2CCC(C1)N2C(C1(O)CCOC1)=O n1(CCC(=O)NCC2CC(C)N(C(=O)C3=COCCO3)C2)ncc2ccccc12 C(=O)(C(CNC(=O)C(=O)N(C)C)CC(C)C)NCC1C(CCC)C1 C(C(F)C(=O)NCCN1CC(C)(O)C1)C1CN(C(C(C)OCOC)=O)C1 C(=O)(C#CC1CCCCC1)NC(C(C(C)C)C)CNC(=O)CN(C)C(N)=O C(=O)(CCCC(CC)NC(=O)C=C1CCCC1)N(CCN(CCC)CCC)CC c1(OC)ccc(OC)c(C(=O)NC2CC2CNC(c2cc(Cl)ncc2F)=O)c1 c1(NC(C2CN(Cc3ccnc(Br)c3)CCS2)=O)ncnc2cc[nH]c12 N1(C(c2cc(C)c(C3CC3)cc2)=O)CC2CC(NC(=O)C=CC3CC3)CC2C1 c1(C(N2CC(NC(C(C)OC)=O)C(C)(C)C2)=O)cnc2sc(C)c(C)n12 Cc1ccc(C)c(CC(=O)NC2CC(C)N(C(C3CC4(C3)CC4F)=O)C2)c1 CC1=C(C(=O)NCC(O)CN(C(=O)CCc2ccc(O)nc2)C)CCS1(=O)=O C1(C(=O)NC2CC(C)C2)CCCC1NC(c1nc(Cl)cs1)=O C1(CCNC(C(F)=C(C)C)=O)CCN(C(=O)CCCCCF)CC1(F)F CC1CC(C(N2CCOC(CNC(=O)CNC(C3CCCC3)=O)C2)=O)CCN1C c1(OC)ncccc1S(=O)(=O)N1CCC2CCC12 N1(C(COCCOC)=O)CCC2CN(C(c3ccnc(OC)c3)=O)C2C1 N1(C(C(CC)SC)=O)CC(Nc2ncnc3c2COC3)C2(CCOCC2)C1 C=C(CNC(=O)C(=O)Nc1ncccc1SC(C)C#N)CC(F)(F)F c1(CC)ccccc1C(=O)NCCN(C(=O)C(C)OCOC)C(C)C CC(C)(C)CCCCCC(=O)NCC1CC2COCC2N1C(c1ncc(Cl)s1)=O c1(C(=O)NC)nc(Nc2ccc(N(C)C)cc2)c2c(n1)CCCC2 c1(C(=O)OC)cc(C)c(NC(N2CCC2c2ccc(Br)cc2)=O)cc1F c12ccc(C)cc1N2.C1(C(N(CCC)C)C)CCCN1C(=O)CCn1cnnn1 Cc1nc2ccccn2c1C(=O)NC12CC(NC(C34CCC(C)(C3)OC4)=O)(C1)C2 c1(CC)[nH]c(=N)sc1C(=O)NC1(C)CC(NC(=O)C(c2cccnc2)O)C1 c1(CC)ccc(C(N2CCC2CC)=O)c(C)n1.N12CC(C1)C2=O C#Cc1cc(C(=O)NC(C)CCNC(=O)C(F)(F)C2CCCC2)cc(F)c1 c1(C(=O)NC(C2(O)CCOCC2)C)ccc(S(=O)(=O)NCc2ccccc2)cc1 C1(C(N2C(C3CCN(C(C4(C=C)CCC4)=O)C3)CCC2)=O)Cc2cccc(F)c2O1 C1(NC(c2ccc(O)cc2)=O)CC2CC1CN(C(c1cn(C3CC3)cn1)=O)C2 c1(C(=O)NCCCNC(C2(F)CC2)=O)sccc1S(=O)(=O)C(F)F C1(CCOC)(NC(c2c(C)nn(CCO)c2C)=O)CCN(C(=O)CSC(F)F)CC1 N1(C(c2ccnc3ccccc23)=O)CCC2C(CCCN2C(=O)CCC2CC2)C1 N1(C(C(C)C2CCOC2)=O)CCC(C(=O)NCc2nncs2)=C(F)C1 c1(CNC(C2N(C)CCC2)=O)ccc(C(=O)NCC2(CC3CC3)CC2)nc1 N1(C(c2c(C)nc(C)[nH]2)=O)CCC(NC(=O)CC2(C#N)CCC2)C(C)C1 C1(CC)CCN(C(=O)CCCF)C1C(=O)NCc1sc(C)nc1C C1(CCC(=O)OC)CCCN(C(c2ccccc2C(C)(C)C)C(=O)NCC(C)C)C1 C(c1nc2ccccc2o1)=CC(=O)N(CC(C)NC(C1CC1(C)Br)=O)C N1(C2CC(C(=O)NC3(CNC(C4CCC4)=O)CCOC3)C2)CCOCC1CO c1(CC(=O)NC(CNC(CCOC)=O)C(C)C)ccccc1Br N1(C(C(C=C)CC)=O)CCCC(C(=O)NCCc2nccc(O)n2)CC1 CC(C#N)C(=O)N1CCC1CC(=O)NC1(CO)CCOC1 CC(CNC(=O)C(=C1CCCCC1)F)CC(=O)NCc1nc(N(C)C)n[nH]1 CC1CCCN(C(=O)CCN2CCOCC2)C1CNC(=O)CCc1cn(C)cn1 Cc1cc(CNC(=O)CCC2CC(NC(C3(C)CCC(C)C3)=O)C2)cc(C)n1 CC1(C)CN(C(=O)C(O)CC2CC2)CC1C(=O)NCC=Cc1ccccc1 c1(OC(c2[nH]cnc2-c2cccnc2)=O)ccc(Cl)cc1Br Cc1sc(Br)c(C(=O)NC2(C(=O)O)CCCSC2)c1C CC(CC1CCC1)C(=O)NC1CC(F)(CNC(C2CCOC2C2CC2)=O)C1 CN1CC(NC(=O)CCC(C)(C)NC(=O)CC(=O)NC2CC2)C2(CC2)C1 c1(NC(C2C(NC(Cc3cccc(C)c3)=O)C2)=O)cnc(Br)c(Cl)n1 C(=O)(C(CCC1CCC1)NC(=O)Cc1csc(C)n1)NCc1cc(C)oc1 C(CN=c1cc(C)[nH]cc1C(=O)OC)C1N(C(c2ccc(CC)s2)=O)CCCC1 N1(C(CCNC(C)=O)=O)CCN(C(C2(C)COCC2(F)F)=O)CC1C Cc1ncc(C#N)cc1NC(C1(C(C)NC(=O)C(C)N(C)C)CC1)=O c1(C(C(=O)NCC2C3CN(C(=O)C(C4CCNCC4)O)CC23)O)ccc(F)cc1 CC(C(=O)N(CCCOCCNC(=O)CCC1CCOC1)C)C1(O)CCC1 c1(-c2cn(C3CN(CC4CCCC(=O)N4C)CCO3)nn2)cc(Cl)c(N)c(Cl)c1 CC1(C)C(CC(=O)NC2(CNC(=O)C(F)(F)C3CC3)CC(F)(F)C2)CC1O C1(O)(CN(C(c2cc(CC(C)C)c[nH]2)=O)CC)CCN(C(C2CC2(F)F)=O)C1 C1(NC(C2(CNC(=O)C3=COCC3)CC2)=O)CCCC1(F)F C(=O)(C(C)(CC1CCC1)O)NC1C(CNC(CN(S(CC)(=O)=O)C)=O)C1.C(C)(C)OC S(=O)(=O)(C1CCOCC1)N1CCC(O)(C(=O)NCCCN2CCCCC2=O)CC1 c1(C(CC)N(C(=O)C=Cc2ncco2)C(C)CC)c(C)cccc1Cl C1(NCc2cc(C)cc(C)c2)CCC2(C1)CN(C(c1cncc(C)n1)=O)C2 C1(C(N2CC(CS(C)=O)C2)=O)C2CCCC2CN1C(C1CCCCC(=O)N1)=O O(NS(=O)(=O)c1ccc(F)cc1)C.Cc1ccc(C2(C)CC2)c(C)c1 c1(OCC(=O)NC2C(NC(c3c(C)snc3)=O)CCC2)ccc(F)cc1Cl C(=O)(C(C)(C)COCC(F)F)NC(C(C)NC(C1CS(=O)(=O)C1)=O)C CC(c1ccccc1F)=CC(N1CCC2(NC(=O)Cc3cc[nH]c3)CC2C1)=O CCN(CC(=O)NCC(F)(F)F)N1CCC(COC)C1 CC(C)(CN=c1[nH]nc(C2CC2)o1)C(=O)NCC1CN(c2ccccc2)C(=O)O1 N1(C(CCc2c(C)n[nH]c2C)=O)CCCN(C(c2csc(O)n2)=O)C(C(C)C)C1 C1(C(=O)NC2CCN(C(c3c(C)n[nH]c3)=O)CC2C(N)=O)CN2CCCC2CO1 C(=O)(CCCC(C)(C)C)NCC12CCC(NC(CC(C)SC)=O)(C1)CO2 c1(N(CC(F)(F)F)C)nc(-c2ccn(CC(F)(F)F)n2)cs1 N1(C(CCOCCOCC)=O)C2CCC1C(C(=O)N(C)CCN(C)C)C2 N1(CC)C(=S)NC(c2ccc(CN(C)C)nc2)C2=C1CC(C)(C)NC2=O Cc1nonc1C(=O)NCc1cc(C(=O)NCCC(C)(O)C2CC2)co1 C(C)(CNC(=O)CC(C)F)(C(C)C)NC(c1nc(C)sc1)=O O=S(=O)(CCN=c1[nH]c(N2CCOC(c3ccc(Cl)s3)C2)nc(=N)[nH]1)C(F)F C1(C(=O)N)CCCN(C(=O)NCCN(C)CC(=O)NCC)C1.C1(OC)CC1 C1(CNC(CC2C(C)=NOC2=O)=O)(CO)CCCN(C(=O)CN=S(C)(C)=O)C1 C1(C(N2CC(COC)(CNC(c3n[nH]cc3C)=O)C2)=O)CCc2nnc(O)n2C1 C1(CNC(C(C=C)(C)C)=O)CCC2(CCC2)CN1C(C1C2CCC(C2)S1(=O)=O)=O C1(NC(c2ccn(CC)c2C)=O)(CNC(=O)C(=O)NCC(F)F)CCC(CC)CC1 N1(C(CC2(NC(c3c(OC)nsc3)=O)CC2)=O)CCC(O)(CN(C)C)C1 N1(C(C(C)C2CC2)=O)CCC2(CC1)CC2c1cn(-c2ccc3ncnn3n2)nn1 c1(-c2ccccc2)nc(N(S(=O)(=O)CC2CNCCOC2)CC)c(Br)c(C)n1 N1(C(C2CN(C(=O)NC)C2)=O)CC2(CNC(c3snc(Cl)c3Cl)=O)CC1CO2 C#CC1(C(=O)N(C(C)(C)CC(=O)NCC(C)C(C)O)C)CCCC1 c1(C(N2CCCC(CNC(C(C(C)C)OC)=O)C2)=O)cccc(Br)c1F C1(n2cc(CNC(C=CC)=O)nn2)CCN(C(c2cc(C#N)c[nH]2)=O)CC1 N1(C(C(=O)NCCCCNC(C=C(C)C2CC2)=O)C)C(=O)CCC1=O c1(NCCCN(C(CCc2onc(CCC)n2)=O)CC)cc(O)nc(O)n1 C1(NC(c2scc(COC)c2)=O)CN(Cc2cccc(Br)c2)CC1(C)C C1(CNC(CCN(C(C(COC)C)=O)C(C)C)=O)CCCC12CCC2 N1(C(c2cnc(C(C)C)o2)=O)CCCC(NC(=O)C(F)(F)c2cnnn2C)CC1 c1(C(=O)NC2(C)CC(NC(=O)C=C(Cl)Cl)C2)ccc(-c2cccnc2)cn1 Cc1cnc(CNC(C2CC(CCNC(C3CCCC(=O)C3)=O)C2)=O)c(C)c1 CC1CCC=C1C(=O)NCC(C1CCN(C(C2CCCCN2C2CC2)=O)CC1)O Cc1cc(CN2CCC3OC(=O)OC3C2)cc([N+](=O)[O-])c1 N1(C(C=CC(=O)N(C)C)=O)CCN(CCNC(=O)Cc2ccno2)CC1 C1(C(=O)NC2CCC2NC(C2(CC3CCC3)CC2)=O)CC(=O)N(c2cccnc2)C1 C1(NC(C2=NOC(C(C)=O)C2)=O)Cc2ccccc2C1NC(=O)CSCC#N n1(CC(N2C(C)(CNC(C3CC34CCC4)=O)CCC2)=O)cc([N+](=O)[O-])ccc1=O N1(C(Cc2cc(C)nn2C)=O)CCC(C)(C)CC1C(=O)NCCC1CC(F)(F)C1 c1(C(N2CC(NC(CC(C)(F)F)=O)C(C)(C)C2)=O)cc(F)cc2ccccc12 Cc1ccc(Cl)c(CNCC23CCCC2C3)c1 c1(OC(c2ncc(-c3ccccc3)o2)C)cccc(CC#N)c1 N1(C(c2c(OC)cccn2)=O)CC(NC(C2CC(OC)C2)=O)CC2(CCOCC2)C1 CC(C)(F)C(C)(F)CNC(=O)NCC1CCCOC1c1cccc(C(F)(F)F)c1 Cc1[nH]c(C#N)cc1C=O.N1CC(C)(C)CC1CNC1C(C=C(C)C)C1(C)C c1(CC(N2CC(Cn3cc(COCC)nn3)OCC2)=O)ncc(F)cc1F c1(C(N2CC(NC(C(C)c3cc[nH]n3)=O)C2)=O)nc(C(C)C)ncc1Cl N1(C(C(C)(C)C#N)=O)CCC2C1CCCN2C(c1cccn2ncnc12)=O c1(C(=O)NC2(C)CC(NC(c3c(C)nsc3N)=O)C2)cccc2[nH]ccc12 N1(CC(=O)NCC2(C(=O)Nc3ccnc(O)c3)CC(=C)C2)C(=O)CCC1=O C1(CC(C)NC(=O)NCCC2CCCC2)CCCCC1n1cc(Br)cn1 c1(C(N(CCOCCN(C(=O)C2=CCC2)C)C)=O)cc(N)c2ncccc2c1 C12(C(N(CCCN(C(c3ccc(CC)o3)=O)C)C)=O)CCCN(CC1)S2(=O)=O n1(CC(N2CC3C(NC(COC)=O)(CCC3)C2)=O)cc(C)c2ccccc12 C1(NC(C2C(C)(C)C2CO)=O)CCCSCC1.C1(C(=O)N)SCCS1 Cc1ncc(NC(=O)C(C2CC2)NC(=O)C(C)CN(C)C)cc1C#N c1(C(C)C)cc(C(N2CC(C)(NC(=O)Cc3cn(C)cn3)C2)=O)n[nH]1 C1(C(N2CCCC(N(C(c3scnc3Cl)=O)CC)CC2)=O)CCc2nnnn2C1 N1(C(CC2ON=C(C)C2)=O)CCC=CC1C(=O)N(CC(O)C1CCC1)C C1(C(=O)NCCCOC2(C)CN(C(CCOCCO)=O)C2)(CC)CCCC1O C1(O)(CN(C(C2CC(C)OC2)=O)C)CCN(C(C2(C)CCNC2=O)=O)CC1 Cc1[nH]ccc1C(=O)NCCN(C(=O)CCN1CCSCC1)CCOCCO N1(C(c2cccc(COC)c2)=O)CC(NC(C2CCC=CO2)=O)C2CCCCC12 N1(C(C(C)OCCCC)=O)CC(C2(NC(=O)CCCCNC(C)=O)CC2)C1 c1(C(=O)NCCC2(CNC(C3(C(=O)NC)CCC3)=O)CC2)cc2cccnn2n1 C12CN(C(C)(C)C1)C2=O.C1(C(=O)NCCCOC(=O)NC)C2CN(C)CC12 N1(C(CCc2n(C)ccc2)=O)CCCCC(NC(=O)CN2CCNC(=O)C2)CC1 C(=O)(CCCCCC(C)C)NCCC.c12nccnc1C(=O)N1CCC(CC1)N2 N1(C(C)=O)CCCC1(C)C(=O)NCC1(F)CN(C(=O)C=Cc2ccsc2)C1 N1(C(c2cccc(C)c2Cl)=O)CCC(C2CC(NC(C3(c4cccs4)CC3)=O)C2)C1 c1(OC)ccc(S(=O)(=O)CC(C)C(=O)OC)cc1.C12Cc3cscc3CN1C(=O)N2 c1(C(N2C(C3CCN(C(c4cnc(CC)s4)=O)C3)CCC2)=O)cccc(F)c1 CC(C)CCC(F)C(=O)N1CCCC1c1ncc[nH]1.C12CCN(CC1)C2=O C1(NC(c2nc(OCC)oc2)=O)CC2CC1N(C(=O)CCc1nc(C)cs1)C2 c1(N(C2CCN(C(C3CC(F)(CO)C3)=O)CC2)C)ncc2scc(Br)c2n1 C12C(C)CN(CC1C)CCNC2=O.C(C(=O)NCCC(C)(C)C)OCC=C.CCO N1(C(C2CC(SC)C2)=O)CC(C)(C)OCC1CNC(=O)Cc1n[nH]c(C)n1 CC(C)(C)C(CC(=O)N1CCCC(n2cc(-c3ncoc3C(=O)O)nn2)C1)NC=O c1(C(=O)NC2COCC2NC(C2CC2C2CC2)=O)cc(Cl)c(O)c(Cl)c1 Cn1nnc2c(NC3CS(=O)(=O)CC3NC(=O)COC(F)F)ncnc12 c1(C(CC)C)nc(C)cc(=NC(C)C2CCN(C(=O)Cc3ccsc3)CC2)[nH]1 c1(CCC(=O)NC2(C)CN(C(=O)CN3CCCC3)C2)cc(Br)ccc1F C1(CC)CN(C(=O)CC2(O)CCC2)CCN1C(c1ccc(Br)cc1)=O c1(OC)ccc(CN2CCC(N(C)C(c3cc(F)ccc3C)=O)C2)c(OC)n1 C1(C(=O)NCC(C)(F)F)(NC(C(C)SC)=O)CCN(C)C1 C1(CC)C(NC(C2(F)CCCCC2)=O)CCCN1C(c1cscc1C1CC1)=O c1(C(N2CC(CC(=O)NCCC(C)(C)C)OCC2)=O)cccc2c1CCCC2 C(=O)(C(C)(C)CCCNC(=O)CC#N)N(C)CC1(F)CCCC1 C1(CNC(C(C)=O)=O)(CO)CCN(C(C2CCCSC2)=O)CC1 c1(CC)noc(C(=O)NC2CCOCC2NC(=O)C(C)OCc2ccncc2)c1C C1(C(=O)NC2(CC=C)CN(C(=O)CC(O)CN(C)C)C2)CC(=O)N(CC2CC2)C1 C1(NC(C2C(CCC)CN(C(C3(C(C)(C)OC)CC3)=O)C2)=O)CC2CCC1CC2 c1(C(N(C(C)=O)Cc2nc(CC)on2)C)ccccc1[N+](=O)[O-] C(=O)(C(C)CC(F)F)NC1(CCNC(CCCSC)=O)CC1 C1(C(=O)NCC2N(Cc3onc(CC)n3)CC2)CCCCC1O c1(C(=O)NC2CN(C(CC3CC(=C)C3)=O)C(C)(C)C2)cc(OC)cc2c1OCC2 c1(C(=O)NCC2CCCN(C(C(C)(O)C(F)(F)F)=O)C2)[nH]nc2ncnc(O)c12 C12(CNC(c3nccc(C)c3)=O)CCCN(C(c3cncc(Br)c3C)=O)C1C2 c1(C(N(CCNC(C2(CC)CNC(=O)C2)=O)C)=O)nn(C)c2c1CCCC2 C(N=c1cc(C)c(C#N)c[nH]1)C1(F)CC(CNC(C2C(C=C(C)C)C2(C)C)=O)C1 CC1CN(C(C2(CCNC(C3(CCCF)CC3)=O)CC2)=O)CCS1=O c1(C(=O)NC(CC(=O)NC(C#C)(C)C)C)ccc(C)n1C Clc1ccc2[nH]cc(CCN=C(NCC3CCC34CCC4)NC3CCCC3)c2c1 C(C)(C(C)(C)NC(C1CC(C)(C(C)(C)CC)C1)=O)NC(C=CC=CC)=O C(=O)(CCS(=O)(=O)N1CCC(C(N2CCCC(CNC(C)=O)C2)=O)C(O)C1)OC N1(C(C=CSC)=O)CCCC2(CNC(=O)CC(C)n3ccnc3)CCCC12 C1(C(CNC(CC(C)C)=O)(C)C)CCCCN1C(c1ccnc(OCCO)c1)=O C1(C(C)C(=O)NCC(C)(C)C2CCC2)CCN(C(c2ccncc2CO)=O)CC1 C(=O)(C1CCCc2nnn(C)c21)NCC1(C(C)NC(=O)C(C)N2CCC2)CC1 C(=O)(CCN(OC)C(=O)CC1CCCC1O)NC(C=C)C1CC1 C(=O)(CCCCCC(C)O)N1CCC(CCNC(CCOCC(C)C)=O)(CF)C1 C(=O)(CCC(C)(F)F)NC1CCC(CCNC(Cc2cn(C)nc2Cl)=O)C1 C1(NC(C2C(O)CCN2C(C2CC3(CSC3)C2)=O)=O)(CO)CCCCCC1 c1(-n2cc(C(=O)NCC#CCNC(C3C(=C)C3)=O)nn2)ccc(Cl)cc1 C1(CC=C)(NC(=O)C(C)N(C)C2CC2)CCN(C(=O)CCC=CBr)C1 C1(COC)COC(C)(C)CN1C(C1CN(C(=O)CC(=O)OC(C)(C)C)CCO1)=O N1(C(c2cncc(OCC(F)F)c2)=O)CCN(C(c2n[nH]cc2Cl)=O)C2CCC12 CN=c1[nH]cc(C(N2CCC3CC23C(N2CC(F)(F)C2)=O)=O)o1 C1(NC(c2occ(C)c2C)=O)CCN(c2nccnc2F)CC1O N1(CC(=O)NC2CN(CC(N3CCC3)=O)C2)CCC(O)C2CCCCC12 c1(CNC(c2cccnc2)CC)ccc(N2CC(F)(F)C2)nc1 CC1(O)CCN(C(C23CC(NC(=O)C=CC4CCCC4)(C2)C3)=O)CC1F CCCC(C(=O)N(CC(O)CNC(c1cccc(C(C)(F)F)n1)=O)C)OC Cc1cc(C)c(C(=O)NC2CCOCC2C(N2CCCC3CC23)=O)o1 N1(C(C2C(CCC)CCC2)=O)CC(O)CC1C(=O)NCCP(C)(C)=O C1(NC(CCc2c(C)ncs2)=O)CCCC1(C)CN(C)C(C1(F)CC=CCC1)=O C1(C(=O)NCC2CN(C(CSCC(C)C)=O)C2)C2(CC2)C12CC2 Cc1nc(NC(c2ccc(OC(F)F)cc2)O)sc1C C12CCCCN1CC=CC(=O)N(C)C2.c1(C=O)cc(OC)n(C)n1.C(COC)OC c1(C(=O)NCC2(F)CC(NC(C3C(=C)C3)=O)C2)ccc2c(c1)NC(=O)CCN2C C1(C2CN(C(c3ccoc3C(C)C)=O)C2)(NC(CCc2cc(OC)no2)=O)CC1 c1(OC)cc(C(=O)NC(C)CCN(C)C(C2CC(CCO)C2)=O)ccc1OC c1(C(N(CC(CC)NC(=O)COc2ccn(C)n2)CC)=O)n[nH]cc1[N+](=O)[O-] O=[N+]([O-])c1ccc2c(c1Nc1cncc(OCCO)n1)CCN2 Cc1ccccc1S(=O)(=O)C1CCN(N2CCN(CC3CC3)CC2)CC1 c1(C(N(CCNC(C=Cc2ccc(CC)cc2)=O)C)=O)cc(N)cc(Cl)c1Cl c1(CC)c(C(=O)NC(C2CC(NC(=O)CC3CC34CC4)C2)C)[nH]c(C)c1C(C)=O N1(C(c2c(C)nc(O)nc2C)=O)CCC2CC1CN(C(c1c(C)noc1C)=O)C2 C(=O)(C(C)(C)CC#N)NCC1(F)CC(NC(c2nc(C)n(C)n2)=O)C1 N1(C(=O)OC(C)(C)C)CCN(C(=O)Cc2nccs2)C(c2ccc(F)cc2)C1 N1(C(C=C2CCN(C)CC2)=O)CCC2CN(C(=O)CSc3nc[nH]n3)CCC2C1 N1(CC)CCC2(C1)CC2(F)F.c12n[nH]cc1C(c1nnnn1C1CCOCC1)N2 C(=O)(C(C)(C)CCOC)NCCCN(C(CCCCOC)=O)C C(=O)(CC(C)(C)NC(c1nn(C)cc1C)=O)NC(C(=O)OC)C1(C)CC1 CC1=C(C(=O)NC2CC(CNC(=O)Cn3ccc(C)n3)C2)CCCC1 O=C1CCC(C(=O)N(CC(=O)NCC2CCCCO2)C2CCC2)C1 C1(C(=O)NC2(COC)CCN(C(C(CC)C(C)C)=O)CC2)CCc2c(ncn2C)C1 C#CCC(CC(=O)N(CC(F)(F)F)Cc1cc(C)nn1C)NC(=O)CC(=O)NC CC(C1CC1)=C(F)C(=O)N(CCNC(C1CC1C)=O)CCOCCO Cc1csc(C(O)CC(=O)NCc2cn(C3CN(S(=O)(=O)CC4CCC4)C3)nn2)c1 N1(C(c2ccnc(OC)c2F)=O)CC2CN(C(C3(C)CC=CC3)=O)CC2(C)C1 C1(C(N(CCOCC#C)C)=O)CC(C)N1C(c1cnc(C)s1)=O N1(C(C(C2(O)CCCCC2)NC(Cc2c(C)n(C)cn2)=O)=O)CC(C)C(C)C1C C(=O)(C1OCCc2ccccc21)NCC(CNC(c1c(OC)n(C)nc1)=O)CO c1(OCc2n(CC(=C)C)nc(-c3cccc(N)n3)n2)cc(F)ccc1F c1(C(N)=O)cc(C(=O)NCC23CCC(C2)C3)cc2nc(C(F)(F)F)[nH]c12 C1(NC(C(CCC)O)=O)CC2CC(NC(c3ccc(SC(C)C)cc3)=O)C1C2 N1(C(c2c(C)con2)=O)CC2CC2C1C(=O)NCC1COCCO1 c1(C(N2CCC23CC(CO)C3)C(=O)NCCOCCCF)cc2n(n1)CCCO2 Cn1ccc(C(c2nnnn2CSc2ccccc2)NCCc2ccco2)c1 Cc1cc(CNC(c2cscc2-c2cnn(CCCO)c2)=O)c(C)s1 c1(C(=O)NCC(CNC(c2cc(COC)no2)=O)CO)csc(S(C)(=O)=O)c1 CC1(C)COC(CC(=O)NCC2CC(NC(=O)C(C)(C)C3CCCC3)C(O)C2)C1 C1(O)(C(N(CC#C)C)=O)CCN(C(c2cccnc2)=O)CC1 C#CC1(NC(=O)C(C2CC2)NC(C2CCC(=O)NC2)=O)CCCCC1 CCC(C(=O)NCCCn1cc(C2(OC)CC(F)(F)C2)nn1)C(C)C c1(C(=O)NC(COCC)C(N2CC(C(N)=O)CCC2C)=O)cnc2n1CCC2 C(C)(CCCCN=c1nc(C)c(C#N)c[nH]1)NC(Cc1c(F)ccc(C)c1)=O c12ccc(cc1)OC2.N1(C(C)C)CCC(CSn2cncn2)C1 CC(C)(C)CCC(=O)NCCC1(NC(C23CC(CO)(C2)C3)=O)CCC1 Cc1cc(C#N)cc(C(N2CCCC(CO)(NC(=O)C=Cc3ncc[nH]3)C2)=O)n1 c1(CCC(=O)NCCN)csc2nc(C)cn12.N1(C(C(=O)CCC)C)CCSCC1 c1(C(=O)OC)nc(=NC2CC3CN(C(c4cc(Cl)nn4C)=O)CC23)c(F)c(Cl)[nH]1 Cc1cc2nc(C(C)OC(=O)C(C)Sc3ncccn3)cn2cc1C C1(CC=C)(N(C(=O)C(C)(C)CF)CC)CCCCC1.C(=O)C(C)=C1CCC1 c1(C(=O)NCC(C(=O)N(CC(C)C#N)C)N(C)C)c[nH]c2cnccc12 c1(OC)cc(C(N2CCN(C(=O)OC(C)(C)C)C(CO)C2)=O)c(F)c(Cl)c1 C1(F)(CC(N2CCC(CCNC(c3cn(C4CC4)cn3)=O)C2)=O)CCCCCC1 CC1(C)CCc2c(C(=O)NC3CCN(C(=O)C4=C(C#N)CCC4)C3)n[nH]c2C1 c1(OCCC)ccnc(CNC(=O)C(C)=C(C)C)n1.C1(C)CCN(C)C(=O)C1 C(=O)(NNc1ccc(S(=O)(=O)C(F)(F)F)cc1)C1CCC(NS(C)(=O)=O)C1 CN1CCC(CC(N2CC(F)CC2CC(N2CC(C)(CC(C)(C)C)C2)=O)=O)C1=O C1(O)(CNC(=O)CN2C(=O)CCC2=O)CCN(C(=O)CC2CSCCS2)CC1 C(=O)(C(C)(O)C(F)(F)F)NCCC(C)NC(c1cccc2occc12)=O CC1(C(=O)NCC(O)C(=O)NC2(CO)CCOC2)CC(=O)C1 c1(C(=O)NCC2CCN(C(=O)CCc3ccc(Cl)cc3Cl)C2)cc(Cl)c(F)cc1Br C1(C(C)NC(=O)Cc2cscn2)CN(C(=O)CSCc2cccs2)CCO1 C(=O)(CCCCC(=O)NC(CCF)C(=O)N1CC(OC)C(F)C1)OC Cc1cc(C)c(C(=O)NCC(Cc2ccccc2)N(C)C(c2c[nH]nc2Cl)=O)o1 C1(OC)CC(CNC(c2cc(C)nn2-c2ccc(Cl)cc2)=O)N(C(=O)CC#N)C1 C1(C(C)NC(c2ccnc(CO)c2)=O)CN(C(=O)CCC2CC(F)(F)C2)CCO1 C(CCC(=O)NC1CCC1NC(C1(OC(C)=O)CCCC1)=O)=CCC=C N1(C(c2c(C)[nH]cc2)=O)CC2CC(NC(C34CCCC3CCC4)=O)CC2C1 CCC(C)C(C(=O)NC(C1CCCCC1)CNC(=O)CN(C)C)NC(C)=O Cc1ccc(CN(C(Cc2cccc(CC(N3CCSCC3)=O)c2)=O)C)cn1 c1(C(C)N(C(=O)CCC2(C(=O)O)CCOCC2)C)ccc(-c2nn[nH]n2)cc1 C(c1cccc(Cl)c1)=CC(=O)NC(C)CC(C)NC(=O)C(CO)N(C)C C(=O)(CCC(F)(F)C(F)F)N(CCNC(=O)CC1CC2(CCCC2)CO1)CC Cc1ccc2c(C(=O)NCC3CN(C(c4occc4Br)=O)C3)coc2c1 c1(CC(=O)NC(CCOC)CNC(=O)C(C)NC(C)=O)cnn2c1OCCC2 c1(C(=O)NCC2C(NC(=O)Cn3cccc3)CCCC2)cnc2ccccn12 N1(C(C(CC)OCC)=O)CC2CCN(C(c3ccc[nH]3)=O)C2C1C C(CC(C)(C)C(=O)N1CC(CO)OCC1C)NC(CCCOCC)=O c1(CC(C(=O)O)NC(c2cncc(C(F)F)c2)=O)ccc(Cl)nc1 C(=O)(CC(F)F)NC1CC(C(=O)NC2CC(CC(=O)NCC3C(C)C3)C2)C1 C=CCCC(C(=O)N1CCC(COCC)C1)NC(C1CC(C)(C)CN1C)=O C(=O)(CCC(=O)NC)N(CC(C)(C)CNC(C1CCSC(C)C1)=O)CC C1(CNC(CC(CCC)CC)=O)CC2(CCN(c3cc(N(C)C)ncn3)C2)CO1 c1(CNC(C2CCN(C(c3c(C)[nH]cc3)=O)C2)=O)cnccc1Cl C1(C(=O)NC2CCCN(CC)C2)CN(C(=O)CC(=O)NC2CC2)CC(C)(C)C1 CS(C)(=O)=NC(=O)C(=O)NC12CCCC1N(C(C1(c3ccccn3)CC1)=O)CC2 C1(C(=O)Nc2ccc(C(=O)NC3CC3)cc2)CC1C1CCCCC1 c1(C(OCCC(=O)N(CC=C)CC2CC2)C2CC2)ncoc1C Cn1ncc(Cl)c1C(N1CC(NC(C2CC2F)=O)CC1CO)=O C1(C(=O)NCCC(C)CCO)CCC(C)(C)N(C(=O)CC(C)F)C1 Cc1ccc(CC(=O)NC(C)CN2CCN(C(c3cc(C)n(C)c3)=O)CC2)cc1F C1(C(C)(C)NC(C(C2CC2)OCC)=O)CCCN1C(=O)CC1(C(F)F)CC1 C1(NC(C(CCC)C)=O)CN(C(c2[nH]cnc2C#N)=O)CCC12CCC2 Nc1ccc(F)c(C(N2CC(NC(C3CS(=O)(=O)C3)=O)CC3(CC3)C2)=O)c1F C1(C(N(CC=C)CCO)=O)CN(C(c2ccc(N(C)C)nn2)=O)C(C)(C)C1 C1(O)(CC2CC2)CCCN(c2ccc(C(=O)NCCNC(C)=O)cc2)C1 N1(C(C)C)CCCC(C(=O)NCCC2CSCCN2C(=O)CS(N)(=O)=O)C1 C1(C(N(C)CC2N(C(C(C(C)C)=O)=O)CCCC2)=O)CC1C1(C)COC1 Cc1cc(F)ncc1NC(c1sccc1NCc1cnccc1C)=O Cc1cc(CC(N2CC3(C2)CN(C(=O)CC2CC(=O)C2)C3)=O)ccc1CO N1(C(c2ccnc(C)n2)=O)CC2CC(CNC(c3cnsc3)=O)CC1C2 C1(CCNC(CC=CC)=O)CCCCN1C(=O)CCSCCC c1(NC(C(C)(CO)NC(COCCCC(C)C)=O)=O)cccc2[nH]ncc12 C1(C)(C(=O)NC(CC=C)CNC(c2cc(C3CC3)on2)=O)CC(C(F)(F)F)=NO1 CON1CC(C(=O)NC(C(=O)N2CCS(=O)(=O)CC2)C(C)(C)C)CC1=O CCC(C)(C)CN=C(NCC(C1CC1)OC)N(C)Cc1ccco1 C1(N(CC#C)C(c2nsc(N)n2)=O)CCN(C(=O)CSC2CCCO2)CC1.C(N)=O c1(C(=O)NC(CC)CNC(C2CCCC(C)(C)CC2)=O)nc2ccccc2nc1C c1(C(=O)NCC2(OC)CN(C(=O)CC3CCS(=O)(=O)CC3)C2)c(O)cccc1F C#Cc1cccc(C(=O)NC2CC(C)CN(C(c3ncn(C)n3)=O)C2)c1F C1(C(N(CC(=O)N(CCOC)CCO)C)=O)(NC(=O)CSC)CCSC1 CC1(C)C(=O)C(C2CC2)C(=O)NC2C(C2)C(=O)N2C1CCC2.C(C)(C)(C)NC1CC1 c1(CC(=O)NCC(C(C)C)(C)NC(C2CCO2)=O)cc(F)ccc1Br c1(C(C(=O)NCC(CO)NC(C(=O)NCC)=O)(C)C)ccc([N+](=O)[O-])cc1 c1(OCC(C)N(C(c2ccc(CC)o2)=O)CCOC)c(C)cc(C)cc1C n1(CC)nnc2c1CCC(C(=O)NC1CC13CC(NC(c1cc(Cl)no1)=O)C3)C2 C=C(C)C1CCC(C)(O)C(C(N2CCC(OC(=O)Nc3ncccn3)CC2)C)C1 n1(CC=C)nnnc1C(C(C)(C)SCC(C)SC)NCCOC(C)=O O=C(CCCCCn1ccnn1)NC1C=CCCC1CO C1(CNC(CCc2scc(C)n2)=O)C2CN(C(C3CC(=C4CC4)C3)=O)CC12 N1(CC(c2ccc(OC)cc2)NCC(=O)NCC#N)C(=O)c2ccccc2C1=O c1(CNc2ccc(NC(C(N3C(OC)CC3)=O)=O)cc2)ccc(F)nc1OC C12(NC(c3c(C)con3)=O)CCCC1N(C(=O)C(C)SCC1CCCCO1)CC2 Cc1nn(C)c(C)c1OCC(=O)NC(C)C(C)NC(c1cc(C2CCC2)[nH]n1)=O O(NC(=O)C(C)(CSC)NC(=O)Cc1cnoc1)CC(=C)C c1(CC(N2CCN(C(Cn3cccc(N)c3=O)=O)C3C2C3)=O)ccc2nn[nH]c2c1 N1(C(C(C)OC)=O)CC(N=[N+]=[N-])CC1C(=O)N(C1CC(C)(C)C1)C Cc1cc2c(C(N3CC4CC4(CNC(C4CCC(=O)C4)=O)C3)=O)ccc(C)c2[nH]1 C(=O)(CCCCC#N)N1C(C(C)(C)NC(C2N(CC(C)C)CCC2)=O)CCC1 N1(c2snc(CCC)n2)CCN(C)C(C2(C3CC4CCC3C4)CC2)C1 N1(C(C(C)OCC#C)=O)CC2CC1CN(C(=O)CCC[N+](=O)[O-])C2 c1(C(=O)NC2CC(CNC(c3c[nH]c(=O)cn3)=O)OCC2)cccc(F)c1O C1(CC(=O)N(C)CC2C(NC(c3cn(CC=C)nc3)=O)CCC2)CC(C)(C)CO1 Cc1cnc2n1C(C(=O)NCC(C)CNC(=O)COCC1CCOC1)CCC2 C1(NC(c2nc(OCC)oc2)=O)CCN(C(=O)C=CC(F)(F)F)C1C C1(C(N2CC(OCCOC)C2)=O)CCCCC1CNC(C1CCOC(CF)C1)=O N1(C(CCC(C(C)C)NC(c2ccn(C)c(=O)c2)=O)=O)CCC2(C=CCO2)C1 Cc1cccc(C(N2CCN(C)C(C(=O)Nc3conc3C)C2)=O)c1C C(c1ccc(NCc2ccc(C)o2)o1)=CC(N1CCNCC1)=O C#CC1CCC(C(=O)Nc2ccc(OCCOCCO)cc2)CC1 C1(NC(C(CC=C)(C)C)=O)Cc2ccccc2C1NC(=O)C(C)C1CCCO1 c1(CC(=O)NCC(CNC(C=Cc2n(CC)ncc2)=O)(C)O)cccc(C)n1 CN1C(=O)C(=O)N(CC(=O)NCCC2CN(C(C3(C)CCCC3O)=O)C2)C1=O C1(NC(=O)OC(C)(C)C)C2CCCC1N(c1cc(O)nc(Cl)n1)C2 N12CCCC(C1C)C(=O)NCC2.c1(C(=O)OCC)cc(COC)no1 N1(C(C2CC(C(C)(C)C)C2)=O)CC(NC(C2(F)CC=CC2)=O)CC2(CCC2)C1 Cc1oc([N+](=O)[O-])cc1C(=O)NC1CC(OC)CN(C(=O)C(C)CC2CC2)C1 c1(CC(N2C(C(C)NC(c3ncc(C)cn3)=O)CCC2)=O)cc(Cl)ccc1O n1(CC)ccnc1CNC(=O)C(C1CCCCC1)NC(C1CC1(C)C(C)C)=O N1(c2nc3c(cc2)C(=O)CC3)CCC2(NC(c3n[nH]cc3Br)=O)CCCCCC12 C(c1cccc(Br)c1)=CC(=O)NCC(C)NC(C1(C)COC(=O)C1)=O c1(CNC(C(C)(C(C)C)NC(C)=O)=O)n[nH]c2c1CN(C(C1CC(O)C1)=O)CC2 N1(CC(=O)NCCCCCNC(CC(C)OC)=O)CCCC(C(F)(F)F)C1=O N1(C(CC)=O)CCC2C(C1)NC(=O)CN2C(c1cc([N+](=O)[O-])oc1C)=O N1(C(COCC(=C)C)=O)CCN(C(=O)CSc2cnn(C)c2)CC1 C(C1CCCCCC1)=CC(=O)NC1CCCCC1CNC(c1cc(CF)on1)=O N1(C(=O)OC(C)(C)C)CCOCC1CC(=O)N(CCSS(C)(=O)=O)C1CC1 c1(CC)nccnc1C(=O)N(CCN)CC.c1(NC(C)=O)cccc(C(C)=O)c1 C1(C(N(C2CCC(CNC(C3CC(C)OC3)=O)CC2)C)=O)CCC2(C1)CC2(F)F n1(CC)ccc(C(N2CCCC(CNC(=O)CCCN(C)C(C)=O)C2)=O)cc1=O C1(C(N2CC(CNC(C3C(CCC)C3)=O)(COC)C2)=O)CC(=O)N(OC)C1 CC(C)(O)C#CC(=O)NC(CCC1CCC1)C(=O)NCC1CC2(CC2)CO1 N1(C(C(c2ccccc2)NC(c2scc(CC)n2)=O)=O)CCCC(CO)C1 O=C1CC2CN(C(=O)C(=O)NCCOCCOCCO)C1=CC=CC=C2.C(CO)OC c1(NC(C(=O)NCc2ccn(CCC(F)F)n2)=O)c[nH]c(-c2ccncc2)n1 CC1(NC(c2cc(C(N)=O)ccn2)=O)CCN(C(C2(S(C)(=O)=O)CC2)=O)CC1 C1(C(=O)NC2(C)C(C)OCC2)CC2(CCN(C(=O)CC(Cl)Cl)CC2)C1 N1(C(C2N(C)CC(C)(C)C2)=O)CC=C(CCNC(c2cc(Cl)cnc2O)=O)CC1 c1(CC(=O)NC(CC)CNC(c2cccc(OC)c2)=O)cn2cccc(C)c2n1 C(=O)(CCC(F)(F)F)NC(c1cnn(C)c1)C(=O)NCCCCCCN(C)C N1(C(c2scc(CNC(c3cc(C)sc3)=O)c2)=O)CC(C)CCC12CC2 C(C(C)(O)CC(=O)NC(C)CC1CN(C(C2CCCCN2CC(F)F)=O)C1)OC c1(OC(CC)C)ccc(C(=O)NC(c2ccno2)C)cc1 C12(CNC(C3N(CCC)CCC3)=O)CCC(C1)N(C(C)=O)C2 CC1(C(=O)NCCCCCNC(=O)CCc2cc[nH]n2)CCC(=O)NC1 C1(NC(C2C(C)(C(C)C)C2)=O)COC2(C1)CN(C(=O)C(C)(C)C(C)(F)F)C2 c12c(noc1C)C2.c12csc(n1)NC(CC)CN(CC)C2=O.C(C)(=O)NC C1(NC(Cc2nc(C)sc2)=O)CCCC(N(C)C(c2cc(Br)c[nH]2)=O)C1 CC(CNC(C1(CF)CC(=O)C1)=O)C(F)C(=O)N=c1ccn(C2CCC2)[nH]1 c1(C(N(CCC(C)NC(C2COCCN2CC(F)F)=O)C)=O)cc2n(n1)CCC2 C12C3CCC(C3)N1C(=O)COC2=O.N12CCN1CC2.Cc1nnc(C)o1.C(C)(C)(C)O C1(C(N2CCC(NC(c3c(CC=C)cccc3)=O)C2C)=O)CCn2nncc2C1 c1(C(N(CCNC(CC2CC(=C)C2)=O)C)=O)cc(OC)cc(F)c1 CCCCCCC(C)C(=O)N(CC(N1CCn2nccc2C1)=O)CC1CC1 C(Cc1nn[nH]n1)(C(F)(F)F)NC(c1ccccc1C(=O)C(F)(F)F)=O C=C1CCC(C(=O)NC(C)CN2CCN(C(c3ccnc(CC)c3)=O)CC2)CC1 c1(C(=O)NC2CCC(C)N(C(=O)C(N3CCSCC3)C)C2)ccnc2ncnn12 c1(C(=O)NCCN(CCC)C(C2(C)C=CCCC2)=O)ccc(C)n(C)c1=O CCC(CO)C(=O)N(C1CCN(C(c2ccnn2CC(F)F)=O)CC1)CC1CC1 C=CCN=c1[nH]cc(Nc2nc(Cl)c(C(=O)OCCC(=O)OC)s2)s1 CCC(CC(=O)NCC1(CC(=O)NCC2CC2(F)F)CC1)CC(C)C c1(C(=O)NCC(CNC(C(C(CC)C)OCC)=O)(C)C)ccc(F)c(C)c1C#N O=C(Cn1ccnn1)NOCC1CC12CC2.C12CN(C1)C2=O c1(-c2cn(C3CN(C(c4cc(C)cc(F)c4)=O)C3)nn2)ccc2nccn2c1 Cc1cc(CNC(c2cc(Cl)c[nH]2)=O)oc1C(N1CCC(C(C)C)CC1)=O N1(C(CCC)=O)CCCC(C(N2CCC(CNC(=O)COC(C)=O)C2)=O)C1.C1CO1 N1(C(c2cnc(CC)nc2)=O)CCC(C(=O)NCC(C2CCCCC2)C)C12CC2 c1(C(N2C(C)CC(NC(C3OCCC3(C)C)=O)CC2)=O)cc2cnccc2o1 C1(C(C)C)CN(C(=O)CN2CCCCC2=O)CCN1C(C1CSCCS1)=O c1(OC(C)C)nc(C(=O)N(CCCNC(=O)C(F)(F)C2CC2)C)cc(O)n1 c1(OC)nccc(C(=O)NCC2CCCN(CCC(F)(F)F)C2)n1 c1(C(=O)NC(CC)(C)CNC(=O)C(C)(C)C2CCOC2)cc(F)ccc1Cl N1(c2nccc(=NCc3ccc4cn(C)nc4c3)[nH]2)CCC2CN(C3CC3)CC2C1 C(CC1=CCN(C(C2(F)CC=CC2)=O)CC1)NC(C(C=C)(C)O)=O C12(C(N3CCC(F)(CNC(C4CCC(=O)N4)=O)C3)=O)CCC(CC1)CC2 N1(C(c2ncn(C(C)C)n2)=O)CCCCCC1CNC(c1n[nH]cc1F)=O CCCC(C(=O)N(C(C)CCSC)C)NC(c1[nH]nnc1C1CC1)=O N1(CC)CC(CNC(N2CCOC(c3cccc(C)c3)C2)=O)OC1=O c1(C(=O)NCC2(NC(C3CCC(C)S3)=O)CCC2)cnn2c1CC(F)(F)C2 CC(C(C)(C)C)=CC(=O)NCC1CCN(C(=O)C(F)(F)c2cncs2)C1 N1(C(CC2CCN(C(C3N(CC)CC3)=O)C2)=O)CCCC(C)(C#N)C1 CCC(CC(=O)N1CCCC1CN(C(=O)C=CC(F)(F)F)C)c1ccccc1 C1(CC#C)(C(=O)NCCCCN(C(=O)C(C)N(C)C(C)=O)C)CCOCC1 N1(C(c2cc(C)ncn2)=O)CCC(O)C(N(C(=O)C=C2CN3CCC2CC3)C)C1 N1(C(c2c(C)nns2)=O)CCCCC1Cc1cn(Cc2cccc(Cl)c2)nn1 CC(C)C(=O)CCc1cn(-c2cn(C(C)Cc3cccc(Br)c3)nn2)nn1 N1(C(=O)NCC(CC)(CC)c2ccccn2)CCC2(C1)CC2(F)F CC(CS(C)(=O)=O)C(=O)N1C(C(=O)NCC(N2CCCCC2)=O)CCC1C C(=O)(C(C)(C)C(O)CC)NC1CC(CNC(C2(C)CC2C(=O)OCC)=O)C1 N1(C(c2c(OC)ccnc2F)=O)CC(CNC(C2CCC2(F)F)=O)OC(C)(C)C1 C1(CC)CN(C(C2CN(C(C)C)CCO2)=O)CCN1C(c1ncc(OC)cn1)=O c1(NC)cnccc1C(N1CC=CC(NC(=O)CN2CC3CC3C2)C1)=O c1(C(=O)NCCCC(C)(C)NC(c2ccsn2)=O)ccc(N)cc1F C(=O)(C1=COCCC1)NC1CC(C(=O)Nc2c(C(C)=O)csc2)C1 C(=O)(C#CC1CCCC1)NC1C=CC(CC(N2CC(C)(C(=O)OC)C2)=O)C1 N1(C(CC=CC(C)(C)C)=O)CCC(NC(=O)C2=CCSC2)CC1c1ccccc1 CC(C(CO)NC(=O)C=Cc1ccco1)NC(C1CCCC1c1cnn(C)c1)=O c1(C(C)=O)ccc(C(=O)NC(C2CCCCN2C(c2cc(CF)on2)=O)C)nc1 C1(C(=O)Nc2cc(C(F)(F)F)ccn2)CC2(C1)CC(C(=O)NCCC(N)=O)C2 CC1CCN(C(C2CCC(C)CC2)=O)CCN1C(=O)C=CI C(CN=c1[nH]c(=NCc2nnc(O)o2)c2ncccc2[nH]1)c1ncc(C)o1 c1(CC(=O)NCC(C)N(C)Cc2n(CCOC)ncc2)ccc(Cl)c(Cl)c1 C(C)(C)(CC(=O)N1CCC(NC(=O)COC2CCCCC2C)C1)OCC c1(NCC(C(C)(C)C)NC(C(CCC)OC)=O)cc(=O)n(C)c(O)n1 N1(C(c2cccc(C)c2C)=O)CC(C(=O)N(C(C)C(C)(C)C)C)CCC1(C)C N1(C(C(CC)Nc2ccccc2)=O)CC(NC(=O)C=CCF)C2(CCOCC2)C1 CNS(=O)(=O)NCC(=O)NCC(C1CCCC1)NC(=O)CCNC(N)=O C(=O)(CC(CC)CCC)NC1(CC=C)CCN(C(c2cc(Cl)cc(Cl)c2)=O)C1 c1(C(=O)NCCC(CC)NC(=O)OC(C)(C)C)ccc2ncc(Br)n2c1 c1(C(N(C)CCNC(=O)C=C(C)C(C)(C)C)=O)cc(C)n(-c2ccc(F)cc2)n1 N1(C(c2n(C)c(O)nc2)=O)CCC2(CNC(C3(S(N)(=O)=O)CC3)=O)CCCCC12 c1(C(N2CC3C(CCNC(C4C(=C)C4)=O)(CC3)C2)=O)cc(C)sc1S(N)(=O)=O C1(c2cn(C(C)C(c3cc(=O)n(C)o3)N(C)C)nn2)CCOC2(CCC2)C1 c1(-n2cc(C(C)(C)N(C(C)C(=O)Nc3ccccc3)C3CC3)nn2)cncc(N)c1 N1(C(C2CC(OCC)C2)C(=O)NC(C)(C)CC)CCOC(CO)C1 c1(CC)nnc(C)cc1C(=O)NCC(C(C)C(C)C)NC(c1cc(C)c(C)[nH]1)=O c1(NCCNC(=O)Nc2ncnn2CC(F)(F)F)noc2c(F)cccc12 N1(C(c2ccnc(C#C)n2)=O)CCC2(CC1)CCN(C(c1ccoc1)=O)C2 CCN=c1[nH]cc(C(=O)NC2CC(CCNC(C3CC(C)(C)CCO3)=O)C2)s1 CC1(C)CCC(CC(N2CC3(NC(=O)CC4(O)CCOC4)CC2C3)=O)C1 C(=O)(C(C)(O)C(F)(F)F)NCCCCCSCCOC.C1(OCC)C(=O)N1 c1(NCCOCC)ccc2c(c1)C(=O)CCS2 Cc1ccc(C(N2CCC(CS(=O)(=O)C(F)(F)F)C2)=O)c([N+](=O)[O-])c1 c1(OC)ncc(C=CC(=O)NCC(C)NC(c2ccc(=O)n(C)c2)=O)cn1 C1(F)(C(N2CC(CC)N(C(c3cc(C)cnc3N)=O)CC2)=O)CC2(CCC2)C1 C(CCCCC)(c1n(CC=C)nnn1)NCC1CC1C1CCCO1 C12(OC)CCC(NC3CCCN(C4CCCCC4)C3)(CC1)CS2(=O)=O Cc1ncc2n1CC(C(=O)NC(C)CNC(=O)CCC1CCCOC1)CC2 C(=O)(CC1=CCN(C)CC1)NC1CCC2(NC(CCC(=O)N(CC)CC)=O)C1C2 C1(C(=O)NCCCN(C(=O)C(C)(C)C2CCC2)C)CC1C1CCOCC1 C1(CNC(C(c2ccccc2)SC)=O)CC(NC(C23CC(C)(C2)C3)=O)C12CCC2 CC(C(=O)NCCOCCN(C(=O)CNC(=O)C1CC1)C)C(F)F CC1CCCCCN1C(C1CCN(C(C2CCNC2=O)=O)C(C)C1)=O C1(CN(C(=O)CCC2(C)CN(CC(F)(F)F)C2)C)CC(=O)C1(C)C C1(C(C)NC(C2N(CC)CC2)=O)CCN(C(C2(OC)CCCC2)=O)CC1 c1(CC(C)(C)C)nnc(C2CCCn3cnnc32)o1 C1(CNC(C(CCC)=CCC)=O)CCCCN(C(=O)CSCc2cccnc2)C1 N1(C(c2cc(-c3cccnc3)on2)=O)CC(NC(=O)C(F)(F)Cl)CC12CCC2 C1(NC(CSc2n(C)nnn2)=O)CN(C(c2ccon2)=O)C2(CCCCCC2)C1 c1(CCC)ccc(CN(N2CCCC2)C(C)C)o1 C=CC(CC)CC(=O)N1CCCOC(CCNC(c2csc(C(C)=O)n2)=O)C1 c1(C(c2nnnn2C2CC2)NCC(=O)NCC)cccc(C#N)c1.C1(N)CCCO1 c1(OC)ccc(C(N2CC3CC2C3NC(=O)C(C)N2CC(C)C2)=O)cc1C(F)F c1(CCC(N2C(CC)CN(C(C3SCC=C3C)=O)CC2)=O)cnc2ccccn12 C1(C(F)(F)C(=O)NC2CC(C)(NC(C3CC(O)C3)=O)C2)(OC)CCCC1 C(N=c1nc2scnc2c(NCC(C(c2cccc(OC)c2)C)SC)[nH]1)SC C12CC13CC(C3)NC2=O.n1(CC(=O)NC2(CSC)CC2)ccc(C)c1 CCC(O)CC(=O)N1CCSCC1CCNC(C1CCCCN1C(C)C)=O C(c1cccc(F)c1)=CC(=O)NC1CCCC(N(C(CCOCC(C)C)=O)C)C1 C1(CC)CN(C(C2(NC(C3CCCO3)=O)CCC2)=O)CCN1C.n12cc(nn1)C2 c1(C(N2C(CN(C(=O)C(C)(C)c3cnsc3)C)CCC2)=O)cc2sccc2s1 N1(C(C(C2CCOC2)NC(CCC=CCC=C)=O)=O)CCCCN(C)CC1 c1(C(=O)NC2CC2CCC(=O)N(CC)Cc2nccs2)nocc1C(C)C c1(-c2[nH]c(N3CCC4(CCCO4)CC3)nc(=NC)n2)ccc2oc(Cl)nc2c1 N1(C(C2CC(C)(C)O2)=O)C(CNC(=O)CCn2ccccc2=O)CC2COCC12 CC1=NOC(C(c2nnnn2CC2CC(OC)C2)Nc2coc(Cc3ccco3)c2)C1 C1(CNC(COCCCCC)=O)CC(NC(=O)Cc2ncoc2C)C(O)C1 C1(C(N(C(C)CNC(C2CC3CC2CC3O)=O)C)=O)CC2(CCCCC2)C1 c1(-c2c(C)cc(Oc3cccc4c3OCO4)nc2)ccc2ccn(CC#N)c2c1 C(=O)(C#CC(=O)N1CCOC(CNC(c2cnn(C)c2N)=O)C1)N(C)C N1(C(c2cnc(Br)n2C)C(=O)NCCOC)CC2CC1CS2(=O)=O c1(NC(C(C)SCCCC)=O)ccc(OC)nn1 Cc1cc(C)c(C(=O)NC2CN(C(=O)CC3CCOC3C)C2)c(C)c1 CC1(C#N)CCC(c2nnnn2C2CC2)(NCCc2nc(CCOC)n[nH]2)CC1 Cc1c(C(=O)NCC2CN(C(C3CC(F)C3)=O)CCC2C)cccc1F C1(CNC(CCc2nnc(C(C)C)o2)=O)CCN(C(C2CC2(F)F)=O)C12CCC2 N1(C(C=CC(C)(C)SC)=O)CCCCC1CNC(c1cc(Cl)cn1C)=O C(C)(c1cccc(Cl)c1)=CC(N1C(CNC(CC(CC)C2CC2)=O)CC1)=O N1(C(C(C)(C)NC(c2cnc(C3CC3)nc2)=O)=O)CC2CC3CC(C2)CC1C3 CC#CC1CN(C(C2CCC(OC)CC2)=O)C1.C12COCCC1NC2=O N(C(=NCCF)NCC1CC2CC1C2)CC1CCC(SC)C1 C1(NC(c2cnc(Cl)c(Cl)c2)=O)CCN(Cc2ncccc2C(F)(F)F)CC1F C1(C(N2C(CC(=O)NC(c3ccn(C)n3)CC)CCC2)=O)CC(C(C)C)=NO1 N1(C(c2c(C)nsc2)=O)C(C)C2CC1C2NC(c1nccn1C)=O C1(CCN(C)C=O)CCCN(C(C2(C)CC=CCC2)=O)C1.C(C)(C)(C)O N1(C(CCC(N)=O)=O)CCC(O)(C2(NC(=O)CC3CCNC(=O)C3)CC2)CC1 CC1(CNC(c2ncsc2C(F)(F)F)=O)CCCN1C(C1(C(F)F)CCCO1)=O C1(C)(CC(=O)NCC(CC)N(C)C(c2cc(-c3ccccn3)[nH]n2)=O)CCCC1 C1(NC(c2ccc(Cn3ccnn3)o2)=O)C2CC1N(C(=O)COCC(F)(F)F)C2 C1(CC=C)(NC(=O)C=C(C)C)CCCN(C(=O)C(c2cncnc2)C)C1 C1(CCCNC(C2C(CC(C)C)C2)=O)CCCCN1C(C1CN(C(N)=O)C1)=O c1(C(=O)NCC=C2CCN(C(=O)CC3(O)CCC3)CC2)nc2c(s1)COCC2 c1(NC(CCC(=O)NC(C=CC(=O)OCC)C)=O)ccc2c(c1)OCO2 C(CCN(C(=O)C=CC1CC1)C)OCCN(C(CN(C)C)=O)C.C(CCO)SCC N1(C(C2OCCN(C(C(C(C)C)NC(C)=O)=O)C2)=O)CCSC2(CCC2)C1 C1(O)(C(N(C)CC2CC2)=O)CCN(C(=O)CCCSC2CC2)C1 C1(CNC(c2nc(CCC)oc2)=O)CN(C(=O)CCn2nc(C)nc2C)CC1C c1(OC)c(C(=O)NC2CCN(C(=O)CC(C)C3CCCC3)CC2O)occc1=O C12(CNC(C(CCC)O)=O)CCC(NC(c3ccnc4nn[nH]c34)=O)(CC1)CO2 N1(C(CCC#N)=O)CCC2CN(C(c3cc4cc(Cl)sc4[nH]3)=O)CCC2C1 c1(C(N2CC(NC(Cn3c(C(C)C)ncc3)=O)C3C2C3)=O)cc(C#N)ccc1F c1(NC(C2C(C(=O)Nc3snc(C)n3)C2)=O)cc(-c2ccccc2)ncn1 CC(C)CC(O)CNC(C1(NC(C2(n3nccn3)CC2)=O)CSC1)=O c1(OCCC)ccc(C(=O)NCCC2(O)CN(C(c3cccc(N)c3)=O)C2)cc1 n1(CC(=O)NCC(CO)NC(C(C)OCCC=C)=O)cc(C)c(C(F)(F)F)n1 c1(C(N2CCC(CC=C)(C(=O)NC3(C)CCCC3C)C2)=O)cc([N+](=O)[O-])n[nH]1 c1(NC(C(C(C)C)CNC(c2cccc(O)c2F)=O)=O)cc(C#N)ccc1O c1(C(N2CC(C(=O)Nc3c(C)cns3)C2)=O)ccc(Cl)nc1OC1CCC1 C1(CN(CCCC)Cc2cccc(F)c2C)CCC(F)(F)CC1 N1(C(=O)CCn2cc(-c3ccccn3)nn2)CC2SCC(C2)C1 N1(C(CCSCCC)=O)CC(C(C)(C)O)(CNC(C2CC2Cl)=O)C1 Cc1ccn(CC(=O)NC2CCN(C(=O)COC3CC(F)(F)C3)C23CC3)c(=O)c1 c1(-c2n(-c3ccn(CC)n3)nc(CCC(C)C)n2)cccc2cnnn12 Fc1ccc2scc(CNC(=NCCc3ncccn3)NCC3CC3Cl)c2c1 c1(NC(c2[nH]cc(C(N)=O)c2)=O)ccc2nc(S)oc2c1 c1(C(N2C(C(=O)NCc3ccc(C)cc3Br)CC(C)C2)=O)nc2ccccc2[nH]1 C1(C)(CCn2cc(C(CC(C)C)C3CC3)nn2)CCC(C)(C)CC1.C1(CNC2CC2)CC1 c1(C(N2C(C(C)NC(CSCCOC)=O)CCC2)=O)cnc2ccc(F)cn12 C1(C(=O)N(CCCNC(c2cc[nH]c2C)=O)C2CC2)(OC)CCCOC1 C1(N(C(=O)CSc2nncn2C)C)CN(C(c2cc(C(F)(F)F)on2)=O)CC1O c1(Nc2ccc(OC(C(F)(F)F)(F)F)nc2)cccc2ccoc12 CCCC(C)CCN=c1[nH]c(N2CCC3(CC2)CN(C)C3)nc2c1CC(C)CC2 c1(CC(=O)OC)ccc(CNC(C2(C#N)CC2)Cc2nnnn2C2CCCC2)o1 CC(C)(C#N)CCCC(=O)N1CCC2(CC2)CC1C(N1CCC(C2CC2)CC1)=O c1(NCC2(CCC)CCC2)cc(NC(C)CC2CCCN2C)nc(C(C)C)n1 N1(C(C2CCN(S(C(C)C)(=O)=O)CC2O)=O)CCC2(CC1)OCC(C)(C)CO2 c1(OC)cc(C(N2CC(CNC(=O)Cc3nccn3C)C3(CC3)C2)=O)cnc1O C(=O)(N=c1cc(Cl)c(C#N)c[nH]1)C1CC2(C(CNC(=O)OC(C)(C)C)C2)C1 CC1CCC(O)CN1C(=O)CC1(NC(C2CC(C)(C)C2)=O)CC1 C(C(O)CC(=O)NCCN1CCCCC1=O)NC(CCC1(C)CC1)=O C1(NC(CNC(C)=O)=O)CCS(=O)(=O)C12CN(C(c1cc(Cl)cc(Cl)n1)=O)C2 C1(=CC(=O)N(C)CC2(NC(C(c3c(C)cccc3)C)=O)CC2)CCC(C)(C)CC1 N(C(=NCC#Cc1cnn(C)c1)NC1CC1)CC1(Cc2c(C)cccn2)CCC1 N1(C(C2(c3ccc(F)cc3)CC(C=O)C2)=O)CC2CN(CC(=O)NC)CC2C1.C(=O)O C(=O)(C1OCCc2c(O)cccc21)NC1(C)CC(NC(c2cc(C)nn2C)=O)C1 N(C(=NCCCSC(F)(F)F)NC1CCS(=O)(=O)C1)C(C(C)C)C C1(CNC(c2cc(CC)no2)=O)CCCCCN1C(C1CC(C(F)F)C1)=O c1(OC)ccnc(-c2cn(C(C)C(=O)NC(c3cnc[nH]3)C)nn2)c1 Cc1nc(C(=O)NCC(O)CCNC(=O)COc2ccccc2O)c(=O)[nH]c1C n1(-c2scc(N(C(c3ncccc3Cl)C)C)n2)cnc2ccccc2c1=O CC1CCOC1CNC(=O)C(C)(C)NC(=O)Cc1ccsn1 C(=O)(CCCC(=O)NC1CCCCN(C(c2c(F)ccnc2Cl)=O)C1)NCCC c1(C(=O)OC)sccc1S(=O)(=O)NCC1C=CCN1C(c1cc(Br)cnc1F)=O c1(C(N2C3CN(C(c4sccc4Br)=O)CC2C3)=O)cnc2ccoc2c1 C1(C(=O)NCCC2CCCN2C(C2CC2C(F)(F)F)=O)COCCC1(F)F C(=O)(CCC(F)(F)Cn1cc(CC(C)O)nn1)NC(C(C)C)C(=O)NCCO N1(C(C(=O)NCC2CC2)=O)CCn2c(CNC(C3(Cl)CC34CCC4)=O)nnc2C1 C(N=c1[nH]c(=NCCC2CCCC2O)c2ncccc2[nH]1)c1cnn(C)c1Br c1(C(N2CCCC(CCCCNC(CNC(C)=O)=O)C2)=O)cc(C)c(O)c(N)c1 c1(C(N(CC(C)NC(=O)CCCc2cnn[nH]2)C)=O)cc([N+](=O)[O-])cn1C c1(C(N2CCN(C(c3cnc(C)[nH]3)=O)C3C2C3)=O)ccc([N+](=O)[O-])c(Cl)c1 N1(C(CC(CC)(F)F)=O)CC2(CC(C(=O)NCc3cc(C)on3)CO2)C1 N1(C(C(CCCC)O)=O)CCCC2(CCN(Cc3ccc(S(C)(=O)=O)o3)C2)C1 C1(C(N2CC3(CN(C(c4ncc[nH]c4=O)=O)C3)C2)=O)CCc2cc(F)ccc2O1 c1(C(C)=O)ccc(O)c(C(N2CC3CC3(C(N3CC(C)OC(C)C3)=O)C2)=O)c1 c1(OC)cc(C(=O)NC2CCCN(C(c3cccnc3O)=O)C2)sc1Br C(C(F)(F)CCC(=O)NC(P(C)(C)=O)c1ccccc1)n1cc(CN(C)C)nn1 C=CCN=c1[nH]cc(C(N2CCCC(NC(=O)C(COC)N(C)C)C2)=O)s1 C(=O)(C1CCCc2nnn(C)c21)NCC1C(CC)CCN1C(=O)C1=C(C)OCC1 N1(C(c2c(C)cn(C)c2)=O)CCCC(C)C1CNC(=O)CCc1ccccc1Cl C(=O)(CCC(N)=O)N(C1CCN(c2ccccn2)CC1)C C(CCCCC(=O)N(C1CCCCC1)C)N(C(C(C)=C(C)C)=O)C N1(C(C2C(CC)N(C)CC2)=O)CCC(C)(NC(C2CCC2(C)C)=O)CC1 N1CCCC(F)(F)C1.c1(C(=O)OCC(=O)Nc2c(CC)cccc2)ccc(Br)c(Cl)c1 C(=O)(C(C)CCCC(C)C)N1CCC(COC)(NC(=O)Cc2ncoc2C)CC1 C1(C(=O)NC(C)(CO)C2CCCC2)CCN(C(=O)C=Cc2cccnc2)CC1O Cc1ccc(Cl)c(OCC(=O)N(C2CCN(C(c3ccc(F)c(C)c3)=O)C2)C)c1 c1(C(N2CCSCC2CCNC(C2CC(N3CCCC3)C2)=O)=O)ccnnc1Cl c1(C(=O)OC)cc2c(NCCCCC(C)NC(C3CC3C)=O)ncnc2[nH]1 C(C(O)CN=c1ccc2ncc[nH]c-2n1)NC(c1c(CC)c(CC)on1)=O C1(NC(C(C)NC(CC)=O)=O)CN(C(c2ccnc(C3CC3)c2)=O)CC1(C)C C1(O)(CNC(C2(C)CCCCC2)c2n(CC)nnn2)CC2CCC1O2 C1(NC(c2cnn(CCCC)c2C)=O)CC2(C1)CN(C(c1occc1CC)=O)C2 N1(C(CC(CC)C)=O)CC=C(C(=O)NC(C)(C)CNC(N)=O)C1 c1(NC(=O)NCCCc2nc(C)sc2)cc([N+](=O)[O-])ccc1COCC(F)(F)F C1(NC(CCC(=O)NC)=O)CC2CCC(C1C)N2C(C1(CC2CC2)CC1)=O CCC(C)(C)CC(=O)NCC1(F)CCC(CNC(c2cn3c(n2)SCC3)=O)C1 c1(CC(=O)NC(C(C)(C)C)CNC(C2COC(=O)N2)=O)noc2cc(F)ccc12 Cc1cn2c(n1)CC(C(N1CCCC1C(C)NC(=O)C(N1CCOC1=O)C)=O)C2 C1(C=O)Cn2c(C)nnc2CN1C.C12(CC=C)CN(C1)N(C)CCCC(=O)N2 C1(C(=O)OC)CC(CN)CN(C(=O)COc2cc(C(C)(F)F)ccc2Cl)C1 Cn1cnc2[nH]c(C(=O)NC3CCC(NC(=O)CC4(C)CC4(F)F)C3)cc12 c1(C(C(=O)OCCC(C)(F)F)O)cccc([N+](=O)[O-])c1.c1(O)cccc(F)c1 c1(SCc2ncon2)c(C(=O)NC2(c3ccncc3)CC2)sc2ccccc12 C=CC(C)(C)CC(=O)N1CC2(CNC(c3ncsc3C(C)C)=O)CC1CO2 c1(C(=O)OC)ccc(NC(c2ccccc2)C2CC(=C3CC3)C2)cc1 C(=O)(CCC(CC)NC(=O)CC1(C)OCCO1)NCC1(CCC)CCC1 C1(CC(=O)NC(C)CCNC(C2(C)CC2)=O)(C(=O)OC)CCCCC1 C1(C(C)NC(C2CCN(C(c3cocn3)=O)CC2)=O)COC2CN(CC3CC3)CC12 C1(NC(CCOCC#C)=O)CN(C(=O)CC2CC(O)C2(C)C)CC(C)(C)C1 C(=O)(CCN=C(NCc1ccc(Br)c(C)c1F)NCC(C)COC)NC C(=O)(C(C)Cn1cccn1)N(CCOCCCNC(C1C(C(=O)OC)CC1)=O)C Cc1ncc(NC(C2COCCN2C(=O)CCc2ccncn2)=O)cc1Cl C1(OC)CC(C(=O)NC(c2ccncc2F)C)N(C(=O)Cc2cnns2)C1 CN1CCCC(CCCC(=O)NCC2CC(n3cc(CC(C)(C)O)nn3)C2)C1 c1(C(=O)NC(CCC(=O)NCCOC(C)=O)(C)C)cc2n(n1)CCC2 c1(C(C)=O)cnc(NC(N2CCCCC2C2CCNC2=O)=O)c(Cl)c1 c1(C(=O)NC2CC(N(C(=O)C(F)=CCCF)C)C2)ccnc(OC(F)F)c1 Cc1nc(Cl)ccc1NC(=O)C(C1CCN(C(=O)CC2NC(=O)NC2=O)C1)F C1(NC(c2c(CCC)occ2)=O)CCCCC1NC(=O)C(n1cc(C)cn1)C N1(C(C=CCN(CC)CC)=O)CCCC(C(=O)NCCOC2CCC(O)C2)C1 CC1CC(C(=O)NCC23CC(CN2C)C3)CN1C(=O)C=Cc1ccsc1 c1(CSC)cccnc1C(=O)NCC(C1CC1)N(C(=O)C(C)c1cc[nH]n1)C CC1CCN(C(C2CCc3ncnn3C2)=O)CCN1C(C1CC2(CCC2)C1C)=O C(c1c(Cl)cccc1Cl)=CC(N1CCC(CNC(COCC=C)=O)C(O)C1)=O C=CCC(C)(C)CC(=O)NCc1nc(-c2ccc(Cl)cc2Cl)cs1 c1(NC(COC(C2C(C(C)C)OCC2)=O)=O)nc2c(s1)CN(C)CC2 Cn1c(=O)nc(O)c2nc(CCCNC(C3CC(O)CN3)=O)[nH]c12 c1(OC)ccc2nc(CN3CC(C)(c4ccccc4)C3)ccc2c1 C(C(F)(C(=O)N1CCS(=O)C(C)C1)C(C)C)NC(C(C)(C)OC(C)C)=O c1(C(=O)NCCC(CC)(CC)NC(=O)CCS(C)=O)cccc2c1OCC(=O)N2 N#CC12CCC(C(=O)OCCC3CCCCO3)(CC1)CC2 C1(NC(c2c(OC)cncc2)=O)CN(C(=O)CC23CCCC2C3)CCC12CCC2 C1(NC(Cc2nccc(OC)n2)=O)CC2(CCN(C(C3(C4CC4)CCC3)=O)C2)C1 CC(CO)C(=O)NC1CC(N(C(=O)CNc2ncccn2)C)C1 CC1(C(=O)NCC2CC23CCOC3)CCCN1C(c1ccc(CO)cn1)=O O=C(CN1C(=O)Cc2cc(F)ccc21)Nc1ccc(F)c(I)c1 c1(NC(C2COCC(C)O2)=O)ccc2c(c1)CCS2(=O)=O CC(CC(C)(C)C)C(=O)N(CC(C)C(=O)NC(C)(C)C)C c1(C(C(=O)NC(CNC(c2ccc(C)[nH]2)=O)(C)C2CC2)C)ccccc1C N1(C(C2CCN(CC(C)(C)O)CC2)C=O)CC(O)CC1c1ccc(F)cc1.CO c1(C(=O)NCCCC(C)NC(Cc2cccc(C#C)c2)=O)cc(S(C)(=O)=O)co1 c1(CN2CC(CN(CCNC(=O)C(=O)Nc3ccccc3)C3CC3)C2)cccnc1 C1(C(C)C)CN(C(C2CC3CCC2O3)=O)CCN1C(c1ccc(C(N)=O)cn1)=O N1(C(C(C2CCN(C(c3ccnc(C)n3)=O)CC2)C)=O)CCCC(C#N)C1 C1(C#CC(=O)NCC2(C)CCC(NC(C3(CF)COC3)=O)C2)(CC)COC1 C1(NC(C(C)(C)C)=O)CN(C(=O)CCN(c2cnccn2)C)Cc2nccn2C1 C(CC(C)CCNC(c1ccc(-n2cccn2)cc1)=O)NC(COCCC#C)=O c1(OCCCC)ccc(C(=O)NCC2CCN2CC2CC(C)CO2)cc1 c1(N(C(CN(C(C(C2CCOCC2)OC)=O)C2CCCC2)=O)C)cccc(C)c1C C1(CCC(=O)NC(C(C)NC(C)(C)C)C)CCCCN1C(c1cccnc1)=O N1(C(c2c(CC(C)C)nc(C)s2)=O)CC2CC1CCC2NC(=O)CC1OCCC1C N1(C(c2n(C=C)ncc2)=O)CC(=O)NCC1C(=O)NCC1CCCO1 c1(CC(=O)NC2COCC2NC(C2(CF)CC2)=O)cnc(C(F)(F)F)s1 N1(C(CC=C)=O)CC(C(=O)Nc2cccc(OCC)n2)CCC1C C1(C(C)(C)C)CN(C(=O)Cc2ccc(Cl)cc2)CCN1C(c1cccc(O)c1Cl)=O c1(CNC(c2cc(Br)n(C)n2)c2n(CCC)nnn2)cccc(C(N)=O)c1 Cc1nc2ccc(F)cn2c1OCc1ccco1 C(c1ccccc1)=C(OC)C(=O)NC1CCC1NC(=O)CCCc1ncco1 C(=O)(C(C)(C)CC(C)C)NC1CN(C(CNC(c2c(C)occ2)=O)=O)CC(F)C1 c1(OC)ccc2[nH]c(=NCC=CC3CC3)[nH]c(=NCC3CC(C)CC(C)C3)c2c1 Cc1ccn(CC(N2CC(NC(=O)CC3CCC(C)(C)C3)C2)=O)c(=O)c1 c1(OC)ncc(C(=O)NCCCC(c2ccccc2)NC(C2CCCOC2)=O)s1 c1(C(N(C)CCNC(=O)C(C)(C)C2(C)CC2(F)F)=O)cnc2cn[nH]c2c1 Cn1cc(C(F)=CC(=O)NCC2CCCC2NC(c2cc(=O)cc(Cl)[nH]2)=O)cn1 C1(OC)CC(NC(C2CC2C)=O)CN(C(=O)CNC(c2cccc(Cl)c2)=O)C1 c1(C(=O)NCCC2CCN(C(CCc3cn(C)nn3)=O)CC2)cc(O)cc(O)c1 CC(CC(=O)NCc1ccsc1)C(C)(C)NC(=O)COCC(F)F c1(C(=O)NCCC(C)NC(=O)CC2CCC(C)(C)C2)coc2cc(F)ccc12 c1(C(=O)NC(C(=O)NCC2(C)CC(C)C2)CN(C)C)ccc(F)cn1 C1(C(N2CCCC(C(C)NC(c3ccc(OC)cc3)=O)C2)=O)CN(C)CCN1C C1(CNC(COC(CC)(C)C)=O)CN(C(c2ccnn2CC(F)F)=O)CCCO1 CC1C(O)CCCN1C(c1nc(C(N2CCC(OC(C)(C)C)C2)=O)cs1)=O N1(C(C2(N(C)C)CCC2)=O)CCCC(CCC(=O)NCCc2nnc(O)n2C)C1 c1(C(N2C(CNC(c3c(C)ccnc3)=O)CCCC2)=O)coc2c1C(=O)CCC2 C1(C)(C(=O)NCC2(O)CCCN(C(c3c(CC)scn3)=O)C2)CCC(F)(F)CC1 CCC(CNC(=O)CC12CCCC1C2)(CC)C(=O)NCC1(C)CC2CC2C1 C123CC(C1)(C2)N3.c1(C(N2CC(NC(CNC=O)=O)C2)=O)csnc1Cl c1(OC)c(C)cc(C(N2CC(NC(=O)CCC3CCCO3)C(O)C2)=O)cc1C CC(C)CCCCCC(=O)N1CCN(C(=O)C(=O)N=S(C)(C)=O)CC1C(C)C N#Cc1sc(=NCC2CN(C(c3nc(-c4cccnc4)no3)=O)CCO2)[nH]c1Cl C(CCC(C(=O)NCCC(COC)NC(C1CC2C=CC1O2)=O)N(C)C)OC C1(C(=O)NCC(C#C)CC)CCN(C(=O)C2OC3CCC2C3)O1 Cc1cc(C(=O)NC2(CS(C)(=N)=O)CCCC2)c(C)o1 N1(C(C2C(=C)C2C(=O)OC)=O)CC2(CO)CC1(C(N1CC=CC1(C)CO)=O)C2 CC1c2ccccc2OC1Cc1cc(N)ccc1C(=O)N.C(CO)N C(=O)(CC(F)(F)C(C)C)NCC1(C)C(NC(c2ccc(COC)s2)=O)CCC1 N1(C(CCCOCC)=O)CCC2CCCC12C(=O)Nc1c(C)nc(O)nc1O Cc1cc(SCC(=O)NC2CC(O)(CNC(C3OCCOC3C)=O)C2)cc(C)c1 C1(CNC(c2nncs2)=O)CC2CC2N1C(c1cc(-c2ccc(Cl)cc2)cs1)=O c1(C(=O)NC(C2(O)CN(C(c3cnccn3)=O)C2)C)cc2c(nc1O)CCOC2 CCCC(O)CC(=O)NCC1CCCCN1c1cc(OC)nc(OC)n1 N1(C(CC(CCC)C)=O)CC2CCCCC2(CNC(c2ccc(CF)cc2)=O)C1 CCCCC(C)CCC(=O)N1CC(O)(CCNC(C23CCOC2CCOC3)=O)C1 c1(CC(C(=O)N2CC(CC(C)NC(C(C=CC)O)=O)C2)C)ccccc1C C1(NC(CC=CC=C)=O)C2CCN(C(c3cnc(N(C)C)s3)=O)C12 N12CC3CN(CC3C1)C1CCCN(C1=O)C(=O)C2.C#Cc1c[nH]nc1NC(C)=O CC(C)(C)C(=O)C(=O)NC1CCCC(CC(N2CC(c3cc(Cl)no3)C2)=O)C1 Nc1cccc(C(=O)NCC(CNC(c2nocc2Cl)=O)C(F)(F)F)c1Br c1(C(N(CCNC(C(C)CF)=O)C)=O)cc(N=S(C)(C)=O)ccn1 C(=O)(C(CO)C(C)(C)C)NCC(C)NC(CN(S(CCCC)(=O)=O)C)=O NS(=O)(=O)N1CC(C(=O)NCCC2COCCN2C(c2cn(CCO)nn2)=O)C1 c1(SC)ccnc(C(=O)NCC2CC(NC(C3CCC3)=O)CCO2)n1 Cc1cccc(F)c1NNC(=O)C1CCCNC1C c1(N(C)CC2OCCN(C)C2)nc(N2CCC3(CCC3)CC2)nc2c1CCC2 CC#CCC(C(=O)NC1CCN(C(=O)OC)C1)NC(=O)COC1CCCCC1 C1(C(N2CC3C(C(N4CCN(C(C)C)CC4)=O)C3C2)=O)(CC)CCNC1=O c1(C(N2CCCC(CNC(CSCC#C)=O)C2)=O)cc(F)cc2cnccc12 c1(C(=O)NCC2(C)CN(C(c3ccc(O)nc3)=O)C2)ccc(C#N)c(C(F)(F)F)c1 N1(C(C(C)C2CC2)=O)CCC2(CCCC2NC(c2ccnc(F)c2)=O)CC1 c1(C(N2CC(CN(C(CC(=C)Br)=O)C)OCC2)=O)cnc2c(c1)CCCC2 C1(C(=O)NCCN(C(C23CCC2C3)=O)C2CC2)CCCOC1 C(=O)(C1CCc2c[nH]nc21)N1C(C(C)(C)C(=O)NCC2(C)CCCCO2)CCC1 c1(C(N2CCC(NC(CN3C(C)CCC3)=O)C(O)C2)=O)cc2cc(F)ccc2o1 c1(C(N(CCNC(c2cn(CC)nn2)=O)CC2(CO)COC2)=O)cc(Cl)c(Cl)s1 C1(CNC(C2CCCN(C(=O)C(F)(F)C(F)F)C2)C)Cc2ccccc2O1 n1(CC(=O)N(CCN(C(C2C(C)(C)C2(F)F)=O)CC)CC)cnc2cc(C)c(C)cc12 C(=O)(CC(CNC(c1ccnc(OC)c1)=O)OC)N(C(C)C(C)C)CC c1(OC)cc(C(N2CCC3CCC23CNC(=O)C=Cc2cc[nH]n2)=O)ccc1C#N C1(C)(C(=O)NC(COC)C2(C)CC2)C=CCN1C(=O)C(C)CC#N Cc1nn(C(C)C)c(C)c1C(=O)NCC(C)NC(c1c(Cl)nsc1Cl)=O c1(C(N2CCN(C(c3cc(C)sn3)=O)C(CF)C2)=O)ccc(O)c2c1CCCC2 N1(C(c2c(F)ccc(CC)c2)=O)CCC(N=c2nc(COC)[nH]s2)C1 c1(CCC(=O)N(CC(CN(C(=O)CCC2CCC2)C)O)C)ncc(C(C)(C)C)o1 [N-]=[N+]=NC1CCC(C(N2CC(O)(CCNC(c3scnc3Cl)=O)C2)=O)C1 c1(C(=O)NCC(CNC(C(C(COC)C)C)=O)C)cc(OC)nc2ccccc12 C1(C(N(CC)CC2CCC2)=O)CC=CCN1C(=O)CC1CCCN1C c1(NCc2cc(OC)nn2C)cc(=NCC2(C(C)(F)F)CC2)[nH]c(C)n1 C1(C(=O)NCC2(OC)CN(C(c3ccon3)=O)C2)C2CN(C)CC12 c1(CC2CCCN2C(=O)CCN2CCC(F)C2)ccccc1F.C12(CC1)C(=O)N2 C#Cc1cccc(C(N2CC=CC(NC(=O)CC3C(C)(C)C3(C)C)C2)=O)c1 N1(C(C=NOC)=O)CCC(NC(=O)CC(C)(C)O)C(C(C)C)C1 C1(OC)CCC2(C(=O)NCCC3CCN(C(C4SCC=C4C)=O)CC3)CC12 C1(CN(C(C2C(C(=O)OC)C2)=O)C)C2CN(C(=O)CCc3ccc(C)s3)CC12 c1(C(=O)NCC(C)(C2CC2)NC(CN(c2ccccc2F)CC)=O)cc(Cl)c(Cl)s1 c1(C(N2CC3(N(C(c4c(C)cccc4F)=O)CC3)C2)=O)ccc(S(C)(=O)=O)s1 C1(C(N(C2CC(C(=O)N(CC(=C)F)CC)C2)C)=O)CC2CCC2C1 c1(C(=O)NC2CC(C)(C(=O)NC(c3nc(C)[nH]n3)CO)C2)cccc(F)c1 C1(C)(C(=O)NCCN2CCN(C(C(CNCC)C)=O)CC2)CC(OC)CN1C CC1CCN(CC=C(Cl)Cl)CCN1C(c1ccc(Br)cc1I)=O Cc1cc(C(N2CC(CNC(=O)Cn3nnnc3C3CC3)C3CC23)=O)c(C)s1 N1(C(CCCOCC)=O)CCCC2(CCN(C(C3CC34CCCC4)=O)C2)C1 C1(CCNC(C(n2cnc(C#N)n2)C)=O)CSCCN1C(=O)CS(C)(=O)=O Cc1nc(C(=O)NC(CCN(C)C)C(=O)NC2CC2CCF)c(C)s1 C1(N(C(C=CC(C)NC(C2(COC)CC=CC2)=O)=O)C)CCN(C)CC1C C1(C(N2C(C3(NC(c4onc(C)n4)=O)CC3)CCC2)=O)CCCSC1C CC1CCC(CC(=O)N(C)CC2(CNC(C3(O)CCCC3)=O)CC2)CC1C C(=O)(C(C)CC(C)(C)C)N1CC(CCOC)N(C(=O)Cc2cncn2C)CC1 N1(C(C(C)NC=O)=O)CCC(CNC(=O)Cn2cnnc2O)C1(C)C CC1c2ccc(F)cc2CCN1C(c1cc(Br)no1)C(=O)Nc1ccccc1Cl N1(C(CCOC(C)C)=O)CC2(C1)CN(C(c1sc3cccnc3c1Cl)=O)CCO2 N1(C(c2c(CC)onc2C)=O)CCCN(C(=O)C(CC)CC(C)C)C(C)C1 C1(NC(C=C(C)C2CC2)=O)CN(C(c2ncoc2C)=O)CCC1C C1(C(C)C)CN(C(=O)CSc2ccc(C#N)cc2)CCN1C(C1CC1C(F)F)=O c1(C(N2CC(CNC(C3C(=C)CC3)=O)OCC2)=O)cc(C(F)(F)F)ccc1OC C12(NC(Cc3cn(CC)nc3)=O)CC1CN(C(=O)CC13CCCC1C3)C2 C#CCC(C)(CC)C(=O)N1CC(NC(=O)CSS(C)(=O)=O)C(c2nccn2C)C1 c1(CC(C(=O)OCC)NC(=O)C(C)CNC(=O)CC)ccc(O)cc1 C(=O)(C1=C2CCCN=C2NN1)NCCN(C)C(c1n[nH]cc1C1CCC1)=O C=C(C)CC(=O)NCCCCNC(C1SCCS1)=O CC1CN(C(=O)CCN2CCCC2=O)CC1NC(=O)C(C)Cc1ccccc1 C1(NC(C(COCC)C)=O)CC2(CCC(NC(c3cc(CC)no3)=O)CC2)C1 C12(C(N3CC(C)C(CNC(=O)C(C)(C)CN(C)C)C3)=O)CCCCC1OCC2 c1(Nc2ncc(CCNC(c3csc(C(=O)O)n3)=O)s2)nc2ccc(O)cc2o1 c1(C(N2CCCC(C(=O)NCC(=O)NC3CCC3)C2)=O)cc2ccsc2s1 C12(NC(C(C)SC)=O)CCCC1N(Cc1c(F)cccc1F)CC2 c1(C(=O)NCC(C)N(C(CC(C)O)=O)C)cccc(O)c1 N1(C(C(C=C)O)=O)CCCC(CC)(NC(c2cn(CCOC)nn2)=O)C1 C1(N(C(=O)CNc2cccnc2)C)CN(C(=O)COCC2CCCC2)CCO1 c1(C(=O)NCC(c2cn(C)nc2)C)cnn2ccc(Cl)c(F)c12 C(=O)(C(C)(C)C(=O)NCc1nc(C(N2CCC(C)C2CC)=O)c(C)o1)OCC Cc1cc(C)c(CNC(=O)NCCCNC2C=CCCC2)cn1 C(CC(C(=O)N1CCC(CN(C(=O)COCC(=O)OC)C)C1)NC(C)=O)SC C(C)(C)(CNC(=O)CN(C)C1CC1)OCCCNC(CNC(CC)=O)=O Cc1cccc(C(=O)NC2CCN(Cc3ccsc3C)CC2)c1F C(C1OCc2ccccc21)C=O.C1(C(C)C)CCCC(N)N1 C1(C(=O)NC(CC(=O)OCC)C)C(C)OCCN1C(=O)C(C(C)OC)OC c1(SCC)ccc(C(=O)N(C2CCN(C(=O)C(c3ccccc3C)C)C2)C)cn1 C(=O)(C(C)(C)CC(C)C)N(CCOCCN(C(c1ccc(SC)o1)=O)C)C C(c1ccc(C)cc1)=C(C(=O)N(CCOCCNC(C1(C(=O)NC)CC1)=O)C)C C1(N(C(=O)C(F)OC(F)(F)F)C)CCCN(C(=O)CC2(O)CCOC2)CC1 c1(N2CC3N(C(c4c(C)c(Cl)ccc4)=O)C3C2)ncnc2sc(C(C)C)cc12 C1(C(N(CC(=O)NC(C)Cn2cc(C)cn2)CCOC)=O)CCC(=O)N(C)C1 C(C)(C)(C(=O)NCCC(O)CNC(C12CCCC1C2)=O)OC(C)=O c1(C(=O)NC2(CO)CN(C(C3CCC(C)(O)CC3)=O)C2)cc2cc(F)cc(F)c2[nH]1 C1(C(=O)NC(C#C)C)CC(C)(C)CCN1C(c1ccncc1N)=O C1CCCC(NC(C)COC)C1.C1(OCC(=O)OCCC)CCOC1 C(=O)(C1CCCn2nccc21)NC1(CCNC(C(C)N(CC(F)(F)F)C)=O)CC1 Cc1oc(Cl)nc1C(=O)NCCCN(CCO)C(c1csc(C(C)OCCO)n1)=O Cc1cc(C)c(C(=O)NCC2(F)CC(CNC(c3c[nH]c(=N)o3)=O)C2)s1 Cc1cnc(C(=O)NCCC2(C(=O)NCC3(O)CC(C)(C)C3)CCCC2)cc1C C12CCC(C)(C1(C)C)C(=O)OC2=O.N1(CC)CCC(N=[N+]=[N-])C1 C(=O)(CCC(C)(C)F)N(C1CN(C(CC(C)Cc2cccs2)=O)C1)C C1(NC(C2CCCO2)=O)CC2CC1CN(C(c1cccnc1I)=O)C2 C(=O)(C#CC1CCCO1)N(C)CC1CCN(C(CC=C)=O)C1 C1(NC(CCNC(COC)=O)=O)CC2CN(C(c3ncc(C)cc3F)=O)CC2C1 N1(C(=O)C(O)C2CCC2)CCC(C2(NC(c3nncc(OC)c3)=O)CC2)C1 Cn1nccc1Cn1cc(CNC(=O)C(O)CC2CCOCC2)nn1 C1(COC)CN(C(C2CC3(C2)CC(C)C3)=O)CCN1C(C1CCN(C)CC1)=O c1(C(N2CCN(C(c3c(C)nco3)=O)CC2C(C)C)=O)ccc2c(c1)OCCO2 N1(C(CC(=O)OCCC(C)C)=O)CCC(C(F)(F)F)C(NC(C2(SC)CC2)=O)C1 N1(C(C(C)n2ccnn2)=O)CC2(CCC2NC(C2(C(N)=O)CC2)=O)C1 n1(CC(=O)NC2(CCNC(CN=S(C)(C)=O)=O)CC2)ccc2nc(O)nc(O)c12 C12(NC(Cn3c(=O)sc(C)c3C)=O)CC(C)(C1)OC21CCN(C(=O)CCF)CC1 c1(C(=O)NCCN(CCOC)C(c2ccc(C)nc2)=O)c(C)nn(CC(C)C)c1Cl c1(CNC(=O)CC2(O)CCCOC2)ccc2c(c1)CCC2NC(=O)C1=COCC1 C1(CC(=O)N(CCC(N)=O)C)CC(C)(C)CN1C(=O)C1=CCCC1 C1(N(C(c2ccc(CC)[nH]2)=O)C)CC2CCC(C1)N2C(c1coc(C2CC2)n1)=O C1(NC(CCCC#C)=O)CCCC(C(=O)NCc2ccc3c(c2)CC3)CC1 C1(NC(C2C(OCC)CC2)=O)CN(C(=O)CCCC2CCCC2)C2CCCC12 c1(CC(N2CC3(CCCC(CNC(C)=O)O3)C2)=O)[nH]c2c(c1C)CCCC2 CCCCC(C(=O)OCC(=O)NC)N(C)C.c1(CC)ccc(OCC)cc1 c1(CNC(C2CCCC(=O)N2)=O)nc(CNC(C2CC3(CCC3)C2)=O)cc(O)n1 C(CC(O)C(=O)N(CC(C)O)CC=CC(=O)NCC(C#N)CC)SC C(=O)(C(O)CCCNC(c1cc2occc2[nH]1)=O)N1CCN(CC#C)C(=O)C1 C12(CNc3cc(C)c(C(=O)NC4CC4)cc3)CN(C(C)C)CC1CS(=O)(=O)C2 n1(CC(C(=O)O)NCCSC)nnc2ccccc12 C1(C)(C(N2C(C)CCC(OC)C2)=O)CC2(C1)CC2(F)F N1(C(C(CC)C)C(=O)Nc2ccccc2)Cc2ccc([N+](=O)[O-])cc2C1 c1(OC)cccc(N(C(C(=O)NC2CCC2)c2cnn[nH]2)C)c1 N1(C(c2nc(CC)[nH]n2)=O)CCC(=CCNC(=O)C(C)CN2CCOCC2)CC1 C1(CC(F)(F)F)(C(=O)OC2CCN(Cc3ccccc3)C2)CCCCC1 C1(C(=O)NCC2(c3cccc(OC)c3)CCC2)CCc2nc[nH]c2C1 c1(N2CCN(C(C=CC=CCC)=O)CC2)cc(=O)n2cc(Cl)ccc2n1 N1(C(CCCN(C)C)=O)CC(CNC(C2CC2CN(C)C)=O)C(F)(F)C1 c1(C(=O)NC2C(NC(C(CCSC)OC)=O)CCCC2)cnn2ccsc12 C123CCC1CN(C2)C3=O.C1(NC(c2ccc[n+]([O-])c2)=O)CCN(C(=O)C2CC2)CC1 N1(C(c2c(C)cc(F)s2)=O)CCCN(C(c2cnc(C(C)C)[nH]2)=O)CC1 N1(C(C2C(C(C)NC(C34CCC(C3)OC4C)=O)C2(C)C)=O)C2CCCC1CN(C)C2 C(c1c(Cl)cccc1Cl)=CC(=O)NC1CN(C(C2(C(C)N(C)C)CC2)=O)C1 C=CC1(CC(C(CCNC(C)C)=O)=O)CN(C(=O)CCc2ccccc2F)C1 N1(C(C(C)C2CCC2)=O)CC(=O)NCC1C(=O)Nc1cccc(F)c1 C1(C(=O)OC)(CNC(=O)Cc2cncs2)CN(C(=O)C(C)Cn2ccnc2)C1 c1(C(N2CCC(O)(CNC(COCCCOC)=O)C2)=O)cnn2c(=N)[nH]cnc12 C1(OC)CN(C(=O)Cc2cnsc2)CC1NC(=O)CC1CC(F)(F)CO1 C(C(CCOC)NC(C1CN(C)C1)=O)NC(C1C(CCC)C1)=O O=C(NNc1c(Cl)cccc1Br)C1CCC12CC2 c1(C(=O)NC23CC(CNC(c4onc(CC)c4C)=O)(C2)C3)ccc(C)c(N)c1 C=C1Cn2c(C(=O)NC(CCN(C(=O)C(C)(C)SC)C)C(C)(C)C)nnc2S1 C1(NC(C2CCC(=O)NC2)=O)(CNC(c2ccc(Cl)cn2)=O)CCCCCC1 c1(C(=O)NC(C2CC=CCC2)C(=O)NCC2CC(F)(CF)C2)cnc(Cl)s1 C1(NC(c2cc[nH]n2)=O)C2CCN(C(c3cn(CCC4CC4)nn3)=O)C12 N1(C(c2cn(C)c(=O)nc2O)=O)C2CCC1C(F)C(NC(=O)CC1(CO)CC1)C2 Cc1cccc(O)c1NC1CN(C(c2cc(C#N)n(C)n2)=O)CC1C CC1(C(=O)N(C2CCNCC2)CC2CC2)CCOC1 O=C(C1=CCS(=O)(=O)C1)NCC1CC2CN(C(=O)C=C3CCCCC3)CC12 C(CC(C)(C)CC(=O)NC(C)(C)CC=CC(=O)N(C)CC1(C)CCC1)OC N1(C(C2C(C)C2C)=O)CC2CCCN(C(C3CCC(=O)N(C4CC4)C3=O)=O)C2C1 C1(CNC(C(c2cn(C)nc2)O)=O)CN(C(=O)Cc2ccno2)CCO1 c1(C(=O)NCC2C(NC(Cc3c(C)occ3)=O)CCC2)ccc(N)c(F)n1 c1(C(=O)OC)ccc2c(-c3ccc(N(CCO)C(C)C)nc3)n[nH]c2c1 CCC(C)(C)CCCC(=O)N1CCCCC1CCNC(=O)CCCF n1(C(C)C)cnc2c(NC(c3nc(CO)cs3)C)[nH]c(=NC(C)c3cnc[nH]3)nc12 c1(C(N2CCC(NC(c3ccc(C)c(C)n3)=O)C2)=O)ccc(C#N)cc1Br c1(C2CNC(=O)CC(=O)N2C)ccc(F)cc1.C(=O)(COC(=O)CO)NC1CC1 c1(C(N2CC(CCCC)N(C(C3C(C)C3C)=O)CC2)=O)ccc2c(c1)CC(C)O2 C(C#Cc1cccnc1)NC(C1C(NC(c2ccc(F)c(F)c2)=O)C=CCC1)=O Cc1nccc(C(=O)NC2(C(=O)NCC3CCCOCC3)CC2)c1C c1(C(=O)OCC)ccc(S(=O)(=O)N2CCC(OC)C2N(C)C)c(C)c1 C1(CNC(C2CC(Sc3ccc(-c4ccc(Cl)cc4)cc3)C2)=O)CCCCC1(F)F N1(C(c2nc(C(C)C)sc2)=O)CC(NC(=O)CC2CCOC2C)CCC1C C1(CCNC(CSCC)=O)CN(C(=O)COC2CC2)CCS1(=O)=O c1(C(=O)NC2CC(OC)CN(C(C3CCC(=O)NC3C)=O)C2)cc(C)cc(O)n1 c1(C(=O)NCC2CN(C(c3c(C)nco3)=O)CC2C)ccc2c(c1)NCCC2=O Cc1csc(C(N2CCCC2CCC(=O)NCCOCCO)=O)c1 c1(C(=O)NCC2C(NC(C(C(C)(C)O)F)=O)CC2)cc(N)c(F)cc1F C12(CCNC(c3c(OC)c[nH]n3)=O)CCC1CN(C(c1cc(C3CC3)cs1)=O)C2 CCCC(C(=O)NCCn1cc(C(=O)NC(C)(COC)C(N)=O)nn1)OC CCCCS(=O)(=O)CC(=O)NCC1CN(C(c2ccoc2Br)=O)C2CCCCC12 c1(CN(C(=O)NCc2ccccc2)Cc2ccc(C)cc2)ccc2[nH]ccc2c1 c1(CCC)cc(C(=O)NC2CC(OC(C)C)C2(C)C)c(C)o1 N(C1CCCc2ccc(C(F)(F)F)cc21)Cc1ccc(F)cc1.n12ccc(n1)C2 c1(C(N(C(CC(F)F)C(=O)NC2C(C)CCC2C)C)=O)ccc(=O)n(C)c1 Cc1cc(O)ccc1-c1cnc(C2CN(C(C3CCC(=O)NC3)=O)C2)nc1 n1(CC)cc(S(=O)(=O)N2CCCC3(CC3)C2)nn1 CC1(C)CC(CC(=O)NCC(F)OC(F)F)CN1C(=O)C=CC(F)(F)F.C(C)(C)C C(CCCCNC(=O)C(CN(C)C)C(C)(C)C)N(CC)Cc1ncnn1CC1CC1 N1(C(CCCC2CC2)=O)CCCN(C(=O)C(C)(C=C)CCNC(C#C)=O)CCC1 CCC(C)C(O)C(=O)N1CCC2C(NC(=O)CC(Cc3ccccc3)CC)C2C1 N1(C(C(C=CC)O)=O)CCN(C(c2cnc(CC(C)C)[nH]2)=O)CC1C(C)(C)C C1(NC(C=Cc2n(C)cnc2)=O)C(CNC(=O)CC2CC=CC2)CCC12CCC2 C1(CCC)CN(C(c2cccs2)=O)CC1C(=O)NC1CCCC1F N1(C(c2c(C)scn2)=O)C2CCC1C(NC(c1ccc(OCCF)cc1)=O)C2 C#Cc1cc(C(=O)NC2(C)CC(NC(C3CN(C(C)=O)C3)=O)C2)ccc1C CCC(C)C(CC(=O)NCC1CCCCO1)NC(=O)CCCc1cc[nH]n1 c1(C(=O)NCCc2cc(C)no2)ccc(C(C)NC(COC(CC)C)=O)cc1 C(CC(C(=O)N(CC(C)(C)OCCO)CC)OC)NC(c1cnc(CC)o1)=O N12CCOCC(C1)NC2=O.C1(CC(=O)NCC=C(C)C)(OCC(C)C)CCC1 N1(C(C(C(=O)OC)OC)=O)CC2(CCC2)CC1CNC(=O)C=Cc1cccnc1 C1(C(N2CCC(NC(=O)NC)C2)=O)CCC2(CC2)N1C(=O)Cc1cn[nH]c1 C(=O)(CCCCC(N)=O)NC(C(=O)NCC(C)CC1CC1)CCN1CCC1 C1(C(=O)NCC(CO)NC(c2conc2C2CC2)=O)(C2CC2)CCCCC1 S(=O)(=O)(c1c[nH]ccc1=NC(C)CCCCCCCO)N1CC(C)=C(C)CC1 c1(C(=O)NC2CN(C(C(C)Sc3nncn3C)=O)C2)cccc2ncnc(O)c12 Cc1cc(C(=O)NCCC2CN(C(C3CC34CC4)=O)CCO2)cnn1 c1(-c2c(F)ccc(C3(NCc4cc(C)ncc4)CC3)c2)ccc2oc(C)nc2c1 C(C(C)CC(F)F)NC(C1(N(C(Cn2c(C)ccn2)=O)C)CC1)=O c1(C(C)O)ccc(C(N2CCCC2CN(C(=O)C(c2ccccc2)F)C)=O)cc1 c1(NC(Cc2cc(C)sc2)=O)ccc(C(C)(C)C)cn1.C12CCC(C1)NC(=O)N2 C1(NCC(c2cccc(C(F)(F)F)c2)(C)O)CCCC1(F)F C1(NC(C2CCSC2)=O)Cc2n[nH]cc2C(C(F)(F)F)C1 O=S(=O)(c1nc(NCc2ccccn2)ccc1Br)NCC CC1=C(C(=O)N2CCCC(O)(CNC(=O)CC(C)CN(C)C)CC2)C(C)(C)CCC1 C1(C(N2CC(NC(C(C=C)(C)O)=O)C2)=O)CCn2cc(C(F)(F)F)nc2C1 CCCC(C)CCCC(=O)NCCOCCCN(C(=O)CCC1CCC1)C C1(C(=O)NCC(CNC(Cc2nc(C)oc2)=O)F)CCCS(=O)(=O)C1 C1(NC(c2c(C)c(C3CC3)on2)=O)CC2CC(C1)N(C(c1csc(F)c1)=O)C2 Cc1cc(O)nnc1C(N1CC(NC(C2CCC(C(F)(F)F)C2)=O)C(F)C1)=O n1(CCC)cc(C(=O)NCC2CC2NC(C2(c3ccc(Cl)cc3)CC2)=O)c(C)n1 CC(C)CC(O)C(=O)NC(CC(=O)NCC1CC=CCC1)C(F)F c1(OC)ccc(C(N2CC3CN(Cc4ccccc4Cl)C3C2)=O)cc1OC C1(C(=O)NC23CC(NC(C4CC(=O)CC45CCC5)=O)(C2)C3)CCC([N+](=O)[O-])CC1 C1(NC(C=Cc2ccc(C)o2)=O)CC1C1CCN(C(=O)C(O)CC2CC2)CC1 CCC(C(=O)NC(C1(O)CN(C(=O)C=CC(F)(F)F)C1)C)OC1CCCCC1 CN=c1[nH]cc(C(N2CCC(C(C)C(=O)NC3CCC(C)(C)C3)CC2)=O)o1 C(C(C)C(=O)N1CCC1C(=O)NCCCc1nncs1)OC C1(CNC(C(C)C(C)(F)F)=O)CCCC2(CN(C(=O)CCCC#N)C2)O1 C1(COC)CN(C(c2ccnc(CO)c2)=O)CCN1C(C1CCC(C)CC1)=O c1(C(=O)NC2C3(CCN(C(C(C)=C(C)C)=O)CC3)CC2)cc2c(cn1)OCCO2 C12(NC(=O)C=C3CCCC3)CCCC1N(C(c1ccc(Cl)cc1F)=O)CC2 C1(CNC(C=NOC)=O)CN(C(C2CC(n3ccnn3)C2)=O)CC(C(F)(F)F)O1 N1(C2CCN(C(C(C)C3CC3)=O)C2)CCN(C(=O)CCOCCN(C)C)CC1 N1(C(c2ccc(OC)nc2)=O)CCCN(C(C2(C)CC(C)OC(C)C2)=O)CCC1 O=C(NOCc1cn(C2(C3CC3)CC2)nn1)C(C)CC1CC(F)(F)C1 c1(C(C(=O)NC(C)CNC(=O)C(F)=CCCF)(C)F)ccc(F)cc1 C1(CNC(C2(C(C)NC(C3CC(C)(O)C3)=O)CCC2)=O)CC12CCC2 N1(C(Cn2ncc(C#C)c2)=O)CCCCC(NC(=O)C(C=C)CC)C1 Cc1ccc(C(=O)NCC23CC2CN(C(c2ccccc2O)=O)C3)cc1Cl N1(C(=O)NCCc2c(C)non2)CCN(Cc2ccccc2)CC1C N(C1CCCOc2cc(Cl)ccc21)C(C(=O)N(C)CC1CC2CC2C1)=O N1(Cc2c(OCOC)cc(Br)cc2)Cc2[nH]nc(-c3cnn(C(C)=O)c3)c2C1 C1(C(N2CCN(C(c3c(OC)ccs3)=O)CC23CC3)=O)CNC(=O)CC12CCC2 C1(CNc2cc(Nc3[nH]cc(NC)c3)ncn2)CCOC(C)(C)C1 C(c1cccs1)=CC(=O)NC1(CCNC(C(C)O)=O)CC1 Cc1sc(Cl)c(C(N2CCSCC2CCNC(=O)CCCC(F)F)=O)c1C N1(C(C(CCOC)C)=O)CCC(C)(NC(=O)C=CC2CCOCC2)CC1 N1(CCC(N2CCCN(C(=O)Cc3ccccc3Cl)CC2)=O)CCC(=O)NC1=O c1(CN2CC(CC)N(C(=O)COC(C)=O)CC2)ccc(C#N)c(C)c1 C(=O)(CCCNC(N)=O)NC1(C(=O)NC2(CC(C)C)CC2)CC1 CC(C)(C)CC(C(=O)NCCN=[N+]=[N-])NC(=O)CC1(N(C)C)CCC1 Cc1nn(C)c(Cl)c1CN=C(NC1CCC1)NC1COCCN(C)C1 C1(NC(c2c(OC)oc(C)n2)=O)CCN(C(=O)CC(=O)NC2CC2)CC1CO c1(N2CC(C(N)=O)OCC2)cccc(S(=O)(=O)NC(Cc2ccsc2)CO)n1 C(=O)(C1CCCc2cccnc21)N(C1CCCCN(C(C2(CCF)CC2)=O)C1)C C(N=C(NC1CC1)N1CCC(C)(C#N)CC1)C1(C)CC(F)(F)C1 C12(CCNC(c3snc(O)c3Cl)=O)CCC1CN(C(=O)CC1CCCCC1O)C2 N1(C(C2N(CCC)CCC2)=O)CCC2C(CCN2C(c2ncc(F)cc2N)=O)C1 C(c1ccc(Cl)cc1)=CC(=O)NC1CN(C(C(c2ccccc2)C)=O)CC1F N1(C(c2ccoc2)=O)CC2CC1CN2Cc1cc(O)cc(F)c1 c1(NCC2CN(C(=O)C(F)CC3CC3)C2)ncc([N+](=O)[O-])cc1Cl C(=O)(C1CCCn2cncc21)N1CCCCC(NC(CNC(=O)OC)=O)C1 CCCCCC(O)C(=O)NCC1(CNC(c2cc(OC)ncn2)=O)CCCC1 C1(N(c2c(C)cccc2)C(C2CC(c3cc(Cl)sc3Cl)C2)C)CC2CCC1CC2 Cc1c(C=CC(=O)N(C)CC2CCCN2C(C2CC(=O)N2)=O)cnn1C Cc1ccc(F)c(C(=O)NC2CCN(C(=O)C(F)=CC3CC3)C2)c1 CC(C)C(CCNC(C1CCN(C(C)C)CC1)=O)NC(C1CC2C=CC1C2)=O c1(C(N2CCC(NC(c3ccc(CC)o3)=O)(CO)C2)=O)cnc(O)c([N+](=O)[O-])c1 C12(NC(=O)C(F)(F)F)CC3CCC(C1C2)N3C(c1cc2c(nn1)CCCC2)=O N1(C(C2N(CC)CCOC2)=O)C2CCC1(CNC(=O)C(C)(F)F)CC2 C(C(C)(C)CC(=O)NC(C)Cn1ccnc1)NC(C(C(C)C)=O)=O CC1(CNC(=O)CN2C(=O)CCC2=O)CC(F)(F)CN1C(=O)C1=CCCCO1 CCC(O)C(=O)NCCC(Cc1ccccc1)NC(c1cc(CO)on1)=O CC(F)(F)C(C)(C)C(=O)N1CC(NC(=O)CCCc2ccccn2)CC(O)C1 CC(C)C(O)C(=O)NCCn1cnc(C(=O)NCc2cscn2)c1 c1(C(=O)NC2CN(C(C(C)SC)=O)CC(C)(C)C2)cc(OC)c(S(N)(=O)=O)s1 N1(C(C(CSC)C)=O)CC2CCC(C1)N2c1cc(Cl)nc(SC)n1 N1(C(c2ccc(CC)nc2)=O)CC(O)(C2CCN(C(C3(O)CCOC3)=O)CC2)C1 N1(C(=O)CC2CCCCO2)CC2(CCN(C(c3csnc3Cl)=O)CC2)C1 C1(NC(C2(Cl)C(C)(C)C2)=O)CCCN(C(c2cc(C(=O)C(F)(F)F)c[nH]2)=O)C1 C1(NC(c2cnc(C(=O)OC)s2)=O)CCCCC1NC(c1ncccc1C)=O Cc1ncn(C)c(=O)c1C(N1CCN(C)C(CNC(c2cnn(C)c2F)=O)C1)=O N1(C(c2ccn(C)c2)C(=O)NC(CC)C)CCCC(C(c2ccccc2)=O)C1 C(=O)(C1=C(Cl)CCCC1)NC1CCN(CCNC(C(c2nc(C)sc2)(F)F)=O)C1 c1(C(=O)NC2CCN(C(C3(C)CC3(F)F)=O)CC2F)sc2ccccc2c1CO c1(Oc2c(NC(C3(C)CC(C(F)(F)F)C3)=O)cccc2)cccc(C#N)c1 Cc1nccc(C(=O)NCC(N2CCC(O)(C(N)=O)C2)=O)n1 c1(S)ccc(C)cc1C.CCC(C)C(=O)N(CCC)CCO c1(CC(N2C(CNC(CC(C)N(C)C)=O)C=CC2)=O)cccc2cnccc12 c1(-n2ncc(CNC(=O)C(=O)NCc3ccccc3O)c2)cccc(F)c1 N1(C(C(CCOC)NC(=O)C2=C(C)CCC2)=O)CCN2C(=O)NCC2C1 C1(C(C(=O)NCCCCC(=O)NC)(C)C)CCCCN(C(C2CCOC2)=O)C1 c1(NC(C)C)ccc(C(N2CC(NC(c3cnn(C4CC4)c3)=O)CC2C)=O)cc1 c1(NCC2CC(=C)C2)cc(=NCC2(C)CCCCO2)[nH]c(C(F)(F)F)n1 C(C(O)CC(=O)NC1C(C)CCC1C)NC(CC1ON=C(CC)C1)=O C1(C(=O)NCC(C)OC(C)C)CCCN1NC(=O)C1COCCC1C c1(SC)nc(O)nc(C)c1C(N1C2CCC1CN(C(C1(F)CC1C)=O)C2)=O C(=O)(C1Cc2ccccc21)N1CC(CCC)C(C(N2CCCC(C)(C#N)C2)=O)C1 N1(C(C2C(=O)NCCC2)=O)CCCC(C2CCN(C(c3csc(F)c3)=O)CC2)C1 c1(C(=O)NC2CN(C(c3c(C)nc(C)[nH]3)=O)CC23CC3)cc2cccc(Cl)c2s1 C1(CNC(C2CC3(CCO2)CC3)=O)CC(F)(F)CN1C(=O)C(c1ccccc1)O Cc1nc(C(F)(F)F)sc1C(=O)NC12CC1CN(C(C1CCCCS1)=O)C2 N1(C(C(c2ccccc2)NC(CC)=O)=O)CC(C)(NC(=O)C(C)(C)OC)C1 CCCC(CCC)CCCC(=O)N1CCC(C(C)NC(=O)C=CSC)C1 O=C(C1=CCCCC1)NC1CN(C(=O)CCC2CCCC2)CC1F C1(SC)CC(CNC(c2ccc(C(N(C)NC(C3(CC)CC3)=O)=O)[nH]2)=O)CN1 N1(C(C2C(NC(c3cc(C)on3)=O)C3CCC2C3)=O)CCN2CCCC2C1 c1(C(N2CCC(CC3C4CCCC34)CC2)=O)ccc(C2CC2)c(Cl)c1.C(=O)(C1CC1)N C1(OC)(CNC(=O)C2=CCCCO2)CCN(C(=O)C(C)c2cc[nH]n2)CC1 C1(C(F)(F)F)(C(=O)OCC2CC2C2CC2)CC2CCC1C2 CN1CC(CNC(C2CC(O)CN2C(c2nn(C)cc2Cl)=O)=O)CC1=O c12ccc(cc1Br)NC(=O)N1CCC(CC(C)C)(C1)C(=O)N2.C(C)(C)(C)O.C(F)F C(=O)(CCCCCCN(C1CCCC1(C)C)C(=O)CC1CC1)Nc1c(C)ncnc1 N1(c2nc(C)cc(OC)n2)CC=C(CNC(C2CCC(C)O2)=O)CC1 c1(NC(=O)NCC2CCN(C(CC)=O)C2)c(-c2ccsc2)noc1C C(=O)(C(C(C)c1ccccc1)N1CCCC1Cc1nnn(C)n1)NCCCCCC CCCCC(F)(F)C(=O)NCCCN(C)C(c1cc(F)cc(F)c1OC)=O c1(C(N2C(CNC(c3cnn(C4CC4)c3)=O)CC(OC)C2)=O)cc(O)ccc1C N1(C(C(CC)CC)=O)CC23CCCC2(C1)CN(C(c1cccc(Cl)c1C)=O)C3 C1(n2cc(-c3c(C)ncs3)nn2)CCN(C(c2ccn(C)c2)=O)CC1 C1(CCOC)CN(C(C(=O)NC(C)C)C2(NCCC(=O)OC)CCC2)CCO1 N1(C(C2C(C(C)(C)C)OCC2)=O)CCC2(CC1)CN(C(c1cscn1)=O)CCO2 C1(c2ncc(C(=O)OC)s2)CCN(c2nnnn2CC2CC2)CC1 C1(CC=C)(C(=O)NC2CCSC2)CN(C(=O)CCc2csnn2)C1 CCCCC(CC)CC(=O)NCCOCCNC(=O)C(c1cc(C)ccn1)(F)F C1(CN(C(=O)C(C)OCC(C)C)C)CCC(CNc2ncc(CC)s2)CC1 n1(CC)ncc2c1CC(C(=O)NC1CN(C(C34CC(C)(C3)C4)=O)CC1(C)C)CC2 N1(C(CNC(C(CC)C)=O)=O)CCN(C(c2sc(C)nc2C)=O)CC1C1CC1 C#Cc1cc(F)c(C(=O)N(C)CCN(C)C(c2ccc(=NCC)[nH]c2)=O)cc1F C1(CCOC)(NC(=O)CSCCC#N)CCN(C(=O)Cc2cscn2)CC1 CCCC(C)CCCC(=O)NC1CC2CCC(C1)N2C(c1cn(C(C)C)nn1)=O N1(C(C(CCSC)OC)=O)CCC2C(C1)CN2C(=O)CN1CCCCC1 c1(NC)ccccc1C(N1CC(N(C(=O)CCC2CCCO2)C)C(O)C1)=O CN1CC2(C1)C(c1nnnn1C(C)(C)C)N2.C1(C)COC(=O)O1 N1(C(C(=O)N(C(C)CNC(=O)CC2CC3CC3C2)CC)=O)CCCC(C)C1 c1(C(=O)OC(c2cccc(C(N(C(CCOC)C)C)=O)n2)=O)cncn(C)c1=O c1(C(N(C2CC(C(C)=O)SC2)C(F)(F)C(F)Cl)=O)nc(C)[nH]c2nccc1-2 CC1(CNC(C2(CC(F)(F)F)CC2)=O)CCC(NC(c2ccc(F)cc2)=O)C1 CC(CC(C)NC(=O)CC(C)c1ccco1)NC(=O)CC(O)C1CC1 C(CC1CCCCC1)(C(=O)NCCCN(C(C1CC1CF)=O)C1CC1)OC C1(CC(=O)N(CC=C)CCC)CN(C(c2ncccn2)=O)CCC1C N1(C(CSCC#C)=O)CCC(C2CCCN(C(=O)C(c3cnn(C)c3)C)C2)C1 c1(C(=O)NCC2C(NC(=O)CC3C=CCC3)CC2)ccc(Cl)cn1 c1(C(N(CC(CC)NC(=O)C(C)Cc2ccnn2C)C)=O)c(F)ccc(Cl)c1F c1(CC(N2CCN(C(C(CC=C)(C)C)=O)CC2)=O)csc2sc(C)cc12 N1(C(COc2cc(C)on2)=O)CCCC(C(C)C(=O)N(CC(O)C(F)(F)F)C)C1 CC1(C)C(NC(C2(C)CC2)=O)CCN1C(=O)C(F)OC(F)(F)F.c1(O)ccc(F)cc1 C(=O)(C(C)(C)CNC(=O)C(C)CNC(=O)Cn1ncn(C)c1=O)OC Cc1nc(NCC2CN(C(c3cc(Cl)c[nH]3)=O)CCC2C)c(Cl)cc1[N+](=O)[O-] C(c1cccc(Cl)c1)=CC(=O)NC1CCC1C(=O)NCCN1CCCCC1 C1(C(=O)NCCCCC(C)NC(C2(C#C)CC2)=O)CCC(N=[N+]=[N-])C1 CCS(=O)CCNC(=O)CC1CC1CNC(C1(CC)CC1)=O C=CC(C)(C)CCN=c1[nH]c(=NC2CCC(C)(CN(C)C)CC2)c2ncccc2[nH]1 c1(NC(C2C(C(=O)NCc3cccc(C)c3C)C2)=O)ccc2nncn2n1 C1(OC)CCCC(C(N2CC(C)(NC(=O)C(c3ccc(C)o3)C)C2)=O)C1 NC1CCCC1N(C(=O)CC1CCN(C(=O)OC(C)(C)C)C1)C1CC1 N1(C(C(CC#C)C2CC2)=O)CCCOC(CNC(c2cc(C)n(C(C)(C)C)n2)=O)C1 N1(C(C(CCC)CNC(=O)C(C)CO)=O)CCCC(C)(C#N)C1 c1(C(=O)NCC2(C(=O)NCc3cc(C)cc(Cl)c3)CC2)cc2ncccn2n1 C1(NC(C(C)OCCC#C)=O)CN(C(=O)Cc2ccc(C)nc2Cl)CC1N=[N+]=[N-] C1(C(=O)NC2CCN(C(c3c(C)nsc3N)=O)C2)Cc2nnc(C)n2C1 CC(C(=O)NC(CNC(c1csc(-c2ncc[nH]2)n1)=O)C(C)(C)C)C(C)S(C)(=O)=O c1(C(=O)NC2CN(C(C3CCC4CC34)=O)CC23CCC3)cnn2cccc2c1 c1(C(=O)NC(C(C)C)CNC(C2CCCN2S(C)(=O)=O)=O)c(O)cccc1F c1(N(CC(=O)NC2CC2)CC2CC2)cc(CNC(=O)CC2C=CCC2)on1 N1(CC(N2C3CC(NC(CCC=CC)=O)(C3)C2)=O)C(=O)NC(CCCC)(CC)C1=O c1(C(N(CC(C)NC(C2(C)CC(C#N)C2)=O)C)=O)ccc2c(c1)NC(=O)C2=O C1(C(=O)NC(C2CCN(C(c3nccn3C)=O)C2)C)CCCCC1(F)F N12CCCC(C1)OCC1(CCC1)C2=O.C(CC(=O)N)SCC.OC C(c1ccccc1N1C(=O)N(C)CC1=O)N1C(C)CC(NCc2ccccc2)CC1 Cc1ccc(C(=O)NC(C)CCNC(=O)C(c2cncnc2)C)c(F)c1C C1(C(=O)NCC#CCC)CCOCCN1C(=O)CCCn1ccnc1 c1(C(=O)NCCC(C)(C)NC(c2scnc2C2CC2)=O)ccc(C2CC2)nc1 C(=O)(C(CC(C)(C)C)N(C)C)NC(C1CC1C(N1CC(=O)N(C)C(=O)C1)=O)C CCS(=O)c1ccccc1C(N1CCCC(N(C(=O)CCN(C)CCO)C)CC1)=O C(C(CC1CC1)C(=O)NCCN1CCCC1=O)NC(C1(C)CC(=C)C1)=O CC1CCN(C(=O)OC(C)(C)C)CC1NCCC(C)(C)N1CCCC1 C1(C)(C(=O)NC(c2n(C)ncc2)C(N2CCCOCC2)=O)CCCOC1 C1(c2c(OCC)cnn2-c2ccccc2C)CCC12CCN(C(=O)OCC)CC2 C(=O)(C1=CCC(C)(C)CC1)NC1CN(C(Cc2cc(C)c(O)cc2)=O)C(C)CC1 N1(C(C(COC)C)=O)CCC(C)(C)C1C(=O)NC1C2CCCCCC12 C(=O)(C1=C(Cl)CCCC1)NCC1C(C(F)(F)F)CCN(C(CC(C(C)C)O)=O)C1 Cc1cccc(CC(=O)C(CC2(NC(C(C)N)=O)CCC2)=O)c1.C1(N)COC(C)C1 c1(CNC(=O)C=Cc2cocn2)cnn2c1CN(c1nccc(CO)n1)CC2 N1(C(CCC2CCC(=O)NC2)=O)CCN(C(c2ccc(CO)cn2)=O)C(CO)C1 C1(NC(c2scc(OC)c2)=O)CC=C(C(=O)NC2(CO)CCSC2)C1 N1(C(CC(C)n2ccnc2)=O)CCOCC1CN(C)C(c1ccncn1)=O C(c1ccc(C)c(Cl)c1)=CC(N1CC2C(CNC(C(C)SC)=O)(C2)C1)=O C1(Oc2ccc(N3CCC(CNC(=O)C(=O)OC)C3)cc2)Cc2ccccc2C1 N1(C(C(CCC)CNC(=O)CP(C)(C)=O)=O)CCn2c(C)cnc2C1 N1(C(CNS(CC)(=O)=O)=O)CC(NC(=O)C(C)SCc2ccccc2)CC1CO N(C(=NCc1ccc(OC(F)F)cc1)NCc1ccsn1)C(C1CCCCO1)C c1(CCC(=O)Nc2c(OCC)ccc(C(N)=O)c2)cccc2oc(C)nc12 c1(CC(=O)NCC2C(CNC(C(CC)C)=O)C2)ccc2c(c1)CCCN2C N1(C(c2c(C)n(C)cn2)=O)CCN(C(=O)Cc2nnc(O)s2)C(CO)C1 CC1(C)CC(C(N2CC3C(CNC(C4CC4[N+](=O)[O-])=O)C3C2)=O)(CO)C1 c1(C(N(CCOC)CCNC(=O)C=C2CCN(C)C2)=O)cc(O)nc(Cl)c1 c1(-n2cc(C(N(CCNC(Cc3c(C)con3)=O)C)=O)nn2)ccc(Br)c(F)c1 C(=O)(CCCc1nncn1C)N(CC(O)CN(C)Cc1nccn1C)CCCC CN1CCC(C2(C(=O)NCCCN(C(=O)Cc3ccc(O)c(Cl)c3)C)CC2)CC1 CC(C(=O)NC)C(C)(C)C.C(C)(C(F)F)=C C1(CN(C(C2CCCN2C)=O)CC)CCN(C(C2CCC=CO2)=O)CC1 c1(OC(COC)C)ccccc1NC(=O)Cc1ccc(C)cc1 N1(C(C(C(C)C)OC)=O)CC2(CCCC2)C1C(=O)NCC(=O)N1CCCO1 c1(C(=O)NC(C(N2CCC(C)(CNC(C)=O)C2)=O)(C)CO)cccc(F)c1C N1(C(c2nc(CC)oc2C)=O)CC2(C)CC1(C(=O)NC(C)CCOC(C)C)C2 c1(CNC(C(C)NC(=O)OC)=O)nc(C)c(C(=O)NCc2cc(F)c[nH]2)o1 c1(CNC(c2cnc3[nH]nnc3c2)=O)n[nH]c2c1CN(C(C1(CF)CC1)=O)CC2 c1(NC2n3nnnc32)n[nH]c(C(C)(C)C)n1.C1(C(C)O)CC2CC2C1.C(C)(C)(C)OCC C(c1cc(C)cc(C)c1)=CC(N1CCC(C(C)NC(c2cnc(CC)s2)=O)C1)=O C(=O)(C(C)(F)C(C)(C)F)NC(CNC(Cc1ccc(C)cc1Br)=O)CO c1(C(=O)NC2C(C=C)CN(C(=O)C(COC)OC)C2)cn(C)c2ncccc12 CCC(F)(F)CC(=O)NC1CC(F)(F)CC1NC(C1(c2ccc(C)cc2C)CC1)=O N1(C(c2n[nH]c(CC)c2C)=O)CCC2(C=C(C(=O)NC3CC(O)(CO)C3)C2)C1 c1(CC)c(C(N2CC3CC3(CNC(=O)C(O)CN(C)C)C2)=O)[nH]c2ccccc12 C(=O)(C(CNC(=O)CC1CCCCC1O)C(C)C)NC1C(C(=O)OC)OCC1 N1(C(Cc2cc(C)ncc2)=O)CCCC2(C1)CN(C(c1oc(CO)cc1C)=O)C2 Cc1cc(C)n(CCC(N2CC(C(=O)NCCCCc3ncc[nH]3)(CC)C2)=O)n1 Cc1cc2cc(C(N3CCN(C(C4CCC=CCC4)=O)C4CC34)=O)[nH]c2cc1Cl N1(C(c2cn(CCOC)nn2)=O)CC(C)CN(C(=O)CC2(O)CCCCC2)CC1C C=Cc1cncc(C(N2CC(NC(=O)C(C)N3CCCC3)C(C(F)F)C2)=O)c1 c1(CC(=O)NCCN(C(C2CCOC2)=O)CC)cccc2nonc12 C(CC)(CCC(=O)NOCC(=O)OC)NC1CC(OCC)C1 c1(CN(CC(=O)Nc2ccc(OC)cc2)C)cccc(OC)c1F C1(NC(CC(C)(C)C(=O)O)=O)C(F)(F)C12CCC2.n12cc(nn1)COCCC2 C1(C(C)C)CCOCCN1C(C1CNC(=O)N1)=O.C12CCN(C1)C2 CN1C(=O)OCC1C(N1CCC(F)(C(=O)NCCC2CC(C)(C)CO2)C1)=O C1(C#CC(=O)NC2(C3CN(C(c4ccnnc4S)=O)C3)CC2)(CC)CC1 C#Cc1ccc(C(=O)NC(C)CN2CCN(C(=O)C(C3CCC3)OC)CC2)nc1 CC1COCCN1CC.C12(CCCCC1)C(=O)N2.C1(CC(=O)NC)CCCCO1 C1(CC)CCCN(C(c2cc(CCNC(c3cncs3)=O)on2)=O)CC1 N1(C(C2C(=C)CC2)=O)CCC(OCCNC(c2scnc2CC(C)(C)C)=O)C1 c1(C(=O)NCC(C2CCN(C(C(CC)(C)C#N)=O)CC2)C)cnc2ccnn2c1 C1(CCC(C)C)CN(CC2(C)CC2(Br)Br)CC(=O)N1 c1(CC)cnc(C(N2CCC(CC(F)(F)F)C2)C(=O)NCC2CC2)[nH]1 C(C1CCC(C)CC1)=C(C)C(=O)NC1CC2CC1CN2C(C12CC(F)(C1)C2)=O c1(OC)cncc(C=CC(N2CCC(NC(=O)C(O)CC(N)=O)C2(C)C)=O)c1 N1(C(C2C(C(=O)OC)CC2)=O)CC(C(=O)NCCC2CC(F)C2)C2(CC2)C1 C(=O)(CC(c1ccccc1)c1ccccc1)N(C1CC(=C)C1)CC(N1CCCC1)=O CCCCC(CC)CC(=O)N1CCC(CCNC(c2scnc2C2CC2)=O)CC1 c1(C(=O)NCC(CC(F)(F)F)NC(C(CCC)N(C)C)=O)cc(Cl)cc(F)c1N C(C(=O)N1CC2CC2C1C(N1CCC2(CC1)N=N2)=O)(C(C)(C)C)OC C1(NC(=O)C(N2CCCC(c3cc[nH]n3)C2)=O)CC2(CCC2)C12CCC2 Cn1cc(CCC(=O)NC2CC2CNC(C2CC(c3ccccc3)C2)=O)cn1 N1(C(CC(C(C)C)O)=O)CC(C2CCN(C(=O)CCNC(C3CCC3)=O)CC2)C1 C1(NC(c2c(NC)nccc2)=O)CN(C(=O)C2CC2)CC12CC2 C#Cc1ccc(C(N2C(C(=O)N(C)CC3(O)CN(C)C3)CC2C)=O)c(C)c1 CC1(C(=O)NCCOC2CCN(C(=O)Cc3ccsc3)CC2)COCCO1 N1(C(C(CC)n2cncn2)=O)CCC(C(=O)NCc2nccnc2C)CC1(C)C c1(COC)cccc(C)c1NC(=O)C(N1CC2CC(NC(=O)OC(C)(C)C)C1C2)=O CC1CN(C(C2(CF)CC2)=O)CC1NC(c1ccc(-c2ccccc2Cl)o1)=O C=C1CC2(C1)CC(C(=O)NC1CCCN(Cc3nc(=O)n(C)[nH]3)CC1)C2 N1(C(c2c(C(F)(F)F)nn(C)c2Cl)=O)CCCC2(CCN2C(c2ccno2)=O)C1 C1(COC)CCCN1C(=O)NC1CCCC1c1ccccc1 c1(OC(c2ccc(C(C)N)cc2)=O)cccc(CN(CCC)CCOC)c1 O=S(=O)(c1cc(F)c(F)c(F)c1)N1CCC(c2nc(-c3ncncc3I)no2)C1 C1(NC(CCOC(C)C)=O)CCC(N(C)C(c2nnn(C)c2N)=O)CC1 CCC1CC(=O)NC2CC(C2)CCCCCC(=O)N1.C1(OC)CC1 N1(C(C(=O)NCC)=O)CCN(CCN(C)C(c2occc2C2CC2)=O)CC1 c1(OC)cccc(NC(=O)C(N2CCC(C(F)F)(OC)C2)c2ccsc2Cl)c1 c1(CC)ccccc1NC(C1CCCN(C(=O)OC(C)(C)C)C1)C(=O)NCCCl N1(C(c2ccc(NC(C)=O)s2)=O)CCN(C(=O)C=CBr)C(C)CC1C c1(C(N2CCC(O)(C(C)NC(c3[nH]cc(CC)c3)=O)C2)=O)cnc2cc[nH]c2c1 C(=O)(CC(c1ccccc1)n1cnnn1)NCC(C)NC(=O)C(C)OC(C)(C)C C1(CNC(CCCC)=O)C2CCCC1N(C(=O)C(C)SCC1CCCCO1)C2 c1(OC)ccccc1CC(C)(O)CNC(=O)NCc1ncc(Br)cn1 c1(OC)ncnc2sc(N3CCC(c4ccc(C(F)(F)F)cc4)C3)nc12 C(=O)(CCC(=O)NC(C)C(C(C)C)NC(C1SCCS1)=O)N(C(C)C)C C(=O)(CCCC(C)(C)NC(c1cc(CO)ccn1)=O)N1CCC(COC)C1 c1(C(=O)Nc2cccnc2)cn2c(n1)CN(Cc1ccc3nc[nH]c3c1)CC2 c1(C(=O)NCC(CNC(c2cnc(SC)s2)=O)O)cn(-c2nccs2)nc1C c1(OC)ccc(Br)cc1CC(N1CCN(C(=O)C(O)C(C)C)C(C(C)C)C1)=O C(=O)(CCC(=O)NN(C)C)NC1CC(NC(C=CC(C)(C)SC)=O)C1(C)C CC1(CNC(C2(CNC(c3nsnc3O)=O)CC3(CC3)C2)=O)CC(F)(F)C1 C1(CCNC(C2CC2c2ccccn2)=O)(OC)CN(C(=O)C=CC2CCCC2)C1 C1(C)(CC(=O)NCC(C)(C)NC(C2(N(C)C)CCCCC2)=O)CC1(Cl)Cl Cn1ncc2c(O)cc(C(N3CCN(C(=O)CC(C)(C)F)CC3C3CC3)=O)cc12 C1(CC(N2CCC(CNC(CC(COC)C)=O)CC2)=O)CCC2(CC1)COC2 C1(C(N(CC)Cc2ccco2)=O)CN(S(=O)(=O)N2CCC(CC(C)C)C2)C1 N1(C(Cn2nnc(C(C)(C)C)n2)=O)CC(NC(C2(O)CCC2)=O)CC2(CCC2)C1 C1(NC(c2c(CC)n[nH]c2)=O)CC=CCC1C(=O)NC1CC1(C)C(F)F c1(C(N2C(C)CCC(CNC(=O)CN3CC=CC3)C2)=O)noc2cc(F)ccc12 N1(C(CC(C)(C)C)=O)CC2(C1)CN(C(=O)CSC)C2.c1(O)cccc(-n2cnnn2)c1 c1(OCCC(=O)NC2C(NC(=O)C=Cc3cc[nH]c3)COC2)ccc(F)cc1 C1(NC(C)=O)CCC(C(N2CCC(CNOC3CCCNC3)CC2)=O)CC1 C(=O)(CC(c1ccccc1)n1ccnn1)N(CCC(=O)NC1CCOC1)C c1(C(=O)NC2CC(CNC(c3ncn(C)c3)=O)OCC2)cc(S(N)(=O)=O)n(C)c1 C1(NC(C2OCC(C)(C)C2)=O)CCC2CCN(C(C3(CCF)CCC3)=O)C1C2 c1(C(N2CCC(N(C(C3CC4CCC4C3)=O)CC)C2)=O)cc2c(cn1)OCCO2 N1(C(C2CC3(CSC3)C2)=O)CCC(C2CC2)C1CNC(=O)C(F)(F)C(F)(F)F N1(C(Cc2nc(=N)[nH][nH]2)=O)CC2CN(C(=O)CC3CC4(CCO3)CC4)CC(C1)O2 CCCC(CCCNC(=O)CCCn1cncn1)NC(=O)C(CCC)N(C)C c1(C(C(=O)NCC(C=C)O)N(C(=O)C(CC)OC)C2CC2)c(C)cccc1Br C1(CCC#C)CCCN(C(C2C=CC(NC(C3C=C(C)CS3)=O)C2)=O)C1 C12(CNC(C3CCCO3)=O)CN(C(c3cnsn3)=O)CC1CS(=O)(=O)C2 CC1CCC(C(=O)NCc2ccno2)N1C(c1c(Br)cnn1C)=O C(=O)(CCS(C)=O)N(CC(C)(C)CNC(c1csc(C2CCCO2)n1)=O)C CC1CCCCC1CC(=O)N(CCCCNC(=O)C=Cc1ccc(Cl)s1)C C1(CCNC(c2ccc(C)nn2)=O)CN(C(c2c(C)csc2C)=O)CC(C)O1 N1(C(Cn2cc(C(C)=O)nn2)=O)CCC(C)C1CNC(c1cc(C)sc1C)=O N1(C(=O)Nc2cnncc2OC)C2CCC1CC1(C2)CC1(F)F c1(C(N(CCCCCCNC(CSC(C)C)=O)C)=O)cnc2c(c1)ncn2C c1(OC)ccc(-c2cn(CSC3COCCO3)nn2)cc1.N12CCCC(C1)CC2 Cc1noc(C)c1CC(=O)NCC1CC(F)CN1C(C1CCCC1)=O c1(C(C)=O)[nH]c2ccccc2c1CC(=O)NCC(C(C)(C)C)NC(C1CC1C)=O N1(C(=O)C2=CCCC2)CCCCC(C2CN(C(c3cncc4ccsc34)=O)C2)C1 C12(C(=O)NC3C(C)CN(C)CC3)CCN(C(C3(C)COC3)=O)CCC1C2 Cn1nnc2c1CCC(C(N1CC(O)CC1CNC(c1ccc[nH]1)=O)=O)C2 c1(C(=O)NC(CC)CNC(c2ccc(Br)nc2O)=O)ccc2ncccc2c1 C1(C(N2CCC(NC(CC(CC)CC)=O)C(C)C2)=O)CC2COCC(C1)C2=O C=C1CC(C(=O)NCCC(C)O)N(C(C2CC3C=CC2C3)=O)C1 C1(C)(C(=O)NCC2(NC(=O)CN(C)C)C(C)CCCC2)CCCCCCC1 C1(CC(=O)NC(CSC)(C)CO)(NC(=O)C(C)CC2CC2)CCCCC1 N1(C(c2cccc(C3CCOC3)c2)=O)CCCCC(N=c2[nH]nc(C3CCC3)s2)C1 c1(N2C(CCNC(C(C(C)C)N(C)C)=O)CCC2)nccc(C#N)n1 N1(C(c2cnc(SC)s2)=O)CCC2(CC1)CC(NC(=O)CCCC1(C)CC1)C2 C(=O)(CCCC(C)(C)CC)N1C(C)CC(CNC(c2cc(CC)nnc2C)=O)C1 N1(C(c2c(C)ccs2)=O)CCC2(CCC(CNC(=O)C(O)C(F)(F)F)OC2)CC1 CCCCC(CC)C(=O)NCC(C)(CO)NC(=O)CCOc1ccc(Cl)cc1 C1(N(C(CC2CCCC(N(C)C(C3(C(N)=O)CC3)=O)C2)=O)CC)CN(C)CC1(F)F N1(C(CNS(CCCC)(=O)=O)=O)CCCC2C1CCN2C(c1ccc[n+]([O-])c1)=O C1(C(=O)Nc2ccc(-c3nn[nH]n3)s2)CCC2(CC1)N=N2 C1(C(N(C)Cc2ncc[nH]2)=O)CN(C(=O)C=Cc2cn(C)nn2)C(C)(C)C1 C(N=c1nc(N(C)Cc2cnn[nH]2)c2[nH]ccc2[nH]1)C1CCCN(C(C)C)C1 CCC(C(=O)NCC1(NC(=O)C=Cc2nc(C)c(C)[nH]2)CC1)C(C)O C1(CC)(NC(c2sccc2CN(C)C)=O)CCCN(C(c2n[nH]cc2F)=O)C1 N1(C(C2CCCN(CC)C2)=O)CC2CC(NC(C3CC(Cl)(Cl)C3)=O)C(C2)C1 Nc1c(C(=O)NC2CC2NC(c2ccc(Cl)cc2)=O)cnn1-c1ccc(F)cc1 N1(C(CC2N(Cc3cnc(C)[nH]3)CCC2)=O)CCC(O)C(F)(F)C1 N1(C(c2c(C)cc[nH]2)=O)CC(NC(=O)C(N2CCC(C)CC2)=O)CC1C c1(N(c2cn3c(n2)SCC3)C)nc2ccsc2c(=NCCSCC(F)F)[nH]1 N1(C(C2(CC#C)CCCO2)=O)CCOCC(C(=O)N(CCCn2cncn2)C)C1 N1(C(CCSC)=O)CC(OC)CC(NC(c2nc(=O)n(C)cn2)=O)C1 Cc1cc(C(=O)NC(C)C(C)(C)NC(C2CCO2)=O)sc1Br C(=O)(C1=C(C)CCCC1)N1C(CNC(c2cccc(OC)n2)=O)CC1 N1(C(CN2C(=O)NCC2)=O)CCC12CCN(C(c1cc(I)c[nH]1)=O)CC2 c1(COC)nnc(C(=O)NCCC2CCN(C(=O)COC3CC=CC3)C2)s1 C1(c2n(C)ncc2)CN(C(c2coc(O)n2)=O)CCN1C(=O)Cc1cccnc1 c1(C(=O)NC2(CNC(C3N(CCC)CCCC3)=O)CC2)cc(S(N)(=O)=O)c(C)o1 c1(OC(C)C(=O)N(C2CN(C(=O)C(C)(C)C3CC3)CC2F)C)ccc(F)c(F)c1 N1(C(c2c(CC)nc(=N)[nH]c2)=O)CCCN(c2nccc(C(F)F)n2)C(C)C1 C1(CC=C)(C(N2CCC(CN(C(=O)Cn3nnc(C4CC4)n3)C)C2)=O)CCCC1 N1(C(C(CCC)O)=O)CCC2(CCC(NC(C3(CO)CC3)=O)C2)C1 CC1(C)CN(Cc2ccccc2CN)CCN1Cc1ccccn1 C1(C(=O)NCCOC(CC)CC)C(C)CCN1C(=O)Cc1csc(C)c1 C1(C2N(C(COC(CC)C)=O)CCC2)CN(C(C2CC(SC)C2)=O)CCO1 N1(C(C=CC=CCC)=O)CCCC(C(C)C(N2CCCC2CF)=O)C1 c1(CC(C)NC2CCCC2N(C(C)(C)C)C(=O)Sc2nnnn2C)nncn1C Cn1ccc(C(=O)NC2(C(=O)NCCCS(N)(=O)=O)CCCC2)cc1=O C(CCN=c1[nH]c(=NCc2ccsc2)[nH]c2c1SCC2)c1ncn(C)n1 C12(NC(C3(NC(C)=O)CCC3)=O)CCC(CC1)N(C(C13CCCCC1C3)=O)C2 c1(C(=O)OC)ccnc(NCC2CCCCC2NC(=O)CC2(CO)CC2)n1 C1(CC#C)(C(=O)NC(CNC(=O)C(C)OCCCC)CO)CCCCO1 C(=O)(C1Cc2ccccc21)NC(C)CCCNC(=O)Cc1cnc[nH]1 CC1CC(CNCC(=O)OCCOC(C2(N(C)C)CC2)=O)CO1 Cc1ccc(C(N2CCC(C)C2CNC(=O)Cc2cc[nH]n2)=O)c(N)n1 c1(C(=O)NCC23C(CN(C(c4ccc(NC)cc4)=O)C2)C3)ccnc2[nH]ncc12 Cc1cc(C(N2CC(CNC(C3(C(C)(C)C)CCC3)=O)CC(C)C2)=O)cc(F)c1 N1(C(=O)COCC2CCCO2)CC2=C(C1)CN(C(C1CC13CCSCC3)=O)C2 C(=O)(C1=CC2CCCCCCC12)NC1CC(CNC(C(=O)NCC(F)(F)F)=O)C1 N1(C(C2(NC(C3(CCN=[N+]=[N-])CC3)=O)CC2)=O)CCC2CCCC2CC1 c1(NCCC2(CO)CCCC2)ncccc1S(=O)(=O)NC(CN(C)C)CO N1(C(CCCn2c(C)csc2=O)=O)CCC2CCN(c3nccnc3F)CC2C1 Cc1n[nH]c(C)c1C(=O)NCc1cn(C2CCN(C(=O)C3=CCC3)CC2)nn1 C=CC(C)(CCOC)C(=O)N1CCCC(O)(CNC(=O)CN2CCS(=O)CC2)C1 C1(CC)(OC)CN(C(=O)CC2CCC(NC(=O)C(C)CC3CCC3)C2)C1 C1(C(N(CCC(=O)NCCC2CCCC2O)C)=O)CSCC(=O)N1 C1(CNC(C(C#C)(C)C)=O)CCC2CN(C(=O)COCc3ccccn3)CC12 CCC(CC)(CCNC(C1CC(C(C)C)=NO1)=O)NC(=O)CSCCC(C)C c1(C(=O)NC2C(CNC(c3[nH]n(C)c(=O)n3)=O)CCC2)ccn2cncc2c1 N1(C(Cn2ccc(C)n2)=O)CC2OCCN(C(c3cc(F)cc(F)c3N)=O)C2C1 CC(C)CC(C(=O)OC(CC(=O)NC(c1cc(F)cc(F)c1)C)C)OC C(=O)(C(C)(C)CSC)NCC(C(=O)NCC1CC=CCC1)OC C1(NC(c2ccc[nH]2)=O)CCN(C(=O)Cc2cnns2)C12CCC2 Cc1ccc(F)c(C(=O)NC(CN=[N+]=[N-])C(=O)NCC2(N(C)C)CC2)n1 C=CCCCCCC(=O)NCC1(OC)CCN(C(=O)CCC(C)O)CC1 C1(c2ccccc2)(C(=O)NC(C)CN(C(=O)CCN2CCC2)C)CCCO1 C1(NC(c2ccnc(OC)n2)=O)CN(C(C2C=CC=CC=C2)=O)C2CCCCC12 c1(C(=O)NCCCCCN(C(C(CC=C)C)=O)C)ccc2c(c1)NC(=O)CCC2 C1(CNC(C=CC=CCC)=O)C(C2CC2)CCN1C(c1nccn1CC)=O N1(C(c2n(C=C)nnc2)=O)CCOC2CN(C(C3CC3CF)=O)CC12 c1(C(N2CCCCC(NC(c3cnc[nH]3)=O)C2)=O)coc2c1CCCC2 N1(C(C(=O)NC(C)C)=O)CCN(C(=O)CCc2ccoc2)CCC1C N1(C(c2ccc(O)cc2)=O)C(C(N2CCCC2c2ccc(F)cc2)=O)C2(CC2)C1 C#CC1CCC(C(=O)N(C)CCNC(=O)Cc2cnsc2)CC1 CC(C)S(=O)(=O)CC(=O)N1CC(NC(=O)Cc2cccnc2Cl)CC(C)C1 C(=O)(C1CCCc2sccc21)N1C2CCCN(C(c3[nH]c(=N)sc3)=O)C2CCC1 c1(C(=O)NC(c2cccnc2)C(=O)N(CCC(C)C)CC)cc2cnccc2[nH]1 C1(C)(CCC(=O)NC2(C(COC)O)CC2)CCCN1C(c1c[nH]nc1Cl)=O CN1CCCC(CCC(=O)N(C2C3CN(C(C4(F)CCC4)=O)CC23)C)C1 C=C(C)CCCC(=O)NC1CCC12CN(C(=O)Cc1ccc(Cl)cc1Br)C2 C#CCCCCCCCNC(=O)C1=CCN(C(C2(C#N)CCOC2)=O)C1 N1(C(CNC(C)=O)=O)CC2(CCC2)CC1CNC(=O)Cc1ccc(F)cc1 C1(NC(CCC#C)=O)CN(C(=O)COCCCCC)C(C)(C)C1 CC1(NC(C2CCC(F)CC2)=O)CCN(C(C2(C)C=CCCC2)=O)CC1 N1(C(CC(C(C)C)OCC)=O)CCN(C(c2cc(OC)ccc2N)=O)CC(CO)C1 N1(c2ncnc(CC)c2F)CCN(C(c2cnc(C(C)(C)C)s2)=O)CC(C)(F)C1 C1(C(=O)OC)CC12CCN(NC(Cc1ccc(CC3CC4C=CC3C4)cc1)=O)C2 C(=O)(CCC1=CCCCC1)NC1CCC(CCNC(c2c(C)snc2)=O)C1 CCC(CC)(CO)C(=O)NCC1CN(C(c2cn(C3CC3)nn2)=O)CCC1(F)F c1(C(N2C(CNC(C=Cc3n(C)ncc3)=O)COCC2)=O)ccccc1N=[N+]=[N-] C1(NC(C=C(CCC)C)=O)CC(CC(=O)NCCC2CCCC2)C12CCC2 O=C1CCCCC(C(N2CCOC(CNC(c3ccn(CC(F)F)n3)=O)C2)=O)N1 c1(OC)nc(C(=O)NC2CCCN(C(=O)CC3(C)CC3)C2)sc1C C(C(C)CC(=O)NC(C)C(C)C(=O)NC1CC(COC)C1)OC N12CCCC(C1)N(c1cccc(C)c1)c1nc(ns1)CC2=O.C(COC(C)=O)OC C1(C(N2C(C(N(CCSC)CC)=O)CSC2)=O)CCC(O)CN1C N1(C(C(C)CN(C)C)=O)CCCC(CNC(c2ccc(OCF)cc2)=O)C1 C(CC(CC)C(=O)NC1CC2(C1)CC2C(=O)NOCC=CCl)=CC Cc1c(CNC(C2CCCN(c3ccccc3)C2=O)=O)ccc2c1NCCO2 c1(C2C(C(=O)NC(C3CCOC3)CNC(c3n[nH]cc3Br)=O)C2)ccccc1 C1(N(CC)CC)CN(C(=O)C=CCN(C2CC2(C)C)C)C1 N#Cc1cccc(NC(=O)COCCc2ccccc2Br)c1 Cc1cc(C(=O)NCC(c2ccc(F)cc2)NC(=O)CC(C)(F)F)cn1C N1(CC)CCC(N(C(=O)C(C)(C)NC(=O)COCc2nc[nH]n2)C)C1 c1(C(N2C(C)CN(C(COCCOCC)=O)CC2C)=O)cncc(S(C)(=O)=O)c1 C1(C(N(C(C(=O)Nc2cscn2)C2CC2)C)=O)C2CN(C(=O)CCC(=O)N(C)C)CC12 C1(COC)(CNC(C2CC(C)CCO2)=O)CCN(C(c2nocc2C)=O)C1 C1(CNC(c2c(CC)nns2)=O)CC(C)CCN1C(=O)CC12CCCC1C2 N1(C(c2ccc(C)n(C)c2=O)=O)C2COCC1CC(NC(C1CCCOC1)=O)C2 c1(N(C(C(=O)N(CCOCCOC)C)=O)C)cc(C(F)(F)F)cc(N)c1 c1(CN2CC(C(=O)Nc3ccc(SC)cc3)OCC2)c(Cl)cnc(Cl)c1Cl C(=O)(CC1=CCCC1)N1C(C2CCN(C(c3c(CC)nn[nH]3)=O)CC2)CCC1 c1(CC(=O)NCC(CNC(C2(N(C)C)CCCC2)=O)O)ccc2c(c1)CCCC2 C1(c2c(CC)csc2)NC(=O)N(CCF)C2=C1C(=O)NC2(C)C C(=O)(CS(=O)(=O)CC(C)C)NCCC1(O)CCCN(C(c2[nH]cc(CC)c2)=O)C1 C1(C)(NC(C(CN(C)C)O)=O)CCCCC1C(=O)Nc1cc[n+]([O-])cc1 C1(NC(c2cncc(C)c2Cl)=O)C2CC3CN(C(=O)C(O)C(C)C)C1C3C2 N1(C(CCCCCCSC)=O)CC(NC(=O)CN(C)C(C)C)CC12CCCCC2 C(C(C)(C)C(=O)NC1CC(NC(c2cc(C3(C)CC3)on2)=O)C1)OC c1(CCOCCOCCOC)ccc(N(C(C)CC)C)cc1.C1CC(=O)N1 N1(C(c2c(CCC)nns2)=O)CCN(C(=O)C(C2CCCO2)OC)C2(CCC2)C1 c1(C(=O)NC)cn(CC(N2CCCC2C(C)NC(c2nnc(C)s2)=O)=O)nn1 C1(NC(=O)CN2CC=CC2)CCCCCC1NC(C1CC12CC2)=O C1(NC(CCNC(CN(C)C2CC2)=O)=O)CC2(C1)CC(C)(C)C2 C#Cc1ccc(C(=O)NCCN(C)C(C2CC23CCCOC3)=O)cc1C C(=O)(C1=C(Cl)CCOC1)N(CCCCC(=O)NCC1CCN(C)C1)C c1(C(=O)NCC(C)(O)CNC(=O)CCS(C)(=O)=O)c2c(c[nH]c1=N)CCC2 CC1(C)CCOC(C(=O)NC2(C)CC(C(=O)NCC3CCC=CCC3)C2)C1 C1(S(C)(=O)=O)(C(N(CCN(C(=O)C=C(Cl)Cl)C)C)=O)CCOCC1 c1(NCCc2ccccc2)ccc(=NCCC(F)(F)c2ccccc2)[nH]n1 c1(C(N2CC3N(Cc4cccc(OC)c4O)C3C2)=O)c(C)nc2ncccn12 N1(C(C)C)CCCCC1C(N1CCC(C(C)(C)NC(=O)Cc2nnc(O)s2)C1)=O c1(C(=O)NCC(C)CNC(=O)Cc2cc(-c3ccccc3)co2)ccncc1O N1(C(C(CC=C)N(C)C)=O)CC2CCC1C(NC(c1ccnn1COC)=O)C2 c1(CC(C)NC(=O)N)ccc(Cl)cc1CCn1cccn1.C12CC(C1)NCO2.CC N1(C(CNC(C(CC)C)=O)=O)CCC(F)(CNC(C2Cc3nccn3C2)=O)CC1 c12cccc(c1)NC(=O)CCc1nnc-2o1.Cc1ncc(C(=O)OC(C)(C)C)[nH]1 CCC(=O)CCC(=O)N1CCC1(C)CC(=O)Nc1cnc(Cl)c(C)c1 C(=O)(C1=NOCC1)NC(C(C)NC(c1c[nH]nc1-c1ccc(Cl)s1)=O)C CC1(C)CCOC1C(=O)NCC1(C)CCN(C(C2(NC(N)=O)CC2)=O)C1 C1(C(=O)NC(CCNC(CCCNC(C)=O)=O)C)CCCCN1CC(F)F C1(C)(C(N(CCCNC(=O)C(C(C)C)OC)CC)=O)CCCCCC1 C(=O)(C(CCCC)NC(=O)C(CC)CCOC)NCC(=O)OCCCC c1(SC)ccccc1.C1(C(=O)OC)CC(CCC(=O)N)(CSCCCC2CCCCO2)C1 C1(O)(CN(CCC(N)=O)C)CCCN(C(=O)C(=O)N)C1.C(c1ccncc1)=CC=O N1(C(C2(C(C)C)CCCN2C(=O)C(C)CCN(C)C)=O)CCCC(C)(N(C)C)C1 c1(C(N2CCCC(O)(CN(C(=O)CC(C)(C)O)C)C2)=O)cc2ccnc(Cl)c2s1 c1(C(=O)NCC2(NC(C(C)(C)c3ccccc3)=O)CC2)ccc2c(c1)CC(=O)N2 N1(C(COCC(C)C)=O)CCN(C(C2CN3CCC2CC3)=O)CC(C)(C)C1 c1(NC2CCN(C(=O)NC(COC)C3CCC3)CC2)nccc(N2CCCC2)n1 c1(C(N2CCC(NC(c3ccco3)=O)C(F)C2)=O)cc2cc(Cl)cnc2[nH]1 c1(C(N2CCCC(CCNC(C3(OC)CCC3)=O)C2)=O)nccc2ncncc12 C1(C(=O)NCCCCNC(CC(C)F)=O)CCC2(CCOCC2)O1 c1(CCN2CC(CN(C(=O)C(C)(F)NC(C3CCC(=O)N3)=O)C)C2)ccccc1 n1(CC)c(NC(=O)NCCc2n[nH]c(=N)s2)nc2c1CCOC2 c1(NC(C2C(CC(=O)N(CC(CC)O)C)C(O)C2)=O)nccnc1CC C1(NC(=O)C(Cl)=CCl)CCCC12CCN(C(c1cnc3ccncc3c1)=O)CC2 N1(C(CCSC)=O)CC2CC1CC2CNC(C1(c2nccn2C)CCC1)=O c1(C(=O)O)c(C(N2CCCc3sccc3C2)=O)nc2n1CCC2 C(=O)(C(CCSC)OC)NC(CC)CNC(c1occc1C)=O c1(C(=O)NCC2(NC(C34CCCCC3CCCC4)=O)CC2)ccc2ccnn2c1 c1(C(=O)OC)ccc2c(=O)n(CCN3CCCCCC3C)c(S)nc2c1 Cc1oc(CO)cc1C(=O)N(CCCSC)C.C1(NC=O)CC(F)(CNC(=O)C(C)O)C1 C1(CC=C)(C(=O)N(CCC(=O)NC2CCC2)CC(C)C)CCCN1C(C)=O N1(C(c2cccc(CCC)c2)=O)CC(NC(c2nc(O)sc2C)=O)CC12CCC2 C1(C(N2CCCC(CC3CCCCCC3)C2)=O)CCC2(CCOCC2)CO1 C(=O)(C(C(C)C)NS(C)(=O)=O)N1CCC(NC(C(c2ccc(C)s2)C)=O)C1 Cc1cc(Br)cc(NNC(=O)NC2CC(C(F)(F)F)CC(C(F)(F)F)C2)c1 CC1CN(C(=O)CCc2nccn2C)C(C)CN1C(=O)C=CC(c1cn[nH]c1)=O CC(C)C(C(=O)N1CCCCC1CN(C(=O)CCNC(N)=O)C)NC(N)=O C1(CC(=O)NCCOCCNC(=O)CCc2ccsc2)COC2CC1C2 C(C)(C)(CC(=O)N1CC(=O)CC1C(N1CC(N(C)C2CC2)C1)=O)OC O(NC(=O)C(C)C(F)(F)F)C(CC(C)C)C(=O)NC(C)(CO)CO CCC(CCC(=O)NCc1ncc(C)o1)NC(C1CCN(CC)C1)=O CN1CCN(C(c2cnn(-c3ccccc3)n2)=O)CC1CNC(C1CC1(C)C)=O C1(C)(C(=O)NCC2C(CNC(CNS(NC)(=O)=O)=O)C2)CC2(CC2)C1 c1(C(=O)NC(CCOC)CNC(=O)C(C)(C)C2CCCO2)cccc(C)c1F c1(C(=O)NCC(CO)NC(Cn2ccc(C)n2)=O)cnc(C(F)(F)F)cc1O c1(CC(=O)NCC2CCCN2C(C2SCCCS2)=O)ccncc1Cl C1(C(=O)NC2CCC(NC(C(C=C)(C)O)=O)CC2)CCC2(CC1)NC(=O)NC2=O C1(C(=O)NC2C(CC)CN(C(C3CCC(NC)CC3)=O)C2)CCc2c[nH]nc2C1 c1(C(=O)NCC2(CCNC(CC(C)SC)=O)CC2)occ2c1CCC2 C(=O)(C1=CCCSC1)NCCC1CN(C(C2(C#N)C(C)C2)=O)C1 C(CCC1CCC1)(C(=O)NCc1c[nH]c(=N)o1)NC(Cc1n(C)nnn1)=O C(=O)(CC(C)C(=O)N1CCN(CCN(C(=O)C(C)(Cl)Cl)C)CC1)OC CCCC(C(=O)N(C1CCCC1)CCCNC(c1coc(Cl)c1)=O)N(C)C c1(C(C)C)cccc(C(c2nnnn2C(C)C)NCC(C)OC(F)F)c1 CC(C)(C)C(=O)NCCN(C(=O)C=Cc1ncco1)CC1CCCCC1 c1(C(=O)NC(CC)CN(C(=O)C(O)C2CC2)CC)cccc2nc(O)ccc12 c1(NCC(COC)(F)F)nc(=NC(C)c2nnc(CO)s2)[nH]c2c(C)nn(C)c12 C(=O)(C(F)C(F)(F)C(F)(F)F)N(CCNC(c1c(C)nc(C2CC2)nc1)=O)C C(=O)(CCC(=O)NC1C2CC(NC(=O)CC3C=CCC3)CC12)NCCC c1(CCN2CC(C)(CC(=O)OCC)C2)nnc(C(C)(C)C#N)o1 c1(C(=O)NC(C(C)NC(c2cn(C)cn2)=O)C)cc2ccccc2c(O)n1 C12CN(CCO1)C2=O.C1(C)(CNC(C2N(C(=O)NC)CCC2)=O)CCCN1C c1(C(=O)NCC(CC)NC(C2CC(O)(C#N)C2)=O)cnc2ncnc(O)c2c1 c1(C(N(C2CCN(C(c3cccc(-n4cccn4)n3)=O)C2)C)=O)ncccc1Br c1(C2N(C(=O)NCCNC(CC3(NC(C)=O)CC3)=O)CC2)ccccc1 N1(C(C2CC23CCC3)=O)CCN(C(C2CCc3nn[nH]c3C2)=O)C2(CC2)C1 C1(NC(c2c(C)cnnc2)=O)CC2CN(C(C3(C)CC4CCC3C4)=O)CC12 C#CCC(C(=O)OCC=CC#N)NC(=O)C(Cc1ccc(C)cc1)N(C)C C1(=O)C(C(C)O)N1.C1(C(N(CC(C)OC)C)=O)CC(C(F)F)C1 Cc1c(F)ccc(Cl)c1C(N1CCOC(C(F)(F)F)C1)=O C1(CCCNC(c2cncc(O)c2)=O)CN(C(c2cnccn2)=O)CCO1 c1(NCC(=O)NC2C3CN(C(CC4(C)CCCCC4)=O)CC32)ccc(F)cc1F C(N=c1cc(Cl)nc(C2CC2)[nH]1)C1CCN(C(c2cnc3[nH]cnc3c2)=O)C1 C1(N(C(=O)CC2(O)CCC2)C)CN(C(c2[nH]ccc2C2CC2)=O)CC1(C)C N1(C(C=C(COC)C)=O)CCC(C(C)CNC(=O)COC2CCC2)CC1 C=CC1OCCCC1C(=O)NCC(CC)NC(=O)C(c1cnccc1C)(C)C c1(C(=O)OC)nc2[nH]c(=NCC(C)Cc3ccco3)ccc2o1 c1(OC)ccc(C(C)C(=O)NCC(C)CNC(=O)C(=O)N(C)C)cc1OC S(=O)(=O)(c1ccc(NCC(F)C2CCC2)nc1)CCOCCOCCOC C1(C(=O)Nc2c(OC)cc(I)cc2)CCC2(CCN(Cc3scnc3Cl)CC2)O1 C1(N(C)C)CCCN(C(=O)C(C)(CO)NC(=O)NC2CC2(F)F)C1 N1(C(CCCC)=O)CC2(CCN(C(c3cccnc3O)=O)CC2)C1C(C)C CCC(CCC(=O)Nc1cccc(Cl)c1O)NC(C1CC1C1CCC1)=O N1(C(c2c[nH]c(=N)o2)=O)CCOC(C(N2CCCC(CCCO)C2)=O)C1 c1(OC)cccc(CC2C3CN(C(=O)C(N4CCSCC4)C)CC23)n1.CC=O Cc1nccnc1C(=O)NCC1COCC1NC(=O)C(O)C1CCC1 C1(C(=O)Nc2cnn(C)c2)(COC)C=CCN1C(C1C=CCCC1)=O C(=O)(C(O)CCC(C)C)NCC1(NC(c2scc(OC)c2OC)=O)CCOC1 c1(C(N2CCC(CNC(C(n3ccc(C(F)(F)F)n3)C)=O)C2)=O)cnnc(O)c1 c1(OC)ncnc(C)c1C(=O)NCC(C)N(C(=O)CN1CC(CF)C1)C c1(CC)nc(=N)[nH]cc1C(=O)NCCN(C)C(c1ccncc1Br)=O O=C(C1=CNC2=NCCC2=C1)N1CCC1CNC(c1cc2c(Cl)nccc2o1)=O N1(C(CCSC)=O)CC(C(C)(C)C)CC(CNC(=O)C(c2cnn(C)c2)O)C1 c1(C2CN(C(CNS(CC)(=O)=O)=O)C2)cn(C2CCc3cccnc32)nn1 N1(C(C2(CCOC)CC2)=O)CC(N(C(=O)CC(C)C2CC2)C)C2(CC2)C1 C1(C(N(CCCC(=O)NC(c2c(C)ccnc2)C)C)=O)CCCC(C#N)C1 C(C(C)(C)C(C)(F)F)NC(c1ccc(CNC(c2c(C)cccc2)=O)cn1)=O c1(C(N2CC(CCNC(C(C)OCC)=O)C2)=O)ccc2ncc(Br)n2c1 c1(SCC(=O)NCC(CN(C(c2c(CC)ocn2)=O)C)C)ccc([N+](=O)[O-])cc1 C1(N(C(Cc2c(C)con2)=O)C)CCC(NC(=O)Cn2cc(Cl)cn2)CC1 c1(CC(N2CCCC(C(=O)NCc3cccs3)C2)=O)ccc2c(c1)OCCCO2 c1(CC)ccccc1-n1nc(CCC(F)(F)F)nc1C1CC2(CC2)C1 C(=O)(C(C)(C)C(N)=O)NC1CCN(C(CC(COC)C)=O)C1C(C)(C)C c1(C(N2CC(C(N)=O)CC(C)(C)C2)C(=O)NCCSC)cc2c(nn1)CCCC2 c1(C(=O)NCC=CCNC(c2nn(C)c(Cl)c2)=O)c([N+](=O)[O-])cnn1C(C)(C)C N1(C(CCCOCC=C)=O)CCC(N2CCN(C(C3CCC(F)C3)=O)CC2)CC1 c1(C(=O)CF)ccc(O)c(C(=O)NC2(CNC(C3C=CCC3)=O)CCCC2)c1 c1(C(=O)NC2CN(C(CCC#C)=O)C(CC)(CC)C2)ccc2c(=O)ccoc2c1 C#CC(C(C)(C)C)NC(=O)C(CC)NC(C1CC(=O)CCO1)=O C1(NC(c2ccc([N+](=O)[O-])cn2)=O)CC2CC(C1)CN(C(c1nocc1Cl)=O)C2 C1(C(=O)NC(CNC(C2CCC(OC)CC2)=O)CC(C)C)CCCC1S(C)(=O)=O N1(C(CCSC)C)CCC1.C12(CCSCC1)C(=O)N2 N1(C(COCCCC#C)=O)CCC(C(=O)N(CCC(C)C)C(C)C)CC1(C)C N1(C(c2c(C)nn(C)c2)C(=O)NC2CCCCC2)CCCCC(CO)C1 C1(C2CC2)(C(=O)NCCCCCCNC(=O)C(F)n2cccn2)CC=CC1 N1(C(Cc2c(OC)cc(Cl)cc2)=O)CC(NC(C2CCCCO2)=O)CC12CCC2 c1(C(=O)NC2C(CC)CN(C(=O)C(F)n3cccn3)C2)ccc(C)c(=O)o1 c1(CCC(=O)NCC2CCC(NC(=O)CC3CCCO3)CC2)cncc(Br)c1 C1(CCC(=O)NCC2(CNC(c3n(CC)ccn3)=O)CCC2)CCCC(O)C1 C1(C)(CC)C=C(C(=O)NC2(N(C3(NC)CC3)C)CC2)C1.C1=CC(C)NC1=O C1(NC(c2c(OC)ccnc2)=O)(CNC(C2CCOC2=O)=O)CC2CCC1CC2 N1(C(=O)OC(C)(C)C)CC2CC(NS(=O)(=O)Cc3ncccc3C)C1C2 C12(CNC(c3nc(CC)oc3)=O)CN(C(C3CC3F)=O)CC1CCO2 N(C(=NCCC1CC1C)NCC1CCOC1)CC1(CC)COC1 c1(NC(=O)NCC2N(C(C3(c4cccc(C)c4)CC3)=O)CC2)cc(C)ncc1C C=CCC(C)C(=O)N(C1CN(C(=O)C(C)(C)Cc2cccc(Cl)c2)C1)C C1(CNC(C(CC#C)C2CC2)=O)CC(C)(C)CN1C(c1nccc(OC)c1F)=O C1(CN(C(=O)C(C#N)CC)CC)CCCN(C(C2CCC(COC)C2)=O)C1 C(c1ccco1)=CC(N1C(CC(=O)NCC2COC(=O)N2)CC1)=O O=S(=O)(CCNC(c1cc(C2CC2)nc2ccccc12)=O)c1ccccc1 c1(C(=O)NCC2C=CC(NC(C(CC)NC(C)=O)=O)C2)nccc(OC)c1F c1(C(N(C2CCN(C(CCC=C=C)=O)C2)CCC)=O)c(C)cc(C)nc1O Cc1ccc(Cl)c(C(N2CCCN(C(c3occ4c3CCC4)=O)CC2)=O)c1O Cc1ccc(C(=O)N(C)CCN(C)C(C2SCCC2C)=O)n1C c1(C(=O)NC2C3CN(C(C(=O)NCCOC)=O)CC32)c(OC)cc(OC)cc1C C1(NC(c2ccnnc2Cl)=O)CCCN(C(c2ccc(CF)cc2)=O)C1 N(C1CCCn2nccc21)C(C1CCN(C(C(CC)C#N)=O)C12CCC2)=O C1(N(C(c2cc(CCC)n(C)n2)=O)C)CN(C(c2cc(CO)[nH]n2)=O)CC12CC2 CC1CCc2nc(C(N3CCC(CCNC(=O)CC(C)(C)F)CC3)=O)cn2C1 C(=O)(CC(C)(C(F)(F)F)N(C)C)NCC1C(NC(Cc2cc(C)[nH]n2)=O)C1 N(C1CCc2c1ccc(Br)c2F)CC(=O)NCc1ccc(C#C)cc1 C1(OC)CC(CCNC(C2(C)CC3(CC3)C2)=O)N(C(c2ccoc2C)=O)C1 N1(C(=O)C2=NOCC2)CCN(C(C2CC(C(F)F)C2)=O)C(C(F)(F)F)C1 c1(CC)cc(-c2ccccc2)n(C(C)C(=O)NCCc2cccc(O)c2)n1 c1(C(=O)NC2C3CN(C(C(C(C)C)SC)=O)C2C3)nnc(O)c(Br)c1O C(=O)(C1CCCc2c[nH]nc21)NC(CN(C(c1c(F)cc(CC)cc1F)=O)C)C c1(C(=O)NC(C2(C(=O)NC3CC(F)C3)CC2)C)c(NC(N)=O)cccc1F C(=O)(C1=CCCC1C)NCC(CCNC(C12CC(C(=O)OC)(C1)C2)=O)OC C(N=c1nc2c(cnn2C)c(NC(C)Cc2ccc(C)nc2)[nH]1)C1(CC=C)CC1 CS(=O)C1CN(C(CCC2CCCO2)C(=O)NC2(CC(=O)OC(C)(C)C)CC2)C1 c1(C(=O)NCCC(CCNC(C(CC(C)C)O)=O)C)cc(S(N)(=O)=O)co1 C12(C(N(CCC)C)=O)CC(C)(CN1C(=O)C(C)(C)CC1CC1)C2 C(C(=O)NCC1CN(C(C2(O)COC2)=O)CC1O)(C(C)C)NC(C)=O Cc1cc(S(N)(=O)=O)cc(Br)c1C(=O)NCC1(Cc2cccc(F)c2)CC1 N1(C(C(COCC)(C)C)=O)CCC(NC(=O)Cc2nn(C)cc2Cl)C(C)C1 C1(NC(c2cc(C)no2)=O)CN(C(C2(C(F)(F)F)CCCCO2)=O)CCC1F C1(NC(c2c(N(C)C)cccc2)=O)CCOC2(CCN(S(=O)(=O)C(F)(F)F)CC2)C1 NC(=O)CCCC(=O)N1CCC(F)C(NC(=O)C=Cc2cccc(CO)c2)C1 CCCCC(O)C(=O)N1CC(=C(F)CNC(c2cccn2Cc2ccccn2)=O)C1 C1(NC(=O)CCSC(F)(F)F)CCCC2CN(C(c3cncnc3)=O)CC12 CC(C)(C#N)CCN1CCC(NC(=O)NCC(C)(C)C)C1=O C1(CC(N2CCC(Sc3cc(Cl)ccc3Cl)C2)=O)(C(=O)O)CCCCCC1 C1(NC(NNC(=O)NC)=O)CCCC2CCCCC12 C(=O)(N=c1cc(-c2ccccc2Cl)o[nH]1)C1(C(N)=O)N(C)CC(O)C1 N1(C(CC(C(C)C)O)=O)CCCC2(CC(NC(C3OCCCO3)=O)C2)C1 c1(C(=O)NCCC2(NC(C=CC(C)C)=O)CC2)cc(O)nc2ncccc12 CC1CC(c2nnnn2C2CC2)(NC2CCC2)CN1CCOC(C)(C)C C1(NC(c2c(C)nsc2C)=O)CCN(C(=O)C2CC2)CC1C CC(CC(=O)NCCC1CCN(C(=O)C(N2CCCC2)C2CC2)CC1)P(C)(C)=O C=CCCCCCC(=O)NC1CC(C)CN(C(c2ncc(C)cc2C)=O)C1 N1(Cc2cn(CC3S(=O)(=O)CCCC3)nn2)CC2CC(F)CC2C1 C(N=c1cc[nH]c(=NCCN2CCCOCC2=O)[nH]1)c1nc(=N)[nH]c2c1scc2 Cc1coc(C(=O)N(CC(C)NC(c2ccco2)=O)C)c1 C=CCC(C)(C)C(=O)NC(C)C(C(C)C)NC(c1nccnc1C(N)=O)=O C1(CC=C)(C(=O)NCCCCNC(N)=O)CCCN1C(c1ccc(CC)cc1)=O C12(C(NOC(C(=O)OC)(C)C)=O)COC(C1)C(NC(C1(C)CCCCCC1)=O)C2 c1(C(=O)NC(C(C)C)CNC(C2CC3C(C2)C3(F)F)=O)ccc2[nH]c(=N)oc2c1 c1(C(N(C(C(=O)NOC2CC3CCC2C3)C2CC2)C)=O)ccc2cccnn12 C(=O)(CC(O)CC(C)(C)C)N1CCC(C(C)C(N2CCN(CCO)C(=O)C2)=O)CC1 C1(C(N2C(C(N3CCCC(OCC(F)F)C3)=O)CCCC2)=O)CC2CC1CC2O C(=O)(C1CCc2nccn21)NCC(C)(C)NC(c1cccc(C(C)(F)F)n1)=O N1(C(c2c(C)nn(C)c2C)=O)CCC2(CC1)CC2NC(=O)Cc1n[nH]cc1Br c1(C(=O)NC2CCC(NC(C3C(=C)C3)=O)CC2)nc2nc(C)cc(C)n2n1 C(=O)(C(C(C)(C)C)NC(C)=O)NCCCNC(C1CC(C#N)(OC)C1)=O CCC(CC)(C(=O)NCC(F)CNC(c1cc(C)cc(C)n1)=O)c1ccccc1 Cc1cc(F)ncc1C(N1CCC(CN(C)C(c2ccccc2Cl)=O)C1)=O C(=O)(C(O)CCSC)NCC1(NC(c2ccc(COC)[nH]2)=O)CCCC1 C1(NC(C2CCN(CC#C)CC2)=O)CCCC(S(=O)C(F)(F)F)C1 C12(CNC(c3nc(CCC)sc3)=O)CC(CC)(CN1C(C1CCCC1O)=O)C2 C(CCC(C)C(=O)N1CC(CNC(c2cccn2C(C)C)=O)C(C)C1)OC N1(C(CC(CC)SC)=O)CC2(CCC(CNC(c3cc4[nH]ccc4s3)=O)O2)C1 CC1(C)Cc2[nH]nc(C(=O)NCCCC3CCCN3C(C3CC=CCO3)=O)c2C1 CC1CCC(OCC(N2CC(CC(C)NC(c3ccc(CO)nc3)=O)C2)=O)CC1 C1(O)(C(C)NC(=O)C=Cc2cc[nH]n2)CCN(C(C2C3COCC23)=O)CC1 N1(C(c2c(COC)noc2)=O)CCCC2(NC(=O)Cn3ccc(C)n3)CCCC12 C1(CNC(=O)Cc2ccns2)CCCCCN1C(C1CCCOC1)=O C1(C(=O)OC(C)(C)C)(CCNCCCCc2nccs2)CCC1 N1(C(CSC(C)C)=O)CC(N(C)C(C2CC3(CC3)CN2C)=O)C(C)(C)C1 CC1CN(C(C2CC2(C)C)=O)CCCN1C(=O)CCOc1c(F)cccc1Cl C1(C)(COC)CC(NC(=O)CC2(CO)CC2)CN1C(c1cnoc1C)=O C1(CC)CN(C(=O)CCN(CC)CC)CCN1C(=O)CC(C)C(C)C c1(N2CCC(CC)C2)nc(=NCCC2CC(=O)N(C)C2)[nH]c2c1SCC2 CCCCCC(O)CC(=O)NCC1=NOC2CN(C(=O)CC(C)(C)OC)CC12 C(=O)(C1=NNC(=O)CC1)N1CC(O)(CN(C(CC(N2CCCCC2=O)C)=O)C)C1 C(=O)(C#CC1CCOCC1)N1CC2(CCN(C(C3CC3c3ccsc3)=O)C2)C1 n1(CC(=O)OC)nccc1OC1CN(C(=O)OC(C)(C)C)C1 c1(C(=O)NCC(CNC(C(C)(C)OCC)=O)(C)O)cc2sc(C(=O)O)cc2[nH]1 CC1CCC(C)N1C(C)C(=O)NC(CNC(C1CC(C)C1)=O)Cn1cccn1 c1(CCC=C)ccc(C(=O)NC(CNC(=O)C(C)CF)CCOC)cc1 C12(C(=O)O)CCC(C(=O)Cc3csc4cncn34)(CC1)CC2 c1(NC(C(=O)N(CCCCC(C)C)C)=O)ccc2ncccc2n1 C(CCCC(=O)NCC1(CC)CCOC1)N(C(Cc1c(CC)con1)=O)C CC1CN(C(=O)Cc2cn(C3CC3)cn2)CCN1C(C1CCSC(C)C1)=O c1(CCC(=O)N(C(C)CNC(=O)C(C)n2cccc2)CC)cccc(C)c1 C1(NC(c2cc(C(=O)OC)ncc2)=O)CCCN(C(C2CCC(F)(F)C2)=O)CC1 C12(CCCN)CC(C(=O)NCCc3ccc([N+](=O)[O-])cc3)(C1)C1(CCC1)O2 C1(C(=O)NCC2C(NC(=O)OCC)C2)(COC)CCC1.C12CN(C1)C2=O c1(C(=O)NCCC(CNC(CSc2ccc(C)cc2)=O)O)cc(C)c(O)c(N)c1 c1(C(N(CCNC(C(C(CC)CC)C)=O)CC)=O)cc(OC)c2c(c1)OCO2 N1(C(CNS(N(C)C)(=O)=O)=O)CCC2OCCN(C(C3CC4CC4C3)=O)C2C1 N1(c2cc(C)nc(N3CCOC(CO)C3)n2)c2ccccc2CCC1C c1(C(=O)NC2CC(C)CN(C(=O)CC3CSCCS3)C2)ccc2c(c1)CCCC2=O c1(COC(C(N2CC3C(NC(C(C)N(C)C4CC4)=O)C3C2)=O)C)ccnc(Cl)c1 N1(C(C(c2cccs2)NC(c2cccn(C)c2=O)=O)=O)CCC2C(O)C(C)(C)C12 Cc1nc(C(=O)NC2(C(=O)Nc3ccccc3C)CCCCC2)cc(O)n1 C(=O)(C(C)CC(=O)N1CC(N2CCN(C(=O)COCC3CC3)CC2)C1)OC Cc1cc(NC(C2CC(F)CN(c3ncncc3F)C2)=O)cc([N+](=O)[O-])c1C C(=O)(C1=CCCC1C)N1C(C)(C(N2CC(C#C)(F)C2)=O)CCC1 N1(C(CN(CCC)C(c2cnc(=N)[nH]c2)=O)=O)CC2(CCCC2)C1 c1(C(=O)NCC2CC(C)CN(C(C3CCC3(F)F)=O)C2)ccn2ccnc2c1 c1(C(=O)NCC(CN(C)C(C2CCCC(CF)C2)=O)O)cccc2nc(O)oc12 Cc1nccc(C(=O)NCc2csc(CNC(=O)C3=CSCS3)n2)c1C c1(OCC)ccccc1C(C)NC(=O)CC1CCCS1 CC1(CNC(c2n[nH]c(C3CC3)n2)=O)CCN(C(c2n[nH]cc2F)=O)C1 N1(C(C(C)=CC2CC2)=O)CCC(C(=O)NCCc2ccccc2O)C(C)C1 c12ncc(C)cc1S(=O)(=O)NN2.c1(C)c2ccc(c1)o2.C=C(Br)COCCO.CC c1(CCC(N2CCC(N(C(C3CC(=C)C3)=O)CCC)C2)=O)cccnc1Cl CON1CCC(CC(N2CC(NC(=O)COCCN(C)C)CCC2C)=O)CC1 c1(-c2n(C(C=C)C)nc(CC(C)CC)n2)ccc(C2=CCCC2)cc1 C(=O)(C1=NOCC1)NCC(C)(Cn1cccn1)NC1COC(C)(C)C1 C1(C(=O)NCCCOCCCNC(C2CC(CC)C2)=O)C(C#N)C1(C)C Cc1cccc(C2(C(=O)NC3CCCC3NC(c3scc(C)c3C)=O)CC2)c1 C#Cc1cc(F)c(C(N2CC3(NC(c4ccc[nH]4)=O)CCC2C3)=O)cc1F C(=O)(CS(=O)(=O)CCO)N1CC(NC(c2c(CC)ccc(F)c2)=O)C(C)C1 CCC(CCC(=O)NC1(C)CCN(C(c2ccc(N)cc2Br)=O)C1)OC c1(C(=O)NC(CN(C(c2nc(C(F)(F)F)ccc2F)=O)CC)C)cccc(O)c1F c1(CC(=O)Nc2c(C)cnc(C)n2)ccc(F)cc1[N+](=O)[O-] c1(C(N(CCNC(C2CC2NC(C)(C)C)=O)CC)=O)ccc(NC(C)C)cc1F C1(NC(Cc2c(C)nccc2)=O)CC(C)CN(C(c2cncc(C)c2)=O)C1 CCCC(CC(C)C)C(=O)NCC1CC(NC(c2ccc(O)cc2C)=O)C1 Cn1nc(-c2c[nH]c3cccc(Br)c23)c2cc(C3=COCCC3)sc12 N1(C(c2c(C)cccc2[N+](=O)[O-])=O)CC2CC(O)C(O)CC2C1 Cc1cn2c(C(N3CCN(C(C4(n5cnnn5)CC4)=O)C(CO)C3)=O)cnc2s1 c1(C(C(=O)N(c2cn(C(CC)C3CC3)nn2)C)C)cc(F)ccc1Br C1(C(N(C(C)C(N)=O)C)=O)OCCC1CNC(C1CCN(C)C1)=O C#Cc1ccc(F)c(C(=O)NCC(C)NC(C2CCN(CCO)C(=O)C2)=O)c1 CCC(C(=O)NCC1(F)CCCN(C(=O)C(C)(C)c2ccsc2)C1)C(C)(C)CC C(C(C)C(C)C(=O)N1CCC(N2CCN(C(C3CCC(F)C3)=O)CC2)C1)OC C(=O)(C(C)(C)C1=CCN(C(=O)C(O)CC2CCCC2)C1)N1CC(C)C(O)CC1 c1(C(=O)NCCOCCCN(C(C2C(C)OCC2)=O)C)ccc(CN=[N+]=[N-])cc1 c1(SC)cc(C)c(C(=O)NCCCC(C)NC(=O)CCOc2ccccc2Cl)o1 C(=O)(C1CCCc2nn(C)cc21)N1C(C(C)NC(c2cc(Cl)no2)=O)CCC1 CC(C)CC(C)C(=O)NC1CN(C(c2ccc(F)s2)=O)C1 c1(C(=O)NC(C)C(CO)NC(N)=O)cccc(NC(=O)CSCC2CCCC2)c1 c1(CC)noc(CCC(=O)N(CCN(C(C2CC2Cl)=O)CC)CC)n1 CC1CCCC1CNC1CCC1(C)C.c1(CC=O)nnnn1-c1ccccc1 Cc1cc(=NC2CN(C(=O)CCc3cc(F)ccc3F)CC2(C)C)[nH]cc1C#N C(=O)(C(CO)C(F)(F)F)NC1CCCC(N(C(Cc2cc(CC)nn2C)=O)C)C1 C1(CC(=O)NCC2CC(N(C(=O)C(O)c3ccco3)C)C2)CCC(=O)CC1 N(C(=NCC(C)C(F)F)NCc1cc(C)on1)CC(C)Oc1c(OC)cccc1 c1(CC(=O)NC(CNC(c2ccn(CC)c(=O)c2)=O)C)c(Cl)ccc(O)c1Cl CCC(Cc1ccccc1)CC(=O)NCCNC(c1cnc(C(F)(F)F)cn1)=O N1(C(C2(CSC)CC2)=O)CCC(C)N(C(=O)COCC2CCOC2)CC1 C1(C(N2CCCC(CN(C(=O)C(O)C(C)C)CC)C2)=O)CCC(O)CN1C O=[N+]([O-])c1ccc(F)cc(N(C2CCCCC2)Cc2cncnc2)c1=O c1(C(N2CCC(C(N3CC(C)(C(F)(F)F)C3)=O)O2)=O)cc2cc[nH]c2cn1 CC1CN(C(=O)Cc2ccn(C)n2)CC(C)C1NC(=O)Cc1ccccc1F C1(NC(C2(OCC)CCC2)=O)CCC(C)N(C(C2CC3(CCC3)C2)=O)C1 c1(C(=O)NCC(c2ccc(Br)c(F)c2)C)cnn2c(C(=O)O)ccnc12 Cc1nn(Cc2nc(COCC(C)N)no2)c(=O)c2ccccc12 c1(C(=O)NC2CC(CNC(c3c(C)coc3C(C)C)=O)C2)c(C)nc(C)n1O C(=O)(CCCC(=O)NCC(C)NC(C1CCCN1CC(C)C)=O)NCCC C12(CNC(C3(CC#C)CC3)=O)CC1CN(C(C1CCCN(C(=O)N(C)C)C1)=O)C2 N1(C(C2C(C(C)C)(CC)C2)=O)CCN(C(=O)CCOCCN(C)C)C2(CCC2)C1 Cc1cc2occ(CC(=O)NC(CCc3ccccc3)CC(F)(F)F)c2cc1C CC1CC(C)N(C(=O)CN(C)CC)CCN1C(=O)CCc1cccnc1F.C1CCC1 Cc1cn(C)nc1C(=O)N(C)CC1(O)CN(C(c2c(C)nsc2NC2CC2)=O)C1 N1(C(c2cc(CC)nn2C)=O)CCOC2CN(C(c3coc(N(C)C)n3)=O)CC12 Cc1nnc(N2CCCC(CCNC(C3CC4CC3C3CC43)=O)C2)c(C#N)c1C N1(C(=O)CC2CCS(=O)(=O)C2)CC(C2CN(C(=O)CCCF)C2)C1 CCCC(CC(=O)N(C)Cc1cccc(C)c1)NC(C1CN(CC)CCO1)=O N1(C(C(SC)SC)=O)CCC1(C)CC(N1CCC(CC2CC2)C1)=O CCC(C)CCC(=O)NCC1(C(N)=O)CN(C(c2cc(C(C)(C)C)on2)=O)C1 N1(C(C#CCNC(C2C(CC(C)(C)C)C2)=O)=O)CCCC(C)(C#N)C1 c1(C(C(C)NC(=O)C(=O)N2CSC2C2CC2)=O)ccc(F)cc1 C(=O)(CC(C)(C)C(=O)NC1CN(C(=O)C(N2CCCCC2=O)C)CC12CC2)OC c1(C(N(C2CCN(C(=O)CCC(C)(C)C)C2)C)=O)cnn2c(=N)[nH]cnc12 Cc1cc(NC(=O)C(C)OC(=O)Cc2cc(C)n(C)n2)cc(Cl)n1 O=C(CN=c1ccc(F)c(Br)[nH]1)NCCCn1c(=O)oc2ccccc12 C12(NC(c3cnn4cccc(Br)c34)=O)CCCC1(F)CN(C(=O)CO)C2 C1(CCNC(c2cnc(S)n2C2CC2)=O)CN(C(C2CCCOC2)=O)CCO1 N1(C(C2(OCC)CCC2)=O)CC2CC(NC(C3COCCN3C=O)=O)CC2C1 c12cnn(c1C)CCN(CC)CCN(C1CC(C(=O)OCC)C1)C2=O.CC c1(C(=O)NCC(C)CN(C)C(C2CC3(C2)CC(O)C3)=O)ccc2c(c1)C(C)CO2 c1(OC)ccc(C(=O)NCc2cccc(CNC(=O)C=CSC)c2)c(N)c1 CC1(C(N2CCC(O)(CNC(C3(N(C)C)CCCC3)=O)C2)=O)CCC(=O)N1 c1(CNC(CC2OCCN(C(C(C)=CC3CC3)=O)C2)=O)nc(C)cc(C)n1 n1(CC(=O)NC2(CNC(CCCCOCC)=O)CC2)cnc2ccc(C)cc12 c1(C(=O)NCC2(C)CCN(C(C(C)C#N)=O)C2)ccnc2ccsc12 C(C(=O)NCC1(C)CC1)(C(C)CC1CC1)N1CCCC(c2nc(C)[nH]n2)C1 N1(C(C(C#C)(C)C)=O)CCC2(CC1)CC2CNC(=O)C(C)(Cc1ccccc1)CC c1(OC)ccc2c(C)c(C(N3CCC(C(C)NC(=O)C=C(C)C)C3)=O)[nH]c2c1 c1(CCC(=O)NC2CN(C(C3(CC)CCCCC3)=O)C2)cc(Br)ccc1F CC1=CCC(C)(C(c2nnnn2C2COC2)NC2C3CCC2CC3)CC1 c1(C(N2C(CCNC(C=Cc3nc(C)sc3)=O)CCC2)=O)cn2ccncc2n1 C1(CF)CC2(CCCC2)CO1.C12(CC=C)CCN(C1)C(=O)CCC1CC1C(=O)N2 CCC1=C(C(=O)N2CCC(O)(C(C)NC(c3csc(Cl)n3)=O)CC2)SCCO1 C1(NC(C2C(=C)C2)=O)CC2CC(NC(=O)NC3CNC3c3ncccc3F)C2C1 c1(C(=O)NC2C(NC(C3CC(OC)C3)=O)CCCC2)cc(F)cc2c1CCC2 C1(NC(CS(CC)(=O)=O)=O)CCCC2CN(C(C3(C#N)CC(=O)C3)=O)CC12 c1(C(=O)NCC2N(C(C(C)S)=O)CCOC2)ccc2c(c1)CCCO2 c1(C(=O)NC2C(CNC(CN(CC)CC)=O)C2)csc([N+](=O)[O-])c1 C1(NC(c2cc(Cl)c(Cl)[nH]2)=O)CN(C(=O)CC2(CO)CC2)CC12CCOCC2 C#CC1(C(=O)NCC(C2CC2)NC(=O)C(C)Oc2ccc(Cl)cc2)CCOCC1 C1(n2cc(CC(C=C)O)nn2)CCCN(C(=O)Cc2ccc(OC)cn2)C1 CCC(CC)C(F)C(=O)NC1CC(C(=O)NCCCCCCCO)C1(C)C N1(C(c2cc(CC)on2)=O)CCC2(NC(c3c[nH]cc3Br)=O)CC2C1 Cn1cc(CNCc2ncon2)cc1C#N N1(CCNC(Cn2cc(CN)nn2)=O)CC2CCCCN2C1=O N1(C(CCCC(=O)NC2(CNC(=O)CC)CC(=C)C2)=O)CCC2CCC(C1)N2 C1(CCCNC(C=CCOC)=O)CCCCN1C(C1CC2(CSC2)C1)=O C(=O)(C(CN(c1ccccc1)C)C(C)C)NCCOCCN(C(C1C(C#C)C1)=O)C c1(OC(C)C(N2CCC(C(O)CO)CC2)=O)cccnc1O N1(C(C2C=C(C)CS2)=O)CCC(C2(NC(=O)CC3(C)CC3(F)F)CC2)CC1 Cc1cc(NC(=O)CCCC#N)ccc1NC(=O)CCC(C)(C)c1ccccc1 N1(C(Cc2cc(CC)no2)=O)CCC(CC)(NC(=O)CC2CCCN2C)CC1 c1(C(C(N2CC(CC(C)NC(=O)CC3CCCOCC3)C2)=O)O)cccc(Cl)c1 C1(C2CCN(C(C3CN4CCCN3CC4)=O)C2)(NC(C(C)CCN(C)C)=O)CC1 C(=O)(C(C)(C)CN(C)C(C1CC1Cl)=O)NCCC1(OC)CCC1 N1(C(C(C(C)C)C#N)=O)C(C(=O)NCC2(C)CSC2)C2CC(O)C1C2 Cc1cnc(C(N2CC=CC2CNC(=O)COc2cc(F)cc(F)c2)=O)c(F)c1 Cc1cc(C)c(CC(N2CC(C3(NC(c4ccns4)=O)CC3)C2)=O)c(C)c1 c1(CCC)n[nH]c(=NC2CCCC3CN(C(=O)C(=O)CC(C)C)CC23)s1 C1(NC(C2N(CC)CCC2)=O)CN(C(=O)C#CC(C)(C)O)CC1N=[N+]=[N-] C1(C(=O)NCc2n(C)ccc2)CC2(CCC2)CN1C(=O)C1=CCCCC1 C(c1cccnc1)=CC(=O)NC(C)C(=O)NCC(C)C.C(C1C(=O)NCC1)OC C(=O)(CC1=CCN(C)CC1)N(CC(CNC(C(CC)CC1CCCC1)=O)O)C c1(CCO)cccc2c(C(C3CCC3)Nc3csnn3)cccc12 c1(OC)ccc2occ(C(N3C(C)C4CC3C4NC(=O)CCC=C(C)C)=O)c2c1 N1(C(COCCCC#C)=O)CC(NC(=O)C(C(C)C)N2CCCC2=O)C(CCC)C1 c1(C(=O)NCC(CNC(C=C(CCC)C)=O)O)ccc(O)cc1C(C)=O N1(C(=O)NCCCC)CCc2c(NC(C3CCOC3)=O)cccc21 CCCC(C)(CC)C(=O)N(CCCCN(C)C(C1CCCC12CCOCC2)=O)C N1(C(C(C)NC(N)=O)=O)CC2CCC(CNC(=O)C(C)(F)C(C)(C)F)C2C1 c1(C(=O)NC(C)CCCS(C)(=O)=O)cnc2c(ccn2C)c1 c1(C(N2C(C(=O)Nc3ccc(CC#N)cc3)CC3CC32)=O)c[nH]c2ccccc12 c1(C(=O)NCCOCCN(C)C(c2cc(C(F)F)on2)=O)ccc(C(F)(F)F)o1 N1(C(c2c(N)cccc2)=O)CCN(C(c2ccco2)=O)CC1CC(F)F C(=O)(CCCC(F)(F)CO)N1CCCCCC1.C1(CNC(COC)=O)CCS(=O)(=O)C1 N#CC1(C(=O)NCc2cc[nH]c2C(N2CCOCC(O)C2)=O)CCCOC1 CCCCCC(O)CC(=O)N1CC2(CCN2C(=O)CSc2cn[nH]c2)C1 Cc1cccc2c1N(C(=O)NC1CCCN(c3ccccc3F)C1=O)CCC2 C(=O)(C1=CCC(C)CC1)NC(CC)CNC(c1c[nH]c(=O)cn1)=O C12(NC(c3cn[nH]c3)=O)CCCN(C(c3ccc(-c4cnn[nH]4)cc3)=O)CC1C2 N12CCC(C(F)(F)F)C(C1)C2=O.C1(O)(CS(=O)(=O)N)CCCC1 c1(C(C(=O)N(CCNC(C(C2CCCN(C)C2)(C)C)=O)C)O)ccc(F)c(Cl)c1 c1(OC)cc(C(N2CC(C3(NC(=O)CNS(=O)(=O)CC)CC3)C2)=O)c(N)cc1F c1(C(N(C2CCN(C(C(C(C=C)C)C)=O)CC2)CCC)=O)cnc2ccsc2c1 c1(C(=O)NC(C(C)NC(=O)COCCN(C)C)(C)C)cccc2nsnc12 C1(CCC)CCCC1NC(C1CC1(C)C(=O)OC)=O N1(C(C2N(C(=O)C3=CCCC3)CSC2)=O)CC2(CCCC2)C1c1ccccc1 CCC(CC)(C(=O)N1CCC2(CC2C(=O)NCC(C)CC(F)(F)F)C1)OC Cc1cc(CN(C)C(C2CCN2C(c2cocc2C)=O)=O)on1 C(=O)(C(CCCC(C)C)N1CCC(SCC(F)(F)F)C1)NCCCC C1(C(N2CC3C(CNC(c4n(C)cnc4)=O)C3C2)=O)C2Cc3ccccc3C12 CC1CC(=O)NC(C(=O)NC(c2ccccc2)CNC(=O)CCCN(C)C)C1 C(CC)(C(=O)NCCOC(C)C(=O)NCC(O)CF)=CC CCCCC(O)C(=O)N1CC(O)CC1Cn1cc(-c2ccc(C(=O)O)cc2)nn1 C(CC(C(=O)NCC1CC1Cl)NC(=O)C=CC1CCCN1C)SC C1(OC)CN(C(=O)CN2CCCS2(=O)=O)C(C)(CNC(=O)CC2(OC)CC2)C1 C1(NC(CCC=CC(C)C)=O)COC2(CCN(C(C3(C#N)CC3(C)C)=O)CC2)C1 C(=O)(C1=CCN(C(c2cccc(O)n2)=O)CC1)NC1C(CCC)C1 c1(C(N2CCCC(C(=O)NCC3C(C)CCC3)CC2)=O)ccc2cc[nH]c2n1 C=C=C(C)CC(=O)NCCCCC1CN(C(=O)CCCCN(C)C(C)CC2CC2)C1 C=CCC(CN=c1nc2scnc2c(NCCN2CSCCSC2)[nH]1)OC N1(C(CCC)=O)CCC2(CC1)CN(C(C1(CO)CC(C)(C)C1)=O)C2 N(C(=NCCCCN1CCOC1=O)NCc1ccnc(CN(C)C)c1)C1C(C)C1 c1(C(=O)NCC2(OC)CN(C(C3(CC)CC3(F)F)=O)C2)cnc(OC)c(F)c1 C1(O)(c2cn(Oc3ccc(OC)cc3)nn2)CCN(C(=O)Cn2cncn2)CC1 N1(C(C(=O)N(C)CC)C)CCC(CO)CC1.c12csc(n1)C(C1CCC1)NC2=O N1(CC)CCCC2CN(C(=O)CCc3cn(C)nn3)CCC12 C1(CNC(C(C)(C)O)=O)CN(C(C2CCC2(C)C)=O)CC1(F)F Cc1ncnc(C)c1C(=O)NCCNC(=O)C(O)CCn1cncn1 c1(OCCCC(=O)NC2CC(NC(c3c(CC)occ3)=O)C2)ccc(F)cc1 C12(NS(=O)(=O)c3ccccn3)CCCCC1OCC2 c1(N(C(CN(C(C2CCC2C)=O)CC)=O)C)nc[nH]n1 CC1=C(C(=O)NC2CCCC(NC(=O)CCc3cccnc3)C2)C(C)(C)CCC1 c1(SC)ccc(Cl)c(C(N2CCC2CNC(c2ccnc(Cl)c2Cl)=O)=O)c1 C1(CNC(C2C(CNC(COCCCC)=O)C2)=O)CC(CC)=NO1 c1(Sc2c(OC)cccn2)ccc2c(c1)CCCC2 c1(C(=O)NCC(C)(C)OCCNC(C(C(C)O)C)=O)ccnc2ncccc12 CC(C)C(C)CC(=O)N1CCCC(N(C)C(c2ccnc(C#N)c2)=O)CC1 N1(C(c2cccn3ncnc23)=O)CCC2(CCN(C(c3cncs3)=O)C2)C1 C1(CC(=O)NC(C2CCOC2)CNC(=O)CC2CC23CCC3)CCC(F)(F)CC1 Cc1cc(Cl)ccc1CC(N1CCCCCC1CNC(C1OCCC1C)=O)=O c1(C(N2C(C)CCC(NC(c3ccc[n+]([O-])c3)=O)C2)=O)nnn2c1C(=O)NCC2 N1(C(Cn2c(N)ccn2)=O)C(CNC(=O)CN2C(=O)CNC2=O)CC2COCC12 C1(NC(C2CC3CCC2O3)=O)CCN(C(c2cnn(CC(F)(F)F)n2)=O)CC1F CCCS(=O)(=O)NCCC(=O)N(CCN(C(CC1CC(NCC)C1)=O)C)C(C)C CCCCCCC(F)C(=O)N1CCC(O)(CNC(C2(CO)CC2)=O)CC1 C12(CCN(C(c3cc(CC(=O)OC)on3)=O)C1)CC2.C1(C)(CC)CC1C(=O)NOC.N.OC.C c1(CC(N2CC(CNC(C3(C)CC4CC4C3)=O)C2)=O)cc2ccccc2o1 CCC(CC(F)F)C(=O)N1CC(O)(C(C)NC(=O)CC2CC3(CCC3)CO2)C1 c1(-c2occ(CC(=O)OCC3CCCC34CC4)n2)ccccc1Cl C(=O)(C1c2c[nH]nc2CN1C(=O)Cc1nc(=N)[nH][nH]1)NC(C)CC(N)=O c1(CN2CC(CC(N3C(C(=O)OC)C4CC4C3)=O)C2)cc(O)ccc1C C1(NC(C2CC(OC)(OC)C2)=O)CC2CC1CN(C(=O)C=C1CCC(C)CC1)C2 C1(C(N2CCC(CF)(NC(c3cn(C)nn3)=O)C2)=O)(CC)CCNC1=O c1(C(N(C(c2nc(C3CCC3)no2)C(=O)NCC)C)C)ccc(S(N)(=O)=O)cc1 N1(C(C=C(C)C2CC2)=O)CCCC(CO)(NC(=O)CCC2CCCCN2C)C1 C1(NC(CSCC(C)C)=O)CN(C(=O)CCc2ncc(F)cn2)CCC1C C(=O)(CCC(C)(C)C(=O)N1CCN(C(=O)CSc2nccn2C)CC1)OC C1(CC#C)(C(N2CCCC(OC)C2)=O)CCN(C(=O)CCc2cnn[nH]2)C1 Cc1cc(F)cc2[nH]c(C(N3C(C)CC(C(=O)O)C(C)CC3C)=O)cc12 c1(NCC2CCN(C(C(C)(C)O)=O)C2)cc2c(cn1)C(=O)CCC2 C12(C(N3C(C#N)CCC3)=O)CCC(NC(c3cc4sccc4[nH]3)=O)(CC1)CC2 c1(OCC)ccc(C)nc1C(=O)NCCC(C1CC1)NC(=O)C=Cc1cnc[nH]1 C1(=O)C(c2ccncc2)C1=O.C1(=O)C(CC)SCCN1.C(COCCN)SCC N(C1CCOc2ccccc21)C(C(c1ncccn1)C)=O C(C(C)(C)CC(=O)N1CCCC(C(C)(O)CNC(=O)Cn2cc(Cl)c(C)n2)C1)OC CC1CN(C(c2cnc(Cl)cn2)=O)CCN1C(c1cccnc1Cl)=O C(C(C)(C)CNC(=O)CSS(C)(=O)=O)N(C(CCN(c1ccccc1)CC)=O)C C1(NC(CC(=C)C)=O)CCSC12CN(C(=O)C(F)=CC1CC1)C2 CC(C)CCC(O)C(=O)NC(C(=O)N(C1CCC1)C)C1CCC1 c1(NC(C(CCC)NC(C2CC2COC)=O)=O)cc(Cl)ccc1OCC C=CC(C)CC(=O)N(C)CCN(C(=O)C=CCCC=C(C)C)C CCCCC(C)N=c1nc(N2CC(CC)OC(C)(C)C2)c2[nH]ccc2[nH]1 Cc1ncc(C(N2CC(CCNC(=O)CC(C)O)C2)=O)n1C C1(C(N2CCCN(CCNC(CCCC(N)=O)=O)CC2)=O)CCn2cnnc2C1 C1(NC(CCCC(=O)NC)=O)CC2CCC(C1)N2C(=O)Cc1cn2ccsc2n1 Cc1ccc(C(=O)NCC(O)CN(C)C(c2cnc(C3CC3)nc2C)=O)cc1N Nc1cc(C(=O)NCC(CO)NC(=O)C=CCn2cncn2)ccc1Cl C1(C2(O)CN(C(c3ccoc3Cl)=O)C2)(CNC(C23CCC(CO)(CC2)C3)=O)CC1 CC1CC2CCC(C(=O)NC3CCN(C(=O)C=CS(C)(=O)=O)C3C)CN2C1 c1(CC2CCN(C(C3(C(C)(F)F)CC3)=O)C2)cn2cc(F)ccc2n1 C1(CC)(NC(=O)CC2CCNC2=O)CCN(C(=O)C(=O)C(C)(C)C)CC1 N1(C(CS(C)(=O)=O)=O)CCC2(CC1)CC(N1CCC3(CCOC3)C1)C2 c1(C2C(C(=O)OC(C(=O)OC)COC3CCCO3)C2)cc(F)cc(Br)c1 c1(C(N(C2CN(C(c3cccc(O)c3)=O)CC23CC3)C)=O)cc2sccc2n1C c1(CNCCC(C(C)C)N)cccc2c1CCOC2 N1(C(C(CCC)O)=O)CCC2(CCN(c3nccc(N4CCCC4)n3)C2)C1 C1(NC(CCC)=O)C2CCC1CN(C(c1cn3ccsc3n1)=O)C2 C1(NC(C2CC(C)OC2)=O)CC2CCC(C1)N2C(=O)CCc1cn(C)nn1 C(=O)(C(CNC(c1cc(C)ns1)=O)CC=C)NC(c1ncccn1)CC c1(C(C(=O)NCC(CNC(=O)C(C)SC)OC)O)cccc(F)c1 c1(CC)cc(C(=O)NC(CNC(C2CC3(CSC3)C2)=O)C(C)(C)C)n(C)n1 c1(C(=O)NCCC(C)NC(C2CC2CF)=O)cc(Br)n2ccccc12 Cc1ccccc1-c1nc(C(N2CCSCC2CO)C(=O)NC2CCOCC2)co1 C=CCC(C)(C(=O)NCC1CC2(CC2)CN1C(=O)CCN1CCOCC1)N(C)C C1(C(=O)NC2CCC(NC(c3c(CC)nn[nH]3)=O)C2)CC(C2CCC2)C1 N1(C(C2(COCC)CC2)=O)CCn2nc(NC(c3cc(Cl)cnc3O)=O)cc2C1 Cc1cc(O)nc(-n2nc(C)cc2C(=O)CC2CC3(CNC3)C2)n1 C1(C)(C(N(CCC(C)NC(C2CCCCN2C)=O)C)=O)CCCC(F)(F)C1 c1(OCC=O)ccccc1Oc1cnns1.C=CCSCCC1CC1 N1(C(C2(COC)CC(=O)C2)=O)CCCC(CC(=O)NCc2cnn(C)c2)C1 Cc1ccccc1OCC(=O)NCCCN(CCCN(C)C)C.N12CCC(C1)C2 c1(C(=O)NC(CC)CN(C(C2C=CCC2)=O)CC)cccc(C2CC(=O)C2)c1 N1(C(c2c(CC)noc2)=O)CC(O)CC1CNC(C1CC2(CCC2)C1)=O c1(C(N(C2CCCC2)C(=O)Cc2ccccc2)=O)cc(F)cc2c1OCOC2 C1(C(NOCCOC)=O)CCC(O)CN1C(=O)C(C#N)C(C)C O=C1CCC2(CN1)CN(C(C1CC(O)C(O)CC1CNC(=O)C1CC1)=O)C2 C12(C(=O)NC3CN(C(C4OCCN(C(C)C)C4)=O)C3)CCC(CO)(CC1)OC2 c1(OC)cc(C#N)ccc1C(N1CCC(NC(=O)CNS(C)(=O)=O)C(CO)C1)=O C1(C(N(CC(C)NC(=O)Cc2ccc(F)c(F)c2F)C)=O)CC1C1CCCCC1 C12(C(=O)NC(C)CNC(=O)C(C)CC(F)(F)F)CCCCC(=O)N1CCC2 C(N=c1nc(C(F)(F)F)cc(C2CC2)[nH]1)C1CN(C(C(C=C)O)=O)CC1C c1(OC)cc(-c2cn(CC(c3ccncc3)F)nn2)ccc1-n1cccn1 c1(N(C)C)ccc(C=CC(N2CCC(C)(NC(=O)C#CC3CC3)C2)=O)cc1 C1(CNC(c2cnc(C)s2)=O)CC2(CO1)CN(C(C1(F)CC=CCC1)=O)C2 C(C(Cc1ccoc1)C(=O)NCCCC1CCOC1=O)OC.C1=CCNC1=O c1(NC(=O)NC(c2ccc(N(C)C)c(Cl)c2)CC(=O)OC)ccc(C(N)=O)c(C)c1 C(N=c1nc2scnc2c(NCc2ccco2)[nH]1)C1CC2(CCC(=O)N2)C1 N1(C(CC(CC)C2CCC2)=O)CCCC(CNC(=O)Cc2cncnc2)CC1 n1(CC)nc(C)c(C(C)NC(=O)NCC(C(C)(C)C)C2CC2)c1C C(CSC)(C(C)C)NC(CCC1N(C(CCOC)=O)CCC1)=O Cc1ccc2c(n1)CN(C(c1cn(-c3cnn(C)c3)cn1)=O)C2 C1(NC(c2nc(OC)oc2)=O)CCC(C)N(C(c2cc(C3CCC3)nn2C)=O)C1 Cn1cc(I)c(O)nc1=NC(=O)NCCc1cccc2cnccc12 CCC(C)(C)CCCC(=O)NC1CN(C(=O)C(c2c(C)noc2C)=O)CC1OC C(=O)(C1=CCCCC1)Nc1cccc(NC(C2C(C)(C)COC2)=O)c1 Cc1cc(C(=O)Nc2ccc(CNCCc3cnn(C)c3)nc2)ccc1[N+](=O)[O-] C1(C(=O)NC2CC(C(N3CC(NS(C)(=O)=O)C3)=O)C23CCC3)CC2(C1)CC(O)C2 N1(c2nc(C)on2)CCCC(NC(=O)NC(c2ccncc2Br)C)C1=O C=CCC(C(=O)NCC(CC=C)NC(c1cc(CC)ccc1Cl)=O)C(C)C C1(C(N(c2ncc(C)cn2)CC2CCNCC2)=O)CCc2nc[nH]c2C1 N1(C(C(C(C)C)C)=O)CCC2(CCCCN(C(c3cnc(S)nc3)=O)C2)C1 N1(C(c2cnc(C)o2)=O)CCN(C(C2(C)C=CCC2)=O)CC1CO c1(C(=O)NCC2CCC(NC(CC(COC)(C)O)=O)C2)ccnc2ncnn12 N1(C(CC2(C)CCOC2)=O)CCCC2(CCCN2C(=O)C#CC2CCC2)C1 CN1C(=O)Cc2cc(S(=O)(=O)NCC3CCCC(C(=O)O)N3)ccc21 C12(NC(C=CC(C)(C)SC)=O)CCCC1N(C(C1CN(C)CCO1)=O)CC2 c1(C(=O)OC)c(C)[nH]c(C(=O)NCC2(NC(c3n[nH]c(C)c3C)=O)CCC2)c1C C(=O)(C(C)(C)CC(C)C)N1CCC(N(C(c2c(C)[nH]c(=N)s2)=O)C)C1 c1(C(N2C(CNC(C(C(CC)C)O)=O)CCCCC2)=O)cc2ccncc2s1 N1(C(C(C2CC2)OCC)=O)CCC(C)=C(F)C1.C1(C)(CSC)C(=O)N1 C(CC(F)(F)Cc1cn(CCOC(F)F)nn1)NC(=O)CC1(C(=O)O)CC1 N1(Cc2c(C)nc(NC(=O)Cc3cc(F)ccc3Cl)s2)CC2CCN(C)CC2C1 N1(C(CCn2ncc(C(N)=O)c2)=O)CCC(NC(=O)C(=O)NC2CC2)CC1CO O=C(C(F)CC1C(CO)C1)NC1CCN(C(=O)Cc2cc(-c3cccs3)on2)C1 c1(C(=O)NC(c2ccc(CNC(C3(C)CC(F)C3)=O)cc2)C)ccn2ncccc12 CCCCC(CNC(=O)Cc1cn[nH]c1)NC(=O)CC(=O)NCC c1(OC)cc(NC(CC(C)C)C(=O)O)cc(F)n1 C1(N(C(CC2(C#N)CC2)C(=O)NC)CCN(C)C)CCN(CC)C1 C1(CCC)CN(C(C2CC2CCN(C)C)=O)CC1C(=O)NC(C)Cc1nn[nH]n1 c1(CN(C2CN(C(c3cnc(Cl)cn3)=O)C2)C)cncc(Cl)c1Cl c1(C(=O)NCC(N2CCOC2=O)(F)F)csc(CO)n1 c1(C(=O)NC2CN(C(C(CC(C)C)O)=O)CC3C2C3)ccc2c(n1)OCCO2 N1(C(Cc2nc(=N)[nH][nH]2)=O)CC(C(=O)NCc2cccnc2)C2(CC2)C1 CC(C)(Cl)CC(=O)NC1CC1NC(=O)CC(c1ccccc1)C1CCCCC1 C12CN(C(c3nn(C)cc3Cl)=O)CC1Cc1cn2nn1.n1(CC)ccnc1C#N c1(OC)ccc(CNC(N(C(c2ccccc2Br)C)CCOC(C)=O)=O)nc1 C(=O)(C(O)C1=CCCCC1)N(C(CNC(C(C)n1cnnn1)=O)C1CC1)C c1(C(C)C)ccc(C(=O)NC(Cn2cncn2)C(=O)N2CC(CF)C2)o1 C(=O)(C1=NN(C)C(=O)CC1)NC1CN(C(c2cc(COC)oc2C)=O)CC1CO N1(C(COC(CC)CC)=O)CC=CC(NC(c2ccn(CCF)n2)=O)C1 O=C(NNc1cc(Cl)ccc1Cl)c1c[nH]nc1C(F)F c1(C(C)C)ccc(F)cc1C(=O)NCC1C=CCN1C(=O)C=CBr N1(C(c2cc(OC)n[nH]2)=O)CCC(C(C)(O)CNC(c2cc[nH]c2C)=O)CC1 c1(CC(=O)NC2C(CC)N(C(c3ccccc3Cl)=O)CC2)cc2ccccc2o1 N1(C(c2c(C)onc2)=O)CCCCCC(NC(=O)C(c2cccc(C#N)c2)C)C1 c1(C(N2CC(CC)C(NC(=O)C(C)(C)CF)C2)=O)cc([N+](=O)[O-])oc1C C#CCC(C)(C(=O)NC(CO)C(N)=O)NC(C1CC2(CCO1)CC2)=O c1(CCC(N2CC3C(CNC(=O)CC4CCC4)(CC3)C2)=O)cnc2ccccn12 c1(CC(=O)NC(C2CCCCC2)CNC(C2CC2[N+](=O)[O-])=O)ncc(Cl)s1 C1(C)(C(N2CC(CN(C(c3cnc(SC)s3)=O)C)C2)=O)CC(C(C)C)=NO1 c1(C(=O)NCCCN(CCCNC(C2(C)COC2)=O)C)cc(F)ccc1Br Cc1nc(C)c(C(=O)NCCC2(NC(C3CC(=O)N(CCN(C)C)C3)=O)CC2)o1 C#CC(C)(C)C(=O)N1CC(O)(CCNC(C2CCN(C(C)=O)C2)=O)C1 C1(CC)CN(C(C2(Cl)CC2)=O)CCC1NC(c1c(C)coc1C(C)C)=O Fc1cc(Br)cc(F)c1CCNC12CC(C1)N(CC=Cc1ccccc1)C2 CN1CCCC(NC(=O)CN(CCC(C)(C)C)CCO)C1=O c1(C(N(C2CCN(C(c3cc(C)cs3)=O)C2)CC)=O)cc2ccccn2c1 c1(C(=O)NCC(C)N(C(c2cc(CSCC)on2)=O)C(C)C)ccc(C)nn1 c1(C(=O)NC(COCC)C(=O)NC(c2noc(CC)n2)C)cccc2c[nH]nc12 C1(C(=O)NCCNC(c2cncs2)=O)CCN(c2ccccc2F)C1=O O=C(C1=CCCCCC1)NCC1CC(O)CN1C(=O)COCC1CCCC1 C(CCCC(C)NC(=O)C(F)(F)C1(C)CCC1)NC(C(N1CCSCC1)C)=O c1(C(=O)N(O)Cc2cn(CC3CCCC3)nn2)cn2ccccc2n1 CCC(O)C(C)(C)C(=O)N1CC(O)(CNC(=O)Cn2ncc(O)nc2=O)C1 C1(CC(=O)NCCCc2c(C)noc2)C2CCCC2N1C(=O)Cc1ccoc1 c1(N2C(C)CC(NC(C3CC4CCCC4C3)=O)C2)ncnc2ccc(Cl)cc12 C1(OC)CC2(CCC(NC(=O)C(=O)NC(C3NC(=O)NC3=O)c3cccs3)CC2)C1 CC1(C)C2CC(C(=O)NC3CCCC3c3cc(F)cc(F)c3)CC12 c1(C(=O)NCCCCCNC(C2(CO)CCC2)=O)ccc(Cl)c(Cl)c1 c1(CNC(=O)CC2CCCN2C(C2CCC2)C)cc(Cl)c(Cl)cc1O C(=O)(C(=O)Nc1ncc[nH]1)NCC(C)N(C(=O)C(C)n1cnnn1)C C1(C(F)F)(CC)CCCN(N(C)CCc2ccc(C)cc2)C1 c1(C(=O)NCCN(C(CNC(C(C)(C)C)=O)=O)C2CC2)cc(Cl)c(Cl)s1 CC1CN(C(=O)CC2CCC2)CC(CCNC(c2csc(C(F)(F)F)n2)=O)O1 O(C1CCc2ccc(Cl)nc21)C(C(C)NC(=O)OCC)=O.c12ccnn1C2 N1(C(c2cc(OC)ns2)=O)CC2(NC(c3ccc(CO)nc3)=O)CCCC2(F)C1 C1(COC)C=CCCN1C(=O)C(CNC(c1cnnc(O)c1)=O)CC1CC1 N1(C(c2n(C(C)C)ccn2)=O)CCCCC(NC(C2(C(C)(C)C)CCCC2)=O)C1 N1(C(C(C)NC(CC)=O)=O)CC(N(C)C(c2cc(C(C)(F)F)n[nH]2)=O)C2(CC2)C1 c1(N)ccc(C)cc1.C12CCN(CC1)C(=O)N(Cc1ccc(C)cc1)CC2F.CO c1(-n2c(C3CCN(C(C)C)C3)nc(C(=O)NC)n2)ccc(N(C)C)c(C)c1 c1(C(C(=O)NC2CCC(CNC(C=CCC)=O)C2)OC(C)=O)c(F)cccc1F c1(OCC(N2CC(CCNC(c3ccccc3)=O)C2)=O)cc(Cl)ccc1Cl S1(=O)(=O)c2ccc(Br)cc2N2CCC(C2)CN1C.C=C(COC)c1ccccc1 C1(OC)CN(C(=O)C=Cc2cc[nH]n2)CCC1NC(c1cnccc1C(F)F)=O CCC(C(=O)N1CCCC1C1(C(=O)N(CCCF)C(C)C)CC1)NC(C)=O N1(C(CCOCC)=O)CC(NC(=O)C(F)=C2CN(C(=O)OC(C)(C)C)C2)CC1(C)C C1(N(C(c2ccc(C)n2C)=O)CCn2ccnc2)CCNCCC1C C12(C(N(C)Cc3ccccc3O)=O)COCC1CN(C(C1CCC(F)(F)C1)=O)C2 C1(C(F)(F)F)(OC)CCN(C(=O)Cc2csc(-c3cccnc3)n2)C1 C1(CC(N2CCC(N(C(c3ccoc3C3CC3)=O)CC)C2)=O)CC2C=CC1CC2 C(=O)(C(C)CCC(C)(C)C)NCCC1=CCN(C(c2cnc(C)o2)=O)CC1 CC(C)(C)C(C#N)C(=O)NCC12CCC1CN(C(=O)CCNc1ccccc1)C2 c1(C(N2CC(O)CC2CNC(C2CC2(Cl)Cl)=O)=O)c(F)cccc1F C(=O)(C(F)CCC(C)(C)C)N1CCCC(NC(C2OCCN(C)C2)=O)CC1 N1(C(C(CC=C)C)=O)CCN(C(=O)CNC(CC(C)(C)C)=O)CC1C1CCC1.C(C)C C1(C(=O)NC(CC#C)(C)C)CCC(C)(C)N(C(=O)CC=C(C)C)C1 Cc1cccn2c(=O)c(C(N3CCOc4cc(O)ccc4C3)=O)cnc12 c1(OC)c(Nc2cnn(C)c2)nc(SC)nc1C.C12(CCC1)CNC(=O)CN2 C1(NC(C(C=C)(C)O)=O)CC(F)CN(C(c2cc(OC)ccc2OC)=O)C1 C12(C(=O)NCCOCCNC(C3Cc4cscc4C3)=O)CCOC1CS(=O)(=O)C2 N1(C(C(C)NC=O)=O)CCC(CNC(C2CN(C(C)C)C2)=O)C1 Cc1nn(CC(F)(F)F)nc1SCC(=O)NC1CC1CNC(C1(CO)CCC1)=O c1(C(=O)NC(CC)CNC(=O)CCc2ccnc(Br)c2)cnc2n1CCC2 O=C(C1=CCN(C(C2(CO)CCC2)=O)C1)NCC1CC(CO)CO1 C1(NC(C2CCC3CCC23)=O)CCN(C(=O)CSC2CCOC2=O)C12CCC2 C1(NC(c2nnc(C)s2)=O)CCN(C(c2cc(C(F)F)ccc2F)=O)C2CC12 c1(C(=O)NCCCC2CC2)ccc2c(n1)CN(C(C1CC(F)(F)C1)=O)CC2 C1(CNC(C(C)NC(C)=O)=O)CCN(C(c2cc[nH]c2)=O)C(C)C1 N(C(=NCC(C)F)NCc1ccco1)C1CCN(Cc2ncc(C(C)C)s2)C1 N1(C(C(CCC)OC)=O)CCC2CN(C(c3cnn(CC4CCCC4)c3)=O)C2C1 Cc1c(C(=O)NC2CC2NC(=O)CCc2nccs2)cnc2c(Cl)cccc12 C=C1CCC1(C(=O)NCc1ccc(-c2ccncc2)s1)NC(=O)OC(C)(C)C C(=O)(C#CC1CCCOC1)N(C(C)C)CCNC(c1cn(C2CCC2O)nn1)=O C(=O)(C(F)C(C)CNC(C1C2CCC(F)C12)=O)NC1CCCC(OC)C1 N1(C(CC(=O)NCCOC)=O)CC(NC(=O)COc2ccsn2)CC12CCOC2 N1(C(CC(=C)C)=O)CCCC(C2(NC(c3cnc([N+](=O)[O-])n3C)=O)CC2)C1 C1(NC(C2(C)N(C(C(OC)OC)=O)CC(O)C2)=O)Cc2ccccc2C1 C=CC1CN(C(=O)CC2C=CS(=O)(=O)C2)CC1NC(C1C=CC=CC=C1)=O c1(C(=O)NC2(C)CCN(C(=O)C3=CS(=O)(=O)CCC3)C2)nccc2c1NCCC2 C1(OC)CC(NC(=O)C(CC(C)C)NC(N)=O)CN(C(C2SCCCS2)=O)C1 C(=O)(C(O)CC(F)(F)F)NC(C(C)C)CC(=O)NC(CCO)C1CCC1 N1(C(C(N2CCC(C(C)NC(c3ccc(F)cc3)=O)C2)=O)C)CCP(C)(=O)CC1 c1(C(=O)Nc2cnc(C(F)(F)F)cn2)ccc(I)c(I)c1 C1(C(N(C(C)C(=O)OC)CC=C)=O)CCN(C(c2cn(CC)nn2)=O)C1 Cc1nc(CCC(=O)NC2CC(CNC(C3(CC(C)C)CC3)=O)C2)oc1C N1(C(CN2CC(C)(OC)C2)=O)CC(CNC(C2(F)CC=CCC2)=O)C(C)C1 c1(C(=O)NCC2(NC(CCCCC(N)=O)=O)CC2)ccc2nnn(O)c2c1 C1(OC)CN(C(=O)CCCn2ccnc2)CC1NC(=O)C(C)N1CCCC1 c1(OC)nc(C(=O)NCCC(C)NC(=O)C=CC2CCCN2C)sc1C C(C(=O)N1CCC1CN=[N+]=[N-])(C(C)C)NC(C)=O.C(CCCO)NC=O CC(C)C(=O)NC(C(=O)NC1CC(Cn2ccnn2)C1)C1CCCC1 C#CC12CCC(C(=O)NCC(CNC(=O)C(C)(C)C(=O)N(C)C)CO)(CC1)CC2 c1(OC)ccc(OC)c(C(=O)N(C)CC2(NC(c3cc(Br)ccc3C)=O)CC2)c1 Cc1ccc(C(=O)NC2CC(C(C)NC(C3CCOC3)=O)C2)cc1N CC1(C)CCCN(C(=O)C(C2CC2)C2CC2)C1C(=O)Nc1cnn(CCO)c1 c1(CN(CCC)CCOCCBr)cc(OC)c(OC)cc1F CCC(C#N)(CC)C(=O)NC1CCN(Cc2nc(C3CC3)nn2C)CC1C C1(NC(C2(Oc3cn(C)nc3)CC2)=O)CCCN(C(c2[nH]cnc2C#N)=O)C1 c1(N2CC(C)C(NC(c3cccc(=O)n3O)=O)C2)ncc2ccsc2n1 CCC(C)C(O)CC(=O)NC(Cn1cncn1)C(=O)NCCC(C)O N1(C(C(C(C)C)O)=O)CC(NC(c2ccccc2CN(C)C)=O)CC2(CCC2)C1 C(C(O)C(=O)NCCCC1(NC(c2cnc(C3CCCCC3)s2)=O)CC1)SC N1(C(C(=O)NC)=O)CCCC(C)(C(N)=O)C1.c12ccc(cc1)CNC(=S)N2 C(=O)(CC1=CCOCC1)NC(C)C(N1CCC(C)(F)C1)=O c1(CN2C(C(=O)Nc3cnncc3Cl)C=CC2)cnc(Cl)nc1Cl c1(C(=O)NCC(CC)NC(C2(F)CCOC2)=O)cncc(C(C)(F)F)c1 C12CCCN(C1)C(CC)C(=O)NC2.C(CCC)=CC=CC=C CCCCC(C)NC(C1(NC(=O)CC2(O)CCCC2)CC(F)C1)=O c1(C(C)NC(=O)NCC2(NS(C)(=O)=O)CCCC2)cccc(C2CC2)c1 N1(C(C=C(C)C(F)F)=O)CCC(C)(C)C(CNC(=O)CC2CCOCC2)C1 c1(C(N2CC(CCCCNC(Cc3cc(C)nn3C)=O)C2)=O)ccc(C)c(Br)c1 C#CCCN=C(NCC(C)(C)OC)N1CCN2C(=O)CCC2C1 N1(C(C2(SC)CC2)=O)CC2CC1C2NC(c1csnc1Br)=O C(=O)(CCCC(C)(C)C)NC1C(C)(CNC(C=CCN(CC)CC)=O)CCC1 N1(C(C2(OC)CCSC2)=O)CCC2CCC(C1)N2C(C12CC(C)(C1)OC2(C)C)=O c1(OC)cc(F)c(S(N)(=O)=O)cc1C(N1CC(C)(C(c2ccccc2F)O)C1)=O n1(CC(=O)NCC(C)CNC(C2COC(=O)C2)=O)ccc(=O)c([N+](=O)[O-])c1 c1(C(C)N(C)Cc2ccccc2OCF)ccncc1Cl C1(CC)C(C)CCN1C(C(=O)NCCCSC)C(C1CCCCC1)OC N1(C(=O)Cn2cnnc2)CC2C(CO)C2C1.N12CCCC1C1(CC1)C2=O N1(C(C(c2cnn(C)c2)NC(C(C)Cn2cccn2)=O)=O)CC(N(C)C)C(O)C1 c1(OC)ccc(C(=O)NC2CN(c3cc(C(C)(C)C)ncn3)CC2(C)C)c(F)c1 c1(OCC)ccc(S(=O)(=O)NC2CCN(Cc3ccccc3)C(C)C2)nn1 Cc1ccncc1SCC(N1CCCC1C(N1CCC(c2ccccc2)C1)=O)=O CCCCC(O)CC(=O)N(CC(C)NC(=O)CCc1cc(C(C)=O)c(C)o1)CC C1(CC(=O)NCCC(=C)CNC(c2ccco2)=O)CCS(=O)(=O)C1 c1(C(N2CCCC(NC(=O)C(F)(F)CC3CC3)C2)=O)coc2c1COC2 Cc1ccc(C(=O)NCC2COCC2NC(=O)C(C)(C)C(C)C)cc1C Clc1ccc(CNC(C2CC3CC3C2)c2ccncc2)cc1.c1(C)nc[nH]n1 c1(CC(C)C)cccc(C(N2CCCC(C(=O)NCC3CC3(C)C)C2)=O)c1 c1(C(N2CC(C(=O)Nc3ncc(F)cc3Cl)C2)=O)cc(F)cc(F)c1Cl CC(C)CC(CNC(=O)CCC(C)(C)C)C(=O)N1CC(C)(C)CCC1CO C(=O)(C#CC1CCCCC1)NC1CC(NC(C(CCOC)C)=O)C1 C1(NC(C2(C(=O)NCCO)CC2)=O)CCN(CC)CC1.c12sccc1CC(=O)N2 C(=O)(CC(C)(C)n1ccnn1)N1C(CNC(C2N(CCC)CCC2)=O)CC1 Cc1ccn2c(C(=O)NCC(C(C)(C)C)NC(=O)CC3CC3C)cnc2c1 c1(C(=O)NCC2CCCN(C(COC(CC)C)=O)C2)cc(O)ccc1C C(=O)(C1=NN(C2CC2)C(=O)CC1)NC1C(C)(CN(C(C(C=C)O)=O)C)CCC1 C=CC1(CC(N2CCOC(CCO)C2)=O)CN(C(=O)C(=Cc2ccco2)C)C1 C(=O)(CP(C)(C)=O)NC(CC)(C)CNC(=O)Cc1nc[nH]n1 Cc1cc(CC(C)NC(=O)N(CCN(C)C)C2CC2)cc(C)c1 c1(OC)cc(C#N)ccc1CN1CCCC(C(N2CCCC(O)C2C)=O)CC1 c1(NC(C(C)NC(c2ccc(Br)cc2)C)=O)cnc(F)cc1NC(=O)OC(C)(C)C C12(C(=O)NCCCCCNC(C3CCC(C)(C)CC3)=O)CCCCC1OCC2 C12(CNC(c3cccc(SCC)c3)=O)CCC1CCN2C(c1c(C)ncn1C)=O N1(C(c2c(N)nccc2)=O)CCC(NC(c2cc3scnc3[nH]2)=O)C12CC2 CC(C)C(C#N)C(=O)NC1(CC(N2C(C)CC2(C)C)=O)CCCCC1 C(=O)(NNc1cccc(F)n1)C1CN(C(=O)OC(C)(C)C)C(C)(C)CC1 c1(CC(=O)N(CC(O)CO)C(C)C)cc2ccccc2s1 CC1=NN(C)C(=O)C1CC(=O)NC1COCCN(C(c2cnn(C)n2)=O)C1 N1(C(C2CCCN(C(C)C)C2)=O)CCC=C(CNC(c2cnn(C3CC3)c2)=O)C1 CC1(O)CCC(NC(c2cc(CNC(c3csc(Cl)n3)=O)cs2)=O)CC1 Cc1ccc(CN(C)C(C2OCCOC2C2CC2)=O)cc1C C(=O)(CC(F)(F)C1CCNCC1)N(C(=O)COC(c1c(C)cco1)=O)C c1(N(C)CC2CCN(C(C(CCC)N(C)C)=O)C2)nc(Cl)nc2cnn(C)c12 C1(C(=O)NCC2(C(N(C3CCCC3)C)=O)CC=CC2)CCOC1(C)C C1(NC(c2c(CNC(c3ccn(C)n3)=O)n(C)nc2)=O)C2CCC3C(C2)CC13 C1(CC)CC(C(=O)OC)CN(C(=O)CC2(C)COCCN2C(C)=O)C1 N1(C(CC(C)c2ccco2)=O)CC(NC(=O)C(Cl)=CCl)C(N=[N+]=[N-])C1 C(=O)(C(F)C(=O)NC(C)(CNC(c1c(C)noc1C)=O)C1CCC1)OCC C12CCCCN1C2=O.CCC(CNC(C)=O)NC(=O)C(C1CCC1)OC C=C=CCCC(=O)NC(CNC(=O)C(c1cn(C)nc1C)O)CCCC N1(C(c2cc(OC)n[nH]2)=O)CCC(CF)(NC(c2ccn(CC(C)C)n2)=O)C1 C1(NC(C(C)C2CCCC2)=O)C2CC3CN(C(=O)Cn4ncn(C)c4=O)C1C3C2 c1(C(=O)NC2CC(C)N(C(=O)CN3CCCC3)CC2)nccc2[nH]ccc12 CC1CN(C)CC(C(=O)NCCNC23CC(CN2C(=O)OC(C)(C)C)C3)O1 C=CCCCCCCCC(=O)NC(CNC(=O)C=Cc1ccc(C)nc1)C(C)C C1(CC(=O)N(CC(F)(F)CC)CC)CC(NC(=O)COCCCF)C1(C)C CC(C)CC(C(=O)NC1CC(F)CN(C(c2cccc(F)c2C(C)C)=O)C1)N(C)C c1(NC(Cn2cc(-c3scc(C)c3)nn2)=O)ccnc(-n2ccnc2)c1 O=S1(=O)c2cc(co2)C(=O)NC2C(CCCC2)N1.c1(C(=O)SC2CC2)cc[nH]n1 C(CN=c1nc(C#N)c(NOCSc2ncc[nH]2)c[nH]1)SC C(=O)(C(F)C(C)C)N1CC(O)(CN(C(C(C)(C)NC(=O)NCCC)=O)CC)C1 N1(C(C2OCCN(C(C3OCCN(CC)C3)=O)C2)=O)CCc2oc(C)nc2C1 C1(C(=O)OC)CC2CC1CC2NC(=O)CC1CCOCC1OC.C12CCN(C1)C2 c1(S)ccc(F)cc1F.N1(C(c2nnc(CO)s2)C(=O)NCCC)CCC(C2CC2)C1 N1(C(C=CCOC)=O)CCC2(CC1)CC(NC(c1cc(C)sc1C)=O)CO2 c1(C(N(CC(CNC(C(COC)(F)F)=O)C)C)=O)cc2scc(Cl)c2[nH]1 CC1(C(=O)NCCC2(NC(C3CN(C(=O)NC=O)C3)=O)CCC2)CCCCO1 CC(CN=c1[nH]c(C#N)c(Cl)s1)NC(=O)CCC(=O)N1CCCC1 c1(OC)ccc(C)c(C(N2CCC(C)(C(N3CCC(n4ccnc4)C3)=O)C2)=O)c1 N1(C(C2(C=C)CCC2)=O)C2CCCC1CC(NC(=O)C(C)(C)C(C)C)C2 C1(NC(CCOC(C)=O)=O)C=CCC(C(=O)N(C)CCN(C)C2CC2)C1 C12(C(=O)NCCC=C=C)CC(CO)(CN1C(C1CC(OCC)C1)=O)C2 CC(CC(=O)NCCCN(C(c1cnc([N+](=O)[O-])n1C)=O)C1CC1)C(F)(F)F C=C(C)C(C)(O)C(=O)N1CCN(CC(=O)N2CCCO2)CC1 CCCC(CNC(c1ccc(F)cn1)=O)C(=O)NCC(C)(O)CCO Cc1cn(C)nc1C(=O)NC(CNC(c1cnc(Cl)[nH]1)=O)C(C)(C)C N1(C(CCCc2n[nH]c(=N)s2)=O)CCCN(C(=O)CCNC(N)=O)CC1 C(=O)(C(CC)CC(F)F)NCC1CCN(C(C(F)=CCC)=O)C12CC2 N1(C(C2C(C)OCC2)=O)CC(NC(=O)Cc2ccc(C(C)(C)C)cc2)CC(F)C1 C(N=c1[nH]c(=NCc2nc(Cl)ccc2Cl)[nH]c2c(F)cccc12)C1N(CC)CC1 CC1(CCC(=O)NCC2(NC(c3ncoc3C3CC3)=O)CCCC2)CCCCC1 C(=O)(C#CC1CCCOC1)N1C2C(NC(c3cc(OC)cc(Cl)c3)=O)CC(C2)C1 N1(C(C2COC(=O)O2)=O)CCCN(C(c2cc3ccccc3[nH]2)=O)C(CO)C1 N1(CC(N2CCC(NC(C(COCC)c3ccccc3)=O)C2)=O)CCCNC1=O CC(C)(C)CC(O)C(=O)N1CCN(CCNC(=O)CC2NC(=O)NC2=O)CC1 C(N=c1[nH]cnc2ccc(OCC3CC3)cc12)C1CCN(C(C(C)OC)=O)C1 CS(=O)CCC(=O)N1CCOCC1CNC(=O)CCc1cncnc1 Cc1cc(C(=O)NC(C2(O)CN(C(=O)Cc3ccc(O)c(C)c3)C2)C)cc(Cl)c1 N1(CC(=O)NCCCCCCN(C)C(c2ccc(F)cc2)=O)CCCCCC1=O c1(C(=O)NCCC(CNC(=O)Cn2cnnc2O)OC)cnn(C)c(=O)c1 c1(C(N(CC(O)CN(C)C(C2CCCC2O)=O)C)=O)c(O)cc(F)cc1F C1(C(CNC(C(n2cc(COCCO)nn2)C)=O)=O)CC2CCC1C2 c1(C(=O)NC(C)C(C)NC(=O)CCSC(F)(F)F)ccnc(C(C)(C)C)c1 N1(C(=O)C=CC(=O)OCCCC2(O)CCC2)CCC(F)CC1OC(C)(C)C C1(NC(C2(SC)CC2)=O)CCCN(C(c2ccnc(OC3CCOCC3)c2)=O)CC1 c1(NC(C2N(C(CC(=O)OC)=O)CCOC2)=O)ccc(Br)c2ccncc12 C1(NC(C(F)=C(C)C)=O)CN(C(=O)CSCCN(C)C)CCC12CCOCC2 c1(NCCN2CCC(CNC(=O)Nc3ccccn3)CC2)cc(Cl)ncc1F c1(-c2c(C(N3C(CC(C)C)(C(=O)OC)CCC3)=O)c[nH]c2)cc(Cl)ccc1Cl C1(CCC(=O)N(C(C(C)SC)C)C)CCN(C(=O)Cc2nccn2C)C1 C(=O)(C(CO)NC(c1cnco1)=O)N(C(C)C1CC1)CC1CC1 c1(C(C(F)(F)F)NC(C2CCNCC2)CC)cc(OC(C)C)ccc1O N1(C(CN2C(C)CCC2)=O)C2CCC1CN(C(c1ccns1)=O)C2 C1(CNC(c2c(C)nc(C3CC3)s2)=O)C(C)CCCN1C(=O)CCNC(=O)CO c1(C(N(CCCOCCNC(=O)CC(=O)NCC)C)=O)c[nH]c2cccnc12 c1(CC)c[nH]c(C(N2CCCC2CN(C(=O)CSC(F)(F)F)C2CC2)=O)n1 C1(C(=O)NC(C2CCN(C(C3CCCC4CC34)=O)C2)C)CCS(=O)(=O)C1(C)C c1(NC(Cc2nc(NC(c3nccc(CC)c3)=O)sc2)=O)nc(C)c(Br)c(Cl)n1 N1(C(C2C(C)CC(=O)NC2)=O)CCC2(C1)CN(C(c1ccc3nc[nH]c3n1)=O)C2 CCCCCC(C(=O)NCCN1CCCC1=O)N1CCC(C)S(=O)CC1 C1(N(C(C(C)=CC2CC2)=O)C)CN(C(=O)Cc2ccn(-c3cccs3)n2)CC1F Cc1cc(CO)oc1C(=O)NCC1CCN(C(=O)Cc2csc(NC=O)n2)CC1 CONC(=O)C(=O)NCc1cccc(NC(=O)C(C)C(=O)Nc2nc(C)cs2)c1 c1(C(=O)NCC(C2CC2)NC(C2(C)CCSCC2)=O)ccc(F)c(C#N)c1 c1(C(=O)NCC(CNC(c2nn(C)c(F)c2)=O)F)noc2c1CCCCC2 N1(c2nnc(CC(C(C)C)(C)O)n2C)CCN2CCCCC1C2.OC(F)F CCC(C)(O)C(=O)NCCC(C)NC(c1cn(-c2ccc(Cl)cc2)nn1)=O N1(C(C=CC(C)(C)C)=O)CC2CN(C(c3ccc(O)cc3F)=O)CCC2(CO)C1 N1(C(CC(=C)Br)=O)CC2CCC(C1)N2C(C1CCCN1S(=O)(=O)CCC)=O c1(C(=O)NCC(C)NC(CS(CC)=O)=O)cnc(Cl)c(F)c1N C1(CCNC(CN(CCCC)CC)=O)(NC(=O)C(C)N(S(=O)(=O)CC)C)CCC1 C1(C(N(CCF)CC)=O)CC1CNC(C1CC1F)=O c1(CCC)nn(C)c(C(N)=O)c1C(=O)N(C)CCC1CCCCN1C(=O)C(C)O c1(C(N(C(C)C)CCNC(=O)CCCC2CC2)=O)cnc2cccnn12 c1(CC)ccc(C(=O)NC2(CNC(C3CC(O)CN3C)=O)CCCC2)nc1 C(C)(C)(CCCNC(=O)C(n1cc(C2CCCN(C)C2)nn1)C)N(CC)CC C1(CC=C)(NC(=O)CCC(F)F)CCCN(C(=O)Cc2ccc(F)c(Cl)c2)C1 S(=O)(=O)(c1cnc(NC2CCC(CO)C2)cc1C)NCC(c1ccc(C)cn1)(C)C C1(CC)(NC(=O)C(F)CC2CCC2)CCCN(C(c2cn(C)nc2OC)=O)C1 N1(C(CC2(C=C)CN(C(=O)CC(Cl)Cl)C2)=O)C2CCC1(C1CC1)CC2 CC1CN(C(c2cc(N)c(Cl)cn2)=O)CCN1C(c1cnc(C(F)F)s1)=O N1(C(C(CCC)OC)=O)CCC2C(C(=O)NC(C3CCCCO3)(C)C)C2C1 N1(C(C(CC)OCC)=O)CCN(C(C2CCC(N=[N+]=[N-])C2)=O)CCC1C CC(CCNC(=O)C(O)CNC(=O)C(N1CCOCC1)C)CCO c1(C(N(C2C(C)CN(C(=O)CC3(N(C)C)CC3)CC2)C)=O)ccc(F)c(C#N)c1 C1(C(N(C2CCCN(C(c3cnc(C)s3)=O)C2)C)=O)C2CC3C(C2=O)C13 c1(C(=O)NC(C2CCN(C(C(CC)COC)=O)CC2)C)cc2n[nH]cc2cc1C C1(C(=O)NCC(C)CNC(=O)C(O)C2CCC2)CSC(c2ccccc2)=N1 Cc1ccc2c(C(=O)NC(C)CC(C)NC(=O)COC3CCCCC3)csc2c1 C1(CC(=O)OC)CCC2(CC1)CCN(C(=O)NC1CCCCC1N1CCCC1)C2 N1(C(CCN(CC)CC)=O)CC2(CCC2NC(c2nnc(C)s2)=O)C1 c1(C(N2C(C3(NC(CC(C)c4cccnc4)=O)CC3)CCC2)=O)ccc[n+]([O-])c1 C1(C(=O)OC)CN(S(=O)(=O)CCN2CCCCC2C(C)(C)C)C(C)(C)C1 C1(NC(CCCC)=O)CN(C(C2CCN(c3ccncn3)CC2)=O)CCC1C c1(OC)ccc2[nH]nc(C(=O)N(C)Cc3ccccc3Cl)c2n1 Cc1cccc(OC(C)C(=O)NCC2CC2NC(c2cccc(C3CC3)c2)=O)c1 Cn1nc(C2CC2)cc1C(=O)NCC1CCN(C(=O)CN2C(=O)CNC2=O)CC1 C1(C(=O)NCCN(C(c2c(CC)ocn2)=O)CC2CC2)SC2C=CC1CC2 C1(NC(c2n(CC#C)cnn2)=O)CC(O)CN(C(C2(C)CCCCC2)=O)C1 Cc1cc(Cl)c(C(=O)NCCC(C)(C)C(C)C)cn1 CC(C)CCC(C)NC(C1OCCC1CNC(C1(F)CCC1)=O)=O N1(C(CC(CC)OC)=O)CCCC(COC)CC1.C12(CCCC1)C(=O)NC2 c1(C(=O)NC(C2CCCN(C(CCCC(C)=O)=O)C2)C)cnc2[nH]c(O)nc2c1 N1(C(CCCOCC)=O)CCC(C)C(CCNC(=O)C(C)C2CCOC2)C1 N1(C(CCCC(CC)C)=O)CCOC2(C1)CN(C(C1CCC(=O)NC1)=O)C2 c1(C(=O)NC(C)CCNC(C23CC4CC2C3C4O)=O)cc(F)cc2cnccc12 N1(C(C(CC)CC)=O)CC2(CCC(CNC(C3(CC4CC4)CCC3)=O)O2)C1 CC(C(=O)NC1CC(CNC(=O)C=CC(=O)N(C)C)CC1O)C(F)(F)F c1(NC(c2ccc(F)cc2)CCC)ccc(-c2cccnn2)cc1 C1(C(N2CC(C)(NC(C(CC)(C)OC)=O)C2)=O)COCC(C)(C)O1 Cc1nn(CC(=O)NCCOCC2(c3ccc(O)cc3)CC2)cc1Br N1(C(C(n2ccc(C)n2)(C)C)=O)CCCC(O)(CNC(c2ncccc2F)=O)C1 C(=O)(C1=Cc2ccccc2C1O)N1CCN(C(C(CCCC)CCC)=O)CC1 c1(CCNC(CC2(CC)CC2)=O)ocnc1CNC(C1CC(OC)C1)=O N1(C(c2ccc(-c3cc(C)sc3)s2)=O)CC2COCC2(CO)C1 c1(C(=O)NCCN2CCCN(C(CC(C)OC)=O)CC2)c[nH]c2cccc(F)c12 N1(C(C2C(NC(Cc3c(C)n[nH]c3)=O)C2(C)C)=O)CC2OCCN(C)C2C1 N1(Cc2ccc(OC)nc2)CCC(NC(=O)C(C)(F)F)C(F)C1 C(C(C)C(F)C(=O)NCC(C)(C)OC(C)=O)NC(C1(CC=C)CCCC1)=O c1(C(N2C(COC)CC2)=O)cnc(CNC(c2snnc2C(C)C)=O)nc1 c1(C(=O)NC(CCC)CCCNC(C2CCC2OC)=O)ccc(F)c(C)c1F c1(C(COC(=O)Nc2cccc(OC)c2)=O)cc(O)ccc1C C(=O)(CCC(=O)NN(C)C)N1C(C(NOCC(=C)Cl)=O)C(CC)CCC1 c1(C(N2CCC(CNC(C3(F)C(C)(C)C3(C)C)=O)C2)=O)cc(C#N)c(N)cc1O N1(C(C(CC=C)CC(C)C)=O)CC23CCCCC2(C1)CN(C(C1CCSC1)=O)C3 Cc1nnc(O)c(C(N2CCC(CO)(NC(C3CC(O)(C(F)F)C3)=O)C2)=O)c1C c1(N2CCC(c3ncc[nH]3)CC2)ncc(Br)c(O)n1.C1(C=O)CCOC1C1CC1 C1(C(N2CC(C(=O)NCCc3cccnc3C)(CC)C2)=O)C2CCC(C2)C1C N1(C(c2nc(CC)oc2)=O)CCC(C)C(CNC(=O)CSc2ccc(Cl)cc2)C1 c1(CC(N2CCC(NC(c3n(C)ccn3)=O)C2)=O)cccc(Br)c1F c1(CNC(CC(C)c2ccco2)=O)cc(C(=O)NCc2cccnc2)ccn1 Cc1coc(C=CC(N2CCCC(N(C(=O)Cn3cccn3)CCF)C2)=O)n1 c1(C(C2(C(C)OC)CC2)NS(CC2(CNC3CC3)CC2)(=O)=O)nnn[nH]1 N1(C(C=CCOC)=O)CC(C(=O)Nc2cccc(F)c2)CC(C)(C)C1 CC1(C)CC=C(C(=O)NCC2(O)CCN(C(=O)CC(F)F)C2)CC1 C#CC(CNC(=O)C(F)C1CC(NC(=O)Cc2ccc[nH]2)C1)C(C)C C1(F)(CNC(=O)COc2ccc(CO)cc2)CCN(C(=O)C2=CCOC2)CC1 C1(c2cn(C)nc2)CN(C(c2cc(Cl)ncc2O)=O)C2(CCC2)C1 c1(C(=O)NCC(C)=CCC2CN(C(=O)N(C)C)C2)cc(CO)c(C)s1 N1(CC(=O)N(CCCNC(=O)C(C)SC(C)C)C(C)C)C(=O)c2cccnc2C1=O N1(C(C2(C(N(C)C)=O)CCCSC2)=O)CCC2(CC1)SCCS2 c1(C(C(=O)NCC(C)NC(=O)Cc2ccco2)O)ccc(OC(F)(F)F)cc1 c1(OC)ccc(CC(N2CC(CNC(=O)CCCOC(C)C)C(O)C2)=O)nc1 c1(C(N(CC(CNC(CC(CC)(F)F)=O)O)C)=O)ccc(O)cc1[N+](=O)[O-] C1(C(=O)NCC2=CCN(C(C3C(OCC)C3)=O)CC2)CCn2nnnc2C1 C(C)(CCCCO)NC(C=CCNC(C1(OC)CCSC1)=O)=O c1(C(N(C2CCN(C(=O)Cc3cn[nH]c3)C2)CCCC)=O)ccccc1C(C)C N1(C(C(c2cccc(Cl)c2)NC(C)=O)=O)CCOCC(NC(=O)CC(C)N(C)C)C1 C(=O)(CC(C)C(F)F)NCC=CCNC(c1occ(C)c1C)=O N1(CC)C2CCCC1CN(C(=O)CC1CC3CC3C1)C2.CC1(N)CCCCC1 CC(C)(C)CC(c1nnnn1CC1CCOC1)NCC(CC1CCC1)CO c1(C(CNC2CC3CN(Cc4ccc(C)o4)C2C3)=O)ccc2occc2c1 c1(C(N2CCC(OC)(CNC(=O)CCc3ncccn3)C2)=O)c[nH]cc(C)c1=O c1(OC)ccccc1NC(c1nnc(C(N2CC(NC(=O)OC(C)(C)C)C2)=O)s1)=O c1(OCCOC)ccc(CNCC2(n3ccnc3)CC2)cc1 C1(C(=O)NC(C2CCCN(C(C3C(OC)CCCC3)=O)C2)C)CN2CCC1CC2 N1(C(C(n2c(C)ccn2)C)=O)CC(C(=O)NCCC(C)(C)C2CC2)CC(C)(C)C1 C1(C(=O)OCC)CN(CC(O)CC)CCC1O.c12cccc(c1)C(CO)O2 Cc1csc(CNC(N2CCCC2CC(c2ccc(Br)cc2)O)=O)c1C N1(C(c2c(C)scn2)=O)CCC(C(N2CC3C(C2)C3(C)C)=O)C(C)C1 Cc1cc(C(N2CCCC2(C)CCC(=O)NCCN2CCOC(C)C2)=O)ncc1N C1(C(=O)NCc2cccc(C)n2)CCCCCCN1C(C1CCC2(CCC2)C1)=O OC1CCN(c2nc3ccccc3c(=NCC3CCCS3)[nH]2)CC12CCOCC2 C12CN(C1(C)C)C(F)C(=O)OCCNC2.C(C)(C)(C)OC(=O)O.CO C(=O)(C1=NOC(C)(C)C1)NCC#CC(=O)NC(CC(=O)OCC)C N1(C(CCNC(=O)NC(C(=O)NC2CC2)C2CCCC2)=O)CC(=O)NC(=O)C1 c1(C(=O)NC(CC(C)C)C(=O)NCc2cnccn2)ccc2c[nH]nc2c1 C1(C(N(CC(C)O)CCNC(c2cncc(C)n2)=O)=O)CCCN2CCCCC12 C1(C(N(CC(O)CNC(c2cc(-c3ccccn3)no2)=O)C)=O)C2(CC2)C12CC2 c1(C2C(N(C(=O)NC(c3ncccn3)C)CCC3CC3)C2)ccccc1 Cn1cnc2c1CCCC2C(=O)N1CCC(C)(NC(c2cnc(C(F)F)s2)=O)C1 N1(C(Cn2c(C)nc(C)n2)=O)CC2CCCC1C2c1cn(-c2ccno2)nn1 C(=O)(C1CCCc2nn(C)cc21)NCC1N(C)CCN(C(c2csnc2Cl)=O)C1 C#CC1(C(N2CC=CC2COC)=O)CN(C(=O)CC2CCCC(O)C2)C1 C1(C)(CC)CC(NC(=O)C(F)C(C)CNC(C2(CO)CCOCC2)=O)CCO1 C(CN=C(NCC1CCCCC1F)NCC1CNC(=O)O1)SC c1(C(=O)NC2(C)CCN(C(C3CCC(C)CC3)=O)C2)cc(N)c(O)c(F)c1 c1(CC)ccc(C(N2CCC(C)(C(=O)N(C(C)C(F)F)C)C2)=O)cc1 C(=O)(CC(CC)NC(=O)CC1(C#N)CC1)NC(CC#C)CC C12(NC(c3c(C)csc3)=O)COC(CNC(=O)C(F)(F)C3CCOCC3)(C1)C2 c1(OC)nc(C)ncc1C(=O)NC1CC(CO)N(C(C2CCC(=O)N2C)=O)C1 Cn1cc2c(C(=O)NCC3(O)CCN(C(C4CC4(F)F)=O)CC3)cc(F)cc2n1 C(CC(=O)N1CC(SCC(F)F)C1)(C(F)(F)F)NC(C(CC)(C)O)=O C(C(CC(C)C)C(=O)NCc1ccncc1Cl)NC(c1cccc(C)n1)=O c1(C(=O)Nc2c(C)ncs2)c[nH]c2ccc(-c3cccc(C#N)n3)cc12 Cc1cnc(Cl)c(C(=O)NCC2CCCN2C(c2ccc(Br)cc2Br)=O)c1 N1(C(CSCCOC)=O)CCCC2(CCCN2C(C2CCC(C(=O)OC)CC2)=O)C1 C12(CNC(CCOC(C)=O)=O)CCC(C1)N(C(=O)CN1CCCCCC1)C2 N1(C(c2c(CC)nc[nH]2)=O)CCC(NC(C2CC(CF)C2)=O)C(CCO)C1 Cc1cc(=NC2CCCC(NC(c3ccc(F)c(Cl)n3)=O)C2)[nH]c(CO)n1 c1(C(=O)NC(CNC(CCc2cnc(C)s2)=O)C2CC2)cc2cc[nH]c(=O)c2s1 CC1CCN(C(=O)CCC2CC(NC(=O)C(C)(C)C#N)C2)CCS1 C=CCCC(C(=O)NC1CCC=CCC1)NC(=O)COCC(=C)C N1(C(c2c(CC)n(CC)nc2)=O)CC2(CCCC2NC(c2ccnnc2C)=O)C1 C(N=c1nc2sccc2c(NCc2ccc3c(n2)NCCO3)[nH]1)c1n(CC)ccn1 c12cn(C)nc1CN2.c1(C(=O)OC)csc(CNC(c2cscc2C)=O)c1 C1(C(=O)NCC(C#C)CC)(CNC(=O)CSc2nncs2)CC12CCC2 C(=O)(C#CC1CCC1)NC(CCCNC(C1CCCN(C(CCC)=O)C1)=O)C c1(OC)ccc(C2CC2)c(C(N2CC3CC3(NC(c3csc(O)n3)=O)C2)=O)c1 c1(OC)cccc2c1C(C(=O)NCC(C)CNC(c1ccc(F)cc1N)=O)CC2 C(CC(=O)NC1CCOCC1(C)C)(C(C)OC)NC(COCCCC)=O CCCCC(O)C(=O)NC(CO)CCCCNC(=O)C=C(C)C1CC1 c1(C(N2CC3(CN(C(C4(OC(C)C)CCC4)=O)C3)C2)=O)cnc(O)n(C)c1=O C(C)(C)(CCC(=O)OC(C)(C)C)N(C1(CF)CCN(c2nc(Cl)ncc2F)C1)C C(=O)(CCC(F)(F)F)N1CCC(CNC(C(CC)Cc2ccccc2)=O)CC1 CCC(N=c1[nH]c2c(c(=NCCNC(C)=O)[nH]1)SCC2)c1nccs1 C1(NC(C=CCCC)=O)CN(C(=O)CCn2ccccc2=O)CCC1CO n1(CC(=O)NC2C(NC(c3cnc(C(C)O)s3)=O)CC2)cc2ccccc2n1 c1(-c2nc(CCC(=O)NCC(CO)OCC)on2)cccc(F)c1 N1(CCC(C2CCC2)N(C)C)CC(=O)N(CC(C)(C)C2CC2)C1=O C1(NC(C2(CC=C)CCN(C(=O)CC3OCCO3)C2)=O)CCCCC1N=[N+]=[N-] c1(C(=O)NC2C(CN(C(=O)OC)C)CC2)cc2n(n1)CCCC2.C1CCC(=O)N1 N1(C(C(F)OC)=O)CCC(C2(NC(c3ccc(CN(C)C)cc3)=O)CC2)C1 c1(OC)cc(C)c(C(=O)NCC2(OC)CN(C(=O)C(C)(C)C(N)=O)C2)cn1 N1(C(C2C(Cl)(C(=O)OCC)C2)=O)CCN(C(=O)Cc2n[nH]c(=N)s2)CC(C)(C)C1 Cc1ccc(C#N)cc1C(N1CC(CC(C)NC(=O)CN2CSCC2=O)C1)=O C(CCCCCC(=O)NCC1CCCC(C)C1)NC(CS(CC)(=O)=O)=O C1(NC(C=C2CCN(C)C2)=O)CCCCN(C(=O)CC2CCCCC2O)C1 N1(C(CC23CC(C(=O)OC)(C2)C3)=O)CCCC(NC(C2CCCOCC2)=O)CC1 C1(C(N(C2CC2(C)C)C)=O)CCC(=O)CC1(C)C N1(C(CS(=O)(=O)NCC)=O)CCC(NC(=O)CN2CCSCC2)C(C)(C)C1 N1(CC(=O)N(C2CCN(C(=O)COc3ccsc3Cl)C2)C)Cc2ccccc2C1 N#CCCCCC(=O)NC12CC1CN(C(=O)COCC(F)F)C2 c1(C(N2CCCC(N(CC(C)(C)NC(C)=O)C)C2)=O)cnc2[nH]cc(C)c2c1 N1(C(C(=O)NCC)=O)C(C(=O)NCC2(CO)CCCC2)CC1C c1(C(N(CC(CN(C(C=CCCC)=O)C)O)C)=O)c[nH]nc1[N+](=O)[O-] c1(OC)ccnc(C(N2CCC(C(=O)NCC(=O)NC3CCC3)CC2)=O)c1 N1(C(C2C(COC)C2)=O)CC2C(NC(=O)CCCc3csc(C)n3)C2C1 N1(C(CCC(CC)OC)=O)CCN(C(c2cnn3ccncc23)=O)CC2(CC2)C1 N1(Cc2cccc(C)c2)CCC(C)(NC(c2sc(N(C)C)nc2C)=O)CC1 C(c1ccnc2ccccc12)=CC(=O)N(CC(CNC(CCC#CC)=O)C)C C1(NC(c2cccc(CC)c2)=O)(CO)CCN(C(c2cc(Cl)cnc2Cl)=O)CC1 N1(C(C(Cc2ccccc2)NC(c2ccc(Cl)cc2)=O)=O)CCC(O)C(F)(F)C1 C1(CCNC(c2cc(-c3cnccn3)[nH]n2)=O)CN(C(C2CCSC2)=O)CCO1 N1(C(Cc2cn(CC)nn2)=O)CCC2(NC(=O)Nc3ccc(Cl)cc3)CCCC12 CC1CN(C(c2cnc(C(C)(F)F)s2)=O)CCN1C(C1CC(C)(C)CO1)=O c1(C(=O)NC(CC(N2CCC(CC#C)C2)=O)C2CC2)cncn(C)c1=O N1(C(c2c(CCC(CC)N)ccs2)=O)CC2CCC(C1)NC2.c1(-c2n(C)ncc2)ccc(Br)cc1.NC C1(NC(CC(=O)NCC#C)=O)CCCC1(C)CN(C(=O)CC1CCCN1C)CC c1(C(N2CC(NC(c3n(C)ncc3Br)=O)C(C#N)C2)=O)c(F)ccc2nc[nH]c12 c1(C(=O)NC2(CF)CCN(C(C=CC(C)(C)C)=O)C2)cncc2ccsc12 C1(N(C(CC(CCC)NC(=O)CCOC)=O)C)CCN(C(=O)C(C)C)CC12CC2 c1(C(N2C(CN(C(CCCN(C)C)=O)C)CCC2)=O)cc(Br)c(Cl)cn1 N1(C(C2(C(C)C)CC2)=O)CCC(F)(F)C(CNC(=O)CC2CCC(F)(F)CC2)C1 CC(C)CCCC(C)C(=O)NC(C(=O)NC1CN2CCCC1C2)C(C)OC C(=O)(C(C(C)C)OC)NCc1ccc(C(N2CC(C#C)C2)=O)o1 c1(OC)cc(C(N2CCCC(NC(c3cnncc3C(F)(F)F)=O)C2)=O)ccn1 CC1(C)CN(C(c2c[nH]c3cc(F)cc(F)c23)=O)CCN(Cc2cccs2)C1 c1(C(N(CCCNC(C(C(CC)C)O)=O)CCO)=O)sc2nccn2c1C c1(C(=O)NC(CC)CNC(c2cncn2C)=O)oc2cc(Cl)ccc2c1C CC(C)CC(CC(C)C)C(=O)N1CC=CC(NC(=O)Cc2ccsc2)C1 CCCCC(C(=O)NC1CCN(C(C2CCC(CC)O2)=O)C1C(C)C)N(C)C Cc1cc(CC(=O)N(C2CN(C(=O)CC3CCOC3=O)CC2(C)C)C)ccc1F c1(SC)ccccc1C(=O)NCC1(O)CCN(C(=O)C(C)C(C)C)C1 c1(OCCC(=O)Nc2ccno2)ccc(C(=O)NCc2cnc(O)o2)cc1 c1(SCC2(C)CC(c3ccc(Cl)cc3)C2)cccc(C2CC2)c1 C1(O)(CC(N2CCCC2CCNC(=O)C(O)CC2CCC2)=O)CCOCC1 N1(C(C=CCC)=O)CC2CCC(C1CO)N2C(c1ccn(Cc2ccco2)n1)=O C(N=c1cc[nH]c(=NCCCc2ccccc2)[nH]1)c1ccc(N)cc1[N+](=O)[O-] C1(CNC(c2cn(CC)nc2C)=O)CN(C(=O)C(C)NC(N)=O)CC(C)(C)C1 C(CC(C(=O)NCCC1(O)CN(C(=O)COC)C1)NC(C)=O)SC C(C(C)C(F)C(=O)NCC(c1nncn1C)C)NC(C(CC=C)C)=O C1(C(=O)NCCOCCCNC(C2CC(C)(F)C2)=O)CC2(C1)CC2(F)F c1(CC)cc(C(N2CC(F)(CNC(C3(CC)CCNC3=O)=O)C2)=O)cc(F)c1 C1(C(=O)NC2CN(C(C)C)CC2C)CCN(C(=O)CC(C)(C)CN(C)C)C1(C)C c1(C(N2CCC(NC(=O)COC3CCCCC3)C(F)C2)=O)ccnc2[nH]nnc12 C(=O)(C(F)C(C)CNC(=O)CC1CC=CC1)Nc1cnc(OCC)nc1 c1(CNC(C(C)Cc2cnco2)=O)ccc(CNC(C2CCOC2)=O)cc1 N1(C(C=CSC)=O)CC2(CCCC2NC(c2cccc(C(C)(C)C)n2)=O)C1 C(=O)(C1=NN(CC)C(=O)CC1)N1CCOCC(NC(C(CCC#C)O)=O)C1 N1(C(C=CCC2(NC(C(CCC)C)=O)CCC2)=O)CCc2ccccc2C1 C(c1ccccc1)(C(F)(F)F)=CC(=O)N(CCCN(C)C(C1CC1(C)C)=O)C C#CC1CCN(CCNC(C(Cc2ccccc2)C(C)(C)C)=O)CC1 C1(CNC(C2C(C(C)C)(CC)C2)=O)C2CN(CCOC3CCOCC3)CC12 Cc1cc(Cl)cc(C)c1C(=O)NCC1(C(C)N)CC1.C(=O)(C(C)CC(C)C)N1CC1 Cc1cc(CN(CCNC(=O)C(C)C(C)C2CCCCC2)C2CC2)nn1C c1(CC)cc(NC(=O)C(C)N(C2CCCC2)C(=O)CC2CC(CF)C2)ccc1C Cc1ccc2[nH]c(C(c3nnnn3C3CCCC3)NC3CC(C4CC4)C3)cc2c1 N1(C(C2CC(NC(C=Cc3cn(C)nc3)=O)C2(C)C)=O)CCN2CCCCC2C1 c1(C(=O)NC2(CCNC(c3c(N)cnc(Cl)c3)=O)CC2)cc(=O)n2ccsc2n1 CC(C)CC(O)C(C)C(=O)N1CC2CC1(C(=O)NC1COCCC1(F)F)C2 N1(Cc2onc(C(C)(C)C)n2)CCC(NC(=O)CCC2CCCCO2)C(O)C1 C1(n2cc(COC)nn2)CC(C)CN(C(=O)CNC(c2ccc(C)cc2C)=O)C1 C1(CNC(C#C)=O)CCN(C(c2cc(Cl)c(C)c(Cl)c2)=O)CC1(F)F C1(NC(CN(S(CC)(=O)=O)C)=O)CC12CCC(NC(c1c[nH]cc1C)=O)CC2 c1(C(=O)NC2C(NC(C(C)Cc3ccccn3)=O)C2)cc2cn[nH]c2cn1 Cc1ccc(C)c(C(N2CCC(C)(C(N3CCC(CC(N)=O)CC3)=O)C2)=O)n1 c1(C(=O)NC(CC)CNC(=O)Cc2ccc(Cl)s2)ccc(Cl)c2cccnc12 c1(Nc2cnn(C)c2)ccc(CNC(C)=O)cc1Br.N12CCCN(CC1)C2=O Cc1ccc(F)cc1C(F)(F)C(=O)NC1CCN(C(c2ccccc2)=O)C12CC2 C(CN=C(NCC1(CO)CC(F)(F)C1)NCC1(N2CCOCC2)CCCC1)SC C(C)(CC(=O)NCCN(C(C1CCC1(C)C)=O)C1CC1)SC N1(C(c2n(CCC)ncc2)=O)CCC(C2CCN(C(=O)C=CCO)CC2)C1 N1(C(CSCCCC)=O)CCC(CN(C)C(c2cnc(OCC)s2)=O)C1.OCC N1(C(c2ccnc(OC)n2)=O)C2CCC1C(NC(=O)CSCc1ccccc1)C2 C=C(C)C(C)(C)C(=O)NC(C(=O)N(C)Cc1ncn(C)n1)C(C)CC C1(CNC(CCCC=C)=O)(OC)CCCN(C(C2CN(C(N)=O)C2)=O)C1 C(=O)(CCS(=O)(=O)CC(C)C)N1CCC(NC(C=CC)=O)C12CC2 CCCCCCC(C)NC(=O)C=CC(C)(C)NC(C1CC2(CCC2=O)C1)=O c1(C(=O)NC(CC(C)NC(C2CN(CCC)C(=O)C2)=O)C)c(N)ccc(Cl)c1F c1(OC)nc(C(=O)NCCCCC2CCN(C(=O)C(F)=C(C)C)CC2)cc(O)n1 C(=O)(CC(=O)OCC)NCC.N1(C(C(c2cccs2)N(C)C)=O)CCC1 N1(C(C2(CCC=C)CN(C(=O)C(C)(C)c3ccno3)C2)=O)CCC(N=[N+]=[N-])CC1 c1(C(C(=O)NCC23CC(NC(c4c(C)occ4)=O)(C2)C3)CO)ccc(Cl)cc1 c1(CCC)c(C(=O)NC(CNC(=O)COC2CCCCC2)C2CCC2)nnn1CC Cc1cncc(C(N2CC(NC(c3oc(CC4CC4)nc3C)=O)C(C)C2)=O)c1Cl C#Cc1cn(C)nc1C(=O)NCC(C1CC1)N(C)C(c1ccncc1Cl)=O c1(N(C)Cc2ccsc2)nc2c(c(=NCCc3cc(Br)no3)[nH]1)COCC2 c1(NC2CC(C)N(C(c3cc(Cl)on3)=O)C2)c(F)cc([N+](=O)[O-])cc1F C1(CC)CCN(C(=O)CC(C2CC2)C2CC2)C1NC(=O)COCCOC.c1ccoc1 c1(OC)cccc(C(CNC(=O)Cn2ccnn2)NC(C2CC2C(F)F)=O)c1 c1(CC(N2CCC(NC(CCN(CCC)C)=O)C2)=O)nn(C)cc1Br C(C(C)(C(=O)NOCc1nc[nH]n1)NC(c1[nH]nnc1C)=O)SC c1(CCC)ccc(C(=O)N(CC(C)(C)CNC(c2ccc(C(=O)OC)[nH]2)=O)C)s1 Cc1[nH]c2cc(Br)ccc2c1C(=O)NC1CC(NC(=O)C2=NOC(C)C2)C1 N1(C(COCCOCC#C)=O)CCC(C)C(N(C)C(c2ccsc2SC)=O)C1 N1(C(C2CCC3(CC3)C2)=O)CCC(C(N2CCC3CC23)=O)C12CC2 C(N=c1[nH]cnc(NCCc2ncnn2C)c1C)c1c(Cl)ccc(C)n1 c1(C(=O)NCC2(C(=O)NC)CC(F)(F)C2)ccc(F)cc1C1CC1 N1(C(CCOCC(C)C)=O)CC(O)CC1C(=O)NCCC(F)F C(c1ccc2c(c1)COCC2)=CC(=O)NC(CC)CN(C)C(c1cnc(S)[nH]1)=O n1(CC)ncc2cc(C(=O)NCC(CNC(=O)COCCCF)CO)cnc12 Cc1cncc(C(=O)NCC2CCCN2C(C2CN(c3ccccc3)C2)=O)c1Cl c1(OC)ccc(C(=O)NC2CC2CNC(C2(O)CCOC2)=O)cc1C1CC1 C1(NC(C2N(C)CCC2)=O)CN(C(c2cccc(C3CC3)n2)=O)CC2(CC2)C1 C1(N(C(=O)CO)CC)CCCN(C(=O)CSC2CC2)CC1 n1(CCCC(=O)NC2CCN(C)C2)c(N(C(C)C)CC)nnc1C1CCC1 C12(NC(C=C(CC)C)=O)COC(CNC(=O)Cn3nc(C)cc3C(F)F)(C1)C2 c1(Cc2ccc(C(=O)Nc3cc(OC)ncc3NC(C)=O)s2)ccc2nnsc2c1 c1(C(N2C(C(C)(C)NC(=O)CN3CCC(O)CC3)CCC2)=O)cc2scnc2[nH]1 C1(C(N2CCCC(CN(C(c3occ(C)c3)=O)C)C2)=O)CCOC(=O)CC1 C(CC(=O)N=c1cc(-c2ccccc2Br)o[nH]1)N(C(=O)Cc1cccs1)CCC c1(C(=O)NC2CCCC(NC(C3CCC(OC)C3)=O)C2)cnc2n1CCCC2 C12(C(N(C)Cc3ccc(CC)o3)=O)CC(CCO1)N(C(c1cn(CC)nn1)=O)C2 C1(OC)CCOCC1NC(=O)CONC(=O)CNC(=O)C1CC1 N1(C(CSCC)=O)CCN(C(=O)C(C)OCOC)CC1C(C)(C)C c1(C(=O)NC(CNC(CNC(CCC)=O)=O)(C)C2CC2)ccnc(F)c1N CN(CCCCC(=O)NC1CC(F)CN(C(=O)CS(C)(=O)=O)C1)N=O CC1C(C(=O)NC2(C(=O)NCC3(F)CCN(C)C3)CCSC2)=NOC1C C1(C(=O)NCC(CNC(C(CCCC)C)=O)(C)C)CC(=O)c2cc(Cl)ccc2O1 C(c1cc(C)c(C)cc1C)=CC(=O)N(CCCN(C(CSCC)=O)C)C c1(CC(N2CC(CC(C)NC(C(CCC)OC)=O)C2)=O)ccc(C)c(Cl)c1 c1(C(=O)NC2CN(C(c3cncc(OC)c3)=O)C3C2C3)ccc(F)c(F)c1C C1(C(C)NC(CCCN(C(C)=O)C)=O)CCCN(C(c2cnoc2)=O)C1 C(=O)(C1=C(Cl)CCCC1)N1CCC(CN(C(=O)CC2CC3(CCC3)CO2)C)C1 CC1CCC(F)(C(N2CC(O)(CNC(=O)Cc3cnc(C4CC4)[nH]3)C2)=O)CC1 N1(C(C(=O)NCc2nnn(C)n2)CC2CCCC(=O)N2)CCOc2ccccc21 N#Cc1ccccc1C(C(F)(F)F)NC(N1CC(C(=O)NCCCl)C(O)C1)=O c1(C(=O)NC2(C)CCN(C(CCn3c(C)ccc3C)=O)C2)ncc2n1CCCC2 C(=O)(C(C)CC(F)F)N1CCC(N(C(c2cn(C3CCOC3)cn2)=O)CC)CC1 C(=O)(C(Cl)=CCl)NCC(Cc1ccccc1)NC(C(C)OCCC(C)C)=O N1(C(C(CC=C)CC)=O)CCC2(C1)CN(C(=O)COc1ccccc1C)CCO2 c1(CC)n[nH]c(CNC(c2ccc(-c3ccc(F)cc3)o2)=O)c1Br n1(CC)ncc(Cl)c1C(=O)N(CCC(=O)NCCCS(C)(=O)=O)CCO C=CCC(C(=O)N(CCN(C)C(C1(C(C)C)CCCO1)=O)CCOC)OC C#Cc1cn(C)nc1C(=O)NCCCNC(=O)Cc1nnc(C)s1 Cn1c(O)nc(N2CCC(NC(=O)C(F)C3CCOC3)C23CCC3)cc1=O C1(NC(C2(C)CCC2)=O)CCCCCC1NC(C1CCC2(CC2)C1)=O N1(C(CCCC(C)C)=O)CCOCC(C)(CNC(C2CCCCCC(=O)C2)=O)C1 c1(N(C2CCN(C(c3cn[nH]c3)=O)C2)C)nc(Cl)nc2c1S(=O)(=O)CC2 CCC(O)C(C)(C)C(=O)N1CC2(CC(C(=O)NCCOCC3CCC3)CO2)C1 C=CC1(O)CCN(C(C2CC(NC(=O)Cc3cncs3)CCO2)=O)C1 C#CCCCCC(=O)NCc1csc(CNC(=O)C(c2ccc(F)c(F)c2)C)n1 N1(C(CCN(C)C)=O)CC=CC1C(N1CC=CC1CN(C)C)=O c1(C(C)NC(N2CC(=O)N(c3cn[nH]c3)C2)=O)ccc(C(F)(F)F)cc1 CCC(CC(=O)NCC(O)C(=O)Nc1ccc(C2CC2)cc1)SC N1(C(Cc2c(C)ocn2)=O)CC(C)(C)OCC1CNC(c1cc(C)n(C)n1)=O Cc1cc(C(=O)N(C2CN(C(=O)CC3C=CCC3)C2)C)c2c(c1)CCC2 C(=O)(C1=C(Cl)CCC1)NCCC1CCN(c2nccc(Cc3cnc(C)o3)n2)C1 c1(C(=O)NCCCNC(CCCNC(C)=O)=O)ccc2c(c1)NC(=O)CCN2 c1(OCC)ccc(C)cc1C(=O)NC1(C)CCN(C(=O)C(C)(Cl)Cl)C1 C12(C(=O)NC(C3CCCC3)CNC(=O)CCC3CC3(Cl)Cl)CCCN1CCC2 c1(C(=O)NC(CN(C(c2c(SC)scc2)=O)C)C)ccc(F)c2occc12 C1(C(=O)NC(C(=O)NCC(C(=O)OC)OC)c2ccoc2)CCCC(O)C1 CC(C)C(F)(CNC(c1cnn2c1OCC2)=O)C(=O)NC1(C2CCC2)CC1 CCCCC(C(=O)NC1CCOC1)NC(c1ccc(CC)[nH]1)=O C1(C(=O)NCCCNC(CCCC)=O)COCCOC1 C1(O)(CNC(=O)COCC(F)(F)F)CCN(C(=O)CNC(=O)C(F)(F)F)C1 CCCCC(CC)C(=O)N1CCC(NC(c2c(I)n[nH]c2C)=O)C1 C1(C(=O)NCC(c2cccc(OC)c2)NC(COCC=C)=O)CCCC(C)CC1 C=C1CCC(C(=O)NCCC2CCCN(C(C3CC(F)CN3C)=O)C2)CC1 c1(C(N(C(CC)CC(=O)NCC2C(C)(C)C2(C)C)C)=O)ncc(F)cc1F CCCC(CC)C(=O)N1CC(C)(CC(=O)NOCCF)CC1(C)C N1(CCC)CCCC(C(N2CCC(N(C(=O)CSCC(F)(F)F)CCC)C2)=O)C1 C1(NC(c2n(CC)nnc2)=O)CC2CCCC(C1)N2C(=O)CN(C)CCO N1(C(c2scc(OC)c2)=O)CCC(C)C(NC(c2ncoc2Br)=O)C1 c12ccc(OC)c(c1)CCSC1(CC(F)(F)C1)CNC2=O.C(C(F)(F)F)OC N1(C(COCc2c(C)cccc2)=O)CCCC(CC(=O)O)CC1 c1(C(NOCC(=O)NC2CCCCC2O)=O)ccn2nccc2c1 c1(C(c2nnnn2CC(F)F)NCc2n(C)ncc2)cc(Br)cc2c1OCCC2 C=CC1(C(=O)NC(C)(C)CC2CC2)CCN(C(=O)CCc2ccoc2)C1 c1(CC(=O)NC(CCNC(c2c(C)nc(SC)s2)=O)C)cc(C)ccc1F n1(CC#C)c(C)cc(C(=O)NC2CC2NC(c2ccnnc2O)=O)c1C c1(CNC(C2CCC(C(=O)Nc3sccc3I)CC2)=O)ccc(Cl)cc1Cl N1(C(C(C2CCN(C(c3cc(OC)nn3C)=O)C2)F)=O)CC(OC)CC1(C)C c12nc(=N)[nH]cc1C(=O)NCCC1N(CCC1)C(=O)CC2.C1(N)CCCSC1.CC c1(C(=O)NC2CCN(CCNC(c3scc(C)c3)=O)CC2)ncc([N+](=O)[O-])n1C c1(OC)ccc(CCC(N2CCC(F)(C(=O)NC(C)C(N)=O)C2)=O)cc1 CC1(CNC(=O)Cn2cc(Br)c(=N)[nH]2)CCCN1C(c1cnsc1)=O c1(CN2C(C)(C(=O)Nc3cccnc3C(N)=O)CCC2)ccnc2ccccc12 c1(C(N(C2CCN(C(=O)Cn3cc(CO)nn3)C2)CC)=O)cnc2cc[nH]c2c1 c1(CN2C(C(=O)Nc3ccnc(Br)c3F)CC(O)C2)cc(F)cc(F)c1O c1(C(=O)OC)ccccc1CCn1nc(-c2cccs2)nc1COc1ccsn1 N1CCN(CCNC(C=CC(C)C)=O)CC1.C1(CCC(=O)N)NC(=O)NC1=O N1(C(c2ncn(C)c2)=O)CCCC(C2CCCN(C(=O)C(O)CC(C)(C)C)C2)C1 C12(NC(c3cc4cnccc4[nH]3)=O)CCCC1CN(C(c1cc(Cl)no1)=O)C2 N1(C(C2(C(=O)NC)CC2)=O)CCC2(CC1)CN(C(=O)CS(N)(=O)=O)CCO2 C1(C(=O)NC(c2nc(C)[nH]n2)CO)C=CCN(C(c2nc(Cl)cs2)=O)C1 c1(C(N(CC#C)CC)=O)cnn(CCNC(c2nc(Cl)cs2)=O)c1 CC1(CNC(=O)CC2CC3CCC2C3)CCCN1C(=O)CC1CCC2CC12 S1(=O)(=O)c2ccc(C)c(c2)C(=O)N1.c1(N2CCC(CC)C2)ncc(Br)c(C(=O)O)n1 c1(C(=O)OC)c(C)[nH]c2cc(OC3CCN(C(c4ccco4)=O)CC3)ccc12 c1(N2CCC(NC(c3cccc(C(N)=O)n3)=O)C2)nc2cc(Cl)cc(Cl)c2o1 C1(CCNC(CN(C)CCO)=O)CCCN(C(=O)CCCC2CCCC(=O)N2)C1 N1(C(Cn2ncn(C)c2=O)=O)CC(CNC(C2CCCS2)=O)C(F)(F)C1 N1(C(C(CC)=O)=O)CCC2CN(C(c3cccc(C(F)F)c3)=O)CC12 N1(N2CC3CCC2CC3)CCC(CC=O)C1(C)C.C(C(C)C=O)SC c1(OC)ccc(OC)c(C(N2CCCC(CNC(C3CCCN3C)=O)CC2)=O)n1 c1(C(C(=O)NCCC(C)NC(C2COC(C)(C)C2)=O)(F)F)ccccc1F C1(NC(CCC=C=C)=O)COC2(CCN(C(=O)CCN(CCCCOC)C)C2)C1 C12(C(=O)NCCC3CCCN3C(=O)C#CC3CC3)CCC(C1)OC2 c1(C(=O)NCC(CNC(C(COC)C)=O)(C)O)nc(OC(C)C)ccc1Cl c1(-n2cc(C(CC)N)nn2)ccccc1CNS(=O)(=O)CC C1(CC#C)CN(C(=O)C(C)N(C(=O)C2=C(C)CC2)C2CC2)CCO1 C1(N)(C(=O)NC(c2nccs2)C)CC2CCC(C2)C1 C1(C(=O)NCC(C)N(C(=O)CN(c2ccncc2)CC)CC)CCC(F)(F)CC1 N1(C(C2(C=C)CCN(C(=O)CCN(C)C)C2)=O)CCC2(CCOC2)C1 c1(C(=O)NC(C(C)C)CCN(C)C(C2(C)CC2(F)F)=O)cc(F)cc2ccoc12 c1(NCC(C)NC(c2c(OCC)nc(C(F)(F)F)cc2)=O)ncccc1[N+](=O)[O-] C(=O)(C1=CCC(F)(F)CC1)N(C1N(C(CCOC)=O)CC(F)C1)C1CCCCC1 c1(C(=O)NCC2C3CN(C(CC(=O)NCC#C)=O)C(C3)C2)ccn2ccnc2n1 c1(CCNC(=O)NCCCC(O)CO)cc(F)c(F)cc1I c1(C(=O)OC)nc(NCCC2CCCCN2C(c2cnc(C)s2)=O)sc1C Cc1ncc(C(=O)NC(CCC(C)C)C(=O)NCc2nn[nH]n2)cc1C#N N1(C(C2CCN(OC)CC2)=O)CC(NC(=O)C(C)C(C)(C)C)Cc2ccccc21 C1(N(C(=O)CCc2cnoc2)C)CCCCN(C(c2cnnc(C3CC3)c2)=O)C1 C12CN(C3COCC3O1)C(=O)C13C4CC1C1C2C4C31.C1(C(=O)NC)CC(O)C1 c1(C(=O)NC(C(C(C)C)C)CNC(=O)C2=CCCCC2)cc2n(c1)CCSC2 c1(C(=O)NC2C(CNC(C(c3cccc(C)c3F)O)=O)C2)cccc2nccn12 c1(C(C(N2C(C(C)C)C(C(C)C)C2)=O)C)cc2ccccc2s1 N1(C(CCC(CC)=O)=O)CC2CCC(N(C)C(c3ccc(C(N)=O)[nH]3)=O)C2C1 C1(C(N2CC(NC(C(CCCC)F)=O)C(C)(C)C2)=O)CCOC2(CCC2)C1 c1(OC)cc(Br)cc(F)c1CN1CCCC(C)(C(=O)NC2CC(C)C2)C1 CC#CC1CCN(C(C2(CC=C)CCN(C(C3CC34CCOCC4)=O)C2)=O)CC1 C#CCC(CC#C)C(=O)N1CC(CN(C(=O)CC2(O)CCC2)C)C2(CC2)C1 C1(C(=O)NC2CN(C(C=C(C)c3ccccc3)=O)CC2F)OCCOC12CCC2 N1(C(c2c(C)nc(CO)s2)=O)CCC(NC(=O)C(C)P(C)(C)=O)C(F)C1 C1(NC(=O)CC2CSC2)CCCN(C(=O)C(CN2CCCC2)c2ccccc2)CC1 C1(NC(c2cc(F)c[nH]2)=O)COCCN(C(C2CCOC2)=O)C1 C1(C2CCN(C(=O)CCCCCCCCCO)CC2)(NC(=O)C(O)C(F)F)CC1 Cc1cc(C(N2CCC(CCNC(=O)C(O)C(C)C)CC2)=O)cc(C)c1C CC12CC(CC(=O)Nc3ccccc3C3CCNCC3)(CO1)C2 N1(C(C(C)(C)C)=O)Cc2occ(C(=O)NCc3cc(O)ns3)c2C1 N1(C(=O)C=Cc2ccc(Br)s2)CC2CCCC(C1)N2C(=O)Cc1cn[nH]c1 C1(NC(C(CC#CC)NC(C2CCCC2OC)=O)=O)CCc2nncn2C1 C(=O)(CCCCCS(N)(=O)=O)NCC(CNC(C1(C)CCN(C)CC1)=O)C(F)(F)F c1(C(=O)NC2C(N(C(=O)C(C)OC)CCC)CCC2)ccnn1CCOC(C)C c1(C(=O)NC2CN(C(C3CCCN(C(=O)OC)C3)=O)CC2O)ccc(F)c(F)c1 c1(C(=O)NCC2(F)CC(CNC(c3c(C)snn3)=O)C2)nccn2nccc12 C1(OC)CCC12CC(C(=O)N(CCCCNC(C1(O)CC1)=O)C)C2 C1(C(=O)NC(CNC(c2scc(C)c2)=O)CCOC)CN=C2N=CNN2C1 CC(CCC(C)(C)C)C(=O)Nc1cc(-c2cccc(F)c2CO)cs1 c1(CC(=O)NC2(C)CCN(C(c3ccc(C)n3C)=O)C2)cc(Cl)ccc1Cl C1(N(CCCn2cc(C3(F)CN(C=O)C3)nn2)C)CC1C1CCCC1.c1cc[nH]n1 c1(C(N2CCC3(CC2)CC3)C(=O)NC(C(=O)OC)C)cccc(C)c1Br C=CCCC(C)(C)C(c1nnnn1C(C)CC)NC(CC)(CC)CO Cc1cc(NC(C2CCN(C(c3cnn4ccsc34)=O)CC2)=O)cc(C)c1C C1(CC(N2CCOC(CNC(=O)CCCc3nccs3)C2)=O)(OC)CCCCC1 c1(CC)ccc([N+](=O)[O-])cc1C(=O)N(C(C)CN(C)C(C1(F)CC1)=O)C C=CCC(CC(C)C)C(=O)N1CCCC1(C(=O)NC(C)C(F)(F)F)C(C)C N1(C(C(C)(C)C2CC2)=O)CC(NC(=O)Cn2nc3c(n2)CCCC3)C2(CCC2)C1 c1(CN2CCC(CN(CCC)C)C2)cc2ccc(Br)cc2nc1Cl CCC(C)(C)C(O)C(=O)NCC1(OC)CN(C(=O)CC2CCCCC2)C1 Cc1ccc(C(C)C)cc1C(=O)NC1CCC(NC(c2cncnc2)=O)CC1 c1(C(C)C(=O)NCCCn2cc(-c3ccc(OCC)cc3)nn2)nc(F)ccc1Cl C(C1CN(C(=O)Cc2ccco2)Cc2ccccc21)NC(C1CN2CCN1CC2)=O CC(C)(C(=O)NCCN(C(=O)C(F)OC(F)(F)F)C1CCCC1)c1cncnc1 C1(NC(=O)CCCCC2CC2)CCCCCN(C(c2c[nH]nc2-c2cccs2)=O)C1 C(=O)(N=c1cc(C2CC2)n(C)[nH]1)C1C(C(N2CCCCC2CN(S(C)(=O)=O)C)=O)C1 c1(OCC(=O)NCC(C2CCC2)NC(C2CCOCC2)=O)ccc(Cl)nc1 c1(C(N(C)CC)=O)c(F)ccc(F)c1NC1CCN(C(C)=O)CC1 C(=O)(C(=O)N=S(C)(C)=O)NCCC1N(C(c2c(OC)cc(F)cc2)=O)CCOC1 c1(C(=O)NCC(=O)NC(C)C(C)NC(c2cn(C)nc2Cl)=O)c(F)cccc1Cl C#CC(C)(C)C(=O)N1CCN(C(C2CC3CCC2C3)C(=O)NC(C)(C)C)CC1 c1(C(=O)NC(CN(C(c2nc(C#C)sc2)=O)C)CC)c[nH]c2nccc(Cl)c12 Cc1nccnc1C(=O)NC(C)(C)CCNC(=O)CSCc1cccnc1 c1(CC(=O)NCCC2CCC(NC(C3CCCSC3)=O)C2)cccc(F)c1F c1(OC)ccc(F)c(C(=O)NC(C2(O)CN(C(=O)CCCN(C)C)C2)C)c1N N1(C(C(N2CCC(C)CC2)=O)=O)CCC2CN(C(c3nc(Cl)cs3)=O)CC12 c1(OCC(=O)NCCn2cc(CSC)nn2)ccc2ccccc2c1 c1(C(=O)OC)c(NC(C2CCN2C(c2ncc(Br)cc2C)=O)=O)sc2c1CCC2 C(C(C(=O)NNc1ccc(C#N)c(F)c1)n1cc(COC(C)(C)C)nn1)OCC C1(O)(CN(C(=O)CC2(C)CC2)C)CCCN(C(C2(C#N)CC23CCC3)=O)C1 C1(N(C(CCN(CCC)C)=O)CCNC(=O)CCNC(N)=O)CCCCC1 c1(C(=O)NC2CN(C3CN(C(CCC#CC)=O)C3)C(=O)C2)ccc([N+](=O)[O-])s1 C(CCCCNC(=O)C(C)(C)N1CCCC1)N(C(CCC1CC(OCC)C1)=O)C N1(C(C2ON=C(C)C2C)=O)CC(NC(=O)Cc2cccn2C)CC(F)C1 C(=O)(C(C)C(C)C(C)(C)C)N1CCC(N(C(=O)CCCS(C)(=O)=O)CCC)CC1 c1(N2CC3C(C(=O)NC4(c5ccncc5)CC4)C3C2)ncnc2sccc12 C(=O)(CCCC(=O)OCC(=O)NC(=O)Oc1cc(F)ccc1N1CCCCC1)OC c1(C(=O)OC)sc2ccccc2c1C(=O)OCc1cc(CSC)no1 CCCC(C(=O)NCC(C)(C)CNC(=O)CSc1nnc(C)n1C)C(C)C CCCS(=O)(=O)CC(=O)N(CCCNC(c1ccc(Cl)nc1Cl)=O)CC Nc1cc(C(N2CCC2C2CCCN(C(=O)Cc3ccncc3)C2)=O)ncc1F CCC(N=c1ccnc(N2CCC=C(C)C2)[nH]1)c1ccc(OC)c(OC)c1 c1(CC(N2CC(C)C(NC(C3(C)CC3C)=O)C2)=O)cc2ccccc2o1 C1(C(N2CCC(C(C)NC(C3CC4(CCOC4)C3)=O)CC2)=O)COCC(C)(C)O1 C=CCN=C(NCc1ccccc1N1CCCC1)NC1CC1 N1(C(C2C(C)(C)CN(C(=O)C(C)(C)C#N)C2)=O)CC2(COC(=O)C2)C1 CC(Cc1cnc[nH]1)C(=O)NCC(O)CCNC(=O)CCc1cncn1C c1(NC(C(=O)NCCN(C(C(C)CC2CCCCC2)=O)C)=O)cccc(C#N)c1 N1(C(c2cncc(C(C)C)c2)C(=O)NCCSC)CCN(C)CC1CCO C1(NCC(C2(C)CC2)OC)C(C#N)C1(C)C.C12(CCCC1)C(=O)NC2 c1(C(N(C2CCN(C(c3coc(N(C)C)n3)=O)C2)CC#C)=O)cc(F)cnc1O C1(O)(CNC(c2ccc(F)cc2)=O)CCN(C(c2ccccc2CO)=O)CC1 c1(OC)c(C)nc[nH]c1=NCC1(F)CCN(C(C2(OC)CC2)=O)CC1 N1(C(c2ccnc(C)c2C)=O)CCC2CCCC12CNC(=O)CC(=O)NC1CC1 CC1C(C)N(C(c2ccncc2F)=O)CCN1C(=O)Cc1csc(S)n1 C1(C(=O)NC(c2nnc(C)o2)C)CN(C(C2CC3(CCC3=O)C2)=O)CC1(C)C N1(C(C(CCCC)C)=O)CC2CCCCC2(CNC(c2nc(Cl)oc2C)=O)C1 C1(NC(CCc2onc(C(C)OCC)n2)=O)CC2CN(C(=O)C(F)(F)CC)CC12 Cc1nc(C(C)(F)F)ccc1C(=O)N(CC(C)CNC(c1cnc(N)cn1)=O)C c1(CC)ccc(OC)c(C(N2CC(O)CCC2C)C(=O)NC2CCOC2)c1 N1(C(C(c2cccc(Br)c2)N(C)C)=O)CCC(NC(C2CCC2)=O)C12CCC2 N1(C(c2nccc(C)n2)=O)C2CCC1CC(NC(c1cccc3nonc13)=O)C2 C(C(=O)N=c1ccn(CC2CC2)[nH]1)C1(C)CN(C(C2C(C)CC(C)O2)=O)C1 N1(C(c2c(CC)ncnc2)=O)CCN(C(=O)CC2(C)CCCC2)CC12CC2 CC1CC(NC(c2cc(C3CCOCC3)[nH]n2)=O)CN1C(=O)C=CC(N)=O C1(CC=C)(C(=O)NC2(C)CC2C)CCN(C(C2(n3cnnn3)CCOCC2)=O)C1 Cn1cc(C(N2CC(NC(=O)CCC3CCOC3)C(O)C2)=O)ncc1=O C12(C(=O)Nc3c(CC)cccc3)CCN(C(=O)CCCCC(N)=O)CCC1C2 C1(C(N2CCCC(NC(C(C)(C)C3CC3)=O)C2)=O)CC(=O)c2ccccc2C1 N1(C(CCCc2ccc(C)s2)=O)CCCCC(NC(=O)COCC2(F)CC2)CC1 N1(C(C2=C(C)OCCC2)=O)CC2CCC1C1CN(C(=O)CN3CCCC3=O)CC21 c1(C(=O)NC23C(CN(C(Cn4cc[n+](C)c4)=O)C2)C3)nnc2ccccn12 c1(C(N2CCCC(CCNC(C(CC)=CC)=O)CC2)=O)cc2nc(Cl)ccc2o1 CC(CNC(C1CCC1CF)=O)(CO)NC(C1(CSC)CCC1)=O C(=O)(C1=CCC2(COC2)OC1)NCCC(=C)CNC(c1cc2ncccc2o1)=O CC(C)(CC(=O)NCCN(C(=O)CN1CSCCSC1)C1CC1)c1ccccc1 C1(NC(c2nc(C)[nH]n2)=O)CC(C2CCN(C(c3cc4c(s3)CCC4)=O)CC2)C1 C1(C(=O)OCC)C2CC1N(N1CCCC(O)C1C)C2 Cc1cc2c(cc1NC(c1occc1Br)=O)CCO2 C12(C(=O)NCCn3cc(C(N(C(CC)C)CCO)=O)nn3)CCCC1CCC2 C1(N(C)C(c2cnn(C3CC3)c2Cl)=O)CN(C(C2CCCS2)=O)CC1(C)C C(=O)(C#CC1CCOCC1)NCC1CCCC(NC(c2nn(C)c(=O)cc2)=O)C1 C1(NC(C=CCOC)=O)CN(C(c2cccc(C(=O)OC(C)(C)C)n2)=O)CCC1F c1(N(C(C)CNC(=O)Cc2ccc(C)cc2)C)ncnc2cnn(C)c12 C(=O)(CC(C)(C)CNC(C1(N(C)C)CCSC1)=O)N(C1CCNC1=O)C C1(C2(C)CC2)(C(N2C(CCC(=O)NC3(CC=C)CCCC3)CCC2)=O)CC1 n1(C(C)C)ncc(C(=O)NCC2(CN(CC(c3ccccc3)C)C)CCC2)n1 CCC(Cc1ccccc1)CC(=O)N(CCC(C)NC(=O)CSC(C)(C)C)C c1(C(=O)NC(CC(C)NC(c2cc(C(F)F)ccn2)=O)C)nnn(C)c1N c1(CC)[nH]nc(Cl)c1C(N1CCC1CNC(=O)CNC(C1CCC(=O)N1C)=O)=O N1(C(C(CN(CC)CC)C)=O)CCC(C)CC1C(N1CCCN(CCO)CC1)=O O(C=CC(=O)NCC1CCCN1C(c1ncccn1)=O)CC N1(C(C2N(C(C3(OC)CCOC3)=O)CCC2)=O)CC(C)CC(C)(C)C1 N1(C(C(C)SC)=O)CCN(C(C23CC4CC2C3C4)=O)C(c2ccccc2)C1 Cc1cc(F)ccc1C(=O)NCC1(O)CCN(C(=O)C2=CCCC2C)CC1 C(=O)(C(CN=[N+]=[N-])NC(=O)C=Cc1ccsc1)N(C)CC1CCN(C)C1 c1(C(=O)OC)cc(C(=O)NC2CC(NC(=O)CN(C)C(C)=O)C(O)C2)n(C)n1 N1(C(c2nccc(OCC)c2)=O)CC2CN(C(=O)CCN3CCOC3=O)CC12 c1(CN2CCCCC2)ccc(F)cc1F.N12CCCC1NC2=O CC1(C)CCN(C(=O)Cc2ccccc2)CC1NC(=O)CC1CSCCS1 CC(C)C(F)C(=O)NCCC(O)CNC(c1cnnc(-c2ccccc2)c1)=O CC(c1cccs1)=CC(=O)NCC1CC(NC(=O)C(C)NC(c2ccoc2)=O)C1 c1(C(=O)NCC(=O)NCCN(C(CC=C)=O)CC(C)O)cccc(Cl)c1 O=C(C(F)CC1CCCC1)NC1CCCC1C(=O)NCC1CC(Cl)(Cl)C1 c1(CC)cc(C(=O)NC2CCN(C(c3cnc[nH]c3=N)=O)C23CC3)ccc1OC c1(NCC(=O)NCC2CC(N(C(C(C)C)=O)C)C2)cccnc1Cl S(=O)(=O)(CC(=O)NCC1(C)CCCN1C(c1coc(C(N)=O)c1)=O)N(C)C N#CC1(C(N2CCC(CF)(NC(C34CC(F)(C3)C4)=O)C2)=O)CC2C=CC1C2 C12(NC(c3c(OC)scc3)=O)CCCC1N(C(C1(NC(C)=O)CCCC1)=O)CC2 C1(CC(=O)N(C2CCOC2)C)CCN(C(C2CC(OCCO)C2)=O)CC1 c1(C(=O)NCC(CC)(CC)NC(=O)CC2(C3CC3)CC2)nccn2ccnc12 C1(NC(=O)C(O)C(F)F)CC2CCCC(C1)N2C(=O)CCCC1CCOCC1 C=CCCC(C(=O)NCCN(C)OC)NC(c1cnns1)=O C1(C(=O)NCC2CCCCN2C(=O)Cc2n[nH]cc2Br)CC12CCSCC2 C(N=c1[nH]c(=NCC2CC(C(F)(F)F)CO2)c2ccccc2[nH]1)c1n(C)nnc1 C(=O)(C1=CNS(=O)(=O)N=C1C)NC1CCC2(CC1)CC2NC(C(CCCC)O)=O CC(CO)C(C)N=c1[nH]c(=NCCN2CCOC2=O)[nH]c2c1COC2 N1(C(CCCC#C)=O)CCC(CO)C(NC(c2ncn3c2CCC3)=O)C1 c1(NC(=O)CNC(c2cnn(-c3ccccc3)n2)=O)ccccc1Br O=C(C1=CC2(CCOC2)C1)N1CC2CCC(C1)N2C(C1C2CCC(F)(F)C12)=O N1(C(COCCC(C)C)=O)C(C(=O)NCC(C)(C)C2CCCO2)C2CC(O)C1C2 c1(C(N2CCC(CC)(NC(=O)CCc3ccsc3)CC2)=O)cc(C#N)c(C)cn1 N1(C(C=NOC)=O)CCN(C(c2ccc(CSn3cncn3)nc2)=O)CC(O)C1 N1(CCC)CC(NC(C2(COC)CC2)=O)CC1=O.C1(O)(CO)CCN(C(=O)COC)C1 C1(C(=O)NC(C2CN(C(c3c(C)cc(C)s3)=O)C2)C)CCc2n[nH]cc2C1 C1(C(C(=O)NC2CC(CNC(=O)C(O)C3CCC3)C2)OC)CCC(F)(F)CC1 C(=O)(C1=CC2CCCCC12)N1C(C)CC(CNC(c2ccn(C)c(=O)c2)=O)CC1 CC(C)(CO)C(=O)N1CC(C)(CNC(=O)CC2CC=CCC2)C1 c1(C(=O)NCCCCCNC(C2(CC#C)CCCCC2)=O)c(OC)cccc1Cl C1(NC(C(COC(C)C)C)=O)CC2CC(NC(c3c[nH]c(C(N)=O)c3)=O)CC12 C1(C2CC2)CC(=O)NCCOCCC(=O)N1.CCCCCOCC C1(NC(c2nccc(CC)c2)=O)CCCCN(C(C2CCNC2=O)=O)C1 C1(C(CNC(C(COC)O)=O)F)CCN(C(c2c[nH]c(C(N)=O)c2)=O)CC1 c1(OC)cccc(C)c1C(N1CCC(O)(C(C)NC(C2CCC2(C)C)=O)C1)=O C(=O)(C1OC(=O)c2ccccc21)NC1C(C)(C)CN(C(C23CC(CO)(C2)C3)=O)C1 N1(C(c2cc(OCC)n[nH]2)=O)CCCC1C1CCCN1C(c1ccnc(C)c1)=O Cn1nc(C(=O)NCC2(F)CC(NC(=O)C3=CCCOCC3)C2)c2c1CCSC2 C1(C(N(C)C)=O)CCN(C(c2cc(C(C)(C)C)no2)C=O)C1.C(COC)N N1(C(C=CC)=O)CCN(C(c2cc(F)ccc2C(C)C)=O)CC1C(F)F CC1CN(C(c2ccco2)=O)CCC1N(CC1CCCN1C)CC1CCCCO1 C1(NC(C(C(C)C)OC)=O)COCCN(C(=O)Cc2cc(C(C)C)no2)C1 CC(CC(F)(F)F)C(=O)N1CCCC1CN(C(=O)C(F)(F)C(O)C1CC1)C C(=O)(CCCC(=O)N(C1CC1)CC1CCCN1C(=O)CCOC)N(CC)CC C1(NC(CCC=C=C)=O)COC2C(NC(c3sccc3OC)=O)COC12 c1(CC)c(C(=O)NC(CC2CCCC2)C(=O)NCC(C)CCC)nnn1C C1(C(=O)NC(C)(CNC(=O)C=CCF)C2CC2)CC2(C1)CC2F N1(CC(C)(O)C(=O)Nc2cccc(C3CCOCC3)c2)Cc2ccccc2C1=O CC(CS(C)(=O)=O)C(=O)N(CC(C)(C)N(C(=O)C(C)Cc1ccccc1F)CC)C CC12CC(CC(=O)NCC(c3ccc(O)cc3)NC(C3CC3(C)C)=O)(CO1)C2 c1(C(=O)NC(CNC(CCc2cnc(C)s2)=O)C)cc(N)ccc1[N+](=O)[O-] c1(C(=O)NC2(C(N(c3c(C(=O)OC)nccn3)C)=O)CC2)ccc(Br)c(C)n1 CC1CC(NC(C2CCC(C)(C)CC2)=O)CN(C(=O)C(Cl)=CCl)C1 n1(C(C)C(=O)O)nccc1NC(=O)C(C)Cc1ccnn1C c1(C(N2CCC(O)(CNC(CC3C(C)(C)CC3)=O)C2)=O)coc2c(F)cc(F)cc12 N(C(=NCc1nnnn1C)NC1COC(C2CC2)C1)C1C2(CC2)C(C)CC1 C(=O)(CS(=O)(=O)C(C)C)N1C(C)CC(NC(CNC(C(CC)C2CCCC2)=O)=O)C1 C(=O)(C(=O)NC1CC1)N(CCN(C)C)CC1CC1 c1(C(=O)NCC2CCC(NC(c3nc(Cl)cs3)=O)C2)cc([N+](=O)[O-])c[nH]1 c1(C(N(C2CCN(C(CSC)=O)CC2C)C)=O)cccn2ccnc12 C(=O)(C(=O)N(CCCCOC)C)NCCC CN1CC2(CCN(C(C3CCC34CN(Cc3ccccc3)C4)=O)C2)CC1=O C1(C(N(CCCCCCC)C)=O)CN(C(c2cc(CO)n(C)n2)=O)C2(CCC2)C1 c1(C(N2C(CNC(=O)CSC(F)F)CCC2)=O)[nH]c2ccccc2c1CC(N)=O N1(C(C(C)C2CCCC2)=O)CCCC(N(C(c2ccc(C(N)=O)o2)=O)C2CC2)C1 c1(C(N2CCC(NC(C(C)C3CC3)=O)(CF)C2)=O)ccn(C)c(=O)c1 Cc1cccc(C(=O)NCC2(CCNC(c3ccc(C)n3C)=O)CC2)c1C(F)(F)F N1(C(C(=O)N(CC)Cc2nn[nH]n2)=O)CC(O)CC1C c1(C(N(CCNC(C2(C=C)CC2)=O)CCOC)=O)ccccc1S(=O)C(F)(F)F C1(C(=O)NC(c2cccnc2)COC)CC(C)C1(C)C c1(C(=O)NC(CC=C)CNC(=O)CCOCC(F)(F)F)cn(C)nc1OC C1(NC(CCC=CC)=O)CCC2CCN(C(=O)C(C)(C)CC3CC3)C1C2 C1(C(=O)NC(COCC)C(C)C)CN(C(c2cn(C(C)C)nn2)=O)CC1F CCC(O)C(C)C(=O)NCCOCCN(C(=O)C(C1CC1)SC)C N1(C(CC2CC(=C)C2)=O)CCCCCC(NC(=O)C(C)(O)C2CCC2)C1 N(C(=NCC1CCOC1C)NCC1(C2CCC2)CC1)C(C)C C1(CNC(C(C(=C)Cl)(C)C)=O)CC2(CCC2)CN1C(c1sccc1C1CC1)=O Cn1cnc(C(=O)NC(C(=O)NCC2CC23CCC3)C2CCC2)c1 N1(C(=O)C(F)=CCCF)CCCCC(CNC(=O)Cc2cnc(C3CC3)[nH]2)C1 c1(OCC#C)ccc(C(=O)NC2CC(=O)N(c3ccc(Cl)cc3)C2)cc1C c1(C(N2CC3(C(NC(=O)Nc4ccc(C)cc4)C3)C2)=O)cccc(S(C)(=O)=O)c1 N1(C(C(CC)NC(N)=O)=O)CC(N(C)C)C(CNC(c2cc(C(F)F)[nH]n2)=O)C1 C1(C(=O)NC2CC(F)(CNC(c3c(C)c[nH]c3)=O)C2)COc2ccc(F)cc2C1 CC1(C)CCC1C(=O)NCCCCCNC(C1(c2ccncc2)CCC1)=O CC12CN(C(c3cccnn3)=O)C(C(=O)NC3CCC4(CCC4)C3)(C1)C2 c1(CC)cccc(C(=O)NCc2ccc(OC(C)C)cc2OCC(C)C)c1N c1(C(N2CCCCC(NC(CC(C=C)(C)O)=O)C2)=O)c(F)ccc(N)c1Br c1(NC(=O)NC2C(N3CCN(Cc4nc(C)oc4)CC3)CCC2)ccc(F)cc1Cl c1(C(=O)NCC2C(C)(C)CCN2C(=O)COc2ccsc2)ccc2c[nH]nc2c1 CN1CCN(C(=O)CC2COC(C(F)(F)F)C2)CC1CNC(c1cnsc1)=O C1(C)(CC)CN(C(=O)CCOCC2CC2)CCO1 C(=O)(C1=CCCC1(C)C)NCC(=O)NC1(C)CC(NC(c2ccc(N)cn2)=O)C1 C(=O)(C(CCC)C(C)C)NCCOC1CCN(C(c2c(C#C)cn(C)n2)=O)C1 C12(NC(C(F)=C(C)C)=O)CCC(C1)N(C(=O)CC(O)CN(C)C)C2 CCCC(C)(CCC)C(=O)NCC1CC(NC(=O)CC2CC(=O)NC(=O)C2)C1 C1(C(=O)NCc2ccc(COC)cc2)C2CN(CCC3CCC(=O)N3)CC12 c1(NC(C(N2CCCC(C(=O)NC)C2)=O)=O)cc(-c2nn[nH]n2)cc(O)c1 c1(OC)ccc(O)c(C(=O)NC(C2CCN(C(=O)C(C)C)CC2)C)c1 c1(OC)cc(C(=O)N(C)CCNC(c2nc(C(F)(F)F)cn2C)=O)ccc1F N1(C(C(=O)NCCCC)C2CC(C(C)(C)C)C2)Cc2c[nH]nc2C1 C=CCC(C)(C)CC(=O)NC1CC(O)(CNC(C2CSCCS2)=O)C1 C(c1ccc(Br)s1)=CC(=O)N(CCCN(C(C(=O)OC)=O)C)C n1(CC(=O)NC(COCC)C(=O)N(C)C(c2cc(C)on2)C)ncn(C)c1=O CCCCC(O)C(=O)NCC1(C)CCN(C(=O)C(c2ccccn2)O)C1 c1(C(=O)NCCN(C(CC(C)SC)=O)CCCN(C)C)ccc(C)nc1 c1(N2C(CNC(C(C(CC)C)OC)=O)CCC2)c(C)c(C)nc2ncnn12 c1(C(=O)NC2C(NC(c3ccc(CCC)s3)=O)CCCC2)cccc(C)c1F C(C(=O)N1CCCO1)C(N1CC(CC)C(C(=O)NC2CCC(=O)N2C)C1)=O c1(C(=O)NC2C(CC)CN(C(=O)C(C)(C)O)CC2)ccc2c(c1)CCCS2 c1(CC(=O)N(CCCNC(=O)COCC2CCOCC2)CC)ccc(C#N)nc1 c1(CN(CC2CC2)C)c(Cl)nn(C)c1Cl.Cc1ccc(C(C)(C)C(=O)O)cn1 c1(OC)cc(Br)ccc1CNC1CC(NS(=O)(=O)C(F)(F)F)C1 N1(C(c2c(OC)occ2)=O)CCOCC1c1cn(CCNS(C)(=O)=O)nn1 Cc1cc(N2CCC(NC(=O)CCCn3ccnn3)C(O)C2)nc(CO)n1 N1(C(COC)=O)CCC(CNC(=O)NC23CC(C(=O)O)C(C2)C3)CC1 c1(C(=O)NCC(c2ccccn2)NC(C(C)C2CCCO2)=O)cc(O)n(C)n1 Cc1c(-c2c[nH]nn2)cccc1Br.c1noc(-c2ccoc2Br)n1 c1(C(=O)NCC(C)NC(c2nn[nH]c2C(F)(F)F)=O)cccn(C2CCC2)c1=O c1(C(=O)NC2(C)CC(NC(C(CC)F)=O)C2)ccc(Cl)c2c1OCCO2 C1(CN(C(COCCC)=O)CCC)CCCN(C(=O)C2CC2)C1 N1(C(c2ccc(C(=O)OC)[nH]2)=O)CCCOC(CNC(C2CC2(C)C)=O)C1 N1(C(CCC=CC)=O)CCC2(CCCC2NC(=O)CN2CCC(NC)CC2)CC1 c1(C(N(C2CC2)CC2N(C(C(F)OC)=O)CCC2)=O)cccc(-c2nc[nH]n2)c1 C(=O)(C(C)(C)CC(F)(F)F)N1C(C2(NC(CC(C)C3CC3)=O)CC2)CCC1 C(c1csc(C)n1)=CC(N1CCC(N(C(C2(C)CC2(Cl)Cl)=O)CC)C1)=O N(C(=NCc1ccoc1)N1CCC(F)(CN2CCCC2)C1)Cc1n(C)ncc1 Cn1cc(CNC(=O)C(C2CCN(C(=O)CSC3CC3)C2)F)nn1 c1(N2Cc3n(cc(C)n3)CC2)nc(NCCCCO)c2ncn(C)c2n1 N1(C(Cc2c(C)con2)=O)CCC2CCCC12C(N1CC2(CCCN2C)C1)=O C1(NC(c2c(C)n(C)cc2)=O)CCN(C(=O)C=Cc2cccnc2)CCC1CO c1(CC)c(C(=O)NC(c2ccccc2)C(C)NC(=O)C(F)=C(C)C)cnn1C c1(C(N2CC3CCCS(=O)(=O)C3(C(F)(F)F)C2)C(=O)O)sc2ccc(Cl)cc2c1C N1(C(COCCOCC)=O)CC(NCc2cc(-c3c(Cl)cnn3C)no2)C(C)C1 Cc1cc(C(=O)N(C2(C(=O)NCC3CCCC(CO)C3)CC2)C)nc(O)c1 Nc1c(C(=O)NCCC(O)CNC(C2C3CC4C(C3)C24)=O)cnc2ncnn12 c1(COC(=O)NNC(c2ccnc(SC(F)F)c2)=O)ccc(F)cc1F CN1CCC(C(=O)NC2CCC2CC(=O)NCC=CC(=O)O)C1 C(=O)(CCCC(F)(F)F)N1C(CCNC(c2cncc(OC)c2C)=O)COCC1 N(C(=NCCOc1ccc(F)cc1)NC(C1(C)CCCO1)CC)CC(=C)C Cc1cccc2c1CCN(C(=O)CC1CC(NC(=O)Cn3ccnn3)C1)C2 Cc1csc(C=CC(=O)NC2COCCC2NC(=O)CN2CCCC2C(N)=O)n1 C=CC1(CC(=O)N(C2CCC2)CC)CN(C(c2ccncc2F)=O)C1 c1(C(N2CC(C(C)C(=O)N3CC(O)C3)C2)=O)cc(Cl)c2cc[nH]c2c1 CC1CCN(CC(=O)NC2CC(C(C)NC(c3cc(C(F)F)cs3)=O)C2)C1 C(=O)(C1=C(Cl)CCOC1)NCC(C)N(C(CN(CCC)C)=O)CC CC(C)(C)CC(O)CNC(=O)C(c1cccs1)NC(=O)CCc1ncccn1 C(CC(N)=O)N(C)C(=O)NCCc1ccc[nH]1 Cc1cc(C)c(CC(=O)NC(CNC(=O)C=CC2CCOC2)C2CCC2)s1 C(C1c2ccccc2CN1C(C1CCCC1O)=O)NC(CSCCC)=O CC1CCC(NC(=O)CN2CCCCC2)CN1C(=O)C(c1nccn1C)N(C)C C#CCC(CC(=O)OC)NC(=O)NCC=CCO.c1(CCN)cc(NC=O)no1 C(CN=c1nc(C2CCCC2)[nH]s1)(C1CCC1)NC(c1ccc(CC)cc1F)=O N1(C(C2C(C)C2)=O)C2CCC1C(C)C(NC(c1cc3c(o1)CCCC3)=O)C2 C#CC1(C(=O)NCCOCC(=C)C)CCN(C(C2CCC(C)O2)=O)C1 C#Cc1ccc(F)c(C(=O)NC(C#N)CC2(C(=O)OC(C)(C)C)CCCCC2)c1 Cc1c(C(=O)NCC(CC(F)(F)F)NC(C23COCC2C3)=O)cncc1N C(C(CCCCC)C(=O)N1CCC(CC#C)CC1)NC(COCC#C)=O CCC(CC)(CC)C(=O)N1CCC(CC(=O)NC(CC2CC2)CC2CC2)C1 C1(CC)CCCC1N=c1[nH]c2c(c(=NC3CCCN(C)CC3)[nH]1)COC2 c1(CC)ccc(C(N2CCC(O)(C(C)CNC(=O)C3=CCCC3)C2)=O)cc1F c1(C(N2CC3(OCC(NC(C4(OC)CC4)=O)C3)C2)=O)nccn2nc(C)cc12 N(C1COc2ccccc21)C(c1cccc(-n2c(C)cccc2=O)c1)=O C(=O)(C1=NOC(C)(C)C1)NCCC1N(C(CCCN(C(C)=O)C)=O)CCCC1C C1(C(N2C(CNC(C3(Cl)C(C)(C)C3)=O)CCC2)=O)Cc2ccccc2NC1=O CC(C)C(F)(CNC(C1(F)CCOC1)=O)C(=O)N(C)CCF c1(NC(N(C)Cc2c(F)cccc2F)=O)cc(=O)n2ccccc2n1 C=CC(CCC)CC(=O)NCCC(C)N(C(=O)C1=CCCCC1)C Cc1[nH]c2ccccc2c1CC(=O)NCC(C)CNC(=O)CCC1CC1(F)F C(C(CC1CCCC1)C(=O)N1CCOC(C(C)C)C1)NC(CC=CC=C)=O C(=O)(CC(C)(C)C(F)F)N1CC2C(NC(Cc3cc(C(C)(C)C)nnc3O)=O)(C2)C1 N1(C(c2cnc(C(C)(C)C)o2)=O)CCOCC1CCNC(=O)CCc1cc[nH]n1 C(C1CCCN1C(=O)CN(C(C)(C)C1CC1)C)=CC(=O)NC1C(C)COC1 C(C)(C(F)(F)C(F)(F)F)N1CC(C(=O)OC)C(F)(F)C1 c1(CC(=O)NC2(COC)CN(C(C3(P(C)(C)=O)CC3)=O)C2)ccc(O)c(Cl)c1 CC1CCC(c2noc(CCCCC(c3ccccc3)c3ccccc3)n2)CC1 N1(C(c2cc(C)nc(C)n2)=O)CCC2(CCC2)C(NC(c2coc(CO)c2)=O)C1 Cc1ccc(C)c(CC(N2CCN(C3COC3)CC2)=O)c1.C1C=CC1 C1(F)(CNC(c2ccn(CC(F)(F)F)n2)=O)CCN(C(C2(CO)CC2(F)F)=O)C1 Cc1c(C(N2CCC=CC2C(=O)N(C)CCN(C)C)=O)nnn1C C(CC1CC1)(C(=O)NC(C)(C)CC)N(C)C(C1CC1C(F)(F)F)=O CC12CCC(CNC(=O)NCC3CCNC(=O)O3)(CC1)CO2 C(C)(N=c1nc(N(CC(C)(C)CC(C)O)C)c2c([nH]1)CCS2)c1cn(CC)nc1 N1(Cc2ccc(CC)s2)CCC(O)(C(=O)NC(c2cncnc2)C)C1 c1(C(=O)NCC(C2CCN(C(=O)CC3CC3(C)C)CC2)C)nccc(Cl)c1O C(=O)(C1CCC(=O)c2ccccc21)N1CC(CCCNC(C(C(C)(C)O)(C)C)=O)C1 C1(CNC(C=CCC)=O)COC(C)(C)CN1C(=O)CN(C1CCS(=O)(=O)C1)C c1(C(N2C(CCNC(c3c(C)oc(CO)c3)=O)CCC2)=O)occ2c1CCC2 N1(C(C(C)OCCC(C)C)=O)CCC2(CC1)C(NC(=O)CSC(=N)N)CS2(=O)=O C1(CC#N)CN(Cc2cc(F)ccc2F)CCN1C(c1ccc(O)nc1Cl)=O CC1CN(C(C2(F)C(C)(C)C2(C)C)=O)CCC1C(N1CCC1(C)CCN(C)C)=O CN1CCN(C(=O)Cn2cc(Cl)c(C(F)(F)F)n2)CC1C1CC1 N1(C(CCNC(=O)OCC)=O)CCCCC1CNC(C1CCC1C(F)(F)F)=O N1(C(CC2CCC(NC(c3snc(C)c3N)=O)CC2)=O)CC(C)(C)C2COCC12 c1(C(C)(C)C(=O)NCCC2CC(NC(=O)CCC3CC3)C2)ccc(F)c(F)c1 c1(C(=O)N(C2CCCO2)CC2CN(C(=O)C(F)=C3CCCC3)C2)cccc(Cl)c1 N1(C(CCCC)=O)CC2(CCOCC2)CC1CNC(=O)Cc1cnsc1 C(=O)(C1Cc2ccccc21)NC1CCC(C(=O)Nc2c(OCC)cccn2)OC1 c1(C(=O)NCC(=O)N(C)CC)c(C(C)=O)cnn1C.c12ccc(o1)SC2 C1(C(=O)NCc2ccn(CC)n2)CC(N=[N+]=[N-])CN1C(c1cc(C#N)oc1C)=O C1(NC(C2ON=C(CC)C2)=O)CN(C(=O)C2=CCCCCC2)C2CCCC12 c1(C(N2C(CNC(C3CC(C)(C)C3)=O)CC3(CC3)C2)=O)ccc2c(c1)NCC2 c1(C(N2CC(C)(CNC(CCCC)=O)C(C)C2)=O)cc2n(c1)CCOC2 Cc1cc(C(=O)NCc2occc2C(N2CCOC(C)C2CO)=O)ccc1F C12(NC(CCc3n(C)cnc3)=O)CCC1CN(C(=O)CSc1n[nH]c(=N)s1)C2 n1(CC(=O)NC2(CNC(c3cc(C(=O)OC)no3)=O)CCOC2)c(C)ccc1C c1(C(C)=O)ccc(C(=O)NCCC(O)CNC(=O)CCCF)c(F)c1 c1(NC(N2CCC(C(C(=O)NC)N3CCCC3)CC2)=O)ccc(F)cc1 Cc1coc(C)c1C(=O)NCC1(C(C)NC(=O)CNC(=O)CC(F)(F)F)CC1 C#CC1(NC(=O)C(C)(C2CC2)N(C(=O)Cc2ccc(O)nc2)C)CC2CCCC12 N1(C(C(C2CCCCC2)NC(C(C=C)CC)=O)=O)CC2CC1CN2C c1(C(=O)OC)cc(SC)ccc1[N+](=O)[O-].C1(=O)C(C)(C)CN(C)CCOCCN1 N1(C(C(CCC)NC(N)=O)=O)CCN(C(=O)Cc2nncn2C)CC12CCC2 Cc1cc(C)c(C#N)c(NC2CC3CC(C2)N(C(C2(O)CC4CCC2C4)=O)C3)n1 C(CCCCCCN(C)C)NC(C(C)N(C(=O)C(c1ccccc1)O)CCC)=O c1(C(N2CCC(CC=C)(NC(=O)CSCC3CCC3)C2)=O)ccnc(F)c1N c1(CC(=O)N(C)CCNC(C2CCC(=O)N2C)=O)cc(Cl)cc(Cl)c1.C1(C)CC1 N1(Cc2ccn(CC)n2)CCN(C(c2ccccc2CC#N)=O)CC1 C1(C(=O)NCCCN(C(c2cn(CC(F)F)cn2)=O)CC)CCCCC1F c1(NC(N(c2ccccn2)C)=O)cnccc1C(=O)OCc1csnc1Br N1(C(=O)NCc2ccnc(OCC)n2)CCC(NC)C(C)C1 c1(C(=O)NC2CCC2CNC(C2CCNC2=O)=O)cccc(OCF)c1 C1(CNC(c2cnc(O)o2)=O)CC(O)CN1C(c1c[nH]c(=S)cn1)=O N1(C(c2c(C)nc(CC)o2)=O)CC(NC(c2cc(OC)n(C)n2)=O)C(C2CC2)C1 C=CCC(C(=O)NCCCC1CCN(C(=O)C(C)OCC)CC1)C(C)C c1(N(C)CC2CCCC2)nc(=NCC(F)CO)[nH]c2c1CC(C)CC2 c1(C(=O)NCC2CC(O)(CNC(C(C=C)C)=O)C2)ccnc(C)c1C Cc1nc(O)c(C(=O)N(CCCCN(C)C(C2(CCF)CC2)=O)C)nc1C c1(C(N2CC(CCNC(CCC(=C)Cl)=O)C2)=O)cc2c(s1)CCCCCC2 C(=O)(C(CNC(=O)C(C)CC1CCCC1)CC(C)C)N1C(C#C)CCCC1 N(C(=NCCc1ccc(F)cc1)NCC12CC(C1)C(C)O2)CC(C)OC N1(C(CN2CCC(C)CC2)=O)CCN(C(C2CCC3CCC2O3)=O)C(C(C)C)C1 C(=O)(CCC1CCc2ccccc21)N1CCN(C(C(C#C)(C)C)=O)CC1CCC c1(C(=O)OCC)cccc(Br)c1-n1cccn1.N12CCC(C1)C(C1CC1)C2 C1(CN(C(C=C(C)C)=O)C)CCCC(NC(=O)CCc2cnc[nH]2)C1 c1(OC)cccc(F)c1CC(=O)NCC(CNC(c1nc(C)ccc1F)=O)OC C(CN=C(NCc1cnn(C)n1)NCC1(OCC)CCC1)OCC Cc1cnc2n1CCC(C(=O)NC1(CCNC(=O)Cn3cccnc3=O)CC1)C2 C1(C#N)(C(N(C)CC2N(C(c3cccc(OC)n3)=O)CCC2)=O)CC12CCCC2 CS(=O)c1cccc(C(N2CC=CC(NC(=O)C(F)(F)c3csc(Cl)c3)C2)=O)c1 C=CCCC(C(=O)NCCC1(C)CC1(F)F)NC(=O)CC1COCCO1 c1(CNC(C2(C)CCCC2)c2nnnn2CCOCC2CC2)ccc(Cl)cn1 S(=O)(=O)(c1cccc(=NCCc2nccs2)[nH]1)N(C(C(CCC)C)C)C c1(NC(=O)Nc2c(SC)c(F)ccc2)[nH]nc2c(=O)n(C)cnc12 c1(CC(C)NC(=O)CCOCCN(C(=O)C(F)=CC2CC2)C)nccn1C C(=O)(CC1=NNC(=O)C1)N1CCCCC(NC(c2c(SCC)cncc2)=O)C1 C1(N(C(=O)Cc2csnn2)C)CN(C(C2CCC(=O)O2)=O)CC1F N1(C(=O)CC2CCC2(Cl)Cl)CCC2(CC1)CCN(C(=O)CCCCC1CC1)C2 c1(SC)ccnc(NC2CCCC2)n1.N12CCC(CC1)OCCCNC(=O)C2=O C1(CC#C)(C(N2CCC(CC(C)C)C2)=O)CCN(C(=O)CCCCOCC)C1 C1(NC(c2c(OCC)cccn2)=O)CN(C(=O)C(F)CC2CCC2)C2CCCC12 C1(CN2C(C(CC)C)CCC2)COC2(CCC2)CN1 C(CN=C(NCCOc1ccccc1Cl)NC1CCCCC1)C1(O)CCOC1 CCC(C)CC(C(=O)NCCN1CCCOC1=O)NC(=O)C(OC)OC C(=O)(C#CC1CCCCO1)N1CCN(C(C=CC=CC)=O)CC1CC N1(c2cc(C)nc(Cl)n2)CCOC2(CCC(NC(c3ccoc3)=O)CC2)C1 Cc1nc(C(=O)NC(C)C(C)(C)NC(c2cc(C#N)c[nH]2)=O)c2ccnc-2[nH]1 c1(C(N(C2CCN(C(C3(C)CCOCC3)=O)CC2)CC#C)=O)cc(SC)nn1C C1(CC(=O)NCc2cnco2)C2CCCC1N(C(=O)C(F)n1cccn1)C2 n1(CC)ccc2cc(CNCC(c3cnnn3C)(C)C)ccc12 N12CC(C)(C1)NC(=O)C1C(C1)C2=O.C(=O)(CCC1CCC1)N.CCO c1(C(C)C)cc(CNC(=O)C(C)(C2CC2)N(C(=O)CCCC2CC2C)C)no1 CC1CN(C(C2(OCC(F)F)CC2)=O)CCC1NC(c1cccc(Cl)c1)=O C1(CC=C)(C(=O)NC2CS(=O)C2)CN(C(C2CC2CC(C)(C)C)=O)C1 O(C=CC(=O)NC1CC1NC(=O)C(C)Sc1ccccc1)CC C1(COC)CN(C(c2c(Cl)cccc2Cl)=O)CCN1C(c1cc(Br)cc(Br)c1)=O C#CCC(C)C(=O)N1CCCC(C(=O)NCC(C)(C)CN)C1 C12(NC(=O)CN3C(=O)CNC3=O)CCCC1N(C(c1ccnc(F)c1F)=O)CC2 C1(C(=O)NCc2c(C)noc2)CC(NC(=O)Cn2nnc(C)n2)C12CCC2 C(=O)(CC1COc2cc(O)ccc21)NC(CC)(CNC(=O)CC1CC(F)C1)CC C1(CC)(NC(=O)CC(C)N2CCCC2=O)CCCN(C(=O)C=C(C)C(C)(C)C)C1 CC1CC(C)CN(S(=O)(=O)N2CCN(S(=O)(=O)CCCl)CC2)C1 C1(NC(CCOCCC)=O)CCOC(C2CCN(C(c3cc(C)no3)=O)CC2)C1 N1(C(c2onc(C)c2C)=O)CC(NC(=O)COCCCC(C)C)C2(CCC2)C1 c1(C(C)C)ccc(C(=O)NC(CNC(=O)Cc2ccc(O)cc2)C(C)C)cc1F Cc1oc(C#N)cc1C(N1CCCC1(C)C(=O)NC1(C2CCCC2)CC1)=O C1(CNC(c2onc(CC)c2C)=O)C(C)CCCN1C(c1cncs1)=O c1(C(N2C(C)CCC(NC(C3CC(C)(O)C3)=O)C2)=O)cc2cnc(Cl)cc2s1 C1(C)(C(NOC(C(=O)OC)CC(C)C)=O)CN(C(=O)C=CCCC(C)C)C(C)(C)C1 C1(CNC(Cc2cn(C(C)C)nn2)=O)CC(C)(C)CN1C(=O)COC(F)F CCC(C)(O)C(=O)NCC(C1CC1)NC(c1ccccc1-n1cccn1)=O C1(CC(=O)N(C)Cc2ccc(F)c(F)c2)CN(C(C2COCCO2)=O)C(C)(C)C1 C1(C(=O)NCC2(C)CN(C(=O)CC3=CCCCC3)CCO2)CCn2nncc2C1 C1(N(CCC)C(C2CC2c2cccc(O)c2)=O)CCN(C(=O)C(C)(C)C)CC1 N1(C(c2scc(C)c2C)C(=O)NCCCC)CCS(=O)(=O)C(C)(C)C1 CCC(COC)C(=O)NCC(C)(C)CN(C)C(C1(C2CCCO2)CC1)=O c1(NC(N2C(NC(C(C)c3ccsc3)=O)CCC2)=O)cc(CO)ccc1Cl c1(C(=O)NC2C(CC)CN(C(C3CC(=O)NC3(C)C)=O)C2)cc(F)c(F)c(F)c1 N1(C(c2cc(C)c(O)nc2)=O)CCC(NC(=O)C(C)CF)C12CCC2 O=S(=O)(c1ccc(Cl)s1)NCCN1CC1.c1(CCCC2CC2)ncc(Br)cc1F n1(CC)ncc(C(=O)N(CCNC(c2cc(C#N)c[nH]2)=O)CC2CC2)c1Cl C(=O)(CCCCCC(C)C)NC1(COC)CN(C(=O)C(c2cccc(C)c2)O)C1 c1(CC(=O)NCC(C)NC(c2cocc2Br)=O)ccn(C)n1 CC1CCC(NC(=O)CCC2CC2)CN1C(C1(C2CCCO2)CCC1)=O N1(CC#CC)CCCC(C2CCN(C(c3ccc(CCN(C)C)cc3)=O)CC2)C1 Cc1cc(=NC2CC(Oc3nccs3)C2)[nH]c(=NCCc2ccc(F)cc2)[nH]1 C1(C(=O)O)CC2CN(c3ncns3)CC2C1.c1(C=O)cc2cc(c1)C1(Cl)C2C1.CO C(=O)(C1=NN(CCO)C(=O)CC1)NCCC(C(C)C)NC(CC1CC(CC)C1)=O N1(C(c2csnc2Br)=O)CCCC2(CCN(C(c3ncncc3Cl)=O)C2)C1 N1(Cc2n(CCC)nnn2)CCCCCC1.c1(S)ccccc1C(=O)N CCC(C)C(O)C(C)C(=O)N(C)CC1CCCCN1C(c1nnsc1C)=O C(=O)(C1=Cc2ccccc2OC1)NC1CCN(C(CC(C)c2ccccc2)=O)C1 C(CCN(C)C)(C(=O)NCC1(O)CC1)NC(C(C)SC)=O C1(N(C)C(c2ccc(COC)c(Cl)c2)=O)CC2CCC(C1)N2C(=O)C1CC1 C1(NC(C2C(C)C2C)=O)CCN(C(=O)CC2CC(F)(F)C2(F)F)C12CCC2 N1(C(=O)CCn2cncn2)CC2CC1CCN2C(c1ccc(C(F)(F)F)s1)=O C1(NC(CC=CC)=O)(CF)CCN(C(c2cccc(CC(C)C)c2)=O)C1 C12(C(=O)NCCOC3CN(C(CC4C(C)CCC4)=O)C3)CC(C)(C1)OC2C c1(N(C)C)c(F)cc(-c2nc(C3CCC3)ncc2C(=O)C2CC2)cc1F C1(C(=O)N)(CO)CCCCC1.C12(F)CC(C1)CN(C)CC(=O)NCCOC2 C12(NC(Cc3c(C)noc3Cl)=O)CC(CNC(=O)C(=O)N(C)C)(C1)OC2C c1(NC)snc(C)c1C(=O)NCCCOC1CCN(C(C2CC3CCC2O3)=O)CC1 C#CCC(C)(C)C(=O)N1CC(OCCNC(=O)C(C)(C)C2CCCO2)C1 C1(N(C(=O)C=Cc2cccs2)C)CCCN(C(=O)COc2cccc(F)n2)C1 Nc1cc(F)c(Cl)cc1C(N1CC2CC(NC(c3nc(Cl)cs3)=O)C1C2)=O C1(=O)C(C)(C)CCO1.C12(N(CC(C)=O)C3CC3)CCC(CC1)C2 C1(C(=O)NCC2(NC(CC(C)C(F)F)=O)CCCC2)CC2(C1)NC(=O)NC2=O Cc1nc(C)c(CNCc2cnc(-c3cccc(C(F)(F)F)c3)nc2)nc1C C(=O)(C1=CS(=O)(=O)CCC1)NCC(C)N1C(=O)c2cn(nn2)CC1.CCSC CC1(CNCC2CCCCC2c2nc(S)n[nH]2)CCCC(F)(F)C1 N1(C(CNS(CC)(=O)=O)=O)CC2(C1)C(NC(=O)C(F)OC)CCS2(=O)=O N1(C(c2c[nH]cc2C(F)(F)F)=O)CCN(C(C2CCS2(=O)=O)=O)C2(CCC2)C1 CC1CCC(NC(c2cc(Cl)nnc2Cl)=O)CN1C(c1cnsn1)=O C1(N(C(CC(C)OC)=O)C)CCCN(C(=O)C(F)(F)CC2CC2)CC1 C1(NC(CCCC#C)=O)CC2(C1)CN(C(c1cnc(C(C)(C)C)nc1)=O)C2 C(C(C)(O)C(=O)NC1CCCC1CNC(c1cn(-c2ncccn2)cn1)=O)OC NS(=O)(=O)c1ccc(C(N2CCC2CNC(c2cc(Cl)c(F)cc2O)=O)=O)cn1 O=C1CCC(C(=O)NCC(C2CC2)NC(C2(c3cc[nH]n3)CC2)=O)O1 C(=O)(C(C(C)(C)C)NC(c1n[nH]cc1Cl)=O)NCC(C)Cn1cccn1 C1(CNC2(CNC(CC(C)c3ccsc3)=O)CC3(CC3)C2)CC2CCCCCC12 c1(CC)cc(F)ccc1C(=O)NC1CCC(C)(CNC(=O)C=CC=C(Cl)Cl)C1 c1(OC(c2nnnn2C2CCOCC2)(CSC(C)C)C)cccc(F)c1 C1(C(N2CCC(O)(C(C)NC(c3c(CC)nc[nH]3)=O)C2)=O)CCC(F)(F)CC1 Cc1cc(C)n2cc(C(=O)NC3CC4CC3N(C(=O)CSCC(F)F)C4)nc2n1 c1(OC)ccc(C(N2CCC(NC(c3ccc(C(C)(C)C)o3)=O)C2)=O)nc1OC Cc1nc2ccc(O)cc2cc1C(=O)Nc1cccc(NC(C2(C)COC2)=O)c1 CCC(C)CC(C(=O)NC1CNC(=O)C1)NC(=O)C#CC(C)(C)O N(C(=NCCCc1ccc(Cl)cc1Cl)NC(C)C1CC1)OCCS(C(C)C)(=O)=O CC#CCCCC(=O)N1CCCC1CCC(N1CCC(C)=C(C)C1)=O c1(C(N2CC(CNC(c3cnn(C)n3)=O)OCC2)=O)ccc2cc[nH]c2c1F c1(N(C2(CC(=O)NCCNC(=O)CC3CCC(=O)N3)CC2)C)ccc(Cl)nn1 N1(C(c2cn(C)nn2)=O)CCC2C(NC(=O)CCC(C)(F)F)C2C1 Cc1cccc(C(O)C(=O)NC2(CNC(=O)COC(C)(C)C(F)(F)F)CCOC2)c1 c1(C(=O)NCC(C)NC(CCn2c(=O)cc(C)nc2)=O)c(F)ccc2ccoc12 Nc1c(C(=O)NCCC2CCN(C(C3(F)CC3)=O)C2)cccc1C(F)(F)F C1(NC(C(c2cccnc2)C)=O)CC2CC(NC(c3coc(C(F)F)c3)=O)CC12 C1(NC(C(C)(C)NC(=O)NCC)=O)CCCN(C(CC(C2CCC2)CC=C)=O)C1 CCCC(C)CC(=O)NC(CNC(=O)Cc1csc(C2CCOCC2)n1)CC N1(CC2OCC(C(=O)OCC)C2)C(C)C(C(N2CCC(C(C)O)C2)=O)CC1C c1(C(=O)NC2(C)CN(C(C3CC3(C)C(F)F)=O)C2)cc2ccccc2s1 C1(NC(c2cc(C)cc(C)c2)=O)CCN(C(=O)Cc2sc(S)nc2C)CC1(C)C C(CC(F)(F)CO)NC(C1CCCN1C(C1COCCN1)=O)=O c1(C(=O)NC(C(CO)NC(CCOC(C)C)=O)C)cccc(C2CC2)n1 C(C(C(=O)NCCn1cc(C(=O)NCc2cc(Cl)no2)nn1)OC)OC c1(C(=O)NC(c2c(OC)cc(OC)c(OC)c2)C)ccc2c(n1)OCC(=O)N2 C(CNC(=O)C=C1CCN(C)C1)(CC(C)C)NC(C(CC)n1cccn1)=O c1(C(=O)NC2CN(C(C3(OC)CCCCC3)=O)CC2C)cc(N)cc(C)c1F C1(NC(c2ccc(CC)[nH]2)=O)CCCC(NC(=O)CC(=O)OC)CC1 C1(O)(C(C)NC(c2csc(CC(F)F)n2)=O)CN(C(=O)C(F)=C(C)C2CC2)C1 CN1N=CC(CC(=O)NCC2CC(F)(CNC(C3CCC(C)CC3)=O)C2)C1=O N1(CCNc2c(S(=O)(=O)NC3CC(C)(C)SC3)cccn2)CCc2ccncc2C1 Cc1ncc(Br)cc1NC(C1CCCC1)=O.N12CCC(O)(C1)C2=O.C1C(=O)N1 N1(C(CC2(C=C)CCC2)=O)CCC2(CC1)CN(C(C1C=CC=CC=C1)=O)C2 Cc1cnc(C=CC(=O)NCC2CC(C)N(C(c3cccc(C(F)F)n3)=O)C2)[nH]1 c1(C(=O)NC2CN(C(c3cc(OC)n(C)n3)=O)C2)cc2c(C)nn(C)c2s1 c1(C(N(CCCn2cc(CC3CCCCC3)nn2)C)=O)c(F)cc(Cl)cc1F Cc1ncc(NC(C2(C)C=CCN2C(=O)C(O)CN2CCCC2)=O)c(C)n1 C=CC(C)C(=O)N1CCCC1CCCNC(=O)CC1CCOC1=O c1(NC(C)=O)ccc(NC(C2CN(C(=O)Nc3ccccc3Cl)CC2C)=O)nc1 C1(C(C)C)CCC(N2CCCC2C2CCOC2)O1 C1(NC(CCSCC)=O)CN(C(c2c[nH]ccc2=O)=O)C2CCCC12 C1(N2C(CNC(=O)CNC(C3CCCCC3)=O)CC2)CC2(CCC2)C1.c12cn-1nn2 N1(C(COC)=O)CCC(CNC(C2CC2C)=O)(OC)C1 C1(NC(C2CC2C(=O)OC)=O)CC(F)(CNC(=O)CN2CCNC2=O)C1 C1(C(=O)OC)N(S(=O)(=O)Cc2ccc(C(=O)O)cc2)CCOC12CCCC2 CN1C(=O)COCC1CNC(c1coc(CNC(c2cscc2Cl)=O)c1)=O N1(C(CCCCCC)=O)CCC(C)C(NC(C2CC3CCC2CC3)=O)C1C C1(C(=O)NC2CC(CC)(CC)C2)C2CCN(C(=O)C=CCO)CC12 C1(CC)CC(C)CN(C(=O)C(CC2CC2)NC(C2CCC(OC)CC2)=O)C1 Cn1cc(C(=O)NCC2(F)CC(CNC(=O)CCC3CCCCC3)C2)cc1Br c1(CNC(c2cnn(C(F)F)c2)CC)ccc(SC)cc1 c1(OC)cncc(C(=O)NC2C3CC2CN(C(C2(C)COC(=O)C2)=O)C3)c1C Cc1nc2cc(C(=O)NCC3(O)CN(C(=O)C4=NOCC4)C3)cc(Br)c2[nH]1 C#CC(CCC)NC(=O)CC1(NC(C2C(OC)CC2O)=O)CC1 c1(C(C(N2CCN(C(COCC#C)=O)CC2CCC)=O)C)nc2ccccc2s1 c1(CC2(COC(F)F)CC2)cc(F)cc(Br)c1 N1(Cc2cccc(OC)c2)CCC(NC(C2CCCC(CC(=O)O)C2)=O)CC1C CC1(C)C(CC(=O)NOCCCOC(F)F)CCN1C(C1CCC2CC12)=O N1(C(C2(CCC=C)CC2)=O)CCC(O)(CNC(=O)COCC(C)(C)C)C1 c1(C(=O)NC(CCOC)CNC(C2CC(O)C2)=O)cccc(-c2ccncc2)c1 C1(NC(c2c(CC)[nH]cc2)=O)C2CN(C(=O)C(C(C)C)NC(C)C)CC12 c1(CC(C)C)cccc(C(=O)NC(C2(O)CN(C(C3CCCS3)=O)C2)C)c1 C1(n2cc(CC(C)(C)OC)nn2)CCC(CNC(=O)CC2CCCCC2O)CC1 C#CCC(C)(C(=O)NCc1ccncc1)NC(=O)C(CC)OC C(=O)(CCC(C)S(C)(=O)=O)N1C(C)CC(CNC(C(=Cc2cccs2)C)=O)C1 c1(C(N2C(CNC(c3ncn(CC)c3)=O)CC(F)C2)=O)ccc(C(C)C)nc1C C1(NC(c2c(C)cco2)=O)CC2CC(NC(=O)C(c3cccnc3)O)CC12 CCCC(C(=O)N1CC(COC)CC1CNC(=O)Cc1cn(C)nc1C)OCC N1(C(CC(C=C)CC)=O)CCC(Nc2ncc(C(F)F)cn2)C(F)(F)CC1 c1(CC)nn(C)cc1C(N1CC(CNC(=O)CC(C)(C)O)CC1C)=O C1(C2(NC(=O)Cc3ccns3)CC2)CCCCN1C(C1CCCS1)=O C#CCCCC(C(=O)NCC1CC1c1ccco1)N1CCOCC1(C)C C1(C(=O)NCC2(S(C)=O)CC2)CCN(C(=O)CN2CCSCC2)CCO1 C1(C(=O)NC2(CF)CCN(C(CCC=CC(C)C)=O)C2)CCC(C2CC2)C1 C1(OC)COCCC1C(=O)NC(c1cccc(F)c1)CF C1(c2cn(NC(c3cccc(OC)c3)=O)nn2)CN(C(c2cnnn2C)=O)CCO1 C1(CNC(C(C)C2CC2)=O)CN(C(c2snnc2C(F)F)=O)CCO1 N1(C(C(=O)NCC(=C)C)c2ccns2)CCC(C(=O)OC(C)(C)C)C1 N1(C(CCSCC)=O)CC(NC(=O)Cc2cc(C)nc(C)c2)CC(C(F)(F)F)C1 N1(C(=O)CCC2CC2)CCOCC1Cc1cn(CC(O)C2CC2)nn1 CC1(C)COC1NC(=O)NCc1ccon1 N1(C(C2=NOC(C)C2)=O)CC(NC(=O)CCN2CCC2)C2(CCS(=O)(=O)CC2)C1 c1(OC)cnc(C(=O)NCCCN(C(=O)CCN2CCCC2=O)C)nc1 c1(CC)nn(C)cc1C(=O)NCCCC(C)(C)NC(=O)COc1ccon1 C1(N(C(=O)CCNC(c2ccc(F)cc2)C2CCC2)CC)CCCOCC1 C(C(CC(F)(F)F)NC(=O)C=CSc1ccccc1)NC(C(C)C(F)F)=O Cc1cccnc1CC(N1CCC(N(C(=O)C(C)Sc2ccc(Cl)cc2)C)C1)=O C(=O)(C1=NNC(=O)C1)NC1CC(O)(CNC(c2cnc(CCCC)s2)=O)C1 C1(C)(NC(c2ccc(OC)s2)=O)CCC(NC(=O)CC2(C(F)(F)F)CC2)CC1 C12(NC(C(COC(C)(C)C)N(C)C)=O)CC3CCC(C1C2)N3C(=O)CC(C)F c1(C(N2CCOCC(CNC(CC(=C)C)=O)C2)=O)cc2n(n1)CCCNC2=O CCC(F)(F)CC(=O)NCc1nc(C)c(C(=O)N(C)CCc2ncon2)o1 C1(C(=O)NCC2C3N(C(CCC(=O)OC)=O)C(CC3)C2)CCc2nccn2C1 N1(C(C(CC)C#N)=O)CCC2(CC1)CCN(C(C1OCC3CCCCC13)=O)C2 N1(C(C2CC(NC(=O)CC3CC(C4CC4)C3)C2)=O)CCN2CC(O)CC2C1 C(=O)(N=c1ccn(-c2nccc(C)n2)[nH]1)C1N(C(c2c(OC)cc(C)cc2)=O)CC1 C1(C(N2CC(C)(NC(c3ccc(CC)c(CC)c3)=O)C2)=O)CC2CCCCN2C1 C1(C(N2C(C(C)NC(=O)CC(C)(C)C)CCC2)=O)COc2ccc(F)cc2C1 N1(C(CCOC(C)C)=O)CCN(C(C2CC2CC(C)C)=O)C(C(C)C)C1 CCC(C)(O)C(=O)NC1CC(CCNC(c2cc(C(C)=O)cs2)=O)C1 CC(C)C(C#N)C(=O)N1CC(=O)NCC1C(N1CC2(CC(F)C2)C1)=O C1(OCC)(CNC(=O)C=CC2CCC2)CN(C(=O)C(C)C2CCCO2)C1 N1(C(C(CC)(C)C#N)=O)CC(C(=O)Nc2cc(C)ccc2OC)CCC1(C)C CCC(C(=O)OC)C(=O)N1CCCCCC1CNC(c1cc(OC)no1)=O C1(C(N2CCC(N(C(C(CCC)O)=O)CCC)C2)=O)CC2(CCCO2)C1 Cc1cc(C)n2ccc(C(=O)NCCNC3(c4ccon4)CC3)c2n1 N1(C(C2(CC)C=CCC2)=O)CC2(CC(NC(=O)C(=Cc3cccnc3)F)CO2)C1 [N-]=[N+]=Nc1ccccc1CCC(N1CC2CCC(NC(c3cn[nH]c3)=O)(C2)C1)=O N1(C(Cn2ncn(C)c2=O)=O)CC2CN(C(=O)Cc3ccco3)CC2(C)C1 C1(C(=O)NC2CCN(C(=O)NCC)CC2)CCC(C)CN1C(C)=O.N12CC(C1)C2=O N1(C(CN(C)C(C2CC(C)(F)C2)=O)=O)CCN(C(=O)CC2(O)CCCCC2)CC1 C1(C(N(C)CCc2nccs2)=O)CNC(=O)CN1C(=O)C=Cc1cccnc1 c1(CC)nn(C)c(Cl)c1C(=O)NCCC(CNC(=O)C(C1CC1)OC)OC N#CC1(C(=O)NCCCNC(=O)CCc2ccccc2F)CCCCC1 C1(C(N2CC(F)C(F)C2)=O)CC(F)CN(C(c2cccc[n+]2[O-])=O)C1 c1(C(=O)NCC(C(=O)OC)CC2CCOC2)cccc2nn[nH]c12 C1(NC(=O)CN2C(=O)CCC2=O)CC2(C1)CC(NC(C1CC3C=CC1CC3)=O)C2 c1(CC(=O)NCC(C(=O)OC)Cc2ccccc2)ccc(OC)c(F)c1 c1(CC)cccc(C(=O)N(C2CN(C(c3cc(CC(C)C)c[nH]3)=O)CC2O)C)n1 N1(C(c2ncc(OC)nc2)=O)CCN(C(c2ccc(F)c(O)c2F)=O)C2(CC2)C1 C(C(=O)N1CCC(C(N2CCC(F)C(F)C2)=O)O1)c1c(C#C)cccc1 N1(C(c2cc(C(=O)OC)oc2C)=O)CCC(NC(=O)CC(O)C(C)C)C(O)C1 N1(C(C=C(COC)C)=O)CC(C)(C)C1C1CCN(C(=O)CCc2cnn[nH]2)CC1 C1(NC(CC2CC(OCC)C2)=O)CC(C)N(C(c2n[nH]c(CC)c2C)=O)C1 c1(C(N2CC(N(C)C(c3sncc3Br)=O)C2)=O)coc(C(N)=O)c1 c1(C(=O)NC2CCCN(C(C(C)SCC)=O)C2C)c(Cl)ccc2c[nH]nc12 c1(OC)ccc(SCC(=O)NC2COCCC2NC(=O)C(C)(C)CF)cc1 C1(CNC(CSCCCC)=O)CN(C(c2nc(Cl)cs2)=O)C2CCN1C2 N1(C(CCn2ccc(C)n2)=O)CCC(C)(C)CC1C(=O)N(CC(F)Cl)C C1(CCCNC(CCC=C)=O)CCCCN1C(=O)C=CCOC C1(NC(N2CC=CC2C(=O)NC2C=CCCC2)=O)CC2C=CC1CC2 c1(CC(C)N(C(=O)CCCCC(=O)O)C)cc2c(Cl)cccc2s1 c1(C(=O)NCCCC(C)NC(c2cnn(C)n2)=O)cn(C)c(=O)cn1 C1(C)(CC)CCC(C(=O)NC2CC3(C2)CC3NC(=O)CN2CC(F)(F)C2)O1 c1(C(CC=C)CC)cc(=NC(=O)C(C)N2CCCCCC2)[nH][nH]1 C1(C(N2C(CNC(c3c(CC)nc(C)[nH]3)=O)C=CC2)=O)CC(S(N)(=O)=O)C1 C(c1cncs1)=CC(=O)NC(C(=O)N(CCCN(C)C)CCC)C1(C)CC1 C1(NC(C2C3CN(C(C(C)(C)CF)=O)C2C3)=O)(CO)CC2CCC1C2 O=C(CC(C(F)F)c1ccc(F)cc1)NC1(CF)CCN(C(c2cc[nH]n2)=O)C1 S(=O)(=O)(c1ccc(C(N2CC(N(C(=O)CCCF)C)C2)=O)cc1)NCCOCC c1(C(=O)NC2CC(CNC(C(CC#C)O)=O)C2)ccc2ncc(Br)cc2c1 c1(C(N2CCC(NC(CS(CCC)(=O)=O)=O)C2)=O)csc2ncnc(O)c12 C1(C(CC)NC(=O)C=CCNC(=O)CSC(F)F)CCOC1 C1(C(N2CC(CCC)C2)=O)CCCCC1(C)NC(c1cc(Cl)n(C)n1)=O Cc1cc(NC(=O)C(C2CCN(C(c3cccn3C)=O)C2)F)cc(CO)c1 C12(CNC(C3CSCCN3Cc3cccc(SC(F)(F)F)c3)=O)CCCN1CCC2 c1(C(C(N2CCC(CCO)CC2)=O)NC(C2CC(OCCO)C2)=O)cccnc1O CCC(C)(C)C(O)C(=O)N(CCC(=O)N1CC(C2CCCCC2)C1)OC C1(C(=O)NCC2CC(O)CN2C(C2CCC2)=O)CC2CC(F)(F)CC(C1)C2(F)F C1(NC(c2cn(CC)nc2)=O)CC1C1CCCN(C(c2cocc2C)=O)C1 CC1CN(C(c2ccccc2NS(C)(=O)=O)=O)CCCN1C(=O)C(F)=C1CCC1 N1(C(CC=C(C)C)=O)CCC2CCN(C(c3ccc(Cl)c(F)c3O)=O)CC2C1 CC1CN(C(C23CC(CF)(CO2)C3)=O)CCN1C(=O)Cc1nncn1C C1(CNC(c2c(C#C)c[nH]n2)=O)CCN(C(=O)C(COC)CC(C)C)CCC1(F)F C1(CNC(CSC)=O)CCC(NC(c2cn(-c3cnn(C)c3)cn2)=O)C1 CCCC(CC1CCCC1)C(=O)NC1CCN(C(C2(COC)CCC2)=O)CC1F C1(CNC(C2CCN(C(=O)Cc3csc(C4CCCCC4)n3)C2)=O)CCCCC1 N1(C(CN(C(COC)=O)C)=O)CC(CC(=O)NCc2cnccn2)CC1C C(=O)(CCN(OC)C(=O)C1(C#N)CC12CCC2)NC(c1ccc(CC)cc1)C N12CC3CC1CN3C(=O)c1cc2ncn1.C1(COC)CCC2(CCC2)C1 N1(C(COC(C)C)=O)CC(NC(=O)CN2CCCCCC2)C(c2ccccc2)C1 C1(NC(CC=CC(C)(C)C)=O)CCCCC1CNC(c1cccnc1N)=O C(C(CC1CC1)C(=O)NCC=CC1CC1)NC(c1cc(C(C)C)no1)=O c1(CC)ncc(C(=O)NCC(C2CC2)NC(=O)CCC#N)s1 c1(C(=O)OCCc2c(C)n(C)nc2)cc(F)c(Cl)c(F)c1 C(C(C)(C)C(=O)NCC(N1CCN(C(=O)CSCCC#N)CC1)C)NC(C)=O C1(CNC(=O)CC2CCSCC2)CCN(C(=O)CCCF)CC1C1CC1 CCCCCCC(F)C(=O)NC1CC(CNC(C2CC2CF)=O)C1 C(C)(CCC(F)(F)F)CNC(=O)C(CC)OC(C(C=C=C)C)=O C(=O)(C1c2ccccc2CN1S(=O)(=O)C1=CCCC1)NCCSC c1(C(=O)NCCN(C(CCOCCOC)=O)CC2CC2)c[nH]nc1C(C)(C)C n1(C(NSc2c3nnn(C)c3ncn2)=O)c(=O)oc2ccccc12 N1(C(c2c(C)c(F)cnc2)=O)CC(C2CN(C(c3c(F)ccc(F)c3Cl)=O)C2)C1 C(CCCNC(=O)C=CCC1(N(C)C)CCC1)N(C)C(C1CC1C1CCCO1)=O C#CC1(NC(=O)CC2CCN(C(=O)CC(=O)OCC)C2(C)C)CC2CCCC12 C=CCCC(CC(C)C)C(=O)N1CCC(CO)(NC(c2cc(CO)on2)=O)CC1 c1(CC(C)C)nc(C(=O)N(C2CN(C(=O)Cc3nncs3)C2)C)cs1 C(=O)(C(C)(C)C(=O)NC1CCC1CNC(=O)CCCc1ccc(C)c(C)c1)NC N(C(=NCCN1CCCS1(=O)=O)NC1CCCCC1C)CCOCC=C N1(C(C2CN(S(CC)(=O)=O)C2)=O)CC2(CC2)CC1CNC(=O)COCCF C1(NC(C(CC)=CC)=O)CCC2(CC1)CN(C(=O)CN1CCC(C)(O)C1)CCO2 C(=O)(C(F)(F)C(F)F)NCc1occ(C(=O)NCC2C(CC)CCCC2)n1 C(=O)(CC(C)(C(F)F)N(C)C)N1CCC(C)C(NC(=O)C=CC(F)(F)F)C1 N1(C(C(CCC)C(C)C)=O)CCn2nc(CNCc3nn(C)cc3SC)cc2C1 C1(C)(C(N(CC(C)NC(=O)CCCSc2ccccc2)C)=O)CC(=O)N(C)C1 c1(-n2c(C(n3nccn3)C)nc(Cc3cccs3)n2)ccc(F)c(Br)c1 N1(C(CC2C(C)C(=O)CC2)=O)CC(CO)C2(C1)CN(C(C13CC(C1)C(C)O3)=O)C2 c1(C(=O)NC2(C3CCN(C(=O)CCCCC4CC4)C3)CC2)n[nH]c2ccccc12 Cn1ccc(C(N2CC(NC(c3sccc3Cc3ccccc3)=O)C2)=O)c1 N1(C(C2(NC(c3c(C)noc3)=O)CCCC2C)=O)C2CCC1CN(C)C2 N1(C(C(C)SCCCC)=O)CC2CCN(C(C3(Cl)CC3)=O)CC2C1 c1(OC)ccc(F)c(C(=O)NC2CCCN(C(=O)C(C)S(C)(=O)=O)C2)c1 Cc1nc2c([nH]1)C(C(=O)NC1CN(C(=O)C=CC(C)C)CC1C)CCC2 c1(C(N2CC(C(=O)NCc3ccc(Br)cn3)OCC2)=O)cc(F)cc(F)c1F c1(C(=O)NCC2(OC)CCN(C(=O)C(C)CC3CCC3)C2)ccc(C)c(Cl)c1F N1(C(CC=CCC)=O)CCCC(C)(NC(C2CCN2C2CCCC2)=O)C1 C(CSCC)(C(=O)NCCCC1CCCC1)NC(=O)OC.c12cc[nH]c1NC2=O c1(CC)ncc(C(=O)NC2(C(=O)NC(C)Cc3ccco3)CC(CO)C2)o1 N1(C(C2(N(C)C)CCC2)=O)CCCC(F)CC1.C12CCC(C1)C(C)(C)C(=O)N2 C1(C(=O)NCCC2(CNC(=O)CN3CCCCC3=O)CC2)CCC=CCCC1 C(=O)(C(C)(CC)C(=O)N1CCC(O)(CCNC(C2(CC)CCC2)=O)C1)OCC C1(CC)Oc2ccc(C(N3CCCN(C(=O)C=NOC)CCC3)=O)cc2NC1=O CC(C)(C(=O)NC1(CCNC(=O)CC(=O)N2CCC2)CC1)c1cncnc1 C1(N(C(=O)CCNC(N)=O)CCCC)CCCN(C(=O)Cc2c[nH]ccc2=O)C1 C(=O)(CS(=O)(=O)CCOC)NC(COC)CNC(c1sc(C)cc1OC)=O c1(C(C(=O)N(CCC(=O)N(C2CC2)CC)C)(F)F)ccc(F)cc1 C1(C(=O)NCC(CC(C)C)NC(C2CN3CCCC2C3)=O)CCC(C)(C)OC1 N1(C(CCNS(CC)(=O)=O)=O)CCCCC(NC(=O)CCC(C)(C)OC)C1 C1(NC(CCC(=C)Cl)=O)CC12CCC(NC(c1cc(CCC)oc1C)=O)CC2 C1(CC)CN(C(=O)CCc2ccon2)CCN1C(=O)C(N1CCN(C)CC1)C C(=O)(C(CO)C(C)(C)C)NCC1OCCCN(C(c2cc(C)sc2C)=O)C1 C1(C(C(=O)NC)F)CCN(C(N2CCC(CSC3CC3)C2)=O)C1 C1(CNC(c2scc(C)c2)=O)CC2(CC(NC(C3COCCC3C)=O)C2)C1 CCCCCCCNC(=O)CC1CCCN(C(C2(C(C)(F)F)CC2)=O)C1 C1(C(=O)NCC(CC)NC(=O)CSc2n[nH]c(=N)s2)CCC(C(N)=O)C1 C(=O)(C1=CCCC1P(C)(C)=O)NC12CC(NC(c3oc(CC)c(C)c3)=O)(C1)C2 C(C)(C)(CC(C)(C)C)NC(CCC(C)NC(c1ccc(O)cc1F)=O)=O c1(C(CC)C(=O)NC2CC(N(C(=O)Cc3cn[nH]c3)C)C2)c(C)noc1C C(=O)(C(C(F)(F)F)C(F)(F)F)N1C(COC)(CNC(=O)C=CCN(C)C)CCC1 c1(C(=O)NC2CCN(C(CCC(C)(C)C#N)=O)C2)cc(O)nc2[nH]c(=N)ccc12 Cc1n[nH]c(C)c1C(N1CCCC(CNC(=O)C=Cc2cc(C(N)=O)co2)C1)=O N1(C(c2cc(C)c(C)s2)=O)CCC=C(C(=O)N2CCN(CC(C)C)CC2)C1 N1(C(C2CCCC(OC)C2)=O)CCCC2(CCCN2C(C2(C)CC(F)(F)C2)=O)C1 C12(CC(=O)NC3CC3NC(=O)CSc3nnc(S)s3)CCC(CC1)OC2 c1(C(=O)NC2CC(C)(C)N(C(C3CC(F)C3)=O)C2)cccc2ncnn12 c1(C(=O)NCCN(C(C2CC(C)C2(C)C)=O)CC)cccc(CO)n1 C(CN=c1cc(C)nc(C(C)(C)C)[nH]1)OCCNC(c1cc(C)c(Cl)cc1C)=O CCC(C)CC(C)C(=O)N1CCC(N(C(=O)CC2(O)CCC2)C)CC1 N1(C(CCCOCC=C)=O)CC(C(=O)N(CC(C)NC(C)=O)C)C(F)(F)C1 CCC1=C(C(=O)N2CCC(NC(=O)Cc3nonc3C)C23CCC3)CCCO1 c1(C(=O)NCC2(C)CC(NC(CCc3cn(C)nc3)=O)C2)cc2scc(Cl)c2[nH]1 CC12CCC(=O)N1C(C(=O)NCC(CNC(C1CCC1)=O)C(F)(F)F)CS2 CC(C)(C)C(C#N)C(=O)NC1(C(N2CCC(F)C(F)C2)=O)CCC1 N1(C(CCn2cc(C(CC)(C)O)nn2)=O)CCCCC1C.N1(C(=O)C)CCCC1 N1(CCC(N2CC(O)(CNC(Cc3scc(C)n3)=O)C2)=O)CCN(C(C)C)CC1 CC1(C(F)F)CN(C(=O)Cc2sccc2Cl)CC1C(=O)O Cc1cn(C)cc1C(=O)NC(C1CCCCN1C(c1cnc(S)n1C)=O)C CON=CC(=O)N(C1CCN(C(C2CC2C(=O)NCCO)=O)C1)CCO C1(C(=O)NCC(C)CN(C)C(c2cc(Br)no2)=O)CCC(=O)N1 C(C(=O)N=c1ccn(C(C)(C)C)[nH]1)(C1CCC1)NC(CCCCCC#C)=O C(=O)(N1CCS(=O)(=O)CCO1)C1C=CC(C(=O)NC(=O)OC(C)(C)C)C1 C1(n2cc(CCCC=C)nn2)CON(C(=O)c2cc(C)nc(O)c2)C1 Cc1cc(OC2C(CNC(CN(C(COC(C)C)=O)C)=O)COC2)on1 Cc1cc(C(=O)NC=CC2CCN2C(=O)CCCC(=O)OC(C)(C)C)nnc1C C(C1C(C(=O)NCCC(C)NC(c2ccc(C(N)=O)[nH]2)=O)C1(C)C)=C(C)C CCC(=O)CCC(=O)N1CC2(CC(=O)NCC(CO)N(C)C)CC1CO2 c1(OCC)ccc2ccccc2c1NCC1CCCN1c1ccccc1 CCCC(CNC(c1ccncn1)=O)C(=O)NCCOCCOC [N-]=[N+]=NCCCC(=O)N1CCOCCC1CC(=O)NCCOC(=N)O C(=O)(C1=CC2(CCOCC2)C1)N1C(CC(C)(C)C)CN(C(=O)COCCF)CC1 C(N=c1[nH]c(=NCCSc2ccccc2)c2ccccc2[nH]1)C1(COC)CCOC1 c1(C2C(NC(=O)NC(c3ccc(F)cn3)C)C2)ccccc1F C(=O)(C#CC1CCOC1)NC(CN(C)C)C(=O)NC1COC(C)(C)C1 c1(C(=O)NCC2CCC(NC(c3cnc(CC)s3)=O)CC2)occ2c1CCOC2 c1(NC(=O)NC2CCOC(C(F)(F)F)C2)ccc(F)cc1OC(F)F C1(C(N2C(C3CCN(C(CSCC)=O)CC3)C(C)(C)C2)=O)C2CCC3C(C2)CC13 C1(C(=O)NCCNC(C(C)N(CCCO)CCO)=O)CCCC2(CC2)C1 c1(OCC)ncccc1NCCNC(C1CCNCC1)=O N1(C(c2cccc(OC)n2)=O)CCCC(CCNC(C2CC2(C)C(F)F)=O)CC1 C1(C(N(CCOCCN(C)C(C2C=CCC(=O)N2)=O)C)=O)CC2(CCO1)CC2 C1(C(=O)NCCCCNC(=O)CCc2cnccn2)Cc2cccnc2C1 C(=O)(C1=NOC(C)C1)N1CC(CC(=O)N(C2(CC(C)C)CC(=O)C2)C2CC2)C1 c1(CC)c(OC)nsc1NC(C1CCCC1NC(=O)NC(C)(C)C)C CCCC(C)(O)C(=O)N1CC(C)C(C)(C(N2CC3CCCC2C3)=O)C1 C1(NC(c2[nH]c(C)c([N+](=O)[O-])c2)=O)CCC12CCN(C(=O)C(F)C(C)(C)O)CC2 c1(C(=O)NCC(C)NC(C(C(COC)C)C)=O)cc2cccnn2c1 C(c1c(Cl)cccc1Cl)=CC(N1CCC(O)(CNC(C2(C)CCOC2)=O)CC1)=O C(=O)(CC(CNC(=O)C(C)(C)C1CCOC1)OC)NC(COC)C(C)C C1(C(=O)NCC2(SC)CCC2)CC(F)CCN1C(=O)CNc1nccs1 c1(C(N2CCC3(NC(c4ccncc4F)=O)C(C2)C3)=O)cc2ccccc2cn1 N1(C(C2(C)CC=CC2)=O)C2CCC1CC(C(=O)NCCCC1CC1)C2 c1(C(=O)NCC2N(C(CCNC(=O)CO)=O)CC=C2)ncc2c(F)cccn12 N1(C(=O)OC(C)(C)C)CC2CC(C(N3Cc4c[nH]c(=N)nc43)=O)CC12 Cc1oc(Br)cc1C(=O)NC(C1CCCCC1)CNC(=O)C(C)NC(N)=O c1(C(N2CCC(NC(c3cnsc3)=O)C2)=O)ccc2nc(O)sc2c1 Cc1cccc(C)c1CC(=O)NCCCC(C)NC(C1CCCCNC1=O)=O CC(C)(CO)C(CO)NC(C1(NC(=O)CCCn2ccnn2)CC(O)C1)=O Cc1nc(C)c(CC(=O)NC2CCC(CN(C)C(c3occc3C)=O)CC2)s1 C12(NC(C3(NC(C)C)CC3)=O)CCN(C(c3cc(Br)n[nH]3)=O)CC1C2 C1(NC(c2c(C)nn[nH]2)=O)CCC(C)(CNC(=O)CC2CC=CC2)C1 c1(NC(N2CCCC(C(=O)Nc3c(C)nsc3)CC2)=O)cnc2ccc(F)cn12 c1(C(C(N2CCSCC2NCCC2CCCO2)=O)OC)ccc(C)c(C)c1 CC1=NN(C)C(=O)C1CC(N1CC(O)(CCNC(=O)CCc2cc(Cl)no2)C1)=O C1(NC(C(CC)OCC)=O)CN(C(=O)CCc2ccnn2C)CCC1F c1(C(c2ccc(N3CCN(S(=O)(=O)CCBr)CC3)nc2)=O)cc(Br)c2cn[nH]c2c1 C1(CNC(CNC(CCC)=O)=O)CN(C(=O)CC(=O)OCC)CCC1(F)F C(CCN(C)C)(C(=O)NCC(F)F)NC(CN(C)C)=O CC1(C)C(NC(C2CCC(=O)N2)=O)CCN1C(c1c[nH]c(=N)s1)=O n1(CCC(OCC)OCC2CCCN(C(=O)C)CC2)ccc2cc(F)ccc12 C1(C(C)C)CCCCN1C(c1ccc(OC)s1)C(=O)NCCOCC1CC1 c1(C(N2C(CN(C(c3scc(C)c3)=O)C)CCCC2)=O)cnc2onc(C)c2c1 C1(NC(C(C2(O)CN(C(C#C)=O)C2)F)=O)CCCC1C(N)=O c1(OC)cc(C(=O)NCC2CC(NC(=O)C(C)(C)F)C2)cc2c1OCO2 C(CNC(=O)C(c1ccc(C)cc1)C)(CC)(CC)NC(C1C(OCC)CC1)=O C(=O)(C(CCOC)NC(=O)Cc1ccccc1O)N(CCCC#C)C C=CC(C)(O)CC(=O)N(C)CC1CCCN(C(=O)COC(F)F)C1 c1(C(=O)NCC2=CCN(C(C(C(CC)C)C)=O)CC2)cccc2c(C)[nH]nc12 Cc1cccc(C)c1C(O)C(=O)NC(C)(CNC(c1ccc(C#N)[nH]1)=O)C1CC1 CON1CC(C(N2CCCCC2CC(=O)N(C)Cc2cccnc2)=O)CC1=O CCC1(CO)C(=O)N1.C1(NC(C2CCC(C(=O)OC)CC2)=O)CC2CC(CO)CC12 C1(C(N(C(CC#C)C)C)=O)CCN(C(c2ccnnc2)=O)CC1(C)C N1(C(C(C2CC(C)(C)C2)OC)=O)CCN(C(=O)C2=NNC(=O)C2)C(CC(F)F)C1 c1(OCC)cccc(C(=O)NC(C2CCCCN2C(c2cn(C)c(O)n2)=O)C)c1 C(=O)(CCCCN=[N+]=[N-])N1C(CC(=O)NCC(=O)N(CC)CC)C2CCCC21 c1(NCC23N(C(=O)OC(C)(C)C)CC(CC2)CC3)nc2c(s1)COc1ccccc1-2 C1(NC(C2CCC(CC)O2)=O)COC2C(NC(=O)CN3CCCNC3=O)COC12 CC1CN(C(=O)C(CF)CNC(=O)CCOC2CCC2)CC1N=[N+]=[N-] c1(NC(=O)C(O)CN2CCCCCC2)cccc(CSc2ccccc2)c1 c1(NCC(C)(C2CC2)OC)nn(C(C)(C)C)cc1C#N N1(C(C2N(CC)CCCC2)=O)CC(CC(=O)NCCC2(C)CCCO2)C2(CC2)C1 N1(C(CCNC(COC)=O)=O)CCC2(NC(=O)C(C3CCCCC3)O)CC2C1 c1(C(=O)NC(CNC(c2c(C)ccc(N)c2)=O)(C)C(C)C)ccc(C#N)cc1O C=CCCCC(C(=O)NC(C)C(C)(C)C#N)NC(=O)C(C1CCOCC1)=O C(=O)(C1=CCC(F)(F)CC1)NC1C(C(C)C)CN(C(=O)C=Cc2cncs2)CC1 C(C(C)(O)C(=O)N(C(C)CCNC(=O)C=C1CCCC1)C)OC c1(CNC(=NCC2C(C)CCC2)NC2CCOCC2)ccc(C2CCCO2)nn1 C(CCC(C)C(C(=O)NC1CCOC1)N1CCN(c2cncnc2)CC1)=C(C)C N1(C(C=CC(C)(C)SC)=O)CC2CC2(CNC(=O)CCC2CC2C)C1 C1(C(=O)NCCC(=C)CNC(=O)CCN(S(C)(=O)=O)C)C2CCC(=O)C12 CN1CCCC(CC(N2CCSCC2C(=O)Nc2ccccc2O)=O)C1 C1(C(=O)Nc2ccno2)CN(C(=O)CCC2CCC2)CCN1 c1(CC(C)NC(C2CCN(C(=O)OC(C)(C)C)C2)C)ccc(Br)cc1 c1(N(CCC(=O)NC2CCOCC2F)C(=O)OC(C)(C)C)ccn2nccc2n1 C1(NC(CCC2COC(C)(C)O2)=O)CC12CCC(NC(=O)CCC(F)(F)F)CC2 c1(C(N2CC(N(C(=O)C(C)CO)C)C2)=O)ccc(-c2coc(=N)[nH]2)cc1 CC(F)(F)CCC(C#N)N(C(C1CCC(C(N)=O)CC1)=O)CC1CC1 c1(C(CNC(=O)NCC23C(CN(C(C)=O)C2)C3)CO)ccc(F)c(F)c1 N1(C(c2cnc(CC)s2)=O)CCC(O)(CN(C)C(C2CCCC2C)=O)C1 c1(OC)ccccc1NC(N1CCOC(CC(N2CC(C)C(F)C2)=O)C1)=O Cc1cn2c(n1)CCC(C(=O)N(CC(O)CNC(=O)C(C)S(C)(=O)=O)C)C2 N1(C(C2N(C=O)CCC2)=O)CCC2CCC(C1)N2C(c1c(Cl)ccc2c[nH]nc12)=O C(=O)(C(CC(F)F)NC(c1ccc(C)cc1O)=O)NCC1(C#C)CCCC1 N1(C(CCC(=O)OC)=O)CCOC2CCN(C(c3ccc([N+](=O)[O-])cc3)=O)CC12 C(CCS(C)(=O)=O)N(C(c1ccc(Cn2cc(CSC)nn2)o1)=O)CC CS(=O)CC(O)CNC(CC(Cc1ccc(C(F)(F)F)cc1)CO)=O S(=O)(=O)(CC(=O)N1CCOC(CN(C(=O)C(C)(CO)OC)C)C1)N(CC)CC CCC(CC(=O)N1CCCC(NCC(n2cc(-c3ncccc3N)nn2)C)C1)C(F)F N1(C(C2ON=C(C)C2)=O)CCC2(CC1)CCN(C(=O)CS(=O)(=O)N(C)C)C2 C1(CNC(C(C(C)OC)NC(C=CCOC)=O)=O)COCC(=O)N1C N1(C(c2cc(CC)sn2)=O)CCC(C(=O)NCCC(C)C(F)F)C1C C=C(C)CC(C(=O)N(C(C)C(=O)NCC1CC(=O)NC(C)C1)C)OC C1(C(=O)NC(CCCNC(C2(C(F)(F)F)CC(=C)C2)=O)C)C(F)(F)C12CCC2 c1(SCC)cccc(F)c1F.C12CCCCC1C(=O)NCC(=O)N2.C(COCCO)S C#CCCCC(=O)NCCOCCOCCNC(C1(c2cc(C)on2)CC1)=O N1(C(c2c[nH]c(=N)s2)=O)CC2(C1)CN(C(C1CN(C3CCC3)C1)=O)CCO2 Cc1cc(NC(=O)C(=O)NCNC2CCOC(c3cccnc3)C2)cc(Br)c1 CC1CN(C(c2ncccc2Cl)=O)CC(C)C1NC(=O)Cn1cnc(=N)[nH]1 c1(CC)cccnc1C(=O)NCC1CC(C)N(C(=O)CCSCC(N)=O)C1 C1(CC#C)(C(=O)N(CC)CC2CCCN2C(c2ccncc2C)=O)CC=CCC1 C1(C(=O)NCC(C2(O)CN(C(C(CC)F)=O)C2)(C)C)CCN(C(=O)OC)CC1 C(c1c(F)cccc1F)=CC(=O)NC1(CNC(CN(CC(C)(C)C)C)=O)COC1 C1(C(C(C)C)NC(C2C(C)=C2)=O)CCN(C(c2ccccc2SCCO)=O)CC1 C(=O)(C(O)C(C)NC(=O)OC(C)(C)C)NCc1c(C)ncs1 c1(CC)occ(C)c1C(=O)OCc1cn(Cc2ncccc2Br)nn1 c1(NCCC2(OC)CCC2)ccc(S(=O)(=O)N2CC(C)C(F)C2)c(Br)c1 CC1NC(=O)OC12CN(C(C1(F)CCN(C(C3(CO)CCCCO3)=O)CC1)=O)C2 C1(C(N(CC(C)NC(CS(CC(C)C)(=O)=O)=O)C)=O)COc2ccccc2O1 N1(C(CCC2(C#N)CCC2)=O)CCCCCC1CNC(C1(CO)CCC1)=O N1(C(c2c(C)nc[nH]2)=O)CCC2(NC(c3nn4ccccc4c3C)=O)CCCCC12 N1(C(C2CCC(=O)NC2)=O)CCC(C2CN(C(C3CS(=O)(=O)CCO3)=O)C2)CC1 N1(C(c2c(C(=O)OC)[nH]cc2)=O)CCOC(C)(CNC(=O)C(F)=C(C)C2CC2)C1 Cc1cc(C(N2CC(C(=O)NCc3ncc(C)o3)C(F)(F)C2)=O)c(C)cn1 c1(N2CCC(NC(C(C)(C)CO)=O)C(CO)C2)ccc([N+](=O)[O-])c(C(N)=O)c1 C1(CN(C2(c3cccs3)COC2)CCOC)CC2C=CC1C2 c1(CNC(CC2CCCN(C(c3c(OC)nn(C)c3)=O)C2)=O)c(C)cccc1F C1(c2n(C(c3ccccc3)(CC)C)nnn2)(NCc2ccc(Br)s2)CC(C)(C)C1 CC1=NNC(=O)C1CC(=O)N(CC(=O)NC(C)Cc1ccncc1)C1CCC1 c1(OC)ccc(N)c(C(=O)NCC(O)CN(C)C(c2ccc[n+]([O-])c2)=O)c1 C(CC(=C)Cl)(C(=O)NCCC=CC)NC(C(C=C)C)=O N1(C(C2CC(=C)C2)=O)CCC(C)(C)C1C(=O)NCC(CCC)OC c1(C2(C(=O)NC(c3cnc(C4OCCO4)s3)C)CCCO2)cccc(Br)c1 C1(CNC(C2CC(SC)C2)=O)CCC(C)CN1C(c1ccnn1C(C)(C)C)=O S(=O)(=O)(c1ccc2[nH]c(=NC(C)CCC=CCSC)sc2c1)N(CC=C)C C(c1ccc(Br)c(Cl)c1)=CC(N1CCC(c2nc[nH]n2)C1)=O c1(C(N2C(CNC(c3c(CC)cc(F)cc3)=O)CCC2)=O)n[nH]c(C)c1[N+](=O)[O-] c1(C(N2CC(N(C)C(=O)OC(C)(C)C)CC2(C)C)=O)cnc2ccccc2c1 C1(CC(=O)N(C2CCN(C(=O)C=Cc3ccoc3)C2)C)CCCNC1=O Cc1nc2n(n1)CCN(C(=O)C(c1cccs1)NC(c1scnc1C)=O)C2 C=Cn1nncc1C(=O)N(C)CC1(O)CN(C(C2COCCO2)=O)C1 c1(C(N2CCN(C(CCCC=C)=O)C(C)C2C)=O)ccc(S(N)(=O)=O)nc1 c1(OC)ccc(OC)c(C(=O)NC)c1.n12cc(nn1)CN1CCC1C(=O)NCC2 C(C(C)(C(=O)N(C1CCOC1)C)NC(=O)CC1CCC(C)(C)O1)SC C(=O)(C(F)(F)CCn1ccnn1)NC1C(C)(CNC(COC(CC)C)=O)CCC1 C1(CC)COCCN1C(C1CCN1C(=O)C=CC(F)(F)F)=O c1(N2CC(=O)NCC2)nc(=NCc2cncc(F)c2)[nH]c2c1CCCC2 c1(C(N2CCC(CNC(=O)CCc3cnn[nH]3)C2)=O)ccc(O)c2ncccc12 C(=O)(C(O)C(C(C)C)OC)N1CC(C#C)(C(N2CC(C)(C#N)C2)=O)C1 O=C1Cc2cc(-c3ccc(C(=O)Nc4cc(F)c(F)c(F)c4)nc3)ccc2N1 C1(C(N(C)CC2CCCN2C(C23CC(O)C2C3)=O)=O)CCC(=O)N1CCC(F)(F)F C(C(C)(C)CN(C(=O)CCC1CCCO1)C1CC1)N(C)C.C12(CC1)CC(=O)N2 C(=O)(CC1=CCCC1)N(CC(C)(C)CNC(c1nc(C2CCC2)oc1C)=O)CC C(N=c1[nH]c(N(C)CC2CCCS2)nc2c1CSC2)C1N(CC(F)F)CCCC1 C(=O)(C1CCCc2nccn21)NC1CC(NC(Cc2c(C)occ2)=O)C1 S(=O)(=O)(c1cnn(C)c1)NC(C(=O)NC(C1CCCN(C(COCC)=O)C1)C)C C(=O)(CS(=O)CC)N(C1CCCN(C(c2ccnc(C(F)(F)F)n2)=O)C1)CC Cc1nc2c(C(=O)NCCC(C)NC(C3CNC(=O)C(C)(C)C3)=O)cccc2o1 C1(NC(C2CC(NC(CCCCOC)=O)C2(C)C)=O)CCN(C)C1(C)C c1(CC(C)C(=O)NC2CN(Cc3c[nH][nH]c3=N)C2)ccc([N+](=O)[O-])cc1 c1(CC)ccc(CCC(=O)N(CC(C)CNC(=O)C(C)OCCF)C)cc1 c1(CC(N2C(C(=O)OCC)C(=O)NCC2)=O)ccc(OCC)c(OCC)c1 Cc1ccc2c(ccn2Oc2ccccc2NCCN=c2cc(C)nc(C)[nH]2)c1 CS(C)(=O)=Nc1cccc(C(N2CC(NC(C34CC(C3)C(C(F)(F)F)O4)=O)C2)=O)c1 C1(COCC)(OC)CN(C(c2cn(CCN(C)C)nn2)=O)C1.C1(=O)C(C2CC2)N1 C12(C(N3C(CCC4(C)CCN(C(COC)=O)C4)CCC3)=O)CCC(CC1)OC2 c1(SCCCC(=O)N(C(C)CNC(=O)Cn2ccnn2)C)ccc(F)cc1 S(=O)(=O)(c1ccc(N2CCOC(C3CCC3)C2)c(Cl)c1)NCC1(C)CCC1 C(=O)(CCCC(=O)NC1CCCO1)N1CC(OCCNC(=O)COC2CCC2)C1 CCCC(CCC)C(=O)NCC1CC(C(N2CC(CCC)C2)=O)C1 c1(C(=O)NC(C2CCCC2)CNC(c2ccoc2Cl)=O)csc2ncnc(O)c12 c1(C(N2CCCC(C(C)NC(CCN(CC)CC)=O)C2)=O)coc(S(C)(=O)=O)c1 c1(OC)cc(C(=O)NCC2CCC(NC(c3cc(O)nn3C)=O)C2)ncn1 CCCCC(CCCC)NC(C1(CCNC(=O)COCCC)CC1)=O N1(C(COCCCCCC)=O)CC2CC(C1)CN(C(c1nocc1C)=O)C2 C=Cc1cc(C(=O)NC2(CN(C)C(C3CCN3C3CCCC3)=O)CC2)cc(F)c1 C1(NC(Cc2cc(CC)nn2C)=O)CC2CC(C1)N(C(c1cccnc1N)=O)C2 c1(OC)ccnc(F)c1C(=O)NCC(O)CNC(=O)C(C)N(C)C(C)=O C1(NC(c2cc(CC)nn2C)=O)CCN(C(C2CC(C#N)C2)=O)CC1(C)C C1(CNC(C(C)SC)=O)C=CCN1C(=O)Cn1cc(-c2cccs2)cn1 C1(NC(Cc2c(C)ccnc2)=O)CCC(O)CN(C(C2(C)CC2(F)F)=O)C1 CC1CC(CNC(=O)CC2C=CCCC2)CCN1C(=O)CCSc1nccn1C c1(C(=O)OC)c[nH]ccc1=NC1(CO)CCCCN(C(c2ccc(C(N)=O)o2)=O)C1 N1(C(C=CC=CCC)=O)CCC2(C=C(C(=O)N(CC(C)CC)CC)C2)C1 C(CC(=O)NC1CC2(CCOC2)C1)(C(F)F)NC(C(C)n1cnnn1)=O C1(C(=O)NC(CN(C(=O)Cc2ccc(F)c(F)c2)C)(C)C)CCn2ccnc2C1 C(=O)(C1=Cc2cc(F)ccc2OC1)N(C(CNC(=O)CSC(F)F)C1CC1)C C(=O)(CC(C)(C)C#N)NCCC(=C)CNC(=O)C(C)Cc1cccc(Br)c1 C1(CCC2(CCC)CCC2)CC(=O)N(C(c2oc(C3CC3)nc2C)=O)C1 C(C(C1CCCCC1)NC(c1cc(C#N)c[nH]1)=O)(C(C)C)NC(CN(C)CC)=O c1(CC)cc(C(=O)NCCC2(C(=O)NC3(C(=O)OC)CC3C)CC2)c(C)o1 N12CC3CCC1C(C3)C2=O.c1(C(=O)Nc2c(OC)ccnc2)cn(C)nc1SC CC1CC(NC(=O)COCCN(C)C)CCN1C(=O)C(O)C1CCC1 N1(C(C(CSC)OC)=O)C(C(=O)NC2CC=CC2)CCC1C1CC1 CCC(F)(F)CC(=O)NCCC1CCCN(C(c2ccc(C(=O)OC)cc2)=O)C1 c1(C(=O)NCC2(OC)CCN(C(=O)C(F)C(C)C)CC2)ccc2[nH]nc(O)c2c1 CC(C)C(=O)C(=O)NN1CCCC1C(=O)NCCOC1CCC1 c1(C(C)C(N2CCCC(NC(C3CCCSC3C)=O)C2)=O)cc(F)cc(F)c1 c1(NC(N(C(CC#C)(C)C)C(C2CCCCC2)c2ccccc2)=O)cc(=O)n(C)cn1 C(=O)(C(O)CC(F)(F)F)N1C(CC)C(NC(=O)CCc2ccccc2Cl)CC1 C1(N(C(=O)C(F)(F)Cl)CC)CC2(C1)CN(Cc1cc(C)cc(O)c1)C2 c1(NC(C2CCN2C(=O)CCC2CCCC2)=O)cccc(F)c1F C1(C(=O)NC(CC2CC2)C(N2CC3CC3C3CC23)=O)CC2C(C1)C2(F)F C(C(C)C(=O)NOC(C)(C)C)NC(c1c(CC)[nH]cc1)=O C(=O)(CC(CC)CC(C)C)NC1CCN(C(c2ncc(OC)cn2)=O)CC1(C)C c1(C(=O)NCc2cc(C(=O)NC3CCCC(O)C3)ncc2)cc(O)cc(F)c1 c1(C(=O)NCC2(NC(C(C)N(C)C)=O)CC2)nnn(C)c1N N1(C(CCC(=C)Cl)=O)CCC(C)C(NC(=O)C#CC2CC2)C1 C(=O)(C(O)C1=CCCCC1)N1CCC(CCCNC(c2c(C)ocn2)=O)CC1 CS(=O)(=O)c1cc(N2CC3CC(NC(C4(n5cncn5)CC4)=O)C3C2)ncn1 C1(C(C(=O)N(CCC)CC)(C)C)CCCN(C(=O)C=Cc2cocn2)C1 C1(C(=O)NCCC2CN(C(CCNC(COC)=O)=O)C2)CCC(C)O1 N12CCCCC1C(=O)NCC2=O.C(C(F)CNC(=O)C1CC1)N(C)C CCCCCCCC(F)C(=O)NCCCC(C)NC(=O)C(O)C(F)F O=C1CC(C(N2CCC(CNC(c3cnc(C4CC4)o3)=O)CC2)=O)CC(=O)N1 c1(C(=O)NCC2C(C)CCN(C(CC3(OC)CCC3)=O)C2)ccc(P(C)(C)=O)o1 c1(C(=O)OC)ccc(NC(=O)CC2CCCN2C(c2ccccc2Cl)=O)cc1 c1(OC)c(Cl)ccc(Cl)c1CNC(c1ccc(F)cc1Br)c1nnnn1C(C)C C(=O)(CC(F)(F)C(F)F)N(CCNC(=O)COc1nn(C)cc1Br)CC C1(C(F)F)(CNC(Cn2cc(CC)nn2)=O)CCN(C(=O)CNC(=O)C(C)C)C1 Cc1[nH]c2ccccc2c1CC(=O)N(C1CN(C(C2(O)COC2)=O)CC1F)C C1(CNC(c2nc(C)sc2)=O)CN(C(C2(C)CCCNS2(=O)=O)=O)CCC1(F)F N1(C(C(=O)NC(c2ncc(C)s2)C)OC)CCCC1Cn1cc(CO)nn1.CO N1(CC)CCOCC1CC(=O)NCC1(OC)CN(C(=O)Cc2cccs2)C1 Cc1cccc(C(=O)NC2CCN(C(c3occ4c3CCC4)=O)C2C(C)C)c1F N1(C(CNS(N)(=O)=O)=O)CCC(C2CC2)C1CNC(c1n[nH]cc1Cl)=O CN1C(=O)CSC1=CC(=O)NCCC1CC(NC(=O)COCCc2cccs2)C1 C1(NC(c2ccoc2C2CC2)=O)CN(C(C2CCC3(CCC3)O2)=O)CC12CC2 C1(CN(C)C(c2ccc(N)cn2)=O)CCCC(NC(=O)Cc2ccc(F)cn2)C1 C1(NC(c2n(C)nc(C3CC3)c2)=O)CC2CCC1CN2C(c1scnc1Cl)=O Cc1ccc(O)c(S(=O)(=O)NCCNCC(c2ccc(Cl)c(Cl)c2)O)c1 C1(CC)CCCN(C(c2nocc2C)C(=O)NC(C)C(=O)OC)C1 N1(C(Cc2n[nH]c(=N)s2)=O)CC=CC(NC(=O)C(c2cccnc2)O)C1 c1(OCC)ccc(F)c(C(N2CCOC(CNC(=O)CCSC(C)C)C2)=O)c1F O=C1COc2ccc(C(=O)NC3(CO)CN(C(C4(CO)CCCC4)=O)C3)cc2N1 Cc1cc(N2CCCC(CNC(C3CCCC3C)=O)C2)n2nc(C)cc2n1 C(=O)(CC(C)CC(C)(C)C)N1CCCC(CCC(=O)NCc2c(C)scc2)C1 c1(NC(C2CCN(C(C3CCCOC3)=O)C2)=O)cccc(O)c1 C1(CN(c2cc(NC(c3c(C)ccnc3)C)ncn2)C)COc2ccccc2C1 N1(C(C=CC(C)(C)SC)=O)CC2CCCC1C2CNC(c1ccc(C)cc1)=O N1(C(C=CCN(C)CC)=O)CC2(CCCC2NC(=O)C(F)C(C)C)C1 c1(CC(=O)NC(C)CCCCNC(=O)C(C)C(C)(C)C)ccc2sccc2c1 C(C)(CC(N)C(=O)NCc1cnc(N2CCOCC2)nc1C)OC c1(C(N2CC(F)CC(NC(C(CC#C)C3CC3)=O)C2)=O)cc(C)c(F)cc1F c1(C(=O)NCC(C)CNC(=O)Cc2cccn2C)cn2cccnc2n1 N1(C(C(C)SC(F)(F)F)=O)CCC(NC(=O)CC2(O)CCOCC2)C2(CCC2)C1 c1(C(=O)NCC2CC(NC(C=C(C)Cl)=O)C2)ccc2c(c1)NC(=O)C2(C)C n1(CC(=O)NC2(CC)CCN(C(=O)C=CCF)C2)ccc(O)nc1=O.C(COC)=C1CC1 C(=O)(C1=NOC(C)C1)NC1C(CNC(c2c(CC(C)C)n(C)nc2)=O)C1 CCCCCC(O)CC(=O)NCCCC(CCC)NC(=O)CCP(C)(C)=O c1(C(N2C(Cn3cc(CC)nn3)C(C)(C)C2)=O)ccc(Br)nc1C(=O)O C1(NC(C(CCC)O)=O)CCC2CN(C(c3ccc4c(c3)CCO4)=O)CCC2C1 CC#CCCCC(=O)NC(CO)C(C)NC(C1(CC)CCCCC1)=O c1(-c2n(CC)nc(CS(C)(=O)=O)n2)c(F)ccc2c1OCC2 Cc1cccc(NCCC(=O)NC(C2CN(C(c3nnsc3C)=O)C2)C)c1 Cn1nc2c(c1C(=O)NC13CC(NC(c4ccc(Cl)c(N)c4Cl)=O)(C1)C3)CCC2 c1(OC(C)C)ncccc1C(=O)NC(C1CN(C(=O)C(O)C2CCC2)CCO1)C Cc1cc(C)c(C(=O)NCc2cc(C)c(C(=O)NCC(C)C(C)C)o2)o1 c1(CC)n[nH]cc1C(=O)N(C1(CNC(c2ccc(CSC)o2)=O)CC1)C c1(SC)cscc1C(=O)Nc1ccccc1.C(CCCC)NC(=O)CN1CCCC1 Cc1ccc(F)c(-n2cc(C(C)(C)OC(=N)ON3CC(C)CS3(=O)=O)nn2)c1F c1(NC(C(N2CCC(CC)C2)n2cc(C(C)(C)O)nn2)=O)ccc(Cl)cc1F c1(C(N2C(CNC(CC(CC)OC)=O)CC(C)(C)C2)=O)cnc2c(c1)NCC2 c1(C(N(C(C)C(=O)NCC=CCOC)CCC)=O)cc(C)[nH]c1C CN(C1=NS(=O)(=O)c2ccc(Cl)cc21)CCOCc1ccc(C(F)(F)F)cc1 N1(C(C(C)Cc2ccncc2)=O)CCN(C(c2ncccc2O)=O)CC1C1CC1 N1(C(CCCc2nc(C)sc2)=O)CCC2(CCCC2NC(=O)Cn2ccnn2)C1 C=C=CCCC(=O)N(CC(C)O)CCNC(c1cnc(N)cn1)=O C(CCCCC(=O)NC1CN(C(C2(N3CCCCC3=O)CC2)=O)CCC1F)OCC N1(C(C2CC(SC)C2)=O)CCSCC1CC(=O)NC(C)CC(C)(C)C c1(C(C(=O)NCC(CC)NC(=O)Cc2scnc2C)O)ccnn1C N1(C(C2(CC#C)CCOC2)=O)CC(C)(CNC(=O)CSCCCC)CC1(C)C N1(C(c2c(C)nsc2)=O)CCC(NC(c2cc(=O)n(C)s2)=O)C(CO)CC1 CCCCC(O)C(C)C(=O)NCC1(F)CCCN(C(c2cnc(C)cn2)=O)C1 Cc1c(N)ccc(C(=O)NC2(CNC(C3CCN(C(C)C)CC3)=O)CCOC2)c1Cl N(C1CCc2cc(F)ccc21)CC1N(CC(c2ccc(Cl)cc2Cl)O)CCC1 O=C1CSc2ccccc2N1CCNS(=O)(=O)c1ccc(NS(=O)(=O)C2CC2)cc1 CCCC(CNC(C1CN(CC)CCO1)=O)C(=O)N1CC=CC1(C)C(=O)OC N1(C(c2c(C)ccs2)=O)CC(CNC(c2n[nH]c(C)c2F)=O)C(C)CC1C CC1CC(CCNC(=O)C(O)CN(C)C)CCN1C(c1csc([N+](=O)[O-])c1)=O Cc1cnc(C(=O)NCCN(C)C)cc1C.C12(CCOCC1)C(=O)N2C Cc1cccnc1C=CC(=O)NCC(C(C)(C)C)NC(=O)C=CS(C)=O c1(C(N2CCC(C(C)(C)NC(COCCC#C)=O)C2)=O)cc(Cl)cc2c1OCC2 CN(C)S(=O)(=O)NCC(N1CC(CCNC(C2(CO)CC2(F)F)=O)C1)=O c1(C(N2C(C)(C)CC(C(=O)NC3CCC3O)C2)=O)ccnc2cc[nH]c12 C1(C(=O)NC(C2CCCN2C(=O)C(=O)C2CC2)C)CCCN(CP(C)(C)=O)C1 c1(C(=O)OC)cc(C)c(C(N2CC3CC3(NC(C3CCCC(O)C3)=O)C2)=O)o1 C12(C(N3CCC(C)(C)C(CNC(C4COC4)=O)C3)=O)CC(C)(C1)OC21CCC1 C(=O)(C(CC)(CC)CO)NCC1CCC(C(=O)NC2CCN(CC)C2)C1 c1(NCC2(F)CC(NC(CC(CCC)(C)O)=O)C2)ncnc2c1cnn2C(C)C C1(NC(CCSCCC)=O)COC2CN(C(C3CCCC(COC)C3)=O)CC12 c1(CNC(CC(C)C2CC2)=O)ccc(CN(C)C(c2ccc[nH]2)=O)cc1 C1(CC(=O)N(C2CCC3(CC2)CC3)C)CC2(CC2)CN1C(=O)CC1CCCO1 c1(C(N(C(C)C(=O)NC(C)(C)CF)CC)=O)cc[nH]c2nccc1-2 C(C(O)C(=O)NC(C)(CNC(C1(CC)CC1)=O)C1CC1)=CC CCC(C)(CCO)NC(=O)C(C1CCCC1)NC(=O)Cn1ccnc1 CCC(COC)C(=O)NCC(N1CCN(C(C2(C)CC2(F)Cl)=O)CC1)=O N1(C(c2c(C)con2)=O)CCCOC(CNC(c2ccncc2F)=O)C1 C(=O)(C1=C(COC)N(CC(=O)O)C(=O)NC1c1cnn(C(F)F)c1C(F)F)OCC N1(C(C=C2CCN(C)C2)=O)CCC(C)(C)C(CNC(=O)C2CC2)C1 C1(CNC(CN(C2CC(C#N)C2)C(C2COCOC2)=O)=O)CC(C(N)=O)=NO1 C1(CN(C(=O)C(CC)N(C)C)CC)CCCN(C(=O)Cn2ccnc2C)C1 c1(COC)ccccc1C(=O)NCC12CC1CN(C(c1cc(F)c[nH]1)=O)C2 C=CCC(CNC(=O)C(C)n1cnnn1)C(=O)NCCCCC1CC1C C#CCCCCCC(=O)NC(C)(CNC(C1CC2OC1C1CC21)=O)CO Cc1cnc(F)cc1NC(=O)NCC1(Oc2cccnc2)CCCC1 c1(CNC(c2nnc(C)s2)=O)cc2ccccc2n1C1CC1 C1(NC(CC(CC2CC2)NC(C(C(C)(C)C)=O)=O)=O)CN2CCC1(C)CC2 C(CC(C)C(=O)NC1CC1NC(c1cc(C)c(C)[nH]1)=O)=CC CCCC(C)(C)CC(=O)NC(C)CCCNC(C)=O.c12cccc(n1)NC(=O)C2 C1(NC(c2c(C)ocn2)=O)CN(C(C2CC3CCCC23)=O)Cc2nccn2C1 c1(OC)cc(C(N2CCc3nnnn3CC2)=O)c2ccccc2c1 C(CCC(C)(C)C(=O)Nc1cnn(C)c1Cl)OC C1(CNC(C2C(C(=O)OC)C2)=O)CCN(C(c2cccc(CF)c2)=O)C12CCC2 c1(N(CCCCC=C)C)nc(N(CCCc2ccc(Cl)cc2)C)nc2c1CSC2 C1(CN(C(=O)Cc2cncn2C2CC2)C)CCCN(C(=O)Cc2csc(S)n2)C1 CCC(CC)C(=O)NCCN(C(=O)CC1(C)CC1(F)F)CCc1ccccc1 C=CCC(CC)C(=O)NCC1CC(NC(c2ccnn2COC)=O)C1 C#CCC(C)C(=O)N1CC2CC2(NC(c2ccc(-c3cccc(F)c3)o2)=O)C1 C1(C)(C(=O)NCC(CNC(C2(C(=O)OC)CCOC2)=O)OC)CC2CC2C1 CC1CC(NC(=O)Cc2cccc(O)c2F)CCN1C(c1cnc(Cl)s1)=O C(=O)(C1=Cc2ccccc2C1C)N1C(CCNC(c2c(C)occ2)=O)CCC1 CC1(C(=O)NCC2CN(C(C3(Cc4ccc(Cl)nn4)CC3)=O)CC2O)CCSCC1 CCC1=NOC(CC(=O)NC(C)(CSC)C(=O)N(C(C)CC)CC2CC2)C1 C1(CC)C(NC(=O)CCc2c(C)cnn2C)CCN1C(=O)Cc1ccc(O)nc1 CC1(C)CC(NC(=O)C(O)c2cnc[nH]2)CN1C(C1(Cc2cccnc2)CC1)=O C12CCCCCC1N2.c1(OCCNC(=O)OC(C)(C)C)ccc(Cl)c(Cl)c1 c1(OC)ccc(C(C)(C)C(=O)NCCNC(=O)Cn2nnnc2C2(C)CC2)cc1 n1(CC)cc(C(=O)NCCC2CN(C(=O)C(C)(C)C34CC(C3)C4)C2)nn1 c1(C(C)C)nc(=N)[nH]c(=NCC2(NNC)CC(CO)C2)[nH]1.c1(S)nc(C2CCCO2)n[nH]1 C1(NC(c2cocn2)=O)COCC1C(=O)NCCCn1ccnc1 CCCCC(CNC(=O)C(C)(O)C1CCC1)NC(C1CCCN(C(C)C)C1)=O C1(SCC(=O)NC2CC(NC(C(c3cncn3C)N(C)C)=O)C2)CCC(=O)NC1 CC1Oc2ccc(C(N3CCC(C4CCC4)CC3)C(=O)NC3(C)CC3)cc2C1C c12ccc(o1)C=CC(=O)N2.C1(C(=O)NC(CN(C(C)C)CC)C)C2CCC1CC2 C=C(C)CN=C(NCCC1CCCO1)N1CCCC(OCCCOC)C1 C1(NC(C(C)OCC)=O)CC2CC1N(C(C1(Br)CC1)=O)C2 CCC(C)(COC)C(=O)NC1CN(C(=O)C(OC)OC)CC1O c1(C(=O)NCC2(F)CC(CNC(c3c(CC)nn(C)c3)=O)C2)ccc(C)nc1O CC1(C(=O)NCC2(NC(=O)CC3(O)CCOC3)CCCC2)COC(=O)N1 C(=O)(CN=c1ccc(Cl)n[nH]1)N(C)CCOCCN(C(=O)C(O)CCS(C)=O)C c1(C(N2CCCC(CN(C(CCC)=O)C)C2)=O)ccc2oc(O)nc2c1 C(C1=CCN(C(=O)CSCC(F)F)CC1)NC(c1cccc(N)c1)=O C(=O)(C1Cc2c(Cl)cccc21)NC(C1CCCC1)CNC(CCOC(C)=O)=O Cc1nc(C)c(-c2cn(CCNC(=O)CCOc3ccccc3F)nn2)s1 c1(C(=O)NC2CN(C(COC)=O)CC3(C2)CC3)cnc(O)c2cccnc12 CCC(O)C(F)(F)C(=O)N1CC(O)(CNC(c2ccn(-c3ccncc3)n2)=O)C1 C1(NC(CC2CC(CC)C2)=O)CC(COC)N(C(=O)COc2ccc(Cl)cc2)C1 N1(C(Cc2c(C)occ2)=O)CCCC(CNC(C2CC=CC2)=O)C1 C1(N(C(=O)CCCN(C)C(C)C)C)CCCN(C(=O)C(C)(C)CC2CCOC2)C1 c1(OCCCC(N2CCC(C(C(=O)NCC=C)C)CC2)=O)ccc(C)cc1 C1(C(C(=O)NCCc2n(C(C)C)c(O)nn2)C)CCC(F)(F)CC1 c1(C(=O)NC2CN(C(C3C(=C)CC3)=O)CC(O)C2)cc(C)c(C)cc1C Cc1nn(C)cc1C(C)C(=O)NCC1(O)CCN(C(c2ccc(C(N)=O)o2)=O)C1 c1(CCC(=O)NCCN(C(C2CCN(S(C)(=O)=O)C2)=O)CC)cc(C)cc(C)c1 Cc1ccc2oc(C(N3CC4(CCCCN4C(=O)C4=NNC(=O)C4)C3)=O)cc2c1 c1(SCC(=O)NC(C2CCN(C(C3CC34CCC4)=O)C2)C)nnnn1C C1(N(C(CC(COC)(C)O)=O)C)CC2CCC(C1)N2C(C1CCCC(CF)C1)=O C=C(C)CC(C(=O)N1CCN(C(c2cn(C)nc2Br)=O)C(C)C1)NC(C)=O C1(NC(CC(=C)C)=O)CC(F)CN(C(C2CCCC2OC)=O)C1 C=CC(C(=O)NCC=CCNC(=O)C(C)Oc1cccnc1)OC c1(OC)nc(C)c(Br)cc1NC(C1CCC(N2CCCCC2)C1)=O c1(C(N(CC(CN(C(C2CC(C#C)(O)C2)=O)C)O)C)=O)ccc(Cl)c(C#N)n1 C1(CC(=O)NCC(C)(C)NC(CCc2cn(C)nc2)=O)OCCC1(C)C N1(C(c2nnc(C)s2)=O)CCc2c(c(CNC(=O)C3=CCCC3)nn2C)C1 C(=O)(C(C)CC1CCCC1)NCC1(CN(C(C2(CC=C)CC2)=O)C)CC1 C=CC(CCC)CC(=O)NCC1(NC(c2cc(C)n(C(C)C)n2)=O)CCCCC1 c1(C(=O)NC2CCC(C)N(C(=O)CNS(C)(=O)=O)C2)noc2ccc(F)cc12 C(CCC(=O)NCc1ccc(C(=O)NC2(C)CC2(C)C)s1)OC(C)(C)C c1(CCC(=O)NCC2CC(NC(CN3CCC(C)(O)C3)=O)C2)nnc(S)nc1O N1(CC(=O)NC(CNC(Cn2ncc(C)c2)=O)CO)CCCCS1(=O)=O C=CC(C)(O)CC(=O)N1CC(CNC(=O)Cc2cccc(OC)c2)CC1C c1(C(N2CCN(C(C(=C)F)=O)C(C)C2)=O)nccc2nc[nH]c12 C=C(C)CC(C(=O)NC1C=CCCCC1)NC(=O)CC1(O)CCOCC1 CC(c1cccs1)=CC(=O)NC1(C)CCN(C(=O)C(C)Cc2cccc(Cl)c2)C1 C(=O)(C1=CC(C)(C)C1)NCC(C1CCN(C(=O)C(C)Cn2ccnc2)CC1)C CCS(=O)(=O)CC(=O)NCC(O)CC(=O)N1CCC(F)(F)C1 N1(C(c2ccc(C)c(O)c2)=O)CCC2(C1)CN(C(c1ccc(C(N)=O)cc1)=O)C2 c1(NC(=O)CNC(=O)Cn2nnc(=O)[nH]2)cnc2c(c1)NCC2 N1(C(CC=CCC)=O)CC(CC(N2CCCC(O)CC2)=O)C2(CC2)C1 c1(CC(=O)NCC(CNC(c2ncoc2C(C)C)=O)OC)cnc(C)s1 C(N=c1ccn(CCO)[nH]1)(c1c(F)cccc1F)c1n(CC2C(=C)C2)nnn1 C1(CNC(C=CC(CC)C)=O)C(O)C(O)CN1C(c1cc(=O)c(OC)c[nH]1)=O c1(OC)ccc(OCC(N2CCC(n3cc(-c4cnsc4)nn3)CC2)=O)cc1F c1(C(N(CC(C)NC(c2cncn2C)=O)C)=O)ccc(-c2ccccc2F)n1C c1(N(C(=O)CC2CCC3CC23)C2CCC2)ccc(NCCn2cncn2)nc1 CC(C)C(CN(CCCCC)C(=O)CO)Cc1ccccc1 c1(OC)noc(C2CC2)c1C(=O)NC(C)C(C)NC(=O)CCc1ccccc1O C(=O)(C1Cc2ccccc21)NC1C2OCC(NC(CC(C=C)(C)C)=O)C2OC1 N1(C(C(C2CC(NC(C3(C)CCNC3=O)=O)C2)F)=O)CC(CO)C2(CCC2)C1 N1(C(CSCCCC)=O)CCN(C(c2cccnc2C)=O)C(C)C1C C1(NC(C23C(C(N)=O)(CCC2)C3)=O)CN(C)C(C)(C)C1.C(=O)(CCCC1CCC1)N C1(C(N(C)CCOCCO)=O)CN(C(=O)CC2CCCC(=O)N2)CC1F C1(O)(CN(C(C(C)C2CCC2)=O)C)CCN(C(c2ccc(C(F)F)o2)=O)C1 N1(C(C2C(C(=C)C)OCC2)=O)CC(CNC(=O)CCSC)C2(CCC2)C1 C1(N(CCC(=O)Nc2cnn(C)c2)C)CN(C(=O)CCC=O)CC1C(F)(F)F C(Cc1ccco1)(C(=O)NCc1cc[nH]c1)NC(C(C)c1ccco1)=O c1(-c2cncc(C(=O)NC(CCC)CCO)c2)n[nH]c2c1CCCC2 C1(N(CCNC(c2c(C)csc2)=O)C(C2CCCC2)=O)CCC(=O)N1CC(=O)OC CCC(CC(=O)N1CC(F)CC1CNC(c1cc(C)c(F)cc1N)=O)CC(C)C c1(C(N2C(CN(C(=O)CC3CC=CCC3)C)CCC2)=O)ccncc1C(F)F C1(C(=O)NC2CCN(C3CC3)CC2)(CNC(C(CN(C)C)O)=O)CC12CCC2 Cc1sc2ncnc(CN(CC(C)C)CCO)c2c1C c1(N(C)CCOCC(c2ccccc2)=O)cccc(F)c1.C(=O)O N1(S(c2cc(C(=O)OC)c(OC)cc2)(=O)=O)CCCc2c(Cl)cccc21 C(=O)(C1CNC(=O)c2ccnn21)N1CCC(CCNC(Cc2c(C)occ2)=O)C1 c1(NC(C(C2(C)CC2)NC(c2cc(C)no2)=O)=O)cc(Cl)ccc1O C1(NC(CC=CCC)=O)CC12CC(NC(C1(c3ccon3)CC1)=O)C2 N1(C(C2(SC)CC2)=O)CCCC(CCC(=O)NC2CC(C)C2)C1 c1(C(=O)NCC(C)NCCC2CCCO2)ccccc1C(C)(C)C C(=O)(C1CCCn2ccnc21)NCC1C2CN(C(CC(=O)OC(C)(C)C)=O)CC21 CC1CC(NC(c2cnc(-c3ccc(Cl)s3)nc2)=O)CCCC1O CC1=C(C(=O)NC2C3CN(C(c4ccc(NCCO)cc4)=O)CC23)CCO1 N1(C(C2CCN(C)C2)=O)CC2CCC2(CNC(c2ccccc2C(F)(F)F)=O)C1 C(=O)(C(C)C(C)CCC)NC(C1CCN(C(c2cc(CCC)ncc2)=O)C1)(C)C C1(c2c(C)n(C)nc2)C(C(=O)NC2CNC(C)C2)CC(=O)N1C c1(CC)c(C(N2CCC(c3cn(CCC4CCC4)nn3)C2)=O)ccn1C CC1(C)C=C(C(=O)NC2CC3(CNC(=O)C(F)(F)CN4CCCC4)CC2CO3)C1 CC1(C)CC(NC(c2sccc2CC#N)=O)CCN(C(=O)CSc2cn[nH]c2)C1 C(=O)(CN=c1[nH]c2ccccc2s1)NCC(C)NC(C(C)OCC#C)=O c1(N(C(C(C)OCC(C)C)=O)C)cccc(C(=O)NC2(CC(N)=O)CC2)c1 c1(C(=O)NC(C2CC2NC(C2COC(=O)N2)=O)COC)ccc(NC=O)cc1 C1(CCOC(C)C(=O)NCCC(N)=O)CCN(C(=O)CS(C)(=O)=O)CC1 c1(C(=O)NCCOCCNC(CC2ON=C(CC)C2)=O)cc2c(Cl)ccnc2s1 c1(CC(=O)N(C2CN(C(C3CCSC3)=O)C2)C)cc(F)cc(F)c1 c1(OC)nc(C)c(C(=O)NC2CCC(CNC(c3cccs3)=O)C2)s1 c1(OC)cc(C)c(C(N2CCCC2C(C)NC(=O)CC(C)CCOC)=O)cn1 N1(C(CC2CC(N=[N+]=[N-])C2)=O)CC=C(CCNC(C2(c3ccno3)CC2)=O)CC1 Cc1nnc(O)c(C(N2CCC3(NC(c4ccn(C(F)F)n4)=O)CC3C2)=O)c1C C(CC(C(=O)N1CCC(CF)C1)NC(c1ncncc1OC)=O)=CC C12(C(=O)NC(CC3CN(C(c4cc(CCC)on4)=O)C3)C)CCCC1C2(F)F CC1CN(C(C2CCC2)=O)CC2(CCN(C(c3sc(Cl)cc3Cl)=O)CC2)O1 C1(NC(C(CC)n2ccnc2)=O)CN(c2nnc(C)s2)CC12CCOCC2 C1(CNC(C(CCC)C)=O)CN(C(=O)C=CCOC)CCC1(F)F C(C)(C)(CN=c1ccc(Br)c(S(=O)(=O)NCCC#N)[nH]1)c1cccc(COC)c1 N1(C(Cc2cc(C)on2)=O)CCC2(CC1)CC2C(N1CCC2(CCC2)C1)=O N1(C(c2c(C)c(=O)cc[nH]2)=O)CC(C)C(NC(C2CC3CCC2CC3)=O)C(C)C1 C1(N(C(CCn2cc(C)nc2)=O)C)CCN(C(C2CCN(C)C2)=O)CC1 C(=O)(C(C#N)C(C)C)NC1CCCC(C(=O)NCc2cc(CC)on2)C1 CCCC(C(=O)NC(C)(C)CN(C)C(C1CC1c1cccc(Cl)c1)=O)NC(C)=O C#CCCCOCCNC(=O)CC1CCN1C(=O)C(C)SC(C)C C(=O)(CCCCCCC(OC)OC)N(C(CNC)CC)c1cncs1 c1(C(N2CC3CC3(C(=O)O)C2)=O)cc2ccccc2o1.c12ccc(F)c(c1)O2 n1(CC)nnc(C)c1C(=O)NCC(CNC(=O)CC1(OC)CCC1)OC C1(N(C(C(C)=C2CC2)=O)C)CN(C(c2c[nH]nc2F)=O)CC12CC2 c1(C(=O)NC2CCCN(C(c3cc[nH]c3C3CCC3)=O)C2)nccn2nccc12 CC1CC(CC2CCCC2C(=O)NCCN(C)C(C)C)CO1 c1(OC)ccncc1C(=O)NC1CCCC1CNC(C1CC(n2cnnc2)C1)=O C12(C(N3CCC(CN(C(=O)C(=O)NC4CCC4)C)C3)=O)COCC1C2(F)F C1(CC)C(NC(C2CC(O)CN2C(C)=O)=O)CCN1C(C1(COC)CCC1)=O N1(C(C2CCN(C(C)C)CC2)=O)CCC(NC(c2c[nH]nc2[N+](=O)[O-])=O)C(F)C1 C1(CNC(C2(CC=C)CCCC2)=O)CC2(CCN(C(C3(CCF)CC3)=O)C2)CO1 CCC(C(=O)N1CCC(CCNC(C)=O)C1)C(C)(C)CC C1(CNC(=O)CC2CC2)CCN(C(C2C3CCC(F)C23)=O)CC1O C1(NC(C2N(C(CC(=O)NCC)=O)CC(O)CC2)=O)CCC2CCCC1O2 C1(NC(CCSCC)=O)CC2(CCN(C(C3(C)CCCS3)=O)CC2)C1 c1(C(=O)NC2(C)CN(C(CC(C)c3ccccc3)=O)C2)cc(N(C)C)ccn1 C#Cc1cncc(C(N2CCC(N3C(=O)C3C(C)C)C2)=O)c1.C(=O)(NC)OCC=C n1(CC)ncc2c(N3CCCC34CCN(C(=O)CCC=C(C)C)C4)ncnc12 C1(CC#C)(C(=O)N(CCC(C)NC(c2cncn2C(F)(F)F)=O)C)CC=CCC1 C=CC1CCN(C(C(=O)N)C2(CC(=O)OC)CC2)CC1.c1(N)ccc(OC)cc1 N1(C(CCN(CC)CC)=O)CC(NC(=O)C(F)C(C)C)CC1CO Cc1cnc(N2CCN(C(=O)CCC(N)=O)C(CCO)C2)nc1O CC1CC(C(=O)NC2(C)CN(C(C34CC(C(C)C)(C3)C4)=O)C2)CCO1 c1(C(N2CCCC(C(C)NC(C(C)NC(N)=O)=O)C2)=O)c(Cl)ccc2c1OCO2 N1(C(CSCCC#N)=O)CC2CCC1C(C(=O)Nc1ccc(Cl)c(Cl)c1O)C2 c1(N2CCC(OC)(CO)CC2)nc(C)nc2scc(C)c12.C12CCN(C1)C2=O C1(C(N(S(=O)(=O)C(F)(F)F)C)=O)(NC2CC2)CCSCC1 N1(C(c2cc(OC)n[nH]2)=O)CCC(NC(=O)CNC(c2ccccc2)=O)CC1C C(=O)(CCC(C(C)C)NC(C1CSCC(=O)N1)=O)NCCC(C=C)C C(CC1NC(=O)c2ccccc21)NC(C1Cc2c(nc(C)s2)CC1)=O N1(C(c2ccc(SC)s2)=O)C2CCC1CC(C(=O)NCc1nncs1)C2 C1(CC(=O)NCc2cnoc2)CCCNC1=O.c12cccc(c1)-c1cn(nn1)C2 C1(C(=O)NCCCN(C(C2CC(F)(F)C2)=O)C2CC2)C2CC3CC(C2)CC1C3 N1(C(C(C)C)=O)CCOCCC1C(=O)NC(c1ccns1)C CCCC(C(=O)N1CCN(C(=O)C(C)Cc2ccccc2F)CC1C)C(C)C c1(C(N2CCC(N(C(=O)CCSC(F)(F)F)CC)C2)=O)cc(F)cnc1O Cc1cc(C(=O)N(C)CCC2CCCCN2C(=O)C(C)C(F)F)c(N)c(F)c1 CC(C(=O)NC1CN(C(c2csc(-c3ncc[nH]3)n2)=O)CCC1F)C(C)(C)C C(CC(C)C(=O)NC1C2CN(C(c3ccccc3C)=O)CC12)=CC NS(=O)(=O)N1CCCCC1C(N1CCN(C(=O)CC2CSC2)C2(CCC2)C1)=O Cn1nncc1CCNC(=O)C(C1CCN(C(=O)CC2CC(N(C)C)C2)C1)F c1(CC)cc(C(=O)N(CC(=O)N(C2CCC(C)C2)C)C)n(C)n1 C1(C(N(CC(CCNC(=O)OC(C)(C)C)OC)C)=O)CCCCN1C C1(C(=O)O)(OC)CCCN(C(=O)C(C(=O)OC)C2=CC=CC=C(OC)C2)C1 C(=O)(C(CCN(C)C)NC(=O)CC1(C)CC1)NC1(C)CC(C)C1 CCC(F)(F)C(=O)NC1CCCC(NC(C2CC(=O)N(CN3CCCC3)C2)=O)C1 c1(C(N2CCCCC(NC(=O)CCCCC3CC3)C2)=O)coc2c(Cl)cccc12 c1(C(N(CCCCC(=O)NC2CC(CC)C2)C)=O)cc(C#N)oc1C N1(C(C(C)SCc2ccccc2)=O)CCC(C)C(NC(C2CC2(F)F)=O)C1 CCC(CC(F)(F)F)C(=O)N1CCN(C(C2CCC2)=O)C(COC)C1 CC1=C(C(=O)NC2CN(C(C3CCCC(=O)N3)=O)CC2CC2CC2)CCCO1 C1(C(=O)NC(CNC(CCN2C(C)CCCC2)=O)CO)CC(F)(F)CCC1(C)C N1(C(C2C(C=C)OCC2)=O)CCCCCC1CNC(c1cncc(SC)c1)=O C1(C(N2CCC(N(C(c3n(C)c(S)nc3)=O)CCO)CC2)=O)CC2CCC1OC2 C1(NC(c2ccc(CF)cc2)=O)CC2CC(NC(C3(F)CCCOC3)=O)CC12 c1(OC)ccccc1CC(=O)C(=O)NCC1(NC(=O)C2=CCSC2)CC1 N1(C(CC=C)=O)CCOC2(CCCN(C(c3nc(C)oc3OCC)=O)C2)C1 c1(CN(C(=O)C(F)C2CCC2)CCNC(C2(C(C)(F)F)CCC2)=O)ccc(Cl)nc1 N1(C(CC=CC)=O)CC(CNC(=O)Cc2coc(C)n2)C2(CCC2)C1 C1(OC)(CNC(=O)CO)CCN(C(=O)Cn2nnnc2-c2ccc(Br)s2)C1 C12(C(=O)NC(c3ccccc3)CNC(=O)CCCC3CCC3)COCC(C1)C2 Cc1cc2ncc(-c3cccc(-c4ccc(C)c(C)c4)c3)cc2[nH]1 CCCCC(C(=O)N(C1(CF)CCC1)CC1CC1)NC(=O)Cn1ncn(C)c1=O C1(NC(COC(CC)(C)C)=O)CCOCC1C(=O)NC1(C)CC(N(C)C)C1 c1(NC(C2C(C)CN(C(C3CSCC(=O)N3)=O)C2)=O)ccc(O)c(N)n1 CC(CCC(F)(F)F)N(C)Cc1cc(OC)[nH]c1Br C1(NC(C(Cn2ccc(C)n2)C)=O)CN(C(c2ncsc2C(C)C)=O)CC1(C)C c1(NC(=O)CN2CCC2)ncnc2[nH]cnc12.CC1C(=O)NCC2N1CC2 C1(C(=O)NC2CCC(N(C(C3CN(C(C)=O)C3)=O)C)C2)CC(=O)NC(=O)N1 N1(C(C2N(C(=O)C=CCCC(C)C)CCC(=C)C2)=O)CCOC2(CCCC2)C1 C1(CCNC(=O)C(C)N2CCC2)(OC)CN(C(c2cc(CCCO)on2)=O)C1 C1(NC(c2ccn(C(C)C)c(=O)c2)=O)CN(C(=O)CC2CCCC2)CC2(CC2)C1 c1(C(=O)NCCCOC(CC)CSC)cccc(CCOC)c1 C1(CC)(NC(=O)C(O)CCCc2ccccc2)CCN(C(=O)CC(C)SC)CC1 N1(C(C=CC(C)NC(C2(SC)CCC2)=O)=O)CC=CC1CF N1(C(Cc2c(C)ccs2)=O)CCN(C(=O)CC2CCCC2C)C2CCCC12 c1(C(N2CCOCC2CNC(C2CCC2C(F)(F)F)=O)=O)ccc(Cl)nc1S C1(NC(c2c[nH]nc2F)=O)CCCC1CNC(=O)C(C1(O)CCCC1)=O C1(NC(=O)C(F)OC(F)(F)F)CCN(C(=O)Cc2cc(Cl)ccc2O)CC1F c1(C(=O)NC(C2CN(C(C3C(CCOC)C3)=O)C2)C)cc(S(C)(=O)=O)oc1C C1(CCNC(=O)NCc2cc(CNC=O)on2)CCCN(C2CCC2)C1 N1(C(CCC=C)=O)CCC(C(=O)NCC(O)C(C)C)C12CC2 C12(NC(c3ccsc3OC(F)(F)F)=O)CCC1CN(C(=O)CC1CC=CC1)C2 N1(C(CCC(C)NC(=O)C=C2CCOCC2)=O)CC2NC(=O)OC2C1 C1(C(N(CCCOCCN(C(c2ccc(C)nc2)=O)C)C)=O)COCC(C)(C)O1 N1(C(=O)Cn2nccn2)CCC(O)(C2CCN(C(c3cccnc3)=O)CC2)C1 N1(C(=O)C(=CC2CCCCC2)F)CCC2(CCN(C(=O)CO)C2)C1 c1(C(CN2CCN(C(CC=C=C)=O)CC2)=O)nc2ccccc2s1 CC(CNC(=O)CC=CC(C)(C)C)C(=O)NCc1cn[nH]c1 C12(NC(CC(=O)OCC)=O)CCCC(NC(c3nc(C)ccc3Br)=O)(C1)C2 c1(OC)cccc2[nH]c(C(N3CCCC3CN(C)C(C3CC34CCC4)=O)=O)cc12 N1(C(C(C)CF)=O)CCC2(C1)c1ncn(C)c1CCN2C(=O)CCCC(=O)C1CC1 N1(C(Cc2nc(C)[nH]n2)=O)CC(C(=O)NCCCN(C)C(=O)C2CC2)OC(C)C1 C(=O)(C(O)CC(F)(F)F)NCC1(NC(c2nc(CC(C)(C)C)oc2)=O)CCOC1 N1(C(CC(C)N2CCCC2=O)=O)CCC2(CC1)OCCC2NC(=O)C(F)F C1(OC)CN(CCNC(=O)C(C)C2CCCO2)C1.C1(C(=O)O)(CC)CCC1 c1(C(N(CC)CC2CCCN2C(C2CCCN2C)=O)=O)cccc2sncc12 C(C(C)(F)CNC(c1ccccc1)=O)NC(COC(C)C)=O C(=O)(C(C)C(C)S(C)(=O)=O)NCCCNC(C(C)C=Cc1ccc(F)cc1)=O c12cc(C(N)=O)ccc1N2.c1(OC)ccc(C(=O)C(F)(F)F)cc1.C1(C)C(=O)O1 c1(SC)nccc(C(=O)NCCOC2CN(C(c3n[nH]c(C)c3F)=O)C2)n1 CC1C(C(=O)Nc2ccccc2)CCCN1C(=O)CSCC(c1cc[nH]c1)=O N1(C(C(C)NC(C)(C)C)=O)CC(F)(F)CC1(C)CNC(=O)C(C)n1ccnn1 C1(CNC(=O)OCCCCC)CCCC2(CCC2)O1 CC(CNC(c1ccccc1Cl)=O)CC(=O)N(c1cccc(Cl)c1)C c1(-n2cc(C3(OCC)COC3)nn2)ccnc(C(=O)NC2CCCC(C)O2)c1 Cc1ccc(F)c(C(=O)NC2CC(C)(NC(c3n[nH]c(C)c3C)=O)C2)n1 Cc1c(Br)sc(C(N2CC(C(n3cc(-c4nccs4)nn3)C3CC3)C2)=O)c1C C1(CNC(c2c(C)cc[nH]2)=O)CCCN(C(c2ccc(C3CC3(F)F)cc2)=O)C1 N1(C(c2c(C)ccn2C)=O)CC2CCC(NC(c3ccn4cncc4c3)=O)(C2)C1 C1(C)(CNC(c2c(CC)cccn2)=O)CCCN(C(c2ccc(SC)s2)=O)C1 c1(N(C)C)ccc(C(=O)NC(C2CCN(C(C3(CO)CC3(F)F)=O)C2)(C)C)cn1 Cc1nc(C)c(CNC2C(C)CN(C(=O)COCCC(C)C)CC2C)c(O)n1 C1(NC(C2N(CCCC)CC2)=O)CCC(CNC(=O)Cc2ccccc2Cl)CC1 C1(C(=O)O)(C(=O)NCC(C2CC=CCC2)N2CCCC2)CCNCC1 c1(CCC(=O)NCC(C(C)(C)C)NC(CC(C)F)=O)ccc(O)c(Cl)c1 Cc1ccc(Cl)c(N)c1CN1CCC(C2CCN(C(C3CC4(CCCO4)C3)=O)C2)C1 C1(NC(=O)C(=O)N(CC(F)(F)F)CC2CCCO2)CCCCC1(F)F C(=O)(C(C(C)C)NC(=O)C(C)(C)C)NCCN(C(=O)CC(C)(C)C1CC1)CCC C1(CC)CN(C(C2(COC)CCCCO2)=O)CCN1C(=O)C#CC(C)(C)C Cc1oc(C)c(C(=O)NCCC2CCN(C(c3ccn(C(F)F)n3)=O)C2)c1C c1(C(=O)NCc2cc(C(N3CCC(NC(C)=O)C3)=O)no2)cnc(C)cn1 c1(-c2cc(CN(C(C3C(C4OCCO4)C3)=O)CCC(C)O)[nH]n2)ccc(F)cc1 c1(C(N2CCC(C(C)NC(=O)C=Cc3cn(C)cn3)CC2)=O)ccc(N)cc1F C1(C(C)NC(C(COC)C)=O)CCN(C(c2ncccc2O)=O)CC1 Cc1ccnc(C(=O)NC2CC(CNC(c3ccc(F)s3)=O)C2(C)C)c1N C12(C(N(CCCO)CC)=O)CCC(NC(=O)COC3CC=CC3)(CC1)C2 C=Cc1cc(C(=O)NCC2CN(C(c3ccn(C4CC4)n3)=O)CCO2)cc(F)c1 CCC(CC(=O)N1CCOC(C(=O)N(CC2=CCCOC2)C)C1)C(F)F C(=O)(C1=CC2(CCOCC2)C1)N(C)CC1N(C(c2[nH]cc(CC)c2)=O)CCOC1 c1(C(=O)NC(Cn2cccn2)C(=O)NCCc2cscn2)ccnnc1O C1(c2nnnn2C)(Sc2c(C)cccc2C)CCCC(C#N)C1.c1cccc(F)n1 S(=O)(=O)(c1cccnc1Cl)N1CC2(CCN(C(=O)CC3CCC(F)(F)CC3)C2)C1 C(=O)(C(F)C1=CCCCC1)N1CCC(C)(CCNC(=O)CC2(CO)CCCC2)C1 C(=O)(CCC(C)(F)F)NC(CN(C(C1CCCCN1C)=O)CC)C C1(NC(C(C)(C)OC(C)C)=O)CCCN(C(C2(C#N)CC2)=O)CCC1 N1(C(c2nc(C(=O)OC)sc2C)=O)CC(NC(=O)C#CC2(C)CC2)CC12CCC2 c1(C(=O)NCC(C)NC(c2nccc(CC)c2)=O)cccc2c1CNC2=O c1(CCC)cc(C(=O)N(CC(O)CNC(c2c(C)n[nH]c2C)=O)C)sc1C c1(C(c2n(CCCC)nnn2)NCCCn2cc(C)cn2)ccccc1F c1(C(c2nc(CCO)nn2-c2ccc(Br)cc2)C)cccc(O)c1 C1(C(N2C(CNC(CCc3n(CC)ccn3)=O)CC(F)C2)=O)CC12CCOCC2 c1(C(N(CC(CC)NC(=O)C(C)=C(C)C)C)=O)cn(C)cc(Br)c1=O CCC(C#N)C(=O)NCC1(F)CC(NC(c2ccc(O)nc2)=O)C1 C12(C(=O)NC3CN(C(C(c4cn(C)nc4)O)=O)CC3F)CCCN(CC1)C2 c1(C(=O)NC2CC(CNC(C3(CC)COC3)=O)C2)cnn2ccc(Br)cc12 N1(C(COC(C)=O)=O)CC(CNC(c2cc(Cc3ccnn3C)[nH]n2)=O)CC1C N1(C(C2(CC(=O)NCCC3(CSC)CC3)CC2)=O)CC(C(=O)NCCO)C1 C1(COC)(CNC(c2cc(C3CC3)n[nH]2)=O)CN(C(=O)CC(C)C2CCCO2)C1 c1(NC(c2n(CC=C)nnn2)CC2CCOCC2)ccc(C2CC2)c(Cl)c1 c1(C(C)NC(=O)C(=O)NC2CCCCC2(F)F)cccc([N+](=O)[O-])c1 c1(C(=O)NC2(CNC(=O)CC3CCCO3)CCOCC2)cc2ccc(F)cc2o1 N1(C(C(CC=CC)C)=O)Cc2[nH]nc(C(N3CCC(C)(C4CC4)C3)=O)c2C1 C1(CC(=O)N)CCCCC12CC2.C1(OCC(=O)NC(C2CC(C)C2)C)CC=CC1 c1(C(N2CCCC(C)(NC(C=CC(CC)C)=O)C2)=O)nc2sc(C)cn2c1C CCCCC(CC)C(=O)N1CCC(O)(CCNC(=O)CN2CC3CC3C2)C1 N1(C(CCC(=O)NC)=O)CCC2(CC1)C(OC)CC2NC(=O)C1=C(Cl)CCC1 c1(C(=O)NCC(C2CCCC2)NC(C(C)NC(C)=O)=O)cnc2ccccc2c1 C(CCN(C)C(C1(C)CCCC1)=O)(C(C)C)N.C(=O)(C(=O)NC)NCCNC(C)=O C1(CNC(c2c(SC)ccs2)=O)CN(C(=O)CCC(F)F)CCC1(F)F C(N=C(NC1CC1)N1CCCC(CN2CCCCC2)C1)C1Cc2n(ccn2)CC1 N1(C(Cn2ncc(C(=O)OC)c2)=O)CC2CC2(CNC(c2ccc(SC)s2)=O)C1 N1(C(C(C)N(C(C(CSC)C)=O)CCC)=O)CCC(C)(C(=O)OC)CC1 N1(C(C(N2CCC(CN(C(Cc3c(C)nsc3)=O)C)C2)=O)C)CCC(O)CC1 C1(CCC)CN(C(C2CCC(F)(F)CO2)=O)CCN1C(C1CCC1c1nc[nH]n1)=O N1(C(CCC2CCC(NC(C(C)(C)C(N)=O)=O)C2)=O)CC2CCC(C1)C2C#N C1(C(=O)NCCCCNC(c2nnn(CC)c2C)=O)CCc2nnc(O)cc2C1 c1(C(=O)NC2CN(C(=O)CCN3CCOC3=O)CC2O)cc2cc(Cl)ccc2s1 N1(C(C(CC)(F)F)=O)CC(C)C(C)(CNC(C2CC2c2ccccc2C)=O)C1 c1(OC)coc(C(=O)NC2CCCCC2CNC(=O)C=Cc2cccs2)cc1=O N1(C(C2(SC)CC2)=O)CC(C(=O)NCC2CCCC(C)(C)C2)C2(CCC2)C1 O=C(NNC(=O)CC(O)C1(N)CCC1)c1cc(Cl)cc(Cl)c1 Cc1nc(C)c(CC(N2CC(CN(C(=O)CCc3ccc(Cl)cc3)C)C2)=O)s1 c1(C(N2CCN(C(C=C(C)Cl)=O)C(C)C2)=O)cccc2nonc12 C(=O)(CCCCCSC)NC(CCCCNC(Cc1cccc(OCC)c1)=O)C C1(C(N2CCC(N(C(c3cc(CSCC)on3)=O)C)C2)=O)CN(CC)C(=O)N1 C#Cc1cccc(C(N2CC3CC2C3NC(=O)CC(C)=C=C)=O)c1Cl Cc1cncc(OCC(=O)N(CC(O)CN(C)C(c2coc(Cl)n2)=O)C)n1 c1(OCCC)ccc2occ(CCC(=O)OC3CC(C(=O)OC)C3)c2c1 N1(CCCCOC)CCC(C(C)NC(c2ccn(CC(C)C)n2)=O)C1 c1(CCC(=O)N(CCC(C)NC(C2CCCCS2)=O)C)cncc(Br)c1 C1(CNC(=O)C=C2CC2)CC2(CC(NC(C3CC3c3cccc(Cl)c3)=O)C2)C1 N1(C(c2cccc(CNC(C3CCO3)=O)n2)=O)CC(CO)CC12CCC2 n1(CC)nc(C)c2cc(C(=O)NCCN(C)C(C3OCCOC3C)=O)sc12 c1(OC)cc(OC)c(C(=O)NC2CC(C(=O)NC3CC(O)C3)C2)cc1Br c1(C(N2C(CNC(COC)=O)CC(F)C2)=O)ccc(OC)c(F)c1 Nc1nc(Cl)ccc1C(=O)NC1CC1CNC(=O)C(F)(F)C(O)C1CC1 C#Cc1ccccc1CC(=O)NCC(C)CC(=O)NCC1CC12CCC2 C1(CC(=O)NCCN(C(C(C)c2cc[nH]n2)=O)C)CC(F)(F)C1 C1(CNC(=O)C2CC2)CC(F)(CNC=O)C1.C12CC(C1)C2.CC(C)(C)O.N c1(OC(C)C)cccc(C(=O)NC2COC(C(F)F)C2)n1 C1(NC(CN(CC)CC)=O)C=CCN(C(=O)CC2(CC)CCC2)C1 N1(CCNC(=O)COCCF)CCC(C(=O)Nc2conc2C(F)(F)F)CC1 C(CCCCC(=O)NCCC1NC(=O)NC1=O)NC(c1cc(COC)nn1C)=O c1(CC(C)C(=O)N2CCC2C(N2CCC(O)C(C)C2)=O)ccc(C#N)cc1 CN=c1[nH]c(C(=O)N(C)CCN(C)C(C2CN(c3nnc(O)s3)C2)=O)cs1 C1(C)(CC)CC(NC(=O)CCc2ncc[nH]2)CN1C(=O)Cc1ccon1 N1(C(c2ocnc2C2CC2)=O)CCN(C(c2occ3c2CCCC3)=O)C2CCC12 C1(CN(C(=O)CCc2cnoc2)C)COCCN1C(=O)C(c1cccnc1)N(C)C c1(C(N(CC(CO)(CO)NC(C2C(C)=CCS2)=O)C)=O)cc2ccncc2[nH]1 CCS(=O)(=O)CCN=c1nc2c(ncn2C(C)C)c(NC2COCC(C)(C)O2)[nH]1 C1(C(=O)NC2C(NC(CNC(CN(C)C)=O)=O)C2)OC2CCC1CC2 C(=O)(CP(C)(C)=O)NCC(C(=O)NC1(CO)CC(C)C1)C C12(NC(C(C3CCC3)OC)=O)CCCCCC1N(C(c1cnncc1C)=O)CC2 C(=O)(C1CNC(=O)c2ccnn21)NCCCC(CCC)NC(=O)C=CCOC Cc1cc(S(=O)(=O)N2CCCCCCC2C(=O)N(C)C)ccc1-c1ccncc1F C1(NC(COC2(C)CCC2)=O)CCC(C(=O)NCC2(C)CCCCO2)CC1 C1(NC(CCCc2onc(CCC)n2)=O)CN(C(=O)COCCCOC)CC1F c1(C(N2CC(O)(CCNC(c3cc(C(CC)C)no3)=O)C2)=O)ccc(Cl)cc1F N1(C(CNC(c2cccs2)=O)=O)CC(O)CC12CCC2 c1(C(=O)NCC(CCOC)NC(C23CC4CC2C3C4)=O)cc(O)n(C)n1 C#CCCN=C(NCC1(F)CC1)NC1CC12CCCC2 CC1(NC(C2(N(c3ccccc3)CCO)CC2)=O)CCN(C(c2sccc2Cl)=O)C1 C1(C(=O)NC2COCC2O)(CC)CCCN1C(=O)CC1CCCNC1=O c1(C(=O)N(C2CC(NC(C3(O)CC3)=O)C2)CC2CCC2)ccc(-c2ccncc2)nc1 N1(C(C(CSC)OC)=O)CCCC2CN(C(c3cc(C)c(N)cc3F)=O)CCC12 CC(CNC(=O)CNC(c1cccnc1)=O)(CO)NC(C1CCCS1)=O C1(C(=O)NC2CC(C(C)C)OC2)(C(=O)Nc2cncn2C)CCN(C)C1 C(C(=O)N1CCC(C(F)CNC(C2(n3ccnc3)CC2)=O)CC1)(C(C)C)SC c1(OC)ccc(F)c(CC(=O)NC2CN(C(=O)Cn3cc(C)cn3)C(C)(C)C2)c1 N1(C(CC(C)OC)=O)CC2CCCC(NC(c3cccc4c[nH]nc34)=O)C2C1 CCC(C)C(C(=O)Nc1ccc(C(=O)OC)cc1)NC(=O)Cc1ccccc1C N1(C(C(=O)NCC)=O)CCC2(CC1)CN(C(C1(CF)CC1)=O)CCO2 C(=O)(CC(C)CC(=O)N1CCOCC1CNC(C12CCCC1CCC2)=O)OC C1(C(N(c2ccccc2F)CCC(=O)OCC)=O)CCOC(c2ccccc2)O1 N1(C(C(=C(C)C2CC2)F)=O)CCC(C)N(C(C2CCCC(C(F)(F)F)C2)=O)CC1 N1(C(c2n(C)ccc2Cl)C(=O)NC)CCC2(CC1)CC2(C#N)Cc1ccccc1Br c1(CNC(C(C)S(N)(=O)=O)=O)cccc2c1CN(C(c1cc(C3CC3)no1)=O)C2 c1(C(N(C2CCCCC2NC(=O)C(C)(C)C2CC2)C)=O)ccc(S(C)(=O)=O)[nH]1 N1(C(c2n(CCOCC)ncc2)=O)CCCC(O)(CNC(C2CCCOC2)=O)C1 N1(C(CC=C)=O)CCC2CCN(C(=O)CN3CCCC3=O)CC12 c1(C(N2CCCC3(CNC(c4ccnnc4)=O)C2C3)=O)cc(F)c(F)cc1F N1(C(Cc2c(C)nc(SCC)s2)=O)C(C)CN(C(=O)C(=O)CC(C)CC)CC1C c1(C2(N(C(=O)CCC3CCCC3)C)CC2)cccc(-c2cn(C3CCC3)nn2)c1 C1(NC(CCc2ccc(C)o2)=O)CS(=O)(=O)CC1NC(C1CCC(O)CC1)=O C1(C(=O)NC(CC=C)C(=O)N(C)CC2CCCN(C)C2)CC(C)CC(C)C1 c1(OCC)cc(NCCC2CCC(NC(=O)CCc3cc(C)no3)C2)nc(C)n1 CCC(C)C(CC(=O)N(C)CC1(C#N)CC1)NC(=O)C(C(C)C)C(C)C N1(C(COCC(=O)NC)=O)CCN(C(c2cc(C)c[nH]2)=O)C(C)C1 Cc1csc2ncnc(NC(C3CN(Cc4ccc(O)nc4)CCN3)=O)c12 C(=O)(C(F)C(F)(F)F)NCC1(CCNC(=O)CCC(=O)c2cccs2)CC1 Cc1cc(C(=O)OCCOc2cnc(C)c(C)c2)n2nccc2n1 c1(C(N(CC(=O)Oc2ccccc2Cl)C)=O)cccc(F)c1 N1(C(c2c(C)noc2Cl)=O)CCCC(CO)(NC(=O)C(O)P(C)(C)=O)C1 c1(C(=O)NC(C2CCCCC2)C)ccc(-c2ccccc2F)cn1 C1(C(N(C)C)=O)CCC(F)(F)C1.C1(C2CCCO2)CCN(C(c2cc(C3CC3)[nH]n2)=O)C1 C1(CNC(c2noc(CC)c2C)=O)CCC2CN(C(c3ccc(F)cn3)=O)CC12 N1(C(C)C)CCC(C(=O)NCC2(CNC(c3cccc(=O)o3)=O)CC2(F)F)CC1 C12(CC)CN(C(C3CCCC3N(C(=O)CC(=O)N(C)C)C)=O)C(COC)(C1)C2 C1(CC)CC(C)CN(C(C2(NC(=O)CCOCC(C)C)CC(O)C2)=O)C1 CC(CCN=c1[nH]c2ccc(N)cc2s1)NC(=O)CC1CC(C)(C)CO1 C1(C)(CNC(CC2(OC)CCCCC2)=O)CN(C(=O)C(C)(C)CC#N)C(C)(C)C1 CC(C)CC(F)C(=O)NC1CC(CCNC(c2n[nH]c(C3CC3)n2)=O)C1 N1(C(CC(CC)C2CC2)=O)CCCCCC1CNC(c1cc(C(N)=O)cn1C)=O Cc1ccnn1CC(N1CC(C(N)=O)(CNC(=O)Cc2ccc(Cl)s2)C1)=O c1(C(=O)NC2C(CNC(c3cccc(C(C)C)c3)=O)C2)ncc(Br)cc1O C12(CCNC(c3c(C)nc[nH]3)=O)CCC(C1)N(C(C1(NC(=O)N(C)C)CC1)=O)C2 C1(NC(c2c(Cl)cccc2Cl)=O)CCCCN(C(C2(O)CCOCC2)=O)CC1 Cc1cc(C(=O)N(C2CCN(c3ncc(Br)cn3)C2)C)nn1C(C)(C)C C(=O)(C(C)CCCCCC)N(CCC(=O)NCC(=O)NCCC)C N1(C(=O)C=Cc2ccsc2)CCC2C(CCCN2C(=O)CN2CC3C=CC2C3)C1 C=CCC(CC(=O)NCC(C)OC(C)=O)NC(C1CCCC(=O)C1)=O C=CCC(C)(C)CC(=O)N1CCOC(C(C)NC(CCc2cncnc2)=O)C1 CCC1=C(C(=O)NCc2ocnc2C(N2CCNC(=O)C2)=O)CCCO1 CCC(CC(=O)NC(C)(C)CC(=O)NCc1coc(C)n1)OC N(C1CN(C(C2CC(C)(C)C2)=O)Cc2ccccc21)C(c1c(C)n(C)cc1)=O C=CCCC(F)(F)C(=O)NCCCCN(CCCNC(=O)CC(C)CF)C C12(C(=O)NC34CCCN(C(C(C#C)(C)C)=O)CC3C4)CC3CC(C(=O)N1)C2C3 C1(C(N(C)CCSC2CCCN2C(=O)C(C2CCCCC2)=O)=O)COCCC1(F)F N1(C(C2(CC)COC2)=O)CCN(C(=O)CCCCCc2ccc(I)cc2)C(CO)C1 C=C1CC2(C1)CC(C(=O)N(CC(C)(C)CNC(C1CC(C)(F)C1)=O)C)C2 O=C(O)C(C(O)C1CC1)NCCCc1cccnc1 N1(C(CCC)=O)CC2CCN(Cc3ccccc3)CC2C1 C(C(COC)C(C)C)NC(c1n(CCC)nnn1)c1cncn1-c1ccccc1 CCC(COC)C(=O)N1CC(C(N2CCOC(CN=[N+]=[N-])C2)=O)C(F)C1 Cc1nnccc1C(=O)NC1CCCCC1C(=O)N(C1(CO)CC1)C C(=O)(C1=CS(=O)(=O)CCC1)NC(C(C)(C)Cc1ccc(Cl)cc1)=O.C12CCN1C2 C(CC)(CC(=O)OCC)NC(CC1CC(=C)C1)=O c1(CN(C)C(c2coc(Cl)c2)=O)cn(CC2(CC3CCC3)CC2)nn1 C1(CC)CC(O)CN1C(=O)CC(C)(C)N(C)C(C1OCCC1C)=O c1(NC(CC2N(C(CCOCC#C)=O)CCC2)=O)cncc(C)c1 C1(C2CCC2)(C(=O)NCC#CCNC(=O)CCCc2ccsc2)CC1 Cc1cccc(F)c1C(=O)N.N1(Cc2ncc(C(C)C)o2)CCCC(N(C)C)C1 C1(NC(C23OCCC(C)(C2)C3)=O)CCC2CN(C(c3cnc(Cl)[nH]3)=O)CCC2C1 c1(CC)ncncc1C(N1CC(N(C)C)C(CNC(=O)CN(C)C(C)=O)C1)=O CC(C)C(CCC(=O)NC(CC1CCC1)CO)NC(C1CC2(CC2)C1)=O C1(C(=O)NCC(CNC(c2c(C)noc2N)=O)O)COc2ccc(Cl)cc2C1 C12(NC(CC=CC)=O)COCCC1CN(C(c1cnc(CC(C)C)[nH]1)=O)C2 CCC1=C(C(=O)N(C2CC(CNC(=O)CCCC(=O)OC)C2)C)SCCO1 CC#CCC(C(=O)N1CCOC(C)(C2CC2)C1)NC(c1csc(Cl)c1)=O CCC(C)C(O)C(=O)NCCCC1CCCCN1C(c1cc(C)n(CC)n1)=O C1(CNC(C2(CC#C)CCCCC2)=O)CC(F)(F)CN1C(=O)C(C)NC(C)(C)C c1(CN)n[nH]c2ccc(Br)cc12.n1(CCN2C(=O)C3CC3C2)cccn1.CO Cc1cccc2oc(N3CCCC3C3CCCCN3C(=O)C3=CCC3)nc12 C1(NC(C2C(C)C2)=O)CC(NC(c2nsnc2O)=O)C(O)C1 c1(C(C)C)[nH]nc(C(=O)NC(CO)C(C)NC(=O)C2=NOCC2)c1Br c1(C(=O)NC2CCCN(C(c3cccc(OC)c3)=O)C2)cc(C)c(O)c(C)c1 C(=O)(C1=Cc2cccc(Br)c2OC1)NCCC(C)NC(C(CCCC)CC)=O c1(NCCCNC(C2CCCCCC2)C)ccc(S(=O)(=O)N(C)C2CC2)c(Cl)c1 C(N=c1cc(NCC2CC(O)CN2C)nc(C(F)(F)F)[nH]1)C1OCC(C)(C)C1 C12(C(=O)NCCCCN(C(=O)Cc3ccc(Cl)cc3F)C)CC1CCC2(F)F N1(C(C(CC2CN(C(=O)OC(C)(C)C)C2)F)=O)CCC2(CC1)CC2C#N C1(N(C(=O)COC(C)(C)C)C)CCN(C(c2scc(C)c2Cl)=O)CC1 C1(C(=O)Nc2cc(C)c(Cl)nc2)CC2C=CC1N(C(c1cccs1)=O)C2 C1(C(N)=O)NC(=O)CCN(CC2CCCCO2)C1=O c1(CC)cnc(Cl)cc1Cl.C12(CC1(F)F)C(=O)N1CCC(C1)CN(C)C2=O N(C1CCCn2cnnc21)C(C)C1CC1.C1(N)CC2CCC(C1)N2C c1(C(=O)Nc2ccc(NC(C3C(OCC)C3)=O)cc2C)cc2c(nc1O)CCC2 CCCC(C(=O)NCC(C1CCCC1)NC(C1CC12CCOC2)=O)OC C#CC1CCN(C(C2CCCN(C(=O)C(C)(O)c3ccccc3)CC2)=O)CC1 N=c1cc(C(N2CC3C(CNC(=O)C(F)CC4CCCCC4)C3C2)=O)nc(Cl)[nH]1 c1(C(=O)NCC2N(C(CNC(c3cn(C)nc3)=O)=O)CC2)cc(Cl)cc(Cl)c1 C(=O)(CC(CN(C)C)C(F)F)NCC(CNC(C1C(CC)C1)=O)F CC1=C(C(=O)N2CC(F)CC2CN(C)C(C23CCC(CC2)CC3)=O)SCCO1 c1(C(N(CCOCCC(=O)N(CCCC)C(C)CC)C)=O)ccnc(CO)c1 C1(C(N2C(CCC(=O)N(c3ccccn3)CCO)CCC2)=O)CC2(CC2)CO1 Cc1nc(CO)ncc1C(N1CC(=C(F)CNC(c2cc(C3CC3)on2)=O)C1)=O C1(CN)C2CC3CC(C2)CC1C3.C1(CC)CN(C(=O)CC(F)(F)F)CCC1(F)F C(=O)(C(F)CCC(C)(C)C)N(C(C)=O)CC1C=CCN1C(=O)C(Cl)(Cl)Cl C1(C(=O)N(C2COC2)CC2CCC2)CC12CCOC2 CCC(CCc1ccccc1)C(=O)N1CCC(N(C(C23CC(C2)C3)=O)CC=C(C)C)C1 CC1CC=CCC1C(=O)NCC1C=CCN1C(c1coc(C(F)(F)F)c1)=O c1(-n2ncc(C(=O)NC(CN(C(CCOCC)=O)C)(C)C)n2)ccc(Cl)cc1 C(=O)(C(C)CCCC(C)C)NCC1CC(NC(c2ccc(NC)cc2)=O)C1 C1(OC)CN2CCCC2CC1CNC(=O)C(=O)NC12CCC(C)(CC1)OC2 CN1CCOCC1CC(=O)N(C1CCN(C(C2(P(C)(C)=O)CC2)=O)CC1)C c1(C(=O)NC2CC(C)(NC(c3ccc(C)s3)=O)C2)cnc2c[nH]nc2c1 c1(C(N(CC(CNC(C(C2CC(F)(F)C2)OC)=O)C)C)=O)cnn2ccn(C)c12 C(CC(=O)N1CCC(C)C(O)C1)(C(F)(F)F)NC(C1(CC#C)CCCC1)=O c1(OC)nccnc1C(=O)NC1(CNC(=O)CN(C2CCC2)C)CCC1 c1(OC)ccc2c(-c3ccc(OC)c(OC4CCC4)c3)cc(=O)oc2c1 N1(C(C2CCC(C(CC)(C)C)CC2)=O)CCC2C(C1)NC(=O)CCN2C c1(NC(C=C)C)cc(=NCc2nc(C(F)(F)F)n[nH]2)[nH]cn1 C(CC(=O)NCC1(C(=O)OC)CC1)(C(F)F)NC(CCN(CCC)C)=O c1(N2CCC(C)(C(=O)Nc3nc4c(s3)CCC4)C2)ncnc2c1CC(=O)N2 Cc1cc(C#N)c(F)cc1CNCc1cc(OC)ccc1C(F)(F)F N1(C(C=CCCCCC)=O)CCC2C(CCN2c2nc(C)nc3ccsc23)C1 c1(C(=O)NCCCN(C(=O)C=C2CCCCC2(C)C)C)[nH]nc2c1COC2(C)C C1(C(N)=O)CC=CCC1CNCC(=O)NC(N)=O.n12cnnc1C2 c1(C(C(=O)NC(=O)CC(F)F)c2cccs2)oc2ccccc2c1CCC1CC1 N1(CC2CC(SC)C2)C(=O)CCN(CCc2cccc(F)c2C)C1=O C1(CNC(CCCCOCCC=C)=O)CC2CN(C(=O)C(C)(C)C(C)C)CC12 C(CCC(C)C(=O)NC(C1CN(C(c2cncc(C)n2)=O)CCO1)C)OC C(=O)(C1=CC2CCC=CCCC12)NCCCN(c1snc(CCC)n1)C1CC1 Cc1ccc2c(C(=O)NCC3OC(=O)NC3C(=O)OC(C)(C)C)cccc2c1 N1(C(C2CC(CC)C2)=O)CCCC(CN(C(=O)C(C)CCOC)CC)C1 C1(NC(CC(COC)C)=O)CC2CN(C(c3ccon3)=O)CC2C1 c1(NC(C2C3CC2N(C(=O)CNC2CCC2)C3)=O)ccc(N2CCCCC2)cc1 C(C1Cc2ccccc21)NC(CC=CCNC(c1nc(C)nc(O)c1)=O)=O C(=O)(C1=NNC(=O)CC1)N(C(CNC(Cc1cc(C)cc(F)c1)=O)C1CC1)C CC1CN(C(c2csc3nccn23)=O)CC(C)C1NC(=O)CCN(C)CCO CC(=O)C(C)CC(C)C(=O)N1CC=C(CNC(c2ocnc2C(C)C)=O)CC1 C1(C(N2CC(OC(C)C)C2)=O)CN(C(=O)CSc2cn[nH]c2)C(C)(C)C1 C1(CN)(CO)CCCN(C(=O)C2=CCCC2)C1.c1(C(C(=O)C(CS)=O)F)ccccc1 N1(CC(=O)NC2CCC(NC(c3ccc(C(F)F)s3)=O)C2)CCCNC1=O c1(C(=O)NC2(CCNC(CCC(=O)NCC)=O)CCC2)ccc(Cl)c(C)c1 C1(C(N2C(CN(C(C3(OC)CCCOC3)=O)C)COCC2)=O)CCCCCCC1 n1(CCOC)c(N2CCN(C3(OC)CCCC3)CC2)nnc1-c1cnc(C)nc1 c1(CC(=O)N(C(CCNC(C(COC)C)=O)C)C)nnc(-c2cnccn2)n1C CCCC(C(=O)NC1CC(C(N2CC(F)C2)=O)C1)OCC N1(C(C(C)OC)=O)CCC2(C1)CN(C(c1nccc(OC)c1F)=O)CCO2 c1(CC(=O)NC2CN(C(C3CC(c4ccccc4)CO3)=O)C2)ccc(Cl)cn1 C1(NC(C2CCC(CC)C2)=O)CCN(CCNC(c2cc(C(N)=O)[nH]n2)=O)CC1 c1(CN2CCC(CC(=O)Nc3cc(C(=O)OC)sc3)CC2)ccc2ncnn2c1 c1(C(N(CC(C)O)CCNC(CC(CC)(F)F)=O)=O)ccc([N+](=O)[O-])cn1 CCCC(C)(O)C(=O)NC1CCCC1C(=O)N(C1CCC(CC)CC1)C C(CS(=O)(=O)CC(=O)NCC(CC1CC1)C(=O)NCC(N)=O)OC C1(CNC(=O)OC(C)(C)C)CCC1C(=O)NC(c1cscn1)CO C1(C(=O)NCC2CCCN2C(C2CCCN2S(C)(=O)=O)=O)(COC)CCCC1 C1(C(=O)NC2CC(NC(C(CC)F)=O)C2)CCC2C(CC1)C2(F)F c1(C(N2C(C3(NC(c4c(C(C)C)scn4)=O)CC3)CCC2)=O)cc(Cl)cnn1 N1(C(C(n2cc(Cl)cn2)C)=O)CCCC2CN(C(=O)C(F)=CC3CC3)CCC12 c1(CNCC2CCC(NC(c3cccc(C)c3I)=O)CC2)ccc([N+](=O)[O-])cn1 C(=O)(C1=CC2CCCC12)NCCCC(N1c2ccc(C#N)cc2CC1)=O c1(C(=O)NCCC2(O)CN(C(Cc3cc(C)no3)=O)C2)ccc(O)cn1 c1(N2CCC(CCOC)(NC(C(C(CC)O)C)=O)C2)ncnc2c(C)csc12 c1(C(C(=O)NCC)N(C)Cc2cccc(F)c2)cc(C(C)(C)C)nn1C c1(C(=O)NC2CCC(CNC(C3CCOC3)=O)C2)nc[nH]c2ncnc1-2 C(C(=O)C(=O)C(N1CCC(C)CC1)=O)(c1ccccc1)=C(C)C.C1(N)CCCC1N C1(OC)CC(CC(=O)NCCC2CCCN2C(c2ncncc2C)=O)C1(C)C C1(C(=O)NCCC2CCN(C(CCC#C)=O)C2)CCCN(CC)C1 C1(C(=O)NC(C)C2CC2)CC2CCC(C1)N2N1CCC1.N1CCC(C=O)CC1 CC(C)C(C(=O)OC(C)(C)C)C(=O)NCC1(C)CCCN1C(=O)Cn1nnc(=O)[nH]1 CC(CC(=O)N1CCN(C)C(C(N2CC=CCC2)=O)C1)C(C)(C)C N1(C(c2c(CC)c(C(C)=O)c(C)[nH]2)=O)CC(NC(=O)CCC2CC2)C(N=[N+]=[N-])C1 N1(C(c2cccc(CC)c2O)=O)CC2CCC(C1)N2C(C1CC(=O)OC1(C)C)=O C(CCCC(Cc1ccccc1)C(=O)N(C)C)N(C(c1ccccc1Cl)C)C c1(OC)ncc(C(=O)NC2CCC(NC(=O)C(F)=CCCF)CC2)cc1C C(=O)(C(C(C)(C)C)N(C(=O)CCN=[N+]=[N-])C)NC(CC(=O)OC)C C1(C(N(C)CC2CCCN(C(=O)COCCF)C2)=O)CCCCC(C)(C)C1 C1(CC)CN(C(=O)C=CC(C)(C)SC)CCN1C(=O)CCc1cccc(O)n1 c1(C(=O)NC2(CCCNC(C(CC)CO)=O)CC2)ccc(C)c(OC)c1 N1(C(c2c(F)cc(C)cc2F)=O)CC2CS(=O)(=O)CC2(CC(=O)OC(C)(C)C)C1 S(=O)(=O)(c1cccc(N2CCCC(C)(CS(N)(=O)=O)C2)n1)N(CCOC)CCF Cc1cccc(C)c1C(C)NC(N1CCCC1c1ccnn1C)=O c1(C(=O)NCCCCNC(=O)Cc2ccc(Cl)cc2)cc2n(n1)CCCC2 CC1(C)CCCC(C(N2CCN(CC(C)(C)NC(c3ccccc3)=O)CC2)=O)C1 c1(C(N2C(CNC(C=C(COC)C)=O)CC2)=O)cc2c(Br)cccc2cn1 c1(C(=O)NC2C(C(=O)NCCN3C(C)(C)CCC3)C2)cc(F)cc(Cl)c1 CCCCCC(O)C(=O)NC1CN(C(C2(c3cccc(F)c3)CCC2)=O)CC1O C1(NC(CCC=CC)=O)COCCC1CC(=O)NC1CC(O)C1OC C(C)(C)(CC(C)(c1nnnn1C1CC(F)(F)C1)NCC1CN(C(C)C)CCO1)OC C1(C(=O)NC(CC#C)C(=O)OCC)C(CC)CCCN1C(=O)CCCC1CC1C C1(C(=O)NC)CCN(C(=O)C(CO)NC(=O)Cc2ccsc2C)C1C c1(OC)cccc(C(=O)NCC2(NC(=O)CCCC(=O)C3CC3)CCC2)c1C C1(NC(C(=O)NC(C)Cc2ccc(N(C)C)cc2)=O)C2CCNCCC12.C(CF)N C1(C(N(CCN(C(=O)Cc2ccccc2[N+](=O)[O-])C)C)=O)CCn2ccnc2C1 c1(C(N2CCC(O)(CN3CCOCC3)CC2)=O)ccc(F)c(CO)c1 C(=O)(CCCCC(C)=O)NC(CC)C(C)(C)c1cn(CCC(C)C)nn1 N1(C(c2ncn(CC)c2)=O)CCN(C(=O)CC(=O)NC)C2CCCCC2C1 C1(n2cccn2)(C(=O)NCC(CCC)C)CCN(C(c2cccnc2)=O)CC1 C1(CCC)CN(C(c2c(C)noc2C(F)F)=O)CC1NC(=O)Cn1cccn1 N1(C(C(C)OC2CCCC2)=O)CCC(C(=O)NCCOCCC2CC2)CC1C C1(C)(C(NNC(C2CCC(SC)CC2)=O)=O)CC(C(C)(C)C)=NO1 c1(C(N(CC(CC)NC(=O)C=Cc2ccccc2Cl)C)=O)ccc(F)c(F)c1 c1(CC)cc(C(=O)NCCCCCCN(C(=O)C(F)=C(C)C)C)cc(Cl)c1 N1(C(C(F)=CCC)=O)CC(C2CCCN(C(C3(C4(O)CCOC4)CC3)=O)C2)C1 c1(CC(N2CCN(C(C3CC(=C(F)F)C3)=O)CC2)=O)c(Cl)cccc1Cl c1(C(=O)NC2(CNC(c3ccc(OC)s3)=O)CCC2)ccc2nc(O)[nH]c2c1F C(=O)(C1=CCC(F)(F)CC1)N(C)CC1CCCN1C(c1nccn2nccc12)=O CC(C)(C(=O)NCCC1CN(C(c2ccc(-c3ccccc3)nc2)=O)C1)C(N)=O C(=O)(CC(CN(C)C)C(F)F)NCCN(C(C1(CCCC)CC1)=O)CC1CC1 CS(=O)(=O)CCCN1CCC(C2(C(F)(F)F)N=N2)CC1 c1(C(N(CCNC(c2sc(F)cc2C)=O)CC)=O)ncnc2c1CCCC2 c1(C(=O)NCCN(CCC)C(c2cnn(CCN(C)C)c2)=O)ncnc(C)c1OC C(CCC(C)C(=O)N1CCN(C(=O)Cc2ccsc2Cl)C(CS(C)(=O)=O)C1)OC c1(COCC)cc(C(=O)NCC2CC3CC(NC(=O)COC)CC32)ccc1OC C(C1(O)CCc2ccccc21)N(C)Cc1ccc([N+](=O)[O-])cc1C(F)(F)F n1(CC)c(O)nc2ccc(C(=O)NCC3CC3CNC(c3cnccn3)=O)cc12 c1(C(N(CC(CC)NC(=O)C2=CCCC2)C)=O)ncnc(OC)c1F C1(CNC(=O)C2=CCOCC2)CC12CCN(C(c1ccc(F)c(Cl)n1)=O)CC2 C1(C#N)(C(=O)NCC2C(NC(C3CN(CCC)C(=O)C3)=O)CCC2)CCCCC1 n1(CC)nnc(C(=O)N(CCO)Cc2ccc(C(F)(F)F)cc2)c1C CC1(C)CC(C(=O)NCC2CCN(C(=O)CSCc3cscn3)C2)CO1 C1(CNC(C2(OC)CC2)=O)CC(C)(C)CN1C(c1sc(C2CC2)nc1C)=O C1(CNc2cccc(C(C)(F)F)n2)COC2(CCC(C)CC2)O1 CS(=O)(=O)c1cccnc1C(N1CC(NC(=O)CC2=CCOCC2)C(O)C1)=O N1(C(C2(CCC)CCC2)=O)CC2CC2(NC(=O)C=Cc2ccncc2)C1 C1(C(=O)NCC2CN(C(c3c(C(C)C)scn3)=O)C2)CC(C)OC(C)C1 c1(OCC)ccccc1C(N1CCCC1C1(NC(c2nccnc2N)=O)CC1)=O c1(NC(C(n2ncc(C)c2)c2ccccc2)=O)nc2ccc(Br)cc2[nH]1 N1(C(C(F)=C(C)C)=O)CCCC(C(C)NC(=O)CSc2cnn(C)c2)C1 CC(C)C(C(C)C)C(C(=O)NCCC1CC1)N1CCC(O)C1.C(=O)C1CC1 c1(CCC)nc(C)c(C(=O)NCC=CCNc2ccon2)o1 c1(CC(=O)NCCC(C)NC(c2ccnn2C2CCOC2)=O)cn(C2CC2)cn1 C1(C(=O)NC(C)CNC(=O)C=Cc2nnn(C)n2)CCc2cnnn2C1 n1(CCC)nc(-c2cccc(Br)n2)nc1-c1coc(Cn2cccn2)c1 CC(C)C(CNC(=O)CCC(C)(C)F)C(=O)NCC1CCC=CO1 c1(C(=O)NC2CCC(N3CCC(N)CC3)CC2)ccc(F)nc1Br CCS(=O)CC(=O)NCC1(C(F)F)CCN(C(=O)Cn2nnnc2C(C)C)C1 C1(NC(Cc2cc(C)ns2)=O)CC2(C1)CC(C(=O)NC(c1cccnc1F)C)C2 C1(CC)(NC(C2CCC(C(N)=O)O2)=O)CCCN(C(c2ccc(Cl)cc2)=O)C1 N1(c2ccc(C(=O)OC)c(C)n2)CC2CN(C(=O)C3=CS(=O)CCC3)CC2C1 N1(C(C2=C(C)CCC2)=O)CCCCC(NC(c2ccoc2Cl)=O)CC1 C1(NC(C(C)OC)=O)(CF)CCN(C(=O)COCc2cccc(Cl)c2)C1 N1(CC(=O)NC(C)(CNC(c2nccnc2CO)=O)C2CC2)CCCNS1(=O)=O C1(NC(C2C(COC)C2)=O)C=CCN(C(=O)Cc2ncc[nH]2)C1 C1(C2CC2)(C(=O)NC2C(C)(C)C(O)C2)CN(C(=O)C(F)n2ccnc2)C1 C=C1CC(C(=O)NCC2=CCCC2)(CNC(c2cc(C)sn2)=O)C1 CCCCCCC(C)C(=O)NC(C)(CNC(=O)CCC(=O)NC)CC C12(NC(=O)OC(C)(C)C)CCCN(CC1CC1COC3(CCC3)CO1)C2 Cc1cnc(F)c(CN2CC3(CC(C(=O)Nc4ccnnc4)C3)C2)c1 N1(C(CN2CCC(C)C2)=O)CC2CCC(CNC(C3CCOCC3)=O)C2C1 c1(CC(=O)OC)c(C(=O)NC2CN(C(C3CC=C(C)CC3)=O)C2)c(C)cn1C c1(C(=O)NCC2CN(C(c3c(C)ocn3)=O)CC2C)c(O)cc(Cl)cc1F N1(C(COCCC)=O)CC2CCCC(CNC(=O)C(O)C(C)(C)CC)C2C1 Cc1c(C=CC(=O)NC2CC23CC(NC(C2CC(=O)NC(=O)N2)=O)C3)cnn1C c1(C(N(C2CCN(C(=O)C(C)CC)CC2)CCCC)=O)cc(C)c(Cl)s1 N1(C(c2ccn(CCC)n2)=O)CCCC(C(=O)NC2CCOC2)CC1 C1(C(=O)NNC(=O)C2CCCC(O)C2)(CC)CCCN1C(=O)CN1CCC(C)C1 Cc1cccnc1CC(=O)NCC1(C)CCC(NC(=O)CC2CCCCC2)C1 Cc1cc(Cl)nc(Cl)c1C(N1CC2(CCCN2C(c2cc[nH]c2)=O)C1)=O C(CCCCCN=[N+]=[N-])NC(C(CC(C)C)N(C(=O)CCC(C)(F)F)C)=O c1(NC(C2N(C(C(C(CC)C)OC)=O)C(C(C)C)CC2)=O)cc(C)c(F)cc1O CCC(CC)CC(=O)NC(c1ccc(F)cc1F)C1CCN(C(=O)CO)CC1 Cn1nc(C(=O)NCC2(NC(N)=O)CCCC2)cc1F N1(C(c2c(CN(C)C)cccc2)=O)CCC2C(C1)CN2C(=O)CC(C)(C)F CCC(CC(C)C)C(=O)N1CC(C(F)Cn2cc(C3(C)CCCO3)nn2)C1 C1(NC(CN(C2CC2)CC)=O)CN(C(c2ccc(C(F)(F)F)cc2Cl)=O)CC12CC2 c1(C(C)C)nnsc1C(=O)N(CCNC(=O)CN(C)C(N)=O)CCc1ccccc1 c1(OC)cc(CN2CCCC(C)(CNC(c3cc(Br)ccc3Cl)=O)C2)cc(C)c1 CC(C)C(O)CC(=O)N1C2CCC1C(NC(C1CCC(=C3CCC3)CC1)=O)C2 C1(C(N2CC(N(C)C)C(F)C2)=O)CCC(C)(C)N(C(=O)CCc2nncs2)C1 C(=O)(C1=CCS(=O)(=O)C1)NC(CNC(c1cc(CC)n(CCO)n1)=O)CC(C)C N1(C(C=COCC)=O)CCCC2(C1)CN(C(=O)Cc1ccc(OC)c(OC)c1)C2 N1(C(=O)Cc2cnc(C3CC3)[nH]2)CCOC2(CCN(C(=O)CC3(C4CC4)CC3)C2)C1 C1(C(=O)NCC(C(=O)NC(C#C)C(C)(C)C)C)CC2CC(=O)C1O2 C(=O)(C1=CCOCC1)NC(CNC(Cc1cccc(OCC)c1)=O)CO Cc1noc(C)c1CNC(=O)C(C)(C)C1CCCN1C(=O)Cc1ccoc1 C(=O)(C(C(C)(C)C)N1CCCC1=O)NCC1CCN(C(CC(C=C)C)=O)CC1 n1(CC(=O)NCCC2CN(C(C(COC)O)=O)CC2C)c(C)nc2ccccc12 CC1CN(C(c2ccc(=N)[nH]c2)=O)CCC1C(N1CC(CO)C(CO)C1)=O C(C(F)(F)F)(C1CC1)N(CC(=O)NCCCCCO)CCO.C12CCC(C1)C(=O)N2 Cc1ccccc1C(C)C(=O)NC1CC1CNC(c1cnn(CC(F)F)n1)=O N1(C(c2cn(CCN(C)C)nc2)C(=O)NCC2CCCO2)CCCOCC1 N1(C(C(C)N(CC)CC)=O)CCN(C(c2cnc(CO)nc2C)=O)CC1C C1(C)(CNC(C(C)CSC(F)(F)F)=O)CCCN(C(c2cnc3sccn23)=O)C1 n1(CCC)ccc2c(C(=O)NC3CC(NC(=O)C(C)(F)C(=O)OC)C3)cccc12 C12(C(=O)NC(CNC(c3c(C)ncn3C)=O)C(C)C)CCC(=O)N1CCS2 C=CCC(C)(O)C(=O)NCCNC(C1CCN(Cc2ccnn2C)CC1)=O N1(C(CC2N(C(CC=C)=O)CCC2)=O)CCc2c(O)noc2C1 N1(CC(=O)NC)CCN(C(C(C)C)c2nc[nH]n2)CC1=O C1(C(=O)NC2CC(NC(c3cc(CC4CCC4)ccc3Cl)=O)C2)CC2OC1C1CC21 Cc1c(C(N2CCC3(CC3CNCc3ncccc3F)C2)=O)oc2ccccc12 CC1(C)C(C(=O)NCC2(F)CC(NC(C3CC4(CCOC4)C3)=O)C2)CCS1(=O)=O CCCC(CC)C(=O)NCc1cn(CCNC(C2CC(=O)N(C)C2)=O)nn1 Cc1c[nH]c(C(=O)N(C2CCN(C(=O)Cc3n[nH]c(=N)s3)C2)C)c1C c1(CSCC)sccc1C(=O)N(C1CCN(C(=O)CC(C)n2cccc2)C1)C C1(NC(C2(n3ccnn3)CC2)=O)CN(C(c2coc(C(N)=O)c2)=O)CC1CO Cn1nc(Br)cc1C(=O)NCC(O)CCNC(C1CC=CC1)=O N1(C(CC(CC)SC)=O)CCCN(C(c2ccc(N(C)C)cc2)=O)CC1CO.OC C1(NC(CCCN2CCN(C)CC2)=O)CC2CC(C1)CN(C(c1ccoc1)=O)C2 c1(C(=O)NC2CCCN(C(C=CSC)=O)C2)coc2c1C(=O)NCCC2 c1(CC(=O)N(CC(C)CNC(=O)Cn2cncn2)CC2CC2)nnn(C(C)(C)C)n1 CCCC(CC)CCC(=O)NC(C)CCN(C(=O)C1=CC(C)(CC)C1)C CCCC(CCCNC(=O)C(O)Cc1ccccn1)NC(=O)CC1CC=CC1 c1(C(N2CCN(C(c3n(C)ccn3)=O)C3C2C3)=O)ccc(=O)n2c1CCCC2 c1(C(=O)NCCN(CC(C)O)C(c2cnns2)=O)cccc(N2CCCC2)n1 c1(C(N2C(COC)CN(C(=O)CSCC(C)OC)CC2)=O)cn2ccccc2n1 N1(C(CN(CCOC)C)=O)CCC(CCC(=O)NCC2CCC(=O)NC2)CC1 N1(C(C(c2ccccc2)C)=O)CCC(C2CCCN2Cc2scnc2C2CC2)CC1 Cc1ccc(C(=O)NCC(=O)N(C(C)CNC(=O)CC2CCC(=O)O2)C)cc1C CC1(C)NC(=O)CC1C(=O)NC1CCC(F)(CNC(c2coc(C3CC3)n2)=O)C1 C(=O)(CC(F)F)N(C1CCCC1)CCOCCCNC(=O)COCC(F)F CC1CN(C(=O)C(C)(C)CO)CC(CCNC(c2cnn3c2OCC3)=O)O1 C1(C(N(CC(N2CCC2C(=O)NC2CCC2)=O)C)=O)CC2COCC2C1 c1(C(=O)NCC2C(NC(CCCc3nc(C)sc3)=O)CCC2)cn(C)[nH]c1=N C1(CN(C(=O)C=CC(=O)NC2CC2)C)CCCN1C(=O)C(O)c1ccco1 C(=O)(CCCCCC(C)(C)C)N(CCCCNC(c1cc(O)ccc1Cl)=O)C N1(N(c2n[nH]cc2C(F)(F)F)C)CCCN(C(=O)OC(C)(C)C)CCC1.C C(c1cccc(Cl)c1Cl)=CC(=O)NC1C2(CN(C(c3c(C)[nH]nc3Cl)=O)C2)CC1 N1(C(c2ccc(N(C)C)nc2)=O)CCC(CO)C(NC(=O)CCn2ccnn2)C1 c1(C(C)=O)cc(C(N2CCC(NC(c3cnn[nH]3)=O)CC2)=O)c(C)o1 C1(CC)C(NC(=O)C2CC2)CCN1C(=O)Cn1nc(C)cc1C(F)F S(=O)(=O)(c1ccc(NC(C)CC(N)=O)c(Cl)c1)N1CC(NC)C(C)(C)C1 c1(C(c2ncnn2C(C)(C)C)NCC(=O)NC(C)C)nc2ccccc2s1 C1(NC(c2c(C)nc(C(C)C)o2)=O)CC(F)(F)CC1NC(=O)CCC(=O)N(C)C S(=O)(=O)(c1cccnc1NCC1CC(C)(C)CO1)N(C)Cc1nnnn1C CC(C)(C(=O)N1CCC(CNC(=O)COCC2CCCO2)C1)n1cnnn1 C1(C(N(C2CCCCC2)CCNC(=O)C=Cc2ccccn2)=O)CC2C(C1)C2(F)F C(=O)(C(C)(C)C#N)NCCC1CC(NC(C(c2ccc(Cl)s2)C)=O)C1 N1(C(C(n2c(C)ncc2)C)=O)CC(CNC(c2cnc(O)s2)=O)OC(C)(C)C1 C1(C(N(C)Cc2onc(CC)n2)=O)COCCN(C(=O)C(O)CCSC)C1 C=CCC(CC=C)C(=O)N1CCC(C(N2CCCCC2(COC)CC)=O)C(C)(C)C1 C1(CNC(COCCC=C)=O)CN(C(C2CCCCN2CC(F)F)=O)CCO1 C1(C(N2C(C)CCCC2C)=O)COC2(CCN(C(=O)C(C)n3cncn3)CC2)C1 C1(NC(C(C)OC)=O)CN(C(c2cncc(Cl)n2)=O)CC12COC2 C1(CNC(Cc2c(C)n[nH]c2C)=O)CC2(CC(NC(=O)C(F)(F)C(C)O)C2)C1 N1(C(c2nc(CC)sc2)=O)CCCN(C(C2CC3C=CC2C3)=O)C(C)C1 c1(CC(=O)NC(C)C(C)(C)NC(C2CCCOC2)=O)ccnc(O)c1 C=CCCC(C)(C)C(=O)N1CCC(C2CC2)(CNC(c2cc(C)ccc2C)=O)C1 N(C(=NCc1ccccn1)NCC1CCN1C1CCCC1)CC1(CC)CC1(F)F c1(C(N2C(CCNC(C3N(C(N)=O)CCC3)=O)CSCC2)=O)ccc(F)c(O)c1 CC(N=c1[nH]c(Cl)ncc1[N+](=O)[O-])NC(=O)CC1(C(F)(F)F)CC1 CCC(F)(F)CC(=O)NC12CC(C(N3CCC(C)C3)=O)(C1)C2 Cc1cccc(-c2nc(-c3n[nH]cc3Br)n(CCF)n2)c1 c1(OC)ccc(Br)c(C(N2CC(CNC(c3nnsc3C)=O)C2)=O)c1C C1(N(CCO)C(c2cccc(OC)c2)=O)CCc2nc(C(F)(F)F)ncc2C1 c1(-n2cc(CNC(c3nn(C)cc3N)C)nn2)cccc(OCCF)c1F Cc1cc(F)c(C(N2CCC(O)(C(=O)NC3CCN(C(C)C)C3)C2)=O)c(F)c1 C1(NS(CC)(=O)=O)CCC2CCCCN12.N12CCCC(C1)N(C)CC2=O C(c1ccccn1)=C(C)C(N1CCC(CO)(CNC(c2coc(O)n2)=O)C1)=O c1(OC)cccc(C=CC(=O)NCCN(C)C(C2CCCC2C)=O)c1 n1(CC(=O)NCC2CC2NC(c2cnn[nH]2)=O)nc2n(c1=O)CCCC2 c1(C(=O)NCC2(F)CCC(NC(C3CCCO3)=O)C2)ccnc2c1CCC2 c1(OC)ccccc1NC(=O)C(C)N.C1CO1 C1(CNC(C2(SC)CC2)=O)CN(C(=O)CC2CC(O)C2(C)C)CC12CC2 CC(C)C(C)(F)CNC(=O)C(C)CNC(C1C=CCS1)=O C1(NC(C2CCC(CC)O2)=O)CCN(C(=O)Cc2cc[nH]c2)CC12CCC2 CCCCCC(C)CC(=O)NC1CCCC1CNC(c1scc2c1OCCO2)=O c1(CC(=O)OCc2ccccc2[N+](=O)[O-])ccc2ccccc2n1 C12(NC(CCCOCC)=O)CCCC1N(C(C1(C3CC3)CC1)=O)CCC2 Cc1c(C(=O)NC2CCN(C(=O)CC(C)c3cnn(C)c3)C2)[nH]c2c1CCCC2 c1(C(N2C(C)CC2C(=O)NC2Cc3ccccc3C2)=O)cccc(C#N)c1C c1(CCC)cc(C(N2CC(CNC(c3cc[nH]c(=N)c3)=O)CC2C)=O)sc1C c1(C(=O)NC2CC(F)(CNC(c3nc(OCC)oc3)=O)C2)cc(C)nc(C)c1 Cc1c(C(=O)NCC2(F)CCN(C(c3ncsc3Br)=O)C2)nnn1C CC1(C)CN(C(c2cnnc(Cl)c2)=O)CC1NC(=O)C(c1cc(F)ccc1F)=O c1(OC)ccc(CN=C(NCC(c2c(C)noc2C)O)NCC(C)(C)C)cc1Br C1(C(N2C(CC)C(C(=O)Nc3cccnc3C(N)=O)CC2)=O)CCCCCN1C N1(C(C(C)OCCC(C)C)=O)CCCCCC1CNC(=O)CCCNC(N)=O Cc1cc(F)cc(C(=O)N(C)C(c2ccc(F)cc2)C)c1I C(=O)(C(CC)C(C)(C)CC)NC(CCCC)CC(=O)NC1(CC)CCC1 C(C(=O)N(CC(C)NC(=O)C=CCOc1ccccc1)C)(C(C)C)SC Cc1nccc(C(=O)NCC(C(C)C(C)C)C2CCC2)c1O.C1(=O)CCN1CCO c12cn(nn1)C2.c1(CC(N2C(CN)CC2)=O)cc(Br)cs1 C1(NC(C(Cc2ccsc2)N(C)C)=O)C=CCN(C(c2ccccn2)=O)C1 C1(NC(COC2CCN(C(C(CC)C#N)=O)C2)=O)CC2CC1CC21CC1 N1(C(C2CC2COC)=O)CC(NC(=O)Cc2cnn(C)c2)CC2(CCC2)C1 C(=O)(CC(C)C(C)(C)C)NCC1C2N(C(C(CC)(F)F)=O)C(CC2)C1 O=C1CC(NC(N2CCN(c3cnccn3)CC2)=O)CN1C1CCCCC1 C1(N(C(CC(=O)NCC)=O)CC)CCN(C(C2COCCC2C(N)=O)=O)CC1 CC1CN(C(=O)CCCCCF)CC2(CCN(C(C3C4CC5C(C4=O)C35)=O)C2)O1 c1(C(=O)NC(CC=C)CNC(=O)C(C)(C)C(C)O)cc2c(nc1O)CCCCC2 c1(C(N2C(CNC(=O)CCCc3cccnc3)CCC2)=O)cccc(F)c1 c1(N(C(Cc2c(C)occ2)=O)CCO)ccccc1S(C)(=O)=O N1(C(C2(CC#C)CCCC2)=O)CC2CC(NC(=O)CCOCC(F)(F)F)C2C1 c1(CN2CC=C(CNC(C(CC)NC(C)=O)=O)CC2)ccc(OC)c(Cl)c1F CC(C)CC(O)C(C)C(=O)N1CC2(CC2)CC1CC(=O)NCC1(F)CCC1 N1(C(C(CN(CC)CC)F)=O)CC2OCC(NC(c3cnoc3C)=O)C2C1 c1(SC)nc(Cl)c(CNC(C2CC(CC(F)F)C2)=O)c(Cl)n1 c1(NC(Cn2c(CCC)ncc2)=O)cc(F)c(Br)cc1C N1(C(C(=Cc2cccs2)C)=O)CCC(NC(C2CCN2C(C)(C)C)=O)C12CCCC2 c1(OC)ccc(C(=O)NC(c2ccc3[nH]ccc3c2)C)c2[nH]ncc12 c1(OCC)cc(CN(C(Cc2cc(OC)cc(C)c2)C(=O)O)C)c(OC)cc1C N1(C(c2cc(C)oc2)=O)CC2CCC1C(NC(c1cc([N+](=O)[O-])nn1C)=O)C2 c1(C(=O)NC(C)C(C)C(=O)NCCc2ccon2)cc(C#N)ccc1N N1(C(c2n[nH]c(C)c2O)=O)CCC(CNC(=O)CC2CSCCO2)C(O)C1 N1(C(C2(CCCC)CC2)=O)CCC(N(C(=O)CN(C2CCC2)C)C)C(C)C1 c1(C(=O)NCCC(CNC(CCOCCC)=O)O)cnccc1Br C1(C(N(C)CCn2cnnc2)=O)CCCCC1(C)NC(=O)CN1C(=O)CNC1=O N1(C(C(C)OCC=C)=O)CCc2c(C(N3C4COCC3C4)=O)n[nH]c2C1 C12(CNC(C=C(COC)C)=O)CC(NC(C3CN(C)C(=O)N3)=O)(C1)C(C)(C)O2 c1(NC(CC(CC)NC(c2cc(OC)cnn2)=O)=O)cc(C#N)ccc1O c1(OC)ccc(C(=O)NC(CN(C(=O)CCC(C)O)C(C)C)C)c(Cl)c1 c1(N2CC(CC)N(C)CC2)nc2cccc(F)c2c(=NCCNC(C)=O)[nH]1 C1(C(C)C)CCC(C)CC1NC(=O)CC1CCN(C(=O)CC2(C)CCCCC2)C1 c1(NC(N2CC3C(CNC(C4CC45CC5)=O)(CC3)C2)=O)c(Cl)ccc(Cl)c1O C1(CNC(C(=O)NC(C(C)C)C2CCCO2)=O)C2C3CC4C1C1C2CC3C41 N1(C(C2COC2)=O)CCCC2(CCN(C(C3CCC4(CCC4)CC3)=O)C2)C1 C1(CCC(=O)OC)CCN(C(C)C(=O)NCC(C)C)C1 O=S(=O)(c1cc2sc(=NCCC3CCCOC3)[nH]c2cc1Cl)NCc1ccoc1 N1(C(C(C)NC(CC)=O)=O)CCC(n2cc(C)nn2)C1.N1(CCC2CC2)CCC1 C(=O)(C(C)(C)C(=O)NC(CN(C(=O)CCCCC1CC1)C)(CO)CO)OC C1(O)(CC(=O)N(Cc2nc(CCC)sc2)CC)CCCN(C)C1 c1(CC)ncsc1C(=O)NC(CNC(=O)CC1CCC2CC12)C1CC1 C1(C(=O)NC2(C3CN(CC)C3)CC2)CC(F)(F)CN1C(=O)Cc1cc[nH]n1 c1(CN2C(C(=O)NC(CC)C(=O)O)C=CC2)cccc(Cl)c1Br c1(C(N(C)CCN(C)C(=O)OC(C)(C)C)=O)ccccc1 N1(NC(C2(n3cccn3)CC2)=O)CCN(C(c2cccc(OC(F)(F)F)c2)=O)CC1 C(=O)(C(C)(C)C(=O)NC1CCCCC1NC(=O)CC(C)C1CCCCC1)OCC c1(C(=O)NC(C)CNC(=O)CCn2ncn(C)c2=O)cc(F)cc2c1NCCC2 Cc1sc(C(F)(F)F)nc1C(=O)NCc1ccc(C(C)(F)F)cc1 CC1(C)CN(C(c2n[nH]c(=N)[nH]2)=O)CC1NC(c1ocnc1C(F)F)=O c1(C(=O)NCC#CCNC(C(C)(C)C2CCCO2)=O)cn2ncccc2n1 Cc1ccc(OC2COC2)cc1NC(c1nnnn1C)C1CC(F)C1 C1(CNC(C(C2CCC2)OC)=O)CCCN(C(c2csc(C(N)=O)n2)=O)C1 N1(C(C(=O)N(CCCO)C(C)C)=O)CCC(C(F)(F)F)(N(C)C)CC1 C(C(=O)NC1CC2(C1)CN(C(c1ccc(N(C)C)nc1)=O)C2)(C(C)(C)C)SC C(=O)(CCCCCCCO)N1CC(NC(=O)Cc2cc(Br)cs2)C2(C1)CCC2 c1(C(N)=O)cccc(NC(c2cncc(CNC(c3n[nH]cc3Cl)=O)c2)=O)c1 C1(NC(C(c2csnn2)N(C(C)CC)CC=C)=O)CCC(F)(F)CC1 C(=O)(C(C)(C)CCCF)NC(c1cccnc1)C(=O)NC1CCCC(CC)C1 c1(C(N2CCC(C)(NC(C3CC3c3ccc(F)cc3)=O)C2)=O)cc2scnc2[nH]1 c1(NC23C(CN(C(C4C(C)(Br)C4)=O)C2)CCCC3)ncnc2cccc(Br)c12 C1(CC(=O)NCC(CC)N(C(=O)CC(C)F)C)(OC)CCOCC1 n1(C(C(N2CC(NC(CSCC)=O)C(SC)C2)=O)C)cc2ccccc2n1 n1(CC)cc(Cl)c(C(=O)NC2CCCC(NC(=O)CC3CCC(=O)O3)C2)n1 C1(NC(Cc2nc(C)sc2)=O)CCCC(NC(c2cn(C)nc2C2CC2)=O)C1 c1(C(=O)NC2C3CN(C(=O)COCc4ccncc4)CC23)ccn2ccsc12 CC#CCCC(=O)NC1CC(NC(c2n[nH]cc2Cc2cccnc2)=O)C1 c1(C(=O)NCC2COCCN(C(C34CC5CC3C4C5)=O)C2)ccc(F)c(F)c1O N1(C(CSc2c(C)ccc(C)c2)=O)C2CCCC1CC(NC(C1(F)CC1C)=O)C2 Cc1ncn(C)c(=O)c1C(N1CCC(NC(=O)COC(F)(F)F)CC(O)C1)=O Cc1c(C(N2CCN(C3CN(C(c4ccc(CO)s4)=O)C3)CC2)=O)cccc1O N1(C(C2(C(C)(F)F)CC2)=O)CCC(N(CCO)C(C2CCCSC2)=O)C1 c1(OCC(=O)NC(C)C(C)(C)NC(=O)C(F)(F)C(O)C2CC2)c(F)cccc1F c1(C(N2CCC(NC(C(C)Oc3ccccn3)=O)C(F)C2)=O)cc(F)c(Cl)c(F)c1 C1(C(=O)NCC(C(=O)N(CCCCO)C)OC)(COC)CCCO1 c1(OC(C(=O)NCCCn2cc(CC(CSC)O)nn2)C)ccc(F)cc1 n1(CCC)nnnc1C(c1ccn(CCF)n1)NCC1CCCCO1 C(=O)(N=c1ccn(C2CC2)cc1C)S(c1ccc(CCC)cc1)(=O)=O n1(CC=C)ncc2ccc(C(=O)N(C(C)C)Cc3cccc(F)c3)cc12 CCC(O)C(F)(F)C(=O)N1CC(NC(c2cc(F)ccc2Cl)=O)CC(C)C1 N1(C(CCNC(C(C)(C)C)=O)=O)CCCC1(C)CNC(C12CC(C1)C2)=O C1(CNC(C(Cn2ccc(C)n2)C)=O)CCN(CCN2CCCC2=O)CC1 C1(CC(=O)N(C2CCN(C(C3CC34CC4)=O)CC2)CC#C)CCn2cncc2C1 c1(C(N(C)CC2CCN(C(C3ON=C(C)C3C)=O)CC2)=O)c(F)cc(Cl)cc1F C1(C(=O)NC(c2ccncc2)C)(CO)CCN(C(c2cnsc2)=O)C1 Cc1cccc(C(=O)NCC(C(C)C)NC(=O)C(C(C)C)n2ccnc2)c1 C1(CCC(=O)N(C2CC(OC)C2)C)CN(C(=O)CN2CCCCC2)CC1C CON=CC(=O)NC(C)CCNC(=O)C=Cc1cscn1 c1(C(=O)NCC2C(Cn3cc(C(CC)O)nn3)C2(F)F)ccc2c(c1)CC(C)O2 Cc1cc2[nH]c(C(N3CCC(CNC(c4cccc(N)c4O)=O)C3)=O)cc2s1 C1(CC)CCC(C(=O)NCCNC(CNC(=O)C(C)n2cncn2)=O)C1 C(CCCCCC(=O)N1CCC12CCOCC2)NC(CCc1ccn(C)c1)=O c1(NC(CCOCC#C)=O)nn[nH]c1C(=O)OC(C)C N1(C(CC(CCCC)NC(C2CCOC2C(C)C)=O)=O)CCN2C(=O)NCC2C1 c1(C(CNC(c2nccc(Cl)c2)=O)F)ccc(Br)cc1.c1(CCC(C)=O)c[nH]nn1 C(=O)(CCCCC(N)=O)N(C)CCNC(=O)COCc1cccc(Cl)c1Cl C(=O)(C(CNC(C1CC1C(F)F)=O)N(C)C)N(CC)Cc1cccs1 Nc1snnc1C(N1CCC1C(N1CC(N2CCCOC2)C1)=O)=O C1(C(N2CCC(CC)(CO)C2)=O)N(C(c2n[nH]cc2Cl)=O)CCCC1(C)C C1(C)(C(=O)NC2CC(NC(C(C=C)c3ccccc3)=O)C2)CCC2CC2C1 CCCCCC(O)C(C)C(=O)NCCC1CCN(C(=O)Cc2cnoc2)CC1 C12(NC(c3c(CC)n(C)nc3)=O)CCCC1N(C(=O)C=C1CCC(C)C1)CCC2 C=CCCCCCC(=O)N(C(CNC(=O)C(c1ccccc1)N(C)C(C)=O)CC)C CC(C)(C)C(C(=O)NC1CN(C(=O)Cc2cccnc2)CC1O)N1CCCC1=O c1(C(N2C(CC)CN(CC(=O)O)CC2)=O)coc2cc(OC)ccc12 c1(N2C(CC)(COC)CCC2)ccc(S(=O)(=O)NC2CCCN(C3CC3)C2)cn1 N1(C(C(C)(C)NC(=O)C(F)(F)F)=O)CC2CCNC(C2)C1 C1(OC)CN(C(=O)CN2CCC2C)CC1NC(=O)Cc1cnn(C(F)F)c1 c1(C(=O)NC2C3(CC(NC(C(C)OCCCC)=O)C3)C2)cc[nH]c(=NC)c1 C1(CNC(c2nc(C)oc2C)=O)CN(C(C23COCC2C3)=O)C2(CCC2)C1 C=CC(CC)CC(=O)NCCOC1CCN(C(c2nccc(C)n2)=O)C1 Cc1nc(CCC(=O)NC(C2CN(C(=O)CCc3cn[nH]c3)C2)C)cs1 C(C)(C(O)C(=O)NCC1CC(F)(CNC(C2CCN(C(C)=O)C2)=O)C1)OC C(CC(C)(C)CC(=O)N(C)CC1CN(C(C2(C)C=CCC2)=O)CCO1)OC c1(NC)ccc(F)cc1C(=O)NC(C1(NC(C2CCCN(C)C2)=O)CC1)C N1(C(C2(COC)CCCO2)=O)CCC12CN(C(c1cccc(C3CC3)c1)=O)C2 c1(CC)ccc(C)c(C(=O)N(CC(C)NC(c2cc(O)n(CC)n2)=O)C)c1 C(=O)(C(CC=CCl)c1ccccc1)NC1C(NC(c2cnc(C(C)(C)C)[nH]2)=O)C1 C(=O)(C(F)C(C)(F)F)NCC1C(CC)CCN1C(c1cccn1CC)=O c1(C(=O)NCCC(C)N(C(C=C(C)C(F)F)=O)C)ccc2c(c1)C(=O)N(C)C2=O N1(C(C2(COC)CC=CC2)=O)CCC(OC)(CNC(C2CCSC(C)C2)=O)CC1 c1(CNC(C(C(C)c2cccc(Cl)c2)N)=O)cc(Cl)cc2c1OCOC2 N1(C(=O)OC(C)(C)C)CCC2(CC2C(=O)OCc2cc(Cl)ccn2)C1 C(CCCCC(=O)N1CCN(C(N)=O)CC1)N(C1CCCN1C)C c1(C(=O)NC(C)C(CO)NC(c2cccc(F)c2)=O)cc2c(s1)CCS(=O)(=O)C2 O=C(C1=CC2CCC(C1)C2)NC(C1CCCCC1)C(=O)N(CC(F)F)C1CC1 C1(CCC)C(=O)NCCN1C(=O)Cc1nccn1-c1cccc(F)c1 C(=O)(CCCCCCCc1nn[nH]n1)NC1CC(OC(C)(C)C)C12CCC2 C(c1cc[nH]c1)=CC(=O)N(CCC(C)NC(=O)Cc1cncnc1)C N1(C(C(C)(C)F)=O)CCCCC2(CCN(CCNS(C)(=O)=O)C2)C1 c1(CNCC2(NC(c3ccc(Br)s3)=O)COC2)cc(Br)cc(Br)c1O c1(OCC)ccnc(CNC(=O)C(=O)NC(C2CCOC2)CN)c1 S(=O)(=O)(c1ccc(Br)cc1NC1C=CC(C(=O)NC)C1)NC(c1n(CC)ccn1)C N1(C(C(C)CC(F)F)=O)CCC(CNC(=O)C(C)Cc2cnc[nH]2)C12CCC2 C1(C(N(C)Cc2nncn2C)=O)(CO)CCN(C(=O)CCC2CCC(=O)C2)C1 c1(C2N(C(C(=O)NCC(=C)C)C3=NOCC3)CCC2)ccc(Cl)c(Cl)c1 CCC(C)C(C(=O)NCCCC1(NC(=O)CCc2ccccc2C)CC1)OC Cc1ccc(C(=O)NC2CC3(C2)CN(C(C2C(C)(C)C2(C)C)=O)C3)c(F)c1 C=CCCCC(C(=O)N1CCNC(=O)C1)NC(=O)COCC(=O)OCC Cc1c(C(=O)NCCC(C)NC(c2ccc([N+](=O)[O-])[nH]2)=O)nn(C)c1N Cc1ccc(C(N2CCCC(NC(=O)C=Cc3ccc(Cl)s3)C2C)=O)cc1C#N CC(F)(F)CCC(=O)NCC(F)CNC(C1CCCN(CC(F)F)C1)=O CC(CO)C(C)N=c1ccnc(N(CCCCCC2CC2)C2CCCCC2)[nH]1 Cc1c(C(N2CC3CC2C3NC(=O)CN2CCCC2C)=O)oc2c(C)cccc12 C1(CNC(C2CC23CC(O)C3)=O)CCCN(C(C2(C3CC3)CCC2)=O)C1 N1(C(CNC(C2N(CC)CC2)=O)=O)CCCC(Nc2cc(C(N)=O)ncn2)C1 C1(F)(C(N2C(C(=O)Nc3cc(C)ns3)CCCC2)=O)CCCCC1(F)F c1(OC)cccc2c(C(=O)NC(C)CCNC(c3cccc(Cl)c3N)=O)n[nH]c12 c1(C(N(C2(CC(N3CCCC(C(C)O)C3)=O)CC2)C)=O)cc(Cl)ccc1Cl c1(N2CCCN(C(=O)CCCc3cnccn3)C2)cccc(Cl)c1 c1(CCOC(C(C)(C)S)=O)c2c(cc3c1CCC3)CCC2.C1CCC(F)(F)CC1 C1(NC(C2CCN(C(c3c(CC)ocn3)=O)C2)=O)CCC2CC2CC1 c1(C(=O)NCC(CC(=O)N(C)Cc2cn[nH]c2)C2CCC2)nnc(O)nc1O N1(C(C2CN(C(CCC(=O)Nc3nccs3)=O)C2)C)CCC(CO)CC1 c1(C(=O)NC2C3(CC(NC(c4oc(CC)c(C)c4)=O)C3)C2)ccn2nccc2c1 c1(C(=O)NCC2C=CC(NC(c3ccc(C(F)F)o3)=O)C2)cnc(S)n1C1CC1 C(CCCCC(=O)N1CCN(C(c2ccc(Br)o2)=O)CC1CCO)OC C1(NC(COCCN(C)C)=O)CN(C(C2(CO)CCOC2)=O)CCC1(C)C N1(C(CC2C(=O)NC(=O)N2)=O)CCc2ccc(COc3ccccn3)cc2CC1 CCC(O)C(C)C(=O)N1CC(C)(C)CC1CNC(C1(C(F)F)CCC(C)CC1)=O CCCCC(C(=O)N1CC2CC2(NC(c2ccc(C)c(OC)c2F)=O)C1)C(C)C C(=O)(C1=CCN(C(=O)Cn2nccc2C)CC1)N(CC)Cc1ncc[nH]1 S(=O)(=O)(c1ccc(N2CCC(CC(C)(C)C)C2)cc1Cl)NCC(C)(CO)OC C(=O)(C(CC(C)C)ONCNCCc1cnn(CNC)c1)SCCSCC.C=CC(C)OC C(CCCC(N)=O)NC(c1c(CNC(C=CC=CCC)=O)c[nH]n1)=O CCCCC(C)CCC(=O)OCC.C12(C)CCN(C1)C(=O)CCCN2C(=O)NCC CCC(F)(F)CC(=O)NCCCCCNC(C1CC1c1ccc(Cl)cc1)=O c1(OC)cc(C(=O)NCC(C)(C)CNC(C2CC3(CCC3O)C2)=O)cnc1C N1(C(c2c(CC)cncc2)=O)CCC2CN(C(=O)Cc3sc(O)nc3O)C2C1 C(CC(C)(C)CC(=O)N1CCCCC1C(C)NC(C1CC=CC(O)C1)=O)OC c1(C(=O)NCC(CC)NC(C2CCC2OC)=O)cc(C(=O)OC)nn1C N1(CCN(C)C(C2(C)CCCCC2)=O)CCN(C(C2CCC3CC23)=O)CC1 N#CC1(C(=O)NC2CCN(CCCNC(C3(CO)CC3(F)F)=O)C2)CCOCC1 N1(C(c2nccc(C)c2)C(=O)NCC2CCOCC2)CCCOC(C)C1 C1(CN(C(=O)CN(C)C(C)=O)CC)CCCN1C(=O)CCCc1ccccn1 C1(CC(N2C(CNC(CCOCC#C)=O)CCCC2)=O)COCC(C)(C)O1 N1(C(C(C=C)(F)F)=O)CCC2(C1)CN(C(=O)CCCCC)CCO2.CCCCOC Nc1cnccc1C(=O)NC1CCCCC1NC(c1coc(O)n1)=O N1(C(C=C(C)C(F)F)=O)CC2CC(O)C1C2NC(C1CC(CC2CC2)C1)=O C1(O)(C(C)C)CCN(C(=O)COC(c2ccc(F)cc2)C)CC1 C1(C(=O)NC(CNC(CNC(c2ccc(C)s2)=O)=O)C2CC2)CCC=CCCC1 N1(C(CC(CC)C)=O)CC2CC3CC2C1C3NC(c1cc(C)no1)=O C12(CCNC(C3CCC(C(N)=O)O3)=O)CCC(C1)N(C(=O)Cc1ccoc1)C2 C12(C(N(CC(C)N(C(=O)CC3(C)CCOCC3)C)C)=O)CCC(C1)C2(C)C c1(COC)cccnc1C(=O)NCC1CC(OC)CN1C(C1(N(C)C)CC1)=O C=CCC(CC(F)F)NC(=O)CN(C(=O)CCn1cccc1)C1CC1 N1(C(CC(N2CCCC2C2(SCC(F)F)CC2)=O)=O)CCCCC(F)(F)C1 C(C)(CCC(=O)NC(C)C(CO)NC(c1coc(C(C)C)n1)=O)OCC C#CCC(C)(CC)C(=O)N1CC2(CO)CC1(C(=O)N(CC(CC)CC)CC)C2 C(=O)(CC(C(F)(F)F)NC(C1SCCS1)=O)NCCC1CCN(C)C1=O CC1CN(C(=O)C=Cc2cnn(C)c2)CCCN1C(C1(C)CC1(Cl)Cl)=O c1(C(C(=O)Nc2ccccc2C)N(CCCC#C)C)cccc(CN(C)C)c1F c1(C(=O)NC2CN(C(CC(CCCC)O)=O)CC2C)ccc2c(c1)NC(=O)NC2 N1(C(c2cc(C)oc2C)=O)CCCC(NC(=O)C(O)C2CCCC2)CCC1 C1(CNC(COC(CC)C)=O)CN(C(=O)C(F)(F)CCn2cccn2)CC12CC2 C1(NC(=O)CC2COC(=O)C2)CCC(O)CN(C(=O)CN2CCCC2)C1 c1(OC)cc(OCC)ccc1S(=O)(=O)Nc1cc(N)ccn1 C1(NC(c2ccc(OCC)c(C)c2)=O)CC2(CCN(C(=O)C=CC(F)(F)F)C2)C1 Cc1nn(C)c(C)c1C(=O)NCC1CC(C(=O)NCCC(C)N(C)C)CO1 c1(C(=O)NC(CC=C)CNC(=O)C(CC)N(C)C)cnc(O)n(C)c1=O CCC(C#N)(CC)C(=O)N1CCC1CNC(c1cnc(-c2cccs2)s1)=O Cc1cc(F)ncc1C(=O)NC1CC(C(=O)Nc2cnc(Cl)nc2)C1 C1(CC=C)(NC(C2CC3(CCCC3)CO2)=O)CC2CCC(C1)N2C(c1cnn[nH]1)=O CCC(C)C(O)CC(=O)N1CCC(O)(CNC(=O)CCC(=O)N(C)C)CC1 C(=O)(C(O)CCS(C)=O)NCC1CC12CCC2.c12ccc(s1)C(=O)NC2C c1(C(N2C(CNC(CCOC)=O)CC2)=O)ccc2c(n1)NCC(=O)N2 C1(C(=O)NC2CN(C(C(C)=CC)=O)CC(F)C2)CCc2ncccc2C1 c1(C(=O)OC)ccc(N2CCC(OC(c3cc(C(C)(C)C)no3)=O)C2)nc1OC N1(C(CCC=CC)=O)C2CCCC1CN(C(=O)CCSCC)C2 CC(CCC(=O)N(C)CCCC(N)=O)Nc1cc(C(F)F)ncn1 Cn1ccc(=NCc2cccc(C(=O)N(CCCO)CCN)c2)nc1O c1(C(N2CC=CC(NC(CCCC)=O)C2)=O)cccc2c1CC(C)(C)C2 CC(C)C(O)(C(=O)N1CC(NC(=O)C(C)CC2CCCC2)CC(F)C1)C(F)(F)F c1cc2n(c1)CCOC2.C1(NC(=O)C=CC(N2CCOCC2)=O)CN(C)CC12CC2 O=S(=O)(c1ccc2[nH]c(=NCC(Cl)(Cl)Cl)ccc2c1)N1CCC(CCO)C1 N1(C(c2c(C)c(F)ccc2N)=O)CCC2CN(C(c3cccn3C)=O)CC2CC1 C(=O)(C(C1=CCSC1)N1CCCCCCC1)NCCN1C(C)CCCC1C C(=O)(CC(C)C(C)(C)NC(C1CCC2CC12)=O)NC1(CC(C)C)CC1 N1(CC(N2C(CC)C(NC(c3cc(C)sc3C)=O)CC2)=O)CCC(=O)NC1=O C(=O)(CC(C)CC(C)C)N1C(C(N(c2cccc(C)c2)C)=O)CSC1 C(=O)(CCCC(F)(F)CO)NC(COC)CNC(c1c[nH]nc1-c1cccs1)=O C(=O)(C(F)C(F)(F)F)N1CCN(C2CN(C(c3ccccc3OC3CC3)=O)C2)CC1 N1(CCC(N2CC(CCNC(=O)CCc3cn[nH]c3)(OC)C2)=O)CCC(O)CC1 c1(SCCC(N2CCC(F)(F)C(F)C2)=O)nc2ccccc2o1 C(=O)(C1=C(C)OCC1)NC1C2CN(C(c3cccc(SCCCC)c3)=O)CC21 C#CC1(C(N2CC(Cc3cccs3)C2)=O)CN(C(=O)Cc2ccc(Cl)cc2)C1 C1(C(=O)NC2C(NC(C3CC(OC)C3)=O)CCCC2)Cc2ccc(F)cc2O1 CC1CN2CCN1C(C(N1CCCCC(NC(=O)C(C)(F)F)C1)=O)C2 n1(CC)nccc1C(=O)NCC(C)(C)NC(C1CC1NC(=O)OC(C)(C)C)=O n1(CC)cnc2nc(N3CCC(c4ccco4)C3)nc(N(C)CC3CC(F)(F)C3)c12 N1(C(CCc2onc(C)n2)=O)CCC(C)(CNC(=O)C(C)C2(O)CCC2)CC1 C1(C(N2CC(O)(CN(C(=O)C=Cc3nccs3)C)C2)=O)CCC2(CCOCC2)C1 N1(C(=O)C#CC2CC2)C2CC1CN(C(=O)C(c1cccc(Br)c1)O)C2 c1(C(=O)NC(c2c(CC)cccc2)CNC(=O)C2=CSCS2)ccc(=O)n(C)c1 CCCCC(O)C(=O)N1CC2CC2(CNC(=O)C(C)NC(C2CCCC2)=O)C1 c1(CNC(c2n(CC=C)nnn2)C2CC2c2ccsc2)ccnc(CO)c1 CCC(C(=O)NC1CC1c1ccoc1)N(C1CNC(=O)C1)C(=O)OC(C)(C)C CCCC(C(=O)NC1CCCN(C(=O)Cn2cc(C3CC3)nn2)CCC1)C(C)C C(CC(C(=O)N1CC(CCCN(C)C)C1)NC(=O)CCNC(=O)CO)=CC C1(NCCCCn2nc(C)cc2C)CC2CC1CN2C(=O)NCCSCCCC N1(C(C=CC=CC)=O)CC(C)CN(C(=O)CCc2ccccc2Br)C(C)C1 n1(CC(=O)NC2CC2NC(=O)Cn2cc(Br)cn2)cccnc1=O c1(C(N(C(C)C)CCNC(=O)CC2C=CCC2)=O)ccncc1N1CCCC1 C1(C(=O)NCc2ccc(C(=O)NC(C)CCN(C)C)o2)C2CCC(F)(F)C12 C1(NC(c2nc(C)c(C)s2)=O)(CO)CCCN(C(c2csnn2)C)C1 c1(COC)nc(C(N2CCOCC2Cc2cn(CC3CC3)nn2)=O)c(C)o1 c1(C(N2CCC(NC(Cc3nnc(C)o3)=O)C(F)C2)=O)c(Cl)cc(Cl)nc1N C1(C(=O)N(CC)CC2CCN(C(=O)CSCCC(C)C)CC2)(OC)CCOCC1 c1(C(N(CC(CC)NC(C2OCCC2C)=O)CC)=O)ccc(N2CCC2)nc1 N1(C(C=CCN(C(C(CCC)(C)O)=O)C)=O)CC2(CNC(=O)C2)C1 c1(C(N)=O)ccc(C(N2CC(CNC(c3sccc3C(F)F)=O)C(O)C2)=O)cn1 C#CC1(N(C(C)C(=O)N)C(=O)C2CC2)CCN(C(=O)CN)C1.C1(OC)CCCOC1 CC1CN(S(C)(=O)=O)CCN1N(C)C1CCC(C2CNC(=O)CC2)CC1 c1(CC)sccc1C(N1CC(CCNC(=O)CC2CCOC2)(OC)C1)=O N1(C(C2CC(C)SCC2)=O)CCC(O)(CNC(=O)C2=C(Cl)CC2)CC1 CCCC(CCC)=CC(N1CCC(O)(CCNC(c2ccc(F)cc2)=O)C1)=O N1(C(C2N(C(CCc3ncn(C)c3)=O)C3(CC2)CC3)=O)CCC2(CC1)CC2C#N N1(C(C=CC(C)NC(C2CCC(F)CC2)=O)=O)CCCCC2(CCC2)C1 C(=O)(C1=NN(C2CC2)C(=O)CC1)NC1CCCN(C(c2c(N)nccc2)=O)CC1F C12(CNC(C3(C#C)CCCC3)=O)CCC1CN(C(=O)C(C)(O)CC)C2 c1(CC(N2CCC(O)(CCNC(C3(F)CC3)=O)C2)=O)ccc(F)cc1Br C(N=c1nc2c(ncn2C(C)C)c(N(CC(C)C#N)C)[nH]1)c1c(C)nc(Cl)cc1 c1(C(=O)NCC(CN(C(C2(COC)CC2)=O)C)O)ccc2nsnc2c1 C(=O)(C(C)C1CC1)NCCOCC#C Cc1cc(Br)cc(Cl)c1C(N1CCCC(C(C)NC(C2(F)CC2)=O)C1)=O C12(C(N3CCC(N(C(c4cccc(N)c4)=O)CCO)CC3)=O)CCCN1CCC2 Cc1nc(-c2nn[nH]n2)ccc1NC(C1OCCNC1)=O.C(C(F)(F)F)SC1CC1 C(C)(CC(=O)NC1C=CCN(C(=O)CC(F)F)C1)(C(F)(F)F)N(C)C C1(CC)CN(C(c2occc2C2CC2)=O)CCCO1.c12cccnc1CNC2=O c1(C(=O)NCC2(C(=O)NCCCN(C)C)CC2)ccc2c(c1)C(C)(C)C(=O)N2 CC1COc2ccc(C(=O)NC3CCCN(Cc4cnc(N5CCC5)s4)C3)cc21 c1(C(=O)NC(C)CNC(=O)C(C)Sc2ccncc2)nnc(O)c2ccccc12 C(=O)(C(C)C(F)(F)C(F)F)NCCC1(O)CCCN(C(C(=O)NC(C)C)=O)C1 C(CCC(C)C(=O)NCC1CC(O)CN1C(=O)CCc1ccc(C)nc1)OC C(c1cccc(Cl)c1)=C(C)C(=O)NCC12CC1CN(C(=O)C(C)(C)c1cscn1)C2 c1(C(N(CCOCCNC(c2cc(C)no2)=O)C)=O)cccc2oncc12 N1(C(CC2CCC(NC(c3nn(C)nc3Br)=O)C2)=O)CCCC(F)(F)CC1 N1(C(c2c(C)nc(CCC)o2)=O)CC(NC(C2CN(C)CCN2C)=O)CC(C)C1 C(=O)(C1=CC2C=CC(C1)C2)N1C(C)CC(NC(CCCCCCC)=O)C1 c1(CNC(C2CCCC(NCc3cn(CCF)nn3)C2)=O)n[nH]c2c1CCC2 C=C1CCN(C(=O)C(=O)N(C)C)C(C(N2CC3CC(OC)C2C3)=O)C1 c1(CN2CCC(N(C(c3cc(CC(C)C)c[nH]3)=O)CC)C2)cccc2ccoc12 S(=O)(=O)(c1ccccc1F)N(c1ncnc(N(C)C)c1[N+](=O)[O-])C1CNCC1O c1(-c2cccc(CN(C)Cc3c(C)ccnc3)n2)cccc([N+](=O)[O-])c1 CN1CCN(C(C2CC(c3ccc(Cl)c(Cl)c3)(C(=O)O)C2)=O)c2ccc(Br)cc21 C1(N(C(=O)CCC2CCOC2)C)CCCCN(CC(C)C2CCC2)C1 C1(NC(C(=O)NCC)=O)CCCC12CCN(C(=O)Nc1n[nH]c3c1CC1CC31)C2 c1(OC)ccc2c(c1C(N1CC(OC)CC1CNC(=O)C=CCF)=O)CCC2 C1(C)(C(=O)NC(CC#C)CC)CCN(C(c2cnc(OC)s2)=O)C1 CC1C(=O)N(CC(=O)NC2CCCC23CN(C(C2CNC(=O)N2)=O)C3)C(=O)C1C c1(C(C)C)ccsc1C(=O)NC(C1CCN(C(C2(CC(F)F)CC2)=O)C1)C CCC(CC(=O)NC1CC(F)CN(C(c2ccc(C3CC3)o2)=O)C1)C(C)C C1(C(N(CC(C)SC)NC(C2CCN(CC)CC2)=O)=O)CC2CCC(C1)S2(F)F CC1CCN(C(=O)CC2(NC(C3CCCCN3C(=O)N(C)C)=O)CCC2)CC1 N1(C(c2nccc(C)n2)=O)CCC(NC(c2ncoc2C2CC2)=O)C(CO)C1 S(=O)(=O)(c1ccc(N2CCOC(C)C2)cc1Br)N1CCCC(C#N)C1 C1(CC(=O)NC2CCC(OCCC)CC2)N(C(C2CC2(C)CC)=O)CCC1(C)C n1(CC(=O)NCC2C3CN(c4ncccn4)CC23)nc(C(F)F)cc1CO CN1CCC(C)(NC2CC(CCNC(c3cccnc3)=O)C2)C1=O N1(C(CN(CCOC)C)=O)CCCC(O)(CNC(c2ncn(C(C)C)n2)=O)C1 C(C(O)(CNC(=O)C(C1(O)CN(C(c2ccc(CO)nc2)=O)C1)F)CO)OC C(=O)(C(C)(C)CN(C(=O)CC1(O)CCCCC1)C)NCC(C(=O)NC)C c1(CNCC2N(C(C3CCC(NC(C)=O)CC3)=O)CCCC2)cnc(C)[nH]c1=N C1(CCOC)CN(C(=O)C(C)Cn2ccnc2)CCN1C(=O)CN1CSCC1=O c1(OC(C)C)ccc(C(=O)NCCN2CCOC(c3ncco3)C2)nc1 Cn1ccc(C(=O)NC(C2CCCCC2)CNC(c2c[nH]nc2Br)=O)c1 c1(NC(C(CNC(C(COC)(C)OC)=O)C)=O)ccccc1SC c1(CCNC(N2CC(Oc3cn(C)nc3)C(O)C2)=O)ccc(Br)cc1C(F)(F)F Cc1cc(CC(N2CC(NC(c3ccc(N)c(N)n3)=O)CC(O)C2)=O)ccc1Cl N1(C(CSCC(C)C)=O)CCN(C(=O)Cn2cnc(C#N)n2)CCC1C c1(C(N2C(CNC(=O)CSCc3cscn3)CCC2)=O)cccc2ccnn12 C1(CN2C(C(=O)NC3CC(C(N)=O)C3)CCC2)CCS(=O)(=O)CC1 C1(NC(C2C(CCC)C2)=O)CN(C(=O)CC2CCOCC2)CC12CC2 Cn1nc(C(N2CC3C(C(=O)NN4CCCOCC4)C3C2)=O)ccc1=O c1(CN(C(C(=O)N(C)C)=O)C)cccc(CNC(C2CC3C=CC2C3)=O)c1 N1(C(C2CN(C(N)=O)C2)=O)CC2CCCC(N)C2C1.C1(=CC(=O)N)CCSCC1 C1(NC(C2(NC(C)C)CC2)=O)CCCCC12CCN(C(c1ccsc1NC)=O)C2 C(=O)(CCC(C)(F)F)N(CCCNC(c1cnc(SC)s1)=O)C(C)C Cn1ccc2c(C(N3CC4=C(C3)CN(C(C3C=CCCC3)=O)C4)=O)[nH]cc2c1=O c1(C(=O)NCCC2(OC)CN(C(C(CCC)CC)=O)C2)cnn2c1CC(C)CC2 C#CCC(C)(CC)C(=O)NC1CCCCC1NC(c1ccc(C(C)C)c(C)c1)=O C1(NC(C(COC)NC(C)=O)=O)CCC(C)N(C(c2n[nH]c(C)n2)=O)C1 N1(C(Cn2ncc(C#N)c2)=O)CCCCCC1CNC(C1CCC(O)C1)=O CP1(=O)CC(NC(=O)NC(c2ccc(Cl)cc2)CC(N)=O)C(O)C1 N1(C(c2ccc(Cl)c(I)c2)=O)CCC2C1CCN2S(=O)(=O)CCC(F)(F)F C1(O)(CN(C)C(C2CC3(CC3)CO2)=O)CCN(C(C2Cc3nncn3C2)=O)CC1 c1(C(=O)NCC2CC(NC(c3onc(CC)n3)=O)C2)cccc(F)c1OC(F)(F)F C12(C(=O)NCCCCC(C)NC(CNC(=O)OC)=O)CCCC1OCC2 c1(C(C)NC(N2CC(C(=O)OC(C)(C)C)C2)=O)n[nH]c(CCO)n1 C(C(F)(F)CN(C(=O)C(c1ccccc1)NC(=O)CCc1cscn1)C)OC Cc1cc(C)c2nc(N3CCCC3(C)C(=O)NC3Cc4ccccc4C3)sc2c1 c1(CNC(=O)NC(C2(O)CCNC2)C)nccc2ccn(C)c12 N1(C(CN(C)C)=O)CC(C(O)C(=O)NCc2cc[nH]n2)C1 C=C(C)C1OCCCC1C(N1CC(Oc2ccc(C(=O)OC)cc2)C1)=O N1(C(C(C)NC(c2ccncc2)=O)=O)CCC2CCC(C1)N2C(=O)C(=O)C(F)(F)F C(=O)(C(C)CCCC(C)=O)NCC(CCC)NC(=O)CS(=O)(=O)CCO C(CCCC(C)NC(c1nc(Br)sc1C)=O)NC(C(C)OC)=O c1(CN2C(C(N(C)Cc3nc(CC)on3)=O)CCCC2)cccc(C#N)c1 c1(C(C)=O)cn(C)nc1C(=O)NC1(CNC(c2cccc[n+]2[O-])=O)CCOC1 CCC(CC)CC(=O)NC(C)(CNC(c1ccnc(O)c1Br)=O)C(C)C C1(CC)CN(C(=O)C(c2ccc(Cl)nc2)(F)F)CCN1C(=O)C(C)C1(O)CCC1 N1(C(CN2C(C)CCCC2)=O)CCN(C(c2snnc2C2CC2)=O)C(CCO)C1 C1(NC(c2ccc(S(C)(=O)=O)o2)c2n(CC)nnn2)CS(=O)(=O)C12CCCC2 n1(CC)nc(C(=O)NC2CN(C(=O)C(C)CCOC)C2)c(Br)n1 C1(NC(C2(COC(C)C)CC2)=O)C=CCN(C(=O)C#CC(=O)N(C)C)C1 CC1(C)CN(C(=O)Cc2ccc(Cl)cc2)CC1CNC(C1CCCC2(CC2)C1)=O C(=O)(N=c1ccn(C2CC2)[nH]1)C1(CC)CCN(C(c2noc(CC)c2C)=O)CC1 CC1(CCC(=O)NC2CC(NC(=O)CC3CC4CCC3C4)C2)CCC(=O)N1 C(=O)(CCCC(C)NC(c1ccc(C#N)cn1)=O)NC1(c2ncc(C)o2)CC1 C1(OC)(CNC(=NCc2ccc(Cl)cn2)NCC(N2CCCC2)C)CCCCC1 N1(C(c2ncn(CC)n2)=O)CCOCC1CNC(C1CC1F)=O C1(C(N2C(CNC(c3cc(O)ccc3F)=O)CC2)=O)CC2CCC1CC2 c1(OC)ccc(C(N2CC(NC(C3(C)CCCN3C)=O)CC2(C)C)=O)nc1Cl CC1CCCC(N(C)C)(CO)C1.C123CC(CN(C1)C(=O)C=CC(C)(C)NC2=O)C3 N1(C(CCSCC)=O)CCC(NC(c2ccnn2CC2CCC2)=O)C(C)(C)C1 N1(C(C2C(NC(C(C)=C3CCCC3)=O)COCC2)=O)CCC(O)CC12CC2 c1(CC)onc(C(N2CC(C(C)(C)O)(CNC(=O)C(C)C3CCOC3)C2)=O)c1C N1(C(COCCCC)=O)CC2CCN(C(c3ccncc3C)=O)CC2C1 N1(C(=O)NCc2cncnc2)CCN(C(C2CCCC2)=O)C(c2cn[nH]c2)C1 C1(NC(=O)COc2cccc(F)c2)Cc2nccnc2C1 N1(C(c2ccc(OC(C)C)nc2)=O)CC(NC(=O)C(=O)NC2CC2)CC(C)C1 N1(C(C#C)CCC)CCC(C2CCOCCN2)CC1.c1(C2CNC2)ccccc1 c1(-c2n(CCC(C)C)nc(Cn3cncn3)n2)cc2c(F)cccc2[nH]1 c1(C(=O)NC2C(F)CCN(C(C(C)OC)=O)C2)sc2[nH]cnc(=S)c2c1C CCCC(C)(C)CC(=O)N1CC(C)CCC1C(=O)NCc1cc(CC)no1 C(C)(c1ccccc1C)=CC(=O)NC(C1CCN(C(C(C=CC)O)=O)C1)C N1(C(C(CC=C)CC)=O)CCCC(C2CN(C(c3ccnn3C)=O)C2)C1 C12(C(=O)NC3CCN(CCNC(C(C)OCOC)=O)CC3)CCC(CC)(CC1)OC2 Nc1c(F)c(F)cc(C(=O)NCC2CC2CNC(c2cnn(C3CC3)n2)=O)c1Cl n1(CCOC)cc(C(N2CCCC2)CNC(c2ccccc2)=O)nn1 c1(C(C(N2CCC(C)(CNC(CSCC#C)=O)C2)=O)C)ccc(F)c(F)c1 C1(C(N(CC=C)C)=O)C2CCN(C(=O)CN3CCCCC3)CC12 c1(NC(CNC(=O)NC(COC)C)(C)C2CC2)ccc(OC)nc1 Cc1nn(C)c(C(F)(F)F)c1C(=O)NC(CNC(=O)CC1CC2CCC1C2)CO C1(C(=O)NCCN(C(CCN(C(C)=O)C)=O)C)CC2(C1)NC(=O)NC2=O C(CCO)(CC(C)C)N(CCNC(c1cc(C(F)F)n(C)n1)=O)CC C1(OC)CN(C(=O)CCC2CCCC(O)C2)CC1NC(=O)CCSC(F)(F)F C1(NC(c2n(C)c(S)nn2)=O)CC2(C1)CC(n1cc(C3CC3CO)nn1)C2 C1(C(=O)NCC2(O)CC3CCC2O3)CN(C(=O)C=Cc2ccoc2)CC12CC2 c1(CN2C(C(N3CCC(CCCO)CC3)=O)CSCC2)ccc(Cl)c([N+](=O)[O-])c1 c1(CNC(C2C(CNC(C(CC)n3cncn3)=O)C2)=O)ccc(O)nn1 C=CCC(CNC(C1OCCC1C(C)C)=O)C(=O)Nc1cncc(N(C)C)c1 C1(C(=O)NCCC2CN(C(C3C(CC(C)C)C3)=O)C2)CC2CCCCC12 CCCC(C(=O)OC)C(=O)NC1CCCCC1C(N1CCC12CC(O)C2)=O c1(OC)cccc2cnc(NC(C3(C)CCCN3Cc3cccc(F)n3)=O)nc12 C1(NC(CCNC(C)=O)=O)CN(C(=O)C=CCO)CC2CCCC12.C(=O)(C(C)C)N C1(NC(c2nc(C(C)OC)oc2)=O)CCCC12CN(C(=O)CC1CSC1)C2 c1(CC(=O)NC2CC(NCc3ccc(F)cn3)C2)cccc(C(F)(F)F)c1 CS(=O)c1ccc(-c2cn(C3C4CC(O)C(C4)N3C(=O)CC(N)=O)nn2)cc1 C1(C(=O)NCCc2cn(CCCCC)nn2)CCC2C(CC1)C2(F)F c1(C(N(CCCCNC(c2ccn(C)c(=O)c2)=O)C)=O)ccnc2c1nnn2C CC(C)C(CNC(C1(C)CC1(Cl)Cl)=O)NC(=O)C(n1cc(Cl)cn1)C c1(C(=O)NC2CC(C(N(C)CC3C(C)OCC3)=O)C2)cnc(N)cn1 C1(CN=C(NCC(C)OCC)NC2CCCC2)CCCC2(CCC2)O1 C1(C(=O)NC2(c3ncc(C(=O)OC)s3)CC2)CC2CSCC(C1)C2 N1(C(CC(C=C)(C)C)=O)CCC(C(=O)NCc2cnc(C)[nH]2)C(C)(C)C1 C1(c2n(CCOC)nnn2)(NCCCF)CCOC(CCF)C1 N1(C(CC2C(C)CCN(C(c3cc(CC)ncn3)=O)C2)=O)CCC2(CCCC2)C1 c1(C(=O)NC2C(NC(C3(C)CCCS3(=O)=O)=O)COCC2)nnn2c1CCCC2 C#Cc1cc(F)c(C(N2CC(CCNC(=O)CC3(N(C)C)CC3)C2)=O)c(F)c1 c1(CC)[nH]ccc1C(=O)NCC1CC1CNC(=O)Cn1cnnc1 c1(CC(C)N(CCC)C(=O)NCc2ccc(Cl)o2)cccc(F)c1 Cc1nc2c(s1)CCCC2C(=O)NC1CN(C(=O)C(=O)Cc2ccccc2)C1 c1(OC)ccc(C(N2CCOC(CNC(C3CCCN3C(C)C)=O)C2)=O)c(F)n1 C1(CNC(c2ccccc2N2CCCC2=O)=O)CN(C(=O)C(F)F)C2CC12 N1(C(CN(C(Cc2c(C)cnn2C)=O)CCO)=O)CCNC(=O)CC1C C1(SC)CC(NC(=O)CNC(=O)COCCF)C1(C)C CCC(C)CC(C)C(=O)NCCCCCCNC(=O)Cc1ccc(C)cc1Cl Cc1cc(C(=O)NCCCC(C)(C)NC(c2cc(CCCO)on2)=O)ccc1Cl C1(NC(c2cn(C3CCCC3)nn2)=O)CCCN(C(c2ncccc2Br)=O)CC1 c1(NC(Cc2cccc(C)n2)=O)ccc2c(c1)CN(C(=O)C(O)CC(C)C)CC2 N1(c2n(CCCCCNC(C)=O)nnn2)C2CC=C(C(=O)O)C1CC2 C1(C(=O)NC2CCOC(C(=O)NCCc3ncccn3)C2)CC2C(C1)C2(F)F CC(C)(CNC(=O)CCNc1ccsc1)C1CCCC1 C1(NC(c2cnc(C(C)=O)s2)=O)(CNC(=O)CSCC(N)=O)CCC(C)(C)CC1 N1(C(c2ncccn2)C)CCC(NC(=O)CC2NC(=O)NC2=O)C(C)C1 c1(C(N2C3(CNC(c4cnc(C)[nH]4)=O)CCC3CC2)=O)nn2c(c1C)OCCC2 C(=O)(CCCC(F)F)NCC1(CO)CCN(C(C(C)SCC)=O)C1 Cn1nncc1C(=O)NC(CNC(c1cn(CC(F)(F)F)nn1)=O)CO C=C1CN2C(=O)CCC2(C(=O)NC2CC2CNC(c2sccc2Cl)=O)C1 N1(c2[nH]c(=NCc3cc(C)c(Br)cn3)cc(C)n2)CCCCC1[Si](C)(C)C c1(CC(=O)NC2C(NC(c3c(C)nc(CC)s3)=O)CC2)ccc(O)c(C)c1 c1(C(N2CCCC2c2nccs2)=O)c[nH]c(=NC2CC(c3ccc(Cl)cc3)C2)cn1 c1(C(=O)NCCC2N(C(C(C(=C)Cl)(C)C)=O)CC(F)(F)C2)cc2ncccc2s1 c1(C(=O)NC2CCN(C(CC(C)OC)=O)C2)ccc(C(C)C)c([N+](=O)[O-])c1 c1(C(=O)NCC(CN(C(C(N2CCSCC2)C)=O)C)O)ccc([N+](=O)[O-])s1 c1(C(=O)NC2CCC(NC(C3C(C)(Br)C3)=O)CC2)cc2c[nH]cnc-2n1 C1(CC)CC(C(=O)NCC2(C(F)F)CCN(C(=O)C(C3CC3)C3CC3)C2)CCO1 N1(C(Cc2nc(C)[nH]n2)=O)CCCC(NC(=O)Cc2nc(C)c(C)s2)C(F)C1 N1(C(C(CCCOC)C)=O)CCC(O)(C2CCN(C(c3ccc(Cl)[nH]3)=O)CC2)C1 c1(OC)cc(C(=O)NC2(CNC(C3CCC34CCC4)=O)CC2)cc(C)n1 N1(C(C2CN(C(=O)CCCc3ccc(F)cc3)C2)=O)CCc2nc(OC)sc2C1 C(N=c1[nH]c(=NCCCn2ccnc2)[nH]c2c1COC2)c1c(OC)cc(Cl)cc1 N1(C(C(C(C)C)(C)O)=O)CCCC2(C1)CN(C(C1CCCCC1)=O)CCO2 c1(CC)cccc(C(=O)N(C)CC2(O)CCCN(C(C3CC3C3CC3)=O)C2)c1O Cc1nc(N2CC=CC(NC(c3cnccc3Cl)=O)C2)ncc1[N+](=O)[O-] c1(C(N(C(C(=O)OC)C)C)=O)ccnc(CNC(=O)CC(C)C2CC2)c1 c1(CNC(C2CCC(NC(C(CCC)NC(C)=O)=O)C2)=O)ccn(C)c(=O)c1 c1(C(N2CCC(C(C)NC(C(CC3CCCC3)OC)=O)C2)=O)ccc(C#N)cc1 C1(OCc2cn(C)nc2)CCCCC1NC1(c2nnnn2C)CCOC1C c1(-c2cccc(C)c2)ccc2sc(NCc3ccc(O)nc3)nc2c1 c12cccc(c1)OCC=CC1(COC1)NC2=O.c1(NCC2CCOC2)cc(Br)ccn1 c1(CC(N2CC(CCNC(CN(CCOC)C)=O)OCC2)=O)ccc(F)cc1Cl N1(C(C2C(CC)CCC2)=O)CCCC(CCNC(=O)CCc2cccn2C)CC1 CC(C(=O)NNC(=O)OC(C)(C)C)SC1CC2COCC12 C1(NC(C(CC)C)=O)CCN(C(c2c(C#N)cnn2C)=O)CC1(C)C C1(C(N(C)CC2CCC(C)CC2)=O)CC2(CCN1C(=O)C(O)c1ccco1)CC2 Cc1ncsc1C=CC(=O)NCC1COCCN1C(=O)Cc1ccc(Cl)cn1 c1(C(N2CCC(CCCCCNC(CC)=O)CC2)=O)ccc(C#N)c(O)c1 C(=O)(CC(C)(C)C)N(CC(C)NC(c1n[nH]cc1Cl)=O)C C1(C(CO)NC(C2(OC)CCOC2)=O)CCN(C(c2cn(C)cc2C)=O)CC1 C1(NC(c2c(CC)ccs2)=O)CCCC(NC(c2coc(C(C)OC)n2)=O)CC1 C1(CNC(c2c(C)nc(C)[nH]2)=O)CC2CCC1N(C(c1cccc(O)c1)=O)C2 c1(C(=O)NC2CCC(NC(c3cnn(C)c3F)=O)C2)ncnc2c1CCC2 C1(C(N2CC(N(CC=C)C)C2)=O)N(C(=O)C(O)CSC)CC12CCCC2 c1(C(=O)OC)cccc(Cl)c1NC(C1CC(C)CN1Cc1cnc(OC)c(C)c1)=O CC(O)C(F)(F)C(=O)N1CC(O)(CCNC(=O)C(F)(F)C(O)C2CC2)C1 C1(C(=O)NC2CC(F)(CNC(c3cnc(C)o3)=O)C2)CCn2ccnc2C1 C(=O)(CCC(C)(C)C)NCCCOCCNC(c1scc(NC(C)=O)n1)=O C(=O)(C(C)(C)CNC(C1CCN(C(c2ncccc2O)=O)C1C(C)C)=O)OC Cc1cc(NC(C2CC2NCc2ccc(CO)cc2)=O)cc(C)c1I C1(C(N2C(C=C)CCC2)=O)(NC(c2cc(NCC)nn2C)=O)CCC(C)(C)C1 C12(C(=O)NCC(C)N(C(=O)Cc3ccccn3)C)CC(C(F)(F)F)C1C2 c1(C(=O)NCCC2(C(=O)NCCn3ccnn3)CC2)c(C(F)(F)F)cccc1Cl C1(CCN(C(CCC#C)=O)C)CCCCN1C(C1CC(OC)(OC)C1)=O C1(C(N(CC(C)C(=O)NCCCC2(C)CC2)C)=O)CCCOCC1 N1(C(c2ccc(CC)s2)=O)CC2CCOC2(CNC(=O)C=CC(C)CC)C1 C1(NC(CNC(=O)NC)=O)CN(C(C2CCC2NC(=O)C(F)(F)F)=O)CC12CC2 CCCCC(O)CC(=O)N(C(C)CCNC(c1cc(C(=O)C(C)C)c[nH]1)=O)C C1(NC(=O)C(c2ccccc2)C2CC2)CN(C(=O)CCCNC(N)=O)CC12CC2 C1(C2(O)CCN(C(c3cc[n+]([O-])cc3)=O)CC2)(NC(C(CC(C)C)F)=O)CC1 c1(-c2ccc3nc(C)sc3c2)ccc2c(c1)CC(=O)N(C)C2 C1(CC(=O)NCCOC2CCN(C(=O)CC3CCC34CCC4)C2)CC2(CCC2)C1 c1(SC)cc(F)ccc1C(N1CC2(NC(=O)Cc3cncn3C)CCC1C2)=O c1(N(CC(N2CCN(C(=O)C=Cc3ncc[nH]3)CC2)=O)C)ccnc2ccccc12 C(CCC(=O)NCCC(C)CCO)(C(C)C)NC(c1cc(OC)ncc1)=O c1(CC(N2C3CN(C(c4[nH]cc(CC)c4)=O)C(C3)C2)=O)ccc2nc(O)[nH]c2c1 CCCC(C)(C)CC(=O)NC(CC(=O)N(CC(c1nn[nH]n1)C)C)C(C)CC CCCCC(C)CCC(=O)N1CCCC(O)(CN(C)C(C2(CC)CC2)=O)C1 N1(C(C=C(CC)CC)=O)CCOC(C2CN(C(=O)CC(O)CC)C2)C1 C1(CNC(C2C(C)(C)C2(C)C)=O)CCCC12CCN(C(C1CCSC1)=O)CC2 C12CC(C)CN(C1)C2=O.c1(OC)cccnc1N1C(=O)CCC1=O.C1(C)C(=O)N1 C12(NC(C3=CC(C)(CC)C3)=O)CCCC1(F)CN(C(=O)CNC(=O)NC)C2 c1(C(N2CCNC(=O)C2CC(C)C)C(=O)NCCOC)cc(C#N)n(C)c1 c1(C(=O)NC2(C)CN(C(C3C(CCOC)C3)=O)C2)ccc2occ(C)c2c1 C(=O)(CC(O)CNC(c1ccc(CNC(=O)C=CCF)s1)=O)OC c1(CC)nc(C(=O)N(CCNC(C2CCCC2C)=O)CC)co1 N1(C(=O)OC(C2(NCC)CC(F)C2)=O)CCCCCC1 C1(C2(O)CN(C(C3CCCC(O)C3)=O)C2)(CNC(c2ccc(N)cc2F)=O)CC1 CC1(C)CCC(C)(NC(=O)CC2CN(C(C3CC(=C4CC4)C3)=O)C(C)(C)C2)CC1 c1(COC)cc(C(N2CCCC2C(C)NC(c2cc[nH]c2C)=O)=O)c(C)o1 NC1CCCS(=O)(=O)C1CC(=O)N(CCCN1CCCC1)Cc1cccs1 N1(C(c2c(OC)cc(N)cc2)=O)CCN(C(=O)CC(C)(C)OC)C(C)C1C C1(C2CCCN(C(=O)CCn3ccnn3)C2)(NC(C(COC)C)=O)CC1 c1(NC(C(=O)NC(c2nn[nH]n2)C)C(C)C)ccc(N)cc1-c1ccccc1 C1(F)(C(=O)NCCOC(CC)CC)CN(C(=O)CCc2cnoc2)C1 C(C(C)(C)C(=O)N1CCC(N(C)C)C1)N(C)C(C1CCCO1)=O CCCC(C)(C)CC(=O)N1C(C(=O)NC2CC(=O)N(C3CC3)C2)CCC12CC2 Cc1ccc(C=CC(N2CC3CC(C2)C3NC(c2nccn2C)=O)=O)c(C)c1 Cc1ccc(C)c(SCCC(=O)NC2CN(C(C34CCC3C4)=O)CCC2F)c1 C1(NC(=O)CCCCCl)CCN(Cc2cnco2)C12CC2 C1(CNC(C=CC(C)(C)NC(C2C(=C)C2)=O)=O)CC12CCCCC2 c1(C(=O)NCCC(C)NC(C2CCC(=O)N2C2CC2)=O)cc([N+](=O)[O-])cnc1N N1(C(C2N(S(C)(=O)=O)CCC2)=O)CC2=C(C1)CN(C(=O)C(C1CCOCC1)F)C2 c1(C(=O)NC(C(C)NC(C=CCC)=O)CO)cc2c(=O)cc[nH]c2s1 c1(C(=O)NC2(CCC(=O)Nc3cccc(SC)c3)CCCC2)[nH]ccc(=O)c1C C=CCCCC(C(=O)NCc1sc(C)nc1C)NC(=O)Cn1ncn(C)c1=O C1(NC(C2N(C(=O)OC(C)(C)C)CCC2)=O)CCN(C(=O)C(O)C2CCC2)CC1 N1(C=O)C(C(N2CC(C(=O)OC)C2)=O)CC1C.C1(CCOC)(COC)CC1 CC(CCNC(=O)Cc1cccc(F)c1)CCNC(=O)CSc1nc[nH]n1 C1(CC(=O)NCCNC(C2(c3ccccc3)CC3(CC3)C2)=O)CC(O)C12CCC2 [SH](=O)(=O)c1cc(C)c(Cl)c([N+](=O)[O-])c1.CCCCC(=O)OCCOCCNCCOCC c1(CN(C(CCCC)C(=O)Oc2ccccc2C)C)cccc2cncn12 c1(OC)cccc(=NC(=O)C2CCN(C(=O)CCCCOC)CC2)[nH]1 N1(C(C2CCN(N(C)CCc3ccco3)C2)=O)CCCCC1.C1(C=O)CCC1 c1(OC)cc(C2CCN(CC3CC3)C2)ccc1C.c1cccc(Cl)c1 C1(C(=O)O)CC2(CCCCC2)C(=O)O1.CN1CCC2(CC1)NC(=O)NC2 Cc1c(C(N2CCC(C)C2CNC(=O)C(c2ccc(F)cc2)(F)F)=O)ncn1C C1(C(=O)NC2CC3(CN(C(COCCSC)=O)C3)OC2)CC(C)(C)CC(C)(C)C1 C1(CNC(CN(S(CC)(=O)=O)C)=O)CCN(C(=O)Cc2cc[nH]c(=N)c2)CC1C C(CCCC(=O)NC1(CCNC(c2cc(C)cc(Cl)c2)=O)CCC1)(OC)OC C1(C2CC2)(C(=O)NC(c2nccc(O)n2)C)CN(C(c2n[nH]cc2[N+](=O)[O-])=O)C1 c1(C(=O)NCC#CCNC(C2OCCN(C)C2)=O)ccc(=O)n(-c2cnn(C)c2)c1 N1(C(C(c2cccnc2)C)=O)CCC(C(C)C)CC1CNC(=O)C(C)CC1CC1 C(CC(O)C(=O)NC1CCCC1NC(c1cnoc1-c1ccccc1)=O)N(C)C c1(SC)cc(F)ccc1C(=O)NC1(C(O)CO)CC1.C12CC3(CC(C3)NC1=O)C2 c1(OCC)cccc(C(N2CCC(CNC(=O)C(O)CF)(CO)C2)=O)c1 N1(C(C)=O)CC(NC(=O)CCC2CC2(Cl)Cl)C2(CCC2)C1 c1(C(N2CC(NCC(C(=O)OC)C)C3(C2)CC3)=O)cc2c(Cl)nccc2s1 C#CC1CC2(CC2)CN1C(C1CC2CCC(C1)N2C(C1CCSCC1)=O)=O C1(NC(CC(C)NC(N)=O)=O)CN(C(=O)CC(C)(C)c2ccccc2)CC1F C1(CNC(C(CCC)CC)=O)CN2CCCCC2CN1C(C1CCCC1)=O C1(NC(C(OC)OC)=O)CC2(NC(c3cccc(F)c3Br)=O)COC1C2 C(=O)(C#CC1CCOC1)N1CCC(CC)(NC(c2cc(C(N)=O)c[nH]2)=O)CC1 c1(CC)ccnc(C(=O)NCCCN(C(c2n[nH]c(O)n2)=O)CC)c1 c1(C(=O)NC2(CNC(C3CC4(CC(=O)N4)C3)=O)CC2)ccn2ccnc2c1 CC1CC(=O)CCC1C(=O)NC1CC(C)N(C(=O)C=CC2CC2)C1 N1(C(C2(OC)CC(CF)C2)=O)CC(NC(c2cc(C)nc(O)c2)=O)C2(CC2)C1 Cc1nc(CCC(=O)NCCNC(=O)CC2CC(CF)C2)c2c(C)c(C)sc2n1 C(CCC(C)C(=O)N1CCC(NC(c2ccnc(NCCO)c2)=O)C(C)C1)OC C(=O)(CC(O)CC(C)(C)C)NCC1N(C(C2(CC)CCNC2=O)=O)CC(F)C1 c1(C(N2C(CNC(C=C(CCC)CCC)=O)CC2)=O)ccc(C2CC2)nc1O c12nc(-c3nccs3)nn1CC2.c1(SCCN(N2CCOCC2)C)nncn1C c1(C(=O)NCCOCCNC(C(CCCC)C)=O)ccc(C(C)=O)cc1Br c1(C(C)=O)ccc(C(=O)NC(CC2CCC2)C(=O)NCCCS(C)=O)o1 C1(NC(C2C(C)(C)C2C(F)F)=O)CC2CCC1N(C(c1cccc3c1OCC3)=O)C2 c1(NC(C2C=CC(NC(c3nc(C)sc3C)=O)C2)=O)ccc2ncnc(O)c2c1 N1(C(C(C)=C(C)C)=O)CSCC1C(=O)NCCCCO Cc1nccc(Cl)c1C(=O)NCC1(CNC(C2CCC(C)CO2)=O)CC12CCC2 c1(C(N(C(C)C)CCNC(=O)CC2CCCC(=O)N2)=O)cncn(C)c1=O Cc1cccc2oc(C(=O)NC3CN(C(=O)CCC4CCC4)C3)cc12 N1(C(CC(C)(C)OC)=O)CCC2CC2N(C(c2c(C(C)C)cnn2C)=O)CC1 C1(C(=O)NCCCN(C(C(C)N2CCCC2)=O)CCO)CCOC(=O)CC1 c1(C(=O)NC2CCN(C(c3n(C)c(S)nn3)=O)C2)cc(F)cc([N+](=O)[O-])c1 N1(C(c2n(CC)ccn2)=O)C2CCC(C2)C1C(N1CCCC(CCO)C1)=O c1(CN(C(C)=O)C)n[nH]cc1C(=O)NC(C)C(c1ccccc1)C c1(C(N2CCC(CNC(C(c3ccn(C)n3)C)=O)CC2)=O)ccc(S(N)(=O)=O)o1 c1(CSCCC2C(=O)OCC2)cc(C(F)(F)F)ccc1O CCCC1CNC(=O)C2(CCC2)CC2CC(C2)CNC1=O.N(C)(C)CC1CC1 C1(C(C(=O)CC2CCN2C(=O)C=CCOC)=O)(CC)CCCCC1.C(C)(C(C)C)N c1(C(N2CCCC(CCNC(c3c(CC)cno3)=O)C2)=O)nccc(C)c1F C(=O)(N=c1[nH][nH]c2nc(C)c(C)cc12)c1cccc(S(=O)(=O)NCCC)c1 C1(NC(CS(CC)=O)=O)CC2(CCC(NC(=O)CC3(OC)CC3)CC2)C1 c1(C(N2CCC(NC(c3cnc(C)s3)=O)(CF)C2)=O)sc2cncn2c1C c1(OC)ccc(F)c(C(=O)NC2CCCCC2NC(C2(CCN(C)C)CC2)=O)c1N C1(CCCNC(C(C)(C)c2cscn2)=O)CCN(C(=O)CC2(C#N)CC2)CC1 N1(C(C(C)n2cnnn2)=O)CCC(NC(c2nccc(C(F)F)n2)=O)C(C)(C)C1 C1(C)(CC)NC(=O)N(CC(=O)NC2CC(CCNC(c3cnn[nH]3)=O)C2)C1=O C(=O)(C1=NOC2(CCC2)C1)N(CC(C)CNC(=O)CCNC(c1ccco1)=O)C C#CCC(C(=O)NCC1CC1CC(=O)NCC(CO)C(C)C)C1CC1 Cc1cc(C(N2CC(NC(=O)Cn3ncc(Br)n3)C3(CC3)C2)=O)cc(C)c1N N1(C(C(C)Cc2cnc[nH]2)=O)CCCOC(CNC(=O)C(C)(C)N2CCCC2)C1 c1(CC(N2CC3CCN(C(C(=Cc4cccs4)C)=O)CC32)=O)ccc(S(C)=O)cc1 c1(C(=O)NCC2C(NC(C=C(COC)C)=O)C2)c(C(F)(F)F)n[nH]c1C C(=O)(C1=NNC(=O)CC1)NC(C)CSC.C(C(F)C(=O)NCCCCCC)N(CC)CC c1(C(=O)NCCCCC2CN(C(=O)CN3CC4CC4C3)C2)coc(C(F)(F)F)n1 N1(Cc2c(C)ncs2)CC2CC1CN2C(=O)CN(CC(C)(C)C)C N1(C(C2CN(C)CC(C)O2)=O)CC2CCCC(C1)N2c1cncc(C#N)n1 CC(CF)CC(=O)NCC1CCC(NC(c2csc(COC3CCC3)n2)=O)C1 c1(CNC(C)COc2cccc(Br)c2)ccc2ncc(Br)cc2c1 C1(OC)CN(C(=O)CSC(F)F)CC1NC(c1cc(C2(C)CC2)n[nH]1)=O c1(OC)ccc(C(=O)NCCN(C)C(C2C(c3ccccc3)C2(F)F)=O)c(F)n1 S(=O)(=O)(c1c[nH]c2cc(Cl)ccc12)N1CC2C(NCCC)C2C1 c1(C(=O)NCC(CC)NC(C2C3CCC23)=O)ccncc1Oc1ccccc1 c1(C2N(C(N3C(C(F)F)CC(C)C3)=O)CCC2)ccnc2cc(Cl)ccc12 O=C(C(O)Cc1ccccn1)NCCN(C(=O)Cn1nccc1C1CC1)C1CC1 c1(-c2ccc(C(=O)Nc3c(C)cc(F)cn3)nn2)ccc2c(c1)CC(=O)N2 c1(C(N2CC(NC(CNC(CC)=O)=O)C(C)CC2)=O)cc(S(C)(=O)=O)co1 C1(CNC(c2c(CC)cns2)=O)N(C(=O)CC2CCCOC2)CCCC1(C)C N1(C(COCCCC#C)=O)CC(C(=O)NCc2oc(C)nc2C)C(F)(F)C1 CC(C)CC(C(=O)N1CCC(CNC(C2(C)CCCN(C)C2)=O)C1)C(N)=O N1(C(=O)COc2ccc(Cl)cc2)CCCC(C2CCN(c3nncs3)C2)C1 C(=O)(C1=Cc2ccc(Cl)cc2OC1)NC(C)CCCCNC(=O)C1=CCCS1 c1(CNC(C(C)C2CCC2)=O)nc(CNC(c2ccc(Cl)cc2N)=O)cc(O)n1 N1(C(C(CC)n2ccnc2)=O)CC(NC(C2CC(OC)C2)=O)C(C)C1 C1(NC(COC2CN(C(CC)=O)C2)=O)CCOC2(CCCC2)C1 c1(C(N(C)CC2CN(C(CCCOCC=C)=O)C2)=O)ccc(O)cc1Cl c1(C(=O)NCC2CN(C(C3CCC(F)C3)=O)CCO2)cccc(C#CCO)c1 c1(C(=O)NCCN(C)C(C2CC2(C)C(F)(F)F)=O)cccc2c1OCC2(C)C c1(C(=O)NC(CNC(C(C)(C2CC2)NC(C)=O)=O)(C)CO)ccn(C)c(=O)c1 N1(C(C2CCN(C(COC)=O)C3C2OCC3)=O)CCCc2ccccc2C1 c1(NC(C(C2CCN(C(C3CCCS3)=O)CC2)C)=O)ccc2ccncc2c1 c1(C(=O)NC(CNC(c2c(C)n[nH]c2)=O)C(C)(C)C)ccc2c(c1)CC2 c1(CCOC)nc(CCN(S(C)(=O)=O)C(C)C)nn1-c1ccc(Cl)cc1 C1(CC(=O)NCC(CNC(CN(CCOC)C)=O)(C)O)N2CCC1CC2 C1(CNC(C2CC2F)=O)CC2(CCC2)CN1C(c1c[nH]ccc1=O)=O CC(O)C(C(=O)N(CC(C1CCCC1)O)C)NC(c1cccc(CC#N)c1)=O Cc1cccc(C(N2CCC(F)(C(=O)N(CCC3CCCN3C)CC)CC2)=O)c1I Cc1cc(F)cc(Cl)c1NC(=O)C(N1CCCC1CNC(=O)OC(C)(C)C)=O c1(C(=O)OC)cc(C)n(CC(N2CC(CNC(=O)CC(C)C)CC2C)=O)n1 Cc1cc2cc(NC(NC3CCc4ccc(F)cc43)=O)ccc2n1C C1(F)(C(=O)NC(C)C(C)n2cccn2)CCN(C(=O)CC2CCC=CCC2)CC1 C1(O)(CNC(C(C(C)C)O)=O)CCCN(C(C2CCC(O)CC2)=O)C1 Cc1ccc(NS(=O)(=O)Cc2coc(C)n2)c(OC2CCCCC2)c1 C(=O)(C1=CCS(=O)(=O)C1)N(CCC(C)NC(=O)Cc1nncn1C)C Cc1cc(C(=O)NC2CCC(NC(=O)C(F)CC3CCC3)C2)cc(Cl)c1Br S(=O)(=O)(c1ccccc1[N+](=O)[O-])NCCCC=C N1(C(c2c(C)n(C)nn2)=O)CCN(C(=O)CCNc2ccccn2)C2CC12 C1(C(N2CC(CC(F)(F)F)C2)=O)CCCCCN1C(=O)CC1CC2(CCC2)C1 C1(C(N(CC#C)CCOC)=O)(NC(=O)Cc2ncccc2F)CCN(C)C1 N1(C(C(C)N(C(C(CC)COC)=O)C)=O)CC2CCC(C1)O2 Cc1ccc(C(=O)Nc2cccc(NC(C3(C(F)(F)F)CCC3)=O)c2)cc1 C1(C(=O)NCC(C2CC2)OC)(NC(COCCC=C)=O)CCCC1C CC(CCC(=O)N(CCCNC(c1cc2n(n1)CCC2)=O)C)S(C)(=O)=O N1(C(COC(C)C)=O)CCOC2(CCN(C(c3nc(C(F)(F)F)cn3C)=O)C2)C1 Cc1cc(CNC(=O)C(=O)NCc2n[nH]c(=N)o2)[nH]n1 c1(C(=O)NCC(C)N(C(c2c(CC)cno2)=O)CC)ccc2ccncc2n1 C1(C)(NC(=O)Nc2nnn(Cc3nc(C)sc3)c2C)CC(C)OC(C)C1 C1(OCCCCOC)CCCN(C(C2C(CNC(=O)OC(C)(C)C)C2(C)C)=O)C1 Cc1ncc(C=CC(=O)NC2CC(CNC(=O)C=Cc3cc[nH]c3)C2)s1 c1(NC(N2CC(OCCCc3cccc(C)c3)C2)=O)c(Cl)cc([N+](=O)[O-])cc1Cl c1(CC)cc(C(=O)NC2C=CC(CNC(C3CCCS3)=O)C2)ccc1O N1(C(Cc2cn(C)nc2)=O)CC2CCCC(NC(C3CSCCS3)=O)C2C1 CC(C)(CNC(c1n[nH]cc1-c1ccncc1)=O)CNC(C1(C)CC1(F)F)=O C#CCC(C)(C(=O)N1CCCC(OCC)C1)NC(=O)C=CC1CCCCC1 CC1CCCC(O)(C(=O)N(CCCNC(=O)CCOc2ccccc2F)C)CC1 C(CCN(C)C(c1cc(C(N)=O)ccc1F)=O)(C(C)(C)C)NC(C=C(C)C(F)F)=O Cc1cc2ccnc(C(=O)N(C)C(c3ccc(C(C)C)cc3)C)c2[nH]1 c1(C(N(C)CC2(NC(C3CC(O)CN3C)=O)CC2)=O)cc2c(cc1Cl)NC(=O)CO2 C1(CC)C(NC(c2c[nH]nc2-c2ccn(C)n2)=O)CCN1C(=O)Cc1ccco1 C(C(C(=O)N(C1CCC2CC12)C)C(C)(C)C)NC(C(C)OCC=C)=O c1(CC(=O)NC2CC(NC(c3cn(C(F)(F)F)nn3)=O)CC2O)c[nH]ccc1=O C(=O)(C1=C(CCCCl)N(CCCSC)C(=S)NC1c1ccc(C#N)s1)OCC N1(C(C(CC2CCC2)OC)=O)CCN(C)CC1NC(=O)CC1CC(O)C1(C)C N1(C(C2C(C)CC(=O)N2)=O)CCCCC(CNC(=O)CC2(C)OCCO2)C1 c1(C2(CC(N(C)CCOCCN3CCCC3)=O)CC2)cccc(Cl)c1Cl c1(C(=O)NC2CCN(C(C(C)(C)NS(C)(=O)=O)=O)CC2F)cc2cccnn2c1 C1(NC(c2c(COC)cco2)=O)CCN(C(c2cc[nH]n2)=O)C1C(C)(C)C c1(C(=O)NCc2cn(C3CCCN(C(N)=O)C3)nn2)ccc2c(n1)CCO2 C1(C(F)F)(CNC(CC2N(C)CCC2)=O)CCN(C(C2(C(C)(C)O)CCC2)=O)C1 c1(CN(C(=O)CC2CN(Cc3ccc(Br)cc3)C2)CC)ccc2ncccc2c1 C1(NC(Cc2c(C)nc(CSCC)s2)=O)CN(C(=O)CN(C)CCO)CCC1C N1(C(CC(CC)O)=O)CCC2(NC(=O)COCC3CCCO3)CCCC12 C#Cc1ccc(C(=O)NCC2CC23CCN(C(=O)Cc2ccsc2)CC3)c(F)c1 C#CCC(C)(C(=O)N1CCSCCC1C)NC(=O)CC1(C#N)CC1 C(=O)(C1=CC2C=CC(C1)C2)N1CC(CN(C(=O)CC2CC2)C)C2(C1)CC2 CC1(C)CCC12CCN(C(c1cc(Cl)c(F)cc1F)=O)C2 C1(C(=O)NCc2cccs2)CC(=O)N(C2CN(C(C3CCCO3)=O)C2)C1 c1(C(CN(C(C2CCCC2O)C(=O)NCC2CCCO2)C)OC)ccccc1Cl CON(C)C1CN(C(=O)CCC2CCN(C(=O)C(C)C(=O)OC(C)(C)C)C2)C1 C1(n2cc(SCC(N3CCN(C(=O)C4=CCCC4)CC3)=O)nn2)CCCCNC1=O c1(C(N2CCC(C(C)NC(CCn3c(C)ncc3)=O)C2)=O)snc2ccccc12 c1(CC(=O)N(CC(=O)Nc2cccnc2)CCO)c[nH]c2ccc(C3=CCOC3)cc12 C1(CC)CN(C(=O)CCn2cc(-c3ccsc3)nn2)CC(C)S1(=O)=O c1(OC(C)=O)ccc(N(C(C(CC2CC2)NC(CCOCCOC)=O)=O)C)cn1 C1(NC(c2c(CCC)nco2)=O)CCC(NC(c2n[nH]c(C)c2Cl)=O)CC1 c1(C(N2C(C(=O)NC3C=CCCC3)CCCC2)=O)cc(F)ccc1F c1(OC)cc(I)c(CNC(C2CCCCC2c2ccc(Cl)cc2)=O)cc1OC c1(-c2ccc(F)c(SC)c2F)cncc2sc(C(=O)Nc3ccc[n+]([O-])c3)cc12 c1(COC)ccc(C(N2CCCCC2c2nc(=O)o[nH]2)=O)c(OC)c1 Cc1ccc(C(N2C3CCC2C(F)C(NC(C2CCCC2)=O)C3)=O)c([N+](=O)[O-])c1 N1(C(C=CC)=O)CCc2sc(C(=O)NC3CCn4cncc4C3)cc2C1 C(C(C)CC(=O)NCC(C1CC1)N(C)C(c1cnsc1C)=O)OC C=CCCC(C(=O)N1CCC(CN=[N+]=[N-])CC1)NC(=O)C(C)CCOC c1(C(=O)NCC(CNC(c2nccc(OC)c2)=O)O)ccc(P(C)(C)=O)o1 c1(C(N2CCCC(CCNC(C(C)OCCCC)=O)C2)=O)cccc(F)c1O C1(CN(C(COC(CC)C)=O)C2CC2)CCCN1C(=O)C(F)n1ccnc1 c1(C(N(C)CC2CCCC(NC(COC)=O)C2)=O)cnc2n[nH]c(C)c2c1 N1(C(c2cc(C(C)C)no2)=O)CC2CCC1C(CO)C2.C12(CCCC1)C(=O)N2 c1(C(=O)NCC2CN(C(C(C)O)=O)CC2c2cncn2C)cccc(N)c1 c1(C(=O)N(C)CC2(n3cc(-c4ncns4)nn3)CC2)cnc2sccc2c1 N1(C(C(C)c2cccs2)=O)C2CCCC1CC(NC(C13CC(CO1)C3)=O)C2 C1(C(=O)NC(CN(C(C2(OC)CC2)=O)C)C)CCCC(C)(C)C1 C12(NC(C3(CNC(c4n[nH]cc4[N+](=O)[O-])=O)CC3)=O)CCN(CC1)CC2 N1(C(CC(CC)C)=O)CCC(C2CCCN(CCC(F)(F)F)C2)C1 C(=O)(C(C)CC(F)F)NC1(CC(=O)NCc2cccc(NC)c2)CCOCC1 N1(CC(=O)N(C)C(c2ccnn2C)=O)CC(=O)Nc2cc(C(=O)C3CC3)ccc21 c1(NC(CC2CN(C(c3cnc(C)s3)=O)C2)=O)c(C(F)(F)F)cccc1Br Cc1cnc(NC(=O)C(COC(C)(C)C)NC(c2cccc(Cl)c2)C)cc1I CC1=NOC(C(N2CC(C(N)=O)(CNC(=O)C(F)C3CCC3)C2)=O)C1 c1(C(N2CCCC(N(C)Cc3ccc(CC)s3)C2)=O)cnc(Cl)cc1C c1(OCCCNC(c2c(NC(C(C)NC(N)=O)=O)c[nH]n2)=O)cccc(O)c1 c1(CNC(=O)NC(COC(F)F)CO)cccc2[nH]ccc12 c1(OC)cc(C(=O)NC2CN(C(c3ncccc3F)=O)CC2C)c(Cl)cc1Cl c1(OC)ccnc(CN2CCCC2C(=O)Nc2nccc(C3(C)CC3)n2)n1 Cc1cc(C(N2CCN(C(C3CC3CC(C)C)=O)CC2C2CC2)=O)c(C)cn1 CC(C)CCCOCC(=O)N(C)CC1CCN(C(=O)Cc2ccsc2)C1 N1(CC(=O)N(CCNCc2ccc(C(=O)O)o2)CC)CCC(F)C1 C1(C(=O)NCC2N(C(CC3C(C)(C)C(O)C3)=O)CCC2)CCC(C#N)CC1 N1(C(C2OCCN(C(CSCCCC)=O)C2)=O)CCC(CO)C1(C)C N1(C(C(CC=C)OC)=O)CCCC(F)(CNC(c2cnccc2Br)=O)C1 C12(C(=O)NCC(C#C)C(C)C)CC(CN(C(=O)CCCc3cnn[nH]3)C1)C2 C1(NC(CCC2CCC(=O)NC2)=O)CCN(C(c2ccc(O)cc2)=O)CC1F C#Cc1ccc(NC(=O)COC2CN(C(c3cc(C)c(C)s3)=O)C2)c(C)c1 c1(CC)[nH]nc(C(N2CC(CNC(=O)CNC(c3ccco3)=O)C(C)C2)=O)c1C C#CCC(C)(C)C(=O)NC(CNC(c1ccc(C2CC2)o1)=O)CCOC c1(C(=O)NCCN(CCC)C(C2CCCN2C(C)=O)=O)cc(Cl)c(SC)nc1OC N1(C(C(C)(F)F)=O)CCC(NC(C2C=CC(=O)N=N2)=O)C(F)C1 C1(C(=O)NC(CNC(c2c(C)ncs2)=O)C(C)(C)C)CCC2(CC1)CC2(F)F c1(OC)ccc(Cl)c(C(=O)NCC(O)CNC2CCOC(C(C)C)C2)c1C C(C)(C)(CCO)N(C(c1ncc(C(=O)OC)s1)C(=O)NCCCC)C.C(CCl)SCCC C(=O)(C1=CC(C)(C)C1)NCc1cn(CCNC(C(C2CCOCC2)OC)=O)nn1 c1(NCC(C)N(C)C)ccc(S(=O)(=O)NC2C=CC(C(N)=O)C2)c(Br)c1 C1(=O)C(C)(C)N1.CC(C(=O)NCCC1(CC2CCCO2)CC1)SCC1CC1 N1(c2cccc(CNCC3CC(OCC)C34CCC4)c2)CCS(=O)(=O)CC1 N1(C(CC(CCC)NC(C2CCCC2F)=O)=O)CCC12CCC(C)CC2 C1(COC)(CNC(=O)CC2CSCCO2)CCCN1c1nnc(C2CC2)o1 C(=O)(CC(C)(C)C(=O)OC)NC1CN(C(C(CC)OCC)=O)CC1O c1(C(N(C2CCN(C(C3(CCOC)CCC3)=O)CC2)CCC)=O)cc(C)sc1C C1(C(N2CCN(CC#C)CC2)=O)CNC(=O)CN1C(=O)COCc1nc[nH]n1 C1(C(=O)NCc2ncn(C)c2)CC2(CCN1C(=O)C=Cc1cscn1)CC2 c1(-c2cccc(N(C)C)c2)cccc2cc(C(=O)Nc3ncc(Br)cc3Cl)sc12 N1(C(=O)C2CC2)CCC2CCN(C)C2C1.C1C(=O)NCC2(CC2)C(=O)N1C N1(C(C(C)C2CCC2)=O)CC(NC(=O)C=Cc2cnn(C)c2)CC12CCCCC2 N12C(=O)C3N(CCOC34CN(C4)C(=O)C1)C2=O.C(C)(C)(C)C(=O)OC(C)C C1(C(N(C2CCCN(C(=O)CSc3n[nH]c(O)n3)C2)CC)=O)COCCOC1 C=CCC(C)(C)C(=O)NC1CCCC(C(=O)NCCCOCCCO)C1 C(=O)(C(O)C(C(C)C)OC)NCC(CC)NC(C1CC(C(C)=O)C1(C)C)=O N1(C(C2CC(C(C)C)C2)=O)CCC2(NC(=O)CC3CCC(=O)N3)CCCC12 Cn1cc2c(C(=O)NCC3CCC3NC(c3ccc(F)o3)=O)cccc2n1 C1(CNC(CSCc2nc(C)sc2)=O)CC(C)(C)CN1C(=O)CC1CCCCC1 N1(C(CC2N(C(C3=C(C)OCC3)=O)CCOC2)=O)CCc2ccccc2C1 n1(CC(=O)NC(CN(C(CCC=CC)=O)C)C)cc(C)c(O)nc1=O c1(C(N2CCCC(CN(C)C(C3CC(F)(F)C3)=O)CC2)=O)cc2sccc2cn1 c1(C(=O)NCCOCCN(C(C=CC(CC)=CC)=O)C)nncc2c1CCCC2 C1(C(=O)NCCCCN(C(C(CCC)OC)=O)C)CCc2cncn2C1 C12CCCC1NC2=O.C(C(F)(F)CC1CC1)NC(=O)CSCC(F)F c1(C(N2C(C(N(C3C(C)CC3)C)=O)CCC2)=O)cc(O)cc(=O)o1 N1(C(C2C(NC(c3cc(C)c(C)nn3)=O)COCC2)=O)CCc2ccsc2C1 c1(OC)ccc(O)cc1C(=O)NCC1CCCC1NC(=O)C(=Cc1c[nH]cn1)F CCN=C(NC(c1ccc(Cl)cc1)c1cccn1C)N1CCCC(C(O)CF)C1 N1(C(CCn2c(C(C)C)ncc2)=O)CCCC(C)C1CCNC(=O)COC(C)C C1(C(=O)NCC2CCN(C(c3ccn(C(F)F)n3)=O)C2)CC(=O)N(C(F)F)C1 c1(CC(N2CCN(CC(c3ccc(C#N)cc3)O)CC2)=O)ccc2nsnc2c1 C1(NC(CC2(OC)CC2)=O)CC2CCC1C(NC(=O)CCc1ccoc1)C2 CC(C)C(O)C(F)(F)C(=O)N1CCCC(C)(CNC(=O)CC2CCCC23CC3)C1 C(=O)(CC(C(F)F)C(C)(C)C)NCCC(=O)Nc1ccc(-n2c(C)ncc2)nc1 N1(C(c2c(C)nc(C)[nH]2)=O)CCC2CCC12CNC(=O)CNC(c1ccoc1)=O N=c1nc2ccc(C(N3CC(NC(c4cnc5[nH]cnc5c4)=O)C3)=O)cn2[nH]1 CCC(C)(CO)C(=O)NCC(C(C)(C)C)NC(=O)CCc1ccccc1C#N c12ccc(cn1)s2.C1(Oc2ccccc2)CCN(NC(C2CC2F)=O)C1 C1(C)(CNC(C(CC)n2nccc2C)=O)CCCN1C(c1cccc(F)c1)=O c1(CCC(=O)NCC2C(CNC(c3c(C)scn3)=O)C2)nc2ccccc2s1 Cc1cncc(C(=O)NC2(C(=O)NCCCOC(=N)O)CC(O)C2)c1 c1(C(=O)NCC2N(C(COC)=O)CCCCC2)c(C)c(O)nc2ccccc12 C(=O)(C#CC1(C)CCCO1)NCC1N(C(c2cccc(C)n2)=O)C2C(C1)COC2 c1(NC(=O)NC(C(=O)NC)Cc2cnn(C)c2O)ccc(C#N)c(I)c1 C(=O)(CCCCNC(C1C=CCN1C(=O)C(F)C1CCCC1)=O)NC C(C(=O)N1CC(CC(=O)N(CCCn2cc(CO)nn2)C)(OC)C1)(C(C)C)SC C(C)(N=c1[nH]c(=NCCCn2cccn2)[nH]c2c1CSC2)c1cn(CCOC)nc1 C1(COCC)CN(C(c2cn(C(C)C)nn2)=O)C(C)(C)C1.C12(CC1)C(=O)N2 n1(C(C)C)ncnc1C(N1CC(F)(CNC(=O)Cc2cnsc2)C1)=O CN(OCc1ccccn1)C(=O)CC1C(NC(=O)CC2CCCCC2O)CC1O c1(C(=O)N(CCSC[Si](C)(C)C)C2CC2)cnc2ccc(F)cc2c1C(F)(F)F c1(C(C(=O)NCC(CNC(=O)CN2CCOCC2=O)CO)O)ccc(Cl)c(F)c1 c1(OCC)cc(CC(=O)NNC=O)ccc1F.[nH]1cc(CCCCC2CC2)nn1 Cc1cc2[nH]c(C(N3CCC(NC(C4CCC(C)(C)OC4)=O)C(O)C3)=O)cc2o1 CN=c1[nH]cc(C(=O)NCC2CCN(C(=O)C(c3c(C)n[nH]c3C)C)C2)o1 C(=O)(C(C)CC(N)=O)N(C1CCN(C(=O)C(COC)OC)C1)CCC c1(SC)cc(C(N2CC3C(NC(=O)C(C)c4cncs4)C3C2)=O)ccc1N c1(NC(=O)C(N2CCC(N3CCC(O)C3)C2)=O)cc(F)ccc1F.C1(=O)CN1CC c1(OC)ccc(CN(C2CCCCC2)C(c2ccc(C3SCCS3)cc2)=O)cc1F CC1=C(C(=O)N2CC(NC(c3ccc(CN(C)C)cc3)=O)CC2C)CCCC1 S(=O)(=O)(c1c[nH]ccc1=NCC1CN(C)C1)N(C)CC1C(C)COCC1 N1(C(C(CC2CC2)NC(C2C(=C)C2)=O)=O)CCOCC1CO c1(NC(C)=O)ccc(Cl)cc1C(=O)NC1CCC(NC(c2occc2Br)=O)CC1 C=CC(C)(O)C(=O)NCCN(C(=O)CCCNC(c1cccs1)=O)CCC c1(C(=O)OC)ccc(NC(C2CC(NC(c3cc(F)ccc3Cl)=O)C2)=O)c(OC)c1 CC(CNC(c1[nH]nnc1C1CC1)=O)C(=O)NCCCc1cc[nH]n1 N1(c2c(C)cnc(C)n2)CC2CCN(C(=O)C(c3ccccc3)F)CCC2C1 CN1CCCC(O)(CC(=O)NC2CCC(N(C)C(c3ccccc3Cl)=O)CC2)C1 n1(CC)cc([N+](=O)[O-])c(C(=O)NC(CNC(=O)CC2CN(C)CC2O)C(C)C)n1 N1(C(c2conc2C2CCC2)=O)CCCC(N2CC2)C1 c1(COCC(=O)NCC(=C2CCCO2)C)cc[nH]c1C1CC1.C1=CCNC1=O C1(C(=O)NCc2cocn2)CCN(C(c2cncc(CO)c2)=O)CC1O CC1CCN(C(=O)C(c2cccc(Br)c2Cl)(F)F)CC1CC(=O)O N1(CC)CCCC(ONC(=O)NC2CC2CNC(c2ocnc2C(F)(F)F)=O)C1 Cc1cc([N+](=O)[O-])ccc1CN=c1cc(NCCn2cc(C3CC3)nn2)nc[nH]1 CC1CN(C(c2cc(-c3cnn(C)c3)no2)=O)CC1NC(C1(C(F)F)CCC1)=O c1(C(=O)NCC(CCOC)NC(=O)CCc2cc[nH]n2)cn2ccccc2n1 C1(C(=O)OC)CC(Cc2cn(CCNC(=O)NCC)nn2)C12CCC2 C1(CNC(c2cc(C)ncc2)=O)CN(C(C2C3CNC(=O)C23)=O)CC(C)(C)O1 S(=O)(=O)(c1ccc(NCc2cc3cccc(F)c3o2)c(Br)c1)NC1CCC(C)O1 Cc1cc(=NCCC(C)(C)CO)[nH]c(=NCC(C)c2cnn[nH]2)[nH]1 C1(C(=O)NC2CC2CC)CC12CC2.CC(C)(C)OC(C)(C)C.C1CCN1C(=O)N C(=O)(C(C)(C)CNC(C)=O)NCC(C)(F)C(C)C CC(CC(C)(C)C)C(=O)N1CCCC(C(=O)NCCCCCC2CC2)C1C Cc1nc2n(n1)CC(C(=O)NC(=O)C(C)(C)n1cc(C3CCCN(C)C3)nn1)CC2 CCCCC(CC)C(=O)N1CC(CC(C)(C)CNC(=O)C2=C(C)OCC2)C1 N1(C(c2ocnc2C(F)F)=O)CC(C2CCCN(C(c3cnns3)=O)C2)C1 C(CC(=O)NC1CC(N(C(=O)CN(C2CCC2)C)C)C1)OCCN(C)C Cc1ccc(C=CC(=O)NC2CCC2CNC(=O)Cc2cccnc2C)o1 C1(C(=O)NCCC(CNC(CN(C)C(c2cccs2)=O)=O)O)CC2(CCCC2)CO1 C1(C(N2C(CC)(CO)CCC2)=O)CCN(C(c2cc(C)c(C)[nH]2)=O)CCO1 c1(OC(C)(C)C)cnc(Cl)nc1N1CCC(NC(C2C3CCCC23)=O)CC1 C(=O)(C(C)(C)C)NCCCCNC(CNS(CC)(=O)=O)=O.C1(C(=O)N)(C(F)F)CC1 N1(C(=O)NC2CCC(c3ccccc3F)CC2)CCCC2(COCCN2)C1 Cc1cc(C(N2CCCCC2C2(NC(C3CCCC3F)=O)CC2)=O)nc(C)c1 CCCCC(CC)CCC(=O)N1CC(NC(C2(C)CC(=O)N(C)C2)=O)C1 C1(C(=O)NCC2C(C(=O)NC(C3(CC)CCCC3)=O)CCC2)CCCC(C)(C)C1 N1(C(c2c(C)[nH]cc2)=O)CCN(CC(=O)NOC2CCN(C)CC2)C(=O)C1 CCC(CC)(C(=O)N1CCC(C(=O)NC(C)(C)CCCF)C(O)C1)OC c1(C(CC)C)ccc(C(=O)NC(C)CNC(=O)CC2OCCOC2(C)C)c(O)n1 C1(C(N2CC(NC(CN(C)C)=O)C(O)C2)=O)CCC(C2CCC2)CC1 c1(C(N(CCCCCC(=O)N(C2CC(C)OCC2)C)C2CC2)=O)cncc2[nH]ccc12 C1(C(N2C(C(N(C)C)=O)C=CC2)=O)CCCC(NC(=O)Cn2ncn(C)c2=O)CC1 c1(C(C(=O)NC(CCCNC(c2cnc(CC)s2)=O)C)C)ccc(C(F)F)cc1 c1(CC(=O)N(C2CCCN(C(c3ccc(C(F)F)s3)=O)C2)C)cccnc1O c1(C(=O)NC(C2CCN(C(C(C)NC(N)=O)=O)C2)C)ncccc1Cl N1(C(CSC)=O)CCC2(CCC(CNC(=O)C(C3CCCN(C)C3)(C)C)O2)CC1 C1(C(=O)NCC(C(C)C)NC(=O)C(c2ccnn2C)C)CCC(=C(F)F)CC1 Cc1cc(NC(N2CCC(CC(N3CCOC(C)C3)=O)C2)=O)ccc1N(C)C n1(CC(=O)NC2CN(C(C(C)CO)=O)CC(F)C2)c(S)nc2ccccc2c1=O N1(C(C(COC)N(C)C)=O)CCC(CNC(c2cccc(=O)n2C)=O)C1(C)C c1(CCC)ccccc1C(=O)NC1CCC(N(C(=O)CC2CC=CC2)C)CC1 c1(NCC(N2CC(CNC(CC=C)=O)C(O)C2)=O)cccc(C#N)c1 C1(CCNC(C2CC2(Cl)Cl)=O)CN(C(c2cccc(=O)o2)=O)CCS1(=O)=O C12(CNC(CCC=C(C)C)=O)CCC1CCN2C(c1cccc(Br)c1N)=O C(C(=O)N1CCC(OCC(=O)NC2CCCSC2)C1)(C(C)(C)C)OC C1(C(N2CCC(NC(=O)CC34CCCN3CCC4)C2)=O)CCc2ccccc2O1 c1(NC(c2ccn(C)c2)C)ncc2n1CCC2 N(C1CSCc2ccc(Br)cc21)C(C)(C)C.N12CCC(O)C(C1)NC2=O C(=O)(C(C(C)(C)C)NC(C1CSCCN1C(C1CC(C)(C)C1)=O)=O)N(C)C N1(C(C=Cc2ccc(CC)o2)=O)CC2(C1)CN(C(c1cc(=O)cc[nH]1)=O)CCO2 c1(CCCC)ccccc1COC(c1cnc(-c2cnccn2)s1)=O C(C(CN)C(F)(F)F)NC(N)=O.c1(C2CN(C(=O)OC(C)(C)C)C2)nn2ccsc2n1 C1(C(=O)NC2CCC(NC(c3c(C)oc(CO)c3)=O)CC2)CCC(N=[N+]=[N-])CC1 c1(C(=O)NCCC(N2CCC(CN(C(=O)OC(C)(C)C)CC)C2)=O)cc(O)ncn1 C(C(CC1CC1)C(=O)N1CCC(OC)C1)NC(CCOCCN)=O.CC(=O)C(C)=O Cc1ccc(C(=O)NCC(CO)NC(=O)C#CC2CC2)c(F)c1Br C1(CNC(c2ccc(C)nc2O)=O)CC2(CCC2)CN1C(c1coc(C#N)c1)=O c1(C(=O)NCCCC(C)NC(=O)Cc2coc(C(F)F)n2)ccc(P(C)(C)=O)o1 C(=O)(C(C)(COC)OC)NC1CC1(C)C.C=C1CC2(C1)C(=O)NC2 C1(NC(C(C)SCCCC)=O)CC(N=c2[nH]c3c(C)cccc3o2)C1 N1(CC(C(C)OC)OC(=O)NC(=O)C(=O)C)CCCCC1(C)C.C(C)(C)(C)O C1(C(N2C(C)C(O)CCC2)=O)C2CCCC1CN(C(=O)Cc1cc(F)ccc1Br)C2 c1(NC(N(CC)CC)=O)cnc(NC2CCN(Cc3ccccc3)C2)cn1 Cc1ccc(COCC(=O)NC(C)C(C)NC(C2CCC2)=O)cc1 C1(NC(CCn2ccc(C)n2)=O)CCC(C)N(C(=O)COc2cccc(F)c2)C1 N(C1c2ccccc2CC1NC(=O)C(C)N1CCC1)C(C=CC)=O C1(NC(CCOC)=O)CN(C(=O)CCSc2nncn2C)CC1n1ccnn1 c1(OCC=C)cccc(C(c2nnnn2C)OCc2ccncc2)c1 c1(C(=O)NCCn2cc(CNC(CC(C=C)C)=O)nn2)cc(Cl)cc2c1OCC2 N1(Cc2snc(OC(C)C)c2Cl)CCCC2(CCCCN2)C1 C1(C(=O)NC2CC(C(C)C)C2)CCN(C(=O)Cc2ccsn2)C(C)(C)C1 C1(CNC(=O)CCOC2CC2)CCCC(NC(c2ccnn2C2CCCC2)=O)C1 Cc1nn(C(C)C)cc1NC(=O)ON1CCC(CCOC(C)(C)C)C1 c1(C(c2cn(-c3nccc(C)c3)nn2)NC(=O)CN(C)C)c(F)cccc1Br C1(NC(c2c(CC)c[nH]c2)=O)CCN(C(C2(C)CS(=O)(=O)C2)=O)CC(C)(C)C1 c1(C(=O)OCC(=O)NC)ccc(S(=N)(=O)C(F)(F)F)cc1 c1(C(=O)NC2COC3(C2)CN(C(c2ccco2)=O)C3)cc2c(Cl)nccc2s1 c1(NC(CC=CC(=O)NCCC2(NC(CC(C)OC)=O)CCC2)=O)ccc(F)cc1 C(=O)(CCCCCNC1CC(O)C1CCO)NCC(n1ccnn1)C c1(C(N2CC(N(C(=O)CCCc3cncs3)C)C2)=O)cncc(CO)c1 n1(CC)ncc(Br)c1C(N1CC(C(F)Cn2cc(-c3ncoc3C)nn2)C1)=O C1(C(=O)O)CC2C(C1)C2(F)F.c1(C(C(=O)NC(CC)CC(N2CCCC2)=O)C)ccn(C)n1 C1(C(N2CCCC(CCOC)C2)=O)CC2CCN(CCC(F)(F)F)CC12 C(c1cc(C)cc(C)c1)=CC(=O)NCC(C)(C)NC(c1cccc(NC)n1)=O C12(C(N3CCCC(C)(N(C)C)C3)=O)CCC(NC(C(C)n3cccn3)=O)(CC1)C2 C1(NC(c2c(C)nc(CC)s2)=O)CCCN(C(=O)COCC2CCOC2)CC1 c1(C(=O)NC(C)CNC(=O)CCC2CC2(F)F)cnc2n1C(C)CCC2 C1(OC)CC(CNC(=O)Cc2cncnc2)N(C(C2SCCCS2)=O)C1 N1(C(C2(CC#C)CCCOC2)=O)CCC(NC(=O)CC(C)(C)C(C)=O)C(C)(C)C1 CP(C)(=O)C1CCCC1C(=O)NCC1CC2CCC1N2C(C1(CN(C)C)CC1)=O N1(C(C2N(CC)CC2)=O)CC2CCC(C1)N2C(C1(C2CCCO2)CCOCC1)=O C1(C(=O)NCC(C)NC(Cc2cnc(C)o2)=O)CCN(S(=O)(=O)N(C)C)C1 CC(C)C(F)(F)CC(=O)N1CCCC1CNC(c1ncoc1C(F)(F)F)=O C#CC1CCN1C(=O)C(Cc1cnc[nH]1)NC(c1sccc1F)=O c1(C(=O)Nc2cc(C)nn2C2CCOC2)ccc(F)c(C(F)(F)F)c1 c1(NCC(C)(C)NC(=O)NC(CC)C)cn(CCN2CCOCC2)nn1 N1(C(C2OCCN(CC)C2)=O)CCCC2(NC(=O)CC3(OC)CC3)CCCC12 N1(C(c2cnc(C)n2C(F)F)=O)CCCC2CCC12Cc1ccccc1 C(=O)(C1CCCc2ccccc21)N1C(CNC(CC2(NC(C)=O)CC2)=O)CCC1 CC1(C)C(C(=O)NCc2cccs2)CCN1C(=O)CC1CCSCC1 C(=O)(C(F)(F)C(C)O)N1CCC(CC(=O)NCC(COCC)(C)C)CC1 C1(C(=O)NCC(C)CNC(c2ccn(CC(F)F)n2)=O)CC2OC(C)(C)OC2C1 O=S(=O)(c1cnc(Cl)nc1)NC1C2CCC1CN(Cc1cccc(Cl)n1)C2 c1(C(=O)NC(CNC(COC(CC)C)=O)C(C)C)cc(Cl)ccc1C(F)(F)F C1(CC#C)(C(=O)NCCCC2CC(F)(F)C2)CCN(C(=O)C=CC(C)C)C1 C(CCCCC(=O)N1CC2CC2(NC(C2CCN(C3CC3)C2=O)=O)C1)OC c1(C2CC(NCc3ccc(-c4onc(C(=O)NC)n4)s3)C2)ccccc1C n1(CCCC)nnnc1C(c1ccnn1CCF)NCCOCC1CC1 c1(C(=O)NC(CN(C)C(C2C3C4CCC(C4)C23)=O)(C)C)c[nH]c2nc(F)ccc12 C1(C(N(C(C)CSC)CC)=O)(CN(C(=O)CC2C=CCC2)C2CC2)CCCC1 c1(N2CCC(OC)C(C)(C)C2)[nH]c(=NCc2cn(C(C)C)nn2)nc2c1ncn2C C12(C(N3CCCC(NC(C(C)C4=CCCC4)=O)CC3)=O)CCCN1S(=O)(=O)CC2 c1(CC(=O)NC(CC)CN(C(=O)C2=CCCOC2)CC)cccc2c1OCCO2 Cc1ncc2c(n1)CCC(NC(=NCCCOC(C)C)NC(C)C)C2 N1(C(CCc2ncc(C)[nH]2)=O)CCN(C(=O)Cc2cccc(C(C)C)c2)C2CC12 Cc1nc(C(=O)NC2(CNC(=O)CC3(C)CC3(F)Cl)CCCCC2)c(C)o1 C1(CN(C(C2(CC=C)CCCC2)=O)C)COCCN1C(c1csc(CC)c1)=O c1(C(=O)NC(CC)CNC(C2OCCC2C(F)(F)F)=O)ccc(C2CC2)c(F)c1 c1(C(C(=O)NC2CCOC2)N(c2cnn(C)c2)CC)ccnc(F)c1 c1(-n2cc(SCCN(CCCCCN=[N+]=[N-])C)nn2)ccc(Cl)cc1F c1(SCC(N2C(CNC(COCC=C)=O)CCC(C)C2)=O)nc2ccccc2s1 C(=O)(CC(C)(C)C)NCC(CC)(C)C(Cn1cc(C(=O)NC(C)C)nn1)=O C1(C(N2CCC(NC(c3c(C)ccs3)=O)(CO)C2)=O)CCCCN(C)C1=O C1(C(=O)NC2(CNC(=O)C(=O)NCC3CC3)CCOC2)CC2(CO1)CC(F)(F)C2 c1(C(N2C3(C(=O)Nc4c(Cl)nc(OC)s4)CC(C2)C3)=O)nn(C)c2ccccc12 c1(OC)ccc(C(=O)NCC2CCCCCN2C(c2c(C)ccnc2O)=O)c(Cl)n1 c1(C(CNC(C(COC)(C)C)=O)NC(C2CCCN(C)C2)=O)cc(F)cc(Cl)c1 c1(CC(=O)NC2CC(NC(C(CC3CC3)OC)=O)C2)sc(Cn2cnnn2)nc1C C=CC1CN(C(=O)CCC2CC2)CC1NC(c1cc(=N)[nH]c(Cl)n1)=O C#CCC(C)(CNC(C1CC(C)CN1C(=O)CCCCN(C)C)=O)CO c1(CC(=O)NC2CCN(CCCNC(COCC#C)=O)C2)ccc(F)c(OC)c1 CCC(C)(CNC(=O)C(C1CC1)OCC)NC(c1cc(C(C)(F)F)on1)=O C1(NC(C(=O)Nc2nc(C)c(CN3CCCC3)s2)=O)CCCC(C)(C)CC1 C1(NC(CNC=O)=O)CCN(C(C2(F)CCCC2)=O)CC1F C1(F)(CNC(C2C=CCC2)=O)CCN(C(=O)CC2COCCO2)CC1 N1(C(C(CCC)NC(C)=O)=O)CC2CCCC2(C(=O)NCC(C)(C)CC2CC2)C1 c1(CC(N2CCCC(NC(CC3CC(OC)C3)=O)C2)=O)c(C)ccc(Br)c1F N1(CC)CC(C(N2CC3(CCN3C(C3CCCN3C(C)=O)=O)C2)=O)CCC1=O c1(C(=O)NCCCCCNC(c2n(C)ccc2)=O)c(Cl)csc1Cl c1(C(=O)N(C(CC2CC(F)(F)C2)CO)C2CC2)ccc(Cn2cccn2)cc1 c1(-n2cc(CN(C(CCCNC(C(CSC)(C)C)=O)=O)C)nn2)ccc(F)nc1C CCC(C)(CCNC(c1nccn1C)=O)NC(c1cnn(C(C)C)c1)=O C1(=O)C#CC(C)(C)CN1.C(=O)(C(C(C)OC)N(C)C)N(CC(CC)(C)OC)C Cn1ccc(C(=O)NC(C)(C)CCNC(=O)CC2CCCS(=O)(=O)C2)cc1=O C1(C(N2C(C(N(CCC(=O)OC)C)=O)CC2C)=O)C2CCC(F)C12 CCC(CC)C(C(=O)N1CC(C(C(=O)NCCC(O)CCO)OC)C1)OC C(C(=O)NCCCNC(c1cc(C)ns1)=O)(C(C)O)NC(C)=O N1(C(C2(C)CC(NC(c3n(CC)nc(C)c3)=O)C2)=O)CCC(F)(C#N)C1 C1(CNC(=O)CCN2CCCCC2)CCCCNC1=O.C1CCCCCC(=O)N1 c1(SC)ccc(C(=O)NC2CC(C(=O)N(CC(O)CN(C)C)C)CC2O)cc1 C1(N=c2[nH]ccn3nnnc23)(CNC(CC2(O)CC(C)(C)OC2)=O)COC1 c1(CC)cc(C(=O)N(C2CCCN(c3nccc(C(N)=O)n3)C2)C)sc1C C12(NCC(=O)NC3C(CNC(CC(CCC)C)=O)C3)CC(C)(C1)OC21CCC1 c1(C(N2CC(N(C)C)C2)=O)ccc(C(F)(F)C(F)(F)F)nn1 C(CN=c1[nH]c(=NCC2CSC2)[nH]c2c1CCC2)n1c(CC)ncc1 C1(NC(C2CC(C)(C)CCO2)C)CCOC12CCCC2 C#Cc1ccc(C(N2CCN(CC(=O)NC3(C(N)=O)CCOC3)CC2)=O)c(C)c1 N1(C(C(c2ccc(Cl)cc2)N(C)C)=O)C2CCC1C1CNCC21 C1(C)(CNC(C(C)n2cccc2)=O)CCN(C(C2CCC(CC#N)CC2)=O)C1 c1(NC2C(C=C)CN(Cc3ccccc3)C2)ncnc2c1ccn2C N1(C(CCNCCCOC)=O)CCCC1C1(NC(=O)CC2CCC2)CC1 CCCCCCC(=O)NCCCC1CCC(NC(c2cc3sccc3[nH]2)=O)C1 CC(C)C(C(=O)N(C)CC1CCN(C(=O)C=CCn2cncn2)C1)n1ccnc1 C(=O)(C1=CC2CCC=CCCC12)N1CC(O)(CNC(c2cccnc2S)=O)C1 C1(C(N2CCc3cccnc3C2)=O)COC2(CCN(S(=O)(=O)c3ccc(Br)s3)CC2)C1 N1(CCN(C(=O)C(COC)COC)CCC)CCCCS1(=O)=O C1(C)CCCN(C(C2CN(N(C)NC(C(C)SCC)=O)C2)=O)C1.C(C)(C)(C)OC=O c1(NC(C2N(Cc3scc(C)c3)CC(O)C2)=O)nc2ccc(I)cc2o1 C1(NC(CN2CCC(C)CC2)=O)CCCC(NC(c2ccc(=O)n(C)n2)=O)CC1 C1(CNC(Cc2c(C#C)cccc2)=O)CCCC2(CN(C(=O)CNS(N)(=O)=O)C2)O1 CCCC(CC)NC(=O)C(C)CN(C(c1ccncc1)=O)C1CC1 CC1C2CCC(C2)C1C(N1CC(C(N2CCN(CC(N)=O)CC2)=O)C(F)(F)C1)=O C1(C(=O)NCC(CN(C(C2C(C)CCO2)=O)C)O)CCC(C(F)(F)F)CC1 CCC(C)C(C(=O)N1CC(CCOC)C1)N(C)C(c1cc(C(C)=O)[nH]n1)=O C=CC(C)CC(=O)N(C(C(=O)NCCCCC(C)SC)(C)C)CCC c1(C(c2nnnn2-c2ccccc2C)NCC(CO)OC)cc(Cl)cc(Cl)c1 N1(C(C(C)(C)N(C)C)=O)CC(NC(c2noc3ncccc23)=O)CC2(CCC2)C1 C1(NC(C2CC(C)OC2C)=O)CC2(C1)CC(NC(=O)C=Cc1ccc(O)cc1)C2 C=CCC(C)(CC)C(=O)NCCCN(C(C1CCS(=O)(=O)C1)=O)C1CC1 C(=O)(C(C(C)CC)N(C(=O)CCN(C)CCC)C)N(CCC#C)CC C1(CNC(c2cn(CCC)nn2)=O)CCCCN(C(c2cn(C)nc2Br)=O)C1 C1(NC(C2N(C(C3(C=C)CCC3)=O)CC2)=O)CCc2nn[nH]c2C1 c1(CCC(=O)NCC2(NC(C(CCC)OCC)=O)CCC2)ccc(Br)c(F)c1 C1(C(=O)NC(C2N(C(CCCOC)=O)CCC2)(C)C)CCCN(c2nccs2)C1 N1(C(C(c2cnn(C)c2)OC)=O)CCC(C(C)NC(=O)CC2COC(=O)N2)CC1 c1(C(N(C(C)CNC(c2cc(C)nc(O)n2)=O)CC)=O)cnn(C)c1S(N)(=O)=O c1(C(N(CCOC)CCNC(c2n[nH]cc2C)=O)=O)cnn(C(C)C)c1C C=C=CCC(=O)NCC(C)N(C(=O)C(O)CN1CCOCC1)C N1(C(C(COC)(F)F)=O)CCCC2C1CCN2C(C1CC(F)(F)C1(F)F)=O c1(CNC(c2ccc(COC)o2)=O)ccc(C(=O)NCC=CBr)cn1 C(C)(N=c1[nH]c(N(C)Cc2ccc(CO)o2)nc2c1CCC2)c1ccc(C)s1 c1(C(C(=O)NCC2CC(F)(CNC(=O)CCNC(=O)CO)C2)O)cccc(Cl)c1 c1(NC(C(c2cc(C)nn2C)(C)C)=O)ccc(F)c(N2CCOC2=O)c1 c1(C(C(=O)NCC(C)(C2CC2)NC(CC=CC=C)=O)(C)C)ccc(CC)cc1 CCCS(=O)(=O)CC(=O)N(C(Cc1ccc(Br)cc1)CO)C c1(COCC)nc(NCCC(C)O)cc(=NC(C)c2cccn2C)[nH]1 c1(NC(N(C(c2nccs2)C)C)=O)ccc(Br)c2nccn12 c1(C(C(C)NC(=O)Nc2ccc(N3CCOCC3)nc2)=O)ccc2c(c1)OCCO2 S(=O)(=O)(c1cc2sc(=NC3CC(C)C3)[nH]c2cc1Cl)NC(C)CF C(=O)(C1=NOC2COCC12)NCc1occ(C(=O)NCc2c(C)nn(C)c2)c1 CS(=O)(=O)C1(C(=O)NCC2CCCCN2C(=O)CNC(C2CCC2)=O)CCC1 N1(CCNC(CCN(C(CCC)C)C)=O)CCOCC1.C(CC(=O)N)=CC=CCO c1(C(=O)NCC2CCN(C(CCSC(C)(C)C)=O)C2(C)C)cc(O)ncc1F C1(NC(C(C2CCN(C(C3(Cl)CC3)=O)CC2)C)=O)CC(=O)N(C)C1 C1(N(C)C(c2cc(C(C)(C)C)no2)=O)CCCC(NC(c2cccs2)=O)C1 N1(C(CCC2N(C(C(CC)C)=O)CCCC2)=O)CCn2c(C)cnc2C1 c1(C(=O)NC2CCC(N(C)C(c3ncoc3C3CC3)=O)C2)c(F)cc(Cl)cc1F N1(C(COCCOC)=O)CCCC(C(=O)NCC(=O)OC)C1 N1(C(CCNC(N)=O)=O)CCC(C(F)(F)F)C(NC(=O)CCn2cccc2)C1 N1(C(COC2CCN(C(C(C)=O)=O)C2)=O)CCS(=O)C(C)C1 CC1(C)CC(CNC(C2CNC(=O)N2)=O)CN1C(=O)CNC(c1ccsc1)=O c1(C(N2CCCC(NC(C(C)Sc3ncccn3)=O)C2)=O)ccc2snnc2c1 c1(C(N(CC(C)NC(=O)C(C)(C)CCSC)CC)=O)ccc2c(c1)N(C)CC2 C12(C(=O)NC3CCN(C(COC(C)=O)=O)CC3O)CCC(C(C)=O)(CC1)CC2 CC(C)C(C(=O)Oc1c(CC(N2CCOCC2)=O)cccc1)OC(F)(F)F c1(N2CCC(CNC(C3CCc4nnnn4CC3)=O)C2)ncnn2c(Br)ccc12 N1(C(C2(C#N)CCCO2)=O)CCCC(CO)(NC(c2ccc(C3CC3)cn2)=O)C1 N1(C(CCC(C)=O)=O)CCN(C)CC1CNC(c1cc(C(F)(F)F)c[nH]1)=O CC1=NC(C)(CNC(C2CCOC2CNC(C2CCCC(O)C2)=O)=O)CS1 c1(OC)nc(=NCCN2CCN(C(=O)C=C(C)C)CC2=O)[nH]cc1C c1(C(=O)OC)ccc(CCC(=O)NCCC(O)CNC(=O)C=C(C)C(C)C)cc1F C1(C(=O)NCc2onc(C)n2)CN(C(=O)C(N2CCOC2=O)C)CC12CC2 c1(CCCNC(=O)CCC2CCCOC2)cccc2c1OCO2 C(C(C(=O)N1CC(CN=[N+]=[N-])C1)C(C)(C)C)NC(CC(C)C1CCCC1)=O C1(C(=O)NCc2ccn(CCC)n2)CC(F)CN1C(C1CC(C)(C)CO1)=O C(c1ncc(C)[nH]1)=CC(=O)N(CCCSC)C(=O)CSCC(F)F.CC C1(CNC(C(CCSC)NC(c2ccsc2C)=O)=O)CC2CCC(C1)C2 c1(C(=O)NCC2CCCCN(C(C(C)CC(F)F)=O)C2)cc2cnccc2o1 N1(C(C(CC=CC)NC(C2CC(F)C(=O)N2)=O)=O)CCC2(CC(CO)C2)C1 C1(C(N2CC(C(C)NC(c3c(C#C)cn(C)n3)=O)C2)=O)CCc2cnc(C)n2C1 c1(CNc2cncc(C(N(CC)Cc3ccncc3)=O)c2)cc(OC)ccc1N C12(CNC(C3CCCCC(=O)N3)=O)CCCC1CN(C(=O)C(F)CC1CCCC1)C2 CCC(C)CCCCC(=O)NCC1N(C(c2cccc(N)c2)=O)CCCC1(C)C C1(NC(c2ncccc2C2CC2)=O)CCN(C(=O)CC2CCCCC2)C1C1CC1 N1(C(Cc2n(C)cnc2)=O)CC2CCC(CNC(C3CC(=C4CCC4)C3)=O)C2C1 c1(C(=O)NCC(C)N(C)C(c2cccc3c2OCC3)=O)cccc2c1CCN2 c1(C(=O)NC2CCCCCN(C(C3(CC#C)CC3)=O)C2)nc(C)n2c1CCCC2 N1(C(C(C)=C(CC)C)=O)CCC2(CCCN2C(c2cn(C(F)F)cn2)=O)C1 N(C1C(=O)Nc2ncccc21)C(c1c(C)oc(C(C)(C)C)c1)=O N1(C(C2COCCN(C(c3cnn(C)c3N)=O)C2)=O)CCC(O)CC12CC2 CCC(CC(=O)OC(C(=O)NCCC1CCCCC1)C)CC(C)C CC(C)C(F)C(=O)N(C(C)(C(=O)NC(C1(O)CCC1)C)C1CC1)C c1(C(C(=O)NCCC(=C)CNC(=O)CC2COCC2O)(C)C)cccc(F)c1 N1(C(C)=O)CC2CN(C(c3ccccc3-c3cnco3)=O)C2C1.c1(C(=O)O)ccc(C#N)s1.CS C1(C(N(CC(CN(C(C(COCC)(C)C)=O)C)O)C)=O)CCC2CC2CC1 C(=O)(CCCCC(=O)N1CCC(C(=O)NCc2cnnn2C)(CO)C1)OC C1(CCNC(C2(SC)CN(C(c3cc(OCC)n[nH]3)=O)C2)=O)CCCN(C)C1 C1(C2CC2)(C(N(CC)Cc2ccncc2)=O)CN(C(c2cc(C(F)F)[nH]n2)=O)C1 c1(C(N2CCC3(CN(C(=O)CC4CSCCS4)C3)C2)=O)cc2n(n1)CCCC2O c1(OC(C)C(=O)N(C)CCN(C(=O)C(C)NC(C)(C)C)C)ccccc1F CC(CCCCC#N)(c1nnnn1CCCOCF)Nc1cccc2c1CCN2 c1(OCC)cc(C(=O)NC(C)C(C)NC(c2ccc(C(F)F)o2)=O)ccc1C c1(C(=O)NCCN(C)C(C2CC=CCC2)=O)c[nH]nc1OCC(F)(F)F N1(C(Cc2nc(C)sc2)=O)CCC(C)N(C(=O)C=CCN2CCOC2=O)CC1 CCC(C)CCCC(=O)N1CCC(CC(C)NC(=O)C(O)C(F)(F)F)CC1 N1(CC)CCC(C(=O)NC2CCCC2CNC(c2ccc(OCC)cn2)=O)CC1 c1(NC(C2C(NC(c3ccc(CSC)cc3)=O)C2)=O)nc2cc(F)ccn2n1 C(=O)(CCC(CF)CF)N1CC(NC(Cc2ccc(C)c(C)c2)=O)C(F)C1 N1(C(C(C(C)OC)N(C)C)=O)CCCCC(C(=O)NCC2CC3CCCC3C2)C1 N1(C(C(=Cc2cn[nH]c2)C)=O)CCC(C)(NC(=O)Cc2noc(C3CC3)n2)C1 CC(C)C(O)C(C)C(=O)NCC1(O)CCN(C(=O)CCN(C2CCCCC2)C)C1 C=C1CCN(C(=O)C(C2CCCC2)N(C)C)C(C(=O)N(CC(O)COC)C)C1 C1(C(N2C(CN(C)C(c3ncsc3C3CC3)=O)CC(F)C2)=O)CC(=O)NC(=O)C1 C1(C(N2CCC(C(=O)NCC)C2)=O)CC(NC(=O)C(C)CCOC)C(O)C1 c1(CN2C(C)(CC)CCC2)ccc(O)c(C2OCCO2)c1 CCC(C(C)(C)C(=O)NOCC1CCCC1)NC(c1cn(C)c(=O)n1C)=O N1(C(C2(C)CC2(F)F)=O)CCC2CCN(C(=O)CC3CCC=CCC3)C2C1 N1(C(c2c(C)scc2)=O)CC(CNC(C2(CO)CCCCO2)=O)C(F)(CO)C1 C1(C(C(=O)OCC(CCCC(=O)OCC)=O)N(C2CCC2)C)CCC2(CC2)CO1 N1(C(c2cnc(O)n(C)c2=O)=O)CCCC2(NC(=O)CC3CCCC3)CCCC12 c12c(cnc3cc(O)nn13)C(=O)N(CC(C)C)C2.CC.OC C1(NC(CCCn2c(C)ncc2)=O)CC(CO)N(C(=O)CCC2CCCO2)C1 CCCCCCCC(=O)NC1CCCC1CNC(c1c(CC)nc(O)nc1C)=O n1(C(C(=O)NC(C2N(C(COCCOC)=O)CCC2)C)CC)cnc(C#N)n1 c1(C(=O)NCC(C(C)C)NC(c2c[nH]c(=NC)s2)=O)cccc2c1OCC(=O)N2 CCCC(C(=O)NC)N(C)C.C12CCC(CC1)N2C(=O)C#CC1CC1 c1(CCCCC)ccc(C(N2CCCC2CC2CCC2)=O)o1 Cc1cc(C(=O)NCC(C2CC2)N(C(=O)CC2(N(C)C)CCC2)C)no1 c1(CN2CC(NC(c3cc(F)ccc3[N+](=O)[O-])=O)C2)c[nH]c2cc(F)c(F)cc12 C(=O)(C(C)(CC)CC)N1C(CCCNC(c2c(CC)non2)=O)CCCC1 C(=O)(C1CCc2cccnc21)N(C)CC1(CNC(c2cc3n(n2)CCO3)=O)CC1 c1(NC2CCC(NC(c3ccc4nc[nH]c4n3)=O)C2)ncc2c(Br)cccc2n1 C1(CC(=O)Nc2cn3ccsc3n2)(COC)CCCNC1=O C(=O)(C1=CCOCC1)N(C1CCN(C(c2ncccc2OC(F)F)=O)CC1)CC c1(C(=O)NCC2OCCN(Cc3c(C)nc[nH]3)C2)n[nH]c2ccccc12 C1(O)(CCNC(CCC(=C)C)=O)CCN(C(c2c(C(C)=O)cnn2C)=O)CC1 c1(CC)cscc1C(=O)NCCCNC(=O)C(CC)C1CCOCC1 c1(C(N(C(CNC(CCCN(C(C)C)C)=O)C)C(C)C)=O)ncccc1Br Cc1cccc(C(N2CC3(C2)CN(C(c2cc(C)c(C)o2)=O)C3)=O)c1N C1(N(C(C2(C)CCCO2)C(=O)NC)C)CCc2cc(Br)ccc2C1 c1(C(=O)NCCN(CCOC)C(C2CCCOC2)=O)ccc(NC(C)C)cc1 CC(C)C(C#N)C(=O)NCCCN(C(=O)COC1CCCOC1)C N1(C(C2N(C(CC)=O)CSC2)=O)CC2CCC1C2NC(c1scc(C)c1OC)=O c1(CNC(c2ccc(Cl)[nH]2)=O)csc(CNC(c2cc(-c3ccco3)on2)=O)n1 c1(CC(N2CC(CNC(c3nc(Cl)cs3)=O)NCC2)=O)ccc2sccc2c1 C1(NC(c2c(SC)scc2)=O)CC2CC(NC(c3cn(C)cn3)=O)C2C1 C=CCC(C)(C)C(=O)NCCC1CCC(NC(c2nccc(C)c2N)=O)C1 c1(C(N2CC(CC)C(NC(=O)C(C)(F)F)CC2)=O)ccc2occc2c1 N1(C(C2CC(=C)C2)=O)CCC(F)(C(=O)Nc2cc(C)on2)C1 Cc1oc(-c2cccs2)nc1CC(N1CC(O)CC1CNC(C1(C)CCCC1)=O)=O CCC(C)(CC)C(=O)NCc1cc(O)nc(CNC(=O)Cc2cc(C)no2)n1 c1(CC(=O)NCC(F)CNC(c2ccc(F)c(O)c2F)=O)ccc2c[nH]nc2c1 C1(C(N(C(C)C)CCNC(=O)CCCC2CCCC(=O)N2)=O)CCC(O)CN1C Cn1cc(C(=O)NCCc2ocnc2-c2ccccc2)nc1O c1(C(=O)NCC2C(NC(C(C)CC3CCC3)=O)CC2)cc2cc(Cl)ccc2o1 c1(CNC2CCC(NC(c3c(C)c(Cl)ncc3)=O)C2)ccncc1[N+](=O)[O-] N1(C(C(CC)CC)=O)CCN(C(=O)CCCc2ncc(C)o2)C(C)C1C N1(C(C(C)C2CCC2)=O)CCC(C(=O)NCCCC2CCC2)C1(C)C c1(C(N2CC(CNC(CCC=C=C)=O)C3C2C3)=O)cnc2c(F)ccc(F)c2c1 c1(C(=O)OCC(N2CCCC2)C)noc2ncccc12 C1(C(=O)Nc2ccn(CC3CC3)n2)(CNC(C2(OC)CCC2)=O)CC12CCC2 C(=O)(C1=NOC(C)C1)NCc1cc(C(N2C(CC)CC(C)C2)=O)on1 Cc1n[nH]c(C)c1CCC(=O)NCC(C)CNC(C1CCN(CC(F)F)CC1)=O CCC(C)CC(C)C(=O)N1CCC2(CNC(c3cnc(C)c(C)c3)=O)CCCC12 C(C(=O)N1CCCC(C(=O)NC2CC3(CC3)C2)CC1)(C(C)(C)C)OC CC1(C)CCCC(CC(=O)NCC(=C2CN(C(c3cnnc(O)c3)=O)C2)F)O1 N(C(=NCCC1CCCCCC1)NCC1(F)CCC1)C(C=C)C C(=O)(C=CS(C)=O)NCC(CNC(c1ncc(Br)cn1)=O)OC C(CCCCCC(=O)NCC1CN(C)CCO1)NC(CSCC=C)=O c1(C(=O)NC(CCN(C(C2N(CC)CCOC2)=O)C)C(C)C)cc(O)cc(Cl)c1 C(CCCC(=O)NC1CC(CNC(c2ccccc2OC(F)F)=O)C1(C)C)OC C1(CC(=O)NCCC2N(C(C(C)C(F)(F)F)=O)CCC2)COc2ccccc2O1 CC1CC2(CCN(C(=O)C(O)C3CC3)CC2)CN1C(C1CCCCCC(=O)C1)=O c1(CC(C(=O)NCCCC(C)NC(C2(CC)CC2)=O)C)cccc(F)c1 N1(C(CCC=C(C)C)=O)CC2CCC(CNC(=O)C#CC3CCOC3)(C2)C1 O=C(CS(=O)(=O)CC1COCCO1)N1CCCOC(CO)C1 C12(CN(CC(=O)OC)C(c3ccc(C(=O)NC)s3)=O)CCCCC1C2 c1(-n2c(C(c3n(C)ncn3)NCCC(O)C3CC3)nnn2)cccc(Cl)c1 N1(CCCC(C)O)CCCC2NC(=O)CC12.C123CCCC1N2C(=O)C3 Cc1nn(C)c(C)c1C(N1CCCCC(N(C)C(c2csc(C(F)F)c2)=O)C1)=O C1(OCCNC(C2CC(F)(CO)C2)=O)CCN(C(=O)CCn2ccnc2)C1 C1(NC(C2(C(F)(F)F)CC2)=O)C=CCN(C(C2CCSC2)=O)C1 c12cnc(Cl)nc1N(C)CC(=O)N2.C1(CC)CN(C(=O)C(C)SC)C1 c1(OC(C)C(=O)NC2CN(C(=O)C(C)(C)CO)CCC2C)cc(F)cc(F)c1 CS(=O)CCC(O)C(=O)NC1CC2(C1)CN(C(c1ccc(Br)s1)=O)C2 C1(NCC2(OC)CC(C(N)=O)C2)CC(C23CC(C2)C3)CN1 c1(C(=O)NC2CCCN(c3snc(SC)n3)C2C)csc2ccccc12 N1(C(C(C)OC(C)(C)C)=O)CCC2(CC1)CC(C)N(C(=O)C=CS(C)=O)C2 c1(CCC(C(=O)NCCOCC)N2CCC(CO)C2)cccc([N+](=O)[O-])c1 c1(C(=O)NC(C(=O)NC2CC(NC(=O)OC)C2)Cc2cnc[nH]2)n[nH]c(C)c1Cl N1(C(C(C)CN(C)C)=O)CC(NC(c2cccc(-c3ccco3)c2)=O)CC(F)C1 c1(C(N(CCCNC(C(C(C)C)N2CCCCC2)=O)C)=O)cccc(Cl)c1N CC1=NN(C)C(=O)C1CC(=O)NC1CC2(C1)CN(C(c1ccc(CO)nc1)=O)C2 O=C1CC2C(=O)NC1=CC=C(Br)C=C2N(CCCCCO)Cc1cn(CCCF)nn1 c1(C(=O)OC)ccc(C(N2CC(C)(NC(=O)Cc3ccc(C(C)=O)s3)C2)=O)s1 C1(C)(CNC(Cc2c(C)cco2)=O)CCCN1C(=O)CCN(S(C)(=O)=O)C N1(C(c2cccc(OC)c2)=O)CCCC2C1CCCN2C(C1CC(Cl)(Cl)C1)=O C(CNC(c1[nH]c(C)nc1C(=O)OC)=O)(CC)(CC)NC(C(C)OCCC=C)=O N1(C(C(C)OCC(C)C)=O)CCCC(N(C)C(c2ccc(=O)n(C)n2)=O)CC1 c1(OC)ccccc1CC(=O)NCC(O)CCNC(=O)C(C)OCCN(C)C C12(C(=O)NCC(CC(=O)N(C3CC(C#N)C3)CC#C)O)CCCC1C2(F)F c1(C(=O)NCC(C)NC(C(CC)CCOC)=O)cccc2c(C#N)c[nH]c12 c1(C(N(CCN(C(=O)C(c2ccccc2Cl)=O)CC)CC)=O)ccc(NC)cc1 c1(N(CC(C)NC(=O)CC(c2nccs2)N(C)C)C)ccc(Cl)cc1[N+](=O)[O-] N1(C(c2cc(CNC(COCCCC)=O)sc2)=O)CC(C)(C)C1C(C)C C(C(=O)N(C(C)CN(C(=O)Cn1cc(C2CC2)nn1)C)C)(C(C)C)OCC C1(CC)CN(C(C2(O)CC2)=O)CCC1CNC(=O)C(c1ccc(F)c(Br)c1)C N1(C(c2c(CC)c[nH]c2)=O)CCN(C(c2ccc(Br)c(N)n2)=O)CC1CC CC(C)(C(=O)NC1CCCC1CNC(c1cc(Br)co1)=O)C1CCCCC1 c1(C(N2CC(NCC34CCN(CC3)C4)C(F)C2)=O)cc([N+](=O)[O-])ccc1F C(=O)(CCCCC(C)C)NCC1CCN(C(CC(C)(C)OC)=O)CC1C Cc1nn(C)c(N2CCOCC2)c1NC(=O)C(C)NC(C)CNC(=O)C(C)(C)F N1(C(c2c(C)occ2)=O)CCN(C(=O)CC#N)C(c2ccncc2)C1 c1(C(N(CCC(=O)NCC(O)CC(C)C)CC=C)=O)ccc2occc2c1 c1(C(=O)NCC(CNC(c2n(CC)cc(Cl)c2)=O)(C)C)cc(F)ccc1N N1(C(C(C)N(C(=O)CCCC2CCCC2)C2CC2)=O)C2CCC1CC(N(C)C)C2 c1(C(=O)NC2CCC(CNC(c3c(C)nccc3)=O)C2)cnc2c(c1)CCCC2 N1(C(c2c(N)nccc2)=O)CCCC2(NC(c3cc(Cl)no3)=O)CCCC12 Cc1nn(C)c(F)c1C(=O)NCC(C(C)C(C)C)NC(=O)CN1CCCCC1=O c1(C(=O)NCC2(C(=O)NCCCCOCC)CC2)cccc(F)c1 c1(NC(CC(C)(C)NC(c2cc(CC)sn2)=O)=O)cc(C#N)ccc1C C1(NC(=O)Cc2sccc2Cl)CC2CC1CN(C(c1c(F)cc(F)cc1F)=O)C2 c1(C(=O)NCC(CN(C(=O)C(c2cccs2)SC)C)O)cnc2ncc(Cl)cn12 C1(NC(CCc2cccc(OC)c2)=O)CN(C(=O)C(CSC)OC)CC12CCC2 C12(C(=O)NC3CN(C(c4cnn(C)n4)=O)C3)CC=CC(C1)OC2 CC1(CNC(=O)C2=CCCC2)CCN(C(=O)CCNC(c2ccccc2Cl)=O)C1 N1(C(=O)NCC2(C(=O)O)CCOC2)CCCCc2cc(Br)ccc21 N1(C(C(SC)SC)=O)C2CCC(C2)C1CC(=O)NOCC1CCCC1 C=C=CCC(=O)NCCCN(C(c1ncc[nH]1)=O)C(C)C c1(C(C2CC2)NC(C2SCCN(C(CCCC=C)=O)C2)=O)cccc2ccccc12 c1(C(N(CCCCNC(c2c(CC)n(C)nc2)=O)C)=O)ccc(OC)nc1F c1(C(N2CCC(CNC(C(C)CF)=O)C2)=O)cc(F)c(F)c(C#N)c1 c1(C(N(CCNC(C(C)(CO)OC)=O)C)=O)cc2ccncc2[nH]1 C1(OC)CCN(CC(=O)NC2(C(=O)N(C)Cc3nnc(O)o3)CC2(C)C)C1 C(=O)(C1=CS(=O)(=O)CCC1)NC1CCC(N(C(Cc2c(C)non2)=O)C)CC1 Cc1n[nH]cc1C(=O)NCC1CC(O)(CNC(C2CC2(Cl)Cl)=O)C1 C(=O)(C(CC)(CC)CO)N(C)CC1N(C(c2c(CCC)occ2)=O)CC(F)C1 C(=O)(C(C)(C)C(C)C)N1CC(CCNC(c2cc(SC)n(C)n2)=O)C(C)C1 N1(C(C=CC(N)=O)=O)C2CCC1CN(C(=O)CCCC1CCOCC1)CC2 C(CC1=CCN(C(=O)CC(C)(C)F)CC1)NC(c1cc(C)c(C)nn1)=O c1(C(N2C(CNC(C(N3CCOCC3)C)=O)COCC2)=O)ccc(S(C)(=O)=O)[nH]1 CC(C)CC(O)C(=O)N1CC(O)CC1CC(N1CCCC(OC2CC2)C1)=O N1(C(C2C(CNC(C(CC3CCC3)OC)=O)CC2)=O)CC2CC1CC2O C(C(F)(F)C(F)(F)F)OCCC(=O)NCCNC(C1C(NC(CSC)=O)C1)=O CC(C)(CCC#N)C(=O)NCCNC(c1c[nH]c2cncnc12)=O C1(C(N2C(CNC(c3occ(C)c3)=O)C=CC2)=O)CCS(=O)(=O)C12CCC2 O=[N+]([O-])c1n[nH]c(=NCc2ccc(OCc3ccccn3)cc2)s1 C1(COC)(CNC(C2C3CCCC23)=O)CCN(C(C2CC2C)=O)CC1 c1(C(=O)NC2C(CNC(C3CN(C)C3)=O)CC2)cn(C)nc1C1CCCC1 N1(C(C(c2n(C)ncc2)O)=O)CC2CCCC2(NC(=O)Cc2cccc(F)c2O)C1 c1(OC)ccc(Br)cc1C(=O)NCCC1(NC(=O)CCC(C)(C)C)CCC1 C1(=CC(=O)NC2CCN(C(CS(CC)=O)=O)C2)CC2CCC(C1)N2C C(C(=O)NNC(=O)C(C)(C)NC(=O)COCC(C)C)=CC.C CCC(C)(CC)C(=O)N(CCN(C)C(c1c[nH]c(C(N)=O)c1)=O)C(C)C N1(C(C=C(CC)C)=O)CCC(COC)(NC(c2sc(C(=O)OC)nc2C)=O)C1 C(=O)(C1=C(Cl)CCC1)NCC(CC(=O)N(CCOCC)CC)C c1(C(=O)NCCC(CNC(=O)COc2cccnc2)O)ncn2c1CCC2 Nc1cc(=O)nc(C(=O)NCCCCNC(C2CCCN2N=O)=O)[nH]1 C(CCN(C(=O)C(C)(Cc1ccccc1)c1ccccc1)C)(C(C)C)NC(C)=O CC1=C(C(=O)NC2CCCCC2NC(=O)C(=Cc2cn(C)cn2)F)CCO1 CC1(C)CCCC1C1CCN(C(c2nnn3ccccc23)=O)C1 C1(NC(CSC(C)C)=O)CN(C(c2csc(Cl)c2)=O)CCC1O Cc1cc(F)ncc1C(=O)NC1(C)CC(NC(C2CN(C(C)C)CCO2)=O)C1(C)C C1(C(N(C)C2CC2)=O)COCCC1NC(=O)CCc1ccc[nH]1 C1(C(F)(F)F)(C(=O)NC2CCC(NC(C)=O)CC2)CC2CCC1C2 CCC(CC(=O)Nc1cn(CCOC)nc1C)N(C)C(c1cncc(CO)c1)=O C=CCC(C(=O)N1CC(CC=C)(NC(c2cnc(C3CC3)[nH]2)=O)C1)NC(C)=O C1(CNC(C(C=C)OC)=O)(NC(c2cnn(C)c2SC)=O)CCCCC1C c1(NC(CC2CCC(NC(=O)Nc3ccc(C)o3)C2)=O)cnn(C)c1Cl O=C(C1=C(Cl)CCC1)NCCC1CCCN1C(=O)C(c1ccc(Br)cc1)O C1(=CC(=O)NC(C(=O)NC(CCOC)C)c2ccco2)CCC(C)C1 N1(C(C2C(COC)C2)=O)CC2CC(NC(c3cccc4nsnc34)=O)CC1C2 c1(-c2c(C(N(CCC)CCNC(=O)CNS(C)(=O)=O)=O)cno2)ccc(F)cc1 CCC(CNC(C1CNC(=O)CN1C(=O)C(=O)NOC)=O)C(C)(F)F C1(CNC(c2cncc(F)c2)=O)CC2(CCC2)CN1C(c1cc(Cl)nnc1O)=O C1(C(=O)NC2CN(C(c3cnc(F)c(Cl)c3)=O)C2)C2C3CC4C1C1C2CC3C41 C1(NC(CCOC)=O)CC(CNC(=O)CCC2CCCCO2)C(O)C1 CN1CC2(CCN2C(=O)CCC2(C)CCCN2C(=O)CCc2ccc[nH]2)C1 C(C(COC)CC(=O)N(CC(C)O)CCNC(C1CC1CC(C)(C)C)=O)OC N1(C(C(C(CC)C)C)=O)CCN2CCN(C(c3cccc4nsnc34)=O)CC2C1 Cc1sc(=O)n(CCC(N2CC(NC(=O)CCc3cnc(O)[nH]3)CC2C)=O)c1C c1(CCN=C(NCC2(SC)CCC2)NCc2ccco2)cccc2c1OCCO2 C12CCCC(C1)CC(=O)N1CCC(C1)CN2.CCS(=O)(=O)N(C(=O)C(F)F)C c1(CCC(=O)NC(C2CCN(C(COCC)=O)C2)C2CCCC2)cccc(Cl)c1 c1(C(=O)NCCCN(C(=O)C(C)CC(=O)NC(C)(C)C)C(C)C)cc(F)c[nH]1 C(CC(O)C(=O)NCCC(O)C(F)F)NC(C(C)(C)c1ccno1)=O C(=O)(C(C#N)C(C)C)N(CC(C)O)CCNC(c1oc(C)c(Br)c1)=O CCC(O)C(C)C(=O)N1CCC(C)(NC(=O)C=CCn2cncn2)C1 c1(C(N2C(CCNC(=O)CCc3nccs3)CCC2)=O)ccc(O)c([N+](=O)[O-])c1 c1(OC)ncc(Cl)cc1C(=O)NC1(C)CCN(C(=O)Cn2ccccc2=O)CC1 Cn1ccc(=O)cc1C(N1CC2CCC2(CNC(c2cc(Br)cnc2Cl)=O)C1)=O C(=O)(CCC1=NNC(=O)CC1)N1CCCC2(CN(C(c3c(CC)[nH]cc3)=O)C2)C1 c1(C(N(CC(C)O)CCNC(=O)Cc2cn[nH]c2)=O)cnc2cccnn12 CC(C)CC(CNC(C1CN(C(N)=O)C1)=O)NC(C1CCC1C#N)=O c1(NC(c2ccc(-c3nncs3)cc2)=O)ccc(F)c(Cl)c1F N1(C(CCOCC)=O)CCCC(CC(N2CC(O)CC2C(C)C)=O)CC1 CS(=O)(=O)CCCCCN=c1[nH]c(NC2CCC3CC23)nc2c1CCCC2 c1(CSc2ccc(OC)cc2F)ccc(C)c(C#N)c1 C(CNC(c1cc(C(C)(C)C)oc1C)=O)(C(C)C(C)C)NC(c1c(C)c[nH]c1)=O Cc1cc(C(=O)NC2CCCN(C(C3CC4CC4C3)=O)CC2)nc2[nH]nc(O)c12 C1(C(=O)NC2(C(C)(C)OC)CC2)CCCCC1(C)NC(c1cc(C)nc(O)n1)=O N1(C(COC2(C)CCCC2)=O)CCC(O)(CNC(C23CC(C#N)(C2)C3)=O)CC1 N1(C(c2scc(C)c2)=O)CCC2CN(C(=O)Cn3ccc(Br)cc3=O)CC12 N1(C(CCc2c(C)noc2)=O)CCC2(CNC(=O)COC3CCC3)CCCC12 C(=O)(CC(C(F)F)n1ccnc1)N1CCC(C(C)(C)Nc2ncncc2Cl)C1 C1(NC(C2(C)CSC2)=O)CCCCN(C(=O)CCCSC(C)(C)C)C1 c1(NCc2cn(C(C)C)nc2)cccc2c1CCN(CC(=O)NCC#N)C2 CCC(C(=O)OC)C(=O)NCC(C1CC1)NC(c1ccc(C)[nH]1)=O c1(C(=O)OCC(=O)C2CC2)c[nH]c2ccccc12.c1(SCC2CC2)ccc(O)cc1 c1(NC(C2CCN(C(C3N(C(C)C)CCCC3)=O)C2)C)c(Br)cccc1[N+](=O)[O-] c1(OC)cc(C(=O)N(C)CC2CCCN2C(C2CCSC2)=O)cnc1O Cc1nc2c(O)cc(C(=O)NCCN(C(C3CC3F)=O)C(C)C)cc2n1C N1(CCCNC(c2cccnc2)=O)CCC(NC(C2CC(F)C2)=O)CC1 c1(C(N2CCOCC2)C)cccc(CN2CCOC(c3cccs3)C2)c1 CCCCCCC(CNC(=NCc1cc(Cl)ncc1Cl)NC1CC1)CC Cn1cnc2cccc(C(N3CCCCC3CNC(C3CC(=O)C3)=O)=O)c12 C1(CC(N2CC(CCC)C2)=O)CN(C(=O)Cc2scnc2C)CC12CC2 C1(CC)COCCN1Cc1cccc(N(C)CC2CCCCN2CC)c1 c1(C(=O)Nc2c(C#N)cc(I)cc2)cn2cccc(-c3cnc(F)c(F)c3)c2n1 C=CCC(C(=O)N1CCCC1C(C)NC(=O)C(C)(C)n1ccnn1)NC(C)=O C(=O)(C(F)(F)CC(C)C)NCC(CNC(c1cc(OC)n(C)n1)=O)CO CCC(C)(CNC(=O)CCc1cnn(C)c1)NC(c1cnc(C2CC2)o1)=O CC12CCC(C(=O)NCC(=O)NC(c3ccccc3)C(=O)O)(CC1)CO2 N1(CC(=O)N(CC=C)CC2CC2)CC(NC(=O)Cc2ccc(C(C)=O)s2)CCC1C Cc1cc(C(N2CCCC(CN3CCCC3)C2)=O)ccc1-n1cncn1 Cc1ccc(C(=O)C(=O)N2CC(C(=O)Nc3cccc(O)n3)C2)cc1 c1(CNC(CC(CNC(CCN(C)CCO)=O)(C)C)=O)ccc2ncnn2c1 Cc1ccc(C(=O)NCC(C2CCC2)NC(=O)COCc2nccs2)n1C N1(C(C=CC)=O)CCC(CNC(C2(c3cnn(CC)c3)CCNCC2)=O)CC1 C(C)(C)(C(=O)NNC(=O)CCS(=O)(=O)NC1C(C)C1(F)F)OC(C)C C1(C(=O)NCC(CCNC(CC(=C=C)C)=O)(C)C)CC2CCCN(C1)C2 Cc1cc(C(N2CCC(NC(C34CC(C)C3C4)=O)C23CC3)=O)cc(C)n1 c1(C2(C(=O)NC3CC(CNC(=O)Cc4ccsc4)C3)CC2)ncccc1F CON1CCC(C(=O)NC(CCOC)C(N2CC3(C2)CN(C)C3)=O)CC1 C=C(Cl)CC(C(=O)NCCNC(=O)CO)NC(=O)CCC(N)=O.C(C)(=O)N S(=O)(=O)(c1ccc(NC(c2cncnc2)C)c(C)c1)N(CCN(C)C)CC N1(C(C=CCCC)=O)CC2(CC(NC(=O)C(O)CCCc3ccccc3)CO2)C1 CC(C(=O)N1CCOC(CN(C)C(c2ccn(CCF)n2)=O)C1)C(F)F c1(C(=O)NCC2(F)COCCN(C(=O)C=CCO)C2)ccc2[nH]ccc2c1F c1(C(=O)NC2CC3(C2)CN(C(C2CC4CCC4C2)=O)C3)csc2ccc(F)cc12 c1(C(N2CCN(C(c3c(C)nsc3)=O)CC2CO)=O)ccc2cnsc2c1 c1(NS(CCOCCOC)(=O)=O)cc(COCC(=O)NC(CC)CCO)ccn1 N1(C(CCCCC=C)=O)C2CC=C(C(=O)NOC3CC3)C1CC2 c1(C(=O)NC(C)(CNC(=O)C(F)n2cccn2)CO)occ2c1CCOC2 CC1(NC(=O)Cc2nc[nH]n2)CCCCC1C(=O)NCCn1cc(CO)nn1 c1(CC)occ(C)c1C(N1CCN(CCN(C)C(c2cc(Cl)sc2Cl)=O)CC1)=O CCCCCC(O)CC(=O)NCC(C)N(C)C(c1c(Cl)csc1Cl)=O N1(C(C(CCCC)O)=O)CC(NC(=O)C=Cc2ccc(SC)s2)CCC(O)C1 C1(C)(CN(C(c2cnc(C(C)C)[nH]2)=O)C)CCCC1NC(=O)CCn1cnnn1 C1(C(=O)NCCN(C(c2c(Cl)cn(C)n2)=O)C2CC2)CC12CC(F)(F)C2 N1(C(CCc2ccc(C#C)cc2)=O)CC2CCN(C(c3nc(C)nn3C)=O)CC12 CC(CC(F)(F)F)C(=O)NC1CC2CCC1CN2C(C1CC(F)(CF)C1)=O C1(C(=O)NC(CCSC)C(=O)NC2CC(C)(C(N)=O)C2)CCC2(CCC2)C1 c1(OC)ccc2[nH]c(C(=O)NC3C4CC5CN(C(=O)C=C(C)Cl)C3C5C4)cc2c1 C(=O)(CC(C)(C)CNC(=O)CC1(OC)CCC1)NCC(CC)N1CCCC1 N1(C(COC)=O)CCC(C(C)CNC(=O)Cc2cc(C)[nH]n2)CC1 N1(C(=O)OCCCC)CCN(CCC(c2cccc(C)c2)CF)CC1.C=O c1(C(N(CCNC(c2ccc(C)cc2)=O)CC)=O)ccc2c(c1)NC(=O)C2 Cc1ccc(CN2CCC(NCc3ccc(OC(F)(F)F)nc3)C2)c(C)c1 c1(C(N2C(CNC(C(CCC=C)(F)F)=O)CCC2)=O)ccc2c(c1)NC(=O)CN2 C1(NC(=O)CCc2cccc(F)c2)CC2CN(C(c3ccnc(F)c3Cl)=O)CC12 N1(C(C=C(CCN(C)C)Cl)=O)CC2CC(NC(c3coc(CO)c3)=O)CC1C2 C#CCC(C)(C)C(=O)NC(C)CCCNC(=O)CNS(=O)(=O)CC CC1CN(C)C(C)CC1NC(c1coc(CNC(=O)Cn2[nH]cnc2=N)n1)=O C12(C(N3CCCC(OCC#C)C3)=O)CC(CO)(CN1C(=O)C#CC(C)(C)O)C2 C1(C(=O)NCC(CO)NC(=O)CNC(c2ccc(Cl)nc2)=O)CCCCCCC1 N#Cc1ccc(NC(C2CC23CCN(Cc2cccc(F)c2I)CC3)=O)c(F)c1 Cc1ccc(CC(C)(CO)NC(=O)CC2(O)CN(CC(=O)OC(C)(C)C)C2)cc1 c1(C(=O)NCC2CCN(C(C3(O)CCOC3)=O)C2)cc2c(F)cccc2s1 C(C(N=[N+]=[N-])C(=O)N1CCN(C(=O)Cc2c[nH]nc2C)C(CCO)C1)OCC C1(CNC(CCOC)=O)CCCC2CN(C(C34CCC(CC3)C4)=O)CC12 C1(NC(C2CCC23CCC3)=O)(CCCNC(=O)Sc2ccccc2F)CCOCC1 C1(C(=O)NCC2(C(N3CCC(C4(C)N=N4)C3)=O)CCCCC2)CCCCC1(C)C C1(C(=O)NC2CC(C)(NC(c3cnc(Cl)s3)=O)C2)CN2CCCN1CC2 c1(C(=O)NC(CNC(C(CC)SC)=O)C2CCC2)cc2c(c([N+](=O)[O-])c1)OCO2 CC(C(=O)N(CCCN(C)CCN(C)C)C(C)CO)C1CC1 c1(C(N2CCN(CCNC(C(C)(C)OC)=O)CC2)=O)sc2nccn2c1C N1(CCC#C)CCC(CC(=O)NCC(C)(O)CNC(C2CC(O)C2)=O)CC1 N1(C(c2cc(C)sc2C)=O)CCc2ccc(CC(N3CCOC(O)C3)=O)cc2C1 C1(C(=O)NC(C)C(C)NC(C2(SC3CC3)CC2)=O)(OC(C)C)CCOC1 Cc1cn2c(n1)C(C(=O)N1CCCC(CNC(c3cc(C)[nH]n3)=O)CC1)CCC2 C(=O)(CS(=O)c1ccc(Cl)cc1)NCC1N(C(c2ncc(C)cc2F)=O)CCC1 c1(C(=O)Nc2cccc(CNC(=O)C(F)=CCCF)c2)cnc2[nH]cnc2c1 N1(C(c2c(OC)c(F)c(Br)cc2)C(=O)NC2CC2)CCc2ccc(C#N)cc2C1 Cc1ccoc1C(=O)NCC(C)(C1CCC1)NC(c1cnn(CCF)c1)=O C(CCC(C)(C)C(=O)NC(CO)C(C)(C)C)NC(c1n(CC)nc(C)c1)=O N1(C(C2C=CCN(C(c3cc(C4CC4)[nH]n3)=O)C2)=O)CC(F)(F)CC1CO c1(OCCC(=O)NC2C3CN(C(C(C)=CC)=O)C2C3)ccc(Cl)cc1CC CC1CC(C(=O)NCCCOCCNC(=O)C2=C(Cl)CC2)C1(C)C C(C)(C(=O)N1CC(C)(NC(=O)CC2CCCOC2)C1)(C(C)C)OC S(=O)(=O)(c1ccc(C#N)cc1)NC1CN(C(c2c(C)nccc2)=O)C1 c1(NC(C(N2C(CC(=O)NCCC(N)=O)CC2)=O)=O)cscc1Cl N1(C(Cc2c(C)ccs2)=O)CCC2(CCN(C(c3cc(CF)on3)=O)C2)C1 CCC(C)(COC)C(=O)NC(CCCNC(=O)C(C)OCOC)C Cc1nnn(C)c1C(=O)NCCC1CCC(NC(=O)C=C2CCOCC2)C1 CCC(C)CC(=O)C(=O)N1CC2CC(NC(=O)C(CC3CCCC3)OC)C1C2 c1(NC(CSC)C)ccc(Br)c(S(=O)(=O)N(N2CCC(C)C2)C)n1.OC CC1=C(C(=O)NCC2CC(NC(c3cc(C(N)=O)ccn3)=O)C2(C)C)CCC1 C1(CC(=O)NC2CC(NC(C(C3CC(F)(F)C3)OC)=O)C2)OCCC1(C)C C1(NC(CC2C(CC)C2)=O)CC(O)CN(C(c2cc(C)nc(C)c2)=O)C1 N1(C(C(C2CCCOC2)OCC)=O)CCCN(C(=O)CCn2ccnn2)CC1 C(CN=c1[nH]c(=NCCC2CSCCO2)[nH]c2c1CSC2)(C1CCC1)OC c1(OC(C(=O)NCCC2CC(NC(c3n(CC)ccc3)=O)C2)C)cccc(F)c1 C=CC1CN(C(C2(C)CCCNC2=O)=O)CC1NC(=O)CCOCC N1(C(c2nc(OC)c(C)s2)=O)C2CCC1(CNC(C1CC(C)C1)=O)CC2 CCCCCC(C)(C)C(=O)NC(C1CC1C(=O)Nc1ccc(C)c(CO)c1)C c1(C(=O)NCC(C)N(C(C(=O)NC(CC)C)C)C)cccc(-c2cnccn2)c1 C=CC(C)(C)CC(NCC1(OC)CCC1)C1CC1 c1(C(C)NC(C2CC2F)=O)n[nH]cc1C(=O)NC(c1nc[nH]n1)C C1(CNC(CSCCOC)=O)CN(C(C)=O)CCC1(C)C.C1(=O)C=CCN1 c1(NC(C(C(C)NC(c2cc(C)ncc2)=O)C)=O)c(C)cc(C)nc1C c1(-n2cc(CC3N(C(c4c(C)cncn4)=O)CCCC3)nn2)noc(=O)n1C C1(CCCC)CN(c2nncn2C2CC2)CCN1 C1(OC)CC(NC(=O)C(C)(C)N2CCCC2)CN(C(c2n[nH]c(C3CC3)n2)=O)C1 C1(NC(C2C(CNC(=O)CCc3cscn3)CCO2)=O)CC2(CCOC2)C1 C1(C(N2CCC(=C)C2)=O)CC(F)(F)CN1C(c1ncn(C)n1)=O C12(NC(c3cncc(C)c3)=O)CCN(C(=O)Cc3cc(CN(C)C)on3)CC1C2 n1(CC(=O)NC(C(C)(C)C)CNC(=O)CNC=O)ccc(O)nc1=O C12(C(N)=O)CCCC1(C(N1CC(O)(CCNC(c3cnc(S)[nH]3)=O)C1)=O)C2 O=C(C(F)CC1CCOC1)NC1COCC1C(=O)NC(C1CCCC1)CO Cc1oc(C(C)C)cc1C(N1CCC(N(C(=O)Cc2ccc(Cl)s2)C)C1)=O Cc1cc(C(=O)NCCN(C(=O)CP(C)(C)=O)C2CCCC2)n(C(F)F)n1 N1(C(C2CCOC2)=O)CC2(CCCN(C(C3(C(F)(F)F)CCCCO3)=O)C2)C1 C1(CNC2C=C(C)COC2)CCC2(CCOCC2)C1O c1(NC(C(CC#CC)NC(c2cc(C)c[nH]2)=O)=O)cccc2ccoc12 Cc1no[nH]c1=NC(=O)CCC(=O)N(C)Cc1cn[nH]c1 N1(C(C(CSC)O)=O)CCCC(C2CCCN2C(=O)CCC2CCCCO2)C1 C1(NC(C(CC)n2ccnc2)=O)CN(C(=O)CNS(C)(=O)=O)CC2(CC2)C1 c1(OC)ccccc1CC(=O)NC(c1ccc(CNC(=O)CC(C)F)cc1)CO c1(C(C(=O)Nc2c(C(C)NC(C3CC(OCC)C3)=O)noc2)=O)ccc(C)cc1 N1(S(=O)(=O)CCC2CC3CCC2C3)CCC(O)C(CN2CCCC(O)CC2)C1 c1(C(=O)NCC2CC(CNC(C(C)SCCCC)=O)C2)cocc1C CC1=NS(=O)(=O)NC(C)=C1CCC(=O)NC1(CNC(C2CC2F)=O)CCCC1 c1(C(=O)Nc2c(OC)nsc2)cccc2c1NC(=O)CC2 CN1CCC2CC1CN2C(c1cc(C(=O)CCCc2ccccc2F)c[nH]1)=O N1(C(CN(C(COCC)=O)CC)=O)CCC(C(N)=O)C(C)(C)C1 C(C)(C)(CC(=O)NCc1cc(CC(N2CCC(C(C)CO)CC2)=O)on1)OC N1(C(Cc2c(C(N)=O)nccc2)=O)CC2CCC(C1)N2C(c1ccc(O)nc1)=O N1(CCNC(C2C(CC)CCC2)=O)CCCN(C(=O)C(C)(C)C(C)O)CC1 c1(CC(C)C)nc(C(=O)NCC2CC2CNC(=O)C=C(Cl)Cl)cs1 C(CC(C)C)(C(=O)NCCc1cn[nH]c1)NC(C1CCC(C)(CC)O1)=O c1(C(N2CC(COC)OCC2)C(=O)NC2CCOC2)ncc2ccccc2n1 N1(C(c2n(C)cnc2)=O)CC2(CCN(C(=O)CSCCC#N)CC2)C1 Cc1nc(C(=O)NCCN(C(c2ccnc(C(C)C)c2)=O)C2CC2)c(C)o1 N1(C(C=CC=CC)=O)C(C(=O)NCc2cncc(F)c2)CCC1C c1(C(N(C)CC=CC(=O)NCC23CC(CO2)C3)=O)cnn(C)c1Br C(=O)(C(C)C(F)(F)F)N1CCC(NC(c2cnc(-c3c(OC)cccc3)s2)=O)CC1 c1(COC)ccc(C(=O)NCC(C(C)C)NC(=O)C(=O)Nc2ncc[nH]2)[nH]1 C(=O)(C(O)COC(C1(CCNC(C=CC)=O)CC1)=O)NCc1ccccc1 C1(NC(c2c(C)nn(CCO)c2)=O)CC2CC1CN2C(=O)Cc1ncoc1C c1(C(=O)NC(CC=C)CNC(c2ccc(SC)s2)=O)cc2sc(Cl)cc2[nH]1 CCC(O)(CC)C(C)(C)CNC(c1cc(OC)nc(C)n1)=O Cc1ccc(C=CC(=O)NC(CNC(=O)CN(C)C(C)C)CC(C)C)cc1 C12(C(=O)NC3(C)CSC3)CC1CN(C(c1ccc(CO)nc1)=O)C2 Cc1n[nH]cc1CC(=O)NC(CC1CC1)C(=O)NCCC(CO)OC(=N)O N1(C(C2(NC(c3ccn(CC)c3C)=O)CCOCC2)=O)CCC2CC1C(=O)O2 C(=O)(C1=C(Cl)CCOC1)NCCCCC12CCC(CC1)S2(=O)=O.CCC(C)(O)C(=O)O c1(C(=O)NC2CC(C(N(C)Cc3cnn(C)c3)=O)C2)cncc(Cl)c1 C(=O)(C(C)(F)C(=O)NC1CCCC1CNC(=O)C(=O)Nc1ccc(C)cc1)OC c1(C(N(CCCCNC(C2(O)CCC2)=O)C)=O)cc(-c2ccccn2)no1 C1(c2nnc(-c3cn(C4(C(C)C)CC4)nn3)o2)COC2CN(C(C)(C)C)CC12 N1(CCCCNC(C=CC=CCC)=O)CCCN(C(c2sccc2Cl)=O)CC1 Cc1ccc(CC(N2CCC(N(C(=O)CNC(=O)CC(C)C)CCO)C2)=O)o1 N1(C(C2C(C=C)C2)=O)CCC(COC)(NC(=O)COc2c(C)occc2=O)CC1 N1(C(COCCSC)=O)CCCCC2C1CCCN2C(=O)CCC(N)=O C(=O)(C1CCc2cc(Cl)ccc21)NCCOCCOCC(=O)NCC(CCCO)O C=CCCCCN(C(=O)CN(C(=O)Cn1nccc1C)C)C C(=O)(C(CC(C)C)N(C(=O)C=Cc1ccc[nH]1)C)NCC(CC)(C)CO C1(NC(Cc2c(C)ncs2)=O)CC2CC(C1)N(C(=O)Cc1ccccn1)C2 N1(C(C(=O)NCCC)CCC2(C#N)CC2)CCOC(C)(C(F)F)C1 C1(NC(c2c(OC)scc2)=O)CCCN(C(c2ccc(C)cc2F)=O)CC1 N1(C(CCc2cn(C)nn2)=O)CC2CCC(C1)N2C(=O)CC1(c2ccccc2)CC1 C1(CC(=O)NCCCC(C)NC(C(CC)C)=O)CC2(C1)CC1(CCC1)C2 N1(C(=O)C=Cc2cocn2)CCC2CCCC12C(=O)NCCC(O)C(F)F Cc1cnc(Cl)[nH]c1=NC(CNC(c1cn(C2CC2)cn1)=O)C1CCC1 CC1CCCC1(c1nnnn1CC12CCN(CC1)CC2)Nc1ccccc1 c1(C(=O)NCCOCCCNC(C2(CC)CCCC2O)=O)ccc(F)c(NC)c1 c1(OC)cccc(C=CC(=O)NCC2(NC(=O)C(C)n3cccn3)CC2)c1 N1(C(C=CC(C)(C)OC)=O)C2CCC(C(=O)NCc3cc(C)c(C)s3)C1CC2 c1(NC(c2c(NCc3ccnc(SC)n3)nccc2)=O)ccc(I)cc1[N+](=O)[O-] c1(C(=O)NCC2CCC(C)N(C(c3ccsn3)=O)C2)ccc(Cl)cc1[N+](=O)[O-] N1(C(C=COCC)=O)CC(C)CN(C(c2ccc(C=CCOC)cc2)=O)CC1C c1(C(=O)NCC2CCN(C(c3n(CC)nnn3)=O)CC2)cc2ccc(Cl)cc2o1 C1(N(C(C=NOC)=O)C)CCN(C(=O)COCC(=O)OC(C)(C)C)CC1 n1(C2(CSC3CCC3)CC2)cc(Br)nn1.C12CC1C(=O)NCCNC2=O CC1CN(C(C2CCC3(CCO3)CC2)=O)CCN1C(c1ccccc1)=O C1(C(=O)NC2C(OC)COC2)CC2CCC1N2C(c1ccccc1CC#N)=O C1(CNC(C=CCC(C)(C)NC(CCOC(C)C)=O)=O)CCC(C)(C)O1 C(=O)(CCCCC(=O)N1CCC(C(C)(C)C)(CNC(=O)C(C)CC(C)C)C1)NC C(=O)(C(C)C(F)(F)C(F)F)N1CCN(C(c2ccc(CC)[nH]2)=O)C(CCOC)C1 O=S(=O)(c1ccc(F)c(F)c1)N1CCc2cccc(-c3ccc(F)nc3F)c2C1 N1(C(c2cc(C)oc2)=O)CCC(C)(C)C(NC(c2ccc(C)c(C)n2)=O)C1 n1(CC)ncc(C(=O)NC2CCC(NC(=O)C(=O)Cc3ccccc3)CC2)c1C c1(OC)ccccc1C(N1CCC1C(c1ncccn1)Nc1sccn1)=O C1(C(C)(O)CNC(=O)CCc2cc(Cl)no2)CCCN(C(c2ccc(O)cn2)=O)C1 N1(C(c2c(Cl)ncc(C)c2)=O)CCC2CN(C(=O)C=CCBr)CC12 N1(CCSC2CC3CCC2O3)C(=O)CN(Cc2ccc(CC)s2)C1=O C1(COC)(CNC(c2cc(OC)ncn2)=O)CCCN1C(C1CCCC(C)C1)=O c1(NC(N(CC(F)(F)C(F)(F)F)CC)=O)cccc2c(C)ccnc12 C1(NC(C(CC)OCC)=O)CN(C(=O)C(C)NC(C)=O)CC2(CC2)C1 N1(C(C=C(CC)C)=O)CCCN(C(C2CCS(=O)(=O)N2C)=O)C(C)C1 c1(C(=O)NC2CCCCC2NC(=O)C(F)F)ccc(F)c2cccnc12 C1(CNC(C(CNC(C(COC)OC)=O)CC2CC2)=O)CC2CCCC2C1 C(CS(=O)(=O)CC(=O)N(C1CCCN(C(c2nonc2N)=O)C1)CCO)OC N1(C(C2(NC(c3ccn(COC)n3)=O)CC2C)=O)C2CCC1CC(CO)C2 Cc1cc(CCN=C(NCc2ccccn2)NC(C)C)ccc1Cl N1(C(CN2CCC(C)(C)C2)=O)CCC2(CCCCN(C(=O)CC(F)F)C2)C1 CC1(C(=O)NCCC2CCCCN2C(=O)C=CC(=O)N(C)C)CC=CCO1 C(=O)(C1=COCC1)NCCC(Cc1ccccc1)NC(Cc1c(C)occ1)=O N1(C(CC2CCC(C)C2)=O)CC2(CNC(c3cc[nH]n3)=O)CC1CCO2 c1(C(C)C(N2CCOC(CNC(=O)CCc3nncs3)C2)=O)ccc(F)c(F)c1 CCCCCCCC(=O)NC1CN(Cc2cccc(I)c2F)CC1F c1(CC(N2CCC(C(C)NC(C(C)NC(=O)NC)=O)C2)=O)ccccc1Cl N1(c2ncc(C(=O)OCC)s2)CC2CCCC(NC(=O)Cc3csc(S)n3)C2C1 C1(C(N(CC(CO)(CO)NC(c2cc(C(N)=O)n[nH]2)=O)C)=O)CCCNS1(=O)=O c1(C(=O)OCC)ccc(CNC(N2CCC2Cc2cc(Cl)c(C)cn2)=O)c(F)c1 C1(CNC(c2c(C)c[nH]c2)=O)CN(C(c2cnn(C)c2C2CC2)=O)CCCO1 N1(C(c2cc(CC)[nH]n2)=O)CCC(C)C1C(=O)NCCCOCC(F)F Cn1c(C(=O)N(C2CCC(NC(C3CC(F)(CF)C3)=O)C2)C)cnc1O C(CC(F)F)(C(=O)NCCC1CC(O)C1)N(C(c1cc(C)sc1N)=O)C c1(C(=O)NCC2(O)CN(C(C3(OC(C)=O)CC3)=O)C2)cccc(C(C)(F)F)c1 CC(C)CCCC(=O)NC1CC(NC(C2CC2C(C)(F)F)=O)C(O)C1 N1(C(CC)=O)CCC(CO)(CNC(C2CCC(=O)O2)=O)CC1 CC1COCCC1CNC(=O)C(c1ccccc1)N1CCCC1 C1(C(N2CC(CC(=O)NCC(=O)OCCCC)OCC2)=O)CC2CCC(C1)O2 C1(CNC(c2nc(C)oc2)=O)CN(C(=O)Cn2cccc2)CC(C)(C)O1 CCCCC(O)C(C)C(=O)NCC1(O)CN(C(c2ccccc2OCCC)=O)C1 c1(CCCC)nc(C)c(C(=O)NC(C)(C)CNC(c2cnc(O)s2)=O)s1 C1(CC=C)(NC(=O)CC(C)(F)F)CCN(C(=O)CC(c2ccc(CC)cc2)C)C1 N1(C(Cc2c(C)cccn2)=O)CC2CC1CCC2NC(c1c(C)nn(C)c1Cl)=O Cc1noc2nc(C(=O)NCC3(F)CN(C(=O)C(S(C)(=O)=O)C4CC4)C3)ccc12 N1(C(C2N(C(c3[nH]c(=N)sc3)=O)CC3(CC3)C2)=O)CCc2ccc(F)cc2C1 c1(C(=O)NC2CCN(Cc3cc(C)ncc3)CC2F)cnn2ccncc12 N1(C(c2c(C)nc(C(C)C)s2)=O)CCN(C(C2OCCN(C)C2=O)=O)C(C)C1 Cc1ccc2oc(C(=O)NCC(C)N(C(=O)C(c3cccnc3)C)C)cc2n1 c1(C(=O)NCCN(C(C2CN(CC)C(=O)N2)=O)CC)ccc2c(c1)NC(=O)CC2 C(CCC(C(=O)NCC(O)CC(C)C)NC(C1CCO1)=O)OC c1(-c2cc(C)cc(C)c2)cc(C(=O)NCC23CCN(CC2)C3)c2cc[nH]c2c1 CN1CCC(C(=O)NCC2CCC2NC(=O)Cc2csc(Cl)n2)C1=O n1(CC(=O)NCC(C(C)C)NC(C2CCCC2CF)=O)nnc2c1CCCC2 N1(C(C2C(CC)N(C)CC2)=O)CC(CNC(C2CC(O)C2)=O)OC2(CCC2)C1 n1(CCC)ncnc1C(CC1CCCOC1)NCc1nnnn1CCCF N1(C(C=CC(C)C)=O)CC(C(=O)NC(C)COCC2CC2)CC(C)(C)C1 c1(OC)ccc(O)c(C(=O)NC2CN(C(=O)CN(C)CCO)CC2O)c1 c1(C(N2CCC(C(C)NC(C(C(C)C)O)=O)C2)=O)cn2c(n1)CCC2 C=CCC(C(=O)N1CCN(CCCCNC(c2cscn2)=O)CC1)OC c1(C(=O)NC2CC3(C(NC(=O)CCF)C3)C2)cnc2c(=O)[nH]cc(CCO)c2c1 N#Cc1ccc(NC(c2sc(-c3ccc(F)cc3O)nc2C)=O)cc1Cl N1(C(CC=C=C)=O)CCCC(CN(C(=O)CCOCC(C)C)CC)C1 O=S(=O)(c1ccnn1C1CC1(F)F)Nc1nnc(-c2ccc(Cl)cc2Cl)s1 N1(C(CCNC(=O)OC)=O)CC(C(=O)NCC(O)C(C)(C)C)C(F)(F)C1.C(C)(=O)O C(c1ccc2nc[nH]c2c1)=CC=O.c1(C(CC(=O)OC)S)ccccc1Cl c1(OC)ccc(C(=O)C(=O)NCC2CCC2NC(C2CCOC2)=O)cc1Cl c1(C(=O)NCC#CCNC(c2ccc(OC)s2)=O)cccc2cccnc12 Cc1cc2c(C(N3CCC(C)(NC(C4C(C)C4C)=O)C3)=O)cccc2o1 c1(C(=O)NCCSCC(=O)NC(COC)CCO)ccc(C)c(C#N)c1 C(C)(N=c1[nH]c(Cl)ncc1Br)NC(C(CCC)Cc1ccccc1)=O c1(OCC(=O)N(C(C(=O)OC)C)C2CC2)nn(C)cc1NC(c1cc(C)n(C)c1)=O C1(C(N(C(C(=O)NC(C)C2CC2)(C)C2CC2)C)=O)C2CC(=O)CC12 c1(C(=O)NCC(C)CNC(C2CCC(C(N)=O)O2)=O)ncc[nH]c1=O c1(C(=O)NC(CC)(COC)c2ccncc2)cc(C(C)C)nc2onc(C)c12 CC1=C(C(=O)NCC2CCCCC2C(=O)NCC2OC(=O)CC2(C)C)COCC1 N1(C(c2n(C)ncn2)=O)CC2(CC(NC(c3noc4ccccc34)=O)CO2)C1 C1(CCOC)CN(C(=O)C(O)C2CCC2)CCN1C(C1C=CCC1)=O Cc1cc(C(=O)NC2CN(C(C3CCN(C)C(=O)C3)=O)CC2C)c(N)c(C)c1 c1(C(C(=O)NCCc2cc(C)no2)NC(=O)CC2OCCO2)c(C)cccc1Br CC(C)(C)C(=O)NCCNC(=S)NCCCNC(N1CCCC1)=O C(=O)(C1OC(=O)c2ccccc21)OCC.C(=O)(C1=CCC1)N1CC2(CC2)C1 c1(C(N2CCCC(CN(C(C(C)N(CC)CC)=O)C)C2)=O)cc2n(c1)CCC2 N1(C(C(C)SC)=O)CC2CC2(CNC(=O)CSc2ccccc2C)C1 C(=O)(C1CCCc2nn[nH]c21)NC1CC(CCNC(c2c(OC)cncc2)=O)C1 CS(=O)(=NC(=O)NCC1CCN1C1CCCC1)C1CCNC2(CC2)C1 C12(NC(c3cc[nH]n3)=O)CCC(CC1)N(C(=O)C(CC(F)F)C1CCC1)C2 c1(C2N(Cc3cn(C4C(=O)NCCC4)nn3)CCC2)ccc(Cl)c(Cl)c1 C1(C(=O)Nc2c(CNC(C(c3ccn(C)c3)C)=O)c[nH]n2)CC2CCCC2C1 C(=O)(CC(C)CC(F)(F)F)NCC1(C)OCCN(C(c2c(C)nncc2)=O)C1 C1(C(N2CC(C3(NC(=O)C(C)CC4CCCO4)CC3)C2)=O)(OC)CCCCCC1 N1(C(c2ccc(OCC)cc2)=O)C2CCC1CC(NC(C1(C)CC(F)(F)C1)=O)C2 c1(OCCC)ccc(C(=O)NCC)cc1.N12CCC1(NC(=O)C(CC)OCC)C2 N1(C(C2CCN(C(=O)NC)C2)=O)CCN(C(=O)CC2CCC(=O)N2)CC12CCC2 c1(NCC#C)ccc(F)c(C(=O)N(C2CCN(C(=O)Cc3ccsc3)CC2)C)c1 C(C(C(=O)N1CCOCC1)NC(=O)CCNc1ccsc1)N(C)C C(C)(C)(CC(=O)NC1CCN(C(C2CCC2)=O)C1)NC(CN(CCC#C)C)=O Cc1ccc(C(=O)NCCCCC(C)NC(C23CC(CN2C2CC2)C3)=O)c(Cl)c1 c1(CNc2c(C(=O)Nc3n(C)cnc3)n[nH]c2)cc(F)ccc1[N+](=O)[O-] C(=O)(C1=NNC(=O)CC1)NCC1N(C(C=Cc2n(C)ccc2)=O)CC1 C(N=c1cc(N2CCOC(C)CC2)nc(C)[nH]1)c1ccc(OC)c(OC)c1 c1(C(N2CCC(NC(CS(=O)(=O)NCC)=O)(CO)C2)=O)cc2ncn(C)c2cn1 C1(CC)CCN(C(=O)CC2CCCN2C(=O)C(C)c2ccco2)CC1 C(=O)(CCCC(=O)N1CCC1)N(CCC(c1cccs1)NC(C12CCC1CC2)=O)C N1(C(Cc2ccc(C(=O)OC)s2)=O)CC2CN(C(=O)CCCc3nccs3)CC2C1 C1(C(=O)NC2CCCC(CO)C2)CN(C(c2cc(O)nc(O)n2)=O)CC1(F)F CCCCCCCCC(=O)NC1COC2(C1)CN(C(C1(C)CC(F)C1)=O)C2 C#CCCCCCCC(=O)NC1CN(C(C2CC(N3CCCC3)C2)=O)CCC1C c1(OCC)ccc(C(N2CCC(F)(C(=O)NCC(O)COC)C2)=O)nn1 c1(CC(C(=O)NC(C)C)N(C2CN(C3CCC3)C2=O)CC)cc(C)cc(F)c1 C(=O)(C(C)(C)C(C)C)N1CCC(C(C)NC(C(CC)COC)=O)C1 CC1(NCC(=O)CCCF)CCCC1c1ccccc1 C1(C(CNC(c2cc(C(C)=O)on2)=O)F)CCN(C(=O)C#CC2CC2)CC1 C(=O)(CC(O)CC(C)(C)C)NCC(CC)(CC)NC(C12COCC1C2)=O c1(C(=O)NC2CC(NC(CC3CCN(C)C3=O)=O)C2)ccc(F)c(S(N)(=O)=O)c1 C1(NC(c2c(CC(C)C)n(C)nc2)=O)CC2CC(NC(=O)C(C)(C)C(C)C)CC12 C1(CCCCNC(c2c(C)scn2)=O)CCCN(C(C2COCCN2C)=O)C1 Cc1cnc(C)c(NC(C2CCN2C(C2CCN(C)C2=O)=O)=O)c1 C1(NC(C2CC(NC(CNC=O)=O)C2)=O)CCn2ncnc2C1 c1(C(N2C(CNC(C#CC(C)C)=O)CCCC2)=O)cn(C)c2ccccc12 c1(C(=O)NC(c2ccsc2)C)ccc(CNC(=O)C(O)CN2CCCC2)cn1 C1(C(=O)NC2CC3CN(C(C4(C(F)(F)F)CCCCC4)=O)CC23)CC2(CCC2)CO1 CCCC(CC1CCCC1)C(=O)NCCCN(C(=O)C(C1CCC1)OC)C S(=O)(=O)(c1cnoc1C)N1CC(C)CC(Nc2cc(C)nc(C)n2)C1 CC(CCC(C)(C)C)NC(c1cc(-c2ccc(F)cc2)nn1C)=O CC1=NNC(=O)C1CC(=O)NCC1(O)CCN(C(=O)CCc2cnn(C)n2)C1 C=CCC(C)(CC=C)NC(=O)CCC(C)(C)NC(=O)CC1CCC(=O)N1 Cc1nc(C)c(CC(N2C3CCC2C(NC(C2CCC(C(N)=O)C2)=O)C3)=O)c(O)n1 c1(C(N2C(CNC(c3nc(C)oc3C)=O)CCC2)=O)cccc2c(C)ccnc12 N1(C(Cc2c(C)scc2)=O)CCC(C(=O)NC2C(C)C2(C)C)C12CC2 N1(C(c2cc(C(C)=O)sc2)=O)CC2CC(NC(=O)CSSC)C(C2)C1 N1(C(CC2CN(C(C)=O)C2)=O)CCC(C(=O)NCc2ccc[n+]([O-])c2)CC1 Cc1cc2c(C(=O)NCC3CCN(C(C4CC5CCC4O5)=O)CC3)nccn2n1 c1(C(=O)OC)cnc(NC(=O)N=c2cc(-c3ccnn3C)[nH][nH]2)c(I)c1 CC1(CNC(=O)CC2CCC(C3CC3)O2)CCCN1C(c1cncn1C)=O C1(CNC(c2cocn2)=O)CC(F)CN1C(=O)CCc1cnc[nH]1 N1(C(CCCN(C)C)=O)CC(=O)CC1C(=O)NCc1cnn[nH]1 C12(OC)CCC(NC(=O)NCc3cn(C4CCC(OC)CC4)nn3)(CC1)C2 CCCC(CCC)C(=O)NC1CN(C(=O)C#CC2CCCO2)C2(CCC2)C1 N12CCCC(C)(C1)C2=O.c1(NC(c2scc(C)c2)=O)ccnc(Br)c1 C1(C#N)(C(=O)NCCCCC2CN(C(CN(C)C(N)=O)=O)C2)CC=CC1 c1(C(N2C(CCNC(=O)C#CC3CCC3)CCC2)=O)ccnc2ccc(Cl)cc12 C1(CCCC)CN(C(=O)CC2CCCCC2)CCN1C(=O)C(c1cncnc1)C c1(C(=O)NCCCN(C(c2cnc(C)o2)=O)C2CC2)cnc(S)n1C c1(C(C)NC(=O)CNC(C2(CNC(=O)C=CCF)CC2)=O)ccccn1 c1(OC)cccc(C(=O)NC2CCC(NCc3c(Br)ccnc3Cl)C2)c1Cl c1(C(N2CC(NC(c3nn(C(CC)C)c(C)c3)=O)C2)=O)cc2n(n1)CCCC2=O c1(C(=O)NC(CN(C(C2C(C)C2C)=O)C)C)coc2ccc(F)cc12 c1(C(=O)NC2CN(C(C=C(C)C)=O)CC2(C)C)c[nH]c2ccc(Br)cc2c1=N C(CCN=C(NCC(N1CCCC(C)C1)C)NCc1ocnc1C)OC C12(C(N(C3C(N)CCC3)C(c3ccccc3)=O)=O)CC3CC(C1)CC(F)(C3)C2 c1(Nc2cnn(CC)c2C2CC2)cc(F)cc(C)c1O c1(CC)ncnc(N2CCC(C)(NC(=O)C=CCN3CCCCC3=O)C2)c1F c1(NCC(CC=C)(C)C)ccc(S(=O)(=O)CN(S(C)(=O)=O)C)c(Br)c1 N1(C(C=Cc2ccc(C)o2)=O)CC2CC(N(C(=O)C(C)CN(C)C)C)C1C2 CC1CCN(C(c2cc(Br)n(C)n2)C(=O)NC2COC2)CC1C c1(OC)ccc(C(=O)NC2C3CN(C(=O)C(C)CF)CC23)cc1[N+](=O)[O-] C1(OCC(=O)NCC2(F)CC(NC(C=CC)=O)C2)CCCC(C)C1 c1(C(=O)NCC2(F)CCCN(C(C(CC)NC(N)=O)=O)C2)csc2cccnc12 CN(S(N)(=O)=O)CC1N(C(CNC(=O)C(C)(C)c2ccno2)=O)CC1 C1(C2CC2)(COC)CN(C(=O)C(=O)NC(c2ccccc2)COC)C1 C#CC1(F)CCN(C(C(=O)NCCCC2CC2)C2CC=CC2)CC1 CCC(CC)C(C)C(=O)N1CCC(NC(c2ccc(CN(C)C)nc2)=O)C(C)C1 N1(C(C(C#C)(C)C)=O)CCC(CCOCC)(NC(C2CC=CCC2)=O)CC1 C1(NC(CCN(CCC)C)=O)CS(=O)(=O)CC1NC(=O)CCc1cccc(O)c1 C(CC(F)(F)CO)NC(C1C(CNC(c2ccc(C3CC3)o2)=O)OCC1)=O C1(CNC(C(=Cc2cccs2)C)=O)CC2CCC1N2C(C1(OC)CCCCC1)=O Cc1ncnc(C(=O)NC2(C(N3CC=CC3)=O)CC(O)C2)c1C c1(NC(C2(C)CCN(C(C3(C)CC3)=O)C2)=O)nc2ccc(C#N)cc2o1 C(CCCC(=O)N1CCN(C2CCCN(C(=O)C(C)CSC)C2)CC1)SC C1(C(=O)NCC2N(C(C3N(C(N)=O)CCCC3)=O)CCC2)CCc2c[nH]nc2C1 c1(C(=O)NCCCCCNC(c2c(OC)noc2C)=O)cc2sccc2[nH]1 N1(C(COCCOC)=O)CC2(CC(CNC(C3CC4CCCCC34)=O)C2)C1 N1(C(CC(C)(C)C)=O)C2CC1CN(C(C1(O)CCSC1)=O)C2 C(=O)(CC(C)CC(C)(C)C)N(CCN(C(C)C)C(C1CCCN1C=O)=O)C C1(C)(C(=O)NC(c2ccccc2)CNC(C(C)(C)c2cnsc2)=O)CC=CCC1 C1(C(=O)NCCOCCCOC)CCN(C(=O)COC(CC)CC)C1CC Cc1ccc(CC(=O)NC2(C)CCCN(C(C3(Cl)CC3)=O)C2)cc1[N+](=O)[O-] CC1(C)OC(=O)CC1C(N1CC(C2CC2C(=O)NCCCN2CCC(O)C2)C1)=O c1(CC)[nH]c(C(N2CC(n3cc(-c4ccc(Cl)cc4)nn3)C2)=O)nc1C(C)C CC(C)CC(C)(CNC(=O)Cc1cccc(C#N)c1)NC(c1cn(C)nc1Cl)=O CC1CC(NC(=O)C=Cc2cncn2C)CN(C(=O)Cn2cnnc2O)C1 C1(CNC(C(F)=CC)=O)CN(C(c2cc(C)ncc2C)=O)CCC1(C)C N1(C(C(CN(CC)CC)F)=O)CCC(CC)(NC(c2cn(CCF)nn2)=O)CC1 c1(NCC)ccc(C)cc1C(N1CCC(NC(c2c(C)ncn2C)=O)C(C)C1)=O C(=O)(C(CC(F)F)N(C)C(C1CC(C)CO1)=O)N1CCC(SC)CC1 O=C(C1=NOC(C2(O)COC2)C1)NC1CCN(CCNC(c2cccs2)=O)C1 c1(C(=O)NCC2N(CC(=O)Nc3ccc(Br)s3)CCC2)ccnc2ccnn12 Cc1cccc(CNC(C2CN(C(c3cn(C)cn3)=O)CC2C)=O)c1C c1(C(N2C(CN(C(CCCOC(C)C)=O)C)COCC2)=O)ncc2n1CCCC2 C1(CNC(C(C)=C(CC)C)=O)CC(OC)CN1C(=O)CCCc1cccs1 c12ccc3c(ncn3c1)NC2=O.C(C(O)C(C)(C)O)NC(C=CC=CC)=O c1(OC)ccc(CC(=O)NC2CC(F)(CNC(=O)CN3CCCCC3C)C2)cc1 c1(-n2ncc(C(N3CC(OCCNC(C(CC)O)=O)C3)=O)n2)cccc(Cl)c1 C(=O)(CCC(=O)NCCOCCCNC(c1cc(Cl)ns1)=O)OC.OC CCCCCC(O)C(=O)NCC(O)CNC(C1(Cl)CC2CCC1O2)=O N1(C(CN(C)CC)=O)CC(C(=O)Nc2c(C)noc2C)CC2OCCC12 c1(SCC(N2C3CN(C(c4nc(OC)oc4)=O)C(C3)C2)=O)ncnc2[nH]cnc12 c1(CCNCc2nc(-c3c(O)ncc(Br)c3)on2)cnn2c1CCCC2 C(=O)(C1CCc2ccc(Cl)nc21)N1CC(CNC(C2C(COC)CC2)=O)C1 Cc1cccnc1CCNC(C1CCC(NC(=O)CCn2cccn2)C1)=O O=C(C=CI)NC1CCC1NC(=O)CCOCC1CCCO1 CC1(C(=O)NCC(CNC(c2ccoc2Cl)=O)CO)CCC(F)(F)CC1 Cc1cc(Cl)ncc1CNC(C1CCN1C(C)C)=O.c12cccc(c1O)N2 c1(C(=O)NC2CC(C)N(C(=O)CC3CC3(C)C)C2)ccc2ocnc2c1 CCCCS(=O)(=O)CC(=O)N1CC(NC(c2ccc(CCOC)cc2)=O)C(F)C1 CN1CC=C(C(=O)N2CC3CC3C2C(=O)NCC2(C(C)(C)O)CC2)C1 c1(OC)cc2c(cc1OC)N(C(C(=O)NCCC1(C)CC1)c1cnsc1)CCC2 c1(C(=O)NC(C)CC(C)NC(C2(Cl)CC2)=O)c(F)ccc2occc12 C1(C=O)CC12CCN(C(=O)C=Cc1cc[nH]n1)C2.C1(C(CC)N)CCOCC1 N1(C(C2CCC(C)CC2)=O)CCC(CO)(NC(=O)CC2NC(=O)NC2=O)CC1 C1(C(=O)NCC2COCCN2C(C2CC2F)=O)CCCC(F)(F)C1 c1(C(=O)NCc2cn(C(C(=O)NC)C)nn2)cnc2n1CC(CCC(F)(F)F)CC2 C(CCCC(F)(F)F)NC(C(C1CCN(C(C(F)=CCC)=O)C1)C)=O c1(C(C(N2CCC(CNC(C(CC=C)OC)=O)C2)=O)(F)F)ccc(F)cc1C CC1CC2(CCN(C(=O)C=CCCCCCCCO)CC2)CN1C(=O)C(Cl)=CCl c1(OC)cc(C(=O)NCC(C2CC2)NC(c2ccccc2C(C)O)=O)ccc1Cl c1(NCCN(C(C)C)C(c2csc(-c3ccccc3)c2)=O)ccc([N+](=O)[O-])cc1 C12(NC(c3ccnc(OC(F)F)c3)=O)CCCC1N(C(=O)C=CBr)CCC2 C(CN=c1[nH]c(=NC2CC(CC)C2)c2ccccc2[nH]1)SCCCC C12(CNC(CSCC=C)=O)CC(CN1C(c1cccc(-c3nccs3)c1)=O)C2 C1(C(=O)NC(CC(C)C)CNC(C2(c3ncco3)CC2)=O)CCCCN(C)C1=O CC1CC(NC(=O)CSc2nnnn2CC(F)(F)F)CN1C(=O)CSC1CCCC1 C1(NC(CCCN(C)C(C2CC3C=CC2C3)=O)=O)CC1C1CCOCC1 N1(C(C2(CC=C)CC2)=O)CCOC2(CCCN(C(C3CC3F)=O)C2)C1 CC1CC(NC(=O)CN2CCCC2)CN1C(c1ccc(C2CCOC2)s1)=O N1(C(Cn2cnc(=N)[nH]2)=O)CCOC2(CCC(NC(C3CCOCC3)=O)CC2)C1 N1(C(CCC(CC)NC(=O)CN2CC=CC2)=O)CCC(C)(C2CC2)C1 CON1CC(C(=O)NCCCN(C(=O)CCn2cc(C)cn2)CCO)CC1=O C1(CC(=O)NC(C2CCCCC2)C#C)CN(C(=O)C(O)C=C)CCO1 C(=O)(CC(C)(C)O)NC(C)CC(=O)NCC(C)(C)C1CC1 CC1(CC(=O)NCCCO)CCN(C(=O)CCc2ccccc2O)C1 CC1=C(C(=O)NCC(C)C(F)C(=O)NC(C)CS(N)(=O)=O)COCC1 c1(C(N(CC(CC)NC(C23CC(OC)C2C3)=O)C)=O)cc2c(=O)[nH]c(C)cn2n1 C1(C(=O)NC(CC)CNC(c2cc3c([nH]2)CCCC3)=O)Cc2c[nH]cc2S1(=O)=O Cc1cc(NC(c2cn(CCNC(C3CC34CC4)=O)nn2)=O)cc(C)c1 C(C(CC(C)C)NC(C1(n2cncn2)CC1)=O)SCC.C1CC(=O)N1 N1(C(CSCC#C)=O)CCC(C(C)(C)C)(CNC(C2C(C(C)=O)C2(C)C)=O)C1 N1(C(C(CC=C)OC)=O)CCC(C)(CNC(c2cncc(C)c2)=O)CC1 C1(NC(c2cc(C)ncc2)=O)CC2CC1CN(C(c1cc(C)c(Br)o1)=O)C2 c1(CNC(C2(c3cccs3)CC(=O)C2)=O)cccc(CC(F)(F)F)c1 C1(NC(C2C(OCC)C2)=O)CCC(C)(NC(C2CCCCC2)=O)CC1 O=C(C#CC1CCCCO1)NCc1ccc(CCNC(c2nn[nH]c2Cl)=O)cc1 C1(C)(OC)CCCN(C(=O)C(C(C)(C)C)NC(=O)COCC2CCCO2)CC1 Cc1cnc(N2CCCC(CN(C(=O)C(F)C3CCOC3)C)CC2)nc1C C(=O)(CCCC(C)CC)NC1CC(NC(CCCC)=O)C(O)C1 N1(C(C(CNC(c2ncc(CC)cn2)=O)(C)C)=O)CCCN(CC)CC1 c1(CCC)ccc(S(=O)(=O)N2CC(C(=O)NCC3CCCO3)CC(CC)C2)cc1 CC1(C)CN(C(=O)CC2C=CC(NC(=O)C=C3CCC3)C2)CCO1 CC1=NOC(CC(=O)NC(CNC(=O)CCC2CCCOC2)C2CC2)C1 C1(NC(C2(NC(c3cnc(OCC)s3)=O)CCCC2)=O)CC(=O)N(C2CC2)C1 C12(C(=O)NC3C(CNC(C4(COC)CCCCO4)=O)CCCC3)CCC(C)(C1)OC2 c1(CC(=O)NC(C(=O)NCCc2cscn2)C2CCC2)cncnc1 N=c1[nH]c(=NCC23CC(CN2C)C3)[nH]c(=NCCN2CCC3CCCCC3C2)[nH]1 c1(C(C)=O)ccc(C=CC(=O)NC2CN(C(=O)CCc3cnn(C)c3)CC2C)o1 CC(CN(C)C)CCC(=O)NC(C1(O)CCN(C(=O)C2=CCCCO2)CC1)C C1(NC(C(C)OCCCCCC)=O)CCN(C(=O)CNS(N)(=O)=O)CC(O)C1 Cc1ccc(OCCCC(=O)NC2(CCNC(c3c[nH]c(=O)cn3)=O)CC2)cc1 C1(NC(C2(c3ccc(Br)s3)CC2)=O)CCCC1NC(CC)=O C(c1cncnc1O)=CC(N1CC2C(N(C(c3c(C)nc(OC)s3)=O)C)C2C1)=O Cc1nc(NCCN(C2CCCCCC2)C(=O)C(C)OCCN(C)C)cc(C#N)n1 c1(C(=O)NC(C(C)NC(=O)CCCc2cnn[nH]2)C)ccc2cnoc2c1 C1(C(N(C(C#C)C2CCC2)C)=O)CCN(C(c2cnc(C)nc2)=O)C12CC2 C(C(C)(C)C(=O)NCC(C)N(C)C(C1CC(=O)N(C)C1)=O)OC(C)C C1(O)(C(N(C(c2n[nH]c(=N)s2)C)C)=O)CCN(c2cncc(C(=O)O)n2)CC1 N1(C(c2ncc(Br)cc2OCC)C(=O)NC)CCS(=O)(=O)CC(C)C1 N1(C(C(C)SCC)=O)CCc2ccc(C(=O)N(C3CCCC(C)C3)C)nc2C1 N1(C(C)=O)CCC(C(=O)Nc2cccc(NC(=O)CC3CCC(=O)C3C)c2)CC1 C(=O)(C1=C(C)CCCC1)NC(CCC)CCCNC(C1CC1F)=O N#Cc1cnn(CC(N2CCCOC(CNC(=O)CC3CCCCO3)C2)=O)c1N c12nnc(o1)SC2.C(=O)(C(C)N(C(=O)CCSC(=N)N)C)OC c1(CCC)cnc(NC(C2CN(Cc3cccnc3)CCS2)=O)nc1 c1(C(N2CC(CN=c3[nH]nc(C4CC4)s3)C2)=O)ccc(F)c2ccccc12 CC(C)(CC(=O)N1CC=C(C(=O)NCC(C)(C)CCCO)CC1)C(F)F C1(NC(CCCCC#C)=O)CN(C(=O)Cn2cncn2)C2CCCC12 C1(C(=O)NCC(C)N(C(c2ccc(CC)o2)=O)C)CCn2nncc2C1 CC1CCc2nc(C(C)NC(=O)NCc3cccnc3Cl)sc2C1 CC1(C)CCC(C(C)(C)C(N2CCCC(CNc3ccc(=N)[nH]c3)C2)=O)OC1 C(=O)(CCC1=CCCCC1)N1CC2CC(NC(C3(CC(=O)OC)CC3)=O)CC2C1 Cn1c(C(=O)NC2(CNC(c3cc4ccccc4o3)=O)CCC2)cnc1[N+](=O)[O-] CC1CC(CNC(=O)CONC(C2CC(=O)C23CCC3)=O)CC(=O)N1 C1(CNC(c2ccc(CC)o2)=O)CC(F)(F)CN1C(=O)C1=C(C)CCOC1 C#CC1CCCC(NC(C2(NC(=O)CCCCCOCC)CC2C)=O)C1 C1(NC(C2CCC(OCCOC)CC2)=O)CCC(C)N(C(=O)CC(C)(F)F)C1 C1(C(N2CCOC(C3CN(C(c4ccc[n+]([O-])c4)=O)C3)C2)=O)CC(C2CC2)=NO1 c1(C(N2CCC(CC(N3C(COC)CC3)=O)C2)=O)ccnc(C)n1 n1(CCC(N2CCCC(F)(CNC(CC(C)(F)F)=O)C2)=O)cnc2ccccc12 C(=O)(CC(CC=C)NC(c1ccccc1CO)=O)NCCCCC#C c1(C(=O)NC(C(C)NC(c2cn(CC=C)nc2)=O)(C)C)ccc(C)n1C CN=C(NCCN1CCOC1=O)N1CCC(C(O)C(F)(F)F)C1 CCC(CC(=O)NC1CN(C(c2ccc(SC)cc2Cl)=O)CC1(C)C)C(F)F c1(C(N2CC(NC(C(c3ccc(OC)cc3)(F)F)=O)C2)=O)cc2n(c1)CCC2 C(=O)(C(C)(C)C(=O)NCC1CCCN1C(C1CC2CCC(C1)S2)=O)OC(C)(C)C C1(C(=O)NC(CC)CN(C(=O)COCCOC)C)CCC(C(N)=O)C1 C1(NC(C(C)NC(=O)NC)=O)CCN(c2nc(C(C)C)nc(C)c2Br)CC1(C)C c1(NCCCCCN(C)C)ccc(N)c([N+](=O)[O-])c1 Cc1cc(C(=O)NC(C)(C)CNC(c2ccc(Br)o2)=O)co1 OCCC(N=c1nc(N2CCc3nocc3C2)c2c([nH]1)CCS2)C1CCOCC1 c1(C(N(CCNC(C2(OCC)CCCC2)=O)CC)=O)ccc(Cl)c(F)c1O C(=O)(CC(F)(F)C(F)F)N1CCCC(CN(C(=O)CCN(S(C)(=O)=O)C)C)C1 CC(C)C(F)(F)CC(=O)NC1CC(CO)N(C(C2CCC(C)CC2)=O)C1 Cc1[nH]c(=N)nc(O)c1CCC(=O)NC(C)CNC(c1cc2ccncc2o1)=O C1(C(=O)NCC2(N(C)C)CC2)(COC)C=CCN1C(c1cc(=N)[nH][nH]1)=O Cc1cc(C(=O)N(CCC(=O)NC2CCS(=O)CC2)C)cnc1O c1(C(C)N)cnc(C(N2CCC(C(C)(C)O)C2)=O)s1 N1(C(C(C)OC2CCCC2)=O)CCN(C(=O)C=C2CCN(C)C2)CC(C)(F)C1 N1(C(C(C)(C2CC2)OC)=O)CCC(O)(CN(C(=O)C=Cc2cc[nH]n2)C)C1 c1(C(=O)NC(C2OCCN(C(CCC(=O)NC)=O)C2)C)c[nH]c(=N)c2[nH]ccc12 c1(C(C(=O)NC2CCCCC2)N(C)CC2CCSC2)cnc(Cl)cc1 CC(CC(C)(C)C)C(F)C(=O)N(CCCCCNC(c1cnn(C)c1Cl)=O)C c1(C(=O)NC(C)CCNC(=O)C(F)n2cccn2)ccc(SCC2CC2)o1 c1(CNC(C2CCC3CC3CC2)=O)cnc2n1CCOC2 C(=O)(C(C(=O)N1CCC(c2cn(-c3occc3OC(F)(F)F)nn2)C1)OC)OC N1(CC(=O)NCCN(C(=O)C(C)(C)C(C)(C)C)CC)C(=O)NC(C)(CC)C1=O CCCN=C(NCC1CC12CCC2)NCC(CC)Oc1ccccn1 C(=O)(C(C)C(C)S(C)(=O)=O)N(CCNC(C1CC=CCC1C(N)=O)=O)CC N1(C(C2C(C)OCC2)=O)CCC2(CCC(CNC(c3coc(Cl)c3)=O)OC2)CC1 Cc1ncc(C(=O)NCC2(CNC(c3n[nH]c(C)c3O)=O)CCOCC2)cn1 N1(C(COC)=O)CC(F)(F)CC1CCNC(C1CC(O)C1)=O N(C(=NCCCOC(C)C)N1CCCC(N2CCCC2=O)CC1)C(C#CC)(C)C C#CCCCCCCC(=O)NC(c1ccc(OC)c(Br)c1)CC N1(C(C(c2cccnc2)C)=O)CC(NC(=O)COC2CC=CC2)C2(CC2)C1 N1(C(c2cc(CNC(C(C(=O)OC)C)=O)nn2C)=O)CC(=O)NC(=O)C1C C1(O)(C(C)NC(C=C(C)C(F)F)=O)CCN(C(=O)C(C)(C)C2CCOC2)C1 C(CCCC(=O)NCc1cc(C(=O)NC2CCCC2O)ccn1)OC CN1CC(NC(=O)CC2CN(C(=O)C3=COCCC3)C(C)(C)C2)C2(CC2)C1 c1(CCC(=O)NC2(C)CCN(C(Cn3c(C)ccn3)=O)C2)ccc(F)cc1Cl N1(C(Cc2c(C)scc2)=O)CCC(NC(C2(c3ccccc3Cl)CC2)=O)CC1C C(=O)(C1CCCn2cnnc21)NCC1CCN(C(C=Cn2cnc(C)c2C)=O)C1 C1(CNC(C=C(CC)C)=O)C2CN(C(c3c(-c4ccsc4)noc3C)=O)CC12 c1(CC)ncc(C(=O)NC(CC2CCC2)C(=O)NC(C(O)CO)C2CC2)s1 N1(C(CC2C(C)(C)N(C(C3CCC(O)C3)=O)CC2)=O)CCOC2COCC12 CC1(C)CCC=C1C(=O)NC1CN(C(c2cc(Br)sc2Cl)=O)CC12CC2 c1(OC)ccc(Br)cc1C=CC(N1CCC(F)C(NC(C2CC(O)C2)=O)C1)=O CCC(CC)C(C)C(=O)NC1(CF)CCN(C(c2ccc(C(F)(F)F)nc2)=O)C1 C1(C(N2CC(C)(O)C2)=O)CCN(C(C2CN(C(N)=O)C2)=O)C12CC2 C1(C#N)(C(N(CCN(C(C)C)C(c2cn(CC(F)F)cn2)=O)C)=O)CCCOC1 C1(N(C(=O)CC2CC23CC3)C)CCN(C(c2cc(C3CC3)ns2)=O)CC1 c1(OCC)oc(C)nc1C(N1CC(CNC(=O)CCCc2ccsc2)(OC)C1)=O c1(CC)noc(C(N2CC(NC(c3ncsc3Br)=O)C(O)C2)=O)c1C C1(NC(C2CCO2)=O)CN(C(c2c[nH]nc2-c2cccc(Cl)c2)=O)CC1O CCCC(F)C(=O)N(C)CCC1CCCCN1C(c1cncc(NC)c1)=O c1(C(N(C)CCNC(=O)CC2(C(F)(F)F)CC2)=O)cnc2c[nH]nc2c1 C1(C)(C(=O)OCC)CCCN(C(=O)CN2CCC(=O)NC2=O)C1 c1(C(N(C)CC2CCCN2C(=O)CCOC2CC2)=O)c(Cl)ccc(Br)c1F CCCCC(CC)(c1nnnn1C1CC1)NC1CCN(C(C2CCCO2)=O)C1 C1(C(N(C(C)C)CCNC(c2ccc(C(N)=O)[nH]2)=O)=O)CC2CCC1C2 N1(C(c2c(SC)n(C)nc2)=O)CCN(C(=O)Cn2cncc2C)C(C)C1C C1(O)(Cc2cn(C3CCN(C(C(C4CCCCC4)OC)=O)C3)nn2)CCOCC1 C(=O)(C(F)(F)C(O)C(C)C)N(C)CC1OCCN(C(C(CCCC)(C)F)=O)C1 CC1(C)CC(NC(=O)C(=O)NC2CC23CCOCC3)C2(CCC2)C1 N(C(=NCC1CCC1)N1CCC(C)(C(N)=O)C1)Cc1c(OC)nc(CC2CC2)cc1 CC1CN(C(c2ncccc2Cl)=O)CC1n1cc(C2CC2)nn1 c1(OCCC(N2CC3C(NC(CN(C)C4CC4)=O)(C3)C2)=O)ccccc1C#N N1(C(=O)NC2CN(C(COc3ccc(CC)cc3)=O)CC2O)CCN(C)C(=O)C1 C(=O)(C1=CCOCC1)NC1CN(C(=O)OC)CC1O.C12(CCCC1)C(=O)N2C C1(CC(=O)NCC(CC)N(C(c2c(C)cc(CC)o2)=O)C)OCCCC1(C)C c1(C(=O)Nc2cccc(CNC(=O)CSC(F)F)c2)cc2c(nn1)CCOC2 n1(CC(N2CCCC(C(C)NC(C(CC)CC)=O)C2)=O)nc2c(n1)CCCC2 CN(CC(=O)N=S1(=O)CC(C(C)(C)C)C1)CCNC=O CC(C(=O)NCCc1ccsc1)NC(=O)C(F)=CC1CC1 C#CCCCCCC(=O)NCCOCCCNC(=O)C(N1CCCC(C)C1)=O c1(C(=O)NCC(CN(C(C2(COC)CCOC2)=O)C)O)c(C)cc(Cl)nc1N c1(C(=O)NCC2C(NC(C3(C(C)C)CCC3)=O)C2)cnc2cc(Br)ccn12 c1(OC)ccc(Cl)c(-c2nc(C(C)NC(=O)Nc3cccc(CF)c3)c(C)o2)c1 Fc1cc(Br)c2ncnc(N3CCN(c4nc(Cl)ns4)CC3)c2c1 Cc1ccc(C(=O)NCC2CCC(C(=O)NCc3ccc(F)nc3)C2)nn1 c1(C(=O)OC)cc(NC(C2CCCC(NC(C3CNC(=O)CO3)=O)C2)=O)ccc1Cl CC12CN(CC3CC4CC4C3)CCC1C2(F)F c1(C(=O)NCC2N(C(c3ccc(C#N)[nH]3)=O)CCC2)cnc(O)c(F)c1 N1(C(Cn2ccc(C)n2)=O)CCCN(CCNC(=O)Cc2cc[nH]c2)CC1 N1(C(C)=O)CCC(NCCCNC(N2C(c3ccc(C)cc3)CCC2C)=O)C1C Cn1cnc2c(N3CCC(OCCNC(C4(CC5CC5)CCCC4)=O)C3)ncnc12 c1(C(N2CC3C(CNC(=O)CC(O)C4CC4)C3C2)=O)ccnn2ccnc12 C(CCC(C)C)(C(=O)N(CC(O)C1CC1)C)NC(c1c(C)coc1)=O C1(NC(CCCOC(C)C)=O)CN(C(=O)Cc2nnc(O)s2)CCC1O c1(C(=O)OCC23OC(C)C(C2)C3)cccc2c1OCCC2 N=c1nc2scc(Cc3nc(C4CCN(c5ncccn5)CC4)cs3)n2[nH]1 C1(C2C(=O)N2)CCOCC1.C1(C(N(CCC)CC)=O)CCN(CC(F)F)C1 C1(OC)(CNC(c2csc(C(F)F)c2)=O)CCN(C(c2ccc(CO)cn2)=O)C1 CCCC(O)(CCC)CC(=O)N(CC)CC1(C)CN(C(=O)C(C)O)CC1C C1(CO)COC2(C1)CN(N1CCCC3(CCO3)C1)C2 n1(CCC(=O)NC2CCCC2NC(C2CCCN2CC(F)(F)F)=O)cnccc1=O c1(NC(CC2N(Cc3cc(C)[nH]c3C)CCC2)=O)ccc2n[nH]cc2c1 C1(NC(Cc2c(C)noc2Cl)=O)CN(C(c2cc(O)nn2C)=O)CCC1CO C12(C(N(C)C(C3COC(=O)O3)=O)=O)C3CC1C1C(Nc4cc(Cl)ncc4Br)C3C21 C1(NC(CNC=O)=O)CCN(C(=O)COC2CC2(F)F)CC1F C(=O)(C1CCCc2scnc21)N1CCN(C(c2ccn3ccnc3c2)=O)C2C1C2 C1(C(=O)NC(C)CC(C)NC(C2(C)CC2)=O)CC2(CCCCC2)C1 N1(C(C2(c3c(C)cno3)CC2)=O)CCC2(CC3CCC(F)C3)CCCC12 N1(C(C)(C)C)CCCC1c1cn(CC2CCN2C(C2C=CCS2)=O)nn1 c1(N(C)C)ccnc(C(=O)NCC2(NC(c3ccccc3Br)=O)COC2)c1 N1(C(CCc2c(C)cccn2)=O)CCC(CO)C(NC(=O)C(O)C(F)(F)F)C1 C(CC(C(=O)NCC(C)(O)CCO)NC(=O)CC1CCC(=O)NC1)OC Cc1cn2c(C(N3CC4C(CNC(C5(N(C)C)CCC5)=O)C4C3)=O)c(C)nc2s1 CCCCCCC(CC)NC(c1c(C(=O)OC)cc(CC)cc1C)=O N1(C(C(CC)N(C)C(C2OCCCC2(C)C)=O)=O)CC2(CC=CC2)C1 N1(C(COC(CC)C)=O)CC(C2CN(C(=O)CC3(C(F)(F)F)CCC3)C2)C1 c1(C(=O)OC)ncc(F)cc1NC(C1CC(O)CCN1C(c1cccc(F)n1)=O)=O C1(CNC(CCC(=O)c2cn(C)nc2)=O)CCN(c2nncs2)C1(C)C c1(CCC(=O)NC2C(OC)CN(C(=O)Cc3ncc(C)[nH]3)C2)ccc(C)c(Cl)c1 c1(C(=O)NCC2N(C(C(N3CCN(C)CC3)C)=O)CC2)cccc2c1NC(=O)CO2 N12CC3CC(C(C3)C1)C(=O)N(C)CC2=O.C1(OC(C)=O)CC1NC.C(C(F)F)C=O N1(C(Cc2cc(C)no2)=O)CC2(CC2)CC1CNC(C1CC(C)(C)CN1C)=O c1(C(=O)NCC2C(NC(C3C4(CC(C)(C)C4)C3)=O)CC2)cccc2c1OCCC2 N1(C(C2C(OCC)C2)=O)C2CCC1CC(CNC(=O)C(O)C1CC1)C2 c1(C(C)(C)NC(NOC(CC)C)=O)cccc(C)n1 c1(C(N(C2CN(C(c3cnc(C(C)C)s3)=O)C2)C)=O)ccccc1F C#Cc1ccc(CC(=O)NCC2CCCCN(C(=O)C(O)c3cnc[nH]3)C2)cc1 c1(C(N2C3CN(C(CCC(C)C#N)=O)C(C3)C2)=O)cc2ccncc2s1 N1(C(CSC)=O)CC(CC(=O)N(C)CCc2cnn(C)c2)CC1(C)C C(=O)(C(C)(O)COC)NC(c1cn(CCCC(=O)O)nn1)CC C1(NC(c2cccc(-n3cccn3)c2)C)CCN(C2CC3CNC2C3)C(C)(C)C1 C1(c2cnn(C)c2N)CN(C(=O)CCCC(F)F)CCC1NC(=O)C=C(Cl)Cl c12cccc(c1)OCCn1cc-2nn1.c1(C(=O)OC(C)(C)C)ccsc1CO c1(C(=O)NCC2C(NC(c3cnn(C(F)F)c3)=O)C2)cccnc1 C(CCCCCC(=O)NC1C2CCC1N(C(=O)C(C)(Cl)Cl)C2)N(C(C)=O)C c12conc1CC(=O)NC2.C1(CNC(C2C(CC)CC2)=O)C(CO)C1(F)F n1(CC#C)ccc(CNC(C(F)(F)F)C2CC2)c1 C1(C)(COC)CC(NC(=O)C(C)(C)C(C)C)CN1C(=O)C=Cc1sccc1C C(=O)(C1CCCc2sccc21)N(CCOC)CCN(C(=O)CC1CCNC1=O)CC C1(COc2ccccc2)CCN(N2CCN(C3CCOC3)C(CC(F)(F)F)C2)CC1 c1(CN2C3CN(c4cc(OC)ncn4)CC32)c(F)ccc(Cl)c1Cl c1(OC(C)C)cccc(CNC(c2cccc(C3CC3)c2)CC(F)(F)F)c1F c1(C(=O)NC2CCC(CCNC(c3ccsc3Cl)=O)C2)ncccc1F CC(CC(=O)N1CC(F)CC1CNC(c1ccc(C(C)(C)C)[nH]1)=O)CC(C)(C)C c1(C(=O)NC2CC(C(=O)NCCNS(CC)(=O)=O)C2)c[nH]cc(C)c1=O C1(CNC(c2ccn(CC)n2)=O)CCC(C)N(C(c2cc(C(C)C)[nH]n2)=O)C1 CC1CCC(NC(=O)C(c2cn(C)nn2)NC(=O)C(O)CC2CC2)C1 N1(C(C(=O)Nc2cccc(F)c2)=O)CC2C(CNC3CCN(C)C3)C2C1 C(=O)(C(F)C(C)(C)O)N1CCC(N(C(=O)CC(C)(C)C2CC2)CC#C)CC1 Cc1c(C(=O)NCC23CC(NC(=O)CN4CCCCC4)(CO2)C3)nn(C)c1N c1(OCCOC)cccc(C=CC(=O)NC2CN(C(C3C=C3C)=O)CC2SC)c1 Cn1cc(C(N2C(C(=O)NC(CC3CCCC3)CO)CCC23CC3)=O)ncc1=O C12(OCC)CC(C(=O)OC)CC1CN(C(=O)NC1CN(CCc3ccco3)C1)C2 n1(CC(N2CC(C)N(C(=O)C(C3CCOCC3)C)CC2)=O)cc(Cl)c(O)nc1=O Cc1nnsc1C(=O)NCC1(CNC(c2cccnn2)=O)CCC1 C12(C(=O)NCC(CNC(c3c(C)cncc3C)=O)O)CCC(CC1)C(C)O2 Cc1cc(C(=O)N(C2(C(=O)NC3CC4CCC3O4)CCCC2)C)nc(C)c1 CCCCCCC(C)(CC)C(=O)N1CC(CC)(NC(=O)CC(C)F)C1 N1(C(CCC=C)=O)CCN(C(C2CCCCN2C(C)=O)=O)C(CC(F)F)C1 N1(C(CNS(CCCC)(=O)=O)=O)C2CCC(C2)C1CNC(=O)C(C)(O)COCC N1(C(CSc2n[nH]c(=N)s2)=O)CCC2(CCCN(C(=O)CC3CCC(=O)N3)C2)C1 N1(c2ncc(C#C)cn2)CCC2(CCC2)C(NC(c2ccccc2CC=C)=O)C1 C#Cc1ccc(C(=O)N(CCC(=O)N(CCC(C)C)CC)C2CC2)nc1 S(=O)(=O)(c1cnc(NCC2CSCCS2)c(Cl)c1)NCc1cn(C(C)(C)C)nc1 C(CCCC(=O)NC1CN(C(=O)C=CCN2CCCC2=O)CC1OC)OCC C1(C(=O)NC(C=CC(=O)NCc2cc(OC)ns2)(C)C)NC(=O)OC1(C)C c1(OC)cc(C)c(NC(=O)Nc2cc(-c3cccc(C)c3C#N)ccn2)cc1Br C1(C(=O)NC(C(C)C)CNC(=O)CCc2ccsc2)OCCC1(C)C c1(CC)ccc(O)c(C(=O)NC2CC(C)CN(C(c3cc([N+](=O)[O-])c[nH]3)=O)C2)c1 O=C(Cn1cc(C2CC2c2cccnc2)nn1)NNC(=O)C1(C(=O)NC)CC1 Cc1cccc(SC(C)C(=O)NCC23CC2CN(C(c2ccncc2O)=O)C3)c1 C1(NC(c2ncc(C)c(Cl)c2)=O)CCOC12CCN(C(=O)CC1CSCCS1)CC2 C(=O)(CCCC(=O)N(C)C)N1CCC(C)(CNC(C2(OC)CCCOC2)=O)C1 c1(C(=O)NC2CC(NC(CSCCN(C)C)=O)CC2O)csc2ccncc12 C1(CC)(NC(=O)NCCC2OCCCO2)CCCC1 c1(C(=O)NCC2CC(C)(C)CN2C(C2CCCS2(=O)=O)=O)nc2ncccn2n1 CN1CCC(C)(C(N2CCC(C)(CNC(C3CC(C)(O)C3)=O)C2)=O)C1=O N1(C(C(C)(C(=O)OC)N(C(C(CC=C)C)=O)C)=O)CC2(C(=O)OC)CCC1CC2 C1(NC(NNC(=O)c2c(C)ccs2)=O)C=CS(=O)(=O)C1 CC1CC(C(N2CCC(F)(CNC(C3CCNC(=O)C3)=O)CC2)=O)CCN1C c1(C(N2CC(C(C)NC(C3CCCC(OC)C3)=O)C2)=O)[nH]c(C)c(C(C)=O)c1C CC1CC(C(=O)NC2CCCOC2)N1C(c1cn(C)nn1)=O c1(OCC)ccc(Cl)c(C(N2CCN(C(c3nccn3C)=O)C(CO)C2)=O)n1 Cc1cc(C(c2nnnn2-c2ccc(F)cc2)NCCSC(F)F)c(C)s1 C1(C#N)(C(=O)NC2CC(NC(c3ccc(COC)cn3)=O)C(O)C2)CCCOC1 C(=O)(CS(=O)(=O)CCOC)N(C1CCN(C(c2ncc(F)cn2)=O)C1)CCC CCCCC(C)C(=O)NCC(O)CNC(C1(c2ccc(O)nc2)CCC1)=O C12(CNC(c3cc(OC)c(O)cc3)=O)CN(C(=O)OC(C)(C)C)CC(F)(C1)C2 C(=O)(C(C(C)C)NC(=O)C(C)C1CCCC1)N1CCC(SC)C1 N1(C(c2c(CC)scc2)=O)CC(NC(=O)CN2CCCC2CO)CC12CCCC2 CS(=O)(=O)c1cccc(C(=O)Nc2cccc(C#N)c2OCCO)c1F CC1CN(C(c2n[nH]cc2C2CCC2)=O)CCN(C(=O)CCC(C)(C)C)C1 C(=O)(C(CC(F)F)NC(c1cnn(C(C)C)c1)=O)N(CC=C)CC1CC1 C(=O)(CC1C(=O)Nc2c(F)cccc21)NC(CNC(c1cnc(COC)s1)=O)C c1(C2C(C(=O)NC3CC(CCNC(=O)C=Cc4nccs4)C3)C2)ccccc1F c1(C(N2C(CCNC(CCN(CC)CC)=O)COCC2)=O)cccc(O)c1F Cc1cccc2cc(C(=O)NC3(CF)CCN(c4nnc(C5CC5)s4)C3)oc12 c1(OC)c(F)c(C(N2CC(NC(c3n[nH]cc3I)=O)C(C)C2)=O)cc(F)c1F C1(CC(=O)NC(CN(C(=O)CCCc2ccncc2)C)(C)C)CCS(=O)(=O)C1 C=CC1(NC(c2nnnn2CCOC(C)(C)C)C2CC2)CCCCC1 c1(C(c2cccs2)NC(C2N(C(C(C=CC)O)=O)CCC2)=O)c(F)cccc1F c1(CC)cc(C(=O)NC2CC(N(C(=O)C=CSc3nc[nH]n3)C)C2)n(C)n1 c1(CC(=O)N(C2CC3CN(C(CSC(C)C)=O)C2C3)C)n[nH]c2c1CCCC2 C(CC(C(=O)N1CCOCC1COCC)NC(=O)COCC(C)C)=CC N1(C(CCCOCCC)=O)CCC2(CC1)CC(NC(=O)CNC(C)=O)CO2 C1(C(N2CC(NC(C(n3ncc(C)c3)C)=O)C(C)C2)=O)CCC2(CC1)CC2 c1(CC(=O)NC2CN(C(C(F)OC)=O)CC2C)c(C)cc(Br)cc1C C1(C(N(CCOCCCN(C(=O)CCCN2CCCC2)C)C)=O)CCC2CC12 C1(NC(C(C)OCC=C)=O)CCN(C(=O)Cc2ccc(CO)c(C)c2)CC1F c1(C(=O)NCC2C(NC(C3C(C)(C(F)F)C3)=O)CCC2)cccc2cnccc12 C1(C(=O)NC23CC(C2)N(C(C2CC2F)=O)C3)CC2CC(O)C(C1)C2 c1(C(=O)NCC2CCN(C(C3CCC(C)O3)=O)C2)cnc2c[nH]nc2c1 c1(N(C)CC2CCCO2)cc(COc2ccc(C(=O)OC)cn2)nn1C N1(C(c2c(C)nc(C)o2)=O)CCC(C)N(C(=O)CN2C(C)CCC2C)CC1 C1(NC(C2(CC)CCCC2)=O)CC(C)N(C(c2ccc(OCC(F)F)cc2)=O)C1 C1(CC=C)(C(=O)N(C)CC2CC2)CCCN1C(=O)CC(C)C1CC1 CC(C)CC(C)C(=O)N1CCCCC1CN(C(=O)Cc1cc(F)cc(Cl)c1)C C1(C(=O)NC2(C)CCC(NC(c3ccnnc3)=O)CC2)CCCCC12CC2(F)F N1(C(CC2CC(OC)C2)=O)C2CCC1CN(C(c1conc1C1CCCC1)=O)C2 Cc1nccc2c(=O)c(C(N3CCc4sc(Br)c(Br)c4C3)=O)c[nH]c12 O=C(C1=CCCCO1)NCCCC(Cc1ccccc1)NC(C1CNC(=O)C1)=O C1(NC(CN(C2CC2)CC)=O)CN(C(c2cccc(SC)c2)=O)CC1O CC1=C(C(=O)NCC2C=CCN2C(c2cc(N)c(F)cn2)=O)CCC1 N1(C(C2C(CNC(CC(=O)OCC)=O)OCC2)=O)CCN(C)CC1C N1(C(C(CC)O)=O)CCCN(C(c2ccnn2CC2CCC2)=O)CC1 C1(C(=O)N(C(C)CC(N)=O)C)(OC)CCN(C(=O)CCn2cccc2)C1 Cc1ccc(C=CC(=O)NC(C)(C)C(=O)NC(CCO)C2CCC2)cc1 CCCC(CCC)CCCC(=O)NCCC1CN(C(=O)CN2CCCC2C)C1 C1(CC(=O)NC2(C)CN(C(c3ncc(OC)nc3)=O)C2)CC(C)(C)CCO1 N1(C(C(CC=CC)NC(=O)C(C)NC(N)=O)=O)CC2CCC2(CO)C1 C(=O)(CCCC(C)(C)NC(=O)CCC1CCCCO1)NC(C#C)C(C)OC CC1CN(C(c2ccn(CCO)c(=O)c2)=O)CCC1NC(=O)CCc1cnoc1 N1(C(CCCCCCSC)=O)CC2(C1)CN(C(=O)C(C)c1ncco1)CC2CO C12(NC(c3cccc(C)n3)=O)CCOCC1CN(C(C1CC13CC3)=O)C2 N1(C(Cc2c(C(C)C)con2)=O)CCC2(C1)CN(C(=O)Cc1ccnnc1O)C2 CC1CC(CNC(=O)CC2(CO)CC2)CN1C(=O)CC1(C2CC2)CC1 C#CCC(C(=O)OCC)NC(C1C(NC(=O)C2CC2)CCN1C(c1ccoc1)=O)=O C(C(C)(COC)C(=O)N(C(C(=O)NCc1csc(CO)n1)C1CC1)C)OC C1(S(C)(=O)=O)(C(=O)NCC(C)N(C(=O)C(C(C)(C)C)NC(C)=O)CC)CCCC1 CCCCCCCC(=O)N1CC2CC1C2NC(c1csc(C(C)OC)n1)=O C1(C)(CC)CCCN(C(C2(NC(c3cc(C)nc(C)n3)=O)CSC2)=O)CC1 C(=O)(C(C1=C(C)C=CCC1(C)C)N(C)Cc1ccc(F)c(Cl)c1)NCCC c1(C(=O)NCC2N(C(c3c(=N)[nH][nH]c3)=O)CCCC2)cc2ccccn2n1 C(=O)(C1=C(F)CN(C(=O)C=Cc2cnccn2)CC1)N1CCC(C(C)(C)O)CC1 C(CC1CCCC1)(C(=O)NC(CNC(C1(OC)CC1)=O)C1CCC1)OC c1(C(N2CCCC(CN(C(C(CC(C)C)F)=O)C)C2)=O)cccn2[nH]c(=N)nc12 C1(NC(c2c(OCC)oc(C)n2)=O)CN(C(=O)CC(C)N(C)C)CCC1(F)F C1(O)(CN(C)C(C2CCOC2)=O)CCN(C(=O)CSCc2csc(=N)[nH]2)CC1 C12(NC(c3n(CC)nc(C)c3)=O)CCN(C(C34CC(F)(C3)C4)=O)CCCC1C2 Cc1cccc(C(N2CCC(C)(C)C2CNC(=O)CC(C)n2ccnc2)=O)c1Cl N1(C(CCCN(C(C)=O)C)=O)CC2CCCC2(C(=O)NC(c2nc[nH]n2)C)C1 C1(C(=O)NCC#CCNC(c2cnc(S)[nH]2)=O)CC(O)CN1C(=O)C(F)(F)F C1(NC(Cc2c(CC)n[nH]c2CC)=O)COCCN(C(C2(C)CCN(C)C2)=O)C1 N1(Cc2cn(CCOC)nc2)CCN(C(c2ncc(C(=O)O)s2)=O)C(C)C1 c1(C(N(CC(C)NC(c2cc(CC)cc(C)c2)=O)CC)=O)c(C)cc(C)cc1C N1(C(CCc2c(C)ncs2)=O)CCC(C(=O)N(C)C(C)C)CC1C C1(NC(=O)C(F)=CC2CC2)CN(C(=O)CCC2CCCCC2)CCC1CO C(=O)(C(C)C(O)C(C)C)NC1CC=C(C(=O)NCC(=O)OCC#C)C1 c1(C(N2CC(NC(c3ccc(N(C)C)cc3)=O)C(O)C2)=O)cc2ccccn2n1 C1(F)(C(N(CCC(=O)NCc2nc(C(C)C)n[nH]2)CC)=O)CC=CCC1 CCCCC(C(=O)NC1CC(C)(C(=O)OC)C1)NC(=O)Cn1nc(C)oc1=O c1(CCOC)n[nH]c(=NC2CN(C(c3ncc(Cl)nc3Cl)=O)C2)s1 c1(OC(N(CCC(=O)N(CC#C)CC#C)C)=O)ccn(C2CC2)n1 c1(C(=O)NC2(CCNC(C(CC)SC)=O)CC2)c[nH]c2ccc(F)cc12 C(=O)(C(C)C(C)NC(C1(CNC(=O)CC2CCC(C)CO2)CC=CC1)=O)OC c1(NC)ccc(C(N2CCC2CNC(c2nccnc2N)=O)=O)c(O)c1 C#CCCC(O)C(=O)N1CCC(C(C)(C)NC(=O)CNc2ccc(Cl)cc2)CC1 c1(C(N2CCC(O)(CNC(CCOCCCC)=O)C2)=O)cccc(F)c1CC N1(C(C)(C)C)CCN(C(=O)CN(C(=O)C2=CCOC2)C2CCC2)CC1 C1(C(N(CC)CC2CCCCN2C(c2nc(Cl)oc2C)=O)=O)CCN(C)C(=O)C1 N1(C(c2cn(C)nn2)=O)C2CCC1C(CNC(=O)CN1CCC(F)(F)C1)C2 C(=O)(C(CNC(C1(F)CCCC1)=O)CC1CC1)NC(COC)C1CC1 Cc1cnc(C(N2CCN(C(=O)C=C(Cl)Cl)CC2c2ccccc2Cl)=O)cc1Cl C1(CC(=O)OC)CC(C)N1C(=O)C(C)CN(C(=O)Cc1ccsc1)C Cc1ccc(OCC(=O)NC2(C)CCN(C(c3[nH]c(C)cc3C)=O)C2)cc1C CCCC(C)C(=O)NCc1ccc(C(=O)NCc2c(C)noc2C)cn1 C1(CC(=O)OCCNC(CNC(C2CC3(CCC3)C2)=O)=O)CCCC12CC2 C(=O)(CC)NCC1C(C(NC=O)=O)C1.c1(NC(C2CC2C(F)(F)F)=O)ccco1 C1(C)(C(N(C2CCN(C)C2)CC)=O)CN(C(c2nc(C)sc2C)=O)C(C)(C)C1 C(=O)(C1=CCC(NC(=O)CCCc2cnn[nH]2)C1)NC(CC)CC1CC1 C1(C(C(=O)NCCN(C(=O)COCC(C)C)CC)SC)CCOCC1 c1(NN(CCC(=O)OC)C)cccc(F)c1Cc1ccc(C)cc1Br n1(-c2n(C)ncn2)nc(CO)nc1C1CCN(c2ccncn2)CC1 c1(C(N2CC(n3cc(CC(O)C4CC4)nn3)C2)=O)ccc(O)c([N+](=O)[O-])c1 C1(C(=O)NCC2(O)CN(C(C(C=C)O)=O)C2)(CF)CCOCC1 CC1CC2(CCCCN2C(N2CCCCC2c2nnc(C3CC3)s2)=O)S1(=O)=O N1(C(CCc2cccc(C)c2)=O)C2CCC1CN(C(=O)C(C1CCC(=O)N1)C)C2 c1(OCCCC)ccc(CNC(=O)CNc2cn(C)nc2Br)cc1 C(#Cc1cccc(Cl)c1)C=CCNCC1CCC2(CCC2)CO1 C(=O)(C#CC1(C)CCCO1)NC1C(C(=O)NC(CC=C)CC(F)F)CC1 Cc1cc(C(=O)NC2(CNC(=O)CC3(O)CCCCC3)CCCC2)cnn1 N(C(=NCc1cccs1)NC1CC1C(F)(F)F)CC1(OCC)CCC1 c1(CNC(C2C(NC(c3c(C(C)C)ocn3)=O)COC2)=O)ccc(O)nc1 N(C(=NCCCF)NC(c1ccccc1)C)CCc1c(C)cncc1 N1(C(C(C)CCO)=O)CCC2(CCC2)C(NC(C2CC(C(F)(F)F)C2)=O)C1 C#Cc1cc(NC(=O)CCCCCNC(c2c(C)cnn2C(C)C)=O)cc(F)c1 c1(C2CCC(CC)O2)nscc1C(=O)NC(C)CCc1cnn(C)c1 C1(CNC(c2cnn(CCCC)c2C)=O)CN(C(=O)C2CC2)C2COCC2O1 N1(C(CS(C)(=O)=O)=O)Cc2ccccc2CC1C(=O)Nc1ccc(C#N)nc1 C1(NC(c2n(CCC)ncc2)=O)CCC2(CCCN2C(=O)C=CS(C)=O)CC1 CC1(C)CC(NC(c2csc(-c3cnc[nH]3)n2)=O)CN(C(=O)CC=C(Cl)Cl)C1 c1(C(=O)NC2CC(CNC(C3C(C)(CC)C3)=O)C2)cc2c(s1)CCC(C)C2 c1(OC)cc(C(=O)NCC(O)CNC(c2cc(O)cc(=O)o2)=O)cc(Cl)c1O c1(C(=O)NC(C(=O)NC(C)CCCNC(=O)C=CCF)C)ccc(Cl)cc1O N1(C(C)=O)CCCC1C(=O)NCCN(CC(F)F)C.C12(CC1)C(=O)N2 C=Cc1cnn(C)c1C(=O)N(CC(O)CNC(C1(C)CC(C(F)(F)F)C1)=O)CC C1(N(CC(=O)NC)C(C)C)CCN(C(=O)C(c2ccccc2)OC(C)C)C1 Cn1ncc2c(NC3COC4(CCC4)C3)nc(N3CCC(F)(F)C(C#N)C3)nc12 C1(CC)OCCC1C(N1CC(CNC(=O)C(=O)C2CCCC2)C1)=O C=CCCCCC(=O)NCC(O)CC(=O)N(C1CC1)CC1CC1 C(=O)(C(C)C(F)(F)F)N1CCC(C)(NC(C(CC)CN(C)C)=O)C1 n1(CC)c(=O)n(C)c(=O)c2cc(C(=O)NC3CCN(c4cccs4)C3=O)cnc12 Cc1cnc(C(N2CCOC(CNC(c3nnc(C)s3)=O)C2)=O)c(F)c1 C(=O)(C(C(=O)OC(C)(C)C)C(C)C)OC.C12CN(CC1C)C(=O)CCC(=O)N2C C1(C(=O)NCC(C=C)O)CN(C(=O)CC(C)C(C)C)CC(C)O1 C1(NC(C(C)(C)CCNC(c2nncs2)=O)=O)CC12CCCCCC2 n1(CC(C)C)[nH]c(CC(=O)N(CC(C)NC(c2cc(Cl)on2)=O)C)cc1=O C1(C(=O)NCC(C2CC2)NC(c2ccn(CC)n2)=O)(OC)CCCOC1.C1(C)CC1 N=c1[nH]cncc1C(=O)NCC1(C(F)(F)F)CCN(C2CCC3CCC23)C1 C(C(C)(C)C#CC(=O)N1CCCC1C1CC1)NC(Cc1nc(C)sc1)=O Cc1cccc2c(C(=O)NC(C)CCNC(=O)CSc3n[nH]c(O)n3)csc12 Cc1ccc2c(c1)N(C1CC3CC1CN3C(=O)OC(C)(C)C)CC2 N1(C(CSCCCNC(=O)Cn2cc(C(F)(F)F)cn2)=O)CCCC(C(=O)O)C1 N1(C(c2c(CC)ocn2)=O)CC(OCC)C(CC(=O)NC2CCCCC2C2CC2)C1 CCC1=C(C(=O)N2CCC3C(CCN3C(c3ccc(OC)cc3)=O)C2)SCCO1 C1(NC(=O)CSc2ccccn2)CCCCC12CCN(C(=O)Cc1cnc[nH]1)C2 c1(C(C(=O)NC(CNC(C(C=C)O)=O)C)(F)F)ccc(F)c(F)c1 C1(CC)CCCCN(N2CC(=O)NCC2C=O)C1.c1(C)ccccc1 c1(CC(=O)NCC(C2CCCN2C(C2CNC(=O)C2)=O)(C)C)cccc(Cl)c1 N1(C(C2C(C=C)OCCC2)=O)CC(CNC(c2coc(CO)c2)=O)C2(CCC2)C1 N1(C(c2c(OC)n(C)nc2)=O)CCC12CN(C(=O)C(C)(C)n1cccn1)C2 c1(C(N2CC(NC(C3C(=C)CC3)=O)(COC)C2)=O)nccc2c(C)cccc12 c1(C(=O)NC2C(CNC(c3cc(C)n(C)c3C)=O)CC2)cnc2ccncc2c1 C(=O)(C1=CCCCC1)NCC1N(C(C(CC)(O)c2ccccc2)=O)C2C(C1)C2 c1(NC(c2c(C)n(-c3ccc(Cl)c(F)c3)nc2)=O)sc2ncccc2c1N Cn1ncc(C(=O)NCCS(=O)(=O)Cc2cn(-c3ccc(F)cc3)nn2)c1Cl c1(CN(Cc2n[nH]c(=N)s2)CC2C=CCN2C(=O)CC(F)(F)F)ccc(F)cc1 C1(NC(C(C)NC(CC)(C)C)=O)CC(C)(CNC(c2ccn(C(C)(C)C)n2)=O)C1 c1(C(N2C(C3CCN(C(c4ccco4)=O)CC3)CCC2)=O)ncn2c1COCC2 C12(N(C)C(C3CC3c3ccco3)=O)CC(C1)N(C(C1CCCN1N=O)=O)C2 Cc1cc(C(=O)NC(C(=O)NCCc2csc(C)n2)C(C)(C)O)cc(C)n1 Cc1c(Br)sc(C(=O)NCCC2CCCCN2C)c1C c1(-c2nc(C3N(C(C4N(C(C)=O)CC4)=O)CCC3)on2)cccc(Cl)n1 C(CCNC(=O)C(c1ccccc1)C)(C(=O)NCCn1cncn1)OC C1(C(=O)NCCc2ccncn2)CCN(C(=O)CN2CCCC2)O1 N1(C(c2occc2Br)=O)CCn2nnc(C(N3CCC(O)CC3)=O)c2C1 N1(C(C(CCCC)N(C)C)=O)CCC2CCN(C(=O)C(C)OC)C2C1 c1(CNC(N2C(c3n(C)ccn3)C(C)(C)C2)=O)ccc2c(c1)CCS2(=O)=O C1(NC(CC(C)OC)=O)CN(C(=O)C=CCCC(C)C)CC1C(F)F c1(C(N2CCC(F)(C(=O)NCc3ccc(Br)s3)C2)=O)ccc(Br)c(I)c1 c1(CC(N2CC(C)C(NC(c3ccnc(F)c3)=O)CC2)=O)cc(F)c(N)cc1F C1(CN=C(NC(C)C)NCc2ccc(P(C)(C)=O)cn2)CC2CCC(C1)S2(=O)=O CC(N=c1cc[nH]cc1S(=O)(=O)NCC1CCCCC1)C1CCC(=O)N1 n1(CC)ncc(C(=O)NC2CC(CNC(c3cc(C)cs3)=O)C2)c1CC(=O)OC CC(C)(CCNCC1CC1)C(=O)N1CCCC(O)(OC(C)(C)C)C1.C1(=O)CC1=O.OCC N1(C(CSc2cccc(OC)c2)=O)CCC(CCNC(=O)C(C)CO)C(F)(F)C1 N1(C(C(CCCC)NC(C23CCCCC2C3)=O)=O)CCCN(CC)C(=O)C1 N1(C(CCN(C)CC)=O)CCN(C(C2CCC3CC3C2)=O)CC1C c1(C(N2CCC(C)(NC(c3ccnc(Cl)c3F)=O)C2)=O)n[nH]c2c1CCOC2 C1(CC(=O)NCCC(C)NC(c2ccnn3ccnc23)=O)CCn2cncc2C1 C1(C)(CC)C=C(C(=O)N2CCCC(N(C(C3CC(=C4CCC4)C3)=O)CC)CC2)C1 c1(C(N(C2CCC(NC(=O)C(F)F)C2)C)=O)ccc(Cl)c(OC(F)(F)F)c1 c1(-n2c(CC3COC(=O)C3)nc(C(C)OCC)n2)ccc(Br)c(F)c1 C1(C(=O)NCC(F)(F)C(N)=O)(CC)CCCN(C(=O)C(C)C2CC2)C1 c1(C(=O)NC2CCC(C)N(C(=O)C=CC3CC3)C2)cnc2c(Br)c[nH]c2c1 CCC(O)C(F)(F)C(=O)NCCCCCC(=O)N(C1CCCC1)C C1(NC(C(CC)(C)COC)=O)CCCN(C(=O)CSCCOC(=O)NCC)CCC1 CC(CN(C)C)CCC(=O)N(C1CCC(NC(C2(C)CC=CCC2)=O)CC1)C C1(CC(C)=O)COCCN1C(=O)CC(c1cccs1)SC.C(C(=O)NNC)(SC)SC S(=O)(=O)(CCC(=O)N(CC(CNC(C1CCCC(C)CC1)=O)(C)C)C1CC1)NC C(=O)(C(C)(CC)C(=O)N1CC(NC(=O)CNC(=O)C2CC2)C(O)C1)OCC CC1(C)CCCC(C(N2CCCC(O)(CNC(c3cn(C4CC4)nn3)=O)C2)=O)C1 C1(CC=C)(C(=O)NCCCSC)CCN(C(=O)CSc2cn[nH]c2)C1 S(=O)(=O)(c1cccnc1Nc1ccc2cc(CC)ccc2c1)NC(CC)CC#N c1(C(=O)NC2CC(C)(C)N(C(=O)CCC3CC3)C2)c(F)ccc(F)c1F c1(C(=O)NCC2N(C(CC3CCN(C)C3)=O)CCOC2)ccc2c(cnn2C)c1 CC1CN(C(C2CCOCC23CCC3)=O)CCCN1C(=O)C(c1ccc(Cl)s1)=O Cc1cc(C(=O)NC(C(=O)NCC(C)CF)C2CC2)n(C)n1 C1(NC(C)=O)CCCCCC1NC(c1cc(C)ns1)=O.C12CCN(C1)C2=O C(CCN=C(NC(C1CCS(=O)(=O)C1)=O)NC1CCN(C(=O)OC)C1)OC c1(C(=O)NC(C2CN(C(=O)CCc3ccncn3)C2)C)ccc(F)cc1[N+](=O)[O-] C1(NC(CN(C(=O)C(C2CC2)C2CC2)C(CC)C)=O)CC(N2CCCC2)C1 C(C(C)C(C)C(=O)N1CCN(CC(C)(C)NC(c2ccc(F)cn2)=O)CC1)OC CCCC(CC(C)C)C(=O)N1CC2(CCC(CNC(c3ccncn3)=O)O2)C1 c1(OCC)cc(C(N2CCCC(C)(C)C2CNC(=O)COC)=O)ccc1[N+](=O)[O-] N1(C(C2C3CN(C(C4CCCC(C)C4)=O)CC32)=O)CCc2cccnc2C1 CN1CC=C(C(=O)N(C2CCN(C(=O)CC3CC4(CC4)C3)C2)C)C1 c1(C(c2n(CCC)nnn2)NC(C)Cn2ccnc2C)c(F)cccc1F CCC(CNC(=O)C=CC(F)F)(CC)C(=O)NCC1(O)CSC1 N1(C(C2CC(OC)C2)=O)CC(NC(c2c[nH]ccc2=N)=O)CC(C)C1 C1(NC(COC(CC)C)=O)CN(C(=O)C=Cc2ccc(C)s2)CC2(CCC2)C1 c1(C(=O)NC(C2CN(C(c3c(CC)occ3)=O)C2)C)ccccc1P(C)(C)=O C1(OCC)CCN(C(=O)CCN(C(=O)CCC2CC2(C)C)CC)C1C C1(C(C)C)(C(=O)NC2CCCC2CNC(=O)Cn2cnnc2O)CNC(=O)C1 c1(CCC(=O)NC(CC(C)NC(CC2(OC)CC2)=O)C)cccc(Br)c1 Cc1cc2ccc(C(=O)NCCC3CN(C(=O)C(C)C(C)(F)F)CCO3)cn2c1 N1(C(Cc2ccn(CC)n2)=O)CC(=O)NCC1C(=O)NCC1CCCS1 C1(CCOC)(NC(c2cc(F)c[nH]2)=O)CCN(C(=O)C(CCO)N(C)C)C1 C1(CC)CN(C(C2(C)CCCC2(F)F)=O)CCN1C(c1ccc(CN(C)C)[nH]1)=O CCC(C)(C)C(=O)C(=O)N1CC2(C1)CN(C(c1coc(C(F)F)c1)=O)C2 Cc1ncc(NC(=O)CCC2CCCCN(C(c3c[nH]nc3Cl)=O)C2)cc1Cl Cc1ccc(CC(N2CC(CCNC(=O)Cc3csnn3)C(C)C2)=O)cc1C CC1CC2(CCN(c3nc(N4CC5CC5C4)c4sccc4n3)CC2)C(=O)N1 C123CC(C1)(OC2C)CNC3=O.C=CC(C)CC(=O)NCC1CC(C(=O)OC)C1 C1(NC(C(c2cccc(NC(C)=O)c2)N(CC(C)C)CC)=O)CCC(F)(F)CC1 N1(CC(c2ccccc2)NC(C)=O)CCC(CC(=O)N(CCC(N)=O)CC(C)C)C1 Cc1[nH]c(C)c(C(=O)NC2CN(C(=O)CCSCC(C)C)CCC2F)c1C c12nc(C3CCCOC3)n(n1)C2.C1CCC(Cn2ncnn2)OC1 CCCCC(C(=O)NC(CNC(=O)CS(N)(=O)=O)C(C)C)NC(N)=O N1(C(C(=Cc2cnc[nH]2)C)=O)CC2CC1CCC2NC(=O)Cc1cscn1 C1(C)(C(=O)NCC(CC)(C)OC)CCCN(C(=O)CSc2nc[nH]n2)C1 CC1(C(c2nnnn2C2CCOCC2)NCC2CC(F)CN2)CCCOC1 Cn1ccnc1C1CC1C(=O)NCC(C1CCCCC1)NC(C1CC1CF)=O Cc1ccc(Br)c(C(=O)NC(C(C)NC(c2c[nH]c(=N)o2)=O)C(C)C)n1 C12(C(=O)NCCNC(c3ccc(C(C)C)cn3)=O)CCCCC1OCC2 C(CC(C)CCOC(c1cnccc1C)=O)NC(C(C)(C)NC(=O)OCC)=O CS(=O)c1cccc(C(=O)NC2CC(CNC(=O)C=Cc3ccncn3)C2)c1 c1(C(=O)NC(CNC(C(CC(C)C)(F)F)=O)CO)cnn2c(Cl)cccc12 Cc1nc(=NC2CC(NC(=O)C(N3CCCC(O)C3)C)C2(C)C)[nH]c2[nH]cnc12 C1C(SC)C(=O)NCC(=O)N(CC)CCS1.C(=O)(C=CCF)NCC.CCCN Cc1ccc(C)c(CN2CC3(CN(C(c4ccc(CO)o4)=O)C3)C2)c1 C(=O)(C(F)(F)C(C)(C)O)N1CCC(CNC(CCCC(=C)C)=O)(OC)CC1 C=C(C)C(O)CC(=O)NC1CCCN(C(C2COCCOC2)=O)CC1 N1(C(C2CCCN(C)C2)=O)CCCN(CCNC(=O)CC(C)(F)F)CC1 N1(C(CN2CCC(C)C2)=O)CCN(C2COCC2NC(=O)CSC2CC2)CC1 N1(C(C=CCN(C)C(=O)OC(C)(C)C)=O)CCCC(C)(NC(=O)C(C)(C)CCCl)C1 C(N=c1[nH]c(Cl)ncc1F)C1CCC(NC(C23CCOC2CCOC3)=O)C1 c1(CNC(C2(F)CCN(C(=O)CSc3nn[nH]n3)CC2)=O)c[nH]c2ncccc12 C1(NC(Cc2ccc(C)cc2)=O)CCSC12CN(C(c1cnc(S)[nH]1)=O)C2 N1(C(c2c(C)nc(O)cc2)=O)CCC(C)(C)C(NC(=O)CC(C)O)C1 CN1CCOC(C(=O)NCCC2CN(C(c3cn(C(C)(C)C)cn3)=O)CCO2)C1 Cc1cnc2cc(C(=O)N(C(C)CNC(c3ncc(Cl)s3)=O)C)ccn12 C1(OC)CC(F)CN(C(C23CC(CO)(CN2C(c2cc(O)ccc2C)=O)C3)=O)C1 C12(C(=O)[N+](N3CCOCC3)(CCC3CN(C(C(CSC)C)=O)C3)[O-])CCC(CC1)CC2 Cc1cnnc(O)c1C(=O)NCC(C1CCCC1)N(C(=O)COC1CCOC1)CC C1(C(=O)NC(C2CCC2)C)CN(C(c2nccc(C)c2F)=O)CC(F)(F)C1 N1(C(CCN(C)C)=O)CCCC1CNC(C1CCOC1)=O c1(C(=O)NCC2CC(O)CN2C(=O)CNC2CCSC2)cc2nc[nH]c2cc1F C1(CNC(Cc2c(CC)con2)=O)CC(COC)CN1C(c1cn(C)nn1)=O C1(O)(CN(C(C2(NC(C)=O)CCC2)=O)C)CN(C(=O)C(C)N(CC(F)(F)F)C)C1 C1(CC(=O)NC2CCC2NC(C2CCSCC2)=O)Cc2ccccc2NC1=O C1(N(C)C(C2COCCN2C)=O)C2CN(C(=O)Cn3cccnc3=O)CC12 c1(C(N2C3C(C(=O)Nc4c(I)ccc(C)n4)C(C3)C2)=O)ccc(F)c(F)c1Cl N1(C(CN2CCN(C(CCC=CCC=C)=O)CC2)=O)CCC(CO)CC1C C1(CC(=O)NC(C)C(F)(F)F)CN(C(c2cscc2C(F)(F)F)=O)CCO1 C(=O)(C1=NNC(=O)CC1)OC.N12CC(C(C)(C)C1)c1nnc(o1)C2=O.N1(CC)CC1 C1(NC(c2cnc(CC)s2)=O)C2CC3CN(C(=O)Cc4ccccc4Cl)C1C3C2 C1(CC(N2CCN(C(c3c(N)non3)=O)C(CF)C2)=O)COc2ccccc2O1 N1(C(c2ccc(OC)cc2)=O)CC2(CNC(=O)C(C3CCCO3)OC)CCC1C2 C1(C(=O)NC2C(NC(CCC(C)OC)=O)COCC2)CC2(CCC2)CO1 C1(C(=O)NCCOCCNC(c2cnc(CCCC)s2)=O)CCCCC1C1CC1 C1(N(C)C)CCCN(C(C2CCC(NC(C3CCCO3)=O)C2)=O)C1 c1(C(N2CCN(c3cccs3)CC2)C(=O)NCC=C)ccc(C2CC2)c(F)c1 C1(C(N2CC(O)(CNC(C3CC(C(=O)OC)C3)=O)C2)=O)CC1C1CCCC1 c1(NC(c2onc(C(c3cccc(OC)c3)CC)n2)C)c(Cl)cccc1Cl Cc1cc(C(N2CC(CNC(=O)CCCC(C)C)C(F)(F)C2)=O)c(Cl)cc1F C1(NC(C(C)NC(N)=O)=O)CC2CCC(C1)N2C(C1CCCC1)=O C1(C(=O)NCc2scc(CNC(C(CC)O)=O)n2)CCC(=O)N1C N1(C(c2c(CC)c[nH]n2)=O)CC2CCC1CN2C(c1cnc(C(C)OC)s1)=O C=CC1CCCC(N=c2ccnc(NCc3ccccc3C3CC3)[nH]2)C1 CC(CC(=O)N(CC(C)O)C)N(C(=O)CNc1ccccn1)C C(=O)(C(O)CC(N)=O)NCC1(OC)CCN(C(=O)C(C2CCOCC2)O)C1 C12(NC(CCCC(=O)OC)=O)CCCC1N(Cc1ccnc(Cl)c1)CC2 Cc1ncc(Cl)c(C(N2CCCC(CNC(=O)Cc3cccc(Cl)c3)CC2)=O)n1 Cc1cn(-c2ccccc2Cl)nc1CN(C(=O)Nc1ccc(Cl)cc1)C(C)C N1(C(=O)CSc2nc[nH]n2)CC2CCCC(C1)N2C(=O)CNc1ccccn1 Cc1c(C(=O)NCC(CC(C)C)NC(C2COC(=O)N2)=O)sc2ccc(Cl)cc12 Cc1noc(-c2cn(CC(N3CC(C)(NC(=O)Cc4cccn4C)C3)=O)cn2)n1 c1(CC(N2CCC(C(C)NC(=O)CS(=O)(=O)N(C)C)CC2)=O)ccc(C)c(C)c1 C1(CSC)CCN(C(C2CC(NC(=O)CC3COCCO3)C2)=O)C1 N1(C(=O)NC(c2cccc(C3CC3)c2)C)CCOC(c2ccco2)(C2CC2)C1 N1(C(c2cnc(-c3ccco3)s2)=O)CCC(CO)c2ccccc21 N1(C(c2nccc(OC)c2F)=O)CCCC12CCN(C(c1ccc(=N)[nH]c1)=O)C2 C1(CC)CC(C(=O)NC(c2nn[nH]n2)C)CCN1C(c1cc(F)ccc1C)=O c1(C(N(C(C)CN(C(=O)CC2CCCCCCC2)C)C)=O)cnc2ncccn12 c1(C(N2CC(COC)(CNC(=O)C(C)OC)C2)=O)cc2c(=O)[nH]ccn2c1 C=CC(F)(F)C(=O)N1CCC(CCNC(=O)C(c2cc(C)oc2C)C)C1 CC1CCCCCN1CCNC(c1ccc(OCCOC)cc1)=O c1(C(C)NCC2CC(C(F)(F)F)CO2)ncc(C(=O)O)o1 N1(CC(N2CC=CC(NC(c3c(C(=O)OC)csc3)=O)C2)=O)CCN(C)C(=O)C1 C1(C(=O)NC(C)(C)CNC(C23CC(F)CC(F)(C2)C3)=O)Cc2cc(Cl)ccc2O1 c1(C(N2CCC(C(=O)OC)CC2c2ccccc2)=O)cnc2c(c1F)CCCC2 N1(C(CC2(C)CCCCC2)C(=O)NCCO)CC2(CCC(Cn3ccnn3)C2)C1 c1(C(=O)NCCCN(C)C(C2CCCN2C2CC2)=O)ccc2c(c1)CCCC2=O N1(C(c2n(CC)nc(C)c2Cl)C(=O)NC2CC(F)(F)C2)CCCC2CC1C2(C)C NC1(C(=O)NCc2cn(CCO)nn2)CCC2CCCC12 c1(C(c2n(C(C(=O)OC)C)nnn2)NCCCCC2CC2)ccc(C#N)nc1 N1(C(=O)CSCC(F)(F)F)CC2CCCC2(Nc2ncnc3c2CCO3)C1 N1(C(c2cc(C(=O)NC)n(C)n2)C(=O)NCCC)CCOCC1C#N c1(CC(F)=C(C)C)cccc(NC(=O)C(C)CF)c1.C12CCCC1C(=O)NC2 C(C(C)C(=O)NC1CC(C(C)O)C1)NC(C(C)OCCCC)=O c1(C(=O)NCC(CNC(=O)CCC(=O)c2cccs2)F)cncc(F)c1Cl CC1CCC(C)(C(N2CC(C(O)C(=O)NCCCCCO)C2)=O)C1 c1(C(=O)NC2CC(NC(C(N3CCC(O)CC3)C)=O)C2)ccc(N)c(C(F)(F)F)c1 N1(CC)CCCC(C(=O)NC2CCC(NC(C3COCCC3C)=O)CC2)C1 N1(C(c2n(C(C)C)ncn2)=O)CCCOC(CCNC(C2CC3C=CC2C3)=O)C1 N#CC1(C(=O)NCC#CC(=O)NCC2(CF)CC2)CC12CCC2 CCC(C)(COC)C(=O)NC1COCC1C(=O)NCC(=O)N(CC)OC C(=O)(CCCN=[N+]=[N-])NC(C1CCCCC1)CNC(C1CC(C)SCC1)=O C1(C)(Cn2cc(C(C)NC)nn2)CCN(C(=O)CCOc2ccc(C)cc2)C1 c1(C(=O)NCc2cc(C(=O)NC3(C)CCCC3O)n[nH]2)cc2ncccc2[nH]1 Cc1ccc(C(=O)NCC2CCN2C(=O)CCCCc2cnn[nH]2)cc1N C12(C(N3CC(Cn4cc(CCOC(C)=O)nn4)OCC3)=O)CC1COC2(C)C c1(C(=O)NCCOCCCNC(CCC(=C)C)=O)cc(C(F)(F)F)ccc1F N1(C(C(CC)NC(C)=O)=O)CC2CC(C(=O)O)C1C2 N1(C(Cc2c(C)scc2)=O)CCC(CSC2CCCN2C(c2cncn2C)=O)CC1 CCCCCCC(C)NC(C1(F)CCCN(C(=O)CC2(O)CCCCCC2)C1)=O c1(CC(N2C3C(CNC(c4c(CC)nc[nH]4)=O)C(C3)C2)=O)c(F)cc(Br)cc1F CC1(P(C)(C)=O)CCCN1Cc1ccc(-c2nn[nH]n2)s1 Cc1cc(Br)ccc1C(N1CCOC(CC(=O)NCC2(C)CCCC2)C1)=O S(=O)(=O)(CCC(=O)N(CCNC(c1cccc(C)c1N)=O)C1CC1)NC C=CCCC(C(=O)N1CCC(CSC)C1)NC(c1cnncc1OC)=O c1(OC)ncc(Cl)cc1NC(N1CCC1C1CCCOC1)=O CCC(C)(C#N)C(=O)NC1CCC(NC(c2ccc(NC(C)=O)cc2C)=O)C1 N1(C(C(=O)N(C)CC=Cc2ccccc2)=O)CCN(C2CCCCC2)C(C)C1 CC1Cc2c[nH]nc2C(C(=O)NCCCCNC(c2cc[nH]c(=N)c2)=O)C1 Cc1ccc(F)cc1C(C)NC1COC(c2ccccc2)C1 Cc1ccc(C(N2CCC2CNCC(C)O)=O)c(C)c1.c1(SCC2CC2)ccccc1.C N1(C(CC(=C=C)C)=O)CC2(CCN(C(c3c(OCC)ncnc3OC)=O)CC2)C1 C=CC(C)CC(=O)NCCC(O)C(=O)N(CC(C1CC1)OC)C n1(CC)cc(C2CC2C(N2CCC2(c2ccccc2)C2CC2)=O)cn1 Cc1nc(C(N2CCC(n3cc(C4(CO)CC4)nn3)C2)=O)nn1-c1nc[nH]n1 CCC(F)(F)CC(=O)NC1CC(C(=O)NCC(C2CC(C)(C)C2)O)C12CCC2 c1(OC)cc(C=CC(N2CC(O)CC2CC(=O)NC2(C)CC2)=O)ccc1O N1(C(C(C)CN(C(=O)C(c2ccn(C)c2)C)C)=O)CCC12CCCOCC2 c1(Cc2nc(CC(=O)N)[nH]n2)ccccc1F.N12CCC(C1)Cn1cc(nn1)C2 N1(C(C(C)SC)=O)CCCC(CN(C)C(c2cc(C)sn2)=O)C1 Cc1cnc2nc(C(=O)NC(C3CCOC3)CNC(=O)CC(F)(F)F)nn2c1 C(CN=c1[nH]c(=NCCCOC(F)(F)F)c2ccccc2[nH]1)c1c(C)c(Cl)ccn1 c1(C(=O)NCC(CC)NC(C2(C(=O)NC)CC2)=O)cccc2sccc12 n1(CCC(=O)N(CC(=O)N(C2CCOC2)CCF)CC#C)ccnc1C N1(C(c2cc(CC)n(C)n2)=O)CCCC(F)(C(=O)NC2CN(C)NC2=O)C1 c1(C(N2C(C(=O)Nc3ncc(Br)nc3Cl)C3CCC2C3)=O)cnc2[nH]ccc2c1 C(C)(C)(CCC(=O)NC1CCC1(C)C)NC(C(C1C(C)C1)C1CCC1)=O N#Cc1nccc(N2CC3CC(NC(=O)C=CSCc4ccco4)C3C2)n1 c1(C(=O)NC2CCN(c3cc(OC)ncn3)C2)ccc([N+](=O)[O-])cc1C c1(CC)conc1CC(=O)N(C1CCN(C(=O)CCC2(O)CCC2)C1)C Cc1ncnc(C(=O)NC2C3CCC2N(C(=O)C(C)OCC2CCCO2)C3)c1C C(=O)(N1CCCc2nncn21)C1C2(CCN(C(C(n3ncc(C)c3)C)=O)CC2)C1 C1(NC(Cc2cn(CC)nc2)=O)CC12CCC(NC(=O)CC1CCOC1)CC2 N1(C(CNC(=O)CN2C(=O)CCC2CC(O)CC(F)(F)F)=O)CCc2ccccc21 c1(CCC(=O)NCC(N(C(=O)Cn2cnc(=N)[nH]2)C)C2CC2)cccc(F)c1Br Cc1ccc2c(CC(=O)NCCC(C)(C)NC(c3coc(CO)c3)=O)c[nH]c2c1 c1(N2C(CC)CN(Cc3ccc(C)s3)CC2)ncc2[nH]ncc2n1 Cc1nc(C(=O)NC(C2CN(C(=O)CC(C)(C)CN(C)C)C2)C)c(=O)[nH]c1C C1(C(N)=O)(CNC(=O)CC2(C)CC2F)CN(C(C2CC(F)(F)C2)=O)C1 C(C1CCCc2ccccc21)NC(NCCCOC)=NCCC(C)P(C)(C)=O N1(C(C=Cc2ncc(C)[nH]2)=O)CC2CC(C1)N(C(=O)COc1ccccc1F)C2 N1(C(CCCOCCC)=O)CCC2CN(C(=O)C(C)(C(C)C)OC)CC12 c1(CC)cc(C(=O)N(CCC(C)NC(C2CCS(=O)(=O)N2)=O)C)ccc1C c1(OC)ccc(Cl)c(CN2CC(F)(F)CC2C(=O)Nc2cccc(O)c2)c1F C(=O)(C(F)(CNC(=O)C1=CCCSC1)C(C)C)N1CC(SC)C1 C(=O)(C(C)CC(=O)NCC1CC1CC(=O)NC(c1c(C)n[nH]c1C)C)OC c1(C(=O)NC(C(=O)N(C)Cc2nnc(C)s2)CN(C)C)cccc2c[nH]nc12 C1(NC(C2CNC(=O)N2)=O)C2CCC1N(C(c1nccn1Cc1ccccc1)=O)C2 Cc1ccc(C(N2CCOCC(NC(c3cc(CC(C)C)[nH]n3)=O)C2)=O)c(C)n1 c1(C(=O)NCC2C(CNC(C(CCCC)O)=O)C2)cccc2oc(=N)[nH]c12 N1(C(C=C(C)C(F)F)=O)CC(CNC(c2ocnc2-c2ccccc2)=O)C(C)C1 c1(C(N2C3CC(NC(C=CCC)=O)C2CC3)=O)c[nH]c2ccc([N+](=O)[O-])cc12 c1(N(CCCNC(c2cn(CCF)nn2)=O)C)cccc2ncnc(O)c12 c1(CN(C)Cc2ccc(CC=C)cc2)cccc(Br)c1F C#Cc1cc(C(N2CC(CNC(=O)CSc3cccc[n+]3[O-])C2)=O)cc(Cl)c1 C1(CN2Cc3c(NC(=O)OC(C)(C)C)ncnc3C2)CC2(CCCCC2)C(=O)O1 Cc1cc(Cl)cc(C(=O)NCC2CN(C(=O)Cc3nc[nH]n3)C(C)(C)C2)c1O N1(C(CC(C)(C)C)=O)CCC2(CNC(C3CC3C(F)(F)F)=O)CCCC12 N1(Cc2cccc(C(C)C)c2)CCN(C(=O)C(C)(F)F)C2(CC2)C1 C#CC1CN(C(C2CC(=C3CC3)C2)=O)CCN1C(c1cccc(SC)c1)=O C1(NC(CCOCC)=O)CN(C(c2ccc(Cl)c(C)c2O)=O)CC(C)(C)C1 c1(C2C(C(=O)NC34CN(C(=O)CC5CC5(Cl)Cl)C(C3)C4)C2)c(Cl)cccc1Cl CCCCC(CN=c1[nH]c2cc(Br)cnc2s1)NC(=O)C(C)N(C)C C=CCC(C)(C)C(=O)N1CCC(CCNC(=O)CC2CCCC(C)C2)CC1 c1(C(=O)NCC(C)CNC(C2COC(C)C2)=O)cc2n(n1)CCO2 N1(C(C(C)OCC#C)=O)CCOCC1CC(=O)NC(C)CC(=O)OCC C(=O)(C1=C(C#N)CCC1)N1C(CCCNC(CC2(OC)CCCC2)=O)CCCC1 C1(CN(C(CCC=C)=O)C)CCCCN1C(c1cc(C#N)c[nH]1)=O c1(C(N2CC(CC)CC(C)C2)C(=O)NCCCC)ccc2n[nH]cc2c1 c1(C(=O)NCC2CCCC2NC(C23CC(C(F)F)(C2)C3)=O)ccccc1[N+](=O)[O-] c1(C(=O)NCC2(NC(CC3C(C)=NOC3=O)=O)CC2)ccc2nc(CO)[nH]c2c1 N1(C(=O)NC(c2ccon2)C)CCC2(CCCC(CO)O2)CC1 C1(CNC(C2(CCC)CCC2)=O)CCCN1C(C1CC1c1ccnn1C)=O c1(-n2c(C3C(OCCOCC)CC3)nc(CC(C)C)n2)ccc(OC)c(Cl)c1 C1(NC(c2ccsc2)=O)(CO)CCN(C(=O)CCc2nncs2)C1 Cc1cnccc1-c1ccc(C(=O)NC2CCC2NC(=O)CC2CC=CCC2)s1 C(=O)(C1CCCn2nccc21)NC(C)CCCCNC(C1(O)COC1)=O N1(C(c2c(OC)c(C)cs2)=O)CCCC(C2CN(C(=O)CNS(=O)(=O)C3CC3)C2)C1 C1(F)(CNC(C(n2cc(Cl)cn2)C)=O)CC(NC(C2CC2(C)C)=O)C1 C1(NC(c2occ(C)c2)=O)CN(C(=O)C(C)NC(C)(C)C)CC12CCOCC2 N1(C(CC=C=C)=O)CCC(C2CC2)C1CNC(c1nc(C)ccc1F)=O c1(C(=O)NC2CN(C(c3cccc4nc[nH]c34)=O)C2)cc(F)c([N+](=O)[O-])cc1F C(CC(C)(O)C(=O)N1CCC(Cn2cc(CC(O)C(C)(C)C)nn2)C1(C)C)NC N1(CC(=O)O)CCCCC(NC(c2ccnc(-n3cccn3)c2)=O)C1=O C1(CNC(=O)CCc2ncc(C(C)(C)C)o2)CCCCC(=O)C1.CC12CCCN1C2 c1(C(=O)NC(CC)CN(C(=O)CC(C)CF)C)ccc(Br)cc1OC C12(C(=O)NC(C)CNC(=O)CC(C)N3CCCC3=O)CCC(C)(CC1)OC2(C)C C=CC1C(C(=O)N(C(C)CN(C(=O)CSc2nnnn2C)C)C)C1(C)C CCCCS(=O)(=O)CC(=O)NCC1CN(C(=O)C(CCO)N(C)C)CC1C c1(C(N2CC(N(C(C(CC)n3cncn3)=O)C)C2)=O)ccc2c(c1)CCN(C)C2 c1(C(N2CC3CCCC3(CSC)C2)C(=O)NCCSC)cccc2sccc12 C(=O)(C1=C(C)S(=O)(=O)CC1)NCC1(CNC(C(C)=C(CC)C)=O)CC12CCC2 CC(C(CO)NC(C1(C)CCC1)=O)NC(C1(C)C=CCC1)=O N1(C(COCCCC)=O)CCCCC1CCNC(=O)C(C1CCC1)SC C1(CNC(C(=O)NC(c2ccc(C#N)cc2)C2CCC2)=O)CCOCC12CCCC2 C(=O)(CC(O)CCCC)NCC12CC(NC(c3c(CC)oc(C)c3)=O)(C1)C2 C1(C2N(C(=O)CCC3CCCC3)CC2)CCN(C(c2cnsn2)=O)CC1 c1(CNC(C(C)C2CCC2)=O)nc(C(=O)NC(CO)C(N)=O)co1 CC1CC(NC(C2CCC(NC(=O)CC3(C#N)CC3)C2)=O)CN1C1CC1 C(C)(C(C(=O)N1CCCC1C(C)(C)C(=O)N1CCC(CN(C)C)C1)N(C)C)OC C1(CCOC)CCN(C(C2(CCNC(c3coc(CO)c3)=O)CC2)=O)CC1 C(=O)(CC(O)(C(F)(F)F)c1ncco1)N(CCN1CCCC(C)C1)C(=O)C1CC1 c1(CNC(C2C(C(N3CCC(CC(=O)OC)CC3)=O)C2)=O)ccc(F)c(F)c1 c1(C(N2C(C)CC(NC(c3ccc(C(N)=O)cn3)=O)C2)=O)cc2occc2s1 O(P(=O)(CNC(=O)NC(C1CCCCO1)C1CCC1)OCC)CC Cn1nc(C(F)F)cc1C(N1CCC(CCNC(=O)CCCC2CCC2)CC1)=O C=C(C)CN=C(NCc1cccn1C)N1CCC(C)(C)C1.C(COC)C1CC1 c1(CC)cc(=NCC2CC(NC(=O)CN(CC)CC3CC3)CCO2)[nH]c(C(C)C)n1 N1(C(=O)CN(C2CC2)CC2CCCCO2)CCN(C(=O)CC23CCCC2C3)CC1 CC1CC(NC(C2(C(=O)NC3CC3)CC2)=O)CN1C(=O)CCSc1ccccc1 c1(C(=O)NCC2N(C(c3c(C)csc3Cl)=O)CCC2)ccc2c(C)[nH]nc2c1 CC1CN(C(=O)CC2CCCC3CC23)CC(C(N2C3CSCC2C3)=O)O1 C1(CN(C(c2ccc(Cl)n2C)C(=O)NCCCSCC)C)CCc2nccn2C1 C(C(C)(C)C(=O)N1CCC1(C)C(N)=O)NC(C(CC)n1cncn1)=O N1(C(C(C)=C2CCCC2)=O)CCC(C)(CNC(c2coc(C(F)(F)F)n2)=O)CC1 n1(C(C)C)cnc2c(NCC(C)(F)F)[nH]c(=NCC3(N(C)C)CCC3)nc12 N1(C(c2c(C)cnnc2O)=O)CCN(C(c2cc(C#N)c[nH]2)=O)C(C)CC1C c1(C(c2n(CC)nnn2)NCC2CC3(CC3)C2)cc(Cl)ccc1OC(F)F c1(C(N(CCCN(C(=O)COCC2CCCO2)C)C)=O)scnc1CCC C1(CCCCNC(C(CC)OCC)=O)CCN(C(=O)C=CC2CCCC2)CC1 c1(OC)ccc(CC(N2CCCN(C(=O)C=C3CCOCC3)C2)=O)cc1F c1(C(N2CCCC(C)(NC(c3c(CC)noc3C)=O)C2)=O)cccc2nonc12 C12(C(=O)NCC3(C(N)=O)CC3)CC1CCN2C(c1cc(C(F)F)no1)=O C(=O)(CCC(C)C#N)N1CCC(N(CCOC)C(C)=O)CC1.C(COC)S C(=O)(CCC1=CCCCC1)NCC(C1CC1)NC(C(C1(OC)CCCC1)(F)F)=O C(=O)(C1=COc2ccccc2O1)N1CCN(C(COCCC)=O)C2C1C2 C(CCCCC(=O)NC(c1ccnn1C)C(N1CCC(c2cnco2)C1)=O)OCC c1(C(=O)NC(CCCC)CNC(=O)CN2CCCC2C)cc2ccnc(Cl)c2[nH]1 n1(CC)cccc1C(=O)NC1COCC1NC(c1ccc(CCCCCC)s1)=O C1(CC(=O)N(C(C)CCNC(c2ccc(=O)oc2)=O)C)CCC(F)(F)CO1 C1(C(C(=O)NC(COC)COC)F)CCN(C(=O)CN(C)C)C1 N1(C(C(C(CC)O)(C)C)=O)CCC(C2(NC(c3cocc3C)=O)CCC2)CC1 Cc1nsc(N)c1C(N1CCC(CCC(=O)NCC2CCCN2C)CC1)=O N1(C(C(C)C2(O)CCC2)=O)CCCC(C(N2CC(CN(C)C)C(O)C2)=O)C1 CC1(C)CCC(C(=O)NCCC2(O)CCN(C(=O)C=Cc3cn[nH]c3)CC2)CO1 C12(C(=O)NC3C=CCN(C(Cc4n(C)ccc4)=O)C3)CC1CCC2(F)F C1(C(=O)NCC(C)N(C)C)CCN(C(C2CC2c2cccs2)=O)C12CC2 C(CCCCC(=O)N(c1ccccc1)CCNC(C1CCC12CCC2)=O)SCC c1(CC)cccc(C(=O)NCC2CC(NC(=O)CCC#N)C(O)C2)n1 N1(C2CCN(C(=O)CC3CC3)CC2)C2CCC1CN(C(=O)Cc1ccc(O)nc1)C2 c1(NC(C(C2CN(C(c3c(CC)nc[nH]3)=O)C2)OC)=O)ccc(C)c(C)c1 C1(C(=O)NCC(C2CC2)NC(=O)CCOCC(F)F)CN2CC3CC2(CO1)C3 C1(CNC(=O)CC2C=CCCC2)CCN(C(=O)C=CC2CCCCC2)CC1(F)F C12(C(=O)NCc3c(C)cc(C)s3)CC(CN(C(=O)CN3CCCNC3=O)C1)C2 N1(C(C2ON=C(C)C2)=O)CC(C(F)(F)F)C(CNC(C2(C(N)=O)CCC2)=O)C1 C#CCCCCCC(=O)N(CC(C(=O)N(CCCO)C)OC)CCCO C(=O)(C1=CCC(F)(F)CC1)NC1CCCC(CNC(C2CN(CC)C(=O)C2)=O)C1 CCC(C)CCCCC(=O)NCC1CCC(F)(CNC(C2(C(C)C)CC2)=O)CC1 n1(CC(=O)NC(CCCCNC(CSCC=C)=O)C)ccc2c(C)cccc12 c1(C(=O)OC)cc(C)[nH]c(=NCCOCC2(C(F)F)CC(N)C2)n1 c1(CNC(C(n2cc(-c3c(OC)cccc3F)nn2)C)=O)cc2c(ncn2C)s1 Cc1ccc(C)c(CCCCNC(N2CCN(c3ccccc3C)CC2)=O)c1 C1(C(N(c2ccccc2CCC#N)CC)=O)CC(F)CN(C(c2cnsn2)=O)C1 c1(C(c2n(CCC(=O)OCC)nnn2)NC2CC2F)cccc(C)c1Cl c1(SC)cccc(-c2cccc(N3CCN(Cc4cnc(CCN)s4)CC3)c2)c1 c1(C(=O)NC(C)CCNC(c2cccn2Cc2cccnc2)=O)nc(=N)cc[nH]1 C(CCCCC(=O)N1CC(N(C)C)C(NC(=O)CCC(C)(C)C)C1)SC c1(NC(N2CCC2Cc2ccccc2Cl)=O)ccnnc1OC1CCCC1 n1(C2CC(C(=O)OCC)C2)c(-c2ccc(O)nc2)csc1=Nc1cccc(OC)c1 N1(C(c2n(CC)ncc2)=O)CCN(C)C(CNC(c2ccc(=O)n(O)c2)=O)C1 N1(C(C2C(CCC)C2)=O)CCOC2(CCC(NC(C3(Cl)CC3(F)F)=O)CC2)C1 C1(C(=O)NCC(CCNC(c2cccc(OC)n2)=O)(C)C)COCCC1(F)F c1(Cc2c(C(=O)NC(CNC(CC=C)=O)C3CCC3)con2)ccc(C)cc1 CC1CCN(C(=O)CCC2CCN(C(c3coc(C(F)F)c3)=O)C2)CC12CCC2 N(C1CCCc2cnn(C(C)C)c21)C(COc1ccc(NC(C)=O)cc1)=O C(=O)(CC(CC)C(C)C)NCCN(CCC)C(c1cc(C)ccc1O)=O Cc1cc(=N)[nH]c(=NCCCN(C)N(C(C)(C)C)C(C2(C)CC(O)CN2C)=O)[nH]1 CC(C)(C)C(CC(=O)NCCNC(c1ccc(C(F)(F)F)c(N)c1)=O)C(F)F c1(C(=O)NCC(CNC(=O)C=CC2CCCO2)O)ccc(=O)n(C2CC2)c1 c1(C(C2(C=O)CC(=O)C2)N2CC(C3CCCO3)C2)cccc(Cl)c1.c1nn[nH]n1 c1(C(=O)NC(CNC(COCC=C)=O)C(C)C)c(C)nn(-c2ccccc2)c1Cl N1(C(C(C)S(C)(=O)=O)=O)CCN(C(=O)Cc2cnc(C3CC3)[nH]2)C2(CC2)C1 C(C)(CC(=O)NCc1cocn1)NC(C1C(CC)C1)=O C1(C(=O)NC2C(NC(c3c[nH]nc3-c3ccncc3)=O)COC2)CCC(F)(F)C1 c1(C(=O)NCCC(C)N(C(c2nn(CC)c(C)c2)=O)C)cccc2ccnn12 C(=O)(C(CN=[N+]=[N-])NC(=O)CC(C)(C)F)N(CCN(CC=C)C)CC C=C1CCC(C(=O)NC2(CC(N3CCC(O)(CO)C3)=O)CC2)CC1 CC1C(NC(C2(F)CCC(=O)CC2)=O)CC2CCC1N2C(=O)Cn1nnc(=O)[nH]1 C=CC(O)C(=O)NCCCCCN(C)C(c1conc1C)=O CCC(C(=O)NCCC(C)NC(N)=O)N(C)C(C1CCC(=O)O1)=O c1(N2C(CNC(c3c(C)noc3C(F)(F)F)=O)CC2)ncnc2c1SCCC2 c1(OC)cc(N)c(C(N2CCCCC(NC(=O)CC=C(C)C)C2)=O)cc1OC C(CCCC(CO)NC(C1(C#N)CC(C)C1)=O)NC(C1C(OC)CC1)=O n1(CCOC)cc(C(=O)NC(C)(Cc2ccccc2)C(=O)OC)c2ccccc12 C1(NC(CSCCCC)=O)CCCCC1CC(=O)Nc1ccc(CCO)cc1 N1(C(=O)CC2CCCN2Cc2cncnc2)CCC2(CCCOC2)C1 N1(C(C(C)CN2CCOCC2)=O)CC(CNC(=O)CSC2CC2)C(C)(C)C1 CCC(C)(O)C(=O)NC1CC(C(=O)NCc2c[nH]nc2C2CC2)CC1O C1(NC(=O)C2CC2)CCCCC1.C12(C(=O)OC)CC(NC(=O)C(C)O)(C1)C2 C1(NC(CCC(=O)NC)=O)CCN(C(=O)COc2ccc(Cl)cc2)CCC1(F)F Cc1cccc(C(=O)NC(C)(CNC(=O)C(F)=CC2CC2)C(C)C)c1Br c1(CSC)ccc(C(=O)NCCCCC2CCCN(C(=O)CC(C)C#N)C2)cc1 c1(C(C(=O)NCCC(C)NC(C2CCC(C(=O)OC)C2)=O)OC)ccccc1Cl CC(O)CCC(=O)NCCC1COCCN1C(C1CC2(CCC2)C1)=O N1(C(C(C2CCOC2)OCC)=O)CC2(CN(C(C3CCCCO3)=O)CC)CCC1C2 N1(C(c2c(C)cno2)=O)CC(CNC(=O)CCC2CC2C)CC1(C)C c1(OCC)ccc(C(O)C(=O)NC(c2ccccc2)NC2CCC2)cn1 N1(C(C2CCCN(C(N)=O)C2)C(=O)NCCCc2ccccc2)CC2CCCC2C1 c1(OCC)ccc(C(N2CCCCC(NC(C3CC(O)C3)=O)C2)=O)cc1Cl C1(C(=O)NCCn2cnnc2C)(OC)CCN(C(c2c[nH]c(=N)o2)=O)C1 Cc1ccc(NC(C2CCN(C(c3ncn(C)c3C)=O)C2C)=O)c(C)c1O c1(C(=O)NC(N)=O)ccc(Br)cc1Cl.CC1C(=O)NCC2(CC2)CN1C C1(CNC(CCc2n(C)cnc2)=O)CN(C(c2ccccn2)=O)CC12CC2 N1(C(c2cncc(C)c2)=O)CC2ON=C(CNC(c3cnc(C(C)C)s3)=O)C2C1 n1(CC)cnc2[nH]c(=NCCS(=O)(=O)CC(F)(F)F)nc(N3CCC(SC)C3)c12 CCC(CC)C(=O)N1CC(F)CC1CN(C(=O)COc1ccccc1CC)C C12(NC(C3(NC(C(C)CC4CC4)=O)CCC3)=O)CC3CC(CC1C3)C2.N1CCOCC1 C1(C)(CC)CCC(C(=O)NCC#CCNC(=O)C(C)CO)CC1 N1(C(CCC(C)=O)=O)C(C(=O)Nc2cnn(C(F)(F)F)c2)CC2CC12 C1(C)(CN(C(c2nnc(NC(N3CCOCC3C)=O)s2)=O)CC)CC2CCC1C2 C1(C(=O)NCC2C(NC(c3n(CC(=O)OCC)ncc3)=O)C2)CC2(CCOC2)C1 N1(C(C2CCCN(CC)C2)=O)CC(NC(C2CSC2)=O)CC12CCC2 CCC(CC)CC(F)C(=O)N1CCCC1(C)C(=O)Nc1cccn2ccnc12 N1(C(c2c(Cl)cn(C)n2)=O)CCC(C(F)(F)F)C(NC(C2(CO)CCC2)=O)C1 c1(C(=O)NCCN(CC(C)O)C(c2c(C)csn2)=O)nc(C)c(C)[nH]c1=O c1(OC)cncc(C(N2CC3CC3(NC(=O)CN3CC4CC4C3)C2)=O)n1 C(CC(=O)N1C2CCC1CC(F)C2)(CC(C)C)NC(C(CCC)C#N)=O CS(=O)(=O)c1ccc2c(c1)C(NC(=O)C1=C(Cl)C=CC=C(Cl)OC(N)SCC1=O)CC2 C1(OCC(=O)OC(C)(C)C)CCCCC1n1cc(C2(C)CCOC2)nn1 N1(C(C2(CSC)CC(O)C2O)=O)CC2(C1)CN(C(c1cc(OC)ccc1Cl)=O)C2 C12CC3CCC1N(C3)C2=O.c1(OC(C)C(=O)NC2(C)COC2)ccc(Cl)cc1 C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CC=CC(NC(C(C)n2cncn2)=O)C1 CCCCC(O)CC(=O)N(C1CCCN(C(=O)CCc2cnc(O)[nH]2)C1)CCO C(=O)(CCCCCC(C)C)N1CCC(CC)C1C(=O)NCC(C)C(=O)OC c1(C(N2C(C(=O)NCC3(OCC)CCC3)CC2C)=O)cc(C)cc(C)c1 c1(SCC(N2CCC(C(C(C)C)NC(=O)Cn3cccn3)CC2)=O)nccc(=N)[nH]1 C(=O)(C(C(C)NC(c1nccn1C)=O)C(C)C)NC(CCCC)C c1(C(=O)NCC2N(C(C(C)S(N)(=O)=O)=O)CCC2)ccc(Cl)c(F)c1N c1(N2CC(N(C)C)C3(C2)CC3)ncc(S(C)(=O)=O)cc1[N+](=O)[O-] Nc1c(Cl)cnc(C(=O)NCCCCNC(C2CCOC2C2CC2)=O)c1Cl N1(C(c2n(C)c(O)nc2)=O)CC2(C1)CN(C(c1nnn3c1CCC3)=O)CCO2 CCCCC(O)C(=O)NC1CN(C(=O)COC2CCCCC2)CC1CC(C)(C)C c1(C(=O)NCCN(CCC)C(c2nsnc2O)=O)cc(S(N)(=O)=O)cn1C c1(CC(=O)N(CC(C)O)CCNC(=O)CCn2cncn2)cccc2ccoc12 c1(C(=O)NCC(CC)NC(C2(OCC)CCOC2)=O)cc2cc(C)cc(C)c2[nH]1 c1(C(=O)NC(C(=O)NC2C(C=C)COC2)Cc2ccoc2)ccc(=O)n(C)c1 C1(C(N2CCC(CNC(=O)CCn3ccnn3)C2)=O)CCN(C2CCSC2)CC1 c1(C(N2C(C(=O)NCC3(C#N)CC3)CC(F)C2)=O)ccc(F)c([N+](=O)[O-])c1 Cc1cc(C(=O)NC(CO)C(C)NC(C2CCCOC2C)=O)c2n[nH]cc2c1 C(c1cncnc1O)=C(C)C(N1CCC(C(=O)NCCn2cnnc2)(C(C)C)C1)=O Nc1cncc(C(=O)NCC2CC(O)CN2C(C2(F)CCOCC2)=O)n1 N1(C(c2c(CC)oc(C)c2)=O)CCC(C)N(C(=O)C(C)P(C)(C)=O)CC1 N1(C(c2ccc(C)o2)C(=O)NC(C(=O)OC)C)CCn2nccc2C1 C(CCCC(=O)NCC1CN(C(C2CCN(c3nccs3)CC2)=O)C1)(OC)OC C1(C(=O)NCCC(=O)NCCN(C(=O)Cc2cc[nH]c2)C)CCCC1O C1(N(C(CC(=O)NCC#C)=O)C)CCCCN(C(c2nc(Cl)cs2)=O)C1 N1(CC(N2CCCC(NC(C(C)(C3CC3)OC)=O)C2)=O)CCCCCC1=O C(=O)(C(C(C)NC(c1cc2ccccc2o1)=O)C(C)C)NCCCCC=C Cc1sc(CN(C)N2CCC2C)nc1-c1ccc(-c2ccccc2)cc1 CN1CC(CC(=O)NCc2occc2C(=O)N(C)CC2CC(F)(F)C2)CC1=O CC(C)CCCCCC(=O)N1CC(O)CC1CNC(c1ncc(C#N)cc1Cl)=O c1(NC(CCc2ccc(C)nc2)=O)ccc(C(=O)NC(=O)C=CC(C)(C)C)c(C)c1 CC1CCCC(CNC(=O)CC(O)CNC(=O)CN(CC(C)(C)C)C)C1 c1(C(N2CC(O)(C(C)NC(c3nccc(N)c3Cl)=O)C2)=O)ccc2cncn2c1 C1(CC)CN(C(=O)CC(F)(F)F)CC1C(N1CCCC(C(C)(C)O)C1)=O Cc1c(N)ccc(C(N2CCCCC2CNC(=O)Cc2cccc(F)c2)=O)c1C C(=O)(C1CCc2nccn21)C.C1(C(C)C)CC(C(=O)NC)CCO1.C1(=O)NCCN1 c1(C(=O)NCC2C(NC(CCNC(N)=O)=O)CCC2)c(NC(=O)CO)cccc1F C(Cn1cncn1)(C(=O)NOCC=C(C)C)NC(C(COCC)(C)C)=O CCC(C)C(C(=O)N(C1CCN(C(c2[nH]cnc2C)=O)CC1)CC1CC1)OC c1(C(N2CCC3CN(S(=O)(=O)CCCCl)CCC23)=O)ccc(I)cc1[N+](=O)[O-] C(=O)(C(CCCC)c1ccccc1)NCC(C1CCCCC1)NC(C(F)=CC)=O N1(C(COCC=C)=O)C2CCC1C(C(=O)NCC1CC=CCC1)C2 CC1CN(C(c2coc(CO)c2)=O)CCN(C(c2c[nH]c3ccccc23)=O)C1 N1(C(C(C)N(C(C)=O)C)=O)CCN(C(c2cscc2C(F)F)=O)C(CCO)C1 N1(C(c2cc(C)cc(Cl)c2)=O)C2CCC1C(C)C(NC(C1CC3CCC1O3)=O)C2 c1(C(=O)NC(CC)(C)C(=O)OC(C)(C)C)cc(C(F)(F)F)cc(N)c1 C(=O)(C(C)(O)CC(C)C)N1CC(C(N2CCC(C)(N(C)C)CC2)=O)(COC)C1 c1(C(N2CC(N(C(c3ccc(CC(C)C)o3)=O)C)C2)=O)c[nH]c2cccc(Cl)c12 c1(CC)nc(C)c(C(N2CCC(C)(NC(C3CNC(=O)N3)=O)CC2)=O)c(C)n1 CC1CC(CNC(C2CC2CNC(=O)CC2CCC2)=O)C1 C1(NC(c2ccnc(Cn3cnnc3)c2)=O)CN(C(=O)CC(F)F)CCC1CO c1(CN(C2CCN(C(COCC)=O)CC2)C(=O)C(O)CF)ccc(F)c(Cl)c1 C1(C(=O)NCC(CC)(C)O)CCN(C(C23CCCN2CCC3)=O)C12CCC2 C(=O)(C1=CCCCCC1)NCC(=C)CCNC(c1cccc(F)c1C(C)C)=O C1(O)(C(=O)NCCN(C(c2cc(OC)ncn2)=O)C)CCCC(C)(C)C1 CCC(C)C(C(=O)OC)N(C(=O)CCc1cc(C)on1)CC.c1cncc(C)c1 N1(C(CCC2(CCC#C)N=N2)=O)CC=C(CC(=O)c2ccccc2)CC1 c1(NC(c2nc(NC(c3c(OC)nccc3I)=O)sc2)=O)cnn2c1CCCC2 c1(C(N2CC(CNC(C(C)OC)=O)C(O)C2)=O)c(C)ncnc1C C(=O)(CC(COC)COC)NC(CN(C(=O)CC1CCCC1)CC)C C12CC(C13CCC3)NC2=O.N1(CC)CCN(C(=O)COCC2CC2)C(C)C1 S(=O)(=O)(c1cnc(N(C)CCF)c(Cl)c1)NC1(C)CCC(C)C1 c1(C(=O)NCC(=O)NC2CC(CC(=O)Nc3c(C)noc3)C2)ccncc1F C#CCCC(O)C(=O)NCC1CCN(C(C2CC(OC(F)(F)F)C2)=O)C1 C#CC1COCCN1C(=O)C(C)CN(C(=O)C(C)(C)C(F)F)C C12(C(N(CCC(C)NC(c3ccncc3F)=O)C)=O)CC3CC(C1)CC(O)(C3)C2 C(CCCC(=O)N1CCCC1CN(C(=O)Cc1nccs1)C1CC1)N(C)C c1(OC)ccc(Br)c(NC(=O)CC2COCCN2c2ncnc3cc[nH]c23)c1F C1(C(=O)NCC2CN(C(C3CC=CC3)=O)CCO2)CSC(c2ccccc2)=N1 C(N=c1[nH]c(=NCC2CC(C)CC(C)C2)c2cccc(F)c2[nH]1)c1c(C)noc1 C(=O)(CCCCCN(C)C(C1(C2CCCO2)CC1)=O)NC(C#C)(C)C1CCC1 N(C1CCCc2ccoc21)C(C(C)(CO)NC(CCOCCOC)=O)=O CC1C(=O)N(CC(=O)NCC2COCCN2C(=O)CN2CCCCC2)C(=O)C1C C(=O)(CCC(F)(F)Cn1cc(NC(=O)C(=O)NOC)nn1)NC(CC)C(N)=O N1(C(COC(CNC(CC=CCCCCC)=O)(C)C)=O)CC2(COC(=O)C2)C1 c1(CCn2cc(-c3ncc(N)cn3)nn2)cc(Cl)ccc1CC(=O)N(CC#N)C c1(C(C(N2CCCC(NC(C(=O)N(CC)CC)=O)C2)=O)O)ccc(F)c(Cl)c1 C1(NC(c2cnn3ccsc23)=O)CCC2(CCN(C(=O)CCc3csnn3)C2)C1 Cc1ncc(C(=O)N(C)Cc2cn(CCN3CCC(N(C)C)C3)nn2)cn1 N1(C(c2c(OC)ccc(F)c2N)=O)CC(NC(=O)CCSC)C2(CCOCC2)C1 C1(C(=O)Nc2ccc(C)cn2)Cc2cc(O)ccc2CN1Cc1ccccc1Br C(=O)(C(C)(CO)NC(=O)CN1CCNC1=O)NC(CC(=O)OCC)C c1(OC(C)C)c(Br)cccc1S(=O)(=O)NCCc1nccn1C C1(C2C(C(=O)NC3CC(C#N)C3)CCO2)CCN(C(=O)CSc2nncs2)CC1 c1(C(N2C(CN(C(=O)COC(F)F)CC)CCC2)=O)cc(C)c(O)c(N)c1 N1(C(c2scc(C)c2)=O)CCCC2CC(NC(=O)C(F)(F)CN3CCCC3)CCC12 Cc1cc(Br)cc([N+](=O)[O-])c1NC(N1CCc2sccc2C1Cc1ccccc1)=O C1(C(=O)NC2C(OC)CN(C(c3sccc3Cl)=O)C2)CN2CCN1C(C)C2 CC(C)(CCC(=O)N1CC(C(N2CCCCCC2)=O)CC1(C)C)[N+](=O)[O-] C1(CNC(c2cncnc2)=O)CC2(CC2)CN1c1cc(C2CC2)ncn1 CC(C)(CC#N)C(=O)NCCC1CSCCN1C(=O)Cc1cccc(N)c1 c1(C(=O)NCC2CCC(NC(C3CC(C#N)C3)=O)C2)ncc(F)cc1F N1(C(COC(C)C)=O)CCN(C(c2sccc2C(F)F)=O)C2(CC2)C1 C1(C(C)(C)C)CN(C(=O)Cc2cccc(Cl)c2)CCN1C(C1CC1F)=O c1(NC(C)=O)cc(S(=O)(=O)NC(C)CCN2CCCC2)c(Br)cc1Br c12sccc1S(=O)(=O)C(=O)N2.C1(C(N(C)CC)=O)(NC(=O)OC(C)(C)C)CC1 N1(C(C2C(=C)CC2)=O)CC2(CCN(C(C3(C(=O)NC)CC3)=O)CC2)CC1C c1(C(=O)NC(CNC(CCOCCOC)=O)C2CC2)oc(CO)nc1C c1(C(C(=O)NCCC(O)C2CC2)NC(CCSC)=O)ccnn1C CC(CNC(=O)C(c1ccoc1)NC(=O)Cc1cncn1C)C(F)F C(=O)(C1CCc2cccc(F)c21)NC1CCN(CCNC(C(CCC)C)=O)CC1 C1(NC(c2nc(C)nc(O)c2)=O)CCN(CC2CCC(C)C(C)C2)CC12CCC2 CC(C)(C)CCCCC(=O)NC1CCC1NC(c1c(O)ccc(F)c1Br)=O CC(C)CC(C)(O)C(=O)NCC1(O)CCCN(C(=O)CN2C(=O)CN(C)C2=O)C1 C1(CC(=O)NC2CC(F)(F)CC2NC(c2ccc(CO)o2)=O)CC2(CCC2)CO1 C1(C)(NC(C2(CNC(c3ncccc3C)=O)CC(=C)C2)=O)CCC(=O)NC1=O C1(N2C(CC3(Br)CC3)C(=O)NCC2)CC(=O)NC1=O.C(C)(=O)NC.CO N1(C(C=CCC)=O)CCC(C2OCCCC2CNC(C2(F)CCCCC2)=O)CC1 S(=O)(=O)(c1cccnc1NCc1ccc(CS(C)(=O)=O)cc1)NCC(C)OC N1(C(C(C)(C)OC)=O)CCCC(n2cc(C(C3CCS(=O)(=O)C3)C)nn2)CC1 C1(C(=O)NCCC2(C(N(C)CC3CCOCC3)=O)CC2)CCCC1(C)C Cc1csc(C=CC(=O)NCCCCCNC(C2(Cl)CC2c2ccccc2)=O)n1 CC1CCC(C)N1CCC(=O)NC1(CO)CN(C(C2C3CCC2CC3)=O)C1 CC#CCC1C(=O)NC(CC(C)C)C(=O)CC(=O)N1.C(C)(C)(C)O N1(C(=O)NC(c2cncs2)C)CCCCC1c1nccn1C N1(C(C(C)OCC(C)C)=O)CC2(CCCC2NC(c2ccc3c(c2)CCC3)=O)C1 CC1CCOC(C(=O)NCC2(C)CCN(C(c3cncn3C)=O)C2)C1 C(=O)(CCCCC(N)=O)NCC(=O)NCC(C)C1CCC1 Cc1c(C(N2CCSCC2C(N2CC(O)CC2C(C)C)=O)=O)ncn1C c1(CC(N2C(C(CNC(=O)CCF)(C)C)COCC2)=O)ccnc(F)c1F c1(C(N2CCC(N(c3nnc(C)o3)C)CC2)=O)ccc(Cl)c(Cl)c1C c1(C(N(C(CCNC(C2(SC)CCC2)=O)C)C)=O)cc([N+](=O)[O-])c(C)s1 c1(-c2scc(NC(c3cnc(OCCC)nc3)=O)n2)cccc2c(C)ccnc12 c1(CNC(C2C(NC(C(C)OCCC#C)=O)COC2)=O)nc(C)n(C)n1 C(=O)(CC(CC=C)NC(=O)C(=O)C(C)(C)C)NC1(C#C)CCOC1 c1(NC(C)=O)ccccc1CNC(=O)CCC1CC1(F)F C1(C(=O)NC2C=CC(CNC(C3CCCC(=O)O3)=O)C2)COC2(CCC2)C1 C1(CC(=O)NC2CCN(CCNC(=O)COC3CCCC3)CC2)CC2(CCC2)C1 C1(C(N(C(C(C)C)C)CC2CC2)=O)(NC(=O)C(=O)NC(C)C)CC(F)C1 Cc1cn2c(C(=O)Nc3cccc(C(=O)NC4CCCS(=O)(=O)C4)c3)c[nH]c2n1 C1(C(=O)Nc2c(C(=O)NC)nccn2)CC12CCN(C(=O)NC1CCCC1)C2 C(=O)(CCCC(C)NC(=O)CCCN(C)C)NCC(CC)CCO CC12CN(C(C3CSCC(=O)N3)=O)C(C(=O)NCC34CCC(CC3)O4)(C1)C2 N1(C(C(C)n2cnnn2)=O)Cc2ccccc2C(NC(c2ccnnc2O)=O)C1 c1(CC(=O)NC(C2CCCN2C(=O)CC2CCNC(=O)C2)C)cccc(F)c1 c1(CCN(C(C(c2ccccc2)NC(CN(C)CC)=O)=O)CCO)cnn(C)c1 C1(NC(C=CC(C)C)=O)CC(C(=O)NCCCCC2CCCC2)C1 C12(CNC(C3(COC)CC3)=O)CC1CN(C(c1ccccc1Br)=O)C2 N1(C(=O)Cc2ccc(F)c(F)c2)CCC2(CCCC2N2CCCC(F)(F)C2)CC1 C1(C(N2C(C(N(C)OC3CCOCC3)=O)CCC2)=O)CC1C1CCOC1 Cc1cc(C#N)cc(C)c1C(=O)NC1COCCN(C(c2nnn(C)c2C)=O)C1 CC1CN(C(c2cn[nH]c2)=O)CCN1C(=O)CCCc1sccc1-c1ccccc1 C(=O)(C(C(C)C)c1ccccn1)NC(CC(=O)Nc1cn(CC)nc1)C1CC1 c1(C(=O)NC2C(NC(C3C(C)C3C)=O)CC(F)(F)C2)nc(O)nc(O)c1F CC1C=C(C(=O)NC23CC(CNC(=O)CN4CC5(CCC5)C4)(C2)C3)C1 C1(C(=O)NC(CC)CNC(C2(C(N)=O)CC2)=O)(OC)CCS(=O)(=O)C1 O=C1CC(CC(=O)N2CCC(NC(c3ccnn3C3CC3)=O)C2)c2ccccc2N1 N1(C(C2CCCN(CC)C2)=O)CCN(C(c2cnn(C3CC3)c2)=O)C(CF)C1 c12nc(cc(C)n1)N1CC(N3CCCC3)C(C1)N2.c1(C(=O)OCC)coc(C)n1 c1(CCCC)ccc(C(=O)NCC2CC2NC(C2(C3(C)CC3)CC2)=O)cc1 N1(C(c2cccc(C)c2C)=O)CCC2(CCCN2C(C2CC2F)=O)CC1 C(c1ccccc1F)=CC(=O)NCCC(CNC(c1c(CC)ccs1)=O)O C1(n2cc(COC(C)=O)nn2)CC(C(=O)O)N(C(=O)Cc2ccc(Br)s2)C1 c1(C(=O)NCCN(C(C2CCNC2=O)=O)CC)cc2c(Cl)c(OC)ccc2[nH]1 Cc1cc(C(N2CCC(C)(NC(c3cnn(C)c3Br)=O)C2)=O)c(C)o1 N1(C(c2n[nH]c(=N)[nH]2)=O)CCC2(CCCCC2NC(c2cc3cscc3s2)=O)C1 C(C1=CCSC1(C)C)NC(c1n(C(C(=O)OC)C)nnn1)c1c[nH]nc1C1CC1 N1(C(c2c(SC)scc2)=O)CCOCC1CNC(=O)CCc1ccncc1 C#CCC(C)(C(=O)N1CCSC2CCC12)NC(c1nc(=N)cc[nH]1)=O C1(NC(c2cc(CO)[nH]n2)=O)COC2(C1)CN(C(=O)CS(=O)(=O)C1CC1)C2 C1(C(=O)OC)CN(C(=O)C(Cn2cncn2)NC(=O)CCOCC(C)C)CCS1 CC(CC(=O)NCc1cc(C(=O)NCC(F)Cl)no1)n1ccnc1 C(=O)(C(C)S(C)(=O)=O)NC1C(C)N(C(C2CCC3CC23)=O)CC1 c1(C(N(C2CCN(CCOCc3nc(C)no3)C2)CCC)=O)ccc(O)c(C)c1 Cc1nn(C)c(C(=O)NCC2CCCN(CC(=O)NC3CC3CC3CC3)C2)c1Cl c1(OCC)c(C(N2CCC(NC(c3ccc(C)c(O)c3)=O)CC2)=O)cccc1F C(=O)(CCC(=O)N(CC)CC)NCCCCC1CN(C(c2nc(CC)sc2)=O)C1 C(=O)(C1=CCCC(C)(C)C1)NCc1ccc(COC)cc1.C1(=O)CCO1 c1(C(=O)NC2C(OC)CN(C(C3(C)C=CCC3)=O)C2)cccc(N=[N+]=[N-])c1 C1(OC)(OC)CC(C2CCN(Cc3ccc4nn[nH]c4c3)C2)C1 C(=O)(C1=NOC(C)C1C)NC(CC#C)C(=O)NC1CCCC(O)CC1 c1(C(N2CC(NC(c3c(C)cno3)=O)C(F)C2)=O)cc(C)c(C)nc1Cl Cc1cnn(CCC(=O)NC2(CN(C)C(C3CC3c3ccsc3)=O)CC2)c1 c1(CN=[N+]=[N-])nccc(N(C2CCN(C(=O)Cc3cnoc3)C2)C2CCCC2)n1 Nc1c(C(=O)NCC2(CNC(C3CCCC(O)C3)=O)CC2)cccc1Br c1(C(C)C)ccc2occ(C(=O)NCCN(C(=O)C(C)OC3CCCC3)C)c2c1 Cc1cc(NC2C3CCCC23)ncc1C#N c1(OC)ccc(C=CC(N2CC(NC(c3cn(C4CC4)cn3)=O)C(F)C2)=O)o1 N1(C(c2cc(OC)ccc2F)C(=O)NCC)CCCC1C1CCCN1C(=O)OC C(=O)(CCC(C)(F)F)NC(C(N1C(C=C)CC1)=O)Cc1ccco1 C(=O)(C1Cc2c(Cl)cccc21)N(CCCNC(=O)CCc1c(C)noc1C)CC C(C(C)(C)CNC(C1CN(S(CC)(=O)=O)C1)=O)NC(=O)CCOC.C1(OC)CCC1 c1(C(c2nnnn2C)NCC(=O)N(C)CC)n[nH]c(C)c1C C(C)(CCC(C)(C)O)(c1n(CCC)nnn1)NC(COC)CCCC(C)C O=C(CC(C(F)(F)F)NC(C12CCCC1C2(F)F)=O)Nc1cccc(Cl)c1 c1(C(CN(C)C(c2ccc(Cl)o2)=O)CNC(=O)CN2CCOCC2)ccccc1 C1(NC(C2C(C)CN(C(C3CC=CC(O)C3)=O)C2)=O)CCn2ccnc2C1 c1(C(=O)NC(CCN(C(c2oc(CC)c(C)c2)=O)C)(C)C)cc(C#N)ccc1F C=CC1(C(=O)NCCCCS(C)=O)CCN(C(C2CC=CC(O)C2)=O)C1 CC1(C)CCc2[nH]c(C(=O)NCC(O)CNC(c3csc(O)n3)=O)cc2C1 c1(C(=O)NC(C)CCCNC(=O)Cc2cnsc2)cccc([N+](=O)[O-])c1 CC1=C(C(=O)NCC2(NC(=O)C(F)C3CCC3)CC2)C(=O)OC1(C)C C(=O)(C1=C(CC)OCCS1)NCC1(F)CCC(NC(CC(C=C)CC)=O)C1 c1(C(C(=O)NC(CNC(C(C(C)C)(C)C)=O)(C)CO)C)cccc([N+](=O)[O-])c1 C#Cc1ccc(C(=O)NCC2CCCN(C(=O)C3=NOCC3)C2)nc1 c1(NC(N2CC(C)(C(=O)OC)CC2(C)C)=O)ccc2ccc(F)c(F)c2n1 N1(C(c2c(CCC)nns2)=O)CC2CCCC2(NC(c2cnsc2)=O)C1 c1(C(=O)NCC(CNC(C=C(C)C(C)C)=O)O)ccc2c(c1)CC(C)(C)C2 C(=O)(C1=CCC(C)CC1)NC1CCCCC1NC(c1ccc(OC(C)C)cc1)=O CC1CCC(CNC(c2ccc(CNC(=O)CCCC3CC3C)s2)=O)CC1 N1(C(C(=O)NC(CC)(C)C)C)CCOC(NCCCN(C)C(C2CCC2)=O)C1 C#CC1(C(=O)NCCCCS(C)=O)CCN(C(c2ccccc2C)=O)CC1 N1(C(CNC(=O)OC)=O)CCCC(N(CCO)C(c2ncsc2Br)=O)C1 C1(NC(C(C)NC(CC2CC(=C)C2)=O)=O)CCC(=O)NC1C C1(OCCC)CCN(N2CCN(C)C(C(F)F)C2)C1 c1(N2CCC(CCOC)C2)cc(S(=O)(=O)N2CCC(SC)C2)ccc1C#N C1(C2CC2)(NC(N(CC(=O)N(C)C)C)=O)CCNC1 c1(CC2(OC)CC2)cc(Br)c(O)c(Br)c1 C#CC1(NC(C2CC2C(C)NC(=O)C(C)(F)F)=O)CCCOC1 Cc1ncc(S(N)(=O)=O)cc1C(=O)NCC1CN(C(C2(C#N)CCCOC2)=O)C1 N1(CCC=CCC)CCC(C(=O)Nc2cccc(OC3CCC3)c2)C1C(C)C N1(C(Cc2c3ccc(C(C)(C)C)cc3oc2)=O)CCC2(CNC(=O)OC2)C1 N1(C(C(CCCCC)O)=O)CCC2(CCCCN(C(=O)C3=CCCOC3)C2)C1 C1(NC(C(CC)OCC)=O)CCN(C(c2cccc(C)c2F)=O)CCC1(F)F c1(OC)ccc(C)cc1C(=O)NC1(CNC(c2ccoc2C(C)C)=O)CCOC1 C1(O)(C(N(CC(C)CNC(C2CC2c2ccccn2)=O)C)=O)CCC(C)(C)CC1 c1(C(N2CCCC(NC(CC(C)N(C)C)=O)C2C)=O)c[nH]c2cc(C#N)ccc12 C1(C(N(CCCCNC(C(CC)(C)COC)=O)C)=O)CCc2cncn2C1 CCCCC(C)CCC(=O)NCC(O)CCN(C(=O)CCCCc1cnn[nH]1)CC c1(C(C)NC(c2n(CCSC)nnn2)c2occc2C)cccc(F)c1F N1(C(c2nc(C)nn2C)=O)CCC2(CCCN(C(c3c(C)ncn3O)=O)C2)C1 c1(CC(N2CCC(O)(C(C)NC(C=C(CCC)C)=O)C2)=O)nc2ncccn2n1 C1(c2cn(CCC(=O)NC3C(OC)C4(C3)CCC4)nn2)CC2(CCCCO2)C1 C12(C(=O)NC34CC(CNC(C(C(=C)Cl)(C)C)=O)(C3)C4)CC(CO)(C1)OC2(C)C c1(C(N(CCC(C2CC2)NC(C2(CC#C)CCOC2)=O)C)=O)cc(COC)c(C)s1 Cc1[nH]nc(Cl)c1C(=O)NCC(C)NC(C1CCOC(C(C)C)C1)=O Cc1onc2sc(C(=O)NC3CN(C(C4(CO)CCOC4)=O)CC3C)cc12 N1(C(C2CC(C)(CC)C2)=O)CCC(CC(C)NC(=O)CSCc2cscn2)CC1 C(=O)(C(CCC)NC(N)=O)NC(CC=C)CNC(=O)C(c1cncnc1)C C1(CC=C)(NC(=O)Cc2cn(C)cn2)CCCN(C(C2CCCC(=O)N2)=O)C1 CN1CCc2cc(C(N3CCC34CN(C(=O)C(C)(C)CC(F)F)C4)=O)ccc21 n1(CC)ccc(CC(=O)NCC2CCCN2C(c2cnc(CC(C)(C)C)s2)=O)n1 C1(CNC(C(C)N(C(CCN(C)CC)=O)CC)=O)CC2C=CC1O2 N1(C(c2ccc(OC)s2)=O)CCCC(N(C(=O)CCc2nnc(S)n2C)C)CC1 c1(C(=O)NC(CC)CN(C(=O)C(CC(C)C)N(C)C)C)cc2c(s1)CCSC2 O=C1NC(=O)N2CCN(c3nnc(-c4ccc(F)cc4Br)n3CCC#CCO)CC12 C1(NC(C(C)OCC)=O)CCOCC1NC(=O)Cc1cc(C)nn1C C(=O)(CC(=O)NC(CN(C(C1CC(NCC(C)C)C1)=O)C(C)C)=O)OC N1(C(c2cc(C(C)=O)oc2C)=O)CCC2(CCCN2C(C2CCC2(F)F)=O)CC1 c1(CC(N2C(CC(=O)NCC3(C)CC(C)C3)C3CCCC32)=O)cnn2ccccc12 C(=O)(CCCC(C)S(C)(=O)=O)N1CC2CC(CN(C(CS(=O)(=O)NCC)=O)C2)C1 CCC(CCC(=O)NC1(C)CN(C(=O)CC2SC(=N)NC2=O)C1)OC c1(CC)ncc(CNC2CCN(Cc3nnnn3-c3ccccc3)C2)o1 C1(O)(CNC(CCN(CCCCC)C(C)C)=O)CC(NC(C2CC2F)=O)C1 Cc1[nH]cc(C(=O)NC2CC(CNC(=O)C3=COCCC3)CC2O)c(=O)c1Cl C1(CN(C(=O)CCCCO)C)COCCN1C(c1scnc1C(F)(F)F)=O c1(C(=O)NC2CC(C(=O)O)C2)ccc2c(n1)COCC2 CC1CCC(NC(=O)CCC(C)(C)C)CN1C(c1cccc(-n2cccn2)n1)=O O=C(CCS(=O)(=O)c1ccccc1)N1CCC2(CC1)OCc1cnccc12 C=Cn1ncc(C(=O)N(CC(=O)NC(c2cnn(C)c2C)C)C2CC2)c1N N1(C(C2N(C(C34CCC(OC)C3C4)=O)CCOC2)=O)CCc2c(O)noc2C1 Cc1ccc2c(c1)CC(C(N1CCC1CNC(c1cc(F)ccc1O)=O)=O)O2 C(=O)(C1=CCS(=O)(=O)C1)NC(CCN(C(C(COC)NC(C)=O)=O)C)C C1(CC(=O)NC(C)Cn2cnnc2)CN(C(=O)C(C)c2ccsc2)CC12CC2 c1(C(=O)NC(C2CCN(C(c3ccc(S(C)(=O)=O)[nH]3)=O)C2)C)cccc2nccn12 c1(OC)ccc(Cl)c(C)c1C(N1CCC(CNC(=O)C(C)P(C)(C)=O)C(O)C1)=O Cc1ccc(SCC(N2CCOC(CNC(C3(Br)CC3)=O)C2)=O)cc1 Cc1csc2c(N3C4CCC3CC(NC(C3CCC(C)O3)=O)C4)ncnc12 C1(C)(COC)CCCN1C(=O)CCCn1cc(-c2nc(C)c(C)o2)nn1 c1(CC)oc(C)cc1C(=O)NCCOCCN(C(=O)CC(C)(C)O)C CC1(C)C2CC(C(N3CC(NC(c4ccc(C(N)=O)o4)=O)C(O)C3)=O)CC12 C1(CCC)CN(C(=O)C(C)N=[N+]=[N-])CC1NC(c1cc(C(=O)OC)c[nH]1)=O C#CCC(C(=O)NC(C)CC(C)(C)O)N(C)C.C12CCN(C1)C(=O)CO2 C(=O)(C#CC1CC(F)(F)C1)NC1CC(NC(Cc2c(C#C)cccc2)=O)C1 Cc1cn2c(n1)CN(C(=O)C(CC1CCC1)NC(C1CCC(C#N)CC1)=O)CC2 CCCCS(=O)(=O)CC(=O)NC12CCC1CN(C(C1CC=CCC1)=O)C2 N1(C(C2CCCC(OC)C2)=O)CC2(CCN(C(c3ccnc(Cl)c3)=O)CC2)C1 c1(SC(C)C(=O)NCCCN(CCO)C(C2CCCC(=O)N2)=O)ccc(Cl)cc1 c1(C(N2CCC(C)(NC(C3(C(=O)OC)CC3)=O)C2)=O)n[nH]c2ccccc12 CC(C(F)C(=O)NCCC1(C)CCN(C(=O)C(F)(F)C2CCOCC2)C1)C(F)(F)F CN1CCC(C(=O)NC2CCC(CCC(=O)NCCCc3cnn[nH]3)C2)C1 N1(C(CC2CC(C)(C)OC2)=O)CCOC2(C1)CN(C(=O)Cn1ccc(=N)[nH]1)C2 c1(C(C2CC2)NC2CCC(C(=O)NC)CC2)c(C)cc(Cl)cc1C C(=O)(C(CCCOC)NC(=O)C=C1CCC(C)CC1)NC(C#C)CC1CCCC1 N1(C(c2c(CCC)occ2)=O)CC2CCCC(C1)N2C(C1CCCC(C#N)C1)=O C1(CNC(C(CC)F)=O)CC(C)(C)CN1C(=O)CC1CSCCS1 c1cncc(Cl)n1.C1(N(CCC)C=O)CN(C(=O)COCCOCCOC)C1 n1(CC)ncc(C(N2CCC(CNC(C3CCC(NC(N)=O)CC3)=O)C2)=O)c1C N1(C(CCN(C)CC)=O)CC2CC1CN(C(c1csc(C)c1)=O)C2 C(N=c1[nH]cnc2ccc([N+](=O)[O-])cc12)C1(C)CCN(C(C2CC2CF)=O)CC1 c1(NCC(N2C(C)C(NC(=O)CSc3nncs3)CC2)=O)ccccc1C#N C1(F)(CNC(C2CCC(C(F)(F)F)O2)=O)CCN(C(c2cccc(N)c2)=O)CC1 C(=O)(CCCC(F)(F)Br)N1CC(CN(C(CCC(=C)C)=O)C)OCC1 C12(CNC(c3c(Cl)c(C)n(C)n3)=O)CCCC1CN(C(=O)C(C)N1CC(C)C1)C2 N1(C(CC(C)c2ccccc2)=O)CCC(NC(c2c(Cl)cncc2Cl)=O)C(F)C1 C(CC(C)(C)C(=O)N1CC(CNC(C2(CO)CCCC2)=O)CC1(C)C)OC N1(C(CCOC)=O)CCC2(CCCC(CNC(=O)C(O)C3CC3)O2)CC1 N1(C(C(C=C)OC)=O)CCC2(CC2)CC1C(N1CC(C)(C)C12CCC2)=O Cc1ccc(S(N)(=O)=O)c(C(N2CCC3CCN(C(=O)C(C)C4CC4)C3C2)=O)c1 c1(NC)nccc(C(N2CC3(CCC3CNC(C3CC3F)=O)C2)=O)c1F C(=O)(C1CCCc2c[nH]nc21)NC1C2CN(C(C(C(C)C)F)=O)C1C2 c1(C(N(CC(C)NC(=O)Cc2cncs2)C)=O)cccc2c1oc(=O)n2C C(=O)(CCCC(CC)NC(=O)C=C(C)C(C)C)NC(C#C)C1CC1 N1(C(=O)C2=CSCS2)CCN(C(=O)C(O)Cc2ccccc2)C(c2cn[nH]c2)C1 c1(C(C2CC2C(C)C)=O)cccc2c(CC(=O)NCC3(COC)CCC3)coc12 CC1CN(C)CCC1NC(=O)C(C(C)(C)O)NC(C1CCC(CO)CC1)=O CC1CN(C(=O)C(=O)Nc2ccc(CNc3ccc(F)cc3)cc2)CCCO1 Cc1ncncc1C(=O)NC(C)C(c1ccccc1)NC(=O)CN(C)C(N)=O C1(C(=O)NCC(CN(C(c2n(CCOC)ncc2)=O)C)O)CC2CCC(C1)C2O C(=O)(C(C)CCCC(C)C)NC(CCC(=O)NC(CCOCC)C)C c1(C(=O)NC)cncc(C=CC=CC(=O)NC2CN(C(=O)COC3CC=CC3)C2)c1 N1(C(CC=C)=O)CCCC12CCCN(C(c1cncnc1)=O)C2 N1(C(C2C(C)(CC)C2)=O)CCN(Cc2ccccc2N(C)C)CC1 Cc1cc(=NC2CN(C(c3snnc3C)=O)Cc3ccccc32)[nH]c(Cl)n1 N1(C(C2C(COC)(CO)C2)=O)CC2(CCC(NC(=O)CC3(C)CC3)CC2)C1 C(C(O)CC(=O)NCC(c1ccccc1)NC(C1CC1C(F)F)=O)N(C)C c1(C(=O)NCC(C)(C)NC(c2nnc(O)cc2O)=O)[nH]cc2c1CCC2 C(C(C)(C)C(F)(F)CC)NC(c1n(C(CC)C)nnn1)c1scnc1C N1(C(c2cc(C(C)C)[nH]n2)=O)CC(NC(=O)C=CCN2CCCC2)CC1C Cn1ncc(C(N2CCCC2C=CC(=O)NCc2nccs2)=O)c1N c1(SCC(=O)NC23CN(C(C(C)OCC#C)=O)C(C2)C3)ncnc2[nH]cnc12 c1(C(=O)NC2CCCC2NC(C2(CN3CCCC3)CCC2)=O)nccc(CO)n1 C(C)(C)(CCC(=O)NC(C(N1CC2(C1)CN(C(C)C)C2)=O)C(C)C)OC c1(C(=O)NC2(C)CCN(C(c3nccs3)=O)C2)ccccc1[N+](=O)[O-] N1(C(C(CCC)(C)C)=O)CCCCC(NC(C2C3COCC23)=O)CC1 C#CCC(O)C(=O)NCC1CCCN1C(=O)C(c1nc(C)cs1)C C1(NC(c2cccc(C)c2F)=O)CCC2CN(C(=O)CC3CC=CCN3C)CC2C1 C(CCCCCC(C)C)NC(C(CCC)NC(C1CCC2(CCC2)C1)=O)=O N1(C(c2nscc2Br)C(=O)Nc2ccc(OC)cc2C)CCn2c(C)nnc2C1 N1(C(c2cscn2)C)CCC(=O)N(CC2CC3C=CC2C3)C1=O c1(N(c2cccc(Cl)c2Cl)C)nc2c(c(=NCC3CC3)[nH]1)CC(C(C)(C)C)CC2 C1(CNC(=O)OC)CCN(C(=O)CNC(C2(CC)CCNC2=O)=O)CC1C C1(C)(C(=O)NCCN(CCCCCC)C(c2c[nH]nc2O)=O)C2CCC(C2)C1(C)C C1(C(N2CCCC(CCNC(C3(CC)CCCC3)=O)C2)=O)Cc2nccn2C1 Cc1cc(C(N2CCCC(c3nnc(O)o3)C2)=O)c(C)cc1Cl O=C(C1CCCc2nn[nH]c21)N1CCN(C(c2c[nH]ccc2=O)=O)C(C(F)F)C1 c1(C(=O)NCC2(F)CCN(C(=O)CC3CSCCS3)C2)cnn2c1OCC2 C12(C(=O)NC3(CNC(C4C5CC6C(C5)C46)=O)CC3)CCCCC(=O)N1CCC2 c1(CC(=O)NCC(=O)NCC=CCNC(CCC(C)SC)=O)c(C)cccc1C Cc1nc2c(s1)C(N(C)C(C(=O)NC1CCCC1)C1CCC1)CCC2 CC(Cc1ccccc1)C(=O)N1CC(C(N)=O)(CNC(=O)Cc2ncccn2)C1 c1(C(C)NC(C2(CCC=C)CN(C(=O)C(C)NC(C)=O)C2)=O)ccnc(F)c1 C1(CNC(CCOC)=O)CCCN1C(=O)CC1CC1(Cl)Cl C12(C(=O)NCc3ccc(C(C)N(C)C)cc3)CCCC1(C(=O)O)C2 Cc1ccnnc1CNC(=O)CN1CCN(C(C2CC2(C)C(C)C)=O)CC1 C12(NC(C=C(COC)C)=O)CCN(C(=O)C(C)C#N)CCC1C2 c1(C(=O)NC2CC(NC(c3ccc(C)nc3)=O)C23CCC3)ccc2n[nH]cc2c1 C#CCC(CC(F)F)C(=O)N1CC(CC)(NC(=O)C(CC(C)C)C(C)C)C1 C1(C(=O)NCCCCC(C)NC(C2(N(C)C)CCCC2)=O)CCc2ccnn2C1 CC(C)C(C(=O)NCC1CCCN(C(=O)COCC2CCC2)C1)C1CCC1 CCC(C#N)(CC)C(=O)NCC(F)CNC(c1cccc2nn[nH]c12)=O C1(NC(c2nc(CC)oc2)=O)C(CNC(c2ccncc2Cl)=O)CCC12CCC2 C1(C(=O)NC(c2cccc(Br)c2)COC)CC(c2cn(C)nc2C)=NO1 N1(C(C(C(C)C)OCC)=O)CC2CC(C1)C2NC(c1cncc(F)c1C)=O C(N=c1[nH]c(C)nc(C)c1C)C1C(CNC(C=Cc2cc(OC)ns2)=O)CCC1 C(N=c1nc2sccc2c(N(C)Cc2c(F)cccc2Cl)[nH]1)c1nc(CC)sc1 n1(CC(=O)NC(C(=O)NC(C#C)CCC)CO)c(C)ccc1C c1(OC)cc(C)nc(N2CCCC(C(C)NC(=O)CCC(C)(F)F)C2)n1 C1(NC(c2cnc3n2CCC3)=O)CN(C(c2ccn(C(F)F)n2)=O)CC12CCC2 C(CNC(=O)C(N1CCCCC1=O)C)(C(C)(C)C)NC(c1c(C)[nH]cc1)=O c1(NC(C(=O)NCCc2nsc(SC)n2)=O)ccc(OCC(F)(F)F)nc1 c1(C(N2CCC3(CCN(C(CC4(C)CC4)=O)C3)C2)=O)c[nH]c2cc(C#N)ccc12 c1(C(=O)NC(CC)CNC(=O)CSCC(N)=O)cccc2nncn12 Cc1cccc(C)c1C(O)C(=O)NCCOC1CN(C(C2CC2(C)C)=O)C1 CC1CN(C(c2cc(Cl)cnc2O)=O)CCC1CNC(=O)CSc1ccncc1 N1(C(CC2C(CNC(CCOCC(C)C)=O)C2)=O)CC(C)C(F)(F)C1 c1(CC)nc(Cl)c(C)c(=NC2CC(CNC(c3cc4n(n3)CCCC4)=O)C2N)[nH]1 C(=O)(C(C)(C(C)C)OC)NCCN(C(CC(CC)C1CC1)=O)C(C)C C1(NC(C2CCNC(=O)C2)=O)CC(CO)N(C(=O)C=CCN2CCC2)C1 Cc1nccc(CCC(=O)NC2(C)CCN(C(C3(c4cc[nH]n4)CCC3)=O)C2)n1 Cc1csc(C(=O)NC2CCC2C(=O)NCCC2=CCCC2)c1C c1(NC(CC2CCCN(C(c3c(C)nc(F)cc3)=O)C2)=O)cc(F)c(F)c(Cl)c1 N1(C(c2ccccc2F)=O)CC2CC2(CNC(C2(Cn3cncn3)CC2)=O)C1 c1(C(N2C(CNC(C3CCC(C)(CC)O3)=O)CC(F)C2)=O)ccsc1S(C)(=O)=O c1(OC)ccc(CCC(=O)N(CC(C)NC(=O)CC2CC=CCC2)C)cn1 C1(NC(C2(C(=O)OC)COC2)=O)C2CN(C(C3CCCN3C)=O)CC12 C1(C(N(CCCNC(c2ccc(N(C)C)nn2)=O)CC)=O)CC2CCC1CC2 Cc1nc[nH]c1CC(=O)NC1(C2CCCN2C(=O)CSC2CCOC2)CC1 c1(C(=O)NCC2CN(C(CCC#C)=O)CC2C(F)(F)F)ccc(Cl)c(S(C)(=O)=O)c1 N1(C(c2nnn(C)n2)=O)CCN(C(c2ccc([N+](=O)[O-])[nH]2)=O)C2CC12 N1(NC(C2CCN(C(=O)C3C(CC)C3(C)C)O2)=O)CC(C)=CC(C)C1 CC1C2CCC(C2)C1C(=O)N(CC(C)C(=O)NC1CC1)C C1(OC)CN(C(c2cnc(S)nc2)=O)CC1C(=O)NCC=Cc1ccccc1 C1(C(N(CC(CC)C)C)=O)CN(C(C2CCOCC2)C)CC1C CC1OC2(CNC(C3C=CC=CC=C3)=O)CC1(C(N1CC(C)(N(C)C)C1)=O)C2 N1(C(C(CN(C)C)(F)F)=O)CCC2(CCCC2NC(=O)C=CC2CCC2)CC1 Cc1nc(C(=O)NC2CN(C(C3CCC(NC(=O)OC(C)C)C3)=O)C2)[nH]c1C C1(C2CC2)(C(N(C2CCCNC2=O)C)=O)CN(C(=O)CCCn2cccn2)C1 N1(C(C=CC(=O)OCC)(C)C)CCC(C(N2CCCC2C(O)C(F)(F)F)=O)CC1 CC(C)(C#N)CC(=O)N1CCC(O)(CCNC(=O)COCC2CCCO2)C1 c1(SC)cc(F)ccc1C(=O)NCC12CC(CN1C(=O)C(c1ccccc1)F)C2 C(C(F)(C(=O)N(C)CCC1CCOCC1)C(C)C)NC(C1CC(C)=C(C)CC1)=O Cc1[nH]ccc1C(N1C(C(N2CC(OCC(N)=O)C2)=O)CC1C)=O C(=O)(CCCC(C)C)N1CCC(OC)(CNC(=O)CCCc2ccsc2)C1 Cc1cc(C(=O)N(C2CCCN(C(=O)CSC(C)C)CC2)C)n2ncnc2n1 c1(Nc2ccc(C(N3C(C)CCC3C(=O)O)=O)cc2)cnn2cccc2c1 c1(C(=O)NCCCC(c2ccccc2)NC(=O)C(F)=C2CCC2)c(F)cccc1Cl c1(CN2CCOCC(C(=O)NCC(=O)N3CCCC3)C2)csc2ccc(F)cc12 O=C(C1Cc2ccc(Cl)cc21)N1CCC(O)C(F)(F)C1 CC1C(Nc2ncccn2)CCCN1C(=O)CC1(C)CC1.C(=O)(CCN1CCCC1)N c1(C(C)(O)Cn2cc(CN(O)C(=O)c3ccoc3)nn2)ccccc1 n1(CC)cc(NC(=O)CC2CCN(C(C3CC(C)OC3=O)=O)CC2)c(C#N)n1 C(=O)(C1=CCCCO1)N1CC(OCCNC(CC(C)N2CCCC2=O)=O)C1 c1(OCC)cc(C(N2CC(CN(C)Cc3c(C)cccc3O)C2)=O)cc(Cl)c1 c1(OC)cnn2cc(C)cnc12.N1CC2CCN(C(=O)C(=O)OC)C2C1.C1(C)CN1C c1(OCC(=O)NC(CNC(CCCOC)=O)(C)CO)ccc(C)cc1OC CON(CCC(=O)N1CCC(n2cccn2)C1)C(=O)CSc1ccccc1 c1(CCC(=O)NCc2cc(CO)ccc2Cl)ccc2c(c1)CCCC2 CC(C(C)C(=O)N1CC(NC(c2ccnnc2O)=O)CCC(O)C1)S(C)(=O)=O C1(C(N2CC(OCC(N)=O)C2)=O)CCCN(C(C2CCC(=O)O2)=O)C1 c1(CNC(c2cccnc2)C(=O)OCC)ccc(I)c(C(F)(F)F)c1 c1(C(=O)NCC(C2CC2)NC(C(C)SC)=O)ccc2cccc(O)c2c1 N1(C(c2cncc(CC)c2)=O)CC2CN(C(C3(CO)CCCC3)=O)CC2(C)C1 Cc1cc(C(O)C(C)NC(=O)NCC2(C#N)CCCC2)ccc1F c1(OCC)ccc(C(=O)NC2CC(CNC(=O)C3=CCC3)C(O)C2)cn1 c1(C(=O)N)n[nH]cc1[N+](=O)[O-].C1(F)(COC)CCN(C(C2C3CC4C(C3)C24)=O)C1 CCC(CO)(C(=O)N1CCC(CC(N2CCC(O)(OCC)C2)=O)C1)OC c1(C(=O)NC(CNC(CCC=CC(C)C)=O)CO)cc2n(n1)CCNS2(=O)=O c1(C(=O)NCC(CCCC)NC(C2CN(C(C)C)C2)=O)cc(C)ccc1[N+](=O)[O-] N1(Cc2cccc(OCC)c2)CCC2C1CCCN2C(=O)Nc1cnccc1Cl c1(OC)ccc2[nH]c(C(N3CC(C)(C(N4CC(O)CC4(C)C)=O)C3)=O)cc2c1 N1(C(CCC=CC(C)C)=O)CCC2(CC1)CC(CNC(c1c[nH]ccc1=O)=O)C2 n1(CC=C)c(N2CCN(CC(F)F)CC2)nnc1C12CC(CC3CC3)(CO1)C2 CC1CN(C(c2cccnc2N)=O)CCN1C(=O)CCc1ccc(Cl)s1 S(=O)(=O)(c1cccnc1)NC1CCC(C)C(NC(=O)OCc2ccccc2)C1 c1(N(C2C(C)COC2)C)cccc(C#N)c1F N1(C(C(=O)NCCCCC2C(C)C2)=O)CCc2c(C)cc(C)cc2C1 CC1COC(C(=O)NCCn2cc(CNC(=O)CCc3cccs3)nn2)C1 C1(CCNC(CCN(C)C)=O)CCCCN1C(c1cn(CCO)nn1)=O C1(C(=O)OC)C(C)CCN1C(=O)C(c1cccnc1)NC(C1CC(F)C(=O)N1)=O c1(C(=O)N(CCSc2cncs2)CC2CCCO2)ccc2cccnc2c1 c1(C(=O)NCC(C)NC(C2CC2C)=O)ccc(Cl)nc1N(C)C C1(CCNC(CN(C2CC(C#N)C2)C(C(C)SCC)=O)=O)COC(C)(C)C1 CC1(C)COC(C(=O)NCCCCNC(C2CC2c2ccccc2)=O)CO1 C1(CNC(C2C(=C)CC2)=O)CC2(CC2)CN1C(=O)C=Cc1ncc[nH]1 N1(C(C(C)(C)C)=O)CCC(F)(F)C(CNC(C2CCCN2CC(F)(F)F)=O)C1 C1(NC(Cc2c(C)noc2)=O)CCS(=O)(=O)C12CN(C(=O)C(C1CCC(=O)N1)C)C2 Cc1nc(N2CC(C)(OCC3CC3)C2)c2cc[nH]c2n1.C1(=O)CCC2CC(C2)N1 c1(C(C(=O)N(CC(C)O)CC(c2ccccc2)O)N)ccc(OC(F)(F)F)cc1 N1(C(=O)Cc2cscn2)CCN(C(=O)CC2CC3(CC3)CO2)C2CCCC12 C1(CNC(c2ccc3n[nH]cc3n2)=O)CC2COCC2N1C(c1ccc(Cl)[nH]1)=O N1(C(C)=O)CCC(CCC(=O)N(CCCO)CCCO)C1.C(CCO)S N1(C(C(C)(C)SC)=O)CCC(C)C(NC(c2ccc(C(F)F)cc2Cl)=O)C1 C1(C)(CNC(C2(C(C)=O)CCC2)=O)CCCN1C(c1cn(CC(N)=O)nn1)=O C1(NC(c2c(C)scn2)=O)CC2CCC(C1)N2C(=O)CCN1CCC(N(C)C)CC1 c1(OC)ccc(C)cc1C(C)NCC1(CO)CC(C)C1 C1(C(C)(C)C)CC=CCC1CNC(=O)Nc1cccc(Cn2ccnn2)c1 n1(CC=C)nnnc1C(c1cnc(C(C)C)o1)NC1(C)CC(O)C1 N1(Cc2c(N)ccc([N+](=O)[O-])c2)CCC2(CCCNC2=O)CC1 N1(C(C(CC)NC(N)=O)=O)CCN(C(C2COCCOC2)=O)C(C2CC2)C1 c1(OC)ccc(C(N2CCCC2(C)C(=O)NC(c2ccno2)C)=O)c(O)c1 c1(SC)cccc(N(C(CO)C(N)=O)C(c2ccncc2-c2cnn(C)c2)=O)c1 c1(C(N2CCC3CCC23CO)=O)ccn2c(C(F)(F)F)nnc2c1 C1(C(=O)NC(CSC)(C)CO)CC2C=CC1N(C(c1ccc(C)cc1F)=O)C2 c1(C(N2CCCC(CNC(CC(C)C3CC3)=O)C2)=O)coc2c1C(=O)NCCC2 N1(C(C2C(C)(COC)C2)=O)CCCCC12CN(C(=O)Cc1cccc(C)c1C)C2 Cc1ccc([N+](=O)[O-])cc1C(=O)N1C2C3CC4C(=O)C4C2N=C3NC1CC1CNCC1 C(=O)(C(=O)C(C)(C)C)NC(C)CCC(=O)N1CCOCC1CCO c1(C(=O)NC(C)COC(F)F)ccccc1-c1nc[nH]n1 N1(C(c2c(N)cc(Cl)nc2)=O)CC2(CCC2)CC1CNC(=O)CCn1cncn1 N1(C(=O)OC(C)(C)C)CCCc2cccc(NCC(C)(C)C(C)(F)F)c21 N1(C(C2C(C)CCC2)=O)CCCC1(C)CNC(C1CCC(=O)N1C)=O c1(CN(C2(c3ccccc3)C(CCC)C2)CC)c(Cl)cc(Br)cc1Br C(=O)(CC(F)(F)C(F)F)N1CCC(C(=O)NC(c2c(C)cccc2)C)C1 C1(C(=O)NCCC(C)NC(=O)CNc2ncccn2)SCCCS1 c1(C(=O)NCCN(C(=O)CCF)CCC)cc(Cl)c(OC)cc1Cl c1(CCC)cc(C(=O)NC2CN(C(=O)C(CC)SC)CC2F)ccc1Cl Cc1cccc2nc(N3CCOCC(NC(=O)C(C)(F)C(C)(C)F)C3)sc12 C#Cc1ccc(C(N2CCC(CN(C(=O)CC(C)C(F)F)C)C2)=O)cc1C C1(C(=O)NCCC(=O)NCC)CC=CCN1C(c1csc(C)c1C)=O N1(C(Cc2c(C)nsc2)=O)CC(CNC(C2CCCN(C)C2=O)=O)CC1(C)C C1(C(=O)NCC(CC)NC(=O)Cn2cc(Br)nn2)OCCC1C C1(NC(c2c(C)oc(SC(F)(F)F)c2)=O)CCN(C(C2CC(F)(F)C2)=O)C12CC2 C1(C2CC2)(NC(C2C(CC)CCC2)=O)CCN(C(c2cccc(C(C)C)c2)=O)C1 n1(CC(=O)OCC)cc(C(=O)NC2COCC2NCC2CCC2)nn1 C1(CC(=O)NC23CC(NC(c4cscc4F)=O)(C2)C3)CCCC1(F)F c1(C(=O)NCC=C(Cl)Cl)cnnc(O)c1.C1C(O)C(=O)N1 C1(C(N2CCC(OC(C)C)C2)=O)CC12CCC(F)(F)CC2 C(=O)(C1CC(=O)Nc2ccccc21)NCCN(C1CCCC1)C(C1N(CC)CC1)=O N1(C(CC2(C=C)CC2)=O)CCN(C(=O)CC2CC2c2ccc(F)cc2F)C2CC12 c1(CC)ncccc1C(=O)N(C1CCN(C(=O)CC2CCCC(O)C2)CC1)C Cn1ccc2cccc(C(N3CCCCCC3CNC(C3CCS3(=O)=O)=O)=O)c12 C(=O)(C(CC1CC1)NC(=O)C(C)N(C(=O)Cc1cncnc1)C)NC CCC(C)CC(C(=O)Nc1cc(C)cc(C)c1C)NC(=O)Cc1cncs1 C(=O)(C(C)(C)n1cc(Cl)cn1)NCCN(C(C1C(C(=O)OC)C1)=O)CC1CC1 c1(NC(C2CN(C(CCc3c(OC)cccc3)=O)C2)=O)cc(Br)ncc1[N+](=O)[O-] C(=O)(C1CCCCc2ccccc21)N1CC(NC(c2c(C)cc(C)c(F)c2)=O)C1 C1(C(N2CCCC2C)=O)(C(=O)N)SCCCS1.C(=O)(CSC)NC(CSC)C1CC1 c1(C(=O)NCC2(COC)CCCN2C(=O)C(C)CC2CC2)cc2cccn2cn1 C1(CC(C)NC(c2ccc(=O)n(C)n2)=O)CC2CCC(C1)N2C(C1(SC)CC1)=O c1(OC)c(Cl)cc(Cl)c(OC)c1C(N1CCN(C(C2(Br)CC2)=O)CC1C)=O S(=O)(=O)(c1ccc(Cl)s1)N1C(C(N2CCCC3(COC3)C2)=O)CCCC1 CCC(C)(C)C(=O)C(=O)N1CCC(CC(C)NC(c2ccn(C)n2)=O)CC1 C(=O)(C(C)(C)CC(C)C)NCCC1OCCN(C(C2N(C(C)=O)CC(O)C2)=O)C1 c1(CCC(C)NC(C2CN(CC(F)(F)F)C2)=O)ccc(F)c(Br)c1 Cc1cc(=NCCCCNC(C2CCC(CN)O2)=O)[nH]cc1C#N CC1COc2c(C(=O)NC(CNC(c3cc(Cl)n(C)n3)=O)C(C)(C)C)cccc21 C=CC(C)(O)CC(=O)NC(C(=O)Nc1cc(OC)ccc1F)C(C)(C)C c1(-c2nc(N3CCC(SCC)CC3)nn2CC2CC2(C)C)cccc2cnsc12 n1(CC)c2ccccc2c2cc(C(N3CCC(NC(c4ccco4)=O)C3)=O)ccc12 c1(C(CC)(C)C)ccc(C(N2CCC(NC(c3cc(NC)ccn3)=O)C2)=O)cc1 C1(C(=O)NCCN(CCOCCO)C(C2CCC2(F)F)=O)COc2ccccc2C1 N1(C(C(c2cccs2)SC)=O)CC(C)N(C(=O)CCc2cc(Cl)cc(Cl)c2)CC1C c1(C(=O)NC2(CC=CC(=O)NC(C)CN3CCCC3)CCC2)cccc[n+]1[O-] c1(CNC(C(C2CCC2)NC(C=CCC)=O)=O)c(F)cccc1F CC(CC(F)(F)F)N(C(=O)C(C1CCN(C(C2(C)CCCC2O)=O)CC1)C)C c1(C(N(CC(=O)NC(CCC)CO)C(C)C)=O)nnc(S)n1C n1(CC)ncc(C(N2CCC(N3CCN(C(=O)CP(C)(C)=O)C3)CC2)=O)c1Cl CCCC(C(=O)Nc1ncnc(SCCC(F)(F)C(C)C)n1)C(C)C N(C1CN(C(=O)C(C)CC(F)(F)F)CCc2ccccc21)C(CS(CC)=O)=O c1(C(C)OC(C2CCCCC2)C(=O)NCCCNC(=O)C(C)C#N)ccc(F)cc1 c1(C(=O)NC2(CNC(c3cn(CCOC)nc3)=O)CCCC2)nc(C)ncc1Cl Cc1[nH]nc2c1CC(C(N1CCN(C(c3cnoc3C(C)C)=O)CC1C)=O)CC2 N1(C(C(F)OC)=O)CCCC2(NC(=O)CCN(S(C)(=O)=O)C)CCCC12 Cc1ccccc1C(N1CCOC(c2cn(C)cn2)C1)C(=O)NCCCF C1(NC(C(CC=C)C)=O)CCN(C(c2ccc(C(=O)OC)c(Cl)c2)=O)CC1(C)C CC1CCOCC1C(=O)NCCCCCN(C(=O)C(N)=O)C CCCC(C(=O)N(C1CCC1)CCN(C)C)NC(c1ccsc1C#N)=O N1(C(C2CC(C(C)=O)C2)=O)C(C(=O)NCC(C)CO)CC1C c1(C(c2n(CCCSC)nnn2)NCc2coc(C)n2)ccc(=O)n(C)c1 N1(C(C2C(C)CC(=O)N2)=O)CCC(NC(c2ccc3c(c2)CC3)=O)C(C)(C)C1 N1(C(C(C)C(C)(C)C)=O)CCCc2ccccc21.N12C(=O)CN(C1=O)CC2 Cc1nc(C(=O)NC2CN(C(=O)C(C)N(C)C(c3ccccc3)=O)C2)n(C)n1 C12(C(=O)NC(c3noc(C)n3)CC)CC(C)(CN1C(=O)CN1CCC(=O)CC1)C2 n1(C(C)C(=O)N(CCCNC2(C(=O)N(C)C)CCSC2)CCO)ccc(C2CC2)n1 c1(NC(=O)Nc2cnc(Br)nc2)[nH]cnc2nc(I)cc1-2 C(=O)(CCCCC(=O)N(C1CCC(NC(=O)CC2C=CCC2)CC1)C)NC c1(CC)nccn1C(C)CC(=O)N1CCC(n2cc(C(N3CCCC3)C)nn2)C1 C1(CNC(c2n(C)ccc2)=O)CN(C(C2CCCN2C2CCCC2)=O)CC1(F)F C1(CNC(c2cn(CC(=O)NC)nn2)=O)CCCCCN1C(C1CCC2CC12)=O CCCC(C)CC(=O)NC(=O)C(CC)NCCC(CN(CC)CC)=C C1(OC)CC2CCC1CC2C(=O)NCC1(O)CN(C(=O)CC(C)(C)OC)C1 N1(C(C2CCC(OC)C2)=O)CC(=O)NCC1C(=O)NCC1(CCO)CC1 c1(C(=O)NC2CC(F)(CNC(CC(OCC)OCC)=O)C2)cnc(SC)cc1C c1(OCC)cccc(C(=O)NC(CNC(c2cc(OC)ncn2)=O)C2CC2)c1C C1(C(N2CCC2CC(C)(C)C)=O)(COC)CN(C(=O)CCc2cnn[nH]2)C1 C=CCC(C(=O)NCC(CO)C1CCC1)NC(=O)C1=CCCC1 N1(CC)Cc2ccc(NC(=O)CS(=O)Cc3ccnc(C(F)(F)F)c3)cc2C1 CC1C(C(N2CC(n3ccnc3)C2)=O)CCCN1C(C1CC1C(N)=O)=O c1(C(=O)NCC2C(C)CN(C(c3ccco3)=O)C2)ccc(=O)n(CC(F)(F)F)c1 c1(N(C(=O)NC(C)CS(C)=O)C)ccnc(O)c1 C1(C(N2C(CNC(Cc3cccc(OCC)c3)=O)C=CC2)=O)CCC2(CCC2)O1 C1(NC(=O)CCCC2CCC2)CC(F)CN(C(c2cn(C3CC3)nn2)=O)C1 c1(C(N(CCNC(C(C2CC2)OC)=O)C)=O)nnn(-c2ccccc2)n1 C12(CNC(CN(C)C3CC3)=O)CC(CN1C(c1cc[nH]c1C1CCC1)=O)C2 CN1CC=C(CC(=O)N2CC(NC(C3CS(=O)C3)=O)C(C)(C)C2)CC1 C(=O)(C(C#N)C(C)(C)C)N(CCNC(C1CCCC12CC2)=O)CC c1(C(C(=O)NCCOC)N(CCF)C2CC2)cccc(OC(F)(F)F)c1 C1(NC(C(C(C)C)NC(C)=O)=O)CC(C)CN(C(C2(CN(C)C)CCCC2)=O)C1 N1(C(C(CC)C)=O)CCC(NCC#N)c2cc(F)ccc21 C1(C(=O)OC(c2cc(F)cc([N+](=O)[O-])c2)CC)CCc2nc(C)nn2C1 C(CNC(C1(C)CCC1)=O)(CC(=O)NC(c1cnc(C)s1)C)OC C1(C(N2CCC(CCOC)C2)=O)N(C(C2C=C(C)CS2)=O)CCCC1(C)C C(=O)(C(O)C(C(C)C)OC)NCC1CC(O)(CNC(CCC(C)OCC)=O)C1 N1(C(C(CC)OCC)=O)CCN(C(C2CC=CCC2)=O)C(C)C1 c1(NC(=O)CSc2cccc(Cl)c2)[nH]c(=NC2CCSC2)nc2scnc12 C1(CNC(c2cc(C(C)C)[nH]n2)=O)CN(C(=O)CN2C(C)CCC2C)CC1(C)C C1(CCNC(c2cccc(CC)n2)=O)CN(C(C2CC2F)=O)CCS1(=O)=O C(=O)(C1CC(=O)Nc2cc(F)ccc21)N(CCCNC(=O)CCCF)CC C(c1ccc(Cl)cc1F)=CC(=O)NC1(CCNC(C(CC)(C)CC)=O)CCC1 N1(C(C(C)OCC=C)=O)CC2CS(=O)(=O)CC2(CNC(c2nnn(C)n2)=O)C1 c1(C(C)CNC(=O)C(=O)N2CC(n3ccnc3)C2)ccccc1 c1(C(=O)NC2C3CN(C(C4(C(C)(C)OC)CC4)=O)C2C3)ncc(N)cc1C Cc1nc(C2(NC(=O)CC3CC3)CC2)no1.C1(=O)CCNCCCN1 C1(CN(C(=O)Cn2ccnc2C)CC)CCCCN1C(=O)Cn1cnnc1O CC(C)CC(C(=O)NCC1CSC1)NC(=O)C(F)CC1CCOC1 c1(CC)ccc(C)c(C(=O)NC(C)(C)CCNC(=O)CC2(SC)CCOCC2)c1 C1(C)(NC(c2scc(C)c2)=O)CCN(C(C2CCCC2C(C)C)=O)CC1 C(=O)(C(C)Cc1ccco1)N(CCC(=O)NCC1CC(C)C1)C C#Cc1cncc(C(N2C3CCC2C(CNC(=O)CC2(C)CCC2)C3)=O)c1 C=CC1CN(C(c2csc(C(=O)OC)n2)=O)CC1NC(C1(C)COCCO1)=O c1(OC)cc2ccc1-2.c12cccc(n1)NC(=O)N1CC2C1.OC.SC c1(C(=O)NC2C(NC(CCC=C=C)=O)CCOC2)cccn(C(C)(C)C)c1=O C(C(F)(C(=O)OCc1cc(C)cc(F)c1)C(C)C)NC(C(SC)SC)=O CCC(CC)OCC(=O)NCC(C)CNC(C1CC(OC(F)F)C1)=O C1(C(N(CCC)CC2CCCC2)=O)(C(C)C)CCCN1C(=O)Cc1cc[nH]c1 N1(C(C2(c3cc(C)on3)CC2)=O)CC2CN(C(=O)CC(C)C(F)(F)F)CC(C1)O2 C12(CNC(C3(OC)CCC3)=O)CC(CO1)N(C(C1CCCO1)=O)C2 C1(NC(C2C(CCOC)C2)=O)CCC(NC(c2cnoc2C)=O)C1 N1(C(CCOC)=O)CCC2(CC2C(=O)NCCc2ccn(C(C)C)n2)C1 N1(C(C2(C)CCC2)=O)C2CCC1(CNC(=O)C=Cc1ccoc1)CC2 c1(C(=O)NCC#CCNC(c2cnc(C(C)(C)C)s2)=O)cscc1C#N c1(C(N(C2C(C)CN(C(C3(C#N)CC=CC3)=O)CC2)C)=O)ccn2c1CCCC2 Cc1cccc(C(N2CCCC2CN(C)C(C2CC3CC2CO3)=O)=O)c1C Cc1cc(CO)c(-c2ncc(Cl)cc2C(=O)Nc2cccc(C)c2I)cc1C C(=O)(C1=COCCC1)N1CCCC(N(C(CCC=C(C)C)=O)C)C1 c1(C(=O)NCC(C)NCC)ccc(OC)cc1.C(=O)(CCN(C)CCO)C(=O)CS C(=O)(C1=CCN(C(=O)CCCCC#N)C1)N(C(C)CS(C)=O)C C=C(C)CCC(=O)N1CC(F)CC1CNC(C1CC(O)CN1C(C)=O)=O c1(C(=O)NC2CC(CNC(C(CC)SC)=O)C(O)C2)c(C)cc(C#N)cc1C C1(CCC(C)C)C(=O)N1.N1(CCOCCOCCOC)CCCC1.C1CS1 c1(C(=O)NC(CCCNC(CCC(=O)NCC)=O)C)ccc(C#N)c(OCC)c1 Cc1c(C(=O)NCC(O)CCNC(C2(F)CC2)=O)nnn1-c1ccccn1 C1(NC(COC(C)C)=O)CC2CC1N(C(=O)Cc1cccnc1)C2 c1(CC(=O)NC2CN(c3nnc(C)s3)CC2(C)C)ccc2cnccc2c1 C1(NC(C(CO)N(C)C)=O)CC2CCCC(C1)N2C(c1ccc(F)cc1F)=O C(=O)(C1CCC(=O)c2ccccc21)N1CCC(N(C(=O)CC(C)C2CC2)CC)CC1 O=C(CC1=CCCCC1)NCC1C2CCC(C2)N1C(=O)COCC1CCCCC1 c1(OC)ccc(C)cc1C(=O)NCCC(C)NC(=O)CCC1CCCCO1 c1(C(=O)NC2CCN(C(C(CC=C)(C)C)=O)CC2C)ccc2c(c1)NCC2 c1(C(N2CC(CCNC(C(COC)O)=O)C(C)C2)=O)nc(C)n(C)c1C C(=O)(C(C)(C)F)N(C1CN(C(C(C)N(CC#C)C(=O)NC(C)(C)C)=O)C1)C c1(NC(N2CCCN(CCN(C)C)CC2)=O)ccc2c(Br)cccc2n1 c1(CC(=O)NC2CCN(c3c(C#N)nccn3)C2)ccc2c(c1)CCCS2 Cc1cncc(CC(=O)NCCN(C(=O)C(C)n2ccnc2)C2CC2)c1 C1(N(C(c2nccc(CC)c2)=O)C)CN(C(=O)CCc2ccc(C)s2)CC1(C)C C1(C(=O)NC(CC)(C)CN(C)C(C)=O)CC2(CC(NC(=O)C(C)SC)C2)C1 CC1CN(C(C2CCS(=O)(=O)C2)=O)C(C)CN1C(c1csc(S)n1)=O N(C(=NCCCCl)NCCNCCC1CNC1)CC(=O)OCC Cc1cc(C(N)=O)cc(C(=O)NC2CC(NC(c3ccc([N+](=O)[O-])[nH]3)=O)C2)c1 c1(C(=O)NCC2CC3(CC(NC(CCOC)=O)C3)C2)nc2ncccn2n1 C(=O)(CC(C)C(=O)Nc1cn(C2CCOCC2)nn1)N(CCCN(C)C)CC CN1CCCCc2ccc(NC(=O)Nc3ccn(-c4ccccc4Cl)n3)cc21 C=CCCC(CO)NC(CCCC=C)c1nnnn1C.C12(CCCC1)C(=O)N2 C=Cc1cc(C(=O)Nc2ccc(NC(c3cncnc3)=O)c(F)c2)cc(F)c1 CC1CN(C(=O)Nc2c(N(C)C(C3CC34CCC4)=O)n(C)cn2)CC(C)S1 C1(CNC(CC(=O)NCC#C)=O)CN(c2nc3ccccc3s2)CC(C)(C)O1 c1(CC)cc(OC)cc(OC)c1C(=O)NC(CNC(c1c[nH]nc1OC)=O)CC CC1C(NC(=O)CSc2cnn(C)c2)CCN1C(C1CC2CC2C1)=O Cc1nc(C(=O)NCC(CNC(=O)CC2CCOCC2)S(C)(=O)=O)cn(C)c1=O N1(C(c2cnn(C3CCOC3)n2)=O)CC2(CCN2C(c2cccs2)=O)C1 C=CCCC(C(=O)NCC1(CC2CC2)CC1)NC(=O)CC1CN2CCC1CC2 C1(CC(N2C(CNC(=O)Cc3c[nH]nc3O)CC2)=O)CC2(C1)C(F)(F)C21CCC1 Cc1nc(NC(c2cccc(-c3cnn(CCO)c3)c2F)=O)cnc1C#N c1(CC)c(C(=O)NC(C)(C)CCCNC(c2ncsc2C2CC2)=O)ccn1C C=CC1(C(=O)NC2CC2NC(c2cc(CC)ccn2)=O)CCCCC1 CCCCC(CNC(=O)CCCF)NC(C1(c2ccccc2)CC1(Cl)Cl)=O c1(C(N2CC=CC2CNC(C2CC(O)C2)=O)=O)cc(Br)c2nccn2c1 C1(NC(c2n(C)ncc2)=O)CC2(C1)CC(CNCC1CCCCN1CC(F)F)C2 CC1C(C)C(=O)NCCC(=O)N1.c1(NC(=O)C(C)(C)C)cccc(O)n1 C1(CC=C)(NC(=O)C(c2cccc(F)c2)C)CCN(C(=O)C=CCF)C1 CCC(O)C(F)(F)C(=O)NCc1occc1C(N1CCSC(C)C1)=O Cc1coc(C)c1C=CC(=O)NCC1CC1NC(C1(CO)CCC1)=O N1(C(CNC(=O)OCC)=O)CCC(C(=O)NCc2nn(C)c(=O)o2)C(C)(C)C1 N1(C(C(F)=CCC)=O)CC2(C1)SCCC2NC(=O)Cn1ccc(-c2ccccc2)n1 CCC(CC)C(C)C(=O)NCCCN(C)C(C1(OCC2CCC2)CCC(C)(C)C1)=O N1(C(c2n(CC)nnc2)=O)CC2(C1)CN(C(c1cc(-c3csc(C)n3)c[nH]1)=O)C2 CCC(CC)CC(=O)N(CCNC(C1CC(C)(C)CN1C)=O)CC C1(CC)CN(C(=O)CC2CCC(F)(F)CC2)CCC1NC(=O)CN1CC(C)C1 c1(-c2c(C)cc(C(=O)NC(C)C#N)nc2)ccc([N+](=O)[O-])cc1 N1(C(CCC(C)OCC)=O)CCN(C(=O)C(C)(F)F)CC1C1CC1 C#CC1(O)CCN(C(=O)C=CC2CCN(C(C3CCN(C)C3C)=O)CC2)CC1 C(=O)(NNC(=O)Cn1ncc(Cl)c1C)C1CC(=C)C1.OC c1(C(=O)NC(CN(C(C(C)NC(C2CCC2)=O)=O)C)(C)C)cc(Cl)c(N)c(Cl)c1 N1(C(C2C(C)=C2)=O)CCC2(CCCN(C(c3cc4cccnc4cc3N)=O)C2)C1 N1(CCCCC)CC2(CC(C(=O)NCC(c3ccc(Cl)cc3)O)CO2)C1 c1(C(=O)NCCC2CSCCN2C(c2cccc(F)c2O)=O)cc2n(n1)CC(F)C2 N1(C(COCc2cccc(OC)c2)=O)CC2(CCCC2NC(=O)CP(C)(C)=O)C1 c1(CN2C(CCC)(CO)CCC2)ccc2c(c1F)CCC2 Cc1cc(C(N2CCCC2C(N2CCN(C(=O)OCC)CC2)=O)=O)c(N)s1 c1(C(C)NC(c2n(CC=C)nnn2)c2cccn2C)c(F)cccc1F O=C(CCC(F)(F)Cn1cc(COC2CCCC2O)nn1)NC1CCCCCC1 CC(C)CC(O)C(=O)N(CCNC(=O)C(O)Cc1ccccc1Cl)C1CC1 C1(CNC(C(C)(C)C)=O)CCCCN1C(=O)Cc1cncnc1.N12CC(C1)C2=O c1(N(C)Cc2c(C)n[nH]c2)nc(N2CCC(C)C(F)(F)C2)nc2c1CC(C)CC2 Cc1ccc(C(=O)NCCOC2CCN(C(=O)CCC3CC3(F)F)CC2)cc1C CCCC(C(O)C(=O)NCc1csc(C)n1)NC(=O)Cn1nc(C)oc1=O C(=O)(C1=NOC(C)C1)NCC(CC)N(C(c1ccc(CC)s1)=O)C c1(CC(N2CC(OCC(=O)NCCOc3ccco3)C2)=O)ccc(Cl)cc1Cl S(=O)(=O)(c1ccc(NCc2ccncc2Cl)c(Cl)c1)NC1CC(C)N(C)CC1 c1(N(CCC)CCNC(=O)CC2(O)CCCOC2)ncnc(Cl)c1[N+](=O)[O-] c1(C(=O)NC2(C)CCCN(C(C3CN4CCC3CC4)=O)C2)cccc([N+](=O)[O-])c1 C1(C(N(C2CN(C(=O)CC(C)C)CC2F)CC)=O)CCC(NC(=O)CC2CC2)CC1 Cc1cccc2c1NCCC2C(=O)N1CC2(CCC2NC(c2ncn(C)n2)=O)C1 C1(C2CCN(C(C3CCCN3C(C)C)=O)CC2)(NC(CS(=O)(=O)NC)=O)CC1 N1(C(CC2C(C)(C)CCC2)=O)CC2CC1CCC2NC(=O)C=Cc1ncc[nH]1 c1(C(N2CCC3(NC(CNS(N)(=O)=O)=O)C(CC2)C3)=O)ccc2nc[nH]c2c1F C1(CNC(c2ccccc2CC(F)(F)F)=O)CC2(CC2)CN1C(C1CCSCC1)=O c1(CC)ccc2c(c1)N(C(c1nonc1C)C(=O)NCC1CCCO1)CCC2 c1(CC)cc(C(=O)N(C)CC2(NC(C3CCNC3=O)=O)CC2)oc1CC C=CC1CN(C(C2CCNC(=O)C2)=O)CC1NC(C1(COCC)CC1)=O c1(N(C)CC2CN(CC)C2)ccc2cc(S(=O)(=O)NCC=CC3CC3)ccc2n1 C(C(O)C(=O)NCCC(O)CNC(=O)C(=O)N(C)C)=CCCC CC(C)(CC(=O)N1CCN(C(c2ocnc2C2CC2)=O)C2CC12)C(F)(F)F C(CCCCCC(=O)NC1CCOC(C(=O)NCC(F)C2CCC2)C1)SC c1(C(n2nnnc2C(c2nccc(C)n2)NCC2CCCO2)C)ccc(Cl)cc1C N1(C(c2cc(Cl)ccc2F)C(=O)NCCC2CC2)CCCc2[nH]ccc2C1 c1(C(N2CC(OC)C(NC(=O)C(F)F)C2)=O)nc(C)n2ccccc12 N1(C(c2ccc(SC)cc2)=O)CC(NC(=O)C(C)Cn2cccn2)C(C)(C)C1 c1(C(=O)OC)coc(C(=O)N(C)CCN(C(=O)C=CSC)C(C)C)c1 N1(C(C2ON=C(C)C2)=O)CCCC(C(=O)NCc2ccc(N3CCC3)nc2)C1 N1(C(C2(C)CN(C(C3C(OCC)CC3)=O)C(C)(C)C2)=O)CCC2(CCOC2)CC1 C(=O)CCCCCn1cc(COC(=N)O)nn1.CC(C)NC Cn1cc(OC)cc1C(=O)NOC1CCCC(CO)C1.c1(C)ccccc1 C(=O)(C(C)(O)CNC(=O)CCC1(C)CN(C(=O)CCSCC(F)F)C1)OC O=C(C1=NOCC1)NC1CC(NC(=O)CCc2nc(-c3ccccc3)no2)C1 C1(CC(N2C(C=C)CCC2)=O)C2CCCC2N1C(c1ccc(C(C)=O)[nH]1)=O N1(Cc2nnc(CC)o2)CC2CC(C)N(C(=O)C(C)(F)C(=O)OC(C)(C)C)C2C1 C=CC(C)(CC)C(=O)NCC(CC(=O)NC1(CCCCO)CC1)OC c1(C(N2CCC(NC(c3ccc(F)s3)=O)(CF)C2)=O)cc(F)ccc1F C#Cc1cncc(C(=O)NC(C2(O)CN(C(=O)CC(O)C(C)C)C2)C)c1 CC1(CNC(c2cnc(C3CCC3)s2)=O)COCCN(C(c2csc(=N)[nH]2)=O)C1 c1(C(N2CC(CNC(c3n(C)cc(C(N)=O)c3)=O)C(O)C2)=O)ccc2nonc2c1 c1(C2C(C(N(CCCNC(C=C(C)C)=O)C)=O)C2)cccc(C)c1 Cc1nc(N2CCC(CNC(c3cccc(F)c3)CO)C2)c2cc(Br)ccc2n1 c1(C(=O)NCC(F)CNC(c2cc(O)cc(O)n2)=O)ccc(Cl)c(C(F)F)c1 C12CCCCCC1C(=O)N2.C(C(C)CC(=O)NC)OC.C12C=CC(C1)C(=O)N2 Cc1cc2c(cc1C(N1CCC3(CC1)CC3NC(c1occc1Cl)=O)=O)OCO2 c1(N2CCC(C)(NC(C3CC3F)=O)CC2)ncnc2scc(Br)c12 C(=O)(C(O)C(C)(C)C)NC(C(N1CCCC(NC)C1)C(c1cc(C)ncn1)(C)C)=O C(=O)(N=c1ccn(C(C)(C)C)[nH]1)N1Cc2ccc(s2)C1.c1(CC)ccncc1F C(=O)(C(Cc1ccccc1)CC)N(CC(CC)NC(C1(c2cccs2)CC1)=O)C c1(C(=O)NC(C2CCN(c3ncccc3[N+](=O)[O-])CC2)C)cc(F)c(F)c(F)c1 N1(C(Cn2cc(C(=O)OC)nn2)=O)CCN(C(=O)C(O)CF)CC1.C1CO1 c1(NC(C2CCN(C(c3ccnc(OC(F)F)c3)=O)C2)=O)ccc(Cl)cc1Cl N#Cc1cc(C(=O)NC2COCCN(Cc3c[nH]c(Br)c3)C2)ccc1Cl c1(OC)cc(N)c(C(N2CCC(C(F)(F)F)CC2)=O)cc1OC C1(N(C(c2c(C)c[nH]n2)=O)C)CCCN(C(c2ncccc2C(C)(C)C)=O)C1 c1(C(N2CCC(C(=O)NC(c3ccc(CC(N)=O)cc3)C)C2)=O)nccnc1Cl c1(C(N(CCCCN(C(CC2C(C)C2)=O)C)C)=O)ccnc(F)c1F C1(CCOC)(NC(c2cnc(O)cc2C)=O)CCN(C(=O)C(COC)OC)CC1 c1(C(=O)NC2CCCC(CNC(CCC=CC)=O)C2)ccc(OC)c(F)c1N Cc1cncc(C)c1C(=O)N(CC(C)CNC(=O)COC(F)F)C CCCC(CNC(c1cc(Br)sc1C)=O)C(=O)NC1CC(=O)N(C)C1=O N1(C(CSCC(=C)C)=O)CC(C)(C(=O)NC(C)(C)C(=O)NC)C1 c1(OC)cc(F)c(C(N2CCC(CNC(c3nnn(C)c3N)=O)CC2)=O)c(Cl)c1 N1(C(c2c(C)cc(O)nc2)=O)CCC2(CC1)CCN(C(=O)C1=CCC1)CC2 C1(CNC(C(C)=C2CCCC2)=O)C2CN(C(C3(C)CCCCO3)=O)CC12 c1(C(C(=O)NCCC)N(c2ccccc2)CCN(C)C)nc(C(C)C)cs1 C(C(=O)NNC(=O)C(C)(C)S(C)(=O)=O)(C(=O)O)NC(C(CCC(C)C)F)=O C=CCCC(C(=O)NC1CC(CC(C)(C)C)C1)NC(C1CC(F)C(=O)N1)=O c12ccnc(c1[N+](=O)[O-])N1CC3C(C3C1)NC2=O.c1(SCC)ccnc(SC)c1 N1(C(c2ccon2)=O)CCC(NCCNC(c2cnc(COC)s2)=O)CC1 C1(NC(c2conc2C(F)(F)F)=O)CCCN(C(C2C3COCC23)=O)C1 C1(NC(Cc2nnc(C)o2)=O)CCCCCN(C(=O)CN(C)C)C1 Cc1nc2cc(C(N3CCCCC(CNC(C4(C)CC4)=O)C3)=O)cc(O)c2o1 C(CC(=O)N(CC(=O)NC1CC(NC(N)=O)C1)C)OCCC Cc1ccc(Br)c(C(=O)NCC2(C(=O)Nc3cnc(Br)cn3)CC2)c1F c1(C(=O)NC2COCCN(C(C3(CC(C)C)CC3)=O)C2)ccnc2ccnn12 C1(C(=O)NCC(CC)(CC)NC(=O)C(F)(F)C(O)C2CC2)CC2(CO1)CC(F)(F)C2 c1(C(N2CCC(CCC)C2)=O)cccnc1CNC(C1CC(=O)C1)=O C12(C(=O)NC(CC)(C3CC3)C3CC3)CCCC1CN(C(=O)Cc1ccns1)C2 C(=O)(CCCC(C)CC)N(C)CC1CCCN(C(C2(OC)CCCC2)=O)C1 C1(CNC(C2CC(OCC)C2)=O)CN(C(c2cc(C(C)=O)[nH]n2)=O)CCCO1 C1(NC(c2n(CCC)nc(C)c2)=O)CN(C(=O)C(C)=CC2CC2)CC2CCCC12 c1(-n2cc(CN(C(C3CCC3)C)CC)nn2)cccc2n[nH]cc12 c1(CNC(C2CC2Cc2ccccc2)=O)ccc(C(F)(F)F)c(F)c1 c1(C(=O)NC(CNC(c2nc(CC)oc2)=O)(C)C2CC2)cnn2ncccc12 C1(C(O)C(F)F)CCN(CCNCc2ccncc2)CC1 N1(C(COCCCC#C)=O)CCC(NC(c2c[nH]c(=N)cc2C)=O)CC1C Cc1sc(C(N2CC(NC(=O)C3=CCCCO3)CC(O)C2)=O)cc1[N+](=O)[O-] c1(CC(=O)NC(CNC(c2nc(C)n(C)c2C)=O)C(C)C)ccc(F)c(Cl)c1F N1(C(c2c(C)cccc2)=O)CCCCCC(NC(c2ccncc2F)=O)C1 N1(OCOC(C)=O)CCC(OC(C)C)CC1 CCC(CNC(c1cc(Cl)cs1)=O)(CC)C(=O)NC(c1ccccc1)C C1(N(C)C)CCC(CNC(=O)NC2(C(F)(F)F)CCCO2)C1 Cc1ncc(C(N2CCCC(NC(=O)CCC3CCOC3)CC2)=O)c(=N)[nH]1 c1(CNC(c2ccc(C3CCCN3)cc2)=O)nn2c(c1Br)CCC2 c1(OCC)ccc(F)c(Sc2c(C(c3nnnn3C3(C)CC3)N)c(C)ccc2)c1 O=C(CS(=O)(=O)C1CC1)NCC1CCCC1NC(c1cc(CO)ccc1Cl)=O C1(CNC(C2CC(NC(c3n(C)cnc3)=O)C(O)C2)=O)CC2C(C1)C2(F)F c1(SC)ccccc1CC(=O)NC1CCCC(NC(c2ccc(Cl)o2)=O)C1 c1(C(=O)NCC2(NC(C(CC)N(C)CC)=O)CCC2)cnc2cc(C)ccc2c1 C1(NC(C2N=C(C)SC2)=O)CCCC2CN(C(=O)C(C)(C)CCC#N)CC12 c1(CNC(CCN(C(C)C)C(C2CC(=O)CS2)=O)=O)cnc2n1CCC2 Cc1cc2sc(C(N3CCCCC3CNC(=O)CCc3ccccc3)=O)cc2s1 N1(S(CC(=O)NC(C)CC)(=O)=O)CCC2(CCC2)C(C(=O)OCC)C1 c1(CC(=O)NCC2C(NC(=O)Cn3cnnc3O)C2)cccc(Br)c1Cl c1(C(N(C2CCN(C(c3nc(=N)cc[nH]3)=O)C2)CC)=O)cc([N+](=O)[O-])oc1C C(N=c1[nH]c(Cl)ncc1F)C1CC1.CC(CC(=O)N)C1CC1c1ccccc1 C1(C(N2CC(CNC(CCc3c(C)n(C)nc3)=O)C2)=O)CNC(=O)CC1C c1(C2C(N(CCCC3(C(=O)OC)N=N3)C)C2)c(F)cccc1F c1(CN2CC3(C(C(=O)N(C4CCS(=O)(=O)C4)CCO)C3)C2)cc(F)c(O)cc1F C1(C)(C(=O)NCC(CCCC)NC(=O)C(=O)NC(C)C)CCN(C)C1=O C12(C(=O)NCc3nnc(CC)o3)CCCC1CCN2C(=O)CCC1CC(C)C1 C1(C(N(CCNC(CC2(C=C)CC2)=O)CCC)=O)CCc2ccc(F)cc2C1 c1(NC(=O)CSCC2CCOC2)cccc(CNC(c2csc(C(F)F)c2)=O)c1 C(=O)(CC(C)CNC(=O)CCc1cccnc1)NCC1(C(C(C)C)O)CC1 N1(C(C2CC(C)(C)OCC2)=O)CCC2(CCC2NC(=O)Cn2ccnn2)CC1 c1(CC)ncnc(CC)c1C(N1CCC(N(C(=O)C(CC)c2ccccc2)CC)C1)=O CC(C)C(CCN(C)C(c1cc(Br)c[nH]1)=O)NC(=O)Cn1ccc(C(F)F)n1 CC(C)(CN=c1ccc(S(=O)(=O)N2CCOC(CCF)C2)c[nH]1)SC1CC1 C1(CC(=O)NC(C)(C)C)CCCCN(C(=O)C#CC2CC2)C1 n1(CC)nc(C)c(C(N2CC(C(N3CCC(SC)C3)=O)CC(C)C2)=O)c1C c1(NC(=O)NC2CC(CC3CCN(C)C3)C2)oc2ccccc2c1OC(F)F C1(F)(CNC(C2(OC)CCC2)=O)CCCN(C(=O)C(F)C(C)(C)O)C1 C1(C(=O)NCC(C)CNC(C23C4CC(CC24)C3(F)F)=O)CCC2C(C1)C2(F)F c1(C(=O)NC(CNC(C2C(=C)C2)=O)CC)ccc(OCCOC)cn1 Cc1nc(C#N)ccc1C(N1CCC(C(C)NC(c2cnccc2Cl)=O)CC1)=O C1(OC)CCCCN(CC(=O)N(C)CCN(C(=O)C=Cc2ccn(C)c2)C)C1=O c1(C(=O)NC(CNC(c2cc(C(N)=O)[nH]n2)=O)C2CC2)cc2c(nn1)CCOC2 N1(C(Cc2n(C)nc(CC)c2Cl)=O)CCC2CN(C(=O)C(O)CSC)CCC12 C(=O)(C1=C(Cl)CCC1)N1CC(CNC(c2cc(-c3ccco3)[nH]n2)=O)C(O)C1 c1(C(=O)NCC2(OC)CN(C(c3nocc3C)=O)C2)noc2ccccc12 C(CC(C(C)(C)C)NC(=O)CNC(=O)CN(C)C)N(C(C(CC)(F)F)=O)C C1(C(=O)OC)CN(C(=O)C(O)C2CCCC2)CC12CCC2.c1(CC=O)cccc(C(F)F)c1 Cc1nn(C)c(N)c1C(=O)NCC1CC(C)N(C(=O)C=Cc2cnc[nH]2)C1 c12ccnc(c1Br)O2.C1(N(C)CC)CCN(C(=O)NC2CC2c2ccccc2)C1 C(=O)(C(F)CC(C)(C)C)NCC(C1CCOC1)NC(c1cncc(CC)c1)=O Cc1cc(CC(=O)N(C)CC2CCCN2C(C2(C#N)CCC2)=O)ccc1Br c1(C(C)C)ccc(N)c(C(=O)NC2CN(C(=O)CN(C3CCSC3)C)CC2C)c1 c1(C(C)(C)C)cccc(C2CC2)c1F.C12CC1CCN(C1CC1)C2 N1(C(c2cnc(COC)s2)C(=O)NCCCCC(=O)OC)CCC(C#N)CC1 C1(CC#C)(C(N2CC3CC3(NC(c3cc(C4CC4)on3)=O)C2)=O)CC=CCC1 c1(C(=O)NCC2CCCN(C(c3ncccc3C3CC3)=O)C2)cc(I)cnc1Cl C(=O)(CCCC(C)(C)C#N)N1CC=CC(C(N2C(C)CCn3ccnc32)=O)C1 c1(C(N2CC3C(NC(C4C(OCC)C4)=O)CC(CC3)C2)=O)cc2c(s1)CC(C)(C)C2 C12C3CN(CC13)C(=O)CNC(C(C)C)CNC(=O)C2.c1(OC2CC2)ccccc1 c1(C(N2CCC(C(C(=O)NC3(CC)CCOCC3)C)C2)=O)cccc(O)c1F c1(OCC)ccc(CCNC(=O)N(CC)CC2CNC(=O)CO2)cc1OC C1(NC(c2cc(CC)on2)=O)C2CC1CN(C(C1CCC(F)C1)=O)C2 N1(C(CCCC)=O)CCCCC1C1(NC(c2cn(C(C)C)cc2C)=O)CC1 C(=O)(C(C)CC(=O)N(CC(O)CNC(c1cc(C(F)F)ccc1F)=O)C)OC c1(C(=O)NC(C2OCCN(C(CC=C)=O)C2)C)cc(Br)ncc1OC c1(C(=O)NCCCOCCCNC(=O)C=Cc2cocn2)ccc2[nH]ccc2c1 C1(CC(=O)NC2CCC(NC(C(C=C)c3ccccc3)=O)C2)COCCN1C N1(C(C2(CC#C)CC2)=O)CCC(NC(=O)CCc2cccnc2Br)C(O)C1 N1(Cc2cn(CCC)nc2)CCC(C(=O)Nc2sccc2CC#N)C(C)(C)C1 c1(OC)ccc(CN(C)CCNC(=O)Cc2nc(=N)[nH][nH]2)cc1Cl N1(c2ncnc(C)c2F)CC2CCC1C(NC(=O)C(c1cccnc1)O)C2 c1(NC(=O)CC2(NC(CNc3cccc(C)c3)=O)CCC2)cc(Br)c(O)cc1O C=C(C)CC(C(=O)NC1CC2CCC1CC2)NC(c1[nH]ccc1COC)=O Cc1nc(C(C)NC(=O)CONC(C2CCC3(CC3)C2)=O)c(C)o1 C(CCCCC(=O)N1CCCC1C(N)=O)N(C)C(c1cc(=O)cc[nH]1)=O C(=O)(CCCC(=O)N1CCC(COC)(NC(c2ccc(C(C)=O)[nH]2)=O)C1)NCC C1(C(=O)NC2CCN(C(Cn3nc(C)oc3=O)=O)C2)CC2C=CCC(C1)C2 C#CCC(CC#C)C(=O)NCC1CC(NC(c2ccc(C3CC3)o2)=O)C12CCC2 c1(CN(CCO)C(N(C)CCc2nn[nH]n2)=O)ccc(Br)nc1Br c1(CC(=O)NCCOCCN(C(CSC)=O)C)cnn(C)c1 C(=O)(C1CCc2nccn21)N(CCCNC(C1CN(C(C)C)C(=O)C1)=O)CCO N1(C(C(C)OCC=C)=O)CC(C(=O)Nc2cnccc2SC)CC1(C)C C1(C(=O)NC2C=CC(C(=O)OC)C2)(CO)CCCN(C(=O)C(C)CC2CC2)C1 c1(C(=O)OCC)nc(C)[nH]c1NC(CN(C)C(c1ncccc1OC)=O)C1CC1 N1(C(C2C(C)C2(F)F)=O)CCC2C(NC(c3cccc[n+]3[O-])=O)C2C1 c1(C(=O)N(CC2=CCN(c3snc(C)n3)CC2)C2CC2)ccc2c(c1)C(=O)NCCO2 C1(CC(=O)NC)C2CN(C(=O)C(c3ccccc3)NCc3cccnc3)CC12 c1(-c2cc(C(=O)NCC3N(C(Cc4c(C)scc4)=O)CC3)no2)cccc(F)c1 CCCCCCC(=O)NCCCN(C(=O)CC1CCCC(C)(C)O1)C(C)C C12(C=O)CC3CC1C2C3(F)F.c1(CC(=O)N(CCOC)CCCOC)ccc(C)cn1 c1(CCC)nsc(N2CCC(CN(C(=O)C=CCOC3CCOCC3)C)C2)n1 c1(C(=O)NC2C3CC2N(C(c2ccn(C4CC4(F)F)n2)=O)C3)ccncc1F c1(C(=O)NCC(CNC(C2(C#C)CC2)=O)O)cn(C(C)(C)C)cn1 N1(CC)CCOCC1C(N1CC(CNC(=O)CCSc2ccc(C)cc2)C1)=O C#CCC(C)(C(=O)NCc1ncnn1CC)NC(=O)CCn1cnnn1 n1(CC)ncc2cc(NC(=O)C(C)NC(c3cnccc3OC)=O)ccc12 Cc1nc2sccn2c(=O)c1CN=C(NC(C)(C)CF)NC1CC1 Cc1cc(Br)sc1C(N1CCOCC1CNC(C1CCC1)=O)=O c1(CC)cc(C(N2CCCCC2C(C)NC(c2nc(C)c(C)s2)=O)=O)cc(N)c1 C(=O)(C(=O)C(F)(F)F)NCC1C(NC(c2c(CC)c[nH]c2)=O)CCC1 Cc1cccc2c(Oc3ccc4[nH]nc(O)c4c3)cc(=O)oc12 c12cccnc1C(=O)NC2.c1(CC)ccc(C(=O)NOCC(F)(F)F)o1 c1(OC)nc2ccccc2cc1C(N1CCN2C(=O)CCC2C1)C(=O)NCC1CC1 CC1CC2CN(C(C3CCCN3C)=O)CC2N1C(=O)CCCC(N)=O c1(NC(c2ccc(CC)cc2)C)nccc(=NC2CCc3nnnn3CC2)[nH]1 N1(C(C(C=CCCC)O)=O)CCCC(N(C(c2cc(C)c(C)o2)=O)CC)CC1 C(C(=O)OC(C)(C)C)(C(=O)N1CC(NC(=O)CN2CCC(C)(C)C2)C(C)C1)OC Cc1csc(C=CC(N2CCCC(CCNC(=O)CCCn3ccnn3)C2)=O)n1 c1(C(=O)NCCC(CCNC(C(C)(C)OC)=O)C)cnn2c1CCCC2 C1(NC(C2N(C)CC(F)C2)=O)CC2CC1CN(C(=O)C(F)=CC1CC1)C2 CC(=O)CCCC(C)C(=O)N1CCCC(N(C(=O)C(C)CF)C)CC1 CCCCC(F)C(=O)NCC(CO)(CO)NC(c1cccnc1N(C)C)=O Cc1cc(O)ccc1C(=O)NC(C(=O)NOCCCO)c1cccnc1 C(=O)(C(C)(O)Cc1ccccc1)N.C12CC(F)(C1)CCCCC21CC1.C(=O)OC C1(C)(C(=O)NC2(C=C)CCC2)CC(O)CN1C(c1csnn1)=O c1(C(=O)NCCC(C)N(C)C(C2CC=CC2)=O)c(N)cc(Cl)cc1F CC1(C)OCCN2C(=O)N(S(=O)(=O)c3ccccc3F)CC2C1 CCCC(CC(C)C)C(=O)NCC1(CCNC(=O)C(C)(CC)CC(F)F)CC1 N1(C(=O)NC2CCC(C)CC2)CC2(CC2)c2cccc(F)c21 c1(C(N(CC(=O)OC(C)(C)C)CCc2cn[nH]c2)=O)ccc([N+](=O)[O-])nc1 c1(CC(N2CCC(C)(NC(C3CCCCN3N=O)=O)C2)=O)n[nH]c2ccccc12 CC1=CC(NC(=O)CN(C)CC2CC(=O)N(Cc3ccccc3)C2)CCC1 Cc1cnsc1C(=O)NCCN(C(=O)C(CN(C)C)N(C)C)C1CCCCC1 N1(C(C2C(=O)OCC2)=O)CCN(C2CN(C(C3(C4CCC=CCC4)CC3)=O)C2)CC1 C1(CN(C(C2C(OC)C2)=O)C)CN(C(C2(c3ccnc(Cl)c3)CC2)=O)CC12CC2 c1(CC)ncc(C(=O)NCC2(C(C)NC(=O)CC(=O)OC)CC2)cn1 c1(C(=O)NCC2OCCN(C(C(CC)F)=O)C2)cc(Cl)ncc1F CN=c1nc(C(N2CCCC(NC(=O)C(=CC3CCCCC3)F)C2)=O)cc(C)[nH]1 c1(CN(C(C(=O)NC)=O)Cc2ccsc2)cccnc1.C1(C)CCCO1 N1(C(COCC(=O)OC)=O)CCC2(CCC(NC(=O)C(O)CCS(C)=O)C2)C1 c1(CN2CC(CC(=O)Nc3cccc(C(F)F)c3)C2)c(Cl)cncc1Cl N1(C(c2cc(OC)ncc2)=O)CCCC(C)(C(N2CCC3CC23C)=O)C1 C(=O)(CCNC(=O)NCC(C)(C)C(=O)OC(C)(C)C)OC(C)C C(=O)(C1=C(Cl)CCC(C)C1)NC(CN(C(c1cnc(S)nc1)=O)CC)C c1(C(=O)N(CC2N(C(CC)=O)CC(C(F)(F)F)OC2)CC)cc([N+](=O)[O-])cn1C S(=O)(=O)(c1ccnc(C(=O)NCC2(COC)CC3(CCC3)C2)c1)NC C1(NC(C2CC3CC3N2C(c2ccc(F)nc2)=O)=O)CCc2ccccc2C1 N1(C(CCc2ccc(C)cc2)=O)CCC(CNC(C23COCC2C3)=O)C(F)(F)C1 C1(N(C)C)CCCN(C(C(=O)NCC2CCOC2)c2cnc[nH]2)CC1 C(=O)(C(C)(C)C1=CCN(C(=O)CC2CCC(C)(C)C2)C1)NCC1CC(C)OCC1 c1(C(=O)NC(C)CNC(C2(c3cc[nH]n3)CC2)=O)ncccc1Br N1(C(C)=O)CCCC(CN(CCC(C)c2cn[nH]c2)CCNc2nccc(C)n2)C1 c1(OCC)ccc(C(N2CCC(COC)(NC(=O)C(F)C3CCCC3)C2)=O)cc1 CCCCC(CC)CCC(=O)OC(=O)CC1(C)CCN1C(C)(C)C N=c1cc(S(=O)(=O)NC(C2CCC(CC(F)(F)F)CC2)=O)cc[nH]1 N1(C(C(C)(C)OCC)=O)CC(NC(=O)C(F)C(C)C)C(O)C1 c1(CCNS(N2CC(C)C2)(=O)=O)nnc2n1CCCCC2 c12ccc(cc1)CN2CCC.C12(CC1)C(=O)NCC(C)NC2=O.C1(C)CC1 Cc1nn(C)c(C)c1C(=O)NCC(C)(C)CC(=O)NCC(c1nncn1C)C CC1CCCCN1CC(N1CC(NC(=O)CNC(=O)C2CC2)(OC)C1)=O C(=O)(C(CNC(=O)CC1CCC(=O)NC1)CC(C)C)NC1CC(C#C)C1 C1(C(=O)NCC(CNC(C(C)N(C(C)=O)C)=O)C)CCCN1S(C)(=O)=O C(=O)(CC=C(Cl)Cl)NC1CC(C)(NC(CCNC(C)=O)=O)C1.C12CC1C(=O)N2 c1(CCC)cc(C(=O)NCC2(C(C(=O)CC3CCCCC3F)=O)CC2)cc(O)n1 c1(C(=O)NC2CCN(C(c3n(C)ncc3C#N)=O)CC2O)ccsc1S(N)(=O)=O c1(C(=O)NC23CC(CNC(C(CC)(C)O)=O)(OC2)C3)cc(Cl)cnc1OC c1(-n2ccc(C(=O)Nc3nc(-c4ccn(C)n4)sc3)n2)ccc(NCCF)cc1 n1(CC)nccc1CNC(=O)COC1CCN(C(c2ccns2)=O)C1 C(CCc1ccccc1Br)(C(C)(C)C)NC(C(C)NC(=O)C(F)(F)F)=O C(=O)(C(C#N)(CC)CC)N(CCNC(c1ccc(CC)cc1Cl)=O)C(C)C C1(C(=O)NCC2CC(NC(c3on(C)c(=O)c3)=O)C2)CCn2cncc2C1 Cc1ccc2c(c1)C(=O)N(C(C)C(=O)N(C1CC1C1CCNCC1)CCO)C2=O CC(C(C)C(=O)NCC1CCCC1CF)NC(c1[nH]ccc1C1CC1)=O C1(NC(CN(C)C)=O)CC2CCC1(Nc1nnc(C(F)(F)F)s1)C2 C(=O)(C1CCCc2ccccc21)N1C(CN(C(CNC(C)=O)=O)C2CC2)CCC1 C(C)(C(C)(C)CO)NC(CCOCCN(C)C(c1cc(CCO)on1)=O)=O c1(C(=O)NC(CC(C)NC(C2(C)CC=CC2)=O)C)cccc2c1CCNC2=O C12(C(=O)NCc3cc(C)n(C)n3)CCN(C(C3CN(C(C)C)C3)=O)CCC1C2 CC(CCO)C(=O)N1CCC(O)(CNC(=O)C(C)Cc2ccc(N)cc2)C1 O=C(NNC(=O)c1cnc[nH]1)NCC1CC1[N+](=O)[O-] C1(NC(CC2CC(=O)NC2=O)=O)CC2CC(NC(=O)C3=COCC3)CC2C1 C1(NC(CSCC(=O)OC)=O)CC2(C1)CN(C(C1CCC(C3CC3)C1)=O)C2 c1(-n2ncc(C(N3CC4C(CNC(C(C)SC)=O)C4C3)=O)c2)ccc(F)cc1F C1(c2n(CCCC)nnn2)(NC(c2nc(C(C)C)no2)C)CCC(CC#N)CC1 c1(C(=O)OC)cc(C)cc(S(=O)(=O)N2CCCC2c2c(C)c3ccccc3n2C)c1 C1(C(=O)NC(CCC=C)CO)CCN(C(C2CC2C2CCC2)=O)CCO1 Cn1cc(C(=O)NC2CCCC(NC(C3CC3F)=O)C2)c(C(C)(F)F)n1 N1(C(C=CC)=O)CCC(C(F)(F)F)C(NC(C2CCCN2C(=O)C(F)(F)F)=O)C1 C1(CNC(C2(C)ON=C(C)C2)=O)CN(C(=O)CN(C)S(N)(=O)=O)CC(C)(C)O1 N1(c2c(C(CC)=O)cccn2)CC(CN=c2[nH]nc(C)s2)C(C)(C)C1 C1(C(=O)NCC(C)NC(c2ccccc2)=O)CCc2nc(O)cc(C(F)(F)F)c2C1 n1(CC(=O)N(C(C)C2CC2)CC2N(C(CSC)=O)CCC2)c(=O)n(C)c2ccccc12 c1(CSCC#C)cccc(C(=O)OCCCN2CCC2)c1 CC1CCC(NC(c2ccc(C#N)o2)=O)CN1C(C1CCC(=O)O1)=O c1(COC(C)C)ccc(C(=O)NC2CCC2NC(C2(CCF)CCC2)=O)cc1 C#CCC(CC#C)C(=O)N1CC(C(N)=O)(CNC(=O)C(F)(F)c2nc(C)cs2)C1 C(=O)(C1=CCC(C)CC1)NCC1(F)CC(NC(C(CCC)CC)=O)C1 CC(CCCCNC(C1CCC1C)=O)NC(=O)C(O)Cn1cncn1 Cc1cc2[nH]c(C(N3CCCCC(NC(=O)C(F)(F)c4cscn4)C3)=O)cc2o1 C(c1cccc(F)c1F)=CC(N1CC(F)CC(NC(C2(C#C)CCCC2)=O)C1)=O c1(C(=O)NC2C(O)CCN(CC#CC)C2)cccc2nc(O)oc12 Cc1ccncc1OCC(C(N1C(C(=O)OCCCCS(C)(=O)=O)CCC1)=O)C C(=O)(C(O)CC[S+](C)C)N(CCCNc1c(NC(C)=O)c[nH]c1C)C N1(C(CNC(c2ccc(CO)nc2)=O)=O)CCN(C(=O)CC2CCOCC2)CC1 c1(CC)cccc(C)c1C(=O)NCC(C)CNC(c1nccnc1N)=O c1(NC(=O)NCc2ccc3c[nH]nc3c2)nnc2cccc(F)n12 c1(C(N(C2CCCN(C(C(CC(C)C)C)=O)CC2)C)=O)cc(F)c2c(c1)CCC2 C(=O)(C1COc2ccc(F)cc21)N1CCCC(C(C)NC(c2ccsc2)=O)C1 C=CCC(CNC(c1ccccc1CC)=O)C(=O)NC(C)(C)CC1CC1 C1(CC(=O)N(C2CCN(C(C(C)N(C(C)=O)C)=O)C2)C)CSc2ccccc2O1 N1(C(c2cc(CC)on2)=O)CCC2CCN(C(c3ccn4c3CCCC4)=O)CC12 C1(C(=O)NCCCCCCN(C(=O)Cn2cnnc2)C)CC2(C1)CC(F)(F)C2 C1(CNC(C(COC)C)=O)CCC2(CO1)CC(NC(c1cn(C)nc1OC)=O)C2 c1(CC(=O)N(CCOCC(=O)N(CC(COC)O)C)C2CC2)cncnc1 Cc1ccsc1C(=O)NC1(C)CC(NC(C2CC2F)=O)C1 c1(OC)ccc(C2CCCCC2C(=O)NCc2cc(OC)nn2C)cc1 C1(CNC(COC(CC)(C)C)=O)CN(C(c2ccc(OC)c(Cl)n2)=O)CCC1(F)F CC(C(=O)NC1CCCN(C(c2ccc(C#N)[nH]2)=O)CC1)C(C)S(C)(=O)=O c1(CC(=O)NCC2(F)CC(NC(c3c(C)nsc3N)=O)C2)nc2ccccc2s1 c1(NC(C2CCN(CCNC(C3(CCOC)CC3)=O)C2)=O)cc(C)cc(C)c1 Cn1nc(C(=O)NC(c2cccc(Cl)c2)CNC(C2CCC2)=O)cc1O C1(NC(=O)C(O)c2ccsc2)CCCC1C(=O)NC(CO)C1CC1 C1(C(=O)NCCC(CNC(C(C(=O)OC)(C)C)=O)(C)C)CCc2c(ncn2C)C1 c1(NC(C(C2CC(F)(F)C2)OC)=O)cccc(CNC(=O)CCc2cnoc2)c1 Cc1ccccc1C=CC(=O)NC(c1ccccc1)C(=O)NCCc1ccon1 Cc1cccc(C(=O)N(C)CCOCCN(C(=O)CC(C)n2cccn2)C)c1C Cn1nnnc1C(CC1(C)CC1)NC1CCOC1 N1(C(CC(C)N(C)C)=O)CCC2(CC1)OCCCC2NC(c1ccc(C(N)=O)o1)=O Cc1ncncc1C(=O)NC(C)C(N1CCC(NC(=O)N(C)C)C1)=O c1(C(=O)NC2CCN(C(C3=NNC(=O)C3)=O)C23CC3)cccc2cccnc12 C1(NC(CCOC(C)C)=O)CC2CN(C(c3ccc(-c4cnn(C)c4)o3)=O)CC12 N1(C(c2c(CC)n[nH]c2)=O)CC2CN(C(c3cc(Cl)c(Cl)cc3N)=O)CC2C1 c12ccsc1OC2=O.C1(N(CCCC)C(C)=O)CCOC1 N1(C(c2c(C)con2)=O)CCN(C(c2ccc(=O)n(C)n2)=O)C(c2cn[nH]c2)C1 N1(C(CSc2cccc(C)c2)=O)CC(NC(=O)CC(C)C(C)C)CCC(O)C1 N1(CC(=O)Nc2nc(-c3c(OC)cccc3)on2)CCC2(CCC(=O)NC2)C1 c1(COC)cccc(CNC(=NCc2ccsc2Br)NC(C)C)c1 N1(C(c2[nH]cc(CN(C)C)c2)=O)C2CCC1CN(C(=O)CN1CC3CC3C1)C2 C1(CC(N2C(CNC(C3CC3c3cccc(F)n3)=O)CCC2)=O)NC(=O)NC1=O c1(C(=O)NCC2(C)C(NC(C(C)SC(C)C)=O)CCC2)ccc2ncccc2n1 C=C(F)C1(CC(N2CC(NC(C3(CC)CC3)=O)C(n3ccnn3)C2)=O)CCC1 CCCCCCCC(CC)C(=O)NCC(C)(C(C)C)NC(c1cnc(O)n1C)=O Cc1ncc(COC(C)(C)C)c(NC(=O)C(=Cc2cccc(F)c2)F)c1O Cc1c(C(=O)NC2CCC3CC2CN3C(=O)C(F)F)oc2ccc(Br)cc12 N1(C(CCC=C=C)=O)CCC(CCC)(NC(C2CN3CCC2C3)=O)CC1 S(=O)(=O)(c1ccoc1)N1CC(CC(=O)OC)C1C c1(CC)onc(C)c1C(N1CC(C)(OCC(=O)N(CC(=O)NC)CC)C1)=O C(CCSC)(C(=O)NCCOc1cccnc1C(=O)OC1(C)CCCC1)OC C(=O)(CC(C)CC(C)(C)C)NCC(C(C(=O)NCC(=O)NC)F)C C1(CNC(C=C(CC)C)=O)CC(C)(C)CCC1NC(c1cn(CC)nc1CC)=O c1(CCC)cc(C(=O)NCCN2CCN(C(C3CCN(CC)C3)=O)CC2)nn1C C1(N(C(=O)C=CC2CCCO2)CCC)CCN(C(c2n[nH]cc2Cl)=O)CC1 N1(C(C(C=C)CC)=O)CC(C(=O)NCC(N2CCCC2)C)C2(CCC2)C1 CCC(O)CC(=O)N1CC(N(C)C(c2cccnc2C(F)(F)F)=O)C(O)C1 C12(CNC(C(COCC)n3cc(CCCCCSC)nn3)=O)COCC1C2(F)F C=CCC(CNC(C1CC(=C2CC2)C1)=O)NC(C1(SC)CC1)=O c1(N2CCC(CN(C(C3(C)CC(=C)C3)=O)C3CC3)C2)c(C)cccc1C C(CC(C(=O)NC(C)C)N1CC(N(C2(c3ccc(F)cn3)CC2)C)C1)SC C1(NC(=O)C2=COCC2)CCC2(CC1)CC(NC(=O)C=Cc1ccco1)C2 N(C1CCOc2ccc(Cl)cc21)C(=O)Nc1nc(Cc2cc(C)on2)sc1 c1(CC(=O)NC(CC)CN(C(=O)CCN(C)C2CC2)C)cccc(OC)c1.COC C1(N(C(=O)C(C)Cc2ccccn2)C(C2CCCCO2)C)CCNCCC1C c1(C2C(NC(N(CCCC)Cc3ccoc3Cl)=O)C2)ccc(Cl)cc1 CCCCC(C)(F)C(=O)NC1CCCN(c2ncccc2C(=O)C(F)(F)F)CC1 Cc1cnccc1C(C)C(=O)N(C1CCCN(C(c2[nH]cnc2C)=O)C1)CCO n1(CC(=O)NC2CC(C)(NC(CC3(C)CC3)=O)C2)ncccc1=O C1(OC)CCCCCC1NC(c1coc(CNC(=O)CC(O)C(C)C)c1)=O C12(NC(C3CC(NC(CCSC)=O)C3)=O)CCC(=O)N1CCS2 C1(CNC(C2(SCC)CC2)=O)(NC(=O)Cn2nccn2)CCCCC1 c1(C(=O)NC2C(NC(=O)CNC(C3CCOC3)=O)CCCC2)nccc(Cl)c1F C#CCC(C)(CC)C(=O)N1CC(NC(c2cc(C)ccc2F)=O)C2(CCC2)C1 C(CC1=CCN(C(c2ccon2)=O)CC1)NC(c1cn(C2CCC2)nn1)=O N1(C(c2ccc(CN(C)C)o2)=O)CC(N(C)C(c2ccncc2F)=O)C(C)(C)C1 N1(C(C(n2cnc(C#N)n2)C)=O)CC(NC(c2coc(Cl)n2)=O)C2(CCC2)C1 C(CNC(c1cn(CC)nn1)=O)(C(C)(C)C)NC(c1c(CCC)nns1)=O n1(CC2N(C(C3(C(C)(F)F)CCC3)=O)CC2)cc(CC2(O)CCSC2)nn1 S(=O)(=O)(c1cnc(NCC2CC23CCC3)c(Cl)c1)NC1CS(=O)(=O)C1 N1(CC2(C(=O)OC)CC(C(=O)NC(CCOC)(C)C)C2)CCCCCC1 CCC(C)(C)C(=O)C(C=Cc1ccccc1)N1CCOCC1CCF c1(CCNC(=O)CC2COCCN2C(C2C3COCC23)=O)cccc(Cl)c1Cl N1(C(CCCOCCOC)=O)CCCN(C(c2c(Cl)cncc2Cl)=O)CCC1 CC1CC(NSS(C)(=O)=O)CN(CCNC(C2CCC(=C3CCC3)CC2)=O)C1 Cc1cnc(C(=O)NCC(C)(C)NC(c2cccc(F)c2)=O)cc1C#N C1(C(=O)NCC2N(C(CCSC)=O)CCC2)CCN(C(=O)C2CC2)CC1 N1(C(CN2C(C)CCC2)=O)CCCOC(CNC(C2(C3CCC3)CCC2)=O)C1 N1(C(CC2CC(=O)NC2)=O)CC2(CCCN(C(c3scc4c3CCCC4)=O)C2)C1 c1(-c2nc(C(CC)CC)nn2CC2CC2)nc2ccccn2c1F c1(OC)cc(C(=O)NCCC(C)NC(C2SC3C=CC2CC3)=O)cc(OC)c1C C1(CNC(c2c(CCC)n[nH]c2)=O)CN(C(C2Cc3nccn3C2)=O)CCN1C c1(C(N2CC(C(=O)OCC)C(C(=O)O)C2)=O)c(C)[nH]c(-c2ccco2)nc1=O c1(-c2nc(C(C)SCC)nn2C)cn(C)c(=O)cc1C(F)(F)F N1(C(CCC=C)=O)CCCCCC1C(=O)NC1C(O)CC1O Cn1ncc2c1C(N=c1nc(N3CCC4(CC4)C3)c3c(F)cccc3[nH]1)CCC2 CCC(C#N)C(=O)NC(C1CCN(C(c2n[nH]c(C3CC3)n2)=O)CC1)C N1(C(C(C)N(CC)CC)=O)CCC(NC(C2CN(S(N)(=O)=O)C2)=O)C(C(N)=O)C1 C=CC1CCN(C(C2CN(C(C3(CO)CCC3)=O)CC(C)O2)=O)CC1 C1(N(C(=O)CCNC(=O)CO)C)CCCCN(C(=O)CC2(C)CCOC2)C1 N1(C(CC(C)SC)=O)CC2CCC1CN2c1nc(C(C)C)cc(C)n1 c1(C(N2CC(C)N(C(c3csc(C(F)F)n3)=O)CC2)=O)ccc([N+](=O)[O-])c(Cl)c1 N1(C(C2(N=[N+]=[N-])CC2)=O)CCC2(C1)CN(C(=O)CCc1ccc(O)nc1)C2 C1(=O)C(C(C)(C)C)N1.c1(NC(N(C(C)C)CC)=O)cc(OC)cc(Cl)c1 C12(CNC(C(C3CCOCC3)OC)=O)CC1CN(C(c1nc(=N)cc[nH]1)=O)C2 Cc1cc(C(=O)NCC2(C)CCC(NC(=O)COC3CCCC3)C2)cnn1 c1(OC)cc(C)c(Cl)cc1S(=O)(=O)N1CCC(CNc2cncc(O)c2)CC1 C12(C(=O)NCC(CCOC)O)CC(CO)(CN1C(C1CC(C)C1)=O)C2 C(CC(C(=O)N1CC(C)(CF)C1)NC(=O)CC1CC(F)(F)C1)OC N1(C(C(COC)(C)O)=O)CC(CNC(=O)CN2CCNC(=O)C2)CC(C)(C)C1 c1(CN2C(C(CC)O)CCCC2)nc2ccccc2n1C N1(NC(C2(CC)CN(C(CSCC=C)=O)C2)=O)CCC2CC2C1 C1(C(N(C)CC2(O)CCN(C(c3cc(OC)n[nH]3)=O)C2)=O)CC(C(C)C)=NO1 C1(NC(C2CCN(C(c3c(CC)onc3)=O)C2)=O)CCCC2(CC1)CC2 CCC(CC(=O)N(N1CCOC1=O)C)N(C(=O)C(C1CCCC1)OC)C c1(COC)nc(=NC2CN(C(=O)CC3COC(=O)C3)CC2(C)C)s[nH]1 CC(C)C(C(=O)NCC1(F)CCN(C(c2ccc(=O)oc2)=O)C1)c1cnn(C)c1 c1(C(N(CCCCNC(=O)CC2CCC2)C)=O)c(F)cc(F)c(F)c1F c1(CNC(C2(n3cc(-c4onc(C)n4)nn3)CC2)=O)ccc(S(=O)CC#N)cc1 C1(CNC(=O)CCC2CCC2)CCCC2(CN(C(=O)CCn3ccnn3)C2)O1 NS(=O)(=O)c1cccc(-c2cn(CCCC(=O)NC3CSCCC3=O)nn2)c1 C1(CN(C(=O)CCOCC(F)F)C)COCCN1C(=O)CCC1CCCOC1 N1(C(Cc2cc(COC)on2)=O)CCC2C(C(=O)NOCC(F)(F)F)C2C1 C(=O)(C(Cc1cccc(Cl)c1)CCCO)NC(CCC)C1CCCC1 Cc1nc(NC(C2CC(NC(c3c(Cl)cccc3Br)=O)C2)=O)ccc1Br C12(CC(=O)N(CCC(=O)N(C3CC3)Cc3ccsc3)C)CCCC1C2 N1(C(C=CC=CC)=O)CC2CCC(C1)N(C(=O)C1=C(C)OCCC1)C2 C1(C(=O)OC)COCCN1C(=O)C(C)NC(c1ccc(NCC(F)(F)F)o1)=O C1(NC(C(CC)C#N)=O)C2CCCN(C(c3c(C(C)C)cnn3C)=O)C2C1(C)C N1(C(c2cc(C)c(C)o2)=O)CC(C)(C)CC1C(=O)Nc1cc(CO)cc(F)c1 c1(OCCC)ccc(C(=O)NCC(F)CNC(=O)CCC2CC2)cc1OC C1(CNC(c2c(CNC(c3c(C)nsc3)=O)cc[nH]2)=O)CC(=O)N(C)C1 CC(C)CCC(=O)NCc1occc1C(N1CCC2CC2C1)=O c1(CNC(CC2(OC)CN(C(=O)CC3(C#N)CC3)C2)=O)nn(C)cc1C C1(C(=O)NCC2C(C)CN(C(c3cncc(CO)c3)=O)C2)CCn2ccnc2C1 C1(O)(CC(N2CC(N3CCN(C(C4CC5(CC5)CO4)=O)CC3)C2)=O)CCCCC1 c1(C(=O)NC(C2CCN(C(=O)CC3C=CCCC3)CC2)C)ccn2nnnc2c1 C(=O)(CC(C)C(C)C(C)C)NCCC1(OC)CN(c2nc(CC)nc(Cl)c2F)C1 Cc1cccc(CN2CCOC(CNC(=O)C=CC(C)(C)C)CC2)c1O C(CCC(C(=O)NCC(=O)NC(C)(C)C)NC(c1cccs1)=O)OC C(=O)(C1CCCc2c[nH]nc21)N(CCN(C)C(C1(c2cccnc2Cl)CC1)=O)CC c1(C(N2C(CNC(CC(COC)O)=O)C=CC2)=O)cccc2nc(C(F)F)[nH]c12 CC1CN(C(C2CCC(C)CC2)=O)CCC1NC(=O)CSC(F)F c1(C(N2CCC(NC(C(CC)NC(N)=O)=O)C2C)=O)ccc2c(c1)COCO2 C(=O)(CCCCCC#N)NCC12CC(NC(C3N(CC)CCOC3)=O)(C1)C2 N1(C(CC2N(C(C)=O)CCCC2)=O)CC(C2CN(C(=O)C(C)C(C)(C)C)C2)C1 c1(C(=O)NCCC2N(C(c3cnc(COC)s3)=O)CCC2)cc2nc[nH]c2cn1 c1(CC(C(=O)NC2CC(CNC(c3c(C)snn3)=O)C2)C)c(C)n[nH]c1C c1(C(=O)OC)ccc2sc(=NCCNC(c3ccc(N(C)C)nc3)=O)[nH]c2c1 c1(NC(=O)NCC23OCC(CC)(C2)C3)ccc2c(c1)C(=O)N(C)C2=O.C(=O)(NC)N C(C)(CCCCNc1nccc(C)n1)NC(CN(C(CNS(CC)(=O)=O)=O)C)=O N1(C(C(C)CS(C)(=O)=O)=O)CCN(C(=O)C(F)CC2CCC2)CC12CCC2 C1(C(=O)NCC(CNC(C2(C(N)=O)CCC2)=O)O)CC12CCOCC2 C12(C(N3CC4(C3)CN(c3cncc(Cl)n3)C4)=O)CC3CC(C1)CC(O)(C3)C2 N1(C(C(C)CC(N)=O)=O)CCN(C(=O)CC2C=CS(=O)(=O)C2)C2(CC2)C1 N1(C(CC2(OC)CN(C(C3CC4CC(=O)C3O4)=O)C2)=O)CCC2(C=CCO2)C1 CCCC(CC(C)C)C(=O)NC(c1ccccc1)C(=O)N(CCCN)C C(CC(O)C(=O)N(C1CCCN(C(c2coc(C)n2)=O)C1)C)SC C(C(C)(O)CC(=O)NC1CC(F)(CNC(=O)Cc2cc(Cl)n(C)n2)C1)OC C1(C(=O)NCC2C3N(C(CC(C)(C)O)=O)C(CC3)C2)CC12CCC1(CC1)CC2 C=C(C)CC(C(=O)NCC1CCCC2(CC2)C1)NC(=O)CC1COC(=O)N1 CON(C)S(=O)(=O)c1ccc(CNC2CCC(F)(CN)CC2)cc1 c1(CC(=O)N(C)CC2CCN(C(C3CC3CF)=O)C2)ccc(NCC(N)=O)cc1 O=C(C1Cc2cc(-c3ccc(C(=O)O)s3)ccc21)NCNc1ccccc1[N+](=O)[O-] C(c1c(C)noc1C)=CC(N1C(c2ncc(COC)s2)CCCC1)=O C1(N(C2CCCC2)C(C2C3CN(CCO)CC23)=O)CCN(c2cnccn2)CC1 C1(CC=C)(C(=O)N(C)CCc2ccccc2)CCCN1C(c1cccnc1O)=O c1(CC(=O)N(C2CCCN(CC)CC2)C)cccc(S(N)(=O)=O)c1 CC(C)CC(C)(C)C(=O)N1CC2CC(CNC(=O)C(C)N(C)C)C2C1 CC(C(=O)N1CCCC1COC(=O)NC1(C(C)(C)C)CCCCC1)S(C)(=O)=O C(=O)(C1=C(Cl)CCC(C)C1)N1C2CC(CN(C(CSC(C)C)=O)C2)C1 N1(C(C2(CF)CC2)=O)CCC(C(=O)NCc2ccccc2SC)(C(=O)NC)C1.CO C1(NC(C(CC)C)=O)CCN(C(C2(C(F)F)CCCC2)=O)CC1O C1(COC)(NC(=O)Cc2ncc(Cl)s2)CN(C(c2ccnn2C)=O)C1 Cc1cc(C(N2CC3(C2)CN(C(c2ccsc2)=O)CCO3)=O)c2n[nH]cc2c1 C1(C(=O)NC(CN(C(=O)CSCC(N)=O)CC)C)CCC(F)(F)CO1 C(C(C(=O)N(CC(=O)N(CC(C(C)C)OC)C)CCO)OC)OC C(=O)(CC(C(F)(F)F)NC(C1CN2CCC1CC2)=O)NCc1ccc(SC)cc1 c1(C(=O)NCC(CN(C(=O)Cn2cncn2)C)(C)C)cc([N+](=O)[O-])c(N)cc1F C=CC1(C(=O)NCCc2cn(C)cn2)CCN(C(=O)CC2NC(=O)NC2=O)C1 CC(C)C(O)C(F)(F)C(=O)N1CCCN(C(C2CCn3nccc3C2)=O)C(C)C1 N1(C(c2[nH]cc(C)c2)=O)CCCC(N(C)C(c2ccc(C3(O)COC3)cc2)=O)C1 Cn1nc(C2CC2)cc1OC(C1CCN(C(=O)C(N2CCCCC2)=O)C1)=O C(=O)(C1=NNC(=O)CC1)NC(C(C)NC(c1c(C)cc(Cl)cc1)=O)(C)C c1(C(=O)NC2CCC2NC(c2ocnc2C(F)(F)F)=O)cnc(C2CC2)nc1O Cc1cc(C(N2CCC(NC(=O)CCCF)C(C)C2)=O)ncc1Cl C(=O)(CCCCCCC1CC1)N1C(C(NOCC(=C)Cl)=O)C(CC)CC1 C(C)(CNC(c1c[nH]cc1C(F)(F)F)=O)(CC(C)C)OC.c12ccc(cc1)[nH]2 N1(C(c2cc(C(C)C)[nH]n2)=O)CC(NC(=O)C=CBr)CC12CCOCC2 Cc1ccc(C=CC(=O)NC2CCN(CCNC(C3CC34CCOC4)=O)CC2)o1 Cc1c(O)ccc(CNC(=O)Nc2occ3c2CCOC3)c1C C(=O)(C1CCCc2nnn(C)c21)N1CC(NC(C2ON=C(C(C)C)C2)=O)(CO)C1 C(C)(C)(C(F)(F)F)OCC(=O)N(C(C)CNC(C1CCOC1(C)C)=O)CC c1(NC2(C)CCN(C(CN(C(C3COC(=O)N3)=O)CC)=O)C2)ccc(C#N)cc1 c1(C(N2CCCC(C(=O)NCC3CC[Si](C)(C)C3)C2)=O)ccc(F)cc1I c1(C(=O)OC)cccnc1NC1CCOCC1C N1(C(CC=C=C)=O)CCC(CCNC(c2ccc(C)cc2Br)=O)C12CC2 Cc1cnc(F)c(C(=O)N(C2CN(c3nccc(C)n3)C2)C)c1 CC(O)C(C(=O)N(CC(C)(C)NC(c1ccsc1C(F)F)=O)C)N(C)C N1(C(C(C)N2CCC2)=O)CCC(O)(CNC(C23CC(O)C2C3)=O)CC1 C(C)(CC(=O)NC(C(=O)NCC(C)(CO)N(C)C)C1CCCO1)SC N1(C(CC(=O)OCC)=O)CCn2ncc(C(N)=O)c2C1C c1(CN2CC3N(C(c4cccc(OC)c4)=O)C3C2)ncnc2[nH]cnc12 N1(C(c2cc3cnn(C)c3s2)=O)CCC2CN(C(=O)CSC(F)(F)F)CC2C1 C(=O)(C(O)CC(N)=O)N1CCC(CC(=O)NCCCNC(C)=O)CC1 C1(CNC(C(c2ccc(C)cc2)C(C)C)=O)CC2CCC(C1)N2C(C1(F)CC1)=O C#Cc1ccc(C(N2CCCCC(CCC(=O)NC3CCC(O)C3)C2)=O)nc1 c1(-n2ncc(C(=O)NC3C(NC(C(C)=C(CC)C)=O)CCC3)c2)ccc(Cl)cc1 C(=O)(C1CCCc2c(O)cccc21)NCC1N(C(C(F)OC)=O)CC(F)C1 c1(C(N2CC(OC)C(C)(C)C2)=O)cccnc1S(C)(=O)=O C1(C)(CCNC(NOCC#C)=O)NC(=O)NC1=O N1(C(CCN(C)CC)=O)CCN(C(=O)Cn2cc(C(C)O)nn2)CC1C(F)(F)F CC(C)C1=NOC(C)(C(=O)NCCc2ocnc2CNC(c2cncc(F)c2)=O)C1 c12csc(n1)COC2=O.c1(CN(C(C(N2CC(C(C)C)C2)=O)=O)C)ccccc1 C1(N(C(C(CC(C)C)N(C)C)=O)C)CC2CCC(C1)N2C(=O)CCc1cccs1 C1(NC(c2c(O)ccc(CC)c2)=O)CN(C(=O)C(C)(O)C(C)(C)C)CC12CCC2 C1(C(N2CCC(SCC(=O)N(C)Cc3nncn3C)C2)=O)CCC2(CCC2)O1 C(=O)(C(CC(CC)CC)N1CCC(CC)C1)N(CC=C)CC C1(C2CCCO2)(C(=O)NCC(CNC(C(c2cn(C)nc2)=O)=O)(C)O)CCCO1 c1(Sc2n(C)ncc2)ccc2cc[nH]c2n1.C12(CCC1)CC(=O)N(CCO)C2=O C1(C(C)=O)CC1(Cl)C(=O)NC1CC1CNC(=O)CCC1CC(C)C1 N1(NC(C(N2CCCC(NC(C)=O)C2)c2nc(Br)cn2C)=O)CC(C)OC(C)C1 c1(C(=O)NC2CC2NC(C2CCSCC2)=O)coc2ccc(F)cc12 N1(c2ccc(C#N)cn2)CCC2(CCCC2NC(C2CN3CCN2CC3)=O)CC1 C1(CNC(c2ccc(SC(F)F)cc2)C)CN(C)CCO1 c1(C(=O)NCC2(F)CC(NC(C3CC3C3CC3)=O)C2)cccc2c1CCC2 c1(CC(F)(F)F)ncncc1N1CCC(O)(C(F)(F)F)C1 CC1(C)C2CCC(C(N3CCC(F)C(NC(C4CC=CCO4)=O)C3)=O)C1C2 C1(C)(CC)CC(NC(=O)CC(C)(C)O)CN1C(=O)C(=O)NCCCc1ccccc1 N1(C(C(=O)NCC)=O)CC2(CCCN(C(=O)Cn3cnc(Br)n3)C2)C1 C=CCC(CC)N(C(=O)C(C1CC1)N(C(=O)CCc1cnoc1)C)C1CC1 c1(CCC(=O)NCC(C)N(C(CN(CC)CC)=O)C)c(C)nc2ncnn2c1C C1(CC(C)C)CCC(CC)CC1.C1(=O)CCCNC(=O)CCOCCN1 CP(C)(=O)CCC(=O)NC(CNC(C1CCCS1)=O)CC(F)(F)F C#Cc1ccc(C(=O)N(CCN(C(=O)C(C)CS(C)=O)C)C(C)C)c(F)c1 c1(C(=O)NC2C(NC(CCCOC(C)C)=O)C2)ccc2ccccc2c1[N+](=O)[O-] CCCCC(CC(=O)NCC(C)C(C)(F)F)NC(=O)CNC(=O)CC N1(C(CC)=O)CCN(C(c2ccc(C3CC3)s2)=O)C(CC(F)F)C1 C(=O)(C1=CCCCC1)N1CC(=C(CNC(=O)NCCl)F)C1 CCCC(C(=O)NC1CC2(C1)CC2C(=O)NCC1(CN(C)C)CC1)C(C)C c1(CC(CC)NC(=O)COCC2CC2)cccc(S(=O)(=O)CC)c1 C#Cc1cc(F)c(C(N2CCN(C(=O)CC(C)(C)C#N)CC(C)(C)C2)=O)c(F)c1 CCCC(C)(O)CC(=O)NC1CCN(C(c2cc(C3CCCN3C)[nH]n2)=O)C1 C1(NC(C2CC23CCOCC3)=O)CN(C(C23CCC(F)(CC2)C3)=O)CC12CCC2 n1(CC(N2CCC(n3cc(C(CC)NS(C)(=O)=O)nn3)C2)=O)c(C)ccc1C c1(CC)ccc(N)c(C(N2CCC(NC(=O)CC=C(C)C)C(F)C2)=O)c1 N1(C(C(C(=O)OCC)F)=O)CC2COCCC2(NC(c2cc(Cl)ccc2Cl)=O)C1 CCC(C)C(C(=O)NCC(C)N(C)C(c1ccn2ccsc12)=O)OC c1(C(=O)NC(CC)CNC(C2(F)CC2)=O)cc2cc(O)ccc2[nH]1 CC(C)CCC(C(=O)NC1CCC(=O)NC1=O)NC(=O)CC1C=CCC1 O=S(=O)(C1CCOCC1)NC1CC2CCC(C1)N2Cc1cccc2ccnn12 N#Cc1[nH]c(=NCC2CCCC2NC(C2(C3CCOCC3)CC2)=O)sc1Cl c1(C(N2CC(NC(C)=O)C(c3cnn(C)c3)C2)=O)ccc2c(c1)C=CS2(=O)=O C1(C)(C)CC(F)(F)CN1C(=O)C(C)NC(c1cc(C(=O)OCC)no1)=O.C1CC1 Cc1n[nH]cc1CSC1CCCN1CCNC(C(C)(C)NC(C)C)=O N1(C(C=CC=CC)=O)CC(NC(=O)C(C)(F)F)C2CCCCC12 C1(C)(COC)CCN(C(C2(CNC(c3coc(C4CC4)n3)=O)CC(C)(C)C2)=O)C1 Cc1noc(Cl)c1CC(N1CCCC(CCNC(=O)C(C)OC2CCCC2)C1)=O N1(CC(=O)N(C2CCN(C(=O)CC34CCCC3C4)CC2)CC(C)C)C(=O)CNC1=O Cc1oc(CNC(c2coc(C(N)=O)c2)=O)nc1NC(C1CCOC(C2CC2)C1)=O CCCC(C)(C)C(=O)NC1CCCN(C(=O)CC(C)CC)CC1 C1(CC(=O)NC2CC(F)C2)CCC(N(C(C2CCC3CC23)=O)CCO)C1 C1(NC(CC2CCC(C)(C)CC2)=O)CC1C1CCCN(C(=O)CC2(CO)CC2)C1 N1(C(CC)C)CCCC(C(=O)NCc2c(-c3cccc(Br)c3)nn(C)c2Cl)CC1 c1(C(C)(C)C)ccc(O)c(C(=O)NC2CN(Cc3ncc(Br)cc3F)CC2F)c1 c1(C(=O)NC2CCCN(C(CC3C(CC)C3)=O)C2C)c[nH]c2cnccc12 N1(C(C=C(C)C2CC2)=O)CCCCC(C(=O)NC2CC2O)C1 c1(C(N2CCC(N3CCN(C(C4(C#C)CCC4)=O)CC3)C2)=O)cc(C)cc(F)c1 C1(C(=O)OC)CCC(NC(=O)CC2CCCC2NC(C2CCCOC2)=O)C1 C1(C(=O)NC2CCC(CNC(C3(CC4CC4)CCCC3)=O)CC2)CCC2CC2CC1 C1(C(=O)NC(C(=O)NCCCc2cccs2)C2CCC2)C2CCC(F)C12 N1(C(C2CCCN(C(=O)OC(C)(C)C)C2)C(=O)NC)CC(CO)CC(O)C1 N1(C(CC=CCC)=O)CCN(C(=O)C(CC)NC(=O)OC)CC1C(F)F C1(C)(C(=O)NCCCC(C)NC(C(C)OCCC(C)C)=O)CCCCO1 C1(NC(C2CCCO2)=O)CN(C(c2nn[nH]c2Cl)=O)CC1c1ccccc1F c1(C(=O)NC(C(C)NC(c2nc(CCC)sc2)=O)C)cc(C)nc2[nH]nc(C)c12 C1(NC(c2c(C)oc(Br)c2)=O)CN(C(=O)C=Cc2ccc[nH]2)CC12CCC2 C(C(COC)CC(=O)NCC(C(F)(F)F)c1ccon1)OC(C)C N1(C(c2nc(C)sc2)=O)CCC(=O)NC2CN(C(c3coc(Cl)c3)=O)CCC12 CC(C)(C)C(C#N)C(=O)NCC1(O)CCCN(C(c2ccc(CO)cc2)=O)C1 c1(OC)ncc(S(=O)(=O)NC2(C)CCCC2CO)cc1Br C(=O)(C(CC1(C#N)CC1)NC(=O)NC1CCOC1)OC c1(-n2cc(CC3CN(C(C4(COC)CCCCO4)=O)C3)nn2)cc(F)cc(Cl)c1 c1(CCC)cccc(C(=O)NC2CC3(C(NC(C4CC4COC)=O)C3)C2)c1 CC(C)(O)C(F)C(=O)NCC(CO)OOC(F)F.C12CCCC1NC2=O N1(C(N(c2c(C)nn(C)c2C)C)=O)CCN(N2CCC(C(C)O)C2)CC1 N1(C(=O)OC(C)(C)C)CCC2(CC1)CC2(CO)C(N1CC(=O)NCC1C(=O)O)=O N1(C(C2CC(C)=C(C)CC2)=O)CC2OCCN(C(=O)CN3CCCC3=O)C2C1 N1(C(c2ccc(CCC)cc2)C(=O)NC(C)(C)CC)CCCC2(CC(=O)N(C)C2)C1 C1(C(=O)NCc2ccoc2)CCC2(CC2)N1C(=O)CCSC(F)(F)F c1(C(N2CCN(C)CC2)=O)cc(C2=CCC(O)CC2)cs1 c1(CC(=O)NC2C3(C(C(=O)OCC)C3C(=O)O)C2)ccc(C)c(F)c1F N1(C(C(C(C)(C)O)F)=O)CCN(C(c2coc(Br)c2)=O)C2CCCC12 N1(C(CC(C)n2cccn2)=O)C2CCC(C2)C1C(=O)NCC(C)(O)C(F)F O=C1CCN(C(C2CCCCC2CNC(=O)CCc2ccccn2)=O)CCN1 Cc1n[nH]c(C)c1S(=O)(=O)N1CCCC(C(N2CCS(=O)CC2)=O)CC1 C1(CC(N2CCC(CCCC)C2)=O)CCCCN1C(C1CC1[N+](=O)[O-])=O C1(C(=O)NCc2nc(COC)on2)CCN(C(=O)C(C)(C)C(C)O)O1 C=CCC(C(=O)N1CCC(N(C(=O)C(C)SC)C)C1C)c1ccccc1 C1(CC)C(C(=O)NC2COCC2CNC(=O)COC2CCCC2)CCN1C n1(C(C(=O)N(CC(C)NC(=O)C=Cc2ncc[nH]2)C)C)cc(Cl)cn1 c1(COC)nn(C)cc1C(=O)NC1CC(CNC(C2CC(n3cccn3)C2)=O)C1 c1(CC(=O)NCCCNCCCNC(C(C)(C)C)=O)cccc(Br)c1 CCCCC(C(=O)N1CCC(CCC)(C(C)C)C1)N(C)C(c1c[n+]([O-])c(C)cn1)=O C1(C(N2CCC(COC)(NC(=O)CN3C(=O)CCC3=O)C2)=O)OC2CCC1CC2 c1(C(N(CC(C)NC(C2(c3ncccc3F)CC2)=O)C)=O)cc(Cl)cnn1 c1(C(C(=O)NCCC=CC)C)ncnc(OC)c1F CC1(NC(C2CCCN2Cc2ccsc2)=O)CCC(NC(=O)CCC(F)F)CC1 Cc1cccc(OCC(=O)NC2CN(C(C3CCOC3(C)C)=O)C2)c1C N1(C(c2cc(NC(C)=O)oc2C)=O)CCC(O)(CNC(=O)CN2CC=CC2)CC1 C1(NC(C(C)NC(=O)C(C)(C)O)=O)CN(C(=O)CS(C)(=O)=O)CCC1(C)C N1(C(COCCC)=O)CCCC(O)(C2(Nc3cc(O)nc(C)n3)CC2)C1 c1(CC)ncc(C(=O)NCC2(C(C)NC(=O)Cc3nc[nH]n3)CC2)[nH]1 C(=O)(C1CCc2c[nH]nc21)N1CCCC(N(C(C(C(C)(C)C)OC)=O)CCF)C1 N1(C(Cc2c(C)ncs2)=O)CCCCC(NC(c2nc(C)sc2Br)=O)C1 C12(CNC(CCCCSC)=O)CC(NC(C3CCC(C)(C)CC3)=O)(CCO1)C2 CC(N=c1[nH]c(N2CCCC(N(C)C)C2)nc2ccccc12)c1cn[nH]c1 N1(CCC(N2CCC(NC(C3(CC(C)C)COC3)=O)C2)=O)CCCC(N(C)C)C1 C1(NC(=O)NCc2nnn(C(C)C)n2)CCC(OC(F)F)CC1 N1(C(CN2C(C)CCC2)=O)CCC2CCCC(C1)N2C(=O)CN1CCS(=O)CC1 c1(C(=O)NCC(N2CCCC(C(N3C(CC)CCC3)=O)C2)=O)c[nH]c(C)cc1=O CC1(CC(=O)NCC2(C)CCCN2C(=O)CCn2cccnc2=O)CC(F)(F)C1 C1(C(=O)NCC(C)(C)NC(C2CCCS2(=O)=O)=O)CCN(C2CC2)C1=O C1(CCC)CN(C(=O)CS(=O)(=O)NC)CCN1CCN1C(=O)CN(C)C1=O c1(CNC(c2ccc(C)o2)=O)ccc(C(=O)NCCNS(N)(=O)=O)nc1 n1(CC)cnc2nc(=NC3CCCC3SC)[nH]c(NCc3cccc(COC)c3)c12 C(N=c1cc(Cl)c(O)n[nH]1)C1CC(NC(=O)Nc2c(F)cc(C)c(F)c2)C1 C1(CC=C)(NC(=O)CC(C)OC)CCN(c2ccnc(C3CCC3)n2)C1 C(=O)(CC1=CCOCC1)NC(C(C)(C)NC(c1c(CC)noc1)=O)C N1(C(C2N=C(C)SC2)=O)CC2(CCC2)CC1CNC(C1(F)CCOC1C)=O c1(CC)cnccc1CNC(=O)CC1CN(C(=O)CC2COCC(C)O2)CC1C c1(C(=O)NC2CN(C(C3CC(C(=O)NC4CC4)C3)=O)C2)ccc(OC2CC2)nn1 C1(OC)CN(C(=O)C=CC(C)C)C(C)(CNC(=O)CSc2cccc(O)c2)C1 Cc1cc2c(cc1Br)N(c1nc(=N)[nH]c(=NCCC3CCC4CC34)[nH]1)CCO2 c1(NC(CN2CCC(NC(=O)CCc3ccsc3)CC2)=O)c(O)ncnc1O N1(C(=O)Cc2cnn(C(F)F)c2)CCN(C(c2cnccn2)=O)CC1 CCC(CCC(=O)N(C1CCN(C(=O)CCCc2ccc(C)cc2)C1)C)NC(C)=O CC1(C)C(NC(C2CCN2C(=O)Cc2cc[nH]c2)=O)CC1(F)F C(=O)(CS(=O)c1ccc(Cl)cc1)NC1CC(CNC(C(=C(C)C2CC2)F)=O)C1 C1(C(=O)NC(C2CCCC2)CNC(c2cccc(F)c2O)=O)CC2(CCOC2)C1 N1(C(CCSCCCC)=O)CCCC(CNC(C2CCSCC2)=O)C1 N1(c2snc(COC)n2)C2CCC1CC(NC(C1CCC(C)O1)=O)C2 c1(C(CNC(c2occ(C)c2)=O)NC(C2(O)CCCC2)=O)ccc(O)cc1 C1(CNC(C2CCCCO2)=O)CCCCCN1C(C1CCCC1F)=O C1(C(=O)NCC2(C)N(C(CC=C=C)=O)CC(F)(F)C2)COc2ccccc2O1 N1(C(CCOCCOCC)=O)CCC(C)C(N(C(=O)C=C(C)C)C)C1 CC(CNC(C1CN(C)CCN1C(c1ccc(O)nn1)=O)=O)CC(F)(F)F c1(C(=O)NCC(CC=C)NC(c2c(C)nn(CC)c2C)=O)sc2cncn2c1C N1(C(C(C=C=C)C)=O)CCCC2C(NC(c3[nH]ccc3CC)=O)C(C)(C)C12 CC1CCCC1(c1nnnn1C1CCC1)NCc1noc(C(F)F)n1 Cc1ccc(CNC(c2cnn(CCNC(c3ccc(=N)[nH]c3)=O)c2)=O)cc1 O=C(CN1CCC(S(=O)(=O)N2CCCC2)C1)NN1Cc2ccccc2C1 c1(CCNC(C2N(C(CSC)=O)CC(O)C2)=O)cccc2ccccc12 C(=O)(C(C)CC(=O)N1CCN(C(C2CC2OC)=O)CC1)NCC N1(C(C(n2ccc(C)n2)C)=O)CC2(CCN2C(c2cnn3c2CCC3)=O)C1 C(CC(F)F)(C(=O)N1CC(O)CO1)NC(C(CC1CN(C(C)=O)C1)F)=O N1(C(c2cc(Cl)ns2)C)CCN2CC1C2.N1(Cc2ccc(CSC)s2)CCCC1C C1(C(=O)N(CCO)CCO)CCC2(CN(C(c3ccnc(Br)c3)=O)C2)O1 CC(C)CC(CCC(=O)N1CCC(n2cncn2)C1)NC(=O)C(F)C1CCCC1 N1(C(c2sncc2C)C(=O)NCCCCCC)CC2CCCC(O)CC2C1 c1(NC)cnccc1C(=O)NCC1CC1CNC(C1CC1C)=O C1(NC(=O)CC=CC(C)(C)C)CCCC(O)C1.C12CC(C1)C(=O)N(C)C2 c1(C(=O)NC2CC3(C(NC(CCCC#C)=O)C3)C2)cc(F)c(C(C)C)cc1F C(=O)(CC1c2ccccc2C(=O)N1C)N(C1CN(C(=O)CC2CCCO2)C1)C C1(NC(C(=Cc2ccncc2)C)=O)CCN(C(c2csc3cncn23)=O)CC1O c1cccc(CC)c1N.C1(CC#C)(NC(CN(C=O)C)=O)CCOC1 c1(CN2C(CCC)CCOCC2)c(OC)ccc(Cl)c1F CC1(C)CCN(C(=O)CC2CCCS2(=O)=O)CC1CNC(=O)CN=S(C)(C)=O C12(C(N(C(c3cccs3)CC)C)=O)CCC(CC1)N(C(C1CC1CC)=O)C2 Cc1nn(C)c2c(N(CC(C)(C)C)C)nc(=NCc3cc[nH]n3)[nH]c12 C(=O)(C(C(C)NC(=O)CN(C)CC1CCC1)C(C)C)N(c1c(C)c(F)ccc1)C C1(C(=O)NCC2COC(Cc3csc(Cl)c3)C2)(OC)CC(CNC(=O)C2CC2)C1 N1(C(C(CC#C)(C)C)=O)CCCN(C(c2ccc(Cn3cccn3)o2)=O)CCC1 CCCC(C(O)C(=O)N1CCC(CC2CCC2)CC1)Cc1cn(CC)nn1 C12(C(=O)NCC3CCCN(C(C)=O)C3)CC(C)(C1)OC2C.N12CCCC(C1)C2=O CC1OC(C)Cc2c(C(N3CC(CCNC(=O)C#CC4CCOC4)C3)=O)n[nH]c21 c1(C(=O)NC(C)C(CO)NC(C2(C)CCC(=O)NC2)=O)cc([N+](=O)[O-])cn1C C1(NC(c2cccc(CS(N)(=O)=O)c2)=O)CCN(C(=O)CNC=O)C(C2CC2)C1 N1(C(c2cc(C(=O)OC)[nH]c2)=O)CCSC2(CCCC2)C1 c1(C(N(C2CC2)CC2(O)CCN(C(CCCC)=O)CC2)=O)ccc([N+](=O)[O-])nc1 C1(NC(C2CC(CC)OCC2)=O)CCN(C(c2n[nH]c(C)c2O)=O)CCC1CO C1(C(N2C(C(=O)OC)CC2)=O)CCN(C(=O)CSc2cccc(Cl)c2)CC1O C1(OCCC)CCCCC1C(=O)NC1CN(C(C2(CN(C)C)CCCCC2)=O)C1 c1(C(N(CC(CC)NC(=O)C(n2cc(Cl)cn2)C)C)=O)nn(C)c(C)c1[N+](=O)[O-] CCCCC(O)C(=O)N1CCOCC1CNC(c1ncc(I)cc1Br)=O CCC(CC)C(F)C(=O)N1CC=CC(C(N2CCC(CN=[N+]=[N-])C2)=O)C1 N1(C(C2CC(n3ccnc3)C2)=O)CCC(n2cc(-c3cccnc3)nn2)C1 CN1C(=O)CCCC1C(=O)NCCC1(C)CCN(C(C2(C3(C)CC3)CC2)=O)C1 C(CN=c1nc(N2CCCC(C)(CO)C2)cc[nH]1)N(CCOC)C C1(NC(=O)NCC2(c3c(OC)nccc3)CCOCC2)Cc2n[nH]cc2CC1C C#CCCCC(=O)N1CCCCC1CNC(=O)CCNC(C1CCN(C)C1C)=O C(=O)(C1=NOC(NC(c2ccccc2C2CCC2)=O)C1)N(C)CC1N(CC)CCC1 C1(NC(Cc2cc(C)no2)=O)CC(NCCNC(c2ccc(F)cc2)=O)C1(C)C N1(C(n2ccc(C(=O)OC)n2)=O)CCC(C(=O)NC2CC(CO)(CO)C2)(CF)C1 N1(C(C2C(COC)C2)=O)CCC(C)C(CNC(c2csc(-c3cnc[nH]3)n2)=O)C1 C#CC1(NC(=O)CC(C(C)(C)C)NC(=O)C=Cc2ccc(C)o2)CCC(C)CC1 c1(CN=c2[nH]nc(C3CC3)s2)cnc(O)c(C)c1.CCC(F)(F)C(=O)N Cc1ccc(C(N2CCC2CNC(c2ccc(Cl)o2)=O)=O)cn1 c1(CC(C)NC(=O)C(N)=O)ccc(CNC(=O)CNC(=O)Cn2ccnn2)cc1 C(=O)(C1=C(C#N)CCC1)NC(C(C)NC(C(CC)(C)COC)=O)C N#Cc1nc(=NC2CC(CNC(=O)CC3CCC(=O)N3)C2)c(Cl)c[nH]1 c1(C(=O)Nc2c(C)cc(NC(C3CC4CCC3C4)=O)cc2)cc([N+](=O)[O-])oc1C C1(NC(C2N(CCC)CCC2)=O)CCN(C(=O)CCCC2CCCC2)O1 C(=O)(C1CN(C)C(=O)c2ccccc21)NC(c1ccc(OC)cc1)C N1(C(c2nc(CCOCC)oc2)=O)CCC(CC(C)NC(=O)C(C)C2CC2)CC1 c1(C(=O)NCCC2(OC)CN(C(=O)C(C)OCC(C)C)C2)ccnc2ncnn12 C(=O)(CC1=NNC(=O)C1)N1CCC(O)(N(C(CC2(NC(C)=O)CC2)=O)C)CC1 C1(CNC(c2cc(C(C)=O)[nH]c2)=O)COCCN1C(c1cncc(COC)c1)=O Cc1nc2cccnn2c1C(=O)NC1CN(C(=O)CC2CSC2)CCC1C CS(=O)(=O)c1cc(C(N2CC(NS(=O)(=O)CC3CC3)C2)=O)ccc1F C(=O)(C(=O)C(C)(C)C)N1CCC(CN(C(C2CC(=O)N(OC)C2)=O)CC)CC1 c1(C(C)C)ccc(C(=O)NCCC2CCC(NC(=O)CCCc3cnn[nH]3)C2)o1 N1(C(c2cc(C)oc2C)=O)CCN(C(=O)CCc2nc(=N)[nH][nH]2)CC(CO)C1 n1(CC)nc(C(=O)NCC2CCN2C(=O)C(C(C)C)n2ccc(C)c2)c(C)n1 c1(CC(=O)N(C2CCN(C(=O)COC3CCCOC3)CC2)CC)nc(C)sc1C C1(C)(CNC(C(C)=CC)=O)CN(C(=O)CC2CC3(CC3)C2)C(C)(C)C1 c1(C(c2nnnn2Cc2ccco2)NCC2C=CCC2)cccnc1OC1CC1 CC1(C)CCN(C(C23CC(C(F)F)(CO2)C3)=O)C1CNC(=O)CC=C(Cl)Cl c1(CC(=O)NCCC2CCC(NC(c3ccccc3)=O)C2)ccc2c[nH]nc2c1 C(=O)(CCCC(C)(C)C)N(C1CCN(Cc2ccccc2I)CC1)CCC CC(C)C(C#N)C(=O)N(C)CCN(C)C(c1c(C#N)cnn1C)=O C1(CCCNC(=O)CC2CCOC2=O)(C(=O)NC2CCCC2CF)CCCC1.COC C(C)(C(CC(=O)OC)NCc1cn(C(CCF)C(=O)O)nn1)OC c1(CC)ccc(C(=O)NC(=O)CCCN2CC(O)CC2CC)c(F)c1 c1(CC(=O)NCC2(O)CCN(C(Cc3n(C)nnc3)=O)C2)cc(Cl)cc(Cl)c1 c1(C(C(=O)NCC(CCOC)NC(c2coc(C(N)=O)c2)=O)O)ccccc1Cl CCC(C(=O)N1CC2CCC2(CC(=O)NC2CC3(CCCCO3)C2)C1)C(C)(C)CC c1(C(=O)NC(C(=O)NCCSCC)C(C)(C)O)cccc2ccnn12 n1(Cc2cc(C)on2)nnc(C(=O)NC(C)(CNC(=O)C(C)O)C2CC2)c1C C(c1ccc(OC)cc1C)=CC(=O)NC1CCC(C)(NC(C(CC)F)=O)CC1 C1(C(=O)NC2C(NC(=O)CC3(CO)CC3)CC2)CC12CCC2 CCC(CC(=O)NCCC(=O)N(C)C)N(C(=O)C(F)C(C)C)C C1(CNC(C(C2(O)CN(C(c3cc(OC)no3)=O)C2)F)=O)(CO)CC(F)(F)C1 C(=O)(C(C)(C)CCCNC(=O)CCC(C)(C)C)N1CCC(N(C)CCOC)CC1 N1(C(c2ccc(CN)cc2)=O)CCn2ccnc2C1 C1(CCC)(C(=O)N(C)Cc2cscn2)CCN(C(C2C(C)C2(F)F)=O)C1 CCCCC(O)C(=O)N1CC(F)(C(=O)Nc2nc(CC)cc(Cl)n2)C1 Cc1cc(NC(=O)C(CN(C)C)NC(=O)C(C)O)c(F)cc1F C1(CNC(C(CC=C)OC)=O)CN(C(=O)CC(C)(C)O)CC12CCC2 N1(C(C2CCN(C(=O)NC)CC2)=O)CCC(NC(c2nccnc2C)=O)CC1C C(N=c1[nH]c(N2CC3CC=CC2C3)nc2cccnc12)c1ccc(OCCC)cc1 C=CC1OCCCC1C(=O)NC(CNC(c1cc(C(F)F)ccc1F)=O)CO C1(CCC)CC(C(=O)N(C2CCN(C(=O)C=CCCC(C)C)CC2)CC)CCO1 N1(C(=O)CC(F)F)CCN(C(c2ccccc2Cl)=O)C(c2ccccc2Cl)C1 N1(C(c2cc(OC)no2)=O)CCN(C(c2sccc2Cl)=O)CC1C1CCC1 CON=C(C(=O)NCC(C)NC(=O)CCc1ccccc1)c1ccco1 c1(CNCC(C(C)C)N2CCCCC2)nc2c(s1)CC(C)CC2 N1(c2nnc(C)s2)CCC(C(CN(C)C)NC(=O)C(F)n2cccn2)CC1 N1(C(C2COCCN(Cc3ccnc(Cl)c3)C2)=O)CCN2CCCC2C1 N1(C(c2n(CC)ncc2)=O)CC(NC(c2ccccc2Br)=O)C2(COC2)C1 C1(C)(COC)CN(C(C2CC=CC2)=O)C1.c12cc(no1)CNC2=O c1(C(N(CC(C)CN2CC(C(=O)O)C2)C)=O)sc(N2CCCC2)nc1Cl C1(OCCNC(c2cnc(-c3ncccn3)s2)=O)CCN(C(=O)C=CBr)C1 n1(CC(=O)NCCN(C(C)C)C(C2CC3CC3C2)=O)nc(C2CC2)cc1C(F)F Cc1coc(C2CC2)c1C(=O)N(CC(C)CNC(C1CCN(C)C1=O)=O)C c1(SC)ccc(CCC(=O)N(CC(C)O)CCNC(=O)Cc2[nH]cnc2C)cn1 CCCC(C(=O)NCC1CC(F)(F)CO1)NC(c1c[nH]c(C)c1)=O c1(C(=O)NC(CC)(C)CNC(=O)C(C2CC2)SC)cc(C)c(C)cc1Cl N1(C(C2C(C)CC2)=O)CCC(C2CCN(C(c3ccc(C4CC4)cc3)=O)C2)CC1 c1(OC)ccc([N+](=O)[O-])cc1CNC12CC(C(=O)Nc3scnc3C(N)=O)(C1)C2 C(C(C(=O)N(CC(C)(C)C#N)C)NC(c1ccc(CC)[nH]1)=O)SCC c1(SCC)ccc(C(=O)OC)cc1COC(=O)CC(C)Cc1cccc(OC)c1 C(CN(C(=O)CN1CCS(=O)CC1)C)(CO)(CO)NC(C1CCN(C(C)=O)C1)=O c1(C(=O)NCCN(C(=O)Cc2cc[nH]c2)C(C)C)cccc(OC(F)(F)F)n1 c1(CC)nn(C)c(CC(=O)NC2(CNC(=O)CCCc3csc(C)n3)CCC2)c1Cl N1(C(c2n(C(CC)CC)ncc2)=O)CCC(N(C(=O)COCCNC(N)=O)C)C1 C1(CNC(CCNC(C(C)=C(CC)C)=O)=O)CC(C)OC1=O CS(=O)CCCCc1nc(-c2cccc(C(F)F)n2)nn1Cc1cccs1 C1(COC)(CNC(=O)Cc2n[nH]c(=N)s2)CCCN1C(c1ccn(C(C)C)n1)=O C(=O)(CC(C(N)=O)c1cnccn1)NC(C)CCNC(=O)C(C)n1ccnc1 O=C(NNc1ccc(F)c(F)c1F)N(c1ccncn1)C1CCCC1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1C(C)CC(NC(c2cc(OC)n[nH]2)=O)C1 c1(C2C(C(=O)N(c3ccccn3)C(C3CC(O)C3)=O)C2)ccc(F)cc1Br n1(C(C(=O)NC(CNC(C2(CC)CCC2)=O)(C)C2CC2)C)c(C)cc(O)cc1=O C(=O)(C1=CC2CC(C1)CC2O)N1CCN(CCN(C(C(C)C(C)(F)F)=O)C)CC1 C(C(COC)CC(=O)NCCC(C)N(C)C(c1cccc[n+]1[O-])=O)OC C1(C(N(CC(C)(C)NC(C2CCCOC2)=O)C)=O)CC2(CCC(CN)OC2)C1 C1(NC(c2n(CC)nc(C)c2)=O)CC2CC1N(C(c1cc(C)n(C3CC3)n1)=O)C2 c1(C(N2CC3C(NC(CC4(NC(C)=O)CC4)=O)C(C3)C2)=O)cc(Cl)c(N)cc1F C(C(COC)CC(=O)N1CCN(C(=O)CCC(=O)NCc2nccs2)C(C)C1)OC Cc1ccc2oc(C(=O)NC3CC(C)(NC(=O)CC4CN(C)C4)C3)cc2n1 C1(CC(=O)NCc2c(C)ccnc2)CN(C(C2CCOC2)=O)C(C)(C)C1 c1(C(=O)NCCCC2N(C(c3c(CC)nns3)=O)CCCC2)ccc(C)nc1N Cc1ccnc(-c2cn(CC(C)NC(c3ccc(F)s3)=O)nn2)c1 C1(C(=O)N(CC(O)CCO)C2CC2)CC2C=CC1O2 c1(CCC)nc(C(=O)N(C(C)C(=O)N(C)CC2CC(O)C2)CC)cs1 C=Cc1cc(C(=O)NC2(C3CCN(C(C4(C)CCC(=O)N4)=O)C3)CC2)cc(F)c1 C1(=CCNC(C2CC2(F)Cl)=O)CCN(C(=O)CCC2CCOCC2)CC1 C(=O)(CCCN(C)C(c1ccn(C)c1)=O)N1C(C)CC1 c1(C(=O)NC(C)CC(C)NC(C2(O)CCSC2)=O)ccc(Cl)cc1O c1(OCC)c(-c2cscc2C(=O)Nc2ccc(F)cc2Cl)cccc1F c1(CC(N2CCC(OCCNC(Cc3ccn(CC)n3)=O)C2)=O)cccc(F)n1 c1(NC(N(C2CCCC2O)CC=C)=O)ccc(C)s1 C1(COC)(CNC(C2CC2c2cncn2C)=O)CCCN1C(c1cscn1)=O C(=O)(C(F)CCC(C)(C)C)N1CC(SCC)C(C(N2CC(=O)NC(=O)C2)=O)C1 C1(CNC(CC(COC)C)=O)CCCCN(C(C2CCCOCC2)=O)C1 C1(NC(C2CCCOC2)=O)CCN(C(c2ccn3nncc3c2)=O)CCC1CO C=CCC(C(=O)N(CC(C)NC(c1ccc(C(N)=O)s1)=O)C)OC C1(C(=O)NCC(CNC(=O)Cn2cccnc2=O)OC)COCC2(CCC2)O1 C1(CC)CN(C(C2CCC(=O)NC2)=O)CCN1C(=O)Cc1ccc(Cl)nc1 C1(CNC(c2cccc(C#C)c2)=O)CC12CCN(C(c1ccsc1OC)=O)CC2 c1(CC2(OCCC)CCC2)ccccc1NC(C)=O.C12(CC1)C(F)NC2 c1(C(=O)NC2CCN(C(c3ccc(CC)o3)=O)C2)cnc(OC)nc1C Cc1ccnn1C(C)C(=O)NC(CNC(c1cccn1C)=O)C1CCC1 N1(C(C2ON=C(C)C2)=O)CC(NC(=O)C=CC2(C)COC2)CC1(C)C c1(CNC(C)=O)cccc(-c2nc(C(=O)NC3CCCOC3)c(C)s2)c1 c1(CC)cccc(OCC(N2CCCC(C(=O)N(c3ccccc3)C)C2)=O)c1 c1(C(=O)NC(CNC(c2c(C(C)C)nns2)=O)C2CCC2)ccc(N)c(Cl)c1O C1(NC(CCNC(N)=O)=O)CCCC(NC(C2CCC(C(N)=O)C2)=O)C1 C#Cc1cccc(NC(=O)CC2CCN2C(C2CCC(C)(C)OC2)=O)c1 Cc1ccc(CC(=O)NCCCC(C)NC(C2(c3ccno3)CCC2)=O)cn1 C(Cc1cnc[nH]1)(C(=O)NOCCOCC)NC(CCN(CCCCC)C)=O N1(C(c2c(SCC)nccn2)=O)CCC(CNC(=O)C=Cc2cocn2)C1(C)C C(=O)(C(C)(CC)C(F)F)NC1(CNC(c2c(CC)c(OC)ccc2)=O)CCCC1 C(=O)(C(F)CC(C)(C)NC(C1C(C)(C)C1(F)F)=O)N(C)Cc1ncc(C)nc1 c1(C(=O)NC(C)CN(C)C)cc2n(n1)CCC2.C12(COC)CC1C(=O)NC2 C(=O)(C(C)P(C)(C)=O)N(CC)CC1CCCN(C(c2snnc2C2CC2)=O)C1 CC1(C)CC(NC(c2cnc(-c3ccccn3)s2)=O)CCN(C(=O)CC(F)F)C1 N1(C(c2ccc(CC)cc2N)=O)CCN(C(c2ccc(CC)cc2)=O)C2CCC12 C1(CCCC)CCCC1N=c1cc(NCCCCCF)nc(C(C)C)[nH]1 c1(C(N2CCCN(C(c3c(CC)occ3)=O)CC2)=O)cccn2ncnc12 C(=O)(C(C#N)CC1CC1)NCC(C)(C1CC1)NC(=O)Cn1ncnn1 c1(OC)cccc(NC(C2CC(NC(=O)Cc3cncs3)C2)=O)c1OC N1(C(C2N(C(c3nc(CC)oc3)=O)CC(O)C2)=O)CCC(C)C2(CCC2)C1 N1(C(c2scc(C#N)c2)=O)CCC(C2CCN(C(C3(CO)CC3(F)F)=O)CC2)C1 Cn1ncc(C)c1N(c1cccc(-n2cncn2)c1)C(C1CCN1C(=O)CC1CC1)=O c1(C(=O)NC2C(CC)N(C(=O)CCCC(F)F)CC2)ccc(C)c(S(C)(=O)=O)c1 C(C)(CC(=O)N1CCC(N(C(=O)CCc2ccsc2Br)C)C1)OC C1(C(=O)NCCN(C(C2CCN(C)CC2)=O)CCOCCO)CCOC(C)(C)C1 c1(CC(C(=O)NCC(CNC(CC=CC=C)=O)(C)O)O)cc(Cl)cc(Cl)c1 C12(C(=O)NC3(C(N(CCCSC)CC)=O)CC3)CCC(OC)C1C2 Cc1nn(C)c(C(=O)NCC2CN(C(C3CC34CCC4)=O)CC2O)c1Br C(CN=c1[nH]c(N2CCCN(C)C(=O)C2)nc2cc[nH]c12)c1c(C)ocn1 C(c1ccc(F)cc1)=CC(=O)NC(CNC(C1(C#C)CCCC1)=O)C(C)(C)C N1(C(CCSCC)=O)CCOCCC1C(=O)NCCn1ccnc1C c1(C(=O)NCC(CC(=O)NC(CC=C)CO)OC)cc(Cl)cc(Cl)c1[N+](=O)[O-] Cc1cc(C(=O)NC2CCCN(C(c3cc(C(F)F)cc(F)c3)=O)C2)ncc1F Cc1oc(-c2ccccc2)nc1C(=O)NCC(C)NC(=O)CC1COCC1O Cn1cc(Br)c(C(=O)NCC2(O)CCN(C(C3C4(CC4)C34CC4)=O)C2)n1 C1(c2ccc(CNC(CC(=C)C)CO)cc2)CCC(=O)NC1=O c1(C(=O)NC2C(C(N(CC=C)CCC)=O)COCC2)cccc(C#N)c1C Cc1cccc(C(=O)NCC2CCC(C(=O)NC3CCCSC3)CC2)n1 c1(COCC)cc(C(=O)NC2(CNC(c3ccc[nH]3)=O)CCC2)cs1 N1(C(CS(CC)=O)=O)CCC2(C1)CN(C(C1CC1(Cl)Cl)=O)CCO2 N1(C(c2c(C)ncc(C)c2)=O)CC2CCN(C(C3CC(=O)N(C)C3)=O)CCC2C1 C=CCCCCCCC(=O)N1CC2CC1CN2C(=O)CN1CCC(F)(F)C1 c1(NC(C2(CNC(c3cncs3)=O)CC23CCC3)=O)cnn2c1OCCC2 N(C(=NCc1cn(C)nn1)N1CCC(OCC(C)(C)C)C(C)C1)C(COC)C c1(C(=O)NCCCNC(C(CC)(C)C(N)=O)=O)ccnc2ccccc12 C(=O)(C(C)(O)C(F)(F)F)NCC1C(NC(COc2c(C)cc(C(N)=O)cc2)=O)CC1 Cc1cc(C(N2CCN(C(=O)CCc3cnn(C)c3)CC2CF)=O)cc(N)c1 Cc1ccc(CN(C(C)C(=O)NCc2noc(NC(=O)C(C)(C)C)n2)C)cc1 Cc1cc(C(N2CCN(C(C3C(C)C3C)=O)CC2)=O)c2c(C)n[nH]c2n1 C(C(C)(C)N=c1ccc(C#N)n[nH]1)N(C(C(C(C)C)OC(F)(F)F)=O)C CC1=C(C(=O)N2CCCN(C(=O)CN3OC(C)(C)CC3=O)CC2CO)CCCO1 C1(NC(C2(C)CCC2)=O)CN(C(c2cnccc2Cl)=O)CCC1C(F)(F)F C(=O)(C(C)NC(=O)CC=CC(C)(C)C)N(CC#C)CC1CC1 Cc1ccnc(C(N2CCC(NC(C3(n4cccn4)CC3)=O)C2)=O)n1 C#CCC(CC(F)F)C(=O)NCC1CN(C)CCN1C(c1cnn(C(F)F)c1)=O c1(C(C(=O)N2CC(CNC(Cc3cnc(C)[nH]3)=O)C2)(C)O)ccc(F)cc1 c1(C(=O)N(C2CC2)Cc2cccc(F)c2)cn2c3c(cc(F)cc3c1=O)CCC2 CCCCCC(O)CC(=O)NCCC1CCCN(C(=O)C=CCOC)C1 n1(CC)cc(C(=O)NC2C3CCN(C(=O)CCc4nc(C5CC5)no4)C23)c(C)n1 C1(NC(=O)CCc2ccccc2)CCCCC12CCN(C(C1CCC(F)C1)=O)C2 C(CS(=O)(=O)NCC(C)NC1CC(C(C)NC(=O)OC(C)(C)C)C1O)OC N1(C(C(CC)(C)F)=O)CC2CCC1C(CNC(C1CC(=O)N(CC(C)C)C1)=O)C2 c1(NC(=O)NC(CC=C)CNC(=O)OCC)ccc(-c2ccncc2)c(F)c1 C(=O)(C#CC1(C)CCCO1)N1C(C(=O)NC2(c3cc(C)no3)CC2)CCCCC1 c1(-n2c(C3CCCC3)nc(C(C)OC)n2)cc(Cl)ccc1C N#Cc1cccc(C(=O)NCC2(C(=O)NCc3ccc(C4CC4)cc3)CC2)c1 c1(OC(C)C(=O)N(C2CCN(C(C3CCCC3)=O)CC2)C)ccc(Cl)cc1Cl N1(C(c2sccc2Br)=O)CC2CCCC(C1)N2Cc1ncsc1Br C(=O)(C1CCCn2ccnc21)NCC(CNC(c1nccc(OC)c1F)=O)(C)C Cc1ccccc1NC(=O)C(c1csc(Br)n1)N(C)C(c1ccco1)C C1(NC(C=NOC)=O)CN(C(=O)C#CC(C)C)CC1F C12CCC(CC1)NC(=O)CONC2=O.c1(CNC(C)=O)cnn(C)c1NC(C)(C)C c1(C(CC)C)nc(N2CC(OCCNC(=O)CCCc3ccc(C)s3)C2)cc(C)n1 C1(C(=O)NCCCCCC)CC(NC(=O)C(N2CCCC2)C2CC2)CCO1 N1(C(c2c(C)nn(C)c2)=O)CCC(C)(CNC(c2cc(C3(C)CC3)n[nH]2)=O)CC1 C1(C(=O)NCc2ccc(-c3c(CC)nc(C)s3)cc2)CC2(CC2)CN1C C1(CNC(CNC(CCCCC)=O)=O)C(C2CC2)CCN1c1ncc(C)c(O)n1 c1(OCC)nc(N2CC(NC(=O)CC3CCOC3)C3(CC3)C2)ncc1C c1(C(N2CC(CN(C(=O)C(O)C3CC3)C)C2)=O)cn2ccccc2n1 c1(C(=O)NCC(CO)NC(=O)Cc2c[nH]nc2O)c[nH]c2cnccc12 C1(C(=O)NC(C(C)SC)C)CC(C)CN(C(=O)Cn2cc(C#N)cn2)C1 N1(C(C(C)OCC2CC2)=O)CC2CC(C(=O)NCC3C(C)(C)C3(C)C)(C2)C1 N1(C(Cc2nc(NC=O)sc2)=O)CC2CC2(NC(=O)C=C2CCOCC2)C1 c1(C(=O)NC2(CCNC(C=Cc3cn(C)nc3)=O)CC2)cccc(C(N)=O)c1Cl Cc1noc(C(N2CC(F)(CNC(c3ccncc3C(F)(F)F)=O)C2)=O)c1C C12(NC(c3c(Cl)n[nH]c3C3CC3)=O)CCN(C(c3c(O)cccc3F)=O)CC1C2 CC1CC(CCNC(c2cccc(N)c2)=O)CCN1C(=O)COC1(C)CCCC1 C1(NC(C2CC(O)C2)=O)COCCN(C(c2cc(C(F)(F)F)cc(Cl)c2)=O)C1 N1(C(C(CC)(C)C(N)=O)=O)CC2CC(C1)C(CO)C2NC(=O)C=Cc1ccc[nH]1 c1(OC)ccc(C(=O)NC2CN(C(C3CCN(C)C3C)=O)C2)c(OC)c1 C(=O)(CCCCc1cccc(O)c1)NC(C(C)NC(C1CC(F)(CO)C1)=O)CO N1(C(CSc2n(C)cnn2)=O)CCN(C(c2nc[nH]n2)=O)C(CO)C1 Cc1cn2c(C(N3C(C(=O)N(C)C)CC4CCCC34)=O)c(Cl)nc2s1 C1(C(N(CCNC(c2c(C(C)C)n(C)nc2)=O)C2CC2)=O)CC2C=CC1CC2 Cc1cccc(C(N2CC(NCc3n[nH]cc3Cl)C3(CC3)C2)=O)c1O C1(NC(CCN2CCCC(N(C)C)C2)=O)COCCN(C(=O)C2=COCC2)C1 C1(C(N2CCN(C(c3c(C)cc(F)cn3)=O)CC2CF)=O)CCC2CC1C2(C)C c1(CC(C)OC(C2OCCN(C)C2=O)=O)ccc(Br)cc1F c1(Cn2c(NCC(CSC)C)nnc2-c2ccc(Br)cc2)ccc2c(c1)CCCS2 CC12CCCC(C(=O)NCC3CCCCC3NC(C3C4CCN3CC4)=O)(CO1)C2 Cc1cc(C)n(CC(=O)NCC(C(C)C)NC(=O)Cc2ccc(F)cn2)c(=O)n1 C(=O)(CC(=O)NC1CC1)NC(C1CCN(C(=O)C=CC2CCOC2)C1)C C1(C(=O)NCCOC2CN(C(Cn3c(=N)nc[nH]3)=O)C2)CCC2(CCCC2)C1 C1(C(=O)NCCCc2ccncc2)C2CN(C(=O)CC3COCCO3)CC12 C1(CC(=O)NC(CCC(=O)OC)C)C2CCCC2N1C(C1CCCCNC1=O)=O n1(CC(=O)NCC(CNC(C(C)OC)=O)F)c(=O)n(C)c(=O)c2ccccc12 c1(C(N2CC(O)(CNC(C(C)(C)C)=O)C2)=O)ccc(Br)c2ncccc12 N1(C(CCC(=O)OCC)=O)CC(CNC(c2cc[nH]c(=N)c2)=O)CC1(C)C c1(C(=O)NC(CCC)CCC(=O)NC2CCc3nncn3C2)cc2cccnc2[nH]1 c1(NC(C)=O)cnc(C)c(C(=O)NC2CCN(C(C3CC34CC4)=O)CC2OC)c1 C1(NC(C(CC)OCC)=O)CN(C(c2coc(CSC)c2)=O)CC1C(F)(F)F Nc1ccccc1C(=O)CCC(=O)NC1CC1CNC(c1csnn1)=O C=CCC(CC)N=c1[nH]c(N2CCCC(CC(=O)NC)C2)nc2c1COC2 C(C(C(C)(C)C)NC(=O)C(=O)NC1CCCN(C)C1)OC C(=O)(C(CO)C(C)(C)C)NC1C(NC(c2c(NC(C)=O)cccn2)=O)CC1 C1(CNC(COCCN(C)C)=O)CC2(CCN(C(=O)CCc3cc[nH]n3)C2)CO1 c1(C(=O)NC(C(C)(C)C)CNC(C2(C)COC(=O)N2)=O)cnc2nccnc2c1 c1(OC)cccc(C(=O)N(CCNC(=O)COc2cccc(C)c2)C2CC2)c1F Cc1ncnc(C(C)C)c1C(=O)N(C(C)CNC(C1(C2CCCO2)CC1)=O)CCF C1(CC)(NC(=O)CC=Cc2ccccc2)CCN(C(C2CCOC2=O)=O)CC1 c1(OC)ccc2cc(C(=O)NC(C)(C)CCNC(c3ncc[nH]3)=O)[nH]c2c1 O=S(=O)(C1Cc2ccccc2C1)N1c2ccc(Cl)cc2CCC1C(F)(F)F C1(C)(C(N(C)CCNC(C2CCCC3(CCCC3)C2)=O)=O)Cc2ccccc2C1 c1(C(=O)NCC2N(C(C(Br)=C(C)C)=O)CC2)ccccc1C1CC1(F)F C(=O)(CCC(F)(F)F)N.C(=O)CN(CCCN(C)C)CCOCCOCC C1(C(=O)NC2CC(C(=O)NCC(F)(F)F)C2)CCOCC1.C12CN(C1)C(=O)CO2 c1(Nc2n(CC)c(-c3nccc4c3CCCC4)nn2)cc(O)c2cnn(C)c2c1 N1(C(C2CCCN(C(C)=O)C2)=O)CCN(C(=O)CCOCC(C)C)CCC1C O(C=CC(=O)NCCc1ocnc1CNC(=O)C(C)(O)c1ccccn1)CC Cc1cc2c(C(=O)NCC(CNC(c3n[nH]cc3Cl)=O)C(F)(F)F)cccc2[nH]1 CC(O)C(C)(C)C(=O)NC1CCCN(C(c2cc(F)ccc2Cl)=O)C1 C1(NC(c2c(C)ocn2)=O)C2CC1N(C(C1(C)CCC(=O)N1)=O)C2 C(Cc1ccoc1)(C(=O)NC1CC1O)NC(C=CC=CC)=O CCC(CNC(=O)C(CCSC)OC)(CC)NC(=O)Cc1n[nH]c(C)n1 C1(CCNC(C(CSCC)C)=O)CCCCN1C(=O)CCN1CCCC1 CC1CN(C(C2(C)CCN(C(=O)C(c3ccccc3)C)CC2)=O)c2cccnc21 CC(C)C(CNC(c1cc(Cl)ns1)=O)NC(c1csc(C(F)F)n1)=O N1(CC)CCCN(C(c2ccnc(C)c2)C(=O)NCC2CC2)CC1=O C1(NC(C(=O)NC(c2cccc(Cl)c2)COC)=O)CCOC2(CCC2)C1 N1(C(CC2N(C(c3ncn(CC)c3)=O)CCCC2)=O)CC2CCCC2C1 CCC(C)CCCCC(=O)NCC1CN(C(c2cc(Cl)c(Br)cn2)=O)C1 Cc1nc(N(C)CC2CCCCN2C(C2CCCCCCC2)=O)ncc1[N+](=O)[O-] N1(C(C(C=C)O)=O)C2CC1CN(C(=O)CC(C)N(C)C)C2 C1(COCC)CCCN(C(=O)CSc2ncc[nH]2)C1.c12cccc(c1)CNC2=O C1(CC(N)=O)(NC(CCCCOC)=O)CCN(C(c2ccc(CO)cc2F)=O)CC1 C1(C(N2CC3CC(O)CC3C2)=O)C(C2CC2)CCN1C(c1ccc(O)cn1)=O Cc1c(F)cc(C(=O)N(C2CCCN(Cc3cccc(Cl)c3)C2)C)c(F)c1F C1(CC)(CC)NC(=O)N(CC(N2CC(NC(=O)COCCF)C3(CCC3)C2)=O)C1=O n1(C2CCN(Cc3ccc(N)c(Br)n3)CC2)c(O)nc2ccccc12 c1(C(C#C)NS(=O)(=O)CCc2ccccc2F)ccc(F)cc1F C(=O)(C1=CCCCCC1)NCC1(C)N(C(CCn2ncn(C)c2=O)=O)CCC1 N1(C(C2CC(=C)C2)=O)CCCC(NC(=O)CC(C)F)C1CCCC C1(C(=O)NCC(CC=C)NC(c2ccccc2CSCCO)=O)C2CCCCC12 C(=O)(CCCC(=O)N1CCN(C(=O)C(F)=C2CCCC2)CC1C1CCC1)OC c1(-c2cn(CC)nc2)cnn2cc(C(N3CCSCC3)=O)cnc12 c1(-n2cc(C(C)(C)NC(=O)Cc3ccsc3Br)nn2)ccc(Br)cc1 C=CCC(CC(C)C)C(=O)NCCCCC1CN(C(c2cc(N)cc(N)c2)=O)C1 Cc1c(C(=O)NCC#CCNC(=O)COC(C)(C)C(F)(F)F)cccc1F C12(C(=O)NC3C(NC(=O)Cn4cnnn4)COC3)CCC(C(F)(F)F)(CC1)CC2 C1(O)(C(C)CNC(=O)NCC(CCO)c2cnccn2)CCCCC1 N1(C(CC=C)=O)CCCCC1CNC(=O)CCNC(c1ncc[nH]c1=O)=O C1(O)(CNC(C(C)(c2ccccc2)N(C)C)=O)CCN(C(C2CCOC2)=O)CC1 c1(-c2nc(C3N(C)CCN3C)on2)c[nH]c2cccnc12 c1(OC)ccc(Cl)c(C(N2CC3(NC(=O)CCN4CCOCC4=O)CC2C3)=O)c1 S(=O)(=O)(c1ccc(C)c(C)c1)N(C(CCC)CO)C N1(C(C2(C(C)C)CCOCC2)=O)CCCN(C(c2cc(Cl)cnn2)=O)CC1 CC1CCc2[nH]nc(C(N3CCC(F)(CNC(c4cnco4)=O)C3)=O)c2C1 C1(C(=O)N(c2ccc(F)cc2)C)(COCC)CCN(C(=O)C2CC2)C1 C1(C(=O)NCC(C)NC(c2ccnn(C)c2=O)=O)CN2CCCCC2CO1 C#CCCCCCC(=O)N1C(C(=O)NCc2nc(C3CC3)no2)CC2CCCC12 CC(C)C(C(=O)NCCC1COCCN1C(c1csnc1Cl)=O)N(C)C CCCCCCC(=O)NC1CS(=O)(=O)CC1NC(c1cnn(CCC#N)c1C)=O C1(CC)(CC)CCN(C(=O)CN(C(=O)CCCC(=O)N(C)C)C)CC1 CC(CCCCNC(C1C(C)(C)C1(C)C)=O)NC(=O)Cc1c(Cl)cnn1C N1(C(c2c(OC)cccn2)C(=O)NCc2ccccc2)CC(OCC)CCC1C CC1CC(CCO)CCN1C(C(N1CCN(Cc2ccsc2)CC1)=O)C1CC1Cl Cc1ccc(C(=O)NCC(CC(C)C)NC(C2CC3CCCCC23)=O)c(F)c1F C(=O)(CC(C(F)(F)F)NC(C1CC(C(=O)N(C)C)C1)=O)NC(C)Cc1ccco1 C1(C(=O)NC(CCOC)COC)CCN(C(c2cnn[nH]2)=O)C1C(C)C N1(C(=O)CN2C(=O)CCC2=O)CCCC2C1CCN2C(c1ccnn1CCF)=O c1(C(N2CC(NC(C3(C)CCCN3C)=O)CC(C)C2)=O)ccc2c(c1)NC(=O)C2 C1(C(=O)NC2(CCF)CC2)(NC(C2CCC2(F)F)=O)CC(O)C1 CCC(CC(=O)NCC(C1CCCCN1C(=O)CCn1nccc1C)(C)C)OC C=CC(O)C(=O)N1CC(O)(C(C)(C)CNC(=O)CCc2cnn[nH]2)C1 Cc1nn(CC(=O)NC2CCCC2NC(C2(c3ccc(O)cc3)CC2)=O)cc1Cl c1(C(N(CCCNC(CCC(=O)NC)=O)C2CC2)=O)cc(C(=O)OC)cc(O)c1 C1(O)(CNC(COCCCC)=O)CCN(C(C2CCC(C(F)(F)F)CC2)=O)CC1 c1(C(N(CC(CN(C(C2(CC)CNC(=O)C2)=O)C)O)C)=O)nc[nH]c2nccc1-2 Cc1nc(C(C)C)nc(O)c1C(=O)N(CC(C)NC(C1SCCC1C)=O)C c1(-n2c(C(N(CC)CC)=O)nc(SC)n2)ccc2nncn2n1 C1(CC)(NC(=O)C(O)Cc2cnc[nH]2)CCN(C(C2CC(=O)NC(=O)N2)=O)CC1 Cc1cccnc1-n1cc(C2(F)CCN(C(=O)CSC(C)C)C2)nn1 C1(C(N2C(CNC(=O)Cn3ccc(O)nc3=O)C=CC2)=O)CCn2nncc2C1 N1(C(C=C(C)c2cccs2)=O)CCC2CC2(NC(=O)Cc2csc(Cl)c2)CC1 C1(NC(=O)C=C(Cl)Cl)CCCC2CN(C(C3CCCC4CCCN34)=O)CC12 C1(CC=C)(NC(c2cc(O)cs2)=O)CCN(C(=O)CC(C)(F)F)C1 N1(C(C2COCCN(c3cccc(CC)n3)C2)=O)CCCc2nc(C#N)ccc21 N1(C(c2cc(C)on2)=O)CC2(C=C(C(=O)NC3CCOC(C(C)C)C3)CO2)C1 Nc1cc(C(N2CCC(OCCNC(=O)CC3CCCCO3)C2)=O)cc(O)c1Cl C1(C(=O)NC2CCC(=C)CC2)CC12CCN(C(C1CC(=O)C13CCC3)=O)C2 C(=O)(C(C)(F)C(C)(C)F)NC1CN(C(c2cn(CC)nc2)=O)CC1(C)C CC1(C(=O)NCc2cnccn2)CCN(Cc2ccccc2Cl)CC1 N1(CCCC=C)CCC2(CC1)CC(NC(=O)CCCCC(C)(C)C)C2 c1(C(C)NC(C2CC(O)(c3ccccc3)CN2)=O)cc2cnccc2o1 c1(SC)cn(C)nc1C(=O)N(C)CCCC(C)O.c12ccnc(n1)NC2=O Cc1ccc(I)c(C(N2CCCC(C(=O)Nc3nc(C)cc(C)n3)C2)=O)c1 C=CC(C)(C)CC(=O)NC1C(C)CN(C(c2cncc(COC)c2)=O)CC1C CCC(CCC(=O)N(CCC(C)NC(C12CC(C)(CCO1)C2)=O)C)OC C1(NC(Cc2c(C)ncs2)=O)CCOCC1NC(C1CC=CCC1C(F)(F)F)=O c1(C(=O)NC2CC(C(C(=O)NCC(=C)F)F)C2)cccn2ccnc12 C1C(F)(F)CCC(=O)Nc2cn1nn2.C1(CCNC(C)=O)CCS(=O)(=O)C1 C(C(O)C(=O)NC(CC1CCCC1)C(=O)N1CCC1C(C)C)SC O=C1CCC(C(=O)N2CCC(CCNC(=O)C(c3cccc(F)c3)CO)C2)=NN1 C(=O)(C1=Cc2ccccc2C1C)NCCN(C(C(CC)CC1CCCC1)=O)C c1(CC)nn(C)c(C(=O)NCC2CCCN2C(c2ccc(OCC)nc2)=O)c1Cl C1(CC)CCCC12CCN(C(c1nc(CCNc3ccccc3)no1)C)CC2 c1(C(N2CC(NC(c3c(C)onc3C(F)(F)F)=O)C2)=O)cc2c(=O)[nH]ccn2n1 c1(NC(C2C(c3n(CC)ncc3)CCC2)=O)ccc2ncccc2c1 c1(OC)cc(OC)c(F)c(C(=O)NCC2(O)CN(C(=O)C(C)n3ccnc3)C2)c1 c1(N(CCN(C(=O)CC2(C)CC2)C(C)C)C)cc(Cl)on1 c1(OC)cc(C(=O)NC2CC(C(=O)NCCCN3C(=O)C=CC3=O)C2)ccc1F C(=O)(C(c1cccs1)=Cc1ccccc1)NC1CC(CNC(=O)Cc2cscn2)C1 N1(C(C2N(CCCC)CCCC2)=O)CCCN(C(=O)Cc2cnsc2)C(CO)C1 C=CCC(CNC(=O)CC1(C(=C)F)CCC1)C(=O)N.C12CN(CCO1)C2.OCC c1(C(COc2ccc(Oc3c(C)cccc3)cc2)=O)coc2cc(F)ccc12 CCCC(O)CC(=O)N(CC(C)(C)CNC(c1cc(OCC)no1)=O)C C12(N)CCCC1CN(C(=O)COCC1CC1)C2.c1(NC=O)cnn(CC(F)F)c1 N1(C(C(CCC)C#N)=O)CC(C2CCCN(C(c3ccnc4[nH]cnc34)=O)C2)C1 C(=O)(C(O)C1=CCCCC1)NCc1scc(C(=O)NC2C3(CC(OC)C3)C2)c1 n1(CCOC)nc(C(N2CCCC2C(C)(C)CNC(=O)CC#N)=O)ccc1=O C(=O)(CS(=O)(=O)CC(F)(F)F)N(C(C)C)CCNC(C1CC1c1cnn(C)c1)=O C1(CNCc2ccc(C)cc2Cl)CCC2(CCC2)C1NC(=O)CCCC(N)=O CC1(C)CC(NC(c2ccc(C(C)C(N)=O)cc2)=O)CN1C(=O)C1=NNC(=O)C1 c1(C(=O)NC(C)CNC(c2cncc(C(N)=O)c2)=O)cc(Br)ccc1F C(=O)(C(C(C)C)[N+](C(C1CCCC1)=O)([O-])NC)NCCCN(C(=O)C(C)C(C)O)CC C1(CO)(NC(=O)Nc2cncc(OCCC)c2)CCc2cc(Br)ccc21 c1(OCc2nc(CC)c(C)o2)ccc(C(c2ccccc2)=O)cc1 CC1C(NC(=O)Cc2ncccn2)CCCN1C(=O)CCc1ccc(F)nc1 Cc1cc(SCc2ccc(F)cc2Cl)c(C(=O)O)cc1[N+](=O)[O-] C1(O)(C(NC(c2c(NCC)cccc2)=O)CC)CCN(C(=O)C2=CCCCC2)CC1 Cc1ccc(Cl)c(C(=O)NC2CCN(C(C3NC(=O)OC3(C)C)=O)C2)c1O C1(C2CCN(C(=O)CCC3CC3)C2)(NC(=O)CC2CCOC2)CC1 C1(NC(C(CSC)C)=O)CCCN(C(c2ccsc2-n2cnnn2)=O)CC1 c1(C(=O)NCC(C(C)(C)C)NC(c2c(CN(C)C)ocn2)=O)nnc(O)cc1O c1(NC)nc(C)ccc1C(N1CCC(NC(c2ccccc2OCCF)=O)C1)=O C(=O)(C1Cc2ccccc21)N1C(CCNC(c2ccc3c[nH]nc3c2)=O)CCC1 C1(CN(C)C(c2ccsc2)=O)CCCCN1C(=O)C=C1CCC1 C(=O)(CC(C)COC)NCC(C)N(C(c1ncc(C(F)F)s1)=O)CC C=C1CC(C(=O)NC)(C(N2CCC(CCO)C2)=O)C1.C(=O)(C(O)C1CC1)OC N1(C(c2c(C)scc2)=O)CC2CC(C)N(C(=O)C3=CCCC3)C2C1 N1(C(c2c(CCC)nns2)=O)Cc2ccc(CNC(C3CC(OC)C3)=O)cc2C1 C(=O)(CCC(=O)NN(C)C)N1CC(CC)C(NC(=O)C(C)OCOC)CC1 n1(CCC(=O)N(CCC)CCNC(=O)CN2CCS(=O)CC2)cnc([N+](=O)[O-])c1 N1(C(CC(CN(C)C)O)=O)CCCC(C)(NC(=O)C(C2CC(F)(F)C2)O)C1 N1(C(C(N2CCC(O)CC2)C)=O)CCCN(C(C2(CF)CC2)=O)CC1CO C1(NC(Cn2ccc(C)n2)=O)CC12CCN(C(c1cc3c(o1)CCCC3)=O)CC2 C(=O)(CCCS(C)(=O)=O)N1CCC(F)(c2cn(CCN(CCCNC)C)nn2)C1 C(=O)(C(C(=O)OC)C1=CCCCC1)OC.c1(CCN2CC2=O)ccc(C)cc1 Cc1nc(NC(=O)OC(C)(C)C)c(NCc2nccn2-c2ccccc2)n1C c1(C(=O)NC2CCN(C(C(CCN(C3COC3)C)O)=O)CC2)cccc2sccc12 C1(C(N2CCC(C(C)NC(=O)C(C)(F)F)C2)=O)CCC2(CC1)CC(=O)C2 CC(=O)CCCCNCc1csc(Br)n1 c1(CC)nc[nH]c(=NCC(C)(C)N(C(=O)OC(C)(C)C)CC)c1F C1(CC)CCSC1.C(C(=O)NCC1CC1CNC=O)=CCOCCOC CC(CN(C)C)CCC(=O)NC1CC(O)C1CC(N1CCCCC1)=O c1(C(=O)NC(C(C)C)CNC(=O)Cn2nccn2)ccc(S(N)(=O)=O)cc1N N1(C(=O)C(F)=C2CCCC2)CCC2CCN(C(c3nc(Cl)c(Cl)s3)=O)C2C1 C1(C(=O)Nc2cc(C)nc(O)n2)(OC)CCN(C(c2ccccc2F)=O)CC1 C1(Nc2ncc(C(=O)OCC)c(C)n2)CCCN(C(=O)C(C)CC2CC2)C1C c1(N(C2CNCCOC2)C(c2cc(OC)c(F)cc2)=O)ncnc2c1CCC2 CC1CC(=O)NCC1C(N1CC(O)(C(F)C(=O)NCCCOC2CCC2)C1)=O c1(OC(C)C)cccc(CNC(=O)NC2(c3cccc(C)c3)CCCCC2)c1 c1(C(=O)NCCOC2CCN(c3nc(C)nc(Cl)c3)C2)ccn2c(O)nnc2c1 c1(C(=O)NCC(C)CNC(c2cncc(C(F)(F)F)n2)=O)ccc2nsnc2c1 N1(C(C(CC)OC(C)=O)=O)CCCN(C(=O)OC(C)(C)C)CC1 c1(C(=O)NC2C(NC(C(C)(C)c3cnsc3)=O)CCC2)cc(O)ncn1 Cn1ccnc1CCC(=O)NCC1CCCN1C(C1(C)CC1(Cl)Cl)=O c1(C(=O)NCCCCc2ccc(C(C)C)cc2)ccc2c(c1)OC(C)C2 S(=O)(=O)(c1ccc(C(=O)NCC2(NC(=O)C(CO)C(C)(C)C)CC2)cc1)N(C)C c1(CNC2CCCN(C(=O)OCC)C2)ccc(Br)cc1Cl C1(C(N2CCC(N(C)CC)C2)=O)CC2(CC(NC(C3(Cl)CCCCC3)=O)C2)C1 Cc1cc(C)c(C(N2CCC3(CCOC3)C2)C(=O)NC(C2(C)CC2)=O)cc1C C(=O)(C1Cc2c(Cl)cccc21)N1CCC2(CCN(C(=O)Cc3nccs3)C2)C1 c1(C(CNC(C(CCC)=CCC)=O)NC(C2COC(=O)O2)=O)ccc(F)cc1F O=C(C1=C(Cl)CCC1)NC1(n2nccn2)CC1.C12CCN(CC1)C2=O C1(CNC(c2cc(CC)no2)=O)Cc2ccccc2CN1C(=O)CC(C)OC CN1CCC(C)(C(N2CCCC(n3cc(CCOC(=N)O)nn3)C2)=O)CC1 N1(C(C(c2cccc(F)c2)C)=O)CCCC(NC(C2(C(F)F)CCC2)=O)CCC1 CCCCC(O)CCC(=O)NCC1CCC(NC(=O)CC(C)(C)CC)CC1 c1(C(=O)NCC2(O)CN(C(c3c(CC)nccn3)=O)C2)cnc(C)nc1OC N1(C(CN(C(=O)OC)C)=O)CC(C(=O)NCCC2CCC(C)(C)CO2)C(F)(F)C1 N1(C(c2ccc(CCC)s2)=O)CC(C)(C)CC1CNC(c1ncsc1OC)=O N1(C(Cc2c(C)nc(C)s2)=O)CCC(NC(=O)C(C)(C)OC(C)C)CC(C)(C)C1 c1(C(=O)NC(c2c(SC)cccc2)CC(=O)O)ccc(N=S(C)(C)=O)s1 C1(NC(c2c(COC)cco2)=O)CC=C(C(=O)NC2(C)CCOC2=O)C1 C(=O)(CCC(CC)NC(c1cc(F)cc(F)c1)=O)N(CC(=O)NCC)C C1(C(=O)NCC(=O)NC(CCN(CCCNC(CCCC)=O)C)C)CCCCC1 C1(C)(CC)CC(NC(=O)NCC(C)(O)C2CCCC2)C1 Cc1nn(CC(N2CCOCC2CNC(c2cc(F)cs2)=O)=O)c(C)c1Cl c1(CNN2C(C(N3C(C(N)=O)CCCC3)=O)CC(O)C2)ccc(O)cc1O N1(C(C2(C=C)CC2)=O)CCCC(C(C)NC(=O)CC(C)(C)OC)C1 CC1CCCN(C(c2ncccc2N)=O)C1CNCc1ncccc1C(F)(F)F CCC(CNC(=O)C(C)C1CC1)(CC)NC(c1cc(C2(C)CC2)on1)=O N1(C(c2c(CC)nns2)=O)CCCCC1C(C)(C)CNC(c1cc(=N)[nH][nH]1)=O N1(C(c2ccc(CCF)cc2)C(=O)NC2CCCC2)CCOCCC1C(F)F N#Cc1ccc(C(=O)NS(=O)(=O)C2CC2c2cccc(Br)c2)cc1F Cc1cc(C(N2CCC(C(C)NC(c3nocc3C)=O)C2)=O)c(N)s1 n1(CC)nc(C(=O)NC2CC(NC(C3(OC)CC3)=O)C(O)C2)cc1C C1(NC(C(F)=CCC)=O)CCC(C)N(C(c2ccnc(OCC)c2F)=O)C1 c1(C(N(CC(C)CNC(C2CCO2)=O)C)=O)cc2cc[nH]c(=O)c2s1 CN1CC(CC(=O)NCC(C)(CO)NC(C2(C3CC3)CCC2)=O)C(O)C1 c1(C(N)=O)ccc(F)nc1NC(=O)NCC1(O)CCOCC1 C12(NC(CCSCC)=O)CC(C1)N(C(=O)CCOCCOC)C2 C(=O)(CC1=CCOCC1)N1CC(C(=O)NC2CCCCC2OCC=CC(C)(C)C)C1 c1(CC(=O)NC2(C)CC(NC(C3C(C)(COC)C3)=O)C2)cccc(F)c1 C1(C(N2CC(F)(CNC(C3CCCCO3)=O)C2)=O)Cc2cc(Cl)ccc2O1 Cn1cc(Cl)c(CCNC(C(Cc2cn[nH]c2)NC(c2ccc[n+]([O-])c2)=O)=O)n1 C(c1ccc(O)cc1)=CC(=O)NCCCN(C(C1(C)CCC(C)C1)=O)C Nc1c(C(=O)NCC2CCCCC2NC(c2ncccc2F)=O)cc(Cl)cc1F c1(C(=O)NCCCN(C(C2CCCN(C(C)=O)C2)=O)C)cncc(Cl)c1C N1(C(CCCOCC=C)=O)C(C(N2CC(F)(C#N)C2)=O)CCC12CC2 c1(C(C(=O)NCCCN(C)C(C2(C(N)=O)CC2)=O)(F)F)cccc2ccccc12 C1(N(CCC)C(c2ccnn2CC(F)F)=O)CCN(CCCC(=O)O)CC1 C(C)(CNC(C1CC1c1cnn(C)c1)=O)(CO)NC(CSCC)=O c1(C(=O)NCCC2(OC)CN(C(=O)CC(C)CC)C2)[nH]c(C)c(C)c1C c1(SC)cc(C(=O)N(C)CC2(O)CCN(C(c3[nH]c(O)nc3C)=O)C2)ccc1F N1(C(=O)CCCc2cnccn2)CCC2(CCN(C(C3(CF)CC3)=O)C2)C1 C(C)(C)(CCC(=O)N(C)OC1CCCC1)NC(C(CCC)C#N)=O C1(C)(CC)NC(=O)N(CC(=O)N(C)CC2CCCN2C(=O)C=C(Cl)Cl)C1=O c1(OC)ccc(Cl)c(C(=O)NC(C)C(C(C)C)NC(c2nncs2)=O)c1 c1(CCC(N2CC3C(NC(C(C)(O)C4CC4)=O)(C3)C2)=O)ccc(Cl)c(F)c1 C(=O)(CC1OCc2ncccc21)NCCC(C)NC(c1cnc(CC(C)C)s1)=O C1(C(=O)NCC2CC(OC)C2)CN(C(=O)C2=COCCO2)CCC1(C)C c1(NCC(=O)NC(C2CN(C(=O)C(C)(C)F)C2)C)c(F)cccc1Cl Cc1cc(C(=O)NCCCC2(NC(C3CSC3)=O)CC2)sc1-c1ccccc1 C1(C(=O)OC)CCCC2(CN(C=O)C2)O1.c1(-c2cn(CC)nn2)cc(F)ccc1F C(CCN=C(NCCNC(C)C)N1CCC(S(=O)(=O)NC)C1)CCCCCC(C)C.O C#CC1CCCC1NC(=O)C(C1(O)CN(C(=O)CCOC2CCC2)C1)F C1(N(c2nnc(O)s2)C)CCCN(C(=O)C(CO)c2ccccc2)C1 CC1CN(C(c2cnncc2C(F)(F)F)=O)CCN1C(=O)Cc1cn(C)nc1Cl c1(OC)ccc(C(N2CCN(C(=O)CCC(C)SC)C(CF)C2)=O)cc1Cl c1(C(=O)NC(C(C)NC(C(C)(C)SC)=O)C)ccc([N+](=O)[O-])c(C)n1 c1(OC)c[nH]c(C(N2CCC(NC(c3ccc(F)o3)=O)C(F)C2)=O)cc1=O C(=O)(C1=CCCOCC1)NC(CNC(C1CC(OC)C(OC)C1)=O)CC(C)C CC1CN(C(C2CCN(C(c3cc(Br)c[nH]3)=O)CC2O)=O)CCN1C c1(OC)cncc(C=CC(=O)NCC2C=CC(NC(C3(F)CC=CCC3)=O)C2)c1 C12CCCCC1C(=O)N2.c1(CC)ccc(C(N2CC(CCO)(OC)C2)=O)s1 C1(CC#N)CN(Cc2ccc(C#N)cn2)CCN1C(c1ccc(O)c(F)c1)=O C(C1=CCCOC1)N(C)CC1CCC(C)(C)C1 Cc1ccnc(O)c1C(N1CC(CNC(=O)Cc2ccccc2Cl)C(C)C1)=O C(=O)(CCCCCNC(=O)C=CCN(C1CC1)CC)NCCC(CCC)C1CC1 c1(C(N2CC(CCNC(COCC)=O)OC(C)C2)=O)nccn2ccnc12 CN1CCCC(CC(N2C(C(N3CCCC3(C)C)=O)CC3CC23)=O)C1 C1(O)(C(=O)NCCC(C(=O)N(C(CC)CC)C)O)CCC(C)CC1 C12(CC=C)CCN(CC1)C(=O)C=CO2.c1(C(=O)OC)ccc(=O)n(CC)n1 C1(C(=O)N(CCCNC(C(COC)O)=O)CC2CCCC2)(C(F)F)CCOCC1 C1(NC(C=CC)=O)CC2C(NC(=O)CCn3cncn3)C2C1 N1(C(CN2C(C)CCC2)=O)CCC2(CC1)CC2NC(c1cc2nc[nH]c2cn1)=O C(CCN(C)C(c1ccc(C(C)(F)F)cc1)=O)(C(C)C)NC(C1CC(SC)C1)=O CC1CN(C(=O)OC(C)(C)C)CC1CO.c12coc(n1)C1N(CCC1)C2 C(=O)(C1=NOC(C)(C)C1)NC(CC=C)CNC(c1ccc(C(F)F)s1)=O c1(C(=O)NC(CNC(C2C(C)C2)=O)CO)cccc(F)c1O C(=O)(C1=NOC(C)(C)C1)NC1CCCC(NC(CCCCCC#C)=O)C1 C1(NC(c2nc(C)n(C)n2)=O)CN(C(C2CC3(CC(=O)N3)C2)=O)C2CCCCC12 C(C)(C(CC(=O)NCCN1CCCCCC1=O)NC(=O)C(c1ccnn1C)C)OC c1(C(C)C)cccc(CC(=O)NCCNC(C2CC3CCC3C2)=O)c1 C=CC1CN(C(c2c(C)coc2C)=O)CC1NC(=O)C(C(C)OC)N(C)C CC1=C(C(=O)NCCC2CCC(NC(C3CCN(C(N)=O)CC3)=O)C2)CCO1 C1(CC(=O)NCCC2(OC)CC2)CC2(CC2)C1.C1(C(=O)N)CSCCS1 Cc1c(C(=O)NCC2(C(C)(C)C)CCCO2)cccc1O c1(C(=O)NC(C(C)NC(=O)COc2cccnc2)(C)C)cc2ccc(F)cc2o1 c1(C(=O)NCCC(CC)(C)NC(=O)CC2CC2)cnc2c(C)ccccc1-2 c1(CC(=O)NCC2OCC(CNC(=O)C=CBr)C2)cc(Cl)ccc1O C(=O)(CS(C)(=O)=O)NCCCCNC(c1cc(NC(=O)OC(C)(C)C)n[nH]1)=O Cc1nn2c(c1Br)N(C(=O)C(=O)NC1CCCCC13NC(=O)NC3=O)CC(C)C2 C1(n2cc(C=O)nn2)CCN(CN)CC1.c1(Cc2n(CC)ccn2)ccncc1C C1(CC(N2C3C(NC(CC4C(C)(C)CCO4)=O)C(C3)C2)=O)CC2CCC(C1)C2 C(CC(=O)NCC1CC(=O)N(C)C1)(C(F)(F)F)NC(c1c(C(C)(C)C)con1)=O N1(CCC2N(C(=O)OC(C)(C)C)CCCC2)CC2(C)CC1CC(C)(C)C2 CC1CCC(C)N1CC(=O)NC1(CNC(C2(O)CCCC2)=O)CC1 C1(COC)(NC(c2occ(C)c2C)=O)CCN(C(=O)C=CC(=O)N(C)C)C1 N1(CC(=O)NCC(CCNC(c2ccn(COC)n2)=O)O)CCn2ccnc2C1 Cc1scc(C(=O)NC2CCN(C(c3cccc(CCO)c3)=O)C2C)c1C C1(OCC)CCC2(C1)CC2C(N1CC(CCNC(c2cccc(SC)n2)=O)C1)=O CC(C)CC(C)(CNC(C1CCC1C(F)F)=O)NC(=O)COC1CCC1 C(=O)(CCCCC1CC1)NCCN(C(C(C)Cc1ccncc1)=O)C1CC1 c1(C(C(=O)OCCC(CC)(C)C)NC(=O)OC(C)(C)C)ccnn1C C1(CC(C)(C)C)CN(C(=O)CCC2CCCO2)CCN1C(c1c[nH]c(C#N)c1)=O c1(OC)ccc(CC(N2CCC(NC(=O)CC3CC3)C(C)C2)=O)c(C)c1 N1(C(c2ccc(Cl)s2)C(=O)NCC(=C)C)CCCC(C(=O)OC(C)(C)C)C1CC C1(CNC(C(C)NC(COC)=O)=O)N(C(=O)C(c2cnn(C)c2)O)CCCC1(C)C CCCNNC(=O)CCCCCCNC(=O)CC(c1ccc(F)cc1)OC c1(C(=O)NC2CN(C(c3c(OCC)scc3)=O)C(C)CC2)cccc2c1NCC2 c1(OC)ccc(C)c(CNCC2CN(C(c3cc(C)cc(C)c3)=O)CC23CC3)c1 N1(C(C)=O)CCC(O)(C(C)NC(=O)CC2CCCN2CCN(C)C)CC1 c1(OCC(=O)NC(C)CNC(C23CC(F)(CO2)C3)=O)cccc(SC(C)(C)C)c1 c1(OC)ccc(NC(=O)C(O)C2CN(C(c3cc(C)sn3)=O)C2)c(O)c1 C(=O)(CC(N=c1[nH]c(N(CCCOC(=N)O)C)nc(=N)[nH]1)c1cccnc1)N(C)C C1(C(=O)NCC(O)C(=O)N2CCC(F)C2)CC12CCCCC2 c1(C(N(C)CC2OCCN(C(CCC=C)=O)C2)=O)ccn2ccnc2n1 Cc1oc(CNC(=O)C(N2CCOCC2)C)nc1C(=O)N(C1CCCC(O)C1)C N1(C(C=CC=CCC)=O)CCC2CCC(C1)N2C(c1cnc(OC)c(C)c1)=O c1(C(C(N2CC(O)(CNc3cc(SC)ncn3)C2)=O)=O)cccc([N+](=O)[O-])c1 C1(C(N2C(C)CN(C(=O)CCc3ncco3)CCC2)=O)CC2(CO1)CC(F)(F)C2 C12(NC(c3ncc(C)nc3)=O)CCCC1N(C(c1ccc3c[nH]nc3c1)=O)CC2 C(=O)(C1=C(C)OCC1)CN(C1CCN(C(C2C(OC)(OC)CC2)=O)CC1)CC1CC1 CCCCC(C)(F)C(=O)NC(CO)C(C)NC(c1cc(C)nn1CCC)=O CC1CN(C(=O)CCCc2ncco2)CCCN1C(c1ccsn1)=O c1(OC)cc(C)c(C(N2CCCC2CC(=O)NC2CC2O)=O)cn1 C12(NC(c3ccsc3)=O)CCN(C(C3(N(C)C)CC3)=O)CCC1C2 n1(CCC)nc(C)c(C(N2CCOCC(CNC(C3CCC3CF)=O)C2)=O)c1C C(CC(=O)NC1C2CN(C(C34CCC(C3)C4)=O)CC12)(C(F)F)OC C12(CCC(C)(C)C1)C(=O)N2.N(C(=NCC1CCNC(=O)C1)NCC)C(COC)C CCC(C)CC(=O)C(=O)N(C)CC1CCCN1C(c1ccccc1OC)=O c1(NC(C(C)=C2CCCC2)=O)nc(CC(=O)C(CNc2ccccn2)=O)cs1 N1(C(c2c(COC)nn[nH]2)=O)CC=C(CNC(=O)C=Cc2cnc[nH]2)CC1 c1(C(C(=O)N(CC(CC)NC(=O)CS(C)(=O)=O)C)C)ccccc1OC Cc1c(C#N)c(N2CCN(C(=O)C(N)=O)C(C)C2)nc2ccccc12 c1ccn(C)c(=O)c1.c1(OC)cccc(CNC(=O)NCCCONC)c1.O c1(C(N(C)C(C)C)=O)ccc(C(=O)NCCCn2cc(CC(C)C)nn2)cc1 N(C(=NCc1ccc(O)cc1)N(C)CC(C1CCOCC1)OC)C(CC)C C(=O)(CC(C(C)C)NC(C1CCCC(C#N)C1)=O)NCCCCCSC N1(C(CP(C)(C)=O)=O)CCCC2CN(C(=O)CC3CC4C=CC3C4)CC12 C(CNC(c1c(C)nn(C(C)C)c1C)=O)(C(C)C(C)C)NC(c1c(C)noc1N)=O C(=O)(C1=NN(CC(C)C)C(=O)CC1)NCCCCN(C(CC1CC(OC)C1)=O)C c1(C(N2C3(CC3)C2)=O)cc(F)ccc1C.c1(COC)cc(CN(C)C2CC2)on1 C1(NC(CC(C=C)CC)=O)CCC2(CC1)CN(C(=O)CCCS(C)(=O)=O)CCO2 C1(C(=O)NCCC2CC(NC(CC3N(CC)C(=O)CC3)=O)C2)CC(=O)NC1(C)C c12ccc(c(Br)c1)S(=O)(=O)NC(=O)CCN2.C12(CO)CC1C2.C(C)(C1CC1)N.CO C1(Cc2ccoc2)C(=O)N1.C1(C(=O)NC(C(=O)OC)C2CCC2)CC1(Cl)C(=O)OC c1(OC(C)C)cccc(C(=O)N(C)CC2(NC(=O)CC3CCCN3C)CC2)n1 c1(CN(C(=O)CCN(C(=O)CCn2cnc(=N)[nH]2)CCO)C)ncccn1 C1(NCC(C)Oc2c(C)cccc2)CCc2nc(C(F)(F)F)[nH]c2C1 N1(C(c2c(C)nns2)=O)CC(CNC(C23COC(CF)(C2)C3)=O)C(C)C1 CCCC(C(=O)NC1CCCC(NC)C1)NC(=O)C=CC(=O)NC1CC1 N1(C(CCOCC)=O)CCC(CC(N)=O)(NC(c2cnc(Cl)cc2Cl)=O)CC1 N1(C(C(C)NC(=O)NC)=O)CC2(CC(NC(=O)CCC(=O)NC)c3nccn32)C1.NC C#Cc1ccc(CC(N2CCCCC2C2(NC(C3(F)CC3C)=O)CC2)=O)c(F)c1 N1(CC(=O)OCc2ccsc2)CCCCC1C(C1CCC1)O C1(NC(C(C)c2ccon2)=O)CCCCN(C(=O)CNc2ccccc2Cl)C1 CC1CN(C(C2CC(O)CN2C(N)=O)=O)CC1CNC(=O)CCc1ccnc(Cl)c1 C1(CC)CN(C(C23CCCC2(C(N)=O)C3)=O)CCN1C(C12CC(CC)(CO1)C2)=O n1(CC(N2CCC(CCNC(C(C=C)C)=O)C2)=O)c(C)c(C)sc1=O C(=O)(C(C(C)CC)N1CCC(=C(F)F)CC1)NC(CCCCC)C c1(CC)ccccc1-n1cc(C(C)N(C)C(c2csnc2Cl)=O)nn1 c1(NC(N2C(C34C(C)(C)OC(C5CC5)(C3)C4)CCCC2)=O)nc2ccccc2[nH]1 c1(C(=O)NCCCCCNC(c2cc(C)no2)=O)coc2c1C(=O)CCC2 C1(C(=O)NCCN(C)C(c2csnn2)=O)OCC2CCCC12 c1(C(N2CCC(C)(NC(C3CCCS3)=O)CC2)=O)c(Br)ccc2ccccc12 c1(C(N(CCCNC(C(C)SC)=O)C(C)C)=O)ccc(Br)o1.C1C(=O)N1 c1(C(=O)NCC2C(CNC(CC3N(C)CCCC3)=O)C2)ncnc2ccsc12 c1(CN(C(C2C=CC(NC)C2)=O)CC)ncc(C(C)C)s1 N1(C(CNS(CC)(=O)=O)=O)CCCC(C2CCN(C(c3cc(C)nn3C)=O)C2)C1 c1(C(N2CC(CNC(c3n[nH]c4c3CSCC4)=O)C2)=O)cccc2ccnn12 N1(C(c2c(CC)c[nH]n2)=O)CCC(C2CC2)(CNC(c2ccc(C)nn2)=O)C1 c1(C(=O)NCC2N(C(C(CSC)(C)C)=O)CCC2)ccc(O)nc1Cl n1(CC)ncc(C(=O)N(C(C)CN(C)C(c2ccccn2)=O)C)c1Br c1(NCC2CC(NC(C(C)(O)c3ccccn3)=O)C2)ccc2nnnn2n1 N1(C(CCOCCCOC)=O)CC(O)CC1CNC(c1ccncc1N(C)C)=O CCCCCCCCCC(=O)N(C)CC1CCN(C(c2cnn(C)c2F)=O)C1 C1(C(=O)NC(C2CCOC2)CNC(CCCOC)=O)CC2C(C1)C2(F)F N1(C(c2c(OC)ccc(OC)c2)=O)CCC2(NC(=O)C=CC3CC3)CCCCC12 N1(C(CCOCCN(C)C)=O)CCOCCC1C(=O)NC12CC=CC(C1)OC2 C1(CN(C)C(=O)NCC2CCCC2CN)CCCC1(C)C C1(O)(CN(C(=O)CCCn2cncn2)C)CN(C(=O)CC2CC(N(C)C)C2)C1 C(CCC)(CCCNC(c1nccc(F)c1Cl)=O)NC(C(C)OCCC=C)=O CC(C)CCCCC(=O)N(CC(C)N(C)C(c1ccsc1C)=O)C c1(C(=O)OCC(c2ccc(C(=O)OC)s2)=O)ccc(S(N)(=O)=O)c(Cl)c1 C(C(=O)N=c1ccn(CC(N)=O)[nH]1)=CC.C12CC(CCO1)C(=O)N2 C12(CNC(C3CCSCC3)=O)CCCCC1N(C(C1(CO)CCCO1)=O)CCC2 C12(CNC(C3CCN(C(C)=O)CC3)=O)CCC(CC1)N(C(=O)CC1C=CCC1)C2 N1(C(=O)NCC#CC)CC(C)S(=O)C(C)C1 C(=O)(C(CC)OC)NC(C(=O)N(C(C=C)C1CC1)C)C1CCC1 N1(C(C2CCN(CC)C2)=O)CC2(C)CN(C(C3CCCCC3(F)F)=O)CC2(C)C1 CC(=O)CCCCC(=O)N1CC(C(=O)NCc2nc(C)cc(O)n2)C2(CC2)C1 c1(C(C(=O)NCCc2occ(C)n2)F)ccc(F)c(Cl)c1 N1(C(C#CC2(CC)COC2)=O)CC2CN(C(C3CCS3(=O)=O)=O)CC(C1)O2 C1(NC(C2C(C)(COC)C2)=O)CCN(C(c2cc(-c3ccccc3)co2)=O)CC1 C(c1ccc(Cl)cc1F)=CC(=O)N(CC(C)NC(C1(COCC)CCCC1)=O)C c1(C(=O)NC(CC=C)CNC(C2CCCC2c2nc[nH]n2)=O)cnnc(O)c1 c1(C(N2CCCC3(NC(c4cc(C)on4)=O)C(C2)C3)=O)cccc(P(C)(C)=O)c1 CN1CCN(CCOCBr)CC1.c12ccc(cc1)NCC2C1CC1 Cc1ccc(C(=O)N(CCCNC(=O)COCC2CCCO2)C)cn1 Cc1cc(O)nc(C)c1C(N1CCCC(N(C)C(c2ccc(CO)o2)=O)CC1)=O C(CCCCCCCCNC(c1nnnn1C1CCOCC1)(C)CSC)OC c1(NC(C)(CNC(=O)C=CCF)Cn2cccn2)ncnc2cc(Br)ccc12 N1(C(=O)C2CC2)CC2CN(C(=O)Cc3cc(O)nc(O)n3)CC2C1.CO O=S(=O)(c1cccc(=NCC2CCCCC23OCCO3)[nH]1)N1CCC(NS(=O)(C)(C)C)C1 C1(C(=O)Nc2cc(F)c(OC)c(F)c2)CCCC1N=c1[nH]cnc2cnccc12 C1(C(=O)NCC(C)(C)C2CC2)(COC)C=CCN1C(C1CCCN1C)=O c1(C(C(=O)NC)N(C2CCC(=O)NC2=O)C)ccc(Br)nc1Cl CC1(C)CC(C(=O)NC2CCCSC2)CN(C(c2cc[nH]n2)=O)C1 CCC(C)(C)C(=O)NC1(CCNC(c2cn(CC)nc2-c2ccc(Cl)s2)=O)CC1 C1(C(=O)NC2(CC)CCCC2)CN(C(=O)CN2CCC(F)CC2)CCC1(F)F Cc1[nH]c2ccccc2c1C(N1CCCCC(NC(C2CCCC(=O)O2)=O)C1)=O NS(=O)(=O)CCCCC(=O)N1CCCCC1CC(F)(F)CO c1(C(=O)NC(CC(=O)N(CC)Cc2ncc[nH]2)COC)ccc(C)c(F)c1 C(=O)(CCS(N)(=O)=O)NCCOC1CC(NC(C23CC(OC)C2C3)=O)C1 C(C#CC(=O)NOCC=CCl)NC(C(C(C)(C)C)O)=O c1(C(=O)NCC2CN(C(c3nc(OC)oc3)=O)C2)sc2nc(C)nc(N)c2c1C C1(NC(c2cc(CCC)[nH]n2)=O)CC2CC(C1)N(C(=O)CSCC)C2 c1(C(=O)NCC(CN(C(=O)Cn2cccc(N)c2=O)C)O)ccc(C#N)cn1 N1(C(C(F)=CC)=O)CCOCC(F)(CNC(=O)C(F)(F)C(O)CC)C1 c1(NC(=O)NC(CSCCCC)C)nc2ccc(S(C)(=O)=O)cc2s1 c1(C(N2C(C(C)NC(c3ccc(C)cc3)=O)CCC2)=O)cc2sccc2cn1 c1(OC)cnc(C(=O)NC2C=CCN(C(c3csc(C4CC4)n3)=O)C2)cn1 Cc1nc(=NC2CCN(C(c3cc4nn[nH]c4cc3F)=O)C(C)C2)s[nH]1 c1(NC(C(COC(C)C)N)=O)ccc2c(cnn2CO)c1 C1(CC(=O)NC(COCC)C(=O)NCC2CC(C)(C)C2)CCCC(=O)N1 c1(C(=O)NC2CC(C(=O)NCC(C)OC)C2)cc(C)c([N+](=O)[O-])cc1C CC(C)C(C(C)NC(=O)C1=CSCS1)NC(c1ccc(OCC(F)(F)F)o1)=O c12ccc(o1)C2NCC=CC(C)(C)C.c1(CSC)nnnn1C1COC1 N1(C(c2nnc(C)s2)=O)CCC2CCN(C(c3sccc3C)=O)CC2C1 C1(NC(COCCOC)=O)CN(C(c2cccc(Cl)c2C)=O)CC2CC12 c1(C(=O)NC2C(F)CCN(C(C3(CO)CC(C)(C)C3)=O)C2)ccn2cnnc2c1 C(=O)(C1=NOC(C2(O)COC2)C1)NC(CC=C)CNC(c1ncccn1)=O CCCC(C)CC(=O)N1CCOCC1(C)c1cn(Cc2ccoc2C(=O)OC)nn1 Cn1ncc2c(C(=O)NC3COCC3NC(=O)C(=O)NCC(F)F)cnc(O)c12 C(CC(=O)N1CC(C)(O)CO1)N(C(=O)CC1CC=CCC1)C(C1CCC1)=O c1(C(C)NC(C2CC(NCc3ccn(C)c(=O)c3)C2)=O)cccc2ncoc12 C12(N(C)C)CCC1CN(C(C1COCCN(Cc3ccc(F)c(Br)c3)C1)=O)C2 N1(C(CSCC=C)=O)CCN(C)CC1C(=O)N(C)Cc1ncc[nH]1 c1(OCCOC)ccc(C(=O)NCC2CCCCC2NC(=O)C(C)(F)CC)cn1 C1(C2CCN(C)CC2)(C(=O)NCC2C(NC(c3ccc(OC)nn3)=O)C2)CC1 C1(c2c(OC)cccc2)CN(C(=O)CC2CNC(=O)C2)CCN1C(C)=O C12(CNC(c3c(OC)nsc3)=O)CCCCC1N(C(c1ccc(CO)o1)=O)CC2 c1(C(N(c2ccccc2)C(Cc2nc(C)on2)=O)=O)cc(N(C)C)ccc1[N+](=O)[O-] c1(C(N2CC(CNC(CC3CC(OCC)C3)=O)C2)=O)c(C)nn(C2CCC2)c1C CC1(CNC(c2cn[nH]c2)=O)CCC(NC(c2c(Br)noc2C2CC2)=O)CC1 c1(CC)cc(OCC2CC2)ncc1F.C1(NCc2ccccc2)CN2CC1O2 N1(C(C=C(C)c2ccco2)=O)CCN(C(c2csc(=N)[nH]2)=O)C(CF)C1 c1(CC)nocc1C(=O)NCCN(C(=O)CCNC(=O)C(C)(C)C)CC(C)O C(C(C)(C)CNC(=O)COCc1cccnc1)N(C)C(c1ccncn1)=O Cc1cc(C(=O)N(CCCCCC(=O)NCCC2CC(C)(C)CO2)C)cnc1C CCCCC(F)C(=O)NCCC1(C(=O)NCC2=NOCC2)CCC1 N1(C(CCSCC)=O)CCCCCC1C(=O)N(C)Cc1cncnc1 C(=O)(C1=C(Cl)CCCC1)NC(CNC(c1cc(C)c(F)nc1)=O)C(C)(C)C N1(C(Cc2cn(CC)nc2)=O)CCC(C2CC(NC(=O)C(O)C(C)CC)C2)CC1 C1(NC(c2coc(C3CC3)n2)=O)CCC12CCCN(C(=O)C=CC1CCOC1)C2 c1(OC)cncnc1C(=O)NCC1(NC(=O)C(C)c2ccco2)CC1 CC1C=C(C(=O)N2CCC(C(C)(C)NC(c3csc(Cl)c3)=O)C2)CC1 c1(C(=O)NCC(C)(CO)NC(C2C(CC)C2)=O)nccc2cc[nH]c12 c1(OC)ccc(CCC(=O)NCCn2cnc(C)c2C)cc1N C1(CCCC)CN(C(C2CC2C)=O)CCN1C(=O)COCc1cccc(Cl)c1 c1(C(=O)NC(C2(O)CCN(C(C(CC=C)(F)F)=O)CC2)C)ncnc2c1CCC2 Cc1ccc(N)cc1C(N1CCN(C(c2ccc(=O)n(C)c2)=O)C(CCO)C1)=O CCCC(C(=O)OC)NC(C1CCCN1C(=O)Nc1ccc(SC)cc1)=O N1(C(C(C)N(C)Cc2ccccc2)=O)CCC2(CCN(C(=O)CC(F)(F)F)C2)C1 c1(CC)nc(C)n(C)c1C(=O)NCC1CC(OC)CN1C(c1cc(CC)[nH]n1)=O CC1CC(C(=O)Nc2cccc(CF)c2)CCN1C(C1CC1C)=O C(=O)(C1Cc2ccccc21)NCC(C)CNC(=O)Cn1cnnc1 CC1(C)C(=O)CC1C(N1CC(O)CC1C(=O)NCCOC(=N)O)=O N1(C(C2N(CC)CC2)=O)CCCCC1CCC1CCCN1C(=O)CC1(C)CC1 C1(NC(c2c(C)nn(C)c2Cl)=O)CN(C(c2ccn(C)c2)=O)CC2CCCC12 c1(C(=O)NC(CNC(c2cc(C)nn2C2CC2)=O)C2CC2)n[nH]c2c1CCC2 c1(C(=O)NCC2CC(F)CN2C(c2ccsc2)=O)ncnc2[nH]cnc12 CCC(CS(C)(=O)=O)NC(c1cc(OC)ccc1C(C)C)C c1(-c2c(C(N3CC(F)(CNC(C(CC)OC)=O)C3)=O)c[nH]n2)ccccc1F N1(C(c2c(C)coc2C)=O)CC(C)(C)CC1CC(=O)NCc1c(C)n[nH]c1C N1(C(=O)Cc2cc3ccccc3s2)CCC(C2CCCNCC2)CC1 Cc1cc(CNC(C23CC(NCc4ccc(C)o4)(C2)C3)=O)cc(C)c1 c1(C(=O)NCCCCCN(C(C2(OCC)CCC2)=O)C)cc(C)nnc1O Cc1ccc(C)c(C(=O)NCCC2CCN(C(C3CC(=C4CC4)C3)=O)CC2)c1N c1(C(N2CC(CCO)(NC(=O)C(c3cccc(F)c3)O)C2)=O)cnccc1Cl C12(CNC(C3(CC)CN(C(c4c(CC)n(C)cc4)=O)C3)=O)COC(C1)C(O)C2 N(C(=NCCc1c(Cl)cccc1Cl)NCC(F)F)C(COC)C1CC1 CCCCC(F)(F)C(=O)NCC(F)CNC(=O)CCNC(=O)CO C1(NC(C2(C)CC2(F)F)=O)CCC2(CC1)CN(C(=O)Cc1n[nH]cc1Br)C2 C1(NC(c2c(C)ocn2)=O)CC(CNC(c2cc(C(C)(C)C)on2)=O)C1(C)C c1(C2N(CC(=C)C(C)(C)C)CCC2)ccc(F)cc1OC c1(CCOCCCN(C)C2CC2)cn(CCC(=O)Nc2c[nH]c(C(=O)O)c2)nn1 N1(c2nnc(C)o2)CCC2(CCC(NC(=O)C(C)Sc3nncn3C)CC2)CC1 c1(C(N(CCOCCNC(C(C)(C2(C)CC2)OC)=O)C)=O)cc(=O)n(C)cn1 c1(CO)cccc(N)c1.C12(CCCC1)CC(=O)NCCN(CC)C2=O CCC(CNC(=O)CNCC1CCCCO1)(CC)NC(=O)CNc1cccnc1 CC(C)CC(C(=O)NC1CCC(C)(CNC(=O)CN2CC=CC2)CC1)N(C)C c1(CC)cc(C(N2CCN(c3nc(C)cc(C)n3)CC2)=O)ccc1F n1(CC(CC(=O)OC)C)c(-c2cccc(CO)c2)csc1=Nc1ccnc(Cl)c1 C1(C(CNC(c2cnc(C)o2)=O)F)CCN(C(=O)CC2C=NN(C)C2=O)CC1 Cc1ccc(C(=O)NCCC2(NC(C3CCC(C)(C)O3)=O)CCOCC2)c(F)c1 c1(CC(N2CC(C(=O)Nc3c(C)csc3)C2)=O)cc(F)ccc1F N1(C(C(C)SCC)=O)CCC2(CC1)CC(CNC(c1c[nH]c(C(F)(F)F)c1)=O)C2 C1(NC(c2ccc(OC(C)C)nn2)=O)C2CCN(C(=O)CC(C)(C)O)CCC12 C1(CC)CN(C(=O)CCc2nncs2)CC1NC(c1sccc1F)=O Cc1ccc(F)cc1C(=O)NCC1CC(NC(C2(C)CCOC2C)=O)C1 CC(CO)C(=O)NCC1(C(=O)N(C)C(C)C2CC2)CC1 c1(SC)ncc(C(=O)NC2(CCNC(=O)C3=CCC3)CCCC2)n1C N1(C(C2(C(C)C)CC2)=O)CCCC(C(C)(C)OC(F)F)C1.N12CC(C1)C2=O C(=O)(C1CCc2c[nH]nc21)NCc1occ(C(=O)NCCCc2ccccc2)c1 c1(C(=O)NC(CNC(C=CC=CC)=O)CC(F)(F)F)cc(S(N)(=O)=O)co1 c1(C(=O)NC(CCNC(c2cc(C(C)=O)oc2C)=O)C)cc2c(cn1)CCCC2 c1(NC(C(N(C)C(C2CCCSC2)=O)C2CC2)=O)ccc2ccoc2c1 N1(C(C(CC=CC)C)=O)CC(NC(c2ccncc2)=O)CC(C(=O)O)C1 c1(C(=O)NC2CCCC(NC(c3sc(CC)c(C)c3)=O)C2)cnc2[nH]cncc1-2 N1(C(c2c(C)cc(C)s2)=O)CCCN(C(=O)CC2SC(=N)NC2=O)C(C)C1 C(=O)(C1=NOC(C)(C)C1)N(CC(C)NC(C12COCC(C1)C2)=O)C N1(C(C=CC(C)C)=O)CC2CC(N)CC1C2.C1(C(C=CC=O)=O)CCC(C)C(C)C1 c1(CC(=O)Nc2cn(C)c(C(=O)NCc3ccc(Cl)cc3)c2)ccc(Cl)cc1Cl c1(C(=O)NC2C3(CN(C(C4C(CCC)C4)=O)C3)CC2)cnc2ccccc2n1 N1(C(CC(=O)NCC#C)=O)CCN(C(=O)C(S(C)(=O)=O)C2CC2)CC1CCO c1(CC(=O)N(CCN(C(C)C)C(c2cscn2)=O)C)cn2cc(F)ccc2n1 O=C(C#CC1CCCOC1)NCC1(F)CN(C(C2(F)CCOC2)=O)C1 C1(NC(c2cccc(C(CC)(C)C)c2)=O)CC(F)CN(C(=O)C(C)NC(N)=O)C1 C1(C(F)(F)F)(C(=O)NCCN(C(C2C(C)CCCC2)=O)C2CC2)CCCCCC1 n1(CCC(=O)OC)cnc(C(=O)NCCCC(c2ccccc2)NC(=O)CO)n1 N1(C(C(CC)C#N)=O)CCCCC(NC(=O)CNC(c2csc(Br)n2)=O)C1 C1(C(N2C(C(C)NC(c3c(C)n[nH]c3)=O)CCC2)=O)CCCN(S(N)(=O)=O)C1 C1(C)(C(=O)OCC)CCN(C(C2(CCNC(c3ccsn3)=O)CCC2)=O)C1 CCC(CCC(=O)N1CC(C)C1(C)C)NC(=O)CCOCC1CCC1 S(=O)(=O)(C1CCOCC1)N(C(COC)=O)C(C1CCNCC12CC2)C c1(C(=O)NCC(=C)CCNC(=O)Cc2nonc2C)c(C)nn2c1CCCC2 c1(C(=O)NCCOCCNC(c2cc(C)on2)=O)nn(C)c2c1CSCC2 C(=O)(CC(C)(C)CC(F)F)NCC(CNC(C1(C)ON=C(C)C1)=O)C(F)(F)F c1(C(N2CC(C(C)(C)O)(CNC(COCC=C)=O)C2)=O)cc(C)c(C)[nH]1 N1(CC(=O)NC(CNC(C2(NC(C)C)CC2)=O)C2CC2)CCCNS1(=O)=O C1(CNC(Cn2c(C)ccn2)=O)CN(C(=O)CC(C)C2CCCC2)CCO1 N1(C(c2ccc(SC)o2)=O)CCC(C(N2CC(F)CC2CO)=O)C12CCC2 C12(CCNC(c3cc(CC)[nH]n3)=O)CCC1CN(C(=O)Cc1ccccc1C)C2 C1(CNC(C=C(C)C)=O)CCN(C(=O)CC2CSC2)CC1C c1(NCc2cc(OC)nn2C)nc2cccc(CO)c2[nH]c1=NC1CC(F)(F)C1 C1(C(=O)NC(CCOC)CNC(=O)CN2CC(C)(C)C2)CSCC(=O)N1 C(=O)(C#CC1CCCCC1)N1CC(C(NOCCOC)=O)N(C)CC1 N1(C(CCc2c(C)cccc2)=O)CCCN(C(=O)CC#N)C(c2ccccc2)C1 C1(CN(C(C(COCC)O)=O)CC)CCN(C(=O)C2=CCSC2)CC1 C1(C(=O)Nc2ccsn2)C=CCN(C(=O)COC2CCCOC2)C1 c1(C(C)(F)F)cccc(C(N2CCCC(NC(c3cnn(C(F)F)c3)=O)C2)=O)c1 c1(CN(C(C(C2CN(C(C=CC(CC)C)=O)C2)OC)=O)C)nc(C)ns1 c1(CNC(C(c2cn(C)nn2)NC(C(C)NC(=O)NC)=O)=O)scc(C)c1C C1(C(N2CC(N(C(=O)CCc3cscn3)C)C3(C2)CC3)=O)CCC2(CCC2)CO1 C1(COC(c2ncc(C)nc2)=O)CN(C(=O)COc2ccsn2)CC1(C)C c1(C(N(C2CCCC(NC(=O)CCC=CBr)C2)C)=O)cnn2c1CCC2 CS(=O)(=O)C(CNC(c1ccc(F)cc1Cl)=O)CNC(C12CC1CNC2=O)=O C1(CC(=O)N(CCCC)CCCO)CC(F)CN1C(C12CSCC1C2)=O c1(C(=O)NCC2(OCC)CN(C(=O)C(C3CC3)OC)C2)cc(C)c(Cl)s1 S(=O)(=O)(c1cc(Br)c(F)cc1Cl)NC(c1cc(Cl)cs1)=O c1(C(N2CCC(CC=C)(NC(=O)C(C)(C)n3cccn3)C2)=O)cc(N)c(Cl)c(O)c1 c1(CC)ncc(Br)cc1NC(C1CC(O)CN1C(=O)Cc1ccccc1Br)=O c1(C(=O)NC2CC(CNC(c3n(C)nc(C)c3Cl)=O)C2)cnc2c[nH]nc2c1 c1(CC(=O)NC)cn(CC(C)(C)CCC(=O)O)nn1.C1(=O)C(C)(C)N1C(=O)OC C#Cc1cccc(C(=O)NC2CC(C)N(C(C3CCCCC(F)(F)C3)=O)C2)c1F c1(C(N2CC(CCCCNC(C3C(C(C)O)C3)=O)C2)=O)cnc2sccn12 C1(C(=O)NC2(C)CN(C(c3c(CC)nns3)=O)C2)CS(=O)(=O)CC12CCC2 c1(C(N(CCN(C(c2cc(C)c(F)nc2)=O)C(C)C)C)=O)ccn2ncnc2c1 C(=O)(C(C)(CO)NC(=O)COCC(F)F)NC1CCN(C(C)C(N)=O)C1 C1(C(N2CC(CN(C(c3c(C)nc(CCC)s3)=O)C)C2)=O)COC2COCC12 CC(C)(CNC(c1ccon1)=O)CC(=O)NC(c1nc[nH]n1)CO CC1CC=C(C(=O)NC2COCC2CN(C)C)CC1.c12cc(c[nH]1)NC2=O C1(OC)CC(NC(=O)CCc2ccncc2)CN(C(c2cc(C)cc(Cl)c2)=O)C1 CC1CC(=O)NC1C(=O)NCC1(CNC(c2[nH]ncc2C#N)=O)CC1 c1(C(=O)NCCC(C)(C)NC(c2cn(C3CC3)cn2)=O)csc(C#N)c1 C(=O)(CC(C)(C)C)N(C1CN(C(C23COC(CC4CCCCCC4)(C2)C3)=O)C1)C c1(C(=O)NCC2(C)N(C(c3cnc(CCC)s3)=O)CCC2)c(F)ccc(N)c1F C1(C(=O)NCC(=O)NCC=C)CCN(C(C2CCC2OC)=O)C12CCC2 C1(COC)CN(C(c2cnc(C)nc2C)=O)CCN1C(c1cccc(F)c1F)=O C(CCCCC(=O)NCC(C)CNC(C1(S(N)(=O)=O)CC1)=O)OC(C)C C12(C(=O)OC)CCC(OC)C1C2.C12(CCC1)C(=O)NC1CC(C1)NC(=O)N2 c1(C(=O)N)ccc(OC)c(Cl)c1.C(=O)(C(F)NC(=O)NC1CC(OC)C1)OCC C1(NC(C2(OCC)CCSCC2)=O)CN(C(=O)CCN(C)C(C)=O)CC1C1CC1 C1(C(=O)NCC2N(C(CSCC#C)=O)CC=C2)CN2CCN1CC2 C1(CNC(CCc2cc(C)no2)=O)CCN(C(c2cn(C)nc2Br)=O)CC1C c1(C(=O)NC(CN(C(CC(CCC)O)=O)CC)C)cnn(C)c1S(C)(=O)=O C1(C(=O)NCC2(NC(C(C)C3CCOC3)=O)CC2)CCOCC1C N1(C(C(CCC=C)(C)C)=O)CCC2CN(C(C3NC(=O)OC3(C)C)=O)CC2C1 C1(NC(c2ccoc2Cl)=O)C2CN(C(C3CC(CCO)C3)=O)CC12 C1(CC(=O)NCC2(CS(C)(=O)=O)CC2)CSCCO1 N1(C(C(C)Sc2ccccc2F)=O)CCC2CCC(NC(=O)C=CS(C)=O)C1C2 CC1(C)C(NC(c2ccc(C3CC3)o2)=O)CC1C(N1CCC(CCF)CC1)=O C1(CNC(CSCC(C)C)=O)CC12CCN(C(=O)Cc1cnoc1)CC2 c12cc3c(cc1CNC(=O)C(=O)N2)OCCO3.N1(S(C)(=O)=O)CCOC(O)C1 N1(C(c2[nH]c(=NCC)sc2)=O)CC2CN(C(=O)C(CO)NC(N)=O)CC2C1 c1(C(N(CCC(C)NC(=O)CCSC(F)(F)F)C)=O)cn(C)c2ccc(F)cc12 N1(C(C2C(OCC)C2C)=O)CC2CC(NC(c3sc(C(C)C)nc3C)=O)CC1C2 C1(NC(COC2CN(C(c3cc(C)oc3C)=O)C2)=O)Cc2nn[nH]c2C(C)C1 n1(CC)nc(C)c(CC(N2CCC(CCNC(c3nnc(C)s3)=O)C2)=O)c1C c1(CNC(C2(CC)CCN(C(c3coc(C(N)=O)c3)=O)C2)=O)c(C)nn(C)c1C c1(C(=O)N(c2ccsn2)CC(C)N(C(CC)=O)C)c(C)sc2ccc(F)cc12 C1(NC(c2ncnc(C)c2C)=O)CN(C(C2CCC2)=O)C2(CCOC2)C1 N1(CC(=O)NC2CC(NC(CC(=O)NCC#C)=O)C2)CCSC2CCCCC12 Cn1c(=O)ccc2c(NC(c3cnc(Cl)nc3C)=O)cccc12 c1(C(=O)NCCCC(C)(C)NC(C(C)SC(C)C)=O)ccc(=N)[nH]c1Cl c1(C(N2CC(C)N(c3ccnc4cc[nH]c34)CC2)=O)cccc2c1nnn2C c1(CN(C)Cc2ncc3ccccn23)c(C#N)ccc(Br)c1F c1(NC(C2CC3CC3N2C(c2c(Br)ccnc2Cl)=O)=O)cccc(S(=O)(=O)O)c1 N1(C(C(C(C)C)OC)=O)CCC2(CC1)CN(C(=O)CCCCCSC)C2C(C)C CC#CCCCC(=O)N1CCOC(CNC(=O)C(C)Oc2cc(F)cc(F)c2)C1 C1CN=C(NCCC2CCN(C)C2)NCC1.c1(O)ccc(Cl)c(F)c1.CC(C)O Cc1nc2c(s1)CN(C(c1cc(C(F)F)[nH]n1)=O)C2.C1(=O)CCC(C(C)C)N1 c1(C(=O)NCC(C2CCN(C(CCC(C)SC)=O)CC2)F)cc(N)c(Cl)cc1C C1(C(=O)NCC=CC(=O)CCOC2COC2)CCCCN1C(=O)C=Cc1ccco1 c1(CC)cc[nH]c1C(=O)N(C)CC=CC(=O)NC(C)COC(F)(F)F c1(C(=O)NC2CCC(F)(CNC(=O)C(F)Cl)C2)ccc2c(c1)OCCO2 C1(C(N(C(CC)CNC(=O)C(C)Cn2cccn2)C)=O)CCCCC1(C)C c1(C(N(CCCN(C)CC2CCCCC2)C2CCC2)=O)n[nH]c2ccc(Br)cc12 c1(C(=O)NCC(C)(CNC(=O)C(C)Cn2ccnc2)OC)c(C)ccnc1O c1(NC(=O)NCCN(CCCO)CCC)cnnc(C2CC2)c1 C#CC1(C(=O)Nc2ccc(O)c(F)c2)CCN(C(=O)CC2(CSC)CC2)C1 C(=O)(C1=CN2CCS(=O)(=O)N=C2C=C1)NC1CCN(C(CC(C)(C)C)=O)CC1O c1(C(N(C2CC(NC(C(C3CCC3)OC)=O)C2)C)=O)ccc2nccn2c1 c1(C(=O)NCC(F)CNC(C2CC=CCC2)=O)ccc(O)cc1Cl C(=O)(CCCCC(F)F)NCCN(C(C1C(C(=C)C)OCC1)=O)CC Cc1c(C(=O)NC2CN(C(=O)C=Cc3cc[nH]c3)CC2C)cc(F)cc1Br C1(C)(SC2CC2c2cc(C)oc2C)CCC(NC(=O)CC2(C)CN(OC)C2)CC1 C1(NC(C2(C)CCCC2)=O)CC2CCC(C1)N2C(C1(F)CCCC1)=O C12C=CC(C1)CC(=O)N2.C1(CN(C(C2(CC#C)CC2)=O)C)CCOC1 C(=O)(C1CNC(=O)c2ccnn21)NCCN(C(c1cc(C)c(C)[nH]1)=O)C c1(CC)ccc(C(=O)N(C)CCNC(C2CC(OC(F)F)C2)=O)c(C)c1 c1(C(=O)NC(C(=O)NC(CCOC)C)c2ccoc2)ncncc1Cl c1(C(=O)NC2CN(C(COC(C)=O)=O)CC2O)cc2c(C)ccc(F)c2[nH]1 Cc1n[nH]cc1CCNC(c1nnnn1C1COC1)(C1CCOC1)C C1(CC=C)CCCN(C(=O)CCCC2(NC(C3(F)CC=CCC3)=O)CCC2)C1 O=C(CS(=O)(=O)CCO)NC12CC1CN(C(c1ccnn1C1CC1)=O)C2 C1(NC(CC(=O)NC)=O)CC1C1CCN(C(c2ccc(NC)cc2F)=O)CC1 c1(NC(Cn2cnc(OC3CCC(C)CC3)n2)=O)c(Cl)ccnc1Br N1(C(c2ncc(P(C)(C)=O)cn2)=O)Cc2c(O)n[nH]c2C(F)(F)C1 Cc1ccc(CC(=O)NCC2(C(N)=O)CN(C(=O)CC3CC3CO)C2)cc1 C1(CC)(CC)CCCN(C(=O)C(C)(C)CNC(=O)C(CO)OC)C1 C(CCSC)(C(=O)NCC1(OCC)CC1)NC(C=CCCC)=O CCCC(CC)CCC(=O)NCC(C)(CC)NC(c1ccc(F)c(F)c1N)=O c1(C(=O)NC(C(C)NC(CC(=O)NCC#C)=O)(C)C)ccc(C2=CCCC2)cc1 c1(C2CN(C(C34N(C(CCN(C)CC)=O)CCC3C4)=O)C2)ccc(C)c(C)n1 N1(C(c2c(C)nn[nH]2)=O)CCC(NC(c2cc(=N)[nH]c(=N)[nH]2)=O)CC1C c1(OCCC(=O)NC2CC(CCNC(C(C)O)=O)C2)cccc(Cl)c1Cl Cc1nc(C)c(F)c(=NCC(C)NC(=O)C2CCOc3c(F)cccc32)[nH]1 C(=O)(CCCCCN=[N+]=[N-])N(CC(=O)N(CC#C)C)C c1(CNCC=Cc2ccc(F)cc2F)ccc2c(ccn2C)c1 C1(=O)C(C(CC)CC)NC(CCC)NC(=O)C(F)CC2CN1C2.c1(C)ccco1 C1(NC(c2ccc(N(OCC)CC)cc2O)=O)CC2CC(C1)N(C(=O)CSC)C2 C(=O)(C#CC1(C)CCCO1)N1CCN(C(c2ccc(C(C)=O)s2)=O)CC(O)C1 c1(OC)cccc(OC)c1C(CC(=O)NCC1CCCN(C(=O)OC)C1)(C)N(C)C N1(C(Cc2nc(C)sc2)=O)CCC(NC(c2cc(C(F)(F)F)n[nH]2)=O)C(CO)CC1 Cc1cc(N2CC(O)(CCNC(c3cnn(CC(C)C)c3C)=O)C2)c(C#N)cn1 Clc1cnc(CNC(c2nnnn2CSc2ccccc2)c2nncs2)s1 CCC(O)C(=O)N1CC(OCCNC(=O)CCn2cnc(=N)[nH]2)C1 C(C1CN(C(c2c(C#N)cnn2C)=O)CC1C(N1CC2C(C1)C2(C)C)=O)=CC c1(C(N2CCCCC(CNC(c3c(C)scn3)=O)C2)=O)csc2c1CCCC2 CS(=O)c1cccc(OCC(C(=O)CC(C(F)(F)F)OC(F)(F)F)=O)c1.OCC c1(CC(C)(C)N2CCCC2)nc(-c2cccc(SC(C)(C)C)c2)nn1C1CCC1 Cn1cc([N+](=O)[O-])c(C(=O)NC2CCC(F)(CNC(=O)C(F)CC3CCC3)C2)n1 N1(C(CC2C(C)(C)OCC2)=O)CC(NC(c2cscc2Cl)=O)CC1(C)C N1(c2c(OC)cnc(Cl)n2)CCC(NC(=O)Cc2cccnc2C)CC(C)(C)C1 Cc1ccc(CC(=O)NCCC2(C(=O)NC3CCCSC3)CCC2)o1 C1(CCNC(CCC)=O)(OCC)CN(C(=O)CNS(=O)(=O)NC)C1 N12CCC(C)N(CC1)C(=O)c1cc(N)ccc1C2=O.C1(OC)CNC(=O)C1 c1(C(N2C(C(=O)NCC3CCCC(OC)C3)CCC2)=O)cc(C)cc(O)c1 CCC(CCN)C(=O)NCC(c1cnc[nH]1)C c1(C(Cc2cn(CC(C(C)(C)C)ON)nn2)(O)C2CC2)cc(F)c(F)cc1 C1(NC(C(CNC(c2cc(COC)[nH]n2)=O)N(C)C)=O)CCCC(OC)C1 c1(NC(CC(C)(C)C)CCc2ccccc2)cccc2nc(C(F)F)sc12 N1(C(c2n(CC#C)ccc2)=O)CC(NC(C2(C3CCCCO3)CCC2)=O)CC1C c1(C(N2CCC(N(C)C(c3cccc4cncn34)=O)C2)=O)ccc([N+](=O)[O-])cc1Cl c1(C(N(CCCNC(C(C=CC)O)=O)CC)=O)c(C)nsc1N c1(OC)ncccc1CNC(=O)C(C)(C1CCC1)NC(=O)CCOCC(C)C CCCC(C)(O)C(=O)NCc1cc(O)nc(CNC(=O)CC23COC(C)(C2)C3)n1 c1(C(N2CCC(C3(NC(C(C=C)O)=O)CC3)C2)=O)cccc2cc(O)ccc12 C(=O)(C#CC1CCC1)NC(C1(O)CN(C(c2csc(-c3ccco3)n2)=O)C1)C CC1(C)CC(C(=O)NC(c2cccnc2)C(=O)NCCOC2CCC2)CCO1 N1(NCC2CC(OCC)C2)CCCC1C1CCCCN1C(=O)OC(C)(C)C c1(CC)cc([N+](=O)[O-])ccc1C(=O)NC(C)CN(C)C(C1(F)CCCOC1)=O C#CCC(C)(C(=O)NC1COC2(CCC2)C1)NC(c1ccn(C)c1C)=O n1(CC(=C)Br)c(N(C)CCC2NC(=O)NC2=O)nnc1C(C)(C)F Nc1cc2c(cc1C(=O)NCCN(C(=O)CCF)Cc1ccccc1)CCC2 C(=O)(C1=CCS(=O)(=O)C1)NC(CNC(c1ccc(C)nc1CO)=O)(C)C1CC1 N#Cc1nc[nH]c1C(N1CCCCC1C1(C(N2CCC(O)CC2)=O)CC1)=O c1(C(N2C(CNC(CC(CC)SC)=O)CC2)=O)ccc(OC(C)C)cc1F C12(CNC(c3cc(C)c(C)nn3)=O)CCC(CN(C(=O)Cc3cncnc3)C1)C2 CC1(C)C2CC(C(=O)NCCCC3CCN(C(=O)CNCC(F)(F)F)CC3)CC12 c1(NC(N2CCC(Oc3cccnc3)CC2)=O)nc2ccc(F)cc2s1 c1(OC)ccc(Cl)c(C(=O)NC(C)CN2CCN(C(=O)C(C)OC(C)=O)CC2)c1 C1(NC(COCCC)=O)(CO)CCN(C(=O)C(c2ccc(COC)cc2)C)CC1 C(C)(CCCCNC(c1cc(C(C)C)[nH]n1)=O)NC(CNC(CNC(C)=O)=O)=O C1(CC(=O)NCCC2CCCN2C(C2COCCO2)=O)CCCC2(CCC2)O1 c1(NC(C2(C)CCN(S(CC)(=O)=O)C2)=O)cccc2nsnc12 c1(C(N(C)CC2N(C(C3C(C=C)C3)=O)CCCC2)=O)cc(C(F)(F)F)cc(F)c1 N1(CC(=O)NCC2CC(O)(CNC(=O)CC3CC3)C2)CCCNS1(=O)=O C(C)(C)(CCC(=O)N(CCCNC(=O)CCCCc1ccccc1)CCO)OC C1(CCNC(CC(=C=C)C)=O)CN(C(=O)CC(C)(C)C#N)CCCO1 c1(OCC)cc(C(N2CC(CC(C)NC(C3(F)CC3C)=O)C2)=O)[nH]n1 CC12CN(C(C3CCCCO3)=O)CC1(C)CN(C(C1CC(n3ccnn3)C1)=O)C2 c1(C(N2C(CC)CN(C(C34CC(F)(C3)C4)=O)CC2)=O)sc([N+](=O)[O-])cc1Cl c1(CNC(c2ccc(NC(C3CCC(=O)NC3)=O)cc2)C)cc(Cl)ccc1O c1(C(=O)NC2C(NC(C(C(C)C)O)=O)C2)cccc(S(=O)(=O)CCO)c1 n1(CC(C)N(C(=O)CC2CCN2C(=O)CCC2CCCC2)C2CC2)ccnc1 N1(C(CN2CCN(C(=O)CSc3nc[nH]n3)CC2)=O)CC(C(=O)O)CC12CCC2 N1(C(C2C3CN(C(CC(C(=C)C)OCC)=O)CC32)=O)CCN2C(=O)CCC2C1 C1(CC(=O)NCC(C2CC2)NC(c2ncoc2Cc2cccs2)=O)COC2CC1C2 NC(=O)CCC(=O)N1CCN(C2CN(C(=O)CCC3CC3(F)F)C2)CC1 C(=O)(C(C(C)(C)C)C1CCCC1)NC(C1CN(C(C2(F)CC2)=O)C1)C C(=O)(C(C)(CO)NC(=O)CC1NC(=O)NC1=O)NCCOCCOC CC(C)C(C)(O)C(=O)NCCOC1CCN(C(C2COC(C)(C)C2)=O)CC1 S(=O)(=O)(CCC(=O)NCCC(O)CNC(=O)C(=O)NC(C)C)NCC c1(CC(=O)NC2(CF)CCN(C(C(C)OCC=C)=O)C2)noc2ccccc12 c1(OCCCNC(c2nncc(OCC)c2)=O)ccc2oc(=O)oc2c1 C1(C(=O)NCC(CNC(c2cc(C)c(C)s2)=O)CO)CC2CCCC2C1 C1(C(C)C)CN(C(c2cnnn2C)=O)CCN1C(c1ccc(C(=O)N(C)C)[nH]1)=O c1(C(N2CCN(C(CCC=C)=O)C(C3CC3)C2)=O)ccc2c(c1)nc(O)n2C C(=O)(C1=Cc2ccccc2C1)NC1(C)CC(NC(c2c(C)c(Cl)c(Cl)cc2)=O)C1 c1(-n2cc(C(C)NC(c3ccnc(C#N)c3)=O)nn2)ncc2n1CCCC2 Cc1nc(=NC2(CO)CCCN(C(C3CCCN3C(C)C)=O)C2)[nH]cc1C#N C(=O)(C1=CCC(NC(=O)Cc2cccc(C#N)c2)C1)NC(C)CCCCO CC(CCCN(C)C)N=c1[nH]n2cc(C3CC3)nc2s1 N1(C(C(CC)C)=O)CC2(C1)CN(C(C1CCC(CCC(=O)OC)O1)=O)C2 c1(C(=O)NCCN(C(C(C)CC2CCCO2)=O)C)cccc2nsnc12 N1(C(C2C(CC)CCCC2)=O)CC2CN(C(=O)Cc3cccc(C)c3)CC(C1)O2 C(CC(=O)NCCN1CCCC1=O)(C(F)F)NC(C1CC(n2ccnn2)C1)=O C1(N(C(CCc2c(C)nn(C)c2)=O)C)CN(C(=O)CC(C)NC(N)=O)CC12CC2 Cc1cnc2cc(C(=O)NCCN(C(=O)CCc3ncccn3)C)sc2c1 CP(C)(=O)c1ccc(C(=O)NCC2CCCC2NC(C2CCCCCC2)=O)o1 C1(NC(C2N(C(CC)=O)CCCC2)=O)CCN(c2nnc(C#N)s2)CC1(C)C c1(C(=O)NC2CCCN(C(c3c(C)ccc(C)n3)=O)C2)cccn2nnnc12 c1(C(N2CCN(OC3(C)CCC3)CC2CO)=O)ccc2c(c1)CNC2=O.C1C(=O)N1 C1(C(=O)NC(C(C)NC(CC2(C(=C)F)CCC2)=O)CO)CCN(C)C(=O)C1 C1(NC(CCCOC)=O)COCCN(C(=O)CC2CCCCCC2)C1 C=CC1CN(C(=O)COC2CCC2)CC1NC(c1csc(C)c1OC)=O c1(C(N2C3CCN(C(=O)CCOCCN(C)C)CC3C2)=O)c(F)ccc(Cl)c1F C1(C(=O)NCCC(C)NC(c2cn(CC3CC3)nn2)=O)CCCC1S(C)(=O)=O C1(C(=O)NC2(CNC(c3ccoc3C3CC3)=O)CC2)CCCCC1O c1(CNC2C(C(=O)Nc3ccc(C(=O)OC)o3)C2)nc(Cl)ccc1Cl CCC1=NOC(C(=O)NC2CCCCC2CC(=O)NN(C)CC2(CO)CCC2)C1 c1(N2CC(O)(CNC(C3CC(N=[N+]=[N-])C3)=O)C2)nc(Cl)nc2sccc12 C1(C(N(C(CN(C(c2c(CC)ocn2)=O)C)C)C)=O)CNC(=O)CC1(C)C C(=O)(C1NCCc2c(C)cccc21)c1nc(-c2c(Cl)cn(CC)n2)on1 c1(CCC(=O)N(CCCCN(C)C(C2CCC3CC23)=O)C)ccc(Br)c(F)c1 Cc1cc(Cl)c(C(=O)N(CCNC(c2cccc(O)c2Cl)=O)CC2CC2)cc1C N1(C(C2(CC)CN(C(C=C(CCC)C)=O)C2)=O)CC2C(C1)C2(C)C C(=O)(CC(C)(C)CNC(=O)CS(=O)CC)C1N(CC)CCNCC1 c1(OC)noc(C)c1C(=O)NCC(C)N(C)C(C1CCCS1)=O C(=O)(CCCCC(F)F)N(CCN(C(C(CC)N)=O)C)C c1(C(=O)NCC(CNC(C2CC3(CC(=C)C3)C2)=O)C)c(F)c(C)cc(N)c1F C(=O)(CCCS(C)(=O)=O)N(C1CCC(NC(c2c(CCC)nco2)=O)CC1)C C1(C(C(C)C)NC(C(N2CCCCC2)C)=O)CCN(C(=O)CCC2CCC2)CC1 C1(c2nnnn2C(C)C)(NCC=CCCOC)CC2CC(OC)CC12 c1(NC(C2CC3CC(C2)NC3)=O)cc(F)c(I)c(F)c1 C(C(CC(=O)N1CCC(OCCF)C1)NC(c1cc(C(C)=O)on1)=O)OC N1(C(c2cc(OC)nn2C)=O)CCC(NC(=O)CC(C)C(F)(F)F)C(F)(F)CC1 CC1(C)CN(C(c2cccc(CF)c2)=O)CC1CNC(C12CCC1CC2)=O Cc1cc(Cl)ccc1OCC(=O)NCC(CO)NC(c1csc([N+](=O)[O-])c1)=O N1(C(Cc2cnc(C)s2)=O)CC(NC(=O)C(C)Cc2ccco2)C2CCCC12 c1(C(C)NC(=O)Nc2ncc(Br)s2)cccc(O)n1 C12(NC(CCS(N)(=O)=O)=O)COCCC1CN(C(=O)C=Cc1ccoc1)C2 C(c1ccccn1)=CC(=O)NC1C(CNC(c2c(CCC)occ2)=O)C1 N1(C(CC(C)SC)=O)CCN(C(c2ccnnc2NC2CC2)=O)CC1C C1(C(N2CC(CCNC(C3COCC3C(N)=O)=O)(OC)C2)=O)CC2CC(=O)C1O2 C1(C(CNC(C2N(C(C)C)CCC2)=O)(C)C)CN(C(c2c[nH]c(=N)s2)=O)CCO1 Cc1coc(C(=O)N(CC(O)CNC(=O)C(F)(F)c2cncs2)C)c1 c1(C(=O)NCC(CNC(C2CCC2)=O)OC)cc(F)c(CC(N)=O)cc1N c1(C2C(C(=O)NCC3(CN(C)C(C4(C)CC4(C)C)=O)CC3)C2)cccc(Br)c1 C1(C(N2CCC(Cn3cnnn3)C2)C(=O)NCC2CCOC2)CC2CCC1CC2 N1(CC(=O)N(C2CCCN(C(C3CC3C(C)C)=O)C2)CC)CCC(C)CC1 Cc1ccc2cc(C(N3CC(CNC(=O)C(C)(F)F)N4CCC3C4)=O)cnc2c1 C1(C(=O)NC2(C(=O)NCC)CC2)(OC)CCN(C(=O)C(C)CC2CC2)C1 N12CC(C(F)C1)C(=O)NCC2=O.C12(CC)CC(C(=O)OC(C)(C)C)(C1)C2 c1(C(=O)NCC2(F)CC(CNC(c3ccncc3)=O)C2)ccc(Cl)cc1Cl N1(C(CCOCC#C)=O)CC(C(F)(F)F)C(CNC(=O)Cc2cncn2C)C1 C(CC(C)(C)C(=O)N1CCC(C(C)CNC(C2(C(F)F)CCCC2)=O)CC1)OC C1(F)(C(=O)NCCC2N(C(Cc3ccn(CC)n3)=O)CCSC2)C(C)(C)C1(C)C Cc1ccc2c(CC(N3CC(NC(c4ccnnc4O)=O)C3)=O)c[nH]c2c1 c1(OC)ncc(F)cc1C(=O)NC(C1CCN(C(c2ccccc2F)=O)C1)C N1(C(CNC=O)=O)CCCC2(CCCN2C(=O)CN2CC=CC2)C1 N1(C(Cc2c(C)cc(C)s2)=O)CC(C2CCCCN(C(c3cn(C)cn3)=O)C2)C1 CC1(CO)CC(O)CN1C(C1CCOCCN1C(=O)CC1CCC(O)C1)=O C1(C(=O)NCc2nccc(C)c2)CC(NC(C23CCC(C2)C3(C)C)=O)C12CCC2 CC1(C(=O)NC2CC2NC(=O)CSCCN(C)C)CCc2ccccc2C1 c1(NC(C2CC2C(=O)NCCF)=O)cc(F)cnc1Cl C1(CN2C(=O)CCC2)CCN(Cc2cc(Br)co2)CC1 Cc1nc(C(F)(F)F)oc1C(=O)NC(C1CCN(C(C2(S(N)(=O)=O)CC2)=O)C1)C N1(Cc2nc(CCC)on2)CC2CN(C(C3CCCNS3(=O)=O)=O)CC2C1 C1(NC(C=CC)=O)COC2(C1)CN(C(C1(n3cc(Br)c(C)n3)CC1)=O)C2 N1(C(Cn2cccc(C)c2=O)=O)C2CCC1CN(C(C1CC=CC(O)C1)=O)CC2 C1(CC)C(C(=O)NC(C)C(C)(C)C)CCCN1C(=O)CC1CC1CC C(=O)(C1CCNc2ccccc21)C(=O)C1=C(Cl)CC1.C12CCCN1C(=O)C21CC1 N1(C(C(C2CCN(C(CC(CCC)(C)O)=O)C2)C)=O)CCC2(COC(C)C2)C1 Cc1cc(F)cc(C)c1C(=O)NCC1(O)CCN(C(c2ccn(C(C)C)n2)=O)C1 N1(C(c2c(OC)csc2)=O)CCC(NC(c2ccnn2C(C)(C)C)=O)C(CO)C1 C1(C(=O)NCC2(CC)CC2)C(C)CN1C(=O)C(O)CSC C1(C(=O)OC)CCC(NS(=O)(=O)CC2(C)CNC2)CN1 N1(C(C(CC=C)C)=O)CCCC(C)(NC(c2ccc(C3CC3)s2)=O)C1 Cc1ccc(Br)c(C(=O)NCC(C)CNC(=O)CC2C(C)(C)C2(C)C)c1N c1(C(=O)NCC(C)N(C(=O)C=C2CCOCC2)CC)ccc(Br)nc1N C1(CC(=O)N(C)CC2CC2(F)F)C2CCCC2N1C(c1cc2occc2[nH]1)=O C1(C(N2CC(CC(=O)NC3CCn4cncc4C3)C2)=O)(OC)CC(C)CC(C)C1 CC1CC(NC(C2CC3C=CC2C3)=O)CN(C(=O)CCCC(F)F)C1 C1(C(=O)NCCCN(C(C2CC2F)=O)C2CC2)(COC)CCC(=O)N1 c1(C(=O)NC2(CC=CC(=O)NCCCP(C)(C)=O)CCC2)cnn2c1OCC2 c1(C(=O)NC(c2cn(-c3cccnc3)nn2)(C)C)nn2cccnc2c1Br C1(C(CC=C(C)C)C(=O)O)CC(C)CN(C(=O)OC(C)(C)C)C1 c1(C(=O)NCC(CC)NC(=O)CCc2nccs2)ccn2c1CCCC2 C(C(C)CN=c1[nH]c(=NCc2ncnn2C2CC2)c2c(F)cccc2[nH]1)OCC c1(CNC(=O)C(=O)Nc2cc(C3(O)COC3)on2)ccc2cccnc2n1 C1(C(=O)NC2CC(CC(=O)NCC3CCC(C)(C)C3)C2)NC(=O)OC1(C)C C1(C(C)(O)CNC(c2ccc(F)cc2)=O)CCN(C(=O)C=CCOC)CC1 C1(C(N2CC(O)(C(C)NC(c3cn(C)cn3)=O)C2)=O)CCCC1S(C)(=O)=O C1(CC(N2C(C(C)NC(=O)CSC(=N)N)CCC2)=O)CCCCN1C C1(CNC(c2c(C)coc2C(C)C)=O)CN(C(=O)C(O)CN(C)C)CC1(F)F Cc1cc(F)cc(C(=O)NCC2CCN(C(=O)CC3CNC(=O)O3)C2(C)C)c1N N1(C(C=C(C)C(F)F)=O)CCN(C(C2CCN(CCS(C)(=O)=O)C2)=O)CC(C)(C)C1 C1(NC(Cc2c(C)ocn2)=O)C=CCC(C(=O)NN2CC=CC2(C)CO)C1 C(C1CCCC1)=CCN.C1(CC(C)C)(C(=O)NCC(=O)N)CCC1 N#CC1CCCN(C(=O)CCCNC(c2csnc2Cl)=O)C1 c1(CC(=O)NCC(CN(C(c2cnn(C3CC3)c2)=O)CC)(C)C)c(C)cccc1C N1(C(C(CSC)C)=O)CC2N(C(C34CC5CC3C4C5)=O)CCC2(C)C1 c1(C(=O)OCC(=O)Nc2c(C(=O)OCC)scc2C)cn2cc(C)c(C)cc2n1 CCCCCCC(C)C(=O)NCC1CCC(NC(C2CCC(=O)C(C)C2)=O)C1 C(=O)(C#CC1CCCCC1)N1C(CNC(c2nc(C)n(C)c2O)=O)C(O)C(O)C1 C(=O)(C(O)C(C)CC)NCC(CN(C(c1c(CC)n(C)nc1)=O)C)(C)C C(C(C)(C)C(=O)NCCO)CC.C1(C)(C(N(CCOC)C)=O)CCCC1O c1(C(=O)NC(CC)CNC(c2cnn(C)c2C2CC2)=O)cc2c(s1)CN(C)CC2 C12(CNC(=O)Cn3cccn3)CC(NC(C3(c4cccnc4Cl)CC3)=O)(CCO1)C2 n1(CC)nc(C(=O)NCC23CC2CN(C(=O)C(O)CN2CCOCC2)C3)cc1C c1(C(N2CC(NC(=O)CCCN3C(=O)CNC3=O)C3C2C3)=O)ccn2ccsc12 N1(C(CC2(C)CC2)=O)CCC2(CC1)CC(NC(=O)Cn1ccc([N+](=O)[O-])n1)CO2 C12(CNC(c3c(CC)csc3)=O)CC(NC(=O)C(COC)N(C)C)(CO1)C2 C=CCC(C)(CC)C(=O)NC(C)(C)CN1CCN(C(=O)C(C)(C)C(C)(C)O)CC1 C(=O)(C#CC1CCCCC1)NC(COC)C(=O)N1CC(C)(C)C1 C1(N(C(c2c(C)cc(C)o2)=O)C)CCN(C(c2cnccc2C(F)F)=O)CC1C CCCC(CCCO)C(=O)N1CCOCC1CNC(C12CC(CO)(C1)C2)=O C12(NC(CC3(CSC)CC3)=O)CC1CN(C(c1ccc(=O)oc1)=O)C2 c1(C(N2C(C)C(NC(c3ncccc3Cl)=O)CCC2)=O)cc(F)cc2c1CCC2 C12(NC(CC(C)(C)C(F)F)=O)CCCC1N(C(=O)CSc1ncccn1)CCC2 N1(C(C(C)O)=O)C2CCC1CC(CNC(c1cncn1-c1ccnnc1)=O)C2 C=C(C)CCCC(=O)NC(C)(CNC(=O)C(C)C=Cc1ccccc1)C1CC1 N1(CCNC(CN(c2ccccn2)C(C(C2CCOCC2)C)=O)=O)CCCOC1=O Cc1nn(Cc2cccs2)c(Cl)c1CNC(c1ccco1)C1CCC1 N1(C(CCc2scc(C)n2)=O)CCOC2(CCCN(C(c3coc(Cl)c3)=O)C2)C1 c1(C(N2CCC(C3N(C(CC(C)C)=O)CC3(C)C)CC2)=O)cc2sccc2n1C N1(C(C2CN(C(C)C)C2)=O)CC2CCC1CN2C(C12CCC(CC1)C(C)O2)=O c1(NC(C2(C(C)C)CN(C(C3CCCOC3C)=O)C2)=O)cc(S(N)(=O)=O)c[nH]1 C1(OC)C(NC(=O)C(C(C)C)NC(=O)C(O)Cn2cccn2)CC12CCC2 c1(OC(C)C(=O)N(C2CCN(C(=O)CNC=O)C2)CCO)ccccc1Cl Cc1ccncc1CC(=O)N(CCC(C(C)C)NC(c1ncc[nH]c1=O)=O)C c1(C(C(=O)NC2CCN(C(=O)CN3CCCC3)C2)(F)F)ccccc1Cl c1(CC)cc(C(N2CC(CNC(C3CCC(SCC(F)(F)F)C3)=O)C2)=O)no1 c1(C(=O)NCCC2(NC(C3OCCC(C)C3)=O)CC2)cc(F)c(C(F)F)c(F)c1 C1(c2n(CC)nnn2)(NCc2[nH]nnc2C)CCCC(c2cnn(C)c2)C1 N1(C(C=CC(C)C)=O)CCCC(N(C)C(C2CCOC2C)=O)CC1 O=S(=O)(c1cccnc1NCCS(=O)(=O)CCO)N1CCC(C(F)F)C1 C(=O)(C1=C(SC)CCCC1)NC1CCN(C(C=CC(CC)C)=O)C1 c1(CN(C2CCCC(C)C2)CCCOCC)noc2c1COCC2 c1(C(N2CC(CO)C3(CCC3)C2)C(=O)NCCCOC)ccc2c(c1)CCC2 C1(C(C(=O)NCCC)N(C2CCCOC2)C2CC2)C2CCCCC12 N1(C(c2nn[nH]n2)C)CCC(O)(CC2CC2)C1 C1(C(=O)NCCCOCCN(C(C)=O)C)CCC(CC(N)=O)CC1CCC c1(C(=O)NCCC2CCN(C(C(CC)O)=O)C2)cc(F)cc2[nH]ccc12 C(c1csc(C(F)(F)F)c1)=CC(=O)NCCCC1(NC(=O)CC2CC=CC2)CC1 N1(C(C(C)C)=O)CC(NC(=O)COCc2nccn2C)C(C(F)F)C1 C1(=O)CC(C)(C)CCN1.c1(CN(C)C)cc(-c2ccco2)on1.N12CC(C1)C2=O N1(C(=O)OC(C)(C)C)CC(NC(=O)NCC2CC=CCC2)COCC1(C)C C1(C(N(C2CCCCC2)CCNC(=O)COCCO)=O)CCC12CCCO2 c1(C(=O)NC(CC(C)C)CNC(=O)C(=O)NCCC(N)=O)ccc2sncc2c1 C1(C2(NC(c3c(SC)nn[nH]3)=O)CC2)CCCCN1C(=O)C=CCN1CCC1 c1(NC(C2CN(Cc3cc(OC)cc(Cl)c3)C2)=O)cc(C)c(OC)cc1Br CCCCCCCCCC(=O)N1CCC(CNC(c2c(C)cc(C)oc2=O)=O)C1 C=CC1(C(=O)NC(c2ncn(CCN3CCOCC3C)c2)=O)CCCC1.C(CSCC)N C1(NC(CCCCC#C)=O)CCCOC12CCN(C(C1CCC(C)CC1)=O)CC2 N1(C(C2N=C(C)SC2)=O)CC2CCCN(C(c3ncc(C(F)(F)F)s3)=O)C2C1 CC1CN(C(=O)COC2CCCOC2)CC(C)N(C(=O)CSCCC(F)(F)F)C1 c1(C(N(C)CC2(O)CN(C(C3(C(C)C)CCC3)=O)C2)=O)cc(O)c2ccsc2c1 c1(C(=O)NC2CCC(CNC(C3(C(F)(F)F)CC3)=O)C2)cc2n(n1)CCO2 n1(CC(=O)N(CC(C)NC(=O)CCc2ccccn2)C)ccc2ccccc12 C1(N(C)C(C2CC2c2cnc[nH]2)=O)CCCN(C(c2cscn2)=O)C1 S(=O)(=O)(c1ccc(Cl)cc1F)N1CC(C)(C(=O)Nc2ccc(C)c(F)c2)C1 c1(-c2nc(CC(C)OC)nn2C2CCC(C)(C)C2)occ2c1CCOC2 c1(OC)cscc1C(N1CC(OCCC(=O)NCCC2CCCC2)C1)=O c1(CN2CCC(NC(=O)NCc3ccc(Br)cc3Cl)CC2)c(Cl)cnc(Cl)c1Cl C1(C(C(=O)NC2CC(N(C)C)C2)N(C2CCCCC2)C)C2CC3CC(C2)CC1C3 c1(CC(=O)NC2(CCNC(C(C)(C)C3CCCO3)=O)CC2)cccc(F)c1 c1(OC)ccccc1C(=O)NC(C)C(C1CCCCC1)NC(c1cc(Cl)no1)=O C(CCC(C)(C)CO)n1cc(N(C(C(C)=NOCC#N)=O)C)nn1 c1(C(N2CCC(O)(CNC(C(c3cnccn3)C)=O)C2)=O)c(N)cccc1Cl C1(NC(Cc2nc(C)oc2)=O)CC2CC1N(C(c1cnc(C(F)(F)F)cn1)=O)C2 C1(C(CNC(CCC)=O)NC(=O)C=CC(=O)NCC)CCCCC1 CCCC(C(O)C(=O)NCCOC(=O)CCC1CCCCC1)NC(=O)OC CC1CCC(CN(C(C2(C#N)CCCCC2)=O)CC)CN1C(=O)CC1CC2CC2C1 Cn1cnc2sc(C(=O)NC3CN(C(=O)CCC4CC4)CCC3F)cc12 C1(C(N2CCCC2)C)CCCN(N2CCC3CNC(=O)C23)C1 c1(C(=O)NC23CCN(C(CC4(C=C)CCC4)=O)CC2C3)cncc2c[nH]nc12 CC(CCN=c1[nH]c(N2CCN(CCN(C)C3CC3)CC2)nc(=N)[nH]1)P(C)(C)=O C=CCC(CNC(=O)C=Cc1ccc[nH]1)C(=O)N1CC(C(C)CC)C1 CC1(C2CCN(C(C3(NC(C4CC5(CCO4)CC5)=O)CC3(C)C)=O)C2)CC1 c1(C(C)C)cc(C(=O)NCc2cc(C(N3CC(C4CCCO4)C3)=O)co2)n[nH]1 C(=O)(CN=c1cc[nH]cc1)N1CC(CCCCC(N2CCC2C)=O)C1.C=CCC=O Cc1cc[nH]c(=N)c1C(=O)N(C)CC1CCCN1C(=O)CC1CCCCCC1 N1(C(C(COCC)C)=O)CCN(CC2CN(C(=O)CC3C(=O)ON=C3C)C2)CC1 c1(C(N2CC(OC)(CNC(=O)CN3CCCC3C)C2)=O)cn(C)c(O)n1 C1(c2nnnn2C2CCCC2)(NCC2NC(=O)NC(=O)C2)COC2(CCC2)C1 C(N=c1nc(N(C)Cc2cnccc2C)c2c([nH]1)c(C)nn2C)C1CC(COC)C1 CCC(C)(CC(=O)N(C)CCOCCNC(=O)Cc1cncnc1O)C(=O)OC n1(CC)ccnc1C(=O)NC(C)C(C)NC(=O)C(C1CCC1)OC c1(C(N(C2CCN(C(c3ccc(SC)o3)=O)C2)CC)=O)cc(C2CC2)ccc1Cl C1(C(=O)NC(CSC2(C)CNC2)=O)CC2(C1)CN(Cc1c(F)cccc1F)C2 C1(CNC(CCC#C)=O)CCCCN(C(C2CCN2CC)=O)CC1 C(=O)(C(F)(F)C(C)(C)C)N1CCC(CNC(c2ccc(OC)c(Cl)c2)=O)C(C)C1 c1(C(=O)NCC(CCCC)NC(=O)CCS(C)(=O)=O)cc2cc(OC)ccc2o1 c1(C(N2CCN(CC3CN(C(C(F)=CC)=O)C3)CC2)=O)cc2occc2s1 C(=O)(C1CCCc2nncn21)NC(C(C)(C)C)CNC(=O)COC(F)(F)F CC(C(=O)N1CC(CNC(=O)CCOCC(F)F)C1)CS(C)(=O)=O c1(C(N(C)CCC2CCCCN2C(C2CC(C)(F)C2)=O)=O)n[nH]c2c1CCC2 c1(C(C)OC)nc(Cl)cc(=NCc2ncc(C)s2)[nH]1 N1(C(c2c(C)snc2)=O)CCCC(N(c2ncccn2)C)C1 C1(C(N(CCCNC(c2c(C)nc(O)cc2)=O)C)=O)CC2(C1)C(F)(F)C21CCC1 n1(CC(=O)NC2C(C)CN(C(c3cnc(O)s3)=O)C2)cccc(O)c1=O C1(C(=O)NCCCOC)(N(C(c2c(C(=O)OC)[nH]nn2)=O)C)CCC(C)C1 C(C(C)(C)C#CC(=O)NC(C)CCCCCO)NC(CC(C)N(C)C)=O n1(CC(=O)NC(CC)C(N)=O)ccc(C)cc1=O.N12CCCCC1C2 c1(NC2C(CO)CCN(C(C(C)OC)=O)C2)ncnc2scnc12 c1(OC)ccccc1OCCCC(=O)NCC1CC1NC(=O)C(O)C1CC1 C1(C(=O)NCC2CC(NC(=O)COCCc3ccc(Cl)s3)C2)CC2CCC(C1)O2 C1(C(=O)NC2C(NC(=O)CCc3cccnc3)CCC2)CCc2ccnn2C1 CC1(C)CCCC(C(=O)NCCC2CCCN2C(=O)C(=O)NCCC(N)=O)CC1 CN1C(=O)OCC1C(N1CCC(C(=O)NCC2(CC3CC3)CCCCC2)C1)=O c1(C(=O)NCC(C2CCCN2C(=O)CCC2CCCC2)(C)C)cnncc1O C1(NC(CCCNC(C)=O)=O)CC2CC1N(C(c1cc(C)c(C)s1)=O)C2 N1(C(C2CC(NC(c3cnc(OC)s3)=O)C(O)C2)=O)CC(F)(F)C(F)(F)C1 C12(c3c(C)cccc3)CCN(CC1c1cccc(NC(=O)NCCC(C)C)c1)C2 C(=O)(C(CCC)N(C)C)NC1(CNC(CC2CC(CC)C2)=O)CCC1 C1(COC)C=CCN1C(c1c[nH]nc1CNC(c1ncn(C(C)C)n1)=O)=O C(=O)(C(C)(C)CC(=O)OCC)NCC1C(C)CCN(C(CC(CC)(C)C)=O)C1 C1(n2ccc(C3CC3)n2)(CNC(=O)C(=O)Nc2ccc(Cl)nn2)CCOCC1 C1(C(=O)NC(C2CN(C(C3CC3(Cl)Cl)=O)C2)C)CC(C)(C)OC(C)(C)C1 Cc1[nH]c(C(=O)NCC23CC(CO2)N(C(C2CCS(=O)(=O)C2)=O)C3)c(C)c1C C(=O)(C1CSc2ccccc21)NCCN(C(=O)C(O)Cc1ccccc1)CC C(CC(=O)NCC1OCC2CCC1C2)(C(C)(C)C)NC(C(C)n1cncn1)=O Cc1c(C(=O)NC(C)C(N2CCN(C(c3c[nH]ccc3=O)=O)CC2)=O)cnn1C Cc1ccccc1C(=O)NCC(=O)OC(=O)CNCC1(C)CCCC1C CCC(C)C(C(=O)NCC1(O)CC=CC1)NC(=O)C(O)CCSC C1(NC(C(C(C)O)C)=O)CCCC12CN(C(c1cc(C3CCCCC3)on1)=O)C2 C(=O)(CC(O)CNC(=O)C(F)C1CC(NC(=O)CC=C(C)C)C1)OC n1(CC)nccc1CNC(=O)Cn1cc[nH]c1=N.C12(CCCC1)CCC(=O)N2 c1(CC(N2CC3C(CNC(C(C=C)CC)=O)(C3)C2)=O)cccc(F)c1CC C(=O)(C(CCNC(c1cnc[nH]c1=N)=O)OC)N(CCCC)C C1(C)(NC(C2CCN(C(=O)NC)CC2)=O)CCCN(C(c2cnc(Cl)n2C)=O)C1 C1(C(=O)NC(C(=O)NCc2ccncc2)c2cccs2)CC(=O)C12CCC2 Cc1ccc(C#N)cc1NC(=O)C(=O)NCC1(C)Cc2ccccc2C1 Cc1c(F)ccc(N)c1C(N1CCCC(NC(C2(C)CCCCO2)=O)CC1)=O c1(CC(=O)NCC(CC=C)NC(c2ocnc2C)=O)ccc(Cl)c(C)c1 C1(NC(=O)C(=O)NC2COCC2n2ccnc2)CC(=O)N(Cc2ccccc2Cl)C1 c1(C(N2CCC(N(CCC)C(C3CCC3C)=O)C2)=O)cc(CO)n(C)n1 Cc1cc(OC(C)(C)C)cc(C)c1C(=O)N(C)CC1CCCC1C c1(C(=O)NCC2CCCN2C(c2c(Cl)n[nH]c2C2CC2)=O)ccccc1F C1(CNC(C(C)Cc2ccncc2)=O)CN(C(=O)CCF)CC2(CCC2)O1 C(CC(C)(C)CNC(=O)C(CNC(=O)CC12CCCC1C2)CC1CCC1)OC N1(CCOC)CC(C#N)C(F)(F)C1.c1(OC(F)F)cccc(N)c1OC c1(OCC(N2CCC(CNC(c3cnc(C)nc3)=O)CC2)=O)nc(O)nc(O)n1 Cc1cc(C(=O)NCC2CC2CC(N2CC(O)(C(N)=O)C2)=O)sn1 C1(OC)CC(NC(c2cnoc2C(C)C)=O)CN(C(=O)C(=C2CCCCC2)F)C1 C1(C(=O)NC2C3N(C(COC(C)=O)=O)CC(CC3)C2)Cc2cccc(F)c2O1 N1(C(c2ccc(C)nc2O)=O)CCC2CCN(C(c3cccc(CO)c3)=O)C2C1 c1(C(c2ccsc2)N(CCCOc2ccc(C)cc2)CC)ccc(Cl)cc1 N1(C(C2(C(=O)NC(C)(C)C)CC2)=O)CC(C)(NC(C(C)=CC)=O)C1 N1(C(C2(NC(c3c(C)cc(N)cn3)=O)CCC2)=O)CCN2CC(C)CC2C1 CC1(C)CC(NC(=O)Cc2cc(Cl)ccc2O)CN1C(C1C2CC3C(C2)C13)=O n1(CC(=O)NC2(CC(=O)NCCc3nc[nH]n3)CC2)cc(C(=O)C2CC2)nn1 N#CC1CC(CNC(=O)CNC(=O)CNC(=O)CCCn2ccnc2)C1 C1(CNC(CC(CC)C)=O)COCCN(C(C2CCC(N=[N+]=[N-])C2)=O)C1 C1(NC(C(C)(C)OC)=O)CS(=O)(=O)CC1N=c1ccc2c([nH]1)CCCC2=O C1(CC)CN(C(c2n[nH]c(C3CC3)n2)=O)CCC1NC(c1nn[nH]c1Cl)=O C(=O)(CCCC(CC)NC(=O)C(O)COC(C)C)N(CCCC)C C12(CC(=O)N(CCNC(CC3CCCC(OC)C3)=O)C)CCC(CC1)C2(C)C c1(C(=O)NC(C)(C)CC=CC(N2C3CSCC2C3)=O)cccn2ccnc12 Cc1sc(O)nc1C(=O)N(CC(C)C(=O)NCC(CC1CC1)CO)C C1(NC(C2N(C)CC(C)(C)C2)=O)CC2CCC1CC2NC(C1(C)CCCCO1)=O N1(C(C(C)NC=O)=O)CCCCCC1CNC(c1ccc(NC=O)cc1)=O CCC(CC(=O)N1CCC(Nc2ccccc2[N+](=O)[O-])CC1)CC(F)(F)F N1(C(C(C(C)C)F)=O)CC2(CCCC2)C1C(=O)NC(c1ccnc(F)c1)C S1(=O)(=O)c2ccc(C#N)c(c2)N1.C1CCN1CCC.C(CCN(C)C)N(C)C c1(CC(=O)NC(CNC(C2(CCCC)CCC2)=O)CO)cc(SCC)on1 N1(C(C23CC2C3)=O)CCc2ccccc2C1.c1(OC)cc(C)cc(C)n1 C1(C(N(CCCNC(c2cc(C3CCC3)[nH]n2)=O)CCC)=O)CCCN(C)C1 Cc1ccc(C(=O)NCCOC2CCN(C(c3cc(C)c(Cl)s3)=O)CC2)nc1F Cc1nsc2ncc(C(N3CCN(C(c4csnn4)=O)CC(CO)C3)=O)cc12 Cc1cncc(C)c1C(=O)NCC(C1CC1)N(C)C(C1CC(=O)N(C(C)C)C1)=O C(=O)(C(C)(C)CS(C)(=O)=O)N1CCC(O)(CNC)C1.C12COCCN1C2=O C(=O)(C=C1SCC(=O)N1C)N(CCCCN(C)C(C1CC2(C1)CC21CC1)=O)C c1(C(=O)NC(CC(C)C)CC(N2CCc3c[nH]nc3C2)=O)cccn2cncc12 CC1(C)CC(C)(NC(=O)C(c2ccns2)NC(CCCC)C2CC2)C1 C1(C#N)(CS(=O)(=O)NC)CN(C(C2COCCC2C)=O)C1 c1(C(N(C(c2ccccc2)C(=O)NCC(C)(C)OC)C)=O)ncccc1N c1(C(=O)NCC=C)cc(CNC(=O)C(C2(O)CCCC2)F)[nH]n1 N1(C(CCN(CC)CC)=O)CCN(C(=O)CC2OCCCC2(C)C)CC1CO c1(OC)ccccc1NC(C)C.c12nc(no1)COC2(C)C C1(CCC(=O)N(CC(=C)C)CC)CCCN(C(=O)C=Cc2cnn(C)c2)C1 CC1CN(C(C2(CNC(=O)C(c3cccc(F)c3)(C)C)CC2)=O)CC1C(N)=O CCS(=O)CC(=O)N1CCC(NC(C2C=C2C)=O)C1C C1(NC(C=CC(=O)OCC)=O)(CNC(c2ccncc2F)=O)CCCCC1C c1(C(=O)NCC2N(C(CN3CCC(C)C3)=O)CC(F)C2)ccc2oc(=O)oc2c1 C1(CCC(N2C(C3(NC(c4cc(C)[nH]n4)=O)CC3)CCC2)=O)NC(=O)NC1=O CCN=c1[nH]cc(C(N2CCC(O)(C(C)NC(C3CC(C(C)C)=NO3)=O)C2)=O)s1 N1(CC)C(=O)CCC1C(=O)N(C)CC1CCN(C(c2nn(C)cc2SC)=O)C1 C1(CC(=O)NC2C(OCC)CC2)CCCCC1NC(C1CC1(F)F)=O Cc1cccc(-n2cc(C3CN(CNC(C(=O)NC(=O)C4CC4)C(C)C)C3)nn2)c1F.O C1(CNC(C(C)NC(=O)NC2CCCC2)=O)CN(C(=O)CC2C=CCC2)CCO1 Cc1nnc2n1CCCC2C(=O)NCCC1CN(C(C2(F)CCOC2)=O)CCO1 C(=O)(CC1=CCCCC1)N1CCC(OCC(=O)NC(C=C)C(F)(F)F)C1 N1(C(C2CCCC(=O)N2)=O)CCC(NC(=O)CCn2cc(Cl)cn2)C12CCC2 C12(NC(C=COCC)=O)CCCCCC1N(C(c1cc3nc[nH]c3cn1)=O)CC2 c1(CCC(N2C(NC(CCOCC#C)=O)CC(OC)C2)=O)n[nH]c2c1CCCC2 C(C(O)CC(=O)C(=O)CCc1cnn(C)c1)N(C(C1(CCC)CC1)=O)C1CC1 N1(c2nc(C)c([N+](=O)[O-])cn2)CC2CCC1C1CN(C(C3(C)CCCC3)=O)CC21 C1(NC(c2cc(CC)ncc2)=O)CCC2(CC1)CCN(C(C1(O)CCOC1)=O)C2 N1(S(CC(C)c2ccccc2)(=O)=O)CCc2ccc(Br)cc2C1 N1(C(c2ccc(C#N)cn2)=O)C2CCC1CN(C(=O)CCc1nc[nH]n1)CC2 C1(CNC(CCNS(C)(=O)=O)=O)CC(C(=O)NCC23CCC(CC2)CC3)=NO1 Cc1cc(F)oc1C(N1CCC(C(C)C(=O)N(CC(O)CO)C)CC1)=O c1(NC(C2CN(C(COCCC)=O)CC2C)=O)ccc(OC(F)(F)Cl)cc1 C(CN=c1cccc(S(=O)(=O)NC(CO)CC(C)(C)C)[nH]1)c1cc(OC)nn1C N1(C(Cc2c(C)ncs2)=O)CC(CCNC(=O)Cc2cnoc2)OC(C)C1 c1(C(C)C)cccc(NCC2COCCO2)c1O C1(NC(C(COCC)NC(=O)CN(CC)CC)=O)CC(=O)N(C)C1 C1(CNC(c2n(CC)ncc2)=O)CC(F)(F)CN1C(c1cnc(CC(C)C)s1)=O N1(C(c2cnc(OCC)c(Cl)c2)=O)CC2CN(C(C3(OC)CCSC3)=O)CC2C1 c1(C(=O)NC(C2CCN(C(=O)CN3CC4CC4C3)C2)C)c[nH]c2cc(N)ccc12 C(=O)(C(C)C(CC)CC)N(C)Cc1cccc(SC(C=CC(=O)OCC)(C)C)c1 N1(C(CC2C(C)CCO2)=O)CCC(NC(c2occ3c2CCOC3)=O)C12CCC2 O=C(C#CC1CCOC1)NCC1CCCC1NC(c1ccccc1)=O C12(C(N3C(CNC(c4ccn(C(F)F)n4)=O)CC3)=O)CC(C1)C(C(F)(F)F)O2 C1(NC(Cc2cn(C)nn2)=O)CCN(C(c2ccc(O)cn2)=O)C1C(C)(C)C CCCCCCC(C)NC(=O)C(C1(C)CC1)NC(=O)COCCSC Cc1ncc(C=CC(=O)NCC(O)CNC(C2COCCC2c2ccccc2)=O)s1 c1(C(=O)NC2CCCC(C(N(CCCCC)CCO)=O)C2)ccc2n[nH]cc2c1 c1(OC)c(Cl)cc(C(N2CCCC2CN(C(=O)CSCCC(C)C)C)=O)nc1Cl c1(C(C(=O)NCC2CCCO2)N(C(c2ccccc2)C)C)csc2c(Br)cccc12 C(=O)(CCCCCn1cnnn1)N1C(C(C)NC(=O)CC2NC(=O)NC2=O)CCC1 C1(NC(c2cc(C)sc2)=O)CC2CN(C(C3CC4(C3)CC4(F)F)=O)CCN2C1=O c1(C(C)C)ncsc1C(=O)N(CC(C)(C)CNC(=O)CSC(F)(F)F)C CC1(C)CC(NC(C2C=CC(NC(C3COC(=O)N3)=O)C2)=O)CCO1 C1(CNC(=O)COCC2(F)CC2)CN(C(C2(C3CCCO3)CCC2)=O)CC12CC2 CC(CC(N)=O)C(=O)NCC1(C)CCCN1C(=O)CCc1nc(C2CC2)no1 Cc1cc(=O)n(CCC(N2CCC(CO)(NC(C3CCCC(=O)O3)=O)CC2)=O)cn1 Cn1c(CCC(=O)NC(C2CCN(C(C3CC4(F)CC3C4)=O)CC2)(C)C)nnc1S Cc1cc(C2CCCC2)ccc1C(=O)NNC(=O)NS(=O)(=O)CCCCl N1(C(C=CCOC)=O)CCC(C2CCCO2)(NC(=O)COC(F)F)CC1 CCC(CC)(C(N)=O)NC(C12CCC(NC(C3CC4(CCC4)C3)=O)(CC1)C2)=O C1(C(=O)NC(CC)C(=O)NCC2CC23CCOCC3)CC12CCCCC2 C1(CCOC(COCC(=O)OC(C)(C)C)=O)CCN(CC(=O)NCC(N)=O)CC1 CC1=NN(C)C(=O)C1CC(=O)NCC1(F)CCCN(C(C2COC(=O)N2)=O)C1 CC(CC(C)(C)C)C(=O)N(C1(C(=O)NCC2(C)CCC(O)CC2)CC1)C CC1CN(C(c2ccncc2)=O)CC(C)N(C(=O)C(=CC2CCCCC2)C#N)C1 C1(NC(CC(OCC)OCC)=O)CC2CCCC(C1)N2C(C1CCC1OC)=O CC1(C)CC(CNC(c2nc(Cl)sc2Cl)=O)N(c2ccnc(CO)n2)C1 CC1(n2ccnn2)CCN(C(N2CC3C(C(N)=O)C3C2)=O)C1.C1(O)CC2(CC2)CO1 C(C(C)(C)C(=O)OCC)(c1nnnn1C(C)(C)C)NCCOC.c12cnn(C)c1C2 Cc1ccc(C(=O)NC2(C(N3CC(O)CCC3C)=O)CCOCC2)cc1C C1(C(C)(C)C)(CNC(c2cnc(C3CCC3)[nH]2)=O)CCN(C(c2ccsn2)=O)C1 N1(C(C(CNC(CCOCC(C)(C)C)=O)CO)=O)CC2(CNC(=O)OC2)C1 c1(N(C)C)cc(C(=O)NC2CC2CNC(=O)C(=O)NCc2ccccc2)ccn1 c1(CC)ccc(C(=O)NC2(C(=O)NC(c3ccccc3F)C)CC2C)nc1 c1(OC(C(=O)N(CCNC(C2CC(OC)C2)=O)C)C)ccccc1Cl N1(C(C(CC2CC2)NC(=O)CC(F)(F)F)=O)CCC2(CCCCC2)C1 C1(O)(CCNC(C2C(=C)C2)=O)CCCN(C(=O)CC2(C)CCOCC2)C1 n1(CCOC)c(SCC(=O)Nc2cccc(N)c2)nnc1-c1ccc(C)o1 C1(C2(O)CN(C(=O)CCCc3nc(CC)no3)C2)(CNC(C(C=C)(C)O)=O)CC1 c1(C(N(C2CN(C(=O)CC3COC(C)(C)CO3)C2)C)=O)cccc2cc[nH]c12 N1(C(COC)=O)CCN(C(c2nc(OC)sc2N)=O)C(c2ccc(SC)cc2)C1 c1(C(=O)Nc2c(C(=O)NCC(C)OC)n[nH]c2)ccc2cc[nH]c2c1 C(=O)(CC(O)CNC(=O)CCn1cc(Cl)cn1)NCC(C)NC(=O)OC(C)(C)C c1(C(=O)NC2C(NC(C(C)(O)CCc3ccccc3)=O)C2)cnc2c[nH]nc2c1 c1(C(=O)NCC2CN(C(CC3CN(C)C3)=O)CC2O)ncccc1S(C)(=O)=O C(CCCCC(=O)NC(C)(C)CNC(c1cc(C)ccc1C)=O)SC Cc1cc(C(N2CC3CC(NC(c4cn(C)cn4)=O)C2C3)=O)c2c(C)n[nH]c2n1 Cn1ncc(C(N2CC3=C(C2)CN(C(C2CC(O)C2)=O)C3)=O)c1S(N)(=O)=O N1(C(CC(CC)NC(=O)Cc2cnsc2)=O)CC2CC=CC1C2 N1(C(c2c(O)ccc(SC)c2)=O)C2CCC1CC(NC(C1(CC(C)C)CC1)=O)C2 c1(N(C(COC(CC)=O)=O)Cc2nn[nH]n2)nscc1C Cc1cnc(C(C)NC(=O)C(=O)NCCC2CCSC2)o1 C(=O)(C(C1CCC1)CC1CC1)N(CC(=O)N(C)CC1CC1(C)C)C c1(C(N2C(CNC(C3CCC3c3nc[nH]n3)=O)CC(F)C2)=O)cc(Cl)nnc1O C1(NC(C2(COCC)CC2)=O)(CF)CCN(C(C2C=CC2)=O)C1.C(=O)OC CCCCCCC(=O)NCC1CCC1NC(C1(OC(C)=O)CC1)=O C(N=c1[nH]c(=NC2CCCS(=O)(=O)C2)c2c(ncn2C)[nH]1)C1OCC(C)OC1 CC(C)CCC(C)NC(C1(C)C=CCN1C(=O)C1=NOCC1)=O N#Cc1cc(F)cc(C#N)c1NCc1noc(C(F)F)n1 N1(C(CCCOCCC)=O)CCC(C(=O)NC2CCOC2(C)C)C(C)C1 N1(C(CN(C(=O)CNC(=O)CC(C)C)CC#C)=O)CCC2(CCCO2)CC1 S(=O)(=O)(c1c[nH]c2nccc(Cl)c12)NC(Cc1cccc(C)c1)C(=O)O CC(C)(CC(F)C(=O)NCC1CCC2(CC2)CO1)NC(c1cccnc1)=O N1(CCCCC(C)C)CCC(=O)N(CC2CC3C=CC2CC3)C1=O Cc1cc(C2CC2)cnc1C(=O)NCCC(C)N(C)C(c1ccc(Cl)cc1C)=O C1(CNC(CC(C)C2CC2)=O)CCN(C(=O)Cc2cccc(C(F)F)c2)CC1O CC1(C)CCN(C(c2cc3ncccc3s2)=O)CC1NC(C1CSCCS1)=O C1(C(N(C(C)CCNC(=O)CC2CCC2)C)=O)CN(S(=O)(=O)N(C)C)CCO1 Nc1cc(Cl)ccc1C(=O)NS(=O)(=O)C(C)c1ccccc1 c1(OCC)nccc(C(=O)N(C)CCNC(c2cc(CC3CC3)[nH]n2)=O)n1 C(=O)(C(C)C(C)C)NCCN(C(C1CCCCN1C)=O)CC CC1(C)CCC(C(=O)NC(C2CCN(C(c3cc(C#N)cs3)=O)C2)(C)C)OC1 C12(NC(c3ccc4ccccc4c3)=O)CCCC1N(C(=O)CCOC1CC1)CCC2 N1(C(C)=O)CCCC2(CNC3(C(=O)OC)CCOCC3)CC2C1 CCCC(C)CC(=O)NCC1CCN(C(c2cc(C(F)F)ccc2C)=O)CC1 C1(COC)(NC(C2Cc3nccn3C2)=O)CCCN(C(c2c(C)cnn2C)=O)C1 c1(NCCc2nc(=N)[nH][nH]2)nc(N2CCN(C3CCOC3)CC2)nc2sccc12 C1(NC(c2cc(C(=O)OC)oc2C)=O)C(C)CN(C(=O)C2CC2)CC1C CCCCC(CC)C(=O)N1CC(OCCNC(=O)CCc2c(Cl)cncc2Cl)C1 C(CNC(c1c[nH]nc1CNC(C1CC(=O)C1(C)C)=O)=O)(C(C)(C)C)OC C1(NC(c2c(C)ocn2)=O)CC2(C(=O)NCCCc3ccsc3)COC1C2 C1(CN(C)C(C2C(C#N)C2(C)C)=O)CN(C(C2CCC2)=O)CC12CC2 c1(CC)cc(N)c(C(=O)NCC2CCC2NC(=O)C(O)CC(N)=O)cc1F C1(CN(C(=O)CCC2CCCCC2)C)CC(F)CN1C(C1CC=CCO1)=O c1(C(N2CCC(C(C(C)C)NC(=O)C(C)C(F)F)CC2)=O)nccc2cc[nH]c12 CC1(C(=O)N(CCNC(c2cnc(S)nc2)=O)C2CC2)CCCOC1 C#CCC(O)C(=O)NCCN(C1CCCCC1)C(c1cc(Cl)no1)=O C1(NC(CNC(C)=O)=O)CCN(C(c2cc(C3CC3)cnc2Cl)=O)CC1CO N1(C(=O)NCC2(C)CCC2)CC(CO)(CO)C1(F)F C(=O)(C1=CCCCC1C)N1CC(O)(CNC(C2CC(C)=C(C)CC2)=O)C1 c1(C(N2CCCC(CCNC(c3nn[nH]c3Cl)=O)C2)=O)cc2cc(F)ccc2[nH]1 N1(C(C(C=C=C)C)=O)CC(N(C)C(c2cc(O)ncn2)=O)C2(CC2)C1 C=CC(C)(C)CC(=O)N(C1CCCC1)CC=C.C(=O)(C(C(C)C)N(CC)CC=CCl)N C(=O)(N=c1[nH][nH]c(C)c1Br)c1c(OC)ccs1.N12C(CC3CC13)C2=O C1(C(N(C)CCOCCNC(C2CC(c3ccccc3)C2)=O)=O)CCN(C)C1=O C1(NC(=O)CC2CC2)CN(C(c2nn[nH]c2Cl)=O)CCC1C(F)(F)F C(N=c1[nH]nc(C(F)(F)F)s1)C1CCCN(C(C(C)(C)C2(O)CCOC2)=O)C1 C12(NC(C3CN(C)C(=O)CC3)=O)CCC(NC(=O)COCCOCCO)(CC1)OC2 c1(C(=O)NC(C2N(C(CC(C=C)C)=O)CCC2)C)ccc2c(c1)CCNC2=O n1(CC(=O)NCC2N(C(C(C)CC3CCC3)=O)CC2)sc(=O)c2ccccc12 N1(C(=O)CC2CCOCC2)CCCC(C2CCN(C(C3(O)COC3)=O)C2)C1 C12(C(N(CCCNC(CC=C)=O)CC)=O)CCC(CC1)CO2 CC1CCN(C(=O)CCC(C)(C)F)C(CNC(C2OCCC2(C)C)=O)C1 S(=O)(=O)(c1ccncc1)NC(C1CCCN(Cc2cc(OC)cc(Cl)c2)C1)C N1(C(CONC(C2C(CN(C)C)CCC2)=O)=O)CCC(O)C(C)(O)C1 CC(C)CCCC(C)C(=O)N1CCC(O)(CCNC(=O)CSCC(N)=O)C1 c1(C(N2CC3C(CNC(c4ccn(C)c4)=O)(C3)C2)=O)ccc(Cl)c(Cl)c1 c1(C(=O)NCC(CN(C(c2cc(C(C)C)no2)=O)C)O)cc(Cl)ccc1F Cc1csc(=NCC(=O)NC(C2CCCCN2C(C2CCN(C)CC2)=O)C)[nH]1 C(=O)(N=c1ccn(CC)[nH]1)OC1(CCF)CCN(C(C(CC)(C)CC2CC2)=O)C1 CCC(CC)C(F)C(=O)N(C)CC1CN(C(C2(C#N)CCC2)=O)CCO1 c1(C(=O)NCC(C2CCC2)NC(c2cc(C(N)=O)oc2)=O)ccc2nncn2c1 c1(C(N2C(CCNC(=O)CCCCC3CC3)CCC2)=O)cccc2c1OCCO2 N1(C(C(CCC)=CCC)=O)CCC2CCN(C(=O)Cc3ncncc3Cl)CC12 C1(C(=O)NCC(CNC(c2n(C(C)C)ncc2Cl)=O)F)OCCN(C)C1=O C12(C(N(C(C)CNC(=O)CCNC(c3cccs3)=O)C)=O)CC(C)(C1)C2 C(=O)(CCCC(=O)N(CCC(=O)NC1CCCNC1=O)C(C)C)NCC C1(CC(=O)NCC2CC(C)(C)C2)CCCCCN1C(C1CCCOCC1)=O Cc1ccc(NC(C2CCC(C)N2Cc2[nH]c(C)nc2C)=O)c(C)c1 c1(C(C)C)nnc2n1CC(NC(=NCCCN(C)C)NC1CSC1)CC2 c1(C(N(C2CN(C(=O)CCOCC3CCCO3)C2)C)=O)cccn2nncc12 Cc1oc(-c2ccccc2)nc1CN(S)NCC(CCO)N(C)C C(=O)(C1=C(CCl)N(CCOC)C(=S)NC1c1nc[nH]c2ncnc1-2)OCC N1(C(C=CC=CC)=O)CC2(CCN(C(c3csc(N4CCCC4)n3)=O)C2)C1 C1(CCC(=O)NC(C(=O)N(CCCN(C)C)C)C2CCOC2)CCC(=O)C1 CC1=C(C)CC(C)(C(=O)NCCC2CN(C(c3c[nH]c(C#N)c3)=O)C2)CC1 N1(C(c2c(C)scn2)=O)CCN(C(C2(C)CCOCC2)=O)CC1C1CC1 C1(O)(CN(C(c2c(CCCC)ocn2)=O)C)CCCN(C(=O)C(F)CC)C1 O=C1OC(C(=O)NCCCCOc2ccc(Br)cc2)Cc2ccc(Br)cc21 N1(CCN(C(=O)C(=O)NC2(C)CC(N(C)C)C2)C)CCOCC1 C1(Cc2cn(CC(=O)NCC)nn2)CCCC(CNC(=O)CC)C1 CCC(C)C(CNC(=O)CCN(C(=O)CC1CC(=O)NC1=O)C(C)C)CO c1(C(=O)NC(C(C)(C)NC(C(Cc2ccc(C)cc2)C)=O)C)c(C)ccnc1C N1(C(c2c(CC)noc2)=O)CCC(N(CCC(C)C)C(=O)CC2CCC(O)C2)CC1 Nc1cc(Cl)cc(Cl)c1C(N1CC=C(CNC(C2CCC(O)C2)=O)CC1)=O c1(C(N2CC(CNC(C3(CC)CNC(=O)C3)=O)C(C)C2)=O)cccc2[nH]ncc12 c1(NC(C2(Cc3scc(C)n3)CC2)=O)ccc2ncn(C)c2c1 n1(CCC(=O)NCC=C)cc(C(C2CCOCC2)C)nn1 C1(CC(=O)N(C)CC2(CN(C)C)CC2)CCN(C(C2CC3CC3C2)=O)C1(C)C C1(NC(=O)COc2cncc(Cl)n2)CC1C1CCCN(C(C2(CO)CCCO2)=O)C1 C1(NC(CNS(N(C)C)(=O)=O)=O)CC2CC1CN2C(=O)CCSC(F)(F)F c1(C(N(C=O)Cc2cc(Cl)ccn2)C)ccc(S(C)(=O)=O)cc1 c1(C(=O)NCC2CCN(C(c3n(CC)nc(C)c3)=O)C2)cnn2c1OCC(C)C2 C(=O)(C1=CCCC1)N1CC(SC)C1.N1(C(CCCC=O)=O)CCC2CC12 c1(C(=O)NC2COCC2NC(c2cn(CC(F)F)nn2)=O)cc2ncccn2n1 c1(CC(C(=O)C(F)C(F)(F)F)=O)cccc2ccsc12.C12(N)CC1CNC2 c1(C(N2CC(C3OCCN(C(C(CCOC)C)=O)C3)C2)=O)c(F)ccc(Cl)c1F CC1CN(C(c2nscc2Br)=O)CC1NC(c1cccc(Cl)c1)=O O=C(CCC(=O)c1cccs1)Oc1ccc(Cl)nc1 C=CC(CC)CC(=O)N(C1CCN(C(=O)C(=O)NCCC(N)=O)C1)C Cc1ccc2c(=O)c(C(=O)NC3CCC(NC(C4CC45CC5)=O)C3)c[nH]c2c1C C1(N)CC2CCC(C1)N2C(=O)CCC1CC1.CN1CCOC(C=O)C1 c1(C(N2CCC(C3CCCOC3)C2)C(=O)NCCSC)cccc2cnccc12 N1(Cc2c(CC)cccc2)CCC(NC(c2c(C)nn(C)c2Cl)=O)C(F)C1 Cc1cc(C(N2CCN(C(c3ncc(C)s3)=O)CC2C(C)C)=O)cc(C)c1 c1(C(N2CC(C3CN(C(C(CC)COC)=O)C3)C2)=O)ccc2c(C)nn(C)c2n1 c1(N2CCC(CSC)CC2)cc(=NCCOc2ccccc2Cl)nc(C(C)C)[nH]1 CN1CCC(C(=O)NCCN(C(C23COCC2C3)=O)C2CC2)c2ccccc21 c1(N2CC3OCC(NC(C4C=CCCC4)=O)C3C2)ccc([N+](=O)[O-])cc1Cl CC1(C)CC(C(=O)NC2CN(C(=O)C(C)(F)C(F)(F)F)C2)CC(C)(C)O1 C12(C(=O)NC3(CC=CC(=O)OCc4ccncc4)CCCC3)CCCC1C2(F)F c1(C(=O)NCCC(C)NC(=O)Cc2ccc(F)cc2F)c[nH]cc(Br)c1=N c1(N(C(CNC(c2nc(C(C)=O)sc2)=O)C)C)nc(C(F)(F)F)cc(C)n1 N1(C(CC(CC)NC(c2[nH]ccc2C)=O)=O)CC2CCC(O)CC2C1 N1(C(C2C(=C)C2)=O)CCC2CCC(NC(c3conc3C(F)(F)F)=O)C12 c1(OCC(N2CCC(NC(C(C)=C3CCCC3)=O)C2)=O)cc(C)ccc1Cl N1(C(C(C)SCC)=O)CC(CO)C2(C1)CN(C(c1ccncc1F)=O)C2 CCCC(C(=O)NOCCCF)NC(C1CC1CC)=O Cc1nc(N2CCC(CNC(c3ccc4c(n3)CCO4)=O)C(C)C2)ccc1C#N C1(F)(CNC(C=CC=CC)=O)CCN(C(=O)CCC(=O)c2ccc[nH]2)C1 c1(CC(=O)NCC2C(NC(CN=S(C)(C)=O)=O)C2)ccc2c(c1)OCO2 N1(CC)CCN(CC(N2CCC(NC(c3c(C)noc3C3CC3)=O)C2C)=O)CC1 c1(NC(c2nc(N3CCC(C)OC(C)C3)cc(OC)n2)C)ccc2cnnn2c1 N1(C(C23CC(C)(C2)C3)=O)C2CCC1C(CO)N(C(c1ccccc1F)=O)C2 C1(NC(Cc2cc(C)[nH]n2)=O)CCC2(CC1)CN(C(=O)CCCCCCC#N)C2 C1(C(C)C)CN(C(=O)CSCCC#N)CCN1C(=O)C=CC1CCCN1C N1(C(c2c(Cl)cn(CC)n2)=O)CCN(C(C2CC2F)=O)C2COCC12 N1(C(c2c(C)sc(O)n2)=O)CCC2CCN(C(C3CN(C)CC(C)O3)=O)CC12 C1(CC)(CO)CN(C(=O)C(c2cccnc2)NC(=O)C=Cc2ccoc2)C1 C(C)(C(C)(C)C(=O)N(C)CCC1CCC1)NC(COCC#C)=O Cc1cc(C(=O)NC2(CN(C)C(C3(CO)CCC3)=O)CC2)c2c(n1)CCCC2=O c1(OC)ccc(C(N2CCC(CNc3ccc(C(F)(F)F)cc3)C2)=O)c(OC)n1 c1(C(N2C3CN(C(CCc4ccc(C)s4)=O)CC32)=O)cccc(F)c1C c1(C(=O)NC2CC(CCNC(C(C)SCCCC)=O)C2)cc(C2CC2)nnc1O N1(C(=O)C(F)CC2CCCCC2)CCCC(N2CCC2)CC1 Cc1cc(C(=O)N(CCCC(N2CCOCCC2C2CC2)=O)C)nc(O)c1 c1(OCC)cccc(CN(C(=O)Cn2cc(CSN3CCCCC3=O)nn2)C)c1 C1(CNC(CC(C=C)C)=O)CN(C(=O)CC2CN3CCN2CC3)C2(CCC2)C1 N1(C(CC2C(C)CCCC2)=O)CC2(C1)CCCN(C(=O)C1=COCC1)CC2 CN(C1CCc2c(F)cccc21)C(=O)CC1NC(=O)c2ccccc21 C=CCCC(C(=O)NC)NC(C1(C)CCCC1)=O.N1(CC(=O)NC)CCC(OC)C1 c1(CN2C(CNC(C(C)Cc3ccccn3)=O)CC2)cc(Cl)ccc1F c1(CC(N2C(C)(CC)CC(NC(c3ccns3)=O)C2)=O)cccc2ccncc12 c1(-c2n(-c3ccn(C)n3)nc(C3CC34CC4)n2)cnn2cnnc2c1 CC(=O)CCCCCCC(=O)N1CCCC(CN(C)C(C2CCCN2N=O)=O)C1 n1(C(CC)(C)C)nnnc1C(C1(c2cccs2)CC1)NCCn1cnnc1 C(C)(CNC(=O)Cc1sc(C2CC2)nc1C)(C(C)C)NC(C1(C=C)CC1)=O C(CC1=CCCCC1)N(C)C(C1COCC1NC(=O)CN1CCCC1=O)=O CC1(C(=O)NCC2CC(NC(=O)Cn3ccccc3=O)C2)CNC(=O)C1 C1(NC(CN(S(C)(=O)=O)CC)=O)CC12CCN(C(C1CCOC1(C)C)=O)C2 N1(C(C(CC)C#N)=O)CCC(CNC(c2ccc(F)c(Cl)c2N)=O)C(F)(F)CC1 c1(C(=O)NC2(CO)CCC2)cncc(CNC(C2CCSC2)=O)c1 C1(S(C)(=O)=O)(NC(CC2OCCN(C(c3cc(CC)nn3C)=O)C2)=O)CCC1 N1(C(CC2(C)OCCO2)=O)CC2CC(NC(c3cc(F)ccc3Cl)=O)CC2C1 C1(NC(c2ncccc2F)=O)CC2CN(C(c3cc(C4CCCC4)on3)=O)CC12 c1(C(=O)NCCCCC2CN(C(c3n(C)nnc3)=O)C2)ccc(C2CC2)cc1 C(c1cccc(F)c1)=CC(=O)NCC1CC2(CC2)CN1C(=O)C1=CCSC1 c1(CNC(N2CC(NC(=O)CCC=CBr)C2)=O)ccc(Br)cc1O S(=O)(=O)(c1ccc(CC(=O)Nc2cnc(C)nc2N2CCCC2)s1)NCC=C c1(C(=O)NCC(CN(C(C(C(C)C)NC(C)=O)=O)C)C)ncc2n1CCCC2 c1(C(C)NCc2cccc(-c3cccnc3)c2)ccc(N)c(Cl)c1 c1(CC)ccc(=NCc2ccc(OC(=O)NCC)cc2)[nH]c1 c1(C(=O)NC(C2CCN(C(c3coc(C(F)F)n3)=O)C2)C)cc(F)ccc1F N1(C(CCC2C(C)C2)=O)Cc2n[nH]cc2C1C(=O)N1C2C=CCC1CC2 N1(C(Cn2ccc(C)n2)=O)CCOCC1CNC(=O)CCc1cnn[nH]1 N1(C(Cc2cccc(OC)c2F)=O)CCC2(CCCC2NC(c2ccoc2)=O)C1 C1(n2cc(CC(C)C)nn2)CC2CCC1(NC(C1CCC(F)C1)=O)C2 S(=O)(=O)(c1cccc(Br)c1)N(C1CCC(N)(c2ccccc2)CC1)C c1(C(=O)NCC2(NC(C3CC(C)SCC3)=O)CC2)cc(F)c2cn[nH]c2c1 c1(NC(C(CCC2CC2)NC(c2cncc(Cl)c2)=O)=O)ccc2nc[nH]c2c1 C(=O)(C1=CCCOC1)NC(C)CC(C)NC(c1ccn(-c2cccc(F)c2)n1)=O N#Cc1ccc(CC(=O)NCC=C2CCN(C(c3csc(O)n3)=O)CC2)cc1 C1(CNC(Cn2c(C)nc(C)n2)=O)CN(C(C2CC2(F)F)=O)CC1(F)F C12(NC(C(C)CO)=O)CC(CO)(C1)OC21CN(C(c2cc(OC(F)F)n(C)n2)=O)C1 c1(OC(C)C)ccc(Cl)cc1C(=O)NCC1CCCN(C(C2COCCO2)=O)C1 C#Cc1ccc(NC(CC(C)C)C(=O)NCC2CC(CN(C)C)C2)nc1 CCC(C)C(C)C(=O)NCCCCCCN(C(=O)CCc1ncco1)C C(=O)(C1=Cc2ccccc2OC1)N(CCN(C(C12OC(C)C(CC1)CC2)=O)C)C c1(SC)cnc(N2CCCC2C(=O)NCc2cnccc2Cl)nc1 c1(C2N(C(C(=O)N(C)CCC3CCCCO3)=O)CCC2)cccc(Br)c1 Cc1ccc(Cl)c(F)c1C(=O)NC1CC1CNC(C1(O)CCSCC1)=O C1(CNC(CCN(CCC)C)=O)COC(CNC(=O)CN(C)C)C1 C1(C(N(C)CC2(C)CCCC2)=O)CNC2CCOCC2C1 Cc1cc(F)cc(Br)c1C(N1CC(CNC(=O)C(C)n2ccnn2)C1)=O n1(CC)c2ccccc2c2cc(-c3cn(CC(=O)NC4CC(F)(F)C4)nn3)ccc12 c1(C(N2CC3N(C(C4(C)CCNC(=O)C4)=O)C(C3)C2)=O)cnc2ccsc2c1 C1(NC(Cc2nc(C)[nH]n2)=O)CC2CC(NC(=O)Cn3cc(C(F)(F)F)cn3)CC12 C(=O)(CC(C)C(F)F)NCC1CCC(C(=O)NC2C(OC)C(O)C2)CC1 N1(C(COc2cc(C)on2)=O)CCCC12CCCN(C(=O)CC1CC=CC1)C2 C12(NC(CN=S(C)(C)=O)=O)CCCC1CN(C(c1cc3ncccc3[nH]1)=O)C2 CCC(C)(CC)C(=O)NC1C=CCN(C(=O)CCc2ccc[nH]2)C1 Cc1ccoc1NC(C=CCC(C)(C)NC1CCN(C(=O)CN2CCCC2)C1)=O C(CC(=O)NCC1(O)CCCC1(C)C)(C(F)(F)F)NC(CCC1CC(C)C1)=O C1(C(=O)NCCC2(NC(C(C)NC(N)=O)=O)CCC2)CCC2(CCC2)CC1 C1(OC)CC(CNC(c2cnc(S)n2C)=O)N(C(c2ccccc2)=O)C1 c1(CC)ncc(I)s1.c12cnn(c1)CCNC2c1nnnn1C(C)(C)CC c1(C(N(C)CC2CCCN2C(c2ccc(NC(N)=O)[nH]2)=O)=O)ccc2sncc2c1.C C=Cn1nncc1C(=O)N(C(C)C(N)=O)C1CC1 C1(NC(=NC)NCC(c2ccc(C)c(C)c2Cl)OC)CCn2ccnc2C1 C1(CCC(=O)N(CC#C)CC2CC2)CCCCN1C(c1nccn1CC)=O c1(C(N2CCN(C(CC3CC(=C)C3)=O)C(C)C2C)=O)ccc2[nH]c(C)c(C)c2c1 c1(C(N2CCCC(NC(C(C)=CC3CC3)=O)C(F)C2)=O)cn2cc(Cl)cnc2n1 CC1(CNC(=O)CCCNC(C2(O)CC(CF)C2)=O)CC2CCC1C2 C(C(O)CC(=O)N1CCC(C2CCCCN2C(C2COC(=O)O2)=O)CC1)N(C)C N1(C(C=C2CCN(C)C2)=O)CC2(NC(=O)CNC=O)CCCC2(F)C1 c1(N2CCC(C(=O)NC(C(=O)NC)C)CC2)ncnc2c1SCCC2 c1(C(=O)NC(C)CCNC(c2cnn(C3CC3(F)F)c2)=O)ccncc1Cl CCC(C(=O)NCCCC1CCCN1C(=O)C=CC(C)C)OC N1(C(Cc2c(C)ncs2)=O)CCC(F)(CNC(=O)C(N)=O)C1 CC(C)(CC#N)c1cn(CC(F)(F)CO)nn1.C(=O)(C(CCl)c1ccccc1)N O=C(O)CCCCc1cccc(-c2nc(-c3ccsc3)nn2CCF)c1 C1(C=O)CCC(n2cc(N(N3CC(O)CC3Cc3ccc(C#N)s3)C)nn2)CC1 c1(OC)ccc(C(=O)N(CCCNC(=O)CN2CCCCCC2)C)cc1Cl N1(C(c2cc(C)no2)=O)CC(C2(NC(c3cc(Cl)ccc3N)=O)CC2)C1 C#Cc1ccccc1CC(=O)NCC1CCN1C(=O)CCC1CCOC1 n1(C(C)CO)cnc2c(NC3(C(=O)OCC4CC4)CCCC3)ncnc12 C1(CNC(c2c(Cl)ncc(C)c2)=O)CCC2CN(C(=O)CC(C)(C)O)CCC2C1 c1(CC)ccc(Cl)c(NC(=O)NCc2nccn2C2(Cc3ccccc3)CC2)c1 c1(C(=O)NC(C(C)NC(c2nc(COCC)sc2)=O)C)cnc2ccnn2c1C C(=O)(C(C)(C#N)CC)NCCC(CC)(C)NC(=O)CCc1nc(=N)[nH][nH]1 C1(CNC(C(C)CNC(=O)CCC2(C)CC2)=O)OCCCC1(C)C c1(NC(C(=O)NC2OCC(CNC(CCC(=O)OC)=O)C2)=O)cc(F)cc(Cl)c1 N1(C(C(C)NC(C)=O)=O)CC(=O)NCC1C(=O)NCCc1ncnn1C N1(C(C(=O)NC2CCN(S(CCCC)(=O)=O)CC2)C)CCCC(O)C1C C(C(CC(=O)NC1(C(C)C)CC1)OC)NC(CCN(C)CC)=O CC(C)CCCC(C)N=c1nc2ncn(C)c2c(NCC2(C)CC3CC3C2)[nH]1 Nc1cc(C(=O)Nc2cccc(CNC(C3CC4CCC34)=O)c2)cnc1Cl C1(CC(N2CCCCC2C2CCCN(c3nnnn3C)C2)C)COCCN(C)C1 CCCCC(C)(F)C(=O)N1CC(NC(=O)CCCF)C(Cc2c(C)n[nH]c2C)C1 C(=O)(CCCC(C)(F)F)NC(C1CCCC1)CNC(C(COC)OC)=O CCC(C(C)CN(C)C)NC(C1C=CC(NC(C23CCC(CC2)C3)=O)C1)=O c1(NC(C23C(CN(c4cc(COC)ncn4)C2)C3)=O)ccc(C(F)(F)F)c(F)c1 CCC(C)CCC(=O)NC(CO)C(C)NC(c1nc(Cl)ccc1N)=O C1(CC(N2CC(Cn3cc(CCn4ncc(C)c4)nn3)C2)=O)CCC(F)(F)CO1 c1(CC)ncncc1C(=O)NC1(C)CC(C(=O)NC(c2cnn(C)c2C)C)C1 C(=O)(CC(C)CNC(N)=O)NCc1cc(C(=O)NC(c2nccs2)CC)n[nH]1 C12(CNC(C(C)OCC=C)=O)CC1CN(C(=O)Cc1ccccc1C)C2 C1(C(=O)NCC(CCOC)NC(C(CC#C)C)=O)CC2CCCC(C1)C2 C(CCCCC(=O)NC(C)CCC(=O)NCC1(CO)CC1)SC C(CC(C)(C)CC(=O)NC1CCC(Cn2cc(CC(C)O)nn2)CC1)OC c1(C(=O)NC2CCN(C(C(C)Cc3ccc(F)cc3)=O)C2)cccc2ccoc12 C1(NC(c2c(C)nsc2)=O)CC2CCC(C1)N2C(=O)CCCc1nccs1 CC1(C)NC(=O)N(CCC(=O)NC2(C)CCCN(c3nnnn3C3CC3)C2)C1=O c1(C(=O)NCC2C(NC(CC3CC(=O)NCCC3)=O)CC2)ccn2ccnc2c1 c1(NC(CNC(=NC)NCCSc2ccco2)=O)ccc(Cl)cc1 c1(OC)ccnc(C(=O)NCC(C)CNC(=O)CCN2CCOCC2=O)c1F C1(C(=O)NCC2CN(C(=O)C=Cc3ccc(C)o3)C3CC23)(COC)CCCCC1 C1(CC)CCN(C(=NCC(c2ccccc2)N(C(C)C)CC2CC2)NC(C)C)C1 c1(C(=O)NCC2CC2NC(C2CC3CC2CC3O)=O)cccc2c1CCO2 c1(C(=O)NC2(CO)CCCN(C(C=C(C=CSC)C)=O)C2)cccc2cncn12 CC1CCC(N)(C(=O)N(CCCC(C)(F)F)C)C1 C=CCC(CC=C)C(=O)NC(C)CN(C)C(C1CCC(NC(C)=O)CC1)=O C1(C(=O)NCCNC(C2CCCC(C(=O)OC)C2)=O)CCc2n[nH]cc2C1 C12(CC(=O)NC)CCC1CN(C(=O)C(C)CC(N)=O)C2.ONC(=O)CCOC(C)C C(C(C(=O)NC1CC(C(C)C)C1)N1CCCC1CC(=O)OC)SCC c1(C(=O)NCCCN(C(C2C3CCN2CC3)=O)C2CC2)nc2ccccc2[nH]1 CC#CCCCC(=O)NC(C1CCCC1)CNC(=O)CCCOc1cccnc1 CCCC(C(=O)NC1CN(C(c2ccc(F)s2)=O)CC1c1cnn(C)c1)C(C)C c1(CC(C)C)c[nH]c(C(=O)NCC2CCCC2NC(c2cc(C(N)=O)c[nH]2)=O)c1 c1(C(=O)NC2CCC2NC(C2CCOC2)=O)cc([N+](=O)[O-])c2nsnc2c1 C(=O)(CC(F)(F)C(F)F)N1C(CC(=O)NOCC(F)F)CC(C)(C)C1 N1(CC)C(=O)c2ccc(C(=O)OCC(=O)NCCc3ccccn3)cc2S1(=O)=O N1(C(c2ccc(C3CCC3)cc2)=O)CC2CN(C(C3CCCC34CC4)=O)CC2C1 C1(NC(c2csnn2)=O)CC(NC(c2cccc(Cl)c2C(F)F)=O)C12CCC2 N1(Cc2cc(OC)no2)CCC(NC(c2cccc(-n3cccn3)c2)=O)C(C)(C)C1 C(=O)(CC(O)CN(C)C)NCC(C1CCN(C(c2cnc(O)s2)=O)CC1)C Cn1cc(CNC(c2ncccc2-c2cccc(F)c2)=O)cc1C#N c1(CC)[nH]nc(C(N2CCC2CO)=O)c1F.N12CCN(CC1)c1ncccc1C2 c1(C(=O)NCCN(C(c2ccc(OC)c(O)c2)=O)CC)ncc([N+](=O)[O-])cc1C C1(N(C(=O)C(N)=O)C)CCN(C(C2CCSCN2C(=O)OC(C)(C)C)=O)CC1 N1(C(CS(C(C)(C)C)(=O)=O)=O)CCC2(C1)CN(C(C1CC(CO)C1(C)C)=O)CCO2 C1(C(C)C)CCOC1C(=O)NC1CCC(CNC(=O)C=C(C)C(F)F)C1 C(=O)(C(C)(F)C(=O)NCC(F)CNC(c1c(Cl)cccc1Br)=O)OC CC(C)CC(C)(C)C(=O)NCC1N(C(=O)CNc2ccccc2)CCCC1(C)C c1(-c2cn(CC)c(=O)cc2)ccc2[nH]cc(C(N3CCOC(CO)C3C)=O)c2c1 c1(C(=O)NCC2(F)CN(C(=O)CCc3nncs3)C2)ccc(-c2cc[nH]n2)cc1 C1(NC(c2scc(OC)c2)=O)CCCC(C(=O)NC(c2ncc[nH]2)CO)CC1 N1(C(C(C)c2cccs2)=O)CCC(NC(c2ccc(F)c(F)c2)=O)CC1C c1(C(N(C(C)CNC(c2ccn(CCC(F)(F)F)n2)=O)C)=O)ccc(Cl)cn1 c1(C(N(CC(CN(C(C2=C(C)OCC2)=O)C)O)C)=O)cccn2nccc12 CC12CCC(C(N3CCN(CCNC(C4(N(C)C)CCCC4)=O)CC3)=O)(C1)OC2 C#CC1CCCN(C(C2(C(C)N(C)Cc3nc(Br)cn3C)CC2)=O)C1 Cc1ccc(C(N2CCC(NC(=O)C3=CC(C)(C)C3)C2C2CC2)=O)nc1C c1(C(=O)NCCCCCNC(C2C(CC)C2)=O)ccccc1SC(C)C C#CCC(CC#C)C(=O)NC1CC2C(NC(=O)CC3CS(=O)(=O)C3)C2C1 CCCCC(CNC(=O)C(F)=C1CCCC1)NC(=O)C(C1CCC1)OC c1(C(=O)NC(C2CCOC2)CNC(C2C3CCC2CC3)=O)ncnc(O)c1Br C1(CNC(c2c(CC)nn[nH]2)=O)CN(C(c2cn(C(C)C)cc2C)=O)CCO1 CC(=O)CCCC(=O)NCCN(C1CCCCCC1)C(C1CC2(CC(=O)N2)C1)=O c1(CN2CC(CNC(C3(C)CC3)=O)C2)ccc2ocnc2c1 C(=O)(CCCC(F)(F)F)N(C1CN(C(=O)Cc2cnc[nH]2)CC1F)C N1(C(C(CC=C)OC)=O)CCN(C)C(C(=O)NC(CN2CCCC2)CO)C1 C1(C(N2C3CC(CN(C(c4ccc(C)cc4)=O)C3)C2)=O)CCc2cnn(C)c2C1 c1(CNC(=O)Nc2nc(C)c(C#N)s2)ccc([N+](=O)[O-])cc1Br C12(C(=O)NC3(CN(C)C)CC3)CCC(NC(=O)C(O)C(F)(F)F)(CC1)C2 N1(C(c2cnc(C)[nH]2)=O)CCC(C)C(NC(C23C4CC(CC24)C3(F)F)=O)C1C CC#CCN=c1[nH]c2c(c(=NC(Cc3ccccc3)CCO)[nH]1)COCC2 C1(N(C)C(C2CC(F)C2)=O)CCC(N(C)C(c2cc(C3CC3)no2)=O)CC1 c1(SC)cn(C)nc1C(=O)NCCCOCCCC.C1(=O)COCCCN1 c1(C(N(C2CCN(C(c3ccc(C)s3)=O)C2)CCO)=O)cccc2[nH]ncc12 C(=O)(CCC=O)NC(C)(C)C1CC1.N1(CC)CCCC1C(C)(C)C N#CC1CN(C(c2ccc(F)nc2F)=O)CC1NC(c1cnon1)=O CCCCCCCC(O)CC(=O)NCC1C(C)CCN1C(c1cc(C#N)c[nH]1)=O N1(C(C(C)(C)C2CCCCO2)=O)CC2CC1CN2C(=O)COc1ccc(Br)cc1 C12(CNC(C3CCC(c4nc(C)on4)C3)=O)CC(C(=O)O)C(CO1)C2 N1(CC)CCN(C)CC1.C(=O)(C(N)CC1OCCO1)N(c1ccccn1)C(C(C)N)=O c1(NC(C2COCCN2Cc2ccc(F)c(O)c2)=O)c(O)cccc1O N1(C(c2c(C)cncn2)=O)CCC(C(=O)N(CC(C)(F)F)C)CC1C(C)C N1(C(c2c(N)sc(C)c2C)=O)CCCC2(CC(NC(C3CC3C3CC3C)=O)C2)C1 C(C1(C)COC1)=CC(=O)NCCCN(C(C1(OC)CCC1)=O)CC C(=O)(CCCCCCC(=O)NC1(CNC(=O)Cc2ccoc2C)CCOC1)OC CCCC(C(O)C(=O)NC(C(=O)OC)C1CC1)NC(C1CC2(CC(=O)C2)C1)=O N(C1CCc2ccc(Cl)nc21)C1C2(CCN(C(C(CSC)C)=O)CC2)CCC1 CC1CN(C(=O)CN2CC(=O)NC2=O)CCC1N=c1ccnc(-c2ccccc2)[nH]1 N1(C(c2sccc2I)C(=O)NCCC2CC2)CCCC2(CC(O)C2)C1 CCC(C)C(C)C(=O)NC1(CC(N2CC(F)(CF)C2)=O)CCC1 C1(C(N(CC(C)(C)NC(CSCC)=O)C)=O)CCN(C(C)=O)C1 c1(CC(N2CCC(CCNC(=O)C(O)C3CC3)C2)=O)c[nH]c2ccccc2c1=O N1(CC(=O)NC(C)CC(C)NC(c2ncncc2Cl)=O)C(=O)CN(C)C1=O n1(CC(=O)NC(c2ccc(CNC(=O)C=NOC)cc2)C)ncc2cccnc12 C1(O)(C(C)C)CCN(C(=O)NN(C)C(c2cnn(CCO)c2)=O)C1.C12CC1C2 c1(COC)c(C(=O)NC(CNC(c2cc(C)nn2C(F)F)=O)C(C)C)cnn1C c1(C(N2C3C(C(=O)NC(C(C)SC)C)C(C3)C2)=O)ccc2[nH]ccc2c1 N1(C(c2c3ccc(OC)cc3[nH]n2)=O)CCC2CN(C(=O)C(C)N(C)C)CC2C1 C#CCC(CC(F)F)C(=O)N1CCC(C)(CCNC(=O)CCCn2cncn2)C1 C(C(C)(C)C(=O)N(CCCOCCNC(=O)C(CC)C1CCC1)C)SC c1(C(=O)NC2C3(CCN(C(CNC(NCC)=S)=O)C3)C2)ccc2cccnc2c1 c1(N2CC(C)C(NC(c3ccc(=O)n(C)n3)=O)C2)nc2cc(F)ccc2o1 C1(OC)CN(C(=O)CCn2cccn2)CC1NC(c1ccn(C(C)C)c1C)=O C12(CNC(c3cnc(C)[nH]3)c3nnnn3C3CCCCC3)CC(C)(CCO1)C2 CC1CCN(C(c2cc3n(n2)CCC3)=O)C(CNC(=O)CCS(C)=O)C1 Cc1ccc(C(=O)NCCN(C(=O)C(C)N2CC(C)C2)C(C)C)c(Cl)c1Cl Cc1cc(Br)c(O)cc1NC(c1sc(NC(c2ccc(I)cc2C)=O)nc1C)=O c1cc(Cl)ccc1CN(C(C1CC1CNC(c1cc(CC)c[nH]1)=O)=O)CC C1(NC(C2N(C(C3(C(=O)NC)CC3)=O)CCCC2)=O)CCCCC1C#N CCC(CC)C(CCNC(=O)C(N1CCN(CC(=O)NCC(C)C)CC1)=O)OC c1(C(=O)NCC(COC)O)ccc2c(c1)NC(=O)C2CC(=O)Oc1ccccc1 CC1(C)CC(n2ccnn2)CN(C(=O)CCCCC#N)C1.N1OC(C)(C)CC1=O c1(C(=O)NCC2(F)CC(NC(C(CCSC)O)=O)C2)cccc2c1OC(C)C2 N1(C(c2cc(CSCC)on2)=O)CCN(C(C2CCNC2=O)=O)C12CCC2 c1(OC)ccccc1CNC1CC(C(=O)Nc2cccc(N3CCCC3=O)c2)C1 C(=O)(CCC(C)(C)F)NC(C(=O)NCC(C(=O)OCC)C)CCC1CCOCC1 CC1(CNC(=O)C(F)(F)CO)CCC(NC(=O)C(C2CC2)C2CC2)C1 CCC1=C(C(=O)N2CCOC(C(C)NC(=O)CSC)C2)CCCO1 C1(NC(C(C2CCC(=O)N2)C)=O)CCC2(CCN(C(=O)Cc3nccn3C)C2)C1 c1(C(=O)NC23CCN(C(c4ccc(C#C)cn4)=O)CC2C3)ccn2cnnc2c1 c1(C(CNC(C(CC)C)=O)NC(=O)CC(=O)N(C)C)cccc(C)c1 Cc1cnc(C(=O)NCc2ncccc2C(=O)NC2(C)CCCC2C)c(C)c1 C(=O)(C(C(C)CC)NC(c1cn(C)c(=O)n1C)=O)NC(CC(=O)OCC)C N1(C(CCC2(C)CC2)=O)CC2CC2C1C(N1CCC(C(c2ccco2)=O)C1)=O O=C(C#CC1CCCO1)NCC1=CCN(C(c2ccc(CO)cc2F)=O)CC1 c1(C(N(C)CC2CCCC(NC(C(F)=CCC)=O)C2)=O)cc(F)c(F)cc1O c1(C(=O)NCCCCNC(C(CC#C)CC#C)=O)cc(Cl)cc2ccncc12 C1(CN(CCCOC)C)CCN(C(C2CCOCC2)=O)CC1.C1(C(=O)OC)CCCO1 C1(C(=O)NCc2cn(C3CC3)nn2)CN(C(=O)CCC2CC2(F)F)CC12CC2 C1(CC(=O)NC2CC3(C2)CC3NC(C2CCC2)=O)Oc2ccccc2NC1=O C(=O)(C1=NOC2(CCOC2)C1)N1C(C)CN(C(=O)CCOC2CCOCC2)CC1 N1(C(CN(C(C)C)C)=O)CC2(NC(=O)C(C)C3CC3)CCC1CC2 CC1=C(C(=O)N2CCN(C(=O)CCc3ccc(C)o3)CC2C)CCCC1 C(=O)(C1CCCc2nccn21)NC.N12CC=C(CC(=O)N3CCCC(C3)C1)CC2 C1(C(C2CN(C(N)=O)C2)=O)CN(C(=O)CNC(=O)NCC2(n3nccn3)CC2)C1 C(CCCCCN=[N+]=[N-])NC(C(Cc1cn[nH]c1)NC(C1(C(=O)OC)CC1)=O)=O c1(C(=O)NC(CCOC)CNC(C2C3(CC3)C23CC3)=O)cc(Cl)cc(Cl)c1 C1(N(C(=O)Cc2ccccc2F)C)CN(C(C2(CC(F)F)CCC2)=O)CC12CC2 N1(C(Cn2c(C)ccn2)=O)CCOCC1Cc1cn(C(C)C)nn1 C=C(C)CCC(=O)N(C1CCN(C(C2CCC2c2c(C)noc2C)=O)CC1)CC CN1CCN(C(=O)CCC2CC2)C(CNC(C2CC3(CC(=O)C3)C2)=O)C1 c1(CNC(c2[nH]nnc2CNC(c2cnc(Cl)s2)=O)=O)cccc(O)c1 S(=O)(=O)(c1cc(NC(=O)NC(c2ccc(F)cc2)C)ccc1C)NC C1(NC(c2nc(CCC)oc2)=O)CCN(c2nc(CC)nc(=N)[nH]2)CC1O N1(C(c2c(Cl)c(C)n(C)n2)=O)CCC2CN(C(c3ns[nH]c3=O)=O)CC12 N1(C(C=C(C)C)=O)CCC(CC(C)NC(=O)C=Cc2nccs2)CC1 CCC1=NOC(CC(=O)NC2(CCNC(=O)C(C)C3CCCC3)CCC2)C1 c1(C(=O)NCC(CNC(C(C)CC(N)=O)=O)C)ccc(O)c2ncccc12 CC1(C)C2CCC1(C(N1CCOC3CCC13)C(=O)Nc1ccccc1)CC2 C(=O)(C#CC1(CC)CC1)N1C(CCCNC(CC(=C)C)=O)CCC1 C(=O)(C(=O)NOC)N1CC(N(C(=O)CCOC(C)=O)C(C2CCCCO2)CC)C1 c1(C(=O)NC(C(C)C)CN(C)C)cnc2cc[nH]n2c1=O Cc1nc2cc(C(=O)NC3CC(NC(=O)C=CC4CC4)C34CCC4)cnc2s1 c1(C2(C(=O)NCC3(CNC(C(CC=C)N(C)C)=O)CC3)CC2)ccc(C)cc1F C#Cc1cnn(CC(N2CC3CC3(NC(=O)CC3(NC(C)=O)CCCC3)C2)=O)c1 Cc1nc(C)n(O)c1C(N1CCCC(C(C)(O)CNC(=O)Cc2ccon2)C1)=O C1(NC(C=CCOC)=O)CCN(C(=O)COc2ccc(Cl)cc2Cl)CC1COC c1(C(N2CC(=CC)C2)=O)ccoc1CNC(=O)C(F)C1CCOC1 N1(C(C2CC(C)(C)OCC2)=O)CCC2(CC1)CC2C(=O)NCC1(Cl)CC1(F)F Cc1nnc(CC(=O)NC(C2CN(C(=O)C(C)(C)C3CCCO3)C2)C)s1 N1(C(c2cnc(C(C)C)[nH]2)=O)CCCC(NC(c2nocc2C2CC2)=O)CC1 c1(C(=O)OC)ncc(C)cc1S(=O)(=O)N1C2CCC(C2)C1c1ccccc1 C1(CNC(CC2CC(C)C2)=O)(CNC(=O)CCc2cccn2C)CCOCC1 N1(C(CC2N(C(CC(C)(C)O)=O)CC(F)C2)=O)CCCC(O)(C(N)=O)C1 N1(C(C2CC(SC)C2)=O)CCCN(CCNC(=O)C(F)CC2CCCC2)CC1 C(=O)(C1CCc2c[nH]nc21)N1CC(CCC)N(C(c2cc[n+]([O-])cc2)=O)CC1 N1(S(c2c(C)cccc2Cl)(=O)=O)Cc2c(Br)cccc2CC1C N1(C(COCC(=O)NC)=O)CC2CC1C2C(=O)N(C1CCOC1C)C N1(C(C2(CCOC)CC2)=O)CCCCC(CNC(=O)CCC(C)(C)OC)C1 c1(SC)nc(=NC2CCN(C(=O)CCc3nc[nH]n3)CC23CCC3)c(C#N)c[nH]1 n1(C(C)C)c(O)nc(N2CCCN(C(=O)Cc3nc[nH]n3)CC2)cc1=O CC(C)CCC(F)C(=O)N(C1CC1)CC1CCCN1C(c1ccc2c[nH]nc2n1)=O C1(CNC(C(CC)(C)C)=O)N(C(c2cnc3n2CCS3)=O)CCC1(C)C CCC(C(=O)N(C)CC1CN(C(=O)CN2CCCCC2)C1)SC.S(=O)(=O)(CC)N c1(C(=O)NCc2nccc(C(=O)Nc3ncc(Br)nn3)c2)nc2ncccn2n1 S(=O)(=O)(c1ccc(C(=O)NCC2CCC2NC(C2CC3(CSC3)C2)=O)cc1)NC CCC(C)(C)CC(=O)N1CCC(F)(C(=O)NCC2(C)CC(F)(F)C2)CC1 c1(CC)ccc(C(N2CCC(F)CC2)C(=O)Nc2c(C)cccc2C)c(OC)c1 CCCC(C(O)C(=O)N1CCCC1CC1CCC1)NC(=O)C(COC)OC N1(C(C2(COC)CC2)=O)CCCC(O)(CC(N2CCC(OC(F)(F)F)C2)=O)C1 C=CCC(C)C(=O)OCC1C=CCN1C(c1onc(OCC)c1Br)=O N1(C(C2CCN(CC)C2)=O)CCN(C)C(C(N2CCC(N3CC=CC3)C2)=O)C1 Cn1nnc2c1CCC(C(=O)NCC1(C)CN(C(c3n[nH]cc3Cl)=O)CCO1)C2 C12(C(N(CCN(C(=O)C3=CCCCO3)CC)CC)=O)CC3CC(CC(C3)C1)C2 c1(OC)cccc(CC(=O)NC(CNC(=O)CCCc2cccs2)C(C)C)c1Cl CCCC(CC)C(C(=O)NCCC1(C)CC1)N1CCC(C(=O)NC)CC1C CCCC(F)(F)C(=O)N1CC(CCNC(=O)CCCN2CCCC2)(OC)C1 N1(C(C2C(OCC)C2)=O)CCC(C2(NC(C3CCOC3)=O)CC2)CC1 c1(SC(C(N2CCC(OCCNC(CC(=C)C)=O)C2)=O)C)ccc(C(C)C)cc1 N1(C(C(C)c2ncco2)=O)CC(NC(C2(C(C)(C)C)CCCCC2)=O)CC1(C)C C(=O)(C(F)(F)C(F)(F)F)NCC1(O)CCN(C(C23CC(C(F)(F)F)(CO2)C3)=O)C1 C1(C(N2CCC(C(C)NC(c3cnc4n3CCC4)=O)C2)=O)CCCCC1C1CC1 c1(OC)ccc(C)c(C(=O)N(C)CC2C3CN(C(=O)Cn4nnc(=N)[nH]4)CC23)c1 CCCCCC(C)CC(=O)N(CCC(=O)NC(CN1CCCC1)CO)CC C1(C(C)C)C(=O)NCC(=O)SCCC(=O)N1.C(CCC(=O)NC1CC1)C1C(C)C1 c1(OC)ccc(C=CC(=O)NCC23CCC2CN(C(=O)Cc2cnoc2)C3)cc1 CCCC(CC)C(=O)NC1CC2(C1)CC2C(N1CCC(C(C)(C)C)CC1)=O CC(C)(CNC(=O)CC1CC2(CC2)CO1)CC(=O)N1CC=CC1C(N)=O Cc1cc(C(=O)NC2CC2c2ccc(Br)cc2)c(Cl)cc1Cl c1(C(=O)NC2C(CNC(CCOCC)=O)COC2)ccccc1CC1CCC1 CC1CN(C(c2ccn(CC(F)F)n2)=O)CCCN1C(c1cccc(N)n1)=O c1(CCC(=O)NCC(CNC(=O)COC2CC(F)(F)C2)O)cnc2n1CCOC2 c1(C(=O)NC(CC)CNC(C2(C#N)CC2)=O)cc(C)c2nc(C)cn2n1 C(=O)(C1CCc2cc(Cl)ccc21)NC1CC(CCNC(=O)CCCC2CC2)C1 c1(CC(=O)NC(C)C(=O)N(C(C)CNC(C23CC(F)(C2)C3)=O)C)cccnc1 Cc1cc(F)ccc1C(c1nnnn1Cc1ccon1)NCC1CC1CO C(CCC(C)CC(=O)NC(C1CC1)C)=CC.N12CC(C1)N(C)C(=O)C2=O.OC CCS(=O)(=O)c1ccc(CNC(C2CCCN2S(C)(=O)=O)=O)cc1 N1(Cc2cccc(OC)n2)CC2CC1CN2C(c1cc(Br)ccc1C)=O C1(NC(c2nncc(C)c2)=O)CCSC12CN(C(C1(C(F)(F)F)CCCC1)=O)C2 C1(CCNC(c2nc(CCC)oc2)=O)CC(F)(F)CN1C(=O)CC1CCSCC1 C(C)(C)(C(C)NC(=O)COCCNC(C12CC(CO)(C1)C2)=O)OC c1(C(=O)NCC2(C)CCN(C(CC=CC=C)=O)C2)[nH]c2c(c1C)CCCC2 CCC(CC)CCCC(=O)NCC#CCNC(C1CC2(C1)CC(CO)C2)=O C1(C(c2cn(CC(CNC(=O)C3=C(C)OCC3)(C)C)nn2)CC)CCCC(=O)N1C c1(CSCC(C)OC(c2ccccc2)C)csc(C)c1C c1(C(=O)NC(CNC(C(c2cn(C)nc2)(C)C)=O)C(C)(C)C)cc([N+](=O)[O-])c[nH]1 C1(NC(=O)Cc2ccccn2)CN(C(c2cnc3[nH]ncc3c2)=O)CCC1(F)F c1(C(N2CC3C(CC(N4CCC(C(C)C)C4)=O)(CC3)C2)=O)n[nH]c2ccccc12 CCCCC(O)C(=O)N1CC(c2cn(C3CCN(C(=O)C(O)CC(C)C)CC3)nn2)C1 Cc1cc(O)c(F)cc1-c1ccc(CN2CCC2CO)s1 n1(CC(=O)NCC2CCN2C(=O)Cn2cc(CC3CC3)nn2)cc(Br)cn1 N12CCN(CC1)c1ccc(cc1)C2=O.N1(CC)CCN(CC(=O)O)CC1.CCCN C(c1ccccc1C(F)(F)F)=CC(=O)NCCCN(C(c1cc(C)no1)=O)CC c1(OC)cc(C(N2CC(NC(C3CC=CCO3)=O)C(F)C2)=O)ccc1F CCCCC(C(=O)NCCCN(C(c1ccncc1N)=O)C1CC1)ON=C(C)C C(=O)(CCC#Cc1ccccc1)NCC(CNC(C1C(C)(C)OCCO1)=O)CO c1(C(N(CC(=O)NC(C)C(C)C2CC2)C2CCC2)=O)c(O)cccc1F c1(NC(c2n(C)cc(NC(CC#C)=O)n2)=O)ccc(Cl)c(C(=O)OC)c1Cl C1(N(C(C(CCOCC)NC(=O)C(=CC2CCCC2)C)=O)C)CN2CCC1CC2 C1(OC)(OC)CC(C(N2CC(C(=O)O)(Cc3cn(C(C)(C)C)nn3)C2)=O)C1 N1(C(C(C)NC(C2CCCC2)=O)=O)CCC2(C1)CN(C(=O)C=Cc1ccncc1)C2 Cc1cc(C(N2CCN(C(=O)CC3CCNC3=O)CC2)=O)c2c(c1)CCCN2 CCCC(CCCNC(=O)CCSCC(=O)NC)NC(c1ccnc(CC)c1)=O C1(NC(C2C(OCC)CC2)=O)C2CC(NC(=O)C(C)OC)CC12 C1(OC)CCC2(C(=O)NC3CC(NC(=O)CSC4CC4c4cccs4)C3)CCC12 c1(C(N2C(CNC(CC(CC)C)=O)CCC2)=O)cc(OC)c2ncccc2c1 Cc1ccc2c(c1)CC(C(=O)NCCCN(C)C(c1cnc3[nH]cncc1-3)=O)S2 N1(C(CC(C)c2cnn(C)c2)=O)CCC(O)(CNC(C2CC=CC(O)C2)=O)CC1 c1(N(C)CCn2cnnc2)cccc(S(=O)(=O)N2CCOC(c3ccsc3)C2)n1 Cc1c(C(N2CCC(CO)(NC(c3cccc(=O)o3)=O)C2)=O)cnn1C1CCC1 c1(C(N2CCC(C)(CCNC=O)C2)=O)nccc(-c2cn(C3(CO)CC3)nn2)c1Cl Cn1ncc([N+](=O)[O-])c1C(N1CC(NC(=O)CCn2cncn2)CC(C)(C)C1)=O Cc1nn(C)c(Cl)c1C=CC(=O)NCC1COC(CNC(=O)C=CCO)C1 N1(C(CS(CC)(=O)=O)=O)CCCC2(CCN(C(C3CCCC3S(C)(=O)=O)=O)C2)C1 N1(C(CCCSC(C)(C)C)=O)CCC(O)C(NC(C2Cc3nccn3C2)=O)C1 c1(C(=O)NCc2ccc(-c3ccsc3)nc2)cccc2c1OCCN2 C1(C(=O)NCCCOCCOC)CC(C)(C)CN1C(C1CCNC(=O)C1)=O c1(C(C)C(=O)NC(C)(C)CNC(C2(n3cccn3)CC2)=O)ccn(C)c1 C1(SC)C(C2CC2)CCN1CC(=O)NC(C)Cn1cc(-c2cncc(C)c2)nn1 C1(C2CC2)(NC(C(C)CF)=O)CCN(C(=O)C(c2cc(F)cc(Cl)c2)=O)C1 N1(C(CN(C(=O)OC(C)(C)C)CC)=O)CCC2(CC1)CN(C(C1CC1C1CC1)=O)C2 C(=O)(CCCC(=O)C1CC1)N1CC(OC(=O)NC)C1.c12cncnc1CNC2=O C1(CC=C)(NC(=O)CC2CCC2(C)C)CCCN(C(=O)CCc2cn[nH]c2)C1 c1(C2(C(=O)OC)CC2)csc(=NCc2ccc(OC(F)F)cc2)[nH]1 c1(C(=O)NCC(CNC(C(C)OCC=C)=O)OC)c(C)oc(Br)c1C c1(C(=O)NCCN(C(CC(CC)O)=O)C2CCCCC2)nc2ncccn2n1 C1(NC(C(C(C)C)O)=O)CN(C(c2ccnc(C(F)F)c2)=O)CC1(C)C CC1(C)C(CC(=O)NC2CCCCCC2)CCN1C(C1CCCOC1)=O CC1C(=O)Nc2ncccc2CN1c1ncnn1CCC(F)(F)F c1(CN2CCCC(NC(c3cnc(Br)s3)=O)C2)cc(F)c(Cl)c(Cl)c1 c1(OC)cc(C(N2CC(C(C)NC(C3(CO)CCC3)=O)C2)=O)ccn1 S(=O)(=O)(c1ccncc1C#N)NC(C(=O)Nc1c(SC)cccc1)C CCCC(CNC(c1ncn(C)n1)=O)C(=O)NCC(C1CCC1)OCC c1(NCC2CCN(C(=O)OC(C)(C)C)CC(C(F)(F)F)O2)nc2c(n1C)CCCC2 c1(OC)ccccc1NC(=O)C(N1CCC(NC(C2(CN(C)C)CCC2)=O)C1)=O CCC(C)(C)CC(=O)N1CC(CNC(c2csc(N3CCCC3=O)n2)=O)(OC)C1 C1(NC(c2c(OCCC)cccn2)=O)CCC(=O)N(CC(F)(F)F)C1 C1(C(N(CCCC(=O)N(CCOCCO)CC)C)=O)OCCC1(C)C C(C(C)(C)CC(C)O)NC(c1c(C)cnn1C)c1n(CCCOC)nnn1 CCCCN=C(NCC(c1ccc(OC)cc1)C)NCCN1C(=O)CCC1=O CC(C)C1=NOC(C(N2CCC(C)(CC(=O)NCCc3cncn3C)C2)=O)C1 CC(F)(F)CCC(C(=O)NCC(F)F)N1CCCC(NC(C2CC(F)(F)C2)=O)C1 C(C(C)(C)C(C)(C)C)NC(C1(C)C(C)C1)=O.C1C(=O)NCCO1 Cc1n[nH]cc1CCCNC(=O)C(CC1CCCO1)NC(=O)CN1CSCC1=O c1(CC)cc[nH]c1C(=O)NC(C(=O)NC1CC(N(C)C)C1)C1(O)CCC1 [N-]=[N+]=NC1(C(N2C3CCC2COC3)=O)CCN(C(C2CC(=O)NC(=O)C2)=O)C1 c1(C(N2CCC(O)(C(CNC(c3c(C)cns3)=O)C)C2)=O)ccc2cnnn2c1 C1(NC(C(CSC)C)=O)CN(C(c2cn(C3CCCCC3)nc2C)=O)CC1O Cc1cc(C)c(CCNC(=O)C(=O)NC(C)C(=O)OC(C)C)s1.C(N)(=O)N C(=O)(C#CC(C)(C)O)N1C2C(NC(C(C)OCC3CCCCO3)=O)C(C2)C1 C(=O)(CCCN(C)N=O)NC(CC)CNC(c1cccc(N2CCOCC2)n1)=O c1(CCC(=O)NC(CCCC)CNC(=O)COCCOC)cc(F)cc(F)c1 C1(C(=O)NC2(CC(=O)NOCC=CCOC)CC2)(SC)CC(=O)C1 Cc1ccc(Cl)cc1NC(=O)NC12CC(C(=O)NC3CC(CO)C3)(C1)C2 Cc1cnn(C)c1CC(=O)NC(C)C(=O)N(CCOCCCF)C(C)C C(=O)(C1CC(=O)N(C)c2ccccc21)NC1CN(C(CSCC)=O)CC(C)(C)C1 CC1(C)OC(=O)NC1C(=O)NC1CCN(C(=O)C=Cc2cncnc2O)CC1O c1(C(=O)NC2CCC(CNC(c3cncc(C)n3)=O)C2)cn(C)ccc1=O C(=O)(C(C)(C)C1CCN(C(=O)COc2ccn(C)n2)C1)NCCn1ncc(C)c1 c1(C(=O)OC)cc(C)n(NC(=O)N(C(CC(=C)C)C)CCOC)c1C Cc1cc(N2CC(O)(CCNC(C3CCCC34CC4)=O)C2)nc(Cl)n1 C1(CC(=O)Nc2csc(C(=O)OC)c2OC)C(OCc2ccccc2)CCC1O Cc1cc(C(=O)NCC2CCC(NC(c3c(Br)ncn3C)=O)C2)c(C)n1C c1(CC(=O)NCCC(CNC(C2=NOC(C)C2)=O)O)ccc2[nH]ccc2c1 C1(N(CCOC)CC)CCC(C)CN1OC(c1cccc(Cl)c1C)=O C1(C(N2CCC(CCOC)(NC(C3CCC(C)C3)=O)C2)=O)CC2OC1C1CC21 c1(OC)ccc2[nH]c(=NC3CCCC(C(=O)NC(=O)C(O)C(C)(C)C)C3)oc2c1 c1(CC2C(=O)N2)c[nH]c2ncccc12.C(C)(C(=O)OC)OCOC.C(C)(C)SC C1(OC)(CNC(C2CCN(C)CC2)=O)CCN(C(=O)C=Cc2ccc(C)s2)C1 C(=O)(C(C)(C(F)(F)F)NC(c1cc(C)cc(OC(F)(F)F)c1O)=O)OC C(=O)(C(O)CC(F)(F)F)NCC(CC(=O)NCCC(C)(C)C(F)F)C1CCC1 C(=O)(C1CCc2cc(F)ccc21)NCC1(O)CCCN(C(c2cn(C)nn2)=O)C1 CC1CN(C(c2cn(C(F)F)cn2)=O)CCN1C(=O)C(C)(O)C1CCC1 N1(C(=O)CC2(NC(C3CC(F)C3)=O)CC2)CC2(CCCC2)C1 N#Cc1cc(F)ccc1NC(C1(F)CCN(C(c2cc(O)cc(Cl)c2Cl)=O)C1)=O CC1CC(NC(c2ccsc2Br)=O)CCN1C(=O)CCc1ccccc1F c1(C(=O)Nc2ccn(Cc3cccs3)n2)ccc(C(F)(F)F)cc1Cl N1(C(C2(O)CCN(C(=O)C=Cc3ccsc3)C2)=O)CCC2COCC2C1 N1(C(C2C(C)(C)C2)=O)CCCCC12CN(C(c1cc(F)c(N)c(F)c1)=O)C2 N1(C(CC2CC(C)OC2C)=O)CC2CC1CN(C(=O)COc1cccc(F)c1)C2 C1(CNC(C2(CC3(CO)CC3)CC2)=O)CC(O)C(O)CC1C(=O)NCC(Cl)Cl c1(C(=O)NC(C(CO)NC(c2cc(CC)c(C)cc2)=O)C)ccc2nccn2c1 Cc1cccc(C=CC(=O)N(C(C)CN(C(=O)CCC2CCCN2C)C)C)c1 CC1CN(C(C2CCN(C)C(C)C2)=O)CCN1C(c1ccc(C(N)=O)nc1)=O C1(C(=O)NC(CN(C(Cc2n(C(C)C)cnn2)=O)C)C)CCN(C(C)C)CC1 CC1(C)CN(c2nc(C#N)ncc2Cl)CCC1NC(c1ccc(Cl)s1)=O C1(O)(CN(C(CCCSC)=O)C)CCN(C(=O)C(C)OC2CCOC2)C1 C1(c2cn(NCCC)nn2)CCC(F)(F)CC1.C1(C)COC1 C1(NC(C2(C)CCCN2C(c2cccc(Br)c2O)=O)=O)CCCC2CCCCC12 C(=O)(C#CC1CCCOC1)NCC1C2CN(C(C(OC)OC)=O)CC21 c1(CCNC(C=CC(C)NC(c2cc(CC)sn2)=O)=O)ncccc1C C1(C(N(C2CN(C(c3nc[nH]c4nccc3-4)=O)C2)C)=O)CCc2ncnn2C1 CC1(C(=O)NCC2(O)CCN(C(C3OCC3(C)C)=O)C2)CCOCC1 c1(C(=O)NCC(CC)(C)NC(C2CNC(=O)C2)=O)cccc(N)c1F N1(C(C(C(C)C)NC(C)=O)=O)CCCC(NC(c2cncn2CC(C)C)=O)CC1 Cn1c(=O)n(CC(=O)NC2CC(F)CN(C(=O)C(N)=O)C2)c2ccccc12 N1(C(C(C)CC2CC2)=O)CCCC12CCN(C(C1CCC3(CC1)CC3(F)F)=O)C2 C(=O)(C(CCN(C)C)NC(=O)Cc1cc(C)no1)N(C)Cc1scc(C)c1 N1(CCNC(C(COC)(C)O)=O)CCCN(C(=O)C=C2CCCCC2)CC1 N1(Cc2ccc(C)o2)CCC(O)(C(N2CCC(C(N)=O)CC2)=O)CC1 Cc1nn(CC(=O)NC(CNC(c2ccccc2Cl)=O)C2CCC2)c(=O)o1 c1(C(=O)Nc2cccc(NC(Cn3c(C)ccn3)=O)c2)cc(Cl)c(N)cc1F N12CC3CCN(CC3C1)Cc1cc(cc(Br)c1)C2=O.N(CCO)(CC)CC C12(NC(C(C)OCC3CCCO3)=O)CCCC1N(C(c1ncoc1C1CC1)=O)CC2 C(F)(c1ccccc1)=CC(=O)NCC(C)CNC(C1(C#N)CCC1)=O C(=O)(C(F)(CNC(c1cscc1OC)=O)C(C)C)NC(CC)C(C)(C)C C1(NC(CC2(C)CCCCC2)=O)CCN(c2ccnc(CO)n2)CC1O N1(C(c2c(F)ccc(C)c2)=O)CCC2CC1CN2C(c1cccc(F)c1)=O c1(NC(CNC(c2c(OC)cc(OC)s2)=O)C)nccc(C#N)n1 C1(C(=O)NCC2(COC)CN(C(=O)CCC3CCC(C)O3)C2)CCn2cnnc2C1 C=C(C)CCCC(=O)NCC1(COC)CN(C(c2onc(OC)c2Br)=O)C1 C1(NC(c2ccc(F)s2)=O)CCC2(CC1)CC2Nc1ncc2c(n1)COC2 CCC(O)CCNC(c1ccc(-c2cccs2)o1)=O C(=O)(C(F)(F)C1=CCOCC1)NCC1C(NC(=O)C2=NNC(C(F)(F)F)C2)CCC1 N1(C(c2c[nH]ccc2=N)C(=O)NCC2CCOC2)CCOCC(O)(C(F)(F)F)C1 N1(C(c2cn(CC)nn2)=O)C(C(N2CC3CCC3(C)C2)=O)CC2CCCC12 C1(C(=O)NC(C(=O)NCC23CCC(CO2)C3)c2ccco2)CC2CCC2C1 C1(CC(=O)NCCN(C(C(n2ccc(C)n2)C)=O)CCCN(C)C)CCCCC1O C1(CNC(C2N(CCC)CCC2)=O)CCC(C(=O)N(C(C)COC)C)CC1 CC1CC(NC(c2ccc(Cn3cc(Br)cn3)o2)=O)CN1C(=O)CC(F)(F)F C1(C(=O)NC2CC(NC(C(C)CC3CCCC3)=O)C2)CCc2ncc(Br)n2C1 c1(C(N(C)CC2N(C(C(C)C3CCCC3)=O)CC(F)C2)=O)ccc(=O)n(C)n1 C12(C(N(C3CCCCC3)C)=O)CCN(C(c3ccncc3Cl)=O)CC1C2 C(=O)(CC(C)C(C)C)NCC1(C(=O)NCC(C2CC2)OC)CCC1 c1(C(=O)NC2CC(C)N(C(c3ccc(=O)oc3)=O)C2)cc(F)c2c(c1)CCC2 C1(C2(C)CC2)COCCN1C(=O)CC(CC1CC1)NC(C1COC(=O)N1C)=O c1(C(=O)NCC(CCC)NC(=O)CCc2cnn(C)c2)ccc(=O)oc1 N1(C(CC=CC)=O)CCCC2CN(C(c3ccc(C(=O)OC)o3)=O)CCC12 N1(C(Cc2ccc(OCC=CC)cc2)=O)CCC(NC(=O)C(F)OC)C(C)C1 C(=O)(C1=C(C)OCCC1)N1C(NC(NOCC(CC)C)=O)CC(O)C1 C(=O)(CCCC(C)C)N(CCC(C(C)C)NC(c1oc(C)c(CO)c1)=O)C C1(NC(C2(CC#C)CCCO2)=O)CC2CN(c3ncnc(C)c3F)CC2C1 c1(CC)ccc(CC(=O)NCC2CC(CNC(=O)CN3CC(C)C3)C2(C)C)cc1 N1(CCN(C(C2(C#C)CCC2)=O)C)CCN(C(=O)CC2CC3CCC2C3)CC1 N1(C(=O)CNC(CNC(CSC)=O)=O)CC2(CCCC2)C1C(N1CCCC1)=O C(=O)(CC(C)(O)COC)N1C(C(=O)NC(c2n[nH]c(C)n2)C)(CC)CCC1 N1(C(C(=O)N(C)C)=O)CC2(CCOCC2)C1c1cn(CC2CC3(CCCC3)C2)nn1 C(C(C)(C)CNC(c1ccncn1)=O)N(C(C1C(C(=O)OCC)C1)=O)CC C(=O)(C1=NNC(=O)C1)NC1C(NC(c2n(C)nc(C3CCCC3)c2)=O)CC1 c1(CC)cc(N)ccc1C(N1CCC(C(C)CNC(=O)C2=CC(C)(C)C2)CC1)=O Cc1cc(F)cc(C)c1C(=O)NC1CCN(Cc2ccc(F)cc2Cl)CC1F CCCC(C(=O)N1CCCCC1CNC(c1ccc(C)[nH]1)=O)C(C)C N1(C(CCN(CCC)C)=O)CCOCC1CC(=O)NCC1CC12CC2 c1(C(=O)N)cnn(CCN(C)C)c1.CC(C)CC1(CC(=O)NC)CC1 N1(C(c2cccc(C(C)C)c2)=O)CC2CC(NC(C3(F)CC=CCC3)=O)C(C2)C1 C(CC(=O)Nn1cnnc1C)C1CCCN(Cc2ncnc(C)c2C)C1 c1(C(=O)NCC(C)(C2CC2)NC(=O)COC2CCCOC2)cccnc1N C1(c2ccc(OC(C)(C)C)cc2)CCN(C(=O)CC2C=CCC2)CC1SCC(=O)O CC1CC(C(=O)NCCN2CCCCC2)CCN1C(c1cnn[nH]1)=O c1(-c2ccc(CCOC)s2)ccc2[nH]nc(C(=O)N(CC#N)CC#N)c2c1 C1(NC(Cc2c(CC)con2)=O)CCC12CN(C(=O)C(C(C)(C)C)N(C)C)C2 c1(C(=O)NCC2CCN(C(C)(C)C)C(CCO)C2)ccnc2[nH]cnc12 c1(NC(=O)NC2C(C(C)C(=O)O)C2)cc(Cl)cc2c1OCC(=O)N2 c1(C(N2C(CNC(c3ccc(OC)c(C)c3)=O)CC2)=O)cc(F)c(Cl)cc1Cl Cc1cc(NC(C(C)(C)C(C)C)c2nnnn2CC2CCCO2)cc(Cl)c1 N1(C(=O)NC(CC)=O)CCC(C(=O)NNC(=O)OC)CC1.c1ccccc1 C1(C(=O)NCC2CN(C(C)=O)C2)(OC)CCN(C(c2cnsn2)=O)C1 CCC(CCC(=O)N(C)Cc1nc(=O)o[nH]1)NC(C1CC1(C)C(C)C)=O C1(C(=O)OC)CCCN(C(=O)Cc2cc(C)ccc2OC)CCC1 CC1(C)CC(CNC(=O)CNC(c2ccsc2)=O)N(C(=O)C=C(Cl)Cl)C1 C1(CC(N2C(C)(C(=O)NC)CC2)=O)CC2(C1)CN(C(C1CCCCN1C)=O)C2 C1(C)CCC(=O)N1.N1(C(C(c2ccoc2)OCC)=O)CC(F)(F)C1 C1(C(=O)O)CCC2(CC1)CC2.c12cccc(c1)C(=O)NCC(O)Cc1cn-2nn1 N12CCC(O)(CC1)C2=O.Cc1cc(CC(N2CCC(CO)CC2)=O)ccn1 N1(C(C(C)OCCOC)=O)CCC(CC2CCN(C(C3(F)CC3C)=O)CC2)CC1 C1(C(=O)NC2C=CCN(C(c3nccc(C)c3)=O)C2)CC2CCCCCCC12 C1(NC(c2ccc(-c3cccs3)o2)=O)CC12CCN(C(=O)CC1=CCCC1)CC2 CC1(C(=O)NCCC2CC(C(=O)NCc3cccs3)C2)CCCC1 C1(C(=O)NCC(C)CN(C(=O)CC2CCOCC2)C)CCc2nnnn2CC1 CC(C(=O)N1CCC(CO)(NC(c2cnc(-c3ccc(Cl)s3)s2)=O)C1)C(C)(C)C C(c1ccc(F)c(F)c1)=CC(N1CC2CCC1CN2C(c1cc(Cl)c(Cl)s1)=O)=O N1(C(C2(C(=O)NC)CC2)=O)CCCCC(NC(c2cc(F)ccc2C)=O)CC1 c1(CC(=O)NCC(C)(C2CCC2)NC(C2CC2C(F)(F)F)=O)cc(F)ccc1F N1(C(c2cc(C(N)=O)[nH]c2)=O)CC2CCC(C1)N2C(=O)CSC(F)F C1(NC(CCCC(CC)C)=O)CS(=O)(=O)C2CN(C(=O)C3=C(C)CCC3)CC12 C1(NC(C(CC)(C)C)=O)CCN(C(c2ccc(F)c(OCC)c2F)=O)CCC1CO N1(C(C=CCC(C)(C)NC(c2cc(C)n(C)n2)=O)=O)CCN(C)C2CC12 C1(C2CCOCC2)(C(N(C)CC2N(C(CCSC)=O)CCOC2)=O)CC1(F)F C1(OC)CN(C(C2CC(F)(F)C2)=O)C(C)(CNC(c2ccoc2C)=O)C1 c1(N2CCC(C(N(c3csc(C)c3)CCC)=O)CC2)cc(=O)n(C)cn1 N1(C(C2C3CN(C(C4C=C(C)CS4)=O)CC32)=O)CCCC12CCNC2=O C(=O)(CS(=O)(=O)C1CC1)N1CCC(F)(CNC(CCC2C(C)C2)=O)C1 C1(C(N2CC3CC2(C(=O)NCc2cc(Cl)ccn2)C3)=O)(CC)CC(C)(C)C1 CN1CCCCC1CC(=O)NC1(C(=O)NC2COC(C(F)F)C2)CC(O)C1 N1(C(C2(C(C)C)COC2)=O)CC2CC(NC(=O)CC(=O)NCC(F)(F)F)CC1C2 c1(OC)cscc1C1c2nnnn2CCCC(C2CC2)N1.C1(SC)CC1 C1(CNC(c2ccc(SC)o2)=O)CC1C1CCCC1.c12c[nH]nc1C(=O)NC2 N1(C(c2ncc(C)cc2F)=O)C2CCC1CC(CNC(C1(CC3CC3)CC1)=O)C2 C1(CN(C(=O)Cc2cn[nH]c2)C)CC(F)CN1C(=O)CCOCC(F)(F)F n1(CC(=O)NC2(C3CN(C(CN(C4CC4)CC)=O)C3)CC2)c([N+](=O)[O-])cnc1C CCCCCCC(C)C(=O)N1CC2CC(C1)CN(C(=O)C(O)CC[S+](C)C)C2 C1(C(=O)NC2CC(NC(c3[nH]cc(C(C)=O)c3)=O)C2)CC2(C1)CC2(F)F C(=O)(CC(C)CC)NC(CC)CNC(C1CCN(c2ccncc2)CC1)=O c1(C(=O)NCC(C)CNC(c2n[nH]cc2C2CC2)=O)ccc(F)c2cccnc12 c1(C(=O)NC2CC(CNC(C3CC(=C)C3)=O)C2)cc2cc(Cl)ccc2n1C C1(NC(C(C)NC(N)=O)=O)CC2CC1CN(C(c1cc[nH]c(=N)n1)=O)C2 C1(C)(NC(CC(C)(C)F)=O)CCCN(C(c2ccc(CNC(N)=O)o2)=O)C1 C(=O)(CS(=O)(=O)CCO)N(CCC(C)NC(c1c(C)nc(CC(C)C)o1)=O)C CC(O)(CNC(=O)CCNC(=O)COC(F)F)CNC(C1(C#N)CC1)=O Cc1ccc(Cl)c(C(=O)NC2CC2CNC(c2cn(C3CC3)nc2C)=O)c1 c1(CC(=O)NC2CC(F)(CNC(CCCC)=O)C2)cccc2c1OCO2 C1(CCC)CN(C(=O)CSc2ccccn2)CCN1C(=O)C(F)n1cccn1 c1(OC)cc(C(=O)NCC2CN(C(C3SCCS3)=O)CC2O)c(F)c(Cl)c1 C1(CNC(C2CCN(C(C)=O)C2)=O)CC2CCC1N(C(=O)CCCC(F)(F)F)C2 C(=O)(CCS(N)(=O)=O)NCc1c(C(=O)NC(c2ccncc2)C)[nH]cc1 c1(N(C)C)c(C(=O)NC(CNC(=O)CC(F)F)C2CC2)cnn1C C1(NC(C2C3(CN(C(c4c(C)oc(C#N)c4)=O)C3)CC2)=O)CCc2n[nH]cc2C1 C#CC1(C(=O)NCCC(C)(C)NC(=O)Cc2cscc2Br)CCCC1 CC1CN(C(c2cc(Br)cc3cn(C)nc23)=O)CC2(CCOCC2)O1 c1(C(=O)NCCCCC(C)NC(=O)CCc2nc[nH]n2)cnc2[nH]nnc2c1 c1(C(=O)OC(C)C(N2CCN(c3ccc(Cl)cc3)CC2)=O)cc(I)ccc1Cl N1(C(C2CC(NC(CCC3CCC(=O)C3)=O)C2)=O)CC2CCC(O)C(O)C12 c1(OC)ccc(CNC(=O)C(c2cccnc2)Nc2ncc(C)s2)cc1 CN1C(=O)CCC1C(=O)NC1(CNC(=O)CCCc2cnccn2)CCOCC1 N1(C(COCCOC)=O)CC2CCN(C(=O)C(C3CCCN(CC)C3)(C)C)C2C1 c1(C(=O)OCCN(CCCN(C(=O)CC)CC=C)C)ccc(OC(F)(F)F)cn1 c1(C(C)=O)nnc(CNC(=O)NC2CC(OCC(C)(C)C)C2)n1-c1ccccc1 c1(C(N(CCOCC#C)C(C)C)=O)cscc1Br C1(C)(NC(c2n(CC(C)C)ncc2)=O)CCCN(C(c2cc(O)nn2C)=O)C1 CS(=O)(=O)c1ccc(C(=O)NC23CC2CN(C(c2ccc4c(c2)CCO4)=O)C3)o1 c1(CC)nc(N(C)Cc2ccc(CNC(=O)CCS(C)=O)cc2)c(F)c(Cl)n1 CCCC(C(=O)NC)NC(C1CCN(C(c2cc(CO)n(C)n2)=O)C1CCC)=O C(=O)(CCC(O)C(C)(C)C)N1C(CCC)CN(C(=O)CCc2ccn(C)c2)CC1 C1(SCC)CCC(C(=O)NC2CN(C(=O)CC3C(=O)ON=C3C)CC2O)CC1 N1(C(CSC(C)C)=O)CCCC(C2CCN(C(=O)C=CCOCC(F)(F)F)C2)C1 C(C(C(F)(F)F)N1CCN(C(=O)C(O)C2CC2)CC1)NC(C1(CC(C)C)CC1)=O C1(CC(N2CC3C(NC(c4cc(F)ccc4Cl)=O)(C3)C2)=O)CC2CCC(C1)C2 c1(C(N(CCN(C2(CC(=O)N)CC2)C)C)=O)ccccc1OCCOC.CO C(CC(C)(C)CC(=O)N(C(CC(F)F)C(=O)NC)C)OC.C1(OC)(OC)CCCCC1 C(=O)(C1CCCc2n[nH]cc21)NC1(C)CC(NC(c2ccoc2)=O)C1 c1(C(C)=O)cc(NC(C2CCN(C(C3CCCCO3)=O)CC2O)=O)ccc1F C(CCN(C)C(C1CC12CCCCC2)=O)(C(C)(C)C)NC(C(CC)CC)=O C1(COC)(CNC(c2cnnn2C)=O)CCCN1C(=O)CC1CCOC1C C1(NC(C(C(CC)C)O)=O)CC2(CCN(C(c3nocc3C)=O)C2)C1 N1(C(C2C(C)N(C(=O)C3=CCSC3)CC2)=O)CC(O)(C2CC2)C1 N1(C(CC2(OC)CCC2)=O)CCN(C(C2CC3CC3C2)=O)C(CF)C1 c1(C(N2CCC(N(C(C(C)=C3CCCC3)=O)C)C2)=O)ccn2ncc(C)c2n1 C12(C(=O)NCC(COC)(F)F)CCC(NC(=O)C(F)OC(F)(F)F)(CC1)C2 Cc1nc(O)ccc1C(N1CCC(C(C)C(=O)NC(c2cnn[nH]2)(C)C)C1)=O C1(CNC(=O)Cc2cccs2)C(C2CC2)CCN1C(c1cc([N+](=O)[O-])c[nH]1)=O C(CC#CC)(C(=O)Nn1cncn1)NC(CCC#C)=O Cc1cc(C(F)F)oc1C(N1CC(O)(C2CCCN2C(C2CC2(F)F)=O)C1)=O CCC(C)(CCC(C)C)C(=O)N1CC2CC2(CNC(c2ccc(Cl)c(O)c2)=O)C1 N1(C(CN2CC(C)(OC)C2)=O)C2CCC1CC(NC(C1(C)CCC(=O)N1)=O)C2 C(C(CC1CC1)C(=O)NCCC1(O)CCC1)NC(COC(CC)(C)C)=O N1(C(c2c(C)ccnn2)=O)C(CNC(=O)CC2CCCCN2C)CC2CCCC12 N1(C(c2cc(C)oc2)=O)CC2(CCCC2)C1C(=O)NCCC1=CCN(C)CC1 CCS(=O)(=O)C=CC(=O)N1CCC(CNC(=O)C(C)(C)NC(=O)C=COC)C(C)C1 C(=O)(CCS(=O)(=O)CC(F)(F)F)NC(CC)CNC(c1cnn2c1OCC2)=O C1(C(=O)NCC23CC2CN(C(c2c[nH]c(C(F)(F)F)c2)=O)C3)(CC)CCNC1=O c1(C(=O)NCCC(C)(C)NC(=O)CSC2CCOC2=O)cccnc1N C(=O)(C(C)(C)CC(=O)N1CCC(O)(CNC(c2cc(Br)n(C)c2)=O)C1)OCC c1(C(=O)NCC(C2CC2)NC(C(C)(C)OC(C)=O)=O)cccc2c1OCC2C C1(C(=O)NCC2(C(N3CCC(C(N)=O)C3)=O)CC(O)C2)CC2CCCC2C1 CCC(C(=O)NCC1CCC(C)CN1C(C1CN(CC(F)(F)F)C1)=O)C(F)(F)F CC1(C(=O)NC2COCC2NC(c2ccc3cc[nH]c3n2)=O)CCCCCCC1 C1(NC(C2C(C)OCC2)=O)CCCCN(C(=O)CN2CCSCC2)C1 C(=O)(C(C)(C)CC(F)F)NCCN(C1CCCC1)C(C1(C=C)CCC1)=O CN1CC(C)(C(=O)NC2CCC2CNC(C2CC(O)C2)=O)CC1=O c1(C(N(C(CCNC(C(C)NC(C)=O)=O)C)C)=O)ccc2c(c1)CCCCS2 c1(C(=O)NCC(C)(C2CC2)NC(C(CC)OC)=O)ccc2occ(C)c2c1 Cc1oc(Br)cc1C(N1CCC(C)(NC(c2cc(C(F)(F)F)cs2)=O)C1)=O c1(NC(C(C)OC(c2c(-c3ccc(F)cc3)nc(C)s2)=O)=O)cc(C)c(C)cc1C c12cc(cnc1Cl)-c1cccc(c1)N(CC)C2.N1(CC)CCN(C)CC1C c1(C(=O)NC2C(CNC(C3(C=C)CC3)=O)CCC2)cnn(CCCC)c1C C(=O)(CCCCC(C)(C)OC)N1CC(F)(CNC(c2c(CC)con2)=O)C1 C(N=C(NC1CCCC1)N1CCC2C(C1)NC(=O)N2C)c1c(OC)nccn1 N#Cc1cncc(C(=O)NCCOC2CCN(C(=O)C(c3cccnc3)O)C2)c1 C(CNC(c1cncc(Cl)c1)=O)(CCCC)NC(CC=C=C)=O c1(C(=O)NC2(CO)CCN(CC)CC2)c(-c2ccnc(COC)c2)cc(F)cc1F c1(C(=O)NC2CC(C)N(C(=O)C(=Cc3cccnc3)F)C2)ccnc2ccsc12 c1(NC(c2n[nH]cc2NCc2cc(F)c(Cl)c(Cl)c2)=O)ccc2ccccc2n1 N1(C(Cc2cnc(C)[nH]2)=O)CCC(C)(CNC(c2ccccc2F)=O)CC1 C(=O)(CCC(=O)NC12CC(NC(=O)C(C)(O)COC)(C1)C2)N(CC)CC Cn1ccc2ccnc(C(=O)NCC3CCCCN3C(=O)CCc3cscn3)c12 C1(C(=O)NC2CCN(CC=C)CC2)CN(C(C23CCCC2C3(F)F)=O)CC1(C)C C(C)(CNC(c1nscc1C)=O)(CC(C)C)NC(c1ccc(COC)o1)=O N#Cc1cc(S(=O)(=O)NC2C3CCCCC23)ccc1NC1CCN(CC(F)F)C1 c1(CN(C)CC2CCN(C(c3nccnc3Cl)=O)C2)ccc(Cl)c([N+](=O)[O-])c1 CC(F)(F)CCC(=O)NC1C2CC1N(C(c1cccn1Cc1cccs1)=O)C2 c1(N(CCCNC(C2(CC)CCCCC2)=O)C2CC2)c[n+]([O-])ccc1[N+](=O)[O-] C12(CC)CNCC(C(=O)Nc3cccn(Cc4ccccc4)c3=O)(C1)C2 N1(C(CCSCC)=O)CC2(C1)CN(C(c1c(S(=O)(=O)NC)cnn1C)=O)CCO2 C(CCCCC(=O)N1CCC(CNC(C2(CF)CCC2)=O)C1)n1c(CC)nnc1 C1(CC(=O)NC2(CCCNC(c3cc(Cl)cnn3)=O)CC2)CCCC(C2CC2)O1 N1(C(CC(C)SC)=O)CC(C(=O)NC(C)(C)CC(C)C)CC(C)(C)C1 c1(C(=O)NC2C(CN(C(C3C(C(C)O)C3)=O)C)CCC2)nn(C)cc1Cl N1(C(c2ccc(C#C)cn2)=O)CCC2CCN(C(=O)CCSCCC)CC2C1 N1(C(c2c(C)noc2)=O)CCN(C(C2CCOC2C)=O)CC1CCO C(=O)(C1=CCN(C(c2c[nH]c3cccnc23)=O)CC1)NC(C)CSC(F)F N1(C(C2CN(C(C)=O)C2)=O)CCC(C)C(CNC(c2cscc2Cl)=O)C1 c1(CN(C)C(c2[nH]ncc2C#N)=O)cnn2c1CN(C(C1(CO)CC1)=O)CC2 c1(OC)cc(SC)ccc1C(N1CC2CC2(C(=O)Nc2cc(C)no2)C1)=O Cc1ccc2c(NC(C3CC3C(=O)NC3(n4cc(Br)cn4)CC3)=O)cccc2c1 CCC(C)CC(=O)NCc1cc(C(=O)NC2C3CCCC23)ccn1 c1(CC)cc(C(=O)NCC2(F)CC(CNC(c3n[nH]c(C)c3C)=O)C2)cc(O)n1 C(=O)(C(O)(C(F)(F)F)C1CC1)N1CCC(CCNC(C(C)OCC)=O)CC1 c1(CCC(=O)NC2CC(NC(C(C)Oc3ccccc3F)=O)C2)cncnc1O c1(C(=O)OC)cc(Br)cn1C(C)C.c12ccc(s1)CNC(=O)C2 C12(C(N(C)CCNC(C3CCS(=O)(=O)CC3)=O)=O)CCC(C)(CC1)OC2 N1(C(C2C(C#N)C2)=O)CCN(C2CCCC2NC(c2cc(Br)co2)=O)CC1 C(=O)(C=CS(C)=O)NC1C(NC(C(=Cc2cccs2)C)=O)COC1 C(CC(O)C(=O)NCc1cccc(O)n1)NC(C)=O C1(NC(=O)C2CC2)CN(C(C2CC(C(F)F)C2)=O)CC12CCOCC2 c1(C(=O)NCC(CNC(C2CC(CC)NC(=O)C2)=O)C)cnc2ccnn2c1N c1(CC)c(NC2(C)CCC(NC(=O)C=CI)CC2)ncnc1Cl c1(C(=O)NCCN(C(=O)CCc2cccc(F)c2)C)ccnn2ccnc12 c1(C(=O)NCC(CNC(c2c(C)nco2)=O)(C)O)cc(S(=O)(=O)N(C)C)c(C)o1 c1(N(CCc2ccc(OC)cc2OC)C)ncnc2c(Br)cc(Cl)cc12 c12cc3ccc(cc3o1)-c1c(noc1C)C2.C1(CC)CCCN(C(=O)C2CC2)C1 CC1CC2(CCO1)CCN(C(=O)C(N1CC(CO)OC(C)C1)=O)C2 CCC(C(=O)N1CC(c2ccncn2)C1)N(C(=O)C(C)CC1CCCC1)C N1(C(C2(OC)CCC2)=O)CCC(C(=O)NC(c2cnn(C)c2)C)C(C)C1 c1(C(=O)NC(CC)CN(C(=O)CC2CCCCC2F)C)cccc2[nH]ccc12 c1(CN2CCC(NC(=O)OC(C)(C)C)(CO)CC2)c(F)ccc(Cl)c1F C(=O)(C(CC(=C)C)OC)NC1CCC(CC(=O)N(CC(C)C)CC#C)C1 N1(C(C(C)OC2CCOCC2)=O)CCC(NC(c2cc(O)ccc2F)=O)C(O)C1 c1(C(CC(=O)NC(C2CC(F)(F)C2)C)C2CC2)ccc(Br)c(F)c1F C1(CC(=O)NC(C)(C)C(=O)NCCC2CCC3CC23)CCCCC1O c1(C(N2C(C(N3CC(C(=O)OC)OCC3)=O)CC(C)C2)=O)cc(C)nc(Cl)c1 N1(C(C2(C)CC(O)CN2C(=O)CC2CCC2)=O)CCc2nnnn2CC1 c1(NC(C2CC(=C)CN2Cc2cc(C)nn2C)=O)ncc(I)cc1I n1(CC(=O)NCC(C)CNC(c2cc(CO)[nH]n2)=O)ccc2cc(F)ccc12 CC(C)(C)CC(O)CC(=O)N1CC(F)CC1C(=O)NC1CCCCC1(C)C C1(NC(C(CC)(C)CNC(=O)CC2CCCCC2O)=O)CCC(=O)NC1(C)C c1(OC)cc(C(=O)NC2CN(C(=O)C(c3ccccc3)C)CC2F)ncn1 C(=O)(C1=CCCCCC1)N(CCNC(c1c(C)n(CC(F)(F)F)nc1)=O)C(C)C C1(c2nnc(C)o2)CCCCCN1C(c1cnn(C)c1)C(=O)NCC(F)F Cc1nn(C)c(C)c1CC(N1CCC(C)(NC(=O)CCc2nc[nH]n2)C1)=O c1(C(N2CC(CN(C(C(C)SC)=O)C)OCC2)=O)cnc2ccnn2c1 C(=O)(C(C)S(N)(=O)=O)NC(C)CC1CN(C(c2cc(C3CCCO3)n(C)n2)=O)C1 C1(CNC(CC2C(N)CC2)=O)C2CC3CC(C2)CC1C3 CC(C)C(C(=O)NCC1CCCN1C(c1ccn(C2CC2)n1)=O)c1cccnc1 O=C(CCCCC1CCNCC1)NC1CCN(c2ccccn2)C1 Cc1nc(Br)ccc1C(=O)NCC1CC(C)N(C(c2c(N)cccc2F)=O)C1 N1(C(C=CC)=O)CCC2(CCN(C(c3cnn4c3CN(C)CC4)=O)CC2)C1 C(CCCC(=O)NC(C(=O)N(C)Cc1ncc(C)o1)C1CC1(C)C)N(C)CC C1(COC)(NC(=O)C(C(C)(C)C)SC)CCCN(C(c2cc(F)c[nH]2)=O)C1 N1(C(C2CCC(NC(c3ccoc3Cl)=O)C2)=O)CCC(O)(CO)C1 N(C1CN(C(=O)C(C)S(C)(=O)=O)Cc2ccccc21)C(c1cc(C)c(C)[nH]1)=O CCC(C)C(CC(=O)NC1CCn2nccc2C1)NC(C1CCCSC1)=O C1(NC(CN(C)S(N)(=O)=O)=O)C2CCC1CN(C(c1cccnc1Br)=O)C2 C(=O)(CCC(=O)N(CCNC(C1(C#N)CC1(C)C)=O)CCOC)NCC CC(C(=O)N1CC2CC(N(C)C(c3coc(Br)n3)=O)C1C2)C(C)(F)F N1(C(c2cnc(C)s2)=O)CCC2CC2(C(=O)NC(C)(CO)CO)CC1 C(=O)(C(C)(CC)CCCCCC)NCC1CCN(C(C(F)=CCC)=O)C1 N1(C(C2(CNC(CC(C)N(C)C)=O)CC2)=O)CC(C(=O)N(C)C)CC1(C)C c1(CSc2cn(C)nc2)ccc(Oc2ccc(C(N3CCCCC3)=O)nc2)nc1 Cc1cc(Br)cn2c(CN3CCCNC(=O)C3C)cnc12 C(=O)(C(C)(O)C(F)(F)F)N(CCNC(C(Cc1ccc(F)cc1)OC)=O)C Cc1cnccc1C(=O)NC1CCC(C)(CNC(=O)CC=CC(C)(C)C)C1 c1(C(=O)NC(C2CCCC2)CNC(CC(C=C)CC)=O)ccc2cccnn12 N1(C(CCC(CC)C)=O)CCC(C2(NC(=O)C(COC)N(C)C)CC2)CC1 CCC(C)(C)CCCC(=O)N(CC(CC)NC(=O)COc1ccsn1)C C1(C)(C(=O)NCc2onc(C)n2)CCCN(C(C2CC2C(N)=O)=O)C1 c1(C(N(C2CCN(C(c3c(CC)non3)=O)CC2)CC)=O)[nH]nc2ncccc12 C1(C(=O)NCC(C)NC(=O)CN2C(=O)C(=O)N(C)C2=O)CCC2(CC1)CC2(F)F N1(C(C2(C)CCCOC2)=O)CC2(CCC2)CC1CNC(c1ncc[nH]1)=O c1(CC(=O)NCC2CC(NC(CCCc3nc(C)sc3)=O)C2)ccc(C)cc1F CC1(C)CN(C(=O)C2=C(Cl)CC2)CCC1NC(=O)C(C)(C)c1cnccn1 CC1(C)CC2CCCOC12.C1(CS(=O)(=O)Nc2nc(SC)n[nH]2)CC2(CCC2)C1 C1(CNC(C(CC)C(C)C)=O)CC2(CO1)CN(C(C1CC3(C1)CC(C)(C)C3)=O)C2 C1(CNc2ncnc(CC)c2F)C(C)CCCN1C(=O)C=C(C)C(F)F C1(NC(c2cn(CCC)nc2C)=O)CC2CC1N(C(C1CN3CCC1CC3)=O)C2 CCCC(C)(CC)C(=O)N1CC2C(CNC(=O)C(F)(F)C(O)CC)C2C1 C1(N(C(c2n(COC)ncc2)=O)C)CCCC(N(C(=O)C=Cc2cc[nH]n2)C)C1 Cc1noc(C)c1C(=O)NC(C)CCNC(=O)COCC1CCC1 O=C(NNC(=O)c1cccc(-c2ccccc2)c1)NCC(C(F)F)n1cncn1 C(=O)(C(C)C(O)C(C)C)NC1(C(=O)NCc2cc(C(=O)OC)no2)CCN(C)C1 CC1CC(O)CN(C(C2CC(NC(c3c[n+]([O-])c(C)cn3)=O)C(O)C2)=O)C1 C12(C(N3CCCC(N(C(CN(C(C)=O)C)=O)C)CC3)=O)CCC(=O)N1CCS2 c1(C(=O)NC(CC)CN(C(=O)COCCO)CC)c(OC)c(Cl)cc(O)c1Cl CC1CN(C(c2cc(F)n(C)n2)=O)CCCN1C(C1CCCCC12CC2)=O c1(C(=O)NC2(CNC(CC(CC)OC)=O)CCOC2)cc(Cl)ccc1N c1(SCC)ccc(NC(=O)CN2CC(C(=O)OC)C2)cc1 c1(C(=O)NCC23C(CN(C(CC(=O)OCC)=O)C2)C3)ccnc2[nH]cnc12 c1(CN(C(C2CCCN(C(c3cnnn3C(F)F)=O)C2)=O)CC)cccc(Cl)c1 Cc1nccnc1-c1cn(C2CCCC2NC(=O)C(C)(C2CCCC2)N(C)C)nn1 N1(CCNC(C2N(CC)CCC2)=O)CCCN(C(C23CC4CC2C3C4O)=O)CC1 c1(SC)cccnc1C(N1CCC(C(F)F)(CNC(C2NC(=O)OC2C)=O)C1)=O N1(C(c2n(CC)cc(Cl)c2)=O)CCCC(C2(NC(C3CC4(C3)CC4F)=O)CC2)C1 C1(CNC(c2cccc(OC)c2F)=O)CCCC2(CCOCC2)O1 n1(CCOC)nnc(C(=O)NCC(C)NC(=O)C(c2cccnc2)O)c1C(F)(F)F N1(C(c2nc(C)sc2C)=O)CCC2C(CCN2Cc2ncc(C(C)C)o2)C1 N1(C(C=CCOCCOC)=O)CC=CC(NC(c2ccncc2)=O)C1 c1(CC)cc2c(NC(c3cccnn3)C(C)C)ncnc2s1 N=c1[nH]c(=NCC(CO)OC(F)F)[nH]c(=NC2CCCN(CC(N)=O)C2)[nH]1 N1(C(C(F)=CCC)=O)CCC(NC(=O)CC2CC3(CCC3)CCO2)C(C)(C)C1 c1(OCCCOC)ccc(NC(c2cc(C)n(C)c2)c2nnnn2C)cc1 N1(C(CS(CC)=O)=O)CCC=C(C(=O)NC(CCCCl)c2ccccc2)C1 Nc1ccc(-c2cn(C3CCCC3NC(c3cnncc3O)=O)nn2)cc1F C1(C(C)C)C(NC(=O)COC2CCCCC2)CCN1C(=O)C=CC1CCCC1 N1(C(C2C(CCC)CCC2)=O)CCC(C)C(NC(=O)CC2(O)CCOC2)C1C n1(CC(=O)NCC2C(CNC(C(c3ccc(Cl)s3)C)=O)C2)cc(CC2CC2)nn1 c1(CNCC(C)(C)NCCSC)nnn(C)c1C(F)(F)F c1(C(=O)NCC2C(C)CN(C(=O)CC3CSCCO3)C2)ccc(O)c(Cl)n1 C1(C)(C(=O)NCC2CC(=C)C2)CN(C(c2nc(Cl)cs2)=O)CC1C C1(F)(C(N(C)CC=Cc2ccccc2)=O)CCCN(C(C2CCCCC2O)=O)C1 c1(C(=O)OC)csc2c(NC(=O)C(=O)NCCN3CCOCC3)cccc12 c1(CC(C)C)nccc(C(=O)NC(C2CCCN2C(=O)CC2(C)CC2)(C)C)n1 C1(C)(C(N2C3C(C2)C3=O)=O)CCOCC1.C(C)(C)(C)O.C(=O)(OC)NCCSC C1(NC(C=CCC)=O)CN(C(C2CC2c2cnccc2C)=O)CC2(CCC2)C1 C(N=c1[nH]cnc2c(Br)nn(C)c12)C1(OC)CCC(C)(C)CC1 N1(C(C(C)CO)=O)CCc2ccccc2C1CNC(=O)C(c1cnn(C)c1)O CC1(C)C(NC(c2cccc(O)n2)=O)CCN1C(c1ccc(C(N)=O)cn1)=O c1(C(N(CCCNC(c2nccc(OC)c2N)=O)C)=O)nccc2cnn(C)c12 c1(NC(CN2CCN(C(C3CCN(C)C3)=O)CC2)=O)cccc2cc(Cl)cnc12 C(=O)(C1COCc2ccccc21)N(C)CC1OCCN(C(CCC=C)=O)C1 CC1(CNC(C2CCCC(CC(F)(F)F)C2)=O)CCN(C(C2(C(N)=O)CC2)=O)CC1 C(c1ccccc1Cl)=C(C)C(=O)NCC(O)CN(C(=O)C(C)(O)C(C)C)C C1(C(=O)NC(C(=O)NCc2c(OC)nsc2)(C)CSC)CCCCC(=O)C1 C(=O)(C(CC1CC1)NC(=O)CCCn1cccn1)N(C1CCCC1)CCC c1(SC(C)C(N2CC(CNC(=O)CC(F)F)CC2(C)C)=O)ccc(F)c(F)c1 c1(C(=O)NC2C3CN(C(c4c(C)nn(C)c4C)=O)CC32)coc2c1CS(=O)(=O)C2 N1(C(c2nc(C)oc2)=O)CC=C(CNC(=O)Cc2c[nH]nc2C)CC1 C1(NC(c2c(N)cncn2)=O)CCCCN(C(=O)Cc2cccnc2Cl)C1 C1(SC)CCCC(NC(=O)COCCNC(C2CCCCC2O)=O)C1 C(=O)(CC(C)CN(C)C)NCCN(CCCN(C)C)C(C1C(C=C)CC1)=O C1(C(=O)NCCC(C)(C)C2CC2)CCCCC1CNC(C1(F)CC1(Cl)Cl)=O CCC(C)(C#N)C(=O)N1CCC(C(C)NC(=O)CC(C)(C)OC)CC1 C1(O)(CNC(=O)C2=CCCS2)CCN(C(=O)Cc2cc[nH]c(=N)c2)CC1 C(=O)(C(CO)C(C)C)N1C(C2CN(C(C3CCC(CC)O3)=O)C2)CCC1 c1(C(=O)NC(CC)CNC(=O)COCC(F)(F)F)ccnn1Cc1ccccc1 C(=O)(C(C)(C)CNC(C1CN(C(C)C)C1)=O)NC(CCOCC)C C(=O)(C1=CCCS1)N(CCN(C(c1cc(C(C)(C)C)oc1C)=O)CC)CC CC(C(O)C(F)F)NC(C1(CO)CCN(C(=O)CCc2cn(C)cn2)C1)=O C(=O)(CCS(C)=O)NC1C(NC(c2ccc(CCC)[nH]2)=O)CCC1 c1(C(=O)NC(C)CNC(=O)CC2CCC(F)(F)CC2)cc(N=S(C)(C)=O)ccn1 C(Cc1ccc(Cl)cc1)(CC(=O)N(C1CC(F)(F)C1)C)NC(C)=O CCCC(CC)C(C(=O)NC1CCCCC1)N1C(C)CCC1(C)C.OC Cc1cnn2ccc(C(=O)NCC3CC3NC(c3ccn4c3CSCC4)=O)nc12 C1(C(=O)Nc2nc(COC)oc2)CC(C)CN(C(=O)CC2CCCC2)C1 CCC(CC(=O)N1CC2CC1(CNC(c1cc(C)nn1C)=O)C2)C1CCC1 c1(C(=O)NCC(C)OC)cc(-c2cccc(C#N)c2C)c2[nH]ccc2c1 N1(OC)CC2CC(C1)CN(C(=O)C(C)C)C2.c12nc3c(s1)CN(CC3)C(=O)N2 CCC(CCC(=O)N1C2CCC(C2)C1CC(N1CC2CC1(C(F)F)C2)=O)OC CC1CN(C(C2CN3CCC2C3)=O)CC(C(N2CCC(CF)CC2)=O)O1 C(=O)(C#CC(C)(C)CNC(C1(CO)CCCO1)=O)N1CCC(O)(CC)C1 C1(C(=O)NC2CN(CC)C(=O)C2)CCN(C(=O)C(C)C2CCC2)CC1(C)C C1(CNC(C2(C)CCC(C)CC2)=O)CC2(CCOCC2)O1 C(=O)(CCC(C)C#N)NC(CNC(c1ncc(CC)cn1)=O)C(C)(C)C CC(N=c1[nH]c(=N)[nH]c(=NC2CCN(C3CC3)C2)[nH]1)C1CCCCC1 N1(C(C(=O)NCC(F)F)CC2C=CCC2)CCCCC1c1ccc(F)cc1 c1(CC)ncoc1C(=O)NC1(C(=O)NCC2CCCCS2)CSC1 c1(C(=O)NC2C(CNC(C3(COC)CCCO3)=O)CC2)ncccc1OC(F)F CC(F)(F)CCC(=O)NCc1cc(C(=O)NCc2c(F)cccc2F)ccn1 c1(OC)ccc(C)cc1NC(=O)CCNS(=O)(=O)CC1(CO)CCC(OC)CC1 C(=O)(CC1=CCN(C)CC1)NC1(CCNC(c2cnc(C)[nH]2)=O)CC1 N1(C(c2ccc(F)c(Br)c2F)=O)CC2CCCC(C1)C2N1CCC(C(=O)O)C1 N1(C(c2c(OC)c(C)sc2)=O)CC2(CCCCN2C(=O)CCC(C)OC)C1 C(=O)(CCC(C)(F)F)NCC(CN(C(C(c1ccc(C)cc1)(C)C)=O)C)C c1(C23CC(C(=O)NCCCC(C)NC(COC(CC)C)=O)(C2)C3)cccc(Cl)c1 C(=O)(CC(C)C(C)(C)C)N(C1CCN(C(C2CCC(C)(C)OC2)=O)CC1)CCC C12(CCNC(COc3c(C)cccc3)=O)CCC(C1)N(C(c1ccnn1C)=O)C2 C1(CNC(Cc2c(C)cccc2)=O)CC(F)(F)CN1C(C1CC(F)C1)=O CN1CC(CNC(=O)C(F)C2CC(NC(=O)Cn3ccnc3)C2)CC12CCC2 C1(CNC(c2ccn(C(F)(F)F)n2)=O)C2CN(C(C3CC3F)=O)CC12 C1(C)(COC)CCN(C(C2CC(O)CN2C(=O)CC2OCCC2(C)C)=O)C1 c1(C(N2CCCC(C(C)NC(c3cc[nH]c3)=O)C2)=O)cc(F)c2cc[nH]c2c1 N1(C(CCCC#C)=O)CC=C(CNC(c2cnc(C)nc2O)=O)CC1 C1(NC(=O)NC(c2c(C)nc(C)s2)C)CN(C)C(=O)C12CC2 C12(C(=O)N(CCc3cc(C(NOC(CC(C)C)C)=O)no3)CC)CCCC1C2(F)F c1(C(N(CCN(C(C2CCC(C)(CC)O2)=O)C(C)C)C)=O)ncc(C#N)cc1C CC1(C)CC=C(C(=O)N2CC3CC2CC3NC(=O)C(C)(C)c2cscc2Cl)CC1 C(=O)(C1CCCc2scnc21)NCC1N(C)CCN(C(C2=C(C)OCC2)=O)C1 N1(C(C(F)=CCC)=O)CC2CCC(C1)N2C(=O)C(C(C)C)NC(C)=O O=C1CC(C(N2CC(C(=O)NCCNC(C3CCNC3=O)=O)C2)=O)CN1 CCC(C)(C)C(=O)C(=O)NC(C1CN(C(C2CCS(=O)(=O)C2)=O)CCO1)C C12(NC(C3C4CN(C(c5cc(CC)on5)=O)CC43)=O)CCC(C1)OC2C N1(C(c2cc(OC)c(C)cc2)=O)CC2CCC(CNC(=O)Cc3cc(C)cs3)C2C1 C1(C)(C(N2CCC(N(C(=O)CP(C)(C)=O)CCC)C2)=O)CC=CCC1 N1(C(CCc2ccn(C)c2)=O)CC2C=CC1C(C(=O)NCCc1ccccc1)C2 c1(C(=O)NC(CCCNC(C(C)OCC#C)=O)(C)C)nccc2nn[nH]c12 c1(C(=O)NC(CC)CN(C(=O)C=C(Cl)Cl)C)ncnc(OC)c1F C(CC(=O)NCCC1CCCN(C)C1)(C(F)(F)F)NC(c1c(C)n(C)nn1)=O Cc1cn(C)nc1CSCC#CCCO c1(CC(=O)NC(C2CCCCC2)C(C)NC(C=CCC)=O)ccc(F)cc1O c1(C(N2CC(OC)(CNC(=O)CC3CC(C)=NO3)C2)=O)cccc2[nH]nc(O)c12 c1(CC(=O)NC2CCC(n3cc(C(C=C)(C)O)nn3)CC2)nn(C)c(C)c1Cl c1(CC)nn(C)cc1C(N1CC(CCCCNC(c2ccn(C(F)F)n2)=O)C1)=O n1(CC)ncc2cc(C(=O)NCC3COCCN3C(=O)C(C)NC(N)=O)cnc12 C1(OCC)(CNC(CC(C)C)c2nnnn2C2CCCC2)CCC(C)(C)C1 C(=O)(CC(C)(O)C(F)(F)F)NC(CN(C(c1ccc(N)c(SC)c1)=O)CC)C C(CC(O)CNC(=O)CCCF)NC(CN(c1ccccc1)C)=O c1(OC)ccnc(C2(CN3CCC(Br)C3)CCC2)n1 c1(C(=O)NCC(C)(C)NC(C2CCCCS2)=O)cnc(-c2ccccn2)nc1 C(CNC(c1cnc2n1CCC2)=O)(C(C)(C)C)NC(C(OC)OC)=O c1(C(N2CCC(C)(NC(C3CCCN(CC)C3)=O)C2)=O)cnc2ccnn2c1O c1(C(=O)NCCC(C)(C)NC(C#CC2(CC)COC2)=O)ccc2sc(O)nc2c1 C1(CNC(c2c[nH]nc2F)=O)CN(C(c2cn(CCCF)nn2)=O)CC12CC2 CC1CN(C(=O)Cn2cncn2)CC1NC(c1ccc(O)c(CO)c1)=O c1(C(=O)NC23CC(NC(CCC#C)=O)C(OC2)C3)cc(F)c2nc(O)ccc2c1 c1(CCC)nc(=NC(=O)N2CCCC(C(N3CCc4ccccc43)=O)C2)n(C)[nH]1 C1(CCCC)CCCCN1C(=O)C(=O)N(C(C)(C)C)C.N12CCCC1C2=O S(=O)(=O)(c1ccc(Cl)c(CNC(C2OCCN(CC(C)CF)C2)=O)c1)NC Cc1c(C(=O)NCC2COCC2NC(C2CC3C=CC2O3)=O)ccn1C1CC1 C1(CNC(=O)C=CC(F)(F)F)C2CN(C(c3n[nH]cc3F)=O)CC12 N1(C(C(CC=C)OC)=O)CCC2CC2(C(=O)NCc2cccc(C3CC3)n2)CC1 c1(C(=O)OCC)cc(C(N2CC3CC2C3NC(=O)CC2CCCO2)=O)[nH]c1C Cc1cc(F)ccc1C(F)(F)C(=O)N1CC=CC1CNC(C1NC(=O)OC1C)=O N1(C(C2CC(CCNC(C3C(SC)CCC3)=O)C2)=O)CCCC2(CC1)CC2 N1(C=O)CC(N(C)C)C2(CC2)C1.c12ccc(o1)C(=O)NC2.CC(C)S N1(C(CNC(C(CC)CC)=O)=O)CC(C2CCCN(C(C3CCC(=O)NC3)=O)C2)C1 C=CCC(CNC(=O)C(CCOC)SC)C(=O)N1CCC(C)=C(C)C1 N1(C(CC)=O)CC(C(=O)OC)C2(CCOCC2)C1.c12cccc(c1)CN1CCC21 c1(C(=O)Nc2ccccn2)ccncc1S(=O)(=O)NC1CCc2c(Br)cccc21 C1(CC)CC2(CCN(C(=O)CC3CC3NC(C3(C(=O)N(C)C)CC3)=O)CC2)C1.OC Cc1cccc(C(O)CNC(C)CC2CCNCC2)c1 C1(C)(C(=O)NCCCN2CCN(C(C(C)(C)O)=O)CC2)C2CCC(C2)C1(C)C N1(C(c2cc(C(C)=O)oc2)=O)CC2C(NC(=O)C(c3ccc(F)cc3)CO)C2C1 c1(C(=O)NCC(CNC(c2cnn(CCO)c2)=O)CO)cnn2c1CCCC2 C12(C(=O)NCCC3(O)CN(C(Cn4ccc(C)n4)=O)C3)CC(CO1)C2(C)C Cc1oc(Br)cc1C(N1CCC(CNC(=O)C(F)=CC2CC2)CC1)=O CCC(CC)CC(F)C(=O)N(Cc1nc(-c2cccc(Cl)c2)no1)CC1CNC1 C(=O)(CCCC(=O)NC(C)(C)C(C)NC(=O)CC1OCCC1(C)C)NC(C)C c1(N(C)C(C2CSCN2C2CCC2)=O)ccc(C2CC2(F)F)cc1 C1(NC(C(C)SCC)=O)CC2CCC1CN2C(c1cccc(Cl)c1)=O C(=O)(C1=CC2CC(C1)CC2O)NCC1(NC(CCCC)=O)CCC1 c1(C(=O)NCC(CC)NC(C2CC23CCCC3)=O)cc(N)cc(O)c1 C(N=c1[nH]cnc(NCC23CCCCC2C3(F)F)c1C)C1CCN(CC)CC1 Cc1noc(C)c1NC(=O)CCC(C)c1ccc(Br)cc1 c1(C(=O)Nc2c(CO)ccc(C)c2)cnc2c(-c3cnc(=N)[nH]c3)cccc2c1 c1(OC)cc(C)sc1C(=O)NCC1(CNC(=O)CC=C(C)C)CCCCC1 c1(C(c2nnnn2CCn2cncn2)NCC2(C)COC2)cc(Br)ccn1 C1(NC(C(C)=C(C)C)=O)(CO)CCN(C(=O)C(=O)Nc2ccccc2)C1 CC1CN(C(c2cnn3cccnc23)=O)CC(C)N(C(=O)C(F)C2CCOC2)C1 N1(C(Cn2c(C)ccn2)=O)CC(C(=O)NCCOc2ccccc2)CC(F)(F)C1 C1(OC)CN(C(=O)CCN(C)C)CC1C(=O)NC1(C(C)(C)NS(C)(=O)=O)CC1 c1(CCC(=O)NC2C(NC(C3C4CCCC34)=O)CCC2)cccc(C(F)(F)F)c1 C1(NC(C(C2CCC2)OCC)=O)CN(C(=O)Cc2cnn(C)c2C)CC1C C=CC1(C(=O)NCC(=O)N(CCN(C)C)CC2CC2)CCOCC1 N1(C(C2CC(C)(NC(Cn3c(C)cc(C)n3)=O)C2)=O)CCSCC(C)C1 C1(=O)NNC(=O)C(C(C)(C)C)n2cc1nn2.C1(C(NOCC=C)=O)CC2C=CC1C2 C1(NC(CSC)=O)CCC2(CCCN(C(c3ccc(C#N)c(O)c3)=O)C2)C1 C(c1sccc1Br)=CC(=O)NC(Cc1n(C)ccn1)C(F)F C12(COC)CC(NC(=O)C(C(C)C)N)(CN1C(C)=O)C2.C(=O)(C1=CCOCC1)C(C)=O CCC(CC)C(=O)NC12CC(CNC(c3cnc(C)[nH]3)=O)(C1)C2 c1(C(CC)=O)cc(C(=O)NC2CCN(C(c3csc(CC)n3)=O)C2)ccc1F CC1CN(C(C2CC(C)OC2C)=O)CC1NC(c1ncnn1C)=O Cc1cc(C(=O)NC2CCCN(O)C2=O)c[nH]c1=N C1(C(=O)NC(C2CN(C(=O)CN(C)C)CCO2)C)(OC(C)C)CCOCC1 C(=O)(C1CCCc2ncnn21)NC1CN(C(c2ncn(CC)n2)=O)CC1O C1(NC(COCC(=O)NC)=O)CC(O)CN(C(=O)CCCOCCNC(C)=O)C1 N1(C(c2cn(CCOC)nn2)=O)CCC(CNC(C2CN(C)CCO2)=O)C(O)C1 C(CC1CCCC1)(C(=O)N1CCC(CO)C1)NC(=O)C=CCN1CCC1 C(CNC(=O)C(C)CC#N)(C(C)(C)C)NC(CC1(OC)CCC1)=O C12(NC(C(C)SC(C)C)=O)CC(C1)N(C(c1cn(CCO)nn1)=O)C2 C(=O)(C1=NOC(CNC(c2cc(C)c(C)nn2)=O)C1)N(C)Cc1n(CC)cnn1 c1(C(=O)NCCN(CCC)C(C2(OC)CCSC2)=O)cnn(C2CC2(F)F)c1 c1(OCC2C(C)(C)CCC2)cccc2c1OCCC2C1CC(=O)Oc2ccccc21 Cn1nc(C(=O)NC2CC(CNC(=O)Cc3ccon3)CC2O)cc1O N1(C(C(C=C)C)=O)CC2(C(=O)NCc3cnc(C)[nH]3)CC1CO2 Cc1nc2ccc(C(N3CCOCC(CNC(=O)C(O)C4CC4)C3)=O)cc2o1 N1(C(CC(c2ccccc2Cl)C)=O)CC(CNC(C2(F)CC2)=O)CC12CCC2 N1(C(c2c(CC)noc2)C(=O)NC(c2ccccc2)C)CC(C)C(C)C1C CC1(CNC(C23CCC2C3)=O)CCN(C(=O)CCN2CCCCC2=O)CC1 C1(NC(C2(OC(C)C)CC2)=O)CCOC2(CCN(c3nnc(C4CC4)s3)CC2)C1 N1(C(CC(C)OC)=O)CCCCC1C(C)(O)CNC(=O)Cn1[nH]cnc1=N c1(C(N(C)CC2CC(F)CN2C(=O)COCC2(F)CC2)=O)ccn(C)c(=O)c1 C12(CCC(F)CC1)c1nnnn1CCN2.n1(CCCNS(CC)(=O)=O)ccnc1C c1(C(N2CC3N(C(c4c(C)cnnc4)=O)C(C3)C2)=O)ccc2occc2c1O C(=O)(C(CC(F)F)NC(=O)C(O)C1CC1)N(C)Cc1cncnc1 c1(C(N2C(C)C(NC(=O)CC3C=CCC3)C(C)CC2)=O)cnn2c1C(=O)NCC2 CCCS(=O)(=O)C(C)C(=O)N1CCC(NC(=O)Cc2ccc(S(N)(=O)=O)cc2)C1 c1(C(N(CC(C)N(C)C(c2nccc3nn[nH]c23)=O)C)=O)cccc2[nH]ccc12 C1(NC(C2(CCOC)CN(C(C3CC(CCC)C3)=O)C2)=O)CN2CCC1CC2 N1(C(c2c(C)ccn2C)=O)CC(CNC(C2CC23CC3)=O)C2(CCC2)C1 c1(C(=O)NCC2(C)CCN(C(C3(CF)CCC3)=O)C2)cc(=N)[nH]c(=N)[nH]1 Cn1ncc2c(O)nc(=NCC=CCNC(=O)CC3CCSCC3)[nH]c12 CC1CN(C(c2csc(CO)n2)=O)C(C)CN1C(c1nocc1Cl)=O c1(OC)n[nH]cc1C(=O)NCC1CC1NC(=O)Cn1ccc(C(F)(F)F)n1 C1(NC(c2ccsn2)=O)CCCCC12CCN(C(=O)C(F)(F)C(F)(F)F)CC2 N1(C(CCOCC(C)(C)C)=O)CCCC(C)(NC(=O)CC2CC3CCC2O3)C1 Cc1ccc(O)c(CC(=O)NC2(C)CCN(C(C3(c4cc[nH]n4)CC3)=O)CC2)c1 C(=O)(C(C#N)C(C)C)NC1C(NC(CC=CCC)=O)CCC1 C=CCCC(C(=O)N(CC(C)(C)C)C)NC(=O)C(C)n1cncn1 CC1(C)CCC(C)(C)N(C(=O)NCc2cccc3ncccc23)C1 C1(C(=O)NC(CC)(CNC(C2CCC(C)(C)C2)=O)CC)CCCCC(=O)N1 Cc1ccc(S(C)(=O)=O)cc1NC(N1C2CCCC1CC(N=[N+]=[N-])C2)=O Cc1cc(C(=O)N(C(C)CNC(c2ncccc2Br)=O)C)ncc1F c1(OC(C)C(=O)NCC(O)CN(C)C(c2cc(Cl)n(C)n2)=O)ccc(F)cc1 c1(C(N2CC(CCNC(C3(CCC=C)CC3)=O)OCC2)=O)csc(S(N)(=O)=O)c1 c1(CNC(C)=O)ccc2c(C(=O)Nc3onc(COC)n3)n(C)nc2c1 C1(CC(=O)N(C(c2ccccc2OC(F)(F)F)C(=O)O)C)CCS(=O)(=O)CC1 c1(C(=O)NC2CN(C(C3C(C4C(C)C4)C3)=O)CC(O)C2)ccc(F)c(C#N)c1 C#CCCC(C(=O)NC(C)CC1=CCCC1)NC(c1cc(C2CC2)[nH]n1)=O c1(CCCC(=O)NC(CNC(c2ccc(Br)cc2)=O)CO)ccc(F)cc1 CCCCCCCC(=O)N1CCCCC1CNC(c1csc(C)c1Br)=O Cc1c(C(N2CCC3NC(=O)NCC3C2)=O)oc2ccc(Br)cc12 N1(C(CCOC)=O)CCCC1C(C)NC(C1CC1C(C)(C)C)=O C1(NC(c2n(CC)nnn2)CC2CCOC2)CCC2(CCCC2)CC1 C1(NC(c2cc(C)on2)=O)COCCN(C(c2cncc(O)c2)=O)C1 C(=O)(C1=Cc2cccc(Br)c2OC1)NC1C(CC)N(C(=O)OC(C)(C)C)CC1 C1(OC)CC2CCC1CC2C(N1CC(Nc2ccccc2)CC1C)=O C1(CNC(CN(CC)CC)=O)COC(C(F)(F)F)C1.c1(C(=O)NC)ccn(CCF)n1 CC1=C(C(=O)NCC2(C)CN(C(=O)CC(C)CC(=O)OC(C)(C)C)CC2C)CCC1 c1(C(=O)NC(CCNC(c2c(C)oc(Cl)n2)=O)C)c(C)nn2c1CCCC2 C1(C(=O)NCC2N(C(c3cc(C)[nH]c3)=O)CCOC2)CCOC(=O)CC1 C=CC(CCC)CC(=O)N(C1CCN(C(c2cn(C)cn2)=O)C1)CCO N1(C(Cc2ccc(C)o2)=O)CC2CCC2(CC(=O)NCCc2c(C)cnn2C)C1 c1(C(C)NC(=O)C(=O)N(C2CC2)CC2CC23CC3)csc(C(F)(F)F)n1 C1(NC(=O)C=CC2CC2)CCN(C2CCCC2)CC1 C(=O)(C(C)(C)CCC(=O)NCC1(F)CC(NC(=O)CCC(C)CN(C)C)C1)OC c1(C(CO)C(c2ccccc2)Oc2nccc(COC)c2)ccc(Cl)c(C)c1 N1(CCCc2onc(C)n2)CCOCC(NC(=O)CC2CCCS2(=O)=O)C1 CN1C(=O)CCCC1C(N1CCC(CF)(NC(c2ncc(C3CC3)cc2F)=O)C1)=O Cc1nc(C(=O)NC2CC(CC(=O)NCC(C)(C)C(C)(F)F)C2)cc(O)n1 Cc1ccc(S(=O)(=O)N2CCCC(C(=O)Nc3cc(F)cc(Br)c3C)C2)c(F)c1 N1(C(c2c(CC=C)cccc2)=O)CCC2(CCCC2C(=O)NCCCCCO)C1 Cn1ncc2c1CCCC2NC(=O)NC1COc2ccc(F)cc2C1 CN1C(=O)CCCC1C(=O)NCCC1CC(NC(=O)CNC(C2CCC2)=O)C1 c1(OC)cccc([N+](=O)[O-])c1C(N1CC2C(C1)N2C(=O)C(C(C)O)N(C)C)=O CCC(CC)CC(F)C(=O)N1CCN(C)C(C(=O)NC(c2cc(C)no2)(C)C)C1 C1(C(=O)NC(C(C)C)CNC(c2ccnn2CC#N)=O)CCC2CCC1O2 N1(C(C2(COCC)CC(=C)C2)=O)CC2C(C(=O)NCCC(C)c3cn[nH]c3)C2C1 c1(CC(=O)NC(C)CNC(=O)C=CC2CCCC2)ccc2[nH]ccc2c1 c1(N(C(c2cc(C)co2)C(=O)NC2CCOC2)CC#CC)cccc(OCC)c1 C1(CC)CC(C(N2CCCC(CC(N3CCC(O)(CC)C3)=O)C2)=O)CCO1 C12(NC(c3cnc(CNC(CC(C)(C)C4CC4)=O)nc3)=O)CCC(CC1)CC2 Cc1c(C(=O)NCCC2CN(C(=O)CCC3CCCOC3)C2)nn2c1CCCC2 CC1(CNC(C2(C)C=CCN2C(=O)CN2CCC(O)CC2)=O)CCCCO1 C1(OC)CC(CNC(=O)C(C)CN(C)C)N(C(=O)Cc2[nH]cnc2C)C1 c1(CC)ccc(C(=O)NC2CC(NC(c3ccc(C(=O)OC)s3)=O)C2)[nH]1 C(=O)(CC(C)CC(C)C)NCC(CC)NC(c1cc(OC(F)F)cc(F)c1)=O CCC(CC(=O)N1CCN(C(C2CC(C)(C)CO2)=O)C(CCO)C1)C(C)(C)C N1(C(C2C3CN(C(C(C)OCCC)=O)C2C3)=O)Cc2cncnc2C1.C(C)(=O)O C(C(C)(C(C)C)NC(=O)COC1CCCOC1)NC(CCn1ccc(C)n1)=O CCCCCC(O)CC(=O)NCC(C)=CC(=O)NC(c1cncnc1)C C1(C(=O)NC2C3(NC(Cc4c(C)nn[nH]4)=O)CCC(C2)C3)CC2CCC(C1)C2O c1(C(N2CCC(C(C)NC(=O)Cc3ccon3)C2)=O)ccccc1P(C)(C)=O C1(CN(C(=O)CC2CC2C(F)F)C)CCN(C(=O)CCc2cc[nH]n2)CC1 N1(C(C(C)C2CCOC2)=O)CCCC(C2(NC(=O)C(C)n3cncn3)CC2)C1 CCCCC(O)C(=O)N1CCSCC1CCNC(c1cccnc1NC(C)C)=O C(N=c1[nH]c(=NC2CCCc3occc32)c2ccccc2[nH]1)c1n(CC)cnn1 N1(C(c2c(C)cc(CNC(c3nccs3)=O)o2)=O)CCN2CCCC2C1 CC1(C(=O)Nc2cncc(Cl)n2)CCCN(Cc2ccc(F)c(F)c2)C1 c1(C2(C(=O)NCCC(C)NC(CCOCC)=O)CC2)ccc(OC)nc1 c1(C(N2CC3C(NC(c4cnco4)=O)(CC3)C2)=O)cccc2c1CCC2=O C1(CNC(c2nc(COC)sc2)=O)(NC(c2sccc2Cl)=O)CC2CCC1C2 C1(CC(=O)NC(COCCOC)C)COCCN(C(C2(NC(C)C)CC2)=O)C1 CCC(CCc1ccccc1)C(=O)N(C1CCN(C(c2sccc2F)=O)C1)C c1(C(N2CCC(NC(C(CSC)OC)=O)C23CCC3)=O)cncc(P(C)(C)=O)c1 N1(C(C(=O)NC(C)C)=O)CC2CC1CC2CNC(=O)CCC(=O)NC1CCCC1 c1(N(c2ncccn2)CC)nccnc1C Cc1ccc(C2(C(=O)NCCCC3CCCN3CCCSC(F)(F)F)CC2)cc1 C1(CC)CCN(C(=O)CS(C)(=O)=O)C(C(=O)NCC2CCCN(CC)C2)C1 N1(C(CC(COC(C)=O)(C)C)=O)CCN(C(C2CC3(C2)CC32CC2)=O)CC(C)C1 c1(C(=O)NC(COC)C2CC2)ccc(F)cc1CSc1ccccc1 N(C1CCOCc2c(Br)cncc21)CCCCCC1(N)CCC1 CC1CCCn2c(C(N3CCCC(N(C)C(C4(F)CCCC4)=O)C3)=O)cnc21 c1(C(=O)OC)c[nH]c(=NCCCC(C)NC(=O)Cc2cc(C(C)C)no2)c(C)c1 CC1CCC(C(=O)N(C)CCN(c2cncn2C)C)N1C(=O)OC(C)(C)C N1(C(C(CC)OC)=O)CCOC2CCN(C(c3ocnc3C3CC3)=O)CC12 C(=O)(C1=NNC(=O)C1)N1CCCC(CNC(=O)CCNC2CCOCC2)C1 C1(CCC(=O)N2CCC2CC2CC2)(NC(=O)CC2(CO)CC2)CCCC1 C1(NC(c2c(OC)n(C)nc2)=O)CCN(C(=O)Cc2cn(C)cn2)CC(C)(C)C1 C1(N(CC)Cc2cnoc2NC)CCN(C(=O)C(C)CC2CC2)CC1 N1(C(C2CCC(=O)N2)=O)CCC(C(F)(F)F)(CNC(C2(CO)CCC2)=O)C1 N1(C(c2c(C)nns2)=O)CCCC12CCN(C(c1n[nH]c(C3CC3)c1Cl)=O)C2 N1(C(C2CC(N(C)C(c3ccsc3C#N)=O)C2)=O)CCC(C)(C2CC2)C1 c1(C(N2CCC(OC)CC2C(F)(F)F)C(=O)NCCC)csc2cc(Br)ccc12 c1(C(=O)NC2CCN(C(c3cc(SC)oc3C)=O)CC2)ccc2c(c1)OCCO2 c1(CCC)ncc(S(=O)(=O)N(C2CC2)CC2CC2)s1 c1(OC)ccc(S(=O)(=O)N2CC3(CCN3C(=O)C(n3nc(C)cc3C)C)C2)cn1 C1(O)(CNC(c2cn(CC)nc2)=O)CCCN(C(c2ncccc2Br)=O)C1 c1(C(N2CC(CN(C(CC(C)CF)=O)C)C2)=O)cccc2c1OC(C)(C)C2 C(CC(=O)NC1(C#C)CCC1)(C(C)C)NC(C1(CC)CCCO1)=O N1(C=O)CC(NC(=O)CCC2(C)CCC(=O)N2)C(C)(C)C1.C1(OCC)CCCC1 CCC(O)C(F)(F)C(=O)NCC1(O)CCN(C(=O)CC(C)CN(C)C)C1 c1(C(=O)N(C2CCCN(C(C(C=C)O)=O)C2C)CC)ccc(CCC)c([N+](=O)[O-])c1 C1(NC(C(C)c2cncs2)=O)CCCC1NC(c1cc(C(=O)NCCO)c[nH]1)=O C1(CNC(c2cocn2)=O)C2CN(C(=O)CC3CCCC(C4CC4)O3)CC12 CC(C)(CCCC(=O)N1CC2C=CC2C1)NC(=O)CCC1(C)N=N1 c1(CC(=O)NC2C(C(=O)NCC(=O)NCc3ccnc(O)c3)C2)cccc(F)c1Cl c1(N(C)C(C2CN(C(C3CCOC(=O)CC3)=O)CCO2)=O)cc2n(n1)CCO2 C(=O)(C1=CS(=O)CCC1)NC(C1CC(NC(c2coc(C(F)(F)F)c2)=O)C1)=O c1(C(N2CCC(F)(C(=O)NCCc3n(C)ncn3)C2)=O)ccnc(O)c1F C1(NC(CNC(C(CC)C)=O)=O)CC2(C1)CC2C(=O)N(CCCO)C.C1CN1 C1(F)(C(=O)OCC)CCN(C(=O)CC(CC)SC)C1 c1(C(=O)NC2C3(NC(c4cc(F)c[nH]4)=O)CCC(C2)C3)csc2ncnc(O)c12 n1(C(C(=O)NC2CN(C(CCCCCNC(C)=O)=O)C2)C)cc2ccccc2n1 C(C)(CCC(C)(C)C)N(CCC)Cc1ccco1 c1(C(N2C(C)CC(NC(c3cc(C(C)C)[nH]n3)=O)C2)=O)cc(F)cc(Br)c1F C=CCC(CC=C)C(=O)NCC(CO)NC(c1ccn(C)c(=O)c1O)=O C12(OC)CCC(C(=O)NCC3(C)CCN(C(C4CCC(C)S4)=O)CC3)(CC1)CC2 CCC(C)CC(=O)C(=O)NCCC1(C(N2CC3CC3C3CC23)=O)CCCC1 C1(C(=O)NCC(CN(C(C(CCC)C)=O)CC)(C)C)Cc2nncn2C1 Cc1cc(C(=O)NC2CC(Nc3nnnn3C)C2)[nH]c1C.C1C(=O)N1C C=CCC(C(=O)NCc1csc(CNC(C2CCN2S(C)(=O)=O)=O)n1)C(C)C C(=O)(CC(C)CNC(c1nc(=N)[nH][nH]1)=O)N(C1CCCCCC1)CC Cc1cccc2[nH]ccc(=NCC3(C)CC3Br)c12 C1(C(=O)NCC2(C(N(C(CC(=O)OC)C)C)=O)CC2)CC(C)(C)CN1C C1(NC(C2(C(=O)NC)CC2)=O)COCC1NC(C1CCCN1C)=O n1(CC(=O)NC2CCCC(N(C(c3ccn(CC)n3)=O)C)C2)cnc([N+](=O)[O-])n1 N(C1CCCc2cc(CNC(=O)C(O)C(F)F)ccc21)C(=O)CCC(F)(F)F c1(C(N2CCC(N(C(C3CC(C)CO3)=O)CC)C2)=O)c(OC)ccnc1F N1(C(c2c(COC)ocn2)=O)CC2CCC1CN2C(=O)Cc1ccc(F)cc1Cl c1(OC)cnnc(C(=O)NCC2CC2NC(c2cnn(-c3ccccc3)c2)=O)c1 Cc1cc(NCC(F)C2CCC2)c(S(N)(=O)=O)c(F)c1 CCCCCCCCNC(=O)C(CC(F)F)NC(c1cc(F)cnc1O)=O c1(NC(c2csc(C(=O)Nc3ncc(Br)c(O)n3)n2)=O)c[nH]c2nccc-2c1 C1(CNC(=O)CC=C(Cl)Cl)CN(C(C23CCCC(CO2)C3)=O)CCC12CCC2 C(CCCCC(=O)NC1CC1NC(c1ccc(-c2ccccn2)nc1O)=O)=CC N1(C(CCCCC=C)=O)CC2CN(C(=O)C(C)CC3CCC3)CCC2(CO)C1 N1(C(=O)N(CCC(C(F)(F)F)c2ccccc2)C2CC2)CCOc2cc(F)cnc21 N1(C(C(CSC)C)=O)CCC2(NC(=O)C=Cc3c[nH]nc3C)CCCC12 C1(NC(c2c(C)coc2)=O)CC(O)CN(C(C2CCCC(C)(C)C2)=O)C1 c1(C(N2CCC3(NC(C(=O)N(C)C)=O)C(CC2)C3)=O)cc(F)cc([N+](=O)[O-])c1 C1(NC(c2c(CC)con2)=O)CC(O)CN(C(=O)C=CCF)C1 C1(N(C)C(c2ccoc2C2CC2)=O)CCCCN(C(=O)CCc2ccccc2)C1 C(c1ccccc1)=CC(=O)NCCC1CC(NC(=O)C(F)CC2CCOC2)C1 C1(C)(C(=O)NCC2CN(C(C3CCCN(CC(C)C)C3)=O)C2)CC2CCC1C2 c1(C(CC2CC2)OCC)cc(Cl)n[nH]c1=NC(=O)c1cccc(C(C)C)c1 C(=O)(C1=CS(=O)CCC1)NC12CC(NC(COc3ccc(OCC)cc3)=O)(C1)C2 N1(C(c2ccc(C)nc2)=O)CCC2C(NC(C3CC(=O)C34CCC4)=O)C2C1 N#Cc1ccc(N2CCC23CN(C(C2CC4(CC(=O)C4)C2)=O)C3)cn1 C(CCC(C(=O)NCCC1(N(C)C)CCC1)NC(=O)Cc1cnnn1C)OC c1(NC(N2CCC(CCC(C)C)C2)=O)ccc(Cl)nc1CC1CC1 N=c1nc(CNC(C2CCNC2=O)=O)[nH]c(=N)[nH]1 c1(C(=O)NC(CNC(C2(COC)CCC2)=O)C)ccc(OCC2CCC2)c(F)c1F C1(NC(=O)CC=C(Cl)Cl)CC(NC(c2csc3cncn23)=O)C12CCC2 c1(C(=O)NCC(C)(C)NC(CCCCOC)=O)c(Cl)cnc(OC)c1Cl Cc1csc(C=CC(N2CC3CC2C3NC(=O)CSC(C)C)=O)n1 C=CCC(CCCCC)C(=O)NCC(N1CCN(C(c2ccn(C)c2)=O)CC1)=O n1(CCC(=O)NCC(CC)Nc2cncc(Cl)n2)cc[nH]c(=O)c1=O N1(C(C=C(C)C(F)F)=O)CCN(C2CCCN(C(=O)CCC3CCC3)C2)C(=O)C1 N1(CC)CC2CCCN(C(c3csc(C(C)(C)C)n3)C3CCC3)C2C1 C12(NCCCNC(CC(C)C)=O)CCC(CC1NC(=O)C(=O)C(C)(C)C)C2 C1(C(N(CC=C)CCO)=O)CCCC1NC(=O)COCCOC Cc1ncc(C(=O)NCCCCNC(C2(n3ccnn3)CC2)=O)c(=N)[nH]1 C1(C(N2C3CCN(C(CC=C(C)C)=O)CC3CC2)=O)CSC(c2ccccc2)=N1 c1(C(=O)NCC(C2(O)CCN(C(c3cccnc3)=O)C2)C)cc(Cl)ccn1 N12CCC(CC1)N(C)CC(=O)N(CCC)C(C)C2=O.S(C)O.SC CON=Cc1ccc(C(=O)NC2CN(C(=O)C(=O)NCC3CC3)CCC2F)cc1 C1(CNC(CCSCC(C)C)=O)(OC)CCCN(C(=O)CCC2CCOC2)C1 C#Cc1cnn(C)c1C(N1CCCC(O)(CCNC(C2COC(=O)N2C)=O)C1)=O N1(C(CCN2CCN(C)CC2)=O)CC(NC(c2ccc([N+](=O)[O-])[nH]2)=O)C2(CC2)C1 C1(C2CCCOC2)(NC(c2n(C(c3ccc(F)cc3)(C)C)nnn2)CC2CC2)CC1 CCN=c1[nH]cc(C(N2CCC2CC(=O)Nc2c(OC)ncnc2C)=O)s1 c1(C(=O)NCCCCCN(C(C(C)c2cc[nH]n2)=O)C)cc(C2CC2)nn1C C1(NC(C2(CC)CCNC2=O)=O)COCCN(C(=O)CSc2cnn(C)c2)C1 N(C(=NCC1(C)CC2(C1)CC(F)(F)C2)N1CCCC2(CCSC2)C1)C1(CO)C(C)C1 C(=O)(CC(c1cccs1)C1CC1)NCCCN(C)CCOCCOCCOCCO Clc1c(CNCCc2cc(Br)n[nH]2)sc2ccccc12 Cc1ccc(C(N2CCCC(C(C)C(=O)NCCC3CC3)C2)=O)nc1 C12(COC(=O)CSCCNC(c3ccccc3)=O)CCCC1OCC2 c1(N(C)Cc2cccc(CC(=O)OC)c2)ncnc2c1nc1n2CCOC1 c1(C(=O)NC2CC(NC(C3CC(C(=O)OC)C3)=O)C2)cc2c(F)c(C)ccc2[nH]1 N1(C(C=C(C)C2CC2)=O)CCC(NC(c2n[nH]c3c2CC2CC32)=O)C(F)(F)CC1 C1(C(C(=O)NC2CC(O)C2OC)C)CCN(C(C2N(CC)CC2)=O)CC1 C(=O)(C1=NOC(C)(C)C1)N(C1CCN(C(C2CC(CN(C)C)C2)=O)C1)CC Cc1cc(C(=O)N(C)CCOCCN(C)C(c2cnc(O)o2)=O)c2occc2c1 C#Cc1cncc(C(=O)NCCCCC(C)NC(=O)C(c2cncc(F)c2)C)c1 N1(CCC(N2CC(C(C)NC(CCSCCCC)=O)C2)=O)CCCC1=O C123CCN(CCC1C2)C(=O)C(=O)N3.Cc1cc(CN(CCC(N)=O)C)co1 C12(C(N3CCCC(C)(NC(C(CC)OCC)=O)C3)=O)C3C4C1C1C2C3C41C CC1CN(C(=O)Cc2cnnn2C)CCN1C(=O)CC1CC(O)C1(C)C c1(C(=O)NC(CC)CNC(C2COC3(C)CC2C3)=O)[nH]c(C)c([N+](=O)[O-])c1C c1(C(=O)NC(CCCCNC(C(CCC)OC)=O)C)c(OCC)nccc1OC c1(C(N(CCCNC(CCNC(=O)OC)=O)C2CC2)=O)cncc(C(F)F)c1 C1(OC(C(C2CC(C(F)(F)F)C2)OC)=O)CC2CC(NC(=O)OC(C)(C)C)C1C2 N1(C(C(C2CCCC2)NC(COCC(=O)OC)=O)=O)CCCCC1C(C)C C1(C)(CC(c2ccc(C)cc2)=O)NC(=O)N(c2cccc(C(=O)C(F)(F)F)c2)C1=O c1(C(=O)NCC2C(NC(C(C)=CC3CC3)=O)COC2)cn2ccccc2n1 C(c1nc(C)c(C)[nH]1)=CC(=O)NC(CC)CN(C(=O)C1=COCC1)C C1(CC(N2CC(C)(NC(=O)CCCCc3cnn[nH]3)C2)=O)COC(C)(C)CO1 N1(C(C2OCCN(C)C2)=O)CC2(CCCC(CNC(=O)Cc3cncnc3)O2)C1 c1(C(N(C(C(=O)NCCCOCC)=O)C)C)ccc(C)nc1C CCCC(C)(O)CC(=O)NCC1COC(CNC(c2cnc(OC)c(C)c2)=O)C1 C1(CC2CCN(c3cc(OC)nc(C(F)(F)F)n3)C2)CCc2n[nH]c(C)c2C1 C1(C(N(C2CC(=C)C2)C2CCC2)=O)CC12CCN(C(=O)C(C#N)CCC)C2 C1(CN(C(c2ccccc2Cl)=O)CC)CCCCN1C(=O)CCOC1CCC1 N1(C(CC(C=C)CCC)=O)CC(C2CCCN(C(=O)Cc3cn(C)nc3C)C2)C1 N1(C(CN(CC)CC)=O)CCCC2(NC(=O)CCNC(C)=O)CCCC12 CC1(C)CC(=O)OC1NC(=O)C(c1ccc(O)cc1)CNC(=O)CCCF C12CN(CCC13CCC3)C(=O)OC2=O.c1(C23CC(C2)C3)cccc[n+]1[O-] C(c1ccccc1)=CC(=O)NC(CNC(=O)CNC1CCC1)C1CCC1 C1(F)(C(=O)N(C2C(N3CCN(C(c4cnns4)=O)CC3)CCC2)C2CC2)CC2(CCC2)C1 C1(NC(C2CCN(C(c3c(CC)oc(C)c3)=O)C2CC)=O)CCCCC1C#N C1(COC)CC(CNC(c2ncc[nH]c2=O)=O)N(C(c2c(C)cnn2C)=O)C1 Cn1ncn(NC(=O)C2CCCC2NC(=O)C2=CCCOCC2)c1=S C(=O)(C1=COCCO1)N(C)CC1CCCC(NC(c2nc(COC)oc2)=O)C1 N12CCC(O)(C1)CN(C)C(=O)C1CCC1C2=O.c1(C(=O)NC(C)(C)C)ccon1 N1(C(C2C(NC(CCc3n(C)cnc3)=O)CCO2)=O)CC(CO)C2(CC2)C1 N1(C(c2c(C)ncnc2)=O)CC2CC3CC2C1C3NC(C1CCOCC1)=O C(=O)(C1CNC(=O)c2ccccc21)NC1CC(C(=O)NCCCCN(C)C)C1 c1(C(=O)NC2CC(NC(=O)C(CC(F)F)C3CCC3)C2)coc2c(Cl)cccc12 C(=O)(C(C)N=c1cc[nH]cc1)NCC12CC(NC(C(=O)NCCOC)=O)(C1)C2 C1(CC(=O)NC(CCC)(C)C)(NC(C2CC2Cl)=O)CCCCC1 c1(C(=O)NCC2CC(F)(CNC(CC(C)c3ccco3)=O)C2)cc2occc2[nH]1 c1(CC(N2C(C)(CNC(C3C(C)(C)C3)=O)CCC2)=O)ccc(F)c(Cl)c1 C(C(CNC(=O)CSc1nc[nH]n1)NC(=O)CCc1ccc[nH]1)OC N1(C(C(CC)F)=O)CCC2(CCN(C(c3ccnc(OCCOC)c3)=O)C2)C1 O=C1COC2(CN1)CN(S(=O)(=O)c1cccnc1NCCc1ccccn1)C2 CC1(C#CC(=O)NCC2(O)CN(C(C3Cc4nccnc4C3)=O)C2)CCCO1 N1(C(c2cc(C3CC3)[nH]n2)=O)CCC2CN(C(C3CC(F)(F)CS3)=O)C2C1 c1(OC(=O)C(F)(F)CC2CCCO2)cc(OC2CC2)ccc1F CC1=C(C(=O)NCC(C)(C2CC2)NC(C2CCCCC2C(C)(C)C)=O)CCCO1 c1(N2CCOCC(CNC(c3cc4sccc4[nH]3)=O)C2)ccc2nccnc2n1 c1(NC(C2CCN(C(c3cc(Cl)cc(Cl)c3)=O)CC2)=O)ncnc2ncncc12 N1(C(C)C)CCOCC1CC(=O)NC(C)(C)CCNC(=O)Cn1cc(Cl)cn1 C12(C(N(C3(CC)CCCN(C)C(=O)CCC=C3)C)=O)CCCC(C)(C1)OC2 c1(C(CNC(=O)NC(CC=C)C)(C)N)cccc(Br)c1 N1(C(C(C=CC)O)=O)CC(C(=O)NCCCNC(=O)OC)CC(C)(C)C1 CC(C)C(O)CC(=O)NC1CC(CNC(c2ccc(OC3CCOC3)cc2)=O)C1 c1(C(=O)NC2C(C#N)CN(c3ncncc3F)C2)c(Cl)ccc(Br)c1F C(=O)(CS(=O)(=O)CC(C)C)NCC(C)NC(c1ccc(OC(F)(F)F)cc1F)=O c1(C(N2CC3CN(Cc4cnc(Cl)cc4F)C3C2)=O)c(F)cccc1I C1(O)(C(CNC(C2CC(SC)C2)=O)(C)C)CCN(C(=O)C2=CSCS2)CC1 CCCC(C(=O)NCCC1(O)CN(C(C2(C)CCC(=O)C2)=O)C1)C(C)C c1(C(C)C)ccoc1C(=O)NC(Cc1cn[nH]c1)C(=O)NCc1cncs1 Cc1cncc(C(N2CCC(CNC(=O)CCC(=O)c3ccccc3Cl)C2)=O)c1 C1(=CC(=O)NC(CCOC)CNC(c2cc(F)c[nH]2)=O)CCC(C)CC1 c1(N(C(C)CNC(c2n[nH]cc2Cl)=O)C)snc(Cl)c1C#N C1(C)(CCC)CCCN(C(=O)CC2CCCCN2C(c2csc(C)c2)=O)C1 c1(C(=O)NCC2CCN2C(=O)C=Cc2ccc(F)nc2)cc2cnccc2[nH]1 Cc1cc(C)c(C(N2CC(NC(C3(C)CC3(F)F)=O)C(CC3CC3)C2)=O)[nH]1 c1(CC)nnn(C)c1C(=O)NC1(COC)CCN(C(C2CC23CC3)=O)C1 C(C(C)(CNC(C1(N=[N+]=[N-])CC1)=O)O)NC(C1(COC)CCC1)=O.C1(C)CC1 N1(C(C2N(C(C(C)NC=O)=O)C3CC(F)C2C3)=O)CCC2(CCCC2)CC1 CC1CCC(NC(=O)CCCCC2CC2)CN1C(c1cnc(N(C)C)s1)=O CC1(C)CN(C(=O)CCc2cnc[nH]2)CCC1NC(C1CC1c1cccs1)=O C(CCF)(C(=O)OC)NC(C(COC)N(C)C(C1CCCC1)=O)=O C1(Cc2nnnn2-c2ccccc2Cl)CN(C)S(=O)(=O)C1.CCCC(CN)CO N1(C(CCSC)=O)CC2CCCC(C1)N2C(c1ccc(C)cc1Cl)=O Cc1cc(OC(c2csc(COc3ccc(Cl)cc3Cl)n2)=O)ccc1Br c1(CNC(C2(C)CCCCO2)=O)nc(CNC(C2(C#N)CCOC2)=O)cc(O)n1 C1(CC(=O)NC2(C(C)NC(=O)CNCCC(F)(F)F)CC2)CC2(CCC2)C1 c1(C(=O)NC(C2CCCN2C(=O)Cn2cnnc2)C)cccc(-c2cncs2)c1 c1(C(=O)NC2(c3ccccc3Cl)CCC2)c(O)nnc2c1COCC2 N1(CC(CCCC)=O)Cc2ccccc2SCC1C CN1CCC(C(N2CC(F)CC2CC(=O)NCc2ncccc2Cl)=O)CC1 C1(C(=O)NCC(CCOC)(C)C)CC2(CCN1C(C1CC3CC3C1)=O)CC2 C(C(CC(F)(F)F)NC(=O)C(=O)NCC(C)O)OC C1(C(C)(C)C)CCC(C(=O)NC(C2CCCC2)CNC(=O)C(Cl)=CCl)CC1 c1(CC(=O)NCC2(O)CCN(C(c3c(C)ccs3)=O)CC2)cnn2c1OCCC2 N1(Cc2ccc(C(=O)N(C(=O)C(O)C3CC3)C3CCCC3)o2)CCCS1(=O)=O CC1(C)C=CC(NC(C2CCCC2NC(C23CCCC2C3(F)F)=O)=O)CC1 N1(C(=O)CN2CCc3ccccc32)CCN(C(=O)Cn2cccc2)CC(O)C1 C12(CNC(c3c(OC)ccc(Cl)c3)=O)CCCC1N(C(=O)CC(F)F)CCC2 C(=O)(CC(C(F)(F)F)NC(=O)C(O)c1ccco1)NC(C=C)C(F)(F)F N1(CCNC(c2ccsn2)=O)CCN(C(C2(C3CCCCO3)CCC2)=O)CC1 N1(C(C(C)N(C(C(CCC)(C)O)=O)C2CC2)=O)CCOC(C)(C)C1C c1(OC)c(F)ccc(Cl)c1CN(CCOC)CC1CCCO1.C1(=O)CCN1 c1(CC(C(=O)N(CCO)CCO)NC(c2ccc(CO)nc2)=O)ccccc1Br n1(CC(=O)NCC(C)CNC(c2cnc3n2CCCC3)=O)ccc(=O)n(C)c1=O C1(CC)CC(C(=O)NCCC2CCCN2c2nccc(CC#N)n2)CCO1 c1(C(N(CC(C)NC(=O)C(F)CC2CCC2)C)=O)nnsc1C(F)F c1(C(=O)NC(C)CNC(=O)C2=CSCCO2)cc2ncccc2cc1Cl C1(NC(C(C)O)=O)CC2CC(NC(c3cc(F)c(Br)cc3F)=O)CC2C1 N(C(=NCCCCC(F)(F)F)NCC1(O)CCCC1)C(NOCC)=O CC(C)CC(C(=O)NC1CN(C(C2CCC(C)(C)OC2)=O)C1)c1ccccc1 C1(OC)C(NC(=O)CCC2CCN(C(=O)CC3(O)CCCOC3)C2)CC12CCC2 c1(NC2(C(=O)Nc3ccc(C(N(C)C)=O)cn3)CCOCC2)ccc(F)c(Cl)c1 c1(C(=O)NCC2CC(NC(COC)=O)C2)sc2ccc(F)cc2c1C c1(C(C)C)nccc(C(N2CC(NC(c3ncccc3O)=O)C(C)C2)=O)n1 C(=O)(C(C)(C)CCC#N)NCC1C(C(=O)NCC(CC)N2CCCC2)CCC1 C(C(CC)(CC)C(=O)NCCc1cnccn1)NC(C(C(C=C)C)C)=O N1(C(C(CC)C)=O)CC(CNC(c2cc3occc3[nH]2)=O)CC(C)(C)C1 c1(C(C(=O)NCC(CNC(CCNC(C)=O)=O)C)(C)C)cccc(F)c1 N1(C(C(CC)(F)C(=O)OC)=O)CCC2(CCC2)C(C(=O)CC2C(=O)N(C)N=C2C)C1 c1(C(=O)OC(c2nc(C)[nH]n2)C)ccc(C)c(C)c1N N1(C(c2ncn(CC)n2)=O)CC2CCC2(CCNC(c2oncc2C)=O)C1 CC(O)C(C)(C)C(=O)N1CCCC(N(CCF)C(c2[nH]cnc2C#N)=O)C1 C(=O)(C1=COCCC1)NC(C1(CNC(CC(C)c2cccnc2)=O)CC1)C CCC(O)(C(=O)NC1CCCC1NC(c1cnn(CC)c1)=O)c1ccc(Cl)cc1 CC1CCCN(C(=O)C(C)(C)C)C1CCNC(=O)Cc1ccc(-c2n[nH]o2)cc1 C1(C(C(=O)NCCN(C(=O)Cc2ncc(C)o2)CC)C)CCC(=O)N1C N1(C(CCC(=C)Cl)=O)C2CCCC1CC(NC(=O)CSc1ccc(C)cc1)C2 c1(C(=O)NC2(CO)CCN(C(C3COCC3C(F)F)=O)C2)cc2cnccc2[nH]1 c1(C(N2CC(C(C)NC(C(n3cc(C)nc3)(C)C)=O)C2)=O)ccnc(Cl)c1Cl CCCCCC(O)CC(=O)NCC1C=CCN1C(=O)Cc1ccc(NS(C)(=O)=O)cc1 C1(C(=O)NCc2c(CC)nns2)C(CC)CCCN1C(c1ccc(CO)nc1)=O C(CC(C)(C)C)(C(=O)NOC1CCOCC1)NC(C1N2C(C)CN(CC2)C1)=O c1(C(C(=O)NCCCC)N(C2CCC2)C2CC2)cnccc1C C1(C(=O)NC(CNC(c2cscc2C(F)F)=O)C2CC2)CCCN(CC(F)F)C1 C1(CNC(C2OCCO2)=O)C2CC1N(C(C1CC1c1ccccc1)=O)C2 C(C)(C(=O)NCCOCCNC(=O)C(C)c1cc[nH]n1)OCC(C)C C1(C(c2ccc(F)cc2)O)CCCCN1CCc1ccncc1 C1(=CC(N2CC(C(=O)NCC(=C3CCCCC3)F)(SC)C2)=O)CC(C2CC2)C1 CC(O)(CC(=O)N1CC2CCC1C(CNC(c1ncc[nH]c1=O)=O)C2)C(F)(F)F c1(C(N2CC(NC(C(C)(C)N3CCCC3)=O)C(O)C2)=O)ccc2cccnc2c1 C1(CC(=O)N(CCC(=O)NCC2(C)CC=CCC2)C(C)C)CCCC2CC12 Cc1cc(Cl)cc(C(=O)NC2CC(NC(=O)CN3CCOC3=O)C2)c1C c1(C(N2CC(CCNC(C3OCCC(C)C3)=O)OCC2)=O)ccc2nn[nH]c2c1 C1(CCOC)CN(C(C2CCC(C)(C)C2)=O)CCN1C(=O)CCCN(C)C(C)C c1(C(=O)NCCCOCCN(C(C(CC)C(C)O)=O)C)cc2cc(Cl)cnc2o1 C(=O)(C1=CCCCO1)N(CC(C)N(C(C(c1cccc(Cl)c1)CC)=O)C)C N1(C(Cn2c(C)ccn2)=O)CC2CCC1CN2C(=O)CCCC#N O=C(C1=CCCOC1)N1CC(C2CN(C(c3ccc(F)o3)=O)CCO2)C1 c1(CN(C(=O)C(F)(F)CC2CCOC2)C)cncc(I)c1 c1(OC)ccc(F)c(C(=O)NCCCCC(C)NC(C2CCCC2SC)=O)c1N N1(C(CCCCC)=O)CCCC2(CNC(c3c[nH]nc3C3CC3)=O)CCCC12 N1(C(CC2CN(C(C3C(F)(F)C34CC4)=O)CC23CC3)=O)CCCC(C2CC2)C1 C1(C(N(C)CC2(OC)CCC2)=O)C(C)CCN1C(=O)CC1CC=CC1 C1(C(=O)NCC2(CC)CC2)(C(C)C)CCN(C(=O)CNC(C)=O)C1 C1(CCNC(Cc2cn(C)nn2)=O)CCN(C(c2csc(C#N)c2)=O)CC1 C(=O)(C(C)C(C)c1ccccc1Cl)NCCN(C(=O)CCN1CCC1)CCC C(=O)(CCCN=c1nccc[nH]1)NC(CC)(CNC(C1CCCC12CC2)=O)CC N1(C(CCC2CCN(C)C2)=O)CCC2(CC1)CC2CNC(=O)CCC(C)(C)F c1(CC(=O)NCCCOCCN(C(c2ccn(CC)n2)=O)C)nc([N+](=O)[O-])n[nH]1 C1(C(=O)NC2(C)CCN(C(C(C3CC(F)(F)C3)OC)=O)C2)CCN(OC)CC1 C1(C)(C(=O)NCc2c(C)cco2)CC(O)CN1C(C1(c2ccccc2)CC1)=O N1(C(C2(COC)CC2)=O)CC(NC(c2ccc(CO)cc2)=O)CC1(C)C c1(C(N2CCC(NC(C(CC)F)=O)C(C)(C)C2)=O)ccc2nc(CC)cn2c1 C(=O)(C#CC1CCCO1)N1CC(O)(CNC(C(c2cc3ccccc3o2)C)=O)C1 N1(C(=O)C2=CCOCC2)CC2COCCC2(NC(C23C4CC(CC24)C3(F)F)=O)C1 CCC(CNC(c1nn(C)cc1C)c1nnnn1C1CCOCC1)CC(C)C N1(C(C(C)(C)C(F)F)=O)CC2CN(C(c3nc(=O)cc(N)[nH]3)=O)CC2C1 N1(C(C2(CC=C)CC2)=O)CCC(CCC)(NC(=O)C(C)CSC)CC1 C1(O)(C(C)NC(CC(=O)OCC)=O)CCN(C(=O)CN2CC=CC2)C1 C(CNC(=O)COc1ccon1)(CC)(CC)NC(C1C(=C)CC1)=O C(CCO)(C(=O)NC1CCC(NC(C2(C#N)CC2)=O)C1)N(C)C CC1CCn2c(C(=O)NC(C3CCCN3C(c3nccnc3N)=O)C)cnc2C1 C1(CNC(C23N(C(C4N(C=O)CCC4)=O)CCC2C3)=O)CC(C2CC2)=NO1 c1(C(=O)NC2CN(C(COCCC)=O)CC(O)C2)ccc2n[nH]cc2c1 C1(C(N2CC(CN(c3ncc(C)cn3)C)OCC2)=O)CCCCN(C)C1=O N1(C(CCc2cnc(C)s2)=O)CC(CN=c2nn[nH]n2C)C2(CCOCC2)C1 C1(C(=O)NCCCC)(N(C(=O)CN(C2CCCC2)C)CC=CCCC)CCC1 Cc1c(C(=O)NC2CCN(C(=O)C#CC(C)C)CC2C)sc2ccc(Cl)cc12 c1(CC)cc(=NC(=O)C2CN(C(c3ccc(Cl)s3)=O)CC(C)O2)[nH]n1C CCCCC(CNC(=O)CCCCc1cnc[nH]1)NC(c1nnc(S)n1C)=O S(=O)(=O)(c1c[nH]c(C(=O)N(CC(C)N(C)C(c2cc(=N)[nH]c(Cl)n2)=O)C)c1)NC c1(N2CC(C)SCC2)nc2cc[nH]c2c(=NCC2C(F)(F)C23CCC3)[nH]1 C1(C(=O)NC2CC(F)(CNC(C=CS(C)=O)=O)C2)Cc2ccccc2O1 C(C(C)CCC=C(C)C)(c1n(CCCOC)nnn1)NCc1cc(Br)ccc1F C(CCCC(=O)NC(CCc1cn(C2CCOC2)nn1)C(=O)O)N(C(C)=O)C CC1COc2c(C(=O)NCC(C)(C)NC(c3cnc4c(c3)CCC4)=O)cnn2C1 Cc1cnn(C)c1CNC(=O)CC1CSCCN1C(C1CC1CC(C)(C)C)=O C#CC1CC2CCC1N(C(=O)COC1CCN(C(=O)CCCCC)C1)C2 N1(C(CN(CCC)C)=O)CCN(CC2CCN(C(=O)CC3CC=CC3)CC2)CC1 C(C)(CC(=O)NC1(CCC(=O)N2CC(C(C)N(C)C)C2)CCCC1)=C(C)C c1(CS(=O)(=O)NC2C(CC(=O)OC)CC2O)cccc(Br)c1 c1(C(=O)NCCCCCNC(c2c(NC)cc(Cl)cc2)=O)cnn2ncccc12 N#CC1(CCC(=O)NC2CCC(NC(c3cc(Br)co3)=O)C2)CCC1 CC1(C)COC(CC(N2CCN(C3(C)CC3)CC2)=O)C1 C(=O)(C(C)CCC(C)(C)C)NC(CCOC)C(=O)N1CC(CN=[N+]=[N-])C1 c1(C(=O)NCc2c(C(=O)NCCC3N(C)CCC3)c[nH]n2)cccc2ccnn12 N1(C(c2ccc(OCC)nc2)=O)CCC(C2CCN(CC(=O)N(C)C)C2)CC1 c1(C(N(CCC(C)NC(c2ccc(CC)o2)=O)C)=O)c(C)nn(CC)c1C C(=O)(C(CC(F)F)NC(C1CC2(C1)CC21CC1)=O)N(CC#C)CC1CC1 C(c1cccc(F)c1F)=CC(=O)NCCCN(C(c1cncc(Cl)c1)=O)C1CC1 Cn1cc2c(n1)C(O)CC1(CCN(C(=O)COc3ccc(O)cc3)CC1)O2 C(C(=O)NCCNC(=O)Cc1cncc(O)c1)(C(C)C)SC CC1CC(C(=O)NC(c2cccc(Cl)c2Cl)CO)CCS1(=O)=O Oc1cc(-n2nc(C(c3ccccc3)O)nc2-c2ncn(CC(F)(F)F)n2)ccn1 N1(C(CCc2n(C)ncc2)=O)CCC(NC(=O)CCCCC(N)=O)C12CCC2 c1(NC2(NC(=O)NCC)CC(O)C2)ccc(S(N)(=O)=O)cc1[N+](=O)[O-] CCCC(C(O)C(=O)NCc1cnc(C)n1CC)NC(=O)CCOC c1(C(N2CCC(NC(C(CCC#C)O)=O)C(C)C2)=O)ccc2nc(O)sc2c1 Cc1c(C(N2CCCC(NC(C3CC(C)(C)C3)=O)C2)=O)[nH]c2ccc(F)cc12 c1(NC(C(CC)N(C)C)=O)ccc(OC)nc1C.C1CCCC(=O)N1 c1(C(=O)NCC(C)(CO)NC(=O)CC2CCCC23CC3)nc2cnccc2s1 N1(C(C(C=C)C)=O)CCN(CCNC(=O)C(C)C2CCCC2)CC1 c1(CC)cccc(C(=O)NCC2COCC2CNC(=O)CNC(=O)OC)c1 CCCCC(O)CCC(=O)NCC(C)(CNC(C1CC2CCC1CC2)=O)OC CCCCCCCC(C)CNC(C1CNC(=O)CO1)c1nnnn1C1CC1 C12(CC=C)CCCN(C1)C(=O)C(CC(C)NS(C)(=O)=O)C1C(C=CC1)C(=O)N2 C(=O)(C1CCc2ccc(OC)cc21)N(CCNC(=O)C1=CCC1)CC N1(C(CC(=O)N2CCOCC2)=O)CCOC2(CCN(C(=O)C(C)=CC3CC3)C2)C1.CO C1(CC(=O)NC2(C)CC(NC(c3ncc(F)cc3F)=O)C2)CCC(=O)NC1=O C(C(CC)CC)(c1nnnn1CCC1(C)CC1)NCCC1(COC)CCC1 Cc1c(C(C)(C)C2(N(Cc3nnnn3C3CCOC3)C)CC2)sc2nccn12 C1(C(=O)NC2CCC(NC(c3cc(Cl)sc3Cl)=O)C2)CC2(CCC2)CO1 N1(CC)CCC(=O)N(CC2CCC2OCc2cc(Cl)ccc2Cl)C1=O.C(C)(C)(C)O c1(COC(C)=O)ccc(C(=O)NCC2(O)CN(C(=O)CCn3cccc3)C2)cc1 N1(C(C#CC(C)C)=O)CC2(C(=O)NCCC3CCN(C)CC3)CC1CCO2 CC(C)(CCC(=O)NC1CC1NC(c1cnc(CC2CC2)s1)=O)[N+](=O)[O-] c1(OC(CC)C)cc(C(=O)N(C)CCN(C)C(c2cc[nH]c2C)=O)ccn1 C=Cn1nncc1C(N1CC2C(CC(=O)NC(CCC)CCO)C2C1)=O c1(C(=O)NCCC(=C)CNC(c2ccc3c(c2)CC3)=O)cc(=O)c(OC)c[nH]1 C(=O)(C(C)(C1CC1)N(C(=O)CSC(C)(C)C)C)NCC(C1CCCC1)OC C=CCC(CC(C)C)C(=O)NC1CC2CC(NC(c3cc(O)cc(=O)o3)=O)C2C1 c1(C(C(N2CC(NC(c3cc(OCC)n[nH]3)=O)C(O)C2)=O)C)cc(C)cc(F)c1 c1(C(=O)NCC(CC)NC(c2ccc3nonc3c2)=O)ccc2c(C)[nH]nc2c1 CCC(CNC(=O)C(C)Cc1ccc(C)cc1)(CC)NC(C1CCN1C(C)(C)C)=O N1(C(C(C(C)O)NC(=O)CCc2cn(C)nn2)=O)CCC(F)(C#N)C1 N1(C(CNC(CN(C)C)=O)=O)CC(NC(c2ccc(N3CCCC3)nc2)=O)C2CC12 C1(NC(C=CC=CCC)=O)CCCCN(C(=O)Cc2ccc(OCC)cc2Cl)C1 N1CCOCCC1CC(c1ccccc1)O.Cc1cc(CC(=O)OC)n[nH]1 Cc1c(CC(=O)NCC2CCN2C(=O)COC2CCCCO2)cnn1C N1(C(CCC)=O)CCC(C(F)F)(CNC(=O)Cn2ncccc2=O)C1 C1(CN(C(C(CC)=CC)=O)CC)CCCCN1C(C1CC=CCO1)=O c1(C(C)Nc2ccnn2CC2(Cc3ccc(F)cc3)CC2)cc(F)ccc1F C1(COCC)CCN(C(C2(C)CN(C(=O)CC3CCC(C)(C)O3)C2)=O)CC1 c1(C(=O)NC2C3(CC(NC(C(CCC)(C)O)=O)C3)C2)nccc2cc[nH]c12 C(=O)(C1=CCCN(C(c2ccccc2F)=O)C1)NC(c1ccc(F)cc1F)C C(=O)(N=c1ccn(C2CC2)[nH]1)C1OCCN(C(C(C)NC=O)=O)C1 C1(C(=O)NC(C#C)CC(C)C)C2CC3C(C2NC(=O)C(c2cnn(C)c2)=O)C13 N1(C(C2(C(F)(F)CF)CC2)=O)CCOCC(C(F)(F)F)C1 C#CC(C(C)(C)C)NC(=O)C(C)(CSC)NC(=O)Cc1ccccc1F Cn1nc(CNC(=O)OC(C)(C)C)c(I)c1C(N1CCC(N2CCC2)C1)=O N1(C(c2ccnc(OC)n2)=O)CCOC2CN(C(c3ccc(C)c(C)n3)=O)CC12 N1(C(C2N(C(C(C=C)C)=O)CCC=C2)=O)CCC(C(=O)OC)C1(C)C N1(C(c2oc(CC)c(C)c2)=O)CCCC2C1CCCN2C(=O)CN(C)C(C)=O c1(-c2c(CC)nn(C)c2)nc(C2CCOc3ccccc32)nn1CC(C)CO c1(C(N2CC(CC=C)(NC(C3CC3c3ccco3)=O)C2)=O)noc(C2CC2)c1C N1(C(C(CCC(N)=O)NC(C)=O)=O)CCCC(C2CN(C(=O)COC3CC3)C2)C1 C(C(F)(CCC)C=O)NC(C)CN(C)C C(CC1CCC1)(C(=O)NC1CCCC1NC(=O)NC(C)(C)C)NC(C(C)C)=O C1(C(N2C(C)(C)CC(C)(CNC(C3CCCCS3)=O)C2)=O)C2CCC1(C)C2(C)C CCC1=C(C(=O)N2C3CN(C(=O)C(C4CCC4)OC)CC23)CCCO1 C=C(C)CCC(C)NC(=O)C(C)=CCNC(c1cncc(O)c1)=O c1(C(N2CC(N(C(c3c(C)nc(CC)o3)=O)C)C2)=O)n[nH]c2cc(C)ccc12 c1(CCC(=O)N(C2CCN(C(=O)CCCC(C)=O)C2)CC)cnc2n1CCCC2 CC1CN(C(C2CCCC2(C)C)=O)CCC1CNC(=O)CC12CCC(CC1)CC2 C1(NC(C(C)N(C(C2CCC(F)CC2)=O)CC)=O)CN2CCC1(F)CC2 c1(C(=O)NCC2CCCCN2C(C2CC2c2ccccn2)=O)occ2c1CCOC2 n1(CC)cccc(NC(=O)C(CC2CCC2)NC(=O)C(C2CCC2)OC)c1=O C1(C(N2C(CNC(Cc3cc(OC)ncc3)=O)C=CC2)=O)NC(=O)C2CCC12 c1(C(=O)NC2CN(C(c3c(C)noc3)=O)CC3(C2)CC3)cc2c([nH]1)CCCC2=O c1(CNC(N2CC(n3ccnn3)C2)=O)ccnc2[nH]ccc12 Cc1ncc(SC2CCN(C(=O)CC3CC3C3CC3)CC2)nc1C N(C(=NCCN1CCC(C)C1)NC1CC(C(=O)OC(C)(C)C)C1)CC=C N1(C(CC(COC)C)=O)CCCCC(CNC(c2cccc(C(N)=O)c2)=O)CC1 C1(C(C)(C)C)CCc2nc(NC(=O)C(=O)NN3CCC(=O)NC3=O)sc2C1 N1(C(c2scc(C)c2)=O)CC(NCc2ncccc2Br)C(C#N)C1 C(C1CCOC1)=CC(=O)NC1CC(F)(CNC(=O)C(O)Cc2ccccn2)C1 Cc1ccc(C(=O)NC(C2CN(C(c3ccc(Cl)nc3)=O)C2)C)cc1C(F)(F)F c1(C(=O)NC2(C)CC(NC(=O)C(C#N)C(C)(C)C)C2)ccc2nc[nH]c2n1 C1(CNC(c2c(Cl)cn(CCC)n2)=O)CN(C(=O)C=CC(C)C)CC2(CCC2)O1 Cc1cc(C(N2CC3CN(Cc4ccsc4Br)C3C2)=O)ccc1[N+](=O)[O-] N1(C(CCCC)=O)CCOC2CCN(C(=O)C(O)c3ccco3)CC12 c1(C(=O)NCC(C)(C2CC2)NC(C(C=C=C)C)=O)ccc(F)c(OC)c1 n1(CC(=O)N(CCC)CCNC(=O)CC2CCOC2)nnc(-c2ccsc2)n1 CC(C)(C)CC(F)C(=O)N1CC(C2(NC(c3cc(C(N)=O)co3)=O)CC2)C1 C(CC(C)(C)C)(C(=O)NC(c1nn(C)cc1O)C)NC(C(C)=CC=C)=O C(=O)(CCS(C)=O)N1CC(C(=O)NC(c2nnc(C)o2)C)(COC)C1 N1(C(C2CC(CCC)C2)=O)CCC2CCN(C(c3cnn(C)c3C(C)C)=O)C2C1 C1(OC)CC2(C1)CC2NC(=O)C(c1ccccc1Br)N1CCCCC1 C1(C(=O)NC2CC(C(C)O)C2)COCCN1C(C1CC2CCC2C1)=O C(=O)(C1CCc2nccn21)NCc1c(C(=O)NC2(C(=O)NCC)CC2)ncs1 Cc1nncc(C(N2CC(OCC(=O)N(C(C)C)C3CC3)C2)=O)c1C C1(C(=O)NC(CC)CNC(=O)C=C(C)c2cccs2)CCCCC(=O)N1 CC1(C)CCCN(C(=O)CC2NC(=O)NC2=O)C1C(=O)NC1CCn2nnnc2C1 c1(OC)ccc(C(N2CCC(OC)C3CC23)C(=O)NC2CC2)c(C)c1 c1(C(=O)NCC=CCC(=O)Nc2c(OCC)nccc2)cccc(C)c1C c1(OC)ccc(C(N2CCN(C(=O)CC3CCC3)C(C(C)C)C2)=O)nc1Br c1(C(N(C)CC2CCN(C(=O)Cc3cccc(Cl)c3)C2)=O)cc2cc(Cl)sc2[nH]1 N1(C(C(CC)SC)=O)CCC2CCN(C(=O)C(F)(F)CC)CC12 CC(O)C(F)(F)C(=O)NCC1(CNC(c2ccc(CN=[N+]=[N-])cc2)=O)CC1 Cc1nn(C)cc1C(C)C(=O)NCC=CCNC(c1cc(C(C)(C)C)ccn1)=O C1(c2c(CNC(=O)Nc3c(I)cnn3C3CCCC3)n[nH]c2)CCC(CO)CC1 CC1CC2(CC(C(N3CCN(C(=O)C#CC4CCC4)C(CC(F)F)C3)=O)C2)C1 C12(CS(=O)(=O)NC(C)=O)CN(C=O)CC1CCO2.c1(C)c(F)cccc1Cl.C12CC(C1)N2 CCCCC(CC(=O)Nc1ccc(O)c(Cl)c1)NC(=O)C=C(C)c1ccco1 N1(C(C(C)=O)=O)CCC2(CC1)CN(C(=O)C(c1ccc(C)cc1)(C)C)C2 C(=O)(CN=S(C)(C)=O)NCCCC(C)NC(C(C)CO)=O N1(C(c2ccc(OC)nc2Cl)=O)CC2CCCN(C(=O)CC3(O)CCCC3)C2C1 c1(CNC(=O)NC(c2nc(=O)o[nH]2)C)csc(Br)c1Br CN1CC2(CCC2)CCC1NC(=O)NCC(C)(C)S(C)(=O)=O c1(C(=O)NC23CC(NC(C45CCCC4C5(F)F)=O)(C2)C3)[nH]c2ccccc2c1Cl C1(NC(C2(F)C3CCCC23)=O)CCN(C(C23CCCC2(C(N)=O)C3)=O)CC1 N1(C(C(C)C(=O)OC(C)(C)C)=O)CC2(CCN2C(=O)Cc2ccc(F)cc2)C1 C(=O)(CCCC(C)(C)C)NCCN1c2ccccc2C1=O.c1(NC(C)=O)csnn1 CC1(CNC(C2CC3CCCC23)=O)CCN(C(=O)CCn2ccc(=N)[nH]2)CC1 N=c1cc[nH]cc1C(N1CCCC(CNC(c2ccsc2C2CC2)=O)C1)=O Cc1cc(=NCc2ccc(Cl)cc2C)[nH]c(=NCCC2CC(C)(C)CO2)[nH]1 CC1CN(C(C2(c3cc[nH]n3)CCC2)=O)CCN1C(=O)Cc1ccc(O)c(F)c1 N1(C(C(C)OC)=O)CCn2c(nc(C(=O)Nc3ccc4c(c3)CCO4)c2Cl)C1 N1(C(=O)NC(c2nn[nH]n2)C)CC2(CCCN(CCO)C2)C1 c1(C(c2n(C(C(=O)OC)C)nnn2)NCC(C)(C)C2CCC2)ccc(C)c(I)c1 C(=O)(CCC(=O)N(C)C(C)C)N1CCC(CCC(=O)N(C(C)C2CC2)C)C1 CC1(C)CC(CNC(C2CC23CC3)=O)CN(C(=O)CCn2cc(Cl)cn2)C1 C1(C(=O)NCC(C)CNC(c2ccc3oncc3c2)=O)CCC(S(N)(=O)=O)CC1 C1(NC(c2c(C)cccc2)=O)CCCN(C(=O)CCc2cnn[nH]2)C1C C1(C2CCC2)(CNC(C2=C(C)OCC2)=O)CCN(C(c2cc(C#N)on2)=O)CC1 N12CC3CC1CN3C(=O)CC(CCCCC)CCC1CC(C1)C(=O)NC(C)C2=O C(=O)(CC1CCCc2oc(C)nc21)NCC1N(C(c2nc(C)sc2)=O)CCCC1 CCC(C(C)CN(C)C)(c1nnnn1C1(C)CC1)NCCc1cc(C)cc(F)c1 c1(CNC(C2CC2C(N2CCCC(F)CC2)=O)=O)cccc(Br)c1Br N1(C(c2c(C)nncc2)=O)CCOC(C(=O)NCC2(C)CCCC2O)CC1 C1(OC)CC2N(C1)C2=O.c1(NC(=O)CNc2ccccn2)cc(Cl)n(C)n1 C1(C(=O)Nc2cccc(OC)c2)CC2(CCC2)CN1C(=O)Cc1cc[nH]n1 N1(C(c2ccc(C)s2)=O)CCN(C(=O)CCC2CC2(F)F)C2CS(=O)(=O)CC12 C1(=CC(=O)NCC(C)CNC(=O)Cc2coc(-c3ccccc3)n2)CCOCC1 C1(NC(C(C2CC2)OC)=O)C2CC1CN(C(=O)CC1CCCN(S(C)(=O)=O)C1)C2 CC(CC(=O)NC(C)(C)CCNC(c1cccc2c[nH]nc12)=O)CC(F)(F)F C(=O)(CCCCCO)N1CC(CNC(CCc2cccc(OC)c2)=O)C(F)C1 C(=O)(C#CC1CCC1)NC1C=CCN(C(CCCCSC)=O)C1 C(=O)(C(C(CC)CC)OC)NC(CC#C)(C)C(=O)NCC1=CCCC1 Cn1ccc(C(=O)NCC2(C)CC(NC(=O)C=Cc3nccs3)C2)c1C1CCC1 N1(C(CC(C)OC)=O)CCC2(CC1)CC2NC(c1c(NC(C)=O)c[nH]c1C)=O C(=O)(C1=CCC(C)(C)CC1)N1CC(NC(c2c(C)c[nH]n2)=O)C(C2CC2)C1 N12CC=C(CN(C)C(=O)CCC(=O)N1C)CC2.Cc1nc(CN2CCCC2)cs1 CCC(C#N)(CC)C(=O)N1CCOC(C(=O)N(C(C)CC2CC2)C)C1 c1(C(=O)NCCCNC(C2C(C)(COC)C2)=O)cc(C(F)(F)F)ccc1N C(=O)(C#CC1(C)CCCO1)NC(CCCCNC(Cc1cc(C)nn1C)=O)C C(C)(N=c1[nH]c(=NC)[nH]c(=NCC2=CCCCC2)[nH]1)c1cc(OC)cc(C)c1 CC1c2c[nH]nc2CCC1C(=O)NCC1CCN1C(C1(F)CCS(=O)(=O)C1)=O C1(CNC(C2(CNC(C3C(CC(C)C)C3)=O)COC2)=O)(CO)CCN(C)C1 C(=O)(C1=CC2(CN(C(=O)CCC(=O)C3CC3)C2)OC1)NCCC1(C)N=N1 CC1C(C(=O)NC2CC(C(N3CCNC(=O)C3C)=O)C2)=NOC1C Cc1nscc1N(C)C(C1(NC(=O)COC(C)(C)C)CC1)=O C1(OCCN(C(C2(CC)CC2)=O)C2CC2)CCN(C(=O)C(C)CSC(F)(F)F)C1 CCC(CC)C(C)C(=O)N1CC(CC(=O)NCc2nnn(C)n2)CC1(C)C C1(CC)CCCN(C(=O)NCc2nc(C)n(-c3cccc(C(F)(F)F)c3)n2)C1C N1(C(C(C2CCC2)OC)=O)CCc2cc(CNC(c3cncnc3)=O)ccc2C1 N1(C(CN(C(C)=O)C)=O)CC2CCCC(NC(c3ccc(CN(C)C)o3)=O)C2C1 c1(C(=O)NC2C(NC(C3(OC)CCS(=O)(=O)C3)=O)CCC2)cc2c([nH]1)CCCC2 C1(C(N(CC(=O)NC(CNC(C2CCCC2)=O)C2CCC2)C)=O)CC12CC2 c1(CC2CCN(C(c3cnc(C)s3)C(=O)NC(C)C)C2)cccc(Cl)c1 N1(C(Cc2cc(C)c(C)nc2)=O)CC(C)N(C(C2CC(=C3CCC3)C2)=O)CC1C c1(N2CCC(SC)C2)nc(=N)[nH]c(=NCC2(N(C)CC)CCC(F)(F)CC2)[nH]1 Cc1cc(O)nc(CNC(=O)CC2N(C(c3ccncc3O)=O)CCC2(C)C)n1 C=C(Cl)CCC(=O)N1CCC(C(N2CCC(F)(CO)C2)=O)C1C(C)C Cc1nccc(NC(=O)CC2CCCN2C(c2cncc(O)c2)=O)n1 C(=O)(CCC(=O)N(C)CCN(C)C(c1ccccc1N(C)C)=O)NC.C(C(C)O)N N1(CC)CCN(C(=O)CC(C(F)F)NC(=O)C(CC)n2cncn2)CC1=O C1(CC(=O)NCCN(C)C(C2(C)CCOCC2)=O)CCCC(F)(F)C1 C1(C(=O)NCCCCCNC(c2c(C(=O)OCC)c[nH]c2)=O)C(C)(C)C1(F)F C(c1ccccc1Cl)=C(C(=O)NC1CC(C(C)NC(CCCC=C)=O)C1)C C1(C(=O)OC)CC(C)=CCN1Cc1ccc(OCCO)cn1 C(N=c1cc(NCc2ccc(-c3cccs3)s2)nc[nH]1)C1(S(C)=O)CC1 c1(C(N2C(CNC(CCc3n(C)ccn3)=O)CCC2)=O)ccc(Cl)o1 N1(C(c2c(N)ncc(Br)c2)=O)CCCCC2(C1)CN(C(=O)Cc1cnoc1)C2 C1(NC(C2(N3CCCCC3)CCCC2)=O)CCC2CN(c3cnc(F)cn3)CC2C1 c1(C(N(CCN(C(C2CC2C(C)(F)F)=O)CC)CC)=O)coc(COC)n1 C12(CCNC(COC)=O)CCC1CN(C(c1cc(C)c(Br)cn1)=O)C2 c1(C(=O)NCC2(O)CC(NC(C3(C=C)CC3)=O)C2)c[nH]c2cccc([N+](=O)[O-])c12 N1(C(c2nc(CC)oc2)=O)CCCC2(CCN(C(=O)CC3CN(C)C3)C2)C1 C(=O)(C1=C(C)N(C)c2nnnn2C1)NC(C(=O)OC)C(C(C)C)OC c1(C(N(CCCNC(C2C(CC)CCC2)=O)CC)=O)ccc2cncn2c1 N1(C(C=CCCC)=O)CC(OC(F)F)C(C=O)C1.C1(CC)CCC(OCO)C1 C(CN=c1[nH]c(=NCCCOC)c2ccccc2[nH]1)c1cn(CCC=C)nn1 C1(NCc2cccc(F)c2)CC2C3CCC(O3)C2C1 c1(OCC(=O)NCC2(O)C(C)CCC2)ccc2c(c1)OCCCO2 Cc1ccccc1CC(N1CCOC(CNC(C2CCCO2)=O)C1)=O Cc1ccc(CN=C(NC(C)C2CC2)NC2(O)CCOCC2)cn1 c1(C(=O)NC2C(C)(C)N(C(c3coc(Cl)c3)=O)CC2)cnc2sccn2c1=O C12(CNC(=O)C(c3cccnc3)O)CCC(CC1)N2C(=O)CCCC(F)F Cn1ccc(-c2nc(C(=O)OCC(C3CC4CC4C3)=O)cs2)c1 C(=O)(C(C)(C)COC)N(CCCNC(C1(CO)CCOC1)=O)CC C1(CC(=O)NCCc2cc(C(N(C3CCC3(C)C)C)=O)no2)CC2(CCC2)C1 C1(COC)CN(C(c2ccn(C)c(=O)c2)=O)CCC1NC(=O)CC1CSCCS1 c1(C(=O)NC(C(C)NC(CCCc2ccc(C)s2)=O)C)cccc2nc(O)[nH]c12 C1(NC(=O)CN2CC(=O)NC2=O)(CO)CCCN(C(=O)CSc2cccs2)C1 c1(C(N2CC(CNC3CN(C(CCSC)=O)CC34CC4)C2)=O)ccc([N+](=O)[O-])n1C C=C(C)CC(C(=O)NCCOc1ccncc1)NC(c1cc(C)ncc1C)=O C(=O)(CC(C)c1ccco1)N(CCN(C(c1csc(C2CCCC2)n1)=O)CC)CC N1(C(C=CCC)=O)CC(C(N2CC=CC(OCC)C2)=O)C(F)(F)C1 c1(C(=O)NCC2C(NC(c3cncc(C)c3)=O)C2)cnc(C2CC2)nc1C C1(NC(Cc2ccc(C)nc2)=O)CC2CC1N(C(c1cc(Br)nn1C)=O)C2 N1(C(c2nc(COCC)sc2)=O)CCN(C(c2nnc(CC)s2)=O)CC1C c1(C(=O)NC(CCOC)CNC(C2CC3CC2CO3)=O)ccc(C)cc1F N1(C(C2CC(C)OC(C)C2)=O)C2CCCC1CC(NC(c1cc(C#N)c[nH]1)=O)C2 C1(CC(=O)NCC2C(CNC(=O)CCSC(F)(F)F)C2)CCCCC(=O)N1 C1(O)(C(=O)NC(C(=O)Nc2c(C)n[nH]c2)C2CC2)CCOCC1 CC1CC2(CCN(C(C3CC3F)=O)CC2)CN1C(C1CCC2(CC2)C1)=O c1(OC(C(=O)NCCC(C)NC(=O)C=C(Cl)Cl)C)ccccc1 c1(OC)ccc(Cl)c(C(=O)NC23CC2CN(C(=O)CC(C)c2ccncc2)C3)n1 c1(C(=O)NCC2C(NC(Cc3n[nH]c(=NC)s3)=O)C2)cc(S(N)(=O)=O)cnc1C N12CCC(CC1)C(c1nnnn1CCCF)CC2(COC)C.C(C=CCl)SC Cc1ccc(-c2cn(CCCCCCC3CCCN3C(=O)CC(C)F)nn2)cc1 N1(C(C2CC(=C)C2)=O)CCN(C(=O)C=C(Cl)Cl)CC1c1cccc(Cl)c1 c1(NC(C(=O)NCCN(C2CCCC3CC23)C(C)=O)=O)c(C)ccc2cccnc12 c1(C(=O)NCC2CN(C(c3cnc(C4CCC4)[nH]3)=O)C2)cc(Cl)nnc1Cl N1(C(CC2(C)N(C(CCN(CC)CC)=O)CC2)=O)CC(C(N)=O)C2(CC2)C1 c1(C(=O)NCC(CNC(C2C(C=C)C2)=O)C)cnnn1C c1(-c2ccn(C)n2)ccc2ncc(-c3ccc4nccc(OC)c4c3)c(=O)n2c1 C1(NC(CSCC=C)=O)CN(C(=O)C(c2ccc(C)cc2)(C)C)CCC1C(F)(F)F C1(C)(C(N(C2CCCC2C#N)C)=O)CC(O)CN1C(=O)C(=O)C(C)(C)C c1(CC(C)NC(=O)C(=O)NC2CCNCC2(C)C)c[nH]c2ccc(F)cc12 CCS(=O)CC(=O)NCC1(CNC(=O)C(CC2CCCC2)CC2CC2)CCCC1 c1(C(=O)NC2C(NC(C(C)CSc3ccccc3)=O)CC2)n[nH]c2c1COCC2 c1(C(N(CCCCCNC(c2n[nH]c(C)c2F)=O)C)=O)ccn2ccnc2c1 c1(C(=O)NC(CNC(C(C)n2cncn2)=O)CO)c(F)cc(O)cc1F C=CCC(CNC(C1CN2CCN1CC2)=O)C(=O)NCc1ncccc1F Cc1ccc(C(N2CC(N(C(=O)CCCN3CCCC3)C)C3(CC3)C2)=O)nc1O C(c1cncnc1O)=CC(=O)NCC1C(CC)CCN1C(C1CC(O)C1)=O N#CC1=C(C(=O)N2CC(CNC(C34CC(F)(C3)C4)=O)OC(C(F)(F)F)C2)CCC1 C(c1cccnc1C)=CC(N1CC2C(CNC(CC=C(C)C)=O)C2C1)=O C(=O)(CCC(C)(C)NC(c1cnc(Cl)n1C)=O)NCC(CC)n1cccn1 c1(NOCCNC(CNC(c2c(OC)n(C)nc2)=O)=O)c(C)ccc(C)c1F.O C(CC(C)C)(C(=O)NOCCC(C)C)NC(CC=C=C)=O C1(C(N2C(C(=O)NC)CC2)=O)C=CCCN1C(C1CCCN1C=O)=O N1(C(C2C(C)(C)C2(C)C)=O)CCC2CN(C(C3(C4CCCCO4)CC3)=O)C2C1 CC1=C(CC(=O)NC2C3CC4CN(c5nnc(O)s5)C2C4C3)c2ccccc2C1 N1(C(CC(C(C)C)OCC)=O)CC(C(=O)NCC23COC(CCO2)C3)C(C)(C)C1 N1(C(c2c(-n3cccc3)cc(C)s2)=O)CC(NC(C2CCCS2)=O)CC(O)C1 O=C1NC(C(N2CCC(C(c3ccc(O)cc3)=O)CC2)=O)C2CCCC12 c1(C(N2CC(N(C(C3CN(CC)CCO3)=O)CC)OCC2)=O)ccc(F)c(I)c1 C#CCCC(O)C(=O)NC1CN(C(=O)C=Cc2ccc(SC)s2)CC1OC CC1CN(C(=O)C(F)CC2CN(C(C3(C#N)CCCO3)=O)C2)CC1N=[N+]=[N-] C1(CCNC(C2(C(C)C)CCC2)=O)CCCN(C(=O)CC2CCCCO2)C1 C1(NCc2nc(C(C)O)nn2-c2cccnc2)CCCN(S(CCC)(=O)=O)C1 N1(C(c2coc(O)n2)=O)CCOCC1CCNC(C1(F)CCOCC1)=O c1(C(=O)Nc2cc(Cl)c(F)cc2F)cc2cccc(C(F)(F)F)c2nc1Cl C1(CNC(C2C(CC)C2)=O)CN(C(c2ccsc2Cl)=O)CCN1C O=C(C(F)CC1CCOC1)NCC1CCN1CC(=O)NC1CCOC1C1CCC1 CC1OCCN(C(c2ncc[nH]2)=O)C1C(=O)NCC1C(CO)C1(C)C C1(F)(CNC(CCc2ccc(C)o2)=O)CCC(NC(=O)CCN2CCC(F)C2)C1 N1(CC(=O)NC(c2cccnc2)C(=O)NC(CC#C)CO)C(=O)CCC1=O N1(C(Cn2nc(C)oc2=O)=O)CCN(C(C2CCC(=O)NC2)=O)C(C)C1 C=CCC(CC(F)F)NC(=O)CC1CN(C(=O)CC2CCCSC2)CC1C=CC C1(N(C)C(c2ccc(F)cc2)=O)CC2CCC(C1)N2C(C1CC1C1CC1)=O N1(C(c2scnc2Cl)=O)CCCN(CCCNc2n(C)nnn2)CC1 Cc1ccc(C)c(C(=O)NC2CCN(C(c3sc(C)nc3C)=O)C(C)C2)c1 C(CNC(=O)CN1CCOC1=O)(CC(=O)N(CC(F)F)CC1CC1)OC c1(CNC(CC=C)C2CC2)ncnc2scc(-c3ccccc3)c12 S(=O)(=O)(c1ccc(Cl)s1)NCCC1c2c(cccc2[N+](=O)[O-])CN(CC)C1=O C1(C(N2CCC(Oc3cccnc3)C2)C(=O)NCC(C)C)CCOCC1 S(=O)(=O)(c1ccc(F)c(C(=O)NCCN(C(=O)C(C)SC(F)(F)F)C)c1)NCC C1(C(=O)NCC(=C)CC(=O)NC(CCC)c2nn[nH]n2)CCC2(CC1)CC2 C(=O)(C(C)CCC(C)(C)C)N(C1(C2CCC2)CC1)C.C#CCC1C(=O)N1 c1(C(C)NC(C2CC(F)(CNC(C3(C)CC3)=O)C2)=O)ccc(NC(N)=O)cc1F N1(C(CCSCCCC)=O)CCC2CCN(C(c3ccncc3F)=O)C2C1 c1(C(=O)OCC)ccc(NC(c2csc(=NCc3cncc(C)c3)[nH]2)=O)c(I)c1 N1(C(=O)Cn2ccnn2)CCCC(O)(C(N2CCCC(OCC3CC3)C2)=O)C1 CCC1=NOC(C(=O)NC(C)(C)CCCNC(C2CC(=O)N(C3CC3)C2)=O)C1 c1(C(=O)OC)cccc2c(CN3CC4(F)CCC3(CO)C4)ccnc12 N1(C(c2cc(C(C)=O)cn2C)=O)CC2CN(C(=O)Cc3ccoc3)CCC2(CO)C1 Cc1cc(CC(=O)NC(C)(C)CC(=O)NCC(F)(F)C(C)O)n(C)n1 C(=O)(CS(=O)(=O)C(C)C)NCC1(C)N(C(=O)CC23CCC(CC2)C3)CC(OC)C1 N1(c2c(C(=O)OC)cnc(C)n2)CC2CCC1C(NC(=O)CC1CC1C)C2 N1(C(C2CC(NC(COC3CCCC(C)C3)=O)C2(C)C)=O)CCCC(F)(COC)C1 c1(OCC)cnc(C(=O)NCCC(C)N(C(=O)C=CCCC(C)C)C)nc1 c1(C(N2CCC(C(C)CNC(=O)Cc3cnccn3)CC2)=O)cnc(Cl)c(F)c1N C(CC(=O)NC1CC(CCC(=O)NCCCc2ncon2)C1)NC(C)=O c1(C(N2CCC(CNC(c3c(C)cc(O)nn3)=O)CC2)=O)cc[nH]c2nccc1-2 c1(C(N2CCCC(CNC(C3(CSC)CC3)=O)C2)=O)cccc2occc12 C(CN=c1cc(C)nc(-c2ccccn2)[nH]1)NC1CN(C(c2cc(CC)[nH]n2)=O)C1 C(=O)(C(C)C(F)(F)C(F)F)NCCCNC(C=C)=O.C#Cc1cc(C(=O)OC)cc(F)c1 N1(C(c2ccc(C#N)s2)=O)CCC2CCN(C(=O)Cn3ccc([N+](=O)[O-])n3)C2C1 c1(C(=O)NCC(C)N(C(c2cc[nH]c2)=O)CC)csc(C(C)(F)F)n1 CCCCCCCCC(=O)NC1C2CC1N(C(c1cnn3c1CCC3)=O)C2 N1(CC(=O)NCC(C)NC(C2(C)CCNC2=O)=O)CCCCCCC1=O C1(N(C(c2cc(C)no2)=O)C)CC2CCC(C1)N2C(c1cncnc1C(C)C)=O C(=O)(CC(O)CNC(C1CC(NC(C23CSCC2C3)=O)C1)=O)NCC CC(C)(C)S(=O)(=O)CC(=O)NC1CC(CNC(=O)CCCc2ccncc2)C1 C(=O)(CN=c1cc[nH]cc1)NC(C1CN(C(=O)C(c2ccccc2)F)C1)C c1(C(N2CC(C(=O)OC)N(C)CC2)C(=O)NCC2CCOC2)cc(C)c(C)cc1C c1(C(CC)NC(=O)C(C)NC(C2(CC(N3CCCC3)=O)CCC2)=O)cnn(C)c1 C1(CNC(C2C(NC(C3C(C)CCO3)=O)COCC2)=O)CC[Si](C)(C)C1 C(C(C(=O)NC1CCC(CCNC(c2ncsc2C)=O)C1)NC(C)=O)OC C1(C(=O)NCC(CN(C(=O)CCn2cccc2)C)(C)C)CCCN2CCCCC12 c1(C(=O)NCC(CC)NC(C2(CC)CC2(F)F)=O)cc(C#N)n(C)n1 N1(C(C(CC(=C)C)NC(C2CC3C=CC2C3)=O)=O)CCn2ncc(C)c2C1 CC1CCCC1(C)C(N1CCN(CCNC(C2CC(F)(F)C2)=O)CC1)=O N(C1CCCn2nccc21)C(CC(C(F)F)NC(CCC=C)=O)=O CN1CCC(C(=O)NC2CC(n3cc(-c4ccccn4)nn3)C2)S1(=O)=O c1(C(=O)OC)cc(C(N2CC(N(C(=O)C(C)CC(C)C)C)C(O)C2)=O)ccc1C c1(C(=O)NC2(CO)CN(C(c3c(C)sc(O)n3)=O)C2)ccc(Br)c(F)c1 N1(C(c2c(C)[nH]cc2)=O)CC2(NC(C3CCCC3C(N)=O)=O)CCCC2(F)C1 N1(C(c2cnc(OC)s2)=O)CC(CNC(c2cc(C)oc2C)=O)CCC1C C1(C(CNC(Cc2ccn(C(C)C)n2)=O)(C)O)CCN(C(c2ccsc2)=O)CC1 C1(N(C)C(C2CCOC2)=O)CCC12CCN(C(c1ccc(OCCF)cn1)=O)CC2 N1(C(C(C)(C)NC(c2ccc(C#N)o2)=O)=O)CC2CC=CC1C2 C1(C(F)(F)F)(C(=O)NCC2(C)CC(NC(=O)Cc3ncccn3)C2)CCCCC1 C(c1cccc(Cl)c1)=CC(=O)NCC(=C)CCNC(c1ccc(C(N)=O)[nH]1)=O C1(OCC)CCN(c2cccc(C)c2)C1=O.C12CN(C1)C(=O)C1(CC1)C(=O)NC2 Cc1ccc(C=CCC(=O)NC(C)C(C(C)C)NC(c2ccc(=N)[nH]n2)=O)cc1 c1(OCC)cc(CN(C)C(c2ccc(SN3CCC(CC)C3)cc2)=O)ccn1 c1(CN2C(C(=O)NCC(O)C(F)(F)F)CC(OC)C2)cc(Cl)ccc1C N1(C(c2cnn(C3CCC3)c2C)C(=O)NCCOCC)CCOC(C)C1(C)C C1(CC(=O)NCCC2(NC(C3CC4(C3)CC(O)C4)=O)CCC2)CC2CCC1CC2 CC1(C)CN(C(C2CCCO2)=O)C(CNC(c2ccn3cncc3c2)=O)CO1 C1(NC(c2c(CC)c(F)ccc2)=O)CCCCN(C(=O)C=Cc2nccs2)CC1 c1(C(C)C)ccc(C(C)CC(=O)NCCCCOc2ccc(Br)cc2)cc1 c1(C(=O)NC2CN(C(c3n(C)cc(C(F)(F)F)n3)=O)C2)cc(Cl)c(O)c(Cl)c1 C1(C(=O)NC2C3CN(C(C4CN(C(N)=O)C4)=O)CC32)CCCCC1C1CC1 c1(NC(C2CCN(CCc3ccc(F)cc3F)C2)C)c[nH]c2cc(C#N)ccc12 c1(-c2cn(Cc3nc(-c4ccc(F)nc4)sc3)nn2)cccc2ccoc12 C1(CN(C(=O)CCCN(C(=O)CC2CCC2)C)C)CCCC(O)C1 C(=O)(CCCC=C)NCC1(OCC)CN(C(c2nc(Cl)oc2C)=O)C1 C1(NC(c2ccn(C(C)C)c(=O)c2)=O)CC2CCC(C1)N2C(c1ccoc1Cl)=O CC1(C)CC(NC(c2ccc(Br)cc2)=O)CCN(C(=O)CCCCCF)C1 C1(CNC(c2cccc(Cl)c2)=O)COCCN1C(c1nc(C(F)(F)F)cs1)=O C#CCCC(O)CCNC(=O)CC(C)CNC(c1cc(Cl)n[nH]1)=O c1(NCC(CCOC)OC)cc(C)c(S(=O)(=O)NCC2CC2(C)C)cn1 C(=O)(CC(C)(O)C(F)(F)F)N1CCCC(NC(CCOCC)=O)(CC)C1 CCC(O)C(F)(F)C(=O)N1CCC(CF)(NC(c2cnn(C(C)C)c2C)=O)C1 C(C(CNC(c1cccnc1)=O)C(F)(F)F)NC(C(C)COC(C)(C)C1CC1)=O C1(CC(=O)NCCC(C)N(C)C)CC(NC(C23CC2CNC3=O)=O)C1(C)C N1(C(CCCNC(c2oc(C)c(CO)c2)=O)=O)CC(C)(C)OCC1(C)C Cc1cc(C)nc(SCC(N2CC(CNC(=O)C=CC(=O)NC3CC3)C(O)C2)=O)n1 c1(C(C(=O)NCC(CNC(c2ccc(F)s2)=O)CO)OC)ccccc1O Cc1ccn2cc(C(N3CCCC(C)(CNC(=O)C(C)C(F)(F)F)C3)=O)nc2c1 c1(CC(C)NC(c2cccc(C(C)N(C)C)c2)=O)cc(I)cc(I)c1 c1(C(N2CC(C)(C)C(NC(c3ccsc3Cl)=O)C2)=O)ccc(O)c(N=[N+]=[N-])c1 CCC(CC)C(C(=O)NCCN(C)C(c1csc(C(F)(F)F)c1)=O)OC C(=O)(CCCC(C)(C)C#N)NC(CCC(=O)N(C)Cc1nccc(C)c1)C CC(CC(=O)NCCCN1CCN(C(C2(C)CC2)=O)CC1)CC(F)(F)F c1(C(=O)NCCN(C(=O)CC2C=CCC2)CC)ccc(C(F)(F)C(=O)NC)nc1 Cn1cc(NC(=O)NCC2(n3cnnn3)CC2)c2ccccc12 n1(CCNC(C2CC2C(=O)O)=O)cnccc1=O C(=O)(C(CC(C)C)OC)NCC1(O)CCN(C(CCN(CCC)C)=O)C1 N1(C(Cc2c(C)n[nH]c2)=O)CCC2(COC(CNC(C3CCN3C)=O)C2)C1 C=CCC(C)(C)C(=O)NCC1C(CNC(=O)CC2CCC3CC23)C1(F)F C1(CNC(c2c(C)scn2)=O)CN(C(c2[nH]c(C3CC3)nc2C)=O)CC12CC2 CC1N(C(c2scc3c2OCCO3)=O)CCC12CCOCC2 N1(C(C=CC(C)=O)=O)CCC(F)C(NC(c2coc(C(C)(C)C)n2)=O)C1 CN1CCC(C)(C(=O)NCC2C=CCN2C(c2cc(C(F)(F)F)cs2)=O)CC1 C1(C(C)(C)CNC(=O)CCC2CC2(Cl)Cl)CN(C(=O)CCc2cn(C)cn2)CCO1 c1(C(=O)Nc2ccc(-c3n(C)nnc3)c(C(F)(F)F)c2)c(Br)c(Br)nn1C N1(C(c2n(C(C)C)cnc2)=O)CCOC(c2ccc(-c3nn[nH]n3)cc2)C1 C12(NC(C3COC4COCC34)=O)CCCN(C(=O)C=Cc3cocn3)CC1C2 N1(C(C(C)(C)C2(O)CCOC2)=O)CCCC(CO)(Nc2cc(O)ncn2)C1 Cc1cc(Cl)cc2[nH]c(C(=O)NC3CN(C(=O)CC4CC5CC5C4)CC3O)cc12 N1(C(C2OCCN(CC)C2)=O)CCCC2(NC(=O)C#CC(C)C)CCCC12 c1(CC(N2C(C(=O)NC)CCC2)=O)cccc(C)c1F C1(CNC(C(CC)CO)=O)CCCN(C(c2nn(C)cc2Cc2cnn[nH]2)=O)CC1 C1(C(=O)NCC(C)(C2CC2)NC(=O)Cn2cc(Cl)cn2)CC2CCC1CC2 c1(C2C(C(N3CCCCC3CCCO)=O)CCO2)cccc(Cl)c1 c1(C(C)(C)C)[nH]cnc1C(=O)NCC(C)(C)OCCNC(=O)CCc1ccccn1 c1(NC(C23C(CN(C(c4c(C(C)C)ccs4)=O)C2)C3)=O)cnc2c(c1)CC(=O)N2 Cc1sc(-c2ccco2)nc1C(=O)NCC(C)CN(C(=O)C(O)C1CCCC1)C c1(CC)ccc(C(C)C(N2CC(O)(CN(C(=O)CNS(C)(=O)=O)C)C2)=O)cc1 c1(NC(C)CCO)cc(N2CCC(C(N3CCCCCC3)=O)CC2)ncn1 N1(C(CC)=O)Cc2[nH][nH]c(=NC(=O)c3cc(C)c(C#N)c(C)c3)c2C1 C1(c2nnnn2C)(NCC2CCC(C)NC2)CCC(C(N)=O)CC1 c1(CCC)ccccc1CNCc1cccc(C(N)=O)c1.N12CCC(O)(C1)C2=O C1(CN2CC(CNC(=O)CC(F)(F)c3ccccc3)C2)Cc2cc(Cl)ccc2O1 C1(CCC)(OC)CN(C(N2CCC(CCF)C2)=O)CCC1O CCCCC(CC)CC(=O)NC1CC(CNC(C2CCCN(CC(F)F)C2)=O)C1 c1(C(=O)NCC2CCC(NC(C3CCN(CC)C3)=O)C2)cnc(C)c(N)c1 c1(C(N2CC=CC(NC(C3C(C)(C(F)(F)F)C3)=O)C2)=O)ccc(S(N)(=O)=O)nc1 C(CC(C)C(F)(F)F)NC(C(C1CN(C(c2ccc(C)o2)=O)C1)O)=O c1(C(=O)NCC(CC=C)NC(=O)C(O)CC2CC2)cccc2c1CC(C)(C)C2 C1(C)(CNC(c2cnc(CCC)s2)=O)CCCN(C(=O)CCc2csc(C)n2)C1 c1(N2CCC(CC3CCCC(=O)N3)C2)cc(NCC)nc(C(F)(F)F)n1.C(F)(F)F CCC(CC)CCCC(=O)N1CC(NC(=O)CC2CCSCC2)CC1C c1(C(N2CC(NC(C=CC=CC)=O)C(OC)C2)=O)ccc2c(c1)CN(C)C2 c1(C(=O)NCC2(C(C)NC(N)=O)CC2)ccnc(O)c1.C(C(=O)NC)CCO C1(NC(C2C3CN(C(C4(CC#C)CCCCC4)=O)C2C3)=O)CCOC(C)(CC)C1 C1(NC(C2(CC(C)C)CCC2)=O)CN(C(c2cscn2)=O)C2(CCCCC2)C1 CCCCCCC(C)C(=O)N1CCN(C(=O)Cc2cc(F)c(N)cc2F)CC1C N1(C(C2CCN(C(CC)=O)C2)=O)CCCC(C)(O)CC1 Cc1cc(CCC(=O)NCC#CCNC(=O)C=Cc2cnccn2)cc(C)c1 C1(NC(CN(CC(C)(C)C)C)=O)C=CCC(C(=O)NCc2ncc[nH]2)C1 c1(N(C2CCN(C(C(C3CC3)OCC)=O)C2)C)nc(Cl)nc2c1CCOC2.OCC CCCCCC(CC)C(=O)NC1CCC2(CC1)CN(C(=O)C(C)C(F)F)C2 C1(C(=O)NC2C(CCOC)C2)COC2(C1)CN(C(c1cnc3[nH]ncc3c1)=O)C2 C(=O)(C(F)CCC(C)C)N1CCCC(C)(CNC(C(CC=CCC)C)=O)C1 Cc1onc(C2CCCC2)c1C(N1CC(NC(=O)CCC2CCCCN2C)C1)=O CCCC(C)(CC)C(=O)N1CC(O)(C2CCCN2C(c2sccc2SC)=O)C1 C12(C(=O)NCCCN(C(CC3(C)CC3)=O)CCO)CCC(C(F)(F)F)(CC1)C2 c1(C(=O)NC(C2CC2C(=O)NCCC2CCOCC2)C)cc(C#N)cn1C C(=O)(CCCCCCNC(=O)CNC=O)NC(CC(C)C)C(=O)N1CCCCC1 N1(CC=C(C)C)CCCC(C(N2CCCC(C)C2)=O)C1 N1(C(Cn2ncn(C)c2=O)=O)CCC2(CCCN2C(C23CCC2C3)=O)C1 Cc1cccc(Br)c1C(N1CC(CNC(=O)CC2CCC2)C(O)C1)=O c1(SCCNC(N2CCC(CN=[N+]=[N-])C2)=O)ccccc1[N+](=O)[O-] CC1CN(C(c2ccc(F)c(CO)c2)=O)C(C)CN1C(c1cc2n(n1)CCC2)=O c1(C(N2CC(COC)(NC(=O)Cc3csnc3C)C2)=O)cnc(=N)[nH]c1 C(=O)(CC(F)(F)F)NCC(CNC(C1C(C(=O)OC)C1(C)C)=O)O Cc1cncc(C)c1C(=O)NC(C)CC(C)NC(=O)Cc1ccc(F)nc1 c1(NC(C(CC#C)NC(=O)Cc2cc(C)cs2)=O)ccccc1N=[N+]=[N-] Cn1cnc(C(N2CCC(N(CCO)C(C3CC3CF)=O)C2)=O)cc1=O c1(CC(=O)NC2(C)CCN(C(C(CC)OCC)=O)C2)cccc2nsnc12 C1(C(=O)OC)CC(C(F)C(=O)NC(C)C(=O)NC2CC(=C3CC3)C2)C1.C1CO1 C1(NC(C)(C)C)CCCC(O)C1O.N1S(=O)(=O)OCCC1 c1(OC)ccc(C)cc1CC(N1CCC(CNC(C2CCCO2)=O)C(C)C1)=O c1(CC)ccc(C(=O)NCCOC2CCN(C(C3CN(C)C(=O)N3)=O)C2)c(O)c1 c1(C(CNC(C2N(C(C(C)N(C)C)=O)CCC2)=O)(F)F)cccc(F)c1 CC1(CNC(C2(CO)CC2(F)F)=O)COCCN(C(=O)CCF)C1 CN1CC(CC(=O)NCCC2CC(NC(C3CCOC3)=O)C2)C1 c1(OC)ccc2c(C(=O)NC3CCC(NC(=O)CC4CCOC4)CC3)cnn2c1 c1(C(=O)NCCC2(C(=O)NCc3ncn(C)n3)CCCC2)cnn2c1OCC2 c1(C(=O)NC2C(CNC(c3n(CCC)ncc3)=O)CCC2)cc(F)n(C)n1 c1(OC)cc(C(=O)N(C2CN(C(c3cc(C#N)c[nH]3)=O)CC2F)C)cc(F)c1F c1(C(=O)NCC(CNC(C2(SC)CC2)=O)CO)cccnc1-c1ccncc1 O=Cc1csc(-c2nnc(N3CCSCC3C3CC3)n2CCOCC2CCCC2)c1 CC(CC(=O)NCCCN(C(C1CC2(CCOCC2)C1)=O)C1CC1)CC(C)(C)C C1(CNC(CSc2nc(C)[nH]n2)=O)CN(C(c2cccc(N)c2)=O)CC1(F)F Cc1nc2cc(C(=O)NC(C)(C)C(C)NC(c3cc4n(n3)CCO4)=O)[nH]c2s1 Cc1ccc(C=CC(N2CC(CNC(C3CC3(F)F)=O)C(F)(F)C2)=O)nc1 Cc1cccc(O)c1C(=O)NC1CN(C(C2(C)CCNC2=O)=O)CC1C N1(C(=O)NCC=C)Cc2nnc(O)n2CC1C(=O)OC C1(OC)CC(C(=O)NC2CC(NC(=O)CC34CCCC3C4)C2)CC1OC n1(CC)cc(Br)c(C(=O)NC2CCC(C)(CNC(c3coc(O)n3)=O)C2)n1 N1(C(C2(C(N)=O)CCC2)=O)CCCC12CCN(C(=O)CN1CCCC1=O)CC2 N1(C(C(C)CC2CCC2)=O)CC2(CC(CC(=O)N(CC(C)(C)CO)C)C2)C1 C1(F)(CNC(C2N(C(CCCN(C)C)=O)CC=C2)=O)CCOCC1 N1(C(C(CC)(CC)CC)=O)CC2CCCC(C1)N2C(=O)Cc1ccc(F)cc1 Cc1cccc2c1CN(C(C1CN(C(c3cncn3C)=O)CCC1O)=O)C2 C(CC)(C(=O)N(C)CC=CC(N1CC(C)(F)C1)=O)OCC C1(CNC(C(CC)CC2CCCC2)=O)CCN(C(=O)CCOC(C)=O)CC1(F)F C1(OC)CCCN(C(=O)CCC2CCCN2C(c2ccc(C)cc2)=O)CC1 C(CC(C)C(=O)N(CC(C)NC(=O)C(C(C)C)NS(=O)(=O)C1CC1)C)OC Nc1nc2c(cc1C(N1CCC(NC(=O)C(F)=C3CCCC3)C1)=O)CCC2 c1(CCC(=O)NCc2cc(C)c(Br)s2)nnc(S)nc1O CC(C)CC(O)C(=O)N1CCC(F)(C(=O)NC2CCOCC2F)CC1 CCC(C)CCCC(O)CC(=O)OC.c12occc1CNC2=O N1(C(CC(C)F)=O)CCOC2(CCC(NC(=O)C=C3CCN(C)C3)CC2)C1 CC(F)(F)C(F)C(=O)NCCn1cc(C(=O)NCC2C3CCCCC23)nn1 C1(C(C(=O)NCCSC)CC(C)C)CCN(CCNC(C)=O)CC1 CC(CNC(c1ccc(O)cn1)=O)CC(=O)NCC1CCC(=O)O1 N1(C(C=CC)=O)CCCC(O)(CNC(=O)CN(C2CCSC2)C)CC1 C1(C(=O)NCCn2cc(CNC(CC(CC)SC)=O)nn2)COCCC1(F)F C1(CNC(c2nnc(O)s2)=O)CCN(C(C2(CF)COC2)=O)C1 c1(COCCNC(C2C(CNC(C3CCC3)=O)CC2)=O)ccnnc1 c1(C(N(C2COCCC2NC(=O)COC(C)(C)C)C)=O)cnn(CCO)c1N C1(CC)CN(C(=O)C2=CCCCC2)CCN1C(C1CCC(OC)CC1)=O C1(C(N2CCC(OCCNC(C(C)CC3CC3)=O)CC2)=O)CC2(COC(=O)N2)C1 C1(C)(CNC(c2occ(C(=O)NC3CC(C)SC3)n2)=O)CCC(=O)CC1 CCCCC(CNC(=O)CC1CC(O)CN1C(c1ccncc1NC)=O)CCC N1(C(CC(C=C)C)=O)CC2(CCN(C(=O)CNC(c3ccc(C)s3)=O)CC2)C1 N1(C(C(Cc2ccoc2)NC(=O)CCc2cn[nH]c2)=O)CCOC2(CCCC2)C1 S(=O)(=O)(c1ccc(Br)c(NC(=O)CS(=O)(=O)CCO)c1)NCC c1(NC(C2C3CN(Cc4cc(C)c(Br)cc4)C2C3)=O)ccc2scnc2c1Br c1(C(N2C(C(C)NC(c3cncnc3)=O)CCC2)=O)ncnc2c1CCC2 Cc1cccc(Br)c1CNC1CCC(NC(C(F)(F)F)c2ccccc2)C1 c1(OC)cnc(C(N2CCC(CC(=O)NC(C(C)O)C(C)C)CC2)=O)cn1 CC1C2CC(C2NC(C2(O)CCOCC2)=O)N1C(=O)C(C)NC(N)=O C1(NC(CC(C)(C)SC)=O)CCC2CC1CN2C(c1cscc1C#N)=O C1(CNC(C(CC=C)OC)=O)(CO)CCN(C(=O)C(C2CCCCCC2)O)CC1 c1(SCC(=O)NCC(C)N(C(C(CC)C)=O)C)ccc(C#N)cc1C C1(CNC(=O)Cc2nc[nH]n2)CCN(C(C2CCCC2)=O)CC1(F)F C(CCCCC(=O)Nc1cn(CCCN(C)C)nn1)N(CC(C)CCCO)C N1(CC)C2CCC1COC2.N1(C(CCN(C)C(=O)C2CC2)=O)CC2C(C(=O)N)C2C1 C(=O)(C1=CS(=O)CCC1)NC1C(NC(=O)CCN2CCCC2)CCCC1 c1(C(=O)NCC(C2CC2)NC(c2cn(C3CC3)nn2)=O)cc(C2CC2)cc(F)c1 C(=O)(C(F)(F)C(C)O)NCC(C(=O)NC(CCC=C)CO)CC1CC1 C1(C)(C(N(C)CC2(O)CCN(C(=O)CCCC3CC3)C2)=O)CCC(C)(C)CC1 c1(CCNC(=O)NCC(C)N(C)C(=O)OC(C)(C)C)nn(C)c(=O)o1 N1(C(CCSC)=O)CC(C(=O)NCCn2nc(C)nc2C)C2(CCC2)C1 N1(C(c2cc(C3CCOCC3)[nH]n2)=O)CC(NC(C2(CO)CCC2)=O)CC(F)C1 N1(C(C(CC2CN(C(c3cc(C)sc3C)=O)C2)F)=O)c2ccccc2CC1C c1(NC(C2(C)CN(Cc3c(Br)ccnc3Br)C2)=O)cc2ccc(Cl)nc2[nH]1 c1(OCc2nn(C)c(C3CC3)n2)ccc(N2CCCS2(=O)=O)c(Cl)c1 CCS(=O)(=O)CCCCCNC(c1nnnn1C(C)(C)CC)c1csnn1 c1(NC)cc(C(=O)NC2CCC(F)(CNC(C3CC4C=CC3C4)=O)C2)cc(Cl)n1 C1(C(=O)NCC2CCC(NC(c3c(CC)non3)=O)CC2)CC2CCCC2C1 C1(C(=O)OCC)CCC(C(=O)OC)C1.C1(CO)C(=O)NCC1=O c12ncccc1N2CC#CCO.c1(S)ccccc1.CO N1(C(c2cc(N)c(Cl)c(O)n2)=O)CCC2(NC(c3ccc(Cl)nn3)=O)CCCC12 C1(NC(Cn2ncc(C(=O)OC)c2)=O)CCN(C(=O)C=Cc2nc(C)co2)CC1C N1(C(C(C)N2CCCC2)=O)CCC(C)(NC(=O)C=Cc2cocn2)CC1 C(=O)(C(O)C(C)C)NC(C)C.C=CCCCNC(=O)CN(C)C(C)=O CC1CN(C(c2ccc(F)nc2)=O)CCN1C(c1ccc(C2CCCO2)[nH]1)=O Cc1cccc(CC(=O)NC2CCOC(CNC(C3CCCC3F)=O)C2)c1Cl C1(=O)C(C(C)C)CN1.c1(C(N(C2(C(=O)OCC)CC2)C)=O)cncc(NC)c1 C(=O)(CC1=CCN(C(c2cnnn2C)=O)CC1)NC(C=C)C c1(-c2cc(C(N3CC(NC(CCc4cn(C)nc4)=O)C3)=O)n[nH]2)ccc(Cl)cc1 C1(CNC(C2C(=C)C2)=O)CCC(C(=O)NCC(F)CO)O1 c1(OC)cccc([N+](=O)[O-])c1C(N1CC2CN(C(=O)C(C)(C)O)CC2C1)=O N1(C(CCSCCCC)=O)CCOC(CN(C(=O)CC2CC(CC)=NO2)C)C1 C1(NC(C(=O)NCC)=O)CN(C(c2cnc(C(F)(F)F)cc2O)=O)CCC1C.SCC C1(C)(CC)CCC(C(N2CC(=C(F)CNC(=O)CC3CCOC3)C2)=O)O1 N1(C(C(COC)(C)OC)=O)CCC2C(C1)CN2C(=O)Cc1cn2ccsc2n1 c1(C(=O)NC(CNC(C(COC)O)=O)C(C)C)cc(Br)cnc1S O=C1C(NC(=O)NCC(O)C(F)(F)c2ccccc2)CCN1C1CCCCC1 CN1CC2CCN(C(=O)CC3CCN3C(C3(CO)CC3)=O)CC2C1 CC1CN(C(C2CCCN2C(=O)CNC=O)=O)C(C)CCO1 N1(C(c2ccc(CCC)s2)=O)CCN(C(c2n[nH]cc2C)=O)C2CCCC12 C1(CNC(CCCSC)=O)CCCCN1C(C1CC1c1cccs1)=O N1(CC#C)CCN(C(=O)C(Cn2cccn2)NC(=O)CCC2CCCO2)CC1=O c1(C(N(CCCN(C(C(C)NC(=O)NC)=O)C)C)=O)ccc2c(c1)C(C)CO2 CCCC(C(=O)NCC(O)CCNC(=O)Cc1cn(C)nc1C)C(C)C CCCC(C(=O)NCC(C)(C1CC1)NC(=O)CCc1nccn1C)OC N1(C(C(C)OCC)=O)CC2(CNC(=O)CC(C)CC)CC1CO2 N1(C(C(Cc2ccoc2)NC(=O)CC2CC3CCC2O3)=O)CCc2nc[nH]c2C1 c1(C(=O)NC2C3CN(C(CC)=O)CC32)ccc2sc(C)nc2c1 CCCCCCC(CC)NC(C1CCCC1NC(c1cc2cc[nH]c2cn1)=O)=O N1(C(C(CC=C)C)=O)CCN(C(c2cccn2Cc2cccs2)=O)C(CCO)C1 c1(SC)cc(C(=O)N(C2CCC(NC(=O)CCCNC=O)CC2)C)c(C)o1 c1(N(C(c2cnn(C)c2Br)C(=O)OC)C)cc(F)ccc1NCCCN(C)C c1(CNC(C2CCN(C(C3(O)CCC3)=O)CC2)=O)ccc(F)c(F)c1Br O=C(C#CC1CCCO1)N.C12CN(C(=O)CC(F)(F)F)CC1n1cc(nn1)C2 C(=O)(C1=CCCC1C)NCC(c1ccccc1OC)NC(COCCSC)=O C1(NC(Cc2ccc(C)nc2)=O)CCCCN(c2ncc(Br)c(O)n2)C1 c1(CNC(CC2CCC(CC)O2)=O)ccc(CNC(=O)C(C)(O)C(C)C)c(F)c1 c1(CC)cc(C(N2CCC(NC(c3c(C)cccc3Cl)=O)C2C)=O)cn(C)c1=O C1(CC)CN(C(c2ncc(Cl)cc2Br)=O)CCN1C(c1[nH]nnc1C)=O CC1CCC2(CO1)CN(C(=O)CNC(c1cc(O)ncc1F)=O)C2 c1(C(C)NC(=O)NCc2nc(Cc3nc(C)n(C)n3)no2)ccnc(O)c1F c1(C(N2CCC(NC(c3cn(CCC)nc3)=O)(COC)C2)=O)nccc(N)c1Cl O=C1CC2C(C(=O)NC3(CCC(=O)NC4CC(CCF)C4)CCC3)C2C1 CC1(NC(C2CCCN(C(c3ccccc3CN(C)C)=O)C2)=O)CCCCC1 C1(C(=O)NC2CC(NC(C(C)CC3CCCO3)=O)C2)COCCOC1 CC(C)(C)C(CNC(C1(NC(c2n[nH]cc2Cl)=O)CCOCC1)=O)CO C1(=O)CC(C)(C)CNC(=O)C2CCCN12.c1(CN(C2CCC2)C)ccco1 c1(CC)cnoc1C(=O)NCC(C)(Cn1cccn1)NC(=O)CCOCC(C)C C(=O)(C1CCc2c[nH]nc21)N1C(CNC(C2CC(F)(F)CS2)=O)CC(O)C1 C1(C(=O)NCCc2cn(C(C)(C)C)nn2)C2Cc3c(Br)cccc3C12 C1(NC(C(=O)NCC)=O)CC2CC1CN(C(c1[nH]ccc1COC)=O)C2 Cn1c(O)ncc(C(=O)NCC2CCC(NC(C3(C)CCCS3)=O)C2)c1=O C(c1ccc([N+](=O)[O-])s1)=CC(N1CC=C(CNC(C2ON=C(C(C)C)C2)=O)CC1)=O C1(NC(CCC2C(C)=NOC2=O)=O)CC2CCC(C1)N2C(c1cscn1)=O N1(c2nnn(C)n2)CCC(O)(CCNC(=O)C(Cc2ccccc2)C2CC2)CC1 CC1CN(C(=O)CCc2cnn[nH]2)CC1CCNC(c1c(Cl)cnn1C)=O C#CC1CCCC(CNC(=O)C(C)(C)C2CCCN2C(=O)CC2CC3CC3C2)C1 C1(OC)CC(CNC(c2cnn(C(C)C)c2)=O)N(C(=O)CC2CCCCO2)C1 CC1C(C(=O)NC2(CF)CN(C(c3ncn4ccccc34)=O)C2)=NOC1C N1(CCCNC(CCC(=O)NC)=O)CC(CO)CCC1C c1(C(N2CC(O)(C(C)NC(=O)CC3CCCCC3F)C2)=O)cn2c(n1)COCC2 c1(NC(c2cnc(-c3cc(O)c(F)c(F)c3)cn2)=O)cccc(Br)c1[N+](=O)[O-] Cc1nc2c(C(=O)NCCCN(C(C3(F)CCN(C)CC3)=O)C3CC3)ccnc2[nH]1 N1(C(C(C)=NOCC#N)=O)CC2CCC(CNC(C3(C)CC3(C)C)=O)C2C1 CC(=O)CCCC(=O)N1CCC(C(C)NC(C2CN(C3CCCCC3)C2)=O)CC1 N1(C(CC(=O)OCC)=O)CCCC1(C)C(=O)Nc1cccc(CC=C(C)C)c1 c1(C(=O)NC2CCN(C(C3CC(O)C3)=O)C2)cc(F)c(Cl)c(Cl)c1 n1(CCC(=O)NC2CC(CCNC(C(C3CCCOC3)OC)=O)C2)cnc(=N)[nH]1 c1(NCc2nnc(-c3cccs3)o2)cccc(CNC(=O)OC(C)C)n1 N1(C(C2CC(OC)C2(C)C)=O)CCC2CC(C(=O)NCC3CCN(C)CC3)C2C1 S(=O)(=O)(c1cc(C)cnc1N1CC2CCC(C)(C)CC2(C)C1)NCC(C)SC C(N=c1[nH]c2ncc(Cl)cc2o1)C1CN(C(C(C(C)C)CCNC(C)=O)=O)CC1C C(=O)(C(CC(C)C)C(N)=O)N1CC2CCN(C(c3c(C)csc3)=O)CC21 C12(SC(C)(C)C)CCCC1(F)CN(C(=O)CCC1CC1)C2.C12CCC1NC2=O C1(CNC(c2cc(CC)c(C)s2)=O)CN(C(C2CCC(N=[N+]=[N-])C2)=O)CCC1C Cc1cocc1C(=O)NCCN(C(C1CC1F)=O)Cc1cccnc1 c1(C(C(=O)NCCC)N(CC(C)COCCOC)C)ccnn1CCF N1(C(=O)OC(C)(C)C)CC(O)(C2(NC(=O)CC3CCCCO3)CC2)C1 N1(C(Cn2c(C)c(Cl)cn2)=O)CCCN(C(c2cnoc2)=O)CC1 C(=O)(CC1=CCCCC1)NC1(C(N2CC(C(=O)OC)N(C)CC2)=O)CC(O)C1 Cc1ccc(CNC(=NCCc2nccnc2C)NCCF)c(Br)c1 C1(CC)(NC(=O)CCSc2cccc(Cl)c2)CCCN(C(=O)COCC(C)C)C1 c1(CC(=O)NCC(CNC(=O)CCn2cc(Cl)cn2)F)cccc2[nH]ccc12 C1(CN(C(=O)CC2CC(F)(F)C2)C)C2CN(C(C3CC4C=CC3O4)=O)CC12 c1(OC)ccc(C(N2CCN(C(=O)CNC(c3csc(C)n3)=O)CC2)=O)cc1 C1(NC(C(C(C)O)NC(=O)CCc2ccc[nH]2)=O)CC12CCOCC2 N1(C(C2CC2F)=O)CCC2CCC(C1)N2C(c1cncnc1C1CC1)=O c1(C(C(CC)OC(c2ccsc2Cl)=O)C)ccc(Br)cc1 C1(C(N2CCN(CCC#C)CC2)=O)CCN(C(=O)CSc2nc[nH]n2)C12CC2 C1(C(C)NC(=O)CNC(=O)NCC2CC2)CCN(C(c2cscn2)=O)CC1 c1(C(=O)NCC2N(C(c3c[nH]c(=N)o3)=O)CC2)cc2c(cc1Cl)NC(=O)CO2 N1(C(CSCC(C)C)=O)CC2CC(C1)C2NC(=O)CCc1ccc(F)cc1 N1(C(=O)NC(C=C)C2CCC2)CC2OCCCC2(CO)C1 C1(C(=O)OCC)(OC)CCN(CC(N2CCOC(C3CCC3)C2)=O)CC1 c1(C(=O)NCC(C)CNC(c2cccc(C3CCOC3)c2)=O)ncnc(O)c1F c1(C(=O)NCC2(O)CN(C(C(CC)(F)F)=O)C2)cccc([N+](=O)[O-])c1NC(C)C C1(NC(c2ccnc(C)c2N)=O)CC2CC(C1)N(C(c1cnc(Cl)[nH]1)=O)C2 c1(CC(=O)NCC(C2CC2)NC(CNC(CCC)=O)=O)c(F)cccc1F C(CC(C(=O)N(C(C)CC(N)=O)C)NC(=O)Cc1csc(C)c1)OC N1(C(CN2CC(C)(OC)C2)=O)CCC(C)(C)C(C(=O)N2CC(C)(O)CO2)C1 c1(C(N2CC(CC(=O)NCC3(CC(N)=O)CC3)(OC)C2)=O)cnc(O)c(F)c1 c1(CC)nc(C(=O)NC(C)(CNC(C2C3CCC2CC3)=O)CC)c(Br)s1 Cc1ccc(C)c(C(=O)NC2CCN(C(c3n[nH]c(C)c3C)=O)C2C)c1C c1(CC(=O)N(CCNC(C(F)=C(C)C)=O)C2CC2)cn2ccsc2n1 CCCCCCC(O)CCC(=O)N(C)CCOCCNC(c1ncccc1C)=O C1(CC=C)(C(=O)NCc2cscc2OC)CCN(C(c2nocc2C)=O)C1 CC1(C)CN(C(=O)CC2CC2(Cl)Cl)CC1NC(c1c[nH]nc1-c1ccccn1)=O C(=O)(C(CCOC(C)=O)N1CC(O)CC1c1ccccc1)NCC(=C)C C(CC)(CCCC(=O)NCC1(C)NC(=O)NC1=O)NC(c1ccn(CCC)n1)=O CC(C)(C(=O)NCC1CCN1C(=O)CSC(F)(F)F)n1cccn1 C1(NC(C=C(CC)CC)=O)CCCN(C(=O)Cc2ccc(C#N)cc2)C1C CC1CCCN(C(=O)C(=O)NCCOCCNC(=O)Cn2cccn2)C1 c1(NCC2CC(=C)CN2c2cc(-n3cncn3)ncn2)cccc([N+](=O)[O-])c1F C(CC)(C(=O)NCC=CC(=O)N(C1CC(C(=O)NC)C1)C)OCC C(=O)(C1CCOc2ccccc21)NCC1(F)CN(C(CC2CC(OCC)C2)=O)C1 C1(NC(C2(CC)CCOCC2)=O)CN(C(C2CCCC(=O)N2C)=O)CC1N=[N+]=[N-] c1(C(N2CCCC(NC(C(C)NC(C)=O)=O)C2C)=O)cnn2cccnc12 Cc1ccc(SCC(N)=O)cc1.C12C3CN(CC13)C(=O)CSC(C)CC(=O)NCC2 c1(C(N(CCNC(CC2(C(C)=O)CCCC2)=O)C2CC2)=O)cccc(C)c1 Cc1c(Cl)ccc(C(N2CCC(NC(=O)C(F)(F)CO)C(CO)CC2)=O)c1O c1(C(C)(C)NCCCC)ccccc1OC(CCN(CC=C)CC=C)=O C(c1nc(C)co1)=CC(=O)NCCCCN(C(CCc1cc(C)on1)=O)C C1(CNC(C2C(C)OCC2)=O)CN(C(C23CC4CC2C3C4O)=O)CC12CC2 c1(OC)cccc2[nH]cc(C(=O)NCCC(C)NC(=O)CC(F)F)c12 c1(-c2cn(CCN(C(C3(OC)CCCOC3)=O)CCO)nn2)ccc(C#N)c(F)c1 C(CCC(=O)OC1CCCCC1C)(c1nnnn1C(C)(C)C)OCC=C C(=O)(C(CC)(CO)OC)NC(CCC(=O)NC(C(=O)NC)CC1CC1)C C(CC(C)C(=O)NCC(C)N(C(=O)Cn1nnnc1C1CC1)C)OC CC(C)C(C)CC(=O)N1CC(NC(=O)CC(=O)N(C)C)CCC1C c1(C(N(CCCNC(C(CC)c2cccnc2)=O)CCO)=O)snc(C)c1N N1(C(C(C2CC(=O)N(C)C2)C)=O)CCOC(C)C1CNC(=O)COc1ccsn1 N1(C(C(C)CCO)=O)CCC2(CC1)OCCCC2NC(=O)CSC(F)F C(=O)(C(C)(C)C(=O)OC(C)(C)C)N(C)CC1(CNC(COCCCC)=O)CC1 C(CN=C(NC(C1CC1)C1CC1)N1CCC=C(c2ccncc2)C1)OCCOC C=CCCCC(C(=O)N1CC=CC1CN(C)C)NC(c1cc(O)n(CC)n1)=O C(=O)(C#CC(C)(C)CNC(=O)CC1CC2C=CC1C2)Nc1cc(C)c(F)nc1 c1(C(N2CCCC(N(C(=O)CN3CC4CC4C3)C(C)C3CC3)C2)=O)ccc(C)c(F)c1 N1(N(C2CCCC2)CCN(CC)CC)CC(=O)NC(c2ccccc2)C1 C(=O)(CC(O)C(C)C)NC1CCC(C)(C(N2CCN(CCC#C)CC2)=O)C1 C1(NC(C(COC)CNC(C)(C)C)=O)CCCCN(C(=O)COCC(=O)OC)C1 C1(=O)C2c3ccccc3CN2N1.c1(C(=O)OC)[nH]c(C)c(C(C)=O)c1C N1(C(CN2CC(C)C2)=O)CCCC(C)(NC(=O)C=CC(=O)N(C)C)C1 c1(C(N(CCCCNC(C2C3CCC(=O)C23)=O)C)=O)cc(OC(F)F)ccc1F C1(NC(CCc2cc(C)on2)=O)CCN(C)C12CCCN(C(=O)CSC(C)C)C2 C1(CC)C(CC(=O)NOCCC(F)(F)F)CCCN1C(C1CCN1C)=O c1(C(N2CCC(C)(CNC(C(C)(C)SC)=O)C2)=O)c(F)cncc1Cl C(=O)(C(O)CC(C)(C)C)NC1(CCC)CCCN(C(=O)CSCC(N)=O)C1 C1(CNC(Cc2c(C)occ2)=O)COCCN1C(=O)CC1CCC(=O)NC1 C1(C(=O)NC2COCCC2C(N2CCC3CC23)=O)(CC)CCCCO1 Cc1cc(C(N2CCN(C)C(CNC(C3CC3(C)C)=O)C2)=O)nc(O)n1 C1(NC(C(C)OC2CCCC2)=O)CCCN(C(c2ccncc2O)=O)CC1 C1(NC(Cc2c(C)nsc2)=O)CCCCN(C(=O)C(C)NC(C2CCC2)=O)C1 C1(CC=C)(NC(=O)Cc2cccnc2)CCCN(C(=O)C(C)CCOCC)C1 C(C(=O)NC(C(=O)N1CC(N2CC(F)C2)C1)C1CC1)(C1CCC1)OCC c1(CN2CCCCC(NC(c3ccnc(F)c3F)=O)C2)n[nH]c2ccc(Br)cc12 C1(OC)(CN(C)C(C2CC2CNC(C2(O)CCOC2(C)C)=O)=O)CCC(C)CC1 N1(C(C(C2CCCO2)NC(C(=O)N(C)C)=O)=O)CCCC(N(C)C)C1 C1(C(C)NC(CCCN(C(=O)OC)C)=O)CCCCN1C(=O)C#CC1CC1 C#Cc1ccc(C(N2CC(CC(=O)NCc3[nH]cnc3C)CC2C)=O)o1 c1(NC(C(=O)N(CCNC)Cc2ccccc2[N+](=O)[O-])=O)c(C)ccc2c[nH]nc12 N1(C(=O)NCCCC)CCN(C(=O)C=Cc2ccccc2Br)C(COC)C1 N1(C(CCCC=C)=O)CC(NC(=O)Cc2c(C)cc(C)nc2O)CCC(O)C1 c1(C(N2CC(CC)C(NC(=O)CCC#N)CC2)=O)cc(S(=O)(=O)N(C)C)c(C)o1 CC(C)C(C(=O)NCCC(C)CCNC(=O)CC1CC1)n1cc(Br)cn1 c1(OC)ccc(Cl)c(C(=O)NC2CN(C(c3ccc(N)c(C)c3)=O)CC2C)c1 C(CNC(C1(SCC)CC1)=O)(C(C)C(C)C)NC(CCC#CC)=O Cc1ccnnc1C(=O)NC1CCC(NC(C2(C)CCC(C)C2)=O)CC1 Cc1cccc([N+](=O)[O-])c1S(=O)(=O)N1CCN(CC(c2ccc(Cl)cc2)O)CC1 C1(C(=O)NC(CCSC)C(=O)NC2CN(C)NC2=O)CCC2CC1CO2 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1(C(=O)NCC2(CC=C)CCC2)CCOCC1 c1(CC)cc(C(=O)NC2CC(C)(NC(=O)C(F)F)C2)ccc1F C(C(C)(C)CNC(c1ccn(CC(F)(F)F)n1)=O)N(C(=O)CC(=O)NC1CC1)C C=CC(CCC)CC(=O)N(CCC(=O)N(C1CCC(CO)CC1)C)CCCO c1(SC)cccc(CNC2CCCC2CSc2cccnc2)c1 C1(C(=O)NC(C(=O)OCC)CO)CC12CCN(Cc1ccc(Cl)c(Br)c1)CC2 C=CCC(C)C(=O)NCC1CCCCC1NC(c1cc(C(F)F)on1)=O C1(NC(CC2(C)CCOCC2)=O)CN(C(=O)COc2cccc(Cl)c2)C(C)(C)C1 c1(SC)cnn(C)c1C(=O)NCC1COCCN1C(=O)CC1CCC1 C1(C)(C(=O)NCC(C)SC)CCN(C(=O)CC2(C#N)CC2)C1 C1(NC(CSC)=O)CCOCC1NC(=O)CC1CCN(C)C1 NS(=O)(=O)CCCC(=O)N1CC(C(N)=O)(CNC(=O)CC2CCOC(CF)C2)C1 c1(C(=O)NCCC2CCN(C(c3ccn(C)c3)=O)CC2)cc(F)cc2nn[nH]c12 CC1CC2(CC(C(=O)N(C3(C(N4CC5CC5(CO)C4)=O)CC3)C)C2)C1 C1(OC)CC(F)(NC(=O)CC2CC2C(=O)NCCNS(C)(=O)=O)C1 N1(C(C=C(C)C)=O)CCN(C(=O)CN(CCCCCC)C(C)C)C2CCC12 N1(C(c2cnsc2)=O)CCC2CCCN(C(c3cc(Cl)c(F)c(Cl)c3)=O)C2C1 c1(C(N2C(CNC(C(C)CC3CCC3)=O)CC2)=O)cc(Cl)cn1C c1(OCC(N2CC(CC=C)(NC(=O)CC3CC(=O)NC3=O)C2)=O)cc(C)ccc1Cl CC1(NC(=O)Cn2cccn2)CN(C(C2CCCS2)=O)C1 c1(N(C(N(C2CCCC2)C)=O)CC2CC2)nc2ccc(C#N)cc2s1 Cc1nc(C(N2CCC(CNC(c3ncoc3-c3cnn(C)c3)=O)C2)=O)n(C)n1 C(=O)(C1Cc2ccc(F)cc21)NC1CN(C(c2[nH]cc(C#N)c2)=O)CC12CCC2 Cn1cc2cccc(CNC(C3CCCN(S(=O)(=O)CC4CCC4)CC3)=O)c2n1 N#Cc1ccc(NC(=O)CC2CCCN(Cc3cc(F)c(Br)cc3F)C2)c(O)c1 C(=O)(CCCCCF)NCC1C(CNC(c2cnc(-c3ccc(C)cc3)s2)=O)C1 C1(C2CCCN(C(C3CC3C3CCC3)=O)C2)(NC(Cc2nnc(C)o2)=O)CC1 C(Cc1ccc(CC)o1)(CC(=O)N(CCC)OC)NC(CCC=C=C)=O C(C(C(=O)OC)c1occ(-c2c[nH]nn2)n1)OCC.c1(CC)nccn1CCF c1(NC(CNC(c2coc(Cl)c2)=O)C2CC2)ncnc2sc3ccccc3c12 C1(COCCOCC)CC(CNC(C2CCCC2)=O)CO1.C1CC(=O)N1 CC1CC(NC(=O)CNC(C2(CF)CC2)=O)CN1C(=O)NCC(F)(F)F N1(CC(C)C)CCCC(C(=O)NCC2(CNC(c3nnn(C)n3)=O)CCCC2)C1 C(C1CN(C(C2CC2C(C)C)=O)CC1C(=O)NC(CO)CCO)=CC c1(OCCC(=O)N(C(CNC(=O)C(F)F)C2CC2)C)ccccc1.C(=O)N N1(CCC)CCC(NC(=O)C(=O)NC2CCCC2c2ccccc2)CC1 N1(C(C2(OC)CN(C(C(CC)OC)=O)C2)=O)CCN(C)C(C(C)C)C1 c1(C(=O)NCC2C(CNC(CCC(C)OCC)=O)C2)ccc2c(c1)CCCO2 c1(C(N2CC(C(=O)OC(C)(C)C)C(O)CC2)=O)cnc2c(F)c(F)ccc2c1 c1(C(=O)NC(CC)CN(C(=O)C(C)OC2CC2)CC)ccc(C)cc1SC C1(C)(C(=O)NC(C)C=CC(=O)Nc2cnn(C)c2Cl)C=CCCC1 C12(NC(CCCOCCOC)=O)CCC(CC1NC(c1cncc(CO)c1)=O)C2 N1(C(=O)CCc2cnn[nH]2)CCCC(F)(C(=O)NC2CC3CC(O)C2C3)C1 C1(C(N2CC(F)(CNC(C(C)c3ccsn3)=O)C2)=O)CCn2nncc2C1 C1(NC(CN(CCC)C)=O)CCN(C2CCN(C(=O)C(=O)NC(C)C)CC2)CC1 c1(N(CCNC(=O)CCCOCC(C)C)CC)cc(C)c([N+](=O)[O-])cc1F c1(C(N2C3C(CNC(=O)COCC4(F)CC4)C(C3)C2)=O)ccc2ccccc2c1 C1(C(CO)NC(CCN(c2ccccn2)C)=O)CCN(C(c2cnc[nH]2)=O)CC1 c1(Cc2ccc(CNC34C(CN(C(=O)CSC(F)F)C3)C4)nc2)cccc(F)c1 c1(C(N2CCOCC(NC(C#CC(C)C)=O)C2)=O)cc(Cl)cc(Cl)c1O c1(OC)nccc(Cl)c1C(=O)NCC1CCCN1Cc1ccc(I)o1 N1(CC)CCN(C(C2CN(C(c3cc(C)ncc3C)=O)C(C)(C)C2)=O)C(C)C1 c1(CNC(NC(C=C)C)=NCCC2CCN(C)CC2)c(F)cc(COC)cc1F N1(C(c2nccc(OC)c2F)=O)CCOC2(C1)CN(C(C1CCC(=O)N1C)=O)C2 C(=O)(CC(C)CC(F)(F)F)NC(CC)CN(C)C(c1cc(F)c[nH]1)=O c1(CC(=O)N(C(CNC(COCCCC#C)=O)C)C)coc2ccc(F)cc12 c1(C(=O)NCC(CC)N(C(=O)C(C)(C)NC(=O)OC)C)cc(C)c(C)cn1 CN1N=C(CC(=O)N2CC3CCC2CN3C(c2cnn(CC3CC3)c2)=O)CC1=O C1(NC(=O)C(C2(O)CCCCC2)F)CCCN(Cc2ccccc2)CC1 c1(C(=O)NCCC2(NC(C3C(C)CCCC3)=O)CC2)ccn2c(O)nnc2c1 O=C1CC(C(=O)NCC(F)(F)C2(O)CCC2)C2(CCC2)C1 c1(C(N(C2CCCC(NC(c3cccc(N)n3)=O)C2)C)=O)ccn2cnnc2c1 N1(C(C2(c3ccc(C#N)cc3)CC2)=O)CCC(NC(C2COC2)=O)C(F)(F)CC1 N1(C(C=NOC)=O)CCC(C2CCN(C(=O)Cn3cccn3)C2)C1 C1(C(N2CC3CC2CC3O)=O)(CC)CCN(C(=O)CN2C(C)CCC2C)CC1 CN1CC(NC(=O)CN(C(=O)C=CC2(C)COC2)CC2CC2)CC1=O c1(C(NOCc2cn(C(C)CNC(N)=O)nn2)=O)ccnn(C)c1=O N1(C(C=CC)=O)CCC(CO)C(NC(=O)CCN2CCCC2=O)C1 C1(CCC)(NC(c2ncc(F)cn2)=O)CCN(C(c2cnc(C(N)=O)s2)=O)CC1 c1(CNCc2ccc(C(C)(C)C)o2)cc(Cl)ccc1N1CCCCC1 c1(CC)c(NC(CNC(c2cc(C)nc(Cl)c2)=O)C(C)C(C)C)ncnc1Cl CC(C)C(C#N)C(=O)NCC1CCCC(CNC(=O)C(C(C)C)N(C)C)C1 c1(CNc2cccc(C(N3CCC(C(N(C)C)=O)C3)=O)c2)csc([N+](=O)[O-])c1 c1(C(N2CCC(N(C(CSCC=C)=O)C)C2)=O)c(C)cc(C)c(Br)c1C C(=O)(C(O)CC[S+](C)C)NCCN(C(C1N(C(C)=O)CSC1)=O)C1CC1 N1(C(CC2C(C)=NN(C)C2=O)=O)CC2CC(NC(c3cc(Cl)ccn3)=O)CC2C1 S(=O)(=O)(c1ccc(Br)cc1N1CCC2(CCCC2)C1)N1CCSC(C)C1C C1(F)(CNC(C2N(S(C)(=O)=O)CC2)=O)CCN(C(=O)C(F)CC2CC2)C1 c1(CC(N2CC(N(C(C=CC(=O)N(C)C)=O)C)C(F)C2)=O)cccc(O)c1F C1(C)(CNC(CCCC#CC)=O)COCCN(C(=O)CC2CCC(OC)CC2)C1 c1(CC(=O)N(CCC(=O)NC2CC2C(F)(F)F)CC#C)cccc(F)c1 CC1CCC(NC(=O)C(F)Cc2ccccc2)CN1C(c1ccc(O)c(Cl)n1)=O c1(C(=O)NC2CC(NC(C(c3n(C)ncc3)(C)C)=O)C2)cncc(P(C)(C)=O)c1 N1(C(C(C(C)C)SCC)=O)CC(NC(=O)CCC[N+](=O)[O-])CC(C)C1 c1(CCC)n[nH]cc1C(=O)NC1CC(CNC(=O)CSc2nnc(S)s2)C1 c1(OCC)cccc(CC(=O)NCCC(C(C)C)NC(=O)Cc2cn(C)cn2)n1 C1(C(=O)NCC(CO)OC)CCC(NC(=O)CC2(C)CCC2)C1 c1(-c2c(C=C)cccc2)ccc2[nH]c(C(=O)N(c3c(Cl)cc(Cl)cc3Br)CC)nc2c1 Cc1ncnc(C(N2CC(C)(C(=O)Nc3c[nH]ccc3=O)C2)=O)c1C N1(C(C(CCC)C)=O)CCC(F)(F)C(CNCc2cc(I)c[nH]2)C1 Cc1cc(CC(=O)NCCCCCNC(C23CCC2C3)=O)nc(NC(N)=O)n1 CC(C)C(CNC(c1cnn(C(F)F)c1)=O)N=c1nc(C2CC2)[nH]s1 c1(C(N2CCCC(N(C(C(C)NS(C)(=O)=O)=O)C)C2)=O)cc(Cl)ccc1F CC(C)CC(C)C(=O)NC1CCCCC1NC(=O)Cc1ccc(C#N)cc1 C1(C(N2C3CC(NC(Cc4ccc(C)cc4)=O)C2CC3)=O)CC2C=CC1C21CC1 n1(C2CCN(CCC#C)CC2)cnc2c1CCN(C(=O)OC(C)(C)C)C2 C(=O)(C1CCCc2ccccc21)NC1CCN(C(C(C)OCC#C)=O)C1C N1(CC(c2ccc(CC(=O)OC)cc2)N2CCCCC2)C(=O)NC(C2CC2)C1=O Cc1oc(C#N)cc1C(=O)NCC(C)(C)CCNC(c1ccc(F)c(Cl)c1)=O C(=O)(NNc1cc(F)cc(Br)c1)NC(C)CCC1CCCCC1 CC1(CS(C)(=O)=O)CCN(C(c2cccn2-c2cccnc2N)=O)CC1 c1(C(=O)OCC2(N(C)C(c3ccns3)=O)CC2)ccc(C(=O)OC)cc1F C12(NC(=O)CNC(C3CCC3)=O)CCC1CN(C(=O)Cc1ccc(F)cc1Cl)C2 C1(NC(Cc2c(C)ccs2)=O)CCCN(C(=O)CNC(=O)NC2CC2)C1 C=C(C)C(O)CC(=O)NCC1CCN1C(c1cc(Oc2ccccc2Cl)ccn1)=O c1(COCC(=O)NCC2N(C(COC)=O)CC3CC3C2)ccc(OC)c(Cl)c1 c1(OCC)ccc(C(=O)NC2CN(C(C3OCC3(C)C)=O)C2)cc1OC S(=O)(=O)(c1cccnc1N1CCS(=O)C(C)(C)CC1)N(C)C(C1CC1)C1CC1 C(CC(C)(C)COC)NC(CC1N(C(c2c(CCC)nco2)=O)CC1)=O C1(CNC(CC(C=C)C)=O)CCC2(CC1)CCN(C(=O)CCF)CC2 c1(C(N2C3CC(NC(CC(C)C)=O)C(C3)C2)=O)cc2n(n1)CCCC2 N1(C(CC(CCC)C)=O)C2CCC1C(C)C(NC(=O)C(C)(C)N1CCCC1)C2 C12(C(=O)NC3(C#C)CC3)CCC(CN=c3ccc(C(F)(F)F)n[nH]3)(CC1)CC2 c1(C2(C(=O)NCC(CCOC)NC(=O)OC(C)(C)C)CC2)ccc(F)cc1C C1(NC(=O)CC2C=CCCC2)C=CCN(C(C2CCC(F)CC2)=O)C1 C(=O)(C1=CCCOCC1)N1C(NC(C2CCC3(CC2)N=N3)=O)CC(COC)C1 C1(C(C2CCCN2C(=O)CCCc2ncco2)C=O)C2CCCCCC12 c1(C(=O)NC2CN(C(C3(SCC)CC3)=O)CC2C)ncc(F)cc1N CN1CCN(CC(=O)NC2(C3CN(C(c4cc(CCO)on4)=O)C3)CC2)CC1=O C1(CNC(CSc2n(C)cnn2)=O)CCCCCN1C(C1(CC2CC2)CCC1)=O c1(CC(=O)NCC2CC(NC(=O)C(c3ccccc3)O)C2)cccc(Cl)c1F C1(OC)CC(CNC(c2ncc(C(F)F)s2)=O)N(C(=O)Cc2cncn2C)C1 N1(C(C(=O)NCc2nnn(C)n2)CC2C=CCC2)CCC2CCC(C1)S2(=O)=O Cc1csc2ccc(CN=c3[nH]c(C(=O)CN=c4cc[nH]cc4)cs3)cc12 C1(CCC)CN(C(C2CC2CC(C)(C)C)=O)CCN1C(c1cscc1Cl)=O c1(CSCC(=O)NCC(O)CCNC(C2CC2(F)F)=O)nc2ccccc2s1 CC(C)(C)CC(Cc1nn[nH]n1)C(=O)N1CCSC2CC12 C(=O)(C1=CCCCC1)N(C1CCC(NC(c2cn3ccsc3n2)=O)CC1)C N1(C(C(C)OCc2cccc(Cl)c2)=O)CC(CNC(=O)C(C)(F)F)C(F)(F)C1 C1(C)(C(N2CCC(NC(c3c(C)scn3)=O)C2)=O)COC(=O)N1 c1(C(c2nnnn2CCCF)NC(C2(OC)CCCCC2)C)cc(C)nnc1O CC(CC(=O)NC1C2CCC1CN(C(C1CCN1C)=O)C2)C(C)(C)C C12(C(N(CCCCCCN(C)C(C3CCCO3)=O)C)=O)CC3CC(CC(C3)C1)C2 N1(C(C2C(C)(C)NC(=O)C2)=O)CCN(C(=O)Cc2csc(C3CC3)n2)CC(O)C1 N1(C(C(CC=C)OC)=O)CC(CNC(c2ncccc2SCC)=O)CC1(C)C c1(NC(C(C)OC(C(CC)SC)=O)=O)ccc(Br)cc1C(C)C c1(OC)c(C(N2CC(NC(C3COCCN3C)=O)CC2CO)=O)cc(F)cc1F CC(C(=O)N1CC(C(=O)NCCNC(=O)C2CC2)C1)C1(O)CCC1 c1(N)ccc(C)n2ccnc12.N1C(=NCC2CCC2)NC2CC12.Cc1ccon1 C1(CNC(=O)OC(C)(C)C)CCCC(Cc2cc(CO)on2)C1 N1(C(c2[nH]n(C)c(=O)n2)=O)CCC(NC(=O)Cc2ccc(F)cn2)C1(C)C C(=O)(C(C)CCC(C)(C)C)N(CCOCC#C)CC#C.C1(=O)C(CCC=C)N1 CCC(C#N)C(=O)N1CCC(C)(NC(=O)CCc2ccsc2Br)C1 CCCC(CC)CCC(=O)NC1CN(C(=O)CCCSC)CC1c1cncn1C C12(C(N3CC(=C(CNC(=O)CCC4CCOC4)F)C3)=O)CC(F)(C1)C2 c1(NCCn2c(N(C)CC3(C#C)CCCC3)nnn2)c(COC)cccc1C c1(C(N(CCOC)C)=O)n[nH]c2c1CCN(C(c1c(F)cc(F)cc1Br)=O)C2 C1(CNC(C2(C#N)C(C)C2)=O)CCCCC1CN c1(C(=O)NC2C(CNC(CC3CN(C)C3)=O)CCC2)cc(N)ccc1C(F)(F)F c1(C(=O)NCC2CCCC(CNC(CCCC=C)=O)C2)cc(F)c(F)c(N)c1Cl N1(C(Cc2c(CC)n[nH]c2CC)=O)CCCN(CCNC(=O)C(F)C2CC2)CC1 c1(C(=O)OC)cc2n(n1)CCC2.C12CCCN1C(=O)C1(CC1)CCCC2 C1(NC(C(CC)N(C)C)=O)CC2(C1)CC(NC(C1CCCN1C)=O)C2 n1(CC)cnc2nc(=NC(C)CCC(C)C)[nH]c(NCC3(CF)CCC3)c12 N1(C(C2N(N3C(C)CC4(CC4)C3)CCC2)=O)CCCNC(=O)CC1 C1(OC)(CNC(c2cnc(Br)s2)=O)CCN(C(=O)C(C)(C)F)C1 c1(C(=O)NC(C2(O)CN(C(C3CCCC(C)(C)C3)=O)C2)C)cnc2occc2c1 C1(CNC(CC(C=C)C)=O)CC(C)CN(C(c2ncccc2C)=O)C1 c1(C(N2CC(NC(C3(C4CCC4)CC3)=O)CC3(CC3)C2)=O)ccc2nccn2c1 c1(C(=O)NC2CCC(C)N(C(=O)C(C#N)C3CC3)C2)cc2ccccc2nn1 C1(Nc2cccc(OCC)c2)CCC12CCNCC2.N12CCCC(C1)NC2=O c1(C(=O)N)cccc(OCCCC2CCC(NC(C3(C=C)CCC3)=O)C2)c1.COC c1(SC(C)C)ccc(Cl)cc1C(N1CCC(CCNC(=O)Cc2cn[nH]c2)C1)=O Cc1cccc(-c2cncc(C3CCCN3C(=O)Cn3cnc(C#N)n3)c2)c1 N1(C(c2nc(NC(C3CCSCC3)=O)sc2)=O)CCc2ccc(Br)cc2C1 c1(C(N2CCC(c3cc(Br)ccc3F)(N)C2)=O)cc(CO)cc(OC(F)(F)F)c1 N1(C(c2ccc(OC)c(C)c2)C(=O)NC2CC2)CCC2(CC1)CC(OC)C2 c1(-n2cc(C(C)N(C(=O)C(C)N(C)C)C)nn2)ccc2nc(C(=O)O)oc2c1 N1(C(C(CCC)O)=O)CC(C2CN(C(=O)CCc3nccn3C)C2)C1 C(CC1CC1)(CCNC(=O)OC(C)(C)C)Oc1csnc1-c1cnco1 c1(C(=O)NCC(CC)NC(C2(O)CN3CCC2CC3)=O)ccc(F)c2occc12 CN1CC=C(CC(=O)N2CCC(CCNC(=O)Cc3nc(=N)[nH][nH]3)C2)CC1 c1(NC(CC)C2CC2)ccc(S(=O)(=O)NC(C2CCC2)C)c(Cl)c1 C(C)(C)(CC(=O)NCC1(C(N)=O)CCOCC1)NC(CCC1CC(OC)C1)=O C1(N(C)C(c2cnc[nH]2)=O)CCC(NC(c2ccc(-c3ccco3)[nH]2)=O)CC1 C(=O)(C1=CC(C)(C)C1)NCCCN(C)C(c1ccc(CN2CCCCC2)o1)=O C=CCC(C)(C)CC(=O)NCC(C)(C(C)SC)NC(c1ccc(F)c(SC)c1)=O CON(CCC(=O)Nc1ccncc1)C(=O)CN(C1CCC1(C)C)C C1(C(=O)NC(C(=O)N(C(COC)C)C)C(C)C)OCCC1CC C(=O)(C(C)(C)CC(=O)N1CCCN(C(=O)COc2cccc(Cl)c2)CC1)OCC Cc1cc(C)n(C(C)C(=O)NC(C)(CNC(=O)CCN2CCCC2)C(C)C)n1 C1(CN(C(=O)Cc2ccoc2)C)CCCN(C(C2(C#N)CC(=O)C2)=O)C1 C12(CNC(C3N(C(C(C)C)=O)CCC3)=O)CC1CN(C(C1(C3CC3)CC1)=O)C2 c1(C2OCCN(CC3(C)CC(OC)(OC)C3)C2)cc(F)cc(F)c1 N1(C(c2c(CC)ccc(F)c2)=O)CCC(C)N(C(=O)C(F)C(C)C)CC1 CCCC(C(O)C(=O)NCCC#CCO)NC(=O)C(C)NC(=O)CC C1(CNC(c2ncc(C(=O)OC)nc2)=O)CCCCN(C(=O)C=C(Cl)Cl)C1 C(CCCC(=O)N1CCCC1CCNC(c1c(C)cccc1F)=O)(OC)OC C12(CNC(C(CC)O)=O)CCCC(CN1C(c1ccc(=O)n(CC3CC3)c1)=O)C2 N1(C(=O)CC2(O)CCOC2)CCC2(C1)CN(C(c1sccc1C(F)F)=O)CCO2 n1(CC)ncc(C(=O)NC2CC(NC(=O)C(C)(C)C3CCCC3)C2)c1Cl C1(C(N2CC3C(NC(C4(CSC)CCC4)=O)C3C2)=O)CCn2nccc2C1 c1(C(=O)NCC(CC=C)NC(=O)CC2(O)CCCCCC2)ccc(C)c(F)c1F N1(C(C=CC(C)(C)SC)=O)CCOCC(C(=O)N(CCO)CC2CC2)C1 Cc1ncnc(C)c1CC(=O)N(C)CCNC(=O)CCCN1C(=O)CN(C)C1=O N1(C(c2cn(CC(C)(CC(=O)O)C(F)F)o2)=O)CCCC2(CCCO2)C1.CC(C)CCC(F)C=O N1(C(CCn2ccc(C)n2)=O)CCC(O)(C(C)C(C)C)C1.c1(C(=O)N)csc(S)n1 N1(C(CNC(C)=O)=O)CCC2(CCCOC2)C1.C1C(O)C(=O)N1 C1(NC(CC2C(OC)CC2)=O)(CNC(=O)CCc2cc(Cl)no2)CCCC1 c1(C(=O)NC(COC)CNC(=O)C(C)CSC)ccnc(OC(F)F)c1 c1(C(=O)NCC2CCCCN2C(c2cnc(C(F)F)s2)=O)cnc2scnc2c1 N1(C(C=CCCC)=O)CC(NC(c2ccco2)=O)CC12CCCC2 c1(CC)ccc(C(=O)NCc2cccc(CN(C)C)c2)nc1N c1(-n2ncc(C(=O)NC3CC3CNC(c3cc(O)no3)=O)c2)ccc(F)cc1 c1(C(=O)NCC(C)CNC(c2ccnc(NC(=O)OC)c2)=O)ccc(Cl)c(O)c1 c1(C(=O)NCC(CNC(=O)CCOC2CCOCC2)OC)ccn(C(C)(C)C)c1 N1(C(C(C)OC)=O)CCN(C(=O)CCc2cccc(F)c2Br)CC1C(F)F S(=O)(=O)(c1cccc2scnc12)NC(c1ccccc1)C1C(c2onc(C)n2)C1 C(=O)(C(C)(CC)C(=O)N1CCC(F)(F)C(CNC(=O)Cc2ccoc2)C1)OCC C12(NC(CCC#C)=O)CC1CN(C(c1ccccc1-n1cc(OC)nn1)=O)C2 c1(CN(c2ccc(-c3ccc(Cl)cc3)s2)CC(=O)NC(CC)(C)C)ccc(C)nc1 CC1CC(CC(=O)NCc2cccc(O)c2)CN1C(c1c[nH]nc1Cl)=O N1(C(c2ccc(NC(C)=O)s2)=O)CC2C(N(C(c3cc(C)c(C)[nH]3)=O)C(C)=O)C2C1 C(=O)(CCCS(C)(=O)=O)N1C(CNC(C2CN(C(C)=O)C2)=O)C(C)CCC1 N1(c2snc(C)n2)CC2CCC1CN2C(C1CCCCC1C1CC1)=O Cc1ccc(CCC(=O)N2CCC2C(=O)NC2CCCC(=O)N2)c(C)c1 C(=O)(CC(C)CNC(=O)CCC1(C)CN(C(=O)CN(C)C(C)C)C1)NC c1(C(N(CC(C)NC(=O)Cc2nc([N+](=O)[O-])n[nH]2)CC)=O)ccn2nccc2c1 C12(NC(c3cnc(SC)s3)=O)CN(C(C3(C)CCOCC3)=O)CC1CS(=O)(=O)C2 c1(C(=O)NCCCCCC(=O)NC)cc2cc(Br)cnc2s1 C=CC1CCCN1C(C1CCOC1CNC(=O)CC(C)C)=O C1(C2(O)CN(C(C3CCC(C)S3)=O)C2)(CNC(c2c(OC)c(F)ncc2)=O)CC1 c1(NC(CC)CC#N)ncnc(N2CCC(NS(C)(=O)=O)CC2)c1C N1(C(CSCCOC)=O)CCC(NC(c2ccncc2OC)=O)C(O)C1 C1(CNC(C2(CC)CCCC2)=O)CCN(C(=O)CC2CCC(=O)N2)CC1C CC1(C)CCc2[nH]c(C(N3CC4C(NC(C5CC(F)(F)C5)=O)C4C3)=O)cc2C1 c12nccnc1C(=O)NC1CN(C1)C2=O.c1(C(C)(C)C)ncc(C(F)F)s1 C1(CNC(c2c(C)n(CC(C)C)nc2)=O)CN(C(=O)C2=CCSC2)CC(C)(C)O1 n1(C(C)C)ncc(CN(C2CCC(N)C2)C)c1Cl C(C(O)C(F)(F)F)NC(C(C)N(C(C1(C=C)CCC1)=O)C1CC1)=O C1(C(N2CC(NC(c3c(CC)cccc3)=O)C(OC)C2)=O)COC2(CCC2)C1 Cc1cnnc(O)c1C(N1CC2CC(NC(=O)CSS(C)(=O)=O)C2C1)=O Cc1cc(F)c(CC(=O)NC2(CO)CCN(C(C3(C#N)CC3C)=O)CC2)cc1F C1(O)(CCNC(c2ccc(C(N)=O)o2)=O)CCN(C(c2ccno2)=O)C1 c1(NC(c2ncc(NC(c3c(C)c(F)ccc3)=O)nc2)=O)nc(Cl)c(C)c(Cl)n1 N1(C(Cc2nc(C)[nH]n2)=O)CC(NC(C23CC(CN2C2CC2)C3)=O)CC(C)C1 C(c1ccccc1Br)=CC(N1CC(CCCCNC(C2(CO)CCC2)=O)C1)=O c1(CC=CC(N2CC(N(C(=O)CNC(=O)C3CC3)C)C2)=O)cccn1C Cc1nc(C(=O)OCc2nnc(-c3cccc(Cl)c3F)o2)c(C)n1C1CC1 C1(CCC)COCCN(C(=O)C(C)(C)C)C1.C12(CO)CCCN(C1)C(=O)C2 c1(C(=O)NC2CN(C(CNC(c3ccco3)=O)=O)C2)cc2ccccc2o1 CCC(O)C(=O)N(CCC(=O)N(CC(C)C(C)C)C)CCCO CC(CN(C)C)CC(=O)NC(C)(C)CCCNC(C1CN(CC(F)(F)F)C1)=O C1(CC)CN(C(=O)CNC(C)=O)CC1C(=O)NC(C)CC1CCOC1=O c1(SC)ncc(C#N)c(N2CCCC2CNC(c2ccc(C(N)=O)cn2)=O)n1 c1(OCCn2c(C(C3CCSC3)NCc3nnc(C)s3)nnn2)ccccc1F N1(C(C2(OCC)CC2)=O)CCC(F)(CNC(c2cccc(C(C)C)n2)=O)C1 C1(CNC(=O)CNc2ccccn2)CCN(C(C2CCCS2(=O)=O)=O)C12CC2 C1(c2nc(-c3nnc(C(F)(F)F)o3)no2)(N(C)C)CCN(CC(F)F)CC1 N#Cc1cc(NC2CN(C(C3CCOC3)=O)CC2C(F)(F)F)c([N+](=O)[O-])cc1F C(=O)(C(F)(F)C(O)CC)Nc1cccc(NC(C(CCC)OCC)=O)c1 CCC1CNC(=O)C1.c1(C(=O)NC(CCC)C2CC2)cc(OC)ccc1OC N1(C(C=C(C)C(C)C)=O)CC2CC(NC(=O)CC3CCC(=O)N3C)CC2C1 c1(OC)cc(C(N2C3CCC2CC(CNC(=O)C(C)CF)C3)=O)c(OC)cc1Cl C1(CNC(c2c(OC)ccs2)=O)CN(C(=O)Cc2ccccn2)CCO1 c1(N(C)C)ccc(C(=O)N(C2CN(C(c3cccn3C)=O)CC2F)C)cc1 C1(N(C(=O)OCCOC)C)(CN(C2(OCC#C)CCC2)C)CCCC1 CC1CC(CNC(c2csc(Br)c2Cl)=O)CN1C(c1ccc(=O)oc1)=O C#Cc1cccc(CC(=O)NCC2CC(C(=O)NCCOCCSC)=NO2)c1 CN1CCC(C(=O)NCC2(O)CN(C(=O)CS(N)(=O)=O)C2)c2ccccc21 O=C(CC(Cc1cccs1)C(=O)O)NC1CN(C(=O)C(c2ccc(O)cc2)=O)C1 C1(NC(CC)=O)(CNC(c2ccn(CCF)n2)=O)CC2CCC1CC2 c1(CC(=O)NC2C(NC(CCSCC)=O)CS(=O)(=O)C2)ccc(Cl)c([N+](=O)[O-])c1 c1(C(N2CC=CC(NC(=O)C(C3CCCO3)C3CC3)C2)=O)ccc2cncn2c1 c1(C(=O)NC2CCCN(C(C(=O)NCC)=O)C2C)cc(O)c2sccc2c1 C1(NC(CCN(C(CC(COC)C)=O)CC2CC2)=O)CCCC(C)CC1 C1(NC(c2cncc(SC)c2)=O)C(C)CN(C(=O)Cn2nnc(C)n2)CC1C c1(CC(=O)N(CCC(=O)NCC(C2CC2)OC)C(C)C)cn(C)cn1 N1(C(c2ccn(C(C)C)n2)=O)CC2(CCC(CNc3cc(N(C)C)ncn3)O2)C1 N(C1CCCc2nc(C)sc21)Cc1ccc(OCC=C)c(OC)c1 c1(OC)cc(F)c(C(=O)N(C)CC2CCN(C(c3cccnc3S)=O)C2)c(F)c1 C(=O)(C(C(C)(C)C)NC(=O)CC1CCC(C)(C)C1)NCc1c(C)coc1 c1(OC(C(=O)NC(CC)CNC(c2cc(F)n(C)n2)=O)C)ccc(F)c(F)c1 C12CCCN(C1)CC1CC21.CC(C)C=CCNC(=O)NC(C)(C)C C(=O)(C(F)(F)C(F)F)NC1CC2(C(NC(c3nccc(N)c3)=O)C2)C1 C(=O)(C(C)C(C)(C)C)N(C)C.N12CC(O)(C1)C(F)C(=O)NC1(CC1)C2=O Cn1c(C(N2CCCC(C(=O)NCc3cnoc3)C2)=O)nnc1S c1(C(N2CC(CNC(C3(OC)CCCC3)=O)C(O)C2)=O)ccc2c(c1)COCC2 CC(C)CCC(=O)NC1CC(F)(CNC(c2ccccc2-c2ccncc2)=O)C1 CC1CCN(C(=O)C(O)Cn2cncn2)C1.C1(=O)CCCCC2(CC2)N1 c1(N2CC(SC)CC3(C2)CC3)ncnc2ncc(Br)cc12 c1(CC)noc(CC)c1CC(=O)NC1CC(NC(c2c(C)cnn2C)=O)C1 CC(C)(CN=c1[nH]c(=N)[nH]c(=NCC(c2ccccc2)OC2CC2)[nH]1)C(C)(F)F N1(C(CC(C)C)=O)CCC(CNC(c2ccc(Nc3nccs3)cc2)=O)C(C)C1 c1(NCC(c2cccc(Cl)c2)OC)nccc(=NCC(C)(C)CC(F)(F)F)[nH]1 c1(C(=O)OC)c(C)sc(C)c1S(=O)(=O)N1CCC(OCc2ccccn2)C1 C(=O)(C(O)C(C(C)C)OC)NCCN(CCOC)Cc1ccc(C)c(O)n1 C#Cc1ccc(C(N2CC(CNC(C3CC(C4CCC4)C3)=O)CC2C)=O)cc1 Cc1cc(F)c(F)cc1-c1nc(C2CC2)nn1-c1ccnc(F)c1 N1(C(C(C)C2CC2)=O)CCC(NC(=O)COC2CCC(F)(F)CC2)C(O)C1 c1(C(N2C(CN(C(C3C(CCC)C3)=O)C)CCC2)=O)cnn2c(Cl)cccc12 c1(NC(C2SCCN(S(CCC)(=O)=O)C2)=O)ccc(OC)c(S(N)(=O)=O)c1 CC1CN(C(c2csc(CNC(C3CC(C(C)C)=NO3)=O)c2)=O)C(C)(C)C1 C1(C(N2CCN(CC(=O)NC(C)CO)CC2)=O)(OC)CC(C)(C)C1 C=CCC(C(=O)N1CCCC(N(C(c2cnc(O)c(C)c2)=O)CC)C1)C(C)C CC1CCN(C(=O)COCCCF)CC1NC(=O)C(C)(F)F C1C(O)CC(=O)N2CC(C(O)C2)c2cn1nn2.c1(C(=O)O)ncccc1Br CN1CCC(NC(c2cc(CCNC(=O)C=Cc3ccoc3)on2)=O)CC1=O N1(C(C(C2CC2)OC)=O)CC(NC(=O)CCC2CCC2)CC12CCCC2 N1(C(c2c(C)c(F)ccc2)=O)CCCC(NC(c2csnc2Cl)=O)C(F)C1 C1(CC=C)(NC(=O)COC2CC=CC2)CCN(C(C2(CF)CC2)=O)CC1 c1(-c2cnc(CC)s2)nc(-c2ccc(C)cc2)nn1C1CS(=O)(=O)C1 c1(Oc2cc(NC(N3CCC(C#N)C3)=O)ncc2)nc2ccccc2o1 Cc1ccc(-c2cccnc2C(=O)NCC(C)NC(C2(CO)CCCC2)=O)cc1 Cc1cc(C(=O)NCC2CCCN(C(C3(CF)COC3)=O)C2)cc([N+](=O)[O-])c1Cl CC(CC(=O)NCCOCc1ccccc1Br)CC(C)(C)C N1(C(c2c(C)n(C3CC3)cc2)=O)C2CCC1CC(NC(C1CC1F)=O)C2 C1(O)(CC)CCCN(C(=O)CC(C)(C)CNC(c2cccc(CO)n2)=O)C1 N1(C(c2ncn(C(C)C)c2)=O)CC2CCN(C(C34CCC3C4)=O)CC12 c1(C(=O)NCCC(C)NC(CCOCC)=O)c(C)ncn(C)c1=O N1(Cc2ccc(C(=O)CN3CCSCC3)o2)CCOC(CO)C1 C(CCCNC(=O)C(C)=CCO)N(C(CN(C(=O)OC)C)=O)C1CC1.C1(SC)CC1 Cc1cc(C(=O)NC23CCC(CC2)N(C(C2CC4CC4C2)=O)C3)n2ncnc2n1 c1(OC)ccc2c(c1)C(N(C)S(=O)(=O)Cc1cc(C)no1)CC2 c1(C(=O)NC2CCN(C(c3cncc(C)n3)=O)C2C)cnc(C)nc1C C12(NC(CN(C(CC3C(C)(C)OCC3)=O)C3CCC3)=O)CCC(CC1O)C2 c1(CC)cccc(C)c1NC(=O)C(c1cn(C)nc1C)N1CC(C)CC1CC N1(C(c2c(C)nco2)=O)CCC(C2CC2)(CNC(=O)C=CC(F)(F)F)C1 N1(C(C2CC(C)(NC(C3CCCN(C)C3)=O)C2)=O)CCCC(C2CCC2)C1 Cn1nc(C2CC2)cc1C(N1CC(CNC(=O)Cn2cncn2)C2CC12)=O CCC(C)(CC)C(=O)NCC1CC2(CC(CNC(=O)CC3CCCC4(CC4)C3)C2)C1 C(=O)(C1=CCCN(C(C2CN(C(C)C)C2)=O)C1)Nc1cc(C)cc(C)c1 c1(N2CC(C(C)NC(c3cc(C)ns3)=O)OCC2)ncc([N+](=O)[O-])cn1 c1(C(=O)N(CCNC(C23CCCC2CC3)=O)CC2CC2)ccc(F)c(O)c1 N1(C(C2CC(CC)(CC)C2)=O)CC2COC(CNC(C3CC4(CCC4)C3)=O)C2C1 N1(C(C(C)Cc2cccnc2)=O)CC2CCC(NC(=O)C(C)C(C)(C)C)CC2C1 C1(C(N2CC(N(CC=C)C)C2)=O)CC(=C)CCN1C(=O)C1=CCCCO1 C12(NC(CC(CC)C)=O)CC(C)(C1)OC21CN(C(=O)Cc2ccc(F)cn2)C1 n1(CCC)cc(C(=O)NCCCN(CCCNC(C2CCC2)CSC)C)nn1 N1(C(C(C)(C2(C)CC2)OC)=O)CCOC(CNC(=O)Cc2conc2C)C1 CCC(C)C(=O)C(=O)NC(Cc1cn[nH]c1)C(=O)NCCCCS(C)=O C1(C(N2C(CNC(COCCOCC#C)=O)COCC2)=O)CCCCNC1=O C1(CC(=O)N(C(C)CNC(=O)Cc2cnn(C)c2)C)CC2COCC12 CC(CN=c1[nH]c(=NCC(C)(C)CC(C)C)[nH]c2c1COC2)C1CCCCC1 c1(C(C(=O)OC)NC(c2cc3n(n2)CCO3)=O)cc2ccccc2nc1Cl C(C(CNC(=O)CC1CC2CCC1O2)C(F)(F)F)NC(C(C)Cn1cccn1)=O c1(C(=O)NC(CC)CNC(c2cc(O)no2)=O)ccc2ncnn2c1 C12(C(N3C(C)(C)CC(CNC(C4CC5(CCC5)C4)=O)C3)=O)CCC(C)(CC1)CO2 N(C1CCCOc2c(Cl)cccc21)C(CCCC1CCC(=O)N1)=O N1(C(C(CC)Oc2ccc3nccnc3n2)=O)C2CCC1C1CC1(NC(N)=O)C2 C(=O)(CCCC(=O)NCC1CCCCN(C(C2CCNC2=O)=O)C1)NCCC c1(CC)ccc(C(N2CCC(CNC(C3(C(F)F)CCCO3)=O)C2)=O)s1 N1(C(C(C)N(C)C(c2cc3ccccc3o2)=O)=O)CC2CCC(O)C2C1 Cc1cc(CN=c2[nH]cc(CCNC(=O)C(C)Cc3ccco3)s2)ccc1Br C1(NC(CC2(C=C)CN(C(=O)CCCC(=O)C3CC3)C2)=O)CC1C1CCCC1 S(=O)(=O)(CC(=O)NCC1CCC(F)(CNC(=O)COC(C)C)C1)NC C1(F)(C(=O)NC(C2CCN(C(c3ccon3)=O)C2)C)CCCCC1 n1(CC=C)cc(C(=O)NC2CCC(N(C(=O)CSc3ccccn3)C)C2)nn1 C1(C)(N(C(=O)CCCCCN(C)C)CCN(C)C)CCCNS1(=O)=O c1(C(N2C(CO)CCC(N)C2)=O)cccn2cncc12 C(CNC(c1cccn1CCCO)=O)(C(C)(C)C)NC(C(C1CCCC1)OC)=O c1(C(=O)NCCN2CCN(C(C(CCC)(C)O)=O)CC2)cccc(N=[N+]=[N-])c1 C(=O)(CCC1=CCCCC1)N1CC(CC(C)(C)C)N(C(=O)C2=CCCSC2)CC1 C(=O)(C(C)(C)CCSC)NCCOCCC(=O)NC1C(C=C)OCC1 c1(CCC(=O)N(CC(CC)c2nn[nH]n2)Cn2nccc2C(=O)O)ccncc1Br C1(CCCCN(CC=C)C(C2CC(C#N)C2)=O)CCCN(Cc2ccc(O)nn2)C1 c1(C(N(CCCNC(c2c(CCC)nns2)=O)CC)=O)nc(CC2CC2)oc1C C1(C(=O)NC(C(N2CCC(CCO)CC2)=O)C2CCOC2)CC(=O)C12CCC2 C1(C(=O)NCC(CC)(C)NC(c2cccnc2O)=O)CCn2c(C)cnc2C1 N#Cc1c[nH]c(C(=O)NCC(O)CNC(=O)C(N2CCOCC2)C2CC2)c1 N12CC3CC1CCC3NC(=O)CONC(=O)NCC2=O.Cc1nc(C(C)(C)C)cs1 c1(C(N2C3C(NC(c4nnn(C)n4)=O)CC(C3)C2)=O)c[nH]c2cccc(C#N)c12 c1(N2CC(NC(C3=C(C)OCC3)=O)CC(C)(C)C2)ncnc2cccc(Br)c12 C1(C(N2CCC(CC(C)NC(C34CCN(CC3)C4)=O)CC2)=O)CN2CCC1CC2 c1(NC(C(C)C)C)cncc(C=CC(=O)OC(C)(C)C)c1 C1(C(=O)NCCCN(C(Cn2c(CCC)nnc2S)=O)CC)CCN(C)C(=O)C1 N1(C(C=C(COC)C)=O)CCCCC(N(C(=O)CCCc2ccc(F)cc2)C)C1 C=CC12CN(C1)C(=O)C1(CC1)C(=O)OC1CN(C1)C(=O)C2.NC.OC c1(C(=O)NC2(CO)CCCN(C(CC#N)=O)C2)cccc2ncsc12 c1(C(=O)NC2(CCNC(c3ccc(C)nc3)=O)CCCC2)ccnc(C)c1O Cc1c(C(=O)NCC(C)(C)NC(=O)C(F)Cc2ccccc2)cnn1C(C)(C)C Cc1ccc(C(=O)NCC2CC2NC(c2cnn(C(C)(C)C)c2C)=O)nc1C C(=O)(C(C)(C)CC(F)F)N1CC(c2cn(-c3c(OC)cccc3F)nn2)(OC)C1 c1(C(=O)NC(CCCNC(c2cnc(CCC)s2)=O)C)nnn(C)c1C C1(C(N(CCN(C(C2(C)C=CCC2)=O)CC)CC)=O)CC(=O)N1C(C)C c1(NC(C2CC(n3cc(CCNC=O)nn3)C2)=O)cc(O)ncn1 c1(C(=O)NCC2CC(F)(CNC(COC)=O)C2)ccc2cnccc2n1 c1(N2CC(OC)(CNC(=O)CCn3cc(Cl)cn3)C2)ccccc1[N+](=O)[O-] N1(Cc2c(CC)nn(C)c2)CC2CCN(C(c3sccc3Cl)=O)CC2C1 C(=O)(CC1=NN(C)C(=O)C1)NC1C(CNC(Cc2cc(C)nn2C)=O)C1 CC(C)CCC(O)C(=O)NCC1CC(F)(F)CN1C(=O)Cc1c[nH]c2ncccc12 C1(CNC(CC(=C)C)=O)CC(NC(=O)C=CC2CCOC2)C(O)C1 c1(CN(CC(C(=O)NC)C2CCCCC2)C2CCCC2)ccccc1C n1(CC)ccnc1C(N1CCCC1C1(NC(c2csc(CC(F)F)n2)=O)CC1)=O c1(CC(N2CC(O)(CNC(C3(C)CCCOC3)=O)C2)=O)coc2ccccc12 C1(C)(C(C)C)CN(C(=O)CC2CC3(C2)CN(C(c2occc2C2CC2)=O)C3)CCO1 Cc1c(C(=O)NCC=Cc2ccccc2)sc2nnc(S)n12 C(=O)(N=c1ccc(OC(C)=O)n[nH]1)C1CC(NC(C(CCCCC)F)=O)C1 c1(C(=O)NCC(CC)NC(=O)CC2COC(C)(C)C2)cc2n(n1)CC(F)C2 c1(-c2onc(N(CCC)CCNC(c3cc(C)n(C)n3)=O)n2)ccc(Cl)c(Cl)c1 c1(C(CNC(C2C(C(C)F)C2)=O)O)ccccc1Br C1(C(=O)NC2C(C)(O)C2)C2CC(O)C(C2)N1C(c1ccc(F)c(F)c1)=O CC1=C(C(=O)NC2CCCCCC2NC(c2ccccc2C(F)(F)F)=O)CCC1 n1(CC#C)c(C)cc(C(=O)NC2CC2C(=O)NCc2ccccc2C(N)=O)c1C CC(C)C(C)(C)C(=O)NCC1CCN(C(=O)C(c2ccc(F)cc2)=O)CC1C c1(NC(c2nc(NC(C(c3cccc(Cl)c3)C)=O)sc2)=O)cc(C#N)ccc1Cl NC(CCS(N)(=O)=O)C(=O)NC1C(c2ccccc2)C1(F)F C1(CC(=O)NCC(=O)NOCC2CCC2)C2CN(CC#CC3CC3)CC12 C(CNC(C1(C#N)CC1)=O)(CC(=O)NC1CN(CC(F)F)C1)OC c1(CO)cccn2c(O)nnc12.c1(OC)ncnc(NC2CCN3CC2NC3=O)c1C C1(C(=O)NCCOC)CN(C(=O)C(C)CC(C)C)CC1(C)C C(C)(C)(CC(C)NC(C1CCC(n2cc(-c3ccns3)nn2)C1)=O)OC CC1CC(NC(=O)C=CC2CCCC2)CN(C(=O)CCSC(F)(F)F)C1 C1(=O)C(C)(C)COC(=O)C2CC(CO2)N1CC=C.c1(OCC(F)F)ccc(F)cc1 N1(C(C=C(C)I)=O)CC2C(N(C)C(c3ccc(O)nc3)=O)C2C1 Cc1oc(COCCCC2CCCN2C(=O)C(O)C2CC2)nc1C(=O)OC CCC(CC)C(C(=O)NCC(O)CNC(c1ncncc1C#N)=O)OC C1(C(=O)NCC(C)CC2CCC2)CN(C(c2c[nH]nc2C(F)F)=O)CC1F C1(CC=C)(NC(C2CC2(C)C)=O)CC2CCC(C1)N2C(=O)C(C)COC N1(C(c2cccc(O)c2)=O)CC2CCC(C1)N2C(=O)C(c1ccc(F)cc1F)O n1(CC(N2CC(NC(C3CC(OC)C3)=O)C(OC)C2)=O)cc2ncccc2n1 C(=O)(CCCCCCS(N)(=O)=O)N1CC2CCC(NC(C3CCN(C)C3)=O)(C1)C2 C=CCC(C)(C)C(=O)N1CCC(NC(=O)CCC2CC(F)(F)C2)C1 N1(C(c2nc(C#C)sc2)=O)CCN(C(c2nc(C)sc2C(F)(F)F)=O)CC(O)C1 C1(C(N2CCCC(NC(C#CC3(C)CC3)=O)(CO)C2)=O)CCc2nc[nH]c2C1 n1(C(C)(C)C(=O)NC2CC3C(NC(c4c[nH]c(=N)o4)=O)C3C2)cnc([N+](=O)[O-])n1 c1ccc(F)cc1.c1(C(N2CC3CC3C2)C(=O)NC(CC)C)csc(COC)n1 c1(OC(C)C)ccc(C(C(=O)Nc2ccsc2)NC(C)CC(C)(C)O)cc1 C1(CC)CCCCC1C(=O)N(C)CCNC(C1(Br)CC1)=O N12CC(OC(F)(F)F)C(C1)C2=O.C(=O)(CC(F)(F)F)NC1C(C)C1 n1(CC(CC)O)cc(C(=O)NCC2C=CCN2C(C2CC(O)C2)=O)nn1 CC1CCC(C(=O)Nc2nccs2)CC1.C1(=O)CCCn2cc(nn2)CN1C N1(C(C2CC3CCC2CC3)=O)CCC2(CCCN2C(C2CCCCC2O)=O)C1 C(C(C)(C(=O)N1CC(C(C(=O)NC2CCC2C(N)=O)OC)C1)OC)OC N1(CC(=O)N(C)CC2(NC(=O)C(C3CC3)C3CC3)CC2)CCCC1=O N1(C(CCCOCCOC)=O)CCC(O)CC1C(=O)NCc1ncccn1 c1(C(=O)NCC#CCNC(C2OCCC(C)C2)=O)ccc(Cl)cc1Br C(CC(F)F)NC(=O)NC(c1cc[nH]c1)C c1(C(=O)NC2(COC)CCN(C(c3ccsc3Cl)=O)CC2)cc(C)cc(Cl)c1N C1(NC(CCC2C(C)=NNC2=O)=O)CCN(C(c2cnn(CCO)c2)=O)CC1F C1(NC(Cc2nc(C)[nH]n2)=O)CCN(C(=O)Cc2nc(C(C)C)c(C)s2)CC1C N1(C(C)=O)Cc2ccccc2CC1C(=O)NCCC1CN(C(=O)CC(C)(C)O)C1 S(=O)(=O)(CCCCS(C)(=O)=O)N(C1CC(N(CCC(=O)O)C2CC2)C1)C c1(C(=O)Nc2ncc(-c3c(N(C)C)nccc3)s2)c[nH]c2ccc(Br)cc12 c1(C(=O)NCC2(NC(CC3C(=O)NCCC3)=O)CC2)ccc2c(c1)C(=O)NC2=O c1(CNC(C2C(CC)C2)=O)ccc(CNC(c2cc(Cl)n[nH]2)=O)cc1 c1(C(=O)NCC2CCN(C(C(C)n3cnnn3)=O)C2)cc(Cl)c(F)cc1F CC(C)CC(C)(O)CNC(C1CCCC(N)CC1)=O CC(CC(=O)N1CC(CO)(NC(=O)Cc2ncn3c2COCC3)C1)C(C)(C)C c1(-c2nc(C3CCCN(CC45C(C(=O)O)CC(C4)C5)C3)on2)ccc(F)c(F)c1 C1(CC(=O)NC2CCC(NC(CC(C)CN(C)C)=O)CC2)Cc2ccccc2O1 C1(C)(C(NOC(CC)C)=O)C=CCN1C(c1cn(C(C)C)cc1C)=O c1(CNC(CNC(=O)NC)=O)ccoc1C(=O)N(C)CCN1CCCC1 C(=O)(C1=CCCCO1)NC(C)CN(C)C(C1(c2cc(Br)ccn2)CC1)=O c1(NC(=O)CC2CCN(C(C3CNC(=O)O3)=O)C2)cc(Cl)ncc1Cl CC(CS(C)(=O)=O)C(=O)N1CC2CCN(C(c3c[nH]nc3-c3ccco3)=O)C2C1 c1(C(=O)OC)cc(C(=O)N(C2CCN(C(=O)CC3CCC(O)C3)C2)C)on1 C1(NC(C2CCCC(OC)C2)=O)CC2CN(c3cc(C(C)C)nc(C)n3)CC12 N1(C(C)=O)CCC(NC(c2cccc(C3CC3)c2C)=O)C12CCC2 N1(C(CC(CN(C)C)O)=O)CC2CC(N(C(=O)CN(c3ccc(Cl)cc3)C)C)C1C2 N1(C(c2ccsc2C(=O)OCC)=O)CC(C)N(C(=O)CN2CCCCC2=O)C(C)C1 C12(NC(C(CC)CCOC)=O)CCC(CNC(c3snc(O)c3Cl)=O)(CC1)OC2 C#Cc1ccc(C(=O)NCCC2COCCN2C(=O)C(C)C2CCC2)c(F)c1 C12(C(N(C)CCNC(c3cc(C(F)(F)F)on3)=O)=O)CC=CC(C1)OC2 C1(c2c(C(=O)NC(c3ncc(Cl)s3)C)cno2)CCN(CC)CC1 CC1CC(C(=O)O)CN(C(=O)CN2CCC(CN(C)C)CC2)C1 C1(CN(C)C(=O)OC(C)(C)C)CCC(c2ccccc2)CC1 C1(NC(c2cnc(COC)s2)=O)CC2CC(C1)CN(C(c1cc[n+]([O-])cc1)=O)C2 Cc1cc(C(=O)NC2(C)CC(NC(=O)CC3(C)CCCC3)C2)sc1C c1(C(=O)NCC2(C)CCCN2c2cncc(Cl)n2)ccc2ccccc2c1 C1(C)(C(=O)NC(C2CCN(C(C=CCC)=O)CC2)(C)C)CC(=O)N(C)C1 c1(OC)ccc(C(=O)NC(C2CN(C(=O)C(C)(C)O)C2)C)c(OC)n1 C1(C(N(C2CN(C(c3cccc(C)c3)=O)C2)C)=O)CC(C)CCC1C(C)C c1(NC(C2CCN(C(c3cnccn3)=O)C2)=O)cc(Br)c(O)cc1Br N1(C(C2CC(C(F)F)C2)=O)CCC2CCCC12C(N1CCCC(F)C1)=O N1(C(C(CC2CN(C(c3c[nH]c(=N)o3)=O)C2)F)=O)CCC(CC(N)=O)CC1 CC12CC(CO1)N(C(C1CC13CC(NC(C1(Cl)CC1)=O)C3)=O)C2 N1(C(c2cnc(C(F)F)nc2)=O)CCC2CCC(C1)N2C(=O)CCOC1COC1 c1(CNC(=O)Nc2cnc(CC)s2)ccccc1SC.C12(CC=CC1)C(=O)C2 n1(CC(=O)NC2CCN(C(c3c(C)ccnc3)=O)C2)[nH]cc2c(=O)ncnc1-2 C1(C(=O)NC2CN(C(CN(C(=O)OC)C)=O)CC2C)CC2(CC(C)=NO2)C1 C(=O)(C1CCC(=O)Nc2ccccc21)NC1C(NC(C2(CC#C)CC2)=O)CCC1 c1(C(=O)OCc2cnc(C(C)(C)C)nc2)cc(F)c(Br)cc1F Cc1ccnc(CNC(C2CCCCN2C(=O)CCN2CCN(C)CC2)=O)n1 C(=O)(C1=CC2CCC(C1)C2)N1C(CNC(=O)C2=CCCSC2)C2CCC1C2 N1(C(c2c(C)nsc2)=O)CC2CCCC(NC(=O)CCC3CCC(=O)C3)C2C1 c1(C(C(=O)NC(C(=O)OC)C)N(C2CN(C(C)=O)C2)C)cccc(F)c1Br C1(NC(C2CC(CCC(=O)O)C2)=O)C2Cc3cc(Cl)ccc3C12 CC1CN(C(=O)CSC2CCCCO2)CCN(C(c2cn(C)nc2Cl)=O)C1 CC1(C)COC(CC(=O)NC(C(=O)NCCN2CCCC2)C2(C)CC2)C1 C(CC(C(C)(C)C)NC(=O)C=C1CCCCC1)N(C)C(C1(C)CCN(C)CC1)=O c1(C(=O)NC(C)(C)CNC(c2ccc(N)c(N)n2)=O)cc(Cl)cc2c1OCC2 CC12CCN(CC1)Cc1cn2nn1.C1(C(=O)NCC(F)(F)F)CCCN1C1CC1 c1(C(=O)OC)cc2c(s1)CCOC2CNCC(COC)OC(C)=O CC1CCC(CC(N2CC(O)(C(F)C(=O)NC(C)CC3CC3)C2)=O)OC1 c1(OC)ccc(OC(=O)C(O)CNC(=O)OC(C)(C)Cc2ccc(C)cc2)cc1 C1(CNC(C2C=CC(NC(c3scnc3Cl)=O)C2)=O)CC2CCC(C1)O2 N1(C(C(C)(C)C2CCCN2C(c2cn3c(n2)CCC3)=O)=O)CC2(CCCCC2)C1 C1(NC(C(CC#C)C)=O)CN(C(=O)C(CCC)OC)CCC1C(F)(F)F CC(C)CC(C)(C)C(=O)NC1CCN(c2cc(C(F)(F)F)ncn2)CC1F C1(CCNC(C(CCCC)F)=O)CC2CCC(C1)N2C(C1COCC(C)O1)=O CC(C)CCC(F)C(=O)N1CCCC(C(=O)N(C)CC2CCOC2)C1 C1(C(N2CC3CC2CS3=O)=O)(CC)CCN(C(C2C=CC=CC=C2)=O)CC1 C1(C)(C(=O)NCC(=C)CCNC(=O)C=Cc2nccs2)CCCNC1=O C(=O)(C(C(C1CC(F)(F)C1)OC)N(C1CCCN(C(C)C)C1)C)NC(C(=O)OC)C C1(CCOC)CN(C(C2CC2C)=O)CCN1C(C12COCC(C1)C2)=O N1(C(C(CCC)OC)=O)CCOC(C)(CNC(c2cccc(F)c2OC)=O)C1 C(C)(CNC(=O)CC1(C)CC(F)(F)C1)(C(C)C)NC(C(C1CCCC1)OCC)=O C1(CNC(C2(F)C(C)OCC2)=O)CN(C(c2cc(O)nc(O)n2)=O)CCN1C C1(NC(C(CC)=CC)=O)CN(C(=O)CSCC)CC12CCOCC2 c1(C(=O)NCC(C)NC(=O)CCS(C)=O)nn2cccnc2c1Br C=C(C)C(O)CC(=O)N(CC(C)N(C)C(c1ccc(SC)o1)=O)C C12(NC(=O)CSc3n[nH]c(O)n3)CCCC1N(C(=O)CCc1cncs1)CC2 C(=O)(N=c1c(Cl)c[nH]cc1I)C1CN(Cc2c(C)ccc(Br)c2)CC(F)C1 C#CCC(C)(CNC(=O)C(c1ccnn1C)NC(=O)C(F)(F)C=C)CO N1(C(C2C(C)C2)=O)CCCC(NC(c2ccn(C3CCCC3)n2)=O)CC1 C1(NC(CSS(C)(=O)=O)=O)(CNC(=O)C(C2CCOCC2)O)CCCCC1 C1(C(=O)OC)C(C)(C)CN(C(=O)NCC2(F)CC(C(=O)O)C2)CC1(C)C C12(C(N3C(CCNC(C4CCN(C)C4)=O)CCC3)=O)CC(C)(CCO1)C2 C(=O)(C(=O)N=c1cc(C)o[nH]1)NCCCN(C(CC(CCCC)O)=O)C c1(-c2[nH]c(=NCc3nnc(C(=O)OCC)s3)sc2)cc(Cl)nn2c(C)nnc12.O C1(NC(Cc2n(C)ccn2)=O)CC2CN(C(=O)CC3CCCNC(=O)C3)CC2C1 c1(NC(c2cccc(Cc3ccc(OC)cc3OC)c2)=O)cccc2c1CCN2 c1(C(N(C)CC2CCN(C(=O)CCc3ccsc3)C2)=O)ccc2c(c1)COC2=O Cc1nc(CNC(=O)C=CC(C)(C)C)ncc1C(N1CCCC1CO)=O C(=O)(C(C)(C)CS(N)(=O)=O)NC1(CCC)CCN(C(=O)C(F)C(F)(F)F)CC1 Cc1ccc2c(=NCC3CCc4cccn43)[nH]c(N(C)Cc3nccs3)nc2c1 CC(C)CC(C(=O)N1CCC(c2cn(CC3CCC3)nn2)CC1)N1CCCCC1 c1(NC(CC)CSC)cc(-c2ccc(O)c(N)c2)c(O)c(Cl)c1 O=C(CCC1CC2(CCOCC2)CN1)NNc1ccncn1 N1(C(c2ccnc(OC)n2)=O)C2CCCC1CC(CNC(=O)C(F)OC)C2 C(=O)(C(CCF)NC(c1c[nH]cc1CC)=O)N1CC(CC(=O)OCC)C1 c1(CCNC(CC2CCN(C(c3c(CC#N)ccs3)=O)C2)=O)ccc(O)cn1 c1(C(=O)OCC)cc(C)c2c(c1)CCCN2C(=O)C(N1CCN(C)C2(CCC2)C1)=O n1(CC)nccc1C(=O)NCC1(C(=O)NCCCC2(C(F)F)CCCC2)CC1 c1(NC(C)=O)ccc(F)c(NC(C(N2CC3CC2(CO)C3)=O)=O)c1 C1(NC(=O)CN2CC3CC3C2)CCC12CN(C(c1ccsc1Cl)=O)C2 C1(N(C(C)C(=O)NCC(F)F)CCC)CC2CCC1CC2 N12CCC(C)C(C1)CNCNc1cn(c(=O)nc1O)CC2=O.CC(C)(C)C1CC1 c1(C(=O)NCCCN(C(C2CC(F)C(=O)N2)=O)CC)ccc2c(c1)C1CCC2O1 C#Cc1cc(C(=O)NCC2CN(C(c3cc(CSC(F)F)c[nH]3)=O)C2)cc(Cl)c1 N1(C(C(CC)NC(N)=O)=O)CC2C(N(C(c3ccncc3Cl)=O)CC)C2C1 c1(CC(=O)NCC23CC(NC(C4(C)COC4)=O)(C2)C3)cccc(Cl)c1F C12(CC(=O)NCC(CC=C)NC(=O)CNS(=O)(=O)C3CC3)COC(CF)(C1)C2 c1(NC(=O)NC23CC(COC4C(C)CCCC4)(C2)C3)cccc2oncc12 C1(CCC)(NC(=O)CCc2ncccn2)CCCN(C(C2CCOCC2)=O)C1 C=CC(C)(O)CC(=O)NCC(C)NC(=O)C(C)(C)NC(=O)C(F)(F)F N1(C(C(COC)NC(C)=O)=O)CC(CNC(=O)C=CCn2cncn2)CC(C)C1 Cc1cccc(C(=O)NCC2CN(C(=O)CC(C)C(C)C)CCC2C)c1F CCC(C)(CC)C(=O)N1CCOCC(C(=O)NC2CCC(C)C2)C1 Cc1c(C(=O)N=c2ccn(-c3cccnn3)[nH]2)ccc(I)c1F Cc1ccccc1NC(=O)NC1CCCN(C(=O)Cc2ncccn2)C1 C(C1CN(C(C2CCC23CCC3)=O)Cc2ccccc21)NC(=O)Cc1cn[nH]c1 C1(CNC(C(C)NC(=O)C(C)(C)C)=O)CN(C(c2nc(Cl)cs2)=O)CC1(C)C c1(C(N2CC(C)C(CNC(=O)Cn3nccn3)CC2)=O)ccnc2c1ncn2C c1(C(=O)NCCC(=C)CNC(=O)CCC2CC2)cncc2ncn(C)c12 c1(C(N2CC3C(C(F)F)C3C2)C(=O)NCCCC)cccc(OC(F)(F)F)c1 c1(CNCc2cc(C(C)(C)C)on2)cc(CO)cc(Br)c1 c1(C(=O)NC(C(N2CC(C(=O)OC)OCC2)=O)C(C)C)ccc(C)cc1O c1(C(C)NCCCCCO)ccn2nnnc2c1.n12ccc-1n2 c1(NC(N2C(CC(=O)OC)COC(C(F)(F)F)C2)=O)cc(C(F)(F)F)cc(Br)c1 N1(C(C(C(=C)C)(C)O)=O)CCC2(NC(c3cnc(N(C)C)cn3)=O)CCCC12 C=CCC(C)C(=O)N(C)CCOCCCN(C(=O)CS(=O)(=O)NC)C NS(=O)(=O)N1CC(C(N2CC3CC3(NC(C3CCC4(CC4)C3)=O)C2)=O)C1 C(=O)(CC(C)(C)CO)NC(CSC)CC(=O)NCC1=NOCC1.C(C)=O CC(C)CC(O)CC(=O)NC1CC2CC1N(C(c1cc(N)ccn1)=O)C2 c1(C(N2C(C3(NC(=O)CCn4ccnc4)CC3)CCC2)=O)cccc(CCO)c1 CC1(C)C(NC(=O)C(c2cccs2)NC(C23CCC(C)(C2)OC3)=O)CC1(F)F N1(C(CC(=O)NC)=O)CCC(NC(=O)C=Cc2ccc(C(N)=O)o2)C(C)C1 c1(C(=O)NCC2(F)CC(NC(C3CN(C)C(=O)N3)=O)C2)ccc2cc[nH]c2c1 C1(NCCC(C)c2ccco2)CN(S(=O)(=O)C2CC2)CC12CC2 CON(CCC(=O)N1CC2C(C)C2C1)C(=O)C(O)c1ccccc1 C1(NC(=O)Cc2ccncc2)CN(Cc2cncnc2)CC(F)(F)C1 C12CC(F)(F)CN1S(=O)(=O)C2.C1(CCNC)CCN(S(C)(=O)=O)CC1 c1(CC)cc(C(N2CCC(NC(=O)Cc3ccc(Cl)cc3F)C2)=O)cn(C)c1=O c1(CC)occc1C(=O)N(C)CCOCCNC(C1COC(C)C1)=O N1(CCCCCOCC#C)CCN(SCC(=O)Nc2cn(C)nc2C2CC2)CC1 c1(C(=O)NCC(CNC(Cc2ncn(C)n2)=O)F)cccc(C(N)=O)c1 c1(C(=O)NC2CN(C(C(C)CN(C)C)=O)CC2C)cccc2nc(CO)[nH]c12 c1(-c2ccc(C(C)NCCn3ccc([N+](=O)[O-])n3)cc2)cccc2[nH]ncc12 Cc1cc(C(N2CC3CC(C2)C3NC(=O)CC2(O)CCOCC2)=O)nnc1C Cc1csc(C=CC(=O)NCC2C(C)CCN2C(=O)CCCc2csc(C)n2)n1 c1(C(=O)NCC2OCCN(Cc3cn(C)nc3)C2)cc2cccnc2cc1Cl N1(C(c2c(C)nsc2)=O)CCN(C(c2cc(NC3CC3)ncc2Cl)=O)C(C)C1 C1(C(CNC(c2cnc(SC)[nH]2)=O)(C)O)CCCN(C(c2coc(Cl)c2)=O)C1 C(CNC(c1ccccc1NS(C)(=O)=O)=O)(CC(F)(F)F)NC(C(C)C)=O c1(C(N2CCCC(N(C(C(CSC)O)=O)C)C2)=O)c(F)cccc1Cl CCC(C)CC(C(=O)NCC#Cc1cnn(C)c1)NC(=O)COc1ccn(C)n1 c1(C(=O)NC(CN(C(COC(CC)C)=O)C)C)cc(Cl)cnn1 c1(CN2CC3C(C(=O)O)(CCOC3)C2)cccc2c1S(=O)(=O)CCC2 C1(C(=O)NC2CC3(CC3)C2)CCCN(C(c2nc[nH]n2)=O)CC1 c1(CCC(=O)NC(C(C)NC(C2CCCC2CC2CC2)=O)(C)C)ccccc1F N1(C(c2c(C)noc2C)=O)CC2CCN(C(c3cnc(Cl)c(F)c3N)=O)C2C1 Cc1nc2cccc(C(=O)NCC3(C)CCN(C(=O)CC4CC5CC5C4)C3)c2[nH]1 C(CN=c1ccnc(Cl)[nH]1)C1CCN(C(c2n(C)c(O)nc2)=O)C1 c1(NCc2c(OC)c(Br)ccc2)cc(Br)ccc1S(=O)(=O)NC(C)(C)CC(N)=O C1(OC)CN2CC1C(=O)NCC(C)(C)C2=O.C(C(C)(C)SC)NC(C)=O C1(C(=O)NCC(CC)NC(=O)CNC(C)(C)C)C(C2CC2)CCN1C(C)=O C1(C(N2CCC(C(C)C)C2C(=O)O)=O)CC2(CC2)CN1C(=O)OC(C)(C)C C1(=CC(=O)NCC2C(NC(CC(CC)OC)=O)CC2)CCCCCC1(F)F CC1CCC=C1C(=O)NCCCOCCN(C)C(C1CN(C2CCOC2)C1)=O C=CC1(C(=O)NC(COC)CCO)CCN(C(C23CC(CO)(C2)C3)=O)CC1 C(C(CC(=O)NC1CCCCN(C(=O)C#CC2(C)COC2)C1)C(F)(F)F)N(C)C N1(C(c2ccc(NC)cn2)=O)CC2CC(CNC(c3ccnc(C)n3)=O)C2C1 c1(C(=O)N)coc(C(F)F)n1.C(C(C)(C)N(C)C)N(C(=O)CSCC(C)C)CCC Nc1cc(F)cc(C(=O)NCCC2CCCN(C(C3CCCCC3)=O)C2)c1F C(CC(C)N=c1nc(-n2c(CO)ncc2)c2c([nH]1)c(C)nn2C)NCCSCC CCC(F)C(=O)NCCCCC1CN(C(=O)Cc2ccsc2C)C1 C1(C(N2CC(C#C)(F)C2)=O)N(C(c2c(C)cccc2O)=O)CCCC1(C)C C1(C(N(C2CCCN(C(c3coc(C(F)F)n3)=O)C2)CC)=O)CCCC1(F)F CCC(C)C(=O)N(C(C)CNC(=O)Cn1cc[n+](C)c1)C N1(C(c2c(CCC)nns2)=O)CC2CC1C2NC(=O)Cc1cn(C)nc1C C(=O)(C1=CCC2CCC1N2C(C1CC2CC(=O)C1C2)=O)N1C(C)(C(F)F)CCC1 C(C)(C(=O)N(CC(C)CNC(C1CC1c1ccsc1)=O)C)=C(C)C C(=O)(C1CCc2ccccc21)NC(C(=O)NC(CC#C)C(=O)NC)CC(C)C C1(CNC(Cc2cc(CC)no2)=O)CN(C(=O)C(C)NS(C)(=O)=O)CCC1(F)F N1(CCNC(CC=C)=O)CC(C)OC(C)C1.C12CCN1C(=O)CCS2 C12(C(N(C)Cc3nc(C)on3)=O)CCC(CC1NC(c1cccc(O)n1)=O)C2 Cc1cc(Br)c(NC(C2CN(C(c3cscc3Br)=O)CCN2)=O)cc1C c1(C(N2CCCCC(CNC(C3(CO)COC3)=O)C2)=O)cnn2c(=O)cc[nH]c12 C(=O)(C(C)(C)CCC#N)NCC1(F)CCCN(C(CC2N(CC)CCOC2)=O)C1 C1(NC23CCC(CNC(=O)OC(C)(C)C)(OC2)C3)CC2(CCC2)CCO1 C(=O)(C(C)C(C)NC(=O)C(CNC(C1(C)CCSCC1)=O)OC)OC c1(C2(CNC(=O)NC3CC(c4ccc(F)cc4)(F)C3)CC2)cncc(F)c1 C#CC1(C(=O)NCC2CCC(CNC(=O)OC(C)(C)C)CC2)CCOC1 C=CC(CCC)CC(=O)NCC1C=CCN1C(c1nnn(C)n1)=O c1(C(=O)NCCC2CCN(C(c3n(C)nc(Cl)c3)=O)C2)cc(Cl)cc(F)c1F C1(CNC(C(CC)n2cccn2)=O)CN(C(c2cnc(C3CC3)s2)=O)CC1(F)F CC1CCC(C)N(C(=O)C=CCNC(=O)C#CC(C)(C)O)C1 c1(OCC)nc(NC2(CNC(c3cncc(C)c3)=O)CCC2)ncc1Cl CC(CC(C1CCC1)NC(=O)OC(C)(C)C)C(=O)NC(C1(CCN(C)C)CC1)=O C(=O)(C1=CN(C)S(=O)(=O)N=C1C)NC(CC)CN(C(=O)CCc1ccccc1)C C1(NC(c2cc(O)nc(Cl)c2)=O)CC12CCN(C(c1csnc1Cl)=O)C2 C(=O)(CCCn1cncn1)N(C(C)C(=O)NCCN(CC)CC)CCC CC(CC(=O)NCC(C)(C)C)C(C)(C)NC(C1CC(=O)CCO1)=O c1(C(N2CCC(NC(C(CCC)(C)C)=O)C2CC)=O)ccc2c[nH]nc2c1 c1(C(N2C(CNC(=O)CC3COCCO3)COCC2)=O)cccc(C=C(F)F)c1 C1(C(=O)Nc2c(CC)ccs2)CC(C)CN1C(C1(C#N)CC1)=O C1(CC)CN(C(=O)CC2(OC)CC2)CCC1NC(=O)CC(C)(C)CC C(=O)(CC(C)(C(F)(F)F)N(C)C)NC1CCC(NC(C(C=C)(C)C)=O)C1 C1(C(C)(C)NC(c2cnc(C)[nH]2)=O)CCN(C(c2ns[nH]c2=O)=O)CC1 C(CC1=CCCCC1)N(C(C(COCC)C)=O)C.C12CC(N(C)C1)NC2=O CC1(C#CC(=O)N2CCC3(CC3C(N3CC(CC(F)F)C3)=O)C2)CCCO1 c1(N(C(CCC2CC(NC(C(CC3CC3)OC)=O)C2)=O)C)cc(Cl)ccc1C c1(OCC)cnc(C(=O)NCC(C)(C2CC2)NC(c2cc(CC)oc2C)=O)c(Cl)c1 N1(C(CCCC)=O)CCC(C)(C(=O)NCc2ccccc2-n2ccnn2)CC1 C(=O)(C#CC1CCCO1)N(CCCCN(C(C(c1cccc(C)c1)=O)=O)C)C c1(SCC=CCCC)ccc(F)cc1.c1(C2C3CC(C3)N2)ccc(Cl)cc1 c1(OCC(=O)N(CC(CNC(C2C(C(=O)OC)CC2)=O)O)C)ccc(Cl)cn1 C(=O)(C1=CCCC(C)(C)C1)N1CCN(C(C(C)CCO)=O)C(c2ccnn2C)C1 Cc1ccc2c(=NCC3CC(C)N(C(C4CCCN4C(N)=O)=O)C3)[nH]cnc2c1 CC(C)C(F)C(=O)NCC1CN(C(c2cncc(-n3cc(Br)cn3)c2)=O)C2CC12 Cn1cc2c(C(N3CCCC34CCN(C(=O)CC3(C)CC3)C4)=O)cccc2n1 N1(C(c2cccc(CC#N)c2)=O)CCN(C(c2cc(O)ncn2)=O)C(C2CC2)C1 CCC(CC(=O)NCCC(C)(C)NC(c1cc(F)n(C)n1)=O)C1CCC1 c1(CC(=O)NC2CCN(C(C(C)CSC(F)(F)F)=O)C2)cn2ccccc2n1 C1(NC(CN(C)C(C2(F)CC=CCC2)=O)=O)CC2CCCCCC12 C(=O)(CC1COc2ccccc21)N1CC(CN(C(CCC(=C)Cl)=O)C)OCC1 c1(C(=O)NC2CCN(C(CC3(C)CCCO3)=O)C2)ccccc1OCC(F)(F)F C1(CNC(=O)C(Cl)=CCl)CN(C(=O)CN2CCOC2=O)CC(C(F)(F)F)O1 N1(C(CCN(C2CCOCC2)C)=O)CCCC(NC(=O)C(F)OC(F)(F)F)CC1 C(N=c1[nH]c(N(CC(F)F)C)nc2c1CCC2)c1cc(C)c(F)cc1 C(=O)(C(C)(CC=CCl)c1ccccc1)NCCN(C(=O)C(F)(F)C(F)F)CCC c1(C(=O)NCC2CC(NC(=O)C3=CCSC3)C2)cc([N+](=O)[O-])c[nH]1 C1(NC(C2CC(C)=C(C)CC2)=O)C2CCCC1CC(NC(=O)Cn1cccn1)C2 S(=O)(=O)(c1cccnc1NCC(=O)Nc1cccs1)NC(C1(C)OCCO1)CO C1(C(N2CCCC2c2c(F)cccc2Cl)=O)C2Cc3c(Cl)cccc3C12 CC1CCCC=C1C(=O)N1CCC(NC(=O)CC2(O)CCCCCC2)C(O)C1 C12CC3CCC(C1)N3CC(=O)NCCNC2=O.C1(N)CCC2(CNC2)O1.CO C1(NC(c2cccnc2S)=O)C2CC3CN(C(c4cc5cscc5s4)=O)C1C3C2 C(=O)(C(c1cccs1)=Cc1ccc(=N)[nH]c1)NC1CCCN(C(C=C(C)C)=O)C1 N=c1[nH]ccc(C(N2CCC3(NC(=O)CCc4cc[nH]n4)CC3C2)=O)c1[N+](=O)[O-] N1(C(CC(COC)(C)O)=O)CC2CN(C3CCCc4ccccc43)CC2C1 C1(C(=O)NC)CCCN(C(=O)C=NOC)C1.c1(C(NCC2CC2)=O)ccn(C2CC2)c1 c1(C(=O)NC2C(C(=O)Nc3ccnc(Cl)c3CO)CCC2)c(Cl)cc(F)cc1Br CC1(C(N2CC(C3CCOCC3)C2)=O)CCCN1C(c1cc(=N)[nH][nH]1)=O C(c1ccsc1Br)=CC(N1CC(CC(C)NC(C2C(C)(C)C2(C)C)=O)C1)=O c1(-n2cc(CC3N(C(C(Cn4ccc(C)n4)C)=O)CCC3)nn2)ccnc(CO)c1 N1(c2ncc(CC)cn2)CC2CCC(C1)C2NCc1ccc(Br)s1 Cc1c(C#N)nn(-c2ccccc2Cl)c1CNCCc1cnc(N)c(Br)c1 CCC(C)(C)CC(=O)N(C(C)(C(=O)NCC(O)CNC(N)=O)C1CC1)C N1(C(COC)=O)CCCCC1C(N1CC(C)(NC(=O)CCC2CC2(Cl)Cl)C1)=O N1(CC)CCOC(C(=O)NCC2CN(C(C3CC3c3ccn(C)n3)=O)C2)C1 C1(C(=O)NCC2(F)CC(NC(=O)Cn3c(C)ccc3C)C2)(OC)CCCCCC1 C1(C(=O)NCC(C(=O)OC)OC)CC2CC1CN(C(=O)COC(C)C)C2 CC(C)C(CCNC(=O)CC1CCC1)NC(C1(c2ccccc2)CC(F)(F)C1)=O C1(NC(C=Cc2ccc(C)o2)=O)CC2CCC(C1)N2C(C1CCCC12CC2)=O CC#CCCCCNC(=O)CC(C)CNC(C1CCNC1=O)=O C1(O)(c2cn(N(C(CCCC#C)=O)CC)nn2)CC2CCC(C1)N2C(=O)CCP(C)(C)=O CC1(CNC(=O)CSCC(N)=O)CCC(NC(c2cnn(C(F)F)c2)=O)C1 C1(C(=O)NCC2(NC(c3c(C)cncc3)=O)CCCC2)CCOCC1(C)C c1(OC)nccc(SC)c1-c1cncc(C(=O)Nc2cc(F)ccc2Br)n1 n1(C(C)CCNC2CN(C)C2)nnnc1C(CC1CCC1)NC(=O)OC(C)(C)C C#Cc1cccc(C(=O)NC2CN(C(c3ccc(Cl)nc3N)=O)CCC2F)c1 c1(OC)ccc(Cl)c(CC(=O)Nc2cccc(NCc3cc(C(C)(C)C)no3)c2)c1 C12(CNC(c3cccs3)=O)CCC1CN(C(c1cccc(-c3cc[nH]n3)c1)=O)C2 C1(CN(C2CCN(C(C3CC3)=O)C2)C(CNS(NC)(=O)=O)=O)CC2CCC1O2 N1(C(C(CC)SC)=O)CCC(CC)(Nc2nc(C#N)c(Cl)s2)CC1 C1(NC(c2ccc(C(F)F)o2)=O)CCOC(C(N2CCC(OC3CCC3)C2)=O)C1 N12CCC(C(F)(F)C1)CN1CC(C1)C2=O.c1(C(=O)O)cccc(F)c1Cl C(=O)(C(O)P(C)(C)=O)NCCN(C)C(C1(CF)CC1)=O N1(C(Cc2ccc(SC)cc2)=O)CCN(C)CC1C(N1CCN(CO)C(=O)C1)=O c1(OCC)cc(C(=O)NC2CCC(CNC(c3ccnnc3)=O)C2)ccn1 Cn1ccnc1CCC(=O)N1CCC1CNC(c1csc(-c2cnc[nH]2)n1)=O c1(SC)[nH]c2ccccc2c1C(=O)NC(=O)CC1CCCN1C(=O)CN(C)C(C)C c1(CN(C)C(C2(C)CCN(C(c3cc[n+]([O-])cc3)=O)CC2)=O)cccc([N+](=O)[O-])c1 N1(C(CNS(CC)(=O)=O)=O)CCC(CNC(c2ncsc2C)=O)C1 C(C)(CCC(=O)NCC1CCN1C(c1c(C(F)(F)F)cnn1C)=O)OCC N1(C(C2CCN(C(C)=O)C2)=O)CCN(C(c2nc(O)nc(O)c2N)=O)CCC1C N1(C(C(C2CCC(=O)N2)C)=O)c2cccn2C(C)CC1(C)C N1(CC(C)NC(c2c(F)cc(OCC)c(OC)c2)C)Cc2ccccc2C1=O C1(C(C)NC(=O)CCCC2CCCCC2)CCCN(C(=O)CSCc2ncc[nH]2)C1 C1(CO)CC2CN(C(C3(NC(=O)CC=C(Cl)Cl)CCCCC3)=O)CC12 c1(C(=O)NC2CC(CNC(c3n(C=C)ncc3)=O)C(O)C2)ccc(C)c(F)c1F N1(C(C(CNC(C)=O)(C)C)=O)CCOCC(CNC(=O)C(O)C2CC2)C1 C(=O)(C1CC(=O)c2ccccc21)NC1C(NC(C2CCN(C(C)=O)CC2)=O)CC1 c1(CC(N2C3CC(NC(c4c(OC)csc4)=O)C(C3)C2)=O)ccc2c(c1)COC2 C1(C(=O)Nc2c(C)c(Cl)ccc2)COC2CN(C(=O)C(C)(N)CN)CC12 C12(CNC(CC(C)C)=O)CC1CN(C(C1CCCN(C(=O)OC(C)(C)C)C1)=O)C2 c1(C(N2C(CCNC(=O)C=C(C)C)CC(OC)C2)=O)c[nH]c2ncccc12 CCC1=NOC(C(=O)N(CCC(=O)N(CC(=O)OC)C)CCCO)C1 CN1CC=CCC1CC(=O)NCC(O)C(=O)NCc1cnns1 C1(C(=O)NC2(CCOCC)CC2)C2CN(C(C3CCC4CC34)=O)CC12 N1(C(C)NC(CC#Cc2cn(C(N3CCCC3)(C)C)nn2)=O)CCc2ccc(F)cc21 c1(OCC(=O)NC(C)C(C)(C)NC(c2cccc(O)n2)=O)ccc(F)nc1 Cc1cncc(F)c1C(=O)NCCCCC(C)NC(C12CCC(C1)C2)=O C(CC(C)(C)CNC(=O)CCOCc1cccc(C)c1)NC(C(CC)SC)=O c1(CC)nnc2cc(NC(C)CCNC(=O)C3=CCCC3)ncn12 Cc1ccc(CC(=O)NC2CC2CNC(=O)C=Cc2nccs2)c(F)c1F c1(CC(N2C(CNC(C(C)CF)=O)C=CC2)=O)ccc(Cl)c(F)c1 c1(OCCCC)ccc(C(N2CCN(C(=O)CC)CC2)=O)cc1 C1(CCCNC(=O)NC(C(OC)OC)C)(NCCCn2cnc(=N)[nH]2)CCOC1 C1(NC(c2cnc(C#N)s2)=O)CN(C(c2cncnc2)=O)CC12CCOCC2 C1(CO)CC2CNC(NC(c3cccc(Cl)c3)Cc3ccccc3F)(C1)C2 N1(C(C(=O)N(C(CCC)C)CCC)=O)CCCC1(C)c1cn[nH]c1 C(CN=c1nc(N(C)Cc2cccc(N)n2)cc[nH]1)c1ccc(OC)cc1 Cc1c(CN(CCCN(C(CC2NC(=O)NC2=O)=O)C)C)cnn1C c1(CC)ncc(C(=O)NC2CCN(C(c3ccc(C#N)n3C)=O)CC2C)c(C)n1 C1(C(=O)NC2CC(NC(C3CCOCC3)=O)C2)CC2(C1)CC2F Cc1[nH]c2ncnc(N3CCCC(c4ncc[nH]4)C3)c2c1C C(=O)(C1=CSCCO1)N1CCC(CC=C)(C(=O)NC(C)C(=O)NCC)C1 C1(CCN(C)C(C2(NC(c3cnn(C)c3)=O)CCSC2)=O)CCCC2CC12 CC(C)CC(C(=O)NCC12CCC(CC1)O2)ONC(=O)CC1CCN(C(N)=O)C1 c1(C(N2CC(NC(C(CCC(=O)OC)C)=O)C2)=O)cc2cccnc2cc1F S(=O)(=O)(c1cc(NC(C2CCC23CCC3)=O)ccc1OC)NC Cc1cc(C(N2CCC2CNC(c2cccnc2F)=O)=O)n(C(C)(C)C)n1 C1(C(N2CC(OCCNC(C(COC)OC)=O)C2)=O)Cc2cccc(F)c2O1 C1(NC(c2noc(C)c2C)=O)C2CCC1N(C(=O)Cc1cccnc1Cl)C2 CC1CN2CCCC2CN1C(C12CCN(C(=O)C3=CCCC(C)(C)C3)CCC1C2)=O C(=O)(CCC(C)NC(=O)OC(C)(C)C)NC(C1(O)CCC1)C CC(F)(F)CC(=O)NCCn1cc(SCCNC(c2occc2Cl)=O)nn1 N1(C(COCCOCC#C)=O)CCC(CNC(=O)C(C)n2cncn2)C12CC2 C1(CNC(c2cscc2C(F)F)=O)CCN(C(=O)C=C(Cl)Cl)CC1 N1(C(CS(CC)(=O)=O)=O)CC(C)CN(C(=O)CC2(O)CCN(C)CC2)CC1C C=CC(CC)C(=O)N1CCCC(Cc2cn(CCN3CCCC3)nn2)C1 C1(CNC(CCCC=C)=O)CN(C(=O)CCCN2CCCCC2)CC(C(F)(F)F)O1 C1(CCC)CN(C(=O)CC(C)(C)CC)CCN1C(=O)CSc1ccc(C)cc1 C1(NC(C2(C)CCNC2=O)=O)CCCCN(C(=O)CNc2cccnc2)C1 c1(OC)ccc(C#N)c(C(N2C3CC2CN(S(=O)(=O)c2cnoc2C)C3)=O)c1 CN1C(=O)CC2CC(NC(C3CCn4nnnc4C3)=O)CCCC12 c1(OC)ccc(Cl)c(CCCNC(=O)COC(c2ccc(Cl)cc2)=O)c1N N1(C(c2cccc(C)c2O)=O)CC(C)N(C(=O)Cc2cnns2)CC1C C=CCCC(F)(F)C(=O)NC1CN(C(c2cccn2C2CCCC2)=O)CC1F CC1CCN(C(=O)CCNC(c2ccccc2F)=O)CC1CO c1(CC)conc1CC(=O)NCCC(C)N(C1CCCCC1)C(=O)COCC(F)F C(=O)(C#CC1CCC1)N1CCC(N(C(=O)Cc2ccccc2F)CCC)C1 c1(C(=O)NC2(CO)CCN(C(CC(CCSC)O)=O)C2)cc2occc2s1 Nc1c(Cl)ccc(F)c1C(=O)NC1CCC(NC(=O)CCC2CCC(=O)N2)C1 c1(NC(C2CC(NC(c3c(CC)cno3)=O)C2)=O)ccn2cnnc2c1 C1(C(=O)NC2(CC(=O)NCC(CCC)OC)CCC2)COCCC1C C1(C)(CC)C=C(C(=O)N2CCCC2C2(C(N3CCCCC3C3CCC3)=O)CC2)C1 N1(C(C(C)c2ccco2)=O)CCC(O)(C2(NC(c3ccnnn3)=O)CC2)CC1 c1(CC(C)NCC2CCC3CC3C2)cccc(Br)c1 c1(C(N2CC(C(=O)Nc3c(C#N)n[nH]c3)NCC2)=O)ccnc(F)c1Cl c1(C(=O)NC2C=CCN(C(c3c(C)cc(F)s3)=O)C2)c2ccccc2nn1C c1(COC)cncc(C(=O)NC(C)CCNC(=O)Cn2ccsc2=N)c1 n1(CC)cc(C(N2CCC(O)(CNC(C3ON=C(C)C3C)=O)C2)=O)c(C)n1 c1(C(=O)NCC2(C)CCN(C(C(CCC)OC)=O)C2)cc2c(F)cc(C)cc2[nH]1 Cc1cc2ccc(C(=O)NC3CN(C(=O)C(C)P(C)(C)=O)CC3F)cn2c1 c1(C2(C(=O)NCC3CCN(C(c4n(CC)ccc4)=O)C3)CC2)ccc(Cl)cc1F CCCC(C(=O)NC1CC2(C1)CC2NC(=O)CC1(CO)CC1)Sc1nc(C)[nH]n1 Cc1nc(N)cnc1C(=O)N(C)CCOCCNC(C1CCCS1)=O O=C1CC(N=c2ccnc(CO)[nH]2)C2CCCCCC12 c1(OC)ccc(Cl)cc1C(F)(F)C(=O)NCC(CNC(=O)CC1CCCO1)CO c1(C(N2CC(CNC(CCCC#C)=O)(OCC)C2)=O)c(C)nn(C)c1SCC C(=O)(CC(C)(C)NC(=O)C=Cc1nccs1)NCc1c(C)cco1 C1(NC(c2ncc(Cl)s2)=O)CC12CCN(C(=O)C(O)Cc1ccccc1)CC2 CCC(C)C(O)C(=O)N1CCC(CO)C1.c1(C2n3cc2nn3)ccccc1Cl Cc1cc2c(C(=O)NCC3CC3NC(c3cc4occc4s3)=O)ccc(C)c2[nH]1 C1(C(=O)NCCC(C(C)C)N(C)C)CCCCC1(C)NC(c1ccc(F)cc1F)=O C1(=CCNC(=O)CC2CCCOC2)CCN(C(=O)COc2ccsc2Cl)CC1 C12(NC(C(N3C(=O)CCC3=O)C)=O)CC(C)(C1)OC21CN(C(=O)C=CCF)C1 c1(CC)cc(C)c(C(=O)N(C)CC2CCCN2C(C2CC2F)=O)s1 c1(C(=O)NCc2c(O)ccc(C)c2)cc(F)c(C)cc1F C1(N(C(C2C(CCC)C2)=O)C)CCC(N(C(=O)C=COCC)CC)CC1 C(=O)(C(C)(CNC(=O)CSC)CC)NCC1CCN(CCC)C1 C1(C(N(C)CC2CCN(C(C(C)=C3CC3)=O)CC2)=O)C2CCC3(COC(=O)C13)O2 N1(C(=O)NCCc2nn(C)c(=O)n2C)CC2CC(OCCN(C)C)CC2C1 C(=O)(CC1=CCN(C)CC1)NC1C(CNC(C(C)NC(CC)=O)=O)CC1 Cc1ccc2c(c1)SC(C(=O)NC1CCC1NC(=O)CC(=O)NCC1CC1)C2 C1(C(N2CCC(F)(CNC(C(C(C)C)N(C)C)=O)C2)=O)CC(S(C)(=O)=O)C1 C1(CC(=O)NC(c2nccs2)(C)C)CC(F)CN1C(=O)CCC1CCC1 CCC(C)(C)C(=O)C(=O)N1CCCC1C(C)(C)C(=O)NCC1CCC(=O)NC1 Cc1cnccc1C(=O)NC1(CNC(=O)CC2C=CCC2)CCCCC1 c1(C(N(CC(=O)NC(CNC(c2ccsc2)=O)CO)C)=O)cc(F)cc([N+](=O)[O-])c1 c1(C(=O)NCCCN(C(c2ccc(NC)nc2)=O)CC)cc2c(s1)CCC(C)C2 C12(C(=O)NCCCC(C)(C)C)CC(CO1)N(C(=O)CC1COCCO1)C2 C(c1cnc(C)s1)=CC(=O)NCC1CCN(C(c2cc(OC)ns2)=O)C1 C12(CNC(c3c(Cl)cn(C)n3)=O)COCCN1C(=O)CN(C(=O)CC1CC1)C2 C1(CCNC(C(C)C2CCC2)=O)CCCN1C(c1csc(CO)n1)=O Cc1cccc2c1CNC(C(N1CCC(c3ccc(C(C)C)cc3)C1)=O)C2 C(=O)(C(CO)C(F)(F)F)N1C(CCNC(c2cc(C)[nH]c2C)=O)CCC1 C1(CNC(C(C)SCCCC)=O)CN(Cc2nscc2C)CCO1 C1(NC(c2c(C)onc2CO)=O)CN(C(=O)Cc2cc(F)cc(F)c2)C(C)(C)C1 c1(OC)nccc(CN(CCCc2ccco2)C(C)C)c1OC(F)F CC(C)(F)C(C)(F)C(=O)N1CCC(O)(CNC(=O)CCSc2cccc(Cl)c2)C1 C12CN(CCC1CO)C(=O)CS2.C1(CC)CCCCO1.C1(=O)CN1.C(=O)C1CC1 c1(C(=O)NC2CCC2C(=O)OCC)ccc(CNC(=O)CC(C)N(C)C)nc1C c1(OC)cc(C)cc(-c2ccc(C(N3CCOC4CC34)=O)cc2F)c1F N1(C(c2ccc(Br)s2)=O)CCC12CCN(Cc1cccc(N3CCCC3)c1)CC2 C1(C)(COC)CC(NC(=O)CCc2cncs2)CN1C(=O)Cn1nnnc1C c1(C(N(CC(CC)NC(C2(CO)CCCC2)=O)C)=O)cnn(CC2CCCO2)c1 C1(CNC(CC2(C)CCCC2)=O)CCN(C(c2ncoc2C2CC2)=O)C12CCC2 N1(C(C(=Cc2ccccc2)C)=O)CCCC(CC(N2CCC(F)(CF)C2)=O)CC1 C1(CNC(C(C)OCc2ccccc2)=O)C2CCCC1N(C(=O)CC(C)F)C2 C1(NC(C(CC2CC2)OC)=O)CC2C(NC(c3cncnc3)=O)C2C1 C(=O)(CCCCN=[N+]=[N-])N(CC(C)(C)CNC(C1CCCC(CC)CC1)=O)CC C(=O)(CC(C)C(F)(F)F)NC(CNC(c1c(O)ncc(CC)c1)=O)(C)C1CCC1 C(CC(=O)N1CCCC(F)(C(=O)NCc2cccc(C)c2F)C1)(C(F)(F)F)OC C1(CNC(C2=C(C)CC2)=O)CC(C(=O)NCc2c(C)cccc2C)=NO1 C(C1CCC(C)CC1)=C(C)C(N1CCC(C)(NC(c2ccc(O)nc2)=O)C1)=O C1(NC(c2cn(CCC)nn2)=O)CC2CCC(C1)N2C(=O)C(c1cccnc1)O N1(C(Cc2c(C(C)C)con2)=O)C2CCC1CN(C(=O)C=Cc1cc[nH]n1)CC2 C(=O)(C1=CCC(C)CC1)NCC1(CO)CCCN(C(c2c(CC)ccs2)=O)C1 C(=O)(C1=CS(=O)CCC1)NCC1C(C)CCN(C(c2cc(C)cc(O)c2)=O)C1 C1(CC)OCCCC1C(=O)NC1CC(NC(c2scc(C)c2OC)=O)C1 C1(O)(CN(C)C(C2(C)CC2C(F)(F)F)=O)CN(C(c2csc(O)n2)=O)C1 N1(C(c2c(CC)con2)=O)CCCC(NC(c2cc(C(F)F)nn2C)=O)C1 c1(CC(N2C(C(=O)NC(C(C)C)CO)CCCC2)=O)cccc(F)c1Cl c1(CC(C)Cn2nc(C3CC3)nc2-c2csc(C(=O)NC)n2)ccc(F)c(F)c1 c1(C(=O)NC(c2cn(C)nn2)C(=O)N(C)Cc2ccn(CC)n2)cc(C)n(C)c1 n1(COCC)nnc(C(N2CC(C(C)NC(=O)COC)C2)=O)c1N C(CCCC(=O)N(CCN1CCCC1)CC)NC(C(CC)n1cncn1)=O c1(C(=O)NC(C)C(C)C(=O)NCC2CC23CCC3)ccc2[nH]ccc2n1 C1(N(C)C)CC2CC(NC(C3CCN3C(C)(C)C)=O)C1C2 c1(C(=O)NCC=CCC(=O)N(C(CSC)C)C)cnnn1C c1(C(=O)NC2CC2CNC(c2c[nH]ccc2=O)=O)cc2ccc(Br)nc2[nH]1 C1(C(N2CCC(NC(CC(C)C)=O)(CO)C2)=O)CC(F)C(=O)N1C c1(OC)ccc(CN2CCCC(C)(C(N3CCOCC(O)C3)=O)C2)c(Cl)n1 C(=O)(CCC(=O)NC1CCCC1NC(C1(C2CC2)CC1)=O)NC Cc1cc(C(=O)NC2CCCCC2NC(c2cc(C)n(C(C)(C)C)n2)=O)c(C)[nH]1 c1(OC)c(C(C)CN(C2CCCNC2)CCF)cccc1F N1(C(C2C(C)(C)CN(C(=O)CC3CCCOCC3)C2)=O)CCC(N=[N+]=[N-])C(O)C1 C12(CNC(c3n(C)cnc3)=O)CC1CN(C(C1(CS(C)(=O)=O)COC1)=O)C2 C1(C(N(CC(C)(O)C2CCCC2)C)=O)COCCN1C(=O)Cc1ccccc1O c1(C(c2n(C(C)(C)C)nnn2)NCC2CCCCC2)ccc(C(C)(F)F)cc1 CC(=O)CC(C)(C)CC(=O)N1CC(CNC(c2cncc(C)c2)=O)CC1C Cn1cc(C(N2CCN(C(=O)C(F)C3CC3)CC2)=O)nc1-c1cccc(Br)c1 c1(C(=O)OCC(=O)NC(=O)C(c2ccc(Cl)s2)=O)cncc2nc[nH]c12 O=C(C1=CCC1)Nc1cn(CCCF)nn1.C12CCN1C(=O)NC2 C(C)(CNC(C1CCCN(C)C1)=O)(CC(C)C)NC(c1c(C)n(CCO)nc1)=O Cc1cc(C(=O)NC(CNC(C2C=CC=CC=C2)=O)C(C)C(C)C)ncc1C#N C(=O)(C(F)(F)CCn1cccn1)N1CC(CN(C)Cc2cccc(Cl)c2)OCC1 Cc1occc(=O)c1OCC(=O)NCc1ccc(CNC(C2CC2CF)=O)cc1 CC1CN(C(=O)C=Cc2ccn(C)c2)CCN1C(c1cc(C2CC2)no1)=O CC1(C)CC(CO)CN(C(=O)C=CCNC(=O)CC2(C)CCOC2)C1 CC(C)C(C)C(C)CC(=O)N1CCCC(NC(c2cc(C(F)F)on2)=O)CC1 N1(C(c2ccc(SC)o2)=O)CCC(C)(C)C(C(=O)NC)C1.C1(CN2CCCC2)CN1 c1(C(c2n(CC)nnn2)NCC2(CO)CC2)cc2ccc(C(=O)OC)cc2o1 N1(C(C2(C(=O)OC(C)(C)C)CCOCC2)=O)CCC(NC(=O)C(C)(C)F)C(F)C1 C1(CC(c2onc(C(=O)OC)n2)OC)CCN(C(=O)Cc2ccoc2C)CC1 c1(OCC)scnc1C(N1CCC1C1C(NC(C2(COC)CC2)=O)C1)=O c1(OC2(C(=O)NCC34CC(NC(C5C(C)C5(F)F)=O)(C3)C4)CC2)cccc(F)c1 N1(C(C2C(OC)C2)=O)CC(O)(CN(C)C(c2conc2OC(C)=O)=O)C1 C1(CCC)CN(C(=O)COC(C)=O)CCN1C(C1(C)COC(C)(C)O1)=O C12(C(N3CCN(C(C4C5CC(=O)CC54)=O)CC3)=O)CCC1CCCN2 C1(C(N2CC(NC(c3cncc(Cl)c3)=O)(CO)C2)=O)C2CC2C2CC12 C1(C(=O)NCc2ccc(-c3ccco3)cc2)Cc2c(F)cccc2O1 C(CO)(C(=O)N1CCCC1CNC(=O)CNC(N)=O)N(C)C C1(C(=O)NC2(CF)CCN(C(C3C(COC)C3)=O)C2)CCS(=O)(=O)C1(C)C C(=O)(CC(C)(O)c1ccccc1)N1CC(O)(CCNC(COCCCC#C)=O)C1 c1(C(c2nnnn2C)NCCC(=O)N(C)C)ccc(-c2ccncc2)s1 C#CC1(C(N2CCC(O)(CNC(=O)Cc3ccno3)C2)=O)CCCC1 Cn1c(C(=O)NC2CC(CCNC(c3cc(CO)ccn3)=O)C2)cc2occc12 N1(C(=O)Nc2ccc(OC(F)F)nc2)Cc2ccccc2C1C(F)(F)F N1(C(C2CCC(C)C2)=O)CCC(C(O)CNC(=O)Cc2cc(C(C)C)no2)CC1 C(=O)(C1=C(Cl)CCOC1)NC1C=CC(CC(=O)NC(C)Cc2cnnn2C)C1 N1(C(C2C3COCC23)=O)CC2CC(C1)N(C(=O)COCCc1cccs1)C2 N1(C(C(C)Oc2ccccc2)=O)CC2C(C1)C2(C)C c1(C(C)=O)cccc(OCC(=O)NC2CC23CC(NC(c2cnnn2C)=O)C3)c1 N1(C(CCNC(C2CCCOC2)C)=O)CCC2CCN(C(=O)OC(C)(C)C)CC12 c1(C(=O)NCC(F)(F)F)cncc(NC(c2cnc(-c3ccco3)s2)=O)c1 C(=O)(C(F)C(F)(F)F)NC1CCC(C(C)NC(c2c(CC)nc(C)s2)=O)C1 N1(C(C(C)c2cccs2)=O)CC2(CCN(CCC3(O)CCCCC3)CC2)CC1C N1(CC=C)CCC(NCCCCOC(C)(C)C)C1=O CCCC(C)(O)C(=O)N1CCC(O)(CNC(=O)C=Cc2cccc(OC)c2)C1 c1(C(=O)NCC(C)(CO)NC(Cc2n(C)nc(C3CC3)c2)=O)ccc(Cl)cc1F C1(NC(c2c(CC)nc[nH]2)=O)CCC(F)(CNC(=O)CCc2cncnc2)C1 CC1C2CCC(C2)C1C(=O)NC(CO)CCC(=O)NCc1ccc(CO)o1 C1(C(C(Cn2ccc(C)n2)C)=O)CCC2CN(c3ncc(I)cn3)CCC2C1 CC1(NC(c2cnc(C3CC3)nc2)=O)CCCN(C(c2ccc(Cl)cn2)=O)C1 CC1(NC(c2nnc(O)cc2O)=O)CCCCC1NC(=O)CN1CC=CC1 Cc1ncnc2c1CC(N=c1cc(C)nc(N3CCOC(c4ccsc4)C3)[nH]1)CC2 c1(C(N(CCCNC(c2cc(C)nn2C)=O)CC)=O)ccc(-n2cncn2)c(C)c1 C1(C(N2CCC(N(CCC(C)C)CCO)CC2)=O)CCC2(CC1)CC2(F)F C1(C(=O)NCCCN(C(CCCc2onc(CCC)n2)=O)C)CCCCN1CC S1(=O)(=O)c2cc(c(Cl)s2)C(=O)N1CCN=[N+]=[N-].C1CC1.CO O=C(CS(=O)(=O)C1CCCC1)NCC1CCCCN1c1ncnc2scnc12 N1(C(C2N(C(CN(C(C)C)C)=O)CCSC2)=O)CCC2=C(CCCC2)C1 C1(C(=O)NC2CN(C(C3(OCC)CC3)=O)CC2OCC)CC2CCC1(O)C2O c1(N(CC(N2CCCC2)=O)C)nccc(=NCC2C(C)C2C)[nH]1 C1(C2CC2)(NC(CCCCC=C)=O)CCN(C(c2cnccc2C)=O)C1 c1(C(=O)NC(CNC(=O)CC2CCOC2)CSC2CC2)cc(O)nc2c1CCCC2 c1(CC)cccnc1C(N1CC(NC(=O)CCOCC(C)C)C2CC12)=O c1(CC)cc(C(=O)NC2CN(C(=O)CNS(=O)(=O)N(C)C)C2)oc1CC c1(C(=O)NCC2(C)N(C(CC3C=NN(C)C3=O)=O)CCC2)cc2cccnn2n1 C(C)(C)(CC(=O)NCCC1CCCCO1)N1CCCC(c2n(C)cnc2)C1 N1(C(c2n(CC)ccn2)=O)CC2CC(C1)N(C(=O)CCC(F)(F)F)C2 c1(OC)cc(S(N)(=O)=O)ccc1NC(N1CC(NC(C)(C)C)C(C)(C)C1)=O N(C(=NCc1cnn(C)c1C)N1CCC(C)(C2CC2)CC1)C(CC)CC C1(NC(C2(c3cc[nH]n3)CC2)=O)CCN(C(C2CCO2)=O)CC1F CC1Cc2cc(F)ccc2C(C)N1Cc1c[nH]nc1Cl C(=O)(C(C)C(=O)OC)NC1(CC(N2CC(OC)C2)=O)CCC1 CC1CC2(CO1)CN(C(C1(N)CCC1)=O)C2.N1(CC(=O)N)CCN(C)CC1 C1(NC(CSCC)=O)CCCC12CCN(C(=O)Cc1ccc(CO)c(C)c1)C2 N1(C(C)=O)CC2CCC1C(NC(=O)Cc1csc(-c3ccccc3)n1)C2 c1(C(=O)NCCN(C(=O)COCCCC(C)C)CC)ccc(C(N)=O)o1 c1(CC)nnc(C)cc1C(=O)NCCCCCCNC(c1n[nH]cc1Cl)=O CCCCCCC(C)(CC)C(=O)NCC1CN(C(=O)C#CC(=O)N(C)C)CC1C C(=O)(C(O)CCC(C)C)N1C(C(N(CC(O)CF)CC)=O)CC(F)(F)C1 C(=O)(CCCCCC(C)(C)C)NC1CN(C(Cc2c(C)nc(S)s2)=O)C1 N1(c2cc(CC)nc(CC)n2)CC2CC(NC(C3(c4cccnc4)CC3)=O)CC2C1 Cc1cc(C(=O)NC2(CCNC(C3C4CC5C(C4=O)C35)=O)CC2)cc(C)n1 C1(CNC(CCC=C=C)=O)CCN(C(C2CCCNC2=O)=O)C1(C)C Cc1oc(C#N)cc1C(=O)N(C)CCN(C)C(c1coc(Cl)n1)=O c1(-c2cn(C(C)C(=O)NCc3cccc(C(C)(F)F)n3)nn2)nnc2n1CCC2 CN1CC(O)CC1CNC(=O)Nc1ccc(Oc2cccc(F)c2)cc1 n1(CC(=C)C)nnnc1C(c1ccns1)NC(C)CC(=O)OCC1CC1 N1(Cc2cc(C)c(F)nc2)CC2CC(CN(C(=O)C(C)CC(C)(C)C)C2)C1 C1(NC(Cc2cn(CC)nc2)=O)CN(C(c2csc(COC)c2)=O)CC12CC2 C1(OC)CN(C(c2cncnc2C2CC2)=O)CC1C(=O)NCC1CCCO1 c1(NC(C2(Cc3cc(C)on3)CC2)=O)ccc2c(c1)CN(C)C(=O)O2 CC1CCC(Cl)=C(C(=O)NC2CC(CNC(=O)CCN(C3CCCCC3)C)C2)C1 c1(NC(CN(C)C(=O)C2CC2)=O)ccc2ncccc2c1.N12C3CCC(C3)C1C2=O O=C(N=c1[nH][nH]c2cccnc12)C1CC12CN(C(c1ccc(F)cc1I)=O)C2 N1(C(=O)NC2(c3cccc(C)n3)CC2)CC2C(=O)CCC2(C)C1 c1(CC)oc(C)cc1C(=O)NCc1cncc(C(=O)NC2CC3(CCC3)C2)c1 CC(C)C(C(C)C)NC(c1ccn(CCNC(=O)C=Cc2nccs2)c1)=O CP(C)(=O)c1cncc(C(=O)NCCC2CN(C(=O)CCc3ccon3)C2)c1 C(C1=CCN(C(C2CN3CCC2CC3)=O)CC1)NC(C1CCCN1C1CC1)=O C1(C(=O)NCC(C)(C)NC(C=C(CCC)C)=O)CCCN1C(=O)OCC C1(CNC(CCCOC)=O)(CO)CC12CCN(C(=O)CN1CC=CC1)CC2 C(=O)(C(C)C(F)(F)F)NC1C(CNC(c2ccc(OCCCC)cc2)=O)CC1 CC(C)C(C(=O)N1CC2C(C1)N2C(C1CN(C2CCC2)C1)=O)C(C)C c1(CC(=O)NC2CN(C(C(C)(C)C3CCC3)=O)C2)ccc(Cl)c(Cl)c1 N1(CC2C(=O)CCC2)CCC(=O)N(Cc2cc(Cl)cc(Br)c2)C1=O C1(CC)CN(C(C2(CNC(=O)C(O)CC3CCCC3)CCCCC2)=O)CC1O n1(C(C)(C)OC)cc(C(N2CCC(NC(=O)Cc3ccno3)C2)=O)cn1 c1(CC(N2CCCCC(NC(CC(C)OC)=O)C2)=O)cn2cc(Cl)ccc2n1 c1(OC)cc2nc(C(C)(C)NCc3nccc4ccccc34)[nH]c2cc1OC C1(C(=O)NC2C(OC)CC2O)CC12CCN(C(C1(C#N)CCOCC1)=O)C2 N1(C(c2c(C)cc[nH]2)=O)CCN(C(c2cn3ccsc3n2)=O)CC1C1CCC1 C(=O)(C(F)C(=O)N(CC(O)CNC(=O)CC1CC2CCC1O2)C)OCC Cc1c(C(=O)NC(C(=O)OC2(C(=O)N(C)C)CCC2)C2CCC2)c[nH]c1C#N C1(CO)CCCCCN(Cc2cc(C(F)(F)F)nc(Cl)n2)C1 c1(C(=O)NCC(CC=C)NC(=O)CC2CCCC2(F)F)c(C)c(C)nn(C)c1=O c1(CC)cc(C(=O)NCC2CCC(C(=O)NOCC(O)CO)C2)n[nH]1 CC#CCCCC(=O)N1CC(NC(=O)CC#CC)C(C#N)C1 C1(C2CN(C(c3ccc(F)cc3Br)=O)C2)(NC(C(C=CCCC)O)=O)CC1 c1(C(N2CCCC(NC(=O)Cc3csc(Cl)c3)C2)=O)nc2ccccc2nc1O CC1(C)OC(=O)NC1C(=O)NCC1(C(F)F)CCN(C(C2CC(F)C(=O)N2)=O)C1 c1(N(C)C)nc(C2CCCN2CC2C3CCCC23)nc2ccccc12 C(=O)(C(=O)N=S(C)(C)=O)NCC(CNC(CCc1ccc(OCC)cc1)=O)CO C(=O)(CCCC(F)(F)F)N(CCCCCNC(C(c1nc(F)ccc1Cl)C)=O)C c1(C(N2CC(CNC(C(C)(C)CC3CCCCC3)=O)C2)=O)cc(N)cc(F)c1 C(C(=O)N1CC2CC2(NC(=O)COc2cccc(F)c2)C1)(C(C)C)SCC Cc1ncc(NC(=O)C(CC(C)C)NC(=O)CN2CCCC2=O)cc1C#N Cc1n[nH]c(C)c1CC(C)C(=O)NCCN(C(=O)CCC1CC1(F)F)C(C)C C1(C(CNC(C2CC3CCC2O3)=O)OC)CCCN(C(c2cc[n+]([O-])cc2)=O)C1 CCC(CCC(=O)NCCCN(CCOC)C(c1cc(OC)n(C)n1)=O)OC N1(C(C2(OC)CC2)=O)CCOC(CCNC(C2CC(=O)N(c3nccs3)C2)=O)C1 C1(NC(C=C(CCC)C)=O)CCN(C(c2ccc(C(=O)OC)[nH]2)=O)CC12CCC2 C(CC(C)(C)CC(=O)N1CC(C)(C)CC1CNC(=O)CCOCC1CC1)OC N12CC3(CN(CCO3)C(=O)c3ccc(cc3)C1)C2.N#Cc1cc(CO)cc(Cl)c1 C(c1ccc(C2CC2)cc1)=CC(=O)NC(C(C)C)(C)CNC(=O)C(F)CC1CC1 c1(C(=O)OC)cc(=NC(=O)C2CC(NCc3nc[nH]c3C(C)(C)C)C2)[nH][nH]1 C1(C(N(C2CCN(C(=O)C(C)(C)c3cnco3)CC2)C)=O)CC(=O)N(C)C1 C(=O)(C(C)CC(N)=O)NC(CNC(C(Cc1ccccc1)NC(C)=O)=O)C1CC1 Cc1ncnc(C)c1C(N1CCN(C(=O)Cc2cnc[nH]2)C(CC(F)(F)F)C1)=O C1(C(=O)NCC2C3CC2N(C(c2ccc[nH]2)=O)C3)CC1C1CCCC1 c1(C(=O)NC(C(C)(C)C)CNC(c2c(F)ccnc2F)=O)ccc2n[nH]cc2n1 c1(C(C)C(N2CC(C(O)C(=O)NC(c3ccnn3C)(C)C)C2)=O)ccncn1 C(=O)(CC(C)C(F)F)NCCCN(C(C(n1c(C)ncc1)C)=O)C CCCCCC(C)(C)C(=O)NCCN1CCN(C(c2cc(CC)ccn2)=O)CC1 N1(C(CC2N(C(c3c(CC)oc(C)c3)=O)CC(O)C2)=O)CCC2(CCCC2)C1 C(=O)(CCC(CF)CF)N(CCC(=O)N(CC#C)C)C(C)C C1(F)(C(=O)NCCCCCNC(c2cc(OC)c(F)cc2)=O)CCC(F)(F)CC1 CC1(C)C(NC(c2cc(Cl)c[nH]2)=O)CCN1C(=O)CC1CCCCC12CC2 C(=O)(C(C)(CO)CC(F)(F)F)NC(C)(C)C1CC1c1cccc(Cl)c1 N1CCN(CCN(C)CCO)CC1.C1(CC(=O)C2CC2C(=O)N)(OC)CC1 N1(C(c2cnc(OC)c(Cl)c2)=O)CC2CCCC1(CNC(c1cnoc1C)=O)C2 Cc1sc(C)c(C(c2nnnn2C2(C)CC2)NCCc2ccnn2C)c1Br c1(NC(=O)CSc2cc(C(=O)NCC(C3CCCCC3)O)[nH]n2)ccccc1O Cc1ccc(S(=O)(=O)NCCCC(=O)N(CCC#N)C2CCC2)cc1 c1(C(N2CC(CNC(c3nncs3)=O)C2)=O)cnc2c(Br)cccn12 CC1CCC(C(C)(O)CN(C(N2CC(c3ccnc(O)c3)C2)=O)C2CC2)CC1 C(=O)(CCC(O)C(C)(C)C)NC(C1(O)CCN(C(=O)CCNC(N)=O)C1)C c1(OC)cc(F)ccc1CNC1CC(NC(=O)Cc2ccccc2C(F)(F)F)C1 C1(C)(CC(=O)N(CCNC(C)=O)C)CCN1C(c1[nH]ccc1C)=O C(=O)(C(F)C(C)(F)F)NCCN(C(=O)Cc1ccco1)CC c1(OC)ccc(C(=O)OC)cc1F.C1C(=O)N1CCCNC(=O)C=C(C)C C(CCC(C)C(=O)NC1CCC(CC(=O)NCC2CC(C)(C)C2)C1)OC C(=O)(CC(C)(O)C(F)(F)F)N(CC(C)NC(COC(CC)C)=O)CC C=CCC(CNC(=O)C(C)NC(=O)OC)NC(c1cnn(CC(=O)OCC)c1)=O c1(C(=O)NC2C(CNC(c3cc(C)c(C(F)F)nc3)=O)C2)cn2cccnc2n1 CCC(CC(=O)NCCN(C(C1(C#N)CC1(C)C)=O)C1CC1)CC(F)(F)F C1(NC(c2nc(C)[nH]n2)=O)CCN(C(c2cc3sccc3[nH]2)=O)CC1C c1(C(=O)NCCN2CCC(NC(=O)CCc3cnco3)CC2)cccc(Cl)c1O c1(C(N(C2CCC2)C)=O)ccc2c(n1)CN(C(C1Cc3ccccc3C1)=O)CC2 C=CCC(C)C(=O)N1CCC(CNC(=O)C(c2ccnc(OC)c2)=O)C1 CCC(C(=O)N1CCCCC1CCNC(c1ncsc1C)=O)C(F)(F)F C1(C(=O)NCC2CC(NC(C34CCOC3CCOC4)=O)C2)CC2CCCCN2C1 CN(C)S(=O)(=O)N1CCCC1c1noc(C2CCC(C(=O)O)C2)n1 O=C1Cc2cc(C(=O)NC3CN(C(c4cc(C5CCC5)[nH]n4)=O)C3)c(Cl)cc2N1 c1(C(N(C(C#C)C)CCCC)=O)ccc2ncc(-c3ccc(OC)nc3)n2c1 C1(NC(C=CC(=O)OCC)=O)CC2CCC(C1)N2C(c1csc(S(C)(=O)=O)c1)=O CC1CCCn2c(C(=O)NC3CC34CC(NC(c3cnccc3Cl)=O)C4)cnc21 Cn1cccc(C(=O)NC(C)(C)CCC(=O)NCC2(C)CCOC2)c1=O N1(C(CCCC(=O)NCC)=O)CCOC2(CCN(C(C3CCOC3C)=O)CC2)C1 CC1(C)CCN(CC(=O)NC(Cc2ccco2)C(=O)NCCC2(O)CCC2)C1 CCCCC(C(=O)OC)N(C)CC1CN(C(c2ccc(C(F)(F)F)nn2)=O)C1 c1(NC2(CO)CCCN(C(CC3C(C)CCCC3)=O)C2)c[n+]([O-])ccc1[N+](=O)[O-] N1(Cc2nnc(C(C)C)o2)Cc2ccc(Cl)cc2C(C)C1 C(=O)(C1=CCCOC1)NC12CC(CNC(C(C=C)OC)=O)(OC1)C2 Cc1cncc(C(=O)NC(C2CCCN2C(C2CCCC2(F)F)=O)C)c1 C12(C(=O)NC3(CC=C)CCN(C(=O)CCCN(C)CC)C3)CCC(C)(CC1)CO2 N1(C(C(C)SCC)=O)CCCC(C2(NC(c3cncc(Cl)c3)=O)CC2)C1 Cc1ccn2nc(C(=O)NC3CCN(C(=O)C4=CCCCCC4)C(C)C3)nc2n1 c1(-c2c(OC)cccc2F)ccc2[nH]nc(C(=O)NCCNC(C)=O)c2c1 N1(C(C#C)C)CCN(C(c2ccc(CNC(=O)C3=COCC3)cn2)=O)CC1 C1(C(=O)NCC2CC(C)N(C(C3(C)CCCN3C)=O)C2)CC2CCC1C21CC1 c1(C(=O)NC2(C)CCN(C(C(C)NC(CC)=O)=O)C2)cc2ncccc2o1 N#Cc1cnc(NCC2CC(NC(C3CC3F)=O)C2)cn1 c1(C(=O)NC(CNC(c2cncc(OC)n2)=O)C2CC2)nn2cccnc2c1Cl C1(NC(C(CC)(C)C)=O)CCN(C(C)=O)CC1F.C12(CCCCC1)C(=O)N2 C1(C(=O)NCC2CC(OC)CN2C(=O)CCN(C)CCO)Cc2ccccc2C1 C(=O)(C(C)(C)CCSC)N(C1CCN(C(=O)CCC=CC(C)C)C1)CC#C C1(COC)(CNC(=O)CC2(C)CC2)CCN(C(C2(O)COC2)=O)CC1 C1(N(C(=O)N)Cc2ccc(C)cc2)CC(C(=O)OC(C)(C)C)C12CC(F)(F)C2 C(=O)(CCC(=O)NCC1CCC1C(=O)NC1(CCO)CCOC1)NCC Cc1ncc(N)cc1C(=O)NC(C(C)NC(=O)Cc1ccc(F)c(F)c1)C(C)C C1(O)(C(=O)NCc2n(CC)ccn2)CCN(C(=O)N(CCO)C2CC2)CC1 CC1(C)CCC(C(N2CCC2CNC(c2cc(CN(C)C)on2)=O)=O)C1 N#Cc1cc(F)ccc1NC(=O)CC1CCCN1C(c1c(Cl)ccc(Br)c1Cl)=O C12C(C)(C)CN(CC1(C)C)C2=O.C12(C(=O)OC)OCCCC1C2(F)F c1(N2CCC(NC(COCc3cc(C)no3)=O)C2)nc2cccc(F)c2o1 C(=O)(C1=CCCC1)NCc1cn(CCOCCNC(CC2NC(=O)OC2)=O)nn1 Cc1oc(C(C)C)nc1C(N1CCC(N(C)C(c2ccnnc2S)=O)C1)=O c1(CC(C)C)cc(C(=O)NCCC(C)NC(=O)CC2COCC2O)n(C)n1 C1(NC(C(=O)N(C)CC2CCCS(=O)(=O)C2)=O)C2Cc3ccccc3C12 C1(NC(CCC=C(C)C)=O)CCOCC1.c1(C(N2CCCC2)=O)cc(C)ncn1 C1(CNC(c2ccc(C)c(CO)c2)=O)COC(C)(C)CN1C(c1cc[nH]c1C)=O c1(CN(C(C(CC2CN(C(C3C(CC)C3)=O)C2)F)=O)CC)ccc(C)nc1 CC1C(CO)CCCN1C(C1(c2ccc(C(F)(F)F)cc2)CC1)=O C(C1COC(C)(C)O1)=CC(=O)NCC(C)NC(=O)CC1CCCC1(F)F c1(CCC)nc(CC(=O)NC2CC2CNC(=O)C(CO)NC(N)=O)cs1 c1(C(N(CCCCCCNC(C2CC(SC)C2)=O)C)=O)cc(S(N)(=O)=O)c(C)o1 N1(C(C(C2CCC2)OCC)=O)CC2CCC(C1)N2C(=O)CC1=CCCCC1 C(=O)(C1=NOCC1)NC(C1CCN(C(c2c[nH]nc2-c2ccoc2)=O)CC1)(C)C CC(C)CC(O)C(=O)NC1COCC1NC(c1cnc(Cl)c(Br)c1)=O c1(C(=O)NCc2ncoc2C2(C)CC2NC(=O)C(F)OC(F)(F)F)ncccc1F N1(C(=O)CC2CC(F)C2)CCC(CCO)(CNC(C2(CO)CCC2)=O)C1 C(=O)(CCC(C)(C)F)NCC(CO)NC(Cc1cc(C)on1)=O N1(C(C(C)(C)C2CCC2)=O)CCC(C)(CNC(C2CCOCO2)=O)C1 N1(C(Cc2cc(C(=O)O)sc2)=O)CC(NC(C2CC2F)=O)CC(O)C1 C1(C(N(OCC(=O)OC)C)=O)CCCN(C(c2ncoc2C)=O)C1 c1(C(N2CCC(CCNC(CC(CCC)O)=O)C2)=O)cc2ccc(C)cn2c1 c1(OC)cc(C(N2CCC(C(C)(O)CNc3nccnc3SC)C2)=O)cc(Cl)c1.OCC Cc1cc(C(=O)NCC2CCN2C(N2CCC(C(C)(C)C)CC2)=O)cnc1Cl C#Cc1ccc(C(=O)N(CC(O)CNC(=O)C(CO)NC(=O)C(F)(F)F)C)cc1 CCCC(C(=O)NC(C)CCCCNC(=O)COCc1ccc(F)cc1)OC CC(c1cnn(C)c1)=CC(=O)NC12CCC1CN(C(=O)COC1CCCC1)C2 N1(C(CC=CC)=O)CC2C(CC(=O)NC(COC)C(=O)OCC)C2C1 C(=O)(C(C(C)C)c1cccnc1)NCC1N(C(c2nc(NC(C)=O)sc2)=O)CC1 c1(COC)cc(C(=O)NCC2CCCN2CCCc2ccccc2Br)ncn1 C(=O)(C#CC1(C)COC1)N1CCC(NC(c2ncc(C)o2)=O)C1(C)C Cc1cccc(C(F)(F)CNC(COC2CCCC2)C(=O)O)n1 C(=O)(CCC(=O)NC1CCCC(CNC(=O)CCCF)C1)N(C)C C123CCC(CC1)(OC2)CNC3=O.c1(OC(C)C(=O)Nc2ccsn2)cccnc1 C1(C(N2CCN(C(C)C)CC2)C(=O)NCCC)CC2(CC(OC)C2)C1 CON(CCC(=O)NC)C(=O)c1cc(C2CCOC2)[nH]n1 c1(C(N(CC(C)NC(=O)CC(C)c2ccco2)CC)=O)ncc(F)cc1F Cc1cc(C(N2CCCC(O)(CNS(=O)(=O)c3cnoc3C)C2)=O)c(F)cc1Br c1(C(=O)NCC(CN(C(C(CC)C(C)C)=O)C)C)cc(Br)n2ccccc12 CCC(C)(C)C(C)CC(=O)NCC1(CCNC(=O)C(C)CN2CCOCC2)CC1 C1(C(=O)NC(CCCNC(c2c(C)c(C3CC3)on2)=O)C)CCC(N=[N+]=[N-])C1 c1(C(=O)NCC2CCC(NC(Cc3nc(C)oc3)=O)C2)ccc(N(C)C)cc1Cl c1(OC)ccc(C(=O)NCCC2CCCCN2c2ncnc(=N)[nH]2)cc1 c1(C(C)=O)cc(C(=O)NC2(CNC(=O)C3=CCCO3)CCCCC2C)ccc1F N1(C(C(c2ccc(C)cc2)C)=O)CC2OCC(CNC(C3(C)CCCC3)=O)C2C1 C1(CC)OCCC1C(=O)NC(C)(CNC(c1cc(O)cs1)=O)C1CC1 CCC(C)(O)C(=O)NC(CNC(c1ccsc1OC)=O)CO N1(C(C(C=C)(C)O)=O)CC(CC(=O)NCCc2ccns2)CC1(C)C CC1(C)CCN(C(=O)C(CC2CC2)NC(c2cccn2C2CC2)=O)CC1CO c1(OCC)cc2c(cc1C(=O)NCc1cn(CC(=O)OC)nn1)OCCO2 C1(NC(C2CC(SC)C2)=O)CN(C(=O)CCc2cnc(C)s2)CCC12CCC2 C1(N(C(=O)CC(F)F)C)CCCN(C(C2CC(F)(CO)C2)=O)CC1 N1(C(c2ccn(C(C)C)c2)C(=O)NCCOC)CCCC2CCC(C)CC12 N1(C(CC2CC(OC)C2)=O)CCCC(CC(N2CCC(C(C)C)(OC)C2)=O)CC1 CCC(C)(C)C(=O)C(=O)NCC(F)(C(=O)N1CC2C(CO)C2C1)C(C)C c1(C(=O)NCCC(C)(C)NC(Cc2cc(C)c(Cl)cc2)=O)cc([N+](=O)[O-])ccn1 C1(NC(C2(N(C)C)CCC2)=O)CN(C(=O)CC(=O)NC2CC2)CC1(C)C CC1(C)CC(NC(c2nc(Cl)ccc2Cl)=O)CCN(C(C2CCC(F)C2)=O)C1 c1(N2CCC(CNC(C3CCN(C)C(=O)C3)=O)C23CC3)ncnc2c1nnn2C c1(C(=O)OCCC(C)=CC(=O)NC2CCC2CNC(=O)C=CC2CC2)ccccc1 C1(F)(CNC(CC)=O)CCCN(C(C2CCCCC23CC3)=O)C1.C1C(=O)N1 C1(C(=O)NC2CCN(C(=O)CC3(NC(C)=O)CC3)CC2)(OC)CCC(C)(C)CC1 N1(C(c2c(C)nc(C)[nH]2)=O)CCC2(CC1)OCCC2NC(=O)CSC(F)F CC(C)C(C)C(CNC(C1CCCC2CC12)=O)N=c1[nH]c(Cl)ncc1C(N)=O C(CC(C(=O)NC(C)C(=O)OC)NC(C1CCC1(OC)OC)=O)=CC C1(C(=O)NC(C2CCOCC2)C#C)CCN(C(=O)CC2CCOCC2)O1 C1(CNC(CC)=O)CCN(C(C2CCCCC2(C)C)=O)C12CC2 C(c1ccccc1Cl)=C(C)C(=O)N1CC(NC(C2(C)CC2C)=O)C1 N1(C(CN(C(C)=O)C)=O)CCCC(NC(=O)CCCC(C)C)C(F)C1 Cc1ccc(C)n1CC(=O)N(C(c1ccc(Cl)cc1)CF)C c1(C(N(C(C)CNC(=O)CCc2nncs2)C)=O)ncc(C#N)cc1Cl C(=O)(C1=C(Cl)CCCC1)NC(C(C)(C)NC(Cc1ccc(C)cc1Cl)=O)C C1(C(C)NC(CC(=O)OCC)=O)CN(C(C2C=C2C)=O)CCO1 c1(OC)cc(C(=O)NCCOCCN(C)C(c2cc([N+](=O)[O-])n[nH]2)=O)cc(C)c1 C1(C)(NC(C=C2CCC(C)CC2)=O)CCCN(c2nnnn2C)C1 N1(C(CC(COC)NC(C2(C)CCCN2C)=O)=O)CC(C)C(C)C1C C1(CNC(CCCN(C2CCCC2)C)=O)CC(NC(=O)COC(F)F)CCO1 n1(CCC(N2CCCC2CCNC(C23CC(F)C2C3)=O)=O)cc(Cl)cn1 C1(C(=O)Nc2ncc(C)cc2Cl)CCCC12CCN(C(c1sc(Cl)nc1C)=O)C2 C1(C)(CNC(C2N(S(CC)(=O)=O)CCC2)=O)CC(F)(F)CN1C(c1sccc1C)=O C1(CC(=O)NCCC(C)F)CCN(C(=O)Cc2ccc(C(=O)O)cc2)CC1 N1(C(c2ccc(SC)cc2)=O)CC(CNC(=O)C(O)CC2CCCC2)C(C)(C)C1 c1(C(N2CCC(NC(C=CC(N)=O)=O)C23CCC3)=O)ccc2c(c1)NC(=O)NC2 Cc1cc(C)nc(NC(C(C)NC(C2CC3CCCC23)=O)C(C)C)n1 c1(C(N2CC(C)C(CNC(c3cc[nH]n3)=O)CC2)=O)ccc(O)c(F)c1F c1(C(N2CCCC(NC(=O)CCC(N)=O)CC2)C)ccc(Cl)c(Cl)c1 C(=O)(C#CC1CCCCC1)NC1(C(=O)NCC(C(C)O)C)CCC1 Cn1cc(C(=O)NC(C)(C)C(=O)NCC(F)CNC(=O)C(F)=CCCF)cn1 c1(CC(N2CCN(C(CSCC(C)C)=O)CC2)=O)cc(F)cc(F)c1 N1(C(c2ccc(C(C)C)cc2)=O)CC2ON=C(CNC(=O)C(F)=CC3CC3)C2C1 C1(C)(CCNC(CN(C(C)=O)C)=O)CN(C(=O)C(O)CC(F)(F)F)C(C)(C)C1 C(CCN=C(NCC(c1ccc(C#N)cc1)C(F)(F)F)NCCCCl)SC C(=O)(C(N)CC(F)(F)F)N(C1CCCCNC1)CC Nc1ccnn1CC(=O)NC1(CNC(=O)CC2CCCO2)CCOC1 CN1CC2(CCN(C(c3ccc(C(F)(F)F)cc3)=O)C2)Oc2ccccc21 Cc1nc(C)n(CC(=O)NC(Cc2cc[nH]n2)C(=O)NCC(C)(C)CCO)n1 C(=O)(C1=CC2CC=CCC12)N(C(CCN(C(c1c(C)[nH]c(C)c1C)=O)C)=O)C(C)C N1(C(c2c(C)scc2)=O)CCC(CNC(C2(C(F)(F)F)CC2)=O)C(O)C1 N1(C(C(N2CCC(C)CC2)=O)=O)CCC2(CCCC2C(=O)Nc2cnc(O)[nH]2)C1 N1(C(CC=C)=O)CC2CC2(C(=O)NC2CC(F)(CO)C2)C1 c1(C(=O)NC(CNC(C2(CC=C)CCOC2)=O)CC(C)C)ccc2c(c1)CCO2 C1(C(=O)NCC2(CCC=C)CC2)CC(O)CN1C(=O)C(C)N1CC(C)C1 N1(C(=O)OC)CC2C=CC1C(C(=O)NCCN(C)C(c1c(C)ncn1OC)=O)C2 c1(OC)cc(Br)cnc1C(=O)NC1CCCCC1CNc1nccc(C2CC2)n1 c1(OC)ccc(I)c(C(=O)NCCCCCCn2cc(CCCC(C)O)nn2)c1 CCC(C)CC(C(=O)NOCCc1ccccn1)NC(=O)C(C)SC N1(C(C(CCC)OC)=O)CC2CCC2(CC(=O)Nc2ccc(F)cc2)C1 N1(C(COCCOC)=O)CCN(C(C2CC23CC(F)(F)C3)=O)C2(CCC2)C1 C(=O)(CC(CC)CC(C)C)NC(CC#C)(C)C(=O)N1CC(=O)NC(CC)C1 c1(CC(NOCC(=O)OCC)=O)cc(Cl)sc1Cl c1(OC)ccc(C(=O)NCC2CN(C(=O)CC3(O)CC3)CC2(C)C)c(Cl)n1 C1(C#CC(=O)NC(C(=O)N2CCCCCC2)C(C)(C)C)(CC)CC1 C(=O)(CCCCNC(N)=O)N(C1CN(C(=O)CC#N)C1)C.n12nccc1C(=O)N2 c1(C(C(=O)NC(C(C)NC(c2cn(C3CCC3)nn2)=O)C)F)ccc(F)cc1 Cc1cc(C(=O)NCC(C)(CO)NC(c2c(F)cccc2F)=O)cc([N+](=O)[O-])c1 C1(C)(NC(CCOCCOC)=O)CCCC1CC.C12CCC1CNC2=O N1(C(Cc2cc(C)no2)=O)CCn2nc(COCC3CCC3)nc2C1 N1(C(c2cc(C)[nH]c2)=O)CC(C(=O)N(C)Cc2c(C)cnn2C)CCC1(C)C N1(C(C2C(=C)CC2)=O)CCCC(NC(C2(O)COC2)=O)C1C N1(C(c2c(C)nco2)=O)CC2CC(NC(c3ocnc3C(F)(F)F)=O)C(C2)C1 C(CC(F)F)(C(=O)N(C)CC1(C#N)CC1)N(C(C(c1ccn(C)c1)C)=O)C c1(CSC)ccccc1C(N1CCC(N(C(C2CC(C)OC2=O)=O)SCC)C1)=O c1(NC(CCCCOC)c2nnnn2C)cc(Br)cc(S(N)(=O)=O)c1C c1(C(N2C(CNC(C3=CC(C)CC3)=O)COCC2)=O)cc(F)cc2nn(C)cc12 Cc1ncc(N)cc1C(=O)NCC(C1CCCC1)NC(c1ccco1)=O CCCCC(C(=O)OCC)NC(c1ccc(C2CCC(=O)N2)cc1)=O Cc1cccc(F)c1CC(=O)NCC(O)CNC(c1[nH]c(C)c(C(N)=O)c1C)=O N#Cc1cccc(NC(C2C3CN(C(C4CCC(=O)NC4)=O)CC23)=O)n1 c1(NC(CSCC(N2C(C)C(C)SC2)=O)=O)ccc(F)cc1Cl N1(C(C(C)N(C(=O)C=Cc2cncn2C)CC)=O)CCC2(C=CCO2)CC1 C1(NC(=O)CC23COCC(C2)C3)CS(=O)(=O)CC1NC(c1cc([N+](=O)[O-])c[nH]1)=O CC(C)(C)CCC(F)C(=O)NCCC(CN=c1ccc(C2CC2)n[nH]1)C(F)(F)F C12(CC(=O)NC3C(CNC(CSCC#C)=O)CC3)CC3CC(CC(C3)C1)C2 C(C(O)CNC(=O)CNC(=O)C1CC1)N(C(=O)Cc1ncco1)C.C(=O)C1CC1 Cc1nc(-c2cn(CC3CCN3C(=O)CC3CCC(O)C3)nn2)sc1C Cc1nc(C(=O)NCC(F)CNC(=O)CCn2cccnc2=O)c2ccnc-2[nH]1 c1(C(=O)NC(CN(C(c2c(C)ncs2)=O)C)C)cncc2sccc12 C(=O)(CC(C)(C)C)N(CCCOCCNC(c1coc(CO)c1)=O)C C(=O)(C1=CCCCCC1)N1CC(NC(c2ccc(CF)cc2)=O)CC(C)C1 c1(C(N2CCC3(CC2)OCCO3)=O)csc2c1CCN(Cc1cccc(F)n1)C2 Cc1ccccc1C1CCN(C(c2ccc(OC(F)F)cn2)C(=O)NC2(C)CC2)C1 C1(C)(COC)CC(NC(C2(C)CC3(CCC3)C2)=O)CN1C(=O)CCCCCSC C(C)(C)(CCCNC(=O)CCc1ccn(C)c1)NC(CC1CCC(C)C1)=O c1(CN2CC(CC(=O)Nc3cccc(C(C)(C)C)c3F)C2)nsc2ccccc12 C1(CC#C)(C(N2CCC(CC=C)(NC(=O)C(O)c3ccco3)C2)=O)CCCCC1 c1(CCC(=O)NC(CN(C)C(C2CC3CCC2C3)=O)(C)C)ccccc1Cl CS(=O)c1ccc(C(N2CCN(C(=O)Cn3cnc([N+](=O)[O-])c3)CC2)=O)cc1 c1(C(N2C3CC(NC(C=CC(=O)N(C)C)=O)C(C3)C2)=O)c(F)cc(O)cc1F c1(C(=O)NCC2C(C)CCN2C(C2CC(O)C2)=O)ccc(N2CCOCC2)c(F)c1 c1(C(=O)NCC2N(C(COc3cc(C)on3)=O)CC(F)C2)cc2ccc(F)cc2o1 c1(C(=O)NC2(CCCNC(C(C=C=C)C)=O)CC2)ccc(F)c(C)c1 c1(C(=O)NCC(CC(C)C)CO)n[nH]c2c1CN(C(=O)Cn1cccc1)C2 C(C)(C(C(=O)NCC(c1cnn(C)c1)O)NC(c1csc(Cl)c1)=O)OC C(=O)(C1=CCc2ccccc21)NC(CC)CNC(=O)C(c1cccc(C)c1)F C1(CC)CCCCC1C(=O)NCC(C1CCN(C(C2(O)CCCC2)=O)CC1)C CS(=O)C=CC(=O)NCCC1CCN(C(C23CCC2C3)=O)CC1 Cn1cc([N+](=O)[O-])c(C(N2CC(F)(CNC(=O)CCc3ccc(F)nc3)C2)=O)n1 CCS(=O)(=O)CC(=O)N1CCCCC1CN(C(c1cn(C)nc1Cl)=O)C1CC1 C1(CCC)CCC(O)(C(=O)NC2CC(N(C(=O)Cc3cnn(C)c3)C)C2)CC1 c1(C(=O)NCC#CCNC(c2ncc[nH]c2=O)=O)[nH]cc2c1CCS2(=O)=O c1(NC(C2C(C)S(=O)(=O)CC2)=O)ccc(F)c2ccccc12 C#Cc1cc(NC(=O)CCOC2CN(C(=O)C(C)C)C2)cc(F)c1 N1(CCC)CCCC1C(=O)NC(C1CN(C(c2ccc(C(F)(F)F)o2)=O)C1)C c12ccc(Cl)c(c1)N2C1CC1.C1(c2n(CC=C)nnn2)(OC)CN2CCC1C2 C(CC(F)F)(C(=O)NCC1Cc2nccn2C1)N(C(=O)CSC(F)F)C c1(CCC(=O)N(C2CCCCC2)CCN2CCCOC2)ccccc1C(F)(F)F c1(C(C2CCCC2)(C)NCC2(C(C)(F)F)CCC2)csc(C(F)F)n1 CN1C(=O)C(C)(C)N(CC(=O)NC2CCOC(C(C)(C)C)C2)C1=O C1(O)(CNC(CCNC(COC(CC)(C)C)=O)=O)CCN(C)C1 c1(C(N2CC(CNC(C=CCCC)=O)C(C)C2)=O)cc(C)sc1S(N)(=O)=O N1(C(c2ccc(C)o2)=O)CCCCC1CC(=O)NCCc1[nH]cnc1C c1(OCC)ncccc1NC(=O)C(C)NC(=O)C(CC1CC1)OC N1(C(Cc2ccc(OC(C)C)cc2)=O)CC(NC(=O)CCF)CC12CCCOC2 c1(C(=O)NC(CCNC(C2(CC)CC2(F)F)=O)C)nnc2ccccc2n1 N1(C(C2(COC)CC2)=O)CC2(C1)CN(C(c1cc(C(F)F)n(C)n1)=O)C2 C1(C(N(C(C)C)CCN(C)C(C23CC(C)(C2)C3)=O)=O)OCCN(C)C1=O c1(N(C)C)cc(C(=O)N(C2CN(C(=O)C(C)(C)OC(C)(C)C)CC2F)C)ccn1 C1(C)(OC)CN(C(=O)CSC(C)C)C1.c12cn(nn1)CCNC2=O c1(C(N(CC(C)NC(C2(C)CC3CCC2O3)=O)C)=O)cn(C)c(=O)nc1O CCC(C)C(O)C(=O)N1CC(C(N)=O)(CNC(C2CCN(C)S2(=O)=O)=O)C1 C1(N(CC(C)C)C(=O)OC(C)(C)C)CCCN(C(=O)CCC2CCCN(C)C2)C1 CC1CN(C2CC(=O)N(c3ccc4cccnc4c3)C2=O)CCS(=O)(=O)C1 c1(C(=O)NC(CNC(CCC(C)SC)=O)C(C)C)cccc2c1ccn2C C(CCCC(=O)NC1(CC2CC2)CC1)(c1nnnn1CCCF)NC(CC)=O CCC(CC)C(F)C(=O)N1CC(C)N(C(C2CCC(C(N)=O)C2)=O)CC1C c1(NC(CC(C)C)=O)cc2ccccc2cc1C(N1CCC(N)C1C)=O Cc1ccc(C(=O)NC(C)CC2CN(C(=O)CSCc3cscn3)C2)nc1F c1(C2N(Cc3c(COC)ocn3)CCC2)cccc([N+](=O)[O-])c1 c1(C(N2CCN(C(c3cc(OC)c(C)cc3)=O)C(C)C2)=O)cccc2nc[nH]c12 C1(CNC(CC(=C)Br)=O)CC2(CCC2)CN1C(c1cc(C)n(C2CC2)n1)=O C1(CCC(=O)N(CCCCN(C(C(C)NC(CC)=O)=O)C)C)CCC(=O)C1 CC(C(=O)NCC1CCN1C(=O)Cn1ccnn1)c1ccsc1 c1(CCC(=O)NC(c2ccccc2C(F)(F)F)CO)cccc2cnccc12 Cc1csc2ncnc(NCCCCNC(c3cc4c(s3)CCCC4)=O)c12 C12(NC(C3(NC(=O)CCN(C)CCO)C(C)C3)=O)CCC(CC1)OC2 n1(CC(=O)NCC(CC=C)NC(=O)CC2CN3CCC2CC3)cc([N+](=O)[O-])cn1 C1(C(=O)NC2CC(F)(CNC(=O)CN3C(=O)CCC3=O)C2)CC2CCC1CC2 CC(C)C(C)C(C)CC(=O)N1CCOCC(NC(=O)CCCCn2ccnn2)C1 Cc1c(C(N2CCCC(CO)(NC(=O)C#CC3CC3)C2)=O)nn2ccccc12 C(C(CNC(c1ncccc1O)=O)C(F)(F)F)NC(c1c(C(C)C)noc1)=O N1(C(=O)Nc2cc(Br)c(C)s2)CC(OCC(n2cnc(C)n2)c2ccccc2)C(C#N)C1 C1(CC=C)(NC(c2cncc(Cl)c2Cl)=O)CCN(C(=O)C(F)=C(C)C2CC2)CC1 c1(C(=O)NCC(O)C(=O)NCCC2CCCCCC2)ccc2nsnc2c1 N1(C(c2c[nH]ccc2=O)C(=O)N)CCCC(C)(C)C1C.CC1CC1 C(C(=O)N1CCC(C(=O)NCc2c(C)noc2C)O1)c1ccc(C)o1 C1(SC)CCCC1C(=O)N(C)CCN(C(=O)Cn1cc(C(C)O)nn1)C C=CC(CCC)CC(=O)NC(C(N(C)C[Si](C)(C)C)=O)C1CCCC1 C(CNC(=O)CC1CCN1C(=O)C=CC(=O)N(C)C)(CO)OC c1(N(C)C)ccc(C(=O)NC2CCCC2CNC(C2CC(C)(C)C2)=O)cc1 CN1CCCCC(C(N2CC3CN(C(c4cc[nH]n4)=O)CCC23)=O)C1=O C(C1CCN(C(=O)C(C)c2ccco2)CC1)=CC(=O)N(c1ccn(C)n1)CC N1(C(C2CCC(CC)CC2)=O)CC2CC(NC(C3(c4cnn(C)c4)CC3)=O)C2C1 C=C1CC(C(=O)NC2CNCC2)(C(F)F)C1.c1(C2(C(=O)OC)CC2)cccs1 c1(CCCC)cc(C(N2CC(NC(c3c(C)nnn3CC)=O)C(C)C2)=O)c(C)o1 N1(C(C2CC(O)(CC#C)C2)=O)CCC(CCOC)(NC(=O)CC(C)C(C)C)CC1 C#CC1CCCN(C(=O)CCOC(c2cc(N3CCC(O)CC3)ccn2)=O)C1 C12(CNC(c3ccc(NC)cn3)=O)CCC(CC1)CN2C(=O)CC1CCCOC1 c1(C(=O)NC2C3(CC(NC(CC(C)CF)=O)C3)C2)cccc(C=C(F)F)c1 C(C)(CN=c1[nH]c(C2CC2)nc(=N)[nH]1)(C(F)(F)F)NC(C=CC=CC=C)=O C(=O)(C1=NNC(=O)C1)N1CC(COC)(NC(=O)Cc2cccnc2)C1 C1(CC=C)(NC(C2(CF)CCC2)=O)CCN(C(=O)CN2CCNC2=O)C1 N1(C(CCC(C)(C)F)=O)CC2C=CC1C(C(N1CCC(C)(C#N)C1)=O)C2 c1(C(=O)NCC(CCOC)NC(C2CC3(CSC3)C2)=O)cccc2sncc12 n1(CC(=O)N(C(c2c(OC)cccc2)C)C)c(=O)oc2ccccc12 C1(NC(c2ccc(Cl)o2)=O)CCN(C(=O)CC(C2CC2)C2CC2)C(C2CC2)C1 C1(CC=C)(C(=O)Nc2cnc(C)nc2)CCCN1C(=O)C(C)CC#N N1(C(c2cn(CC)nc2)=O)CC2CC(C1)N(C(=O)CCC(C)NC(C)=O)C2 C1(NC2(C)CN(C(c3ccc(CONC(CSC)=O)[nH]3)=O)C2)CCCC1(F)F CS(=O)(=O)CCCCN=c1[nH]c(=NCCN2CCCC2CO)c2sccc2[nH]1 CCC(C(=O)NCCN(C1CCCCC1)C(c1nscc1Br)=O)OC N1(C(C2N(C(CN(CC(C)(C)C)C)=O)CC(=O)NC2)=O)CCC(C)(C#N)CC1 C1(NC(C2C(C)C2)=O)COC2(CNC(=O)CCC(=O)c3ccccc3N)CC1C2 C(C(C)(C)C(=O)N(C1CCCC1)C)NC(C(CC)SC)=O C(N=c1[nH]c2c(c(=NCc3nc(C(F)(F)F)cs3)[nH]1)SCC2)C1C(C)(C)OCC1 Cc1cc2[nH]c(C(N3CC(NC(C4CCCO4)=O)C4(CC4)C3)=O)cc2s1 CCCCC(O)C(=O)NCC(C)(CC)NC(c1cccc(-c2nccs2)c1)=O c1(N(C(C(C2CCN(C(c3cccc(Cl)c3)=O)CC2)C)=O)C)ccccc1C(F)F N1(C=O)CC2CC1CC2NC(C1CC(NC(COC)=O)C1)=O C(=O)(C(O)C(O)C(C)C)NCC(CC)Oc1ccc(C(C)(C)C)cc1.C1CCCCC1 c1(NCC(C)C)ncccc1S(=O)(=O)N(C1CCCCC1)C(C)CN1CCCC1 C123CC1CC1CN(C2)C(=O)CC(CCC(=O)NC)C(=NC=CN=C1C)C(=O)N3 CN1CCC2(CCCN(C(C3CCC4(CC3)CSC4)=O)C2)C1=O CC1CCC=C1C(=O)N1CC(CNC(c2ccc(F)cc2F)=O)C(O)C1 C1(C2CCCCC2)(C(=O)NC2CC(CCNC(c3c(C)nc(CO)s3)=O)C2)CC1 CC1CCCN(CCNC(=O)NCc2nc(C(=O)OC)cs2)C1 Cc1nn(-c2ccccc2)cc1C(N1CC(N(C(=O)C(C)N(C)C)C)C(O)C1)=O N1(C(c2nccc(CC)c2)=O)CCC(C)N(C(=O)C(c2cncnc2)C)CC1 CCC(C)(C(=O)N1C2CCC1C(CNC(c1ccnc(CO)c1)=O)C2)C(F)F C1(NC(COCC)=O)CC(F)CN(C(=O)CNC(c2ccoc2)=O)C1 N1(C(C23N(C(C4(OC)CCOC4)=O)CC(C2)C3)=O)CCN2C(=O)NCC2C1 Cn1nc(C(=O)NCc2cc(O)nc(CNC(C3CC(C)(O)C3)=O)n2)ccc1=O C1(NC(C(CC)CO)=O)CCC2CCN(C(=O)C(c3ccc(F)cc3)=O)C1C2 N1(C(Cc2c(C)cco2)=O)CCN(C)C(CNC(=O)CC2CC3(CC3)C2)C1 C1(NC(C(C)c2cccs2)=O)CC2CC(NC(C3(C#N)CCOCC3)=O)CC2C1 CCC(C)(C)C(=O)C(=O)N(CCCOCCC(N1CCC(c2ccco2)C1)=O)CC CC1Cc2cc(S(=O)(=O)NCCCC#N)ccc2O1 Cc1cnc(C(=O)NCC2CC2CNC(C2(CCO)CC2)=O)nc1 [N-]=[N+]=NC1COCC1NC(C12CC(CN(C(=O)CC3CCC3)C1)C2)=O C1(C2N(C(CCN(C(CSC)=O)C)=O)CCC2)CCN(C(C23CC(CO2)C3)=O)CC1 C1(n2nnnc2C)=C2CN(C1=O)C2.c1ncc(C#N)o1.CC=C N1(C(COC)=O)C2CCC(C(=O)NCC3(N4CCNC4=O)CC3)C1CC2 CC(C)C1=NOC(C(=O)NC(CCN(C)C)C(=O)NC2C(C)OCC2C)C1 C1(NC(C2CN(CCC)C(=O)C2)=O)CN(C(=O)C(F)=CC2CC2)CC12CCC2 S(=O)(=O)(c1c[nH]c(=NCCOC)cc1C)N1CCC(CN(CC)CC)C1(C)C N1(C(C)C)CCC(C(=O)NCC2CCC2NC(=O)CC2C=NN(C)C2=O)CC1 C1(OCCNC(C2(CCOC)CCC2)=O)CCN(C(=O)CC2CC2(C)C)C1 C1(F)(CC(=O)NC2CON(CC)C2=O)CCN(C(C2(CC)CCCO2)=O)CC1 N1(C(C2C(=C)CC2)=O)CC(C)OC2(CCN(C(C3CC(C)(C)C3)=O)CC2)C1 c1(COC)ccncc1NC(C1CC(O)(CNC(C2CCCCS2)=O)C1)=O C1(CNC(C(CCOC)C)=O)CC2COCC2N1C(c1ccc(CF)cc1)=O C(=O)(C(C)(F)C(C)(C)F)N1CC(C)C(C(N2CCC3(CC2)CC3)=O)C1 c1(CC)ncsc1C(=O)NCC1(NC(=O)C(CC2CCC2)OC)CCCC1 N#CC1=C(C(=O)NCCCNC(C2(C(F)(F)F)CCCCC2)=O)CCC1 N1(C(C2C=CC(NC(C(C)OCCN(C)C)=O)C2)=O)CC=CC(O)C1 N1(C(CC2C=NN(C)C2=O)=O)CC(CO)C2(C1)CN(C(C1(C)CS(=O)(=O)C1)=O)C2 N1(C(=O)Cc2ccc(F)cn2)CC2OCCN(C(C3CC4CCC3C4)=O)C2C1 N1(C(CC(C)(C)O)=O)CC2CCOCC2(NC(C2C=CC=CC=C2)=O)C1 C#CCCCC(C)C(=O)NCCCNC(c1ccc(Br)s1)=O N1(C(C(C(CC)O)(F)F)=O)CCC2CN(C(=O)C(C)(C)CC(F)F)CC2C1 CCC(O)CC(=O)N1CC(=O)CC1C(N1CCC(F)CC1)=O C1(CNC(CCC2C(C)C2)=O)CN(C(=O)CSCC#N)CCC1(F)F N1(C(CCC(=O)OCC)=O)CCOC2(C1)CN(C(=O)C(c1cnn(C)c1)O)C2 C(CC1=CCN(CC(=O)OC2CCCCC2)CC1)NC(=O)OC C(=O)(N=c1nc(-c2ccccn2)[nH][nH]1)NC1C(C(=O)OC)C(O)C1 c1(C(=O)NCC2CN(C(C3CCCC(F)C3)=O)CCO2)cnc2cccnn12 C(=O)(C1=CNC2=NCCC2=C1)NCC(CC=C)NC(c1cnc(C2CC2)s1)=O c12nn(c(=O)o1)CC2.c1(CC=C)nc(-c2ccc(Cl)nc2)nn1CCS(N)(=O)=O C1(NC(c2nccc(COC)c2)=O)CC2CC(C1)N(C(C1(C)CCOCC1)=O)C2 N1(CCCNC(C(C)n2cncn2)=O)CCN(C(=O)CC2CCC(O)C2)CC1 N1(C(CCCN(C(C)C)C)=O)CC2CC(CNC(C3CCC(C)(F)CC3)=O)C2C1 c1(C(=O)NC2C(NC(CC3(C=C)CCC3)=O)CCC2)occ2c1CCOC2 c1(CCC)nc(C(=O)NC23CC(NC(C4CC4c4ccccn4)=O)(C2)C3)co1 c1(CN(C(c2c(OC)ccc(Cl)c2)=O)C)ccc(S(=O)(=O)NC2CNC2)cc1 C(c1ccccc1)=CC(C(=O)OC)NC(c1ccncc1Oc1cccnc1)=O CC12CCC(C(=O)NC(C(=O)OC)C3CC3)(CO1)C2.C12CCCCC1CC(=O)N2 N1(C(C(CC)CC(F)F)=O)CCC2CCN(C(=O)CCC3CCCO3)CC2C1 C1(=CC(=O)N(CCCCN(C(=O)C(F)C2CCOC2)C)C)CCSCC1 c1(C(N2CC(O)(CNC(C3C(C)(COC)C3)=O)C2)=O)cccn2[nH]c(=N)nc12 Cc1c(C(=O)NCC(C)(C2CC2)NC(=O)Cn2cnc(=N)[nH]2)cnn1C1CC1 CCCCC(O)CC(=O)NCC1C2CN(C(c3ccc(C)cn3)=O)CC12 Cn1cc(C(=O)NCCC2COCCN2C(=O)C=CCF)n(C)c1=O c1(OCCC)ccc(CCC(=O)NC(C)(C)C(C)NC(=O)C2=CCSC2)cc1 C1(COC)CN(C(=O)CCC(C)OC)CC(C)(C)O1 CC#CCC(C(=O)NCc1cc(COC)no1)NC(=O)C(CC)OCC Cc1cc(C(N2CC3(CC(NC(=O)CCCC(C)C)C3)C2)=O)n2ncnc2n1 N1(C(C2C(C)(Br)C2)=O)CCC(C(F)(F)F)C(N=c2[nH]nc(C3CC3)s2)C1 N1(C(C2(SCC)CC2)=O)CC(NC(c2cc(Br)cnc2O)=O)CC(C)(C)C1 C(=O)(NNC(=O)C(C)(C)N)NC(C)COc1ccccc1[N+](=O)[O-] C(=O)(CC(C)C(F)(F)F)NCC1CCCC(NC(CC2CC(N(C)C)C2)=O)C1 O=CN1CCCC1CNC(=O)CC1CCCC1.N12CCCC1C1(CC1)C2=O CC(C)(C)CC(=O)N1CC(O)(CCNC(C2CC(N3CCCC3)C2)=O)C1 CC1(C)CCC(CNC(C2CC2CF)=O)N(C(=O)C(F)(F)C2CC2)C1 c1(C(=O)NC(CCCNC(CCCc2onc(CC)n2)=O)C)sc(F)cc1C c1(CNc2c(F)ccnc2F)ccc(F)c(F)c1O.CC1CC2CN1C(=O)N2 CS(=O)(=O)c1cnn(CC(N)=O)c1.c12ccc([nH]1)C(=O)NCC=CCNC2=O C(=O)(CCCCC(F)(F)F)N1CCN(C(=O)CC2CCOC2)CC1CF CC1(O)CCC(C(N2CCC(F)C(NC(C3CCS(=O)(=O)CC3)=O)C2)=O)CC1 C12(C(=O)NCc3cn(CCOC)nn3)COCC1C2(F)F C(=O)(C(C)(C)CCNC(=O)C(C)(C)N=[N+]=[N-])NC(c1nc(C(=O)O)co1)C C(=O)(C(c1cccs1)=Cc1cccs1)N1CCN(C(C2CC(O)C2)=O)CC1CF CC1(C)CCC(F)(F)CC1C(N1CC2(CC2)CC1CNC(=O)CCC1(C)N=N1)=O CN=c1ccc(C(=O)NC23CC(CNC(=O)CCc4cnn[nH]4)(C2)OC3C)c[nH]1 N1(C(c2c(C)nncc2)=O)CCCC(F)(CNC(C23CC(C(C)C)(CO2)C3)=O)C1 C(=O)(C(CO)C(C)(C)C)NCC(CNC(C(CC)(C)COC)=O)(C)C c1(C(C)=O)ncc(C(=O)NCCN(C)C(c2cnc(-c3ccccn3)s2)=O)s1 O=C1NC(=O)C(CC(N2CCCC(N(C(=O)Cc3cccc(Cl)c3)CC3CC3)C2)=O)N1 N1(C(=O)Cn2cc(Br)c(Br)n2)CCCc2cc(Br)c(Cl)cc21 c1(OCC)cccc(OC)c1CNC1(C)CCCCC1 C1(C#N)(C(=O)NC(CNC(c2ncc(C)cn2)=O)C2CC2)CC2(CC2)C1 N1(C(c2cn(C(C)C)nc2)=O)CCC2CC12C(N1CCC(CC(C)(C)C)C1)=O Cc1c(C(=O)NC2CC2NC(=O)CNc2nccs2)[nH]c2c(Cl)cccc12 c1(C(N2CCC(CCNC(C=NOC)=O)C2)=O)cc2ccccc2c(=O)n1C C(N=C(NCc1cc(C(C)(C)C)on1)NC1CCS(=O)(=O)C1)CC1CC(C)C1 C1(C(=O)NCC2CC(C)N(C(=O)CN3CCOCC3=O)C2)COCCN1C=O Cc1cc(C(=O)NCC2(O)CCN(C(C3CC3C)=O)C2)c2c(C)nn(C)c2n1 Cc1ncc(F)c(N2CC3CC2CN3c2nc(C)ncc2Br)n1 C1(CNC(C(c2ccncc2)C)=O)CCN(C(=O)CSc2nncs2)C(C)C1 Cc1cc(N)n2ncc(C(N3CC(NC(=O)C(C)SC(C)C)CC(F)C3)=O)c2n1 N1(C(CC(C)OC)=O)CC(CNC(c2cc(C)oc2C)=O)C2CCCCC12 c1(NC(N2C(C(=O)OCC)CC(O)CC2)=O)cc(P(C)(C)=O)cs1 C1(C(=O)O)(NC(c2cncc(CCCC)c2)=O)CC2CCC1CC2 C1(NC(c2c(C(C)C)cccc2)=O)Cc2ccccc2C1NC(=O)C(C)C1CC1 N1(C(CCN2CC3N(C(C)=O)C(C3)C2)=O)CCC2CCCCC2C1 c1(C(N2CCC(C3CCCN3C(C3CC(n4cnnc4)C3)=O)C2)=O)csc(O)n1 CCC1=C(C(=O)NCC2CCN2C(C2=CC=C(C3=CCCC3)CC2)=O)CCCO1 c1(C(=O)NC2C3CCN(C(=O)Cc4cccc(Cl)c4)C23)ncn2c1COCC2 C1(C(N2CCN(C(=O)Nc3cccc(OC(F)F)n3)CC2)=O)CC2CC1CC2=O CCCC(C(O)C(=O)N1CCCC1C(=O)NCC)NC(c1c[nH]c(C#N)c1C)=O N1(C(C(CC=C)(C)N(C)C)=O)C2CCCC1CC(NC(=O)CN1CCOCC1)C2 c1(C(N2C(CCNC(C3CCN(C)C(=O)C3)=O)CCC2)=O)cc(F)c(N)cc1F C(=O)(CCCCCC(C)O)NCCC(C)NC(c1cnc(C2CC2)nc1)=O N1(C(C(C)SC)=O)CCC2(CC1)CN(C(C1CCN(S(C)(=O)=O)C1)=O)C2 c1(C(N2CC(C)C(CNC(=O)C(C)(C)F)CC2)=O)cnc2ccoc2c1 N1(C(c2ncc(OC)cn2)=O)CCC(NC(c2ccc(C(F)F)s2)=O)C12CCC2 C1(NC(CN(C)OCC)=O)CCN(C(c2cnc(C3CC3)nc2C)=O)CC1C CC1(CNC(c2cc(CO)ccn2)=O)CCC(NC(=O)C=CCO)C1 c1(C(N(CCC(C)NC(C2(C(C(C)SC)=O)CC2)=O)CC)=O)ccc(COC)o1 N1(C(C(C=C)(C)O)=O)CCC2(C=C(C(=O)Nc3cnn(CCO)c3)C2)C1 n1(CC)c(=O)sc2ccc(-c3nc(-c4noc(C(F)(F)F)n4)cs3)cc12 N1(C(c2c(C(C)(C)C)nccc2)=O)CC2(C1)OC(=O)Nc1ncccc12 N1(C(c2ccccc2SCCO)=O)CCCC2(C1)CN(C(C13COC(C1)C3)=O)C2 c1(C(C)=O)cnc(C(=O)NCC2CCCC2NC(=O)C(C)(C)O)cn1 N1(C(C2(C#C)CCC2)=O)CCC2(CCC2NC(=O)CCCN(C)C)CC1 C1(CC(N2CC(CCNC(c3c(CC)ncs3)=O)C2)=O)NC(=O)NC1=O C#Cc1cc(F)cnc1NC(c1c(C)[nH]c(C(=O)NC2CSCC(=O)N2)c1C)=O c1(C(N2CC(NC(=O)CC3CSCCS3)C3(C2)CC3)=O)ccc2c(n1)COCC2 C1(NC(C(C)C#N)=O)CCC12CCN(C(c1ccc(Br)c(F)c1)=O)CC2 Cc1ccc(C(=O)NC2CN(C(=O)COc3cc(Cl)ccc3Cl)C3CC23)nc1C CCCC(C(O)C(=O)NC(C)CCCO)NC(c1cc(C)n(CC)n1)=O Fc1ccc(CNCc2cc(-c3cccc(Br)c3)no2)cc1N1CCCC1 N1(Cc2ccc(C)c(O)c2)CC2OCCN(C(c3cccc(CO)n3)=O)C2C1 Cc1nc(O)c2cc(NC(=O)C(=O)NCC3(C)CCCCC3)ccc2n1 c1(OC)cc(C(N2CC(CNC(c3ccc(F)nn3)=O)C2)=O)cc(F)c1OC Cc1cc(=NCCN2CC3CCC2C3)[nH]c(NC(c2nccs2)C)n1 c1(C(N2CCC(CC)C2C(N2CCC2(C)CC)=O)=O)nc(C)ccc1C C1(NC(C(N)=O)=O)CN(Cc2cccc(Cl)c2F)CC1C#N C1(CC(=O)NCc2ccn(CCC)n2)CCCN(C(C2CCC2COC)=O)C1 c1(CC)nc(C(=O)NCc2ccc(C(F)(F)F)cc2)c(C)o1.C12CC1CNC2=O C1(NC(CN(CCOC)C(c2ocnc2C2CC2)=O)=O)CCCC1C(N)=O Cc1ccc(C(=O)NC2(CC(=O)NC3CC3CC(C)(C)C)CC2)nc1O N1(C(C(CCC)OC)=O)CCC2(CC1)CC(NC(c1cn(C3CC3)cn1)=O)CO2 N1(C(C2(C=C)CCN(C(c3csc(CO)n3)=O)C2)=O)CCC(C)OC(C)C1 c1(CC(N2C(CNC(C(CC)(C)O)=O)COCC2)=O)ccc(Br)c(O)c1 c1(OC)cnc(C(F)(F)F)cc1C(=O)NCCC(O)CNC(=O)C(C)CF CN1N=C(C(=O)NC2CCC(C)(CNC(=O)CCC=CC(C)C)C2)CCC1=O CCCCC(CCC)NC(c1c[nH]nc1CNC(C1OCCCC1(C)C)=O)=O c1(C(N2CC(NC(C3(C(C)C)CC3)=O)C(O)C2)=O)ccc(S(N)(=O)=O)cc1 c1(C(N2CCC(C)C(NC(c3ccoc3Cl)=O)C2)=O)ncc([N+](=O)[O-])n1C CC(CCC(=O)N(C)CC1CCCN1C(=O)C(C)(C)CO)c1ccccc1 N1(C(CC(=C)C)=O)CCN(C(=O)CCc2ccc(=N)[nH]c2)C2CCC12 CC12CC(C(=O)NC3CC(n4cc(CC5(C)CCCCC5)nn4)C3)(C1)C1(COC1)O2 c1(CC(=O)NC2(CNC(CCCCC#C)=O)CCOCC2)ncnc2sccc12 c1(C(=O)NCC2CC(NC(c3c(OC)n[nH]c3)=O)C2)cccc(S(C)(=O)=O)c1F N1(C(C(C)NC(=O)NC)=O)CC2CN(C(=O)C(C)Sc3ncccn3)CC2C1 N1(C(CC(=O)OCC)=O)CC2CCC(C1)C(NC(=O)C(C1CC1)N(C)C)C2 Cc1cccc2c1NCCC2C(=O)NCCCNC(C1CCC(C)CC1)=O C1(C(N2C(CNC(C(C)(Cl)Cl)=O)CC2)=O)CCn2nnnc2C1 c1(OCC(=C)C)ccc(NC(N2CC(Sc3ccc(Cl)cc3)C2)=O)cc1 N1(C(C2(CC)CC2)=O)CCC2(CCCN2C(c2c(OC)cccc2Cl)=O)CC1 C(=O)(C1=NOC(CNC(=O)CC2CCC(=O)C2C)C1)NCCC(C)C C(=O)(C1CCCc2ncnn21)NC1CN(C(C=C2CCC(C)C2)=O)C(C)C1 C12(C)CCN(CC1)C(=O)OCCNC2=O.C1(C)(C)C(=O)N1.CCCNC(C)=O CCCCCC(=O)NC(C)C(C)NC(c1cn(CC(F)(F)F)nn1)=O N1(C(Cn2nc(C)c(Br)c2)=O)CCC2(CCCC2NC(=O)C2=CCC2)C1 c1(CC(=O)N(CC(C)N(C(=O)C=C(Cl)Cl)C)C)sc(O)nc1O c1(C(N(C)CC2N(C(CC(C)SC)=O)CCCC2)=O)cnc(O)c(C)c1 c1(CC(N2CCC(NC(C(C(C)C)C#N)=O)C2)=O)cc2ccccc2cc1O C1(CNC(C2(C#C)CC(=O)C2)=O)CC(C(=O)NC(C)CC(C)n2cccn2)=NO1 C(=O)C1Cc2ccccc21.c1(-c2cn(CCN(CCC)CC)nn2)ccncc1C O=S(=O)(c1c[nH]ccc1=NCC1CC2(C1)CC21CCC1)N1CCCCC1CO CCCN(OC)C(=O)C(C1(C)CC1)NC(C1CCCC12CCC2)=O C=C(C)C1OCCCC1C(=O)NC(c1ccc(Cl)cc1)c1ccccn1 c1(OC)ccc(C(N2CCCC2CCC(=O)N(C2CC2)C(C)C2CC2)=O)cc1OC Cc1cc(C#N)nnc1N1CCC(C(=O)NC2CCCCN2C)C1 C1(CC(N2CC=CC(NC(C#CC(C)C)=O)C2)=O)CCOC(C)(C)C1 N1(Cc2cc(-n3ccnc3)c(Cl)cc2)CC2CC3CC(C2)CC1C3.C1CN1 CC1CC2CN(C(C3(C)CN(C(c4ccc(C#N)[nH]4)=O)C3)=O)CCN2C1 c1(-c2onc(CC(C(=O)NC(C)C)(C)C)n2)ccc2ccn(CCO)c2c1 C1(CNC(C(C)(C)C)=O)CCCC(NC(c2ccc(NS(C)(=O)=O)nc2)=O)C1 C1(O)(CNC(=O)NCCCNC(c2ccco2)=O)CCCNC1 c1(OCCNC(=O)NC2COCC2N2CCCC2)ccc(Cl)c(Cl)c1 C(=O)(C1=C(C)C(C)(C)OC1=O)NCC(C)(C1CC1)NC(C(COC)CC(C)C)=O S(=O)(=O)(c1ccc(C(F)(F)F)cc1)N1C(C(=O)Nc2ccccc2I)CSCC1 N1(C(c2cccc(CC)n2)=O)CCN(C(c2cnc(C)[nH]2)=O)C(C)C1 CC(F)(F)C(C(=O)NC1CC1NC(c1c(Cl)cccc1Cl)=O)c1ccccc1 c1(C(N2CC(C)C(NC(=O)CC(C)CN(C)C)C2)=O)cc2cn[nH]c2cn1 CC1CCN2CCN(C3CC4CCCC4C3)CC2C1 C1(NC(c2c(Cl)cc(C)s2)=O)C(C)CCN(C(c2cc(N)cnc2Cl)=O)C1C N1(C(C2CC(=O)N2)=O)CC2(C1)C(NC(c1noc3ccccc13)=O)CCS2(=O)=O C1(CN(C(c2cccc(C)c2)=O)C)CN(C(c2nc(C)nn2C)=O)CC12CC2 C1(NC(CC)=O)CC(C(=O)NOCCc2ncoc2C)C1(C)C C#Cc1ccc(OC)c(C(=O)NC2CN(C(=O)C(O)CCCC)CC2F)c1 CONC(=O)CCOCC(=O)Nc1ccnc(Cl)c1 c1(C(=O)NC2CCC(CNC(C(C)SCCCC)=O)CC2)cnc2scnc2c1 C1(CNC(c2nc(C(C)=O)sc2)=O)CCCCN(C(C2(C)C=CCCC2)=O)C1 c1(C(=O)NCCC(CNC(CC(=C)C)=O)O)cc(F)cc(Cl)c1N C#Cc1ccc(C(=O)NCC2(NC(c3ccc([N+](=O)[O-])s3)=O)CCC2)c(F)c1 C1(NC(c2cc(C)oc2)=O)COC2(CCN(C(c3ncn4ccccc34)=O)C2)C1 c1(OC)ccc(F)c(S(=O)(=O)NC(=O)NCC2CCCCN(C)C2)c1F c1(CCC(=O)NCCC(C)NC(c2cc(C)[nH]n2)=O)c(F)cc(Br)cc1F C1(NC(C2C(=C)C2)=O)CC2CCC(C1)N2C(=O)COC1(C)CCCC1 Cn1nc2ccccc2c1C(N1CC(NC(=O)C(O)P(C)(C)=O)C2(CCC2)C1)=O CCC(O)C(F)(F)C(=O)N1CC2CC2(NC(c2cc(-c3ccccc3Cl)on2)=O)C1 N1(C(CCc2scc(C)c2)=O)CC2CCC(NC(c3cnc(O)n3C)=O)CC2C1 C1(NC(CC(COC)(C)O)=O)CCC2(CC1)CC2NC(c1cnn(C)n1)=O C1(CC)CC(C)CN1c1nnc(C2(CC#N)CCCCC2)n1CCC#N C(=O)(CCCC(=O)N1CCOCC1CCNC(C1COCCC1(F)F)=O)OC c1(C(=O)NCC(F)CNC(=O)C(F)CC2CCCC2)cccc2c1OCCO2 Nc1ccc(C(N2CC(O)CC2C(N2CCCC2CC2CCC2)=O)=O)nc1 c1(N2C(C(N)=O)CCC2)nc2cc(F)cc(F)c2o1.C12CCCN(C1)C2=O Cc1cccc(C(=O)NC2COCC2NC(=O)C(C2CCCCC2)F)c1 C1(NC(C2(F)C(C)C2)=O)CCN(C(c2cc(C(N)=O)c[nH]2)=O)C1C(C)(C)C C1(C(=O)NCC(CC)NC(=O)CSc2c(C)n[nH]c2C)Cc2nccnc2C1 C12(NC(CN(CCC)C(C3CC(C)OC3=O)=O)=O)CC3CC(CC1C3)C2 c1(C(=O)OC)ccc(NC(C2CCCO2)=O)cc1.C12CCCC1NCCC(=O)N2 CCC(C)(C(=O)NC)NC(=O)CC1CCCN1C(=O)OC(C)(C)C.C(C)(C)(C)C(=O)O c1(C(=O)NC2CCN(C(C(CC)O)=O)C23CCC3)[nH]c2ccccc2c1C n1(CC(=O)NCCCC2CCCN(C(C3(C(N)=O)CC3)=O)C2)cnc2c1CCCC2 C(=O)(C(C)(O)CC(C)C)N1CC(CCNC(c2ccc(SC)s2)=O)C(C)C1 C(C1CCCN1C(c1ccsn1)=O)=CC(=O)NCCCN1C(C)CCC1 CC(C)CS(=O)(=O)CCC(=O)N1CCN(C(=O)Cc2cccc(F)c2Cl)C(C)C1 c1(NC(C2CCCCN(C(C(C)NC(COC)=O)=O)C2)=O)cn(C)c(=O)nc1O c1(C(=O)OC)ccc(C(N2CCC(CCNC(C3CCC3OC)=O)C2)=O)cc1 C1(CNC(=O)Cc2cc[nH]c2)CC2CCC1N(C(c1ccnc3ncnn13)=O)C2 N1(C(C2CC(NC(C)=O)C2)=O)CCC(N(C(=O)CN(C2CCCCC2)C)C)CC1 CC1CCN(CC(=O)Nc2cc(C#N)ncn2)C(C)C1Nc1cc2ncccn2n1 C1(C(N2C(CNC(c3ccn(CCC)n3)=O)CC2)=O)CCOC2(CCCCC2)C1 C(C(CC(C)C)NC(c1cn(C)nc1O)=O)NC(C1(COC)CC1)=O C(=O)(C(F)(F)C(F)(F)CCl)N1CC(CCn2c(C)nnn2)C1.C1(CC=O)CC2(CC2)C1 C1(CCOC)CN(C(c2onc(C)c2C)=O)CCN1C(=O)Cc1ccnn1C n1(CC(=O)NCC(CC)NC(C2CCN(C(=O)NC)C2)=O)ncn(C)c1=O CC(CCc1ccc(F)cc1)C(=O)N(C(C)CN(C)C(C1(CCF)CC1)=O)C Cc1cc(C(=O)N(C)CC2CCCN2C(=O)CC2C=CCC2)cc(C)c1C CC12CN(C(c3cc[n+]([O-])cc3)=O)CC1CN(C(=O)C(F)(F)Sc1ccccc1)C2 CC(C)(C)CCCCC(=O)NC1CC(NC(c2cnc3n2CCCC3)=O)C(O)C1 c1(N(CCCCC=C)C)nc(N(C(c2ccc(C)cc2)CC)C)nc2c1COC2 C1(CNC(C=C(CC)CC)=O)CC2(CO1)CN(c1ncc3ccnc-3[nH]1)C2 S(=O)(=O)(c1ccc(NCCCSC)c(C#N)c1)N1CCC(OC(COC)C)C1 C(=O)(CC(C)(C)CC)N1CCCC(N(C(c2ccc(CCC=C)cc2)=O)CC)C1 Cn1cc(C(=O)NC2C=CCN(C(=O)CCN3CCOCC3)C2)nc1C(F)F Cc1nn(C)cc1C(C(=O)NC1CCC1)N(c1sccc1Br)C c1(C(N(CCCN(C(C(c2cccc(C)c2)O)=O)C)C)=O)cnn2cccc2c1 Cc1nccc(C(N2CC(CNC(c3c(C)cnn3C)=O)C3CC23)=O)n1 C1(CN(C(=O)C(O)C2CC2)CC)CCN(C(=O)C(C2CCOCC2)O)CC1 C(CC(C)(C)C)(C(=O)NCC1(CNC(=O)CC2COC3CC2C3)CC1)OC C(=O)(CCC(F)(F)F)N1CCC(N(C(=O)COc2ccccc2)C)CC1 N1(C(c2c(CNC(CC(=O)NCC#C)=O)nccc2)=O)CCC2CCC(C1)N2C c1(CCC(=O)NC2CN(C(c3nc(C)c(C)s3)=O)C(C)C2)cccc(F)c1Cl c1(NC(C(CCC)C)c2nnn[nH]2)ccc(C(N)=O)c(F)c1.c1ccccc1 c1(N2CCCC(=C)C2)nc2cccnc2c(=NCCCN2CCCC2)[nH]1 CCCC(CCC)CC(=O)N1C2CCC1(CNC(=O)CC1CC3CCC1C3)CC2 CC1Cc2cc(CC(N3CCCCC3CCNC(=O)C=CC3CC3)=O)ccc2O1 C1(C(=O)NCCC2CN(C(C(C(CC)O)(F)F)=O)C2)CCc2ncccc2C1 c1(C(N(C)CC2CCCN(c3cc(C(N)=O)ncn3)C2)=O)cc(F)c(Cl)cc1F CC(C)C(C)C(N)C(=O)NCC(c1cc(Br)ccc1Cl)=O c1(CCC)noc(CCC(=O)NCCC(C)N(C)C(C2CC(C(N)=O)C2)=O)n1 c1(C(C(=O)NCC(F)(F)F)Nc2cc(C(C)(F)F)[nH]n2)ccccc1OC(F)F C(=O)(C1=C(C)OCC1)N(C(C(C(C)=O)c1ccccc1)=O)C C1(CCC)(N(C(c2ccc(C#N)o2)C(=O)NCCOC)C)CCN(C(C)=O)CC1 C(CCCCC(=O)NCc1ccc(C(=O)NC2CC2(C)C)s1)SC C1(N(C(C(C2CCCCC2)C)=O)CCNC(C2CC=CCC2)=O)CCCCCC1 CC1(C#CC(=O)NC(C)(C)CCCNC(C2(c3cccnc3)CC2)=O)COC1 N1(C(C2N(C(c3c(C)[nH]cc3)=O)CCOCC2)=O)CCCC(C)(C#N)C1 S(=O)(=O)(c1ccc([N+](=O)[O-])cc1F)N1CC(CC)Oc2c1cccc2 c1(C(=O)NCC2N(C(c3scc(C)c3Cl)=O)CCCC2C)cccc2sncc12 C(=O)(C(C(C)CCCC)NCC(=O)NC1CCCCC1)N1CCC(C#C)C1 N1(C(C2(C)CC2Br)=O)CCC(C2CN(C(=O)CC3(O)CCOCC3)C2)CC1 c1(NC(C2(C)CCCN2Cc2ccc(F)cc2F)=O)cnc(Cl)c(Br)c1 C(=O)(C1=NNC(=O)CC1)NCCOC1CCN(C(c2cc(OC)cc(F)c2)=O)C1 Cc1cc(CC(=O)NC2CCCC(C(=O)Nc3cnc(Br)cc3C)C2)cc(C)c1 C1(NC(c2n(C)c(=O)ccc2)=O)CC2CCC(C1)N2CC1CC2CCC1C2 C(CC(=O)NC(COC)CCOC)(CC(C)C)NC(C(CCC)C#N)=O C1(NC(C2C(C(N(CC(C)C)C(C)C)=O)C2)C)CCCN1CCCO c1(C(N2CCCC(N(C(C(C)CN(C)C)=O)CC3CCCO3)C2)=O)ccc(F)cc1 c1(NC(C2CC(O)CCN2C(c2cc[nH]n2)=O)=O)c(Br)cc(F)c(F)c1F C1N=C2NC(=NCCCc3c(N)cccc31)Nc1ccsc12.C1(CO)CCOC1 c1(OCC(=O)NCC(C)(C2CC2)NC(Cc2ccc(C)s2)=O)cc(Cl)ccc1Cl CCC(C)CC(C(=O)N1CC2CC2C1COC(c1cc(C)[nH]c1C)=O)OC N1(C(C2C(c3ccc(C)cc3)CC2)=O)CCc2ccnc(N(C)C)c21 CCC(C)CCC(=O)N1CCCC(CC(=O)N(CC(Cl)Cl)C)C1 c1(CNC(C(c2c(C)noc2C)C)=O)ccnc(C)c1O C1(NC(COCc2cc(C)on2)=O)CC2CCC(C1)N2c1ccc(C#N)nn1 C1(O)(C(C)NC(Cc2cnc(C)o2)=O)CCN(C(C2CCCCC2(F)F)=O)CC1 N1(C(c2c(N)cncn2)=O)CC2CC1CCC2NC(=O)C(O)Cc1cnc[nH]1 N1(C(c2c(C)nc(CSCC)s2)=O)CC(CNC(=O)C(CC)OC)C2(CCC2)C1 C1(CCC=C)(C(=O)Nc2c[nH]nc2OC)CN(C(=O)C(N2CCOCC2)C)C1 C(=O)(CCCC1CCC1)N(CC)CC1CCN(C(=O)CC(C)C2CCCO2)C1 C12(NC(Cn3c(=N)nc[nH]3)=O)CCC1CN(C(c1sccc1C(F)F)=O)C2 c1(NC(C2CC3CC3N2C(c2csc(Br)c2)=O)=O)cccc2c1CCC2 C(CN=C(NCc1c(O)cccc1F)NCC1CCCO1)OCC=C C1(CNC(C2(CCC)CCC2)=O)CC(OC)CN1C(=O)C(C)SC(C)C C1(C(N2CCCC(N(C(=O)CNC=O)C)C2)=O)CN(C)C(=O)CCO1 CC1(CNC(c2ccnn2C(C)(C)C)=O)CCN(C(=O)CCOCC(F)F)C1 C12(NC(CCNC(C)=O)=O)CCN(C(c3cc(C)cc(N)c3)=O)CC1C2 N(C1CCCn2cnnc21)C(CC(CC=C)NC(=O)CN1C(=O)CCC1=O)=O C=CCC(F)(F)C(C)(C)C(=O)NCC1CC1NC(=O)C1CCc2c[nH]nc21 N1(C(CCOC2CN(C(C3N(C)CC3)=O)C2)=O)CC1(C)COC1CC1 C1(=O)C(C(=O)SC)OCC(C)(CC)CN1.C(C)(C(=O)CC(=O)N(C)C)OCCOC c1(C(=O)NC(C)CC(C)NC(C2CC(C3CC3)=NO2)=O)nc2ccccn2c1F c1(C(=O)NC2CCN(C(C3CC4(CC4)C3)=O)CC2)ccc2nn[nH]c2n1 N12CCC3C(C13)N(C(=O)O)CC2=O.c1(C(=O)NC(C)(C)C)cc(C2CC2)on1.CC C1(CNC(CCCCC#C)=O)CC2CCCC2N1C(C1CC(F)(F)CN1C)=O c1(C(=O)NCC2CCN(C(C(CC)O)=O)C2(C)C)cc2nn[nH]c2cc1F C(C)(C)(CC(=O)NCCC1CC2CCC1C2)N(C(c1c(C2C(C)C2)noc1)=O)C C#CC(CNC(=O)C(C)NC(c1nccs1)=O)CC c1(CC)ccc(O)c(C(=O)NC2CC2CNC(c2ccc(C(C)C)nc2O)=O)c1 C(=O)(C(C)(C)CN1C(=O)CCC1=O)N(CCCCN(C)C(C1CC(C)(C)O1)=O)C n1(CC)nnnc1CNC(=O)CC1CCCN1C(=O)CCF c1(SCC(=O)NC2CC(CNC(C(c3cnn(C)c3)OC)=O)C2)nnc(S)n1C N1(C(CC(C)OC)=O)CCn2c(C(=O)NCc3ccc(F)cc3Cl)cnc2C1 C1(CC(=O)NC(CC(C)C)CNC(C2C3COCC23)=O)CC2(CCO1)CC2 c1(SC)cn(C)nc1C(=O)NCC12CC1CN(C(c1cnoc1C)=O)C2 CCCCC(O)CC(=O)N1CCN(C(c2ccnc(O)c2)=O)CC1CCO N1(C(C2C(C)(C)N(C(C3CC4CC4C3)=O)CC2)=O)CCN2CCC1CC2 CC(CCCC(F)(F)F)(c1nnnn1C(COCF)N)C1CC1.C1CC1 C1(NC(CCCC)=O)CC(NCc2cc(C)nn2C(F)F)C1(C)C Cc1nc(NC2(CN(C)Cc3ccn(C)n3)CCC2)nc2ccc(Br)cc12 C(CCCCCNC(=O)C(N1CCCCC1=O)C)N(C(COCCOC)=O)C C1(CF)CC(c2nnnn2C2CCOCC2)(NC2CCC2)CCO1 CCC(CC)CCCN(C)C(c1cncc(CNC(c2nnn(C)c2N)=O)c1)=O C(CCCCNC(C1CC(CF)C1)=O)N(C(C(C)SC)=O)C C=CC(C)(O)CC(=O)NCCCN(C(=O)C(CC)C(=O)OCC)CCO C(=O)(CC(P(C)(C)=O)c1ccccc1)NC(C)CCNC(C1CC2(CC2)C1)=O C1(F)(CNC(C(C)NC(C2CCC2)=O)=O)CC(CNC(C2CCCN2C)=O)C1 c1(NCCCNS(N(C)C(C2C3CS(=O)(=O)CC23)C)(=O)=O)cc2nccnc2[nH]1 CC1(C)CCC(C(=O)NC2CCC(CNC(=O)CC3CC4C=CC3CC4)C2)CO1 c1(OC)cc(S(=O)(=O)N(C)CC2(CCO)CC2)sn1 C1(C(=O)NCCC2CCCN(c3snc(C(C)C)n3)C2)CCC2(CCCC2)C1 C1(CN(C(c2c(C(C)C)con2)=O)C)C2CN(C(c3cc(C#N)c[nH]3)=O)CC12 C(C(C)(O)CC(=O)OCC12CNC(CNC(=O)OC(C)(C)C)(C1)C2)OC c1(OC)cc(C)c(Cl)cc1-c1c[nH]nc1CN1CCOCC1 C(=O)(C1CCCc2c1ncn2C)NCc1c(Cl)cc(C)nc1 n1(CC)cc(NC(=O)C(=O)NCCNS(=O)(=O)N(C)C)c(C#N)n1 C12(C(N(C3CCN(C(c4c(CC)sc(=N)[nH]4)=O)CC3)C)=O)CC(C)(CCO1)C2 N1(C(c2c(C)snc2)=O)CCCC2CN(C(c3n[nH]cc3C3CC3)=O)CCCC12 c1(C(N(C(=O)CC2CCCC(C)O2)CCCC)=O)c(-c2ccccn2)noc1C Cc1cc(NC(=O)NCCc2ccc3cc[nH]c3c2)ccc1S(C)(=O)=O C1(N=[N+]=[N-])(C(=O)NC2CN(C(CC(C)(C)SC)=O)C(C)CC2)CCOCC1 c1(CC)cncc(C(N2CCC(C(C)NC(C3(OC)CC(O)C3)=O)C2)=O)c1 Cc1coc(C)c1C(=O)NCC1CCCN1C(c1csc(S)c1)=O c1(OC)cccc2ccc(C(=O)Nc3ccc(OCc4ccccc4)nc3C)nc12 C(=O)(CC(C(=O)NCC(c1ccco1)N1CCCC1)N(C)C)OC CCCC(C)CC(=O)NC1C=CCN(C(=O)CC2CC(n3cnnc3)C2)C1 C(CNC(c1cnncc1C)=O)(CC)(CC)NC(C(C1CCC(C)CC1)CC)=O N1(C(CC(C2CC2)NC(c2nc(C)oc2C)=O)=O)CCN(C)CC(O)C1 N1(C(C2CC(F)C2)=O)CC(C(N2CCC(OCC3CC3)C2)=O)C(F)(F)C1 c1(OC)cccc(CN(C(C2CC(n3ccnn3)C2)=O)C)c1.C1CC(=O)N1 C(=O)(CCCC(=O)N1CC2CC2(CNC(c2cncc(C(N)=O)c2)=O)C1)NCC c1(CNC(Cn2cnc(=N)[nH]2)=O)cccc(CNC(C2CC(CC(F)F)C2)=O)c1 CC1(CNC2CCN(C3CCCC3)C2)CC2CCC1C2.N12CCC(CC1)C2 C1(C(N(CC(C)(C)NC(CN(C(C(C)C)=O)C)=O)C)=O)CCCN1C c1(CNC(C=C(C)C(F)F)=O)cc2n(n1)CCN(C(=O)C(c1ccccc1)C)C2 N1(C(c2cc(C(C)C)c[nH]2)=O)CC(NC(c2nc(COCC)sc2)=O)C(C)C1 C1(C(=O)NCC(CC(C)C)O)CCCCC1(C)NC(=O)C=Cc1ccsc1 n1(CC(=O)N(C)CCC2CCC(COC(C)=O)CC2)ncc2cccnc12 c12cccc3c1CCN(C3)C2.C(CC(C)C)(C(=O)NCc1cccc(I)c1)OC CC(CC#N)C(=O)N1CCC(NC(c2ocnc2C(F)F)=O)C1 C=C(C)C(CC(=O)Nc1nccc(CO)n1)OCC.C12(C)CCC(C1)NC2 N1(C(C2CCN(C(CN(C(C(C)C)=O)C)=O)C2)=O)CC2CCN(C)C2C1 N1(c2nc(CC)c(C)s2)CC2CCCC1C2CNC(=O)Cc1cccc(C)n1 C(=O)(CC(O)CCCC)NC(C(=O)NCC(C#C)OC)(C)C1CCC1 C1(CNC(C(CC)N(C(=O)Cc2coc(C(F)F)n2)C)=O)CCC(NC)CC1 N1(C(C(COC)OC)=O)CCN(C(c2nc(C)n(C)n2)=O)C(C(F)F)C1 N#Cc1cc2c(sc1=O)CCN(C(=O)NCCOC1CCCCO1)C2 C1(NC(C2CC2(F)F)=O)CCN(C(C2CC23CCSCC3)=O)CCC1CO c1(C(N(CCN(C=O)CC)CCN2CCCC2)=O)ccc2nncn2c1.OC C#Cc1cccc(C(=O)NC(C(=O)NCCC#C)c2ccoc2)c1 C1(CNC(c2nccc3[nH]ccc23)=O)CN(C(C2CS(=O)(=O)C2)=O)C2(CCC2)C1 N1(C(C=CC=CC)=O)CCCN(C(c2cnncc2C)=O)C(C)C1 CCC(C)CCC(=O)NC(C1CN(C(c2cnc(CC)[nH]2)=O)CCO1)C C#Cc1ccc(C(N2CCN(C(c3ccc(O)cc3)=O)CC2CC2CC2)=O)nc1 CC1=C(C)CN(C(c2cncc(-n3ccc(C(F)(F)F)n3)n2)=O)CC1 c1(C(C)NC(c2cccc(C3(C#N)CC3)c2)c2nnnn2C)ccc(F)cc1F N1(C(c2c(C)cno2)=O)CCC(O)(CNC(C2(N3CCCCC3)CCCC2)=O)C1 C1(C(C)NC(Cn2c(C)ncc2)=O)CCCCN1C(c1c[nH]nc1Cl)=O c1(C(N2CCCC(CN(C)C(c3cncs3)=O)C2)=O)cc(C(F)(F)F)ncc1Br C1(C(=O)NCCCOCCNC(=O)CC2CCSCC2)CC(=O)N(C(C)(C)C)C1 Cc1ccc(C(=O)NC(C)C(C)NC(=O)CC2C=CCC2)cc1C#N c1(CNC(C2CCCCC2NC(c2ccnc(CO)c2)=O)=O)ccncc1CO C12(CNC(=O)CCC3CCCO3)CC(NC(c3ccccc3)=O)(CO1)C2 C1(CN(CCNS(=O)(=O)Cc2ccccc2Br)CC)Cc2ccccc2C1 CCC(Cc1cccc(C)c1)C(=O)NC1CCC(C)(NC(=O)C(C)(C)CO)C1 C(CN=C(NCc1c[n+]([O-])c(C)s1)NCC1CCOC1C)OCC N1(C(c2c(OC)ccc(Br)c2)=O)CC(NC(=O)C(Cl)(Cl)Cl)CC(F)(F)C1 C1(CNC(COC(CC)C)=O)(OC)CCN(C(=O)CC(C)(F)F)C1 N1(C(COCCCC(C)C)=O)CC2CCCC(NC(c3c[nH]c(=N)s3)=O)C2C1 CC1CC(C)(C(=O)NC2CCN(C(c3cn(C)nn3)=O)CCC2CO)CC(C)O1 c1(SCC(=O)NCC2C(NC(C(CC)(C)C)=O)C2)ccsc1[N+](=O)[O-] c1(C(N(CC(C)NC(=O)C(CO)SC)CC)=O)cc(C)nc(N2CCOCC2)n1 C1(C)(C(=O)NCC2C3CN(C(Cn4cnc(C(=O)OC)n4)=O)CC32)SCCCS1 N1(C(COCCCOC)=O)C(CNC(=O)Cc2ncoc2C)CC2COCC12 C1(C(N2CCC(C)(C(N3CC(O)(CO)C3)=O)C2)=O)CCc2n[nH]cc2C1 N1(C(C(C)(F)F)=O)CCC2CC2(NC(C2CN(CP(C)(C)=O)C2)=O)CC1 c1(C(N(CC(CC)NC(c2cnc3n2CCC3)=O)CC)=O)cc([N+](=O)[O-])oc1C N1(C(c2csc([N+](=O)[O-])c2)=O)CCCC(N=c2[nH]c(Cl)ncc2C(F)(F)F)C1 N1(CC(=O)NC(C)C(=O)NCCF)CCCC(NC(=O)CC2CCCN(C)C2)C1 CC1CCCC(OCC(N2CC(CCNC(=O)Cn3ncn(C)c3=O)C2)=O)C1 C1(CNC(c2ccc(C)s2)=O)COCCN1C(c1cn(CC2CCCO2)nn1)=O C=CC1(C(=O)NCC2C(C)(C)C2(F)F)CCN(C(c2csc(O)n2)=O)C1 C(CNC(=O)C(C)Oc1cccc(Cl)c1)(CC(C)C)NC(C1(COC)CCC1)=O C(=O)(CC1OB(O)c2ccccc21)OC.C1(=O)CC(C)(c2ccon2)C2CC2N1 C(=O)(C1=C2CCCN=C2NN1)NCCCN(C(C(C(C)OC)O)=O)CCO N1(C(CC=CC)=O)CCC2C(C1)NC(=O)CN2C(=O)C(C)OC1CCCCCC1 C#CC1(C(=O)NCC(C2CC2)N(C(=O)CCc2ncc[nH]2)C)CCC1 n1(CC(N2CC(C)C(CCNC(=O)C3=CCCOC3)C2)=O)ccc(O)nc1=O N1(C(C(C(C)C)F)=O)CC(NC(=O)OC(C)(C)C)Cc2ccccc21 C1(NC(CCc2ccc(C)s2)=O)CC2(C1)CN(C(=O)CC(C)(C)C1CC1)C2 C1(CC)CC(C(=O)NCCCN(CCCNC(C2SCCCS2)=O)C)CCO1 c1(C(=O)NCCCCCCNC(c2cnn3ccsc23)=O)cc2c(nn1)CCC2 n1(CC)cc(Cl)c(C(N2CC(CC(C)NC(=O)COc3ccccc3F)C2)=O)n1 c1(CNC(CCC=CC)=O)ccc2c(c1)CCC2NC(=O)C(C)NC(=O)COC N1(C(C2(C)CC(O)(C(F)F)C2)=O)CC2CCOC2C1.C1(CN)C2C3CCC(C3)C12 C12(C(=O)NCCC3CN(C(c4ccc(C)nn4)=O)C3)CCCCC1C2(F)F N1(C(C(=O)NCCNC(C)=O)=O)CCN(C(C2CC2F)=O)CC1C C12(CNC(COCC=C)=O)CCCC1CCN2C(=O)CCOc1ccccc1C N1(C(CC(C=C)C)=O)CCC2C(NC(=O)CNC(c3ccoc3C)=O)CC12 Cc1ccc(CCC(=O)NC2CC3(C2)CC(NCc2ncc(C)s2)C3)c(C)c1 Cc1nc(C(N2CCC(CF)(NC(=O)CS(=O)(=O)NC3CC3)C2)=O)cn1C Cc1nn(C)c(C(=O)NCCN(C(c2cc(Cl)ns2)=O)C(C)C)c1Cl C(CN=c1[nH]c(=NCc2cnns2)c2sccc2[nH]1)c1c(C)ncs1 N1(CC(c2cccnc2F)C)CC(O)CC2CCCCC12 N1(C(C=CC)=O)CCCCCC(NC(c2cc(C3CC3)oc2C2CC2)=O)C1 CC1CC(CNC(=O)COc2ccccc2Br)CN1C(=O)CCCC1(C)N=N1 Cc1nc2cncc(C(=O)NC3COCCN(C(C4CN(C)C4)=O)C3)c2[nH]1 c1(CC(N2C(CNC(c3c(C)onc3C3CC3)=O)CCC2)=O)noc(C)c1C#N c1(C2(C(=O)NCCCCCCC)CCC2)cccc(C2=CCN(C)C2)c1 CC12CC(C(=O)NC3CC(O)(CNC(C4(c5ccno5)CC4)=O)C3)(CCO1)C2 CC#CC1CCN(C(=O)C(CC=CC=CC)NC(=O)COCC)C1 c1(C(=O)NCCC2CN(C(CCOC(C)=O)=O)CC2C)[nH]nc2c1COC2(C)C c1(OC)cc(C)c(C)cc1-c1ccnc(CC(=O)Nc2cccc(CO)c2)c1 N1(C(C2(CSC)CC2)=O)CCCC(CCC(=O)NCCC2CC(C)(C)CO2)C1 C1(OC)CCSCC1.c1n[nH]cc1C.C1(OC(=O)OC(C)(C)C)CN2C1NC2=O Cc1onc(-c2ccncc2)c1C(=O)NCC(C)N(C)C(C1CCCC1(F)F)=O Cc1c(C(=O)NC(C(N2CCCCC2c2ccccc2)=O)C2CCC2)ncn1C O=C(O)C(O)C(Cc1ccccc1)NC(C(=O)NCc1ccc(CO)o1)=O C1(CC)C(NC(c2cncc(C)n2)=O)CCCN1C(=O)C(C)CC1CCCC1 N1(C(C(CC)SC2CCCCC2)=O)C2CCC1CN(C(C1CC1OC)=O)CC2 C=CC1(C(=O)NCCCC(C)NC(C2C3CN(C)CC23)=O)CCCCC1 CC1(CNC(c2ncc(Cl)cc2F)=O)CCCN(C(C23CC=CC(C2)OC3)=O)C1 C#CC1CC2(CC2)CN1C(=O)C(C)(C)NC(C1OCCC1C(C)C)=O O(NC(=O)C(C)n1cc(CNC2CCCC2C(=O)O)nn1)CC1CCC(=C)CC1 c1(CC)cc(CC)nc(N2CC(CO)(NC(=O)CCc3ccc(F)c(Cl)c3)C2)n1 C1(C(=O)NC(CC(C)C)C(N)=O)CCC(C)(C)N(C(C2(C(=O)C3CC3)CC2)=O)C1 Cc1ccc(C(=O)NC(CNC(=O)C(C)(O)C(C)(C)C)C(C)C)c(F)c1F O=C(C#CC1CCCC1)NC1(CNC(c2cccc(-c3cc[nH]n3)c2)=O)CCC1 C1(NC(=O)CC2=CCCC2)CC2(CCNCCO2)C1 C1(CNC(=O)C(F)=C2CCC2)C(C2CC2)CCN1C(=O)C(O)CC(F)(F)F C1(CNC(c2ncc(C)nc2)=O)CCN(Cc2cc(O)ccc2C)CC1O CC1C(NC(=O)C(=O)N(C)C)CCCN1C(c1ncc(Br)cn1)=O Cc1cc(CC(=O)NCCCC(C)NC(=O)C(C)Cc2cnn(C)c2)n[nH]1 C(C1=CCN(c2ncnc(Cl)c2Br)CC1)NC(C(C)(C)SC)=O N1(C(CC=CC)=O)CC2(CC(NC(c3sc(F)cc3C)=O)CO2)C1 C1(CCNC(C=CCC)=O)CSCCN1C(C1CC(O)(c2cccnc2)C1)=O N1(C(c2ccc(C)nc2Br)=O)CCC(F)(F)C(NC(c2cccc(F)c2O)=O)C1 S(=O)(=O)(c1cc(C)cnc1NCC(C)(C)CC(C)O)NC(CCCC)C C1(CNC(c2c(CC)occ2)=O)N(C(c2ccc(F)cc2F)=O)CCCC1(C)C CC(C)(C)C(C#N)C(=O)N1CCCC(F)(C(=O)NCC2C3CCCC23)C1 CC1(O)CC(=O)NCC1NC(=O)C=CI.C1(C2CC2)CC1 c1(CC)[nH]nc(C(N2CCSCC2c2nc(C)no2)=O)c1Br c1(CCC)nc(C)c(C(=O)NC(C)(CNC(C2(COC)CC2(F)F)=O)CC)o1 C12(CNC(c3ccc(C(C)C)o3)=O)CC(CO1)N(C(=O)CSCCC#N)C2 N1(C(C2N(CC)CC2)=O)CCCCC(NC(=O)COC(C)(C)C)CC1 C(=O)(CCC(=O)C(C)(C)C)NCC1(CN=c2cc(C)nc[nH]2)CCCC1 C(=O)(C1CCCc2n[nH]cc21)N(CCCNC(c1c(C)cccc1)=O)C(C)C c1(CC)noc(CC)c1CC(=O)NC1CCC(F)(CNC(=O)C(C)CC2CC2)C1 N1(C(C(CC)NC(C)=O)=O)CCN(C(=O)C(F)CC2CCOC2)C(CO)C1 N(C(=NCCc1nccs1)N)CCCC1C(C)C1.c1(C2(C)CCC2)ccc(Cl)cc1 CCC(C)(C)CC(=O)N(C(C)C(=O)N(CCCCCO)C)CC C1(NC(=NC)NCc2ccc(COC)cc2C)CCc2nnc(C)n2C1 C=CCCCCCC(=O)NC1CC(F)(CNC(c2ccc(C)c(CC)c2)=O)C1 CC1(C(=O)N2CCC(C)(NC(=O)CCC(F)F)C2)OCCc2ccccc21 N1(C(C2N(C)CC(C)(C)C2)=O)CC(NC(=O)CCC2(C)CC2)Cc2ccccc21 C=CCC(C)(CNC(=O)CCOCCN(C)C(c1n[nH]c(C)c1Cl)=O)CO N12c3ccccc3CC1C2=O.C1(N(C)C(C2(COC)CC2)=O)CCN(C(N)=O)C1 C(CCC(C)C(=O)N(CCCCCC(=O)NCC(F)C(C)(C)O)C)NC(C)=O Cc1cccc(CN2CCC(CC(F)F)(C(=O)O)CC2)c1[N+](=O)[O-] c1(C(N2CC(NC(C3(O)CCOC3)=O)C2)=O)csc(-c2ccsc2)n1 C1(CBr)NC(=S)N2C(C3CCN(c4cc(F)cc(Cl)c4)C3)=C1C2=O.CCS(=O)C1CC1 CC1Cn2nccc2CN1C(=O)COC1CCN(C(C2(C#N)CCCOC2)=O)C1 C1(C(=O)NCCCN(C(=O)CS(=O)(=O)N(C)C)C)CC12CCC1(CC2)OCCO1 C1(N(C(C)=O)Cc2n[nH]cc2Br)CCCN(CC2CCCO2)C1 CCC(C)(C)CCNC(=O)CC1CN(C(=O)C=CC(C)C)CCO1 C1(NC(C2C(C=C)CC2)=O)CN(C(=O)C=CC(C)C)Cc2nccn2C1 CN1CCC(C2CCCN(C(c3cn(CCC4N=N4)nn3)=O)C2)CC1 O=C(C#CC1CCCCO1)N1CC(N2CC(NC(C3CC(CF)C3)=O)CC2=O)C1 C1(C(=O)OC)CCCN(CC(=O)NC2CC2NC(c2cnnn2C2CC2)=O)C1 c1(C(=O)NCC(C)=CC(=O)N(C)CC2CN(C)CCO2)cnncc1O N1(C(c2c(C)cc[nH]2)=O)CCC(CCNC(=O)CC2CCCO2)C(F)(F)C1 C1(CNC(=O)Cn2nnc(=O)[nH]2)CCC(NC(C2C3CCCCC23)=O)CC1 CC(O)(CC(=O)NCc1cccc(CNC(C2CCCCS2)=O)c1)C(F)(F)F CC1(CNC(c2csnc2Br)=O)CCCN1C(C1OCC1(C)C)=O C(=O)(C(C)(C)CC(F)(F)F)NCC(C)(CNC(c1cnn(CCF)c1)=O)OC C1(O)(CNC(c2cncnc2)=O)CCN(C(c2cc(Br)ccn2)=O)C1 C=CCC(C(=O)NC1(C)CCCC1C)NC(=O)C=Cc1ccncc1 C1(C(=O)OC(c2ccc(OCC)c(Cl)c2)=O)COCC1P(C)(C)=O Cc1cc(=NC2CC2C2CCCCC2)[nH]c(N(C)Cc2ccnn2C(C)C)n1 c1(CCNC(c2n(CC)nnn2)c2csc(Cl)c2)ccc2c(c1)OCCCO2 c1(C(N2C(CNC(=O)CC(C)(O)c3ccccc3)CC2)=O)cc(Cl)c(Br)cn1 N1(C(C2C(=O)NCCCC2)=O)CC=C(C(=O)NCC(O)C(F)(F)F)CC1 c1(OC)ccc(Cl)c(C(F)(F)C(=O)N2CCC(N3CCN(CC=C(C)C)CC3)C2)c1 C1(NC(c2nc(C)[nH]n2)=O)CN(C(c2ccncc2C)=O)CC12CCOCC2 CCCCC(F)C(=O)N(C1CCCN(C(=O)CC2(C)CCCCC2)CC1)C C1(CC(=O)NCC2C(CC)C2)COCCN1C(C1CC(F)C(=O)N1)=O c1(C(C)C)ccc(C(=O)NCC2CCCCCN2C(=O)CC(O)C(C)C)c(F)c1 C1(NC(c2cn[nH]c2)=O)CN(C(=O)CCc2nc3ccccc3o2)C2(CCC2)C1 C1(NC(C(c2ccc(Cl)s2)OC)=O)CCC(C)(NC(=O)C(F)CC2CCC2)CC1 c1(OC)cc(C(=O)NCC(c2ccc(Cl)cc2)NC(=O)C(CO)NC(N)=O)n(C)n1 C1(CC)CN(C(C2CC(F)C(=O)N2)=O)CCN1C(c1ccc(N(C)CC)nn1)=O C(c1c(F)cccc1F)=CC(=O)NC1CN(C(C23CC(O)C2C3)=O)CC1O C1(C(NC(c2ccc(C)c(Cl)c2)c2n(CCOC)nnn2)CC)CCCC(C)(C)C1 CCCCC(O)CCC(=O)N1CCCCC1CNC(c1ccc(CSC)o1)=O Nc1cc(C(N2CC3(C2)CN(C(C2COC2)=O)C3)=O)cc(Cl)n1 C1(C(=O)NC(c2cn(CC3CCCCC3)nn2)(C)C)C(C(=O)O)C1(C)C c1(C(N(CC(CN(C)CCc2ccccn2)O)C)=O)cc(=O)cc(Cl)[nH]1 C1(N(C(C2C(CC)C2)=O)CC)CCN(C(c2cc(C)c[nH]2)=O)C1 Cc1nnc2n[nH]c(NC(N3CCOc4ncccc43)=O)c2c1C c1(C(=O)NCCC2COCCN2C(c2csc(O)n2)=O)cc2cccn2c(O)n1 c1(CC)cnc(O)c(C(=O)NC(C)CN2CCN(C(=O)C(F)C(C)(F)F)CC2)c1 Cc1ccc(O)c(COCC(=O)Nc2cccc(SCC3CCC3)c2)n1 C1C(CCCC)NC(=O)C(CC)O1.C12(CC(=O)NC(C)=O)COCC(C1)C2 C1(C(=O)NCC(C2CCN(C(C(C)SCC)=O)CC2)C)(C(F)F)CCOCC1 C1(NC(c2c(C)scn2)=O)CCOC(CNC(=O)CCCc2cccs2)C1 N#Cc1ccc(N)c(C(=O)NCCCNC(=O)CCOCC(F)F)c1 CC1CN(C(c2cnc(C3CC3)s2)=O)C(C)CN1C(=O)Cc1cccc(F)c1F Cc1cc(CC(=O)NCCNC(=O)C(C)Oc2cccc(Cl)c2)n(C)n1 c1(CC(=O)NC(C)CC(C)NC(C2CC(N(C)C)C2)=O)nc([N+](=O)[O-])n[nH]1 N1(C(C=CC(C)NC(C=CCC)=O)=O)CCC(N2CCCC2)C1 C1(NC(C2(C)C=CCC2)=O)CN(C(C2CC3(CCC3)C2)=O)CC1F Nc1nc(Cl)ccc1C(=O)NCCC1CN(C(c2csc(-c3nc[nH]n3)n2)=O)C1 c1(CCC)cc(C(=O)NCCC2CC(NC(=O)C(CC)N(C)CC)C2)n[nH]1 C1(C(N2CC(C)C(C)(CNC(=O)CCc3cn[nH]c3)C2)=O)CC2(CCC2)CCO1 c1(C(=O)NCCc2c(C)cn(C)n2)ccc(CN2CCOCC2)c(F)c1 C12(CNC(C3CC(SC)C3)=O)CCCC1N(C(c1cc(C3CC3)ns1)=O)CCC2 CC(O)C(C(=O)NCCC(C)NC(=O)CCc1ccoc1)NC(N)=O n1(CC(=O)NC2(C)CN(C(c3cc(C)c(Br)o3)=O)C2)cc(Br)c(O)nc1=O c1(NC(CC=CCNC(C(C2CCC2)OCC)=O)=O)ccccc1O N1(C(CCNS(C)(=O)=O)=O)CCC2(NC(=O)Cn3cccc(N)c3=O)CC2C1 N1(C(=O)N(CCC(c2ccc(F)cc2)O)CC2CCCO2)CCC2CCC(C1)S2 C1(CNC(CNC(CC)=O)=O)CN(C(=O)CCc2nnc(S)n2C)C2COCC2O1 C1(NC(C(C)NC(CC)=O)=O)CN(C(c2cccc3occc23)=O)CC1N=[N+]=[N-] c1(C(=O)OC)cc2c(nc1N1CC(C)(NC(C3CCCSS3)=O)C1)CCC2 Cc1nc2ccc(C(=O)N(CC(C)NC(=O)C(C)(C)c3sccc3Cl)C)cc2s1 Cc1c(C(N2CCCC(CNC(=O)CC(=O)N(C)C)C2)=O)cccc1CO C1(OCC(N2C(C)CCCC2)=O)CCN(C(=O)CCc2ccoc2)C1(C)C c1(OC)cncc(C(=O)NC23CC2CN(C(C2CN(C4CCCCC4)C2)=O)C3)n1 Cc1ccc(COC(C)(C)C)c(Br)c1.C1CC(C)CCNC(=O)C(=O)N1 C1(CS(=O)(=O)NC(CC)CCCO)CCC2(CCOCC2)CO1 c1(C(=O)NS(CCC(CC)CC)(=O)=O)cc(C#N)cc(S(C)(=O)=O)c1 N1(C(C(C)O)=O)CCC2(CC1)OCCC2NC(c1ccc(C(F)(F)F)c(Cl)c1)=O CC(C(=O)N1CCOCC1)C(=O)N(C)CC1(CNC(C2(N(C)C)CC2(F)F)=O)CC1 c1(C(=O)NC2C(CNC(c3c(N)ccc(C)c3)=O)CC2)cccc2ccnn12 C12(NC(c3ccc(C)cc3)=O)CCCC1N(c1ncnc3c1ncn3C)CCC2 C1(CNC(CCN(CCC)C)=O)CCC2CN(C(=O)C=CC=C(Cl)Cl)CC12 N1(C(CCCC(OC)OC)=O)CCC2(NC(=O)C(C(C)C)C(C)C)CCCC12 Cc1nc2ccc(C(=O)NCCCN(CCO)C(C3CCCC(C)CC3)=O)cc2s1 Cc1cc(C(=O)NCCN(C(C2CC3CC3C2)=O)CC2CC2)c(Cl)cc1N c1(C(=O)NCC(CC(F)(F)F)NC(C(C)OC)=O)ccnc2ccc(F)cc12 c1(NC(CCC)=O)ccc2cc(-c3noc(C4CCC(O)C4)n3)[nH]c2c1 C(C(C)C(=O)N1CC(CNC(C2COCCO2)=O)C1)SC C(=O)(CCCC(=O)N1C(CNC(C2(c3ncccn3)CC2)=O)CC2CC12)N(C)C N1(C(CCN(C(c2c(OC)ccs2)=O)C)=O)CC2(C1)CC(C)(F)C2 C(=O)(C1Cc2ccc(C)cc21)N1CCC(O)(CCNC(CSC)=O)C1 C(=O)(C(CC(C)C)C(N)=O)N(CCCOCCNC(c1cccc(C)n1)=O)C S(=O)(=O)(c1cccc(Cl)c1)N1CCC(N(C)C(c2nc(C)on2)(CC)NC)C2(C1)CC2 Cc1c(C(=O)NC2CCN(C(=O)Cc3cnccn3)CC2C)cc(O)cc1N Cc1cc(=O)n(CCC(=O)NC(C(C)NC(C2(CO)CC2)=O)C(C)C)cn1 C1(C(N2CCCCC(NC(c3c(C#N)ccs3)=O)C2)=O)CC2(CCCCC2)CO1 C1(CN)CC(CN)CN1C(=O)C(=O)NC1CCC(c2ccc(F)cc2)CC1 CN1N=C(C(=O)NC2CC(C)(NC(C3CC(=O)N(CC4CC4)C3)=O)C2)CCC1=O Cc1cc(C(=O)NC2CCN(C(c3cnn(C)c3)=O)CC2O)c(C)n1NC(N)=O C1(NC(C(C)C#N)=O)CCCC12CCN(C(c1cc(C(F)F)no1)=O)CC2 C(=O)(C(CC1CCCC1)NC(C1C=CCCC1)=O)N(C)CC1CC1(F)F Cc1nc2cc(CCNCCS(=O)(=O)CCOc3ccccc3)ccc2o1 CCC(CC(=O)NCc1ncc(C(=O)NCC(C)C2CCC2)cn1)C1CCC1 c1(COC(c2c(C)c(Br)cc(Cl)c2)=O)n[nH]c2ccc(Br)cc12 N1(C(C2CCN(C(C(CC)NC(N)=O)=O)C2)=O)CC2CCC1C(O)C2O CC1NC(=O)OC12CN(C(C1CC(O)CN1C(=O)CCc1cccnc1)=O)C2 Cc1occc1C(=O)NCC(=O)NC(CNC(c1cscc1C(F)F)=O)C1CC1 N1(Cc2nnc(C(C)(C)C)o2)CC2CCCN(C(=O)Cc3nn(C)cc3Cl)C2C1 N1(C(CC(O)Cn2ccnn2)=O)CCN(C2CCCCC2)C(=O)C1 N1(C(C(C)C)=O)CCCC(C(=O)NCCOC2CN(C(C3CC(Cl)(Cl)C3)=O)C2)C1 c1(C(=O)NCc2ccc(C(=O)O)o2)cccc(S(=O)(=O)CCO)c1 c1(OC)c(N2CC(OCCN(C(=O)C(C)C3CCCO3)C)C2)ncnc1Cl c1(OC)nn(C)cc1C(N1CCC(O)C1C(=O)NCC1(O)CCC(C)C1)=O C1(NC(CC(C(N)=O)NC(C)=O)=O)CC2CCC1N(C(=O)CC(O)C(C)C)C2 N1(C(c2n(C)c(S)nn2)=O)CCC(NC(C2CC(S(C)(=O)=O)C2)=O)CC(O)C1 CCCC(CCC)CC(=O)N1CCCC1(C(=O)N(C)C(C1CCCC1)C)C(C)C CCCC(O)(CCC)CC(=O)N(C1CN(C(C2C=CCCC2)=O)C1)C N1(C(c2cn(-c3cccc(C)c3)nn2)=O)C2CCC1CC(C(=O)NCCNC=O)C2 N1(C(CNC(C)=O)=O)CCOCC(C)(CNC(C2(CF)CCC2)=O)C1 c1(C(=O)NCC(C)CN(C(=O)CN(C2CCC2)C)C)cc(F)cnc1Cl c1(C(c2snnc2C)NC(C(=O)NC(CC)(C)C)C)ccc(C)s1 c1(SC)ccc(C(=O)NCC2CN(C(=O)Cc3csc(C)c3)CCO2)c(Cl)c1 C1(CC)CN(C(c2coc(C)n2)C(=O)OCCC2CC2)CCN1CC(F)F c1(OC)ccc(C(C)C(N2CCCC(CCNC(C3CCOCC3)=O)C2)=O)cc1 N1(C(c2cn(C(C)C)nc2)=O)CC(CNC(c2cn(C)cn2)=O)C(F)(F)C1 C(=O)(C(C)Cc1ccncc1)NCCN(C(C(C)OCC=C)=O)CCC c1(CN2C(C(=O)NCc3c(C#N)cccc3)CCCC2)cnc2ccccc2c1Cl C(=O)(CC(C)C(F)(F)F)NC1C2CN(C(C(C)SCc3ccccc3)=O)CC1C2 Cc1cnc(C(=O)NCC(C)(C)C(=O)N2CCC(N3CC(O)C3)C2)c(C)c1 O=C1CCC(C(=O)NC2CC3(C2)CC3NC(C2SCCCS2)=O)CCO1 N1(C(c2c(C)csn2)=O)CCN(C(C2CCN2C)=O)C2(CC2)C1 C1(NC(CCC(=O)N(CC)CC)=O)CCCN(C(c2c[nH]nc2F)=O)C1C c1(C(=O)NC(CCN(C(C(c2scc(C)n2)C)=O)C)C)cc2sccc2n1C C(=O)(C(C)C(C)COC)NC(CCC)C(=O)N1CCC(OC(C)C)CC1 C(CC(C)(C)C(=O)NC(c1ccccc1O)C)NC(CC(C)CN(C)C)=O C1(C)(CNC(CC2(C)CN(C(=O)CC3CCCSC3)C2)=O)CCOCC1 c1(OC)cn(C)c(C(N2CC(NC(=O)Cc3cnc[nH]3)C3(CC3)C2)=O)cc1=O CCCC(CNC(c1ccc(SC)o1)=O)C(=O)NC(c1ccccn1)C c1(C(N2CC(NC(c3c(CCC)n(C)nn3)=O)C(C)C2)=O)cnc(C)c(N)c1 C1(C(=O)NCC2N(C(C#CC(C)(C)C)=O)CCCC2)CCc2nncn2C1 C(C(F)(F)CN=c1[nH]c(=N)[nH]c(=NC(C)c2nncs2)[nH]1)OC Cc1ccc2c(c1)CCC(C(=O)Nc1ncc(Br)c(C)c1C)O2 CCC(CCC(=O)Nc1cccc(F)c1F)NC(=O)Cn1nc(C)oc1=O Cc1nc(C(N2CCC(C(=O)NCC(=O)NCCC#N)CC2)=O)sc1C.C(N)(=O)N.O CCC(C)CC(=O)NC1CCC(NC(=O)Cc2sc(C3CCC3)nc2C)C1 N1(C(c2cc(C)oc2)=O)CCC(=CCNC(C2CCCC(O)C2)=O)CC1 CCCCCCCCCCC(=O)NC12CC(NC(=O)CCCC(O)C(C)C)(C1)C2 c1(CC)cc(N)c(Cl)cc1C(=O)NCC1CCC1CNC(=O)CC1(CO)CCC1 c1(NC(=O)NCC2C(c3n(C)ncc3)OCCC2)ccc(O)cc1F Cc1cnc(CCC(=O)N(C)CCN(C(=O)C(C)CC2CCCC2)C2CC2)[nH]1 c1(C(=O)NC2CN(C(C3(C)CC(C)=C(C)CC3)=O)C2)cc2c(=O)[nH]ccn2c1 C1(C(=O)NCC2(CC)CN(C(=O)C(c3ccccc3)C)C2)(OC)CCCOC1 C1(CNC(C2C(c3c(C)nn(C)c3)C2)=O)CCN(C(=O)C2=CCCC2C)C1(C)C c1(C(N2CC(NC(C(C)OCC)=O)C(OC)C2)=O)cc(C)ccc1C CC1CN(C(=O)COC2CCCC2)CC1CNC(=O)C=Cc1ccc(C(N)=O)o1 c1(C(=O)NCCC(C)NC(c2ccc(-c3cccs3)o2)=O)ccc(N)c(Cl)c1O c1(C(CCOC)NC(c2nnnn2CCCOC)C2CCC2)cc2ccccc2o1 C(=O)(CCCCN1CCOCC1)N1CCC(C(C)NC(c2cc(OC)n[nH]2)=O)C1 c1(-n2cc(C3CN(N4CCC(C)(F)C4)C3)nn2)cc(F)cc(Br)c1 N1(C(C23CC(C(=O)Nc4c[nH]ccc4=O)(C2)C3)=O)CCc2c(ccc(F)c2Br)C1 C1(NC(C2CCN(CC)C2)=O)CN(C(c2cn(CC)nn2)=O)CC1F C(N=c1cc(Cl)nc[nH]1)C1CN(C(c2cc(CC)no2)=O)C(C)C1 N1(C(c2cn(CC=C)nn2)=O)CCCCC1CCN(C(=O)CN(C)S(N)(=O)=O)C C1(C(C(C)C)NC(CCCOCC=C)=O)CCN(C(=O)C(CC)NC(C)C)CC1 c1(C(N2CC(CNC(c3c(C)occ3)=O)C(O)C2)=O)cc([N+](=O)[O-])cnc1N c1(C(N2CCC(CCNC(c3ccc(CC)[nH]3)=O)C2)=O)c[nH]c2nccc(Cl)c12 C1(CC)C(C(=O)N(CC(C)(C)NC(=O)C=CBr)C)CCN1C CC1CN(C(=O)C=Cc2cc[nH]n2)CC1C(N1CCOC(C)C1)=O C1(NC(CCCOCC)=O)(CNS(C)(=O)=O)CCN(C(=O)C(C)(C)NC)C1 Cc1csc(C(N2CCN(C(c3cn(C)nc3-c3ccoc3)=O)CC2)=O)c1Br c1(C(N(C2CCC(CNC(=O)CNC(=O)OC(C)(C)C)C2)C)=O)cnc(Cl)s1 c1(C(=O)NCC2C(C)(C)N(C(C3CCCC3)=O)CC2)cn2ccccc2n1 Cc1ccc(CNC(C2CCOC2)CO)cc1Br c1(C(N2CCC(NC(CSCC(C)C)=O)C2C2CC2)=O)cccc2c1OCCC2 C1(C(=O)O)(NC(=O)NC(c2cccnc2)CC2CCOC2)CCCCC1 CC(C)(C)CCCC(=O)NC1(CNC(=O)COc2ccccc2F)CCOC1 C=CC(C)CC(=O)NCCCC1CCCN1C(c1sccc1-n1cnnn1)=O c1(C(=O)NCC(CN(C(=O)C(C)SC)CC)(C)C)cn2c(n1)SCC2 c1(NC(C2N(C(CC(C)O)=O)C3C(C2)C3)=O)cc(O)nc(Cl)n1 Cc1c(CNC(=O)C(=O)NC(c2c(Br)c(C(F)(F)F)nn2C)C)cccc1Cl N1(C(c2ccn(C)c(=O)c2)=O)CC2CCCN(C(C3C4CC5C(C4)C35)=O)C2C1 N1(C(C2CC(CNC(CCC(C)OCC)=O)OC2)=O)CCC2(CC1)N=N2 C(CCC(C)C)(C(=O)NCCC(C(C)C)N(C)C)NC(c1c(OC)cc(C)s1)=O c1(CNC(=O)CC2CC(O)CN2C(=O)CC2CCCO2)cc(F)cc(Cl)c1 C12(CC(=O)NCCCCC(C)NC(C(COCC)C)=O)CC3CC(CC(C3)C1)C2 N1(C(CC=CC)=O)CC23CCCC2(C1)CN(C(=O)C(=O)N=S(C)(C)=O)C3 C1(O)(CNC(c2cncnc2C2CC2)=O)CCN(C(c2coc(O)n2)=O)C1 N1(C(C(C=C)O)=O)CCOC2CCN(C(c3ccccc3NC(=O)OC)=O)CC12 C=CC1CN(C(=O)CC(C)C(C)C)CC1NC(=O)C(C(=O)OCC)OC C1(N(C(=O)CCC=CC)CC#C)CCN(C(=O)C(O)C2CCCC2)CC1 c1(CNC(=O)NCC2(COC)CC(C)(C)C2)cc(OC)ccc1C C1(C)(C(=O)NCC2N(C(c3c(CC)scc3)=O)CCC2)CC2CCC1C2 N1(CC(=O)N(CC(C)O)CCNC(=O)Cc2cnns2)CCCNS1(=O)=O C1(C(=O)NCC2(CC(N3CCOC(CCO)C3)=O)CC2)(CC)CCCCC1 CCC(C(=O)N1CCCCCC1C(=O)NCc1cc(C)cc(F)c1)C(F)(F)F S(=O)(=O)(c1cccc2cnc(Cl)cc12)NC1CCCN(C)C1 c1(OC)cc(C)c(C(=O)NC(C)C(C)NC(C2(C3CC3)CC=CC2)=O)c(F)c1 C1(NC(c2ncn(C(C)C)c2)=O)CCC(CNC(c2nn(C)cc2Cl)=O)CC1 C1(CC)CN(C(=O)C(n2ncccc2=O)C)CC1C(=O)NC1CN(C2CC2)C1 CC#CCC(CO)NC(=O)COCCCCn1cc(CC(O)C(C)C)nn1 C1(F)(C(=O)NCC(CNC(C2CC(CF)C2)=O)OC)CCC(F)(F)CC1 CCCCCC(C(=O)N(CCCNC(c1csc2ccncc12)=O)CC)C(C)C C(=O)(C(CNC(C1CC(CNC(C23CC(C#N)(C2)C3)=O)C1)=O)CC(C)C)OC S(=O)(=O)(c1cccnc1Cl)NCC1CCC(NCc2ncn(C)c2)CC1 C(C(O)C(=O)NCCOC1CCN(C(=O)Cc2ccn(C(F)F)n2)C1)=CC N12CCCCC1CC2=O.c1(C(NOCc2cn(CC=C)nn2)=O)cc(Cl)n(C)n1 C(=O)(C(F)CC(C)C)N(CCOCC)CCN(C(C1(C#N)CC2(CC2)C1)=O)CC CCC(CC(=O)NCCN(C(C1CC(=O)CC(=O)N1)=O)C1CC1)CC(C)C C1(NC(=O)NC(C)C(=O)NCc2n[nH]c(-c3ccccc3)n2)CCOCC1 C1(NC(CC(C)CF)=O)CC2(C1)CN(C(C1OCCC1c1ccccc1)=O)C2 N1(C(c2c(CNC(C3CC(C)C(=O)CC3)=O)cc[nH]2)=O)CC2CC(C1)N(C)C2 Cc1ncsc1C=CC(N1CCCCC1CCNC(=O)C(c1cncnc1)C)=O c1(C(C)C)nnc(C=CC(=O)NCC(CNC(=O)Cc2nc[nH]n2)CO)o1 N1(C(c2cc(C)n(C)c2)=O)CCC2(C1)CN(C(=O)C(C)CSC(F)(F)F)CCO2 c1(C(=O)NC2CCC(NC(=O)COCC3CC3)CC2)nnn2c1C(=O)NCC2 C12(CNC(C(N3CCC(C(C)C)C3)=O)=O)CCOCC1C2 c1(C(N2C(C(=O)NC(C)CC)CC(=C)C2)=O)c(C)ccc(I)c1C c1(N(CC(CN(C)C(C2(C)C=CCC2)=O)O)C)cc(Cl)nc(-c2ccccn2)n1 C1(NC(COCCN(C)C)=O)CC1C1CCCN(C(C2(CO)CCOCC2)=O)C1 C(=O)(C(C)C(O)C(C)C)N1CC(C(C)NC(c2c(C)ccc(CC)c2)=O)C1 CCC(O)(CC)CCNC(C1CC2CCC1N2C(=O)COC1(C)CCC1)=O C1(C(C(=O)N(C2CCCC2)CC=C)C)CN(C(=O)CC(C)(C)C)CCO1 C1(C(N2C(CCNC(CCSC)=O)CSCC2)=O)Cc2ccccc2NC1=O C1(CNC(=O)OC(C)(C)C)CC2(C1)CN(N1CCCC3(C1)N=N3)C2 C1(C(=O)NC2CN(C(C3CCCN(CC)C3)=O)CC2F)CCC(=O)N(C(C)C)C1 Cc1cccc(C(=O)NCc2ccoc2C(=O)NCC=C(Cl)Cl)c1O C(CO)(CCCCNC(c1ccc(=O)n(C2CC2)c1)=O)NC(=O)Cn1ncnn1 C=CC(CCC)CC(=O)NC1(C)CCN(C(c2nc3c(s2)COCC3)=O)C1 c1(SC)nccnc1C(N1CCN(C(C)CNC(C2CCC(=O)C2)=O)CC1)=O C1(C(=O)NCC(C(=O)NCC2=CCCOC2)N(C)C)CCCCC(=O)N1 C(CC(C)(C)C(=O)N1CC(CC(F)C(=O)NC(C(O)CO)C2CC2)C1)SC C1(C(=O)NC(C2CC(NC(c3cc(OC)no3)=O)C2)C)CCCSC1C c1(C(c2n(CC)nnn2)NC(C)CCCOC)ccc([N+](=O)[O-])c(C)c1 C(=O)(C(C)CC(F)(F)F)NCC1CCC(NC(C(N2CCCCC2)C)=O)CC1 Cc1ncc(C#N)c(N2CC3C(C(=O)N(CCCOc4ccccc4)C)C3C2)n1 C1(NC(C(CC)OCC)=O)CCN(C(=O)Cc2cc(C)on2)C(C)C1 N1(C(CCc2ccc(OC)c(OC)c2)=O)CCC2(CC1)CC2C(=O)NCC(C)C C(=O)(C(C)S(N)(=O)=O)N(CC(CC)NC(C(=O)NCC)=O)C C1(C(=O)NCc2ccn(C3CCC3)n2)(CNC(c2cnc(O)o2)=O)CCCC1 CCCCC(C)CCC(=O)NC(C)(CNC(=O)CCCCCCOC)C1CCC1 C1(NC(C(C=CC)O)=O)CC2CN(C(C3(c4ccc(OC)cc4)CC3)=O)CC2C1 C=C(C)CC(C(=O)N(C1CCN(C(=O)C(C)NC(C)=O)CC1)CC)OC c1(NC(CNC(c2cc(C)on2)C)=O)ccc(N2CCOCC2)c(C)c1 N1(S(c2ccc(C)c3c2nccc3)(=O)=O)CCC2(CC1)COC(C)(C)OC2 CCCC(CNC(=O)Cc1ccc(O)cn1)C(=O)NC1C2CCN(CC2)C1C C1(C(N(CCC(=O)Nc2cn(C3CC3)nn2)CC=C)=O)C=CCCC1 C(=O)(C#CC1CC1)NC(c1ccccc1)C(C)NC(COCCC)=O C#CCCCCC(=O)N1CCC(NC(=O)C(c2ccccc2)=O)C(C)C1 c1(C(=O)NCC2(F)CC(NC(C3N(N=O)CCCC3)=O)C2)ccc2occc2n1 C1(N(C(=O)C(O)CC2CCOCC2)C)CCC(NC(c2cccnc2)=O)CC1 C(=O)(CCC(C)CC)N1CCC(CNC(CCC(=C)Cl)=O)CC1 O(N1CCC(N=c2[nH]c(=NC(C)c3csnn3)[nH]c3ccc(OC)cc23)CC1)CC C1(OC)CC(C(=O)NNC(=O)C2CCC(F)CC2)C1(C)C C1(=O)C(C)(CC(C)C)N1.C12(CNC(CCCC)=O)C3C4C5C3C1C5C24 c1(C(=O)NC(CC(C)NC(Cc2n[nH]c(=NC)s2)=O)C)ccc2c(n1)CCCN2 c1(OC)cccc(C(N2CCC2C(=O)N(C)CCN2CCCC2=O)=O)c1 N1(C(c2ccc(C(C)=O)cc2F)=O)CC2(C1)SCCC2NC(=O)CCF c1(NCC(c2cn(CON3CCCC3)nn2)OC)nn(C)c2c1CC(C)(C)CC2 C1(C2CCCOC2)(NC(C2(F)CCCN(C(Cc3cn(C)nc3)=O)C2)=O)CC1 c1(NC2C(NC(=O)CCC(=O)N3CCC(O)CC3)C2)ncc2c(n1)CCNC2 C=CC1(C(=O)NCC(C)(CC)C(N)=O)CCN(C(C2CN(C3CCC3)C2)=O)C1 N1(C(c2nc(CC)[nH]n2)C)CCCC(C(C)NC(c2cc(C3CC3)n(C)n2)=O)C1 C=C=CCC(=O)NC1(COC)CN(C(c2ccnn2CC2CC2)=O)C1 C1(CNC(C2(CCOC)CCC2)=O)CCN(C(C2CC2C(F)(F)F)=O)CC1(F)F C1(S)CCC(F)(F)CC1.N1(C(c2csc(C)c2)C(=O)NC)CCCC(N(C)C)C1 C(=O)(C(F)C(=O)NCC12CC(NC(c3ccc(O)nc3)=O)(CO1)C2)OCC C(=O)(CC(C)(C)C(F)(F)F)NCC1(OCC)CN(C(C2CCCC(=O)N2)=O)C1 C(=O)(C1c2c[nH]nc2CCC1C)N1CCC(NC(c2c(C)ccc(Cl)c2)=O)CC1 C12(CC)CN(C(C3CSCN3C)=O)CC(C(=O)O)(C1)C2 c1(N2CCC(OC)(COC)C2)nc(N2CCC3(CCCO3)C2)c2c(n1)CSC2 CCC(CCC(=O)NCC1N(C(=O)CCCc2ccc(C)o2)CCC1(C)C)OC C(=O)(C1CCOc2ccccc21)N(CC(O)CNC(C1(C#N)CCSCC1)=O)C CC(C(F)F)=CC(=O)NC1CCC1C(=O)NC1(CC2CC2)CC1 c1(C(=O)NCC(N(C(C(CC=CC)C)=O)C)C2CC2)cc2sc(C)nc2[nH]1 O=C(N=S1(=O)CCC2(CC1)CNC(=O)C2)c1cccc([N+](=O)[O-])c1 CCCC(CCC)CC(=O)NC(C)CN(C(=O)C=CC1CCCCC1)CC Cc1ccc(F)c(NC(=O)C(C)NC(c2cn(-c3ccc(F)c(Br)c3)nn2)=O)c1 C1(CCC)(NC(=O)CCn2ccnn2)CCCN(C(c2cc(C)c(C)o2)=O)C1 C1(NC(c2cnns2)=O)CCN(C(C2CCCC2)=O)CC1 N1(C(=O)CCCN2Cc3ccccc3C2=O)CCCc2c1ccc(Br)c2F c1(C(=O)OC)ccc(C=CC(=O)N(C)CC2CN(C(C3CCCS3)=O)CCO2)o1 O=C(C1=CSCCO1)NC1CCN(C(c2cn(CC3CCCO3)nn2)=O)CC1F N1(C(CCSC)=O)CC2CC(CNC(=O)COc3ccc(Cl)c(C)c3)CC1C2 c1(NC(C2OCCN(Cc3c(OCOC)cccc3)C2)=O)ccc2ncnn2c1 N1(C(C2C(CC(C)C)C2)=O)CC2CC(C(=O)NC(C3CCOC3)CO)C(C2)C1 c1(CCC(N2CCC(N(C(=O)CCF)CC)C2)=O)ccc(Cl)cc1Cl Nc1ccc(C(=O)NC2CC(F)(CNC(c3nc(Cl)sc3Cl)=O)C2)cc1Cl c1(OC(CC#C)C)cccnc1NC(c1cccnc1C(F)(F)F)=O c1(C(=O)NCC(C)N(C(=O)CC2C=CS(=O)(=O)C2)C)cncc(C(=O)N(C)C)c1 c1(C(=O)NC(CNC(c2c(C)cc(F)s2)=O)C(C)C)ccc2c(O)nncc2c1 N1(C(c2ccn(C)c2)=O)CCC(C)(CCNC(=O)CC2CC3CC3C2)C1 CC(C)(C)C(C)(O)C(=O)N1CCC(O)(CCNC(=O)CSC(F)F)C1 C(C1CCCC1)=C(C)C(=O)NCCNC(c1cc(-c2cccs2)cs1)=O C1(CNC(C2C(C)CCC2)=O)CC2(CO1)CN(C(=O)Cc1ccc(C#N)nc1)C2 c1(C(N2CCC(CNC(C3(CO)CCC3)=O)C2)=O)csc2cccnc12 C=C1CCN(C(C2CCC2OCC)=O)C(C(=O)N(CCCCCCC)C)C1 C1(NC(CC2C(OCC)COCC2)=O)CCCN(C(=O)Cn2cc(C)cn2)CC1 ONC(=O)CSC(CC)C.C1(CC)CCC1 Cc1cc(C)c(C(=O)NCCCOCCCNC(C2CN(C)C2)=O)c(C)n1 c1(C(=O)NC(CN(C(c2csc(S)n2)=O)CC)C)cc(Cl)ccc1C(F)F c1(C(=O)NC2(CC)CCCN(C(C(CC)C(C)C)=O)C2)c[nH]c2cccc(Cl)c12 c1(C(=O)NCC(CN(C(=O)CCCN(C)C)C)(C)C)cccc(C(F)(F)F)c1 C1(C(N(C2(CC#N)CCN(C(C)=O)C2)C)=O)CC2(CC(NC(=O)OC(C)(C)C)C2)C1.CO N1(C(CNC(C)=O)=O)CC2CC2C1C(=O)NC(C(C)(C)O)C1CC1 C1(C(=O)Nc2cn(C)nc2)CN(C(=O)Cc2ccccc2C#N)CCC1O N1(C(Cc2cccc(C)c2Cl)=O)CCCC2(NC(c3cccc(Cl)n3)=O)CC2C1 CCC(CC)(CCNC(C1CC2(CC(N(C)C)C2)C1)=O)NC(=O)CCS(C)=O c1(-c2ccccc2)nc2nn1C2.c1ccccc1.n1(C)cncn1 N1(C(C(COC)N(C)C)=O)CC(C(=O)NCCCC2CCC2)C(F)(F)C1 CCC(C)(C)C(O)C(=O)NC(C)CCNC(=O)CCC(=O)N(C)C(C)C Cc1ncnc(C)c1CC(=O)NC(C1CCCC1)CNC(=O)C=Cc1ncc[nH]1 c1(C(N(CC(C)NC(C2(F)CCCCC2)=O)CC)=O)ccc2[nH]c(C)c(C)c2c1 c1(OC)cc(O)ncc1C(=O)NC1CC1NC(=O)Cc1cccnc1C c1(C(N2CCC(CNC(c3c(C)ncnc3)=O)C2)=O)ncncc1C#N N1(C(c2ccc(C)cn2)C(=O)NC(C)(C)C)CC(=O)NC2CCCC2(C)C1 Cc1c(C(N2CC(O)(CNC(c3ccsn3)=O)C2)=O)c(Cl)nn1C c1(CCC(=O)NC2CC(NC(c3n(C(C)C)nnc3)=O)C2)ccc(F)c(F)c1 N1(C(C2C(C(C)C)OCC2)=O)CC2CCCC2(NC(C2CN3CCC2CC3)=O)C1 C1(NC(=O)Cc2cccnc2O)CC2CCC(C1F)N2C(c1ncc[nH]c1=O)=O CC1CCN(c2nc(NCCc3nccs3)c3ncsc3n2)CC12CCC2 C1(C(=O)N(C2CC2)CC2CCCN2C(c2cc(Cl)ccn2)=O)(OC)CS(=O)(=O)C1 Cc1ccc(CC(=O)NCC2CCCOC2(C)C)cc1Cl N1(C(c2cnc(C)s2)=O)CCC2(CCCC2NC(C2CN(C(N)=O)C2)=O)CC1 C1(NC)CC(C(=O)NCC(=O)NC(C)COC)N(S(C)(=O)=O)C1 c1(CC)nc(Cl)cc(=NC2CCCCN(C(=O)C3=C(C)S(=O)(=O)CC3)C2)[nH]1 Cc1cc(C(=O)NC2CCN(C(=O)C3=NOC(C)C3)CC2O)cc(F)c1 C12(C(=O)N)C3C4C1C1C2C3C41C(N)=O.c1(COC)nc(N2CCNCC2)cc(C)n1 C1(=CC(=O)N(C(C)C(C)n2cccn2)CCO)CN2CCC1CC2 N1(C(CCSCC)=O)CC2CC(NC(c3ccc(N(C)C(C)C)cc3)=O)C2C1 C1(CC)CN(C(=O)CCC2CCC(=O)C2)CC1NC(C1(C)CCOC1)=O CC1CN(C(=O)CCCOc2ccccc2)CC1(C)CNC(c1nsnc1O)=O C(=O)(C(C)(C)CC(F)(F)F)NC1C(CN(C(=O)C(c2cccn2C)=O)C)CC1 C#CCCN=C(NCC(c1ccc(C)cc1)C1CCC1)N1CCC(NC(C)=O)C1 N1(C(C2C3CCN(C(C(CC(=C)C)OC)=O)CC32)=O)CC2CCCC(C1)N2C C1(NC(C2(C(=O)NC)CCOCC2)=O)CCN(c2ncc(C)cn2)CC(C)(C)C1 C1(CCCNC(C2CN(CC)C2)=O)CCCN1C(=O)CCc1cc(C)no1 N1(C(Cc2ccn(C)n2)=O)CCC(NC(=O)Cn2nnc(C3CC3)n2)C12CCCC2 C(=O)(CC(C)(O)C(F)(F)F)NCCN(C(c1c(C)cccc1Cl)=O)CC1CC1 C=CC(Cc1nc(C(C)O)nn1-c1ccc(OCC)cc1)CCC CCCCCCC(O)CCC(=O)NCC(C(C)C)NC(c1ccn(CC)c1C)=O C(=O)(C1=CCC(C(F)(F)F)OC1)NCCCC(C)(C)NC(=O)CC1CC2CC2C1 C1(NC(C2CCCS2)=O)CCC2CN(C(C3(F)CCS(=O)(=O)C3)=O)CCC2C1 C1(NC(C2(N(C)C(C3COCOC3)=O)CC2)=O)CCC(CC2CC2)CC1 C1(C(=O)NC(C(N2CC(C#CC)C2)=O)c2cccs2)CCC(=O)N(C)C1 C1(CCNC(C(=O)NC(C)C)=O)CCCN(C(=O)CCN2CCC(F)C2)C1 C1(C(NCC)C)CCN(C(=O)C(C)CCN(C)C)CC1.C1(C=O)(CF)CC1 N1(C(c2nc(C)oc2C)=O)CCC2(CC1)CCN(C(=O)C(C)Oc1ccccn1)C2 N1(C(C(CC)F)=O)CCCC(CCCCNC(=O)CNC(=O)CN(C)C)C1 C=CCN=C(NCC1(C)CCC(C)(C)CC1)N1CCC(OC(=O)N(C)C)CC1 C(CN=c1nc2n([nH]1)CCN(C)C2=O)OC(CCN1C(C)CCCC1)=O C1(COC)(NC(c2[nH]nnc2C)=O)CCN(C(c2cc[nH]c2)=O)CC1 N1(C(c2ccnn2C2CC2)=O)CC2OCC(NC(C3(Br)CC3)=O)C2C1 N1(C(c2n(CC)ccc2)=O)CCC(CNC(c2cc(C(C)C)n(C)n2)=O)C1(C)C N1(C(c2n(CC)ccc2)=O)CCCC(N(C)C(c2sc(C(C)C)nc2C)=O)C1 N1(CCC)CCC(N(CCC)CC2CC(F)(CN)C2)C1.C1(=O)CN1C Nc1cc(Cl)cc(Cl)c1C(=O)NC1CCN(C(C2CC3C=CC2C3)=O)CC1 Cc1c(C(=O)NC2CN(C(C3CCCN3C(C)C)=O)CC2O)sc2ccccc12 C(=O)(CCCC(C)(C)NC(C1COCC1C(N)=O)=O)NC1C2(CC(OCC)C2)C1 c1(N2CCC(C)C2)cc(C(=O)NC2CC(NC(=O)C=CCN(C)C)C2)ccn1 Cc1ccc(C(N2CCOCCC2C(N2CC(N3CCC3)C2)=O)=O)c(C)c1 c1(NC2C(C)CN(C(=O)CCOCC(F)F)C2)cc(C(F)(F)F)nc2ncnn12 C(F)(C(=O)Nn1cccn1)C1OCCN(C(C(C2CCC2)OC)=O)C1 N1(C(c2nc(C3CCOCC3)no2)C)CCOC(C(=O)O)C1 c1(NC(C2(COC)C=CCN2C(=O)C(O)C(F)(F)F)=O)cnc(C)c(C)c1 C1(NC(CC2(OCC)CCC2)=O)(CNC(C2CCCO2)=O)CCCCCC1 c1(OC)noc(NC(=O)NC(C)C(C)n2cncn2)c1Br S(=O)(=O)(c1cccc(C)n1)N1CCN(Cc2ccc(NC)c(Cl)c2)CC1CO C1(C(=O)NCC2(CO)CCN(C(C3CC(F)C3)=O)C2)OCC2COCCC12 C1(N(CC#C)C(C2CCCC2C)=O)CCN(C(c2ccc(Cl)o2)=O)CC1 C1(CNC(C2(S(C)(=O)=O)CC2)=O)CCCCN(C(=O)CC2(O)CCCCC2)CC1 c1(C(N2CCCCC(CNC(CC3C(C)(C)C3)=O)C2)=O)c(F)ccc(N)c1F c1(NC(C2CCC(CNC(CCCOC(C)C)=O)C2)=O)ncc([N+](=O)[O-])cc1F N1(C(c2cnc(C)n2C)=O)CCC2(CCCC2NC(=O)COC2CCC2)C1 c1(C(=O)NCC(=C)CCNC(c2ccnn2CCC)=O)csc(C)c1CC c1(CC)cnn(CC(=O)NCC2(F)CN(C(=O)CC3CC(C)=NO3)C2)c1 c1(CNC(c2ccnc(Br)c2)C(=O)O)cc(Br)cc(F)c1F C1(COC)(CNC(=O)C(=O)NCC(F)(F)F)CCCN1C(=O)CNC(C)=O C12(C(=O)NCC3(OC)CCN(C(=O)Cn4cc(Cl)cn4)C3)CC1COC21CCC1 C1(C(=O)NC(C)CC(C)NC(=O)CN2CCCCC2)CC(=O)OC1(C)C c1(C(N2C(CNC(C3C(C)CC3)=O)CC2)=O)csc(C(C)(C)C)c1 c1(C(N2C(CCC)CN(C(C3(SC)CC(O)C3)=O)CC2)=O)cc2c(=O)[nH]ccn2c1 Cc1ccc(COCC(N2CCCC2CCNC(C2(C)CCOC2)=O)=O)cc1 CC1C(=O)Nc2ncccc2N1c1cc(-c2ccc(N(C)C)cc2)cc(F)c1 Cc1ccc(C(N2CCCC(O)(CCNC(C3CC3C(C)C)=O)C2)=O)c(F)c1C N1(C(C2(C(=O)OC)C(=C)CC2)=O)CCC(NC(c2sc(O)nc2C)=O)C(CO)C1 N1(C(C(C)SC)=O)CC(C)(C)CCC1CNC(c1ccc(C(F)(F)F)c(C)c1)=O C1(CNC(c2n[nH]c(C)c2Cl)=O)N(C(=O)CC2(C#N)CC2)CCCC1(C)C C1(C(C)C)CCCCC1N=c1[nH]c(=N)[nH]c(=NCc2csc(CC3CC3)c2)[nH]1 C1(C(N2CCCC(N(CCOC)C)C2)=O)Cc2cccc(Cl)c2C(=O)O1 c1(NC(C=C)C2CCC2)ccc(S(=O)(=O)NCC2COC(C)(C)CN2)cc1Br CCC(CC)CCC(=O)NC(C1CCCN(C(=O)CN2CCCC2=O)C1)C N1(C(Cc2c(C)scc2)=O)CC(CNC(C2(F)CCCCC2)=O)C2CC12 C(C)(C)(CCCC(=O)N(C1CCCC(C)C1C)C)NC(CSCC(=O)OC)=O C#CC1(C)CCN(C(=O)CC2CCC(O)CN(CC(=O)OC)C2)CC1.C(C)(C)C c1(CNC(N2CCCC2c2cccc(I)c2)=O)cc2c(s1)C1CCC2C1 CC1CCN(C(=O)CCCc2nccs2)CC1NC(=O)Cn1nnc(C2CC2)n1 CCCN=C(NCCCCC(=O)N(C)C)NC(c1cc(Cl)ccc1O)C c1(NC(C2CCN(C(c3cncc(Br)c3)=O)C2)=O)ccc(Br)cc1[N+](=O)[O-] N1(C(C(N2C(C(CCC)C)CCC2)=O)=O)CCC(C)(CO)C1.n12cc(nn1)C2 C=C(C)CC(C(=O)N(CCC(=O)OC(C1COC2(CCC2)C1)=O)C)OC C1(CNC(C2(OC)CC2)=O)(NC(c2sccc2Oc2ccccc2)=O)CCCCC1 C(C1=NOC2CN(C(C3(F)CCCCC3)=O)CC12)NC(c1cnc(O)cc1O)=O N1(C(CC(CC#C)NC(=O)CCc2nc[nH]n2)=O)CCCC(C)(C)C1C C1(NC(CCN(CCCCOC)C)=O)CCN(C(c2c[nH]nc2C(F)F)=O)C1 N1(C(CSCCC)=O)CC2CCCC1(CNC(c1cc(CC)c(CCC)s1)=O)C2 C=C=CCCC(=O)NC(CN(C)C)C(=O)NCCC1CCSC1 c1(C(N2CCCC(Cc3cn(CC4CCOC4)nn3)C2)=O)nc(Cl)c(Cl)s1 c1(OC)ccc(S(=O)(=O)NC2CCCC(Oc3c(F)cccc3Cl)C2)cc1 c1(C(=O)NC2C(NC(c3c(CC)onc3C)=O)CCC2)cc2cn[nH]c2cn1 C(CC1=CCCCC1)NC(C1C(CNC(C(NOC)=O)=O)OCC1)=O C1(NC(=O)CSC2CC2)CC2CC1N(C(c1cnc(C3CCOC3)s1)=O)C2 C1(OC)CC(NC(=O)CSc2nc[nH]n2)CN(C(C23CC4CC2C3C4O)=O)C1 CCC(CC(=O)C1(C(=O)NCCOCC2CCCO2)CC1)SC.C(C)(C)O N1(C(C(CC)(C)CNC(=O)C(c2ccn(C)n2)C)=O)CCC2(CCCC2)C1 c1(NC(C2(C)CCCN(C(CSCC=C)=O)C2)=O)cc(C)c(O)c(C)c1 c1(C(=O)NC(COCC)C)ccc(Cl)c(C)c1O CC1CCCC(CC(=O)NCCc2cc(C(N3CCC4CC34)=O)no2)C1 C(CC)(CC)(CCNC(=O)C=Cc1cnc[nH]1)NC(C1CC(CCC)C1)=O N1(C(C=CC2(C)CCOCC2)=O)CCC2(CC1)CC(NC(=O)C=CCO)CCO2 c1(-c2cnc(C(=O)Nc3nc(O)ccc3F)nc2)ccc2c(c1)OCO2 c1(NC(C2CC(OC)CN2C(c2c(Cl)cnc(Cl)c2Cl)=O)=O)cc(C)c(Cl)cc1C N1(C(CCSCC)=O)C2CCC(C(=O)OC(C)C)C1CC2.C1(C(=O)NC)CCC1 C1(NC(=O)COCCF)CCCCN1C(=O)C(F)(F)F c1(SC)ccccc1C(=O)NC(C)CN(C(=O)CCc1cncn1C)C Nc1cc(C(=O)NCC2(NC(C3CC4(CC4)CO3)=O)CCOCC2)c(F)cc1F N(C1CCCn2cnnc21)c1c(C)c(N2CC(C)C(F)(F)C2)ncn1 C(CS(=O)(=O)C1=CCOCC1)NC(c1n(CCSC)nnn1)c1conc1C1CC1 C(CC(=O)NCC1CC(C2CC2)=NO1)(C(C)(C)C)Nc1c(C)c(Cl)ccc1 C(C(C)(C)C(=O)NC(Cc1cccs1)CCNC(=O)CCc1cnco1)N(C)C C1(OC(C2CCCC(C(F)(F)F)C2)=O)CN2CCC1C2 C1(NC(c2cc(COC)on2)c2nnnn2CC(F)F)C(C)(C)C(O)C1(C)C CCC(Cc1cn(CC(=O)NC)nn1)C(=O)NOCCOCCOC N1(C(COC)=O)CC2CCN(C(c3cn(CCC(C)C)nn3)=O)C2C1 O(N1CCC(CC(=O)NCC2CN(C(=O)Cc3cc[nH]c3)CCN2C)CC1)CC c1(C(=O)NC2CC3CN(C(C(CC)(C)NC(C)C)=O)C2C3)[nH]c2ccccc2c1Cl C1(OC)CN(C(c2cc(C)[nH]n2)=O)CCC1NC(=O)C(F)(F)C(O)C1CC1 C1(C(N2CC3(CCC3O)C2)=O)(CC)CCCN(C(=O)CCNC(=O)OC)C1 c1(-c2c(C)cc(C#N)cc2)nc2c(s1)CCN(Cc1ccn(CCN(C)C)n1)C2 CC(C(=O)NCC1CCN(C(C2CN(c3cnn(C)c3)C2)=O)C1(C)C)C(F)(F)F c1(NC2CC(OCC)C2)cccc(C2(C)CC2(F)F)c1 C12(CCOCC1)C(=O)N2.C1(CN(C2CCOCC2)C=O)CCCC(F)C1 C12(C(N3CCCC(N(C(c4c(CC)nns4)=O)CCF)C3)=O)CC1COC2(C)C O(NC(=O)C1=CCC(NC(C23CCN(CC2)CC3)=O)C1)C(C=C)C N1(C(c2ccn(C(C)C)n2)=O)CC2CCN(S(=O)(=O)c3cnn(C)c3)C2C1 c1(C(c2nnnn2C2CC2)NCc2nc(COC)oc2)n[nH]c(C)c1SC C#Cc1ccc(CC(=O)NC2CN(C(=O)C#CC3CCC3)C(C)(C)C2)c(F)c1 Cn1nc(CCC(=O)NC(=O)CN(CC(=O)O)C(=O)CN2CCNC2=O)oc1=O C(C)(C)(CCC(=O)NCC(C)(C)OCCNC(C1(C)CC1F)=O)OC N1(C(C(C)C#N)=O)CCC(C)(NC(c2cc(CS(C)(=O)=O)on2)=O)CC1 CCCCC(C)(F)C(=O)N1CCCOC(CNC(c2ccn(C3CC3)c2C)=O)C1 c1(NC(C(CNC(c2cnc(C)nc2)=O)OC)=O)cnc2[nH]ncc2c1 C(O)(CN=C(NCC(F)F)NC1CCOCC1)c1ccc(OC)cc1 C#Cc1ccc(OCC(=O)NCCCCCN(C(=O)CCC(=C)Cl)C)cc1 C1(C(N2CC(C#C)C2)=O)C2CC1N(C(C1(OC)CCOCC1)=O)C2 c1(N2CCN(c3cccnc3)CCNC(=S)NCC2)cccc2ncccc12.CC.OC C1(C(N)=O)C2CCC(C2)N1C(=O)CN1CCN(C(c2cc(Br)c[nH]2)=O)CC1 C(=O)(C1=NN(C)C(=O)CC1)NCC(CNC(=O)C(C)(C)CN(C)C)OC C1(C(N(C2CCC(F)(F)C2)C)=O)CCCCCN1C(C1CN(C2COC2)C1)=O C1(CCC(=O)NCC2(O)CN(C(c3noc(C4CC4)n3)=O)C2)CCC(=O)N1 Cc1cc(C)n(CCC(=O)NCCN(C(c2cnc(CO)s2)=O)C(C)C)n1 c1(C(=O)NC2CN(C)CC23CC3)ccc2c(n1)CN(C(=O)C=CCF)CC2 c1(C(=O)NCC(CCCC)NC(=O)CS(=O)C(F)(F)F)ccc(C#N)c(C)n1 c1(C(N2CC(CCNC(C(CCOC)C)=O)C2)=O)ccc2c(c1)CC(C)(C)O2 O=C(CS(=O)(=O)CCO)NC1COCCC1NC(C1(CC(F)F)CC1)=O c1(OC)ncc(CN2CCC2C(=O)NCc2nc(Cl)sc2C)cc1C c1(C(=O)NCC(CC)NC(C2(CC)CCC2)=O)csc(Cc2ccccn2)n1 c1(C(=O)NCC(C)(Cn2cccn2)NC(=O)C=C2CCC2)ccc(C(N)=O)cc1 C=C(Br)CC(C)(C)C(=O)N1C2CCC1C(CNC(c1ccc(C)c(C)c1)=O)C2 C1(NC(CCN(S(C)(=O)=O)C)=O)CC(OCF)CN(C(=O)Cc2csnc2C)C1 C1(NC(c2c(C)c[nH]n2)=O)CCN(C(C2CCC=CCC2)=O)CCC1CO C#CCC(C)(C(=O)N1CCCC(NC(C)=O)CC1)NC(c1cccc(O)c1)=O N#Cc1ccc(=NCC2(NC(=O)CC3=CCOCC3)CC2)[nH]c1C(F)(F)F c1(C(=O)OC)cc(Br)ccc1[N+](=O)[O-].C1CC(=O)N1CC#C C1(CC(N2CC(O)C(F)C2)=O)CC2(C1)CN(c1ncccn1)C2 C1(C(N(C(CNC(c2cc(C)sc2C)=O)C)C)=O)Cc2ccccc2C1 C1(NC(C2CC(OC)(OC)C2)=O)CC(NC(c2cccc(C(N)=O)c2)=O)C(O)C1 c1(C2(C(N3CCCC(CNC(C=CCC)=O)C3)=O)CCCC2)ccc(F)cc1F Cc1cc(CN(C(=O)C(CN(C)C)NC(=O)Cc2ccc[nH]2)C)no1 C(=O)(CC(C)C(=O)NC1COC2(CNC(C3CCN(C)CC3)=O)CC1C2)OC c1(CC)nc(O)c(C(N2CC3CC(C2)C3NC(c2ccsc2C#N)=O)=O)cc1C N1(Cc2c(CC)ocn2)CCC(C2CC2)C1Cn1cc(CC(=O)C(CC)CC)nn1 C(C(N=[N+]=[N-])C(=O)N1CCCC(N(C(=O)Cc2cnn(CC)c2)CC)C1)OCC C(=O)(C(C)CC(F)(F)F)N1CCC(CC#C)(C(=O)NCC(C)(C)CC#N)C1 C(c1ccncn1)=CC(=O)NCCCCN(C)C(C1(n2nccn2)CC1)=O c1(C(=O)NCC(COC)NC(c2ccc(C)c(Cl)c2N)=O)cccc2c1CCC2 C(CN=C(NCC1(N(C)C)CCCC1)NC1CCCC1O)N(CC=C)CC C(CC(F)(F)C(=O)NOCC)c1n(CC)ncc1 C(CO)(CCCNC(=O)C1=NOCC1)NC(C=CCN(C)CC)=O CC1CCC(C(=O)NCCc2ncon2)CN1C(c1cncn1C)=O C1(C(N(CCNC(c2c(CC)c[nH]n2)=O)C)=O)CC(c2ccncc2)=NO1 C12(C(=O)NC3C(O)CCN(C(C(C)=C4CC4)=O)C3)CC3CC(C)(C1)CC(C)(C3)C2 Cc1ccc(CCC(N2CC(CO)(NC(=O)CCC3CNC(=O)N3)C2)=O)cn1 Cc1ccnc(-n2cc(C(N3CCCC(C(=O)O)CC3)=O)nn2)c1Br N1(C(c2cc(C)[nH]n2)=O)CC(NC(=O)CNC(C2CCC2)=O)CCC1C N1(C(CCCOCC=C)=O)CCC2(CCN(C(C3(N(C)C)CC3)=O)CC2)C1 C(=O)(C(C)C(F)(F)F)N1CC2C(C(N3CCCC(OC)C3)=O)C2C1 C1(NC(COCC)=O)CCC(C)N(C(c2csc(-c3cccnc3)n2)=O)C1 Cn1cc(S(=O)(=O)NCc2cccs2)c(CCO)n1 n1(CC)nc(C)c(CC(N2CCOC(CNC(C3CC4CC4C3)=O)C2)=O)c1C C1(C)(C(N(C)CC2N(CC)CCC2)=O)CC(O)CN1C(c1ccc(C)c(F)c1)=O CC1=C(C(=O)N2CC(NC(=O)CN(C3CCCC3O)C)C3(CC3)C2)CCS1(=O)=O C1(C(N(C2CCCN(C(c3ncncc3Cl)=O)C2)C)=O)CCCC1(F)F c1(C(=O)NCC(CN(C(=O)CC(C)(C)OC)CC)(C)C)c(F)ccc(C)c1F N1(C(C(CC)CCOC)=O)CCC(C2(NC(c3cncc(Cl)n3)=O)CCC2)CC1 c1(N(CCC(C)NC(=O)CC2CN3CCC2CC3)C)cccc(F)c1C#N C1(C2CCOCC2)(C(=O)NC(CCNC(c2c(C)cccc2O)=O)C(C)C)CC1 C1(NC(C2C(C=C)C2)=O)CCCN(C(c2ccccc2CN(CC)CC)=O)C1 NS(=O)(=O)CC(=O)NC1COCC1CNC(=O)CCCc1ccco1 C1(CN(C(CC(C)C2CCCO2)=O)C)CCN(C(C23CC(C)(CO2)C3)=O)CC1 C1(n2cc(C(C)(C)OC)nn2)CN(C(c2sccc2C(F)F)=O)CC1SC C1(NC(c2c(CC)sc(=N)[nH]2)=O)COCCN(C(c2oncc2CC)=O)C1 N1(C(c2[nH]c(=NCC)sc2)=O)CC2CN(C(=O)C(n3cc(Cl)cn3)C)CC2(C)C1 N(C(=NCCC1(C)CC(C)C1)NCC1CCCO1)Cc1c(C)scc1 CC(C)(CC(=O)NCCCCCCNC(C1OCCOC12CCC2)=O)C(F)(F)F N12CCOC3C1=CC=CC=C3C(C(=O)O)CCC(O)CCC2 c1(N2CCCC(C(C)NC(=O)CC(F)F)C2)nnc2c(c1C#N)CCCC2 C1(NC(C(C2CC2)SC)=O)CCN(C(c2cn(C)cn2)=O)C1C(C)C N(C(=NCCc1cn(C)c2ccc(F)cc12)N1CCC(SC)C1)C(C=C)C c1(C(N2CCC(CNC(C3(C4CCC4)CC3)=O)C2)=O)cc2nc[nH]c2cn1 N1(C(C=Cc2ccc(CC)o2)=O)CC2(CCCC2NC(c2c(Cl)cnn2C)=O)C1 C1(F)(C(=O)NCC2CCCN(C(C3(C(F)F)CCCO3)=O)CC2)CC2(CCC2)C1 C(=O)(NN1CCCC1C(=O)NCC(F)(F)C(N)=O)C1CCCC(C#N)C1 CC1(C)CC(NC(C2CC(F)C2)=O)CN1C(C1CCC1)=O C(C)(CNC(=O)CCN1CCCC1=O)(C(C)C)NC(c1c(OC)csc1)=O Cc1nsc(N2CCC(C(C)(C)NC(c3cn(CCO)nn3)=O)CC2)c1C#N CC1CCC(CNC(c2ccc(F)s2)=O)N(C(c2cccc(Cl)c2O)=O)C1 C1(NC(C2CCCCS2)=O)CN(C(=O)CCc2ccccn2)Cc2nccn2C1 CCC(CC)(CO)C(=O)NC1CCCC1CNC(c1cn(C2COC2)nn1)=O c1(CC)nncn1CCC(CC1CN(C(=O)NC(c2ccnn2C)CO)C1)=O CC(C)(C)C(C)(O)CNC(=O)NC1CC(Cl)(Cl)C1 N1(C(CCNC(N)=O)=O)CC2(C1)SCCC2NC(C1CC2(C1)CS(=O)(=O)C2)=O C1(C(N(CCC#C)CC)=O)CC(C)N1C(=O)C=Cc1cc[nH]c1 c1(C(N(CCCN(C)C(c2scnc2C2CC2)=O)C)=O)cccc2cc[nH]c12 c1(CC(C(=O)NC2CN(C(c3ccc[nH]3)=O)CC2O)O)c(F)cccc1Cl C1(C(=O)NC2(CN(C(C3(OC)CC3)=O)C)CC2)CCCN(C(N)=O)C1 N1(C=O)CCCC(N(C)C)(CC)C1.n1(CCC)nc(C)cc1C1N(C=O)C(C)CC1 Cn1nc2c(c1C(=O)NC1CC(C)(NC(=O)CC3NC(=O)NC3=O)C1)CCCC2 CC(=O)C(C)(C)CC(=O)N1CCCC(C)C1CNC(c1ccc(C)cc1)=O C1(C(=O)NCC(CC)NC(C)=O)CN(C(c2cncs2)C)CCO1 c1(C(N2CCC(NC(CCCC)=O)(CO)C2)=O)c(Cl)nc2sc(C)cn12 c1(NC)cc(C(N2CCC(CNC(c3cc(OC(F)F)n(C)n3)=O)C2)=O)ccn1 CC1(C)CC(NC(=O)C=CBr)CN(C(c2cc(C3CC3)ccc2F)=O)C1 C1(C(N2CCC(N(OC)C)C2)=O)CCCN1NC(=O)C1CCCOC1 CC1CN(C(=O)C(C)(C)C2CC3(CC3)C2)CCCN1C(C1CC(F)(CO)C1)=O N1(C(C=CCOC)=O)CC(CNC(C2CC23CCC2(CC2)CC3)=O)C2(CCC2)C1 C(=O)(C(O)CCC(C)C)NC1CCN(C(c2c(C)ccc(SC)c2)=O)C1 C1(CC(=O)NC(C=CC(=O)NC(c2nc(C)sc2)C)C)CC2CCCC2C1 Cc1c(Br)ccc(C(N2CCC(CNC(c3nccnc3Cl)=O)C2)=O)c1C c1(CC)cccc(-c2cn(CC(C)NC(C3CCOC3C)=O)nn2)c1 c1(NS(C)(=O)=O)ccc(C(=O)NCCN(C(=O)CC2CCCSC2)CCF)cc1 C(=O)(C(O)CC(C)(C)C)NCC(CNC(C(C)(C)OC(C)=O)=O)O N1(C(=O)OC(C)(C)C)CCC2C(CCCN2C(=O)Nc2ccc(Cl)s2)C1 C(=O)(C(C)CC(C)C(C)=O)N(CC(=O)N(C(CC)C)Cc1nc[nH]n1)C c1(C2C(C(=O)NCCC3CN(C(C(C=CC)O)=O)C3)C2)cc(F)ccc1F CCCC(C(O)C(=O)NOCC1(F)CCC1)NC(=O)CCCCOC(C)C N1(CC(C)C)CC(C(=O)N(C)CC2(NC(c3cncn3C)=O)CC2)CC1=O N1(S(c2ccn(C)n2)(=O)=O)CC2CCN(C(c3cnccc3Cl)=O)C2C1 C1(Cn2cc(CN(CC=C)C)nn2)CN(C(C2CCCOC2)=O)CCCO1 N1(C(C2(C)N(C)CCC2)=O)CCCC2CN(C(c3ccnnc3O)=O)CC12 N1(C(N2C(=O)CCC2CC)=O)CCC2(C1)CN(C(=O)CS(=O)(=O)N1CCCC1)C2 N1(C(C(CC)n2cncn2)=O)CCN(C(=O)C=CCN(CC)CC)C(CO)C1 c1(C(=O)NC(CC)(C)CNC(=O)C(F)OC(F)(F)F)cc(F)cc(N)c1F N1(C(C2C(C)(C)COCC2)=O)CCCC12CCN(C(c1ncccc1Cl)=O)C2 n1(CC)ncc(C(=O)NC2CC(NC(=O)C(C)CCOC)C2)c1Br CC1(C#N)CN(C(=O)CCC2CCCN(C(C3(C)CCCO3)=O)C2)C1 N1(C(CCc2c(C)n[nH]c2C)=O)CCOCC(CNC(C2CCC3CC3C2)=O)C1 c1(C(=O)NCC2N(C(CN(CC)CC)=O)CC(F)C2)ccc2ncc(Br)n2c1 C(=O)(C(F)C(C)(C)O)NCC1C(NC(c2cccc(N(C)C)c2)=O)CCCC1 C1(C(N(C2CCCN(C(=O)C(C)=CC3CC3)C2)CC)=O)CC2CCC(C1)C2O C1(C(CNC(c2nc(C)sc2)=O)(C)O)CCN(C(=O)C(C)C)CC1 CCCCC(C(=O)NCC(CC)(CC)NC(=O)Cc1cccs1)NC(N)=O C(CC(=O)Nc1ccc(F)c(C)c1)(C(C)C)NC(c1ncn(CC)n1)=O c1(C(N(CCCNC(c2cn(CC=C)nc2)=O)C2CC2)=O)ccc2c(c1)CC2 C1(C(N2CCN(C(C)=O)CC23CC3)=O)CCn2c(cnc2Br)C1 c1(OC)cc(OC)c(C(N2CCC(CNC(=O)C(C)C(F)F)C2)=O)cc1OC C1(C(N2CC3C(NC(CC(CC)(F)F)=O)(CC3)C2)=O)CCc2c(n[nH]c2C)C1 C(=O)(C1=CS(=O)CCC1)N1C(C(C)C)CN(C(=O)CC(C)(C)O)CC1 c1(CCC)cccc(C(N2CCCC(CN(C)C(C3CCNC3=O)=O)C2)=O)c1 C(CC(C)C(=O)NCC1CC(O)CN1C(c1ccc(C(C)(C)C)s1)=O)OC c1(CC(N2CC(CN(C(CC)=O)C)C2)=O)cc(OC)c(O)c(OC)c1 c1(OCC#C)ccc(SCCN(C(CCOC(C(=O)NC(CC)O)C)=O)CCC)cc1 Clc1ccc2c(c1)CN(Cc1cccc3ccccc13)C2 N1(C(C2N(CC)CCC2)=O)CCC2C(CCN2C(c2ccc(F)cc2)=O)C1 c1(C(=O)NCC2(C(N)=O)CN(C(CC3CC(OC)C3)=O)C2)cn2cccnc2n1 c1(NC(C2N(C(c3cnn(C)n3)=O)CCOC2)=O)cccc2c1CCO2 c1(CC)cc(F)ccc1C(=O)N(C1CCC(NC(=O)C2=CC(C)(C)C2)CC1)C N1(C(C2C(CC(C)C)C2)=O)CC(CNC(=O)CCC(=O)c2cnn(C)c2)C(C)C1 C1(C(N(C)Cc2cc(C)on2)=O)CCCCN(C(c2cnc[nH]c2=N)=O)C1 CCC(C(=O)N1CCCC1CC(=O)NOCC(O)CO)OC N1(C(COCCCC(C)C)=O)CC(NC(=O)CSc2ccccn2)C2CC12 Cc1cc(=NCc2cn(C3CN(C(C4CCC(C)C4)=O)C3)nn2)[nH]c(C)c1C#N c1(OC)nc(Cl)ccc1C(C)NC1CC2C=CC1O2 c1(C(C)C(=O)NCCCNC(=O)CC(C)(C)C2CC2)cccc([N+](=O)[O-])c1 Cc1nsc(C)c1C(=O)N(C)CC1(NC(c2ccnc(-n3ccnc3)c2)=O)CC1 c1(C(=O)NC2CCN(C(CCC3N(C)CCCC3)=O)C2)cnc2c(c1)CCCO2 C1(C(C)C)N(C(c2ccc(C#N)[nH]2)=O)CC12CCN(C(=O)C(F)C1CCC1)CC2 C(CCN=c1[nH]cnc2ccc(C(F)(F)F)cc12)NC(C1C(C)(C(F)F)C1)=O c1(SC)ccc(C(=O)NCCC2CN(C(=O)Cc3cc[nH]n3)CC2C)c(Cl)c1 C1(CNC(C(C=C)OC)=O)CCN(C(c2conc2C2CC2)=O)C12CCC2 c1(OC)cc(C)ccc1C(F)(F)F.C1(=O)CCC(=O)NC(=O)NCC2(CC2)CO1 C12(CNC(N(C3CCN(C(CCCc4scc(C)n4)=O)C3)C)=O)CCC(CC1)OC2 C1(C(=O)NCC2CC2c2ccc(F)cn2)CCN(Cc2ncc[nH]2)C12CCC2 CCC(C(=O)Nc1coc(C)n1)n1ccnc1.C1C(=O)NCC1=O.NC CC1(C)CCCOC1C(=O)NCC1CCN1C(C12CC(F)C1C2)=O CC(C)(C)CC(O)C(=O)NC1(CO)CCN(C(c2ccc(-c3cc[nH]n3)s2)=O)C1 Cc1[nH]c(C)c(C(N2CCCC2CCC(N2CC(F)C(F)C2)=O)=O)c1C CC(C)CCCC(=O)NCC1COCCN1C(=O)CCc1ccc(O)c(Cl)c1 CCC(CC(=O)N1CC(CNC(c2cc(C3CC3)nn2C)=O)C2CC12)SC CCC(CCN(C)C)C(=O)NCC1(O)CCN(C(=O)CC2CC3CC3C2)CC1 C1(C(N(C2CCCC2)CCCNC(C(C(C)C)O)=O)=O)CC2(COCCO2)C1 C1(N(CCC)C(c2csc(C3CC3)n2)=O)CCN(C(C2COCC(C)O2)=O)CC1 CC1C(NC(=O)C(C)(C)c2cccs2)CCCN1C(=O)Cc1csc(C2CC2)n1 c1(NC(C2CC(c3ccc(Br)cc3)C2)=O)cnc2cccnc2c1 C1(C(N(CC(CNC(c2c(C)ccnn2)=O)(C)C)C)=O)CN2CCC1(C)C2 N1(C(C2(C(C)C)N(C(CC(C)N(C)C)=O)CC2)=O)CC(CO)C2(CC2)C1 O=C1Cc2c(C(=O)NCCCn3cc(C4CCCCC4)nn3)ccnc2N1 N1(C(CN(C(C)=O)C)=O)CC(N(C)C(c2c[nH]nc2-c2ccco2)=O)C(O)C1 c1(C(=O)Nc2cnn(-c3ccncc3)c2)cccc2ncnc(O)c12 C(=O)(CC(C)CC(F)(F)F)N1CCC(CCNC(C(C(C)C)F)=O)CC1 N1(S(CC#N)(=O)=O)CC2(CN(C(c3cnc(Cl)cc3F)=O)CC2C(=O)O)C1 C1(CCNC(c2coc(C)n2)=O)CNCCS1(=O)=O.CCC(CC)C1CC1 C1(C(=O)NCC=CCNC(c2[nH]cc(CC(C)C)c2)=O)CCCCC(F)(F)C1 c1(NCCSCCC=C)ccc(S(=O)(=O)NC2CCN(C)C2)cc1Cl c1(C(N2CCC3CN(S(=O)(=O)CC4CC4)CC23)=O)cn2ccc(Br)cc2n1 CC1CN(C(=O)OC(C)(C)C)CCCN1C(C1CCN(c2nc(=N)[nH][nH]2)C1)=O c1(N2CCC(COCCC)CC2)ncnc(N2CCCC(C)(N(C)C)C2)c1C N1(C(c2c(CC)nn[nH]2)=O)CC2CN(C(c3cc(F)cc(F)c3O)=O)CCC12 O=C(C1CCc2c[nH]nc21)NCC(O)CCNC(=O)Cc1cc2ccccc2s1 Cc1ncn2ccc(C(N3CCC(N(CCO)C(C4CC=CC4)=O)CC3)=O)cc12 N1(C(CC2(O)CCCN(C)C2)=O)CCC(C2CCN(C(c3cscn3)=O)C2)CC1 c1(C(N2C(Cn3cc(CCC(N)=O)nn3)CCCC2)=O)onc2c1CCCC2 c1(CC)ccc(C(F)(F)F)cc1NC(=O)NCCCOc1ccc(F)cc1 c1(NC2CCN(CCNC(c3ccccc3F)=O)CC2)cc(O)ccc1[N+](=O)[O-] c1(OC)cc(NC2CCN(C(=O)CC(F)(F)C(F)F)C2)c([N+](=O)[O-])cc1OC CC1C(C(=O)NC(C2CCN(C(=O)CCc3cncn3C)CC2)C)CCN1C c1(C(=O)NCC(C)CNC(c2ccoc2)=O)cc(S(=O)(=O)CC(N)=O)ccc1Cl C1(CC)CN(C(C2C3(CC3)C23CC3)=O)CCC1NC(c1cscc1Br)=O n1(CC(N2CC(F)(C(=O)NC(CC#C)CO)C2)=O)cccnc1=O C12(C(=O)NCC(CNC(c3c(C)csc3)=O)C)CC1COC21CCC1 c1(N2CC(CNC(C3(C)ON=C(C(C)(C)C)C3)=O)C2)ccc(C#N)cc1[N+](=O)[O-] Cc1noc(C)c1C(N1CCC(CF)(NC(C2CCCC(N(C)C)C2)=O)C1)=O c1(C(=O)NCC2C=CCCC2)ccccc1F.C12(CCCC1)C(=O)N1CC(C1)C2 CC(C)C(C)C(CNC(c1cc(Br)oc1Cl)=O)NC(C12CCC(C1)C2)=O CC1CC(C)OC1C(N1CC(C(C)NC(=O)CCC2(C)N=N2)C1)=O CCC(C)(CNC(=O)C=Cc1nccs1)C(=O)NCc1cc(C)c(C)o1 c1(CSCC)c(O)ccc(CNCC2CC2C(=O)Oc2ccccc2)c1[N+](=O)[O-] C1(NC(C(C)c2ccsc2)=O)CC(F)CN(C(=O)C=C2CCN(C)C2)C1 C(CCC(=O)NCC1=NOC(C)C1)(C(C)C)NC(c1c(C)coc1)=O c1(C(=O)OC)ncc(C)c(CNc2cn(CC3(C)CCCC3O)nn2)c1Cl C1(CC(=O)NC(C)C(=O)N(C)C)CCCN(C(=O)C=CC(=O)N(C)C)CC1 N1(C(C2(C(CC)=O)CC2)=O)CCN(C(c2cnc(O)o2)=O)CC1C c1(C(=O)NCC(C)(C)NC(C2CC3COCCN3C2)=O)ccc2ncsc2c1 C1(CC#C)(C(=O)N(C(CNC(=O)CN2CC3CCC2C3)C2CC2)C)CCCCO1 n1(C(C)C)ncc(Cl)c1C(=O)NC1CCCN(C(=O)CCc2cccs2)C1 Cc1nn(CC(N2CC(CO)(NC(c3ccc(F)o3)=O)C2)=O)cc1Cl N1(C(C(C)SCC)=O)CC(NC(c2cc(N)ccc2Cl)=O)CC12CCCC2 N1(C(C(C)=CC2CC2)=O)CC(N=c2[nH]nc(C3CC3)o2)C(C)(C)C1 C1(NC(C2CCC(=C)CC2)=O)COCCN(C(=O)C=Cc2cnccc2C)C1 C(=O)(C1=CC2CCC(C1)C2)N1C2CC(C(F)C(=O)N1)C2.c1(N)cc(F)ccc1F C1(NC(C(CC)C#N)=O)CCC2(CC1)CN(C(=O)CCCC(C)(C)CC)CCO2 CS(=O)(=NC(=O)CN1CC(O)C(O)C1)c1ccc(F)cc1.c1(C2CC2)ccccc1 CCC(C)C(C)C(=O)N1CCCCC1C(C)(C)CNC(c1ccn(C)c1)=O C(=O)(C(C)(C)C(=O)NCC1C2CN(C(=O)C(C)(C)c3ccno3)CC12)NC N1(C(C(c2ccoc2)NC(=O)Cc2cc[nH]c2)=O)C2CCC1CC2 c1(CNC(C2OCCN(C(c3cc(CC)[nH]n3)=O)C2)=O)cccc(C#N)c1 C(=O)(CCCN=[N+]=[N-])N(CCC(C)O)C.Cc1ccccc1CCS(C)(=O)=O C(=O)(C1=CCCC(C)(C)C1)N1CC(CNC(c2c(CC)scc2)=O)OCC1 C1(C(N(CC(CC)NC(=O)C(O)CC2CCCCC2)C)=O)CC(=O)N(OC)C1 CCCCCCC(C)CC(=O)N1C2CCC1CC(NC(=O)C(C)OC)C2 N1(C(C(C)OCC#C)=O)CCOC2(CCC(NC(=O)Cc3nncn3C)CC2)C1 CC(C(=O)N1CCC(NC(=O)CC(C)(C)c2ccccc2)C(CO)C1)S(N)(=O)=O CCCC(CC(=O)NCC1(CO)CC12CCC2)NC(=O)C(c1ccn(C)c1)C CC(CC(=O)NCc1cn(C2CN(C(=O)CCC3(C)CC3)C2)nn1)C(F)F C1(C(=O)NCc2cc[nH]n2)C=CCN1C(=O)C(O)CC1CCCC1 CC(CC(=O)NCC(=C1CN(C(C2CCCCS2)=O)C1)F)n1cc(Br)cn1 C#CCCCCC(=O)NCC1CC(C(F)(F)F)CCN1C(=O)C=NOC c1(C(C)=O)cc(C(=O)N(C2CC(NC(c3ccc(C(F)(F)F)o3)=O)C2)C)no1 C(=O)(C(C(C)C)NC(N)=O)N(CCC(=O)NCC(C)OCC=C)CC C1(NC(c2cccnc2)CCC)CC2CCCC2(CO)C1 C1(CN(C(C=CCOC)=O)C)C2CN(C(=O)C(N3CCCCC3)C)CC12 C1(CNC(CC(C=C)C)=O)CCN(C(=O)CSc2ccccn2)CC(C)(C)C1 C1(C)(OCC(=O)N(CC(=O)NC)CC)CN(C(c2cccnc2)=O)C1 C1(CNC(=O)CCOC2CC2)COC(CNC(=O)CC2CCC2)C1 C(=O)(C=CS(C)=O)N.CC(O)CN1CC1.C(C)=O c1(SCC(=O)N(C2CN(C(C3CCOC3=O)=O)CC2O)C)ccc(O)cc1 C(CC(C)C)(C(=O)N(C)CCOCCCNC(=O)Cc1ccsc1[N+](=O)[O-])OC C(C(C)C)(C(O)C(=O)N1CC(O)CC1(C)C(=O)NC1(C)CCC(C)=C(C)C1)OC Cc1cc(Cl)c(C(=O)NCC23CC(NC(=O)C4=CCCC4C)(C2)C3)cc1C c1(CC)noc(C)c1C(=O)NCC1(NC(=O)COCP(C)(C)=O)CCOC1 c1(CNC(CC(=O)NC(C)C)C2CCC2)ccc(O)cc1 n1(CC(CC)Nc2ccccc2)nc(CCCO)nc1-c1ccsc1C(=O)NC C(C(=O)NCCC1CC(NC(c2cscc2C(N)=O)=O)C1)(C(C)(C)C)SC C(CCCCCNC(c1cccn1CC1CCC1)=O)NC(c1cc(CO)[nH]n1)=O N1(C(c2c(OC)scc2)=O)CC(NC(=O)CCC(C)(C)C)C(F)(F)C1 N1(C(c2c(C)ccc(C)c2)=O)CCN(C(=O)C(c2ccc(F)cc2)C)CCC1C C1(C(N(CC)CC2CCCO2)=O)COC2(C1)CN(C(=O)CCOCC1CCC1)C2 C1(CNC(CCN(C(C)=O)C)=O)CCC2(CC2)C1.c1(C=O)ccn(C2CC2)n1 c1(C(=O)NC(C2CCN(C(c3sccc3F)=O)C2)C)cccn2c(O)nnc12 N1(C(CC=CCNC(C(NOC)=O)=O)=O)CCC(O)CC(C)C1 C(=O)(CCCCC(C)CC)N(CC1(CN(C(c2ccc(CC)c(Cl)c2)=O)C)CC1)CC C1(CC(=O)NC(CC)(CC)CCNC(=O)CCn2cnnn2)COC2(CCC2)CO1 C(CCCCC(=O)N1CCCC1CN(C)C(C1CC(O)(C(F)F)C1)=O)N(C)C C1(C(=O)NCC(C(C)(C)C)NC(C=CC(C)=O)=O)CCc2nnc(C)n2C1 n1(CC)cc([N+](=O)[O-])c(C(N2CCN(C(c3cc[nH]n3)=O)C3CCC23)=O)n1 C(=O)(C(O)C(F)(F)F)N1C(CNC(CCN2CCC(C(N)=O)CC2)=O)CCCC1 c1(CN2CC(N(C(c3ccc(C(=O)NC)cc3F)=O)C)C2)cc(C#N)ccc1O C(=O)(C(C(C)(C)C)NC(c1cnc(C(C)C)o1)=O)NC(c1cn(CC)nn1)C c1(C(=O)NC(CS(CC)(=O)=O)CC)c(C)ccc2cc(C)ccc12 c1(OC)c(C(=O)NCCN(C(=O)CC(C)(C)F)C)sc(Cl)c1Cl N1(C(C2CC2CC2CCOC2)=O)CCC(c2ccc(Br)cn2)CC1 c1(C(=O)NCC2N(C(CCC#N)=O)CC(O)C2)cc2cc(Cl)cnc2[nH]1 C1(NC(COCC(C)(C)C)=O)CCN(C(=O)CCF)CC1c1ccccc1 C1(CNC(C2C3CCN2CC3)=O)CC(F)CN1C(=O)CC1CCCC1 S(=O)(=O)(c1ccc(O)cc1)NCC12C(CN(C(c3cc(Br)ccc3Cl)=O)C1)C2 c1(C(N2CC(C)C(NC(c3nc(Cl)ccc3Cl)=O)C2)=O)cc2n(n1)C(C)CCC2 C(C(C)(C)C(F)F)NC(C1(CCC=C)CN(C(=O)C(COC)N(C)C)C1)=O C12(CNC(c3[nH]cc(OC)c(=O)c3)=O)CCCCC1CN(C(c1cocn1)=O)C2 C1(CNC(C(C)(C)CO)=O)CN(c2ncnc3c2CCO3)CCC1(F)F c1(CC(=O)N(C23C(CN(C(C4C(C=C)C4)=O)C2)C3)CC)ccc2sccc2c1 c1(C(=O)NCc2c(OC)cc(O)nc2)c[nH]c2ccccc12.C(C)(C)O C(=O)(CC(C)CCC=CCl)OCC.N1(C(C=C)=O)CCCC1Cn1cc(C(C)OC)nn1 Cc1cc(Cl)cc([N+](=O)[O-])c1C(=O)OCCCc1cccnc1 C#Cc1ccc(CC(=O)NCC(F)CNC(C2CCN2C2CCCC2)=O)cc1 N1(C(c2cccc(C#C)c2)C(=O)NCCCC)C2CCCC1CC(O)C2 C1(CNC(C(C)OCOC)=O)OCCC1C(=O)N(CC(C)O)CCF C1(C(=O)NC2(C)CN(C(CCOC)=O)C2)CC2(C1)CC2C(=O)O c1(C(N2CCCC(NC(CCC)=O)C(F)C2)=O)ccc(S(N)(=O)=O)n1C C1(CC=C)(NC(c2cnn(CC(F)F)c2)=O)CN(C(c2cn(C(C)(C)C)nn2)=O)C1 C1(C(=O)NC(CN(C(c2ccn(CCCC)n2)=O)CC)C)CC(C2CCC2)C1 CON(CCC(=O)N1CCC1COC)C(=O)C1(C)CCC(=O)N1 C1(OC)CN(C(=O)C(c2c(C)ncn2Cc2ccc(F)cc2)=O)CC1CN CCCCC(O)CCC(=O)N(C1CCN(C(c2cn(C)nn2)=O)CC1)CCC C(N=c1cc(Cl)nc(C2CCOCC2)[nH]1)C1CCN(C(CSC(C)(C)C)=O)C1 C(CC)(CCC(=O)Nc1ccc(O)nc1)NC(C=C(CC)CC)=O N1(C(CCc2c(C)noc2)=O)CCC(CNC(c2ccc(Cl)nc2O)=O)CC1C CCC1=C(C(=O)N2CCN(C)C(CNC(=O)CC3CSCCS3)C2)CCCO1 CC(C)(C)C(CO)NC(=O)CC1C=CC(NC(C2CCC2(F)F)=O)C1 C1(NC(C(CCSC)NC(=O)C=CC(F)(F)F)=O)CC2(CCCC2)C1 O=C(C(F)C(F)(F)F)NC1CC2CC1N(C(C1(CN3CCCC3)CCCC1)=O)C2 c1(C(N(CC(CC)NC(c2ccnn2CCN(C)C)=O)C)=O)cnncc1OC N1(Cc2ccc(CCCCC)cc2)CC2CCC(C1)N2C(C1CNC(=O)N1)=O CCC(CC(=O)NCC=CC(N1CCOC(C2(C)CC2)C1)=O)SC C1(CCO)(CNC(C(n2cc(CCOC)nn2)C)=O)CCCCC1 CC1(OCC(=O)NC2CC(F)(NC(=O)CN(C3CCCC3)C)C2)CCCC1 CC1CCC(CNC(C2CC3(CC3)C2)=O)N(C(c2nnc(C(F)(F)F)s2)=O)C1 Cc1ccc(C(=O)NC(Cc2cn[nH]c2)C(=O)NC(C)Cc2nncn2C)cc1 CCCCCC(O)C(=O)NC1CCCC1NC(=O)CN1CCCC1CC C(C)(CCCC(=O)NC(C)Cc1nc[nH]n1)NC(c1c(C)n(C)cn1)=O CC(CS(=O)(=O)N1CCCC1)N=c1nc2sccc2c(NC2CCC2)[nH]1 C1(CC(N)=O)CCCC12CCN(Cc1nn[nH]n1)CC2 N(C1CCc2c1ccc(Br)c2F)C(c1cc[nH]n1)C(=O)Nc1c(C)c(Cl)ccc1 C1(C2CN(C(=O)NC(CCC=C)C)C2)CCCCC1=O C(CC(C)C)(C(=O)NC(C1CCCCO1)C)NC(c1ccnc(C)n1)=O C(N=c1[nH]nc(-c2ccon2)s1)C12OCC(NC(CCCOC)=O)(C1)C2 c1(C(N(C(C(=O)NC(CC)(C)C2CC2)c2ccco2)C)=O)cnn(C(F)F)c1 C1(C(=O)NC(CNC(c2c(CC)noc2)=O)CCOC)CCn2nncc2C1 C1(C(N2C(CNC(CCCN(C(C)=O)C)=O)C(C)CC2)=O)CC2(CCO1)CC2 CC1C(C)N(C(CCCOCCCNC(=O)CC(=O)OC(C)(C)C)=O)CCS1=O N1(C(C2(C(=O)OC)CC2C)=O)CC(CNC(C2CC=CCO2)=O)C(O)C1 C(C(C)(C)C(C)(C)C)NC(N1CC(CCC=C)(C(=O)OC)C1)=O N1(C(C2N(CC)CCC2)=O)CC2OCC(NC(=O)CN3CCCCC3)C2C1 Cc1cccc2c(C(N3CCC(O)C(NC(C4C(C)C4C)=O)C3)=O)n[nH]c12 c1(OC(c2cn(Cc3cccnc3)nn2)=O)nnc(C(F)(F)F)s1 c1(C(=O)NCC2CCC(NC(=O)CC3C=CS(=O)(=O)C3)C2)ccc2c(c1)CCO2 c1(C(=O)NC2CC(F)C2)ncnc2c1cnn2C1(OC)CCC1 C1(CC=C)(NC(c2nc(C)ncc2Cl)=O)CCN(C(=O)CS(N)(=O)=O)CC1 c1(C(N(C)CCN2CC=CC2)=O)cnc(CNC(C2CCN2C(C)(C)C)=O)nc1 CC1CCN(C(=O)C=CC2CCCC2)CC1NC(C1CCC(=O)N1C)=O C(N=C(NCC(N1CCCC1)=O)NCC(C)OC)C1N(CC)CCC1 N1(Cc2c(OC)ncc(Br)c2)CCC2(CC1)CC2NC(c1ccc(C)c(I)c1)=O C1(NC(C(C)NC(=O)NCC)=O)CN(C(c2ccn(C3CCC3)n2)=O)CC1F C1(NC(CC(CC)OC)=O)CC=C(C(=O)NCC(N2CC=CC2)=O)C1 c1(OCCCC(=O)NC2CC(C)OC(C)C2)ccc(S(N)(=O)=O)cc1F N1(C(C)=O)CCN(CCNc2ccccc2)C2(CCC2)C1.C(=O)(C(N)C(C)CC)N c1(CNC(c2cc(C)ncc2)=O)nc2c(s1)CCN(C(C1CC3(C1)CC3F)=O)C2 c1(C(=O)NCC2C(C)CCN2C(=O)CCNC(=O)CO)cncc(P(C)(C)=O)c1 CC(CC(=O)N1CC2C(NC(=O)C=Cc3ccccn3)C2C1)C(F)F C1(NC(C)(C)CNC(C2CC(=O)N2)=O)CC2CCCCC2NC1=O C(=O)(C1CCCc2ccnn21)N1CC2C(CNC(c3c(SC)cccn3)=O)(C2)C1 c1(C(=O)NC(CN(C(C(C)OCC2CC2)=O)C)(C)C)cc2ccc(O)nc2s1 C12(CNC(C(CC)O)=O)CC(CN1C(=O)CC(C)F)C2 C12(NC(c3c(Cl)cnc(C)n3)=O)CCCCC1CN(C(C1CC=CC1)=O)C2 C12COCC1n1cc(nn1)CN(C1CC1)C(=O)N2C.C1(C)CC1(F)F.CO N1(C(c2cc(C)c(C)[nH]2)=O)CC(C2CCCN(C(=O)CSc3nncs3)C2)C1 Cc1c(C(=O)N(C2CCCCC2)CCO)cc(C(F)(F)F)cc1N C1(F)(C(=O)NCCC(C)(C)NC(C2CC(OC)C(OC)C2)=O)CCCN(C)C1 N1(C(CC(CC)C)=O)CC2CC(NC(c3cnc4sccc4c3)=O)CC2C1 c1(C(N2CC(O)(CNC(C=CS(C)=O)=O)C2)=O)ccc(F)c(-c2ccccc2)n1 N1(C(C(CCC)NC(c2ncn(CC)n2)=O)=O)CCC2(C=CCO2)CC1 CC12CCC(C(N3CCC(n4cc(CC[NH2+][O-])nn4)CC3)=O)(CC1)CO2 N1(C(c2ccc(SC)o2)=O)CCCC(NC(=O)C(c2ccccc2)=O)C1C c1(C(=O)NCCN(C(C(C)SC)=O)CC2CC2)cnc2c(C)cc(C)cc2c1O c1(C(=O)NC(CC(C)NC(CCCNC(=O)OC)=O)C)[nH]ccc(=O)c1C C(CCC(=O)NC1CC(O)C1O)(C(C)C)NC(C1(CC#C)CCC1)=O CCC(CNC(c1ccc(F)cn1)=O)(CC)NC(=O)Cc1cn(C2CC2)cn1 C(=O)(C1CCc2cc(OC)ccc21)N(CCNC(c1cc(COC)no1)=O)C Cc1cc(-c2cn(CCC(N3CCC(C)(O)C3)=O)nn2)ccn1 CC1(C)C(NC(c2cnc(-c3cccs3)s2)=O)CC1CNC(=O)Cn1nccn1 N1(CC)CCOCC1C(=O)NCC1CC(NC(=O)Cc2ccnn2C(C)(C)C)C1 C1(CNC(C(C)OCC#C)=O)CCCCCN1C(=O)CC(C1CCC1)C1CCC1 C1(F)(CNC(C(N2CCN(C)CC2)C)=O)CC(N=c2[nH]nc(C(C)(C)C)s2)C1 N1(C(c2c(C)nccn2)=O)CCC(C(=O)NCC(O)(C2CC2)C2CC2)CC1(C)C Cc1ccnc(Cl)c1C(=O)Nc1ccc(-n2cccc2)c(Cl)c1 C#CC1(N(C)C)CN(C(=O)CN(C(c2ccc(C(C)=O)o2)=O)CC2CC2)C1 c1(C(N2C(C)CCC(CNC(=O)COC(F)F)C2)=O)cnc2c(c1)NC(=O)CS2 N1(C(C2(COC)CC=CCC2)=O)CCN(C(=O)CN(C)C(C)C)CC(C)(F)C1 O=C(CCc1cnc[nH]1)NNc1ccc(-c2cccs2)nc1 N1(C(c2ncc(OC)nc2)=O)CC(=O)NCC1C(=O)NC(C)Cn1cnnc1 C=CCCN=C(NCC1CCC(OC)CC1)N1CCC(N2CCCCC2)C1 Cc1cc2cccc(NC(C3(C)CCN3C(=O)C3CC3)=O)c2cn1 C(=O)(CC(C)CC(C)C)N1CC(OCCC(=O)NCC=CC(CC)C)C1 C1(C(N2CC(C3C(=O)N3)C2)=O)CCCN1C.C1(N(C(C)=O)C)CCC2CC12 c1(SCC)cc(NC(=O)C(CN(C)C)NC(=O)OC(C)(C)C)ccc1Cl C1(C(=O)NCC2CCC(CN(C(C34CC(C)C3C4)=O)C)CC2)CCCNS1(=O)=O c1(C(=O)NC(C2CCN(C(c3scnc3Cl)=O)C2)C)cc(Cl)cc(Cl)c1N C(=O)(C(F)C(F)(F)F)NC(C(=O)N(C)CC1CCCC1O)C1CCC1 O=C(CS(=O)(=O)C1CC1)NC1CCCC1NC(C1CCN1Cc1ccccc1)=O c1(CC)ccc(NC(=O)C(C)(C)CNC(c2cnns2)=O)c(C)n1 Cc1cc(F)ccc1CC(=O)NC1(Cn2cc(CCC(C)O)nn2)CC1 C12(C(=O)NC(C(C)C)C(=O)NC(C)CCn3cncn3)CCCC(CO1)C2 S(=O)(=O)(c1cccs1)NC(C(=O)NC(CN(C(c1ccn(CC)n1)=O)CC)C)C CCC(CC(=O)N1C(C(=O)NC(COCC)C(C)C)CCC1C)CC(C)C CS(=O)(=O)CCCC(=O)NC1CCCN(C(=O)C(c2ccccc2)=O)CC1F c1(C(N2CC(OC)(CNC(C3(F)CCOC3)=O)C2)=O)cncc(Cl)c1Cl C1(C)(NC(C(C)OCC#C)=O)CN(C(=O)Cc2coc(CCOC)n2)C1 N1(C(C2C=CCN2C(c2csnn2)=O)=O)CCOC2COCC12 c1(CNCc2cccc(-c3ccc(C(C)=O)cc3)c2)cc(Br)cc(I)c1 C1(NC(c2c(CC)nn[nH]2)=O)CN(C(=O)C(C)(O)C(C)C)CC(F)(F)C1 C(C)(N=c1[nH]c2c(c(=NCC3CCCCN3C)[nH]1)CSC2)c1ccc(OC)cc1 c1(C(=O)NCCN(C(CC2(CS(C)(=O)=O)CC2)=O)CCOC)ccc(Cl)nc1O CCC(C)(C)C(=O)NCc1csc(C(=O)N(C)CC2(N(C)C)CC2)c1 C1(C(=O)NC2CCCC2)CC1(F)Cl c1(C(=O)NCC2CN(C(CC(C)CF)=O)CC2(F)F)ccc2c(c1)ncn2C c1(C(=O)NC2CN(C(C=C(C)Cl)=O)CC2O)cc(C)cnc1C C1(CCNC(C2CC(N(C)CC)C2)=O)COCCN1C(=O)Cn1nc(C)oc1=O C=CCCCC(C)(C)C(=O)N1CCC(NC(c2csc(C(C)=O)n2)=O)C1 C1(NC(C2C(C=C)OCC2)=O)CCC2CC1CN2C(c1cc(OC)cc(F)c1)=O N1(C(CC)=O)CSCC1C(=O)NCC(C(C)C)NC(c1ccc(Cl)[nH]1)=O c1(C(N2CC3C(CNC(=O)Cc4cc[nH]c4)(C3)C2)=O)cnc2ncccn12 CCCCCCCCC(=O)N1CC(O)CC1(C)C(N1CC(C#N)(SC)C1)=O N1(C(C(C)(C)c2cnc[nH]2)=O)CCC(CO)C(NC(c2cccc(Cl)c2)=O)C1 c1(OC)cc(OC)c(C(=O)NCC2(F)CN(C(C3CC=CCO3)=O)C2)c(OC)c1 CC1C(C(=O)N(CC(C)(C)NC(c2cnn(C)c2Br)=O)C)CCN1C C(=O)(CCCCC(F)(F)F)N1CC(CNC(CC=CCC)=O)CC12CCC2 C(=O)(C(C)(C)CC(C)(C)C)N1CCC2(CC(C(=O)NCC(C)SC(F)F)C2)C1 N1(C(C2CCCCN(C(=O)CCc3ccoc3)C2)=O)CCc2c(F)cccc2C1 c1(C(CNC(c2cnn(C3CCC3)c2)=O)NC(C(C)SC)=O)cccc(C)c1 CCC(C)C(O)C(C)C(=O)NC(C)(C)CCC(=O)NCC1(CCO)CN(C)C1 c1(C(CNC(CC2C(C)OCC2)=O)NC(c2cnccc2)=O)ccccc1F Cc1ccc(C(N2CC3CC2CC3NC(=O)CCC#N)=O)cc1O N1(C(CCC(C)OC)=O)CC2OCCN(C(c3ccc(C(C)C)nc3)=O)C2C1 N1(C(CC(=C)Br)=O)CC=CC(NC(C2C(c3ccccc3)C2(C)C)=O)C1 N1(C(CCC=CCC=C)=O)CC2(C1)CN(C(c1ncccc1OC)=O)C2 c1(C(=O)Nc2n(C)ncc2I)ccc2c(C(N3CCOC4CC34)=O)n[nH]c2c1 C(=O)(C1CCCc2ccccc21)NC(C1N(C(CC(C=C)CC)=O)CCC1)C C1(C(N(CCC)CCC)=O)CN(C(=O)C(c2cnn(C)c2)=O)CC(C)(C)C1 c1(CCOC)n[nH]c(=NC2CC(F)(CNC(c3ccn(C)n3)=O)C2)s1 N#Cc1ccc(C(N2CC3(C2)SCCC3NC(=O)CCSC(F)(F)F)=O)c(F)c1 CC1CC(N=c2[nH]nco2)CN1C(C1CCC=CCCC1)=O Cc1cc(OC(c2cc(S(C)(=O)=O)ccc2F)=O)nc2ccccc12 CCS(=O)c1ccccc1C(=O)N(CCCCCNC(c1cc(F)c[nH]1)=O)C N1(CC(=O)NCCN(C(=O)C(O)C2CCC2)C(C)C)CCS(=O)CC1 C(c1cc(F)c(O)c(F)c1)=CC(=O)NC1C(C(=O)O)C2CCCCC12 c1(C(=O)NCc2c(C3CCN(C(C(C)=O)=O)CC3)cccc2)cc(C)cc(Cl)n1 N1(C(CCC#N)=O)CCC(NC(=O)C(C2(O)CCCC2)F)C(C(N)=O)C1 c1(CNC2N(C(COCCOCC)=O)CCC2O)ccc2c(c1)nc(C)c(=O)n2C C1(NC(C2CC(SC)C2)=O)CN(C(c2ccccc2OCCF)=O)CC1(C)C N1(C(C(=O)NCCOC2(C#C)COC2)=O)C(C)CC(C)CC1C CC1(NC(c2cnc(Cl)cn2)=O)CCCN(c2cc(Cl)nc(C(F)(F)F)n2)C1 Cc1n[nH]c(C)c1CC(=O)NC1CC(CNC(C2CCCN2C)=O)CC1O N1(C(C=C2CCN(C)CC2)=O)CC2CCCC2(NC(c2cnc(C(F)F)s2)=O)C1 c1(N2CCC(CCC)=C(F)CC2)nc(N2CCOc3ncccc3C2)c2c(n1)CSC2 CC(C(C)C(=O)NCC1(C(=O)O)CCCC1)S(C)(=O)=O c1(C(=O)NCCC2(CNC(c3cnc(OC)s3)=O)CC2)csc2c(O)ccnc12 CC1(C)CCC(C(=O)NC2CC(CF)C2)CN1C(C1(O)CCCC1)=O C1(COC)CN(C(c2cnc(N)cn2)=O)C(C)(C)C1 C1(CNC(=O)Cn2cc(C3CC3)cn2)CCCCN(C(=O)CC=C(Cl)Cl)CC1 n1(CCOC)cc(NC(=O)CCNC(=O)CCNO)ccc1=O c1(C(N2CCCC(N(CCF)C(c3cn(C4CC4)nn3)=O)C2)=O)cnnc(Cl)c1 N1(CC(CC)NC(=O)NCC2(c3ccccc3C)CCC2)CCCC(O)C1 N1(C(C(CC)(F)F)=O)CC2(CNC(=O)C=C3CCCCC3)CC2(C(F)(F)F)C1 C(=O)(CS(=O)(=O)c1ccccc1F)NC1(CC)CCCN(C(CSCCCC)=O)C1 Cc1cc(C(=O)NC2CCC(O)CN(C(=O)C(C)C3CCC3)C2)c(S(N)(=O)=O)s1 c1(C(=O)NCC2CC(NC(C3(SC)CC3)=O)C2)cc(Cl)cc(Br)c1N C(=O)(CCC(C)CN(C)C)N(CCN(C(COCC(=O)NC)=O)C)C(C)C C1C(C)(OC)C(=O)Nc2nccc(c2)CC1=O.C12(CC1)C(=O)NC2.CO C1(NC(COCC)=O)CCC(NC2(C)CCN(c3ncc(OC)cn3)C2)CC1 c1(C(N2CCC(C)(C(=O)Nc3ccc(Cl)nc3Br)C2)=O)cnn2ccccc12 C(=O)(CCCCC#N)N(C(C)C)CCNC(=O)CC(C)CC1CCC1 C12(C(=O)NC(CNC(C(C)=C3CCCC3)=O)C)CC(C)C1C2 c1(NC(CC(C)N(C(C(C)S(C)(=O)=O)=O)C)=O)cnc2ccccc2c1 CC1(NC(c2nonc2N)=O)CCCN(C(=O)C=Cc2ccco2)C1 N1(C(=O)OC(C)CN(C)C)CCCCC1C1CCCN1C(=O)NC(C)(C)C N1(C(CC2(CSC)CC2)=O)CC(N(C)C(C2COCCN2C(C)=O)=O)C(F)C1 c1(C(=O)NC23CN(C(c4cncc(C)c4)=O)C(C2)C3)ccc([N+](=O)[O-])c(C)c1 C1(CC)(NC(C2CC(C)(C)CCO2)=O)CCCN(C(=O)C=Cc2sccc2C)C1 c1(C(=O)NC(CCOC)CNC(C2CC2C(N)=O)=O)c(C)nc2ccnn2c1C c1(CC)ccc(C(=O)NCC2CCCN(C(=O)CCNC(N)=O)C2)c(N)c1 C1(CNC(c2cc(O)ccc2Br)=O)CCN(C(c2cncc(O)c2)=O)CC1(F)F C1(CNC(=O)CN2CCCC2)CC2CCC1N2C(c1ccc(C(F)F)cc1Cl)=O c1(-c2c(C)nc(C(=O)Nc3ncc(F)cc3Cl)cc2)c(F)ccc(Cl)c1F C1(CNC(c2nc(CC)oc2)=O)CCCC2(CN(C(=O)C=C3CCCCC3)C2)O1 N1(C(C(c2ccnn2C)C)=O)CCC2CN(C(c3nnc(O)cc3O)=O)CC2C1 C(C(C(F)(F)F)N1CCN(C(=O)Cc2ccon2)CC1)NC(C(Br)=C(C)C)=O C(C(=O)NCCNC(=O)C(C)C1CCCC1)(C(C)(C)C)N(C(=O)OCC)C Cc1ncnc(N2CCOCC(CNC(C3(O)CC3)=O)C2)c1C#N c1(C(=O)NCCCC)ccc2nc(CSC)cn2c1.C(=O)(C(C)CN(C)C)NC1CC1 N1(C(C(CC)OCC)=O)CCN(C(c2nn(C)cc2S(C)(=O)=O)=O)CCC1C Cc1ccc(C(=O)NCC(O)CC(=O)N2CCN(C3CC3)CC2)n1C C1(C(=O)OC)C(C2CC2)CCN1C(c1cc(F)ncc1F)C(=O)NCCCSC Cc1cc(CNC(=O)C(C)(C)C2CCN(C(c3cc(=O)cc[nH]3)=O)C2)nn1C N1(C(Cc2n(C)cnc2)=O)C2CCCC1CN(C(c1coc3c(F)cccc13)=O)C2 C12(NC(CN(S(CC)(=O)=O)C)=O)CCC1CN(C(C1CCC1)=O)C2 C1(NC(=O)CCCN2CCCCC2)CCOCC1NC(C12CC(F)C1C2)=O C1(CC)CN(C(C2OCCC2(C)C)=O)CC1C(=O)NC(C)(C)C(=O)OC.CC CC1=NOC(C(=O)NCC(=O)OC(C2CCCC2)C)C1.C(C)C C1(NC(c2ccc(C)nn2)=O)CCN(C(c2cnoc2C)=O)CC1C(C)C C(=O)(C#CC1CCCCO1)NC1COCCN(C(Cc2ccc(C)cc2F)=O)C1 CCCCCCCCCC(=O)NCC(CNC(=O)Cc1ccns1)CO Cc1cc(C(N2CC(NC(c3cnn[nH]3)=O)CC2C)=O)c(C)c(C)c1 c1(NC(C2(NC(C3(C#C)CCCC3)=O)CCN(C)C2)=O)cc(CC)ccc1C CC1(C)CC(CNC(=O)Cn2nccn2)CN1C(=O)C(=O)NCC1CC1 n1(CC)ccc(C(=O)NC2(c3ccccc3)CN(C(=O)C=CCOC)C2)cc1=O C12(C(=O)OC)CN(C(=O)C(=O)Sc3cccc(Br)c3)CC1S(=O)(=O)C2 n1(CC(=O)NCCC(C)NC(c2cc(Br)ns2)=O)cc(C2CC2)nn1 CCCC(C(=O)N1CCC(C)C1C(N1CC(COC)C1(C)C)=O)N(C)C C(=O)(C(O)CC(C)(C)C)N1CC(C)(CCC(=O)NC2CCCC23CC3)C1 C1(C(=O)NCCOCCNC(c2cn(C3CCC3)nn2)=O)COCOC1 c1(CC)cc(C(=O)NC2CCN(C(=O)CCOC3CCCC3)C2)ncn1 c1(CNC(C2(C3N(C(C(CC(N)=O)O)=O)CCC3)CC2)=O)cn2cccnc2n1 N#CC1(C(N2CCC2CNC(=O)Cc2cccc(C(F)F)c2)=O)CC2CCC1C2 CCCCC(C(=O)NCC1(NC(=O)CCC2CCCOC2)CC1)NC(N)=O S(=O)(=O)(CC(=O)NC1CC(NCC(CC(=O)OC)O)C1)NCC N1(C(C(C(C)C)S)=O)CCC2(CC1)CC(C(N1CCCC(F)(F)CC1)=O)CO2 C1(C(=O)NCC2(O)CN(C(C(n3c(C)ccn3)C)=O)C2)CC2(CC2)CO1 N1(CC(=O)NC2C(CCC3(NC(C4CC(=O)C4)=O)CCC3)C2)CCOC1=O c1(CCC(C(=O)NC(C)C(=O)NC(=N)N)NS(CC)(=O)=O)cc(Cl)cc(Cl)c1 C1(C(N(CC(C(C)C)C)C)=O)COCCC1NC(c1cnsc1)=O c1(C(=O)NC(CCCC)CNC(=O)CC(=O)NCC2CC2)ncnc2c1CCC2 N1(C(CCCN(C(C)C)C)=O)CC(NC(C2COCCN2C(C)C)=O)CC(O)C1 C1(C(N2CC(OC)C(F)C2)=O)(NC(=O)C(F)OC(F)(F)F)CCC(C)(C)C1 c1(C(=O)NCCOCCNC(C2C(CCC)CCCC2)=O)ccc(N)c(OC)c1 c1(CC2CN(C(C3C(C)(CC)C3)=O)C2)cn(Cc2ccsc2)nn1 Cc1ccc(O)cc1C(=O)NC1C2CCC1N(C(=O)CC1CN(C)C1)C2 C12(C(=O)NCC3(CCC)CCC3)CCCC1CCN2C(C1CC1(C)C(F)F)=O N1(C(C23CC(CN(C(C4(Cl)C(C(C)=O)C4)=O)C2)C3)=O)CCC(F)(F)C(F)C1 N1(C(C(CC)NC(C)=O)=O)C2CCC1C(C(=O)N(CC(F)F)CC1CC1)C2 N1(C(=O)NCCc2nc(C)on2)CCc2sc(Cl)cc2C1 N1(C(c2ccc3ncn(C)c3c2)C)CCOC2(CCN(CC#N)CC2)C1 C=CCC(C)C(=O)NCCC1CCCN(C(c2ocnc2C2CC2)=O)C1 C12(C(=O)NCC3CC(C)OCC3)CC(CN(C(=O)CCC3CCCCC3)C1)C2 c1(OCC(=O)NCC2CC2NC(c2coc(Cl)n2)=O)ccc(F)c(Cl)c1 c1(NCC)cc(Cl)ccc1C(=O)NCC1CCC(NC(C23CC4CC2C3C4)=O)C1 C1(OC)CN(C(=O)C(CC(F)F)NC(=O)C(C)C2CCCC2)CC12CC2 c1(C(=O)OC(CCCC)COC)ccc(C(C)=O)cc1C N1(C(c2c(C)cc(C)nc2)=O)CCC(C2(NC(c3ccnc(C)c3C)=O)CC2)C1 C(C(CCO)N=c1[nH]c(C)cc(=NCCc2sc(C)nc2C)[nH]1)OC C1(CC)CN(C(=O)NC(C)Cc2cc(F)cc(F)c2)CCN1CCOC c1(CC(=O)N(CCNC(CCCOC)=O)C(C)C)csc2c(Cl)cccc12 N1(C(C(C)C2CC2)=O)CC2(COC(CNC(c3ccc(=O)oc3)=O)C2)C1 c1(C(N2CC(OC)C(NC(C3(C)CC4CCC(C3)S4)=O)C2)=O)ncnc(O)c1F c1(N(C)Cc2c(OC)nsc2)nc(=NC(C)Cn2cccn2)[nH]c2c1CSC2 C1(NC(C(C)OCCC(C)C)=O)COCCC1NC(c1ccnc(C(C)C)n1)=O C(CC(=O)NCC(C)(CO)OC)(C(F)F)NC(CC(C)CN(C)C)=O c1(CC(=O)C(N2CC3C(NCC4CC4c4ccccc4)C3C2)=O)ccccc1Cl Cc1ccc(F)cc1-c1csc(C(N2CCN(C(=O)C(C)C)CC2)=O)c1 C1(CNC(C2CC(C(C)C)C2)=O)CC2CCC1N2C(=O)CC1C=CS(=O)(=O)C1 C12(NC(C#CC)=O)CCN(C(=O)Cn3cc(Cl)cn3)CC1C2 CC1CC(NC(c2nn(C)cc2Br)=O)CN1C(=O)CCOC1CC1 c1(C(N(CC(CO)(CO)NC(C2(C#N)C(C)C2)=O)C)=O)cnc(N)c(Cl)c1 C(C1C(C(N2CCCC(N(C)C(c3cscc3F)=O)C2)=O)C1(C)C)=C(C)C N1(C(C2(OC)CCSC2)=O)CC(C)OC2(CCN(C(=O)Cc3cccnc3)C2)C1 N1(CC)CCOCC1CC(=O)NC1CC(NC(=O)CC2CCC(C(F)(F)F)O2)C1 N1(C(C2CC(CCC)C2)=O)CCCN(C(=O)CN2CCCS2(=O)=O)CC1C c1(CN2CCC3(C(C(=O)NC4C(C)OCC4)C3)CC2)ccc2ncccc2c1 c1(OC)cccc(C(=O)NCC(C)N(C(c2cn(CC)nc2C2CC2)=O)CC)c1 Cc1cc([N+](=O)[O-])c(NC(C2CC2C(=O)NCCOCCCO)=O)nc1Cl c1(C(N2CCCC(CCCCCC)C2)C(=O)NC2CC2)cc(OC)c(OC)cc1Cl CCCC(F)(F)C(=O)N(C)CC1CN(C(=O)Cc2ccn(CC)n2)CCO1 N1(C(=O)OC(C)(C)C)CCC(C(=O)N2C3CCC2CC(O)(CNC(N)=O)C3)=C(F)C1 C12(NCC3CCC4(CC(C(=O)OCC)C4)O3)CC1CN(S(=O)(=O)CC)CCO2 c1(CC)nc(C(=O)N(CC(C)O)CCNC(=O)C(F)CC)c(C)o1 C1(C(=O)NCC(CCC)OCC)CC(=O)N(c2ccnn2C(C)CC)C1 C1(CNC(CC=CC)=O)(CO)CCN(C(=O)CNc2cccnc2C)CC1 C1(NC(CC2(OC)CCC2)=O)CCC2COC1O2 N1(C(CC(CNC(C=CC=CCC)=O)C2CCC2)=O)C2CCCC1COC2 n1(CC(N2CCC(O)(CN(C(CCCN(C)C)=O)C)C2)=O)ccc(O)nc1=O Cn1nc(CNC(=O)CC2CC3C=CC2C3)c2c1CCN(C(c1ccns1)=O)C2 CC1(C)COC(CC(N2CCC(C)(CNC(=O)CCCSC(C)(C)C)C2)=O)C1 c1(C(N2CCN(C(COCC)=O)C(C)C2C)=O)cc([N+](=O)[O-])cnc1C N1(C(C=C(C)C)=O)CCCC1C1(NC(=O)COCCc2ccc(Cl)s2)CC1 c1(C(C)NC(C2C(CNC(=O)C(C)(F)c3ccccc3)C2)=O)ccc(F)cc1 C1(C(N2CC(N3CCN(C(Cn4c(C)ccn4)=O)CC3)C2)=O)CCC(=O)N(C)C1 Cc1ccc(C2(O)CCN(C(CC3(C)CC3)C(=O)NC3CCC3)C2)cn1 N1(C(C(C2CCC2)NC(c2c(C)c(=O)cc[nH]2)=O)=O)CCC2(CC(F)C2)C1 Cc1cc(C(c2nnnn2CC2CCOCC2)NCC(Cl)C(F)(F)F)ccc1F Cc1oc(C)c(C(N2CC(C(N3CC(C)(CCO)C3)=O)CC2(C)C)=O)c1C CC(C)CCC(=O)C(=O)N(CC(N1CCC(C)OC(C)C1)=O)C1CCC1 CCC(C)CC(C(=O)NCC(F)Br)NC(c1sc(O)nc1C)=O c1(C(=O)NC(c2cn(C)nn2)C(=O)N(C(CC#C)C)C)cc(C)c[nH]1 c1(SC)cc(C)ccc1C(=O)NCC1CN(C(=O)C=Cc2ncc[nH]2)CC1C c1(C(N2CCN(C(C=CSC)=O)C(C(C)C)C2)=O)cc([N+](=O)[O-])c(C)cc1C c1(C(=O)NC(C2CCN(C(C(C)=C(C)C)=O)CC2)(C)C)cc2cccc(Cl)c2o1 C1(N(C(=O)Cc2nn[nH]n2)Cc2ccccn2)CCC(CC(=O)Nc2cnsn2)C1 C1(NC(C(CSC)(C)NC(C2CN(C)CCO2)=O)=O)CC2COCC(C1)C2 N1(C(C2C(C)C2)=O)CCC2CN(C(c3ncccn3)=O)CCC2C1 c1(CC)cccc(CC)c1NC(=O)NC1CCN(Cc2ccc(C)nn2)C1 Cc1ccc(C(F)C(=O)N2CC(N(C(=O)C(C)(C)NS(C)(=O)=O)C)C2)cc1 C(c1ccc(=N)[nH]c1C)=CC(=O)NCC(C)NC(c1c(CC)oc(C)c1)=O C(=O)(CC(C)CC(F)(F)F)NCC(CNC(Cc1c(CC)nn(C)c1CC)=O)F N1(C(CCOCC)=O)C2CC1CN(C(=O)CC1CCC(C)(C)O1)C2 CC(CC(=O)NC1(NC(=O)CC2CCN(CC=C(C)C)C2)CCC1)c1ccccc1 CC1(C)CCC(N(C(c2ccc(Br)cc2-n2cncn2)=O)CC2CCC2)CC1 Cc1cc(O)ncc1C(=O)NCCC1CN(C(=O)C=CCO)CC(C)O1 c1(CC)ncoc1CNC(C1(NC(=O)CCc2cncs2)CCCC1)=O c1(OC(CC(C)O)C)ccc(C(=O)Nc2nnn(C3CC3)c2C(F)(F)F)cc1 N1(C(C(CN(C)C)N(C)C)=O)CCN(C(c2ccn(CO)c(=O)c2)=O)C(CO)C1 Cc1cccc2c1CN(C(=O)CONC(C1CN3CCN1CC3)=O)C2 c1(C(N2CCCC(NC(C3(C)C=CCCC3)=O)C2)=O)cc(C(F)(F)F)cc(N)c1 CCC(C)(CCNC(c1ccnnc1)=O)NC(=O)Cc1ccn(C)n1 C12(C(=O)NCC(C#C)CC)CCC(CN(C(=O)CCCC(F)(F)F)C1)C2 c1(-n2c(-c3cc(Cl)c[nH]3)nc(CCO)n2)ccc2cnccc2c1 Cc1cc(C(N2CCCC(N(C(=O)Cc3cnsc3)C)CC2)=O)c(S(N)(=O)=O)s1 c1(C(=O)NCC(C2CCCN2C(c2ccon2)=O)(C)C)ccc2scnc2c1 C1(NC(CCC)C2CC2)CCCCC1NC(C1CC(SC)C1)=O C(C(CC(F)(F)F)NC(C1(CC)CC1(F)F)=O)NC(CC(=O)NCC#C)=O C(=O)(CC(C)C(C)C)NCC(=O)NC(CCSCC)C(=O)NC1CC1 Cc1cc(Cl)cc(C)c1C(=O)NC12CCCN(C(=O)CC(C)C3CC3)CC1C2 c1(NC(C)COC(F)F)ccc(S(=O)(=O)NCc2nn(C)nc2Br)cc1Cl n1(CC#C)cccc1C(=O)NC(c1cnn(C)c1)C(=O)NCC1CSCCO1 CCCC(CNC(c1ccc(SCC)cc1)c1nnnn1C1CCC1)CCO CC1(C)CN(C(c2ccc(F)c(CO)c2)=O)CCC1NC(C1(C)CC2CC2C1)=O C1(CNC(C2CCC(N(C)C)CC2)=O)(CO)CCN(C(C2CC(F)(F)CS2)=O)C1 C1(CNC(C(C)NC(=O)NC)=O)CN(C(=O)OC(C)(C)C)CCC12CCOCC2 N1(CCOC)CCOC(C)C1C(=O)Nc1cc(C(=O)OC)[nH]n1 O=C(C1=CC2C=CC(C1)C2)NC1(CCCNC(C23CCCCC2C3(F)F)=O)CC1 n1(CC(=O)NC(CC)CNC(=O)C(c2cccc(Cl)c2)C)ncc(O)nc1=O C1(C)(NC(c2cc(CNC(C(C)=C(C)C)=O)nn2C)=O)CCCCCC1 N1(C(C2(C#C)CCN(C(C3OC4CCC3C4)=O)C2)=O)CC(C)(C2CCC2)C1 N1(C(c2cc(C#N)c[nH]2)C(=O)NCCCCCC)CCCC(C)C1C.C(=O)(C(C)C)NCc1ccco1 C1(NC(C(CC)OCC)=O)CN(C(=O)CCCc2nnc(C)n2C)CC(C)(C)C1 CS(=O)c1cccc(C(N2CC3CC3(NC(c3cc(CN(C)C)c[nH]3)=O)C2)=O)c1 CC1C(NC(=O)CCc2nc[nH]n2)CCN1C(=O)Cn1ccc(C(F)F)n1 c1(C(=O)NCC(CNC(C(CC)CC)=O)C)cnc2ccccc2n1 c1(C(N(C(C)CN(C)C(C2CC23CCOCC3)=O)C)=O)cc2c(ncn2C)[nH]1 c1(C(C)NCC2CCN(CC(C)C)CC2)ccc2ncoc2c1 N1(C(CONC(Cc2nc(=N)[nH][nH]2)=O)=O)CCc2ccccc2C1 N1(C(C(c2ccc(O)cc2)C)=O)CCN(C(c2cnn3ccsc23)=O)CCC1C C1(NC(C2(CCC)CCC2)=O)CC(O)CN(C(c2cc[nH]c2C2CCCC2)=O)C1 c1(CC(=O)NC(C2N(C(c3ccc(CC)[nH]3)=O)CCCC2)C)cc(F)ccc1F C(CC(C)C)(C(=O)N1CCC(O)(CCNC(=O)CCc2cnoc2)C1)NC(C)=O c1(C(=O)NCC)[nH]cnc1CCC(C)N(C(=O)COC1CCC1)C c1(CNC(C(C2CCN(C(=O)C(O)c3ccsc3)CC2)C)=O)ccnc(Cl)c1 c1(CC)cc(C)c(C(N2CCOC(CN(C)C(C3(CO)CC3)=O)C2)=O)o1 c1(CNC(C(C2CCCO2)NC(C(C)n2cccc2)=O)=O)cnn(C)c1O C12(C(=O)O)CCCCC1(C(=O)NC1CCN(c3ncccc3F)CC1)CC2 CC1(C)CCC(CNC(=O)C(Cn2ccnn2)NC(c2ccc(C#N)o2)=O)OC1 c1(C(N2CC(C(C)NC(c3nc(OC)c(C)s3)=O)C2)=O)cc2n(c1)CCC2 Cc1cc(=NC(=O)C(=O)NCC2(F)CC(NC(C3OCC3(C)C)=O)C2)[nH]o1 CC1CCCCC1C(=O)NCC(O)CNC(c1n[nH]c(C2CC2)n1)=O N1(C(C(C(C)C)c2cccnc2)=O)CCC(F)C(NC(c2csc(CO)n2)=O)C1 c1(C(=O)NC(C)C)cc2c(s1)CCCC2.n1(C(COC)COC)cc(C)nn1 c1(C(N(CCN(C(c2c(C)cco2)=O)C)C(C)C)=O)ccc2c(c1)CN(C)CC2 CC(C)C(C)CC(=O)N1CCCCC1CN(C(=O)CCNC(C1CCCC1)=O)C C12(NC(c3ccc(OC)cn3)=O)CCCC1N(C(c1ccno1)=O)CC2 n1(CCCC=C)cc(NC(C23CC(F)C2C3)=O)nn1 C1(C(C(=O)N(CC=CC(=O)N(C)CC2CCOC2)C)O)CCCCC1 c1(C(C(=O)NCC(CC)NC(=O)C=Cc2cc[nH]c2)(C)C)cccc(OC)c1 C1(CC(=O)NCCN(C(=O)Cc2cc(C)[nH]n2)CC)CS(=O)(=O)C1 C1(C)(CNC(CCOCC(C)C)=O)CN(C(=O)CC2CC=CCN2C)C(C)(C)C1 C1(COC)C2CCCC1N(c1nc(-c3cnccc3C)ns1)C2 N1(C(C23C(C)OC(CC2)C3)=O)CCCCC2(CCN(C(C3CC=CC3)=O)C2)C1 Cc1n[nH]c(C)c1C(C)C(=O)NC1CC1CNC(c1csnc1Br)=O c1(C(N(CCCNC(C2Cc3nccn3C2)=O)C)=O)sccc1S(N)(=O)=O Cc1nc(CC(N2CCCC(NC(=O)Cc3ccccc3Cl)C2)=O)[nH]c1C C1(C(N2CCC(OCC3CC3)C2)=O)CC=CCN1C(=O)Cn1ccnc1 C12(NC(c3onc(C)c3C)=O)CCCCC1N(C(=O)CCc1ncc[nH]1)CC2 C1(OC(C)C)CC(F)(CNC(C2C(C(F)F)C2(C)C)=O)C1.C1(C)CCN1C=O C(=O)(C(C)CC(=O)OC)NCC1C(CC(=O)N(C(CO)CO)CC)C1 C(CCCC(=O)NC1CCOC1=O)N(C(Cc1cc(C)[nH]n1)=O)C N1(C(CCCOCC)=O)CC2CCCC1(CNC(c1cc(OC)n(C)n1)=O)C2 c1(C(=O)NCCC(C)NC(CS(=O)(=O)NCC)=O)nnc2ccccc2n1 c1(C(N2CC(CNC(C3(CC)COC3)=O)N(C)CC2)=O)cc2n(n1)CC(F)C2 N1(C(C(C=C)O)=O)CCCCC(C2CN(C3CCN(c4ccccc4)C3=O)C2)C1 c1(CNC(c2n(C(C(=O)OC)C)nnn2)c2cc(C(C)C)no2)c(Cl)cccc1Cl c1(C(C(=O)NC2CCCC2)N(CCC)C2CC2)cc(C2CC2)cc(C)c1 c1(CC)nc(C)c(C(N2CCC2CC(=O)NC2CC3CCCCCC23)=O)c(C)n1 c1(C(N(C2CCCN(C(c3cc(O)ncn3)=O)C2)CC)=O)ccc(C)nc1C C1(C(N2C(C)(CCC(N3CC(C)(C)C3C3CC3)=O)CCC2)=O)C2CCCC(=O)C12 Cn1ncc(Cl)c1CC(=O)NCC(C)(C)CCNC(=O)C=Cc1cnc[nH]1 C(=O)(CC(F)(F)Cl)N(C1CCN(C(=O)Cc2nocc2C(C)C)CC1)CCC N1(C(c2cn(C)nc2OC)=O)CCCC(C)C1.C1C(C)NC(=O)C=CCN1CC N1(C(C=Cc2ccc(OC)c(O)c2)=O)CCOc2ncc(C(C)C)c(C)c21 c1(C(=O)NC2C3(CN(C(CC=C)=O)C3)CCC2)ccc2c(c1)OCCN2C C1(C(N2CCC(NC(C(C3(O)CC(C)(C)C3)(F)F)=O)CC2)=O)C2CCCCCC12 N1(C(CC2=NNC(=O)C2)=O)CCC(C2CN(C(=O)CC3CC=CCC3)C2)CC1 c1(C(N(CC(CN(C(=O)C(F)(F)c2ccccn2)C)O)C)=O)cc2n(n1)CCO2 CCC(CCC(=O)N1CCC(C)(C(C)C)CC1)NC(C1CCCCC1(C)C)=O c1(C(=O)NCCC2N(C(C(C)OCC#C)=O)CCCC2)ccc(F)c2[nH]ccc12 N1(C(C=C(C)C)=O)CCC2(CC1)COC(CNC(c1cc[n+]([O-])cc1)=O)C2 c1(C(N2CC(CNC(c3c(C)nco3)=O)C(C)(C)C2)=O)cc(F)cc2ccoc12 C1(=O)CCC(C)(C)CCO1.C1(CC(=O)NCCC2ON=C(C)C2)CC(=O)NC1=O C(CCCCCC(=O)NCc1cc(O)ncn1)NC(CC)=O C1(CN(C)C(=O)NCc2nc(C#N)cs2)NC(=O)CC1(C)C C(=O)(C1=CCCN(C(=O)C(C)(C)N2CCCC2)C1)N1CCC(C2(C)N=N2)C1.S(C)(=O)(=O)NC C12(C(=O)NC3C4CC(NC(CCCCC)=O)CC43)CC3CC(C(=O)N1)C2C3 O=C1CNc2cc(C(N3CC(NC(=O)C=CBr)C4CCCCC34)=O)ccc2N1 N1(C(CCOC(CC(C)C)C)=O)C2CCC1CN(C(C13CC(CCO1)C3)=O)C2 N1(C(CCC#C)=O)CC(O)CC1CNC(C1(N(C)C)CCCC1)=O c1(SC)ccccc1C(=O)NCCC(C)CCNC(=O)CCc1cnn[nH]1 CCC(CC)CCCNC(C1CCN(C(c2cc3n(n2)CCC3)=O)CC1O)=O c1(NC(C2N(C(COCCOC)=O)CC2)=O)cnccn1 N1(C(c2ccc(C)c(Br)c2)C(=O)NC=O)CCC(C)(C)CC(C)(C)C1.C1(C)C(=O)N1 N1(C(c2ccc(CC)[nH]2)=O)CC2CCCC2(CNC(=O)Cc2nnc(C)o2)C1 C1(C)(C(=O)NC(C)CCCCNC(C2CCC(C)C(C)C2)=O)CC(C)OC(C)C1 C1(C(N2CCC(C(C(=O)NC(c3ncccc3F)C)(C)C)C2)=O)CC(=O)CCO1 c1(SCC)cccc(C(=O)OCCCc2ncccn2)c1 C1(CN(C(=O)Cc2ccc(F)cc2)C)CCCN(C(=O)CSC2CCCCO2)C1 c1(OCCOC)cc(C)[nH]c(=NC(=O)OCC2COC2)n1 C=C(C)CC(C(=O)N1C(CO)CC1CO)NC(c1cccnc1)=O C(=O)(CCCN(C)N=O)NC1CC2C(NC(c3ccc(OC)cc3C)=O)C2C1 c1(C(=O)NCC2C(NC(C(F)=CC)=O)CCCC2)ccc(P(C)(C)=O)o1 C12(NC(=O)C(C3CCOCC3)c3ccccc3)CCCC1C2 C(=O)(C(C)C1CCCO1)NCCN(C(=O)CN(C1CCCC1)C)C(C)C c1(OC)ncc(C(=O)NCCOC2CCN(C(=O)C(=O)NCC(F)F)C2)nc1C Cc1cc(=O)c(C(=O)N(C)CCOCCN(C)CC2CCCC2)c[nH]1 C(=O)(CC1=CCN(C)CC1)N(C1CN(C(=O)COC(C)(C)C)CC1(C)C)C N1(CC)CCCC(NC(c2cc(CNC(c3n(CC#C)ccc3)=O)[nH]n2)=O)C1 CC(=O)CCCC(C)C(=O)NCCN(C(C1CC1C1(C)COC1)=O)C(C)C CC1CCC=C1C(=O)Nc1cn(-c2ccc(OC(F)F)cc2)nn1 c1(NC(c2c(NC(C(c3cn(C)nc3)O)=O)c[nH]n2)=O)cc(F)ccc1[N+](=O)[O-] c1(C(CC)NC(=O)NC(C)CN2CCSCC2)ccncc1 CC1c2nccn2CCN1C(=O)C1=CCC(NC(=O)CCn2cnnn2)C1 C12(C=O)CCCC1CCN2C=O.N1(N(C(C)(C)C)C)C2CCC1CC2 C(=O)(N=c1ccn(C2CN(C(C3CC34CCCCC4)=O)C2)[nH]1)c1c(C)cco1 c1(C(CC)C(=O)NC23CCOC(CNC(C)=O)(C2)C3)ccc2c(c1)OCCO2 C1(C)(C(=O)NC(c2ccccc2)CC)CCN(C(=O)Cn2nnnc2C)C1 c1(NC(C2CCC(C(C)C)CC2)=O)ccc(Cl)cc1CN1CCOC(O)C1 c1(C(=O)NC23CC(NC(C4C(C)CN(C)C4)=O)(C2)C3)cc2c(Cl)cncc2s1 CC(C)(C)CC(O)CC(=O)N1CCCC1C=CC(=O)NCC1CCc2nccn21 N1(C(C=Cc2c(C)n(C)nc2)=O)CC(C)CN(C(c2cn(C)nc2Cl)=O)CC1C CC(C)CC(O)C(=O)N1CCC(C)(NC(c2cnc(=N)[nH]c2)=O)C1 c1(C(=O)OC)cc(C)cnc1N1CC(NC(=O)C=CCO)C(O)C1 N1(C(C2CC=CC(NC(C3(C)CCCN(C)C3)=O)C2)=O)CC2(CCOC(=O)N2)C1 C1(CNC(C2CC(=O)NC2)=O)CN(C(C2C3CC4C(C3)C24)=O)CCCO1 CN1CC(C(=O)NCC=CCNC(=O)CCCc2nccs2)CCC1=O c1(C(N(CCC)CCNC(=O)C=C2CCOCC2)=O)ccnc2cc[nH]c12 C=CCC(CNC(c1csc(CO)n1)=O)NC(C1(Cl)CC1(F)F)=O N1(C(C2CCC(=O)N2)=O)CC2(C1)CN(C(=O)C(F)(F)C=Cc1ccccc1)C2 c1(OC)cc(CN2CCC(NC(c3c(Cl)cccc3Cl)=O)CC2)ccc1C(F)F N1(C(c2c(OC)scc2)=O)CCN(C(c2coc3c2COC3)=O)C(C)C1C Cc1cc(C(=O)NC(C2CCN(C(=O)C3=C(Cl)CC3)C2)(C)C)cc(C)c1Cl C1(NC(C(C)NC(C)(C)C)=O)COC2(C1)CN(C(=O)CCCCCn1cnnn1)C2 C1(CNCc2cc(C)n(-c3ccccc3)c2C)CC(C)(C)CCC1O c1(C(N2CCCC(NC(C3(C)CCC(C)C3)=O)C2)=O)ccnc2ccsc12 c1(CC)ccnc(C(=O)N(C(C)CNC(=O)Cn2cc(C3CCOC3)cn2)C)c1 c1(CCC(=O)NC2(C)CCCCC2C(=O)O)ccc2c(n1)NCCC2 N1(CC#C)CCC(C(=O)NC2CN(C(=O)C(C)CN(C)C)CC2C)CC1 C(C(CN=c1nnn(C)[nH]1)C(F)(F)F)NC(CCC(C)N(C)C)=O C(CCC)(C(=O)NCCCC(c1ccccc1)NC(C1(C(C)=O)CC1)=O)=CCC N1(C(c2cc(C)[nH]n2)=O)CCCC(NC(=O)C(C)(C)c2cc(Cl)sc2Cl)C1C C1(NC(=O)Cc2cc[nH]n2)C2CCC1N(C(=O)CCc1cccc(F)c1Cl)C2 C(CC)(C(=O)NC1CC(C(F)C(=O)N(C2CCC(C)C2)C)C1)=CCCC CN1CCC(C(N2CC3CCC3(CCNC(=O)Cn3cnc(=N)[nH]3)C2)=O)S1(=O)=O CCC(C)C(=O)C(=O)NC1CC1NC(C1(CC)CCNC1=O)=O CN1CCC(C)(NC(N2CCCC2Cc2cc(F)ccc2F)=O)CC1 C(=O)(C1=CCCCO1)N(C1CC(NC(c2ccc(N)c(Br)n2)=O)C1)C c1(OC)ccc(C(=O)NCC(F)(F)C2(OC(F)F)CC2)c(OC(F)F)c1 n1(CC2(C(=O)NC3CC(C(C(=O)NC(C)(C)C)F)C3)CC2)c(O)nnc1O C1(NC(C2N(CC)CC2)=O)CC2CC(C1)N(C(c1ccn(CC(F)(F)F)n1)=O)C2 C=CCCCCC(=O)N1CCC(C=CC(=O)NC(COC)C(C)C)CC1 C1(C(N2CCCC(C3CCCN3C(c3cnsc3)=O)C2)=O)Cc2nccn2C1 Cc1cnc(C(=O)NCCCCN(C)C(c2nc(C(C)(C)C)no2)=O)c(C)c1 C1(C(=O)Nc2ccc(C(C)(C)C(F)(F)F)cc2)CC2(CC2)CN1C(=O)CN c1(NC)cnc(C(N2CCC(C)(NC(=O)CN(c3ccccc3)C)C2)=O)cn1 C(F)(F)(C(=O)NC1(CNC(c2csnc2-c2ccccc2)=O)CCC1)SC c1(NS(=O)(=O)CC2CCN2CCOC)cc(Cl)cc(Cl)c1 CC1OCCN(C(=O)CC2CCCN2C(C2CC3CC(=O)C2C3)=O)C1C N1(C(CCCCSC)=O)CC2(NC(c3ccc(S(N)(=O)=O)[nH]3)=O)CCCC2(F)C1 N1(CC(N2C(C(C(=O)NCCCCCSC)(C)C)CCC2)=O)CCNC(=O)C1 N1(CC)OCC(NC(=O)C(CCC2CC2)NC(=O)NC(C)C)C1=O N1(C(CCc2nc(C)oc2)=O)CC2CN(C(=O)C(C)(F)c3ccon3)CC(C1)O2 C1(C(=O)NCC=CCNC(CC(C)OC)=O)CC(=O)N(CCc2ccccc2)C1 C(CC(C(C)(C)C)NC(c1cn(C(F)F)c(C)n1)=O)N(C(CCOCC#C)=O)C C1(C(=O)NCC2CN(C(c3ccoc3Cl)=O)C2)CC2CC(O)C(C1)C2 C(=O)(C(C)C(C)(C)C)N1CC(N(C(C(C(C)C)c2ccc(F)cc2)=O)C)C(O)C1 C1(CNC(C2CC2(F)F)=O)CC2(CCN(C(c3cc(=O)cc(Cl)[nH]3)=O)C2)CO1 CCC(CCCC(=O)NCC(C)(CC)C(N)=O)NC(c1nnsc1N)=O c1(NC)cc(C(=O)NC(C2CCN(C(C3CC(=C(F)F)C3)=O)C2)C)cc(Cl)n1 Cc1ncccc1C(N1CCC(C(C)(C)NC(=O)Cc2ccccc2C)CC1)=O Cn1nnnc1N1CC(C(=O)NC2(CCCNC(=O)CSC3CC3)CC2)C1 CCC(O)C(C)C(=O)NCC(CC)(CC)NC(=O)CN1CCCCC1 c1(CC)noc(C(=O)NCC(C)(C)OCCNC(=O)C(n2cc(Cl)cn2)C)c1C c1(C(=O)NC(CNC(C(C)(C)N2CCCC2)=O)(C)C2CCC2)cc(F)cc(F)c1 C(=O)(CC(CC(N)=O)CC(C)C)NCC(CC)(CC)NC(=O)COC1CC=CC1 C1(C2CCN(C(=O)C=CC(C)C)C2)(NC(CN2CCCCC(OC)C2=O)=O)CC1 c1(NC(c2c(C)nccc2)C)nc(N(C)CC2COC(C)(C)O2)c2ccsc2n1 CCC(C(=O)OC)C(=O)NC(C)(C)C=CC(N1CC=C(C)C1)=O c1(-c2cc(OCC)no2)nc(-c2cc[nH]n2)nn1CCc1cccc(F)c1 C1(C(N2C(C(=O)NCC3=CCCC3)CCC2C2CC2)=O)CC2(CCC2)CO1 N1(C(Cc2c(C)cnn2C)=O)CC2CCCC2(NC(=O)C(F)=C2CCC2)C1 c1(C(=O)NCC2(F)CCN(C(c3cc(C)ns3)=O)CC2)c(C)sc(C)c1C#N CCC(C)(CNC(=O)OC(C)(C)C)C(=O)N1CCCC(C)(CNC(=O)C(N)=O)C1 N1(C(C2COCC(C)(C)O2)=O)CC(O)(C2(CNC(=O)C3CC3)CC2)C1 C(CC(=O)NC12CCCC1CN(C(=O)Cn1c(C)csc1=O)C2)(C(F)(F)F)OC c1(NC(=O)C2CC2)ccccc1S(=O)(=O)NC1C(C=C(Cl)C(F)(F)F)C1(C)C C1(C2CC2)(C(=O)NCCCOCCN(C(C(C)S(N)(=O)=O)=O)C)CCOCC1 C1(O)(C(=O)NCCC2(CNC(C(n3cc(Cl)cn3)C)=O)CC2)CCCC(C)(C)C1 C(=O)(CCN(C)C1CC1)N(CCCNC(C=C(C)I)=O)CC.C(=O)(CO)N C1(NC(C=CC=CC)=O)CCCC12CN(C(C1CCCSC1)=O)C2 c1(CC(=O)NC2C=CCN(C(C(n3cc(Cl)cn3)C)=O)C2)ccc2c(c1)CCO2 CP(C)(=O)CCC(=O)N1CC(O)CCC1C(N1CCCC(C(N)=O)C1)=O N1(C(=O)COc2ccccc2O)CCC2OCCN(C(=O)CCc3nncs3)C2C1 C12(CC(=O)NCCC(C)NC(C3CCCC3c3cnn(C)c3)=O)COCC(C1)C2 c1(C(=O)NC(CNC(C(c2c(C)n[nH]c2C)C)=O)C)cc2c(nn1)OCCS2 c1(OC)c(C(=O)NCC(CO)NC(=O)C(C)Cc2cnn(C)c2)cc(F)cc1F N1(C(c2n(CC)nnc2)=O)CC(NC(C2(F)CC3(CCC3)C2)=O)CC2(CC2)C1 C1(OC(C(C)c2ccco2)=O)CN(C(c2ccc(Cl)cc2)=O)C(=O)CO1 C(C(C)C(C)(F)F)NC(CC1C(NC(C(C)C2CCC2)=O)CC1O)=O CN1CCC2(CC1)CN(c1nc(NCc3ccncn3)c3ccsc3n1)CCO2 c1(-n2cc(CN(CC#C)CC=C)nn2)c(Cl)cccc1Cl C(C(CC(=O)NC1COCC1O)OC)NC(c1c(OC)scc1)=O c1(C(=O)NCC(C)N(C(c2cc(CC(C)C)[nH]n2)=O)C)c(F)c(C)cc(N)c1F C(=O)(CC(C)COC)NC(C1(C(=O)NC(CCC=C)C2CC2)CC1)C C#CC1(O)CCN(C(c2ccoc2CNC(C2CC3(CSC3)C2)=O)=O)CC1 Cc1ccnc(C)c1CN1CCCC(N(CCCCO)C(C2CC2)=O)CC1 C(=O)(C(C)(C)CC1CCCO1)N(CCCNC(C1CC1C(C)(F)F)=O)C(C)C.CO C1(C(=O)NCC2(CCNC(C3CC(OC)C3)=O)CC2)CCCCS1 C1(C(=O)NC(CC)CNC(=O)C(F)n2cccn2)CC2(CCC2)C1 CCC(CC(=O)N(C1CCCC1)CCCNC(=O)C(COC)OC)C1CC1 C(=O)(C1=NOC(C)(C)C1)NCC1N(C)CCN(C(C2(C)CC=CC2)=O)C1 c1(NC(=O)NC)cccc(C(=O)NCC(C)N(C(=O)C(F)(F)C2(O)CCC2)C)c1 c1(OCC(CNC(=O)C(c2cccc(Br)c2)O)O)cc(O)c(Cl)cc1Cl N1(C(C(C(=O)OCC)F)=O)CCN(c2ncnc(CC)n2)CC1C c1(C(=O)OCCSc2cn(C3CCC3)nn2)cc(Br)c(C(C)(C)C)s1 CC1(CNC(=O)N)CC(F)(F)C1.C1(C)CC(O)(CC#N)C1 N1(CC(=Cc2cccs2)C)CC=CC1(C)C S(=O)(=O)(c1cc(Br)ccc1F)N1C(C(=O)Nc2ncc(Cl)nc2Br)CC(O)C1 c1(CC)ccc(F)c(C(=O)NCC(C)NC(c2ccc(C(C)C)o2)=O)c1F c1(CN(C)C(c2sccc2C(C)(C)C)=O)ccc(CNC2(CC3CC3)CC2)cc1 C1(C(N2CC(OC)C(NC(C3(C)CC(O)CN3C)=O)C2)=O)CNC(=O)CC1C n1(C2CC(N)C2)ncc2ccc(CCCCNC=O)cc12 Cn1nc(C(=O)NCCC2CCCN2C(=O)CCn2ccnc2)cc1O c1(OC)cc(NC(C2CCN(C(c3cc(C(C)(C)C)on3)=O)C2)C)ncn1 C12(CC)CC(CN1C(=O)OC(C)(C)C)C2.c12cnccc1CC(C)NC2 CC(=O)C(C)(C)CC(=O)NCCc1cncc(C(F)(F)F)n1 CC1CC(=O)NCC1C(N1CCCC(Cn2cc(CCN3CCCC3=O)nn2)C1)=O C1(C)(NC(CC(C=C)C)=O)CCN(C(=O)COc2ccc(Br)cn2)CC1 C1(O)(C(N2CC(CN(C(=O)COCP(C)(C)=O)C)OCC2)=O)CCCC(C)(C)C1 c1(CNC2C(C(=O)Nc3onc(C)c3C#N)C2)cc(C#N)ccc1O N1(C(C(C=C)O)=O)CCC(O)(CCNC(c2cc(C)on2)=O)C1 C(CN=c1[nH]c2ncnc-2c(C(F)(F)F)[nH]1)(N(C(=O)Cc1cnc[nH]1)C)C1CC1 CC1CC2(CCC2)CN1C(C1CCC(C)N(C(C2CCCCC2)=O)C1)=O N1(C(CN(C)C(C2CCCCO2)=O)=O)CCN(CC2CC2)CC1 C(=O)(C(O)CCN1CCCC1)NC(CC(C)NC(CCCC)=O)C CC1CN(C2CC(=O)N(C3CN(C(C4CCC=CO4)=O)C3)C2=O)S(=O)(=O)C1 N1(C(COCC(C)(C)C)=O)CC2CC2(NC(=O)CC2CCOCC2)C1 C(=O)(C1=C(Cl)CCC1)NCC1N(C(c2cn(CC)nc2C2CC2)=O)CC(OC)C1 c1(CC(=O)NCCC(C)(C)NC(C#CC2(C)CC2)=O)c(F)c(F)cc(F)c1F c1(C(=O)NCC(C)NC(CCC(=C)Cl)=O)oc2ccc(C)cc2c1C C(=O)(C(C)C(C)NC(=O)CC1CC(N(C)C)C1)NCC=C(CC)C n1(CC(=O)NC2CCC(NC(C(CC)(C)O)=O)C2)c(C)cc2ccccc12 C(=O)(C1=NOC2(CCC2)C1)NC(C(=O)NCC(CC)NS(C)(=O)=O)(C)C(C)C C12(C(=O)NCC(CC)NC(C3(CC(C)C)CCNC3=O)=O)CC(C)(CO1)C2 c1(C(C(=O)NCCC2CC2)N(CC)CC)cccc2c1CCO2 C1(C(=O)Nc2nc(C)nc(O)c2)CCCC12CCN(S(=O)(=O)CCCCl)C2 c1(CC(N2CC(CC(=O)NC)N(C(=O)C3=C(Cl)CC3)CC2)=O)c(C)cc(C)nc1O Cc1ccc(CC(N2CCC2CC2C(C(=O)N(C3CCOCC3)C(C)C)C2)=O)s1 C(CC(=O)NOCc1ccccn1)(C(C)C)NC(c1cncc(C)c1)=O N1(C(C(C)CF)=O)CCN(C(c2cccc(C(F)F)c2)=O)CC1C1CCC1 N(C(=NCCCC(C)(C)O)NC1CCN(c2ccc(Cl)cc2)C1)C1CC(OC)C1 C(=O)(CC(C)(O)COC)NC1(CF)CCN(C(C(C)NC(=O)OC)=O)C1 Cc1cc(CCC(=O)NC(C2CCN(C(c3conc3C)=O)C2)C)cc(C)c1 c1(C(C(=O)NCC=CCCNC(C2CC2CF)=O)N2CCCC2)ccccc1 N1(C(CC2N(C(C3CC(=O)NC3)=O)CCC2)=O)CC2CCC(O)C(O)C12 N1(C(CSCCC)=O)CCCC(CCNC(c2[nH]ccc2CC)=O)CC1 N1(C(C(OC)OC)=O)CC2(CCC2)CC1CNC(C1CCCC1C(F)F)=O N1(C(=O)C(C2CCOCC2)F)CCC2CCN(C(C3CCS(=O)(=O)CC3)=O)C2C1 C1(NC(CCSCCCC)=O)C2CCN(C(c3occ(C)c3C)=O)CCC12 Cc1nn(CC(N2CCC(C)(CNC(c3ccn(C)c3)=O)C2)=O)c(C)c1[N+](=O)[O-] Cc1cc(F)ncc1C(=O)NCC1(F)CC(NC(c2[nH]ccc2C)=O)C1 N1(C(C2(COC)CCOCC2)=O)CCC2(CC1)CCN(C(C1CC1C)=O)C2 c1(N2CC(C)(C(=O)NCCN3CCS(=O)(=O)CC3)C2)ncnc2c(F)cccc12 N1(CC(=O)N(C(C(=O)NC(C)C(C)n2cncn2)C)C2CC2)CCOCC1 CC(C(=O)N1CCCC1CC(=O)NCCC(C)(C)N(C)C)S(N)(=O)=O c1(C(N2CCCCC(N(C(C=NOC)=O)C)C2)=O)cc(C)c(Cl)cc1Cl C1(C(C)C)CN(C)CCN1C(c1ncoc1Br)=O C1(NC(CCSCC(C)C)=O)CCCCN(C(=O)CO)CC1 c1(C(=O)NCC(CC)NC(=O)Cc2cn(C)nc2Cl)c[nH]c2cccnc2c1=O c1(C(C(=O)NCC(C)(O)CNC(C2CCNC2=O)=O)O)ccc(O)c([N+](=O)[O-])c1 C1(C(N2C(CC(c3ccco3)=O)CCC2)=O)CCOC2(CCOCC2)C1 CC(C)(C)CC(O)C(=O)N1CCC(NC(c2ccc(C3CCCO3)[nH]2)=O)C(O)C1 C#CC1CN(C(=O)CC2CCCN(C(c3c(C)nsc3C)=O)CC2)CCO1 C=C=CC(C)C(=O)NCC(C)(C)CN(C)C(C1CCN(c2nc(=N)[nH][nH]2)C1)=O N1(C(c2ccc(OC)c(F)c2)=O)CCCC2(CCCN2Cc2cnc(Br)s2)C1 CC(C)C(N)CCNS(=O)(=O)C1CC1c1ccccc1Br C(=O)(C1=CC2CCCCC12)NCC1CCC2(CN(c3nc(CC)nc(=N)[nH]3)C2)O1 c1(NC(C(CC)C(CC)CC)c2n(CCCC)nnn2)cccc2c1OCCO2 C1(C(=O)Nc2cc(COc3cnn(C)c3)on2)(CNC(C2C(=C)C2)=O)CCOC1 N(C(=NCC(C)OC)NCC(F)F)CCOC1(CC=C)CCOCC1 C(CCCCC(=O)NCCCN(C(C1CCC2C1C2(F)F)=O)CC)OCCC=C C1(C(=O)NC2(C)CN(C(c3cccnc3S)=O)C2)CC(O)C(F)C1 C=CC(CCC)CC(=O)NCC1CCCN1C(c1cc(-c2ccncc2)on1)=O C(=O)(C1CCc2cccnc21)N1CC(NC(c2c(CC)non2)=O)C(N=[N+]=[N-])C1 n1(CC)nc(C(=O)NC2CC(NC(C3(C4CC4)CCC3)=O)C2)c(C)n1 c1(C(C)OCS)c[nH]ccc1=NS(=O)(=O)c1ccccc1 N1(C(CC(CCC)C)=O)CC2CC(NC(=O)C3=CCCCC3)CC(C2)C1 c1(C(N2C(C(=O)NCc3nnc(C)o3)(C(C)C)CCC2)=O)cn(C)ccc1=O N1(C(COC)=O)CC2CC(NC(C3(C(F)(F)F)CCC3)=O)CC2C1 C(N=c1nc2sccc2c(Nc2nc3ccccc3s2)[nH]1)C1CC(C)C1 N1(C(C(=O)NCc2c(C)cc(F)cc2)=O)CC2CC(N)CC1C2 C(=O)(C1=CS(=O)(=O)CCC1)NC(c1ccccn1)C.CC1C(=O)N1 C(=O)(CCCCCCNC(=O)CC1CCCCO1)N(C1C(C)CC1)C c1(C(N(C(C)CNC(C2(O)CCC2)=O)C)=O)cc(Cl)nn1C CCCCC(O)CC(=O)NC1CCN(C(c2cncnc2)=O)C1(C)C N1(C(C2C(CC)N(C(c3cc(C)sc3C)=O)CC2)=O)CC2CCCC2(CO)C1 C1(C)(C(N(CC=C)CCC)=O)CN(C(=O)C(C#N)CC)C(C)(C)C1 C1(NC(Cc2ccc(SC)s2)=O)C2CCN(C(=O)C(N3CCOC3=O)C)C12 c1(CN2C(CC=C)(C(=O)OC)CCC2)n[nH]c2ccc(NC(=O)C(F)(F)F)cc12 C1(NC(CCC2C(C)C2)=O)CN(C(c2ccccc2F)=O)CC1CC(C)(C)C c1(OC)cc(C(=O)NC2CCCC2NC(=O)CCSC(F)(F)F)ccc1O N(C1c2ccccc2C2CC12)NC(c1n(C)nnn1)(C)Cc1c(Cl)cccc1Cl C1(S(C)(=O)=O)(C(=O)NCCCC(C)NC(=O)CC=CC(C)(C)C)CCC1 N(C(=NCC1CC1)NCC(c1ccc(Cl)cc1)CC)N(CC(C)OC)C(C)C.CO c1(C(N2CCCC(COCC)C2)=O)ccc(C)c(Cl)c1N.C12C=CC(C1)NC(=O)C2 c1(C(=O)NCC2CN(C(c3cnc(C4CCCO4)s3)=O)C2)cccc2c[nH]nc12 CCCC(CC)CC(=O)N1CCN(C(C23CCC(F)(CC2)C3)=O)CC1C(C)C N1(C(C2(C=C)CC2)=O)CCC(NC(=O)CC2(CC=C)CC2)C(C)C1 CCC(CCC(=O)NCc1nc(C(N)=O)co1)NC(C1CCCCNC1=O)=O c1(N2CC(C)(C)C2)ccn2ncc(S(=O)(=O)NCC3CCCC(N(C)C)C3)c2n1 CC(C)(C)C(=O)C(=O)N1CCC(n2cc(NC(=O)COCCN(C)C)cn2)C1 N1(C(c2c(O)ccc(N)c2)=O)CCOC2CCNCC12 Cc1nc[nH]c1CNC(=O)CN(C1CC1)C1CC1 C1(C2CCCC2)(C(=O)NCCCCCCn2cc(C(CC)O)nn2)CCNC1=O N1(C(C2CN(C(C(C)(C)N=[N+]=[N-])=O)CC(C)(C)C2)=O)CC2(CCC(O)CC2)C1 c1(NC(C(=O)N(CCNC(c2nnnn2C2CC2)=O)CC)=O)c(F)cccc1F C1(C)(CNC(C2C(=C)CC2)=O)CN(C(=O)CCc2ccc(F)cc2Cl)CCO1 Cc1ccc(N)c(C(=O)NC2CC(NC(=O)Cc3sc(C4CCC4)nc3C)C2)c1 c1(CC)cc(C)c(C(=O)NCCN(C(=O)C#CC2CC2)Cc2ccc(F)cc2)o1 N1(C(C2(C)CC(=C)C2)=O)CCC(C)(C)C(NC(=O)C(=O)NC(C)C)C1 N1(C(c2cnc(C)o2)=O)CC(NC(=O)C(O)C2CC2)CC2(CCC2)C1 C(=O)(C1=CC2(CCOC2)C1)NC1CC2(CC(N)C2)C1.Cc1ccc(C)c(C(=O)N)c1 C1(NC(CCN(c2ccncc2)C)=O)CCCCN(C(C23COCC(C2)C3)=O)C1 C1(CC)COCCN(Cc2cn(C3CCOC3(C)C)nn2)C1 Cc1c(C(=O)NCCCN(C)C(C2(C)CC2)=O)nnn1C CN1C(=O)CCCC1C(=O)NC1CCC12CN(C(=O)COC1(C)CCC1)C2 CN=C(NCc1ccccc1)NC1CCN(CC(C)(C)C(C2CCCCC2)OC)C1 C(=O)(C1CCc2cc(Cl)ccc21)NCC#CCNC(C(C(C)C)NC=O)=O c1(C(=O)NC2CC2C(=O)Nc2cncc(Cl)c2Br)cccc2ccncc12 CON(C)C1CN(C(C2(NC(=O)CCCN3CCCC3)CCN(C)C2)=O)C1 C1(C(N(CC(CC)OC)C)=O)CN(C(=O)CCCCCSC)CC1(C)C N1(C(c2nc(COC)[nH]n2)=O)CCC2(CCCN2C(=O)Cc2cc(C)ns2)C1 c1(C(N2CCCN(C(C(C=C)O)=O)CC2C)=O)cccc2cc(O)ccc12 N1(C(c2cccc(C)n2)=O)CC2CC1CN(C(C1COCCN1C)=O)C2 C1(CC(=O)N(C(C)C)C2CC2)CCN(C(=O)C=CC2CCOCC2)CC1.C(C)S N1(C(C(C)CC(C)(C)C)=O)CC2(CCCCN2C(C2CC2CN(C)C)=O)C1 c1(CCCCN(C(=O)Nc2cccc(OC)c2)C)nccc2ccccc12 C1(NC(c2cc(C3CC3)[nH]n2)=O)CC2CCC1CN(C(=O)C(C1(O)CCCC1)F)C2 CC1(C)CC(CNC(N2CCC(Cn3cccn3)C2)=O)OC(=O)N1 Cc1noc(C)c1C(C)C(=O)NC1CCC(F)(CNC(=O)C(=O)NC(C)C)C1 CCC(C)(C)C(O)C(=O)N1CCN(C(=O)CCn2cnc([N+](=O)[O-])c2)C(CF)C1 N1(C(C#CC)=O)CC2CN(C(=O)COc3cccc(CC#N)c3)C2C1 Cc1sc(O)nc1C(=O)NCCCN(C(=O)C=CCO)CC1CCCO1 c1(C(N2CCC(OCC(N)=O)C2)=O)ccnc(CNC(c2ccc(F)s2)=O)c1 C12CCCN(C1)C(=O)CN(CCOC)C2=O.c1(CC(=O)NC)ncn(C)c1C CC1C(Cc2ccccc2)CCN1.C1(CO)CC1Cl C12(C(=O)Nc3cn(CC=C)nc3)CC(CO)(CN1C(=O)C(C)(C)n1cncn1)C2 C1(OCC(=O)NC2CCCOC2)CN(C(=O)CCn2cnnn2)CCC1CO C(c1cc(Br)cs1)=CC(=O)N(C(CNC(CC1(CSC)CC1)=O)C)C c1(CN2CCOCC(C(=O)Nc3cncc(C)c3)C2)cnc2cc[nH]c2c1 C1(CC)CN(C(c2ccc(COC)cc2)C(=O)NC(C)(C)C)CCO1 c1(SC)nc(Cl)c(C)c(=NC2CC(CNC(=O)C3=CCCCO3)C2)[nH]1 C1(C)(C(=O)NC(C2CN(C(c3nnc(S)n3C)=O)C2)C)C=CCCC1 C1(C(=O)NC(C)CCCCO)CCCN(C(=O)CCn2cccn2)C1C c1(CNC(c2nc(C(=O)NC(C)CCO)sc2)=O)c(F)cccc1F N1(C(C2CC(C(=O)OC)C2)=O)CCC2CCN(C(C34CCOC(C)(C3)C4)=O)C2C1 N1(C(c2[nH]cc(C)c2)=O)CCC(C)C(CNC(C2(n3cncn3)CC2)=O)C1 N1(C(Cc2ccc(C)o2)=O)CC(CNC(c2nnn(C(C)(C)C)n2)=O)CC1(C)C c1(C(N2C(C)CC(NC(=O)C=Cc3cccs3)CC2)=O)cnn2c1NCCC2 CC1(C)CC(C(=O)N2C3CCC2CC(NC(=O)CC2CC(C(F)F)C2)C3)=NO1 N1(C(c2onc(OC)c2Br)=O)CCCC(C2CN(C(C3CCC3)=O)C2)C1 CC(C)(C)C(CNC(C1(CNC(=O)Cc2nc(=N)[nH][nH]2)CCC1)=O)CO C(=O)(C1=CC2(CCOC2)C1)N(C1CN(C(c2cnc(Cl)cc2Cl)=O)CC1(C)C)C N1(C(CCCCCC)=O)CCN(C(c2cn(C(C)C)nc2C2CC2)=O)CC(O)C1 C1(C(N(C)CC2(C)CC2)=O)CCC(N(C)S(N)(=O)=O)C1.C(C(C)(C)C)OCC(=O)N C1(C(=O)NCCOCCCNC(C(c2ccn(C)n2)C)=O)CCC2CC2CC1 N1(C(c2c(COC)nn[nH]2)=O)CCN(C(C2CCCO2)=O)CC1C(F)F c1(CC(=O)N(C(C)C)CCNC(c2cc(F)cs2)=O)cccnc1O n1(CC)ncc(C(N2CCCC2C2(NC(c3ccc(Cl)s3)=O)CC2)=O)c1Cl C(=O)(C1(C)CCCc2ccccc21)N(C1CN(C(C)=O)C1)C.C1(C)CN1 n12nc(Br)nc1C2C(=O)NC(C)C.N1(CC)CCCC(C(C)(C)C)C1 O=C(C1=NN(C2CCCCC2)C(=O)CC1)NCCCNC(c1cnc[nH]1)=O Cc1cc(CN2CC3C(C2)N3C(=O)Cc2c(C)cccc2C)c([N+](=O)[O-])c(C)c1 N1(C(c2c(C)sc(Cl)n2)=O)CCN(C(c2ccc(F)c(CO)c2)=O)C(C(C)C)C1 Cc1ccc2nc(C)c(C(=O)NCC3CCN3C(=O)C(C)NC(N)=O)cc2c1 c1(C(=O)NCC2CC(COC)CN2C(c2ccco2)=O)cccn2c(O)nnc12 N1(C(C(C=C)(C)O)=O)CCN(C(=O)CNC(c2ccoc2)=O)C(c2cccnc2)C1 C1(CC)C(C(=O)NCCCC2(O)CC2)CCCN1C(c1ccc(O)cn1)=O c1(C(=O)NC(C2(O)CN(C(c3cc(C4CC4)no3)=O)C2)C)cnc2sccn12 c1(C(=O)NCc2ccc(NS(=O)(=O)CC3CC3)nc2)ccc2ncccc2c1 Cc1oc2ccccc2c1CC(=O)NCC(=O)NC1CCCN(CC2CC2)C1 C1(C2(O)CCC2)(CNC(C2N(C(C3N(C(C)=O)CSC3)=O)CC(F)C2)=O)CC1 C1(C(N2CC(CNC(c3nnc(CC)s3)=O)C(C)(C)C2)=O)CC(=O)CC12CCC2 C1(N(C)C(c2cc(CO)n(C)n2)=O)CC2CC1N(C(C1(N3CCOCC3)CC1)=O)C2 C1(COC(=O)NCC(C(=O)OC(C)(C)C)F)COC2(CCCC2)C1 c1(OCCOC)ccc2c(c1)CCN(C(=NCC1CC1)NCc1ccnn1C)C2 C1(CC)CC2CCC(C1)N2C(=O)Cn1nc(Cl)ccc1=O c1(OC)ccc(F)c(F)c1-c1cncc(CN2CC(C)OCC2C)c1 CC1CN(C(C2(F)CCCN(C(=O)C(O)CC3CCCC3)C2)=O)Cc2c[nH]nc21 C1(C(N(C2CCN(C(=O)CCCN(C)C)CC2)CCC)=O)COC2COCC12 CC(C)C(F)(F)CC(=O)NCC1CN(C)CCN1C(C1C2C3CCC(C3)C12)=O c1(OCC(N2CC(CC)C(NC(c3ccoc3)=O)C2)=O)cccc(F)c1F Cc1cc(NC(C2CCC(NC(c3cc([N+](=O)[O-])cs3)=O)C2)=O)cc(Cl)c1 N1(C(c2n(CC)cnn2)=O)CC(NC(=O)Cc2ccsc2C)CC(C)C1 N1(C(C2(OC)CC2)=O)CCCN(CCNC(C2(CC#C)CCC2)=O)CC1 c1(N2CCN(C(C(=O)NC(CC(=O)OC)C)c3csnn3)CC2)nnc2n1CCC2 C(=O)(CCCS(C)(=O)=O)NCCCC(c1ccccc1)NC(c1c(CC)nns1)=O C1(C(=O)NC2(C(=O)OC)CC(CO)C2)CCCC(CNC(=O)C(C)(C)O)C1 CC1CN2CCN12.C12(C=O)CC(CO)(CN1C(C1(C#N)CCSCC1)=O)C2 C1(C(N(CCC)CC)=O)CCC(C)(C)N(C(=O)CN2CCC(OC)C2)C1 S(=O)(=O)(CCCNC(C1(c2ccc(CN)cc2)CC1)=O)N(C)C c1(OC)cc(C)c(C(N2CC(N(C)C(c3cncc(CC(C)C)c3)=O)C2)=O)cn1 c1(C(=O)NCC2N(C(=O)OC(C)(C)C)CC(O)C2O)cc(F)cc(Cl)c1N C=CC1COCCN1C(C1(NC(C2CC23CC3)=O)CC(F)C1)=O c1(OC)c(Cl)cc(C(N2CCC2C(N2CC3CCC2CN(C)C3)=O)=O)c(OC)c1Cl N1(C(C(CC)F)=O)CCC(OCCNC(=O)CNC(c2cncn2C)=O)CC1 C1(NC(C2CC2(F)F)=O)COCCN(C(c2cc(Cl)on2)=O)C1 N1(C(C(CCCC)ON=C(C)C)=O)CCCC2CN(C(=O)C(=O)N(C)C)CC12 C1(C(=O)NCC2C3CC2N(C(c2ccc(CO)cn2)=O)C3)CCCCC1C1CC1 CC(C(=O)NC(c1ccc(F)cc1C(F)(F)F)C)P(C)(C)=O C#CC1(C(=O)NOCc2ccsc2)CCN(C(=O)Cc2cnns2)C1 C1(C(N2C(C(C)NC(c3ccoc3)=O)CCC2)=O)C(C(F)(F)F)C1[N+](=O)[O-] CCC(COC)C(=O)N1CCC(C(C)NC(=O)C=Cc2ccccc2)CC1 c1(C(N2CC(F)(CNC(C(C)OCCOCC)=O)C2)=O)cn(C)c(=O)n1C N1(CC(C(C)(C)C)CO)CC2(CCOC(=O)N2)C1 Cc1ccc(Br)cc1NC(=O)NCC(C1CCCCC1)CO Cc1nn(CCCN2CCC(CO)CC2)c(C)c1S(=O)(=O)Nc1ccc(C#N)cc1 N1(C(c2c(NCC)scn2)=O)CCC(CO)C(NC(c2cc(O)nn2C)=O)C1 C(CC(CC)C(=O)NCC1CC(OC)CN1C(=O)CCNC(=O)OC)=CC c1(-n2cc(C3CCN(C(Cc4ccc(C)nc4)=O)CC3)nn2)cc(Br)ccc1Br C12(C(N3CC(F)(CNC(C=CCOC)=O)C3)=O)CCCC1CC(F)(F)CC2 CC1CN2CCN1C(C(=O)NCC1CN(C(=O)CCn3cccn3)CCO1)C2 C1(NC(c2ccccc2)CNC(c2cncc(C#N)n2)=O)CC2CCCC(C1)C2 C1(C(N2CC(CNC(C3(SCC)CC3)=O)C2)=O)CN2CCN1CC2C c1(CC(=O)N(C(CNC(CSCC#C)=O)C)C)csc2ccc(C)cc12 Cc1cc(Cl)c(C(N2CCCN(C(c3cc4c(s3)COCC4)=O)CC2)=O)cc1F N1(CC#CC)CCN(C(=O)C(CCOC)NC(C2CCCSC2C)=O)CC1 Cc1ccc(C=CC(=O)N(C)CC2CCCN2C(=O)C=Cc2ccncn2)cc1 CC1ON=C(C(=O)N2CC(NC(=O)CCC(=O)NCCC(N)=O)C(C)(C)C2)C1C C#Cc1cccc(NC(=O)C(F)CC2CN(C(=O)CC3OCCCO3)C2)c1 c1(C(=O)NC(CNC(CCc2onc(C)n2)=O)C2CC2)cc2sccc2[nH]1 C(C(F)(F)CCC(=O)OC1CCN(C(N)=O)C1=O)n1cc(CCCC)nn1 CC(N(C)N1CCCC(C)C(CO)C1)c1csc2ccccc12 CC1CCN(C(c2ccn(-c3cccnc3)n2)=O)CC1N(C)C(C1CC1F)=O CN1Cc2ccc(C(N3CC4CCC3CN4C(=O)CNC(=N)N)=O)cc2C1 N1(C(c2ccc(OC)c(O)c2)=O)CC(C)N(C(c2n[nH]c(=N)[nH]2)=O)CC1C Cc1cc(N2CCC(CN(C)C)C2)ncc1S(=O)(=O)NC(c1cccc(Cl)n1)C Cc1ccncc1CC(N1CCCC1CN(C(C1CC1(C)Br)=O)C1CC1)=O C(CCC(=O)NC(CNC(=O)C(C)Sc1nnnn1C1CC1)CO)OC C(=O)(C1CCc2cccc(Cl)c21)N1CC(NC(C=CC(C)C)=O)C1 N1(C(c2ccc(SC)o2)=O)CCOC(C(=O)N(C)CCSc2ccccc2)C1 c1(C(N2CCC(NC(c3cn[nH]c3)=O)C(CO)C2)=O)cc(F)cc2nc[nH]c12 c12ccc(C(F)(F)F)c(c1)NC(=O)CS2.c1(OCC)ccc(C(=O)N(C)C)cc1 N1(CC)CC(C(=O)NCC(CC(C)C)NC(c2cc(C)c(O)nn2)=O)CCC1=O CCC(C)CC(C(=O)NC1(CO)CC(O)C1)NC(=O)Cc1cnccc1C Cc1cc(N2CCC(C)(NC(c3cc(C4CC4)n(C)n3)=O)CC2)nc(C(C)C)n1 N1(C(C2N(C(CC)=O)CSC2)=O)CCCC2CN(C(=O)CC(C)C(C)(C)C)CC12 C12(C(N3C4CC(NC(COC)=O)CC3CC4)=O)CC3CC(C)(C1)CC(F)(C3)C2 C=CCCC(C(=O)NC1CN(CCC)C1)NC(C1(C)CNC(=O)C1)=O C1(C(N(C2CCCCC2)CCNC(C2(C=C)CC2)=O)=O)CN2CCC1CC2 C(CCCCC(=O)NCCN(C(C1CCCSC1C)=O)C(C)C)NC(CC(C)C)=O N1(C(Cc2nnc(C)o2)=O)CCOC(C(C)NC(c2c(C)noc2C)=O)C1 N1(C(c2cncc(SCC)n2)=O)CC(C)N(C(c2sncc2C)=O)CC1C Cc1cc(Cc2cn(-c3ccccc3)nn2)c(C)n1CCc1cc(Br)ccc1O c1(C(=O)NC(CC=C)CNC(=O)CCSC)cc(C(F)F)ncn1 N1(C(=O)NCCS(=O)(=O)NC(C)C)CCCC(C2CC2(F)F)C1 C1(NC(C23CC(CN2C2CC2)C3)=O)CCN(c2ncnc(C(F)(F)F)n2)CC1F CC(C)C(F)C(=O)NC1(CNC(c2ccnc(C(=O)OC(C)(C)C)c2)=O)CCC1 CC1COCC(C(=O)NCCN2C(=O)C3(CC3)C2)O1.C(C)(C)(C)NC(=O)OC C(=O)(CCC(F)(F)C(F)F)NCC1=CCN(C(c2c(C)scc2)=O)CC1 c1(C(=O)NC(CC(C)C)CNC(C23CCC(CO)(CC2)C3)=O)cc(F)cc(F)c1F CC1CC(NC(C2CCCN2C(C2CC(C)(C)CCO2)=O)=O)CC(C)(C)C1 c1(C(=O)NC(CNC(c2ccsc2C(F)F)=O)CO)ccnc2ncccc12 C(=O)(C1=NN2CCC(C)N=C2N1)NCC(CNC(c1c(C)nc(O)[nH]1)=O)CO C1(C(N2CC(CCC)C2)=O)CC(O)C(O)CC1CNC(C1CCC2(CCC2)C1)=O CC1(C)C(CNC(=O)CCc2cnn[nH]2)CCN1C(c1ncn(C(C)(C)C)n1)=O c1(CC)cccc(C(=O)NCc2cccc(OC3CCNC3)n2)c1O c1(NC(CNC(C(=O)OC)C2CCOC2)=O)cccc2c1S(=O)(=O)CCC2 N1(C(=O)NC(c2cccc(C#N)c2)C)CCN2CCC1C2 CCCC(CNC(C1CCCC1C(C)C)=O)C(=O)NCc1nnn(CC)n1 C1(CNC(COC(CC)C)=O)CCN(c2cc(C)ncn2)CC1C N1(C(C2CCC(C)O2)=O)CCN(C(c2ccccc2OCC#N)=O)C(CF)C1 c1(OC)cccc(C(N2CC3(C2)CN(C(=O)Cc2cccc(C)c2F)C3)=O)c1O C(=O)(C(C)(C)COc1ccc(C(F)(F)F)cc1)OCC(C)NC c1(CC)oc(C(N2CCC(CN(C(=O)CSS(C)(=O)=O)C)C2)=O)cc1C N1(C(CC(CNC(CC2OCC(C)(C)C2)=O)O)=O)CCOC(C#N)C1 c1(C(c2n(CCSC)nnn2)NCC(C)(C)CCC(C)O)ccc2c[nH]nc2c1 C(=O)(C(CC)C(=O)N(C(C)CCC)CCNC(C1OCCC1CC)=O)OC N1(C(C(=O)NCCOCC(=C)C)=O)CCC2CCC1C2 O=C(CCCCc1cccc(O)c1)NCCCCCNC(c1cocn1)=O N1(C(C(C)OCC#C)=O)Cc2ccccc2C1CNC(=O)C1=NOCC1 N1(C(C(C(C)(C)C)O)=O)C2CCCC1CC(NC(C1(CO)CCC1)=O)C2 C(=O)(C(CNC(C1C2CC3C(C2)C13)=O)CC(C)C)Nc1cccc(SC)c1 Cc1ccc2c(=NC3CC4CCC34)[nH]c(N3CC(CO)C4(CCC4)C3)nc2c1 C(=O)(C1=NN(C)C(=O)CC1)N1CC2(CC(NC(C3(COC)CC=CCC3)=O)C2)C1 CCCCCC(O)C(C)C(=O)NC1CCCCC1C(N1CCC(F)(F)C1)=O Cn1ncc2c1CN(C(=O)CNc1ncccn1)C2 c1(CC(=O)NCC(CNC(C(COCC)C)=O)F)c(OC)cccc1OCC C(=O)(CCCC(=O)NCC1CCC(NC(c2ncc(F)cc2C)=O)C1)OC N1(C(C(C=C)OC)=O)CCC(C)(C(=O)NC2CCOC(C)(CC)C2)CC1 c1(NC(C23CCCCC2C3(F)F)=O)ncc2c(n1)CCCCC2 N=c1[nH]c2ccccc2cc1C(=O)NCC1CC2CCCC2N1C(=O)CC(F)F c1(NC(C2N(C(c3ccc(OCC)nc3)=O)CC(O)C2)=O)cnc(C#N)c(Cl)c1 C1(C(=O)NC2(C(N(C)CC3CCCCO3)=O)CC2(C)C)C2CC(=O)CC12 C1(C(=O)NC2(CC#C)CCC2)(NC(C2SCCS2)=O)CCOCC1 C1(C(=O)OC(C)(C)C)(COC(CC(C)N(C)C2CC2)=O)CCCCO1.C(C1CC1)O C12(C(=O)NCCCN(C(CCCc3c(C)ccs3)=O)CCO)CC1COC21CCC1 N1(CC)CCC(N=c2ccnc(NCCC(=O)N(C)C(C)C)[nH]2)CC1C n1(CC(=O)NCCC2(O)CN(C(c3ccc(SC)s3)=O)C2)nc(Cl)ccc1=O c1(C(C(=O)NC(=O)CCn2cnnn2)=O)cc(CNCCCCOC)oc1C C=CCC(C)C(=O)NCCC1(CNC(c2cc(OC)no2)=O)CCC1 C1(C(NC(C(n2c(C)ccn2)C)=O)CC)C2CN(C(=O)CC3CCC(C)(C)C3)CC12 c1(C(C)OC)noc(CNC(=O)CC2(C)CCN2C(C2(CF)CC2)=O)n1 C=CCCCC(C(=O)N1CC2CCC(CC2)C1)NC(=O)C#CC(C)C N1(C(CNS(NC)(=O)=O)=O)CCC(CNC(=O)Cc2c(C)n[nH]c2C)C(CO)C1 N1(C(CSCCN(C)C)=O)C2CCC1C(CNC(c1nc(Cl)ccc1Cl)=O)C2 Cc1cnn(C)c1CNC(C1CC=CCN1C(=O)CCC(C)N1CCCC1)=O CN1CCC(C#N)(C(=O)NCC23CCCC2CCN3C(c2cn[nH]c2)=O)CC1 C1(CC(=O)N(C)CC2CC(F)CN2C(=O)CC2CC=CCC2)(OC)CCCCC1 C(=O)(C(C)(C)C(O)C(C)C)NCC1CCC(C(=O)NCc2nccc(OC)c2)C1 C1(C(N2CC(COC)(NC(C3CC3c3nc[nH]n3)=O)C2)=O)CCc2nc[nH]c2C1 C1(C2CC2)(C(=O)NCCCNC(c2ncoc2C(F)(F)F)=O)CCC1 c1(C(N(C2CCN(C(=O)C(C)(C)CF)C2)CC)=O)ccc2c(c1)N(C)CCO2 N1(C(c2cc(Cl)cc(Cl)c2)C)CCC2(CCOC(C)C2)C1 Cn1[nH]c(=NC(=O)NCC(F)C2CCC2)cc1Cl c1(COC)ccc(C(C)C(N2CCC(C(F)Cc3cn(C(C)C)nn3)CC2)=O)cc1 C1(C)(C(=O)NCC(C)C)CC(O)CN1C(c1ccccc1C#N)=O C1(n2cncn2)CCN(C(=NCc2cnc3n2CCC3)NC2CCOCC2)C1 O=C(CCCC1CCCCC1)NCCN(C(C1CCCCC1)=O)C1CC1 N1(CC(=O)NCCC(CNC(C2C(=C)C2)=O)O)C(=O)CN(C)C1=O CC(F)(F)C(F)C(=O)N1CCOC(C(=O)NCCCCC2CCCC2)CC1 C(c1cccnc1)=CCNC(CC1(NC(=O)C=Cc2cc[nH]n2)CC1)=O N1(C(COCCC#C)=O)CCCC(N2CCN(C(=O)C=C(C)C(C)(C)C)CC2)C1 c1(C(N2CC3C(C2)C3(F)F)C(=O)Nc2c(C)cccc2)ccnc(Cl)c1Cl C1(NC(c2c(C)nc(C(C)C)s2)=O)CCN(C(c2ccn(C)c2C)=O)C12CCC2 c1(C(N2CCC3CN(C(=O)C(F)Cl)CC23)=O)ccc2nc(Br)nn2c1 CC1CCC(C(=O)NCC2CCCN(C(c3n[nH]cc3[N+](=O)[O-])=O)CC2)CC1C C1(NCCCCCCC(=O)OC)CCC(C(C)C)N(C(=O)OCc2ccccc2)C1 N1(C(C(CCSC)NS(C)(=O)=O)=O)CC2(C1)CN1CC2NCC1=O.CCCCN c1(NC(C(CC2CCOCC2)NC(CN(CC(C)(C)C)C)=O)=O)cccc(F)c1 c1(N(c2cc[nH]n2)C)ccc(S(=O)(=O)NNC(=O)C2C3C4CCC(C4)C23)cc1 C12CCC(CC1)C(=O)NC2=O.c1(NC(C(C)S)=O)ncnn1-c1ccccc1 N1(C(c2n(CC)ccn2)=O)CC(F)(F)CC1C(N1CCN(C)CC1C(C)C)=O N1(C(C2(C(=O)OCC)CC2)=O)CCN(C)CC1CNC(C1OCCN(C)C1=O)=O c12ccccc1C(C)N2.c1(CSCC)cccc(-n2cc(C(O)CC)nn2)c1 N1(C(CCC(C)=O)=O)CCN(C(C)C(=O)NC2CCCCC2)CC1C C1(C(=O)NC(c2ccc(F)cn2)C)CC2(CC(NC(c3sccc3Cl)=O)C2)C1 Cc1ccncc1C(=O)NCC1CCN(C(C2C3CCC23c2ccccc2)=O)CC1 C1(NC(C2N(C(C)=O)CC(O)C2)=O)CCN(C(=O)CC2CCOCC2)C(C)C1 Cc1cc(C(N2CCN(C(C3CC3C3CC3)=O)C3CC23)=O)c(F)c(F)c1 N1(CCC)CCCC1C(=O)N(C)CCN(C)C(c1ncc[nH]1)=O C1(NC(c2cscn2)=O)CC(NC(c2ccc(F)nc2)=O)C12CCC2 C(N=c1cccc(S(=O)(=O)NCc2cnn(C(C)C)c2)[nH]1)c1snc(C)n1 C1(NC(c2cc(CC)sn2)=O)CC2CCC(C1)N2C(=O)Cc1cnc(C)nc1O N1(C(CC2(C=C)CC2)=O)CC(C2CCCN(C(c3nn(C(C)C)cc3Br)=O)C2)C1 C1(C(=O)NC(C(C(=O)OC)C)C)CC12CCN(C(C1CC3(CC3)CO1)=O)CC2 CCCC(C(=O)NC(C)CCNC(c1cnn[nH]1)=O)NC(N)=O C1(C(CNC(C2CCC(N(C)C)C2)=O)F)CCN(C(c2ccnc(O)c2)=O)CC1 c1(C(N(CCC)CCN(C)Cc2nc(=O)n(C)[nH]2)=O)cncc(C2CC2)c1 c1(C(N2CC(O)(CN(C(C(CC)F)=O)C)C2)=O)cc(Cl)c(O)c(Cl)c1 Nc1cc(Cl)nc(Cl)c1C(=O)NC1CC(NC(=O)Cc2ccccc2Cl)C1 C1(CC(C)NC(C2CCC(CCCCO)C2)=O)(CCNC(=O)COC)CCCC1 c1(C(=O)NCCC2(NC(C(C)OCCC#C)=O)CCC2)oc(CC(C)C)nc1C c1(C(=O)NCCOCCCCNC(C2CC3C=CC2C3)=O)ccc(Cl)cc1Cl O(P(=O)(COC(c1ccc(C(C)NC(=O)N(C)C)nc1)=O)OOC)CC c1(C(=O)NC2CC(NC(CC3CCCC(=O)N3)=O)C2)c[nH]c2cccc(F)c12 Nc1nccnc1C(=O)NCCNC(c1ccc(CN2CCCC2=O)cc1)=O c1(C(N2CC(CC(=O)NC)N(C(C3CC3F)=O)CC2)=O)cc(F)c(C#N)c(F)c1 CC1CC2(CCO1)CC2C(=O)NCC1CC(NC(=O)COC2(C)CCCC2)C1 n1(CC(=O)NC2CCN(C(c3c(C(C)O)cccc3)=O)C2)ncc2ccccc12 C=CCN=C(NCc1ccccc1COc1ccccc1)NCC(F)F CCC(CNC(=O)NCc1c(C)cc(C)nc1O)(CC)C(F)(F)F C1(NC(c2cc(SC)c(N)cc2)=O)CN(C(c2cocc2C)=O)CC2(CC2)C1 C1(C)(CCNC(C(c2c(C)noc2)C)=O)CCN(C(=O)C2=CCCO2)C1 C1(C)(C(=O)NCCN2C(C)CCC2)CCN(C(C2(C#N)CC(=O)C2)=O)C1 N1(C(C(F)=CC)=O)CCN2C(=O)C(NC(=O)Cc3ccc(Cl)nc3)CC2C1 c1(NC(CC)C(O)c2ccccc2)ncccc1S(=O)(=O)NCc1cccnc1 C(=O)(CCCCCSC)NC1(CC=C)CCN(C(C2CC(C)CC(=O)N2)=O)C1 c1(C(=O)NC23C(CN(C(CCCOCC)=O)C2)C3)cc(Cl)ccc1-n1ccnc1 n1(CC(N2CC(CNC(COC)=O)OCCC2)=O)cc(OC)c(=O)cc1C.CC=O Cc1ncc(CNC(=O)C(=O)NCCC2(CC3CC3)CC2)s1 N1(C(C(n2cc(C)nc2)(C)C)=O)CC(NC(=O)CC2CCC3CC23)C(C(F)F)C1 c1(C(=O)NCC2N(C(CN(c3cccc(O)c3)C)=O)CC2)ccc(N(C)C)nc1 C1(C(N2C(CNC(CCc3cnc(C)o3)=O)CC2)=O)CCCCCN1C c1(OCCC)ccccc1C(N1CCOC(C(=O)N(CC(C)OC)C(C)C)C1)=O CC(C)(C(=O)N1CC2CC(NC(C3CC34CCSCC4)=O)C1C2)C(N)=O C=CCCCC(C(=O)NC(C)(C)C(O)CO)NC(c1csc(C)c1C)=O c1(C(N(CCOCCCNC(CSCCC)=O)C)=O)cc(C#N)cc(C)n1 C1(C(N(C2CN(C(C3(Cc4ccc(F)cc4)CC3)=O)C2)C)=O)CCCCS1(=O)=O O=C(C1Cc2ccccc21)NCCC1CSCCN1C(c1cncc2c[nH]nc12)=O C1(CNC(CN(C(C(COC(C)=O)C)=O)C2CC2)=O)CCN(CCO)CC1 c1(C(C)NC(=O)CC2C=CCC2)ccnc(NC(=O)CNC(=O)N(C)C)c1 C(=O)(CS(=O)(=O)NC1CC1)NCCCOCCCNC(c1cc(C)ns1)=O C=CCC(C)(C)CC(=O)NCC1CC1NC(c1ccc(C)cc1C1CC1)=O C(C(F)(F)CC1CCCC1)(c1ccccc1)NC(C1CCCC1(F)F)=O C(=O)(C(C)CCc1cccc(F)c1)NCCCC(C)NC(c1ccc(C#N)[nH]1)=O N1(C(C(C)NC(c2ccco2)=O)=O)CC(CO)(NC(C2(O)CCOC2)=O)C1 CC1CCSCCN1C(C12CCC1CN(C(=O)C=CCO)C2)=O CC1CCC(C)(C(=O)NCC2CN(c3nnc(C(F)F)o3)CCO2)C1 CCC(C)(C)CCCC(=O)NC(CC(C)(C)C)C(=O)NCc1ccon1 c1(CC(=O)NCc2ccc(C(=O)O)o2)cc(O)ccc1C(=O)O Cc1cc(C(=O)NC2CCN(C(c3cncnc3C)=O)CC2CO)cc(N)c1 n1(CCNC(C2N(C(C(n3ncc(C)c3)C)=O)CC(O)C2)=O)cc([N+](=O)[O-])cn1 N1(C(C2C(OC)C2)=O)CCC2CN(C(C3CC(C)(C)C3)=O)CCC12 Cc1cc2c(cc1C)OC(C(=O)NCC(C)N(C(=O)CSCCC(F)(F)F)C)C2 C(CCC(C)(C)C(=O)N(Cc1cn(C(C)C)nn1)CC1CC(F)(F)CO1)OC N1(C(c2c(OCC)cccn2)=O)CCC2(CC1)CC(NC(=O)OC(C)(C)C)CO2 C1(CC)CC(CNC(=O)NCC2CCCN2c2ccccc2)CCO1.CC(F)F C(=O)(CC(C)C(C)(C)C)NC(CC)(C)CNC(c1c[nH]c(=N)o1)=O CC1(C(=O)NCCC2CCC(NC(c3cn(CCF)nn3)=O)C2)CNC(=O)C1 C(=O)(CCCN(C)C)N(C1CCN(C(=O)Cc2cnnn2C)C1)CC c1(C(N2CCCN(CCNC(CCS(C)=O)=O)CC2)=O)ccc2sncc2c1 C(CC(=O)N1CCC(COCCC(=O)NO)O1)OCC c1(C(=O)Nc2[nH]c(C)c(C(N3CCOC(C)C3)=O)c2C)cccc(Cl)c1C#N C#CCC(CC(=O)NCC=CC)NC(=O)C(=O)NOC Cc1cc(C(F)F)n(CC(N2CC(NC(=O)CN(C)C(C)C)CC2CO)=O)n1 N(C1CCCc2ccoc21)C(C1COCCC1NC(C1CCNC1=O)=O)=O C#Cc1ccc(OCC(=O)NCC(CNC(=O)C(O)C=C)CO)c(OC)c1 c1(C(N2CC(NC(=O)CCCCc3ccsc3)(CO)C2)=O)cc2c(Cl)cccc2[nH]1 CC1(C)CC(CC(=O)NCC2(CF)CCC2)CN1C(c1n[nH]c(=N)[nH]1)=O n1(C2C(C)C2)nc(C2CCCCC2)nc1-c1cn(C)nn1 C(CNC(=O)C(C)C)(CC(F)(F)F)NC(c1cc(-c2ccc(C)cc2)n(C)n1)=O N1(C(c2ccc(F)c(F)c2)C)CC2CN(C(C3CCCCO3)=O)CC2C1 C1(C(=O)OCC(=O)NC(c2ccc(F)cc2)CCn2c(C)ncc2)CC2(COC2)C1 C1(NC(CCC2CCN(C(CC)=O)C2)=O)CC(C)OC1=O c1(NC(N2C(C(=O)NS(=O)(=O)CC)CC2)=O)ccc2c(O)nnc(O)c2c1 CCCC(CCCNC(=O)C(C)(C)CO)NC(=O)CCNC(=O)C=CCl Cc1cn2c(=O)c(C(=O)NC3CC4CCC(C3)N4C(=O)COC(C)C)cnc2s1 N1(C(C(C)N2CCCC2)=O)CC2C(C(=O)NCCc3ccn(C)n3)C2C1 c1(C(N(CCNC(c2c(CC=C)cccc2)=O)CCOC)=O)cnc2n1CCS2 c1(C(=O)NC2C(F)CCN(C(C(CC)O)=O)C2)cnc2c(c1)CCCC2 c1(C(=O)NCCC2CN(C(COCCCC)=O)CC2C)cc(F)c(Cl)c(N)c1Cl C1(NC(CC2CC(SC)C2)=O)CCC2(CC1)CN(c1cc(C)ncn1)C2 O=C(CCCCc1ccccc1)N1CC2CC2(CNC(C2CC(F)C2)=O)C1 N1(C(C(=O)NC(c2cccc(N3CCCC3=O)c2)C)=O)CC2(C)CCCCN2C1 c1(C(=O)NC(CCC)CCCNC(C2CC(F)(CO)C2)=O)cnc2cccnn12 C=C1CCN(C(=O)CC2CC(OC)C2)C(C(=O)N(CCCO)C2CC2)C1 C(C1CN(C(=O)CC2CCCCN2C)CC1C(=O)NCCn1ccnn1)=CC c1(C(=O)Nc2cccc(NC(c3c(CC)non3)=O)c2)cc(C)c(F)cc1F S(=O)(=O)(c1cc(NC(C)=O)c(C(=O)O)cc1Br)NCC#CCOC C=C(C)CC(C(=O)N1CC(NC(c2ccnc(C3CCC3)c2)=O)C1)OC CC(C(=O)NC1CCC(CNC(c2ccccc2OCC#N)=O)CC1)C(C)(F)F C12(NC(c3cccc(=O)o3)=O)CCC(NC(C3CC3Cl)=O)(CC1)C2 C1(NC(Cn2nnc(C)n2)=O)CN(C(C2(C)CC2)=O)CC1CC(C)(C)C C1(CC=C)(NC(=O)C(C)n2cncn2)CCN(C(=O)CC=CCC)CC1 c1(OC)ccccc1C(C)(C)C(=O)N(C(CO)C(C)C)C C(=O)(C1=CCc2ccccc21)NCC(C)(C)CNC(c1scnc1C(F)(F)F)=O N1(C(C(C2CN(C(C(C)C3CCC3)=O)C2)O)=O)C2CCC1CC2 N1(C(c2nc(C)sc2)=O)CCC(NC(=O)C(C)SC(C)C)CC1 C(=O)(CCCCN(C)C)NC1CCC(CC(N2CCC(=CCC)C2)=O)C1 N1(C(c2nc(CC(C)C)sc2)=O)CC(CNC(=O)C=Cc2ccc[nH]2)CC1C n1(CCOC)nccc1C(=O)NCC(C)NC(c1cc(-c2ccco2)c[nH]1)=O C1(C(=O)Nc2c(C(N(CCN(C)C)CC)=O)scc2)CC2C=CC1C2 C(=O)(C(C)C(O)C(C)CC)NCC(CC)N(C)C(c1cnc2[nH]nnc2c1)=O c1(C(=O)NCC(CO)NC(C(C)OCCC#C)=O)cn(C)nc1COC c1(C(=O)NCCN(CCCN(C)C)C(C2(CC=C)CCC2)=O)cccc2c(C)[nH]nc12 Cc1noc(C(C)C)c1C(N1CCC(O)(CNC(=O)CCOCC2CC2)C1)=O C1(CNC(C(=O)NC2CCC(C(=O)OC)CC2)=O)CCCN2CCCCC12 C1(NC(C23OCC(C)(C2)C3)=O)CCSC12CN(C(=O)CC1CCCC1(F)F)C2 C(=O)(C(C)(C)CCC#N)NC1CCC(C)CN1C(=O)CS(C)(=O)=O C=Cn1nccc1C(=O)NC1CCN(C(c2cccc(C(F)F)c2)=O)C1C C1(CN(CC(C)(C)Cn2cc(CN3CCCC3C(=O)O)nn2)CC)CCCC1O C1(C(N(C(C(C)SC)C)C)=O)CN(C(c2cn(C3CC3)cn2)=O)C(C)(C)C1 N1(S(=O)(=O)c2ccc(O)cc2)CCC2(CCCN(Cc3cc(Cl)cc(I)c3)C2)C1 c1(C(N(CCCNC(C2C(F)(F)C23CCC3)=O)CC)=O)cc2c(s1)CCCC2 Nc1ccc(NC(c2n[nH]cc2-c2ccccc2OC(F)(F)F)=O)cc1 C1(CC)CCCCC1C(N1CCN(C(c2nc(C3CC3)oc2C)=O)CC1)=O c1(C(N2CC(C=C)(CC(=O)NCC(C)Cn3ccnc3)C2)=O)c[nH]c(C)cc1=O C1(NC(C2CC(F)C2)=O)CN(C(=O)Cc2ccc(CO)cc2)Cc2nccn2C1 CC1CCC(CNC(c2cc(O)ncn2)=O)CN1C(=O)C1=CCCCO1 Brc1cnccc1-c1nc(CCc2ccncc2)nn1CC(F)(F)F CC1CCN(C(=O)CC2CC(=O)NC(=O)C2)CC1CNC(=O)C=C1CCN(C)C1 c1(C(=O)NC2CC2CNC(C2(C(F)(F)F)CC2)=O)cccc(=O)o1 C1(C)(CNC(C(CC)C(C)O)=O)CN(C(c2ccsc2SC)=O)C(C)(C)C1 Cc1ccc(CC=O)c(F)c1.N12CCN(CC1)C(=O)C(=Cc1ccccc1)N2 C1(CNC(c2nc(C)[nH]n2)=O)(NC(=O)Cc2csc(NC=O)n2)CCCCC1C C=CC1(C(=O)NC(CNC(c2ccc(C#N)cc2)=O)C2CC2)CCOCC1 C(C)(C)(CN=C(NCC1CCCCC1(F)F)NC1CCS(=O)(=O)C1)SC Cc1cccc2oc(C(N3CC(N(C(=O)CCCS(C)(=O)=O)C)C(F)C3)=O)cc12 N1(C(c2c(C)c[nH]n2)=O)CC2CCCC(C1)N2C(=O)CNc1cccnc1 n1(CC)ccnc1C(N1CCC(C(C)NC(=O)C(CN(C)C)N(C)C)C1)=O N1(C(C(C)C(C)O)=O)CC(N(C)C(C2CC3(CCC3)C2)=O)C2(CC2)C1 C=CC(COC)N=c1ccnc(NCC2CCCN(c3ccc(C)cc3)C2)[nH]1 N1(C(CCOCCOC)=O)CC(C)(C)OCC1CNC(=O)CSC(F)(F)F c1(OC)ccc(C(C)C(=O)N(CCCNC(=O)C(CO)c2ccccc2)C)cc1 Cc1cnc(C(=O)NCC(C(N2CCCCC23CC3)=O)N(C)C)cc1C c1(C(N2C(C)(C)C(CNC(=O)CC(=O)N(C)C)CC2)=O)ccc2[nH]c(=N)[nH]c2c1 c1(C(=O)NC2CN(C(c3[nH]cc(C(C)=O)c3)=O)C2)nccc(C)c1O c1(CN2C(C(=O)NC(C(=O)NC)C)CC(F)C2)cnc2ccc(Br)cn12 C1(C#CC(=O)N2C3CCC2CN(C(=O)CC2CCN(C(C)C)CC2)C3)(CC)COC1 N1(C(C23CC(C)C2C3)=O)CC(N(C)C(C2(C)COC2)=O)C(O)C1 Cc1ccc(F)cc1-n1nc(-c2ccc(F)cc2)nc1C1CC(C(F)(F)F)C1 c1(C(N2CC(NC(C3OCCN(C(C)=O)C3)=O)C2)=O)c(I)ccnc1F N1(C(c2cnn3c2CCC3)C(=O)NCCOC)CCOC2CCOCC12 N1(C(CCCC)=O)CC(NC(=O)CC(O)c2ccccc2)C(C(F)F)C1 N1(C(C(C)C(F)(F)F)=O)CCOC2CN(C(=O)NCc3ccccn3)CC12 N1(C(c2n(C(C)C)ccn2)=O)CCN(C(=O)C(C)SC(C)C)CC(C)(C)C1 CCC(C(=O)OC)C(=O)N1CC(C(=O)NCCC(C)(C)C)CCC1C N1(C(c2ccc(COCC)o2)=O)CC2CC2(NC(=O)NCC(CC=C)CCO)C1 C1(NC(C(CC)=CC)=O)CC(C(=O)NCC2CCSC2)C12CCC2 C(C1CCCc2ccccc21)N(C(C)C)Cc1cccc(Cl)c1 c1(COC)ncc2c(n1)CCC(C(=O)N(C)CC1CNCCC1(C)C)C2 c1(-n2cc(OC(c3ccc(Br)cc3F)CO)nn2)cccc2c(Br)cccc12 C1(NC(C2CC(OC)(OC)C2)=O)CCCCCC1NC(c1[nH]c(O)nc1C)=O C1(CNC(C2(OC)CCCOC2)=O)CC(C)CN(C(=O)CC2COCCOC2)C1 N1(CCNC(c2c(CC)ncs2)=O)CCCN(C(=O)Cc2cncc(O)c2)CC1 CCCS(=O)(=O)CC(=O)NC1CN(C(=O)C(c2cnccn2)C)CCC1CO Cc1ccc2c(c1)CCC(C(=O)NC1CC3(C1)CC3NC(=O)C(F)=CC1CC1)O2 NC1CN(CCC(=O)Nc2ccccc2CO)CC1O N1(C(c2ccnc(CC(C)C)n2)=O)CCCC(C)C1CCNC(c1cnns1)=O N1(C(CCC(C)=O)=O)CC2CC(NC(=O)CCC3CCC(C(F)(F)F)O3)CC2C1 C1(NC(C(n2cnc(C#N)n2)C)=O)CC12CCN(C(c1c[nH]nc1C1CC1)=O)C2 CC(C)CCC(=O)C(=O)NC1CC2CC(NC(=O)CSc3nncs3)C2C1 C(=O)(C(C)(C)C(F)F)N(C(=O)CNCC(C)(CC)NC(CNS(CCCOC)(=O)=O)=O)CC C(=O)(C(C)C(C)(F)F)NC(CCCC)CNC(=O)CCOc1ccccc1Cl C1(C(=O)NCC23C(CN(C(CCc4nc(=N)[nH][nH]4)=O)C2)C3)COCC2(CCC2)O1 C1(CC)CCC(O)(C(N2CC(O)(CCNC(c3conc3C(C)(C)C)=O)C2)=O)C1 N1(C(c2c(COC)scc2)=O)CC(CNC(c2n[nH]c(C)c2C)=O)C(F)(F)C1 C1(NC(C(C)OCC=C)=O)CCN(C(=O)C=C2CCCC2)C1C1CC1 Cc1oc(C(=O)NCCC2(CNC(=O)Cc3ccccc3F)CC2)cc1Br N1(C(CN(C(c2cn(C3CCCCC3)nn2)=O)CCO)=O)CCC2CCCC12 CC(C)CC(C(=O)NCC1(C)CC1)ONC(=O)C1CCN1C(C)(C)C c1(C(N2CCCC(CN(C(C(C)OCCC#C)=O)C)C2)=O)cc(C)cnc1N c1(C(N2CC(CNC(c3ncoc3C(F)F)=O)C2)=O)cnc(O)nc1O C#CCCCC(C)C(=O)NC1(CC(=O)N(C2CCC(C)C2)C)CC1 N1(C(c2cnn(CC)n2)=O)CC(N(C)C(c2ccnnc2)=O)C2(CC2)C1 c1(CC)cccc(C(=O)NC(C)CC(C)NC(=O)CCc2nnc(C)n2C)c1N N1(C(C(=O)O)C)CCN(C(=O)NC2CC2SC(C)(C)C)C(C)C1=O.CC(C)C C1(C)(CNC(Cc2c(C)cccc2)=O)CCN(C(C2CCCC(C)CC2)=O)CC1 N#Cc1cc(Br)c[nH]c1=NCCCCNC(=O)CCCC1CCCC1 N1(C(CC(C)C)=O)CC(CNC(=O)CCCSC)C2(CC2)C1 c1(C(=O)NC2CCN(C(C3CCCC3C(F)F)=O)CC2F)ccc([N+](=O)[O-])cn1 c1(NC(C(=O)CCC2CCCN2)=O)ccccc1OC(F)F.C1(C)CC1 C(=O)(C(C)(C)CCNC(=O)CCCN)C(C=C(C)C(C)C)=O.C1(O)CCOCC1 c1(C(=O)NC2CC(NC(C=CCC)=O)C2)c(F)cccc1Br N1(C(C(=O)Nc2sc(CCC)c(C)n2)=O)CCC2(CCSC2)C1 C=CCC(C)(CC)C(=O)N1CCCC(CCNC(c2cnc(SC)n2C)=O)C1 N1(C(CC(=O)NCC)=O)CCC(C)C(NC(C2C(C)C2(F)F)=O)C1 N1(C(c2n(C)ccn2)=O)CCCC2(CCN(C(c3cnc4c(c3)CCC4)=O)C2)C1 CCC(CC)C(C(=O)NC1(CNC(=O)C(C)Oc2ccccc2F)CCC1)OC C1(F)(CNC(CC(=O)NCC)=O)CCC(CNC(=O)CC(C)c2ccco2)C1 C1(NC(=O)CCC2CC(F)(F)C2)C2CCC1N(C(c1cnn(C3CC3)c1Cl)=O)C2 C(C(C)CN=C(NCc1cnc(C(=O)OC)s1)NCC(C)(C)C)OCC N1(C(C2(C)CCCC2)=O)CCn2ncc(-c3cccc(C4(C)OCCO4)c3)c2C1 C1(C(=O)NC2C(NC(=O)CCc3ncc[nH]3)CC2)Cc2cccc(F)c2O1 N1(C(CCC)=O)CC(C(=O)NCCOCC(C)(C)O)C(CC)C1 CCCC(CCC)CC(=O)NC1(CNC(C23CCCN(CCC2)C3)=O)CCC1 C(=O)(N=c1c(F)c[nH]cc1Cl)C1(c2onc(-c3cccc(S(N)(=O)=O)c3)n2)CC1 c1(NC(C2C(C)CN(C(=O)C(=O)NCC(F)F)C2)=O)ncnc2ccc(Cl)cc12 C1(C(F)(F)C(=O)NC(C)C(C)NC(c2cc(C)[nH]n2)=O)(OC)CCCC1 C12(NC(C3C(NC(CCCOC(C)=O)=O)COC3)=O)CCC(O)(CC1)CC2 c1(C(N2CCCC(NC(CC3(C=C)CC3)=O)C2)=O)cc(C(F)(F)F)cc(C)n1 C1(C(=O)OC)CCC(c2nc(C(N3CCOCC3)=O)c(C)o2)CC1.C1C(=O)N1C C1(NC(c2cnc(C)s2)=O)CCC12CN(C(=O)COCC(c1ccccc1)C)C2 n1(CC(=O)NCC2CC(NC(C(c3cnn(C)c3)C)=O)C2)cc(CC2CC2)nn1 C(=O)(CC(CC(C)C)NC(=O)CCNC(C)=O)OC(C)=O.C1(=O)C(C)O1 C1(NC(=O)NCC2C=CCCC2)CCCN1c1ncccn1 C1(CC(N)=O)CC(NC2NC(=O)CC23CCC3)C12CCC2 C1(C(=O)OC)CN(Cc2cc(Cl)cc(OC)c2OC)CC(F)(F)C1 C(CC(CC)C(=O)NC1(CCCNC(=O)CCCn2c(O)nnc2O)CC1)=CC c1(SC)ncccc1C(=O)N(c1nnc(Br)s1)C1CC1.C12CC(C1)NC2=O c1(C(=O)NCC(COC)NC(c2cccc(CO)c2)=O)cc2c(=O)[nH]ccn2n1 c1(C(=O)NC(CCNC(C2(Cc3ccc(OC)nc3)CC2)=O)C)c[nH]c(=N)cc1C c1(SCC(=O)NC2CC(n3cccn3)C2)ccc(-c2noc(C3CCCO3)n2)cc1 CCCCCS(=O)(=O)CC(=O)N1CC2CN(C(=O)CC3OCCC3(C)C)CCC12 c1(OCC)ccc(C(=O)Nc2cc(C)oc2C)cc1.C12CC3(C1)CC3NC(=O)N2 c1(C(=O)NC2C(NC(C3C4CCC(=O)C43)=O)COC2)ccc(F)c(Br)c1 C#CC1CCC(NC(C2CC(N(C(c3cn(C4CC4)cn3)=O)C3CC3)C2)=O)C1 N1(C(C(COC)NC(C)=O)=O)CCC(C(C)C(=O)N2CC(COC)C2)CC1 C(=O)(C(C)CC(C)(F)F)NC1C(F)CCN(C(C=Cc2ncn(CC)c2)=O)C1 C1(COC)CC2CCC(C1)N2C12C(C1)C(=O)NC2.CCC(C)=CCSC c1(C(N2CCN(C3CCOCC3)CC2)C(=O)N(C)C2CC2)ccc(C)c(I)c1 c1(C(C)C(=O)NCCCC(N2CCCCC2CO)=O)ccc(F)c(F)c1 C1(NCCc2c(C)nn[nH]2)CN(c2ccncc2)CC1C(=O)O C1(C)(CNC(Cc2c(C)nc(S)s2)=O)CN(C(c2cc(Cl)ccn2)=O)CCO1 C1(CC(=O)NCC(CNC(COCCOC)=O)CO)COCC1(C)C CCCCC(O)C(C)C(=O)NCCN(C)C(c1ccc(O)c(C)c1)=O N1(C(C(C)OCCCC)=O)CC(OC)CC1CNC(C1(CCCC)CC1)=O C1(CC#C)(NC(C2(CC3CC3)CCCO2)=O)CCCN(C(=O)C2=COCCC2)C1 C(=O)(C(CC(C)C)C(C)C)N1C(CNC(c2ccc(C)cc2C2CC2)=O)C=CC1 C1(NC(c2ccco2)=O)CCN(C(=O)CC2CCS(=O)(=O)C2)C12CCCC2 C12CCC(C3CC3)N1C2=O.c1(C(N2CC(CCCCNC(=O)O)C2)=O)cnns1 Cc1cc(C(N2CCN(C(=O)Cc3cncn3C)CC2CC2CC2)=O)ccc1Cl C(C(C)(C)C(=O)NCC(Cc1ccccc1F)N(C(=O)Cn1nccn1)C)OC c1(CNC(C(C2CC2)NC(C(C)C)=O)=O)nccn1CC(C)C C1(CNC(N(C)Cc2ccc(Cl)cc2)=O)CC2CC(=O)C1O2 C12(C(=O)NCCN(CC(C)O)C(c3cccc(C(F)(F)F)n3)=O)CC3CC1C2C3 c1(OC)cc(C(=O)NC2CC2CNC(c2ncoc2C2CC2)=O)nn1C c1(C(=O)NCc2c(C(C)C)nn(C)c2)c2ccccc2nn1C C1(C2CC2)(NC(c2cccc(OC3CC3)c2)=O)CCN(C(=O)CC2CCCCC2)C1 N1(C(C(C)Sc2nnc(C3CNC(=O)C3)o2)=O)CCCCC1C(N)=O C1CN=C(N(C)CC2CCS(=O)(=O)C2)NCC(=O)N1CC.C1(C)CC1.NC CC(CC(=O)NC1(CCNC(=O)Cc2ncc(Cl)s2)CCCC1)P(C)(C)=O c1(OC)ccccc1C=CC(=O)NCCCCN(C(=O)C(C1CCOCC1)F)C C1(C)(C(=O)NC(C#C)C)CN(C(=O)C(C)COC)CC1C C(C(C)(C)CCNC(=O)CCOCCN(C)C)OC c1(CC(=O)N(CCCOCCC2(Br)CC2)C)cc2ccccc2s1 C12(NC(Cc3ccc(CC)cc3)=O)CCC(CC1)N(C(=O)C(C)(C)OC1CC1)C2 c1(COC)ccc(C)c(NC(C2CC(=O)N(Cc3ccncc3)C2)=O)c1 c1(NC(C(=O)N(CC(=C)I)CC2CCC2)=O)ccc(F)c(C(F)F)c1 O=C(CCCCC(F)F)NC1CCN(C(=O)CCC2CCCCC2)CC1F N1(C(C2CCCN(C(c3c(OC)cc(F)cc3)=O)C2)=O)CCC2(CCCC2)CC1 CC1CN(C(=O)CN2CC=CC2)CC(C)C1NC(C1(N(C)C)CCC1)=O C1(C(N2C(C)(CC(=O)NCCCCCN(C)C)CC2)=O)COCC1(C)C c1(C(N2CC(NC(C=CCOC)=O)CC2(C)C)=O)ccc(S(C)(=O)=O)o1 C(COc1ccccc1)(C(=O)NC1(CF)CN(C(=O)Cn2cc(Cl)cn2)C1)OC CC(C)(CCl)C(=O)NC1CCC(C(=O)NCC2(C#N)CCC2)CC1 C(CC(C)(C)CC(=O)N1CC(CC(C)NC(C2Cc3ccccc3O2)=O)C1)OC Cc1nc(N)cnc1C(=O)NC1COCC1NC(=O)CCn1ccccc1=O c1(C(=O)NC2(COC)CN(C(C3(SC)CCC3)=O)C2)cc([N+](=O)[O-])ccc1O c1(C(=O)NC2N(C(c3c(C#C)c[nH]n3)=O)CC2C)occ2c1CCCC2 N1(C(C(c2cccnc2)C)=O)CCCCC1C(=O)NOC(C)(C)C CCCCC(C)(F)C(=O)NCCC1(OC)CCN(c2nnc(O)s2)C1 C(=O)(CCCCCN(C)C)N(CCCNC(=O)C(C)(C)C1CCOC1)C(C)C c1(C(=O)NC(C(C)(C)O)C(=O)N2CCC(C)(O)C2)ccc2occc2c1 c1(N2CCCC(NC3(C)CC=CC3)C2)ncccc1S(=O)(=O)N1CCCC1 N1(C(C2ON=C(C)C2)=O)CCCC1(C)CNC(C1CCCC(C)O1)=O N#Cc1ccc(S(=O)(=O)N2C3CN(Cc4cc(Br)cs4)CC23)c(Cl)c1 N1(C(C(C)C)=O)CC(O)CC1CNCc1c[nH]ccc1=N N1(C(=O)C(O)Cc2cnco2)CC2(C1)CN(C(c1cnc(S)nc1)=O)C2 C1(CCC)CN(C(C2CCCCN2C(C)=O)=O)CCN1C(=O)CCC=C(C)C C1(CNC(c2ncc(C(F)(F)F)s2)=O)CC(F)(F)CN1C(C1CCCSC1)=O C(=O)(CC1c2ccccc2C(=O)N1C)N1CC2CN(C(C(CC)SC)=O)C2C1 c1(OC)ccc2nccc(C(=O)NC(C)CCNC(=O)C(C)(C)CF)c2c1 c1(C(N2CC(F)(F)C2)=O)cc2c(C(=O)O)cccc2[nH]1 c1(NCC(CC)O)ncc(C)cc1S(=O)(=O)N1CCOC2(CCN(C)C2)C1 O=C1CCC(NC(=O)CCC2CCCN2C(c2cccc(Cl)c2Br)=O)C(=O)N1 c1(CC(=O)NCC2C3N(C(CCS(N)(=O)=O)=O)C(CC3)C2)cc(F)c(F)c(F)c1 C(C(=O)N=c1ccn(C2CCC2)[nH]1)C1(C)CN(C(=O)C=C2CCOCC2)C1 C12(CC(=O)NCCCN(C)C(C3CC(F)(CF)C3)=O)CC3CC(CC(C3)C1)C2 c1(CNC2CCCC(CCN)C2)ccc([N+](=O)[O-])cc1Cl Cc1ncsc1C=CC(=O)NC1(CNC(C2CC2Br)=O)CCC1 N1(C(CC2(N(C(C(C3CC3)OC)=O)C)CCC2)=O)CCC(C(N)=O)C1 C(CCCCCNC(C1C2CCC1(c1ccncc1)C2)=O)NC(C=C(CSC)C)=O c1(C(=O)NCC2CN(C(c3cnc(Br)s3)=O)C2)cc2c(nn1)CCC2 C(=O)(C(C)CCCC(C)=O)N1CCC(C(N(CC(=O)OC)C)=O)C1(C)C C1(CC=C)(NC(c2ncccc2F)=O)CCN(C(=O)CCC(C)OC)CC1 Cc1nc(C(=O)NCC(O)C(=O)NCCC(=O)N(C)C2CC2)c(C)o1 Cc1cn2nc(N3CCC(F)(F)C(CNC(c4cc(Cl)ccc4Cl)=O)C3)sc2n1 C1(CC(=O)N(CC(C)(C)NC(=O)COCP(C)(C)=O)C(C)C)CCCC(O)C1 c1(NCc2cn(-c3ccc(C)cc3)nc2)coc2cc(Cl)ccc12 Cc1cnn(CC(=O)NC2CCC2NC(c2cc(C)co2)=O)c(=O)c1 c1(C(C)=O)ccc(COC(c2ccnn2C2CC2)=O)c(F)c1 C(C(C(C)C(C)C)NC(c1cnc(OCC)s1)=O)NC(C(CC)CC)=O N1(C(C(CC)(C)O)=O)CCCC2(CCCN(C(C3CC4CCC3O4)=O)C2)C1 c1(CN2CC(CCCCNC(c3ccnc(Br)c3)=O)C2)ccc2cc(F)ccc2n1 N1(C(C=NS(CC)(=O)=O)=O)CCN(C(C2CN(C(C)C)CCO2)=O)CC1C C(C(O)CC(=O)N1CC(CCNC(C2CCCN2C(=O)C(C)C)=O)C1)SC CC1OC2(C(=O)NCC(C)(C)NC(=O)C(c3ccc(C#N)cc3)C)CCC1CC2 c1(NC(C2CCCCN2C(c2ccc(Cl)o2)=O)=O)nc(Cl)cnc1Br C1(C(N(C(CNC(C2C(=C)CC2)=O)C)C)=O)CC(=O)NC(CC(C)C)C1 N1(C(Cn2cc(C(C(=O)C(C)C(C)(C)C)C)nn2)=O)CCC(C2CC2)C1CO N1(C(CCCOCC=C)=O)CCC(NC(=O)Cn2c(C)csc2=O)C(F)(F)CC1 Cc1cnc(N2Cc3ccc(Cl)cc3C2)c(S(=O)(=O)N2C3C=CCC2CC3)c1 N1(C(=O)CCN2CCOCC2=O)CCC2CCCN(C(=O)Cc3cncs3)C2C1 c1(C(=O)NCC(C2CC2)NC(C(CC)F)=O)ccnc(O)c1 c1(C(=O)NCC2N(C(CS(CC)=O)=O)CCC(C(F)(F)F)C2)nnc(O)nc1O c1(OCC(=O)NCCNC(C(C)c2ccsc2)=O)cc(C(F)(F)F)ccc1O c1(C(N2C(c3onc(NC(C)=O)n3)CCC2)=O)cnnc2ccccc12 c1(Cc2cn(C3CCN(C(=O)CCCOC4CCOCC4)C3)nn2)ccc(Cl)cc1 N1(C(c2ccc(C)c(Br)n2)C(=O)NC(C)(C)C)CCc2ccc(Cl)c(F)c2C1 Cc1ccc2c(c1)CC(C)N(CC(=O)NCCc1ccc(Cl)cc1Cl)C2 C1(C(N(CCNC(C2CCSC2)=O)Cc2ccccc2)=O)CCCC2C1C2(F)F C1(OCC)CN(C(c2cncnc2C)=O)CC1CNC(=O)C(CSC)OC N1(C(C2(CC=C)CC2)=O)C2CCCC1CN(C(c1ccn(C(C)C)n1)=O)C2 c1(OC(C(=O)NC2(CCO)CN(C(C(C)OC)=O)C2)C)cccc(COC(C)C)c1 C1(S(N)(=O)=O)(C(N(CCN(C(=O)C(c2cccc(Cl)c2)C)CC)CC)=O)CC1 C1(CCCNC(C(C)OCCCC)=O)CCCCN1C(c1occc1C)=O CC(C)(C)CCC(F)C(=O)N1CCC(NC(=O)CC2CCCC2)C(O)C1 C1(CC#C)(C(=O)NC(CO)C(=O)OC)CCCC1.C1(CC)CN1 CC(C)(CNC(=O)NCCC1CCCOC1O)C(=O)OCC(F)F C1(NC(c2c(C)ccs2)=O)CCC(C)(CNC(=O)CC2CCOC2)CC1 c1(OCC)ccnc2sc(C(N3CCC(C)(NC(=O)C(F)CC)C3)=O)cc12 C1(OC)CN(C(=O)Cc2oncc2C)CC1NC(c1cnc(C(=O)N(C)C)s1)=O Cc1cc(Br)ccc1NC(c1ccc(NC(=O)N(CC(O)CN)C)cc1)=O CCCN=C(NCc1cc(Cl)cn1C)N(C)CCSC C(C)(CCCF)(c1nnnn1CC(F)F)NCC(=O)N(C(C)(C)C)Cc1cccs1 C(=O)(C1CCC(NCC(C2CCCCC2)C(F)F)c2ccccc21)OC C1(C2CCCN(C(C3CC3C3CC3)=O)C2)(NC(CSCCN(C)C)=O)CC1 C1(C(C(=O)NCC2CC(OCC)C2)(C)C)CCCN(C(C2CCCCN2C)=O)C1 C1(C(N2CC(CC=C)(NC(=O)CC(C)(C)C3CC3)C2)=O)Cc2c(F)cccc2O1 c1(N2CCN(C(C(=O)NCc3nc(CCC)[nH]n3)=O)CC2)cc(C)cc(C)c1 N1(C(CN(C(CC2CC(=C)C2)=O)CC(C)C)=O)Cc2nncn2C(C)C1 C1(C(=O)NCCN(C(c2c(C)onc2Br)=O)C)CC2(C1)OCCO2 C=CCCCCCNC(=O)NC.C12CCCC(C1)NC(=S)NC2 CP(C)(=O)C(O)C(=O)NCC1CCCN(C(C23CCC(CC2)C3)=O)C1 C1(OCC)CCCN(C(C2(C)CCN(C(c3cc(OC)ns3)=O)C2)=O)C1 N1(C(c2cccc(OC)c2C)=O)CC2OCC(NC(=O)C3=CCS(=O)(=O)C3)C2C1 C(CCCCC(=O)NC(c1nocc1C(=O)NC(C)CC(C)(C)CO)C)=CC c1(C(=O)NCC2CN(C(C(COC)COC)=O)CC2C)n[nH]cc1[N+](=O)[O-] CC(CCNC(C1CCCCC1CNC(=O)CCc1cccnc1)=O)C(F)F C(=O)(C(C)CCCC(C)C)NCCC1(C)CCN(C(CCCN(C(C)=O)C)=O)C1 C(CC(=O)NC1CC2C=CC1C2)(C(F)F)NC(c1c(COC)noc1)=O c1(C(N2CCC(N(C(CNC(=O)NC)=O)C)C2)=O)cc2c(F)c(F)ccc2s1 CN1CCN(C(C2(C)CCC(=O)N2)=O)CC1CNC(C1CCCC(C)(C)C1)=O N1(S(=O)(=O)Cc2csc(Cl)c2)CC2CC1CN2CC(F)(F)F C(CC(F)F)(C(=O)NCC(C)C(=O)NC)N(C(C(C=C)C)=O)C c1(N2CC(NC(CC(C(C)C)O)=O)C(C)C2)ncnn2c(Br)ccc12 c1(NC(C2CC(NC(C=C(C)C(C)C)=O)C2)=O)nc(C)nc2sc3c(c12)CCC3 Cc1ccc(C(C)C(=O)NCCC2CCN(C(=O)CCOC3CCC3)C2)s1 c1(CC)c(C(N2CCCC(NC(=O)C(=O)C(C)(C)C)C2)=O)[nH]c(C)c1C(C)=O C(=O)(CCCC(C)C)NC1CCC(CNC(c2n(CC)cc(Cl)c2)=O)CC1 C(CN=c1[nH]c(CC(=O)N(C)C)cs1)C1(C)CC2CCC1C2.C1CO1 N1(C(CC(CCC)(C)C)=O)CCCC2(C1)CN(C(=O)C(CC)N(C)C)C2 C12(CNC(CN(CC)CC)=O)CCC(CC1NC(C1SCCS1)=O)C2 C1(C)(C(=O)NCC2C(CCC)C2)CCN(C(c2ccc(Cn3ccnn3)o2)=O)CC1 Cc1cccc(O)c1NC(c1ccccc1NC(C1CCC1(C)C)=O)=O CCCCCC(O)CC(=O)N(C)CC=CC(=O)NCCCF Cc1ccc2c(=NCc3nc(C(C)C)cs3)[nH]c(N(CC(F)(F)Br)C)nc2c1 N1(C(Cc2cc(COC)on2)=O)CCOC(CNC(=O)C(C)N2CC(C)C2)C1 CCCC(C)CC(=O)NCC1(NC(c2cnoc2C2CCC2)=O)CCOCC1 N1(C(C(C)NC=O)=O)CCC(C2CC2)(NC(c2ccc(C(C)(C)C)s2)=O)C1 C(C(C)C(=O)NC1CN(C(=O)CSCc2cccnc2)C1)SC S(=O)(=O)(c1ccc(NCC2=NOC3(CCC3)C2)cc1Cl)NCC1CCC(C)C1 N1(C(c2c(NCC)scn2)=O)CCC(F)(F)C(CNC(=O)C(CC)C(C)C)C1 C1(C(N2CCN(C(C3(C)COC(=O)N3)=O)CC2)=O)CC2(COC(=O)N2)C1 N1(Cc2n(C)cnc2)CC=C(CNC(c2cc(F)ccc2Br)=O)CC1 CC1(CO)CCN(C(C2CN(Cc3cnc(Cl)c(C(F)(F)F)c3)CCO2)=O)CC1O c1(NCc2ccc(CC(C)C)s2)cc(I)c(Cl)cn1 C(=O)(C(C)(C)C(=O)N1CCC(CC)C1CC1(C#CC(=O)NC)CC1)NC1CC1 C1(C(=O)NC(c2c[nH]ccc2=O)C)(CNC(C(C)OCC#C)=O)CCOCC1 N1(C(C=CC(CC)=CC)=O)CCC(F)(CNC(C2SCCC2C)=O)CC1 C1(CC(=O)NCc2c(C(=O)NC(C(C)SC)C)c[nH]n2)C=NN(C)C1=O n1(CCOCCOC)cc(C2(O)CN(C(c3cn(C4CC4)cn3)=O)C2)nn1 N1(C(c2cc(C)ncn2)=O)CCOC2CCN(C(c3ccc[n+]([O-])c3)=O)CC12 c1(C(N(CCN(C(C(CC2CC2)NC(C)=O)=O)C)C)=O)ccc(C2CC2(F)F)cc1 C1(C(=O)NC2C(CC(=O)NC(c3c(C)ncs3)C)CCCC2)CC12CCCCC2 N1(C(c2c(C)ccc(C)c2)=O)CCC2CCN(C(c3sccc3SC3CC3)=O)C2C1 c1(CCCC(=O)NCC2(NC(CNC(CC(=C)C)=O)=O)CC2)cc(O)ccc1C n1(C2CN(C(CC(CC)NC(C3CC(F)C3)=O)=O)C2)ccc2ccccc12 CC(C(=O)NCC1CCN(C(C2CSC2)=O)C1)S(N)(=O)=O c1(C(N2CC3(CCN(C(C4CC5(CCC5)CO4)=O)C3)C2)=O)ncnc2cc[nH]c12 N1(C(c2ncccc2Br)=O)CCN(C(c2cc[nH]n2)=O)C2CC12 Cc1cc2[nH]c(C(=O)NCC(C3CC3)NC(C3CCN(C4CC4)C3=O)=O)cc2s1 CCC(C)(C(=O)N=S(C)(=O)c1cc(Br)ccc1Br)c1cnccn1 CC(C(=O)N(C)CC1CCCN(C(C23CC(C(F)(F)F)(C2)C3)=O)C1)C(F)(F)F c1(C(C)NC2OC(C)CC2C)ccc(CNC(c2ccc(Br)o2)=O)cc1 N1(CC(=O)N(CC(C)NC(C)C)CC)CC2CCOC2(CC)C1 S(=O)(=O)(c1ccc(S(=O)(=O)N2CCCCC(CO)C2)cc1)NC(COC)C c1(C(=O)NCCC(=C)CO)ccc(-c2ccc(C(=O)OC)cc2)cn1 C(C)(CC(=O)NCC(C)(C)CC1CN(C(c2cnns2)=O)C1)OC c1(C(=O)NC2CC(F)(CNC(C3N(C(C)C)CCC3)=O)C2)ccc(Cl)cc1 N1(C(C2CCCCCC2)C(=O)NC(C(=O)OC)C)CCC(S(=O)(=O)CC)C1 c1(OC)ncc(S(=O)(=O)N2CCC23CCCOCC3)cc1Cl C(=O)(C(C)(C)CS(C)(=O)=O)NCC1CCN(C(C2=C(C)OCC2)=O)CC1C CC(C)CC(C)C(=O)N1CCC(NC(c2n[nH]c(C(F)(F)F)n2)=O)C1(C)C N1(C(c2c(C)n(CCO)cc2)=O)CCCN(C(=O)C(C)c2cccs2)C(C)C1 N1(C(CC23N(C(=O)OC(C)(C)C)CC2CCCC3)=O)CCC2CCC(O)C1CC2 N1(C(C2C(C(=O)OC)C2)=O)CCC2(CCCCN(C(C3CSCN3C)=O)C2)C1 c1(C(=O)NC2C(NC(=O)C=CBr)C2)cccc(Cl)c1O CCC(CC(=O)NCC1(C(=O)NC2CCSC(C)C2)CCCC1)C1CCC1 C(=O)(CC(F)(F)C(F)F)N1CC(C2N(C(CCc3nc(=N)[nH][nH]3)=O)CCC2)(O)C1 c1(NCC)cncc(C(=O)NCC(C(C)C)NC(c2cnn(C3CC3)c2C)=O)c1 C1(C(=O)NCCn2ccc(C(=O)N(C3CCCC3)CCO)c2)CCC2CC1CO2 Cc1nc(-c2ccco2)ccc1C(N1CC2CC(O)CC12)C(=O)NC(C)(C)C C(C(=O)NCC(C)(C(C)C)NC(C12CC(F)(C1)C2)=O)(C(C)C)OC C1(CC)(NC(=O)C(C)(F)F)CN=C(N2CCC(N(C)C)CC2)O1 Cc1cc(C)c(C(=O)NC(C)CCN(C(=O)CSCc2ccccn2)C)c(C)n1 C1(C=C)(CC(N2CC(CN(C(C3(CCC=C)CC3)=O)CC)C2)=O)CCC1 C1(CNC(CCC(C)OCC)=O)CN(C(=O)C(c2ccc(Cl)cc2)=O)CC1(F)F CCCCCS(=O)(=O)CC(=O)N(C)CCN(C)C(c1c(COC)nn(C)c1Cl)=O N1(C(C2C(OC)CC2)=O)CC(NC(C2CCS(=O)(=O)C2)=O)C2(CCOCC2)C1 N1(CCC)CCC(C(=O)NCC2CC(O)(CNC(C3CCC=CCC3)=O)C2)CC1 C1(C(N(C2CCN(c3ccc(F)cc3)CC2)C)=O)C2CC2C2CC12 CC(CS(C)=O)C(=O)NC1(C)CN(C(C2CN(C3CCN(C)CC3)C2)=O)C1 c1(C(=O)NC(CN(C(C(N2C(=O)CCC2=O)CC)=O)C)C)ccc(C)n1C C1(n2cc(C(N3CCSCC3)C(N)=O)nn2)CCCCC1O c1(CC)cc(C(N2CCC2(C)CCO)C(=O)NCC(F)F)on1 CC(CNC(=O)C(c1cn[nH]c1)C)CC(=O)NCCCN1CCOC1=O N1(C(c2c(C)ncs2)=O)CCC(CNC(=O)C(C)C(F)F)(CN(C)C)C1 Cc1cc(=NCC2CC2CNC(=O)C=CCF)[nH]c(-c2ccccn2)n1 C12(C(N(C)CCN3CCCC3=O)=O)CCCC1N(C(C1SCCS1)=O)CC2 N1(CCN(C)C(c2csc(F)c2)=O)CCN(C(c2coc(C(N)=O)c2)=O)CC1 C1(C(=O)NC(C(=O)NCC(C)C(C)(C)C)C2CCCO2)CC2(C1)CC(O)C2 CC(C)CCCCCCNC(=O)NCCc1nnc(C2CC2)s1 CCCCC(CNC(c1ccc(C)n1C)=O)NC(=O)Cn1cnc(Br)n1 C1(C(=O)NC(C)Cc2cncnc2)(CNC(C2C=CCC2)=O)CC12CCC2 N1(C(C2CCN(C(C)=O)CC2)=O)CC(C2(NC(=O)CCCCC#N)CC2)C1 C1(C(C)NC(CN(CC)CC)=O)CCN(C(=O)CN(C)C(=O)OC)CC1 C(=O)(CC(CNC(C1CC1c1cncs1)=O)OC)NCc1cnc(CC)[nH]1 C(=O)(C(O)CCCNC(=O)C(N)=O)N1CC(CC(C)C)C1 c1(CC)nn(C)c(NC(=O)CNC(=NCC2CCCC2O)NC2CCOCC2)c1Cl N1(C(C(C)C2CCCC2)=O)CC(CC(N2CC(S(C)(=O)=O)C2)=O)C2(CC2)C1 c1(NC(C2C(COC)(COC)C2)=O)ccc(CNC(=O)Cc2n[nH]c(C)n2)s1 C1(N(C(CC2(NC3CC3)CC2)=O)C)CCN(C(c2cc(C(F)F)no2)=O)CC12CC2 c1(CC)nc2c(s1)CN(C(C(=O)NCCCF)C(C)C1CCCOC1)CC2 N1(C(C2CCCN(CCc3ccc(OCC#C)cc3)C2)=O)CCCCC(F)(F)C1 C1(C(C(N2C(CN(C(C(CN(C)C)(C)C)=O)C)CCC2)=O)O)CCS(=O)(=O)CC1 c1(NCCC=C=CC)[nH]c(=NC2CCC(S(C)(=O)=O)C2)nc2scnc12 C1=C(I)C(CN=S(C)(=O)NC2CCCCC2)=NN=C2N1CCCC2 C1(CCCNC(C(n2ccc(Br)n2)C)=O)CCN(C(C2COC2)=O)CC1 C(=O)(C(C)(C)C(N)=O)N1CCC(C(C)(C)NC(CCc2onc(CSC)n2)=O)C1 c1(CC(C)NC(C(c2cccs2)NC(C2CC(SC)C2)=O)=O)cnccn1 c1(NC(CN(CCC)C(C2CS(=O)C2)=O)=O)ccc(O)cc1F C1(C2CC2)CCN(C(C2N(C)CC(F)C2)=O)CC1n1cc(-c2cnn(C)c2)nn1 C1(CNC(=O)CCc2nccs2)CCCCN(C(c2ccc(F)s2)=O)CC1 C1(C(=O)NCc2c(C)cco2)C2CCC(C2)C1NC(C1SCCS1)=O C=CC1CCCCN1N1CCN(c2c(C)cc(C)cc2C)CC1.c12cnn(c1)C2 N1(C(=O)Cc2cnsc2)CCCCC(C2CN(C(=O)Cn3cnc([N+](=O)[O-])n3)C2)C1 C1(CNC(c2[nH]cc(C)c2)=O)CCN(C(c2cnncc2C)=O)CC1O N1(CC(=O)NC(C(=O)NC(CC)CCOC)C2CCCC2)CCCNC1=O CCCCCC(O)CC(=O)NC1CC1NC(=O)C(C1CCCC1)NC(C)=O N1(C(CSCCC)=O)CC(NC(=O)CNC(c2ccc(O)cc2)=O)C2(CCC2)C1 C12(CNC(=O)Cc3cncnc3)CC(CNC(C3C4CCN3CC4)=O)(CO1)C2 C#Cc1cccc(NC(=O)C=CCNC(=O)CC2(O)CCC2)c1 N1(C(C23CCCC2C3)=O)CCN(C(=O)CC2CCC2)C(C2CC2)C1 N1(C(C2CCOCC2)=O)CCCC12CN(Cc1ccc(F)nc1)C2 C1(C(N2CCCC(CCNC(C(C(=C)C)(C)C)=O)C2)=O)Cc2ccccc2S1 c1(C(=O)NCC2CC2NC(C(N2CCC(C)C2)=O)=O)cccc(S(N)(=O)=O)c1 CN1CCc2cc(-c3nc(-c4cnn(C)c4)nn3C3CCCSC3)sc2C1 C(=O)(CC(C(F)(F)F)OC)N(C1CCN(C(c2cc(O)cc(=O)o2)=O)C1)CCC CC1CC(c2nc(C3(C4CC4)CCCN3)no2)(C2CC2)CCO1 c1(NCC(CN(C(c2c(C)coc2C)=O)C)O)c(C#N)cnc2c(Cl)cccc12 CC1(C)CCN(c2cc[nH]c(=NCCOC3CCC3)n2)CC=CS1(=O)=O c1(C(N2C(C#C)CC2)=O)ccccc1-c1nccc(=N)[nH]1 Cc1cc(NC(C2(CCNC(c3ccn(C)c3)=O)CCCC2)=O)cc(C)c1 C(CC1=CCN(C(=O)Cn2cc(Cl)cn2)CC1)NC(C1(OCC)CCSCC1)=O C(=O)(C1=NNC(=O)CC1)NCCCN(C(C(CO)N(C)C)=O)C1CC1 N(C1c2ccccc2CC1NC(C1CNC(=O)N1C)=O)C(C(CCC)(C)CC)=O Cc1nc(CN(C(=O)CCC2CCCN2C(=O)CC2(N(C)C)CC2)C)no1 c1(OC)cccc2c(C)c(C(=O)NC3CC3CNC(=O)C=Cc3cc[nH]c3)oc12 c1(CC)occ(C)c1C(=O)NC1COCC1CNC(=O)C(C)Nc1cccnc1 CC1(C(=O)N2CC(CCNC(C3CC3[N+](=O)[O-])=O)C2)COc2ccccc21 C1(NC(C2OCCN(C(CSCC)=O)C2)=O)CCN(OC)CC1 c1(C(=O)NCC2C(O)C(O)CN2C(=O)CN2CCOC2=O)cccn2nnnc12 N1(C(CCSC)=O)CC(NC(c2cnc(C(C)C)n2C)=O)CC1(C)CC Nc1c(C(N2CCN(C(C3CC3(F)F)=O)C(c3cccnc3)C2)=O)cccc1Cl C1(C(=O)OCC2CC(=O)NCC2)CN2CCN1CC2 C1(NC(CCOCC=C)=O)CC(OC)CN1C(=O)CSCC(C)C C1(C(N2CC=CC2Cn2cc(CCc3ccccn3)nn2)=O)CCCC12CCC2 c1(CC)ccc(O)c(C(=O)NCC(C)(CO)NC(=O)C(C)C2CCC2)c1 CCC(CC)CCC(=O)N1CC(NC(c2oncc2C)=O)CCC1C N1(C(c2cccc(Cl)c2Cl)=O)CCC2CN(C(C3(F)CCOCC3)=O)CC2C1 c1(CN2C(C(=O)Nc3ccc(O)c(F)c3)CC3CC32)cc2ccccc2[nH]1 N1(C(C(CC)N(C)C(c2ncnc(O)c2F)=O)=O)CCC2(CC1)N=N2 C1(NC(CC2(C=C)CCC2)=O)CC2CC(NC(=O)CC3(O)CCC3)CC12 C1(C(=O)NCCCc2nc(C)[nH]n2)CCCCN1C(c1ccncc1)=O C1(CC)CN(C(=O)Cc2cn(C)nn2)CCC1CO.c12ccnc(n1)OCCO2 C=CCC(CNC(c1nccnc1CC)=O)C(=O)NCc1cccc(O)c1 S(=O)(=O)(c1ccc(NCC(c2cnn(C)c2)(C)C)cc1Br)NCCC C(=O)(CC(C)CC(C)(C)C)N1CCN(Cc2ccc(C)c(C)c2)C(C)C1 c1(C(=O)NCC(CC(C)C)NC(CCCCC#C)=O)ccc2c(c1)C=CS2(=O)=O N1(C(C(CCN(C)C)N(C)C)=O)CCC2C(NC(C3CCC(CO)O3)=O)C2C1 C1(C(=O)NCC(N(C(=O)CSCC#N)C)C2CC2)OCCCO1 C=CCC(F)(F)C(=O)N1CCC(CC(=O)NCC(O)CCC2CC2)CC1 CC1C(=O)N(C)CCN1C(=O)C(=O)NCc1cccc2c1OCC2 S(=O)(=O)(c1ccc(Cl)nc1C)N1C(COC)CN(C(c2scc(C)c2Cl)=O)CC1 CC1=C(C(=O)N2CCCC2C2(NC(=O)C(O)C3CC3)CC2)C(C)(C)CCC1 C1(C)(CCC)CCCN(C(C2CC2CNC(=O)CC(C)n2ccnc2)=O)C1 c1(C(=O)NCCC(C)NC(C2CCN(C)C2)=O)cnc2occc2c1 C(=O)(C=CS(F)(F)(F)(F)F)N1CC(NC(CSc2cccc(C)n2)=O)C1 N1(C(CN(C(C)C)C(c2cc(C(C)C)no2)=O)=O)C2CCC1CCSC2 c1(OC)ccc(CCCC(=O)NC2CCCCC2CNC(=O)CCCSC)cc1 c1(C(=O)NCCC2CC(NC(C(COC)OC)=O)C2)nccc2cccnc12 Cc1ncc2ccccc2c1C(=O)NC(C)CCc1cccnc1 CCC(CC)(CCNC(=O)CCCCSC)NC(=O)C=Cc1cocn1 CCC(CC)C(=O)NC1(C(=O)OC)CC1.N1(C)CCN(C(=O)CC(C)CF)CC1 N1(C(c2nn(C)c(F)c2)=O)CC(NC(c2c(F)cc(F)cc2F)=O)C(C2CC2)C1 c1(C(N2CC(CCOC)N(C(=O)CC3CCOC3)CC2)=O)ccc([N+](=O)[O-])cn1 n1(CC(=O)NC2CN(C(C3CCC4(C3)N=N4)=O)C2)nnc2c1CCCC2 C(=O)(C#CC1CCOC1)N(CCN(C(C)C)C(C1CC12CCCC2)=O)C N1(C(C(C)(F)F)=O)C2CCC1CN(C(=O)COC1CCC1)C2 N1(C(CN(C)C)=O)CC(F)(F)CC1(C)CNC(c1cc(-c2ccns2)on1)=O c1(C(=O)C(N2CCOCC2)NCSc2ccccc2)ncc(SC(F)(F)F)cn1 C1(CNC(C(C)(C)N(C)C)=O)C(C2CC2)CCN1C(c1nccn2nccc12)=O c1(NC(CN2CCC(C(=O)NCc3ccc(C)cc3)C2)=O)ccc2nonc2c1 C1(C2(C(=O)NCCOCC3(O)CN(C(C(C)O)=O)C3)CC2)CCCCC1O C1(NC(=O)CN2CC3CC3C2)(CNC(c2csc3cncn23)=O)CC2CCC1C2 c1(OCCOCC)ccc(-c2cn(C(CSC)CCNCS(C)(=O)=O)nn2)nc1 c1(OCC#C)ccc(NCC2CC3CCC2C3)cc1 C(CCN(C(=O)C(F)(F)C1CCCC1)C)(C(C)C)NC(C(C=C)O)=O C=CCC(C)(C)CC(=O)N1CCC(C)(C)C1C(=O)N(CC(=O)NC)CCC C(=O)(CC(SC)N)NCC1(C(=O)Cc2ccc[nH]2)CCC1.C(=O)(C)OC C(CCCCC(=O)N1CCC(O)(C(C)CNC(c2ccc(C)cc2)=O)C1)OC N1(C(c2cn(C)c(Br)c2)=O)CCC2CCCC12CNC(=O)CC#N c1(SC)c(C(N2CCCC(N(C(=O)C(F)F)C)C2)=O)cccc1Br CC1CC(C(=O)NC2CC(CC(=O)NCCNC(=O)CC3CCCC3O)C2)CCO1 c1(C(=O)NCCN(C(C(CC)n2cccn2)=O)CC2CC2)cc2oc(C)cc2[nH]1 c1(C(=O)NCCC(CNC(CNS(NC)(=O)=O)=O)O)ccc(C#N)nc1C c1(C(CC(=O)NC(CF)CF)N2CCOCC2)cc(F)ccc1F c1(C(=O)NCC(C2(O)CN(C(CCCC#C)=O)C2)(C)C)ccc(C)c(CO)c1 CCC(C(c1nnnn1Cc1nnn(C)n1)NC(C)CC)=Cc1ccsc1.C(c1ccsc1)=C C(C)(C(C)(C)C(=O)NC1(C2CCC2)CC1)NC(C(C)OCCC=C)=O c1(C(=O)NC2CC2CC(=O)NC(COC)CO)cc(N)ccn1 c1(CC(=O)NC(C(=O)NC(C(C)(C)OC)C)CC2CC2)cccc(F)c1 N1(C(CSCCCC)=O)CC(CNC(=O)CC(C)(C)c2ccccc2)CCC1C C(=O)(CCCCC(C)CC)NC(CCC=C)C(=O)NCc1c(C)cccc1C c1(NC(=O)NCCC2C(C(C)C)CCCC2)ccc(Cl)cc1C(F)(F)F C1(C(C)NC(=O)CSc2cn[nH]c2)CCCN(C(=O)Cc2cccs2)C1 C(=O)(CC(CC1CC1)NC(=O)COc1ccsn1)NCCCc1onc(C)n1 Cc1csc(C=CC(=O)NC(CCNC(c2cnc(Cl)n2C)=O)C(C)C)n1 N1(C(C(C)(C)C2CC2)=O)CCC2(C1)CN(C(C1CN3CCC1CC3)=O)C2 c1(C(=O)NC2CN(C(COC(C)=O)=O)CC2C)ccc2c(c1)-c1ccccc1C2 c1(C(N2CC(NC(C3(OC)CCSC3)=O)C2)=O)ccc(N2N=C(C)CC2=O)cc1 C(=O)(CC(C(F)F)NC(=O)OC(C)(C)C)N(C1CC1(F)F)C N(C(=NCCC1(OCC)CCOC1)NC1CCC1)C(C=C)C CCCC(CC)C(=O)NCC1(F)CCN(C(=O)CCCCC2CCCCC2)C1 c1(CC)cccc(C(=O)NCC2CCC2(F)F)c1O.C12CCCC1C(=O)N2 CC(C)CC(C(=O)N(C1CCN(C(C2C(C3CC3)C2(F)F)=O)C1)C)NC(N)=O c1(C2C(=O)N2)cc2sccc2s1.N1(C(C)C)CCCC1CN(C)CC1CCCO1 c1(OC)ncc(C(N2CC(O)C(O)C2CNC(c2ccc(Cl)cc2)=O)=O)c(C)n1 C=CCCCC(=O)N(C(CC)C(=O)NC)C.C1=CCNC(=O)C1 N1(C(C(C)NS(CC)(=O)=O)=O)CCC(NC(=O)C(C)(C)c2ccncc2)C(C)C1 Cn1cc([N+](=O)[O-])c(CC(N2CC(=O)NCC2CO)=O)n1 C1(NC(c2cccn3cncc23)=O)CN(C(=O)C2=CSCS2)Cc2nccn2C1 C1(C(CNC(C=CCOC)=O)C(C)C)CCN(C(c2ccc(CO)cn2)=O)CC1 C1(S(C)(=O)=O)(C(=O)NC(C)CCCNC(c2ncoc2-c2cccs2)=O)CCC1 NS(=O)(=O)N1CCC(C(=O)NCC2CN(C(C3CCN4CCCC4C3)=O)C2)CC1 C(=O)(CCCCC(C)(C)C)N1CCN(CCNC(CCc2ncc(C)[nH]2)=O)CC1 C1(NC(CC2CC(C)(C)CN2C(=O)CC2CCOC2)=O)CCC([N+](=O)[O-])CC1 N1(CC(O)CN)CCN(CCO)C(C)C1.c1(CCC(C)C(=O)NCC)ccccc1 N1(C(C=Cc2c(C)nccc2)=O)C2CCC1CN(C(c1ncccc1CO)=O)C2 N1(C(C(CCNC(C(C)N=[N+]=[N-])=O)O)=O)CCCC(F)(CO)C1 N1(C(c2c(N)cco2)=O)C2CCC1CC(N)C2 C1(C(N2C(C(CNC(c3c(C)csc3)=O)(C)C)CCC2)=O)CCOC(C)(C)C1 c1(CC(N2CC(C)C(NC(c3cc(O)cc(O)c3)=O)C2)=O)ccc2nonc2c1 C(C1CCCCC1)=CC(=O)NCCn1ccc(C(=O)NCC(O)C2CCC2)c1 FC1CC(N=c2[nH]ccnc2-c2nc3ccccc3o2)C12CCC2 O=C1CCN(CC2(c3ccncc3F)CC2)SC1CC1CCC1 FCC(N=c1[nH]c(N2CC3CC2C3)nc2c1COC2)c1ccccc1 C(CNc1nc(CC)cc(C)n1)(C(C)C(C)C)OCCOCC c1(C(=O)NCC2CN(C(C(=O)NCCNC(C)=O)=O)C(C)C2)ccc(O)c(F)c1F CC1CN(C(c2c(Cl)nsc2Cl)=O)CC1N=c1ccc(C#N)c[nH]1 C(=O)(CCCC(F)(F)C(F)(F)F)N1CCCN(C(CN2C(=O)NCC2)=O)CC1 Cc1nn(CCC(=O)NCC(C2CCC2)NC(C2CCC3(CC3)C2)=O)c(C)c1C c1(CC(=O)NC(C(C)NC(C2(SC)CCC2)=O)CO)cc(C)cc(F)c1 C1(C(N(CC(C)C(N2CC=CC(O)C2)=O)C)=O)CCCC(O)C1 N1(C(c2c(CC)c[nH]n2)=O)CCC(C(=O)NC2CC(CN(C)C)C2)C12CCC2 N1(C(c2cc(C3(F)COC3)no2)=O)CCc2ccncc21 C12(CNC(CCCC#C)=O)CC(NC(c3ccc4c(c3)CC4)=O)(C1)C1(CCC1)O2 C1(CCC(=O)NCC2CC2C(=O)N(CCCO)CC2CC2)CCCCC1 C1(C2CCN(C(=O)C(C(C)C)NC(=O)COC)C2)(NC(CCOC)=O)CC1 C1(NC(C(CC)(C)C(N)=O)=O)CCC2(CC1)CN(C(=O)CCCNC(C)=O)C2 C1(NC(C2(SC)CC2)=O)(CNC(=O)CCn2cnc(C)cc2=O)CCCCC1C C1(C(=O)NC2CCCN(CC)C2)CC(C)(C)CCN1C(=O)C(C)=CC(C)(C)C N1(C(C2C(CC)CCCN2C(=O)CCc2ccccc2)=O)CCC(O)CC(C)C1 c1(OCC)cccc(NC(c2ccc(F)cc2)CNC(=O)CC(C)(C)OC)c1 C(c1ccc(Br)o1)=C(C)C(=O)NC(C)(C)CN(C)C(c1c[nH]c(=N)o1)=O c1(C2C(C(=O)NCCCN(C(c3cncc(C)c3)=O)CC)CC2)ccc(F)cc1 c1(C(N2CCN(C(CC(CC)O)=O)CC2)=O)c[nH]c2ccc(Cl)cc2c1=O Cc1cccnc1C(=O)NC(C1CCCN1C(=O)CCn1ccnc1C(C)C)C C1(OC)CC(F)CN1C(c1cnc(-c2cnn(-c3ccccc3)c2)cn1)=O C(=O)(CCCC(=O)N1CCCC(NC(=O)CCCCNC(N)=O)C1C)N(C)C CC(C)(C)CC(F)C(=O)N1CC2(CCC2)CC1C(=O)NOC1CC1 C1(C(C)C(=O)N(C2CCN(C(=O)CNC(c3ccccn3)=O)C2)C)CCCCC1 n1(CC)ccc(C(=O)N(CCCNC(c2c(C(=O)OC)cnn2C)=O)C)cc1=O C1(CCNC(=O)Cc2ccccc2Cl)CCCCN(C(=O)CC2CC3CC3C2)C1 C(=O)(C(O)CCNC(=O)CSCCC#N)NC1(CCOC)CCOC1 C1(Cc2cn(CC(COC)O)nn2)COCCN1C(C12CCCCC1C2)=O C(=O)(C1=CCC(F)(F)CC1)N1CC=CC(NC(CCCCCOCC)=O)C1 C12(NC(c3c(OC)cccn3)=O)CCN(C(c3cscc3Br)=O)CCC1C2 c1(C(=O)NCC(C)C(N2CCC(C)C2(C)C)=O)ccn2ccnc2c1 c1(C(=O)NCC2CC3CN(C(C4CC=CCC4)=O)CC23)cc2cc(F)ccc2o1 N1(C(C=CC=CCC)=O)CC=CC1C(=O)NC1CN(C(=O)OC)C1 CC#CCC(C(=O)NCc1cnc(C)[nH]1)NC(c1cnc(C)cn1)=O C1(N(CC(C2CCSCC2)NC(C)=O)C(=O)CC2CC=CC2)CC2CC2C1 C1(C(=O)NC(C2CN(C(=O)C(O)C(C)(C)C)CCO2)C)C2CCC(C2)C1(C)C c1(C(C2CCCC2)NC(=O)NC(C)(C)C2CCC2)cc2c(nn1)CCC2 CC(C)S(=O)c1ccc(C(=O)NC(C)CCNC(c2ccc(F)c(N)c2)=O)cc1 c1(SC)cc(C(=O)NCC2C3CN(C(c4ccn(CC(C)C)n4)=O)CC23)oc1C c1(N(CCCF)C)nc2cc[nH]c2c(=NCC2CCCc3cncn32)[nH]1 CCCC(C(=O)NC1CN(C(C2(C(C)C)CC2)=O)C1)S(N)(=O)=O.C1CO1 c1(NC(C2C(c3n(C(C)C)ncc3)C2)=O)cccc(CCCCF)c1.C1(=O)CN1 c1(C(C)=O)n[nH]c2ccc(C(=O)NC3CC4CC3CN4C(=O)C(Cl)=CCl)cc12 C1(CC(=O)NC(C(C)C)(C)CNC(=O)Cn2cnc(=N)[nH]2)OCCOC1(C)C c1(C(N2CCC(CC(=O)NCCO)C2)=O)cccnc1CNC1CC(N(C)C)C1 N1(CCCN)CSCCSC1.c1(C(=O)OC)ccoc1NC(=O)N(C(C)C)C c1(CC)ccc(C(CCC[Si](C)(C)C)C(=O)OC)cc1.C(C)(CC)NC c1(C(=O)NC2CC(NC(CCC(=O)c3ccncc3)=O)C2)coc2ccccc12 c1(C(=O)NC2CCCCCN(C(C(C)C)=O)C2)ccc(=O)n2c1CCC2 N1(C(COC)=O)CCC2(C(=O)Nc3ncc(-c4ccc(F)cc4F)n3C)CC2C1 c1(OC)cc(CN(C)CC2CCN(C(c3csnn3)=O)C2)ccc1C(F)F C1(C(=O)NCC(C)N(CC)CC)CCCCN1Cc1cc(C(=O)OC)ns1 C1(NC(c2ccc(CF)cc2)=O)CCCCN(C(=O)Cn2cc(C3CC3)nn2)C1 C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NC1CN(C(CP(C)(C)=O)=O)CC1O C1(C(N2CC(CCC#C)C2)=O)CC(F)(F)CN1C(=O)CCC(C)CC c1(CN(C)C(C2CC(NC(=O)CSc3nc[nH]n3)CCO2)=O)cncc(F)c1 c1(C(=O)NC(C(C2CCC2)NC(c2ccnc(C)n2)=O)C(C)C)cccc(F)c1F N1(C(c2cc(CC)nn2C)=O)CCN(C(c2cc(OC)ccn2)=O)CC12CC2 C1(NC(C(c2cnccn2)C)=O)CCN(C(=O)CC2CN(C)C2)CC(C)(C)C1 C(N=c1[nH]c(=NC(C)CSC)[nH]c2c1CSC2)C1(CC)CC1 Cn1cc(C(=O)NCC(C(C)(C)C)NC(=O)Cc2cccs2)c(C2CCCO2)n1 Cc1nc(=NC(=O)c2ccnn2CC(=O)NC2CCS(=O)(=O)C2)o[nH]1 C1(NC(c2c(CC)n[nH]c2)=O)CC1C1CCCN(C(c2cc(C3(C)CC3)n[nH]2)=O)C1 CCC(C(=O)OC)NC(C1CC(CNC(c2cnn(C(C)C)c2)=O)C1)=O CCCCCCCCCCCC(=O)N1CCCCC1CNC(c1snnc1C)=O C1(NC(c2cccc(C#C)c2)=O)CCN(C(=O)CCc2csc(=N)[nH]2)CC(O)C1 C(=O)(CC(C(=O)NC(CO)C(C)NC(=O)C=Cc1ccsc1)NC(C)=O)OC N1(C(c2ccccc2)C(N)=O)CCN(Cc2sccc2-c2nn[nH]n2)CC1 C1(C(N2CC3C(C(=O)OC)(C3)C2)=O)CCN(C(=O)C2(CO)CCCCO2)O1 N1(C(C(CC#C)C)=O)CC(NC(=O)C#CC2(C)COC2)C2(CCC2)C1 c1(C(=O)NC2(CNC(C3C(CC)OCCC3)=O)CC2)cc(OC)cc(Br)c1 Cc1ccc2nc(NC(=O)C(N3CC(C4CC4)CC3C3CC3)=O)cn2c1 C#CC1(C(=O)NCCCCN(C)C)CCN(C(C2CCCCC(=O)N2)=O)C1 C1(CC)CN(C(=O)CCc2cncs2)CCN1c1ncc(C)c(O)n1 C1(C(=O)NCCN(C(c2cc(C)[nH]n2)=O)CCOCCO)CC2CCCCN2C1 C1(CNC(CN(CCOC)C)=O)C(C)CCCN1C(=O)CCOC(C)=O N1(C(C(C(CC)CC)OC)=O)Cc2ccccc2CC1CNC(=O)CC(C)C C=CCC(F)(F)C(=O)NCC(c1cccc(C)c1)NC(C1(CCF)CC1)=O S(=O)(=O)(c1ccc(N(C)CC2CCSC2)c(F)c1)NC(c1cccnc1)C(C)C C(C(C)(C)[N+](=O)[O-])n1cc(C2CN(C(c3c(COC)c[nH]n3)=O)C2)nn1 C(=O)(CC(C(F)F)N1CCOCC1)NC1C(NC(C2CC(=O)NC2)=O)COCC1 C(N1CCN(C(c2ncccn2)c2ccccc2)C1=O)N1C(=O)NCC1 Cc1cn2c(n1)CC(C(=O)NCCC1(C)CCN(C(c3ccncc3)=O)C1)CC2 C1(c2nnc(C)o2)CN(C(=O)OCC2CCCS2)CCO1.N12CCC(C1)C2=O N1(C(C(N2C(=O)CCC2=O)C)=O)CCC(C)(NC(=O)C(=CC(C)(C)C)NC2CC2)C1 O=C(C1=C(Cl)CC1)NCC1CC(CNC(c2ccccc2Cl)=O)CO1 C=CCC(C)(C)CC(C(=O)NCCCC(C)(C)C)N(C)C(c1ccccc1)C C=CCC(CNC(=O)C(CC=C)OC)C(=O)NC(C)C(C)(C)OC C(C)(C(C(C)C)NC(=O)CSCc1scnc1C)NC(Cc1cnc(C)[nH]1)=O N1(C(c2c(C)nn[nH]2)=O)CCCC(C)(NC(c2scnc2-c2ccccc2)=O)C1 c1(OC)cc(C(=O)NCCNC(=O)CC2CC(SC)C2)ccc1S(C)(=O)=O c1(C(=O)NC(CN(C(Cc2c(C)cc(C)s2)=O)C)(C)C)ccc(C)nc1O c1(OC)ccc(C(N2CC3(C2)CN(C(=O)CCN2CCC2)C3)=O)c(Br)n1 C(C1CCCCC1)=CC(=O)NCC(C1CCCCC1)NC(C1CC2CCC1O2)=O c1(CC(N2C(C(N(C(C)C)Cc3cccc(OC)n3)=O)CC2)=O)cccc(F)c1O CC(C)C#CC(=O)N(CCCCNC(=O)CCC1CCCC(O)C1)C N1(C(C=C(CCC)C)=O)CCC(C)(C(=O)NCC(C)(C2CC2)OC)CC1 c1(C(=O)NC2(C)CC(NC(C(CCC)OC)=O)C2)ccc2ncsc2c1 C1(C(N(C2CC2)CC2(NC(C3CC(SC)C3)=O)CCC2)=O)CC1C1CCOCC1 c12cncn1C2NCC(Cc1nnnn1C(C)(C)C)OC.C(COCCO)OC.C1CC1 c1(C(=O)NCCN(C(CCn2ncc(C)c2)=O)C)cc(C)c(F)c(S(C)(=O)=O)c1 C1(NC(C2CC(C)(O)C2)=O)CN(C(=O)CCc2ccc(Br)cc2)C2(CCC2)C1 C1(C(=O)NC(C)C(C)(C)NC(C2CC(F)(F)C2)=O)CCC2(CCCC2)CC1 c1(OC)ccc(C(N2CCN(C(c3cc[nH]c(=N)c3)=O)CC2)=O)cc1 CCS(=O)(=O)c1ccc(CC(=O)Nc2ncccc2OCc2ccccc2)cc1 C#Cc1cccc(C(=O)N(CC(N2CCCC(C)(N(C)C)C2)=O)C2CCC2)c1C c1(C(N2C(COC)CN(C(c3cnc(C)nc3)=O)CC2)=O)scc2c1OCCO2 c1(C(=O)OC)ccncc1C(=O)NCc1ccc(CNC(=O)CN(C)C)cc1 C1(COC)(CNC(=O)CC(C)n2ccnc2)CN(C(C2(CF)CC2)=O)C1.N(C)C C1(CNC(Cc2c(C)con2)=O)CCC(N(C(=O)Cc2ccc(F)cn2)C)CC1 C1(C(=O)NC2C(NC(c3ccncc3)=O)C2)CCc2nnnn2C1 CC(Cn1ccnc1)C(=O)NCC1CCCC1NC(=O)CC1CCCCO1 c1(OC)ccc2c(c1)C(C(=O)NCC(C(C)(C)C)NC(c1cnc(Cl)s1)=O)CC2 CC1=NOC2(C1)CC(C(=O)NC1CC(CNC(c3cn(C(C)C)cn3)=O)C1)C2 C1(C(CNC(c2c(CC)cco2)=O)(C)O)CCN(C(=O)Cc2nc(=N)[nH][nH]2)CC1 N1(C(c2c(C)cccc2)=O)CCCC(C)(C)C1C(=O)NC(C)CC(F)(F)F C1(CN2C(C=C)CC2)CN(C(=O)OC(C)(C)C)C2(CCC2)C1 c1(CCNC(C2C(C)OCC2)=O)ccc(CNC(=O)CC(F)(F)F)cc1 N1(C(C(CC)(C)C)=O)CCC=C(C(=O)NC(c2ccc(Br)cc2)C#N)C1 c1(C(=O)NCC2N(C(c3ccc(SCC)cc3)=O)CC2)csc(S(C)(=O)=O)c1 C1(CNC(CCSCCC)=O)CCC2(CCC2)C1NC(=O)C=CC(F)(F)F C1(N(C(=O)C=Cc2cnc[nH]2)C)CCC(NC(c2csnc2Br)=O)CC1 C1(CC(=O)NCCC(C)(C)NC(Cc2n(C)ncc2)=O)CCC(C)(C)OC1 c1(-n2cc(CC3CN(C(CC=C)(C)C)C3)nn2)ccccc1[N+](=O)[O-] n1(CC)ncc(C(=O)NCCCN(C(=O)CSCc2ncc(C)o2)C2CC2)c1C c1(C2C(C(=O)NCC(C)(C)NC(c3c(CCC)[nH]cc3)=O)C2)ccc(C)nc1Cl CCC(C)C(C(=O)NC1C2CN(C(c3c[nH]nc3C3CC3)=O)CC12)N(C)C C(=O)(C1=NNC(=O)C1)N1CCC(NC(c2cnn(CC)c2Cl)=O)(CF)C1 CC(CCC(=O)NCCc1cc(C(=O)N(C2CCCC2(C)O)C)no1)N(C)C c1(NC(CNC(CCC(C)OCC)=O)C(C)C)cc(C)nc(S(C)(=O)=O)n1 C#Cc1ccc(C(N2CC3CC2C3NC(C23CC(OC)C2C3)=O)=O)cc1 Cc1cnn(C)c1C(=O)NCCCCNC(c1ccc(Cl)s1)=O C(C)(CCC(=O)N(C)CCO)OC.C(=O)(C(=O)NCC(F)F)NCCC(C)SC N1(C(=O)COc2ccsn2)CCC(C2CCCN2C(=O)C(F)C2CCC2)CC1 Cc1cc(C)n(Cc2ccc(CNC(=O)Nc3cc(C4CCCC4)ncn3)o2)n1 C(=O)(C(C(C)C)NC(=O)C(C)Cn1cccn1)NC(Cc1cc(C)[nH]n1)C c1(OC)cc(Br)ccc1CNC(c1nnnn1C1CCOCC1)C1CC=CC1 c1(C(=O)NCC(C(C(=O)N2CC(C#C)(F)C2)F)C)ncc2ccccn12 c1(C(=O)NC2CN(C(CCC(C)OCC)=O)C3C2C3)c[nH]c2ccc(F)cc12 CC1CC(NC(c2cccc(F)c2Cl)=O)CCN1C(=O)CC1CC(C2CC2)C1 N1(C(=O)NCCCCCCCC)Cc2ccccc2C1CCO C1(N)(CN2CCCC(c3nc(C(C)C)on3)C2)CCCCCC1 C1(CNC(c2cccnc2)CNC(C(=O)NC(CC(C)C)C)=O)C2CC3C(C2)C13 c1(C(N2C(CN(C)C(C3CCC(=O)N3)=O)CCC2)=O)cc(C#N)ccn1 c1(C(=O)NC2(CC=C)CCN(C(C(CC#C)(C)C)=O)C2)cccc2c1OCCO2 c1(CC)ncc(C(N2CC(CCNC(=O)CSCC(C)C)C2)=O)c(C)n1 C1(C(=O)N(C)CCF)(NC(=O)NC(c2ccn(C)n2)C)CC1(C)C C1(NC(C2(C#C)CC2)=O)C=CC(C(=O)NC2CC(C)(C(=O)OC)C2)C1 C1(NC(Cc2cc(CC)no2)=O)CCN(C(c2cnc(=N)[nH]c2)=O)CC1F CC(C)C(CNC(c1cncn1-c1cnn(C)c1)=O)NC(=O)CC1CCOC1 C1(C(=O)Nc2cccc(-c3cn(C)nc3)c2)C2CC1CN(C)C2 C1(C(=O)NC(CNC(c2n(C(C)C)ncc2)=O)C2CCC2)CCCNC1=O c1(C(=O)NCC(CCC)NC(c2cnn(C(C)(C)C)c2)=O)nccc2[nH]ccc12 c1(C(N(CCCOCCNC(Cc2cc(CC)no2)=O)C)=O)ccc(F)cn1 c1(C(N2C3CN(C(CC4ON=C(C)C4)=O)C(CC3)C2)=O)cccc2c1CC(=O)N2 C(=O)(CCCCCC(C)(C)C)NC1(CNC(C(C)CC(F)(F)F)=O)CC1 c1(C(N(C2CC(NC(C3CCC(C)(C)OC3)=O)C2)C)=O)cc(C#N)c(N)cc1O c1(C(=O)NCCCN(C(=O)CC2CCSC2)C(C)C)ccc[n+]([O-])c1 C(C(F)(C(=O)N(C)CCN1CCCC1=O)C(C)C)NC(c1scc(C)c1)=O C1(NC(CC2N(CC)CCOC2)=O)CCN(C(=O)C(C)c2cccs2)CC1C c1(C(=O)NCC(N(C(C(CCC)N(C)C)=O)C)C2CC2)ccc2nn(C)cc2c1 N1(C(COCCOC)=O)CCCC1(C)CNC(c1ccccc1C1CCC1)=O c1(C(=O)NC(C(C)C)CCN(C(=O)CC2CCN(C)C2)C)cc(C#N)ccc1O C1(NC(CCNC(=O)OCC)=O)CCCCN(C(c2cc(C(N)=O)no2)=O)C1 C1(NC(=O)CC2CCN(C(C)C3CC3)CC2)(Cc2ccc(O)nc2)CCOCC1 c1(-c2ccc(C(N(CC(C(=O)C(O)C3CCC3)=O)C3CC3)=O)o2)nc2ccccc2s1.OC C1(NC(C(C)OCCCCCC)=O)CCCCN(C(c2cc(C)ccc2O)=O)C1 c1(N(CCNC(CCC)=O)CC)c(Br)cccc1[N+](=O)[O-] C1(C)(C(=O)NC2C3CN(C(c4cccc(OC(C)C)c4)=O)CC32)CCN(C)C1=O c1(C(N(C2CC(NC(CC3(CC=C)CCCC3)=O)C2)C)=O)cc2ccnn2cn1 C1(CCC#C)CN(C(c2cc(I)cn2C)C(=O)NCCOCC)CCO1 N1(C(c2n(C)nnc2Br)=O)C2CCC1CN(C(=O)C#CC1CCOC1)C2 C1(C(C)C)CN(C(=O)CC2CNC(=O)C2)CCN1C(=O)C(=O)NC1CCCC1 C(=O)(CCCS(C)(=O)=O)N1CCC(NC(Cc2cc(C)on2)=O)C(C(N)=O)C1 C#Cc1cccc(CNC(=O)C(C2CCCCC2)NC(=O)CCS(C)(=O)=O)c1 c1(OC)cccc(F)c1CC(=O)NC(CNC(C1(Cl)CCCCC1)=O)CC(C)C C1(=CC(=O)NC(C2CCN(C(c3c[nH]c(C(N)=O)c3)=O)C2)C)CCC(C)C1 c1(NCc2ccc(C)cn2)cnc(Br)c(Br)n1.C12CCCN(C1)C2=O c1(C(N2C(CNC(Cc3ccn(CC)n3)=O)C=CC2)=O)cccc2c1CCO2 Cc1cccc(Br)c1C(=O)NC1C=CC(CNC(=O)CC2CCCOC2)C1 C1(CC)CN(C(=O)C=Cc2nccs2)CCC1NC(C1(C(F)(F)F)CC1)=O C=CC(CCC)CC(=O)N1CCCC(CC(N2CCC(C)=C(C)C2)=O)C1 Cc1cc(F)c(C(=O)NCCC2CCCN(C(c3cc(F)cs3)=O)C2)c(F)c1 N(C(=NCC1CCCC1)N(C)CC(=O)NC)C(C#C)C1CC1 c12cn(nn1)CCS2.C(C(C(=O)O)C1CCCN1)NC(C1CCCCC1)=O C1(CNC(CCOC)=O)CCCC2(CN(C(C3CCCN3S(C)(=O)=O)=O)C2)O1 CCCCCC(C)(CC)C(=O)N1CC2CC(C1)N2C(c1cccc[n+]1[O-])=O c1(C(=O)NCC2(F)CN(C(C(CCCC)C)=O)C2)cnc2nccnc2c1 c1(OC)ccnc(NC(C2CCCN2C(=O)C=CCBr)=O)c1I c1(OC(C(=O)NCC2CN(C(CC=CC=C)=O)CC2C)C)ccc(Cl)cc1C Cc1cc(Cl)cc(C(=O)NC2CCCC2CNC(=O)CSCC2CCCO2)c1C c1(OC)ccc(Br)c(F)c1CN1CCCC(C(=O)NCC(C)(C)F)C1 c1(CC(=O)NCC(CNC(=O)C=Cc2cc[nH]n2)O)cncnc1O C(C(C)(C)CN(C(=O)Cn1cnc(C(N)=O)n1)C)NC(C1C(C(=O)OC)C1)=O c1(C(=O)NC2(COC)CN(C(c3n[nH]c(CC)c3Cl)=O)C2)cncc(C)c1 C(=O)(CC(C)P(C)(C)=O)NCC(CNC(C(=Cc1cccnc1)C)=O)O N1(C(CNC(C2CCC(C)O2)=O)=O)CC2CC1C2C(=O)NCC(F)F c1(C(C(=O)NCC(C)CN(C)C(C2(C)CC(F)C2)=O)=O)cc(F)cc(Cl)c1 CC(C)CC(CC(=O)NCC(C)(C)CCO)NC(C1(n2cnnn2)CC1)=O c1(C(C(C)C)=O)cccc(NC(c2c[nH]nc2SC(C)C)=O)c1 c1(C(N2CC(CN(C(=O)CC3CCCC(=O)N3)C)C2)=O)coc2cc(F)ccc12 N1(C(CC2CCC(=O)NC2=O)=O)CCC(C2CN(C(c3cc(Cl)c[nH]3)=O)C2)CC1 C1(CNC(C(C)NC(=O)NC)=O)(NC(=O)C(CC)C2CCOCC2)CCOCC1 c1(C(=O)NC2(C)CC(C(=O)NCC3(C)CCOCC3)C2)ccc([N+](=O)[O-])o1 c1(C(=O)NC2(C)CC(NC(=O)COC3CCC3)C2)cnc2ccsc2c1 c1(OC)cc(O)c(C(N2CCN(C(=O)C(C)C3CCCO3)CC2)=O)cc1Br C1(C(=O)NCC2C(NC(c3nc(OC)oc3)=O)CC2)CC(=O)N(C2CCCC2)C1 C(N=c1cccc(S(=O)(=O)N2CCOC(C(F)F)CC2)[nH]1)C1CC(C)(C)C1 C12(C(N3CC4C(NC(CSc5n(C)ccn5)=O)(C4)C3)=O)CCC(F)(CC1)C2 N1(CC(=O)NCCN(C(C)C)C(C2CCN(C)C2C)=O)Cc2ccccc2C1=O C1(CNC(c2c(C)nc(C(C)C)s2)=O)CC(C)(C)CN1C(=O)CC(C)F N1(C(CC2C(C)(C)C(O)C2)=O)CC2(CCN(C(=O)CCc3ccoc3)CC2)C1 C1(C(N(c2c(C)nsc2)C)=O)CCN(C(C2C3CCC(F)(F)C23)=O)C(C)(C)C1 C=CCCCC(C(=O)N1CCNC(=O)C1C)NC(=O)Cc1cc(CC)no1 C1(NC(C(=O)NCC)=O)CN(C(=O)CSCc2ncc[nH]2)CC1C C(CCNC(C1(NC(C2C3CCCOC23)=O)CC(F)C1)=O)(C(C)C)OC C1(OCCC2CC3(N(C(C=NC(C=CC(C)C)=O)=O)CC3)C2)CCC(=O)C(C)C1 c1(C(=O)NCC2C(NC(C(C)(CC3CCC3)OC)=O)C2)ccc(Br)cc1C#N CCC(CC(=O)N1CC(NC(C2CC(SC)C2)=O)C(C)(C)C1)C(C)(C)C Cc1ccc(C(F)CNC(=O)NCCCCCN2CCNC2=O)cc1.C(C)(C)O N1(CC(=O)NC(CC2CN(C(C3(C)CCC(C)C3)=O)C2)C)CCCCCCC1=O N1(C(c2nc(C)[nH]n2)=O)CC2CN(C(c3nncn3-c3ccccc3)=O)CC2C1 O(NC(=O)C(CC1CCCC1)NC(c1cnn(C)c1)=O)CCCC c1(C(=O)NCC2N(C(CCC(=O)OCC)=O)CC(O)C2O)nnn2c1COCC2 N1(CC(=O)N(C2CC2)CC2CCCC2NC(=O)CCOC2CCC2)C(=O)CNC1=O c1(C(=O)OC)[nH]c(=NCC23CC(NC(c4nnsc4C(F)F)=O)(CO2)C3)sc1C c1(CCC)nc(C(=O)NC(C)(CNC(C)=O)CO)co1.C1(C)C(=O)N1 c1(NC(C)=O)ccc(S(=O)(=O)NC2(C)CCC(C)C2)o1 CCC(C)C(CC(=O)NCC1CC(NC(=O)Cc2cccnc2C)C1)OC(C)=O c1(C(=O)OCC2COCC(C)O2)cnc(OC(F)F)c(N(C)C)c1 c1(OC)ccc2cc(C(N3CCCC(NC(=O)C(CCO)N(C)C)C3)=O)[nH]c2c1 c1(-c2c(OC)cc(C(N3CCC(C(F)F)CC3)=O)cc2)cnc2ccncc2c1 c1(NC(c2ccccc2-c2cn3c(n2)SCC3)=O)cnc2[nH]cnc2c1 C1(n2cc(C(C)OC)nn2)CC2CCC(C1)N2C(c1c(F)cccc1F)=O N1(C(C(C)c2cccs2)=O)CCC(C2(O)CCN(C(=O)C3=CCCS3)C2)CC1 C(CC(C)N=c1[nH]c2c(c(=NCCCc3cnn[nH]3)[nH]1)CSC2)SC CCC(CCOC(=O)OCCN(C(=O)CC)C)CC C1(C(=O)NC2CCN(C(C3(OCC)CCC3)=O)C2)CCCN(S(C)(=O)=O)C1 C1(C(N(C(C(=O)NCC)C)C)=O)CCCCC1CNC(=O)COCCF c1(C(C(=O)NCCC(=C)CNC(c2cc(CCC)n(C)n2)=O)=O)ccc(F)cc1 C1(C(=O)Nc2n(CC)ncc2)CCN(CCCNC(=O)OC(C)(C)C)CC1 c1(C(=O)NCCNC(c2cccc(OC)c2OC)=O)cnc2snc(C)c2c1 N1(C(c2c(C)[nH]nc2C(C)C)=O)CCOCC(NC(=O)C(C)Cc2ccccc2)C1 CN1C2CCC1CN(C(C1(CNC(=O)Cn3cnc(C#N)n3)CC=CC1)=O)CC2 C1(NC(C=CC(C)NC(c2ccc[nH]2)=O)=O)CCCC(C)(C)C1 C=CCCCC(CNC(=O)C(C)(C)C1CC1C#N)CCCN1CCOCC1 c1(N(C(=O)NCCC(CCOC)C)CCN2CSCC2=O)ccc(F)cc1F O=C(CN1CCCN(c2nccnc2C(=O)O)CC1)C(=O)NNC(=O)c1ccon1 c1(C(=O)OC)ccc(Br)cc1CCNC(c1ccc(OCCO)cc1)=O n1(CC)ncc([N+](=O)[O-])c1C(=O)NC(CCS(C)=O)C(C)C C1(C)(C(N2C(C)CC2CO)=O)CCCN(C(=O)CN2CCNC(=O)C2)C1 N1(C(c2c(C)cc[nH]c2=N)=O)CCC2(CCCC2CNC(C2C(C)C2C)=O)CC1 C1(CNC(C2(C)CCCC2)=O)CCCN(C(=O)C(O)CF)C1 c1(CCN(C(C(COC)O)=O)c2ccccc2)ccc2c(c1)OCO2.C1C(=O)N1 N1(C(CCc2nnc(C)n2C)=O)CCC(O)(CNC(=O)C(C)C2(O)CCC2)CC1 N1(C(C2(C)CCCS2(=O)=O)=O)CC2CCCN(C(c3n[nH]c4c3CCC4)=O)C2C1 CP(C)(=O)CC(=O)NCc1occc1C(=O)NCC(O)C(F)F C1(NC(c2c(C)ccnc2O)=O)C(C)CCN(C(c2ccc(N)cc2F)=O)C1C CCC(C)(CC)C(=O)NC1CCCN(C(c2ccc(C(F)(F)F)cc2O)=O)C1 C1(CNC(C2ON=C(CC)C2)=O)CCCC2CN(C(=O)C=Cc3cscn3)CC12 C(=O)(C(C)C(O)CC(C)C)NCCN=c1[nH]nc(C2CC2)o1.CCO C12(C(N3CC(OCC(=O)N(C)CCN4CCCC4=O)C3)=O)CC1CNC2=O c1(C(=O)NCC(CC)NC(=O)CCc2nnc(C(C)(C)C)s2)ccc(C)cc1C C12CCCN(C1)C2.C1(C(N2C(N(C)C)CC2)=O)COC(=O)N1.C(=O)(NOCCO)O C(c1cn(C(c2cccc(CNC(=O)C(=O)C(C)C)c2)C)nn1)=CC CC1(C)CC(CNC(c2cnco2)=O)CN1C(c1nc(=N)cc[nH]1)=O C12CN(CCC1CO)C2=O.N1(CCN(C)CC2(N(C)C)CC2)CCOCC1 C1(CNC(C(C)(C)Nc2nccs2)=O)CCCCN1C(=O)CNc1ccncc1 C(CCC(N)=O)(C(=O)NC1CCC(C(=O)NCC(F)(F)C(N)=O)C1)N(C)C c1(OCC(=O)NCC(C)CN(C)C(c2csc(=O)[nH]2)=O)cccc(F)c1F C#CC1CCN(C(C2OCCC2CNC(=O)Cc2cnn(CC)c2)=O)C1 c1(C(=O)NC(CNC(C(=O)NCC)=O)CO)cncc2ccsc12 CCCCCC(O)CC(=O)N(C)CC=CC(=O)NCc1ncccc1Cl c1(C(N2C(CNC(CCN(C)CC)=O)CC(F)C2)=O)cc(O)cc(O)n1 N1(C(CC=CC)=O)CCC(C(N2CCC(C)(O)C(O)C2)=O)CC1(C)C C(CC=CC)(C(=O)N1CCC(CC=CCC)C1)=CNC(C(CCC)=CCC)=O N1(C(C=Cc2n(C)ccc2)=O)CCN(C(=O)Cn2ccccc2=O)CC1C(F)F c1(OCC)cccc(-c2nc(-c3ccncc3C)n(C3CCOCC3)n2)c1 C1(C(=O)NCC2CCC(NC(C3(C)CC(=C)C3)=O)C2)CCC2(CCOCC2)O1 Cc1cnc(C)c(C(N2CCN(Cc3ccccc3-c3cnco3)CC2C)=O)n1 c1(CNC(CSC(C)(C)C)=O)ccc(CNC(C2(F)CCOC2)=O)cc1 n1(CC(=O)NC(CC)CN(C)C(C2CCC(C(N)=O)C2)=O)cc(C2CCOC2)cn1 C#Cc1cn(C)nc1C(=O)NC(C)C(C)NC(=O)CCc1cnn[nH]1 c1(NC(C(N2CCN(c3n(C)nnn3)CC2)=O)=O)cc(P(C)(C)=O)ccc1F c1(C(=O)NC(CC)CNC(=O)C(O)CSC)c(C)nc2ccnn2c1C c1(OCC)ccnc(N2CCC(CCNC(=O)Cc3nc(C)cs3)(C(=O)NC)C2)n1 CC(C)CC(C(=O)N1CCC(c2cn(C3CCCCC3CN(C)C)nn2)C1)C(N)=O C(CNC(c1cncc(C)c1)=O)(C(C)C(C)C)NC(c1nc(CCC)sc1)=O C1(C(=O)N)CC2CCC2C1.c1(C(NC)=O)cc(CNC(C)CN(C)C)no1 CCCN=C(NCc1cnc(-n2nc(C)cc2C)s1)NCC1(O)CCCC(C)C1 C1(C#N)(C(N2CCC(O)(CCNC(C3CC(SC)C3)=O)C2)=O)CCCCCC1 N1(C(=O)Cn2cc([N+](=O)[O-])cn2)CCC2CCCN(C(=O)CCC3CCC3)C2C1 C1(NC(c2cc(CC)on2)=O)CC2(CCN(C(C3C(C)CC3C)=O)CC2)C1 C(=O)(CCCC(C)O)N1CCC(N(C(=O)C(C2CCOCC2)F)CC#C)CC1 N1(C(=O)NCCC2COCC(C)O2)CCCc2sccc2C1 N1(C(C=CC(C)C)=O)CCCN(C(C2CCOC(C)C2)=O)CCC1 Cc1ccc(Br)c(-n2cc(C(N3CC(C4(NC(=O)C(C)O)CC4)C3)=O)nn2)c1 N(C(=NCCc1cn[nH]c1)NCC(c1ccccc1F)C1CC1)C(C)C c1(CN2CC3CCN(C(c4cc5c(s4)CSC5)=O)C3C2)c[nH]c2cc(F)ccc12 c1(OC)ccc([N+](=O)[O-])cc1NC(c1nnnn1C)(C1CCCCC1)CF N1(CC(CN2CCC(OC)CC2)O)CCn2ncc(S(C)(=N)=O)c2C1 C(C)(C)(CCC(=O)NCCCC(C)(C)NC(C1CC1CC(C)(C)C)=O)N(C)C CCC(C)C(O)C(=O)N1CCN(C)C(CNC(c2nccs2)=O)C1 CN1CCC(CCNC(C23CC(NC(=O)CC4CC(F)C4)(C2)C3)=O)C1 c1(CCC)onc(C)c1C(N1CCN(C(c2cccnc2N)=O)CC1)=O N1(C(=O)NCC2(C#C)CCCC2)CCN(C)C(c2nc(-c3ccccn3)no2)C1 C1(C(CN(C)C(c2cnns2)=O)=O)CC12CCOCC2 CCC(CNC(=O)CSC1CC1)(CC)C(=O)N1CCC(F)(CO)CC1 N1(C(c2cc(C)oc2C2CCC2)C=C)CC2CCC(C1)N2C(c1ccccc1)C c1(C(N2CC(C)(C)C(NC(=O)CCCCCF)C2)=O)csc(=NC2CC2)[nH]1 Cc1cc2[nH]c(C(N3CCN(C(C4CC4F)=O)C(c4ccccc4)C3)=O)cc2s1 CCCCCC(=O)NCCN(C(c1cc(C)sn1)=O)CC C12(CC)CC1CN(C(c1sccc1CNC(=O)CC1CCCC(=O)N1)=O)C2 c1(C(N2CC(COC)(NC(c3ccc(CF)cc3)=O)C2)=O)ccnc(C)c1O CC1OC2(C(=O)NCCNC(c3cc(C4CCCC4)n(C)n3)=O)CCC1C2 c1(CC)nnc2c(C(=O)NC3CCCN(C(c4cc(C)co4)=O)C3)cccn12 C1(C(=O)OC)CCC(C)N(C(=O)Nc2nnnn2C2CCC2)C1 C12(C(=O)NCC3C4CN(C(C5(CC(C)(C)C)CC5)=O)CC43)CCC(O)(CC1)CC2 C1(N(C(=O)C(C)CCc2cccc(F)c2)C2CCNCC2)CC(C(=O)OC)CCO1 CCC(C(=O)N1CCCC1CN(C(=O)C(C)Cn1cccn1)C1CC1)SC CC1=CCC(C)(C(=O)NC2CCN(C(c3cccnc3Cl)=O)CC2F)CC1 C1(C(=O)NCC2CCC2)(CC)CCCN1C(=O)CC1CC1C1CC1 c1(C(N(C2CCN(C(C3CCC(C)(O)C3)=O)CC2)C)=O)cccc2cc(Cl)ccc12 C(=O)(CC(C)C(F)F)NC1C(NC(CC2(NC(C)=O)CCCCC2)=O)CCCC1 C1(CCC(=O)NCC(C)C2CC2)CCN(C(=O)CN(C)C2CC2)C1 N1(C(C2C(CC)C2)=O)CCC(NC(c2cc(C3CC3)nc(Cl)c2)=O)CC(O)C1 N(C1CN(C(c2cc(C)c(F)c(C)c2)=O)CCc2ccccc21)C(C(F)OC)=O C1(N2C(C)CC2)CCCCCC1.c1(OCCNC(=O)NC(C)CO)ccccc1 Cc1cccc(Br)c1CC(=O)NC(C)C=CC(N1CCSC(C)C1)=O N1(C(C(C)N2CCCC2)=O)CC(C(N)=O)(CNC(=O)COCC2CCCO2)C1 CC1=CC(C(F)(F)F)(NC(=O)Nc2ccc(Nc3ccncc3)cn2)C=C1I C1(NC(c2c(OC)noc2C)=O)CCCCCC1C(=O)N(C(CO)C(C)C)C Cc1ccc2sc(N3CCC(CO)(NC(=O)Cc4c(C)n[nH]c4C)CC3)nc2c1 C(=O)(C(O)CC(C)(C)C)N1CCCC(CCNC(c2occ(C)c2C)=O)C1 N1(C(C(C(C)C)NC(C)=O)=O)CC(C)CN(C(c2csc3cncn23)=O)CC1C C12CC(C1(C)C)CC(=O)N2.c12cc(cs1)NC2=O.C1(N2CCCC2)(C(C)=O)CCC1 N1(C(c2c(C)nns2)=O)CC2(CCN(C(c3cn(C(C)(C)C)nn3)=O)CC2)C1 Cc1cc(C(N2CC(NC(c3cc(N)cc(F)c3)=O)C(C)C2)=O)nc(C)c1 N1(C)CCN(CCF)CC1.n1(CCOC)c(N2CC(O)C2)nnc1-c1ncn(C)n1 c1(C(=O)NCCC2(OC)CN(C(=O)C(Cl)=CCl)C2)ccc2c(n1)CCCN2 CC1CC(NC(C23CCOC(C)(C2)C3)=O)CCN1C(=O)CC(O)c1ccccc1 c1(OC)ccc(Cl)c(C(=O)NCC(C)(C)CNC(C2(C)C=CCC2)=O)c1N C1(CNC(COCCC=C)=O)CCC2CN(C(C3CC(Cl)(Cl)C3)=O)CCC2C1 C(C)(CC(=O)N1CCCC1CNC(=O)Cc1ccn(C(F)F)n1)OC c1(CN(C2CC3CNC2C3)C(C(=O)Nc2ccsc2)=O)cccc(Cl)c1 C1(C(=O)NCCC2CCC(NC(=O)CC(C)CF)C2)(COC)CCOCC1 c1(C(=O)NCC2(CNC(C3=C(C)CC3)=O)CC2)cc(N(C)C)nc(Cl)c1 C#Cc1ccc(F)cc1C(=O)NC(C)CN(C)C(C1CCC1C(C)(C)C)=O CCC(C)(CNC(=O)C(O)CC1CCCC1)C(=O)NCCc1cccnc1C c1(OC)nccc(SC)c1CN1CCCC1(C)C(=O)Nc1ncc(Cl)nc1Cl C(=O)(C1=CCC(NC(=O)CC2CC(F)(F)C2)C1)NCCc1onc(C)n1 c1(CN2CC(C(=O)NCC(F)(F)F)C2)c(F)ccc(Cl)c1Cl Cc1ncc(C)c(N(C(C)CCNC(C2(C3CCCO3)CC2)=O)C)n1 C1(NC(C2CC(C)(C)CN2C(=O)C=C(C2CC2)C2CC2)=O)CC2CC1C(O)C2O N1(C(C2C(CCC)C2)=O)CC2=C(C1)CN(C(=O)C(C)n1nccn1)C2 C1(C(N2CC(n3cc(SCC4C(=O)NC(=O)N4)nn3)C2)=O)COC2(CCC2)CO1 c1(OCC(=O)NCC2C(NC(=O)C=C3CC3)COC2)ccc(Cl)cc1 c1(NC2C(C(=O)NCc3ccc(OC)c(OC)c3)C2)c(OC)cccc1C#N N1(Cc2cc(C)ncc2)Cc2ccccc2C1C(=O)N1CCNC(=O)CC1 C1(O)(CNC(C(C)(C)CO)=O)CCCN(C(C2CCCN2C2CC2)=O)CC1 C1(NC(=O)CC2CCCCCC2)CC(CNC(c2occc2Cl)=O)C12CCC2 c1(C(=O)NCC(CNC(CCSCCC)=O)C)cccc(Nc2ccc(C)s2)c1 C(=O)(C(C)=Cn1ccnn1)N1CC(CCNC(c2c(CCC)nco2)=O)C1 c1(C(N2CCS(=O)(=O)C(C)C2)C(=O)NCCCC)cnc2cc(C)nn2c1 N1(C(c2cc(N)sc2)=O)CC2CCC(C1)N2C(=O)CC(O)C1CCCC1 c1(CC)ccc(C=CC(=O)NCC2C3CN(C(C4(C)CC4(Cl)Cl)=O)CC23)o1 N1(C(C=C(CC)CC)=O)CCC2(CC1)CN(C(=O)NC1CC(n3ccnc3)C1)C2 c1(NC(C(N(C(C(CC)C)=O)C)C2CC2)=O)ccc(F)nc1 c1(C(=O)NCCN(C)C(C2(C#N)CCOCC2)=O)cnc2onc(C3CC3)c2c1 c1(CC(=O)NCC(C)(O)CNC(c2cccnc2)=O)c[nH]c2cc(Cl)ccc12 c1(C(N2CCC(CNC(C3CCN(CC#C)CC3)=O)C2)=O)c(Cl)sc2nnsc12 n1(CC)cc(C(=O)NCC(C)N(C)C(C2CCCC2CF)=O)cc1C1CC1 N1(C(c2cccc(OC)c2)=O)CC(C)(C)CC1C(=O)NCCC(C)CCO N1(C(CC2CC(C(=O)OC)C2)=O)CCCN(C(=O)CCC2CC2)CCC1 c1(C(C(=O)N(CCNC(=O)C(CO)c2ccccc2)CC)O)ccc(Cl)cc1F N1(C(CSCc2ccc(C)s2)=O)CCC(C2CC2)(NC(C2CCCN2C)=O)C1 N1(C(CNC(CC)=O)=O)Cc2ccccc2C(NC(c2c(C)noc2C)=O)C1 N1(CCc2cccc(OCC#C)c2)CCC(CC)OC(C)C1 C(=O)(C(O)C(C)(C)C)N(CCN(C(C(C)CNC(=O)CC(C)(C)C)=O)C)C C(CO)(C(=O)N1CCC(OC2(CSC3CC3)CCC2)C1)NC(N)=O c1(N(C2CN(C(C(C)CC3CCC3)=O)C2)C)ncnc2c1nnn2C c1(NC(=O)Nc2ccc(SCC)cc2C)nc2c(n1C)CCOC2 C1(C(=O)NCC(C)(C)NC(COCc2nnc(C)s2)=O)C(C)(C)C1(F)F C12(C(=O)NCC3(F)CN(C(C4(CC)CC4(F)F)=O)C3)CCCCN1CCC2 C#Cc1ccc(C(=O)NC2(CC)CCCN(C(C3CC34CC(O)C4)=O)C2)cc1 C(=O)(C(CC(C)C)CC(C)C)c1ncc2c(N)n(ncn1)NCC(CC)NC2=O C(=O)(C(O)CCC1CC1)N(C(=O)Cn1cc(CNC(C(C)C)=O)nn1)C(C)C C(C#CC(=O)NCCC1CCCN(C(C2CCCC2C)=O)C1)(OCC)OCC c1(C(N2C(C)CC(NC(CCSCC)=O)C2)=O)cc(NC)c(C2CC2)nn1 C#Cc1c[nH]nc1C(=O)NC1CC(CCC(=O)NCC2(c3cccc(F)c3)CC2)C1 Cc1ccc(C(N2CCCC(CCNC(=O)CCS(C)=O)C2)=O)cc1S(C)(=O)=O C#CCC(O)C(=O)Nc1cccc(NC(C2CCC(C(C)(C)C)CC2)=O)c1 CC1CC(CNC(c2ccc(C(=O)CF)cc2)=O)CN1C(c1cc(O)cs1)=O C(=O)(C1CCCc2nn[nH]c21)N1CCCCC(NC(c2cncc(NC)c2)=O)C1 N1(C(CC(CN(C)C)O)=O)CCC(F)(F)C(NC(=O)CNc2ccccc2)C1 C1(CN(CCOCC)Cc2ccc(Cl)cc2F)Cc2ccccc2N1 C(CC(F)F)(C(=O)NC(c1nnc(O)o1)C)NC(CN1CCC(OC)C1)=O c1(NCCC(C)N(C)C)[nH]c(=NCCC(C)S(C)=O)nc2ncn(C)c12 c1(C(=O)NC(CCCNC(C(C)OCCOCC)=O)C)ccc(C)cc1C C1(N(C2CCCC2)C(c2ccc(CC)nc2)=O)CCN(C(c2ns[nH]c2=O)=O)CC1F C1(CC(=O)NC2CCN(N(C)CCO)CC2)CC2(C1)C(F)(F)C21CCC1 C1(CC)CCN(C(=O)C=CCNC(=O)Cc2cccc(C)c2)CCO1 C1(NC(CCC)C(=O)OC)CN(C(=O)OC(C)(C)C)C2(CCCC2)C1 C1(C#N)(C(=O)NC(CCOC)CNC(c2cn(CC(F)(F)F)nn2)=O)CCCC1 C1(CNC(C(C)(C)c2cscc2Cl)=O)(NC(=O)CSC2CC2)CCCCCC1 c1(NC(=O)NC2CCN(C(=O)OC)C2)cc(S(C)(=O)=O)ccc1F N1(C(c2ncc(C#C)cn2)=O)CCC(C)N(C(C2CSCCS2)=O)CC1 C(CC(=C)C)(C(=O)N(C1CCCC1)CCO)NC(CC=C)=O c1(CC(N2CC(CNC(c3c(CC)noc3)=O)C(C)C2)=O)ccc2c(c1)CCC2 C(c1ccc(F)c(Cl)c1)=CC(=O)NCC1N(C(c2occ(C)c2)=O)C2CCC1C2 Cc1cc(Cl)ccc1CC(=O)NC1CCCN(C(=O)CN2CC(=O)NC2=O)CC1 CC(C)(C(F)(F)F)c1ccc(OC(=O)CCCOc2ccc(F)cc2)cc1 c1(C(=O)NCCN(C(c2c(OCC)ccs2)=O)C(C)C)ccn2cc(C)nc2c1 N1(C(C(CC2CCCC2)NC(C(C2CCCCC2)C)=O)=O)CC2CC1(CO)C2 C1(NC(C(C2CCCCCC2)OC)=O)CN(C(=O)CC(C)CF)CC1N=[N+]=[N-] c1(CC)cc(C(=O)OCCCCc2ccc(C(F)(F)F)cc2)n(C)n1 c1(C(N2C(C)CC(CNC(=O)Cc3ccncc3Cl)C2)=O)ccnc(Cl)c1O Nc1cc([N+](=O)[O-])ccc1C(N1CCCN(C(c2c[nH]cc(Cl)c2=O)=O)CC1)=O N1(C(=O)OCC)CC2(C1)CN(C(=O)C(Cc1ccccc1)N1CCOCC1)C2 c1(CNC(c2ccc(C3N(C(=O)OC(C)=O)CCCC3)o2)=O)ccc(O)nc1C c1(-n2c(C)cc(C(=O)C(C)SC(F)(F)F)c2C)ccc2c(c1)CCN2C C1(C(N2CC(COC(C)=O)C2)=O)CCN(C(c2cc(=N)[nH][nH]2)=O)C1(C)C c1(C(N2CC(CNC(C3C(OC)CCC3)=O)C(C)C2)=O)nn(C)c(C)c1Cl c1(COC)cncc(C(=O)NC2CCCCC2NC(c2conc2C)=O)c1.C1(C)CC1 C1(C(=O)NCc2occ(C)c2)C=CCN(C(c2nnsc2C)=O)C1 c1(CNC(C2CCC(c3nn[nH]n3)C2)=O)cccc([N+](=O)[O-])c1 N1(C(CCCOC)=O)CCCC(C2CCN(C(c3cccn4cnnc34)=O)C2)C1 C(CCCCC(=O)NC(C(N1Cc2ncsc2C1)=O)c1cccs1)=CC N1(CCNC(C2(C#N)CC2)=O)CCC(NC(=O)CCCc2nccs2)CC1 c1(CC)c(C(=O)NCCCN(CCCCNC(=O)C(C)(C)CO)C)nnn1C C1(CC)CN(C(=O)CSC)CCN1C(C1CCN1CC)=O N1(C(C2C(C)(C)C2c2nc(=N)[nH][nH]2)=O)C(CNC(c2cc[nH]n2)=O)CC2CC12 Cc1nc2sccn2c1C(N1CCC(CNC(C2CC3(CC3)CO2)=O)C1)=O C1(n2cc(CCC(=O)NC(c3ccc(C)cc3)CCC)nn2)CCCC1(C)O c1(NC(N2C(c3c(C)n[nH]c3C)CCC2)=O)ccc2c(c1)OCCO2 n1(CC#C)ccc(C(N2CCC(CC(C)C)C2)C(=O)NC2CCC2)c1 Cc1nc(=N)[nH]c(C)c1C(=O)NCC1CN(C(=O)CC(=O)NC2CC2)CCO1 c1(C(=O)NCC(CC(C)C)NC(C(CCOC)NC(C)=O)=O)cnc2[nH]ccc2n1 c1(NC2CN(NCC)C2)[nH]c(=NCc2nccc(OC)n2)nc2sccc12 N1(C(CCNC(COC)=O)=O)CCC2C(NC(c3ccc(CN(C)C)[nH]3)=O)C2CC1 c1(CCC(=O)OC(c2ccc(F)cc2F)C)cccc(S(N)(=O)=O)c1 C1(NC(N2CCOC(C(O)CO)C2)=O)C=CC2CC1CO2 C1(NC(c2c(C)coc2)=O)CC2(C1)CC2C(=O)N(C1CCNC1=O)C(C)C CC(CN(C)C)C(=O)NC1CCCC1NC(c1cc(C(F)(F)F)no1)=O c1(C(N2CC(C)C(NCc3nccnc3Cl)C2)=O)cc(Br)cc(Cl)c1Cl Cn1ncc(NC(=O)COC(F)F)c1C(=O)NCCN1CCC(n2cncn2)C1 c1(C(N2CCC(CN(C(C(CN(C)C)O)=O)C)C2)=O)cc2n(n1)CCO2 CCC(C(=O)NC(CCCOC)C(=O)N1CC(S(N)(=O)=O)C1)C(C)(C)CC Cc1c(C(N2CC(NC(c3cnsn3)=O)CCC2C)=O)oc2c(F)cccc12 N1(CCOC)CC(c2nc(-c3ncccn3)nn2CCC(F)(F)F)CC1=O N1(C(C(C)OC)=O)CCCCC(CNC(=O)COc2cccc(C(N)=O)c2F)C1 N1(C(=O)NC)CCC(C(=O)NCC(F)CNC(C2(COC)CC=CC2)=O)C1 c1(CC)cnc(O)c(C(=O)NC(C)CCNC(c2[nH]nc(OC)c2Cl)=O)c1 C1(CC=C)(C(=O)Nc2csnc2C)CN(C(=O)C(C)n2ccnn2)C1 c1(NC2CCC3CN(C(C4CC(C)=C(C)CC4)=O)CC32)nc(C)nc2scc(C)c12 N(C(=NCC(C)N1CCCCC1)NC1CCOCC1)CC(CCC)OC C(=O)(C1=CCSC1)NC(C(C)NC(C1CC1Sc1ccccc1)=O)CO c1(CC2(F)CN(C(c3n(C)ncc3CN)=O)C2)cc(F)ccc1F C1(NC(C2C3CN(C(c4cc(C)[nH]n4)=O)C2C3)=O)CCCCC1(C)C C(=O)(CC(C)(C)C(C)=O)N1C(C(N(C)CC2CCN(CC)C2)=O)CC2(CC1)CC2 C1(C(=O)NC2CCC2)CCCN1NC(=O)C1CCC(C2CC2)C1 N(C1CC2(CN(C(=O)C(C)CC)C2)n2ccnc21)C(c1c(CC)nn(C)c1)=O c1(SCC)cccnc1C(N1CCC(NC(=O)CCCC2CCC2)C1C(C)C)=O c1(C(N2CC(CNC(C3(CO)COC3)=O)CC2(C)C)=O)cc(Cl)nnc1O Cc1ncc(Cl)c(C(=O)NC(C2(O)CCN(C(c3cn4c(n3)CCC4)=O)C2)C)n1 C#CC1(NC(=O)C(F)C2CC(NC(=O)CCCC(=O)OC)C2)CC2CCCC12 N1(C(c2c(CCC)[nH]cc2)=O)C2CCC1CN(C(=O)CCC1CC1(Cl)Cl)C2 C12(C(=O)NC34C(CN(C(c5ncsc5Br)=O)C3)C4)CC1CCC2(F)F N1(C(C(C)NC(C)=O)=O)CC2CC(C(=O)NCC3CCC=CO3)CC1C2 c1(C(N(CCN(C(C2CC=CC2)=O)CC)CC)=O)c(C)nn(C2CC2)c1O N1(C(C2CC2C(F)F)=O)CC2OCCN(C(=O)CCOC3COC3)C2C1 c1(OCC)cc(C(=O)NCC2CN(C(=O)COc3cnn(C)c3)CCO2)ccn1 Cc1cc(CC(=O)NCCCN(C(=O)Cc2cncnc2)C)ccc1Cl C1(NC(C2CCN(C)CC2)=O)C2CCN(C(c3cc(N)ccc3Cl)=O)CCC12 N1(C(C(C)Oc2ccccc2Cl)=O)Cc2n[nH]cc2CC1C(=O)O C=Cc1cncc(C(N2CCC(CCNC(=O)C(C)(CC)OC)CC2C)=O)c1 c1(OC)cc(Cl)cc(F)c1CN1CC2CC2(C(=O)Nc2ncccc2Cl)C1 CCCCC(CC(=O)N(C1CCN(C)C1=O)C)NC(=O)COC(CC)CC c1(C(=O)NCC(c2ccc(C)cc2)CNC(CCCOC)=O)nccc(CO)n1 C12(NC(c3cccc(C)n3)=O)CCC(CNC(=O)C(C)C3CCCC3)(CC1)OC2 C=C1CCC(C(=O)NCCNC(C2CCCN2C(=O)C(C)O)=O)CC1 C=C(Cl)C(C)(C)C(=O)NC1CCCCC1NC(C1CC1Br)=O c1(C(C(=O)N(C)CC2(CNC(C3CC3)=O)CC2)O)ccc(C(=O)CC)cc1.SC C1(c2cn(CC(=O)NC(C)CC3CC3)nn2)C(C)(C)C1(C)C CCCCC(C)CCC(=O)N1CCC2CN(C(c3cc(C4CC4)on3)=O)CC2C1 C=CC1(C(N2CCC(C(=O)NC(C(O)CO)C3CC3)C2)=O)CCCCC1 CC(CC(=O)NC(C(=O)NCc1ccccc1C#N)c1ccoc1)C(F)F c1(C(=O)NCC(C(C)(C)C)NC(C(C(C)C)F)=O)cc(F)c(F)c(C#N)c1F c1(-c2n(CC3N(CC=C)CCOC3)ccn2)cc(F)cc(F)c1F C(S(=O)(=O)CCNC(=O)CC1(O)CCOC1)c1cn(CCC=C=C)nn1 n1(CC)cc(C(=O)NC2CC(C)(NC(=O)C=CC3CCCO3)C2)c(C)n1 C(C(C)(C)C(=O)NC(C)Cc1cnn(C)c1)N(C(C(CC1CCC1)OC)=O)C c1(C(=O)NC2(CO)CN(C(c3cn(CC(F)F)cn3)=O)C2)ccc2c[nH]nc2n1 c1(CC)ncsc1C(=O)NCc1occc1C(=O)NCC1CCOC1C Cc1ccc(-c2cn(C3CN(C(N)=O)C3)nn2)cc1.C12CCN(CC1)CC(=O)N2 Cc1cc(-c2cn(CCNC(=O)CCc3cc(OC)cc(Br)c3)nn2)ccc1F CCCN=C(NCc1ccc([N+](=O)[O-])cc1)N1CC2C(C)C2C1 N1(C(CCC2(CCC#C)N=N2)=O)CC(NC(c2ccncn2)=O)C(C2CC2)C1 CCC(C(=O)N1CCC(N(C(=O)Cn2cc(N)cn2)CC)C1)c1ccccc1 c1(N(C)CC2C(OC)CCC2)nc2c(c(=NCCN3CCC3)[nH]1)COC2 c12cnc(F)cc1C(=O)O2.c1(N(CCC)C)cc(Br)cnc1C N1(C(COCCOC)=O)CCC(NC(=O)C(C)N2CCC2)CC1 c1(C(=O)NCC=CCC(=O)NC(C(CC)C)CO)ccc2nccn2c1 c1(CCC(N2CC(N(C)C(C3C4CC4C4CC34)=O)C2)=O)ccc(O)c(F)c1 N1(Cc2cn(C(C)C)nc2)CCN2C(C1)C2=O.c1(CO)c(O)cccc1O c1(CC(C(C)C)NC(=O)Cn2cc(CC(O)C3CC3)nn2)ccc(F)cc1 N1(C(CCC2CC(C)C2)=O)CCC(O)C1C(=O)NCC1CCOCC1 N1(C(c2scc(OC)c2)=O)CC2(CCN2C(C2COCCC2(F)F)=O)C1 C1(C)(C(=O)NCCCC(C)NC(c2cc(O)cc(O)n2)=O)CC(O)CN1C C(=O)(C(F)C(C)CNC(=O)CN1CC(C)(C)C1)N(c1sccc1C)CC c1(CC(N2CCC(N(c3ncc(F)cn3)C)C2)=O)ccc(Cl)nc1F c1(C(=O)OCC)n[nH]c(C)c1CNC(=O)CN1CCCC1C CC1CN(C(C2CC3CCC2O3)=O)CCC1NC(c1cnc(S)n1C)=O N1(C(CP(C)(C)=O)=O)CCC2CCC(NC(=O)CCS(=O)(=O)N3CCOCC3)C12 c1(C(=O)Nc2c(C(=O)Nc3ncccc3F)n[nH]c2)ccc2cccc(F)c2n1 C1(NC(Cc2c(C)noc2)=O)CCC2(CCCN2C(=O)C(C)c2ccco2)CC1 C1(NC(c2cn(CC(=O)OC)nn2)=O)CCCCN(C(C2CC23CCOCC3)=O)C1 C=CCC(C(=O)NCC(=O)N(CCCCCSC)C)NC(C)=O N1(CCC(=O)NCC2CCCC2NC(c2ccc(C(F)(F)F)s2)=O)CCOC1=O C(=O)(C1=NN2CCCN=C2N1)N1C2C(NC(=O)CSC3CCCO3)CC(CC2)C1 N1(C(c2ncc(SC(C)(C)C)s2)C(=O)NC(C)(C)C)CCC2CSCC2C1 C(c1cc(Cl)ccc1Cl)=CC(N1CC2(CN(C(c3cc(C)no3)=O)C2)C1)=O N=c1cc[nH]c(C(N2CCC2C(N2CCC(OCCF)C2)=O)=O)n1 c1(C(N2C(CO)CC(NC(c3c(CCC)nco3)=O)C2)=O)ccc(C#N)cn1 C1(NC(C(c2ccc(C)o2)C)=O)CN(C(c2ccncc2Br)=O)CCC1F C=CC(C)CC(=O)N(CCCNC(=O)Cc1cnn(-c2ccccc2)c1)C(C)C Cc1nc(N2CCCC(C(C)NC(c3cc(Cl)sc3Cl)=O)C2)c(F)c(C)n1 C1(CC(=O)N(CCCC(C)(F)F)C)CCCN(C(=O)CC(C)O)CC1 C1(CN(C)C(C2CC3(CCCC3)C2)=O)CN(C(=O)CN2CCCC2)CC12CC2 c1(CC)cc(C(=O)NCC2CC2CNC(c2ccccc2OC(C)C)=O)c(C)o1 C#CCC(O)C(=O)NC(CNC(=O)COCC1CCCC1)CC(C)C c1(C(C)C)cc(C(=O)NCCC2(C(N3CCC3C3CCC3)=O)CCC2)no1 N1(C(C2C(C)(C)CCCO2)=O)CCCC2CN(C(C3CCCS3(=O)=O)=O)CC12 C(=O)(C(C(=O)N1CC(CO)(NC(C2OCC3CCCCC23)=O)C1)C(C)C)OCC c1(OC)cc(C(C(=O)NC2CCOC2)N(C2CCC2)C(C)C)c(F)cc1Cl C1(C(NOCCCC#C)=O)(NC(=O)CCOC2CCCC2)CCC(C)(C)C1 N1(C(C(C)Oc2ccc(C)cc2)=O)CC2CCCC1(CNC(C1CC1F)=O)C2 c1(NC(C(CC)Sc2ccccc2)=O)cc(Cl)c(O)c(Cl)c1 c1(N(CC(CNC(CCSCCC)=O)O)C)ccc(C#N)nc1 C=CCC(C)N=c1[nH]c(=NCC2(Cl)CC23CCC3)[nH]c2c1COC2 c1(CC)cc(C(N2CCC(C(C)NC(c3ccc(CC4CC4)s3)=O)C2)=O)on1 c1(C(=O)NCCOCC)n[nH]c2c1CN(C(=O)CC(C)N1CCOC1=O)CC2 C1(C)(NC(Cc2c(C)ncs2)=O)CCC(NC(=O)CN(CC(C)(C)C)C)CC1 C(=O)(CCCC(=O)N(C)C)N1CCC(N(C(c2ccc(F)s2)=O)CC)C1 C1(NC(C2(C)CCC2)=O)CCC2(CC1)CN(C(c1cc[nH]c1C1CC1)=O)C2 C1(COC)(NC(=O)C(C)SC(C)C)CCN(C(c2cc(CO)n(C)n2)=O)C1 C1(C(=O)Nc2ccn(C)n2)(NCC(CC)(C)c2ncc[nH]2)CCN(C(=O)NC)C1 c1(CC)nc(NC2(CCNC(=O)CCOc3cccnc3)CC2)c(C)c(C)n1 C1(CNCc2n[nH]c(C)c2C)CC(C)(C)OC(C)(C)C1 Cc1ccc(-c2ccc(C(=O)NC(C)C(C)NC(=O)CCn3cncn3)s2)o1 c1(CC(=O)N(CCOCCCNC(c2c(C)cc(C)o2)=O)C)c[nH]c(=N)nc1O N1(C(C)=O)CCCCCC1CNC(=O)CC(c1ccc(F)cc1)NC(N)=O CC(C)(C)CCCC(=O)NCCOCCCNC(C1CCC(O)C1)=O c1(C(=O)NC2(C(=O)Nc3ccn(CC)n3)CCCOC2)ccc(O)c(C)c1 N1(C(C2C(NC(C3C(C(=O)OC)C=C3)=O)CC2)=O)CC(C)C(F)(F)C1 C1(NC(=O)CCc2cccc(F)c2)(CO)CCCN(C(c2nocc2Cl)=O)C1 c1(NC(C2OCCN(C(C3C(=O)CCC3)=O)C2)=O)nc2c(s1)COCC2 N1(C(c2[nH]cc(C(N)=O)c2)=O)CC2CCCC1(CNC(C1CCOC1C1CC1)=O)C2 c1(C(=O)NCCN(C(=O)CC2(O)CCCCC2)CCOCCO)ccc(C#N)nc1O c1(C(C)NCc2c(C)scc2)ccc2c(O)nccc2c1 N1(C(c2ccccc2C(F)(F)F)C(=O)NCCCC)C2CCC1C(C)C(CO)C2 c1(CC(=O)NC2(C)CN(C(C=CS(C)=O)=O)C2)coc2ccc3ccccc3c12 N1(C(C)=O)CCC(=CC(N2CCOC(CCc3ccccc3)C2)=O)CC1 c1(C(C)(C)C)cc(C(C)(C)C)cc(CN2CCNC(CS(C)(=O)=O)C2)c1O c1(CNC(=O)NC2CCNc3ccccc3C2)ccc2c(n1)COCC2 CC(C)C(C)C(C)CC(=O)N1CC=CC(CC(=O)NOC(=O)C2=CCCCC2)C1 Cc1ccc(C(C)C(N2CC(C)(NC(c3cnn(CC(C)C)c3)=O)C2)=O)s1 n1(CCC(=O)NC(C2CCN(C(=O)COC3CCCCC3)CC2)C)cnccc1=O C(=O)(C1=COCCO1)NC(C1CCCN(C(c2c(OC)cccc2)=O)C1)C C1(C)(C2(NC(C(C)Sc3ncccn3)=O)CC2)CCN(c2cc(O)nc(O)n2)CC1 C1(CCNC(c2n(CCC)nnn2)c2nocc2Br)COC(C)(C)OC1 N1(C(C(C)=O)=O)CCC(NC(c2cc(C3CCOCC3)n[nH]2)=O)C(CO)CC1 c1(C(N2C(C(=O)OC)CC2)=O)n[nH]c2c1CN(C(c1cc(F)c(F)c(Cl)c1)=O)C2 N1(C(c2cc(OC)n(C)n2)=O)CCC(O)C(NC(C2COCC2(C)C)=O)C1 c1(Nc2cc(C(=O)NS(CCOCC)(=O)=O)ncc2)cc(C#N)c(Cl)cc1F C1(NC(CC(C=C)CC)=O)CC1C1CCCN(c2cc(CC)nc(CC)n2)C1 c12cccc(c1)C(O)c1cn(nn1)CCCC(=O)N2C.c1(SC)sc(S)nc1C CC1(NC(C23CCCC2C3)=O)CC(NC(c2c[nH]c(Br)c2)=O)C1 c1(C(N2CCC(C(C)NC(c3n[nH]c(C)c3F)=O)CC2)=O)nccn2ccnc12 N1(C(C(C(C)(C)O)NC(c2ccncc2Cl)=O)=O)CC2CCC2C2(CC2)C1 C1(CC)CCN(C(c2ncc(OC)cn2)C(=O)NC(C)C)CCO1 c1(NCc2c(CC)con2)nccc(=NCCCc2cccc(O)n2)[nH]1 C1(C(C)CNC(=O)C(=O)NC2CCC(F)(F)C2)CCC(F)(F)CC1 CC1=C(C(=O)N2CCC(NC(=O)Cn3nc(C)c(Cl)c3C)CC2C2CC2)CCO1 C(C(C(=O)NCC1CN(C(c2cncc(F)c2Cl)=O)C1)C(C)(C)C)OCC=C C1(NC(c2nccnc2Cl)=O)CC2CC(C1)N(C(C1CC=CCO1)=O)C2 c1(CNC(c2occ(C)c2)=O)ccc2c(c1)CN(C(=O)CSc1ccncc1)C2 c1(C(N(CCCCN(C)C(c2cn3c(n2)SCC3)=O)C)=O)cn(C)c(=O)nc1O C(=O)(C1CCCc2ncnn21)NCC(C)NC(C(C(=O)OCC)C(C)C)=O C1(NC(Cc2c(C)nsc2)=O)CCCCN(C(c2cc3sccc3[nH]2)=O)C1 C(CCc1ccccc1)(C(C)NC(=O)CCCF)NC(C(C)=C(C)C)=O c1(C(=O)NC23CCC(C2)N(C(=O)C=CC2CCC2)C3)ccc2n[nH]cc2n1 C(=O)(N=c1[nH]c(Br)ncc1N1CCCC1)c1ccc(C=Cc2n(C)ncc2)cc1 C1(CC(=O)NC(c2cnns2)(C)C)CCC(NC(C2(C)CCNC2=O)=O)CC1 CC1(C(=O)NC2CC(O)CN(C(=O)CC3=CCCC3)C2)CCC(=O)NC1 Cc1n[nH]c(C)c1C(N1CC(C(N)=O)(CNC(C2CC(C)N(C)C2)=O)C1)=O C(=O)(C1=CS(=O)(=O)CCC1)N1CCC(C)(NC(COC(CC)(C)C)=O)CC1 N1(C(c2ccn(CCNC(C(c3ccnn3C)C)=O)c2)=O)CCOCC(C)(O)C1 c1(C(N2C(CNC(C(C)CCO)=O)CC3CC32)=O)cnn2c1OCCC2 N1(C(COC(CC)C)=O)CC(NC(C2(O)CCSC2)=O)C(C)(C)C1 C1(CCC(=O)NC(C)CCNC(C2CNC(=O)C2)=O)CCN(C)CC1 C1(NC(C(=Cc2cccnc2)C)=O)CN(C(c2nc(=N)cc[nH]2)=O)CC1(C)C C(=O)(C(F)C(C)CNC(c1cccn1C1CC1)=O)N1C(C)CC1 CC1(C)CCN(C(=O)C=CC2CC2)C1CNC(C1OCCO1)=O N1(C(c2cccc(C)n2)C(=O)NC2(C)CC2)CCCCC(CO)C1 C1(C(=O)NCc2cc(C)ns2)CC(O)C(O)CC1CNC(=O)C(C)(C)C(C)O C(=O)(CCCCC(C)(C)C)N(C(C)C(=O)NCC=C(C)C)CCC C1(C)(NC(c2nc(C(C)OC)sc2)=O)CCCN(C(=O)CN2CCCNC2=O)C1 C(=O)(C(F)CC(C)(C)C)NC(CC(=O)N(c1ccc(O)cc1)C)C1CC1 c1(-n2c(C(CCC3CCCC3)NC(C)CC(=O)O)nnn2)cccc2cccnc12 C1(C(=O)NC(C=C)C2CCC2)C2CCCC1NC2 Cn1nc(C(N2CC(O)(C3CCCN3C(=O)CSCC#N)C2)=O)cc1C(C)(C)C C1(N(C)C(C2CCCCC2)=O)CC2CCC(C1)N2C(=O)Cc1ccno1 C=CCC(C)(C)C(=O)N1CCN(CC(N2CCC(C(=O)NC)C2)=O)CC1 c1(NC=O)ccc(CC(=O)NCC(CNC(=O)Cc2ccc(F)cc2)CO)cc1 c1(C(=O)NC2(C)CCCN(C(C(C(C)C)=O)=O)C2)cnc2[nH]ccc2n1 c1(N2N3CC(C(C)C3)NC(=O)CC3CC2C3)c(C)cc(C)cc1N.C(C)(C)(C)CC C(=O)(C(C)CCC(C)(C)C)N1CCC(C)C(Nc2cc([N+](=O)[O-])ccc2N)C1 Cc1csc(C=CC(=O)NC2CC(NC(=O)CCCN3C(=O)CCC3=O)C2)n1 c1(C(=O)NC(C)(C)CNC(=O)CCC2CNC(=O)N2)cc(F)c(O)c(Br)c1 N1(C(c2c(CC)sc(=N)[nH]2)=O)CCC(F)C(NC(c2ccn(C)c2)=O)C1 N#CC1C2CCC1CN(C(c1sccc1CNC(C1CCCO1)=O)=O)C2 C(=O)(C1=C(Cl)CCC1)NCCCN(C(C1CCN(CC(F)(F)F)C1)=O)CC C1(C(N(C)CC2CCCN(C(c3csc(S)n3)=O)C2)=O)CCCC1S(C)(=O)=O Cc1cc(C(N2C(C(=O)O)CC2C)=O)on1.C(=O)NOC1CCC1 N1(C(c2cc(C)[nH]n2)=O)CC(CNC(c2cnn(C3CCC3)c2)=O)CC1(C)C c1(N(C(C)C)C)nc(=NCCCNCc2ccccn2)[nH]c2c1CSC2 N1(C(C)=O)CCOC2(CCN(C(C3CN(C)C3)=O)C2)C1 c1(C(N2CCN(C(C(CCN(C)C)O)=O)CC2CCO)=O)ncc(C#N)cc1Cl C(=O)(CC(C)C(=O)N(C(C)(C)CC(=O)NC(C1CC1C(=O)OC)C)C)OC C1(C(=O)NCC2(C(C)(C)C)CCN(C(c3cnco3)=O)C2)CC2(CCCCC2)C1 C1(CN(C(c2cnc(N(C)C)o2)=O)CC)CCCN1C(C1CC1C(C)(C)C)=O N1(C(C(C)N(C(C)=O)C)=O)CCC2CCCC12C(N1CCC(F)(CO)C1)=O n1(CC(N2CCCC(CN(C)C(C3CCC(=O)N3)=O)C2)=O)cc(F)ccc1=O CC(C)S(=O)(=O)N1CCN(C(c2ccc(Br)cc2)C(=O)NCCC#N)CC1 C12(O)CCN(C1)C2=O.C1(N(C)CCO)C2CN(C(C)CN3CCCCC3)CC12 C1(C(=O)NCC(CNC(C=C(C)C2CC2)=O)O)CCc2cccc(F)c2O1 Nc1nc2c(cc1COCC(N1CC(O)(c3cn(CCCO)nn3)C1)=O)CCC2 C1(C(N(CCC(F)F)C)=O)CCN(C(C2CCNC(=O)C2)=O)C12CCC2 C(C#Cc1ccccc1Cl)NC(C(C(C)(C)C)NC(C1C(C(=O)OC)C1)=O)=O C(=O)(CCC(F)F)NCC(CCOC)NC(=O)C(F)(F)c1cncs1 C(=O)(C1=CCN(C(=O)CC2CCC(=O)C2C)CC1)NCC(C(=O)OCC)O C1(C(N2CCCC(NC(C(C)(CO)NC(C)=O)=O)C2C)=O)CC2(C1)CC(C)(C)C2 c1(C(N(CCC(C)NC(C23CC(C)(C2)C3)=O)C)=O)cccc2nonc12 N1(C(c2[nH]nc(OC)c2Cl)=O)CCC2(CC1)CC2CNC(=O)CC1CC1(C)C C(=O)(C1=NOC2COCC12)N1CC(C(NOC(C(=O)OC)C)=O)C2(C1)CC2 n1(C(C)CN(C)CCc2ccccc2)cnc2c(C(O)C(C)C)ncnc12 N1(CC)CCN(C(=O)C(C2CCC2)NC(c2ccc(=N)[nH]c2)=O)CC1=O C1(CC(=O)NC(CC)CN(C(=O)C(=O)NC2CC2)C)CCCCO1 Cc1ccc(C(=O)NC2CCCN(C(C)C(=O)NC3CCOC3)C2)cc1Br N1(C(c2n[nH]cc2Cl)=O)CC2CC1CCN2C(C1CC2(CCC2)CO1)=O C1(OCC)(CNC(=O)C(Cc2cnc[nH]2)SC)CN(C(=O)CN2CCC(C)C2)C1 CC(C)C(CNC(C1CCCCN(C)C1=O)=O)N=c1ncc2ccccc2[nH]1 C1(COC)(NC(=O)CCC2CC2CC2CC2)CN(C(=O)CC2CCCOC2)C1 N1(C(CSCCOC)=O)CCC(NC(=O)CCOc2cccc(Cl)c2)C12CC2 CC(C)C(O)C(F)(F)C(=O)NC1CN(C(c2ccc3c(c2)CCN3)=O)CC1(C)C c1(CN2CCC(CC(=O)OC)C2)ccc2c(n1)NCCC2.c12ccc(cc1)[nH]2 c1(C(N2C(CNC(C(c3scc(C)n3)(F)F)=O)CC2)=O)cc([N+](=O)[O-])c(C)s1 Cc1ccc(C(CNC(=O)C(O)C2CCCC2)NC(c2cnc(C)[nH]2)=O)cc1 C(=O)(C(C(=O)NC1CCC(C(=O)NOC(C)C)CC1)OC)OC C(=O)(C1=NOC(C)(C)C1)NCC(C1CCCCC1)N(C(=O)CC1CCCN1C)C N1(CC(N2CC(C)C(CCNC(=O)CN(C)C(N)=O)C2)=O)CCCCS1(=O)=O c1(C(=O)NCC2N(C(C(c3ccccc3)C)=O)CC2)ccc(C(N)=O)cn1 C(=O)(C(CC)C(=O)NC(CO)C(C)NC(c1cc(F)ccc1C(C)C)=O)OCC c1(N2CC(C)OC(C(N)=O)C2)ccc(S(=O)(=O)N2CCS(=O)C(C)C2)cc1Cl C1(NC(C23OC(C)C(C2)C3)=O)CCCC(NC(=O)C=Cc2cnn(C)c2)CC1 C(=O)(C1Cc2ccc(Cl)cc21)NCCC(C)(C)NC(c1cn(C2CC2)cn1)=O CN1CCC(C)(C(=O)NC2CCCN(C(c3cnn(C4CC4)c3C3CC3)=O)CC2)C1=O c1(C(=O)NC2CCC(NC(CC=CC=C)=O)CC2)cc(C(F)F)ccc1Cl CCCCC(CNC(=O)C(O)C(F)F)NC(=O)C(C)(C)CC1CC1 c1(C(=O)NCCC2(O)CN(C(CC3C(CC)C3)=O)C2)cc(C)ccc1S(N)(=O)=O n12cc(cn1)NC(=O)C2.C1(CCC(=O)OC)CCN(C(=O)CC2CCCC2)C1 O=S(=O)(c1ccc(NCc2ccco2)c(Cl)c1)N1CCC1CF c1(CCC)noc(CCCC(=O)NCCC(O)CNC(C2CCSC2)=O)n1 N1(C(CCC2CCCN(C(CC3CCCN(C)C3)=O)C2)=O)CC(C2=NOCC2)C1 c1(C(N2CCC(N(C(=O)C(O)C(C)CC)CCC)C2)=O)ccnc2ccccc12 c1(C(N2CCN(C(C)(C)C)CC2)=O)ccc2[nH]nc(-c3cn[nH]c3)c2c1 N1(C(=O)CCC2CCOC2)CCN(C(=O)COc2ccc(Cl)c(Cl)c2)CC(CO)C1 N1(CC(CCC)NCC(=O)Nc2nc(C)ccc2I)C(=O)c2ccccc2C1=O C1(NC(C=CC(C)NC(c2c(CC)cno2)=O)=O)CCCCC1(F)F N1(C(C2(C(C)C)CC2)=O)CCC2CCN(C(=O)CC3CCC(=O)N3)C2C1 C1(NC(C(C)n2ccnc2)=O)CCN(C(=O)CCc2cccs2)C1C(C)(C)C C(=O)(C1=NNC(C(F)F)C1)N(CCC(=O)NC1CCOCC1)CC C1(C(=O)NC2CN(C(c3cnc(CC(C)C)s3)=O)C2)CCc2nnc(O)cc2C1 N1(c2cc(C)c(Cl)cc2)C(=O)NC(c2ncco2)C2=C1C1(CCSC1)NC2=O CC(C(C)C(=O)N1CCC2(CC2)C1)NC(=O)CN1CC2CC2C1 C1(CNC(c2cc3c[nH]cnc-3n2)=O)CC12CCN(C(c1coc(Cl)n1)=O)CC2 c1(CC(=O)N(CCNC(C2(OC)CCC(C)C2)=O)C(C)C)n[nH]c2c1CCCC2 c1(C(=O)NCCCOCCNC(CC(C(CC)C)O)=O)cc2cc(Cl)ccn2n1 C#CC1(C(=O)NCC2CC3CC3C2)CN(C(=O)C(C2CCCCC2)C)C1 n1(CC#C)c(C)cc(C(=O)NC2COCC2NC(C2CC2C(C)(C)OC)=O)c1C N1(C(C2(C)CC=C(C)CC2)=O)CC2(CCN(C(c3c(C)cncc3C)=O)CC2)C1 N#Cc1sc(=NC2CC2c2ccc(F)cc2C(F)F)[nH]c1Cl C1(CCNC(C(CC#C)O)=O)CN(C(=O)COC2CCCC2)CC(C)O1 c1(CC)c[nH]c(C(=O)NCC(C2CCCN2C(=O)C=C2CCN(C)C2)(C)C)c1 S(=O)(=O)(CC(=O)NC(CCNC(=O)CC1CCCC12CC2)C(C)C)NC CC1CC2CCC(C(=O)NCCC3CSCCN3C(=O)Cc3cc[nH]c3)CN2C1 c1(NC)nc(C)ccc1C(N1CCC(NC(=O)C(F)(F)C(O)C2CC2)CC1)=O C12(NC(CCSC)=O)CCCC1N(c1nnc(O)s1)CC2.C1(=O)CCC1=O.OC N1(C(COCC(=C)C)=O)CCC(CC=C)(NC(c2nsc(OC)n2)=O)CC1 C1(O)(CNC(C2(SC)CC2)=O)CCCN(C(c2ccnn(C)c2=O)=O)CC1 C1(C(CO)NC(COCCC)=O)CCN(C(c2cc(OC)cs2)=O)CC1 c1(NC(C2CC(NCc3c(C)cc[nH]3)C2)=O)cc(Cl)ccc1C#N C1(NC(c2ccnc(F)c2)=O)CC12CCN(C(c1cnc(OCF)cn1)=O)CC2 C1(C(N(CCCNC(CCN(CCCCC)C)=O)C)=O)Cc2nn[nH]c2C(C)C1 C=CC(C)(O)CC(=O)NCC(CCC)C(=O)N1CCOC(C(N)=O)C1 C1(C(N2C3C(NC(c4c(CC)n(C)nc4)=O)CC(C3)C2)=O)CCn2ccnc2C1 C=C(Cl)CC(C(=O)N1CCCC(C(C)C)C1)NC(c1sccc1NC)=O C1(C(=O)NC)C=CCN1C(C1CCCC1CNC(=O)CCc1nncs1)=O C=C(C)CC(C(=O)NCc1cc(C)n(C)n1)NC(=O)Cn1cc(Cl)cn1 CC1CCC(CNC(C2(C3(O)CCC3)CC2)=O)CN1C(=O)Cc1cnn(C)c1 Cc1cc(N)c(C)nc1C(=O)NC1CCC(O)CN(C(=O)CC2CCOC2)C1 N1(C(c2c(C)cc(C(=O)OC)o2)=O)CC2=C(C1)CN(C(=O)C=Cc1ccc(C)s1)C2 N1(C(c2cccc(CCC)c2)=O)CC2CCC(NC(=O)CC3(C4CC4)CC3)(C2)C1 c1(C(N2CC(CC)C(NC(c3cnccc3C)=O)C2)=O)cnc(O)c(Cl)c1 CC1CC=C(C(=O)NC2CC(C)(C(N3CCOC(CO)C3)=O)C2)CC1 CC1CCc2nc(C(N3CCCC(NC(C45CC6CC4C5C6(F)F)=O)C3)=O)cn2C1 Cc1ccc2c(c1)CC(C(=O)Nc1c(C)nc(-c3cnn(C)c3)nc1C)CO2 C(CCC(C(=O)NCC(=O)N(C)C1CC1)NC(c1cc(C#N)c[nH]1)=O)OC C1(COC)(CNC(c2[nH]ccc2CO)=O)CCN(C(c2[nH]ncc2C#N)=O)CC1 c1(C(N2CC(NC(CC(=O)NCC#C)=O)C2)=O)cc(N)ccc1O c1(OC)ccc(Cl)c(OC)c1C(=O)NCCC(C)N(C(=O)CC1CCCC1)C C(=O)(C1Cc2ccccc21)NCC1N(C(c2c(C)cc(N)cn2)=O)CC1 c1(C(=O)NCCN(C(c2c(C(=O)OC)ccnc2)=O)C)noc2c1CCCC2 CC(c1cccnc1)=CC(=O)NCC(C1CCCCC1)NC(=O)CC1(C)CCCO1 c1(CNC(=NC)NC2CC3(CCC3)C2)cccc(C2COC2)c1 C(CC(C(C)(C)C)NC(=O)CC1CCOC1)N(C)C(C1CN2CCC1CC2)=O C1(CNC(C(CC)NC(C)=O)=O)CCCC2CN(C(=O)CC(C)(C)O)CC12 N1(C(COCCSC)=O)CC(NC(=O)Cn2cc([N+](=O)[O-])cn2)CC(F)C1 O=C(C1=CCCCC1)NCCCCNC(=O)C(c1c(F)cccc1F)(F)F O=C(CCC1CCN(C(c2ccncc2)=O)C1)NOCc1cnsc1 c12ccnc(c1)CC(=O)N2C1CC2CNC1C2.C=CCCC(=O)OC C1(F)(CNC(=O)CC2CCOC2)CCN(C(C2(O)CCSCC2)=O)CC1 C(=O)(CCC(C)(C)NC(C1CC1(F)Cl)=O)N(C)CC1CCN(C)C1 C1(C(=O)NCC2C(NC(c3c(O)nc(CC)c(C)c3)=O)C2)Cc2cccc(F)c2O1 C(=O)(CCCCC(F)(F)F)N1CC(CC(C)NC(CCC(CC)C)=O)C1 CC1C(NC(c2cc[nH]c2)=O)CCCN1C(=O)Cc1c(Cl)cccc1Cl Cc1sc(Br)nc1C(N1CCC(NC(=O)Cc2nnc(O)s2)CC1)=O C1(CNC(CCCCCC)=O)CC2(CO1)CN(C(=O)C(CCC)NC(C)=O)C2 N1(C(c2cc(C(=O)OC)c(F)cc2)=O)CC(C)N(NC=O)CC1C N1(C(C(C)C(=O)N(CC(C)C)C(C)C)=O)CC2C(C1)C2(F)F c1(C(=O)NCC(CNC(C2CCSC2)=O)OC)cncc2nc[nH]c12 Cc1csc(C(=O)N(CC(O)CN(C)C(C2CC23CCC3)=O)C)c1Br C1(C(C)C)(C(=O)NCC2(C)CCCC2)CCN(C(c2ccon2)=O)C1 c1(C(N2CCC(C)(CNC(=O)C=Cc3ccccn3)C2)=O)cc2n(n1)CCCO2 C1(CNC(C2C(C)(CC)C2)=O)CC(C)(C)CCN1C(=O)CC1CCC2(CC1)CC2 c1(C(=O)NCC(C)NC(C2CC3CCC2O3)=O)csc2cc(Cl)cnc12 c1(C(N(C(CCNC(c2cnc(C(C)C)[nH]2)=O)C)C)=O)ccc2cccnc2c1 CC1CN(C(c2cc(CNC(=O)CCc3nncs3)nn2C)=O)CCC1O c1(NC(C2CN(Cc3ccc(O)cc3Cl)CCC2O)=O)ncc2[nH]ncc2n1 Nc1ccc(C(=O)NC2CC(CNC(c3cc4sccc4s3)=O)C2)nc1F C1(C(N(CCNC(COCC)=O)C2CC2)=O)C2CCC1(c1ccccn1)C2 C(=O)(C1CC=Cc2ccccc21)NC(C)CCNC(=O)CC(C)(F)F C1(C(C)(C)C)CCCC(CC(N2CCC(c3cn(Cc4ccccn4)nn3)C2)=O)C1 CC(CCC(C)(C)C)C(=O)NC1(C)CCN(C(c2cnn(-c3cccnc3)c2)=O)C1 N1(C(C(C)C2CCC2)=O)CC2(CNC(=O)C=Cc3ccsc3)CC1CO2 N1(C(c2c(C)nn[nH]2)=O)CCOC(CCCNC(C2CCCN2C)=O)C1 c1(C(N2C(CC(=O)N(C(C3CCCO3)C)C)CCC2)=O)ccc(O)cc1 C1(NC(CC=C=C)=O)CC(C)N(C(=O)C(=O)Cc2cccc(OC)c2)C1 c1(CCC(=O)N(CC(C2CCC2)C2CCC2)CCO)cc(Cl)no1.C(=O)C(F)F Cc1cnc(C(N2CC(C)CCC2C(=O)NCc2csc(O)n2)=O)c[n+]1[O-] N1(C(c2nc(CCC)oc2)=O)CC(CNC(C2(CO)CC2(F)F)=O)C2(CC2)C1 N1(C(Cc2c(C)ocn2)=O)CCCC(CN(C)C(C2COC(=O)N2)=O)C1 O=C(CC1OCCc2sccc21)NCC12CC1CN(C(=O)CSC(F)F)C2 CC1=C(c2cc(CNC(c3nn[nH]n3)=O)c3[nH]ccc3c2)CCCC1 CCC(C)(C)C(C)CC(=O)NCCCN(C(=O)CC(F)F)C1CCCC1 CC(C(=O)N1CCC(CF)(NC(=O)CC2CN(C)C2)C1)S(N)(=O)=O N1(c2n(CCOCC)c(C3CCC(=O)N3)nn2)CCCc2cccnc21 N1(C(C(c2cn(CC)nc2)=O)=O)CC2CCN(C(c3cn(C)nc3SC)=O)CC12 CC(CC(C)N=c1ccn2ccnc2[nH]1)NC(C1CCCS1(=O)=O)=O c1(C(=O)NC(CC)CNC(=O)C(C)Cc2cnco2)cccc2nonc12 CC(CNC(=O)CC1C=CCC1)C(=O)NCC1(O)CC(O)C1 N1(C(=O)C2=CCN(C(=O)C=Cc3ccsc3)C2)Cc2cccc(F)c2C1 Cc1cc(C)n2cnc(C(=O)NCC(=C3CN(C(=O)COC(F)F)C3)F)c2n1 CC1CN(C(=O)CN2CCCNS2(=O)=O)CC(C)CN1C(=O)C=Cc1cscn1 C(c1ccsc1Br)=CC(=O)NC(C)CCN(C(=O)CCc1cnco1)C Cc1n[nH]c(C)c1CC(C)C(=O)NC1CC1CNC(c1cc(Br)cn1C)=O C1(NC(C(CC=C)CC)=O)COC2(C1)CN(C(c1ccc(OC)c(CC)c1)=O)C2 C1(C)(C(=O)NCC2CN(C(C(CC)OC)=O)CC2C)CCCNS1(=O)=O c1(C(=O)NC(CNC(CCCNC(=O)NCC#C)=O)C)ccc2nc(O)[nH]c2c1 C(CC1=CCOCC1)NC(C1OCCCC1(C)C)=O.c12nc(co1)C(=O)NC2C N1(C(c2c(CC)oc(C)c2)=O)CCC(C)C(CNC(=O)COC2CCC2)C1 N1(C(CN(CC(C)(C)C)C)=O)CCC(NC(C2(O)CCOCC2)=O)C(F)C1 c1(CCC(=O)NCC2(NC(C(c3ccccc3F)C)=O)CCC2)ccnc(Cl)c1 C12CN(CC1C)c1nnnn1C2.c1(CN(C)CC)c(C)noc1C c1(C(=O)NC(C2CCN(C(=O)C(C)n3ccnc3)CC2)C)cnc(N(C)C)c(Cl)c1 CP(C)(=O)c1sccc1C(=O)NC1CC(NC(=O)CCc2ncc[nH]2)C12CCC2 C=C(C)CCCC(=O)N1CCC(C(=O)NCCN(C)OC)CC1CC c1(C(=O)NCC2C(NC(=O)C=CCO)C2)cccc2c1CCC(=O)N2 n1(CCOC)cc(C(=O)NCC(C)(C)NC(C23CC(F)C2C3)=O)nn1 CC1CN2CCN1CC2C(N1CCC(C(C)NC(C2(CC3CC3)CC2)=O)CC1)=O Cc1nn(C)cc1C(N1CCC(NC(=O)C(C)NC(=O)C(C)(C)C)C1C)=O C1(C(N(CCC)CCNC(=O)C(c2ccc(F)cc2)=O)=O)CC2CC1C1CC21 c1(C(N2CC(OCC)C(CNC(C3CCCC3(F)F)=O)C2)=O)ccc(F)c(Cl)c1 c1(CN(CC(=O)Nc2ccc(OC)cc2)C)ccc(F)c(Br)c1 c1(C(=O)NC2C(CNC(C3(CC)CCOC3)=O)CCC2)cc(O)nc(Cl)c1 Cc1cc2cc(-c3ccc(C4CCCN4)cc3)ccc2nc1C(c1ccsc1)=O Cc1noc(C)c1CC(N1CCOC(CNS(=O)(=O)CC2CC2)C1)=O c1(C(N2CC(CC)N(C(=O)C(C)n3ccnc3)CC2)=O)cccc2nn(C)cc12 N1(C(C)=O)CC(C)(CO)CC1(C)C.C(CCC(=O)NC1=CCC1)OCCC N1(NC(CSc2ccc(NCC)cc2)=O)C(=O)NC(C)(c2ccccc2)C1=O c1(C(=O)NCC2CC(NC(COC3(C)CCC3)=O)C2)cnc2scnc2c1 C1(C(=O)NCCCCCCNC(C=CC(C)(C)SC)=O)CC(C(C)C)=NO1 C1(CNCc2cncc(-c3cccc(C)c3)c2)N(C)CCCC1(C)C C(=O)(CCCC(=O)NCC1CN(C(C2(C3CC3)CC=CC2)=O)CC1(C)C)NCC Cc1ccc(Cl)c(F)c1C(=O)NC1CCC(N(C(=O)CS(=O)(=O)N(C)C)C)CC1 C(=O)(C1=CCCCC1C)NC(CN1CC(NC(C(C)OC)=O)C(C)(C)C1)=O C(=O)(C(C)(C)C(=O)NC1CCCN(C(C2CCN(C)S2(=O)=O)=O)C1)N(C)C N1(C(CC(C)C(=O)OC(C)(C)C)=O)CCC(C2CCC2)C1 c1(C(=O)NCC2C3CN(C(c4c(CCC)n[nH]c4)=O)CC32)ncc([N+](=O)[O-])n1C N1(C(CNC(=O)OCC=C)=O)CCOCC1CN(C)C(c1cccnc1C)=O c1(C(=O)NCCC2CCC(NC(=O)CCC3CC3)C2)cccc2c1CCCC2=O S(=O)(=O)(c1cccc(F)c1)NCCNC(=O)NC1(NC(=O)NC)CCCC1 CC(C(C)(C)NC(c1c[nH]nc1C1CCCO1)=O)NC(c1cocn1)=O C1(NC(c2nc(C)sc2)=O)CN(C(=O)C(C)N(C)Cc2ccccc2)CC1O C1(NC(=O)Cc2n[nH]cc2Br)CC2(C1)CC2NC(c1ccns1)=O C1(CNC(C2(C=C)CC2)=O)CC(C(C)(C)C)CCN1C(=O)C=Cc1ccco1 c1(C(C)C)ccc(NC(c2cn(CCNC(=O)C(N)=O)nn2)=O)cn1 Cc1ccnc(O)c1C(=O)NC1CCC1C(=O)NC(c1cscn1)C c1(CCCC(N2CCC(NC(CCC(CC)C)=O)CC2)=O)nc2ccccc2o1 c1(C(=O)NC(CN(C(c2cnn(CC)c2C)=O)C)C)ccc([N+](=O)[O-])c(C)n1 C1(C(N(C)CCn2cc(Cl)cn2)=O)CCCC(C(F)(F)F)N1 N1(C(CC(C)OC)=O)CCCC(C2(NC(=O)Cn3cc(Cl)c(C)n3)CC2)C1 C(=O)(C1=CCC2(COC2)OC1)NCC1CN(C(C=Cc2ccc(C)o2)=O)CC1O C(CC(=O)N1CCN(C(C2CCC3(CCC3)O2)=O)CC1)(C(N)=O)NC(C(C)C)=O C1(CNC(CSCCC)=O)CCC2CN(C(=O)C(O)C3CC3)CCC2C1 C(C(C)(C)C(=O)N1CCC(OCc2cn(-c3cncc(Br)c3)nn2)C1)SC CN1CC2CC1CN2C(C12CC1CN(Cc1ccccc1N1CCOCC1)C2)=O N1(C(c2c(CC#N)ccs2)=O)CC(CNC(c2nsnc2O)=O)C2CC12 C1(NC(COC(C)=O)=O)CCC(F)(CNC(=O)CN2CCCCC2=O)C1 C1(NC(C(CO)NC(C(C)OCCC=C)=O)=O)CC2(CCCCO2)C1 CC(CF)C(=O)NCC(c1ccccc1)NC(c1c[nH]c(SCCC(N)=O)n1)=O c1(C(N2CC(C(F)(F)F)CC(F)C2)=O)cccc2c1CCC2.c12ccsc1CN2 n1(CCC(=O)NC(C2CCN(C(=O)Cc3ccccc3Cl)C2)C)ncn(C)c1=O c1(C(N(C(C2CCN(c3nnc(CC(=O)OC)s3)C2)=O)CC)C)ccc(Cl)s1 C(=O)(CC(F)(F)C(C)C)N1CCN(CC(N2CC3(C2)CN(NC(C)=O)C3)=O)CC1 N#Cc1c[nH]c(C(N2CCCC(C3CCCCN3C(C34CC(C3)C4)=O)C2)=O)c1 c1(C(=O)NCc2ncoc2CCNC(c2coc(Cl)c2)=O)cccc(F)c1F CCC1=CCN(C(=O)C2=NOC(CNC(c3cc(OC)n[nH]3)=O)C2)CC1 c1(CC)cccc(C(=O)NC(C)C(C)NC(c2ccc(CSC)o2)=O)c1F CC1=C(C(=O)N2CC(NC(=O)CCCc3nc(C)no3)C(C)C2)CCCC1 c1(C(C)C)ccc(NC2CCCC2C(=O)O)c(-n2ccnc2)c1 N1(C(C(C=CC)O)=O)CCC2(CC1)CN(C(c1cc(Cl)cc(Cl)c1O)=O)C2C(C)C n1(CC)nc(NC(C2CN(C(=O)Nc3ccc(CO)cc3)CCO2)=O)c(Br)n1 CC(F)(F)C(C(=O)NC1CC(CCNC(c2cc(Cl)n[nH]2)=O)C1)c1ccccc1 C1(CC(=O)NCCOC)CCN(CCOC)CC1.N12CC(C1)NC2=O N1(CC)CC(C(=O)NC2CCC(NC(=O)C(F)(F)C3(O)CCC3)C2)CCC1=O Cc1cnc(C(N2CC(CN(C)C(c3cc(O)cc(Cl)c3)=O)C2)=O)c(F)c1 C(CCC1CCC1)(C(=O)Nc1ccc(Cl)nc1)NC(=O)CN1CCSCC1 C1(OCC)CCN(C(=NCCNc2ccc(CC(C)C)cc2)NCC)CC1C Cc1cc(O)c(C(N2CCC(NC(=O)C#CC(C)(C)C)C2(C)C)=O)cc1F CC(CC(C)(F)F)C(=O)N1CCCN(C(=O)C=C2CCSCC2)C(c2cn[nH]c2)C1 C1(C(N(C(C)CCNC(=O)CCNC(C2CCOCC2)=O)C)=O)CCCN1C=O C(CC1=CCN(C(C2(CN(C)C)CC2)=O)CC1)NC(c1c(C)nn(C)c1Cl)=O C(C)(C)(CCN(C1CCN(CC(=O)NC2CCCN2C2CC2)C1)C)N(C)C N1(C(CNC=O)=O)CCC(NC(=O)Cc2cnc[nH]2)C1 C1(C(=O)NCC(CNC(CCc2onc(C)n2)=O)O)OCC2CCCCC12 n1(CCC)ccnc1CCC.C12(CCCC1)C1C(CC(=O)NCCN(C)C2=O)C1 N1(C(c2[nH]cc(CC)c2)=O)CCC2CCC(C1)N2C(=O)CC1CCC=CCC1 C(=O)(CCCCCN=[N+]=[N-])NCCN(C(C1N(C(=O)OC)CCC1)=O)C1CC1 N1(C(C(=O)NC(CC)C)c2cc[nH]n2)CCS(=O)(=O)C(C)C1 c1(C(=O)NC(CC=C)C(N2CC3(CCOC3)C2)=O)ccc(F)cc1C c1(C(=O)NCC(C)CN(C(=O)C(F)(F)c2cscn2)C)cnc(N)c(N)c1 C12(CNC(c3ccc(COC)s3)=O)CC(CCO1)N(C(=O)Cc1ccccc1)C2 CCC(C)C1C(=O)N(C)CCC(C(C)C)OC(=O)N1.C1(C(=O)NC2CC2)CCCO1 Cc1cc(F)ccc1S(=O)(=O)N1CCN(C(c2ccc3sccc3c2)=O)CC1C Cc1cc(C(=O)NC2CC(NC(C3CC(C)(C)C3)=O)C2)nn1C1CCOCC1 N1(C(c2c(CCC)nco2)=O)CCC(O)(CNC(c2nnn(C(C)(C)C)n2)=O)C1 C(=O)(C(C)(C)CCOC)N(C(C)CNC(c1coc(C(C)C)n1)=O)CC c1(C(N2C(C)CC(NC(=O)CSc3n[nH]c(O)n3)C2)=O)cn2cc[nH]c(=O)c2n1 C1(C(=O)NCCCCCCN(C(C(CC)(C)F)=O)C)Cc2ccc(OC)nc2N1 C1(C2(O)CCN(c3ncnc(Cl)c3CO)CC2)(NC(CC(COC)(C)C)=O)CC1 C12(C(=O)NCC(CNC(=O)CSC(F)(F)F)OC)CC(N=[N+]=[N-])C1C2 c1(C(=O)NCC2C(NC(Cc3cccc(C)c3)=O)CCCC2)cccc(F)c1Cl c1(C(N(c2nccc(C)c2)C)=O)cc(F)c(F)cc1Cl c1(CC)noc(CC)c1CC(=O)NCC1CCN(C(=O)C=CC(C)C)CC1 n1(CCCOC)nnnc1C(c1ncnn1C1CCC1)NCCCC1CC1(Cl)Cl Cc1ccc(N)c(C(=O)NCC2CCCC2NC(C2CCC(=O)N2)=O)c1F Cc1ncccc1-c1cccc(C(=O)C2CC2)c1.N1CCCC(F)CC1 C(=O)(CC(C)C(=O)N1CC2C(CN(C(=O)CC(C)(F)F)C)C2C1)OC C1(COC)CN(C(=O)C(C)(C)CNC(c2[nH]ccc2C)=O)CCO1 N1(C(C2C(C#C)C2(C)C)=O)CCN(C(=O)C=CC(F)(F)F)C(c2ccnn2C)C1 c1(CC(=O)NC(C)C(C)NC(c2cnsn2)=O)cc(Br)ccc1F C1(C)(CC(=O)NCC2ON=C(C)C2)CCN(C(C2CC(C#N)C2)=O)C1 C(CCC(C)(C)C(=O)N1CCCC(CCC(=O)NOC2CC3CCC2C3)C1)OC CC#CCCC(=O)NC(C)(CNC(c1ncccc1F)=O)Cn1cccn1 C(=O)(C(C)(C)CC#N)N(C1CC(NC(=O)C(C)(C)OC(=O)CO)C1)C Cc1c(C(=O)NC2CC3CC2N(C(C2CC2CF)=O)C3)cncc1Cl c1(OC)noc(C(N2CCCC(CNC(C3(c4ccccn4)CC3)=O)C2)=O)c1Br c1(C(N2CC(CCNC(=O)CC3(O)CCC3)OCC2)=O)cnc2c(c1)CNC2=O CC1(C)CCCN(C(=O)COCC2CCC2)C1CNC(=O)CC(F)(F)C(F)F C1(CNC(C(C)NC(=O)C2CC2)=O)CCN(C2CCN(C(=O)C=CBr)C2)CC1 CC(C(=O)NCCC1CC(NC(=O)Cc2cc(Cl)cc(Cl)c2)C1)C(C)C(C)(C)C c1(OCCC(=O)N(CCNC(c2ccccc2)=O)CCC2CC2Cl)ccccc1 CCCS(=O)(=O)C(C)C(=O)N1CCC(NC(=O)C2=CCCC2)C1C(C)C N1(C(C2CN(CCC)C(=O)C2)=O)CCN(C(=O)Cc2cncs2)CC1CO N1(C(c2nccn3ccnc23)=O)CCCC2(C1)CN(C(c1cc(=O)cc[nH]1)=O)C2 C1(CCOC)(NC(=O)CSc2cccs2)CCN(C(=O)CS(=O)(=O)NC)C1 c1(C(=O)NCCCCCCN(C)C(C2CCCOCC2)=O)ccc(C#N)cn1 CCCCCC(F)C(=O)N1CCCC1CN(C(=O)CCCCCF)C C1(O)(CNC(CCSCCC)=O)CCCN(C(=O)Cc2ccc(C)s2)C1 c1(C(N2CCC(N(C(=O)Cc3ccno3)CC#C)C2)=O)ccc(C(C)=O)cn1 c1(N2C(CC)CCC2)nnc(COC)n1CCCOCc1ccccc1 C(=O)(C(F)C(C)CNC(=O)C(C)N(C)C(C)=O)NC(CCSC)C N1(C(C(COC(C)C)NC(C)=O)=O)CCC(C(C)NC(=O)C(F)=C(C)C)CC1 CCC(CC(=O)NCCC1(NC(C2CCC3(CCC3)CC2)=O)CC1)C(C)C CC1(CNC(c2cc(CNC(=O)CC3CCSC3)on2)=O)CC=CCC1 C1(CNC(=NCCC=C)NCCC(=C)C)COC2(CCOCC2)O1 N1(C(C(CCC)n2ccnn2)=O)CC(CNC(=O)Cn2nnc(C)n2)C2(CC2)C1 O(C1CCc2cc(C(=O)N(CCCNC(C3CC3C)=O)C(C)C)ccc21)CC c1(C(N2CCCC(NCC3CC3)C2)=O)ccc2c3c(cccc13)CC2 CN=C(NCCCOc1nc2ccccc2s1)N1CCC(O)C1 c1(CNCC2CN(c3nc(C)c(Br)cn3)CC2F)c[nH]c2cccc(C)c12 Cc1cc(C)n(-c2ccc(NC(=O)C(=O)NC3CCC3C(=O)OC(C)(C)C)cn2)n1 N1(CC)CC(CC(C)(C)NC(=O)OC(C)CSCC(F)(F)F)CC1=O c1(-c2nc(-c3ccc(-c4c(O)cc(F)cc4)cc3F)on2)ccc2nc[nH]c2c1 C(CCCC(=O)N1CCN(C(=O)C(N)=O)CC1c1cn[nH]c1)(OC)OC c1(C(=O)NCC(CC(=O)NCCOc2ccncc2)OC)cnn(C)c(=O)c1 N1(C(c2nc(C)n(C)c2)=O)CCCC2C(NC(C3C4CCC3CC4)=O)C(C)(C)C12 [N-]=[N+]=NCCCCCC(=O)N1CCOC(CNC(c2cnc3[nH]cnc3c2)=O)C1 c1(C(=O)NC(CC(C)NC(=O)CCc2csc(=N)[nH]2)C)cnccc1C(N)=O c1(OCCNC(C2CN(c3nncs3)C2)=O)cc(Br)ccc1Cl N1(C(C2CC(CSC)C2)=O)C2CCC(C2)C1CC(=O)NOC(c1ccccn1)C Cc1cc(C#N)cnc1NC(=O)NCC1CC2(CC2)CO1 C1(CC(=O)NC2CC(O)(CNC(CCCOC)=O)C2)CCC(=O)C1C C1(C(=O)NC(c2cccs2)C)CCc2nc(NS(=O)(=O)c3cccs3)sc2C1 c1(C(N2C(CNC(CCC=C)=O)C=CC2)=O)cccc(CO)n1 CC(C)(C)C(O)CNC(=O)CC1(NC(C2CCC(=O)NC2)=O)CCCCC1 c1(CC)ccccc1N(C(c1ccc(OC)cc1)C(=O)NC1CC1)CC1CCC1 c1(SCC(=O)NCC2(F)CN(C(C(CC)F)=O)C2)ccc(C#N)cc1 C1(C(N2C(CCC(=O)NC3CC(O)C(O)C3)CCC2)=O)Cc2ccccc2C1 c1(OCCNOC)nc2cc(F)ccc2s1.C(=O)(C1C2CN(C2)C1=O)NCC.OC C=CC1(C(=O)N(CC(Cl)Cl)C)CN(C(=O)COCCCF)C1 c1(C(C(=O)NC2CN(C(CC3(OC)CCCC3)=O)C2)=O)ccc(F)c(Cl)c1 N1(C(c2ccn(COC)n2)=O)CCC2CCCC12C(=O)NC(CO)C1(C)CC1 c1(C(N(C2CCCC2)CCNC(C(C=CC)O)=O)=O)cnn(C)c1OC CCC(CC(=O)NCCC1CCN(C(C)C(=O)Nc2cccc(C)c2)CC1)OC C(c1cccs1)=C(C)C(=O)NCCOCCN(C(=O)C(C)=CC1CC1)C N1(C(C2CCC(CC)O2)=O)CCC(NC(=O)Cc2ccc(F)nc2)CC1 C(=O)(CC(F)(F)F)N1CCC(C(C)(C)NC(CC(=O)OCCC(C)C)=O)C1 Cc1cscc1C(N1CC(C(N)=O)(CNC(c2ocnc2C2CC2)=O)C1)=O C=C(C)CC(C)C(=O)N(CCCC(=O)N1CCOCC1)C.C12CCC1NC2=O S(=O)(=O)(c1cccnc1NCCC1CCN(C2COC2)C1)NC1CCC(C)(C)C1 c1(OCCC(=O)N(C(C)CNC(=O)CCC2CC(C)C2)CC)ccc(F)c(F)c1 N1(C(C(CC)=CC)=O)CCC(Nc2ncnc(Cl)c2F)CC(C)(C)C1 N1(c2nc(CC)on2)CCC(c2cc(C(N3CCNC(COC)C3)=O)n[nH]2)CC1 C1(CC(=O)NC(CCSC)C(=O)NCCC2(O)CCCC2)CCCC2CC12 C(=O)(C(C)(C)C(=O)N(CCCNC(C1CCN(C2CC2)S1(=O)=O)=O)C)NC CCC(CN1CCC1C1CCOCC1)CCC1CCCCC1 C1(CC(C)(C)C)CN(C(=O)C=CCO)CC1NC(=O)COC1CC1 N1(C(CC(C)SC)=O)CC2(CCN(C(=O)CC3CCCS(=O)(=O)C3)C2)C1 Cc1cc(Cl)cc(C(=O)N(CC(C)N(C(=O)C(C)C(F)F)C)C)c1C C(CN=c1nc(N2CCC(C#N)C2)c2c([nH]1)c(C)nn2C)c1c(C)cncc1 N#Cc1ccc(CN=c2cc(-c3ccccc3Cl)[nH][nH]2)c(Br)c1 C1(OC)CN(C(=O)CCCc2ncco2)CC1NC(c1cc(O)nn1C)=O Cc1ccc(C)c(C(=O)NCCC2CN(C(=O)C(C)N(C)C)CC2C)c1O C(C(C(F)(F)F)N1CCN(c2ccncn2)CC1)NC(=O)Cc1cccc(Cl)n1 c1(C(=O)NCCCCNC(C(COC)COC)=O)cnc2n1CC(C)CC2 c1(C(C)C)ncncc1C(=O)NCC(O)CN(C(C1CC1c1ccsc1)=O)C1CC1 C1(F)(CNC(C2CCC(F)(F)C2)=O)CCN(C(C2CC3CCC2C3)=O)CC1 C1(NC(C2(OC)CCOC2)=O)CC2CCC1CN(C(c1cc(C)[nH]n1)=O)C2 C1(CC=C)(NC(=O)Cn2nnc(C)n2)CN(C(c2coc(OCC)n2)=O)C1 C1(C(N2CC(CNC(C=Cc3cnc(C)s3)=O)C(C)C2)=O)CCOC2(CCC2)C1 CON1CC(C(=O)NCc2ccc(C(=O)N(C)C(C3CCCO3)C)s2)CC1=O C(=O)(CCCCn1ccnn1)NC1(CN(C)C(C2CC2C(C)(C)C)=O)CCC1 c1(C(=O)NCC(=O)NCC(N2CCC(C(N)=O)C2)=O)cnc2[nH]cncc1-2 c1(OC)c(C(N2CCC(CC3CC3)C2)C(=O)NCC(C)C)cccc1Br N1(C(COCCC)=O)CCC(CC(=O)NCc2noc(C)c2C)C1(C)C c1(OC)ccc(C(=O)CNC2CNCCN2Cc2cccc(F)c2)cc1Cl N1(C(C2(C)ON=C(C)C2)=O)CCC2CN(C(c3cnn(CCO)c3)=O)C2C1 C(=O)(CCCCCN(C)C)N(C)C1CC1.C1(CSC)CCN(C(CC)C(N)=O)C1 N1(C(c2c(CC)nn(C)c2)=O)CCCC(C)(NC(=O)CC2CCC(F)(F)C2)C1 C1(C(=O)NC2CN(C(c3c(CC)non3)=O)CC2C(F)(F)F)CCC(O)CN1C c1(CC(=O)NC(C)C(C)NC(c2cc(CF)on2)=O)cccc2cccnc12 C1(C(=O)NC2COCCC2C(N2CCC=C(F)C2)=O)(CC)CCCCO1 CCC(CCCC(=O)NCC1CCCCC12CC2)NC(c1ccc(C(F)F)o1)=O S(=O)(=O)(c1ccc2nc(Nc3nnc(CN(C)C)o3)sc2c1)N(CCOCC)C C1(NC(Cc2c(C)nc(S)s2)=O)CCN(C(C2(C3CCC3)CCC2)=O)CC(O)C1 c1(CCC(=O)N(CC(C)N(C(=O)CNC(N)=O)C)C)ccc(Br)cc1F c1(C2(C(N3CCC(CC)C3)=O)CC2)cccc(OC(F)(F)F)c1 c1(NCC(=O)N(CCC(C)NC(=O)C=CC(=O)NCCC)C)ncncc1Cl CC(C)C(O)C(F)(F)C(=O)N1CC(NC(=O)C(F)(F)C(C)O)C1 C1(NC(C(Cn2ccc(C)n2)C)=O)CC2(C1)CC1(CC(NC(=O)CC3CC3)C1)C2 C1(CNC(C2CCCN(C)C2)=O)CC2CCC1N(C(=O)C(c1ccccc1)O)C2 C1(C(NOCC(=O)NOCCF)=O)CC2(CC2)CO1 c1(C(=O)NC2C(NC(CNC(=O)OC)=O)CCCC2)c[nH]c2ncnc(O)c12 C1(NC(=O)CC2CSC2)CC2CN(C(C3COCCN3C3CCCC3)=O)CC2C1 c1(C(N2CCC(NC(C3C=CC=CC=C3)=O)(CF)C2)=O)cnc2c(n1)CCCC2 c1(CCC(=O)NC(C(=O)NCC2(C(N)=O)CC2)C2CCCO2)ccncn1 c1(C(=O)NC(CC)CNC(=O)Cc2ccc(C)nc2)ccc2nc(S)oc2c1 C1(NC(c2cn[nH]c2)=O)CC2CC1CN2C(c1cc(C2CCCC2)no1)=O c1(NC(N2CCC(O)(C(=O)NC(CC)C(=O)OC)CC2)=O)ccccc1[N+](=O)[O-] C(=O)(CCCCN=[N+]=[N-])N1CCC(N(C(c2nccc(OC)c2)=O)C)C1 c1(C(=O)NC2C3CC(NC(C(CC)(C)CC)=O)CC32)ccc2nnn(O)c2c1 C1(NC(C2(F)CN(C(=O)C3=COCCC3)C2)=O)CC(CO)C(O)C1O c1(C(=O)NCCC2CCCN2C(=O)CCc2ccsc2)noc2ccccc12 C#Cc1cnc(C(N2CCN(C(c3cn(C4CC4)cn3)=O)CC(O)C2)=O)c(C)c1 c1(C(=O)NCC2(CNC(C3(OC)CC3)=O)CC2(F)F)cc2c(ncn2C)s1 N1(C(C=CCC)=O)CCCC2C1CCCN2C(=O)CN1C(=O)C(=O)N(C)C1=O C(C)(C(=O)N1CCCC(N=[N+]=[N-])C1)(C(C)C)NC(C)=O CN1CCCC(O)(CNC(C2(C)CCC(NC(=O)CC34CCCC3C4)CC2)=O)C1 N1(C(C2C(=C)C2)=O)CCN(C2CN(C3(C(c4cc(C)sn4)=O)CCC3)C2)CC1 C(=O)(C(C)P(C)(C)=O)NCC1CCCN(C(CCCOCCOC)=O)C1 C#CCC(CC(=O)NC(C)(C)C#CCC)NC(=O)C(F)=CC1CC1 C1(NC(C2(F)CCN(C(C3C(CCOC)C3)=O)CC2)=O)CCn2cnnc2C1 C1(NC(c2csc(-c3ccoc3)n2)=O)CN(C(c2cnc[nH]2)=O)CC1F C(=O)(C(CCC1CCC1)N(CC#N)CCn1nnnc1SCCOC)NC Fc1ccc2[nH]cc(-c3cc(-c4nccn4CC4CC(O)(C(F)(F)F)C4)n[nH]3)c2c1 C1(C2(O)CCN(C(c3cccc4c3CCC4)=O)CC2)(NC(C2CN(C)C2)=O)CC1 N1(C(c2cc(C)oc2)=O)CCN(C2(NC(=O)C(F)Cc3ccccc3)CC2)CC1 c1(OC)cscc1C(=O)NC1COCC1C(=O)NCC(C)CC1CCC1 Cc1nnc2n1CC(C(N1CCOCC1CNC(c1cnccc1Cl)=O)=O)C2 CC1COc2ccccc2C1C(=O)NCC1CC(NC(c2cnc[nH]2)=O)C1 C(=O)(CC1=NN(C)C(=O)C1)NCC1CCC(C)N(c2cc3nncn3cn2)C1 c1(C(N(CC(=O)N(CCCO)CCC)C2CC2)=O)ccc(O)c(OC)c1 c1(C(N2CCCN(C(c3csnn3)=O)CC2CO)=O)c(F)ccc2occc12 C12(C(=O)NCC3C(C)CN(C(c4cnn(C)n4)=O)C3)CCC(C1)OC2C Cc1cc(C(=O)NC2CC(NC(c3csc(C(C)C)n3)=O)C2)no1 C1(C(=O)NCCN(C(C(Cn2cncn2)OC)=O)CC2CC2)CCC(C)(C)C1 N1(C(C(CSC)(C)C)=O)CC2CC(NC(=O)Cn3cc([N+](=O)[O-])cn3)CC1C2 c1(C(=O)NC2(CNC(c3n(CC)ccc3)=O)CC2)cc(C)c2ccccc2n1 CC(C)C(O)C(=O)N1CC(OC)CC1CCNC(C1(OC2CCCCC2)CC1)=O CC#CCCC(=O)NCC(C)CNC(c1csc(Cl)c1OC)=O N1(C(C(C)NC=O)=O)CC=CC1CNC(=O)C(=O)NCC(F)F CC1CCCN1C(=O)CCC1(NC(C2CC2C(F)F)=O)CCCC1 CC(CN(C)C(C1CNC(=O)O1)=O)C(=O)NCC1CCCO1 c1(C(=O)NC2CCN(C(CCN(C(CCC)C)C)=O)C2)ccc(=O)n(C(C)C)c1 c1(C(=O)NCC2(O)CCCN(C(C(CCCC)=O)=O)C2)c(F)ccc2c1OCC2 C1(C(N2C(C)(CCO)CC2)=O)CCNC(=O)C1.C1=CC(=O)NC1(C)C C1(NC(c2cc(C)no2)=O)CC(NC(=O)C(c2ccc(Cl)cc2)C)C(O)C1 C(=O)(C(C)S(N)(=O)=O)NC(C1(O)CCN(C(=O)COCC2CCCCCC2)C1)C c1(C2(NC(C3CC(C#N)C3)=O)CC2CO)cc(F)ccc1F C1(F)(C(=O)NCC2(C(N)=O)CN(C(C3(C)CCCC3)=O)C2)C2CCCCC12 C1(C(N2CC(C(=O)NCCSCC)OCC2)=O)CCOCC1(C)C C1(NC(c2c(C(=O)OC)c[nH]n2)=O)CCN(C(C2(c3ccno3)CC2)=O)CC1 c1(SCCC(=O)NC2CCN(C(C3C(C#C)C3(C)C)=O)C2)ccc(C)c(C)c1 N#Cc1ccc(S(=O)(=O)N2CCCC2Cn2cncn2)cc1NC(CO)CCF C12(CC(F)(F)C1)C(=O)N2.N1(CC)CCCC1C(=O)NCCCC=CC C1(C)CCN(NC(C2CC(C)(C)CCO2)=O)CC1C.c1(C(C)=O)cnc(F)nc1N C1(C(N2CC(C)(NC(C)=O)C2)=O)CCC(NC(C2CC(O)C(F)C2)=O)CC1 N1(C(C(=C)C(F)(F)F)=O)CC2=C(C1)CN(C(c1cccc(Br)c1OC)=O)C2 C1(CNC(C(CSC)C)=O)CC2(CCN(C(=O)CC(O)C(Cl)(Cl)Cl)CC2)C1 c1(OCC=C)ccc(Cl)nc1C(=O)NCC(C)NC(=O)C(C)S(C)(=O)=O C(C)(CCC(=O)NCc1ncccc1CNC(=O)C(C1CCCCCC1)F)OC N1(C(C(CCC)=CCC)=O)CC(CNC(=O)C2CC2)OC2(CCC2)C1 c1(COC)oc(C=O)cc1C.C(=O)(CC(C)(O)C1CC1)N1CCC(CCOC)C1 C(=O)(CCCC(F)(F)F)NCc1cn(CC(N2CCC(CC)C2C)=O)nc1 c1(C(N2CC(C)(NC(c3cc(C)cc(C)c3)=O)C2)=O)c(C)cc(F)cc1C C1(CC)CN(C(c2cc(Cl)ccc2C(F)F)=O)CCN1C(=O)C=CCN(C)CC C1(C(N(CC(C)NC(c2ncoc2-c2ccco2)=O)C)=O)CCOC2(CCC2)C1 C1(C(N2CC3C(N(C)C(c4cnc(CF)s4)=O)C3C2)=O)CC2CCCN2C(=O)N1 Cc1cc(F)cc2[nH]c(C(=O)NCC3(O)CN(C(C4COCCO4)=O)C3)cc12 C(=O)(CCC(C)(C)C)NC1C(CC)CN(C(c2cc(-n3cccc3)ccn2)=O)C1 c1(N2CCC(c3cc(C)on3)C2)nccc(=NCCCCCF)[nH]1 CCCC(O)(CCC)CC(=O)N1C2CCC1C(NC(=O)CC1CCSC1)C2 c1(OC)cc(O)ccc1NC(=O)C(Cc1ccco1)NC(c1ccon1)=O C1(C#CC(=O)N2CCC(O)(CNC(c3cc(C4CC4)ns3)=O)CC2)(CC)COC1 C(=O)(C(C)(C)CC(=O)N1CC(NC(=O)C(C)(C)C(C)C)C(O)C1)OC C(=O)(CCCC(C)C)NC1C(OC)CN(C(=O)CCCc2ccncc2)C1 C1(N2CCN(C(CC3(OC)CCC(F)(F)CC3)=O)CC2)CCCCC(C)(C)C1 c1(OC)cnc(Cl)cc1C(N1CCOCC1C(=O)Nc1nnco1)=O C(=O)(C(C)(C)COC1CC1)NC(c1ccccc1)CN(C(=O)C(F)=CCCF)C Cn1ccc(C(=O)NCC2(O)CC(CNC(c3ccccc3)=O)C2)n1 O=C(C#CC1CC1)NCc1ccc(CCNC(C2OCCC2C(F)(F)F)=O)cc1 N1(C(CNC(=O)OCC=C)=O)CCOC2CN(C(=O)CC3CC=CCC3)CC12 N1(C(c2c(C)cccc2)C(=O)Nc2ccc(OC(F)F)cc2)CC2CCC(N)C2C1 c1(CC(C)NC(=O)C(CNC(=O)CC=CC(C)(C)C)N(C)C)nncn1C C1(NC(CCC)C(C)CC)COC2C(SC)COC12 c1(C(=O)NCC2CCCCN(C(CC(C)C(F)F)=O)C2)cc2ccccc2n1C Cc1ccc2c(=NC3=CCC4(CC3)CC(O)C4)[nH]c(=NC3CCN(CCF)CC3)[nH]c2c1 CCC(C)CC(=O)NC1(CCNC(=O)C(C)C2CC2)CCC1 C(=O)(C(C)(CO)N(C)C)NCC(C(=O)N(C)CC)NC(=O)COCCCC(C)C C(=O)(C(CC(F)F)NC(c1ccc(C)cc1C)=O)N1CCCC(NC)C1 c1(C(=O)OC)cccc(C(=O)NCC2(N)CCC2)c1F CC(C)C(C)(CNC(c1ccccc1-n1ccnn1)=O)NC(=O)CCC1CC1C c1(C(=O)NCC(CNC(C(CC)(F)F)=O)(C)O)cccc2nonc12 CS(=O)(=O)CCC(=O)NC1CCC(Oc2cccnc2)C1 C(=O)(NNC(=O)N=c1nc(C2CC2)[nH]s1)c1c(Cl)ccc(SC)c1 C1(C2CCCC2)(C(=O)NCCN(C(C(C)CC(F)F)=O)CC2CC2)CCNC1=O c1(CC(=O)NCC2CC3CN(C(c4cnccn4)=O)CC23)cnc2cccnn12 CC(CCNC(=O)C=Cc1ncc[nH]1)CCNC(c1ccsc1C(F)F)=O C(C1CCCC1)=C(C(=O)NCCCN(C(=O)C(c1nncn1C)C)CC)C CCCCC(C)CCC(=O)N1CC(CNC(C2(CC)COC2)=O)CC(C)C1 c1(C(=O)NC(C2(O)CCN(C(C=CSC)=O)C2)C)cnc2[nH]c(C)nc2c1 c1(C(=O)NCCSC)ccc(CNC(=O)C(O)c2ccsc2)o1 C1(C)(C(=O)NCC2C(NC(C3(OC)CC(CF)C3)=O)CC2)CCCCC1 C(=O)(C1=CC2C=CC(C1)C2)N1CCC(CCC(N2CC(C)CC(OC)C2)=O)C1 C1(CNC(c2ncn(CC)c2)=O)CN(C)CCN1C(=O)CCc1cnc[nH]1 Cn1c(C(=O)NCCCNc2ccc(C(=O)O)cn2)nc2cc(Br)ccc12 C1(OC)(CNC(=O)C(C)N2CCC2)CCN(C(=O)Cc2cncnc2O)C1 C1(C(=O)NCC2(O)CN(c3ncccn3)C2)CCC=CCCC1 C(CCCCCC(=O)N1CC(O)(C(F)(F)CO)C1)c1cccc(OC)c1 N1(C(COCCC=C)=O)CC(C)N(C(=O)Cc2cn(C)nc2C)CC1C c1(C(=O)NCC2(C)CCN(C(=O)CCc3ccc(Cl)nc3)C2)cc2sccc2s1 C1(C(=O)NC(CCNC(c2c(C#C)cn(C)n2)=O)C(C)C)CCc2nn[nH]c2C1 N1(C(c2cccc(C(C)=O)c2)=O)CCC(NC(c2oc(C)cc2C)=O)C(C)(C)C1 C(=O)(C(F)CCCC)N1CCC(n2cc(CNC(c3c(C#C)c[nH]n3)=O)nn2)C1 N1(C(C=CC(C)C)=O)CCC2CCN(C(c3cc4c(nn3)CCCC4)=O)CC12 Cn1c(C(=O)N(C(C)(C)C)CCO)cnc1C(F)(F)F.N12CC3C(C3C1)C2=O C1(C(=O)NCC2(CCNC(C=C(CCC)C)=O)CC2)C2CCC(F)(F)C12 N1(C(C(CC)C)=O)CCC2CCN(c3ccc(C(=O)OC)c(C)n3)CC2C1 N1(C(c2csc3cccnc23)=O)CCC2(CC(NC(C3(O)CCC3)=O)CO2)C1 c1(CN2C(C(=O)NCc3cc(C)nc(Cl)c3)CCCC2)cnn2c1CCCC2 Cc1c(C(N2CCCC(N(C(=O)CC(C)CF)C)C2)=O)cc(C(C)C)n1C C1(C#N)(C(N2C(CCC(=O)NC3(C(C)(F)F)CC3)CCCC2)=O)CCCCC1 Cc1c(C(N2CCCC3C2CCN3c2nnc(C3CC3)o2)=O)cnc2nncn12 Cc1cnc2cccc(C(=O)NC3CCN(C(=O)Cc4cncs4)C(C)C3)n12 C(C)(C(O)C(=O)Nc1cccc(CNC(=O)Cc2cccnc2C)c1)SC C(=O)(C1CCCc2ccnn21)NC(CCNC(C(C)Oc1cccc(Cl)c1)=O)C C(=O)(C(C#N)CCc1ccccc1)NC(C1CCN(C(=O)CCCC(=O)NC)C1)C Cc1cc(C(=O)N(C(C)C(N2CCC(C(=O)N(C)C)C2)=O)C2CC2)c(C)[nH]1 C1(C(=O)NCC2=CCCN(C)C2)(NC(C(CC#C)C2CC2)=O)CCC(C)(C)C1 c1(CC(=O)NCC2CCN(C)C2c2ccc(Cl)cc2)cnc(N)c(N)c1 c1(C(C(=O)NCC(CC(C)C)NC(C=CC(CC)C)=O)C)cc(C)ccc1C c1(C(=O)NCC(C)CNC(c2cnnc(Cl)c2)=O)cc2c(nc1O)CCSC2 Cc1ccc(F)c(C(=O)NCCCN(C(c2scnc2Cl)=O)C(C)C)n1 N1(C(C(CCC)OC)=O)CC2CCC(C1)N2C(c1ccc(SC)s1)=O CC1CCc2[nH]c(=NC(C)C(F)F)nc(N3CCC4(CCC(=O)NC4)CC3)c2C1 CC(CC1CCC1)C(=O)NC(Cn1ccnn1)C(=O)NC1CC(C(C)C)(CO)C1 c12cc(cc(F)c1)Oc1c(Cl)ccc(c1)C(CC)(C)N2.C(COCC)(CF)OC C1(NC(C(C)C(F)F)=O)CCN(C(c2ncccc2N)=O)C12CC2 C(=O)(CC(=O)NCC1(C(=O)NCC(O)C(C)O)CCCO1)OC N1(C(C(C)(C)C)=O)CC(C2CCN(C(c3noc4cc(Cl)ccc34)=O)CC2)C1 c1(C(N(C)CCNC(C2COC3COCC23)=O)=O)cnc2ncc(Cl)cn12 Cc1cc(O)ncc1C(=O)NCC1(F)CC(NC(=O)C(C(C)O)N(C)C)C1 O=C(CCS(=O)(=O)C(F)(F)F)NC12CCCC1CN(C(c1ccc[nH]1)=O)C2 N1(C(C2N(C(C)C)CCC2)=O)CC(C)CN(C(=O)C2=CCOC2)C(C)C1 C1(CNC(c2c(C)scc2)=O)CN(C(=O)Cn2nccc2C)CC12CCOCC2 CC1(C)CC(CNC(C2(C#N)CC=CC2)=O)(NC(C2CC2c2ccco2)=O)C1 N1(C(C2C(C=C)OCC2)=O)CC(C)C(C)(CNC(=O)CCOc2cccnc2)C1 CC(C)(C)C(C)(O)C(=O)NC1CC(CNC(=O)CCc2cn[nH]c2)C(O)C1 C(=O)(C1CCc2c[nH]nc21)N(C(CC(C)C)C(=O)NCCc1cnn(C)c1C)C N1(C(C2CCC(N(C)C)C2)=O)CCC2(CCCC2NC(c2cnsc2)=O)CC1 n1(NC(C)CCCc2ccco2)c(C)cc(O)cc1=O.C12CCCN(C1)C(=O)N2 C1(C(N2CC(COC)C2)=O)C2Cc3cc(Cl)ccc3C12.[nH]1cc(-c2cscn2)nn1 c1(C(N(CCOCCNC(c2c(C)nn[nH]2)=O)C)=O)cnc2c(c1)NCC2 c1(CC(N2CC(C)(NC(c3ncccc3O)=O)C2)=O)ccnc(Cl)c1F C1(C)(NC(C(Cc2cc[nH]n2)NC(C2C(C)CC2)=O)=O)CCCC1(C)C C1(C(N2CCC(N(C)C(C3(CCF)CCC3)=O)C2)=O)(OC)CCSC1 CN1CCCCCC1C(=O)NCCCCCNC(=O)CN1CC=CC1 C1(SC(CCCn2cc(-c3c(C)nn[nH]3)nn2)=O)CCOC(C(C)(C)C)C1 CC(=O)CCCC(=O)N1CCC(NC(C2(CS(C)(=O)=O)CCC2)=O)C(C)C1 N1(C(c2c(C)scn2)=O)CCN(C(C2CCNC(=O)C2)=O)CC1c1ccccc1Cl C1(C)(CCCC)NC(=O)N(CC(=O)N(C(c2cccc(C#N)c2)CC)CC)C1=O C1(CCNC(c2cc(C3CC3)[nH]n2)=O)CCN(C(C2CCN(C3CC3)C2)=O)C1 C(=O)(C1=CCN(C)C1)N1CCC(NC(C(C)(C2CC2)OC)=O)C1 c1(C(=O)NCC2N(C)CCN(C(=O)CCS(C)(=O)=O)C2)cn2cccc(F)c2n1 c1(C(N2CC3C(NC(c4cscn4)=O)(CC3)C2)=O)c[nH]c2ccncc12 N1(C(C(C(C)O)C)=O)C2CCCC1CN(C(=O)C(c1cnn(C)c1)=O)C2 c1(C(=O)NCCCN(CCCNC(CC)=O)C)ccccc1C(F)(F)F N1(C(C(CCSC)N(C)C)=O)C2CCC1(CNC(C1CCC3CCC1O3)=O)CC2 C1(CNC(c2ccc(OC)nn2)=O)C2CCCC1N(c1nccc(CO)n1)C2 N1(C(c2cn(CC)nn2)=O)CCC(C(N2CC(OC)CC2C(=O)O)=O)C(OC)C1 C(CCCC#C)(c1nnnn1CC1CCCO1)NCCCC1(CC=C)CCCC1 N1(C(c2ccc(CO)o2)=O)CCN(C(=O)CC(c2cccs2)C2CC2)C2CCC12 c1(CN2CCC(CC(N3CCC(CNC(C)=O)C3)=O)C2)ccc(F)cc1Cl C(=O)(C(C(C)C)n1ccnc1)NCC1(F)CC(NC(CN(C)C(=O)C2CC2)=O)C1 N1(C(c2n(C)ccn2)=O)CC(C2CCN(C(=O)C=Cc3cncn3C)CC2)C1 C1(CC=C)(NC(=O)CNC=O)CCCN(C(=O)C(C)(C)CCc2ccccc2)C1 c1(OCC(=O)NC(C)CCN(C(=O)C(O)CF)C)ccc(F)cn1 N=c1[nH]c(C)c(C(N2CCC(CNC(C3CC(C(F)(F)F)C3)=O)CC2)=O)s1 c1(CCC(N2C(C(N3CCC(N(C)C)C3)=O)CC2)=O)cccc(Cl)c1 c1(C(=O)NCC(c2ccccc2)CNC(C2(N(C)C)CCCC2)=O)csc(Cl)c1 c1(NC(C2(OC)CC2)C)ncccc1S(=O)(=O)NC1CCC(N(C)C)CC1 C(=O)(C1CCCc2nn[nH]c21)NC1C(C)CCN(C(CN(C(=O)OC)C)=O)C1 c1(NCc2c(C)ccc(C(=O)O)c2)cc2c(cc1Br)OCO2 N1(C(c2c(C)ccnn2)=O)CCC(C(=O)N(CCCCCO)C)C(C)(C)C1 C1(C(N(CC(C)CNC(=O)CN2CCS(=O)(=O)CC2)C)=O)CC(=O)C12CCCC2 Cc1cc(F)cc(C(=O)N(CCCNC(=O)C=CC2CCC2)C)c1O C1(NC(C(CC)F)=O)CS(=O)(=O)C12CCN(C(c1cn(C(F)F)c(C)n1)=O)CC2 C12(CNC(C(C#N)C3CC3)=O)CCCC1CN(C(c1cc3scc(Cl)c3[nH]1)=O)C2 N(C1CCCc2ccoc21)C(C=CC(C)NC(C(CCCC)CC)=O)=O C1(NC(=O)CC2(O)CCOC2)C=CCCC1C(N1CCC(CCCO)CC1)=O c1(OCC)ccc(F)c(C(N2CC3CC3(CNC(=O)Cc3cccnc3)C2)=O)c1 C(=O)(C(C)(C)CCCNC(CC)C(N1CC2CC1(C(NC)CC)C2)=O)NC(C)=O c1(-c2cn(CCCCCC)nn2)cccnc1C#N.C1(C2CC(=O)N2)COC(C)C1 N1(C(c2ccn(CC)c(=O)c2)=O)CC2CCCC1C2CNC(=O)C(C)CO Cc1[nH]c(C)c(C(N2CCCC(CNC(=O)CC3CCOC3)CC2)=O)c1C Cc1cnn(CC(N2CC(O)(C(C)NC(C3CCC(F)C3)=O)C2)=O)c1 Clc1ccc2c(c1)CC(CSC1(c3ccccc3I)CC1)C2 c1(C(N2CC(Nc3ccnc(C)n3)C(C)C2)=O)cc2cc(Cl)ccc2[nH]1 C=CC1(CC(=O)NCC(C)CNC(=O)C(C)n2ccnn2)CCCCC1 c1(Nc2ccc(O)nc2)ncc(Cl)cc1F.C1(OC(C)(C)C)CC2C1NC(=O)N2 CC(=O)CC(C)(C)C(=O)NC1C(C(=O)NCC2C3CCCCC23)C1(C)C C(=O)(CC(O)CC(C)(C)C)N1CCCC(C(C(=O)N(C)Cc2nc[nH]n2)(C)C)C1 C1(C(=O)NC(C2CCN(C(CC=CC=C)=O)CC2)(C)C)CC2(CC(OCC)C2)C1 O=C(C1=C(Cl)CC1)N(C1CCCN(C(=O)Cn2ncccc2=O)C1)CCF N1(C(C(C)(C)CO)=O)CC2CCCC(C1)N2C(C12CCC(C)(C1)OC2)=O C(C1CCCCCC1)=CC(N1C(C2CCCN(C(CCOCC)=O)C2)CCC1)=O C1(CC)CC(C)CN(C(c2ccoc2CNC(=O)CCc2ccnn2C)=O)C1 c1(NC(C(C(C)OC)NC(CCCOC)=O)=O)cccc(C)c1O c1(NC(C(=O)NCC(CC)NC(=O)C(C)Cn2ccnc2)=O)ccccc1 c1(C(=O)NCC2CCN(C(=O)CCCCc3cnc[nH]3)C2)[nH]nc2cnccc12 C1(NC(=O)CCc2nncs2)CCOC12CCN(C(=O)C=CC1CCCO1)CC2 C1(C(N2CC(NC(C(C3CCOCC3)OC)=O)C2)=O)CCCSS1 C1(CNC(=O)CCOCC(F)F)CN(C(=O)C=Cc2cccs2)C2CC12 C12(NC(CCN(CCC)C)=O)CCCN(C(=O)CCn3cncn3)CC1C2 c1(N(C)C)ccc(CCC(N2CCC(CNC(c3cnc(O)o3)=O)C2)=O)cc1 c1(C(C(=O)NCC=C)N2CCC2c2ccc(OC)cc2)cc(Br)cc([N+](=O)[O-])c1 Cc1cccc(C(C)NC(c2cnc(CNC(=O)CCC3CCCO3)nc2)=O)c1 N1(C(C(C)(C)CC2CC2)=O)CC2CCCC(C1)N2C(c1ccc2c[nH]nc2n1)=O C=CCC(C(=O)NCC12CC1CN(C(=O)CC1CC(C)CC(C)(C)C1)C2)C(C)C c1(C(C(=O)N(CCCN(C(CCCC)=O)C)C)(C)O)ccc(F)c(Br)c1 C1(CC)(Nc2ncnc(CO)c2C)CCN(C(C2CCC(CC)O2)=O)CC1 CC(N=c1[nH]nc(C2CCCC2)s1)C1CN(C(=O)CC2CCCCO2)C1 C(c1cccc(Cl)c1Cl)=CC(=O)NC1CN(C(Cc2nnc(C)o2)=O)CC1C N1(C(C=CC=CCC)=O)CCCC(C(=O)NCC(C)(F)C(C)(C)F)C1C N1(C(C(C)C2CCC2)=O)CCCC12CCN(C(c1cncc(Br)c1)=O)C2 C(=O)(C(C)(C)CO)N(C1CCN(C(C2(C(C)(F)F)CCC2)=O)C1)CC C1(CC(=O)NCC(C)(C)NC(c2cnc(=N)[nH]c2)=O)CCCC(C2CC2)O1 Cc1cc(=O)ccn1CC(=O)NC1CC(NC(c2occc2F)=O)C12CCC2 C(C)(C)(CCCC(=O)NCC1CCC(C)(C)CC1)NC(CC1N(C)CC=CC1)=O C1(C(=O)NC(c2ccncc2F)C)C=CCCN1C(=O)CN(C)C(N)=O c1(C2CC(C)(F)C2)cccc(C(N2CCSC2)=O)c1 C1(CNC(C#CC(C)(C)C)=O)CCC2CN(C(c3ccncn3)=O)CC12 Cn1nc(CNC(C2CC(OC3CC3)C2)=O)c2c1CCN(C(C1CCO1)=O)C2 CN=S(C)(=O)c1cccc(C(N2CCC(C)(CCNC(=O)CSC(C)C)C2)=O)c1 c1(C(N2CCC(C)(CNC(C(CCCOC)C)=O)C2)=O)c(F)ccc2n[nH]cc12 N1(C(c2c(OC)ccs2)=O)CCN(C(C2CC3(C2)CC3(F)F)=O)CC1CC(F)F C1(C)(C(N2CCN(C(C(C)C)=O)C(CF)C2)=O)COCC2CCCN12 N1(C(C(CCNC(CS(CC)=O)=O)OC)=O)CC(F)(F)CC1CO c1(C(=O)NCCC(C)N(C(C(C)OC)=O)C)c(F)ccnc1Cl c1(C(C)C)cc(C(=O)NC(=O)NCCc2csc(Cl)n2)on1 Cc1cc(C(=O)NC2C3CC2N(C(C2(C4CCCCO4)CC2)=O)C3)c(C)o1 C1(NC(C(c2cn(C)nn2)NC(C(C2CC2)OCC)=O)=O)CCn2nnnc2C1 c1(N(CCCSCC)CCNC(C2CCOC2)=O)cc2[nH]c(C)cc(=O)n2n1 N1(C(CC2C(=O)OCC2)=O)CCC2C(CCCN2C(=O)Cc2c[nH]nc2O)C1 N1(NC(=O)NC)CCN(C(=O)C(CCSC)C(=O)C=Cc2cnc[nH]2)CC1 C(=O)(C1=CC(O)CCC1)NC1(C)CCCN(C(C(=O)N(C)C)=O)C1 c1(CN2CCC(NC(c3c(Cl)cccc3I)=O)C2)cnc2ccc(F)cn12 C#Cc1cnn(CC(=O)NCC2CCN2C(=O)C(C)COC)c1 Cn1nc(C(=O)NC2CCCC2NC(c2ccc(Cl)cc2)=O)ccc1=O N(C1c2ccccc2CC1NC(C1CCCCC1O)=O)C(COCCC(C)C)=O C1(CNC(COCC#C)=O)CC(C)CCN1C(=O)C(C)Cc1cnco1 Cc1ccc(O)c(S(=O)(=O)Nc2ccc(O)c3ccccc23)c1 C1(C(=O)NCC2(NC(C(c3cn(C)nc3)(F)F)=O)CCC2)CC2C=CC1O2 C1(F)(CNC(=O)CCc2ccoc2)COCCN(C(=O)CCCC2CCCO2)C1 N1(C(C(c2ccc(Cl)nc2)(C)C)=O)CC(NC(C2CC2C(N)=O)=O)C(N=[N+]=[N-])C1 N1(C(C(C)OCCC=C)=O)CCCC1CCNC(C1CCCC1CC)=O c1(C2(NC(C3(C)CC(NC(C(C)NS(C)(=O)=O)=O)C3)=O)CC2)cccc(C#N)c1 C(=O)(C(CCC1CC1)NC(N)=O)NCC(CNC(CCCCCCC)=O)F c1(C(=O)NC2(CC=C)CN(C(=O)CCN3CCOC3=O)C2)c(C2CC2)cnn1C C(CCC(=O)N(C)C)C(C)SCC1(NC(=O)COCC2CCCOC2)CC1 N1(C(Cc2nc(C)[nH]n2)=O)CCCC(NC(=O)CC(O)C(C)C)C1C c1(C(=O)NC(CNC(CC2(CN(C)C)CCC2)=O)(C)C2CC2)cc(Cl)cs1 c1(C(N2C(C)CCC(CNC(c3c(C)ncs3)=O)C2)=O)nccc2c[nH]nc12 C1(NC(=O)Nc2nc(C(F)(F)F)c(Br)s2)COC2C(O)COC12 C(=O)(C1Cc2ccccc21)N1CCCC(CN(C)C(c2cccnc2)=O)C1 C#Cc1ccc(F)c(C(=O)NC2CCN(C(c3ccccc3C)=O)CC2CC)c1 c1(OC)c(C)cc(C(=O)NCC2(NC(C3(F)CCS(=O)(=O)C3)=O)CC2)cc1Cl CCC(C(=O)NC(CC(F)F)C(=O)N1CC(CO)C(O)C1)C(F)(F)F C#CCC(C)(C)C(=O)NC1CC1CNC(c1ccnc(CO)c1)=O Fc1c(-c2cn(C3CCN(Cc4cc(Cl)ccc4Cl)C3)nn2)cccc1Br C1(NC(C(c2ccc(C)o2)C)=O)CC2CC1N(C(=O)Cn1ccc([N+](=O)[O-])n1)C2 CC(C)(C)S(=O)(=O)CC(=O)NC1CC(CNC(C2CC23CCC3)=O)C1 CC1(C)OC2CC(N3CCOCC3)(c3nnnn3C3CC3)CC2O1 c1(C(C(=O)NCC2CCOCC2)N(CC(C)(C)CCO)C)nn(C)c2c1CCCC2 c1(CC(N2CCC(C)(NC(CSCC)=O)C2)=O)ccc2c(c1)CCC2 C(=O)(CCCCCN(C(=O)CCS(C)(=O)=O)C)NC(c1ncc(C)[nH]1)CC c1(C(=O)NC2C(C)CN(C(c3csnc3C3CC3)=O)C2)cc(Br)ccc1O c1(C(N(CCSCC(=O)NC2CCCO2)C2CC2)=O)cccnc1OC(F)F c1(CC(N2CCC(CNC(C(C)SC)=O)C2)=O)c[nH]c(=N)nc1O C1(CNC(COCC)=O)CN(C(c2cc(C(F)F)no2)=O)CCC1(F)F N1(C(C)=O)CSCC1C(=O)NCCCC(C)NC(=O)Cc1csc(C)n1 CC1CN(C(=O)Cn2cnc(C3CC3)n2)CC1CNC(C1CC2CCC2C1)=O N1(C(C2(SCC)CC2)=O)CC2CC2(NC(=O)C(C)(C)n2ccc(C)n2)C1 c1(C(N(C2CN(C(CNC(=O)OCC)=O)CC2(C)C)C)=O)cc2cccnc2o1 c1(C(C)=O)ccc(C(=O)NCC2(F)CCCN(C(C3CCC4CC34)=O)C2)c(F)c1 S(=O)(=O)(c1ccc(NC)cc1Br)NCC(CC)N(C)CCn1cccc1 c1(OC)cccc(C(N2CCCC2CC(=O)NCc2ccnn2C)=O)n1 C1(C(N(CC(CC)NC(C2(CC)CCC2)=O)CC)=O)CCc2nn[nH]c2C1 C1(C)(NC(CCCOC(C)=O)=O)CCCN(C(=O)CC2CCCNC2=O)C1 c1(C(N2CC(C)(NC(c3cnn(C)c3Cl)=O)C2)=O)ccc2nc(N(C)C)sc2c1 N1(C(c2nc(C)[nH]n2)=O)CCOC2CCN(C(c3ccc4nonc4c3)=O)CC12 C1(C)(NC(=O)NCC(C)(C)c2nn[nH]n2)CCOC1 c12cnc(nc1)C(=O)N(CC)CC(O)CNC2=O.C(=O)(CCSC(F)(F)F)C(C)C N1(C(CC=CC)=O)CCCC(CC(N2CCN(CCO)CC2C)=O)CC1 CC(=O)CCCC(C)C(=O)NC1CCCC1NC(=O)CCc1cccnc1 c1(OC)ccc(F)c(CC(N2CC(NC(c3cc(Br)ccc3N)=O)C(O)C2)=O)c1 c1(C(=O)OC(Cc2c(C)noc2C)C)nc(O)c2ccccc2n1.C1(=O)CCN1 c1(N(CCCCN(C)C(c2ccccc2)=O)C(C)=O)cccc(F)c1C c1(C2C(C(N(CCCCN3CCCC3)C)=O)C2)ccncc1.C12(CC1)C(=O)NC2.O=C C(CC(C)C)(C(=O)NC1CC1CC(=O)NC(CO)CCF)OC CCCC(C(=O)OC)C(=O)N1CCCCCC1CNC(c1ccoc1)=O N1(C(CN2CCCC(O)(OC)C2)=O)CCN(c2nc(OC)c(C)c(C)n2)CC(C)(F)C1 c1(NC2(CNC(c3c(C)nns3)=O)COC2)c(Br)cc([N+](=O)[O-])cc1Br c1(C(N2CC(CNC(C(C(C)C)N(C(C)C)C)=O)C2)=O)cccc(F)c1I c1(C(=O)OCC)ccc2nc[nH]c2n1.C12CC3CC(C1C3)N2 c1(C(c2nnnn2C2CCC2)NCC(=O)NCCC)cccn2ccnc12 c1(C(C2CC2[N+](=O)[O-])NC(N(CC(C)O)C(C)C2CC2)=O)cnc(O)c([N+](=O)[O-])c1 CC1CC(=O)NCC1C(N1CC(F)(CNC(c2cnc(Cl)[nH]2)=O)C1)=O N1(C(c2ccc(=N)[nH]n2)=O)CC(C2CC3(C(C(=O)NC)C3)C2)C(C2CC2)C1 C1(CN(C(c2ccn(CC)n2)=O)CC)CCCCN1C(=O)CC1(C)CCCC1O C1(O)(C(=O)OC)CCN(C(=O)C(=O)Nc2conc2-c2ccccc2Cl)C1 N1(C(CC(C(C)C)OCC)=O)CCC(C)N(C(c2cc(F)ccc2F)=O)CC1 Cc1nc2nnnn2c(C)c1CCCN(C)Cc1ccon1 C12CC(F)CN1CC(=O)N2.Cc1nccn1C1CCN(c2nc(C3CC3)ns2)C1 C=CC(C(=O)NC1(C(=O)N(CC)Cc2ncc[nH]2)CSC1)OC C=CCCCCC(=O)N(C1CCCC(N(C)C(c2ncoc2CC)=O)C1)C C1(CNC(=O)CCCn2ccnn2)CCC(NC(=O)Cc2cnccc2Cl)CC1 N1(C(C2C(C)C2C)=O)CCC(C)(NC(c2cc(-c3ccccc3)on2)=O)C1 C(C)(C)(CS(=O)(=O)NC(C1CCCO1)Cc1ccccc1)OC(C)=O C1(NC(=O)C2=CCCO2)CCC2CN(C(=O)CN3C(=O)CCC3=O)CC2C1 C(=O)(C(C)(CO)NC(CCCl)CF)NC(C1CCCCC1)C c1(CNC(C23CC2CN(Cc2nc(C(=O)OC)sc2)C3)=O)ccc2ccccc2n1 c1(CN(C2(C)CCCC2)C)ccc2c(c1)C(=O)N(C1CCCCC1)C2=O c1(C(=O)NCC(C(C)C)NC(C(C2CCC2)OCC)=O)ncc(C2CC2)cc1F C1(C(=O)NCCCCN(C(C(CC2CCC2)OC)=O)C)Cc2nnc(C)n2C1 C1(NC(c2c(NC)nccc2)=O)CCCCN(C(=O)C(c2c(C)noc2C)C)C1 N1(C(c2cc(CCOC)on2)=O)CCN(C(=O)CCP(C)(C)=O)CC1C1CCC1 c1(Oc2cnc(COC)[nH]2)cccc2c1CCN(C(C1(OC(C)C)CCC1)=O)C2 C=C(C)CC(C(=O)N1CC(Cc2ccoc2)C1)NC(C1CCOC1(C)C)=O C=C(C)CC(C(=O)NC12CC1CN(C(c1cnc(O)cc1C)=O)C2)OC Cc1[nH]c2ccc(F)cc2c1C(=O)N(CC(O)CNC(=O)CC1(C)CCCO1)C C1(C)(C(N2CC(c3cn(CCC=C)nn3)(O)C2)=O)Cc2ccc(Br)cc2C(=O)O1 c1(C(=O)NC2C3(CC(NC(CC(C)O)=O)C3)C2)cn2cc(Cl)cnc2n1 N1(C(C(C2CCCOC2)OC)=O)CCCC(NC(c2ccc(C(C)C)nc2)=O)C1 C1(NC(c2c(C)cnn2C)=O)CCN(C)C12CCCN(C(=O)C(C)C1CCC1)C2 N1(C(C(=O)Nc2cc(CC3CC3)cs2)=O)CCOCCC1CCc1ccncc1 c1(OC)cccc(S(=O)(=O)NCc2ccc(F)c(F)c2)c1-c1cccc(C#N)c1 C(CC1CCOCC1)(C(=O)NC1CC(F)(F)C1)NC(C(C)C1CCCC1)=O C1(C(=O)NCCN(c2ccccc2Cl)c2ccccc2)CC2(COC(=O)N2)C1 N1(C(CC(C)n2cccc2)=O)CCC(C)(CNC(=O)CC2CCC(F)(F)C2)C1 Cc1cc(C(=O)N(C2CCCCN(C(C3CCCCC34CC4)=O)C2)C)ncc1F N1(C(CC(CC)SC)=O)CCCC(C(=O)NC2CCC(C(=O)OC)CC2)C1C N1(C(C2CN(C)C(=O)N2)=O)CC(O)(C2(CNC(C3CC4C=CC3O4)=O)CC2)C1 C1(CC(N2CCC(N(C(CCC(CC)C)=O)C)CC2)=O)CCCC2(CCC2)O1 Cc1cccc(F)c1CC(=O)NC1CC(C(C)NC(=O)C(C)CC2CCCC2)C1 Nc1cc(F)c([N+](=O)[O-])cc1C(N1CCCC(NC(=O)C=CC2CCC2)C1)=O C(=O)(C1=NOC2(CCOC2)C1)NC(c1ccc(F)cc1)C(=O)NC N1(C(CC(C)C)=O)CC(NC(c2ccc(OC(F)F)cc2)=O)C(CC(C)(C)C)C1 CN1CCCC(C(=O)NCC(O)C(=O)NC2CC2c2cn(C)cn2)C1 C(=O)(C1=CCS(=O)(=O)C1)NCC(CNC(CCn1ncc(C)c1)=O)(C)O C(=O)(CC(F)(F)C(F)F)NCC1(C)CCCN1C(c1ccc(Cl)c(N)c1)=O c1(C(N(CC(CC)NC(=O)CN2CCCC2)C)=O)cnc(-c2cccs2)[nH]1 c1(C(=O)NC(CNC(c2cc(CCC)on2)=O)(C)CC)ccnnc1O C1(C(=O)NCC2N(C(C(c3cccnc3)OC)=O)CC2)OCCC1C CC(Cc1ccccn1)C(=O)NCC1(NC(c2cnn(C)n2)=O)CCCC1 Cc1cnn(CC(=O)NC(C2CC2C(=O)NC2(CCCF)CC2)C)c1 N1(C(C2CCN(C(N)=O)C2)=O)CCN(CCNC(c2c(C)ncs2)=O)CC1 C1(C(N(CCCC)C2CC2)=O)CCN(C(C2CSCN2C(=O)C(C)CC)=O)C1 C1(C=O)CN(CC2CC(F)C2)CC1C.c1(C2CC(C)C2)ccc(Br)cn1 S(=O)(=O)(c1ccc2[nH]c(=NC(C)CC3CCCC(=O)N3)sc2c1)N(C(C)C)C C1(NC(C(=O)OC)=O)CN(c2nc(C(F)(F)F)nn2C)CC1C C(=O)(CC(CC)NC1CCN(c2cccc(OC)c2)CC1)N(CC=C)C1CC1 N1(C(C2CCCCCC2)=O)CCC(C(=O)NCC(F)CO)(CC2CC2)C1 C1(C(N2C(COC)CN(C(=O)Cn3nccn3)CC2)=O)CC(C2CCCC2)C1 C(=O)(C(C(C)(C)C)NC(c1ccc(Cl)s1)=O)NCc1snc(CC)n1 c1(CC(=O)NNC(=S)Nc2ccc(F)c(F)c2)ccc2[nH]ccc2c1 C1(C(=O)NCc2nnn(-c3ccccc3)n2)COC2(CCCNC2)C1 c1(SC)c(C(N2CCC(N(C)C(C3CC3CF)=O)C2)=O)sc2ccccc12 C1(C(=O)OC(C)(C)C)C2CCC(O2)C1CC(=O)NOCCC(F)F C#CCCCCC(=O)N1CCCC(NC(c2cn(CCC(F)(F)F)nc2C)=O)C1C N1(C(CN(CC=C)C(c2n(CC#C)ccn2)=O)=O)CCC(C)=C(F)C1 N1(C(Cc2onc(C)n2)=O)CCC2(C1)CN(C(C13CC1COC31CCC1)=O)C2 N1(CCc2n(C)ncn2)CCC(=O)N(CCc2cccc3cc[nH]c23)C1=O C1(CNC(Cc2c(C)occ2)=O)N(C(C2CCS(=O)(=O)N2)=O)CCCC1(C)C N1(C(CC2ON=C(C)C2)=O)CC(N(C(=O)Cc2cn[nH]c2)C)C2(CC2)C1 N1(C(C(C(C)C)n2cc(C)nc2)=O)CCC(NS(C)(=O)=O)C(O)C1 C(=O)(CCCC(=O)N1CCC(C(C)NC(=O)C(c2ccccc2)C)C1)NC C1(NC(C(C)N(C(=O)CN2CCOC2=O)CC)=O)CCC(=O)NC1C c1(NCCCC(C)NC(=O)OCC)cnc(C2CCC2)nc1O N1(C(CC(C)F)=O)CCC(C)(C)C1C(=O)NC1CC(=O)NC(=O)C1 C=CCC(C(=O)N1CCC(C(=O)NC(CC(=O)NC)C2CC2)C1)NC(C)=O c1(NCCCCC2(C)NC(=O)NC2=O)nccc(=NCCCF)[nH]1 C1(C)(CNC(C2CCN(CC)C2)=O)CCCN1C(=O)Cc1cc(C2CC2)no1 C1(C)(CNC(C(C)C2(O)CCC2)=O)CCN(C(C2CC2C2CC2)=O)CC1 O=C(C(O)CC(F)(F)F)N1CC(NC(C2CC3CC3C2)=O)C1 c1(CNC(c2nccs2)=O)ccccc1-n1cc(C(=O)O)nn1 c1(C(N2CCC(N(C(C3CCOC3)=O)CC)C2)=O)ccnc(C)c1N C12(CC(N3CC(CC)N(C(c4ncn5c4CCC5)=O)CC3)=O)CCC(CC1)OC2 c1(C(=O)O)ccc(F)cc1Cl.C12(OC)CC1CN(C(c1ncccc1O)=O)C2 C1(NC(Cc2ccc(OC)nc2)=O)CC2CCC1N2C(=O)CC1(O)CCCC1 Cc1nc(C(N2CCCC2Cn2cc(CN3CCOCC3=O)nn2)=O)c(C)n1C CCCCCCCC(=O)NCC1CC2(CC(NC(=O)Cc3ccccc3F)C2)C1 C1(CNC(c2cccc(F)c2)=O)CCCCCN1C(c1nc(Cl)ccc1Cl)=O c1(C(c2nnnn2C(C)CC)NCCSCCCCCC)cnn(CCO)c1C c1(C(C2CC2)NC(=O)NCCC(=O)NCCC)ccc(F)c(F)c1 c1(C(N(C)CC2(NC(c3cc(C)ncc3)=O)CC2)=O)n[nH]c2c1C(O)CCC2 N1(C(CCCCN(C(c2ncn(C(C)C)c2)=O)C)=O)CCCC(C)(N(C)C)C1 Cc1nn(C)cc1C1OCCC1CNCCCC1CCCNC1 C12(CNC(C=C(C)C)=O)CC(C1)C(NC(=O)CCc1ccc(C)c(C)c1)CO2 c1(C(C)NC(=O)COCCNC(C2(C3CCCOC3)CC2)=O)ccc(C#N)cc1 N1(C(C)CNC(=O)CCc2ccc(Br)nc2)CC2CCNC2C1 Cc1cc(C(=O)NCCCN2CCOCC2CO)nc(C)n1 n1(CCC)nc(C)c(C(N2CCC(C)C2CNC(=O)CC(C)(F)F)=O)c1C C1(CNC(c2nc(CCC)oc2)=O)C2CN(C(C3CC34CCC4)=O)CC12 c1(SC)ncc(C(F)(F)F)c(N2CC(NC(c3cc(O)ccc3F)=O)C(F)C2)n1 N1(C(Cc2n(C)cnc2)=O)CC2CC1CCN2C(=O)CCNC(C1CCC1)=O c1(C(=O)NC2CCCC(NC(CCSCC)=O)C2)c[nH]c(=NCC(F)(F)F)cn1 N1(C(=O)C=CC(C)(C)C)CCC(c2ncc[nH]2)C1.CC(C)CN1CC1=O C(=O)(C1=CCOCC1)NC(CCOCC)C(=O)NCc1nc(C)co1 N1(C(C2(C(C)C)CCC2)=O)CCOC(Cn2cccn2)C1 CCC(CC(=O)NC(CNC(=O)C(C)OC1CCCCC1)C(C)C)C1CC1 C(=O)(C#CC(C)(C)CNC(c1c(C)ccnc1C)=O)N(CCCCCC=C)C N#Cc1ccc(CC(N2CCCC2CCNC(c2cscc2F)=O)=O)cc1 c1(NC(C2CN(C(=O)C3=CC(O)C(O)C(O)C3)C2)=O)ccc2ccncc2c1 C1(O)(COC)CCCN(C(=O)C=CCNC(C2CCCCN2C)=O)C1 c1(CNC(C(C(C)C)NC(c2c(C)nns2)=O)=O)ccc(F)cc1F C1(CCNC(c2cn(CCNC(=O)Cc3cncnc3)cn2)=O)CCCC1O Cc1cccc2c1OCC2C(=O)NCCOCCNC(=O)CC(C)(C)C1CC1 C(CNC(=O)C(C)(C)CNC(C)=O)(CC(C)C)NC(C(C=C)O)=O c1(C(=O)NCC2(O)CN(C(C=CCC)=O)C2)ccc(N2CCCCC2=O)cc1 C1(CC)(NC(=O)C(C)O)CN(CCc2nccn2C)C1 Cn1cnc2ccc(C(=O)NCC3CCCC(NC(=O)CP(C)(C)=O)C3)nc12 c1(C(N2CCC(CNC(c3cc(COC)sc3)=O)C2)=O)ccc2nnn(C)c2c1 c1(C(=O)NC2(CC)CN(C(c3cnc(SC)s3)=O)C2)cc2ccccn2n1 C(=O)(C1=C(C)N(C)c2ncnn2C1)N(C1C2CN(C(C(COCC)C)=O)CC21)C C1(NC(=O)CCCOCc2ccccc2)CC(C)N(C(=O)OC)CC1C C1(NC(C2CC(O)(CC#C)C2)=O)CCSC12CN(C(c1ccnn1C1CC1)=O)C2 C1(CC(=O)N(C2CCN(C(=O)C=Cc3cnn(C)c3)CC2)CC)CCC(C)(C)O1 N1(C(C(C)S)=O)CC2C(C1)N2C(c1cc(C(C)(C)C)on1)=O C(C(CNC(=O)CC1CCOCC1)C(F)(F)F)NC(CCc1cn(C)nc1)=O C(=O)(CC(C(C)OC)NC(c1cnncc1OC)=O)N(C(CC)CC)C N1(C(c2c(CC)nc(C)o2)=O)CCCC(NC(=O)CC2CCCCC2O)C1C N1(CC(=O)NC(CC(C)C)CNC(=O)Cc2ccnn2C)CCCCC(O)C1=O C1(C)(COC)CC(NC(=O)C(C2CC2)C2CC2)CN1C(c1ncc(N)nc1C)=O C1(CC(=O)OC)CN(CC(C)Cc2cccc(OC)c2)CC(C)O1 N1(C(c2cc(C(C)C)nn2C)C(=O)NCC2CCCO2)CCCCCC1C c1(OC)ccc(CNC(=O)NC2CCOCC2F)c(Cl)n1 C#CCC(C)C(=O)N1CCCC1CN(C)C(C1OCCOC1C(F)(F)F)=O Cc1ccc(OCC(=O)Nc2nnc(CC#N)n2CCN2CCSCC2)cc1 c1(OCC)ccccc1C(=O)OCC(=O)NC(c1cccc(O)c1)C n1(CC)ccnc1C(F)(F)C(=O)NCCNC(C1(CC)CCC1)=O CCC(C(=O)NCC1CCN1C(C1CC1C)=O)NC(N)=O CCC(CC#N)C(=O)NCCCN(C)C(c1ccc(F)cc1SCC)=O c1(C(=O)NCC(CC=C)NC(C2CCN(C)C(=O)C2)=O)cncc(Br)c1C C(N=c1nc(N2CC3CC2CS3(=O)=O)c2cc(F)cc(F)c2[nH]1)c1nnc(C)o1 C(=O)(C(CC(C)C)CC(C)C)N1CCC(N(C(Cc2nc(C)[nH]n2)=O)CCO)C1 Cc1nc2cc(C(=O)NCC(O)CNC(=O)CC3CCOC3)ccc2n1C1CC1 c1(N2CCC(C(=O)NC(CC)C)CC2)nccc(=NC2C=C(C)CCC2)[nH]1 C1(NC(C(C)OCCN(C)C)=O)CCN(C(C2CCCS2(=O)=O)=O)CC1F c1(CC)oc(C(N2CCC(C(=O)NC(c3cc[nH]n3)C)(CC)C2)=O)cc1C CC12CCC(NC(C3CN(C(=O)Cc4cc[nH]c4)C3)=O)(CC1)C2 c1(NC(C(CC2CN(C(C(COC)N(C)C)=O)C2)F)=O)cc(C)c(O)cc1C c1(C(=O)NCCOCCN(C)C(C23CC2COC3(C)C)=O)ccc(F)c2occc12 C1(CNC(CN(CCOC)C(C2CC2C2CC2)=O)=O)CCC(O)CC1 C(=O)(C(C)(C)CC(=O)N1CC(O)(CCNC(=O)Nn2cc(C)cn2)C1)OC C(C(C)(C)OC)NC(c1ccon1)=O.N12CC(C1)C(C)OCC2=O.C(=O)NCCO c1(C(=O)NCC2(CNC(CC(CCC)C)=O)CC2)cnc2n(c1=O)CCS2 N1(C(c2[nH]cc(C#N)c2)=O)CC2CCC(C1)N2C(c1conc1C1CC1)=O c1(NC(N(CC)CC)=O)ccc(Cl)c(C(N2CCOC3CCCC23)=O)c1 CC(CC(F)(F)F)C(=O)NC1(CNC(=O)Cn2cnc(=N)[nH]2)CCCCC1 N1(CCNC(C2(CCNC(C3C(C)CC3)=O)CC2)=O)CCC(C)(C)C1 c1(C(N2CCCC(F)(C(=O)NCCSCCO)C2)=O)cc2scnc2[nH]1 CCCS(=O)(=O)c1ccc(S(=O)(=O)NCC(=O)Nc2ccc([N+](=O)[O-])c(Br)c2)cc1 N1(C(c2c(C)[nH]nc2C(F)F)=O)CCC(C)(CNC(C2CC(F)C2)=O)CC1 C1(O)(C(CNC(CN(C)C(=O)C2CC2)=O)C)CCN(C(=O)COC(F)F)C1 c1(CNC(CCC(=C)C)C)cccc2c1CCC2N C(C)(C(=O)NNc1cccc(C(F)(F)F)c1C)Oc1ccc(C)cc1C c1(CNCC(C)S(C)(=O)=O)sc2ccccc2c1Br c1(C(C(=O)N(c2ccsc2)CC)NC(C2CCC(C(=O)OC)C2)=O)cn(C)nn1 N1(C(CN(C(C)=O)C)=O)CCC(F)(CNC(=O)CC2CCCCCC2)C1 N1(C(C2(C#C)CC2)=O)CC2CCC2(CCNC(=O)C(C)Cc2ccnn2C)C1 C=C1CC2(C1)CC(C(=O)NC(C)C(C)NC(c1cc(C#N)[nH]c1C)=O)C2 c1(C(=O)NC2CCC(NC(=O)C=CC(F)(F)F)CC2)ccc(F)c2ccncc12 C1(CN2CCC(C(CC)CC)CC2)COCC(=O)N1C c1(C(=O)NC(C)=O)cc(N)ccc1F.c1(CN(CC)CC)cc(C(C)C)no1 C1(CNC(c2ncn(C)n2)=O)CN(C(c2cc[nH]c(=N)c2)=O)CC12CCC2 Cc1nn2c(c1NC(=O)CCn1cc(C3CCCCC3O)nn1)CCCC2 C1(C#CC(=O)Nc2cccc(NC(=O)C(C)NS(C)(=O)=O)c2)(CC)CC1 c1(NC(C)=O)ccc(C(=O)NC2CCCN(C(=O)C(C)Cc3cnc[nH]3)C2)nc1 N1(C(COC(C=C)C)C)CCN(c2nnnn2CC(C2CCC2)OC)CC1 N1(C(C(C)SC)=O)CC(C)(C)OCC1CNC(c1c[nH]nc1[N+](=O)[O-])=O CCCC(C(=O)NCC1C(C(=O)NCC(c2ccsc2)C)C1(C)C)NC(C)=O C#Cc1ccc(OCC(=O)NCC(C(C)C)NC(C2CCN(C)C2)=O)cc1 c1(NC(c2c(C)[nH]c(C(=O)NCC3COC3)c2C)=O)ncc(Br)c(C)c1[N+](=O)[O-] C1(N(C(CSC)=O)C)CCN(C(C2(F)CCOC2)=O)CC12CC2 Cc1cc(O)ncc1C(=O)N(C1CCCN1C(C1CN(c2nnc(C)s2)C1)=O)C C1(C(=O)NC2CCCC2CNC(C2(c3cc[nH]n3)CCC2)=O)CCOCC1 C(=O)(C1=CCC(C)CC1)NCCC1(OC)CN(C(c2c(OC)csc2)=O)C1 c1(C(N2C(C(N3CCC(OCCC)CC3)=O)COCC2)=O)cnn2c1OCC2 N1(C(c2c(CC)nc[nH]2)=O)CCC2OCCN(C(c3ccc(N)c(Cl)c3)=O)C2C1 C#CCCCCCC(=O)NC(c1ccccc1)C(=O)N1CCC1CC1CC1 C1(C(=O)Nc2ccccn2)CC(NC(c2sc(Br)nc2C(F)F)=O)C2CC12 c1(CCC(=O)NCCC2(O)CCN(C(c3ccccc3F)=O)C2)ccc(F)nc1 N1(C(CSCCC)=O)CCC(C2CC2)(CNC(=O)C(C)(C)OCCOC)C1 C(=O)(C(C)(O)C(F)(F)F)N1C(CCCNC(C(CCC)O)=O)CCC1 c1(O)ccc(OCc2ccccc2)cc1F.CN1C(C(=O)O)CCC1C(C(=O)O)N c1(C(=O)NC(CC)(C)CNC(C2CCCN2C)=O)ccc(Br)c(C)c1 c1(C(=O)NCC2CCC(NC(C=C(C)Cl)=O)C2)[nH]c2ccccc2c1C(F)(F)F C1(N(C)C(c2ccc(-n3cncn3)cc2)=O)CN(C(=O)Cn2ccnn2)CC1F C(=O)(C1=COCCC1)NCC1CCC(C(N2CCC(OCC)C2)=O)C1 c1(N(C(c2cn(CCNC(C3C(C)CC3)=O)nn2)=O)C2CC2)cncc([N+](=O)[O-])c1 c1(-c2cn(CC(CNC(c3cccnc3F)=O)OC)nn2)ccc(F)c(Cl)c1F C1(NC(C(CC)OC2CCCC2)=O)CC(NC(=O)CC(C)C)C12CCC2.C1CN1 N1(C(c2ccc(C)nc2C)=O)CC(NC(=O)CC2OCCO2)CC2(CCC2)C1 C1(CCC)CN(C(=O)C=CC(=O)OC(C)(C)C)CC1C(N1CC(CCOC)C1)=O c1(C(=O)NCC2C(C(N3CC(C)(COC)C3)=O)C2)c[nH]c(=S)cn1 c1(C(=O)NCC2C(NC(c3ccc(NC)cn3)=O)C2)nsc2ccccc12 CC1CCC(NC(C2CC(O)C2)=O)N1C(C1CC1c1ccccc1)=O CC(C)CC(F)C(=O)NC1CCCC1NC(=O)CSCc1ccc(Br)cc1 n1(CC(=O)NCC2(NC(C(C)O)=O)CC2)ccc(=O)c([N+](=O)[O-])c1 CC(C)C(CC(=O)NCCCO)NC(C12CC(C(=O)OC(C)(C)C)(CO1)C2)=O Cc1nc(F)ccc1C(N1CCC(NC(C2CCC2)=O)C(F)C1)=O N1(c2cc(OCC)ncn2)CCC2(CC1)CC2CNC(c1nnc(C)s1)=O C(c1cncnc1O)=CC(=O)NC1(CNC(c2ccc(OC)nc2)=O)CC1 C1(C#N)(CC(=O)NCCN(C(C(N2C(=O)CCC2=O)CC)=O)CC)CCCC1 C12(C(N(C)CC3N(C(C4C(C=C)OCC4)=O)CCC3)=O)CCCCC1C2(F)F C1(C(C)NC(C2CC(OC)CN2Cc2ccc(C)[nH]2)=O)CCC(F)(F)CC1 C123CCOC(C1)(C2)CNC(=O)C1OCCC1C(=O)N3.C1(C)(CC)CC=CCC1 C=Cc1cncc(C(=O)NCCOCC(N2CCC(C)C(O)C2)=O)c1 C1(CC(=O)NC(CC2CC2)CSC2CC2)(CNC(=O)OC)CCC1 CC1COc2c(C(=O)NC3CCC(CNC(c4cnc(=N)[nH]c4)=O)C3)cccc21 c1(CCC(=O)N(CC(CNC(CC(CC)C)=O)C)C)cccc(C)c1Br C=C(C)C1CN(C(C2(CNC(C3CN(C(C)=O)C3)=O)CC(=C)C2)=O)CCO1 c1(C(N2CCC(C)(C(=O)NC3CC4CC4C3)CC2)=O)c[nH]c2cccnc12 C(=O)(C1=CS(=O)(=O)CCC1)NCCC(C)NC(Cc1cc(OC)c(Cl)cc1)=O C1(NC(C(C)OCCN(C)C)=O)CCN(C(=O)CCc2cnn[nH]2)C12CC2 C1(C(N(CCCN(C(c2[nH]cc(C(N(C)C)C3CC3)c2)=O)C)C)=O)COC(=O)N1C N1(C(c2cnn(C)c2Cl)=O)CC(C)(C)C(NC(c2cnn[nH]2)=O)C(C)(C)C1 c1(C(=O)NCCOC2CCN(C(=O)C(F)=CC3CC3)CC2)ccc2cccnn12 n1(CC)nnc(C)c1C(N1CCN(CC(C)NC(=O)C(C(=O)OC)OC)CC1)=O N1(C(C(CN(CC)CC)F)=O)CCC(NC(=O)C(F)(F)C2(OC)CCC2)C(F)C1 c1(C(=O)NCCC(C)NC(C2CCN(C)S2(=O)=O)=O)c(F)cccc1Cl N1(C(CC=C=C)=O)CCC(NC(=O)CC2(C#N)CCOCC2)C(F)(F)CC1 c1(C(CC)NCCCCCC2CC2)ccc(OC(C)C)c(F)c1 C(=O)(N=c1[nH][nH]cc1-c1cccnc1)c1nc(C(N2CCN(C=O)CC2)=O)sc1 C=CC(C)(O)C(=O)N(C1CCN(C(=O)C(O)C2CCCC2)CC1)CC1CC1 C1(C(=O)NC2CCN(C)C2)COC2(C1)CN(CCOCc1ccccc1)C2 CC1(C)COCCC1CN(C=O)Cc1cnn[nH]1 C=CC(CC)CC(=O)N(C1(CC(=O)NC2(NC(C)=O)CC2)CC1)C N1(C(C2CCN(CC)C2)=O)CCN(C(c2cccc(N)c2)=O)CC1CC(F)F c1(N(C)C)cncc(C(N2CCCC2(C)CNC(=O)CN(C)S(N)(=O)=O)=O)n1 CC1(C)OCCC1CC(N1CCCC(CNC(=O)CC2(C)OCCO2)C1)=O C1(C(=O)NCCCOCCNC(c2c(=N)[nH]cnc2)=O)CCCS(=O)(=O)N1 N1(C(c2cc(C)ncc2)=O)CCN(C(=O)CCCCOC(F)(F)F)CC1C c1(CC)ccc(C(N2CCCCC2CNC(c2c[nH]c(=NC)s2)=O)=O)c(OC)c1 CCCC(C)CC(=O)N1CCC(O)C(NC(=O)C(O)Cn2cncn2)C1 c1(C(=O)NC)cccc(CCC(=O)N(C2CCCN(C(=O)C(F)(F)CO)C2)C)c1 C(=O)(C(C)CCC(C)(C)C)N1CCCC(CC)(NC(c2cc(F)ccc2C)=O)C1 C1(C(=O)NCC(CNC(c2cc(C)oc2C)=O)C)CCC(=O)N(CC(F)(F)F)C1 c1(C(C(=O)NC2CC(NC(CN(C)CCO)=O)CC2O)O)cc(Cl)cc(Cl)c1 c1(C(F)(F)F)cc2c(s1)CCCN(c1nccc(=NCCC3CC3C3CC3)[nH]1)C2 CCCCC(C)(F)C(=O)NC1CN(C(=O)COc2ccc(C)cc2C)CC1O c1(NC(C(C2CC=CCC2)NC(CSCC=C)=O)=O)cnccc1Cl c1(C(=O)NC2CC(C)N(C(=O)CCCCc3cnn[nH]3)C2)csc([N+](=O)[O-])c1 c1(C(=O)NCC2C(CNC(=O)Cc3ccccn3)C2)cc2c([nH]1)CCCC2 C(=O)(C1=CCN(C(=O)C(F)(F)C2CC2)C1)NC1(C)C(C)(C)C1 c1(CC)nc(C(N2CCCCC2CN(C(=O)CCOC)C)=O)c2ccccn12 N1(C(c2cc(SC)c(F)cc2)=O)CC(C)(C)OCC1CNC(=O)CCS(C)=O C(C(C(=O)NC1CCN(C(=O)C(CC)CC)C12CCC2)C(C)(C)C)OCC=C c1(C(N2CC(NC(C(CSC)C)=O)C2)=O)cc(C)cc(Br)c1O c1(C(=O)N(c2ncc(F)cn2)C2CNCC2F)ccc2[nH]ccc2c1 CN1CCOc2c(C(=O)Nc3cscc3Br)cccc21 N1(C(c2c(CC)cno2)=O)C2CCC(C(=O)NCC3(O)CN(C(N)=O)C3)C1CC2 c1(SCC)ccc(CC(=O)NCC(C)(O)CNC(=O)C=Cc2ccc[nH]2)cc1 C1(NC(=O)CN2CCCNC2=O)CCC2CC1CN2C(C1CCC1)=O c1(C(=O)NC2C(NC(c3c(OC)cncn3)=O)CCC2)cc(Cl)ncc1O C1(NC(C(F)OC)=O)(CNC(=O)CCOc2ccccc2)CC2CCC1CC2 CCC1=C(C(=O)NC(C)CN(C)C(c2cc(F)c(C3CC3)c(F)c2)=O)CCCO1 N1(C(c2c(C)n(C)nn2)=O)CCC(O)C(N(C)C(c2cc(CN(C)C)c[nH]2)=O)C1 c1(C(=O)NCC(CC)NC(=O)CCOCC(F)(F)F)cccc2cnsc12 C1(NC(C(C(C)C)NC(C)=O)=O)CC=C(C(=O)NC(C)(C)C)C1 c1(CCC(=O)NCCCCCNC(C=CC(CC)C)=O)cc(COC)c(C)o1 Cc1cc(=NCC2COCCN2C)[nH]c(NC2CC(=O)N(C3CCCCC3)C2)n1 c1(C(N2C(CNC(C=Cc3scc(C)n3)=O)CC2)=O)ccc(C2=NOC(=O)C2)cc1 c1(NC(C2(C#N)CCC2)=O)ccc2ncnn2c1.N12C3CCC(C3)C1C=CC2=O c1(CC)[nH]nc(C(N2CCC(CCC(=O)N(C3CCNC3=O)CC)C2)=O)c1C c1(C(=O)NCCC2CCCN(C(c3nncs3)=O)CC2)cc(F)c2cn[nH]c2c1 c1(C(=O)NCC(CNC(c2n(CC)ccc2)=O)(C)C)ccc2c(C#N)c[nH]c2c1 CCC(CC(=O)N(CCC(C)NC(c1cc(Cl)n(C)n1)=O)C)C(C)(C)C Cc1c(C(=O)NC2CC3CCC2N(C(C2(C)C=CCC2)=O)C3)oc2ccccc12 C(=O)(CN=c1cc[nH]cc1)NCC(C(N1CCOC(C(C)C)C1)=O)OC CCCC(O)CC(=O)NCc1cccnc1CNC(C1CCN(CCC)CC1)=O c1(C(N2C(CNC(CC3(NC(C)=O)CC3)=O)CCC2)=O)cn(CCC(F)F)nn1 c1(C(=O)NCC2(COC)CCOC2)ccc2c(=O)c3ccccc3sc2c1 C1(NC(c2n(CC=C)ccn2)=O)(CF)CCN(C(C2CCCC2C2CCC2)=O)C1 C(=O)(N=c1[nH][nH]c2c1CN(C(=O)CCc1ccoc1)C2)c1ncc(C)c(Br)c1 C#Cc1c[nH]nc1C(=O)NC(CO)C(=O)N1CCCC1CNC(N)=O CSC1=C(C(=O)NC23CCCC2CN(C(C2CCCN2C=O)=O)C3)CCCC1 c1(CCC(=O)NCC2(F)CCN(C(=O)CNc3nccs3)C2)cc(F)ccc1F C(=O)(CC(C)(C)C(C)=O)NCC1CCC(CNC(C2CCCC(OC)C2)=O)CC1 C1(CNC(Cc2cc(C)nn2C)=O)CCC2(CO1)CC(NC(c1cnco1)=O)C2 N1(C(CC(CC)C)=O)CC(NC(c2scnc2C)=O)C(N=[N+]=[N-])C1 C(CC(=O)NCCC(C)N(C)C(c1cnc(C(C)C)s1)=O)(C(C)C)OCC C1(OC)C(OC)CN2C1CNC(=O)CC1CC2C1.c1(C(=O)OC)csc(CO)n1 C1(NC(c2n(CCCOC)nnn2)c2csc(C)c2)CC(=O)N(C(C)C)C1=O c1(C(=O)NCCC2(CNC(C(C)n3cnnn3)=O)CC2)csc2nccn12 O=S(=O)(c1ccc(NCc2ccccc2CO)c(F)c1)NCC1=CCCOC1 NC(=NCCCF)NC1CSC1.O=S(=O)(CCOC(F)F)C(F)F c1(COC)noc(CCC(=O)NC(C2CCCN2C(c2cnoc2C)=O)C)n1 c1(CN2C(CNC(=O)CCc3nncs3)CC2)cccnc1 c1(NC2CCC(CC)CC2)cccc(S(=O)(=O)C(F)F)c1 C1(CNC(C(C)O)=O)CC2(CCC2)CN1C(=O)C(O)C(F)(F)F C(CN=C1NC2=C(CC(C)CC)C(=NCCCCC3(CC2)CCO3)N1)SC N1(C(C2(F)CCN(C(C3(C)C(C)C3)=O)CC2)=O)CCC(CO)C(C)(C)C1 CC(C)(C)CCCC(=O)NC1CCCC(C(=O)NC2CN(c3ncco3)C2)CC1 C(=O)(CN=S(C)(C)=O)NC(C1CCN(C(C(C)NC(=O)C2CC2)=O)C1)C N1(C(C(CC)=CC)=O)CCC(NC(=O)CC2CCN(C(=O)C(C)C)CC2)C(C)C1 C1(CC(=O)NC2(COC)CCCC2)C2CCCC2N1C(=O)C(C)CC(F)F N1(C(c2c(CC)c[nH]n2)=O)CCOC(CN(C)C(C2CCC(C(F)(F)F)C2)=O)C1 c1(OC(C(=O)NCC2CCC2C(=O)NCc2cc(C)on2)C)ccc(C#N)cc1 CC(C)CC(O)C(C)C(=O)OCC.C1(C)(CCO)CCN(C(=O)OC(C)(C)C)C1 C(C1CCCc2ccccc21)NC(c1n(CC=C)nnn1)c1n[nH]cc1C Nc1ccc(C(N2CCC(CNC(=O)C(c3ccccn3)O)C2)=O)c(O)c1 C(=O)(CS(=O)(=O)CCO)N1CC2(C(NC(c3ccc(CCCCCC)s3)=O)CC2)C1 C1(NC(CN(C)C2CC2)=O)CC2CCC(C1)N2C(C1CCN1C1CCCC1)=O C1(CNC(C(C)(C)c2ncco2)=O)CCN(C(=O)Cc2csc(=N)[nH]2)C12CCC2 C1(CC=C)(NC(C2CCS(=O)(=O)N2)=O)CCN(C(=O)CCc2ncc[nH]2)CC1 Cc1nc(C(=O)NC2(CNC(C3CCN(C)C3=O)=O)CC(F)(F)C2)c(C)o1 C1(C(=O)NC2(CCC(=O)NC3CCNC(=O)C3)CCCC2)CC2(C1)CC1(CC1)C2 c1(C(N2CCCC(N(C(=O)Cc3nc[nH]n3)CC)C2)=O)cnn2c1CC(F)(F)C2 N1(C(c2[nH]cc(C)c2)=O)CCCCC1C1(NC(c2n[nH]c(C)c2F)=O)CC1 c1(C(=O)NCC2N(C(c3c(C(C)=O)cccc3)=O)CC2)nccc2ccncc12 c1(-c2c(C(=O)NC(C)CCNC(C3CC(N(C)C)C3)=O)[nH]cc2)ccc(F)cc1 C1(C(N(CC(CC)(C)OC)C)=O)CCN(C(=O)CC23CCC(CC2)C3)O1 C(CN=c1nc(N2CCCC(COCCOCC)CC2)c2c([nH]1)CSC2)=CC C1(NC(Cc2cc(C)on2)=O)CC(N=c2[nH]c(Cl)ncc2C(N)=O)C1(C)C Cc1nocc1C(=O)NCC(C)(C)CN(C)C(C1CCOC1C(F)(F)F)=O C1(CC(N2CCC(N(C(=O)Cc3nc(=N)[nH][nH]3)CC)C2)=O)CCC(C)(C)CC1 c1(CC)noc(C)c1C(N1CC(CNC(C2(CO)CC2)=O)(OC)C1)=O C#CCCCCCC(=O)N1CCC(C)(C)C1C(=O)NCCC(C)(C)C c1(OC)ncc(Cl)cc1C(=O)N(C(C)CNC(c1cc(C)ccc1Cl)=O)C c1(N2CCC(CC)C2)cc(N(C)C)nc(C)n1.c12ccccc1NC(=O)NC2 C(C)(C(=O)N(CC(=O)NC(C)CN1CCCC1)C(C)C)=CC CCCC(O)CC(=O)NC1CC(O)(CNC(c2c[nH]nc2OCC(F)(F)F)=O)C1 C(=O)(CCC(=O)NC1CC1)N(CCC)CCN(C(c1cc(Cl)c[nH]1)=O)CC1CC1 c1(C(N2CCC(O)(CCNC(C(C)C(F)F)=O)C2)=O)c(F)cc(F)cc1F N1(C(CCOCCCOC)=O)CCC(C(=O)NC(=O)CC(C)C)=C(F)C1 C(=O)(C#CC1CC1)NCC(C1CCC1)NC(CCCOCCC)=O c1(C(N2CCC(C(=O)NCc3n(C)nnn3)C2)=O)ccnc(OCC(F)(F)F)n1 Cn1ccc(COCC(=O)NC(c2ccccc2)c2cccs2)n1 N1(CCCC(=O)NCC(CO)NC(c2n(CC#C)ccc2)=O)C(=O)CNC1=O C#CCCCCCONC(C1(F)CCN(C(c2c[nH]nc2Cl)=O)C1)=O C1(NC(C2(C)CC=CC2)=O)CC2CCC(C1)N2C(C1Cc2nncn2C1)=O C1(CNC(CC)=O)N(C(C2CC23CCC3)=O)CCCC1(C)C C1(CC(=O)N(C)CC2(COC)CC2)CC(NC(=O)Cc2ccn(C)n2)C1(C)C C1(NC(C(C)N(C(C)=O)C)=O)C=CCN(C(c2cnn(C(C)C)c2N)=O)C1 C1(NC)CCN(CC(N2CC(CC(C)NC(=O)C=CBr)C2)=O)CC1 c1(CNC(=O)NC(c2ccc(O)nc2)C)cc(C#N)n(C)n1 CC1(C)CCCOC1C(=O)NC1CC(CC(N2CC(n3ccnn3)C2)=O)C1 c1(C(=O)NCC(C2CC2)NC(C(COC)C)=O)c(Br)nc2n1CCCC2 c1(OC)cccc([N+](=O)[O-])c1C(=O)N(c1ccc(N)cn1)CCN1CCOCC1 c1(C(=O)NCC2C3CN(C(c4c(N)nccc4)=O)C2C3)cnn2c1OCC(O)C2 C#CC1CC2(CC2)CN1C(=O)CCCNC(C1CC2C(C1)C2(F)F)=O C1(CN(C(=O)CC2C=CS(=O)(=O)C2)C)COCCN1C(=O)C=Cc1cn(C)nn1 c1(C(=O)NCC2CC(NC(C(=O)NC)=O)C(O)C2)cc(C)n(C)c1C C1(O)(CCNC(C=CCOCCOC)=O)CCN(C(=O)C=Cc2nccs2)C1 c1(CN2CC(C)(C(=O)NCC3CCCO3)C2)cccc(O)c1O c1(OC)cccc(Cl)c1CCNC(=O)C(N1CC(O)(CO)C1)=O C1(NC(c2ncn(CC)c2)=O)CCCC(CC(=O)NOCCC(F)F)C1 C1(C(N2CC(n3ccnc3)C2)=O)CCC(O)CN1C(c1ccc(C(F)F)o1)=O C#CCCC(=O)NN1CCCC1C(N1CC2(CCC(=O)NC2)C1)=O N1(C(C(CC)F)=O)CC(NC(C2(COC)CCNC2=O)=O)C(C)C1 C#Cc1ccnc(C(=O)NC2CC(C(=O)NOCC(N)=O)C23CCC3)c1 C1(CN(CC(O)CN2CCCCC2)C)CCCCC12CC2 c1(C(N2CCOCC(CCNC(=O)COC3CC3)C2)=O)cnn2cc[nH]c(=O)c12 C1(NC(C(C)CC2CCC2)=O)CC2CCC1N2C(c1ccc(-c2ccco2)s1)=O N1(C(=O)OCC)CCCC(NCCCC2=CN2)CC1 CCC(N=c1[nH]c(=NC2COC3(CCC3)C2)c2ncccc2[nH]1)c1ccncc1 Cc1cc(C#N)cc(C(N2CCCCC2CCNC(c2cc(Br)no2)=O)=O)n1 c1(CC(C)NC(c2cc(CC)[nH]n2)=O)ccccc1Br CCC(O)CC(=O)N1CCCC1CCCNC(=O)CCc1cnn(C)c1C N1(C(c2c(CCC)nco2)=O)CC2CCCC(C1)N2C(C1CCS1(=O)=O)=O C=CC1(C(=O)NCc2cnc(C)c(C)c2)CCN(C(c2ccc(=O)n(C)c2)=O)C1 C1(NC(C(CC(C)C)C)=O)CN(C(c2cccc(CCO)c2)=O)CC(F)(F)C1 N1(C(CN2CC(CC)C2)=O)CCOCC1CCNC(=O)CNc1ccc(O)cc1 c1(CC)cc(-c2nc(CC(C)OC)nn2-c2ccc(F)cc2)cc(Cl)n1 c1(CCC)cc(C(=O)N(CCNC(=O)CCc2cccc(C)c2)CCOC)n(C)n1 CCCC(CCCNC(c1cc(C)n(C(F)F)n1)=O)NC(=O)CCN(C)CCOC Cc1cc(CCCNC(C2(CNC(C3COC3)=O)CCOC2)=O)cc(C)c1 C1(CC#C)(C(=O)NCC2CCCN2C(=O)C(C2CCOCC2)OCC)CCCC1 c1(CN(CCNc2cnn(-c3cccnc3)c2)CC)ccc(F)cc1Br N1(C(C(CNC(C(C)=C(CC)C)=O)C)=O)CC2CC(O)CC1C2 c12nc(cc(O)n1)N1CC(O)(C1)CCN2.C(=O)(C(C)OCC1CC1)OC CN1CCC(F)(C(=O)OCc2ccc(CN(C)C)cc2)CC1 c1(OC)cc(C(=O)NC2CCCC(NC(C3CCSCC3)=O)CC2)cc(F)c1C#N C12(C(=O)NCCC3CN(C(=O)CC(F)(F)F)C3)OCCCC1C2(F)F C(c1ccc(C(F)F)o1)=CC(=O)N(C)CC1(CNC(C(F)=CCC)=O)CC1 C12(NC(c3cc4n(c3)CCOC4)=O)CCCC1N(C(=O)C=CC=C(Cl)Cl)CCC2 c1(C(=O)NC2(C)CC(NC(C3CCNC3=O)=O)C2)cccc(OCC(F)(F)F)c1 C1(CC)CN(C(c2ccccc2C(C)=O)=O)CCN1C(=O)C(CN(C)C)C(C)C CCCCC(C(=O)N(CC(CC)NC(c1cn(C)ccc1=O)=O)C)NC(=O)NC c1(C(N(C2CCN(C(c3c(C)ccnc3)=O)C2)C)=O)cc2c(F)ccc(F)c2[nH]1 C(=O)(CCCC(F)(F)F)N1C(C(N(CCCC)C)=O)C(CC)CC1 Cc1nn(C)cc1CC(N1CCCC(C(N2CC=CC2C(=O)N(C)C)=O)C1)=O c1(C(CC)C(=O)NCCC(O)CNC(c2ccn(C)c2)=O)ccc2c(c1)OCO2 C(=O)(C(C#N)CCC)N1CCC(CC#C)(C(N2CC(SCC)C2)=O)C1 C12(C(N3CC(C(C)NC(=O)CS(C)(=O)=O)C3)=O)CCOC1CC(=O)NC2 c1(CC(N2C(CCNC(C(CC)C)=O)CSCC2)=O)ccc2nonc2c1 C(=O)(C#CC1CCOC1)NCCC(C)NC(CCOC)=O C=CCCCC(C(=O)NC1C=CC(C)(C)CC1)NC(c1ccc(C#N)c(C)c1)=O C(c1c[nH]cn1)=C(C(=O)N(CC(C)N(C)C(c1cnc(O)s1)=O)C)F N1(C(COCc2n(C)nnc2)=O)CC2CCC(C1)C2CNC(c1cc(C#N)cs1)=O c1(C(=O)NC2CCOCC2NC(C2CC=CCO2)=O)n[nH]c2c1COC2 C=CCCC(C(=O)N(C)CC1OCCC1(C)C)NC(c1ccc(Cl)o1)=O C1(C)(NC(CC2(OCC)CCC2)=O)CC(NC(=O)COC2CCC2)C1 c1(OCC)cc(CNC(=O)C(CC)N2CCCC2=O)on1 Cc1nc(O)nc(O)c1CC(=O)NC1CCCCN(C(=O)CCc2ccsc2)C1 N1(C(c2ccc(OC)nn2)=O)CCCCC(NC(C2C(C)C2C)=O)C1 C(=O)(C(CO)C(F)(F)F)NCC1CC(NC(c2ccc3ocnc3c2)=O)C12CCC2 C(=O)(CC1=CCCCC1)N1C(CCNC(C2CNC(=O)N2)=O)CCC1 c1(CCC)nnc(S)n1CC(=O)NC1(C)CC(NC(=O)C(C(C)C)SC)C1 c1(NC(c2cc(Br)ccc2F)C)ccc2nonc2c1 N1(C(c2c(F)ccc(C)c2)=O)CCC2(NC(C3CCCC34CCC4)=O)CCCC12 N1(C(c2n(CC=C)ccc2)=O)CCCC12CCN(C(c1ccc(C)nn1)=O)CC2 N1(C(c2ncn(CC)n2)=O)CC2CC2(C(N2CCC(CCO)C2)=O)C1 c1(C(N(CC(C)O)CCNC(CC(C)OC)=O)=O)nccc2c1NCCC2 N1(C(C23C(NC(c4cnc5n4CCC5)=O)CC(CC2)C3)=O)CCC(O)CC12CC2 C=CCC(C(=O)NNC(=O)C(C)(C)C)C(C)OC(=O)C(c1ccccc1)=O CC(=O)CCCCCCC(=O)NC(c1ccccc1)CNC(C1COC(=O)O1)=O c1(C(=O)NCc2c(C(N(C)CC3CCCO3)=O)n[nH]c2)ccc(F)cc1F Cc1cc(Br)ccc1C(=O)NC1CC1C(N1CCOC(C(F)(F)F)C1)=O C1(CNC(=O)Cn2cnnn2)CCN(C(c2cn(CCO)nn2)=O)C12CC2 C1(C(=O)OC)CN(C(c2ccccc2OC)=O)CCC1NC(c1cccc(Br)n1)=O CCC(C)C(C)(c1nnnn1C1CCCC1)NCCc1nncn1CC c1(NC(C2CSCCN2Cc2cccnc2F)=O)ccnc(C(F)(F)F)c1 c1(NC(CC2C(C)(C)C(O)C2)=O)c(N)cc(Cl)nc1Cl.C12(C)CCN(C1)C2 CC(C)CC(C)C(=O)NCC1CCCN1C(C1(c2nc(F)ccc2Cl)CCC1)=O C12(CNC(CCCOCC=C)=O)CCCC1CCN2C(=O)C1=CCCOC1 C1(C)(CC)C=C(C(=O)NCC(C)(C2CC2)NC(c2cccc(C3CCC3)c2)=O)C1 N1(C(CCC=C(C)C)=O)CC(NC(C2CC(=O)N(C)C2)=O)C(CC2CCCC2)C1 Cn1ncc(Cl)c1CNC(=O)C(O)CCNC(c1csc(Cl)n1)=O c1(N2C(C(=O)NCCC#N)CC3CC32)ccc2nccnc2n1 CC1CC2CN(C(=O)CCN(S(=O)(=O)c3ccc(Br)cc3)CCCN(C)C)CC2N1 c1(C(CNC(=O)NC23CC(C(C)(C)O)(C2)C3)NC(CC(C)C)=O)ccc(F)cc1 c1(C(=O)NC2CC(F)(CNC(c3n(OC)cnc3C)=O)C2)cnc2cccnn12 c1(C(C)C)ncc(C(=O)NCCN(C(=O)C(C)OC2CC2)C(C)C)[nH]1.C(C)(C)C C1(CC(=O)N(c2ccnc(CC3CC3)n2)CC2CCNC2)CCCC(=O)N1 c1(C(=O)NCC(C)(C)NC(C(C(C)C)CC2CCCC2)=O)ccc2cnnn2c1 N1(C(c2cc(OCC)no2)=O)CCN(C(c2ccc3c(c2)CC3)=O)C(CF)C1 N1(C(C2(COC)CCC2)=O)CCCC(N(CC(O)C(F)(F)F)C)C1 CC1(C(=O)NCCC(O)CNC(=O)C2=CCSC2)Cc2ccccc2NC1=O c1(OC)cccc2cccc(C(=O)N(C3CCN(C(=O)C(C)CC(F)F)C3)C)c12 Cc1cccc(C)c1CC(=O)NC(C)CNC(c1csc([N+](=O)[O-])c1)=O N1(c2nnc(C#N)s2)CC2CCC1C1CN(C(c3cc4ccncc4s3)=O)CC21 N1(C(CC2C(C)OCC2)=O)CC(C2CC2)(C(=O)NCc2ccn(C)c2)C1 c1(C(=O)NCC(C)NC(C2(COCC)CC2)=O)c(F)cncc1Br c1(C2(N3CC4CC(F)CC4C3)N(C(C(CC=C)C)=O)CCC2)cccn2cncc12 c1(C(F)(F)F)ccc(C(O)CF)cc1.N(CCN)(CCN(C)C(C)=O)CC N1(C(c2nscc2Br)C(=O)NCc2c(OC)cccc2)CCc2nn[nH]c2C1 C(Cc1cnc[nH]1)(C(=O)NCC1(C(=O)O)CCC1)NC(C1CSC1)=O N1(CC)CCN(C(C2CC(C)CN(C(=O)CN=[N+]=[N-])C2)=O)C(C)C1 C(CN=c1[nH]c(N2CCOCC2)nc2c1COCC2)OCC(=O)NCC1CCC1 C1(NC(C2N(C)CCN(C(c3cc(C)nc(C)n3)=O)C2)=O)Cc2ccccc2C1 N1(C(C2C(C(=O)OC)CC2)=O)CC2CN(C(=O)C=Cc3nccs3)CCC12 C(C(CO)(CO)NC(C1CCCCN1S(C)(=O)=O)=O)NC(c1cnc(C)o1)=O C#Cc1ccc(F)cc1C(=O)NC1(CCNC(=O)C(C)(C)C(=C)C)CCC1 Cc1cnc(C(N2CCC(C(C)NC(C3(F)CCCCC3)=O)C2)=O)cc1Br c1(CCC(N2CCC(C)CC2)C)ccn2c(C(F)(F)F)nnc2c1 C#CC1CCCN1C(=O)CNC(=O)OC(C)(C)C.c12oc(cc1C)[nH]c2=O c1(C(=O)NCC2(C)CCCN2C(=O)COCC2CCOC2)ccsc1S(N)(=O)=O c1(N2C(C3CN(C(C(N4CC(C)C4)C)=O)C3)CCC2)ccc(C#N)cn1 Cn1nc(C(C)(C)C)cc1C(=O)NC1(CNC(=O)CC2COCCO2)CCCC1 N1(C(Cc2ccc(C)o2)=O)CCC2(CC1)CCN(C(c1sc3nccn3c1C)=O)C2 N1(C(C(C)C2CCCO2)=O)CCC(CCN(C)Cc2csc(=N)[nH]2)CC1 c1(CC(=O)Nc2cccc(NC(=O)CC3CSCCS3)c2)cccc(Cl)c1 C1(CCC)CN(C(c2cn(C)nc2C)=O)CCN1C(C1C(F)(F)C12CCC2)=O CCC(C)CCCCC(=O)NC(CC(C)C)C(=O)N(C)CC1CCOCC1 c1(C(C(=O)NCCC)N(N2CC(OCC)C2)C)ccc(C(F)F)c(F)c1 c1(N2CCC(N(C)C(c3ccc(=O)n(C)n3)=O)C2)ncn(C)c(=O)c1Br N1(C(C(C)OCC)=O)CCN(C(=O)Cc2cnc[nH]2)CC1c1ccccn1 C1(CNC(=O)NC(C)(C(F)(F)F)c2ccccc2)CCC2COCCC2C1 C(CCCCN=C(NCc1cnn(C)n1)NC(C)C1CC1)NC(C)=O CCC(C(=O)NC1C=CC(CNC(C2(C3(C)OCCO3)CC2)=O)C1)C(C)O C1(C)(NC(C(C2CN(C(CC3(OC)CCCC3)=O)C2)O)=O)CC2CCC1C2 N1(C(c2ccc(NC)cn2)=O)CC(NC(C2CC2F)=O)CC12CCCCC2 C1(C(=O)NCCC2CCCN(C(COC)=O)C2)CC(c2ccc(Cl)cc2Cl)=NO1 c1(C(=O)NC2(CO)CCCN(C(C(C)(C)OC)=O)C2)ncc(F)c2ccccc12 C1(NC(=O)C(F)OC(F)(F)F)CC(=O)N(CC2CC2)C1.O c1(C(=O)NC(C2CCCCN2C(=O)C=CC(F)(F)F)C)n[nH]c2c1CSCC2 C=CCC(C(=O)NCCCC(C)(C)NC(C1CC12CC2)=O)NC(C)=O C1(NC(CC)=O)COCC1NC(C1(COC)CC1)=O c1(C(N2CCC3CN(Cc4c(F)cccc4Cl)CC23)=O)ccc2ncccc2c1 c1(CC)cc(C(=O)NCCC2(NC(c3ccc(F)s3)=O)CCCC2)ccc1Cl N1(C(CCCC)=O)CCCC(F)(CNC(C2CCCC(C)C2)=O)C1 C(CN(C(=O)CCCSC(C)(C)C)C)(CO)(CO)NC(C(C)=C1CCC1)=O C1(C(N(C)CCNC(C2CC(C)(C)CO2)=O)=O)CN=C2N=CNN2C1 CCC(CC(=O)NCC12CC(C1)C(NC(c1nc(O)sc1C)=O)CO2)C(C)(C)C C=CCCCC(C(=O)NC)NC(=O)CS(=O)(=O)NC.C(CF)N Cc1ccc2oc(NCC3CCCCN3C(c3cccc(N=[N+]=[N-])c3)=O)nc2c1 C1(NC(c2ccc(Cl)cc2)=O)CCC2(C1)CN(C(c1ccnc(F)c1Cl)=O)C2 C1(CC=C)(NC(=O)C(CCC)NC(C)=O)CCN(C(=O)C(=O)NCCOC)CC1 c1(C(C)C)ccc(C(c2nnnn2C2(C)CCCC2)NC2CCC2(F)F)c(F)c1 C(=O)(C1Cc2c(Cl)cccc21)N(CCN(C(C1(COC)CC1)=O)C)C C#CCCC(O)C(=O)N1CCC(C(=O)N(c2ccc(F)cc2OCC(C)C)CC)C1 C1(C2(C(C)NC(CC)=O)CC2)CCCN1C(=O)CCN1CCOC1=O N1(CC(=O)N(C2CC3CC2CN3)C(C)(C)CN2CCNC(=O)C2)C(=O)CCCC1=O c1(C(N(CC(C)NC(C2(C)CCCN(C)C2)=O)C)=O)cn(C)c(=O)n1C Cc1ccccc1CCC(N1CCC(CNC(C2CC2c2ccccc2)=O)C1)=O NC(=O)CC(O)C(=O)NC1CCC(NC(=O)Nc2ccnn2CC(F)F)C1 N1(C(C2C(C)(C)CCO2)=O)CCC(O)CC1C(N1C2CCC1COC2)=O N1(C(C2CC3N(C(C4CC(O)C4)=O)C(CC3)C2)=O)CC(C2CCCCC2)C1 c1(C(=O)NC2CC(NC(C3C(CC)OCC3)=O)C2)cc2ncccc2o1 C1(NC(c2nc(C(C)C)oc2)=O)CCCCN(CC2CCCN(C)C2)C1 c1(C(=O)NC(C)CN(C)C(C2(C)CCN(C)C2)=O)csc2cccnc12 C(C(=O)NCc1ccccc1)(C(C)CC1CCC1)N(C(CC)C)C1CC1 Cc1c(NCCCC2CCOC2)nc[nH]c1=NCc1cc(C(F)(F)F)nn1C C=CCC(C(=O)NCC(=O)N(C)NCC(C)C)C(C)C.CCC c1(C(c2n(CC(=C)C)nnn2)NCc2cc(Cl)ccc2Br)ccc(Cl)c(C#N)c1 C12(CNC(c3ccn(C)n3)=O)CC1CN(C(C1CC1c1ccsc1)=O)C2 c1(OC)ccc(NC(=O)NCC=CCNC(C)=O)cc1N1CCCCC1=O c12cccc(n1)S2.C(CCC(c1nnnn1C1CC1)NCC=C(C)C)OC C12(CO)CCOCC1CN(c1ccnc(-c3cn4cc(Cl)ccc4n3)n1)C2 Cn1cc([N+](=O)[O-])c(CC(=O)NC2CCCCC2CN=c2ncc(Br)c[nH]2)n1 C1(C(N2C3C(NC(CCOCC)=O)CC(CC3)C2)=O)CC(C)c2nc(C)cn2C1 c1(C(N2CCC(C(=O)OC)C2C)C(=O)NCC(=C)C)cc(F)c(OC)cc1Br c1(NC(c2ccc(Sc3ccncc3)cc2)=O)ncc(F)c(I)c1F c1(C(N2CC(C(C)NC(C(Cc3c(C)n[nH]c3C)C)=O)C2)=O)c(O)ncnc1O c1(C(=O)NC2CN(C(C(COC)(C)C)=O)C2)cc2c(Br)[nH]nc2s1 C(CC)(C(=O)NC1CC(C)(NC(c2cnc(C(C)(F)F)s2)=O)C1)OCC Cc1nc(-c2cnn(C)c2)oc1NC(c1ccccn1)=O C1(C(=O)NCC2C(NC(=O)CN3CCCC3)CCC2)CCC2CC1CO2 C1(COC)(NC(c2cnn(-c3ccccc3)c2)=O)CN(C(C2CC2(C)C)=O)C1 c1(C(N2CCC(O)(CNC(c3onc(C)c3C)=O)C2)=O)ncnc2ccsc12 c1(C(N(C)CC2N(C(C(CC3CC3)OC)=O)CCC2)=O)nccc2[nH]ccc12 N1(C(CC)=O)CCOC2(C1)CN(C(=O)C(C)(C)C)C2.Cc1nc(C=O)c(=O)[nH]c1C c1(C(=O)NC2CCC(CNC(CCn3ccc(C)n3)=O)C2)cccc(C(N)=O)n1 C1(C(=O)NC2C3CN(C(COC4CN(C(C)=O)C4)=O)CC32)CCCCC(=O)N1 c1(C(=O)NC)cccc(C(=O)NC2CC2CNC(c2cc(C)c(Br)o2)=O)n1 C#CC1CCCN(C(=O)CC2CCCN(C(=O)CCC=CC(C)C)C2)C1 C1(CNC(C(C)C2CCCC2)=O)CN(C(c2cc(Cl)nnc2O)=O)CCC1(C)C C1(NC(CC=C)=O)CCC2(CCN(C(c3cc(-c4ccncc4)no3)=O)CC2)C1 CCCCC(C(=O)N1CCCC1CN(C(=O)CC1CC1C)C)NC(N)=O c12cccc(c1)CS(=O)(=O)N2.c1(C(C)=O)c(-c2ccsc2)noc1C N1(C(C(CC)CO)=O)CC(C2CCCN(C(c3cnn(C4CCC4)c3C)=O)C2)C1 C1(NC(=O)NC)CCN(C(C2(NC(C3CC(F)C3)=O)CC2)=O)CC(C)(C)C1 CC1(C)CN(C(C2CCOCC2)=O)CC1C(=O)NCc1c[nH]ccc1=O c1(CC)o[nH]c(=NC(=O)C2=NOC(c3ccccc3)C2)c1C CC(CCc1ccc(F)cc1)C(=O)N(C1CN(C(=O)COc2ccsc2Cl)C1)C Cc1cc(C(=O)NCC2(CNC(c3c[nH]ccc3=O)=O)CCC2)ccn1 C(=O)(CCC(C)(C)C#N)N(CC(C(=O)NC(C)Cn1cncn1)(C)C)C C1(C(C2N(C(CCC)=O)CCC2)=O)CCCN(C(=O)CCC#N)C1.C1C(=O)N1 C1(NC(CCOC)=O)CC(NC(=O)C(F)(F)n2cc(Br)cn2)C12CCC2 c1(CNC(C2(F)CCN(C(=O)CCCC3CCC3)C2)=O)cccc(O)c1 C(=O)(CC(C)(C)CC)N1CCC(CC=C)(NC(C2CCN(CCC#C)CC2)=O)C1 C1(CN(CCC#C)C)CCN(C(=O)CC2CCCC23CC3)CC1C N1(C(N(CCCC(=O)OC(C)(C)C)C)=O)CCOC2COCC12 C=CC(C)(C)CC(=O)N1CCC(N(C(c2sccc2OC(F)F)=O)CC2CC2)CC1 C(=O)(C1=CS(=O)CCC1)N1C(CN(C(C2(COC)CCCO2)=O)C)CCC1 C(N=c1[nH]nc(COC)s1)C1(CCNC(C(C2CCCOC2)OCC)=O)CC1 N1(C(C2(CNC(C3CC(F)(F)CS3)=O)CC2)=O)CCOC(C2CC2)C1 c1(C(N(CCC(C)NC(c2cc(OC)n(C)n2)=O)C)=O)ncc2[nH]ncc2n1 N1(C(c2c(CC)occ2)=O)CCC2(C1)CN(C(c1cccc(F)c1C)=O)C2 c1(SCCNC(=NCC)NC(C)CC)cc(F)cc(F)c1 C1(CNC(C2CN(C)C(=O)C2)=O)CN(C(C2CCCC2)=O)CCC12CCOCC2 CS(=O)(=O)C1(NC(C2CC(n3cc(C4(CO)CC4)nn3)C2)=O)CC(=O)C1 C(=O)(C(C)(C)S(C)(=O)=O)N(CCCC(=O)NC1CCCC(N(C)C)C1)C CCC(C)C(O)CNCc1cn(-c2cccc(Cl)c2)cn1 Cn1ncc(C(=O)NC2CCC(CC(N3CCCC3C(N)=O)=O)C2)n1 C1(CCC)(NC(=O)CN2CCNC(=O)C2)CCN(C(C23CC(C)(CO2)C3)=O)CC1 C(C(CC(C)C)C(=O)NCC1CCC(NC(c2ccc3nsnc3c2)=O)C1)OC C1(CCCC)CCC(C(=O)NC(C)CN(C(=O)CNC(=O)OC)CC)CC1 N1(C(C(C)C2CCCO2)=O)CC2CC(C1)CN(C(=O)Cc1csc(C3CC3)n1)C2 C(CC1=CCN(C(=O)CN2CCC(C)C2)CC1)NC(c1c(CC)nn(C)c1Cl)=O CC1CC(O)CN1C(=O)C(C)N(C(c1nc[nH]n1)=O)C1CC1 Cc1c(N(C(=O)C(C)C)C(=O)Cn2cc(C(C)O)nn2)cccc1F C(CCC(=O)N(C1CC1)CC1CCCN1C(C1CC1OC)=O)OCC=C Cc1ccc(C(=O)NC(CNC(=O)CC(C)NC(C2CCCC2)=O)C2CC2)s1 Cc1c(NCC(N(C)C)C2CC2)ncnc1NCCCCC1CCCC1 Cc1cc(C(=O)NC(C(=O)NCC(Cl)=CCl)C2CCCO2)ccc1F c1(C2(NC(=O)NCC3CCC(CCC(=O)O)CC3)CC2)cccc(O)c1 c1(C(=O)NCC2(NC(=O)CC3CCC4CC34)CCC2)cc(F)cc2cnccc12 C1(C(C)OC(c2cnn(C)c2-c2cnccn2)=O)CCCC(F)C1 c1(CCC)cccc(C(N2CCCC(CNC(=O)C(C)(C)c3ccns3)C2)=O)c1 CC(C)S(=O)(=O)C(C)C(=O)NCC(=O)NCc1cn(CC2CCCC2)nn1 C1(C(=O)NCCNC(C(C)OC)=O)CCCN(C(=O)Cc2cscn2)C1 C1(C(N2CCC23COC3)=O)CS(=O)(=O)C1c1ccccc1 C(=O)(C1CCCc2c1ncn2C)N1CCC(C)(NC(COC(C)=O)=O)CC1 N#Cc1cccc(CC(=O)NC2CCCN(C(=O)C=Cc3cncc(F)c3)C2)c1 c1(CC(N2CCC(COC)(NC(c3cscc3C)=O)C2)=O)ccccc1[N+](=O)[O-] N1(C(C(C(C)C)=O)=O)CC(NC(c2ccc(NC=O)cc2)=O)CC12CCC2 c1(CC)ccccc1NC(CCN(C(C)CC1CCNC1=O)C=O)=O.C(C)(C)(C)O C1CCCCC(=O)NCCN1C(=O)CC1CCCCC1C.N1(CC)CCCC1 C=C1CC2(C1)CC(C(=O)NCC1(F)CCN(C(C3(N(C)C)CCCC3)=O)C1)C2 CC(C)N(O)C(=O)C(=O)NC1(C)CC(NC(C2CCC(CCO)CC2)=O)C1 C1(NC(C(C(CC)C)N(C)C(C2C(C)(C)C2(C)C)=O)=O)CCn2cncc2C1 N(C1=NCC(CCc2ccccc2)N1)=CCCC Cc1coc(C)c1CNC(=O)Cc1csc(NC(=O)Cc2ccccn2)n1 N1(C(C2CCCN(C(C(C)SCC)=O)C2)=O)CC=C(C(C)(C)C)CC1 N#CC1(C(=O)N(CCC(=O)NCC2(n3cccn3)CC2)C2CC2)CCOC1 C1(CNC(C2COCCC2NC(=O)CSc2nc[nH]n2)=O)CC2C=CC1C2 C1(CNC(C2OCCN(C)C2)=O)CCN(C(=O)CN2CCOC2=O)C1(C)C N1(C(c2nc(C)[nH]n2)=O)CCC2OCCN(C(=O)CCc3ccon3)C2C1 c1(C(=O)NC(CN(C)C)C(=O)NCC2CC2)cccc(F)c1F C1(CNC(=O)OC(C)(C)C)(N(C2CCC23CCCC3)C2CC2)CC2CCC1C2 C1(F)(C(=O)NC2C(NC(c3cnn(C4CCCC4)c3)=O)CC2)CC12CCCCC2 N1(C(CC)=O)CCC(CO)(NC(=O)C(CC)NC(=O)C2CC2)C1.c1(N)ccccc1 N1(C(c2cc(CC)no2)=O)CCOCC(C)(CNC(=O)Cc2cccc(F)c2)C1 C1(C(=O)NC2(C)CN(C(c3cn(CC(F)(F)F)nn3)=O)C2)CCC(=O)CC1(C)C c1(C(CNC(CSCC)=O)C)ccccn1.C12(CCC1)C(=O)N2 Cc1ccc2cccc(C(N3CC(CNC(=O)Cn4cncn4)C(C)C3)=O)c2n1 c1(OCC)cccc(C(=O)NC2CCC(NC(=O)CSc3ccc(C)cc3)C2)c1 C1(CC)CN(CCC2C=CCC2)CCN1C(C(=O)NC(C)(C)C)c1ccco1 C1(OC)CN(C(=O)Cc2cc(C)on2)CCC1NC(c1cnccc1C)=O CCC(F)(F)C(=O)N1CCC(C)(NC(c2cnn(C3CCC3)c2C)=O)C1 c1(C(COC(c2cc(C)on2)CC)=O)ccc(Oc2ccc(F)cc2)cc1 Cc1cc(OCC(N2CC(CNC(C3CCOC3)=O)CC2C)=O)c(C)c(C)c1 CC(C)CCC(F)C(=O)N1CCC(C(N2CC(O)(CCO)C2)=O)CC1(C)C C(CCC1CC1)(C(=O)NC1(CCF)CC(O)C1)NC(COCCCN(C)C)=O Cc1ccc2n1CCN(C(C(=O)Nc1ccccc1)c1cncs1)C2C c1(C(=O)NCC2C(C(=O)Nc3ccccc3F)CCC2)cccc2ccnn12 n1(CCOC)cc(C(=O)NC23CC(C2)N(C(=O)C(C)O)C3)c2ccccc12 c1(CCCOCCN(C)CC)ccccn1 c1(C(=O)NCc2c(C)ocn2)c(CNC(c2ccnn2C(F)F)=O)nnn1C n1(C(C)C)ncc(C(N2CCC(OCCNC(=O)CC=C(Cl)Cl)C2)=O)n1 Cc1cc(F)cc(C(=O)NCCC(C)N(C(=O)C(CO)C(C)(C)C)C)c1O C1(COC)(NC(=O)C2=CCOC2)CCN(C(c2cncc(C)c2)=O)CC1 Cc1nn(C)c(=O)c(C(N2CCCC(CO)(NC(=O)CC3CC(C)C3)C2)=O)c1C c1(CCC)ncc(C(=O)NC(C)(CNC(c2ccn(C3CC3)n2)=O)CO)s1 N1(C(c2cc(CNC(CCC#C)=O)[nH]n2)=O)CC(F)(F)CC1CO N1(C(C(C)OCCC=C)=O)CC2CC(C1)N(c1nc(SC)ns1)C2 Cn1nc(CNC(=O)Cc2cnccn2)cc1C(=O)NCC1CC1(F)F c1(N2CC(N(C)C)C(C3CC3)C2)nc(N(CCC(N)=O)C)nc2cccnc12 c1(C(N2CC(F)(CNC(Cc3c(C)nn(C)c3Cl)=O)C2)=O)ccc2ncn(C)c2n1 C1(C)(NC(CNC(CC)=O)=O)CCN(C(C2CC(=O)C2)=O)CC1 N1(C(C(CN(CC)CC)F)=O)CC2CN(C(=O)C3=NNC(=O)CC3)CCC12 C(=O)(CCCCC1CC1)NCCNC(C1C(CN(C)C)C1)=O c1(C(N(CCCOCCN(C(C(C)C(F)F)=O)C)C)=O)scc2c1CCCC2 CC(C)C(O)C(=O)N(C1C2CN(C(c3ccccc3-c3ncc[nH]3)=O)CC12)C c1(C(=O)NC(CN2CCN(C(C(C)C#N)=O)CC2)(C)C)cc2c(nc1O)CCC2 N1(C(c2c(CC=C)cccc2)=O)CC2(COC(CNC(C3(CCF)CC3)=O)C2)C1 N1(C(C=C(C)C(C)C)=O)CC(CNC(=O)COCc2cccnc2)C2CC12 c1(CNC(=O)COC2CCCCC2)c(Cl)n[nH]c1C.C12(COC)CN(C1)C2=O CCC(COC)C(=O)N(CCN(C(=O)C(C)(c1ccccc1)N(C)C)C)C(C)C N1(C(c2cccc(CSC)c2)=O)CC(C)(C)CCC1CNC(=O)CCCC(F)F N1(C(CNC(c2c(OCC)cccc2)=O)=O)CCN(C(C)=O)CCC1C C1(NCCCC)CCCCC1CNC(c1nnnn1C1CCOC1)C1COC1 c12ccc(cc1)CNC2.c1(C(=O)OC)ccsc1NC(=O)CN(C)C(C)C N1(C(c2[nH]cc(C(N)=O)c2)=O)CCC2(CC1)CCN(C(=O)CC=C(Cl)Cl)CC2 C(C(=O)NN1CC2CCCC2C1)n1cc(C2CCCC(C)(O)C2)nn1 C1(O)(C(C(=O)N(CC(F)Cl)C)NC(C2CS(=O)C2)=O)CCCCC1 C(=O)(C(O)CC(C)(C)C)NC(C)C(CO)NC(c1ocnc1C(F)(F)F)=O CC(C)(CC(=O)N1CCC(CO)(NC(C2CCSCC2)=O)C1)C(F)F N1(C(CC=C=C)=O)C2CCC(C2)C1CNC(c1ccc(N)c(F)c1)=O Cn1c(C(=O)NCC(C)(C)OCC(=O)NCC#CC(F)(F)F)nnc1S N1(C(C2CCC(=C)CC2)=O)CC(CNC(C2NC(=O)OC2C)=O)C2(CC2)C1 C(=O)(C(CC(C)C)NC(c1ncccc1Cl)=O)NC(CCOC)COC C1(C(=O)NCc2oc(C(N(C(CO)C3CC3)C)=O)c(C)n2)CCCC12CCC2 c1(C(N2CCN(C(C(C)=CC)=O)CC2CC(=O)NC)=O)ccc2c(c1)nnn2CC C1(C)(C(N(CCN(C(C(CSC)C)=O)C)C(C)C)=O)CC(=O)N(C)C1 N1(C(CC=CCC)=O)CCC(C)(CC(=O)NCC2(C(C)C)CC2)C1 C1(NC(C(C(C)C)n2cncn2)=O)CCCCN(C(c2ncccn2)=O)C1 CC(C)CC(CC(C)C)C(=O)N1CC(C(n2cc(CCC(C)(C)O)nn2)C)C1 C(=O)(C(CC=C(Cl)Cl)OC(c1cn(C)nc1-c1ccccn1)=O)OC(C)(C)C N1(C(=O)Nc2cccc(C(C)C)c2)CCN(C(C)(C)C)CC1CC#N c1(C(C)NC(Cc2cccc(C)c2)C)cccc([N+](=O)[O-])c1 C12(C(=O)NCC3C(CNC(=O)CCC4CCCCC4)C3)CCCC1CCC2 c1(OC)cc(C(=O)NC(CO)C(C)NC(=O)CC2CC=CCC2)cc(Cl)c1O c1(C(=O)NC(C#C)C(C)C)cc[nH]c2nccc1-2 c1(OC)cc2c(cc1C(=O)NC1CC3CC(OC)C3C1)CCC2 c1(CC)ccc(NC(N2CCC([N+](=O)[O-])CC2)=O)cc1[N+](=O)[O-] c1(CC)sc2ccccc2c1NC(=O)CSc1ccc(C)cc1C CC(C)CC(C(=O)OC(=O)C(c1ccc(F)cc1)CO)N(C)C C1(CC=C)(NC(=O)CCOCC(F)F)CCN(C(=O)C(O)CSC)C1 CC(C)CCC(C(=O)N1CCC=C(F)C1)NC(=O)CC1CCN(C)C1=O c1(C(=O)NCCC(C(C)C)NC(CC=C)=O)cc(F)c(Cl)cc1F c1(OC)noc(C(=O)NCCCCN(C(=O)CNC(c2ccccc2)=O)C)c1Br CC1CCN(C(C2C=CC=CC=C2)=O)CC1CNC(c1ccc(C#N)[nH]1)=O c1(C(N2C3CCC2CC(OCCC)C3)C(=O)NCC)ccc2c(c1)CC(C)(C)O2 CC1(C)CC(NC(C2(C)CC2(F)F)=O)CCN(C(=O)CC2(O)CCCCC2)C1 C1(OC(C2(CCC)CCCC2)=O)CCN(C(c2cc(CSC)cn2C)=O)CC1C c1(C(C)F)cccc(NC(C2CC(CCNC(C34CC(C3)C4)=O)C2)=O)c1 C1(CCC)CN(C(C2CCC3(CCC3)C2)=O)CCN1C(=O)CN1CC2CC2C1 C=CC(C)(CC)C(=O)NCC(C1CCCC1)NC(=O)C(C)Cc1ccncc1 C1(C(N2CCC(c3ccc(F)cc3)CC2)=O)CCN(c2nnc(C(F)(F)F)s2)CC1 c1(C(=O)NC2CC3(NC(=O)C(O)C4CCC4)COC2C3)cc(O)c2ccsc2c1 c12cc3cc(cc(Br)c3o1)CNC2=O.c1(C(C(=O)OC)SCC)ccccc1F C(=O)(C(CNC(c1cccnc1)=O)(CC)CC)NCC(=O)N(C)CC N1(C(C2(CC3CC3)CN(C(CCCC=C)=O)C2)=O)CCOC(C2CC2)CC1 N1(C(C2C(=C)C2)=O)CC2CC(C1)C(CO)C2NC(=O)C(C)(CC)CC c1(C(N2C(CC(=O)Nc3c(C)ccc(Cl)c3)CCCC2)=O)cc(Cl)cc2cc[nH]c12 C12(CNC(C3(CC#C)CCOC3)=O)CC(CO1)N(C(=O)CCC(C)C)C2 C1(NC(CC)=O)CC(OC)CN1C(=O)C(C)OCC(C)C c1(C(=O)NCCN(C(C2CNC(=O)N2C)=O)CC)ccc(C(C)=O)cc1 CC1(C(=O)Nc2c(C#N)cnn2C(C)(C)C)CCN(S(=O)(=O)c2ncc[nH]2)CC1 N1(C(CCc2onc(CC)n2)=O)CCOC(CNC(=O)CC(C)N2CCCC2=O)C1 N1(C(=O)COc2ccc(CO)cc2)CC2CCCC2(NC(=O)C2=COCCO2)C1 C12(CNC(C3N(C(COCC(=C)C)=O)CCCC3)=O)CCCC1OCC2 N1(C(C(C=C)O)=O)CCC2CCCC12C(N1CCC2CC12)=O c1(NC(N(C(C)C(=O)NC(c2cn[nH]c2)C)CC)=O)cccc2ccoc12 c1(OC)nccc(C(N2CCN(CCN(C(=O)C(=O)NC(C)(C)C)C)CC2)=O)n1 c1(CN2C(C(=O)NCCCCCO)COCC2)ccc2nccn2c1 N1(C(Cc2ccc(C)s2)=O)CC2C(C(F)(F)F)CC2(NC(C2CC2C(N)=O)=O)C1 c1(CC(=O)NCCC(O)CNC(=O)CSC(F)(F)F)cccc(Cl)c1F C1(O)(C(=O)NCC(C)NC(C2CCCN2c2ccccc2)=O)CCSC1 N1(C(CSc2ccc(C)cc2)=O)CCC2(CCCCC2CNC(=O)CC2CC2)C1 C1(N=[N+]=[N-])(C(=O)NC2(C)CCOC2)CCN(C(=O)CC23CCCC2C3)C1 C(=O)(C1=NOC2(CCOC2)C1)NCCCN(C(CC(CC)C1CCC1)=O)C(C)C c1(CN2CC3(C(C(=O)N(CCO)C4CC4)C3)C2)ccc(Br)cc1F N1(C(C2C(CC)CCN2C(C2CC(CF)C2)=O)=O)Cc2nc(C)sc2C1 Cc1c(Cl)c(C(=O)NC2CC2CNC(c2ccccc2C(C)(C)C)=O)nn1C c1(NC(=O)C(=O)NC23CC(C(=O)C(F)(F)F)(C2)C3)c[nH]c2ccc(Cl)cc2c1=O CCCCC(C)CCC(=O)NC1CCCC1C(=O)NC1CCCN(C)C1 C1(NC(c2cc(CC)oc2C)=O)CCC12CN(C(c1ccccc1CO)=O)C2 CC1CC(CNC(c2ccc(C(C)(C)C)[nH]2)=O)CN1C(=O)CSc1nnc(S)s1 C1(NC(=O)CN2CCCCCC2)CCC(O)CN(C(C2CCOC2C2CC2)=O)C1 CCCC(CCC)=CC(=O)N(C)CC1C2CN(C(c3ncoc3CC)=O)CC12 C#CCC(CC(=O)Nc1ccc(C#N)o1)NC(=O)CNC(=O)OC c1(CCC(=O)NCC(C)NC(=O)Cc2conc2COC)ccc(OC)cc1.C(=O)OC C1(C)(C(=O)NC2C=CCN(C(c3[nH]n(CC(C)C)c(=O)c3)=O)C2)CCOC(C)C1 C(=O)(C(C(=O)N(CC(CC)NC(C1CN(CC(F)(F)F)C1)=O)C)C1CC1)OCC c1(C(=O)NCCCC(C)NC(C(CCSC)NC(C)=O)=O)c(F)ccc(F)c1Cl c1(C(=O)NC(C)CC(C)NC(=O)C=C2CCOCC2)cnc(O)c(Cl)c1 C1(NC(C2CCC(C)CC2)=O)CCN(C(=O)CC2CCOCC2)C12CCC2 c1(C(N(C)CC2(NC(c3scc(C)c3C)=O)CC2)=O)cc(Cl)ccc1-n1cncn1 C1(NC(Cn2ccc(C)n2)=O)CCC2CCN(C(=O)C=CBr)C1C2 N1(C(C(C)N(CC)CC)=O)CCC2CC12C(=O)NC12CCCC1C2 c1(NC(C2C(CNC(=O)Cc3cncs3)CCC2)=O)c[nH]c(=O)c2ccnn12 c1(NC(C(=O)NCC(C)(C)NC)=O)cc([N+](=O)[O-])ccc1Sc1ccccc1 N1(C(C2C(NC(c3c(C)scc3)=O)CCCC2)=O)CC(CO)C(C2CC2)C1 CC(C(=O)N1CC(C)C(C)(CNC(c2cc(C(F)(F)F)ncc2Cl)=O)C1)S(C)(=O)=O Cc1[nH][nH]c(=N)c1C(=O)NCC1CCCC(NC(C2(CCF)CC2)=O)C1 c1(CC)cc(NC(C2CCN2NC(C(OCC)OC)=O)=O)nn1C.C12CCN1C2=O c1(CC)ncc(C(=O)NCCCCCN(C(c2sccc2F)=O)C(C)C)[nH]1 c1(NC2(C)CC2)cc(F)c(NC(CCCC2CCCCC2O)=O)c(F)c1F Cc1cncc(CCC(=O)NC(C)(C)CNC(c2sccc2C#N)=O)c1 N1(C(C2C(C)CC(=O)N2)=O)CCCC(CO)(CNC(=O)CC=CC(C)(C)C)C1 C1(CC#C)(C(N2CC3CCC3C2)=O)CCN(C(c2c[nH]nc2Cl)=O)C1 Cc1ccc(CC(C)C(=O)N(C)CCN(C)C(C2CC23CCC3)=O)cc1 C12(C(=O)NCC(CN(CC)CC)(C)C)CC(C)(C1)OC21CCC1.C12CC1NC2=O N#Cc1ccc(NCC(=O)NC2(CNC(=O)CC3C=CS(=O)(=O)C3)CCC2)c(F)c1 c1(CNC2CC(C(F)F)NC2)cc2c3c(ccc2[nH]1)OCO3 Cn1ccc(CCC(=O)NCCCCNC(c2ncoc2C(F)(F)F)=O)n1 C1(CNC(C(CCC)(C)C)=O)CC2(CCC2)CN1C(C1CN(C)C(=O)CCO1)=O CC1CCC(NC(C)(COCCc2nn[nH]n2)c2cccs2)C1 N1(C(C(CCCC)N(C)C)=O)C(CNC(=O)CCc2ncc[nH]2)CC2COCC12 CCCCCCCCC(=O)NCC1CC(NC(CC2(C)CCCS2(=O)=O)=O)C1 c1(C(=O)NCC(C2CCOC2)NC(C=CC(N)=O)=O)cn2c(n1)CCC2 C(CCCCC(F)(F)F)NC(c1ccc(OCC)c(OC)c1)c1cccnc1 c1(NC(c2cc(OC)c(F)cc2)=O)cnc2c(c1)CN(C(C1CCCS1)=O)CC2 c1(C(N2CCN(Cc3ccc(Cl)c(Br)c3)C3CC23)=O)ccc(Br)cc1CO C(=O)(C1=CC2CCCCCC12)N1C(C)CC(NC(c2c(C)sc(O)n2)=O)C1 c1(C(N(CCOC)CCNC(c2csc(C(C)C)n2)=O)=O)nc(Cl)sc1C c1(OC)ccc2c(n1)NC(C(=O)N(C)CC1CN(C(C3CCCCO3)=O)C1)C2 N1(c2snc(CCOC)n2)CCC(O)C(C(=O)Nc2c(C(F)(F)F)ncn2O)C1 C12(NC(C=C(COC)C)=O)CCCC1N(C(=O)CSc1ccncc1)CC2 C(=O)(CCS(C)(=O)=O)NC(C)CN(C)C(c1cscc1Br)=O c1(C(=O)NCC2CCCN(C(C(CC)(F)F)=O)C2)ccc(C)c(O)n1 C1(C(=O)NCc2c(F)cncc2F)C2CCC1CN(Cc1c(C(=O)O)ccs1)C2 CCC(F)(F)CC(=O)NCCC1CC(OC)CN1C(c1csc(Br)n1)=O C1(c2ccccc2)(CNC(CSC)=O)CC12CCN(C(C1CC13CC3)=O)CC2 Nc1c(NCc2ccc([Si](C)(C)C)s2)cc(F)cc1[N+](=O)[O-] C(=O)(CCC(=O)C1CC1)N(CCCCNC(c1cnco1)=O)C C(=O)(C1=NN2CC(C)CN=C2N1)NCC1(NC(COCCCCC)=O)CC1 Cc1c(NCCN=[N+]=[N-])ncnc1NC1CC2CSCC2C1 C1(C(=O)NCC2CN(C(c3onc(COC)n3)=O)C2)CCOC2(CCOCC2)C1 N1(C(C(CC)SC)=O)CC2COCC(C1)C2NC(c1cc2nccn2c(O)n1)=O NS(=O)(=O)CC(=O)NCCC1(O)CCN(C(c2ncc[nH]c2=O)=O)C1 C12CCN(C13CC3)Cc1cn2nn1.C1(Cc2nccc(OC)c2)COCC(=O)N1C C(=O)(C1CNC(=O)c2ccccc21)NC(C1CCN(C(=O)C=CS(C)(=O)=O)C1)C c1(C(N2CCC(C)(CNC(CC=C=C)=O)CC2)=O)cccc2ncsc12 c1(C(=O)OC)cc(C(=O)N(C)C2CC2)nn1C.n12cc(nn1)CC(CO)C2 C(=O)(CCC(C)SC)NCc1c(C(=O)Nc2cc(OCC)no2)nco1 O=C(C1=CCCN(C(c2cnns2)=O)C1)NCCC1=CCCCC1 C1(NC(C(CC)c2ccccc2)=O)CN(c2ccc(C(F)(F)F)cn2)CC1C c1(CC)cc(C)ccc1C(N1CC(CCOC)(NC(=O)C(C)=CC2CC2)C1)=O CC(C)(C(=O)NCCc1cc[nH]n1)C1CCCN1C(=O)Cc1cccs1 N1(C(=O)CC2(O)CCC=CC2)CCOC(Cn2cncn2)CC1 n1(CC)nc(C(=O)NC2CCCC2CC(N2CC(NC(N)=O)CC2C)=O)c(C)n1 Cc1cc(Cl)nc(N)c1C(=O)NCC(C)(C)CNC(C1(C)C=CCC1)=O N1(CC(=O)NCCCCNC(CC2CCCC(C)C2)=O)CCCCCC1=O c1(NC(C2(C)CN(C(C3C(C(=O)OC)CC=CC3)=O)C2)=O)ccc([N+](=O)[O-])cc1I N1(C(CC)C)CCCC(C)C1.C12CCCN1C(=O)CN(C)CCCN2C N1(C(C(CC)N(C)C)=O)CC(CC(=O)NCCC(O)CO)C2(CC2)C1 C(CC(C(=O)NCCCCOC)NC(=O)C(C1CCCC1)OC)OCC.OC N1(C(CSC)=O)CC(C(N2CCC(CC(N)=O)C2)=O)CC(C)(C)C1 C1(CNC(C(CSC)C)=O)CCC2(CCC2)CN1C(=O)CC(C)(C)O Cc1cc2scc(CC(=O)NCCC3CN(C(=O)CC4CN(C)C4)CC3C)c2s1 CC1Oc2ccccc2OC1C(=O)NCC1CC1NC(=O)CCSC(F)(F)F c1(OC)ccc(F)cc1C(=O)N(C(CNC(C1CCCC(C)CC1)=O)C1CC1)C c1(-c2nc(Cn3c(C)nc(C)c3C)nn2-c2cnn(C)c2)cncc2nccn12 c1(CC(=O)NC2CC(CNC(c3ccc(C(C)(C)C)[nH]3)=O)OC2)cn2ccsc2n1 c1(CNC(C(=O)NC2C(C#N)CCCC2)=O)nnc2ccc(Cl)cn12 CCS(=O)(=O)CCNC(C1(NC(c2csnc2C)=O)CCCC1)=O CN1C(=O)CCC1C(=O)NCCC1(C(=O)NCCC2CC(C)(C)CO2)CCCC1 C1(N2C3(CN(CC)C3)C2=O)Cc2ccccc2O1.c1(CC)cnc(SC)nc1Cl C1(CC(N)=O)(NC(CCOCC#C)=O)CCN(C(C2CC(=O)N2)=O)CC1 N1(C(C2(C)ON=C(C)C2)=O)C2CCC1C(C)C(NC(=O)CCS(C)(=O)=O)C2 c1(C(C)C)ccc(C(C)CC(=O)N(CCNC(c2ccnnc2)=O)C2CC2)cc1 n1(CCCOC)cc[nH]c(=NC(=O)c2ccn3c(N)cnc3c2)c1=O C(=O)(C(CCF)C(=O)OC)N(CCCNC(=O)C(C)(C)C1CCCC1)CC C1(NC(C(F)=CC)=O)CCCN(CC(N2CC3C(C(=O)O)C3C2)=O)C1CC c1(OCCOCC)ccc(CNC(C2CCCNCC2)=O)cc1 C1(CC)CC(C(N2CCC(NC(=O)CCC(=O)NC)CC2C)=O)CC(=O)N1 N1(C(C(CCCC)NC(N)=O)=O)CC2(C1)SCCC2CNC(=O)C1=CCCC1 Cc1cc(O)nc(C)c1C(=O)N(CC(O)CNC(C1CC(C)(F)C1)=O)C C1(CC)CCN(C(=O)C(C)C(C)=O)CC1C.C1(C(=O)OC)CC(CBr)CCO1 Cc1ncccc1C=CC(=O)NC1CC(CNC(C2COCC3(CCC3)O2)=O)C1 C1(NC(c2ccc(CC)[nH]2)=O)C2CCC1N(C(c1ccc(C(C)C)c(Cl)c1)=O)C2 c1(C(N2CCC(C)(C(=O)NC)C2)C(=O)NCc2cccs2)cccc(F)c1C c1(CC)ccc(C(=O)NCCc2n[nH]cc2C(=O)N(C2CCN(C3CC3)C2)C)o1 N1(C(CN2C(C)CCCC2)=O)CCN(C(C2CC2C2(C)COC2)=O)CC1C1CC1 CCC(C)CC(C)C=O.c1(C(N2CC3(N)CC2C3)=O)ccc2occc2n1 C(=O)(C1=NN(C)C(=O)CC1)NCc1cc(C(=O)NCC2CCCCN(C)C2)no1 Cc1csc2c(C(N3C4CCC3CN(C(C3CC(=C(F)F)C3)=O)C4)=O)cccc12 N1(C(C(CCCCC)O)=O)CC2(NC(=O)C(CC)CC)CCCC2(F)C1 S(=O)(=O)(c1ccc(NCc2nccc(Cl)c2F)nc1)NCC(CCC)(C)C C(=O)(CC(C)C(C)C(C)C)NCC(=C)CCNC(c1cc2n(n1)CCCC2)=O C(=O)(C#CC1(C)CCCO1)NC(CNC(C1C(CC)CCCC1)=O)C(C)(C)C C1(C)(CC)CC(NC(c2cc(CNC(C3CCCSC3)=O)on2)=O)C1 N1(C(C2C(CC(C)(C)C)C2)=O)C2CCC1CN(C(=O)C=Cc1ccccc1Cl)C2 c1(C(=O)NCCCN(C(=O)CN2CCSCC2)C)nc(Cl)sc1Cl Cc1noc(C)c1NC(=O)C(CCc1ccccn1)NC(=O)CN(C)C N1(C(CC(CCC)NC(=O)C(C)S(N)(=O)=O)=O)CCc2cccnc2C1 Cc1[nH]c(C#N)cc1C(=O)N(C)C(c1c(F)cccc1Cl)C1CC1 N1(C(c2ccc(C)nc2)=O)CC(CNC(=O)CCCN2CCCC2)CC(C)(C)C1 c1(OC)cccc2c(C(N3CCN(C(=O)C4=CSCS4)CC3CO)=O)c[nH]c12 n1(CCC(=O)NCC(O)CO)ncc2c(Nc3ccc(OCC)cc3)ncnc12 N1(c2cc(C)c([N+](=O)[O-])cn2)CC23CCCC2(CN(C(c2ccccn2)=O)C3)C1 N1(Cc2c(OC)ccs2)c2ccccc2OCC1C(F)(F)F C1(C(=O)NC(C(CO)NC(c2c(CC)[nH]cc2)=O)C)CCc2nn[nH]c2C1 C1(CNC(C2(CN(C)C)CCCCC2)=O)CN(C)CCN1C(C1CS(=O)C1)=O C1(CNC(CCNC(=O)OC)=O)(NC(=O)COC2CCCCO2)CC(O)C1 C1(N=[N+]=[N-])(C(=O)NC(C2(CO)CC2)C)CCN(C(c2scnc2Cl)=O)C1 C1(C(N2C(CCCNC(C3(C)CC(C)(C)C3)=O)CCC2)=O)CCc2nncn2C1 Cc1ccc(C(=O)NCCC2CN(C(C3CCC4CC34)=O)CCCO2)c(C)n1 N(C1c2ccccc2CC1O)C(C(=O)NC1CC2(C1)CC(F)(F)C2)=O C#CCC(CC#C)C(=O)NCc1nnc(C2CCCN(C(C3CC3=C)=O)C2)s1 c1(C(=O)NCC(CC)NC(C2NC(=O)OC2C)=O)cnc2n1CCCC2 c1(C(=O)NCC(CC=C)NC(=O)C(C)SC)cc(C)n(-c2ccn(C)n2)c1C C1(C)(C(=O)NCC2(O)CC(NC(C=C(CC)C)=O)C2)CC(C(C)(C)C)=NO1 CC(C)(C(=O)NCCCOCCNC(C1(C)CC(O)CN1C)=O)C(F)F C1(CC(N2CCC(NC(C)=O)C2)=O)CCCCN1C(C1(CO)CCCC1)=O c1(C(N2CCN(C)C(CNC(=O)CNS(N)(=O)=O)C2)=O)nnc2n1CCCCC2 n1(CC)nc2cc1C(=O)N1CCCC21COCC=CCCC(C)C.N(C)(C)CC c1(CC(=O)NCCC(CNC(c2cc(CC)sn2)=O)O)cc(OC)ccc1Cl c1(C(=O)NC2C(CNC(CC3(C#N)CC3)=O)CCCC2)ccnc2ccccc12 c1(C(N(C2CCN(C(CC(CC(C)C)C)=O)C2)C)=O)cccc2cccc(O)c12 CC(C)(C)CC(=O)NCC(=O)NCCCNC(C)(C)CNC(C1C=CCC1)=O N1(C(Cn2nnc(=N)[nH]2)=O)CCC(O)(CNC(=O)CCc2cccc(Cl)c2)C1 C1(CN(C(=O)CNc2ccc(O)cc2)C)C2CN(C(=O)C(F)(F)CO)CC12 N1(C(C(C=CC)O)=O)CCC2(CC1)C(NC(=O)CC1CCCOC1)CS2(=O)=O Cc1nc(CNC(c2csc(CNC(C3CCCCS3)=O)c2)=O)sc1C C(CNC(=O)CCc1ccc(C(N)=O)cc1)(CC(C)C)NC(C(CC)C)=O Cc1nocc1CNC(c1[nH]ccc1CNC(=O)CCn1ccnn1)=O C1(CC(=O)NC2C3CC(C(=O)OCC)C(C3)C2)COC2(CCC2)CN1C(C)(C)C N1(C(C(c2c(C)noc2C)C)=O)CCN(C(c2csc(C(C)(F)F)n2)=O)C(C)C1 C1(OC)CN(C(=O)CCC2CCC2)CC1NC(=O)Cc1cccc(Cl)c1 C(=O)(CC(CNCCCCCNC(=O)CC(C)(C)C)N(C)C)OC C(=O)(CS(=O)(=O)NC)NCC(CNC(C1(CC)COC1)=O)OCC c1(C(N(CCNC(C(CC)n2cncn2)=O)CC)=O)cccc(CO)c1 C1(CC)CCCC1(C)C(=O)NCCCCN(C)C(c1ccc(C(C)C)s1)=O C1(NC(N(CCNC(N(C)C)=O)C)=O)CNC(=O)C(C)(C)C1 N1(C(C2N(C)CC2)=O)CCCCC1C1CCN(C(=O)Cn2nnc(=O)[nH]2)CC1 CC1CCC(NC(c2cc[nH]c(=N)c2)=O)CN1C(C12CCOC(C)(C1)C2)=O c1(C(=O)OC)ccc2nc(C(=O)NC3CCOCC34CCC4)cn2c1 CC(C#N)C(=O)NCc1cc(C(=O)NC2(c3ncccn3)CC2)cs1 CCS(=O)(=O)C=CC(=O)N1CCCC1(C)CNC(c1cccc(CN=[N+]=[N-])c1)=O Cc1onc(C(C)(C)C)c1C(=O)Nc1cccc(-c2cccc(F)c2)c1 c1(NC2CCCN(C(C3C(C)(Br)C3)=O)C2)ncnc2ccc(Cl)cc12 C1(CNC(=O)C(F)Cc2ccccc2)CC2(CC2)CN1C(c1ccc(O)cn1)=O c1(C(N(C2CCCN(C(c3scc(C)c3Cl)=O)C2)C)=O)cn2c(n1)CCC(C)C2 N1(C(C(CC)(C)OC)=O)CCC2CN(C(c3cc(C)ccc3C)=O)CC2CC1 c1(C(=O)NC2C(C(N3CC(C)OCC3)=O)C2)cc(C(F)(F)F)ccc1Br C1(O)(C(=O)NC2CCN(C(C(C)(C)C)=O)C2)CCCCC1 C1(NC(C2CC(NC(=O)CSc3ccccn3)C2)=O)CCc2n[nH]cc2C1 Cc1cnc(CCNC(=O)C(C)(C)C2CCCN2C(C2CC(C)N(C)C2)=O)nc1 n1(CC(=C)C)c(N(CCCN(C)C(=O)OC(C)(C)C)C)nnc1-c1c[nH]nc1C N=c1[nH]c(Cl)c(Cl)cc1C(N1CCC2CCC12CNC(=O)CC1CCC1)=O C1(C(=O)NCC(CCC)O)CC12CCN(C(c1sc(C)nc1C)=O)CC2 N1(C(Cc2n(C)ccn2)=O)CCCC(N=c2[nH]c(Cl)nc3c2COCC3)CC1 N1(C(c2c(CNC(C(COC)OC)=O)ocn2)=O)C2CCC1(CO)CC2 c1(C(=O)NCC2CCN(C(C(C(C)(C)O)(C)C)=O)C2)ccc2nc[nH]c2c1F N1(C(C(CC)N(C)C)=O)CC(C)N(C(c2csc(Cl)c2)=O)CC1C c1(CC(=O)NCCCOCCNC(CC2CCC(C)CC2)=O)cccc(F)c1F Cc1cc(N2CC(C(=O)NCc3ccc(C(C)C)s3)C2)nc(C)n1 c1(C(N2CC(C(N3CCC4(CCC4)C3)=O)C(O)CC2)=O)ccc2ocnc2c1 c1(OCC(c2ccccc2)CC)ccc(C(=O)OCC(N)=O)cc1 Cc1cc2c(SCC3CCCCC3)nccc2n1C N1(C(CCOCC(C)C)=O)CC(NC(=O)CCCC2CCCC2)CC1C C(=O)(C#CC1CCCCO1)NCC(C)(O)CNC(=O)Cc1nnc2n1CCCC2 CC(C(=O)OCC(c1cc(F)c(F)c(F)c1F)=O)C(C)S(C)(=O)=O c1(C(F)(F)F)noc(CCNCc2cc(-c3ccccc3)sn2)n1 c1(C(=O)NC2CCc3n(C)nnc3C2)cnn2c1NC(C1CC1)CC2C(F)F c1(CC)ccc(C)c(Cl)c1F.C12CCCN1C(=O)C1CN(C1)CC(=O)NC2 C1(F)(CNC(C2(Cl)C(C)(C)C2)=O)CCN(C(=O)CCCn2ccnc2)C1 c1(Nc2ccccc2)cccc2c1CCCC(NS(=O)(=O)C1CCC(F)(F)C1)C2 C(c1ccc2c(c1)OCO2)=CCOC(C1C(CC(C)(C)C)CCC1)=O C(=O)(CCC(=O)N(C)C)NCC(C)CNC(c1ocnc1Cc1cnn(C)c1)=O C1(C=O)COc2ccc(F)cc2C1.N1(C(=O)C(F)(F)CO)CC2CC(N)CC1C2 C1(C(=O)NCCc2ccncc2)(COC)CCCO1 N1(C(C(CCC)N(C)C)=O)CCCCCC(NC(c2conc2CC)=O)C1 CC1(C)C(C(=O)NC2CCOCC2NC(=O)C=Cc2ncc[nH]2)C1(C)C c1(C(C)C)cc(C(=O)NC(C)CCNC(C2(CC3CC3)CCCO2)=O)ccc1F Cc1cc(C)c(CC(N2CC3CC3(NC(=O)COC3(C)CCCC3)C2)=O)c(C)c1 N1(C(C(CC)NC(C)=O)=O)CCCC1C=CC(=O)N(C)CCSC CC1CC(=O)NC(C(=O)NC(CNC(=O)CCOc2ccc(F)cc2)C2CC2)C1 c1(CNC(CC(C)OC)=O)cc(C#N)oc1C.c12ncccc1CNC2=O C1(NC(C2C(=C)C2)=O)CCS(=O)(=O)C12CN(C(=O)CSc1ccc(F)c(F)c1)C2 N1(C(C(CCSC)O)=O)CC2CN(C(c3cc4ccc(F)cc4[nH]3)=O)CC2(C)C1 c1(C(=O)NC2CC(NC(CC(n3ccc(C)n3)C)=O)C2)cccc2cccnc12 c1(CCNC(c2ccncc2Cl)c2n(C(C)C)nnn2)ccc(F)nc1 c1(C(=O)NC(CNC(C2(CC#C)CCCC2)=O)CO)cnc(=N)[nH]c1 c1(OCC(=O)NCCCN(C(=O)C(CO)N(C)C)CC)ccc(Br)nc1 c1(OC)c(C(N2CCCCC2C(C)NC(c2ccc(C)cn2)=O)=O)cnn1C c1(C(=O)OC)ccc(NC(N2CCCC2(C)CO)=O)cn1 C1(C(=O)OC)COCCN1C(=O)CC1(C)CCN1C(=O)Cc1ccco1 C(CC(C(N)=O)NC(=O)C#CCNC(=O)CN1CCCCCC1)OC c1(C(CC)NC2(c3nc(C(=O)OC)no3)COC2)nnnn1C(C)CC C1(NC(C(=O)NCCOC)=O)CC(C)N(C(=O)CSCc2c(C)noc2C)C1 CC1CN(C(=O)Cc2ccns2)CC1(C)C(=O)NCc1cc(C#N)cs1 C(=O)(C(O)CF)N1CC(CCNC(C2CC(=O)N2)=O)C1 C1(C(=O)NCC(O)CF)CCCN1C(c1cn[nH]c1)=O N1(CC(CC(=O)NCCCOC)O)CCOc2ccc(COC)cc2C1 C(=O)(CCCN=c1[nH]c2ccccc2o1)N1CCCC(NC(C(=O)NCC)=O)C1 C1(CNC(C(COC)C)=O)CCN(C(c2cc(C)c(C)cn2)=O)CC1O c1(C(N2C(CCNC(C(CCC)NC(N)=O)=O)CSCC2)=O)cc(C)nc(C)c1 N1(C(C=C(C)C)=O)CC(C)CC1C(=O)Nc1ccc(-n2ccc(C)n2)cc1 C1(CCNC(c2c(CC(=O)OC)occ2)=O)CCCN(C(C2(C#N)CC2)=O)CC1 c1(CC)cccc(C)c1.C1(CCC(C)C)n2nnnc2N1C n1(CC)nc(C(N2CCCC(C(C)NC(=O)CSCC(F)F)C2)=O)cc1C N1(C(C2COCC(C)O2)=O)CCC2(C1)CN(C(c1ccccc1)=O)C2 c1(CNC(=NC)N2CC(CN(C)C(=O)OC(C)(C)C)C2)ccccc1F C1(C)(CNC(C(C)(C)OC(C)C)=O)CCN(C(c2ccccc2CC#N)=O)C1 CCC(CCC(=O)NCC1CC2CC2N1C(c1cnc(C(C)(F)F)s1)=O)OC c1(CC)ccc(C(=O)NC2CCCC2CC(=O)NCc2cscn2)o1 CCCC(C(O)C(=O)Nc1cc(C#N)ccc1C)NC(c1cccnc1)=O C1(CCOC)(NC(=O)CN(C)C(C)=O)CCN(C(c2ccc(Cl)cn2)=O)C1 C(CC(C(=O)NC(C1(CO)CC1)C)NC(=O)CN1CCCC1)=CCC N1(C(C=CC)=O)CCC2CCN(C(c3c(SC)cnn3C)=O)CC2C1 C(=O)(CN1C(=O)Cc2cc(F)ccc21)N1CCC(c2cn(CCCC(C)C)nn2)C1 C1(C(N(CC(c2ccccc2)NC(=O)CC2OCCO2)CC)=O)CCC12CCC2 C1(C(=O)NC2CC(C(C)(C)O)C2)CCCCC1(C)NC(C12CSCC1C2)=O C1(C(=O)Nc2cc(CC3CC3)cs2)COCCN1Cc1ccc(-n2cncn2)cc1 C1(N(C(=O)CCC2CCCCO2)CC#C)CCN(C(C2CCCC(=O)C2)=O)CC1 CCS(=O)(=O)CC(=O)NC1CCCCC1NC(c1[nH]ccc1-c1ccccc1)=O CC(C)(C)C(CNC(c1cc(O)nc(O)n1)=O)C(=O)N1CC(C)(NC=O)C1 CCCCCC(O)C(=O)N(C1CCN(C(c2nccc3occc23)=O)C1)CCC c1(C(=O)NCC(CCCC)NC(C(=O)NCCCC)=O)cc(Br)cnc1O c1(C(=O)NC(C)CCN(C(=O)CCCCCN(C)C)C)cccc2c1ncn2C C1(CNC(=O)NCc2c(C)ncs2)(CNC(=O)OC(C)(C)C)CCCCC1 C1(C(=O)NCCc2n(C)ncn2)CN(C(c2cc[nH]n2)=O)CCC1(F)F c1(CC#N)cccc(NCCC2CC2C2CC2)c1 N1(C(C(C(=O)OCC)F)=O)CC2COCC(C1)C2NC(c1cc(F)cc(Cl)c1)=O C(=O)(C1=CC2C=CC1C2)NCC(CC(=O)N(CCN(C)C)CC)C1CCCC1 c1(OC)cccc(OC=CC(=O)Nc2nc(OC(C)CCC=C(C)C)c(C)s2)c1 N1(C(CNC(N)=O)=O)CCC(NC(c2cc(C3CC3)on2)=O)C(CO)CC1 C(=O)(C1=CC2(CCOCC2)C1)N(CCC(=O)OC(C)C)C C1(CC(=O)NCC2CC(O)CN2C(=O)CC2(C(F)(F)F)CC2)CC(C2CC2)C1 c1(CCC)n[nH]cc1C(=O)NC(C(=O)NCCSC(F)F)C1(C)CC1 CN1CCn2ncc(C(N3CC4(CNC(C5CCC(=O)NC5)=O)CCC3C4)=O)c21 c1(CC)cscc1C(=O)N(C(C)CNC(C1CC1C(C)(C)C)=O)CC N1(C(C2C(CC)CCN2C(=O)Cn2ccccc2=O)=O)CCCNC(=O)CC1 C12(C(=O)NCC3(CNC(C4(C)CC=CCC4)=O)CCC3)CCC(CC1)C2(C)C N1(Cc2onc(CC)n2)CCC2(CCCN(C(c3ccc(CC)o3)=O)C2)C1 C(c1ccccc1)=CC(N1C(C(C)NC(C=CCN(CC)CC)=O)CCC1)=O C1(C(=O)Nc2cnc(C(N)=O)s2)C2CCC(F)(F)C12.C12CCN(CC1)C2=O Cc1noc(C)c1C=CC(=O)N(C(C)CCNC(=O)C(F)(F)c1cccnc1)C c1(OCCC(=O)NCC2(F)CC(NC(C3CSCCS3)=O)C2)cccc(F)c1 c1(C(N2CC(NC(CCOCC)=O)(COCC)C2)=O)cc(C(N)=O)cn1C Cn1nc(OC2CN(C(C3CCCN(C(=O)C(C)(Cl)Cl)C3)=O)C2)ccc1=O C1(CC(=O)N(C)CC2(CNC(C3(O)CC3)=O)CC2)(OC)CCCC1 c1(C(N2CC(C3N(C(c4c(C)cns4)=O)CCC3)(O)C2)=O)cc(Cl)ccc1F C1(C(=O)NC2CCC(NC(=O)CCc3cn[nH]c3)CC2)Cc2ccc(F)cc2C1 C1(C=O)CCN(C(=O)c2ccccn2)O1.C1(=O)C(C)N1C1CC1.CO C1(c2n[nH]c(=NCc3c(C)c(Cl)ccc3)s2)C2Cc3ccccc3C12 N1(C(C2CC(C)(C)N(C(C3CCS3(=O)=O)=O)C2)=O)CCOc2ccccc21 C(=O)(CC(C(F)F)NC(=O)C#CC(C)(C)O)N(C)CC1CCN(CC)C1 c1(C(=O)OC(C)C(=O)Nc2ccc(C#N)cc2F)ccccc1S(C)(=O)=O Cn1[nH]c(=NC(=O)c2ccnn2CC(F)F)cc1CC1CCC1 Cc1c(F)cc(C(N2CCOC(C(=O)NCc3ccnc(Cl)c3)C2)=O)cc1Br C1(C(=O)NCCC(C)(C)NC(CNC(CNC(C)=O)=O)=O)OC(C)(C)OC1(C)C c1(OC)cccc(SC(C(=O)NCC2CCN2C(c2onc(C)c2C)=O)C2CC2)c1 C(=O)(C1=Cc2ccccc2C1C)NCCC(C)CCNC(c1csc(CO)n1)=O Cc1cc2c(cc1C)C(C(=O)NCC(C)N(C)C(c1cn(C(C)C)cn1)=O)CO2 C1(C2CCOCC2)(CNC(CCN(C)CC)=O)CCN(C(c2cc(C)[nH]n2)=O)C1 C(=O)(CC(C)(C(F)F)N(C)C)NCC(C)NC(c1c[nH]nc1C(C)(F)F)=O C=C(C)C1OCCCC1C(=O)NCCCC(CCC)NC(=O)C(C)(C)CF C(=O)(C1=CC(C)CC1)N1CCC(CN(C(=O)CCc2cccc(O)c2)CCC)C1 C(=O)(C1CCCc2c[nH]nc21)NC1CC2(CCCN(C(C3(C#N)CC3)=O)C2)C1 c1(OC)cccc(CNC(CCCO)=O)c1.C(=O)(CC(C)(F)F)NCC(C)(C)CSC C(=O)(CCC(C)NC(c1cc(SC)n(C)n1)c1nnnn1CCCF)OC C(=O)(C1CCCc2ncnn21)NCC(CO)NC(Cc1c(C)occ1)=O c1(C(N2C(CNC(c3ccc([N+](=O)[O-])[nH]3)=O)C=CC2)=O)ccn2nnnc2c1 c1(NC2CC(NC(c3c(C)c[nH]n3)=O)C2(C)C)ccccc1[N+](=O)[O-] Cc1c(C(=O)NCCCC(C)NC(C2CCCN2C(C)C)=O)cnc2ccnn12 C(C)(CCC(=O)N(CCNC(=O)Cc1ccn(C(C)C)n1)CC1CC1)SC C1(F)(CNC(c2cc(OC)no2)=O)CCN(C(c2nccnc2N)=O)C1 N1(C(C)=O)CC(O)(CC(=O)NC(c2cnns2)C2CC2)C1 C1(CC)CN(C(=O)Cc2cnn(C)c2)CCN1C(=O)CC=CC(C)(C)C N1(C(CCCCC(N)=O)=O)CCC2(CC1)CC2(CO)CNC(C1CCC(=O)N1)=O C1(CC(N2CCC(C(C)NC(C3(CC)CCC3)=O)CC2)=O)CCC2(CCC2)O1 Cc1cc(=NC(C)C(C)CO)[nH]c(=NCc2cncc(Cl)c2)[nH]1 Cc1ccc(CCCC(=O)OCCC2(CNC(=O)OC(C)(C)C)CC2)cc1 N1(C(C2(CC)COC2)=O)CCOC(C)(CNC(=O)CC2OCCCC2(C)C)C1 c1(C(N2C(C)CC(CC(=O)NC(C(CC)CC)C)C2)=O)ccc2[nH]ccc2n1 N1(C(COCCC)=O)CCCC2(CCN(C(=O)Cc3ccc(F)cc3F)CC2)C1 c1(CCCOC)cccc(OC(=O)Nc2ccc(CC)cc2)c1OC C1(NC(C2N(C(Cc3ccn(C)c3)=O)CC(O)CC2)=O)CCCCC1N=[N+]=[N-] C1(C(=O)N(C2(CC(=O)NCCCOC(=N)O)CCC2)C2CC2)C2CCCCCC12 C1(C(=O)NC(C)CCCCNC(C2C3CCC(C3)C2C)=O)Cc2ccccc2C1 c1(CCC)cc(C(N2CCCC(c3cc(C(F)(F)F)n[nH]3)C2)=O)c(C)o1 c1(C(=O)NC)ccc(C(=O)N2CC(n3cc(C(O)C(C)(C)C)nn3)CO2)nn1 c1(C2(OC)CCN(Cc3cccc(CC)c3)C2)ccc(C(F)(F)F)c(OC)c1 C1(COC)CN(C(=O)Cc2nc[nH]n2)CCN1C(C1CCOC(C)(C)C1)=O C12CCC(O)CN1C2.O=C1CN(CC(=O)NCC(F)(F)F)CCN1 c12ccc(Cl)c(c1)C(c1n(CCOC)nnn1)N2.C1(CC(C)SC)CCOCC1 S(=O)(=O)(c1cccc(C(=O)NCc2ncn(C)n2)c1)NCC c1(CCC(N2CC(C)(NC(=O)Cc3cscn3)C2)=O)ccc(CO)cc1 C12(CC3(CC3)C1)CN(c1ncccc1C(C)=O)C2.C(=O)(NCC)NCC C12(OC)CCC1CN(C(=O)C(O)CCCNC(=O)C=CC(F)F)C2 CC1(CNC(=O)CN2CCSCC2)CCN(C(c2csc(C(F)(F)F)c2)=O)CC1 C1(NC(C2(C)CCOC2)=O)CC(N=c2cc(Cl)nc(C3CCC3)[nH]2)C1 N1(C(C(C)OCCOC)=O)CC(CNC(=O)C2=CCCS2)C(F)(CO)C1 c1(C(N2CC=CC(NC(C3(OC)CCCCCC3)=O)C2)=O)ccc(P(C)(C)=O)o1 CC1CN(C(=O)CNC(C)=O)CCC1C(=O)N(C)CCc1cccnc1 C=CCC(CC(=O)NCC(CC)NC(C1CC(OC)(OC)C1)=O)NC C12CCCC1C(=O)N2.n1(CCNC(CN(C(=O)OCC)C)=O)nncc1C c1(CC2(NC(C(=O)NCCNCCOC)=O)CC2)cccc(CCC#N)c1 C1(CNC(Cc2c(C)scc2)=O)CCN(C(=O)Cn2nnc(=N)[nH]2)CCC1(F)F c1(C(N(C)CC2(NC(CC3CCC(C)O3)=O)CC2)=O)ncccc1Cl C(C)(C)(C(=O)NC(C1CCCN1C(C1SCC=C1C)=O)C)OCCC c1(C(=O)NCCc2nc3c(s2)CCCC3)cc2cc([N+](=O)[O-])ccc2cc1O c1(-c2n(-c3ccn(C)n3)nc(CCN(C)C)n2)ccc2c(CC(F)(F)F)n[nH]c2c1 c1(N(C(=O)NC(C(=O)OC)Cc2csc(Br)c2)C2CC2)ccc(C)cc1 Cc1ccc2c(C(N3CC(NC(c4nc(Cl)oc4C)=O)C4CC34)=O)c[nH]c2c1 CC(CCCCO)NC(=O)CCC1(C)CCCN1C(c1cnc(Cl)n1C)=O N1(C(CN2CCC(C)C2)=O)CC2CCC1CN2C(=O)COc1cn[nH]c1 c1(OCC)ccc(OC)c(C(=O)NNC(=O)c2cc(NC(C)(C)C)ccn2)c1 CCCC(C)CC(=O)NC(C)C(C)(C)NC(=O)Cc1cccs1 N1(C(CC2CC(C(N)=O)C2)=O)CC(C2(NC(=O)Cc3ccn(C(F)F)n3)CC2)C1 C1(C(=O)NC2CC(N3CCN(C)CC3)C2)CCN(C(=O)C(O)CF)CC12CCC2 CCC1=C(C(=O)NCCCN(C(=O)C(O)C(C)c2ccccc2F)C)CCCO1 c1(C(=O)OC)cc([N+](=O)[O-])ccc1NCc1c(Cl)ccc(Cl)c1O c1(CSCCNC(C2N(CCCCC)CCC2)=O)cccc(OC)c1 C1(CNC(C(=O)NCCn2ncnn2)=O)CCCC2(CC2)C1 n1(C(C)C)ccc(C(=O)N(C)CC2CCCN2C(=O)COc2ccsc2)n1 C1(CCNC(c2c(C)cno2)=O)CN(C(C2CN(C)CCO2)=O)CCS1(=O)=O c1(OC)cc(NC(C2C3CC2(c2ccc(F)cc2)CO3)=O)ccc1C C1(C(=O)NC(CNC(c2ccc(OC)nn2)=O)CC(=O)OC)COCC(C)(C)C1 C(=O)(CS(=O)(=O)N1CCCCC1)NC(CC)CN(C(=O)C(C)NC(N)=O)C c1(CC(=O)NCCN(C(=O)C(F)=C(C)C)CC)cccc(Cl)c1 CCC1=C(C(=O)NCC2C(C)CCN2C(=O)CC(C)(C)C#N)CCCO1 C1(CCNC(C=COCC)=O)CC(F)(F)CN1C(=O)CN1CCC(CO)CC1 Cc1[nH]nc2c(O)cc(C(=O)NCC3(C)CCN(C(c4ccc(Cl)o4)=O)C3)cc12 C(CC(CNC(=O)CCOC)NC(C1CCC(=O)N1)=O)OC C1(NC(C2(SC)CN(C(c3ccc(O)nn3)=O)C2)=O)CC(C)(C)C12CC2 N1(CCCC)CCCCC1C(=O)NC1CCN(C(=O)CC2(CSC)CCCC2)C1C CC(C)C(C(=O)NCC(C)(C)NC(=O)Cn1cnc(C#N)n1)c1ccc(Cl)cc1 C(CC1CCCC1)(C(=O)NC1CCN(CCCNC(=O)CC2CNC(=O)C2)C1)OC C1(OC)CN(C(=O)CCSc2ccccc2)CC1C(=O)NC1CN(CC)CC1C C1(C(N(CC(O)CN(C)C(C2(N(C)C)CC2)=O)C)=O)(CCF)CCOCC1 C1(NC(C(c2cccs2)N(C)C)=O)CC(F)CN(C(=O)CN2CSCCSC2)C1 CC1CCC(C)C1NC(C1CC(C)N1C(=O)C=CCN(C)C)=O C(=O)(C(O)CC(C)(C)C)N1CCC(C)(CNC(C2N(C(CC)=O)CCCC2)=O)C1 C(=O)(N=c1ccn(CC(=O)NC2CC3(CO)COC2C3)[nH]1)C1(NC(C)=O)CCC1 C1(C(=O)NCC(C)CN(C(=O)Cc2cccc(Cl)c2F)C)CCC(N=[N+]=[N-])C1 c12cccc(c1)-n1cc(nn1)CN(O)C2=O.c1(NC(C)=O)cnc(N(C)C)nc1 N1(C(C2(C)CS(=O)(=O)C2)=O)CCCC2(NC(c3cc(F)ccc3O)=O)CC12 c1(C(=O)NCC23C(CN(C(C(CCC)O)=O)C2)C3)cccc(Cl)c1F C1(CNC(c2c(Cl)nc(OC)s2)=O)CN(C(C2CCCCC2F)=O)CCN1C c1(OC)ccc(CC(=O)NCC(C)N(C)C(c2ncc(Cl)cc2F)=O)c(OC)c1 O=C(CCCCCCCCCO)N1CCC12CCS(=O)(=O)C2 N#Cc1cccc(CC(=O)NC2CC(C(F)C(=O)NC(CF)C(F)(F)F)C2)c1 C(C(CC1CC1)C(=O)NCC1(O)CC(O)C1)NC(C(C)=C(CC)C)=O C#CCC(CC(F)F)C(=O)N(C1CN(C(c2ccn(CC(F)F)n2)=O)CC1O)C C(C)(C)(CCC(=O)NC1CC(CNC(=O)C(C(C)(C)C)N2CCOC2=O)C1)OC C1(C)(CCC)CCN1C(=O)CCCC1(NC(=O)COCC(=O)OC)CC1 CC(CC(C)(C)C)C(=O)N1CC(OCCN(C(C2CN3CCCN2CC3)=O)CC)C1 C1(N(C(C(CC)C2CCOCC2)=O)C)CCCCN(C(=O)COCCCOC)C1 C1(COC(CCCOc2c(OC)cccc2)=O)CN2CCC1CC2 N1(C(c2c[nH]nc2Cl)=O)CCC2(CCN(C(c3ccn4nccc4n3)=O)C2)C1 c1(OC)ccc(C=Cc2nc(-c3ccccn3)no2)cc1 N1(C(CCOC(C)C)=O)CC(NC(=O)CC2CC(c3ccccc3)C2)CC1C N1(CCC(=O)NCCCN(C(=O)C(CC2CCC2)N(C)C)CC)CCCC1=O N12CCC(C1)CN(C)CC2=O.C1(C#N)(CCC(=O)NCCF)CCC1 C12(CC(=O)NCCCCNC(Cn3ncc(C#C)c3)=O)CCCN1CCC2 CC(CN(C)C)CC(=O)NCC=CC(=O)N(C(C)(C)CF)C(C)C C1(F)(C(=O)NC2CC(C(=O)OC)C2)CCCN(C(=O)CCC(C)(C)C)C1 c1(C(=O)NCC2OCCN(C(CC3(C=C)CC3)=O)C2)ccc(OC)c(C(C)=O)c1 C1(Cc2cn(CCCOC)nn2)CCCN(C(=O)CC(C)c2ccncc2)C1 CC1(C)COC(C)(C(=O)NCC2CN3CCN2CC3)CO1 N1(C(c2n(CC)ncc2Cl)=O)CC(CNC(=O)C2=COCC2)C2(CCC2)C1 c1(C(N(C(=O)NC(c2nc(C)[nH]n2)CO)C)=O)sc(C)nc1C.C1CCOC1 C1(C(=O)NCCC(C)(C)O)CCN(C(C2(C)CCCCO2)=O)CC1 c1(OC(c2ccc(F)cc2)c2nnc(SC)o2)cccc2nn[nH]c12 N1(C(c2cccc(C)c2Cl)=O)CC(NC(c2cc(Br)no2)=O)C2(CCC2)C1 C1(NC(=O)C(c2ccccc2)F)C=CCN(C(C2(CCF)CC2)=O)C1 Nc1cccc(C(N2CCC2CNC(c2ccc(C3CCCCO3)cc2)=O)=O)c1 c1(OCn2cc(-c3ccc(F)nc3)nn2)ccc(Br)cc1.N12CCC(CC1)NC2=O CCCCC(O)C(=O)NCC(N1CCN(C(=O)C(C)C(C)C)CC1)C Cc1ccc2c(N3CCC(NC(c4c(O)cccc4Br)=O)C3)ncnc2c1 N1(C(c2cc(=N)[nH]cc2)=O)CC=C(CNC(C2(F)CCCCC2)=O)CC1 c1(C(N(CCCC)C(C)CC)=O)coc2c1CN(C(c1cn[nH]c1)=O)C2 CCC(C)CCCCC(=O)NCC1(CNC(c2ccc(OC)c(OC)n2)=O)CC1 c1(C(=O)NCCC(C)(C)NC(COC(CC)(C)C)=O)cc2cc(Cl)ncc2[nH]1 C1(C)(C(=O)NC(C(C)C)CNC(=O)C(C)N2CCC2)CCC(=O)NC1 C1(CC(F)(F)F)(NC(=O)NC(CC)C)CCN(CCOC(C)(C)C)CC1 N1(CCN)Cc2c(O)ccc(OC)c2C1.C(=O)(C(CCC(=O)OC)N(C)C)OC C1(C)(NC(C=C(CC)CC)=O)CCCCC1C(=O)N(C)Cc1cncs1 c1(NCc2ccc(Br)s2)ncc(C2CC2)cc1Br.c12cncc(c1)N(C1CC1)C2=O N1(C(c2c(OCC)nccc2)=O)CCC2(CC1)CC2NC(=O)C=Cc1cccs1 C(=O)(C1=CC2(CCOC2)C1)NC(CCCNC(c1nc(OC)c(F)cn1)=O)(C)C Cc1cc(C(N2CC=CC(NC(C3CC4CC4C3)=O)C2)=O)c(C)n1NC(N)=O c1(C2(NC(C3CCN(C(c4cc(C)ncc4)=O)C3)=O)CC2)cc(F)ccc1F N1(C(c2ccc(C)cc2C)=O)CCN(C(=O)C(c2ccc(N)cc2)C)CC(O)C1 C(=O)(CP(C)(C)=O)NCC1(CNC(CC2CC(N(C)C)C2)=O)CC1 C=CC(C)(O)C(=O)NCCc1n[nH]cc1C(=O)NC(C1CCCC1)C c1(-c2ccc(F)cc2)nc(NCc2cnccn2)cc(N2CC3CC3(C(F)F)C2)n1 O=C(N1CC(O)CCO1)C1CC=CCN1C(c1cc(Cl)ns1)=O C1(C(=O)NCC(C)NC(CCc2cc(C)on2)=O)CCN(C2CCCCC2)CC1 C1(C(=O)NCC(C(CC)C)O)CN(C(=O)C#CC2(C)COC2)CC12CCC2 Cc1ccn2cc(C(=O)NCC3(C)CCN(C(c4cncc(N)n4)=O)C3)nc2c1 Cn1ccc(C=CC(=O)NC23CC(CNC(=O)CN(C4CCCC4)C)(C2)C3)c1 C1(CC=C)(NC(=O)CC2CC=CC2)CCN(C(=O)C(F)=CC2CC2)C1 Cc1noc(C)c1CC(C)C(=O)NCC12CC1CN(C(=O)CC1CCCC1)C2 c1(NC(C(CCC)NC(=O)CC(C)SC)=O)c(C)[nH]c(C)cc1=O N1(C(COCC(C)(C)C)=O)CCCCC1CCC(C)(C)NC(c1sccc1F)=O N12C(CCC3CCCCC13)C2=O.Cc1c[nH]c2ncnc(NC(C)CCO)c12 c1(C(=O)NC2(CCNC(c3scc(C#N)c3)=O)CC2)n[nH]c2ccc(O)cc12 c1(C(=O)NC2CC3(CN(C(CCSCCC)=O)C3)C2)nccn2ccnc12 c1(C2C(C(=O)N)C2)cccnc1.c12ccc(o1)C(C1CC1)CCCNC2=O.C(F)F N1(C(C2C(CNC(=O)Cn3cncn3)CCO2)=O)CCC=C(F)C1 C(C(F)(F)C(F)(F)c1ccccc1)NCC(=O)NC(c1c(C)nccc1)=O C(N=c1cc(Cl)nc(NC(=O)C(C(C)C)OC)[nH]1)C1CCN(CCC)C1 N1(C(CC2(C)CCOCC2)=O)C(C(=O)NCC2CCCCC2)CCC12CC2 CC1(C)CC1(C(=O)NCC(C1CC1)N(C)C)NC(=O)Cn1[nH]cnc1=N C1(CC)CC(O)CCN1C(=O)Cn1cc(CCN(C2CCOC2)C)nn1 Cc1cccc(N(CC(C)(C)C)C(C2CC2c2cccc(Br)c2)=O)c1 c1(C(=O)NC2C(C(=O)NC3C(OC)COCC3)OCC2)ccc(C)c(O)c1 CCCC(O)CNC(=O)CN(C(=O)CCCC1CC1)CC(C)C C1(C(N(CC(N2C(C(C)C)CC2)=O)C2CC2)=O)CCCC1O c1(C(=O)NC2CN(C(CCC#C)=O)C3(C2)CCC3)ccc2c(c1)N(C)C(=O)C2 N(C1c2ccccc2OCC1F)C(C(=O)NCc1cn(C)[nH]c1=N)=O c1(C(=O)NCC(C)CNC(c2cc(F)c(F)cc2F)=O)ccn2[nH]c(=N)nc2c1 C1(C(=O)NC(C)CC(C)NC(C2CN(S(C)(=O)=O)C2)=O)CCCOCC1 C=CC(C)CC(=O)NC1CCN(C(=O)Cn2cccc2)C1c1ccccc1 C1(C(=O)NCC2(CNC(c3c(CC)ncnc3)=O)CC2)CCCC1S(C)(=O)=O C(C)(C(F)(F)C(F)(F)F)=CC(=O)NC1CC(NC(CCC=C)=O)C(O)C1 C1(C(N2C3CC(NC(C4N(C=O)CCC4)=O)(C3)C2)=O)CCc2ccc(F)cc2O1 C(=O)(C#CC1(C(F)(F)F)CC1)NC(C1N(C(CCNC(C)=O)=O)CCC1)C CC(CC(=O)N(CCC(C)NC(=O)C=C1CCCC1)C)c1ccccc1 C1(OC)CC(C(=O)OCC(N2CCCC2(CO)Cc2cccc(F)c2)=O)C1(F)F C1(CO)C2CC(CN=c3nc[nH]s3)CC12 N1(C(CCC=C)=O)CCC(CNC(=O)COCCSC)CC1C c1(C2CN(CC(CCOC)NC(=O)CCc3ccncc3)C2)ccc(Cl)c(Cl)c1 N1(C(c2c(-c3ccc(C)o3)onc2)=O)CCC(NC(=O)C=CC=C(Cl)Cl)C(C)C1 C1(CC(C(=O)OC)F)CCC(F)(F)CC1.n12ccnc1C(N1CCCC1)C2 Cc1cc(C)c(CC(=O)Nc2cc(C(=O)O)cc3c2OCC3)c(C)c1 C1(NC(C(N2CCC(C)C2)=O)=O)C2CN(C(c3ccc(C#N)o3)=O)CC12 CCC(C)(COC)C(=O)NCC#CCNC(=O)C(C(C)(C)C)n1ccnn1 C(=O)(C(C(C)C(C)C)NC(=O)NC1(CC2CCC2)CC1)OC CC1CC(CNC(C2CC23CCOC3)=O)CN1C(c1ccn(C(C)(C)C)n1)=O c1(C(=O)NCC2(CNC(C3CCS(=O)(=O)N3)=O)CC2)nc(Cl)ccc1OC(F)F n1(CC=C)cc(C(=O)NC2CC(N(C(=O)CCc3c[nH]c(=N)[nH]3)C)C2)nn1 S(=O)(=O)(c1cnc(N2CCS(=O)(=O)NC2)c(Cl)c1)NCCCn1c(C)ncc1 c1(C(N)=O)ccc(NC(=O)C(=O)NC2CC(OCC(C)(C)C)C2)c(OC(F)F)c1 Cc1noc(C(C(C)(C)C)N(C(C)C(c2ccccc2)N)C(=O)C)n1 c1(C(=O)NC(CNC(C(=O)NCC)=O)(C)CO)cc(OC(C)C)cc(Br)c1 Cc1cccc(CC(C)NCCCN2CCN(C)CC2)c1.C=O O=S(=O)(Oc1cccc(Cl)c1C1CCC1)c1ccc(C2CC2)c(Cl)c1 CC(C)CC(C)(CNC(=O)CC(C)(C)c1ccc(F)cc1)NC(=O)C1=CCC1 c1(OC)ccc2[nH]nc(C(=O)NCCCCNC(C3CC4CCC34)=O)c2c1 c1(CC)ncnc(CC)c1C(=O)NCC1CCN(C(=O)CC23CC(C2)C3)C1 N1(C(C(C)OC2CCCC2)=O)CCC2(C1)CN(C(c1cccc3nsnc13)=O)C2 Cc1ccc(F)c(C(N2CCC(N(C(=O)Cc3nn(C)cc3Cl)CCO)C2)=O)c1N N1(C(C(CC)O)=O)CCC2(CC1)CN(C(c1ccnc(C)c1N)=O)C2 N#CCS(=O)(=O)NC(C1CCN1Cc1ccc(C(F)(F)F)s1)=O N1(C(C(C2CC2)NC(CN(CC)CC)=O)=O)CCC(C)C(C)(C)C1 C(CCC(O)C(=O)NC(C)(C)CC(N)=O)NC(CC(C)SC)=O C(=O)(C(C)(C)C1CCN(C(C2CC23CCC3)=O)C1)NCC=C C1(C)(C(N2CCCC2)CN2CCC(CC(=O)OCC)CC2)CC(C(C)C)=NO1 Cc1cc(C(=O)NC2CN(C(=O)Cc3ccc(O)cn3)CC2F)cc2ccoc12 C1(C(N(C)CC2(C)CCOCC2)=O)N(C(C23CCC(C2)C3)=O)CC12CCCC2 n1(CC)cc(C(=O)NC(C)(CNC(=O)C(c2cccc(Cl)c2)C)C(C)C)c(C)n1 Cc1cncc(C(N2CCOCC2CN(C)C(C2CC3CCC2O3)=O)=O)c1 c1(CC)[nH]nc(Nc2ccccc2NC(c2cccc(C(N)=O)c2)=O)c1C c1(C(=O)NC2(CF)CCN(C(C3(C#N)CCOC3)=O)C2)ccc(F)c(F)c1F c1(CC(=O)OCC2CC3(C2)CC3(F)F)csc2ccc(F)cc12 N1(C(c2n(C(C)C)ccn2)=O)CCC(CNC(C2CCCS2(=O)=O)=O)CC1 C1(NC(C2C(C(C)(F)F)C2)=O)CCC(NC(=O)CCc2cnoc2)CC1 C1(F)(CN(C)C)CCC(NC(=O)NCCC2CC2)C1 CCCCCC(O)C(C)C(=O)N1CC(F)(CNC(c2cc(SC)c(C)o2)=O)C1 C1(NC(C2(c3cccc(Cl)c3)CC2)=O)C2CC(O)C1N(C(=O)C#CC1CCC1)C2 C1(OC)CCN(C(=O)CCC2CC(NC(=O)Cc3cncc(C#N)c3)C2)C1(C)C C1(OC)(COC)CN(C(=O)COC)C1.C1(C)(CCOCCNC=O)CC1n1cccn1 c1(C(=O)NCC(C2CC2)NC(c2nc(C(=O)OC)sc2)=O)ccnc(C)c1 c1(C(=O)NCC(=O)NC(CNC(=O)CCc2nccs2)C2CC2)ccc(F)cn1 C1(C(=O)Nc2cnn(C(F)F)c2)CCC2(CC2)N1C(C1CC2(CCC2)C1)=O c1(C(N2C(C(C)NC(c3cncc(C)n3)=O)CCC2)=O)cnn(C)c1S(C)(=O)=O N1(C(c2ncccc2C(F)F)=O)CCCC1C1CCCN1C(=O)Cc1ccsc1 c1(C(=O)NCC2N(C(CC(C)OC)=O)CC(C)(C)C2)c(C)ccc2nsnc12 c1(C(=O)NCC2(NC(C3C(C)(C(C)C)C3)=O)CCC2)ccc2c(=O)cc[nH]c2c1 c1(CNC2CCC(NC(c3cnc(OC)nc3)=O)C2)cc(F)cc(F)c1[N+](=O)[O-] c1(NC(C2C(NC(c3ccc(C(F)(F)F)cc3Cl)=O)C2)=O)[nH]nc2cnccc12 N1(C(C2C(CN(C)C)C2)=O)CCN(C(c2cnn(C)c2N)=O)CC1C1CC1 c1(CC2(C)CC2(F)F)cccc(=O)o1.c12ccc(o1)C2NC(=O)OC(C)(C)C N1(C(C23CC(C(=O)OC)(C2)C3)=O)CC2COCCC2(NC(c2cccc(C)n2)=O)C1 C12(C(=O)NCC(CC)NC(=O)CCCN(C)C(C)=O)CCC1CC2 c1(C(N2CC3C(Nc4ncnc(CC)c4F)C3C2)=O)cc(C)c2nc(C)nn2c1 C1(C)(N(C2CCN(CCCCCC)C2)C(=O)C=Cc2ccncc2)CC(OC)CN1C C1(NC(CC=CC=C)=O)CC(O)(C2CCN(C(=O)COCC)C2)C1 C1(CNC(CCCC(C)=O)=O)CCC2(CCC2)C1NC(C1(N2CCCC2)CC1)=O c1(CC)cc(C(N2CC(O)(C(C)NC(c3cc(COC)oc3C)=O)C2)=O)sc1C CCCC(C)(CCC)C(=O)N(C)CC1(NC(=O)CSc2ccoc2C)CC1 N1(C(C2CCCC(C)C2)=O)CCCC2(CCCN(Cc3ncc[nH]3)C2)C1 CC1CN(C(c2ccn(C3CC3)n2)=O)CC(C)N(c2ccc([N+](=O)[O-])c(O)n2)C1 C1(CNC(C(CC)NC(C)=O)=O)CC2CCC1N2C(=O)CC1(CO)CCCC1 C1(NC(C(C)NC(N)=O)=O)CCN(C(=O)CCCc2n[nH]c(=N)s2)CC1O c1(C(=O)NCC(C(=O)NC(CC)CN2CCOCC2)O)cc(C)c(C#N)cn1 C=C=C(C)CC(=O)N(CC(=O)NCC1CCC(=O)NC1)C1CC1 c1(C(=O)NCC2N(C(c3c(OC)cc(O)nc3)=O)CCC2)cc(Cl)c(N)c(Cl)c1 c1(OC)ccc(C(=O)NCCN(C(=O)C=Cc2ccc(C)s2)C(C)C)nn1 C12(NC(c3c(C)ccs3)=O)CC1CN(C(c1cnc(CC3CC3)s1)=O)C2 c1(SCC)cnccc1C(=O)NC1CN(C(c2c(C)coc2C)=O)CC1F Cn1c(O)nc2ccc(C(N3CC(O)(CNC(c4cc(Cl)no4)=O)C3)=O)cc12 C1(NC(C(=O)NCC)=O)CCCCCN(C(c2ccc(C(F)(F)F)nc2)=O)C1 N1(C(c2c(C)scc2)=O)CCCC1C1CCCN1C(c1cnc2[nH]ncc2c1)=O c1(C(N2CC(NC(=O)C(F)(F)C(O)C3CC3)C2)=O)cccc2c1CCNC2=O n1(CC(=O)N(C(CNC(c2c(CC)cno2)=O)C)C)ccc(O)nc1=O Cc1ccc(C(N2CCN(C(C3CC3CC3CCC(N(C)C)CC3)=O)CC2)=O)cc1 n1(CC(=O)NCCCN(C(COCCCCC)=O)CC)cc(Cl)c(C(F)(F)F)n1 c1(C(=O)NC2CCN(C(C(CCC)C)=O)CCC2CO)nn(C)c2c1COCC2 C1(C)(C(N2C(C)(CC(NCP(OCC)(C)=O)=O)CC2)=O)CCCCC1C c1(C(N(C)Cc2cn(CC3CC3)nn2)=O)c2ccccc2nn1C N1(C(C(C)N(C)C)=O)CCCC12CCN(C(C1CCc3cnn(C)c3C1)=O)C2 c1(C(N2CCC(C)C(CO)C2)C(=O)NCC)c2ccccc2nn1C C1(C(=O)NCC2CCN2C(=O)C(F)(F)c2csc(Cl)c2)(CC)CCCCO1 C(=O)(C1=Cc2ccccc2C1)NCC1CC(C(=O)NC2CCCC(C)C2)C1 CC(C)C(C(=O)N(CC(F)(F)Cl)C)C(C)NC(c1cnn(C2CC2)c1)=O N1(C(c2c(C)cccn2)=O)CCC(NC(=O)C(C)S(N)(=O)=O)CC(O)C1 C1(C(C(=O)NCCCSCC)N(C)Cc2ncnn2C)C2(CCC2)C12CCC2 CS(=O)(=O)C1CN(C(c2cc3ccc(Br)cn3n2)=O)C2(CCOCC2)C1 C1(OC)(CNC(=O)CC2CCC(O)C2)CCN(C(c2cnn3ccsc23)=O)CC1 C(=O)(CS(=O)(=O)C(C)(C)C)NCC(CNC(c1c(C)nn(C2CCOC2)c1)=O)C N1(C(C2CN(C(C)=O)C2)=O)CC(CC(=O)NC(CCO)CC(C)C)CC1(C)C c1(CC)cc(C(=O)NCC2(NC(=O)CN3CCS(=O)CC3)CCOC2)ncn1 C(=O)(N=c1ccn(C(F)F)[nH]1)C1(NC(c2cnc(C)o2)=O)CCC(C)(C)C1 N1(C(C2CCC(CC)CC2)=O)CCN(C(=O)C2=NNC(=O)CC2)C2(CC2)C1 C1(C(N(C(C)C)CCNC(=O)COc2ccsn2)=O)CCCC2(C1)CC2(F)F N1(C(c2c(C)con2)=O)CCC(C)(CC(=O)N(C2CCC2)C)C1 c1(C(N2CCC(C)(NC(c3cocn3)=O)C2)=O)ccc2nn[nH]c2c1O Cc1cc(O)c(Cl)cc1C(=O)NC1CC(CNC(C2(C)CCCCC2(F)F)=O)C1 c1(OC)cc(C(N2CCN(C3CCN(C(=O)C(C)O)C3)CC2)=O)c(F)cn1 C1(NC(c2cc(Cl)ccc2O)=O)(CO)CCCN(C(C2CC3CCC(C2)S3)=O)C1 N1(C(CC(COC)OC)=O)CC(=O)NCC1C(N1CC2CC1C2)=O c1(C(=O)NC(CC)CNC(c2cnc(O)s2)=O)cc(C(F)(F)F)ccn1 C(CCCCCNC(c1ccc(SC2CC2)cc1)=O)OC.C12(CC1)C(=O)NC2 CC1(CNC(N2CCc3ncc(Cl)cc32)=O)CCCc2ccccc21 c1(C(=O)NCC2(OC)CN(C(c3ocnc3C3CC3)=O)C2)cccc2c1OCO2 c1(C(N2C(C)CC(NC(CCc3n(CC)ccn3)=O)C2)=O)[nH]c(=N)ccc1C c1(C(N(CC(O)CN(C)C(c2ccc[nH]2)=O)C)=O)nccc2ncccc12 N1(C(COC(C)(C)C)=O)CCN(C(c2cc3cccnn3c2)=O)C2CCC12 C1(NC(CCc2cnc(C)s2)=O)CN(C(c2sc(C)cc2C)=O)CC1F c1(OC)cccnc1C(=O)NC1(CN(C)C(C2CC3C=CC2C3)=O)CC1 N(C(=NCC1CCSC1)N1CCC(F)(c2ccccc2)C1)(C(C=C)C)CC C1(CN(C(c2cn(C3CC3)cn2)=O)CC)CCN(C(=O)CCCC2CCCO2)CC1 c1(SCC(=O)NC(C(C)NC(C(C)N(C(C)=O)C)=O)C)ccc(C)c(C)c1 C(=O)(C1=NN(C)C(=O)CC1)NCC(CC(=O)NC1C(CC)OCC1)OC CC(C)(CC(F)(F)F)C(=O)N(C(=O)CCCCN(C)C)C1CCOC1 C1(CC=C)(NC(c2cnncc2C)=O)CCN(C(=O)C(c2ccc(C)cc2)=O)C1 C1(C(=O)OC)CCC(n2nnnc2C(C2CC2)NCCCC2(C)CC2)C1 C1(N(C(C2CN(CCC)C(=O)C2)=O)C)CN(C(c2ccc(C)s2)=O)CC12CC2 c1(CNC(c2c(CC)con2)=O)cnn(C)c1C(=O)NCC(O)CC(C)C c1(COC)ncc(C(c2nnnn2C(C)CC)NCCCc2cccs2)cn1 C(c1cccc(C=O)c1)=CCOCC(=O)NCC(C)CNCc1cccs1 C=CC(C)(C)CC(=O)NCC1(F)CCC(NC(c2cc(C(C)C)ccc2O)=O)C1 N1(C(C(N2CCCCC(NC(C)=O)C2=O)(C)C)=O)CC2(CCC(=O)NC2)C1 CCCC(CCC)CC(=O)NC12CC1CN(C(C1CCC3(CCC3)O1)=O)C2 Cn1ccc(C(=O)NCC2CC3(C2)CN(C(C2CC(C4CC4)C2)=O)C3)cc1=O c1(OCC2OCCN(C(=O)Cn3cc(CO)nn3)C2)ccc(Br)c(Cl)c1 C(=O)(C(C)(C)C(=O)NCC1CCN1C(=O)CCCNC(c1cccs1)=O)NC c1(CC(=O)NC(C)(C)CSC)ccnn1C.C1(C(C)CNC(=O)COC)CCCCC1 C(=O)(C(CCC(N)=O)n1cc(-c2ccc(N)cc2)nn1)NC1(C(F)F)C(C)C1 C1(NS(CC)(=O)=O)CCC(=O)NC1=O.C1CCNC(=O)O1 Cc1c[nH]c(C(N2CCC(CCNC(C3CC(F)C3)=O)C2)=O)c1 Cc1[nH]nc2ncc(C(=O)NC3CC(C)(NC(c4cc(Br)c[nH]4)=O)C3)cc12 CCC(C)C(CC(=O)N1CC2(C1)CN(C(c1ncc(OC)cn1)=O)C2)SC CS(=O)(=O)C1(C(N2CC(O)(CCNC(c3cc(Br)n[nH]3)=O)C2)=O)CCCC1 N1(C(c2c(C)nc(CC)s2)=O)CCCC2(CC(NC(c3cncc(F)c3)=O)C2)C1 CC1(C)CCN(C(=O)CCc2cnccn2)CC1CNC(C1(O)CCSC1)=O c1(C(=O)NC(CNC(c2ccc(C)n2C)=O)CC(C)C)ccc(F)c(F)c1F C1(NC(Cn2c(C(N)=O)cnc2)=O)CCCC(NC(C2CC2C(N)=O)=O)C1 c1(CNC2CCC(NC(c3cnc(C)nc3)=O)C2)cc(F)ccc1[N+](=O)[O-] O=C1NC2(CO1)CC(C(N1CCCN(C(C3CSCCS3)=O)CC1)=O)C2 C12CCN(CC1)C(=O)CNC2=O.C1C(=O)N1.C(COCC1CC1)OCC C1(C2CCN(C(=O)C(CC(C)C)OC)C2)(OC)CC1.C12CC(C1(C)C)CC(=O)N2 CCCC(C)(CC)C(=O)NC(C)CCN(C(=O)Cc1coc2ccccc12)C c1(NC(=O)NCc2cc(Br)cnc2Cl)ccc(C(F)(F)F)cc1-c1nn[nH]n1 O=C(CC(CNC(c1ccncc1O)=O)C1CCC1)NCC12CC(F)(C1)C2 c1(C(N2CC(CCNC(c3ccc(OC)cc3)=O)(OC)C2)=O)ncc(N)nc1C C1(C(=O)NCCSCCC=C)(CO)CCN(C(=O)CCC=C(C)C)C1 CC(C)(C)C(C(=O)NC1CC2C(NC(=O)C(=C3CCCCC3)F)C2C1)NC(N)=O C(=O)(C(O)CCC(C)C)NCC1CCC(C(=O)Nc2cnc(OCC)nc2)C1 C1(C)(C(N(CCC(=O)OCC)C)=O)CCN(C(C2CCOCC2)=O)CC1 c1(OC)c(C(N2CCCC2C(F)(F)CO)=O)ccnc1F C(C(C)(C)CNC(=O)CSc1ccccc1)N(C(CCOCCOC)=O)C(C)C CC1C(C(=O)NC2(CF)CN(C(=O)CC3CCCOCC3)C2)CCN1C C1(CC)C(C(=O)NC(C)CCNC(c2ccc(CC3CCC3)cc2)=O)CCN1C c1(CC(=O)NC(CN(C(=O)COC2(C)CCCC2)CC)C)ccccc1[N+](=O)[O-] C1(N(C(c2cnc(=N)[nH]c2)=O)CC2CCCCCC2)CC2CCCC(C1)N2 C#CCC(C)(C)C(=O)N1CCCCC(NC(=O)C(CO)C(C)C)C1 c1(C(N(C(CC)CNC(C2COC(=O)C2)=O)C)=O)cnc(OC)c(Cl)c1 Cn1c(C(=O)NCC2(F)CC(CNC(=O)CC3CCOC3(C)C)C2)cnc1O C12(CNC(c3c(OC)ccs3)=O)CCC(CC1)N(C(c1cc(C)ccc1O)=O)C2 N1(C(CCC=C)=O)CC2CS(=O)(=O)CC2(NC(=O)CC2(CC)CCC2)C1 c1(CC)c[nH]nc1C(=O)NCC(C)NC(=O)Nc1ccc(Oc2ccccc2)s1 C(N=c1nc(-c2cc(F)ccn2)[nH]s1)c1c(CC)cccc1 C12CN(CC1(F)F)C2=O.C(=O)(CC(=O)NCCCCNC(=O)C1CC1)OCC CC1=NOC(C)(C(=O)NCCCCN(C)C(C2(C3CCCO3)CC2)=O)C1 O(C=CC(O)(CNC(c1cnc(C(F)(F)F)s1)=O)C(F)(F)F)CC Nc1c(F)ccc(Cl)c1C(=O)NCCCN(CCO)C(C1CC1c1ccccc1)=O N1(C(C(C)=CCC)=O)CC(C(=O)NC(c2cccnc2)C)CCC1(C)C C1(OC)CN(C(c2ccc(C(N)=O)[nH]2)=O)CC1NC(c1oc(CSC)cc1C)=O C1(C(=O)NCCc2ccoc2)(CNC(=O)C(F)C2CCC2)CCCCC1 C1(C(N(CCCCNC(C2(CO)CCC2)=O)C)=O)CC12CCC(C(C)(C)C)CC2 C1(CNC(C(CC)COC)=O)CN(C(c2ccnc(CO)c2)=O)CC(C)(C)O1 N1(C(CNC(=O)OCC)=O)CC2CCC(NC(=O)CCS(N)(=O)=O)CC2C1 Cc1c(C(=O)NCCN(C(=O)C2=CCCC2)CC(=O)N(C)C)sc2[nH]cnc(=O)c12 Cc1ccc(OCCCC(=O)NCC2COCC2NC(=O)C(=O)NC2CC2)cc1 C(=O)(CC(C)(C)c1ccccc1)NCC(C)(C)NC(C12CSC(C1)C2)=O C1(CC(=O)N(CC(C)(C)C)CC)CN(C(c2cccc(F)c2O)=O)CCC1C N1(C(C(CC)C(C)(C)CC)=O)CCC2(CCCN(C(=O)C3=CCCC3C)C2)CC1 C1(OCCNC(c2c(C(C)C)c[nH]n2)=O)CCN(C(=O)C(C)(C)CF)CC1 O=C(N=c1c(F)c[nH]cc1F)c1ccc(F)cc1Br N1(C(c2ccc(CC)[nH]2)=O)CCC2C(C1)CN2C(C1CC1(F)F)=O N1(C(c2c(C#C)c[nH]n2)=O)CCN(C(c2c[nH]nc2C(C)(C)C)=O)CC1C1CC1 N1(C(c2cc(C)c(Br)c(C)c2)=O)C(C(=O)NCCF)CC2CCCCC12 Cc1cccc(CC(=O)NC2CC(NC(=O)CC3(O)CCCC3)C23CCC3)c1Br C12CN(CC13CC3)C(=O)CC1CCN21.N1(C(=O)CC2CC2)CCC(F)CC1.CO N1(C(C2N(C(c3n(C=C)ncc3)=O)CC(F)C2)=O)CCn2nncc2C1 c1(NC(C(=O)NC(CC(C)NC(CN(CCC)C)=O)C)=O)cccc(C)c1F C(=O)(C1=Cc2ccccc2C1O)NC1CC(CCNC(CCNC(N)=O)=O)C1 C12CC(=NO1)C(=O)N1CCC1C2.C1(ONC(=O)OC(C)(C)C)CCCC1 C12(NC(c3c(Br)cc(C)s3)=O)CCCCC1N(C(=O)CCC#N)CC2 c1(C)ccc(Br)cc1.O=C(CC(O)c1cn(CC2CCC2)nn1)N1CCC1C(=O)N c1(CNC(C2(N(C)C)CCC2)=O)ccc(C(=O)NCC2(CCO)CC2)cn1 N1(C(COCCOCC#C)=O)CCCC(C2CN(C(=O)CSC(F)(F)F)C2)C1 C(C)(C)(C(=O)NCc1nc(CNC(=O)Cc2csc(S)n2)cs1)OC(C)=O C(C)(CCC(=O)N(C)CC=CC(N1CCC(n2cccn2)C1)=O)OC C1(NC(CC2=CCN(C(C=CC3N(C)CCC3)=O)CC2)=O)CCc2nccn2C1 Cc1ccc(CC(=O)NCC2CCCCN(C(C3CCCO3)=O)C2)cc1C N1(CCC(=O)N(C)CCN(C)C(C2C=CCCC2)=O)CCCS1(=O)=O c1(OC)ccc(C(=O)NCCCN(C(=O)Cn2nc(C)cc2C(F)F)C)c(Cl)n1 C1(CCC)(CO)CCN(C(=O)C(C2CCOC2)NC(=O)C(C)=NOCC#N)C1 C(=O)(CCC(CC)OC)NCc1c(C(=O)NCc2c(CC)onc2C)n(C)nc1 C=CC1OCCC1C(=O)NC(C)CNC(=O)CP(C)(C)=O Cc1ccc(Cl)c(C(=O)NCC(CO)NC(c2c[nH]nc2C2CCOC2)=O)c1 c1(C2C3(CCC3)N2)nnnn1CC1CCCO1.C1(C(C)C)(CCC)CC1.CSC CN(C)NC(=O)CCC(=O)N1CCC2CCC12CNC(c1cc(C(N)=O)co1)=O N1(C(C2CC3(CC(=C)C3)C2)=O)CCC2(CC1)CN(C(c1ccnnc1)=O)CCO2 S(=O)(=O)(c1cc(Cl)ccc1F)NCC1CC(F)CN(S(=O)(=O)CC2CCC2)C1 C1(CC(=O)NCC(C)NC(C2(Cl)CC23CCC3)=O)Cn2ccnc2NC1=O C1(CCC=C)(NC(=O)N(CCO)CCOc2ccccc2Cl)CCN(C)CC1 c1(CC)[nH]c(C(=O)NCC2CC(NC(C3(N4CCCCC4)CCCC3)=O)C2)nc1Cl C(C)(CCCC(=O)Nc1ccc(O)cc1)NC(C1(C)CC(=C)C1)=O N1(C(CCC2OCC(C)(C)C2)=O)CCC2(CCCN2C(C2CC(=C3CC3)C2)=O)C1 Cc1nnc2n1CC(C(=O)Nc1ccccc1-c1cn(CCOCCO)nn1)CC2 N1(C(CC=C)=O)CC(NC(=O)Cc2cncn2C)CC1C C1(N(C(=O)CC2CCCN(C(c3ccc(CO)cn3)=O)C2)C)CS(=O)(=O)C1(C)C c1(C(N(C2CN(CC=CCC)CC2O)C)=O)cnc2c(cnn2C(C)CC)c1 c1(CC(=O)NCCN(C(c2cc(C)c(N)cc2F)=O)CC)cn2c(n1)CCCC2 C1(NC(c2c(C)nsc2)=O)CCCC12CN(C(=O)CCCn1ccnn1)C2 N1(C(C23CC(C)C2C3)=O)CCN(C(c2ccsc2)=O)CC1C CC(C)(CC(F)(F)F)C(=O)N1CC(n2cc(CNC(C3C(C)(C)C3(F)F)=O)nn2)C1 N1(C(C(=O)N(C)C)=O)CCc2nc(O)cc(C(N3CCc4sc(Cl)cc4C3)=O)c2C1 NS(=O)(=O)c1sccc1C(=O)NCC1C2CCCC1N(C(c1cnco1)=O)C2 CC1(C(N2CC3(CCC3NC(c3cccc(Cl)c3F)=O)C2)=O)CCCS1(=O)=O N1(C(CSCCCC)=O)CC(NC(=O)CS(=O)(=O)CCOC)C2(CCC2)C1 C(=O)(CC(CC)SC)NCC1(CNC(C2CC(=C)C2)=O)CCC1 c1(OC)ccc(SC)c(OC)c1C(=O)NC1CC1NC(=O)C(O)CC[S+](C)C C1(CNC(C2C(CC)N(C)CC2)=O)CCC12CCN(C(c1oncc1C)=O)CC2 C=CCC(C(=O)NCCC(C)(C)NC(c1cc(C(C)(C)C)c[nH]1)=O)OC n1(CCCNC)c(N(C)CCc2c(C)noc2C)nnc1C(C)OC N1(C(c2cc(OC)n[nH]2)=O)CC(NC(c2cnc(C)s2)=O)CC(O)C1 C1(NC(C(C)OC)=O)CN(C(c2ccnn2CC(C)C)=O)CC1n1ccnn1 c1(C(=O)NC2CCCN(C(C3(CF)CC3(F)F)=O)CC2)ccc2c(O)n[nH]c2c1 c1(-c2cn(C3CCN(C(C4(SCC)CC4)=O)C3)nn2)ccc(C(=O)O)cc1F c1(N2CCCC(N(C(C=Cc3c(C)ccnc3)=O)C(C)C)C2)ccnc(C#N)n1 C(=O)(C1=CCC(F)(F)CC1)N1C2CC(CNC(C(C)(C)OC(C)C)=O)CC1CC2 N(C(=NCC1CCOC1)NC(C)Cc1cccnc1)CC1(C=C)CCC1 c1(CNC(C2C(C)C2)=O)cnn2c1CN(C(C1(C#N)CCOC1)=O)CC2 CCC(C(=O)N1CC(O)(C(F)C(=O)N(CCCN(C)C)C)C1)NC(N)=O n1(CCN(C(C(=O)N(C2CSC2)CC=C)C)C)cc(C)cn1 N1(C(COCCC=C)=O)CC(NC(=O)COCCCF)CC1CO Cc1nn(C2CC2)c(Cl)c1C(N1CCCC(NC(=O)CCn2cccn2)CC1)=O CC(F)(CC1CCCC1)C(=O)NNC(=O)c1ncc[nH]1 c1(CC(=O)OCC)cccc(NC(=O)COC(c2cncnc2CC)=O)c1 C(=O)(CC(C)CCC=C(C)C)N(CC)CC.c1(CCO)cccs1.C1(=O)CO1 c1(CC)ncsc1C(=O)NC1CCN(C(=O)Cc2cnc(CC3CC3)s2)C1 Cc1nc(C)c(C(=O)NC2(C(=O)N(C(C)CN(C)C)C)CC2(C)C)o1 N(C(=NCc1ccccc1)NC1CCCC1)CC(C)C.n1(CC)ncc(C#N)c1N c1(C(=O)NCC2N(C(CCc3ccc(C)nc3)=O)CC2)cnc2ccnn2c1C C1(O)(CNC(CCCC)=O)CCN(C(c2n[nH]c(Nc3ccccc3)c2Cl)=O)C1 c1(C(C(=O)NCCCN(C(=O)CN2CCC(O)CC2)CC)O)ccc(Br)cc1 C1(CNC(C2CCCN(C(C)=O)C2)=O)CN(C(=O)C2CC2)CC1(F)F C1(C(N2CCC(CN(C)CC)C2)=O)C=CCN(C(=O)CC2CCOC2=O)C1 c1(NC(C2CN(C(CCc3onc(C)n3)=O)C2)=O)ccc2n[nH]cc2c1C Cc1cc(F)ccc1C(F)(F)C(=O)N1CCC(NC(C2CCC(=O)O2)=O)C1 C1(C(=O)NCCN(C(C2C(=C)C2)=O)CC)COC(=O)C1 C1(C(N2CC(NC(COC)=O)C2)=O)CCCCCCN1C(c1ccoc1)=O C1(NC(C(CO)OC)=O)CCN(C(=O)CC2=CCCCC2)CC(C)(C)C1 N1(C(c2cscc2Br)=O)CCN(C(c2n[nH]cc2F)=O)C2CC12 C1(C2CCCN(C(c3ccc4c(c3)COB4O)=O)C2)(NC(CC(C)(F)F)=O)CC1 c1(C(N2CC(O)C(F)C2)=O)cnc2ccsc2c1 CC1c2c(ccc(Cl)c2F)CCC1N=c1ccc(C(=O)NOC(C)(C)C)n[nH]1 N1(C(Cc2nc(C)sc2)=O)CC(C(=O)NCC2NC(=O)NC2=O)C(F)(F)C1 c1(N(C2CCCCC2)C=O)cccc(-c2cccc(N3CCCCC3)c2)c1 CCCC(O)CN(C(=O)CCCN(C(=O)C(c1cccnc1)O)C)C C(CCCC(C)NC(c1cc(C)sn1)=O)NC(C(CC)SCc1ccccc1)=O N1(C(C2(C)CC2(F)F)=O)CCN(C(c2cccc(F)c2O)=O)CC1c1cn[nH]c1 C1(C#N)(C(=O)NCC2N(C(C3ON=C(C)C3)=O)CCC2C)CC2C=CC1C2 C(=O)(C1=C(C#N)CCC1)NC(CN(C(C1CCCN1C)=O)CC)C c1(OC)ccc(C(=O)NC(c2ccc(OC)nc2)CC2CCCCC2)c(C)c1 Cn1cc(C(=O)NC2CN(C(=O)CN3CCOC3=O)CC2N=[N+]=[N-])c(O)nc1=O c1(NC(C)=O)cc(C)cc(F)c1-c1cc(-c2cc(O)nc(Cl)c2)n[nH]1 C1(CCC(=O)NC2CCC(CCNC(C3CCC3)=O)C2)(N(C)C)CCCC1 N1(C(=O)CCc2cccc(C(F)(F)F)c2F)CCCC(C2CCNCC2)C1 CCC(C)(C)CC(=O)N1CC(CC(=O)NOC(COC)COC)OC(C)C1 N1(C(N2CCC(C(F)F)C2)=O)CCc2c(N)cccc21.c1(C(N)=O)csc(C(F)(F)F)n1 N1(C(C(CC)CC2CCCC2)=O)Cc2occ(C(=O)N(C3CCOC3)C)c2C1 Cc1cc(C(N2CCN(C(c3ccc(C4CC4)cc3)=O)C(CO)C2)=O)cc(Cl)c1 O=c1cc(CN2CC(F)(c3cccnc3)C2)oc2ccccc12 c1(NC(C2CC(F)CN2C(=O)CCCC(F)(F)F)=O)ncc([N+](=O)[O-])cc1I c1(SC)ncc(Br)c(N2CCCC(C(=O)NC(C3CNC(=O)O3)C)CC2)n1 N1(C(Cn2c(C)cnc2)=O)CCC2(NC(=O)CCc3cccc(F)c3)CC2C1 C12(C(N3C(NC(=O)OC)CCCC3)=O)COCC1CN(C(C1CCCC(=O)N1)=O)C2 N1(C(c2cc(C)cc(Cl)c2)=O)C2CCC1CC(NC(C13CCCC1C3(F)F)=O)C2 C1(N(C)C(C2(C(N)=O)CC2)=O)CCCC(NC(=O)CC2(C#N)CC2)C1 C(=O)(C(C)(CSC)NC(C1CC(C)(CC)C1)=O)NCCCOCC=C CC1CN(C(=O)CC2CCC2)CCC1CNC(=O)CCCC1CCCCC1 Cc1cc(NC(=O)C(C)OC2COC2)ccc1C(F)(F)F.c12ccc(cc1)o2 N#Cc1cc(C(=O)NC2CCCN(C(=O)CCN3CCC(F)C3)C2)c[nH]1 N1(C(C(CC(C)C)NC(=O)Cc2cccc(F)c2)=O)CCC(C2CCCC2)C1 C=Cn1nccc1C(N1CC(NCC2CCCO2)C(CNC(=O)C(C)=CC)C1)=O C12CN(CCO1)C(=O)NC2C.C1(NC(C2CC(OC)C2)=O)=CC=CCCC1 N1(C(CCC(C)=O)=O)CC2(C)CC1(C(=O)NC1C=CCCCC1)C2 c1(C(N2CCCC3(NC(C4C(=C)CC4)=O)C(C2)C3)=O)cnc2c(Cl)cccn12 N1(C(CCC(=O)N(C)C)=O)CCc2c(C(=O)NC3(CO)CCOC3)cccc2C1 N1(C(Cc2ccc(C)cc2O)=O)CCCC2(NC(=O)C=CC(F)(F)F)CCCC12 c1(C(N2C(CN(C(CN(C(C)C)C)=O)C)CCC2)=O)cnc2ncccn12 n1(CC(N2CCC(N(C(=O)CCSCC(N)=O)C)C2)=O)nc(C)c(Cl)c1C c1(NC)c(C(=O)NC(CNC(=O)C(C)(C)C(F)F)C(C)(C)C)cccc1N c1(SCC#C)cnccc1NC(C1CC(=O)C1)=O N1(C(C2CC(CC)(CC)C2)=O)CCC(NC(c2cnc(C)cn2)=O)C(C)C1 C1(NC(C(c2cnn(C)c2)OC)=O)CC2(CCN(C(=O)C=C(Cl)Cl)CC2)C1 C1(NC(C(C)n2cccc2)=O)CCN(C(C2(C(C)(C)O)CC2)=O)CC1C c1(C(N(CCCNC(C2CC23CC(O)C3)=O)C)=O)ccnc2[nH]ncc12 Cc1cc(N2CCC(NC(=O)COc3cnn(C)c3)CC(O)C2)ccc1[N+](=O)[O-] Cc1nc2cc(C#N)ccc2cc1-c1cccc(C(O)C(=O)O)c1 C1(C)(CNC(Cc2cn(CC)nc2)=O)CCCN(C(C2CC(CN(C)C)C2)=O)C1 C1(C(N(C2COCC2O)C)=O)CCN(C(=O)C(O)CC(N)=O)C(C)(C)C1 N1(C(C(=O)NCCNC(C)=O)=O)CC2CCC2(NC(=O)C(O)C(C)(C)C)C1 N1(C(CNC(c2c(C)csn2)=O)=O)CC(C)C12CCOCC2 C1(O)(C(N2CCC(CNC(c3cnc(COC)s3)=O)C2)=O)CCCCCC1 N1(C(CC(C)C2CCCCC2)=O)CC2(NC(=O)CN3CCCC3=O)CC1C2 CC1OCCC1(C)C(=O)NCc1cccc(C(=O)Nc2cnn(C)c2)n1 N1(C(c2snc(OC)c2Br)=O)CCC(CNCC2(C(F)(F)F)CC=CCO2)C(C)C1 Cc1cnc(C(N2CCCC(CCC(N3CC(O)(CCO)C3)=O)C2)=O)c(F)c1 CCCCS(=O)(=O)NCC(=O)NC(C)CC1CCCN1C(=O)COC(C)=O c1(C(N2CCCC(C)(NC(CN3C(C)CCC3)=O)C2)=O)cc([N+](=O)[O-])c(O)cc1N Cn1cc(C(=O)NC2(CNC(C3(C4CC4)CC(=O)C3)=O)CCOCC2)n(C)c1=O c1(NCC=CCNC(CCc2onc(COC)n2)=O)nc(Cl)ncc1C(C)C C1(CNC(c2cc(C(C)(C)C)on2)=O)CN(c2nccnc2F)CCO1 C(C(CC(F)(F)F)NC(C1CCCCC1O)=O)NC(c1ccns1)=O N1(C(C2C(C)SCCC2)=O)CC(CNC(=O)Cn2ncnn2)C2(CC2)C1 n1(C(C(=O)NCC#CCNC(C(C(C)SC)O)=O)(C)C)cc([N+](=O)[O-])cn1 CCCCC(C(=O)NCC(C)(C(C)C)NC(=O)CC1CCOC1)ON=C(C)C n12cc(nn1)CC(=O)N1CC2C1.c1(COCC)cn(CC)nn1.C1(C=O)CCCCS1 c1(OC)cc(C(=O)NC2CC2C(=O)NCc2cccnc2O)cnc1O N1(C(C2CC3(CC3)CN2C(c2[nH]cc(C)c2C)=O)=O)CCn2cc(O)nc2C1 N1(C(C2C3(CC(NC(c4cc(C5CC5)no4)=O)C3)C2)=O)CC(F)(F)C(F)(F)C1 C1(C(=O)NCC2CCCN(C(c3cnc(C4CC4)s3)=O)C2)CC2(CCCC2)CO1 CC1CCCCCC1C(=O)NCC1(C)CCCN1C(=O)C(CN)n1cccn1 N1(C(C(CC)=CCCC)=O)CCC2(CCCN2C(c2csc(C)n2)=O)C1.CCC C(CO)(CO)(CN=c1[nH]c2c(c(=NCc3cc(Cl)cc4c3OCC4)[nH]1)SCC2)OC c1(CCC)c(C(=O)NCC(CC)NC(=O)Cc2ccn(C)n2)[nH]c(C)c1C(N)=O C1(C(=O)NCCN(C(C2CCCN2C(C)=O)=O)CC)(C(F)F)CCCCC1.C(N)(=O)N c1(CC(=O)NC2CCCCN(C(C3C(=C)CC3)=O)C2)ccc(C)c([N+](=O)[O-])c1 CN1CC(C)(C(=O)NC2CN(C(=O)CC3(C)OCCO3)CC2O)CC1=O c1(C(=O)NCC(CN(C)C(c2ccnn2C2CC2)=O)O)cccn1C C(=O)(C1CCCc2cccnc21)N1CC(CC(C)CNC(C2(C)CC(C#N)C2)=O)C1 C(=O)(C1=CC2C=CC1C2)NC1CCCC(C(=O)NCC2(C)CCOCC2)CC1 c1(C(N2C(C)(C(=O)Nc3c(OC)ncnc3)CC2)=O)cc(F)cc(F)c1O C1(C(=O)NC(CC)(C)CNC(=O)CC2CC3(CCO2)CC3)CCC2(CCC2)CO1 c1(N(C(=O)NCC2(C(=O)OC)CC2)C2CC2)cc(C)nn1-c1ccccc1CC C(CN=c1nc2c(cnn2C)c(NCc2ccc(Br)cc2F)[nH]1)c1c(C)ocn1 N1(CCCNC(C2N(C(C3CC(C(=O)OC)C3)=O)CCC2)=O)CCCCC1=O C1(NCC2CCC(CN=[N+]=[N-])O2)C2CC3CC1CC(O)(CC2)C3 N=c1[nH]c(N2CCC(NC(c3ccc(Cl)nc3)=O)C(F)C2)ncc1[N+](=O)[O-] c1(SC)cc(C(N2CCC(n3cc(CNC(=O)C#CC(C)C)nn3)C2)=O)sc1C c1(-n2c(C3OC(=O)NC3(C)C)nc(CC(OC)OCC)n2)cnn2c1CCCN2 c1(OC)cc(Cl)cc(F)c1CN1CC2C(C1)N2C(=O)Cc1cccc(Cl)c1F CCCC(CC)CCC(=O)N1CC(CC(N2CC(C#N)C2)=O)C2(CC2)C1 C1(N(C(=O)Cc2cnc[nH]2)CC2CC2)CCN(C(C2CN(C(N)=O)C2)=O)CC1 Cc1cc(C(=O)NC2COCC2NC(C2CC=CC2)=O)c(C)n1NC(N)=O c1(C(=O)NCCOC2CCN(C(c3cnsc3)=O)C2)cc2n(c1)CCCC2 c1(C(N2CC3C(NC(C4CCC(CC)O4)=O)(C3)C2)=O)ccc2nncn2c1 C(C(CNC(=O)C(c1cncc(F)c1)C)C(F)(F)F)NC(c1c(C)nn(C)c1)=O N1(CC(C)C)CC2(C)CN(C(=O)CC3CC3(C)C)CC2(C)C1 c1(C(N2CCSC(C(F)(F)F)C2)C(=O)NCCCC)cccc(OC2CC2)c1 n1(CC(CC)O)cnc2c(C)cccc2c1=O c1(N2CCCC(CCC=C)C2)nccc(=NCCC2(CO)CCC2)[nH]1 C#Cc1ccc(C(N2CC(OC)C(C(=O)NCc3nncn3C(C)C)C2)=O)cn1 C1(CC(=O)Nc2ccsc2C(=O)Nc2ccsc2-n2cncn2)CC=CCC1 c1(NCCC(=O)N(C(C2(C3CCCO3)CC2)C)C)ccccc1 C12(COC)CC(CO1)N(C(C1CCCN(C(c3c(Cl)ccnc3F)=O)C1)=O)C2 c1(CCC(N2CC(C(N(C3CCOC3)CC)=O)(CCOC)C2)=O)cc(C)n(C)n1 c1(C(N2CC(N(C(c3ccc(C)cc3)=O)C)C(C)CC2)=O)cnc2[nH]cnc2c1 Cc1nnc(CC(=O)NC(CNC(=O)Cn2nnnc2C(C)C)CO)o1 C1(C(N2CCCC(O)(CNC(c3ccncc3F)=O)C2)=O)CCn2nccc2C1 CC1(C)C(CC(=O)NCC2(n3cc(-c4ccsc4)nn3)CC2)CC1O CC(O)C(F)(F)C(=O)N1CC(CCCCNC(C2CN(C)CCCO2)=O)C1 c1(C(=O)NCCCNC(c2c(C(C)C)noc2)=O)csc(N=S(C)(=O)N(C)C)n1 c1(C2N(C(C3CC(=C(F)F)C3)=O)CCC2)ccc2ccccc2n1 N1(C(COc2c(C(C)C)cccc2)=O)CCC(NC(C2(C#N)CCC2)=O)C(O)C1 c1(CC(=O)NC(CCNC(C2C(CCC)C2)=O)(C)C)cc(C(F)(F)F)n(C)n1 N1(C(C(=O)OCc2c(Cl)ccc(OC)c2)=O)CCn2nncc2C1 C(=O)(CS(=O)(=O)C1CCCC1)N1CCN(C(c2c(Cl)cc(C)s2)=O)C(C)C1 C1(NC(CC(=C=C)C)=O)CC2CCC(C1)N2C(=O)CCCOc1cccc(F)c1 C(=O)(CCCCC(N)=O)N1CCC(NC(C(C)Cc2ccccc2)=O)C(C)C1 C1(F)(CNC(C(CNC(C)=O)(C)C)=O)COCCN(C(=O)C(C)(C)C(C)C)C1 N1(C(C)C)CC(CN2CC(C3(C)CCC(=O)N3)C2)CC1=O.c12ccccc1S2 C1(CC=C)(NC(C2CCCC2(F)F)=O)CCCN(C(c2sccc2C#N)=O)C1 C(=O)(CS(=O)(=O)CCOC)N(C)CC1(NC(Cc2n(CC)ncc2)=O)CC1 C1(C(=O)NC(C)CN(C)C)(CC)CN(C(=O)C(C)c2ccsc2)C1 c1(OC)ccc(CN2CCC(O)C(C(=O)NCCc3ccccc3C)C2)nc1Br C=CCCC(C(=O)NCCCCC(=O)NCC(C)(C)CC(C)C)C(C)C N#CC1CCCN(C(C2C=CCN2Cc2ccccc2Cc2ccccc2)=O)C1 Cc1ocnc1C(N1CCCC1Cn1cc(CCC(N)=O)nn1)=O c1(OC)cc(C)cnc1C(N1CC2C(CN(C)C(c3nc(O)c(C)s3)=O)C2C1)=O c1(CN(CCN(C(=O)C(=O)NC)CC)CC)nccs1 N(C(=NCC(C)(C)C1=CCOCC1)NC(C)C)Cc1c(C)ccc(C(F)(F)F)c1 C1(NC(C2C(C(N)=O)C2)=O)CC(NC(=O)CCc2cc(F)cc(Cl)c2)C12CCC2 C(C(C)N=c1nc(N2CC=CCC2)c2sccc2[nH]1)SC CC(C(=O)NCCC1CC(NC(=O)COCC2CCOCC2)C1)C(F)F C(=O)(C(=O)C(C)(C)C)NCCCCCC1CCN(C(Cc2cnc(C)[nH]2)=O)CC1 C(=O)(CC(C)C(=O)OC)NC1CCC(NC(C2CCN(CC)C2)=O)CC1 c1(C(=O)NC(CCC)C(=O)NC2COCC2C(N)=O)cc(C)nc(O)n1 N1(C(CNC=O)=O)CC(NC(c2ccc(OC3CCC3)cn2)=O)CCC(O)C1 N1(C(c2cc(C)[nH]n2)=O)CC2CC1CC2NC(=O)C(C)OCC(C)C N1(C(Cc2c(C(=O)OC)csc2)=O)CCOCC(NC(c2cnc(S)n2C)=O)C1 c1(C(N2C(CC)C(NC(C3(C)CC3(Cl)Cl)=O)CC2)=O)ccc2c(c1)nnn2C N1(C(=O)C(c2ccc(Cl)cc2)O)CC(c2nc[nH]n2)C(C2CCCC2)C1 S(=O)(=O)(c1cccc(OC(F)F)c1)NC(C1(c2cccc(F)c2)CC1)=O c1(OC)cccc(OC(c2ccnn2C(F)F)=O)c1.C12CCC(C1)C(=O)NC2 C(CCC(C)C(=O)NC1CN(C(c2ccc(-c3cccs3)[nH]2)=O)CC1C)OC C12(C(=O)NCC(C(C)(C)C)NC(=O)CCn3ccnc3)CCC(O)C1CC2 CC(CCN(C)C(C1(Br)CC1C(=O)O)=O)NC(=O)OC(C)(C)C c1(CC)cc(C(=O)NC2CCCCC2CNC(C2(C#N)CCCO2)=O)cc(O)n1 c1(NC(c2c(CCC)[nH]cc2)=O)cccc(NC(C2CCCC(CC)O2)=O)c1 N1(C(c2cnc(OC)s2)=O)CCN(C(C23CC(C)C2C3)=O)CCC1C c1(NC(c2ccc(CNC(=O)Nc3cccnc3Br)cc2)=O)ccc(Br)cc1Br Cc1[nH]c2ccc(Br)cc2c1C(=O)OC1CCC(F)CC1 c1(C(N2C(C)CC(CNC(C(C=C)(C)O)=O)C2)=O)ccc2c(c1)CCCS2 N1(C(C2C3CC(=O)CC32)=O)CCN(C(c2cncc(F)c2)=O)C(C2CC2)C1 C1(C(C)O)CCN1C(C1(CNC(=O)CCn2ccnc2)CC1)=O c1(C(N(C2CN(C(C3(OC)CCC3)=O)C2)C)=O)cc(C)ns1 N1(C(C(C)OCCC=C)=O)CCC(C(C)NC(=O)NCCSC)C1 C1(CNC(c2ccc(OC)s2)=O)CCN(C(=O)Cc2cnnn2C)C(C)C1 C1(F)(CNC(C2CCC(O)C2)=O)CCC(CNC(C2CC(O)C2)=O)C1 C1(CO)CC2CCCC2N1C(=O)N=c1[nH][nH]c(-c2ccccc2)c1Br C1(CCC(C)C)CCC(N(C2CCCN(C(=O)OC(C)(C)C)C2)C)CC1 c1(NC(C2CC(C)CN2C(C2CC2c2ccccc2)=O)=O)cc(F)c(F)cc1Cl C1(C(N(C)CCNC(=O)Cn2ccc(C(F)(F)F)n2)=O)CCc2nnc(O)n2C1 N1(CCC)C(=O)CC(C(=O)Nc2cn(C)c(C(=O)OC)n2)C1c1cccnc1 C1(NC(CCC#N)=O)CCN(C(=O)C=Cc2cccc(Cl)c2)C12CC2 CCC(O)C(C)C(=O)NC1C(C(CCc2ccc(Cl)s2)NC(=O)COC)CC1 C1(C(=O)OC)CN(c2cc[nH]c(=NCCC3CC3)n2)CC12CCOC2 N=c1[nH]nc(Cl)cc1C(N1CC2CC2(CNC(=O)Cc2cnc[nH]2)C1)=O N1(C(CCCC(=C)C)=O)CC(NC(=O)CCc2cnc[nH]2)CC2(CCOCC2)C1 C1(C(=O)NC(CCC=C(C)C)c2nnnn2CC2CC2)Cc2ccccc2S1 CP(C)(=O)C(CC(=O)NC1CC1CNC(=O)C(c1ccc(O)cc1)=O)C(F)(F)F N1(C(Cc2c(OC)ccnc2)=O)CCCC2(C1)CN(C(=O)C(C)(O)C1CC1)C2 C1(NC(c2ccc(COC)[nH]2)=O)CN(C(=O)CSCC2CCCO2)CC1C1CC1 N1(C(C2C(C)OC(=O)N2)=O)C2CCC1CN(C(=O)C(=C1CCCCC1)F)C2 C1(CC(=O)N(C2CCN(C(CCc3scc(C)n3)=O)CC2)C)CCCC(C)(C)O1 O=[N+]([O-])c1ccc(C2(NC3CC3c3ccc(Cl)cc3)CCCC2)nc1 C(CC(CNC(=O)CSC1CCCC1)NC(C1CN(CC(C)C)C1)=O)OCC C(=O)(C1=CCCN(C(=O)CC2NC(=O)NC2=O)C1)N(CC(C)O)CCO Cc1nc(C(C)NC(=O)C(CN(C)C)NC(=O)CCCN(C)C)no1 N1(C(C2(CC)CC2)=O)CCC(CC2CC(CC(=O)Nn3cncn3)C2)C1 CC1(C)CC(CNC(C2CCOC2)=O)CN1C(=O)C1=CCCC1 c1(CNC(=O)Nc2[nH]nc(C(CC)N(C)C)n2)cc(OC(C)(C)C)ccc1Cl c1(C(N2C(CNC(CCS(C)(=O)=O)=O)CCC2)=O)ccc(O)cc1[N+](=O)[O-] c1(CC)cc(=NC(=O)c2ccccc2Nc2cncc(C#N)c2)[nH][nH]1 C1(NC(C2CCC(F)(F)CC2)=O)CC12CCN(C(=O)Cc1ccnc(O)c1)CC2 c1(C(=O)NCC2CC3(CC(NC(C4CC4(F)F)=O)C3)C2)ncc2cc(Cl)ccn12 N1(C(C(=O)NCCC)C(C)C2CCC2)CCCC(O)(C(F)F)C1 N1(C(c2cccc3nsnc23)=O)CCC(C2CCN(CC3CCCCO3)C2)CC1 N1(C(c2cnn(C(C)(C)C)c2)C(=O)NC(CC)C)CCC(CC(C)C)(CC)CC1 N1(C(=O)CCCc2nccs2)CC(C2CN(C(c3ccc4c(c3)CCC4)=O)C2)C1 N1(C(=O)OC(C)(C)C)CCC(C)(CNC(=O)NC2(c3nn[nH]n3)CCCOC2)C1 C(=O)(CCCC(C)(C)NC(c1cc(O)cc(F)c1)=O)NC(c1cnn[nH]1)C C(CCN(C(CC)C(=O)NCCN(CC)CC)C)(C(=O)SCC)N(CC=C)C C=C(C)CCCC(=O)N(CCC)CCNC(c1ccc(C)cn1)=O Cc1cnc(CNC(C2CC(F)CN2C(=O)Cc2ccccc2)=O)c(F)c1 Cc1ccsc1C(N1CC(O)(CCNC(C2C=CCC2)=O)C1)=O C(=O)(CCCCC(F)(F)F)NCCc1c(CNC(n2c(C(N)=O)ccn2)=O)nco1 c1(C(=O)NCC(CNC(CCC=CC)=O)O)cc(Br)ccc1NC(C)=O N1(C(c2n(C)nc([N+](=O)[O-])c2)=O)CC2CC(NC(C3CCC(=O)N3)=O)CC1C2 C1(CC)CCC(C(=O)NCCCCCn2cc(CC(C)(O)CC)nn2)CC1 C1(CC(=O)NCC2CCC(NC(C3CCN(C)CC3)=O)C2)CCC(C)(C)CO1 Cc1nn(C)c(F)c1C(=O)N(CCCNC(c1conc1C1CC1)=O)C N1(C(C)=O)CC(O)CC1C(N1CC(N(C(=O)CN(C2CCCCC2)C)CCO)C1)=O C1(NC(CCN(C)CCNC(=O)COCC(F)(F)F)=O)CCc2nc(C)ncc2C1 C1(CNC(c2c(N)cc(F)cc2)=O)CC2CCC1N(C(C1CC13CC3)=O)C2 c1(C(=O)OC2CC(F)C2)cc2cc(F)ccc2s1 N1(C(C=Cc2n(CC)ccn2)=O)C2CCCC1CN(C(c1oc(C)nc1C)=O)C2 c1(NCCc2cc(C)ncn2)cc(=NCCOc2ccncc2C)[nH]c(C)n1 N1(C(C(C)N(C(C)=O)C)=O)CC2(CC(CC(=O)NC3(CO)CC4CCCC34)C2)C1 C1(C(N2C(C)(CCO)CC2)=O)CCN(C(=O)C=Cc2ccoc2)CCO1 C1(OCCNC(c2cc(C(=O)OC)[nH]c2)=O)(C)CCOCC1.C1(C(=O)N)CCC1(F)F CC12CC(C(=O)NC3CCC(C)(CNC(c4coc(Cl)n4)=O)CC3)(CCO1)C2 c1(OC)ccccc1C(N)CC(=O)NC1CC1c1ccccc1 C1(C(=O)NCC2N(C(CSC(C)C)=O)CC(O)C2)CCc2ccccc2O1 Cc1c[nH]cc(C(N2CC(CNC(=O)CCCCC3CC3)CC(C)C2)=O)c1=O c1(CC(=O)NC2CCCC2NC(c2ccc(F)o2)=O)nc2c([nH]1)CCCC2 N1(C(C2(SC)CC2)=O)CC(CNC(=O)CC(c2cccc(F)c2)O)C(O)C1 N1(CC(C)NC(=O)C(C)(Cl)Cl)CCN(C(C2CC2C(F)(F)F)=O)CC1 c12cc(C)c(cn1)o2.c1(OC(C)=O)ncccc1-c1ccnn1C C1(CNC(c2nn(C)c(Br)c2)=O)CCN(C(=O)Cc2ccnc(O)c2)C12CC2 C12(C(N3CC(NC(=O)C=Cc4c[nH]cn4)(COC)C3)=O)CC3CC(CC(C3)C1)C2 c1(NCC=C2CCN(C)C2)nc(N2CCC(C#N)C2)c2c(n1)CCCCCC2 Cc1nc(C(=O)NCC2CCC(C)N(C(c3cc(O)nc(C)n3)=O)C2)cc(O)n1 C1(NC(c2c(C)n(C)nc2)=O)CCN(C(c2cnn(C)n2)=O)CC12CCC2 C1(OCC)CN(C(=O)Cc2nc[nH]n2)CC1Sn1ncc(C(=O)OC)c1C1CC1 c1(C(N(CCN(C(c2c(NCC)scn2)=O)C)C)=O)cccn2nccc12 CCC(CC)CC(F)C(=O)NCC(CC(=O)NC(COC)CCO)OC CN1CCN(C(c2cnco2)=O)CC1C(N1CCC(CC2CCC2)C1)=O C1(C)(N(C)CC)CCN(C(C2CC(O)CN2C(=O)C(C)C(F)F)=O)C1 c1(CC(=O)NCCCCN(C(C(F)OC)=O)C)csc(Cl)n1 N1(C(C2N(C)CCCC2)=O)CCC2(C1)CN(C(c1cscc1C1CC1)=O)C2 N1(C(C(=C(C)C2CC2)F)=O)CCC(NC(c2cnccn2)=O)CC1C Cc1cc(Cl)ccc1C(=O)NCCCCC1CCCN(C(=O)Cc2ccsn2)C1 c1(N2CC(C(N(CC(C)C)CC(C)C)=O)CC(F)(F)C2)ncnc2c1ncn2C C1(N(C(C=C(C)C)=O)CC2CC2)CCCN(C(=O)CC(C)n2cccn2)C1 C(=O)(C(C)(CC)CCCCC)N1CCC(CNC(C(C=C=C)C)=O)C1 C1(CCC)CCN(C(C2CCNC2=O)=O)CC1NC(=O)COCCOCC CC(C(C)(C)C(=O)NC1C=CCCCC1)NC(=O)Cc1cc[nH]c1 N1(C(c2c(CNC(C)=O)nccc2)=O)CCN(Cc2c[nH]cc2C)CC1C1CC1 C(C)(N=c1nc2scnc2c(NCCN2CCC(C)C2)[nH]1)c1c(C)sc(Br)n1 Cc1n[nH]c(C)c1C(=O)NC1(CNC(=O)CCc2cnc(O)[nH]2)CCCC1 C=Cc1ccc(CC2=NOC(COC(=O)CCCc3nc(C)no3)C2)cc1 N1(C(C2C(C)C2C)=O)CCN(C(=O)CN(C)C2CC2)C(C(F)F)C1 C1(NC(C2C(C=C)CC2)=O)CN(C(=O)C(=O)NCCNC(C)=O)CCCC1 N1(C(c2c(C(C)NC(CCCC)=O)noc2)=O)CCC12CCN(C)C2 c1(C(=O)NCC2(NC(C3C(C)CCCC3)=O)CCC2)cccc2c1COCCN2 C1(NC(C2(SC)CC2)=O)CN(C(c2noc3cccc(C)c23)=O)C2CCCCC12 Cc1cnc(C=CC(=O)NC(C)(C)CN(C)C(c2ncccc2C(F)(F)F)=O)[nH]1 C1(NC(CC2CCCN(C(CC3N(C)C(=O)CC3)=O)C2)=O)CCCCC1(C)C C(C)(C)(CCCCNC(=O)CC(C)O)NC(c1c(CC)cno1)=O N1(C(C(C)n2cncn2)=O)CCCC(CCNC(=O)CCc2ccc(F)nc2)C1 N1(C(c2cncs2)=O)CC2CCC1CN2C(c1ccc(-c2ccncc2)o1)=O C12(CNC(CCCC)=O)CC1CN(C(=O)CCOC1CCCOC1)C2 C(=O)(C(CNC(=O)C(C)CC)C(C)(C)C)NCc1cnc(COC)[nH]1 CCCC(CCN=c1nc(N2CCC3(CCCO3)C2)c2c([nH]1)COC2)=C C(=O)(Nn1nnc2c1CCCC2)C1(C=C)CCN(C(=O)CCC2CC2(F)F)C1 c1(OCC)ccc(S(=O)(=O)N2CC3CCC(C2)N3C(=O)C(C)CN)cc1 N1(C(C(C)N=[N+]=[N-])=O)CCCC(N(C)C(c2coc(Br)n2)=O)CC1 CC1Cc2cc(C(=O)N(C)CC3CCN(C(=O)CCC4CC4)CC3)ccc2O1 C(=O)(C1=Cc2ccccc2C1)N1C(C)CCN(C(C(C=CC)O)=O)CC1 C1(F)(C(=O)OC)CC(N=C2C=CC(c3ccc(C(F)(F)F)cc3)=NNN2)C1 C1(C(C)C)CCCCCN1S(=O)(=O)Cc1c[nH]nc1Cc1ccccc1 CCC(COC)C(=O)NCC(CC)NC(c1cnn(C)c1-n1cnnc1)=O c1(C(N2CCC(NC(CCC=C)=O)C2c2ccccc2)=O)cnc2ccnn2c1 N1(C(c2c(C)cc[nH]2)=O)CCC(C(=O)NC(c2ccnn2C)C)C12CCC2 C1(NC(C2CCN(Cc3ccccc3)C2=O)=O)(CO)COc2ccccc2C1 c1(C(=O)NC2CCCC(NC(CCC(C)OC)=O)C2)cccc2c1NC(=O)CO2 C(=O)(C(N)C(C)(C)N(C(c1ccco1)CSC)CC)OCC C(=O)(C1=C(Cl)CCC1)N1C(C(C)(C)NC(=O)Cc2ccsc2)CCC1 N1(C(c2cc(C)c(O)cc2)=O)CC(NC(C2(C3CC3)CCCO2)=O)CC(C)(C)C1 N1(C(c2cc(OC)no2)=O)CC2(CCC2)CC1CNC(C1CCC(=O)N1)=O N1(C(CCc2c(C(=O)NCCOC)c(C)[nH]c2)=O)CC(CO)C2(CC2)C1 C1(NC(C2CC(OC)C2)=O)CC2(C1)CN(C(=O)C=C1CCCCC1(C)C)C2 c1(C(N(C2CCN(Cc3nc(C4CC4)cs3)C2)CC)=O)[nH]nnc1C CCCCCCCCCC(=O)NCC(C(C)C)NC(=O)CCCCNC(C)=O C(CN=c1ncc(Cl)c[nH]1)(C1CC1)OC(c1ncc(OCC)nc1)=O CC1=CCC(C)(C(=O)NC(CCN(C(=O)C2=CCCC2)C)C(C)C)CC1 c1(C(=O)NC2CCN(C(=O)COC3COC3)C(C3CC3)C2)nc2cnccc2s1 c1(C(N2CCN(C(c3ccc(C#C)cn3)=O)CC2C)=O)cc2nc(=O)ccn2[nH]1 c1(C(=O)NC(CNC(CC(CSC)O)=O)C(C)C)cccc(P(C)(C)=O)c1 C(=O)(C1=CC2(CN(C(=O)C(C)(C)N=[N+]=[N-])C2)OC1)N1CCC(C)C1C C12(C(=O)NC34CC(NC(c5nc(C(C)C)oc5)=O)(C3)C4)CCCCC1C2 C1(c2ccccc2)(NC(C2C(CC)CC2)=O)CCN(C(C2CCCOC2)=O)C1 C1(C)(NC(C(CCC)NC(C2CC(CC)C2)=O)=O)CC(C)(C)OC1=O c1(C(N2CCN(CC(C)(C)NC(=O)CO)CC2)=O)c(Cl)nc2cc(Cl)ccn12 c1(CC(C(N2C(CC(CC)(C)O)CC2)=O)C)ccccc1 CC1CCC(C(=O)NCC#CCCC#N)N1C(c1ccc(CC#N)cc1)=O c1(C(N(CCN(C(C)C)C(C2CC(C)CO2)=O)C)=O)cnn(CC(C)C)c1 N1(C(C)CC(=O)NCC2CC2CNC(=O)CCc2nncs2)CCc2ccccc21 N1(C(c2sc(C)c(O)n2)=O)CCN(C(C2(F)CC2)=O)CC(CO)C1 c1(C(=O)NC(C(C)NC(CC2(NC(C)=O)CC2)=O)C)ccc(CF)cc1 C1(C(=O)NC2CC2C(C)O)COC(C)C(=O)N1.C=C1C(C(=O)O)C1C(=O)OC N1(C(C2CN(CCC)C(=O)C2)=O)C2CCC1C(CNC(=O)CC(C)(C)C)C2 C1(NC(c2c(C)nc(C)[nH]2)=O)CCN(C(c2ncsc2C(C)C)=O)CC1(C)C C1(CNC(COCCC)=O)CC2(CCC2)CN1C(=O)CCCc1cc(C)sc1C C1(C(=O)NCCOCCN(C)C(C2CCCOCC2)=O)CCC(=O)N(C2CC2)C1 C12(NC(CCc3ccc(OC)cc3)=O)CCCC1N(C(c1[nH]nnc1C)=O)CC2 C(C(O)(CO)CO)NC(N1CCOCC1C(c1ccccc1)C1CCOC1)=O C1(C(=O)NC2C(CNC(c3ccncc3)=O)C2)CCn2c(O)nnc2C1 C(=O)(C1=NN(C)C(=O)CC1)NCCC(C)N(C(c1cc(C)c(O)nc1)=O)C n1(C(C)C)cnnc1CC(=O)NC(C)CC1CN(C(=O)CC2(C#N)CCC2)C1 N1(C(C(=O)N(C)C)=O)CCC(C)(NC(C2CC(CF)C2)=O)C1 c1(C2(N)CC2)cccc(NC(C2CCCCC2c2cccc(F)c2)=O)c1 C1(CC(=O)NCCN(C(c2c(COCC)cc[nH]2)=O)C)CCCCN1C(C)=O c1(C(N2C(CNC(c3cc4ccncc4[nH]3)=O)CCC2)=O)c(O)cc(O)cc1O N1(C(C(CCSC)O)=O)CCC(CNC(=O)Cc2cnoc2)C(C)C1 C1(C(=O)NC2C(C(=O)OC)C2)CCCC1C(=O)NCc1c[nH]c(=O)s1 c1(CNC2CC(C(=O)NCc3c(C)cccc3O)C2)ccc(F)c(S(C)(=O)=O)c1 c1(CC(O)CNN2CCCC(N3CCCCC3)C2)cccc(Cl)c1 CCCCCC(CC)C(=O)N(C)CC=CC(=O)NOCCCOC C#CCC(C)C(=O)NCc1cn(CCNC2(C3CCCC=C3Br)CC2)nn1 c1(OC(C(=O)NCC(CC)NC(C2CN(CC3CCC3)C2)=O)C)cccc(F)c1 C#CCC(C)(CC)C(=O)NCC1CCC2(CN(C(c3cccc(=O)o3)=O)C2)O1 CC(F)(F)CC(=O)NC(C)(C)CN1CCN(C(c2ccc(OCF)cc2)=O)CC1 c1(CC)c(C(N2CCC(N(C)C(C3CCCC3C(C)C)=O)C2)=O)ccn1C c1(C(N2C(CNC(c3c(N)c(Cl)ncc3)=O)CCC2)=O)noc2cc(F)ccc12 c1(C(=O)NC2CN(C(c3cc(C(C)C)[nH]n3)=O)CC2(C)C)cc(O)cc(C#N)c1 C1(C2CC2(F)F)(CNC(C2C(CNC(=O)OC)CCCC2)=O)CC1 N1(C(CC(C)N(C(C2CCN(CC)CC2)=O)C)=O)CCOC2C(O)CC12 C(=O)(C(C#N)C(C)(C)C)NCC(C(N1C(CC)CNC(=O)C1)=O)OC c1(OC(C)C(F)(F)F)ccccc1Cl.C1(C)(C)C(N)CN1 c1(OC)cc(C(=O)N(C)CC2(O)CCN(C(C3(NC(N)=O)CC3)=O)C2)ccc1F C12(C(=O)NCC3N(C(c4c(C)cc(C)o4)=O)CCC3)CCC(CC1)C2(C)C c1(NCc2c(-c3cc(C)c(F)nc3)ccc3c2OCO3)c(F)cc(C#N)cc1Br CC1CCN(C(C2CCCCC2)=O)C1CNC(c1ccc(NC=O)cc1)=O N1(CC(=O)N(C2CCCN(C(c3cnnn3C3CC3)=O)C2)C)CCCCCC1 N(C1CCCc2cc(C#N)ccc21)CCN1c2ccc(C)cc2SCCC1.C(CO)O c1(N(CC(C)NC(=O)CC2CCCCCC2)C2CC2)ccc(C#N)nc1 CC12CN(C(=O)C(c3ccc(F)cc3F)(F)F)CC1(C)CN(C(C1CC1F)=O)C2 N1(C(CCC(C)C)=O)CCC(F)(F)C(C(=O)Nc2cc(F)c(Br)c(F)c2)C1 c1(C(N2CCCC(C(N)=O)CC2)C(=O)NCC2CC2)ccc(F)c(Br)n1.C1(C)CC1 N1(C(C(C=C=C)C)=O)CCOCC(C)(CNC(c2cn(C3CCOC3)cn2)=O)C1 C1(C(N(CCN(C)C(c2cc([N+](=O)[O-])c[nH]2)=O)C)=O)COc2cc(O)ccc2C1 C(=O)(C(C)S(N)(=O)=O)NC1CN(C(c2ccc(SC)o2)=O)CC1C.c1ccccc1 C1(CC(C)NC(C(F)OC)=O)CC2CCC(C1)N2C(=O)CC(C)n1ccc(C)n1 C(=O)(CCCCCCCCCO)N1CCN(C(C2CCC(C)(C)O2)=O)CC(O)C1 C=C=CC(C)C(=O)NCCC1COCCN1C(=O)CNC(C1CCCCC1)=O C(=O)(C1=CC2CCC=CCCC12)NC1(C)CC(NC(c2cccc(C)c2F)=O)C1 CC(CS(C)(=O)=O)C(=O)NCC1(C)CN(C(=O)CCc2cn(C)nn2)C(C)(C)C1 N1(C(CC2N(C(C(CC)C)=O)CCOC2)=O)CCC(C)(N(C)C)CC1 C1(C(=O)NCC(C)OCc2ccccc2)CCN(C(=O)CC2CCOC2)CC1 C(C1CCCN1C(=O)COC1CCOCC1)=CC(=O)N(C1C(C(C)C)C1)C1CC1 c1(CC)cnc(Cl)[nH]c1=NCCCNC(=O)C1=CS(=O)(=O)CCC1 C12(C(=O)NC(CC)CS(C)(=O)=O)C3C4C1C1C2C3C41C(=O)NC CC1CCC(NC(=O)C=Cc2cccs2)CN1c1cc(=O)n(C)cn1 C(CC1CCC1)(C(=O)N=c1ccn(CC2CC2)[nH]1)NC(C1CC(C)(CC)C1)=O N1(C(C2(CC)CC2)=O)CCOC2(CCCN(C(C3(C#N)CCN(C)CC3)=O)C2)C1 C1(NC(COCCSC)=O)CCN(C(=O)Cc2cc[nH]n2)C1C(C)C c1(C(=O)NC(C(C(=O)NCCOCC(C)C)C)C)cc(C#N)n(C)n1 c1(C(N2CCC(C)(NC(CSCCCC)=O)CC2)=O)cnc2c(cnn2C)c1 Cc1ccccc1C(C)C(=O)NCC1(C(C)NC(c2cncs2)=O)CC1 CC1(CNC(=O)CSCC(N)=O)CCCN(C(C2CC3C=CC2CC3)=O)C1 CC(C)CC(C)CC(=O)NCCN(C(c1nc2cccnc2s1)=O)C(C)C c1(COC)n[nH]c(=NC2CC(F)(CNC(c3[nH]nc4ncnc(O)c34)=O)C2)s1 N1(C(C=Cc2n(C)ccc2)=O)CC(NC(c2cn(CC3CC3)nn2)=O)C2(CC2)C1 c1(C(=O)NCCN(C(=O)CC2CCC(=O)NC2)CCC)ccc(Cl)c(C)c1 N1(C(COCCC(C)C)=O)CC2C(CC(=O)N(c3cccs3)CC3CC3)C2C1 N1(CC(N2C(C)C(NC(=O)CCc3cc[nH]n3)CC2)=O)CCn2nccc21 n1(CC)nc(C)cc1C(=O)NC1CCC(NC(=O)CC2CCCC2O)C1 C(c1cncc(C)c1)=CC(=O)NCC1C(NC(c2nc(CC)sc2)=O)CC1 c1(OC)ccc(S(=O)(=O)N2CC3CN(C(c4c(C)cccc4C)=O)CC23)c(F)c1 C(C)(CCCCNC(=O)CCCn1ccnc1C)NC(C(C)=C1CCCC1)=O N1(C(CCC2CC(NC(C=CCN(CC)CC)=O)C2)=O)CCCC(CCO)CC1 C1(NC(C2CCC=CO2)=O)CCN(C(c2cc3ccncc3[nH]2)=O)C12CCC2 N1(C(C2C(CC)CC2)=O)CC(NC(c2c(C)cnn2C(C)C)=O)CC12CCOC2 N1(C(C2C(OC)CCCC2)=O)CCC(C)N(C(c2ncc(F)cn2)=O)CC1 c1(C(=O)NCC2OCCN(C(C(CSC)C)=O)C2)cncn(C)c1=O N1(C(C(CC)c2ccccc2)=O)CCSCC1CCNC(=O)CCN(C)CCC C12(C(=O)NCC3OCCN(CC)C3)CC(CCO1)N(C(C1CC1(C)C(F)F)=O)C2 CC(C(=O)NC1CC1NC(C1CN(C2CCCC2)C1)=O)NS(C)(=O)=O N1(C(CC(Cc2ccccc2)SC)=O)CCC(O)C(C2CCCC2)C1 c1(C(C(=O)NC(=O)CS(=O)(=O)N2CCCC2)OC)cc(Cl)cc(Cl)c1 CCCC(C(=O)OC)C(=O)N1CCC(CCC(=O)NCc2cc(C)sc2C)CC1 N1(C(COCc2cc(C)on2)=O)CCCC(NC(=O)CC(O)C(C)C)CC1 C1(NC(=O)CCCC2CCCCC2)(CO)CCCN(C(c2ccncn2)=O)C1 c1(C(=O)NC2CCC(F)(CNC(CCCNC(C)=O)=O)C2)cnc2sccc2c1 N1(C(CC2CCC(C)C2)=O)CCC(O)(CNC(=O)COc2cncc(Cl)n2)CC1 CCC(CCOC)C(=O)N1CCC(NCc2ccnc(Cl)c2F)C(C)C1 N1(C(C2CC3CCC3C2)C(=O)NCCCC)CCCNC(=O)C(F)(F)C1 N1(C(C(c2cn(C)nc2)=O)=O)C2CCC(C(=O)NOCc3cc(O)no3)C1CC2 CN(C)S(C)(=O)=Nc1nc(C(N2CCC(NC(C3CC3F)=O)C23CCC3)=O)cs1 c1(OC)ccc(F)c(C(=O)OC(C(N2CC3N(C(C)=O)C3C2)=O)=O)c1F C1(CC(=O)NCC(CCOC)NC(c2noc(C3CC3)n2)=O)CCC(C)CO1 Cc1cccc(O)c1C(=O)N(C1CCN(C(=O)CSS(C)(=O)=O)C1)C C#Cc1cnc(C(N2CCC(C(=O)N(C)Cc3nncs3)CC2)=O)c(C)c1 N1(C(c2cc(COC)[nH]n2)=O)CCC(C)(C(=O)NCC2CNC(=O)CO2)C1 c1(C(C)OC)ccc(C(=O)NCC23CC(CO)(CN2)C3)cc1 N1(C(C(CC)C)=O)CCOC2CN(C(C3(C#N)CCC3)=O)CC12 N#Cc1cccc(CNC(C2(O)CCN(C(c3cccc(CO)c3)=O)C2)=O)c1 C1(N(CC=C)C(C2CCNCC2)=O)CC(=O)N(C(=O)Cc2ccccc2)C1 N1(C(c2cccc(C)c2F)=O)CCC2(CC1)CCN(c1ncnn3cccc13)C2 c1(C(=O)NC(c2ccccc2)C#N)c(Cl)oc2ccccc12 CCCCCCn1nnnc1CNC(C)(CCCO)c1nnnn1C1(C)CC1 c1(C(=O)NCC2C(NC(c3c(C(C)C)onc3)=O)COC2)nnn2c1CSCC2 C1CC2(CCC2)CO1.N1(C(C)COC)CCOCC1.C12C(C1(C)C)NC2=O C#Cc1cccc(C(=O)NC2CCC(C(=O)N(c3nc(C)cs3)C)C2)c1 CCCC(CC(C)C)C(=O)NCCC1COCCN1C(c1cc(O)n(CC)n1)=O N1(C(CN(C)CC)=O)CC(NC(=O)COc2cc(C)ccc2C)CC(O)C1 n1(CC(=O)NCCCNC(C2CCCC(C)CC2)=O)cc(S(C)(=O)=O)cn1 C1(C(=O)NC(CC)CC)CC12CCN(C(C1CCC(N)C1)=O)CC2 CC1=C(C)CC(C)(C(=O)NC2CN(C(C34CCN(CC3)CC4)=O)CC2F)CC1 c1(OC)ccc(Cl)cc1C=CC(=O)NC1CCOC(CC(C)C)C1 N1(C(C2(C)ON=C(C)C2)=O)CCCC(C2(NC(C34CC3C4)=O)CC2)C1 C(=O)(C#CC1CCCCC1)N1C(C(C)NC(c2cc(CN(C)C)on2)=O)CCC1 S(=O)(=O)(c1ccc(CN=C(NCC2CC2)NCC2(C)CCS(=N)(=O)CC2)cc1)NC C1(C)(CC)CCC(C(=O)NCC2CN(C(=O)C=C3CCCC3)CC2C)O1 c1(C(=O)NCC23C(CN(C(c4c(C)nsc4C)=O)C2)C3)ccc(C(C)C)cc1F N1(C(C(C)NC(=O)NC)=O)CCC(N2CCC(NC(=O)CSC(F)F)CC2)CC1 c1(NC(C(CC=C)CNC(=O)C(C(C)C)SC)=O)cccc(N=[N+]=[N-])c1 NS(=O)(=O)c1ccc(C(CF)NC(=O)NC23CCC(CC2CO)C3)cc1 c1(CC)cc(F)c(C(=O)NC(C2CCCN2C(C2(Cl)CC2)=O)C)c(F)c1 N1(C(C2C(C=C)C2)=O)CCCN(C(=O)CCc2cnccn2)C(C(C)C)C1 c1(SC)nc(C)cc(=NC2CC(F)(CNC(=O)CSc3cccs3)C2)[nH]1 C#CCCCCC(=O)NC1CN(C(c2cn(C)c(C(F)F)n2)=O)CC1OC CC(C)C1=NOC(C)(C(=O)NC(C)CCCCNC(=O)Cc2nc(=N)[nH][nH]2)C1 CC1CCc2c(C(N3CC(F)(C(=O)Nc4cc(F)c(Cl)cn4)C3)=O)n[nH]c21 c1(CCC(N2C(C(=O)OCC)CC(CC)CC2)=O)cccc([N+](=O)[O-])c1Cl N(C(=NCCc1ccc(Cl)cc1Cl)NCCN(C)C)C1CC(C)SC1 CS(=O)(=O)c1cnc[nH]1.c1(N2C3CCN(CC3)CCCCC2=O)c(F)cccc1F N1(C(c2nc(C)[nH]n2)=O)CCCC(C)C1CNC(=O)CC1CCC(C2CC2)O1 C1(NC(CC)=O)CCN(C(=O)CCN(C(=O)C(C)c2ccsc2)C)C1 N1(C(C(C)OCCC=C)=O)CCCCC(N(C(=O)C(C)(C)c2cc[nH]n2)CC)C1 C=CC1CCCC(NC(=O)C(Cc2cc[nH]n2)NC(=O)C(C)C#N)C1 C1(CNC(C2N(C(CCC)=O)CSC2)=O)CCCN(CCc2cccc(C)n2)C1C C#Cc1cc(CNC(=O)Nc2ccc(C(=O)OC(C)(C)C)c(C)n2)cc(F)c1 N1(C(COCCOCC)=O)CCOC2(C1)CN(C(c1cccc(C=O)c1)=O)C2.C(C)=O N1(C(c2ncc(C)cc2F)=O)CCCC2C1CCN2C(=O)CCc1cnn(C)n1 N1(C(C(c2ccc(OC)cc2)O)=O)CC2CN(Cc3cccc(Cl)c3F)CC12 CCCC(CC)C(=O)NCCCCC(=O)NCC(C)(C)CC(F)F CC1(C)C=C(C(=O)N2CCC(O)(CCNC(c3csc(C(F)(F)F)c3)=O)C2)C1 C(=O)(C1CCCc2nccn21)N(CC(CC)NC(=O)C1=CCCCO1)C N1(C(C(C)NC(C)(C)C)=O)CCCC(NC(c2csc(-c3ccco3)n2)=O)CC1 C=CCC(CC=C)C(=O)N1CCC(NC(C2(C3CC3)CCOCC2)=O)C(F)C1 Cn1c([N+](=O)[O-])cnc1C(=O)NC1CCCC1CNC(C1CCC(F)(F)CC1)=O C(=O)(CCS(C)(=O)=O)N1CC(=O)NC2CC(C2)C1.CCSSC C1(NC(Cc2c(C)nc[nH]2)=O)CN(C(C2CCCCN2C)=O)CC1F C(=O)(C(F)CCC(C)C)NC1(C(=O)NC(C=C)(C)CC)CCCC1 C(=O)(C(C(=O)NCC(F)CNC(=O)C(C)=CC1CC1)C(C)C)OCC C1(NC(c2ccc(OC)cn2)=O)CC2CN(c3nnc(C4CC4)s3)CCN2C1=O c1(C(N2CC(C(N3CCC(C(=O)OC)C3)=O)C(F)C2)=O)ccc2nc(Cl)sc2c1 c1(C(=O)NC(C)CNC(COCC)=O)cc(C(=O)NC23CC(C2)C3)cc(CC)c1 N1(C(C2=CCC(NC(C(C(C)(C)C)N(C)C)=O)C2)=O)CC2(CCOCC2)C1 Cc1ncc(NC(=O)CC2CCN(Cc3ccncc3)C2)cc1Cl c1(COCC)cn(CC(O)CNC(=O)C(c2ccccc2)O)nn1 C=CCCCCCCC(=O)N1CCC(NC(=O)CS(=O)C(F)(F)F)C1(C)C C(=O)(CCCCCNC(c1nc[nH]n1)=O)NC1C(CC)CCC1 c1(NC)c(C(=O)N(C)C(C2CC2F)=O)sc2nccnc12.C1(CO)CC1 c1(C2CC(C(=O)NC(CC)CNC(C3(CF)CC3)=O)C2)ccc(O)cc1 C1(C(C)NC(C2C=CCCC2)=O)CN(C(=O)CC(C)(C)C2CC2)CCO1 N1(C(c2ccccc2)=O)C2CC1CN(C(=O)COc1noc(CC)c1C)C2 c1(C(N(C(C)(C)C)CC2CN3CCCCC3CO2)=O)cc(C#N)c(N)cc1O CN1C(C(=O)NC(CNC(c2cnn(CCO)c2)=O)C(C)(C)C)CCS1(=O)=O C12(O)CCN(C1)C(=O)C1(CC1)C2.C=CC(O)C(=O)N1CCC(OCCN(C)C)C1 N1(C(c2nc(COC)oc2)=O)CCC(CN(C)C(C2CCC(F)C2)=O)CC1 c1(C(=O)OC)cc(NC(=O)CSCC(=O)NC2CCC(=O)CC2)ccc1O C12(C(=O)NCC(C)OCC=C)CCC(NC(=O)CSCC(=O)OC)(CC1)CO2 C1(C(N2CCC(C)(C(N(C3CCCC3)CCCC)=O)C2)=O)CC(C2CC2)=NO1 CC(C)C(C)C(C)CC(=O)N1CCC(CCNC(=O)CCn2cccnc2=O)C1 Cc1nn(C)cc1CC(N1CC(N2CC(NC(=O)C3CC3)CC2=O)C1)=O c1(CC(C)N(C)C)cn(C(C)CNC(c2coc(C(F)F)n2)=O)nn1 CS(=O)C=CC(=O)NC1C2CN(C(c3c[nH]nc3-c3ccco3)=O)CC12 c1(C(N(CCC(=O)NC)C)=O)coc2c1CN(C(=O)CSC1CC1)C2 C1(C(=O)NCCN(CC(C)O)C(C2CC(F)(F)C2(C)C)=O)CC2C(C1)C2(C)C Cc1nnsc1C(C)NC(=O)C=CC(C)NC(=O)C(c1cnn(C)c1)=O CCC(C)C(C(=O)NC(c1ccc(F)cc1)C(N)=O)c1ccccc1 c1(OC)cc(Cl)ccc1C(C)NC(c1ccc(C)c(Br)c1)C N1(C(N)=O)CCCCC1.C(CCC(=O)NCC1CC(NC(C23CCC2C3)=O)C1)N(C)C N1(C(c2cn(CC)nc2)=O)C(C(=O)NC2(CC(C)C)CC2)CC2CC12 c1(C(N(C2CCN(C(=O)CC(C)OC)C2)CC)=O)scnc1Cl Cc1cc(C(=O)NCC2CCN(C(=O)Cc3cncs3)C2)ncc1CO c1(C(=O)NC(C2CC(NC(=O)CCNC(C3CCC3)=O)C2)C)cnco1 N1(C(CCC=CC(C)C)=O)C2CCC1CN(C(=O)CC13CCCC1C3)CC2 C(CCC(C)(C)C(=O)NCC1CCC(C(=O)NC(c2ccccc2C)C)C1)OC N1(C(Cc2n(C)ccn2)=O)CCN(C(c2cc[nH]c(=N)c2)=O)C(c2ncc[nH]2)C1 c1(OC)ccc(Br)c(S(=O)(=O)NC(=O)NC2CCN(C(C)C)CC2)c1Br C1(NC(C2OCC(C)(C)C2)c2ccccn2)CC2(CCCNC2)C1 C(=O)(C1=NOC2(CCC2)C1)NCC(CNC(C(c1ccc(CC)cc1)C)=O)OC CC1=NN(C)C(=O)C1CC(=O)NCC1(F)CC(NC(=O)CC2(C)CCCCC2)C1 C1(NC(C(C(=O)OC)OC)=O)CC2CC1CC2C(N1CC(N2CC(F)C2)C1)=O N1(C(c2nccc(OC)c2)=O)CC(C(=O)N(CC(C)CN(C)C)C)C(F)(F)C1 C1(C(=O)NCCn2cc(COC)nn2)OCCCC1(C)C.C12(CC1)CC(=O)NC2 CC(C(=O)NC(C)CC1CCN(C(=O)CCC2CCOC2)CC1)S(N)(=O)=O C1(CC(=O)NC2CN(CC#C)C(=O)CC2)CCC2(CCCC2)O1 c1(C(=O)OCC)oc2ccccc2c1C.c12ccsc1C(=O)O2 C1(NC(Cn2cnc(C(N)=O)n2)=O)COC2(CCCN(C(c3csc(S)n3)=O)C2)C1 c1(C(=O)NCC(N(C)C(C2CCOCC2)=O)C2CC2)ccc2nccnc2c1 c1(CNC(C=C(CCC)C)=O)cc(C(=O)N(C2CCC2C)C)co1 N1(C(CCNC(=O)OCC)=O)CC2OC(=O)N(C3CCOCC3)C2C1 N1(C(CCSCCCC)=O)CC(N(C(=O)CCOCCOC)C)C(O)C1 CCCC(C)CCCC(=O)N1CC(NC(c2cnc3cc(C)ccn23)=O)C(C)C1 c1(NC(C(CCC)CNC(c2ccc(CO)cn2)=O)=O)ccn2nccc2c1 C1(NC(c2c(C)nc(COC)s2)=O)CC2CN(C(c3ccc(C(F)F)s3)=O)CC12 CCCS(=O)(=O)CC(=O)NC(C)(CNC(c1csc(O)n1)=O)CC(C)C Cc1nc2c(s1)CCCC2C(=O)NC1CCC(NC(C2CC(O)CN2C)=O)CC1 C1(C(N2CCC(NC(C3(CO)CCOC3)=O)C2)=O)CCC2(CC2)CO1 C(=O)(CC(CN(C)C)CC)NCCSCC(=O)NCC1(C#C)CCCC1 C1(CC(=O)NC(C)C2CC2)CCCN(C(C2(F)CC=CCC2)=O)CC1 CC(C)CC(CNC(c1cn(Cc2cccnc2)nn1)=O)NC(C1C(C)C1C)=O C(C(=O)NCCC1CC1)(C1=NOC2CCCCC12)N(C)Cc1cccc(Cl)c1 C1(C(=O)NC2(CNC(CCc3c[nH]c(=N)[nH]3)=O)CCC2)CN2CCN1CC2 N1(C(CC=CC)=O)CC(CNC(C2(OC)CC2)=O)(OC)C1 c1(C(N2CC(C(N3CC=CCC3)C(=O)OC)C2)=O)ccc(F)c(C2CC2)c1 C1(C(=O)NCC(CC)N(C(COCCOC)=O)C)CC12CCOCC2 N1(C(=O)N2CCC(C(C3C4CCC(F)(F)C34)=O)O2)CC2CC(O)CC2C1 N(C(=NCc1ccc(OCC)c(F)c1)N1CCC(C(=O)OC)(C(C)C)C1)CCC C1(COC)CCN(C(=O)C=CCCCSC)C1.C12(CCC1)C(=O)N2 c1(-c2cn(NC(C(C(C)NC)CO)=O)nn2)ccc2c(c1)OCO2 C1(NC(=O)CC2CCOC2)CC2CC(C1)N(C(c1cc3ccsc3[nH]1)=O)C2 c1(N2CCCCC(NC(=O)CCn3cccn3)C2)ncnc2c1nnn2C1CC1 c1(C(=O)NCC23CCCN(C(C=CC)=O)C2CCC3)cc(C)c2nc(C)cn2n1 C=CC(CC)CC(=O)N(C)CC1CCN(C(c2cnc(O)cc2C(F)(F)F)=O)C1 c1(C(=O)OC)ccc(CNC(C)(C)C(C)NC(=O)Cc2cccn2C)o1 CC(CCCCNC(=O)C=Cc1cc[nH]n1)NC(=O)CC1(n2ccnc2)CC1 c1(CC(N2CCC(CCNC(CN(CCC)C)=O)CC2)=O)csc2nccn12 C1(C)(C(=O)NCC23C(CN(C(c4n(C(C)C)ccn4)=O)C2)C3)CCCNS1(=O)=O c1(CC(=O)N(CCN(C(=O)CC2COC(C)(C)C2)C)C)cc(F)ccc1Cl C1(C(=O)NCC2ON=C(C(C)C)C2)CCC2(CCN(C(=O)CN3CC=CC3)C2)C1 c1(C(N2CCC(NC(C(C)OCCC=C)=O)C2C)=O)cn2ccncc2n1 c1(C(N2CCC(CNC(c3c(CC)[nH]nc3Cl)=O)C2)=O)ccc(F)c2occc12 C(=O)(CC(C=C)CC)N1CCC(CC=C)(C(=O)NCc2nccnc2CC)C1 C(=O)(CCCCCCCBr)NC(C1C2CN(C(C)=O)CC1CC2)c1ccccc1 CCC(CNC(C1CC(C)CN(C(c2scnc2C)=O)C1)=O)(CC)CO CCCC(F)C(=O)NC1CN(C(=O)C(CO)N(C)C)CC1C(F)F c1(OC)cc(N)c(C(=O)NCCCCNC(=O)CC2CCC3CC23)c(F)c1 Cc1cccc2c(C(N3CCC(NC(=O)C=C4CCC4)C(C)C3)=O)nccc12 CCCCCCCCC(=O)NCC1CC(NC(c2ccc(C(F)(F)F)nn2)=O)C1 C(=O)(C(O)P(C)(C)=O)N1C(C(C)(C)C(=O)N2CC(N3CC(=O)NC3=O)C2)CCC1 C1(CNC(c2ccc(C)cc2)=O)CCC(C)CN1C(c1ccc(Cl)c(C)c1)=O N1(C(C2CC(NC(C(c3ccn(C)c3)C)=O)C23CCC3)=O)Cc2c[nH]nc2C(C)C1 C1(O)(CNC(=O)NC2CN(CC3CCCO3)C2)CCCC(C(F)(F)F)C1 CCC(C)(CCC(C)C)C(=O)N1CCC2CN(C(=O)C(N)=O)CC12 C1(NC(=O)Nc2ccnc(N3CCOCC3)n2)CNCC2(CCC2)C1 C1(NC(Cc2c(CC)noc2CC)=O)CN(C(c2cccc(Cl)c2Cl)=O)CCC1O N1(C(C2N(C(c3c(C)ncc(C)n3)=O)CC3(CC3)C2)=O)CCc2ccsc2C1 C1(C2CCN(C(=O)CSCC#N)CC2)(NC(C)=O)CC1.C12CC3CCC(C1)N23 Cc1nnc2ccc(C(=O)NCc3cnsn3)cc2c1C C(=O)(C#CC(C)(C)C)N1CC(CNc2nc(C3N(C)C(=O)OC3)sc2)OCC1 C(=O)(C#CC1CCOC1)N1CCC(N(C(=O)COCc2ccccc2)C)C1 c1(OC)cc(NC(C2CSCCN2C(C2CC2C)=O)=O)cc(C)n1 C(=O)(CC(C=C)CCC)N(C1CCCC1)CCCNC(COCC#C)=O c1(C(C)NC(N(C2CSC2)C(C)C)=O)ccc(Cl)c([N+](=O)[O-])c1 N1(C(c2[nH]cc(C)c2)=O)CCC(O)(CCNC(c2cn(CCF)nn2)=O)C1 C1(CNC(CC(C)c2ccccc2)=O)CCCCC1NC(C1CN(C)CCO1)=O c1(CC(=O)NC2(CO)CN(c3ncc(I)cn3)C2)sc(O)nc1O c1(C(=O)NCC2CN(C(C3(F)C(C)OCC3)=O)C2)cc2c(=O)[nH]ccn2c1 CCCCCC(O)C(=O)NC1CC(CNC(c2cc(Cl)c(OC)c(Cl)n2)=O)C1 c1(NC(C2N(Cc3ccc(OC)cc3O)CC(F)C2)=O)cc(C)c(OC)cc1C N1(C(c2n(CC=C)ccc2)=O)CCN(C(=O)CCC(C)(F)F)C2CC12 C=CCCC(F)(F)C(=O)NCCCN(C1CCCC1)C(C1CCCCC1C)=O C1(C(=O)NCC(CCOC)NC(c2ccns2)=O)CCC(=O)N1C(C)C Cn1cc(Cl)c(C(N2CCOC(CCCNC(c3ncccc3CO)=O)C2)=O)n1 CCC(C)(C)CCCC(=O)NC(C)(C)CCCC(=O)Nc1cnc(Cl)c(C)c1 Cc1ccc2c(C(=O)OCCSn3ccnc3C(C)(C)C)cnn2c1C Cc1cc(C(=O)N(C)CCOCCN(C)C(c2cocc2C)=O)ncc1Cl C1(NC(C2CCCN(C)C2)=O)CCN(C(c2[nH]nnc2C2CC2)=O)CC1CO N1(C(Cc2n(C)cnc2)=O)CCCC(n2cc(CCNC=O)nn2)CC1 C1(C(=O)NCCN(C(c2cncc(N(C)C)c2)=O)CC)COC(C)(C)CO1 S(=O)(=O)(c1cccc(Cl)c1Cl)Nc1cccc(-c2c(COC)cn(C)n2)c1 N1(C(C(C)C2CCC2)=O)CCC12CN(C(=O)CSc1nncs1)C2 c1(C(=O)NCC2CN(C(c3n(CC)cnn3)=O)CC2(C)C)ccc(Cl)c(F)c1F C=C(C)C1OCCC1C(=O)NCC1CC(F)(CNC(C2CC2C2CCC2)=O)C1 C1(C(=O)NC(C(C)(OC)CO)C)CN(C(=O)C2=NOCC2)CC2(CCC2)O1.C(C)(C)(C)O c1(C(N2CC(CN)C2)=O)cccc(Cl)c1Br.c1(CN(C)C=O)cccc(C2CC2)c1 c1(OC)ccc(C(C)CC(=O)NCC=CCNC(=O)CCSc2nnnn2C)cc1 C12(NC(c3cc(C)[nH]c3)=O)CCN(C(=O)CCCc3cccs3)CCC1C2 c1(C(C(=O)N(C)Cc2cn(CC3(COC)CCC3)nn2)(F)F)ccc(F)cc1C N1(C(c2nc(C(=O)OC)sc2)=O)CCC2(CC1)CC2CNC(=O)C(C)CC(C)C C12(C(=O)Oc3nc(-c4ccc(OC)cc4)sc3)CCCCC1OCC2 O=S1(=O)CC2(C(F)(F)F)CN(N3CCC(c4ncc(Br)cn4)C3)CC12 c1(C(=O)NC2C(CNC(c3c(C)n(C(C)C)nc3)=O)CCC2)ccc(=O)n(C)c1 C1(NC(CCCSC)=O)CC(C2CCN(C(C3CN4CCN3CC4C)=O)C2)C1 CCC(CN(C)C(n1cc(C2CCCN2C)nn1)Cc1ccc(C)cc1)C(=O)OC c1(C(=O)NCCCN(C(=O)CC2CCCCC2)C2CC2)cccc2c1NCC2 C(c1cncc(O)c1)=CC(=O)NC(C1CCN(C(C2CCC(F)CC2)=O)C1)C N1(C(c2cc(SC)ncc2)=O)CCOC2(C1)CN(C(c1cn(C)nc1C)=O)C2 C1(C(=O)NC2C=CC(C(=O)NC3CCN(C)CC3)C2)CC2(CC2)CN1C C(=O)(C(C)(C)NC(C1CCCOC1)=O)NCC(C1CC1)SC C(=O)(C1CCCc2nc[nH]c21)NC1(CNC(=O)CCn2cncn2)CC1 c1(OC)cc(CN(C)Cc2cccc(CN(C)C)c2C)c(Br)cn1 CC1(C)CCN1C(=O)C(Cc1ccoc1)NC(c1cc(C(N)=O)c[nH]1)=O N1(C(=O)COC(F)F)C2CCC1CC(NC(C1(Sc3ccccc3)CC1)=O)C2 C1(NC(C2CN(C)C(=O)CC2)=O)CN(C(=O)CC2CCCC2)C2CCCCC12 C#Cc1cncc(C(=O)NC(CCCC)C(=O)NC2(C)CCC(C)(C)C2)c1 Cc1ccc(CC(N2CC(O)(CNC(c3ccn(-c4ccccc4)n3)=O)C2)=O)s1 C1(NC(=O)Cn2nccn2)CN(C(=O)CCn2cncn2)CC1n1cccn1 c1(C(N(C)CCN(C)C(c2csc(C(C)(C)C)n2)=O)=O)cnc2cnccc2c1 c1(NC(c2cc(C(=O)O)no2)=O)cccc(OCCF)c1 Cc1nc2ccccc2c(=O)n1C.O=S(=O)(NC)N1C2CCCCC2C1 CC1(C(=O)NCc2cnc(Cl)s2)CN(C(C(C)(C)C)=O)CCO1 C=C(C)C(CC(=O)NC(C1CCCCO1)C(=O)N(C)CCOC)OCC c1(OC)cc(C(=O)NC2C3CN(C(c4nccc(C)c4N)=O)CC23)ccc1C C1(NC(=O)CC2(CO)CCCC2)CCCCCC1NC(=O)CC1CCCOC1 C(N=c1[nH]c(C2CC2)nc(=N)[nH]1)c1c(CNC(CCSC)=O)cccc1C C1(NC(C(C)(C)NC(=O)NCCC)=O)CCC12CN(C(c1cnc(S)nc1)=O)C2 c1(C(=O)NC2CCCCN(C(c3c(C)snc3)=O)C2)nnn2c1CSCC2 CCC(C)C(C(=O)N1CCC1C(C)C)N(C(=O)Cc1ccc2c(c1)CC2)C C1(C(=O)NC(C)CCC2CC2)N(C(=O)Cc2ccc(O)cn2)CC12CCCC2 C(CCC1C(=O)N(C)CC2(CC(=O)N1)CC2)OC.C(C(C)OC)SC c1(C(=O)NC2(CO)CN(c3nncs3)C2)ccc2cnccc2c1 c1(OC)ccc(C(=O)NCC2CCC(=O)N2C(C2CCN(C(C)=O)C2)=O)nc1Br C1(NC(C(C(C)C)CNC(C2(CF)CC(=O)C2)=O)=O)CC1C1CCCCC1 C1(CC)CN(C(c2ccc(F)c(C)c2)=O)CCN1C(c1cn(C)c(=O)nc1O)=O N1(C(c2c(CC)ncnc2)=O)CCCOC(CNC(=O)CCc2cncn2C)C1 N1(C(C=CC(C)C)=O)CCC2C(NC(=O)CCCCOc3ccc(Cl)cc3)CC12 N12CCN(CC1)CCc1nc(nn1C)C2.N1(C(=O)OC(C)(C)C)CCC2CC12 C1(N(C(=O)C(=O)NC2CCNC(=O)CC2)C)CCCC12CCNCC2 c1(C(=O)NCC2(NC(C(C)CC3CC3)=O)CCOC2)cc(F)c(N)c(F)c1 N1(C(c2nc(C)[nH]n2)=O)CCN(C(c2snc(O)c2Cl)=O)C2CCCCC12 c1(C(=O)NCC2CCN(C(C3(COC)CCCO3)=O)C2)cccc(Cl)c1 C1CC(C)N=C2C=CN=C(N2)N1.S(=O)(=O)(c1cn(C)cn1)N(CC)CC C1(CN2CCCC(C(=O)Nc3n(C)ncc3Br)C2)CCc2cc(Br)ccc2O1 N1(CC)CCC(c2nnnn2C(C)C)(NCCC2CC(C)(C)CO2)CC1C C1(C(=O)NC2(C)CN(C(c3c(CC)scc3)=O)C2)OCCOC12CCC2 c1(C(=O)NCC2OCC(C(=O)NC(CC)C(C)(F)F)C2)cc[nH]c(=NC)c1 c1(C(NNC(c2c(OS(=O)(=O)CBr)nc(C)s2)=O)=O)ccc2c(c1)CCC(=O)N2 Cc1nc(C(C)C)ccc1C(=O)NCCC(C)NC(=O)CC12CCCC1C2 C1(CNC(C2(N(C)C)CC2)=O)CC2CCC1N2c1ccnc(Cl)n1 C1(C(=O)NCC23CC(NC(C(C)(C)C)=O)(C2)C3)Cc2cccnc2C1 c1(C(N2C(C)(C(N3CCC3CO)=O)CCC2)=O)c(Cl)cccc1Cl Cc1cc(O)ccc1C(=O)NC1CC2CC1N(C(c1ocnc1C(C)C)=O)C2 N1(C(CN(C(=O)C(CC2CCCC2)OC)CCC)=O)CCOC(CC)C1.C(C(=O)OC)O N1(C2(NC(N3CC(C(C(=O)OCC)F)C3)=O)CC2)CCCC1=O C1(CC)CCCCCCN1C(=O)CC(=O)NCCSCC(F)(F)F N#CC1C2CCC1CN(C(C1CCOC1CNC(c1cc[nH]c1C1CC1)=O)=O)C2 C(=O)(C1=NOC2COCC12)NCC(C)(CNC(c1cc(C)ns1)=O)OC c1(C(N(C)CC2CCCN(C(C3N(CCC)CCC3)=O)C2)=O)cc2scnc2[nH]1 c1(C(=O)NCC(Cn2cc(C(CC)(C)C)nn2)(F)F)cc(Cl)n(C)n1 Clc1cc(-c2nnc(Cn3ccnn3)n2Cc2noc(CC3CC3)n2)ccc1Br C(C)(CCC(=O)NCC(C(C)(C)C)NC(C1(CC(C)C)CCC1)=O)SC O=C1CCC2(CN(C(C34CC(CN3C(C3OCCC3C(=O)O)=O)C4)=O)C2)O1 C(=O)(C#CC1CCOC1)NCC(C(C)C)(C)NC(=O)Cc1cc(C2CC2)on1 CC(C)S(=O)(=O)CC(=O)N1CCC(NC(C2CC2CF)=O)C(C)(C)C1 CC(C)CCCCCCNC(c1cc(CCNC(=O)C(C)(O)C(F)(F)F)on1)=O c1(C(N2CC(NC(c3ccc(OC)nn3)=O)C(F)CC2)=O)cn2ncccc2n1 CC1CN(C(=O)C(CCC2CC2)NC(c2ncccc2O)=O)CCC1O C1(NC(c2cnc(C)o2)=O)CC(O)CN(C(=O)Cn2ccc(=O)cc2C)C1 c1(CNC(C2CC(O)CN2C(=O)Nc2ccccc2)=O)ccc2occc2c1 N1(C(CCOCCCOC)=O)CC2CCCCC2(CNC(=O)C=CBr)C1 c1(CNC(C2C(NC(=O)OC(C)(C)C)CCCC2)=O)ccc(C(C)(C)C#N)cc1 C(C(=O)OC)(c1csnn1)N(CC(=O)NCC1CC1)CC=C C1(F)(CNC(CCC)=O)CCCN(C(=O)C=Cc2c(C)cc(C)cc2C)CC1 Cc1ncc(Br)cc1C(N1CC2(C(=O)NCCc3ccccn3)CC1CO2)=O C1(C(=O)NC(CC(=O)NC(C)C)C)CN(C(C2CC2(C)C(F)F)=O)CC1C C1(O)(CC(=O)NC2(C)CC(NC(=O)CCCn3ccc(C(F)F)n3)C2)CCOCC1 n1(CC(=O)NC2(C)CN(C(=O)CCC(N)=O)C2)ncc(O)nc1=O C1(C(N(CCCN(c2cc(COC)ncn2)C)C)=O)COc2ccc(F)cc2C1 C1(NC(CCC(=O)NCCC)=O)CCN(C(=O)CC2CC(CC)=NO2)C12CCC2 N1(C(C(C(C)C)OC)=O)CC2(C(=O)NC3(CO)CCOC3)CCC1CC2 c1(C(=O)NCC2CCC(NC(C=CSC)=O)C2)cncnc1C(C)C C1(S(N)(=O)=O)(C(=O)NC2CCN(C(C(C)OCc3scc(C)n3)=O)CC2)CCC1 CS(=O)(=O)C1CCCN(C(C2CCC(CO)CC2)C(=O)NCCC#N)C1 C(=O)(CC1=CCCCC1)NC(C(=O)N(CC(F)Cl)C)Cn1cccn1 C(=O)(C1=CC(C)(C)C1)NC1CCC(N(C)C(C2CC3(CCC3)CO2)=O)CC1 c1(NC(=O)CC2CCCN2C(C2C=CCS2)=O)ccc(F)cc1I C1(C(=O)NCC2CC(NC(c3cc(CC)sc3)=O)C2)CC2C=CC1O2 Cc1cc(NC(C2CC(C)CN2Cc2cnc(Br)s2)=O)cc(C)n1 C(=O)(C1CCCc2ccnn21)NC(C)(C)CNC(C1(c2ccc(Cl)nc2)CC1)=O Cc1cc(C(N2CCC(CC(=O)NCCC3CCN(C)C3)C2)=O)n[nH]1 C(=O)(C1CCN(C)c2ccccc21)N1CCC(=CC(=O)NCC(C)C)CC1 c1(C(N2CCCC(CC)(NC(c3ccc(C)nc3)=O)C2)=O)ccc(C#N)c(O)c1 c1(N(CC(=O)O)C)ccc(Br)cc1I.C1(=Cc2ccccn2)CCN(C=O)CC1 c1(C(=O)NCCN(C(=O)C(C)Cc2cccnc2)CC)cc[nH]c1C1CC1 c1(C(=O)NC(C2CCCN(C(C(CC)N(CC)CC)=O)C2)C)cnn2c1OCC2 Cc1oc(C(C)C)cc1C(=O)NC1(C)CCN(C(=O)C(F)(F)C2CC2)C1 CC1CN(C(=O)CCc2cncs2)CCN1C(=O)C(CC(F)F)C1CCC1 N1(C(CN(C(C)C)C)=O)C(CNC(=O)C(C)n2cncn2)CC2CCCCC12 C=C(C)CC(=O)NC(C1CCCCC1)CNC(=O)CC1(CO)CC1 C1(NC(c2cc(C(F)F)ccn2)=O)CCCC2CN(C(=O)Cn3cnnc3)CC12 N1(CC(=O)NCCC(C)CCNC(C2(C)CCOC2C)=O)CCC(=O)NC1=O C1(C(N2CCN(CC(C)NC(=O)CC(C)(O)C3CC3)CC2)=O)CCCCN1N=O C=CCC(C)N=c1[nH]c(N2CCOC(c3ccccc3F)C2)nc2ccsc12 c1(C(=O)Nc2ncc(Br)cc2Br)nnc2c(F)cccn12 N1(C(C2C(C)=C2)=O)CC2CCC1C2NC(c1cccc(C(C)(C)C)n1)=O N1(C(CCNC(=O)OC)=O)CCCC2(NC(c3snc(Cl)c3Cl)=O)CC2C1 C(=O)(NNC(=O)CCOC1CCC1)Nc1ccc(C)cn1 c1(C(N2CCC(N(C(c3csc(C)c3)=O)CC)C2)=O)cc(Br)ccc1Cl c1(C(=O)Nc2ccc(C(=O)Nc3cc(Cl)ccc3O)nc2)cccc2occc12 Cc1ccc2sc(C(=O)NC3CC(C)N(C(=O)Cc4cnc(C)s4)C3)c(C)c2c1 C1(C(N(CCCNC(=O)CCc2ccsc2)C2CC2)=O)CC2CC(=O)C1O2 C=CC1(NC(=O)NCCC(=O)NCC2C3CCCCCC23)CCOCC1 N1(C(=O)NCC(NOCC)=O)CC(O)CC1C(C)C N1(C(c2c(C)n[nH]c2)=O)C2CCCC1CC(NC(c1csc(CO)n1)=O)C2 Cc1ncc(C(N2CC(NC(C3NC(=O)OC3(C)C)=O)C(F)C2)=O)cc1Cl C(=O)(C1Cc2ccccc21)NCC(C(C)(C)C)NC(C1(F)CCS(=O)(=O)C1)=O c1(C(N(C(C)C)CCN(C(=O)C=CS(C)=O)C)=O)ccc2[nH]ccc2c1 C(=O)(C(C)C(F)(F)F)N(CCC)CCNC(=O)CC1(C#N)CCC1 N1(C(C2CCN(CC(C)C)CC2)=O)CC(CN(C)C(c2ccco2)=O)C2(CC2)C1 C1(CNC(C2CC(n3ccnc3)C2)=O)CN(C(c2n[nH]cc2Br)=O)CC1O C1(C(=O)NCC(CNC(c2nc(C(C)(C)C)[nH]n2)=O)O)COCCN1C1CCCC1 C(=O)(C#CC1CCCOC1)N1C(CN(C)C(C2CC3(CC(=O)N3)C2)=O)COCC1 C1(NC(COCCN(C)C)=O)CN(C(C2CCC([N+](=O)[O-])CC2)=O)C2(CCC2)C1 c1(CC(=O)NC(CC)CNC(c2cc(=O)n(C)cn2)=O)cc(Cl)cc2c1OCC2 C=CCC(CNC(=O)Cn1cc(Cl)cn1)NC(c1cn(C2CC2)cn1)=O Cc1nn(C)c(C)c1CC(=O)NC1C=CCN(C(=O)CN2CCN(C)C(=O)C2)C1 Cc1cccc(C(N2CCC(C(C)NC(c3cnc(O)c(Br)c3)=O)C2)=O)c1F C1(NC(c2cc(SC)oc2)=O)CC2CN(C(C3CCCC3(C)C)=O)CC12 N1(C(=O)C#CC2CCC2)CCC2CN(C(=O)CS(=O)C(F)(F)F)CC2CC1 c1(C(=O)NC2CCN(C(COCC#C)=O)C(C)C2)[nH]c2ccc(F)cc2c1Cl c1(C(=O)NCC(CNC(C(CSC)OC)=O)(C)O)cnn(C2CC2)c1C C1(NC(=O)COCc2ccnnc2)C=CC(C(N2CC(c3ccccn3)C2)=O)C1 CC(C)CC(C)CC(C)C(=O)N(C1CCCN(C(=O)CCF)C1)C C1(C(=O)NCC2(F)CC(NC(c3n(CC)cc(Cl)c3)=O)C2)(OC)CCCCCC1 Cc1c(NC(=O)C(C)NC(=O)NC2CCCN(S(C)(=O)=O)C2)cccc1Cl CC1=CCC(C(N2CCC(CF)(NC(C3CCC(C)(C)O3)=O)C2)=O)CC1 C1(C(=O)NCCC(CCC)O)CCCCN(C(=O)CC2CC(N(C)C)C2)C1 N1(C(C(C)CNC(=O)CC2CCCNC2=O)=O)CCn2c(O)nnc2C1 C1(NC(CONC(=O)OC(C)(C)C)=O)CN(C(=O)CN(C2CC2)CC)CC1C.C1(C)CC1 C1(CC(=O)NC(C2CCC(Sc3nnnn3C)C2)C)CCN(C(=O)CNC=O)C1 Cc1cc(C(=O)NCC(C2(O)CCN(C(=O)Cc3cc[nH]c3)C2)C)ccc1O C=Cn1ncc(C(=O)NCCOCCCN(C)C(C2(CC)CCCO2)=O)c1N N1(C(CCC(C)C)c2n(CCCCSC)nnn2)CCc2ccccc2C1 c1(NC(=O)NC)ccc(S(=O)(=O)CCN=C(NCCF)NC2COC(C)C2)cc1 c1(C(C(=O)NCC(CNC(CC2C(C)C2)=O)O)=O)ccc(Cl)cc1 Cc1nn(C2CCOCC2)cc1C(=O)NCC#CCNC(=O)CC1CCCC1C CC1(C)C(C)(C(N2CC3CC(NC(=O)CCc4nccs4)C2C3)=O)C1(C)C C1(COC)(NC(=O)CCC(C)(F)F)CCCN(C(=O)CC2CCCCC2(F)F)C1 N1(C(C2(OC)CC(C)C2)=O)CCC(C(F)CNC(c2cc(C)no2)=O)CC1 C1(C(=O)NCC2(O)CN(C(c3cc(C)nn3C)=O)C2)CN2CCCC1CC2 C(=O)(CCCC(=O)NCC(O)CCNC(c1cc(C(C)C)no1)=O)NC(C)C N1(c2nccc(OC)n2)CCC2(CN(C(=O)CC(C)(C)CCOC)CC(C)O2)C1 N1(C(C(C)(C(C)C)OC)=O)CCC2(C1)CN(C(c1cnc3sccn13)=O)C2 N1(C(C(C(C)C)NC=O)=O)CC2CC(NC(=O)CC3CSCCO3)CC(C2)C1 CC1(C)CN(C(c2cc(O)ccc2F)=O)CC1NC(=O)COC1CC(F)(F)C1 C1(NC(N2CC(C(C(=O)OC(C)(C)C)OC)C2)=O)CC2CCC(C1)O2 c1(C(N2C(CNC(CCNS(CC)(=O)=O)=O)CC2)=O)cc(OC)cc(C)n1 c1(NCC(C)NC(=O)C(C)OC2CCCCC2)ncnc2cccc(F)c12 N1(C(C2C(=C)C2)=O)Cc2ccccc2OC2(C1)CN(C(c1cscc1C)=O)C2 C1(NC(C2(N(C)C)CC2)=O)CCN(C(c2cc(-c3ccco3)c[nH]2)=O)CC1CO c12ccoc1CNC2=O.c1(C(=O)NC(C(=O)NCCC)C)ccoc1Cl c1(-c2cc(C(=O)NCC3C(C)(C(C)C)C3)on2)cccc(C#N)c1 CCCC(C(=O)NCCC1CCC(NC(C2(C(F)F)CCOCC2)=O)C1)C(C)C c1cccc(F)c1[N+](=O)[O-].C(=O)(CC(F)(F)F)NCCSC(C(=O)NC)CC1CC1 N1(C(C)=O)CCC2CN(C(c3cc(Br)cc(C#N)c3N)=O)CCC2C1 C#CCC(C(=O)NCCCC(C)NC(c1c(C)noc1C(F)(F)F)=O)C1CC1 Cc1cccc(Cl)c1C(c1nnnn1C1CCC1)NCCOC.c1(C)ccn(C)c1 c1(C(=O)NCCN(C(C2SC3C=CC2CC3)=O)C2CC2)n[nH]c2cc(Cl)ccc12 c1(C(=O)Nc2cccc(C(N3CCCC3)=O)c2)ccc2n[nH]cc2c1F c1(C(N2CC3CC(Nc4ncc(Br)cn4)C2C3)=O)ccc2cccnc2n1 C1C(C(C)C)C(=O)N1.C12(CSCCOC3(C#C)COC3)CCCC1OCC2 N1(C(C2N(C)CCC2)=O)CC(NC(c2cccc(N3CCCC3)n2)=O)C(O)C1 c1(C(C)NC(C2CCCC(CC3CCCO3)C2)=O)ccc2ccccc2c1 c1(OC)ccc(F)cc1C(=O)C(=O)NCCCCCNC(c1cc(C)c(C)[nH]1)=O Nc1ccc(C(=O)NC2CN(C(=O)Cc3cnccc3Cl)C2)nc1F c1(OC)cc(OC)nc(C(=O)NCC(CNC(=O)CC(O)(C2CC2)C2CC2)CO)n1 C1(NC(C23CC(CO2)C3)=O)CCS(=O)(=O)C12CN(c1ccc3c(n1)CCC3=O)C2 CC1CCC(F)(F)CN1C(c1sccc1CNC(C1CC(=O)C12CCC2)=O)=O Cc1cc(Cl)c(C(=O)NC2CCCN(C(c3cc(C)nnc3O)=O)C2C)cn1 C1(CNC(C(COC(C)C)NC(C)=O)=O)N(C(=O)CNC=O)CCCC1(C)C C1(C(=O)NC(c2c(C(=O)NC(CC)C)con2)C)(COC)CC(F)(F)C1 Cc1cn2c(CC(N3C4CCC3C(C(=O)N(C3CCCC3O)C)C4)=O)csc2n1 c1(C(C)(C)C)ccc(O)c(NC(C2CC(N)C2)=O)c1 C1(NC(=O)CC2CC2C2CC2)C2CC3C1C3C2C(=O)N(C1C2CCCC12)C1CC1 c1(SC)cc(F)c(OS(=O)(=O)NCCOC(C)=O)cc1[N+](=O)[O-] N1(C(CSCCCC)=O)CCC(C(=O)Nc2ccncc2OC)C(O)C1 c1(CC)cnc(O)c(C(=O)NCC2CCC2NC(C2CC2CC(C)C)=O)c1 C12(C(=O)NCC3CC(NC(C(CC(=C)C)C)=O)C3)CC(CO)(C1)OC2(C)C c1(OC)ccc(C(O)CCC(=O)NCCc2cc(OC)ncn2)cc1OC C#CC(CNC(=O)CCC1(NC(=O)C(C)C(C)(C)C)CCCC1)CC(C)(C)C N1(C(Cc2cn(C)nc2)=O)CCCC(NC(=O)CN2CC=CC2)C(F)C1 CCC(CC)=CC(=O)NCCC(C)NC(=O)C=C(C)Cl C1(NC(c2cn(CCC)nc2)=O)C(C)CN(C(c2cscc2Cl)=O)CC1C Cc1cnn2ccc(C(=O)NC(CNC(c3cccn4nccc34)=O)CO)nc12 c1(C(C)C)csc(CNC(C)CCN2CCCCC2)n1 C1(Cc2cn(Cc3nc(C(=O)OC4(C=C)CCC4)c(C)o3)nn2)CCCCC1(C)C C(CCC(=O)NCC1CN(C(C2COCCO2)=O)C1)SC c1(C(N2C3C(NC(CCCCN(C)C)=O)C(C3)C2C)=O)cc2cc(Cl)ccc2s1 Cc1cc(CC(=O)NC2CC(C)(NC(=O)CSCC(F)(F)F)C2)cc(F)c1 N1(C(C2C(C)(C)CC2)=O)CCC2(CCN(C(=O)CN3CCC(=O)NC3=O)C2)C1 C1(C(N2CC(O)(CCNC(C3CC(C)(C)C3)=O)C2)=O)CCN2CCCC2C1 c1(CCCCNC(=O)Nc2cccc(CC)c2)ccc(N2CCCC2=O)c(F)c1 C1(C(N2C(c3cn(C(c4ccccc4F)C)nn3)CC2)=O)CC(=O)NC(=O)C1 CC(C)(O)C(F)C(=O)N1CCC(CCNC(C2(C#N)CCOCC2)=O)C1 c1(C(=O)NC2CC2CNC(C2CC3CCC3C2)=O)cc(F)cc2nc[nH]c12 Cc1ncnc2c1CC(C(N1CCN(CCS(=O)(=O)N(C)C)CC1)=O)CC2 C1(CC)(CNC(=O)CCOC2CN(C(=O)Cc3coc(C)n3)C2)CCCC1O c1(C(=O)NCC(C)NC(=O)CC2C=CCCC2)nc(Br)sc1C1CC1 N1(C(CCC2CCN(C(CC3(CSC)CC3)=O)C2)=O)CC(=O)N2CCCC2C1 CCCCCC(O)CC(=O)NCCCC(CO)NC(C1CC1(Cl)Cl)=O N1(C(c2ncn(C)n2)=O)CC2COCC(C1)C2NC(=O)C=Cc1ccccn1 C1(C)(CC)C=C(C(=O)N2CCCC2C2(C(=O)NCC3CC4(CC4)CO3)CC2)C1 CC1CCc2[nH]c(=NCc3ncco3)nc(N3Cc4cnc(CO)nc4C3)c2C1 C1(CNC(C2(CC=C)CC2)=O)(OC)CCN(C(=O)CCSCC)C1 N1(C(c2c(CC)ocn2)=O)CCC(CNC(C2CS(=O)(=O)C2)=O)C12CCC2 Cc1ccc(C(=O)NCC2CCC2NC(=O)CC2CSC2)cc1N N1(C(C2CC(C)(CC)C2)=O)CC(NC(C23CC(C)(C2)C3)=O)C2(CCC2)C1 N1(C(C(C)Oc2cc(C(=O)N(C)CCSC(F)F)on2)=O)CCCC(CO)C1 c1(CS(=O)(=O)NC(C2CCOC2)(C)C)nn(C)cc1Cl C=CCCC(CC(C)C)C(=O)NCCN(C(=O)CC1C=CCCC1)CC1CC1 N1(C(C2(CNC(CN(CCOC)C)=O)CC=CC2)=O)CC2(C=CCO2)C1 CC1CN(C(=O)C=C2CCN(C)C2)CCCN1C(=O)C=CC=C(Cl)Cl c1(C(=O)OCC(=O)N(C2CCN(C(=O)CCCOC)C2)CCC)cccc(OC)c1 c1(C2C(CCOCCNC(C(COCC)OC)=O)C2)cccnc1O N1(C(C(c2ccc(C)s2)C)=O)CCC(F)C(NC(c2coc(CO)c2)=O)C1 c1(C(C(=O)NC2CC(NC(C(C)SC)=O)C2)C(C)C)cccc([N+](=O)[O-])c1 C1(C(N2CCC(c3ccco3)C2)=O)CC2CC2N1C(C1CC(=O)CCO1)=O Cc1cc(C(C)C)nc(N(C)CC2CCCN2C(c2cccc(=S)n2O)=O)n1 c1(N2CC(=C(CNC(C(c3ccc(F)cc3)OC)=O)F)C2)ccc2c(n1)CCC2=O c1(NC(=O)CC2CC(NCc3cc(Br)c(O)cc3O)C2)cc(Cl)c(Br)cc1F Cc1nc(N2CCSCC2CCNC(C2CCCNS2(=O)=O)=O)c(C)c(Cl)n1 C1(CCCNC(C2(C(=O)NCC)CC2)=O)CCCN1C(c1sccc1C)=O N1(C(c2ccc(C)o2)=O)CCC(C(N2CC(N3CCNC3=O)C2)=O)(C(C)C)C1 c1(OCCC(=O)NCC(CC=C)NC(=O)COCCOC)ccc(Cl)c(Br)c1 N1(C(c2ccccc2O)=O)CCCN(CC2(C(CC)(F)F)CC2)CC1C c1(C(N2CCCC(CNC(=O)C(O)C3CCC3)C2)=O)cc(C(F)(F)F)ccc1O c1(C(N(CCOCCCNC(C(C=CCCC)O)=O)C)=O)ccc(C(C)C)cn1 c1(C(=O)NCC2N(C(C=C(C)CN3CCOCC3)=O)CCC2)ccc(O)nc1Cl N1(C(c2c(CC)ccs2)=O)CCCC12CCN(C(C1CCC3(CCC3)O1)=O)CC2 CC1CC(C)CN(C(c2ccc(F)cc2I)C(=O)NCC2CCCO2)C1 c1(C(N2CCCC(O)(CNC(CCCC)=O)C2)=O)ccc2c(n1)CCCC2 C12(C(=O)NC3(CNC(c4cc(C(C)(C)C)on4)=O)CCCC3)CC(C#N)(C1)C2 N1(C(C2(CCC=C)CC2)=O)CCN(C(C2CCC2C(F)(F)F)=O)CC1CC N1(C(C#CC)=O)CCC(O)C2(CCN(C(=O)C=Cc3cc[nH]c3)CC2)C1 C1(NC(C(C(C)(C)C)NC(C)=O)=O)C2CCC1CN(C(=O)Cc1cccnc1)C2 C1(C(=O)NC(C2CCN(C(c3cc(N)ccn3)=O)C2)(C)C)Cc2ccccc2O1 C1(OC(c2c(CC)cc[nH]2)=O)CC(F)(F)C1C N1(CC)CCCCC1C(=O)NCC1C2CN(C(=O)CC3CNC(=O)C3)CC12 C(=O)(CCC(=O)N(C1CN(C(C2CC3CCCC23)=O)C1)C)N(C(C)C)C C(CC(C(=O)Nc1cnn(C(=O)OCC)c1)NC(=O)C(C)SCC)=CC c1(NC2CC(NC(c3ccc(C)nc3)=O)C2)c([N+](=O)[O-])cccc1[N+](=O)[O-] C1(C)(CNC(c2cc(OC)no2)=O)CCN(C(c2cc(C3CCOC3)[nH]n2)=O)C1 C1(C(=O)NCCCCC#C)CC(OC)CN1C(C1CCC(C)(C)C1)=O N1(C(CN(S(C)(=O)=O)C)=O)CCC2(CCCN(C(c3cncc(C#N)c3)=O)C2)C1 c1(C(=O)NCC2C(NC(C(CO)N(C)C)=O)CCCC2)ccc2nncn2c1 N1(C(CN(CC#C)C(c2n[nH]c(C)c2Cl)=O)=O)CCC(C)C1CO N1(C(C2CN(C(C)=O)C2)=O)CCCC2(CNC(c3cc(Br)n(C)c3)=O)CC12 c1(C(N2CC(NC(c3nc(N(C)C)oc3)=O)C(F)C2)=O)cnn(C)c1C#N c1(C(=O)NCC2(CN(C(C(C)O)=O)C)CCCC2)ccc(Cl)c(F)c1 n1(-c2ccc(C)cc2)nc(C)c(C=CC(=O)NC23CCC(CC2CO)C3)c1Cl N1(CCC)CCCCC1C(=O)NCCNC(c1csc(COC)n1)=O c1(-n2cc(CN3CCCC(=C)C3)nn2)cccc2ccc(C)nc12.C(C(CC)C=O)SCC c1(C(=O)NC2(C(C)NC(c3cn[nH]c3)=O)CC2)cc(-c2ccncc2)nn1C c1(C(N(CCNC(C2C(OC)CCC2)=O)C2CC2)=O)ccn(CC(F)F)c(=O)c1 c1(-c2cn(CCN(C)C)nc2)cc(NC(=O)C(N2CNC(=O)C2)=O)ccn1 C1(C#N)(C(=O)NC2C(NC(COCCCOC)=O)CCC2)CCCO1 N1(C(C(C)Sc2ccc(O)cc2)=O)CCC(O)(CNC(=O)C#CC(C)(C)C)CC1 C1(C)(CC)CC(NC(=O)Cn2cc(Cl)cn2)CN1C(c1cnc2sccn12)=O c1(C(N(C2CN(C(c3ccnc(Cl)c3N)=O)C2)C)=O)ccc2[nH]c(=O)cnc2c1 Cc1cnc(Cl)c(C(=O)NC2CCCC2NC(=O)Cc2nnc(C)s2)c1 N1(C(C2(CC#N)CC2)=O)CC(C(F)F)C2(CC2)C1 C1(C(=O)NCCN(C2CCCC2)C(C2C(C)C2c2ccccc2)=O)CS(=O)(=O)C1 N12CC3(C1)CN(C(c1ccoc1)=O)CC3CN(C(=O)CC(F)(F)F)CC2=O.CO C12(CNC(CC(C(C)C)O)=O)CN(C(=O)C(C)(F)C(C)(C)F)CC1CCC2 N1(C(CCCOC)=O)CCC(O)(C(C)NC(=O)Cc2ccon2)C1 N1(C(C(N2CCNC2=O)C)=O)CCOC(C)(CNC(C2CCCCO2)=O)C1 N1(C(c2nnc(CC)o2)=O)CCC2C(C(=O)NCCc3nccs3)C2C1 c1(C(=O)NC(C(C)NC(C(CC)=CC)=O)C)ccnc(OCC(F)(F)F)c1 Cc1cc2ncc1CC13N(CC(C1)C3)C2=O.C(CC1=NOC(C)C1)NC(=O)CSC C1(NC(C(CC=C)C)=O)C2CC3CN(C(c4cnc5c(c4)ncn5C)=O)C1C3C2 C(=O)(CC1=CCOCC1)N(C1(CC(=O)NCC(C#C)CC2CC2)CC1)C c1(NC(CC2(C)CCN(C(=O)CCS(N)(=O)=O)C2)=O)ncc(Cl)cc1O C(C(C)(C)CCCNC(=O)Nc1cc(C#N)no1)OCC C1(OC)CC(C)CN(C(=O)C(C)(C)CCNC(c2cc(O)n(CC)n2)=O)C1 C1(NC(C#CC(C)C)=O)CC12CCC(NC(c1nnc(C(C)(C)C)s1)=O)CC2 Cc1ccnc2c(C(=O)NC3CCCC3NC(=O)C(O)c3ccsc3)cnn12 N=c1[nH]cc(CCC(=O)NCCCCCNC(=O)Cn2cc(Cl)cn2)[nH]1 c1(N(CCC)C)ccc(S(=O)(=O)NC2CN(C(C)C)CCO2)cc1F N1(C(CC(C)(C)OC)=O)CCC(NC(c2ccc(SC(F)(F)F)cn2)=O)CC1C C1(C(=O)NC(CCNC(C2(OC)CC(CF)C2)=O)C)CCC(OC(F)F)CC1 CCCC(C(=O)OC)C(=O)NCC1(NC(=O)CSc2nnc(S)s2)CCC1 C1(c2cccc(OC)c2)CN(C(C2(C)C=CCC2)=O)CCN1C(=O)CCC1CC1 C(=O)(C1Cc2ccc(F)cc21)N(C1CCCCC1Nc1ncnc(O)c1Br)C c1(CC(=O)NCCCCN(C(c2nc(C(=O)OC)sc2)=O)C)cc(C)ccc1F Cc1nc(C(C)NCCNc2nnc(C(C)(C)C)s2)c(C)o1 c1(C(N2C(C)CN(C(=O)Cc3cnc[nH]3)CC2)=O)ccc2c(c1)CCCO2 C1(O)(C(N2CC3(CN(C(C4OCC(=O)C4)=O)C3)C2)=O)CN2CCC1CC2 C1(NC(CN(C2CCCC2)C)=O)CCC(NC(=O)CC2(C)OCCO2)C1 n1(CC)nc(C(=O)NCC(C2CC2)N(C(=O)C(F)C2CCC2)C)ccc1=O N1(C(c2ccc(C(=O)OC)o2)=O)CCC(NC(=O)CC(C)(C)O)C(O)C1 N1(C(c2c(C(=O)OC)nn(C)n2)=O)CCC(CNC(C2CC2F)=O)CC1C c1(C(=O)NCC2(O)CC(NC(=O)CC3C=CS(=O)(=O)C3)C2)ccc2scnc2c1 N1(C(C(=O)NC(C)C)=O)CCC(C(=O)NCCCc2nncs2)C1C C1(NCC=C(CC)CC)C(C(=O)NCC2(CO)CC2)C1(C)C C1(C(C)(C)C)CN(C(c2cnsn2)C2CC2)CC1c1ccccc1.C12CC1NC2=O CC1=C(C(=O)N2CCC(CNC(=O)Cn3ccnc3C(C)C)C2)CCC1 c1(NC(C2CCCN(C(CC(C=C)CC)=O)C2CC)=O)cc(C)c(C)cc1C C1(C(=O)NCCCCCN(C(=O)CC2CC(C)(C)CCO2)C)CC(=O)CC(=O)C1 N1(C(c2c(C)scc2)=O)CCC(O)(C(C)NC(C2CC(C)(C)C2)=O)CC1 N1(C(C23N(C(c4cn(CC)nc4)=O)CCC2C3)=O)CCC(C)(N(C)C)CC1 Cc1ccc(C)c(C(=O)NC(C(C)NC(=O)C(C)(C)C2CCCC2)C(C)C)n1 c1(C(N2CC(OC3CCN(C(C4C(=C)CC4)=O)CC3)C2)=O)c(C#N)cnn1C c1(C(=O)NC(C)(CNC(C2(S(N)(=O)=O)CCC2)=O)CO)cc2c(=O)[nH]ccn2n1 C(=O)(C(C)C(O)C(C)CC)OCCNC(=O)CC(=O)OC.CCC(C)C1C(=O)N1 S(=O)(=O)(c1ccccc1F)NCC(=O)NCC(C)N(C(Cc1c(C)noc1)=O)C CC1CN(C(C2CCCSS2)=O)CCN1C(c1coc(Br)c1)=O CN1CC(C(=O)N(C2(C(N3CCCCC3(C)C)=O)CC2)C)CCC1=O N1(C(C2N(C(CCC#C)=O)CCC2)=O)CCC(CO)(CO)C1 C1(NC(c2cnc(C(C)C)[nH]2)=O)COCCN(C(=O)C(C)Cc2ccnn2C)C1 C1(CCCNC(CNC(CC)=O)=O)CN(C(c2ccc(OC)o2)=O)CCO1 c1(C(N2CCCC(COC)(OC)C2)C(=O)NCC(=C)C)ccc(F)c(Cl)c1 c1(Cn2cc(C(N3CCC(OC)C3)C(=O)O)nn2)c(C)cccc1Cl Cc1ccc2c(C(=O)Nc3cc(O)ccc3CO)ccnc2c1 C1(O)(NC(=O)NC(C)Cc2ccco2)CC(NS(C)(=O)=O)C1 C12(NC(COCCC(C)C)=O)CCCC1N(c1ccc(C(F)(F)F)cn1)CC2 C(=O)(C(Cc1ccccc1)CN)NC(c1noc(CCC(C)C)n1)CCC c1(NC(C2(C(=O)OC)CCC2)=O)cc(Cl)cc(Br)n1.C12CC1C(=O)N2 C1(NC(C2(COCC)CC2)=O)CC(C(=O)N2CC(C(C)C)C2C(C)C)=CC1O C1(CNC(=O)NCC(c2cccc(Cl)c2)N(C)C)CCC2(CCC2)O1 c1(NC2(C(=O)NCC=CCNC(C3CCN(CC(F)(F)F)C3)=O)CC2)ccncc1 Cc1cnc(CC(=O)NC2(CN(C)C(c3ccc(CN(C)C)o3)=O)CC2)o1 c1(C(=O)NCC=CCNC(C=CC(=O)OCC)=O)sc(C)cc1Cl CC(=NOCC#N)C(=O)NC1COCCC1C(=O)N(CCS(C)(=O)=O)C c1(CSCC(=O)NCCN(C(CC(CC)O)=O)C)cc(C)ccc1C N1(C(C(C)N(C)C)=O)CC(N(C)C(c2cnn(C)c2Br)=O)C(F)C1 C1(NC(c2c(C)cnn2C)=O)CCCN(C(=O)Cc2[nH]cnc2C)CC1F c1(C(N(CCN)C(C2CCC(OC(F)(F)F)C2)=O)=O)cnn2cc[nH]c(=O)c12.CC Cc1nocc1NC(=O)CNCC(C)(C)C1CCOC1 C(C(=O)N1CC(C2(NC(c3nc(Cl)sc3Cl)=O)CC2)C1)(C(C)(C)C)N(C)C c1(C(=O)NCC2N(C(c3cc(C)n(C4CC4)n3)=O)CC=C2)cccc2nn[nH]c12 c1(C(=O)NCC(C)(CNC(c2cscc2C(C)C)=O)OC)cn(C)[nH]c1=N N1(C(COCC(=O)NC)=O)CCCOC(NC(=O)CC(C)=C(C)C)C1 c1(C(=O)NCC2(F)CCN(C(=O)CC3CCCCC3O)C2)nccc(Cl)c1F c1(NC(COc2cccc(C)c2)C)ccc(S(=O)(=O)NCc2sncc2Br)cn1 C(=O)(CCC(F)(F)F)NC1CCCN(C(Cc2n[nH]c(=N)s2)=O)C1 N1(C(C(F)=CCC)=O)CCC(CNC(=O)CCS(C)=O)(COC)C1 C1(CC)CN(C)C(=O)CN1C(=O)OCc1ccccc1.C1(N)(C)COC1 C#Cc1ccc(C(N2CCCC2C2(NC(=O)Cc3c[nH]ccc3=O)CC2)=O)cn1 c1(OC)ccc(C(=O)OCC23CC(C(C)CCO)(C2)C3)c(Cl)n1 Cc1cnc(Cl)nc1NC(C1CCN1C(c1cnccn1)=O)=O N1(C(C(C)OCC(C)C)=O)CC(N=[N+]=[N-])CC1C(=O)NCC=C(C)C C(=O)(CCCCCC#N)NCC1CN(C(CN(C(C)C)C)=O)CC(C)C1 C(c1ccccc1)=CC(=O)N(CCCNC(C(N)=O)=O)C1CC1 c1(-n2ccnn2)ccc(C)c(-c2ncccc2F)c1.C(c1ccc(Br)s1)=C(C)CSCC N1(C(=O)OC)CCN(C(=O)CC(C)NC(C2CCCC2C)=O)CC1 c1(CCC(=O)NCCCNC(C2CCN(C)C2)=O)cc(F)cc(F)c1 CCC(C)(CC)C(=O)N(CCCCC(=O)NC1C(=O)C1CC)C.OC C(CS(=O)(=O)CC(=O)NCCC(=O)NOCCO)OC N1(C(CCC(=O)NC2CC(C)OC2)=O)CCN(Cc2ccccc2)CC1c1ccco1 c1(C(=O)NC2CCCN(C(Cc3c(C)cccc3C)=O)C2)ccn2nnnc2c1 CS(=O)(=O)c1ccccc1CN(C(c1[nH]ccc1-c1cncs1)=O)C1CC1 C1(C(=O)NC(C2CN(C(C3C(=C)C3)=O)C2)C)CCCC1C(C)C Cc1ncc(CCNC(C2CC(C)N2C(=O)CCCC2CCC2)=O)s1 N1(C(Cc2c(C)nsc2)=O)CC(C(=O)NCC(C)(C)N2CCCC2)C2(CC2)C1 c1(NC(C(c2ccccc2)NC(C2(CC)CCCN2)=O)=O)ccc(C)c(C)c1 c1(C(=O)N(C)CC2COC(=O)N2)cnccc1C(=O)NC1C(OC)CCO1 c1(C(N2CCC(OCCNC(CC3(C)CC3(F)Cl)=O)C2)=O)ccc(N)c(O)c1 CC(C(CO)NC(=O)CCc1cn[nH]c1)NC(C1CCC(n2ccnc2)O1)=O c1(C(N2C3CN(C(C(C(C)(C)C)OC)=O)C(CC3)C2)=O)ccc2cnc(C)n2c1 c1(SC)cc(F)ccc1C(N1CC(NC(c2occc2C)=O)C2CC12)=O N1(CCC(=O)NC(C)(C)CCNC(=O)C=CC2CCC2)Cc2ccccc2C1 c1(C(=O)OC)cncc(C(N2CC(O)(CNC(c3ccncc3C)=O)C2)=O)c1C c1(C(CN(C(=O)CSC2CCN(C)C2=O)C)O)cc(Br)ccc1Cl N1(C(CCCCCC)=O)CCC2CCN(C(C3CN(C(C)C)CCO3)=O)C2C1 c1(C(N2CCC(C(C)NC(c3ccc(CC)[nH]3)=O)CC2)=O)ncnc(O)c1F C(=O)(C(C(CC)CC)OC)N(C)CCOC.N1(C(CCCC#C)=O)CCCC(O)(CN)C1 C(c1cccc(O)c1)=CC(=O)NC(N1CCN(C(C2CC23CCC3)=O)CC1)C C12(CNC(CC(C)C(F)F)=O)CCCC1CN(C(c1ccc(CO)nc1)=O)C2 C12(CNC(C3CCC(C(=O)OC)C3)=O)CCC(CC1)N(C(C1(C)CC1(F)F)=O)C2 c1(C(N2CCC(O)(C(C)NC(=O)C=CC3CC3)C2)=O)ccc(N)c(N)n1 C1(c2cn(CCC(CC)C(=O)NC(=O)CC3CCN(C)C3)nn2)CC2(CCC2)C1 C1(C)(C(N(CCCCCCNC(c2ccon2)=O)C)=O)CCC(F)(F)C1 C(=O)(C1=C(Cl)CCC1)NCC1CC(NC(C2CN(CCC)C(=O)C2)=O)C1 c1(OC)c(C(N2CCC(NC(=O)CC3CC34CC4)C(F)C2)=O)ccnc1Cl c1(OC)ccc2nnc(CCC(=O)NCCCn3cnccc3=O)n2n1 c1(C(N(C)CC2(NC(=O)CC3COCCO3)CC2)=O)occ2c1CCCC2 C#Cc1cccc(C(N2CC(NC(=O)C=Cc3ccccc3OC)C2)=O)c1F C=CCC(C)(C)CNC(c1oc(CNC(C2CCC(F)(F)C2)=O)nc1C)=O C(C(C)C(F)C(=O)Nc1ccccc1C#N)NC(COCCSC)=O c1(CCC(=O)N(CC(C)N(C)C(C2(F)CCC2)=O)C)ccnc2ccccc12 C1(NC(=O)CN2C(=O)CCC2=O)CC(F)CN(C(c2cnsc2)=O)C1 N1(C(C)C)CCN(C(C2CN(C(C3CC(C)CCC3)=O)CC2N(C)C)=O)CC1=O C(=O)(CC1=CCCCC1)NCC(C)N(C)C(c1ccc(C2CCC2)cc1)=O c1(C(c2nnnn2C)NCC(C(=O)NCC(=O)NC)C)ccnn1CCF n1(CC)ncn(NC(=O)C(CC)NC(=O)CC2CCC(=O)NC2)c1=O c1(C(N2CC(CC=C)(NC(=O)CCC(F)F)C2)=O)cnc2c(cnn2C)c1 c1(C(N2CCC(OCc3nc(C)on3)C2)=O)cccc2c(Br)cccc12 N1(C(c2cccc(C)n2)=O)CCC(CNC(c2ccc[nH]2)=O)C(C)C1 C(=O)(CC1COc2ccc(Br)cc21)OC1C2(COC(C)(C)C)C(C1)ONC2=O C1(NC(C(C)OCCCC)=O)CC2CC(NC(c3ccc(OC)cc3Cl)=O)CC12 CC(C(=O)N1CCC2CC12C(=O)NOCc1ccccc1)S(C)(=O)=O N1(C(C=Cc2c(C)ccs2)=O)CCCC(NC(=O)CN2CCCC2=O)C1C C(=O)(CCC1=NNC(=O)CC1)NC(C1CCN(C(C(C)CN(C)C)=O)CC1)C C1(NC(C2C(C)C2)=O)CCN(C(c2nc(Br)c[nH]2)=O)C1c1ccccc1 C=CCCC(=O)NC1CCCC1CNC(c1cn(CC(O)CC)nn1)=O Cc1cc(CC(N2CC(NC(=O)COc3cccnc3)CCC2C)=O)ccc1F C(N=c1[nH]c(=NC2CN(C)C3(CCOCC3)C2)c2ncccc2[nH]1)c1c(C)noc1 C(CN=c1[nH]ccn2nnnc12)N(C)C(c1cncc2nc[nH]c12)=O Cc1cccnc1C(F)C(=O)N(CC(CO)(CO)NC(=O)Cc1cnoc1)C n12cc(nn1)C#CCC2.c1(C2C(N(CCOCC)C(=O)OC)CC2)nc(S)n[nH]1 c1(C(N(C(c2ccccc2)CNC(=O)C(Cl)=CCl)C)=O)nnn2c1CCC2 CC(C)(CCCF)C(=O)NCC1CCN(C(=O)CCOCC2CCC2)C1 N1(C(C(CC=C)C)=O)CC2(CO)CC1(C(=O)Nc1ccccc1CCO)C2 N1(C(CN2CCN(CC)CC2)=O)CCC2CN(C(=O)C=Cc3cccc(Cl)c3)CC12 N1(C(CC(=O)C(C#CC)C)=O)CCCN(c2ccncc2)CC1 c12cccc(c1)S(=O)(=O)NC1CCCN21.C(C(=O)N=c1cco[nH]1)(C1COC1)OC c1(C(N2CC(CC(N3CC(CC(C)C)C3)=O)(OC)C2)=O)ccc(O)nc1 CC(CC(=O)N1CCN(C(=O)C#CC(=O)N(C)C)CCC1C)CC(F)(F)F C1(CNC(c2cc(CNC(=O)C=C3CCC3)sc2)=O)(CO)CCOCC1 C(=O)(CC(C)(O)C(F)(F)F)N1CC(c2c(CNC(C(C)CC3CC3)=O)nco2)C1 N1(C(C23C(C(N)=O)(CCC2)C3)=O)CCC2(CCC2)C(CNC(C2(Br)CC2)=O)C1 C1(CCC)CC(OCCCCNC(=NC)NCCF)C1(C)C C12(C(=O)NC3CN(C(C(C)(C)C4CC4)=O)C4(C3)CCC4)CC3CC(C(=O)N1)C2C3 c1(C(c2n(CCC)nnn2)NC(c2ccsc2)C2CC2)nc2ncccn2n1 C=CC1(C(N2CC3(CNC(=O)CC4C(=O)NN=C4C)CCC2C3)=O)CCOCC1 C(=O)(C(C)(C)C(C)(F)F)NCC1CC(C(=O)NCc2cc(C)no2)C1 c1(OC)ncc(F)c(N(C2CC3CNCC23)C(c2ccc(C3CC3)nc2)=O)n1 c1(C(=O)NCCC2CC(NC(C(C)CS(C)=O)=O)C2)ccc(F)c2[nH]ccc12 C1(CCCCNC(C(COC)OC(F)(F)F)=O)CCCN(C(=O)C(F)OC)C1 NS(=O)(=O)c1c[nH]c(C(N2CC3CCC3(CNC(=O)CC3CC(F)(F)C3)C2)=O)c1 Clc1ccc(C2COCCN2Cc2nnnn2CC2CCCO2)cc1 Cc1ccc(Cl)c(C(=O)NC2(CCNC(c3nn(C)nc3Br)=O)CC2)c1 c1(CN(C(C)C)C(C2CCN(c3cccnc3)C2)=O)nc(-c2ccccc2)no1 N1(C(CCCC=C)=O)CC(=O)NCC1C(=O)NCC1(C)CCCOC1 C(=O)(C1=NOC(C)C1C)NC1CC(NC(C(CC#C)C)=O)C1 C1(C(=O)NC(CNC(C)=O)CC(C)C)CCCN1S(=N)(=O)N(C)C c1(NC(N2CCCC(OCCCl)C2)=O)sc(Cl)cc1Br c1(N2CCCC(CN(C(C3N(CC#C)CCC3)=O)C)C2)nc(Cl)ncc1Cl C12(NC(C(CC=CC)C)=O)CCC(C(=O)NC3CCN(CC4CC4)C3)(CC1)C2 N1(C(CC(CC#C)NC(C2CC2C#N)=O)=O)CC(O)C(C2CC2)C1 C(=O)(CCCCC(F)(F)F)N1C(CC(=O)N(C2CC3CC3C2)C)CCC1 c1(OC)cc(C)ccc1C(N1CCCC1C(=O)Nc1nc(F)ccc1Br)=O c1(C(N2CC(N(C(=O)CC3CCCO3)C)C2)=O)cncc(C2CCOC2)c1 C1(CNC(Cc2nc(NS(C)(=O)=O)sc2)=O)CN(C(C2(Cl)CC2)=O)CCN1C N1(C(c2oc(C)c(CO)c2)=O)CC(NC(c2cc(F)cnc2O)=O)CC(C)C1 N1(C(CC2C(OC)COC(C)(C)OC2)=O)CCOCC1C1CCCO1 C1(CNC(c2c[nH]nc2C(F)F)=O)COCCN1C(c1cccnn1)=O c1(C(N2CCCC(CNC(C(COC)COC)=O)C2)=O)cccc2c1C(C#N)C2 c1(OC)cc(OC(C)=O)cc(NC(C2CCN2C(C2(N)CC2)=O)=O)c1 C(c1c(F)cccc1F)=CC(=O)NC1CCN(C(CC2CCC(OC)CC2)=O)C1 Cc1ccc(C(=O)NCCCN(CCO)C(C2CC(C)C2)=O)cc1C(F)(F)F C1(C(N2CC(C(=O)NC)C2)=O)CC2C=CC1N(C(=O)C1=COCCC1)C2 n1(CC)c(C)nn(CC(=O)NC2(C)CN(C(c3cnc(C(F)F)cc3C)=O)C2)c1=O C(C(CC(=O)N=c1ccn(CC(C)C)[nH]1)NC(=O)CCCCC1CC1)OC CCCC(C(=O)NC(C)Cc1cccs1)NC(C1(CC(C)C)CC1)=O c1(CN2C(C(=O)Nc3c(C(N)=O)n[nH]c3)C=CC2)ncc(Br)cc1Br CCC(C(=O)N1CC(O)CC1CNC(=O)CC(C)(C)CCOC)C(C)(C)CC c1(SC)cnc(OC)nc1.N12CCC1C(=O)N(CCC)CC2=O CC1(C)CC(C(N2CCN(C(c3ncccc3F)=O)CC2CCO)=O)CNC1=O N1(C(C2(C=C)CCC2)=O)C2CCC1CC(N(C(=O)CCC1C(=O)NN=C1C)C)C2 C(=O)(C(CC(=O)NC1CC(CNC(C2CCNC2=O)=O)C1)C(C)=O)OCC C1(NC(C(CC)(C)O)=O)CN(C(C2(CNC(=O)NC(C)C)CC2)=O)CCC1(C)C C(=O)(C1=NOC2(CCOC2)C1)N1CC(OCCNC(C(C)CS(C)(=O)=O)=O)C1 c1(C(=O)NC(CC2CN(C(C=CSC)=O)C2)C)cc2c(=O)cc[nH]c2s1 c1(C(=O)NCCOCCCC#C)ccc(C(=O)N(C)CC2(CO)COC2)s1 Cc1cc(CNC(=O)C(C)C(C)NC(=O)C=CC(C)(C)C)cc(O)n1 c1(C(N(C(C)CNC(C2CC2C(F)F)=O)C)=O)ccc2c(c1)nc(O)n2C C1(C(=O)NC)CC(O)CN1C(=O)C(n1cc(-c2cc(O)ncn2)nn1)C C#Cc1cccc(C(N2CC=CC2(C)C(=O)NCC2(O)CC(CO)C2)=O)c1C N1(C(c2ccc(NCCCC)cc2)=O)CCS(=O)CC1C(=O)O N1(C(C2C(C3C(C(=O)OCC)C3)CC2)=O)CCC(c2cn(C3CC3)nn2)C12CC2 C1(C(=O)N(CC(CC)NC(=O)C(C)C)C)(CC)CCC(F)(F)CC1 c1(NC(N2CCC(F)C2)=O)cc(F)c(Br)cc1Cl.Cn1c2ccc1C1COCCN21 C(=O)(C1=C(C)OCCS1(=O)=O)NCCNC(C1CCCN(CCC)C1)=O C(=O)(C1Cc2c(Cl)cccc21)NC1(CNC(c2c(=O)ccn(C)c2)=O)CCCC1 c1(C(=O)NC(CNC(c2nc(C)c(C)[nH]2)(C)C)C)ncnc2sccc12 C1(C(=O)NCc2ccc(CC)o2)CC2C=CC1N(C(=O)CCC1OCCO1)C2 N(C1c2ccccc2C2CC1C2)C(C1C(C)C1)=O.N12CSCC1C2=O c1(C(=O)NC(CNC(Cc2c(C)ccnc2)=O)(C)CO)coc2cc(F)ccc12 c1(OCC)cccc(C(=O)Nc2cccc(NC(c3c(O)cccc3Cl)=O)c2)c1O c1(C(=O)NCCCCC(C)NC(c2cc(Cl)ccn2)=O)ccc(Cl)nc1N c1(-c2cn(C(C)CNC(C3CC3c3ccn(C)c3)=O)nn2)ncnc2sccc12 CCCS(=O)(=O)C(C)C(=O)NCC(CC)NC(c1ccc(-c2cccs2)[nH]1)=O N1(C(c2c(C)nsc2)=O)CCCCC(C(=O)NC2CCCN(C(=O)N(C)C)C2)C1 c1(CNC(CC(C)SC)=O)cc(C(=O)N(C)CC2(C#N)CC2)ccn1 c1(C(N2C(C)CC(NC(C3CCC(CC)O3)=O)C2)=O)c[nH]cc(Cl)c1=O C1(NC(C(COC)O)=O)CCCC12CN(C(C1CCOC(C)C1)=O)C2 N1(C(C(CC)C(C)C)=O)C2CCC1CC(CNC(C1CC3(CCC3)C1)=O)C2 C1(F)(CNC(CCC(N)=O)=O)CCCN(C(C2CCOC2c2ccncc2)=O)C1 C1(NC(=O)CCc2nncs2)CCN(C(=O)CC(F)F)C1C1CC1 Cc1cc(O)c(C(=O)NCC(Cc2ccccc2)C(N)=O)nn1 N1(C(C(C)(C)c2cscc2Cl)=O)CCC2(CCN(C(C3COC(=O)N3)=O)C2)C1 CCC(C)C(CN(C)C)NC(C1(NC(=O)CN2CCN(C)CC2)CC(CO)C1)=O C1(C(=O)NCC2(OC)CN(C(C3C(CCC)CCC3)=O)C2)CC1C1CCCCC1 O=C1CN(C(=O)C(O)Cn2cncn2)C(C(=O)NC2CCC(F)(F)C2)CN1 C1(NC(CNC(C(CC)C)=O)=O)CN(C(=O)CCn2ccnc2C)C(C)(C)C1 O=C(CCC(=O)N(C)CCc1cn(CC2CCCO2)nn1)c1cccs1 C(=O)(CCCC#N)N(C(CCNC(c1n(CC)ccc1)=O)C)C CC(C)C(C(=O)NC(C1(n2cc(CCCN(C)CCO)nn2)CC1)=O)SC(=N)N c1(C(=O)NC2C(CNC(C(C)Cc3cnc[nH]3)=O)C2)ccc(=O)n(C)c1 c1(C(N2CC(C(C)NC(=O)COC3CCCOC3)C2)=O)cccc2c1CCC(=O)N2 c1(C(N2CC3=C(CN(C(CC(C)OC)=O)C3)C2)=O)ccc2c(c1C)OC(F)(F)O2 N(C1c2ccccc2CCC1F)C(C1(C)CCCN1)=O c1(OC)cccc(C2(NC(=O)C(=O)NC(C)C(C)NC(C)=O)CCC2)c1 C1(C(=O)NCC23CC(NC(C(C)OCCC(C)C)=O)(C2)C3)CCC(F)(F)C1 N1(C(c2ccc(Cl)c(F)c2O)=O)CCC2(CCCN2C(C2CCCC(O)C2)=O)C1 C1(CC)CN(C(=O)C2=COCC2)CC1C(=O)NC(Cc1cnn(C)c1)CO c1(C2C(NC(c3nnnn3C)CCC)CCC2)ccccc1Cl C=C(C)CC(C(=O)NC1CC(N(C)C)C1)NC(=O)CCSCCCC N1(C(CC)C(=O)N(CC(C)CNC(c2nnsc2C)=O)C)CCN(CCO)CC1 C#Cc1ccc(SC(C)C(=O)N2CC(C(=O)NCCC(C)(C)C)C2)nc1 C1(CC(N2CCC3C(NC(c4[nH]cc(C(=O)OC)c4)=O)C32)=O)CN2CCC1CC2 c1(N2C(C(=O)Nc3c(O)cccc3Cl)CC3CC32)ncc2sccc2n1 N1(C(C(OCC)OC)=O)CCN(C(=O)CC2(c3ccccc3)CC2)C2CCC12 c1(C(=O)NCCNC(CCC=C=C)=O)cc(O)ccc1N(C)C c1(C(=O)NCCC(C)N(C)C(C2CCC3CC23)=O)coc(CO)c1 c1(C(=O)NC2CC(NC(c3cc(OCC)no3)=O)C2)nc(CC)ncc1Br C(=O)(CC1OCCc2sc(Br)cc21)OCC(=O)Nc1sc2c(c1)CC(C)CC2 N1(CC)CC(C(N2CCCC2CNC(=O)Cc2cncc(C)c2)=O)CCC1=O C1(OC)CC(C(=O)NCC2CC=CCC2)N(C(=O)C=Cc2cn(C)nn2)C1 c1(C(N(C)CC2(CNC(=O)C3=C(C#N)CCC3)CC2)=O)cc([N+](=O)[O-])cnc1O c1(OC)ccc(NC(=O)NC(C(=O)NCc2ccccc2)C2CC2)cc1.c1ccco1 c1(C(N2CCC(C(N)=O)C2)=O)cc2n(n1)CCN(C(C1CNC(=O)C1)=O)C2 C(C(=C)CCNC(=O)C(C)(C)N(C)CCC)NC(CNC(COCC#C)=O)=O CC1CC(C(N2CC=CC(NC(C3CCC(=O)N(C)C3)=O)C2)=O)CC(=O)N1 c1(C(=O)NCC2C(CNC(CNS(N)(=O)=O)=O)C2)ccc(C(F)(F)F)o1 C1(C(=O)NCCNC(c2csc(C(F)(F)F)n2)=O)CCCCS1(=O)=O CC(C)(CCCNC(=O)Cc1ccc(Cl)s1)NC(C1CC1c1cccs1)=O C(=O)(C1=CC2(CN(C(c3cncs3)=O)C2)OC1)NC(C=C)(C)C C(=O)(C(C)(C)O)NCC(CNC(c1cnn(C(C)C)n1)=O)OC c1(NC(=O)CC2CCCCO2)cccc(N2CCCCC2)c1 C(=O)(CCS(=O)(=O)N1CCOCC1)NCC(CNC(c1cc(CC)oc1C)=O)O c1(C(=O)NC2CCC(NC(C(CN(C)C)N(C)C)=O)C2)nccc2c[nH]nc12 C12(CNC(C3C(C)CCC3)=O)CC1CN(C(c1cc(CO)on1)=O)C2 C1(CNC(=O)COC(F)F)(CNC(c2occc2CCO)=O)CCOCC1 C1(CNC(c2nn[nH]n2)C)CC(C)CCN1Cc1ccccc1 C(C(O)C(=O)NCc1cc(C(N2CCCC2C(=O)NC2CC2)=O)no1)SC C(=O)(CCCCN(C(=O)C(C(=O)OCC)OC)C)NC(C(=O)N(C)CC)C CC(CCC(C)(C)C)C(=O)NCC1(O)CC(NC(C2(C(F)(F)F)CC2)=O)C1 CN1CCn2ncc(CNC(=O)NCC3(CO)CCO3)c2C1=O C12(C(=O)NC(c3ccc(-c4cccc(C)c4)cc3)CCO)CC=CCN1CCC2 C1(C(N2CC(C)C(CNC(=O)C(F)C3CCOC3)CC2)=O)CCCC12OCCO2 c1(C(N2CCC(CCNC(CN(C3CC3)CC)=O)C2)=O)ccc(C(N)=O)cc1 c1(CCN2CCC(NC(c3ccccc3)=O)C2)ccc(F)cc1F C12(CC)CCC(C1)N(C(c1cccc(OC)c1)CNC1CCCC1)C2 c1(C(=O)OC)ncccc1NC(c1ccc(SCc2cncs2)cc1)=O N1(C(C)Cc2csc(-c3ncccn3)n2)CC2(CCN(c3nnnn3C)C2)C1 c1(C(N2CCC(=CCNC(C3C(=C)C3)=O)CC2)=O)cccc2ncnc(O)c12 CCC(CC)C(=O)NC(C1CCN(C(C2CC(N3CC(O)C3)C2)=O)C1)(C)C C1(O)(CNC(C(C)CCN(C)C)=O)CCN(C(C23CC(F)(C2)C3)=O)CC1 C1(CNC(C(C)C2CC2)=O)(NC(c2cc(F)cc(F)c2)=O)CCC(F)(F)CC1 c1(N(CCC(C)(F)F)C)nc(=N)[nH]c(=NCC2CCOc3ccccc32)[nH]1 c1(CCC(=O)NC(C2CC=CCC2)C(=O)NC2(CSC)CCC2)ccn(C)n1 C(CCC(O)C(=O)N(CC(C)(C)C)CC1CCCCC1)NC(C)=O n1(CC(N2CCC(N(C(=O)C(O)c3ccsc3)CCC)C2)=O)c(O)nnc1O N1(Cc2scc(COC)c2)CC2CCCCC2C1.c12cc(ncn1)N2 c1(C(=O)NCC(C)NC(=O)CC23COCC(C2)C3)nncc2c1CCCC2 N1(C(C(c2n(C)ccc2)=O)=O)CCCC(C2CN(C(=O)CC3CCCC3)C2)C1 CCCCC(O)CC(=O)N1CC(NC(=O)C(C2CCCC2)OC)CC1CO Cc1cnc(N2CCOC2C)c(S(=O)(=O)NC2CC3(CCC(C(N)=O)CC3)C2)c1 c1(C(=O)NC23CC(NC(C4=C(C)CC4)=O)(C2)C3)ccc(F)c(N)c1 c1(CC)cc(C(=O)NC(C)(C)CCCNC(c2ccc(F)s2)=O)cc(Cl)n1 N1(C(C2CN(OC)C(=O)C2)=O)C2CCCC1CN(C(c1cc(Cl)no1)=O)CC2 N1(C(CNC(C=CSC)=O)C)CCN(C(C2OCCC2c2ccccc2)=O)CC1 N1(C(CCN(CC(C(C)C)C)C)=O)CC2CCCN(C(=O)CCN(C)C)C2C1 C#Cc1ccc(C(N2CC(NC(c3cnc(C4CC4)s3)=O)CC(C)C2)=O)cc1Cl C1(C(N2CC=CC(NC(c3cccc[n+]3[O-])=O)C2)=O)CCc2ncnn2C1 Cc1[nH][nH]c2ncnc(=NC(C)C3CCN(C(c4scnc4Cl)=O)C3)c1-2 C(=O)(C(CC(C)(C)C)NC(=O)C(C)SC(C)C)N(CCCC#C)C c1(C(N2CCN(C(c3cc(CC)on3)=O)C3C2C3)=O)c[nH]c2c(CC)cccc12 C(=O)(C1=CCCC1)NCC(C)N(C)C(c1cn(C)nc1C(C)(C)C)=O c1(CCC(=O)NCC2CCC(NC(c3cc(C4CC4)on3)=O)C2)cncc(F)c1 C(CCC)(CCCNC(=O)Cn1ccc(Br)n1)NC(C(CC#C)C)=O C12(CCCCC1)C(=O)NCC1CN(C1)C(=O)C1C(CC1)OC2.O(C(F)(F)F)CC c1(-c2cc(C)nn2C)ccc2[nH]c(C(=O)NCc3cscn3)c(C)c2c1 C1(CC(=O)N(C)Cc2ccon2)CCCCN1C(=O)CC1CCCSC1 C(=O)(C(C)(C)COC)N(CCCCCNC(C1C(=C)C1)=O)C C1(C(N(CCCCCC)C2CC2)=O)C=CCN(C(=O)CC2CCOC2)C1 c1(C(=O)NC2(CNC(C(CC#C)C)=O)CCCCC2)cc2cccnn2n1 c1(C(N2CCC(N(C(C=C=C(C)C)=O)CCO)C2)=O)cccc(F)c1C(C)C C(CN=c1cc(Oc2ccccc2)c2ccccc2[nH]1)(OCC)OC C1(NC(C(C)=C(C)C)=O)(CNC(c2nn(C)c3c2CCC3)=O)CC2CCC1CC2 c1(C(=O)NC(C(C)NC(C2CC(CF)C2)=O)(C)C)ccc2nc[nH]c2c1F C(C)(C)(CCCC(=O)NCCC(CC)OC)NC(CCCCC=C)=O n1(CC(=O)OC)nccc1C1CC1C(=O)N(CCOC)CCOc1ccccn1 C123CCC(CC1)(C2)C(=O)N3.c1(C2CN(C(C(C3CC3)SC)=O)C2)noc(SC)n1 Cn1nnc(CNC(C23C=CC(CC2)C3)=O)c1C(=O)NCC12CC(CO1)C2 c1(C(N(CCN(C(C2(COC)CC2(F)F)=O)C)C)=O)cc(Cl)nnc1O C1(NC(CCC2(C)CCOC2)=O)CC2CC1N(C(c1cnn(CCF)c1)=O)C2 N1(C(CSC)=O)CCC2(CC1)COC(C)C2NCC1CC(O)CN1 C1(CNC(c2nc(C)sc2)=O)CCCN(C(c2c(N)cccc2Cl)=O)CC1 c1(C(=O)OC)cn(CC(=O)NC2CC2NC(=O)C(F)(F)C(F)(F)F)c(=O)nc1O c1(NC2(CNC(c3c(C)noc3)=O)CCCCC2)cc2nncn2cn1 C(C(=O)N1CC(C(=O)NCC(C2CC2)NC(=O)OC(C)(C)C)C1)(N(C)C)NC N1(C(CC(=C)C)=O)CCC2CN(C(c3ccc(N4CCCS4(=O)=O)cc3)=O)CC12 c1(OC)ccc(C)c(C(=O)NC2CCN(C(=O)C3=CCSC3)CC2CO)n1 c1(C(N2C(CNC(=O)CCc3cnoc3)CC2)=O)cnccc1Br Cn1nc2c(c1C(N1CC(CNC(=O)CN3CCOCC3)C1)=O)CCCC2 c1(C(N2CCCC(C)(CNC(C3CC(F)(F)CS3)=O)C2)=O)cccc2sncc12 C(C)(N=c1ccc(Oc2ccc(F)cc2)n[nH]1)c1ccc(CCC)cc1 C(c1cccc(OC)c1)=CC(=O)NC(CNC(C1CCC(CC)C1)=O)CCC c1(OC)ccc(-c2nc(-c3ccccc3)nn2CCC(C)C)cc1C N1(C(C(N2CCC(C)C2)=O)=O)CCC(CNC(=O)CN2CCCCCC2)CC1 c1(C(N(CC(C)N(C(c2cc(CCOC)on2)=O)C)C)=O)c(C)cc(C)nc1O Clc1ccc(-c2nc(CC3C=CCC3)n(C3CCCOC3)n2)nc1 Cc1cc(C)c(C#N)c(NCC2CCN(C(c3n[nH]c4c3CCSC4)=O)C2)n1 c1(C(=O)NCC2(NC(CC(C)CN(C)C)=O)CCCC2)cc2cn[nH]c2cn1 C12(C(=O)NC3CC(CCNC(c4n(CC)ccc4)=O)C3)CCC(F)(CC1)CC2 c1(CC(=O)NC2C(CNC(CCc3cnc(C)o3)=O)CC2)cc(F)ccc1Cl C1(C(=O)NCCN(CC(C)O)C(c2c(C)nc(CCC)o2)=O)CCC(C#N)CC1 C1(C(F)(F)F)(OC)CCOCC1.C12CC(CN1C(C1CC(F)(F)C1)=O)COC2=O C1(=CC(=O)N(CCCNC(c2[nH]c(=N)ccc2C)=O)CC)CN2CCC1CC2 N1(C(C2(C#C)CCCC2)C(=O)NCCCOC)CCOC2(CCSC2)C1 N1(C(C(CCC)OC)=O)CC2CC(C1)CN(C(c1cccc(C(F)F)c1)=O)C2 C(C)(C(O)C(=O)N(C)CCN(C(=O)CN(C1CCCC1)C)C)OC C(C(C(C)C)C(C)C)N.n1(CC)nncc1-c1ncno1 c1(C(C(=O)NCC2CC2)N(C(C(C)SC)C)C)csc(C(C)(C)C)n1 C(=O)(CC1=CCOCC1)NCCN(c1ccc(Cl)nc1)C(CC1C(C)OCC1)=O N1(C(CCCC(C)C)=O)C2CCCC1CN(C(C1CS(=O)(=O)CCO1)=O)C2 Cc1cc(CC(N2CC(NC(c3ccn(C(C)C)c3C)=O)C(C)C2)=O)ccc1Cl c1(OC)ccccc1CCC(=O)NCC(N1CC(CNC(=O)C(C)C)CC1C)=O CCC(CC)C(c1cccs1)NC(c1cn(CC(=O)OC)nc1-c1cccs1)=O c1(C(=O)NCCN(CC(C)O)C(C2CN(C)C2)=O)ccc2occc2c1 [N-]=[N+]=NCCCCC(=O)NCCCCNC(c1ccccc1C(F)F)=O N1(C(C2(NC(C)=O)CCC2)=O)CC(C(=O)Nc2sccc2CC#N)C2(CC2)C1 N1(C(c2nc(OCC)oc2)=O)C2CCC1C(NC(=O)C(O)C1CCC1)C2 CC(C)C(C)(CNC(=O)CC(c1cccc(F)c1)O)NC(=O)C(C)SC(F)(F)F c1(CN2CC(CNC(c3nn(C)c(O)c3)=O)OCC2)cc(C(F)(F)F)cc(O)c1 N1(C(C2CC(C(=O)OCC)C2)=O)CCC(N(C(=O)CC2CCCC(C)C2)C)CC1 c1(C(N2CC(NC(c3ccc(C4CCCO4)[nH]3)=O)(CO)C2)=O)ccc2c(c1)COC2 c1(NC)ccc(C(N2CC=CC(NC(=O)Cc3cc(C)[nH]n3)C2)=O)cc1F C(CCC(=O)NOC(C)(C)C(=O)O)NC(C(COC(C)(C)C)N)=O C1(CNC(C2(CC=C)CC=CC2)=O)(COC)CCN(C(=O)CCNC(N)=O)C1 c1(CC)nc(C(=O)NCC2C=CCN2C(c2cnn(CC3CC3)c2)=O)c(C)o1 c1(C(N(C2CC(NC(C34CCCN(CCC3)C4)=O)C2)C)=O)cc2sc(Cl)cc2s1 c1(C2C(C(=O)NCC3(C(=O)OC)CC3)C2)ccccc1N1CCC(N)C1 C1(CNC2C3(C(=O)OC)CCC(C2)C3(C)C)CCC2(CCC23OCCO3)O1 N1(C(N(C2CCCC2Cc2ccc(F)cc2)CC(N)=O)=O)C2COCC1CC(F)C2 c1(CC(=O)NC2C(C)N(C(=O)C=Cc3nccs3)CC2)ccc(C#N)nc1 c1(C(=O)NCC2(C)CN(c3cc(SC)ncn3)C2)c(Cl)ccnc1Cl CCCCCCOCC(=O)NCCOCCN(C)C(C1CSCCS1)=O CC1CCC(NC(c2ccc(C(F)F)cc2)=O)CN1C(=O)C(F)C1CC1 C1(NC(CN2CC(=O)NC2=O)=O)CCN(C(C2CC2(Cl)Cl)=O)C12CC2 c1(OC)cnccc1CN1CC(NC(c2ccc(CO)o2)=O)C1 C1(NC(C(C)(CO)NC(C)=O)=O)CC2(C1)CN(C(=O)Cc1ccsc1)C2 c1(NC(C(CNC(c2c(OC)cnnc2)=O)OC)=O)cc(C)cnc1O Cc1cc(CNCC2CCCN2C(=O)C(c2cccnc2)O)cc(Br)c1 N1(C(C(C(CC)CC)F)=O)CCC2CN(C(C3CCCN3C)=O)C(C)C12 c1(CC)[nH]nc(C=O)c1C.C12(CC(C)(C)C1)N1CCC(C1)OCCNC2=O.COC N1(CCNC(CC2CC(CC)OCC2)=O)CCCN(C(c2nncs2)=O)CC1 Nc1cc(C(=O)NC2CC3C(NC(=O)CCCc4ccsc4)C3C2)ccc1Cl CC(CC(C)NC(c1ccnnc1Cl)=O)N=c1nc[nH]s1 C1(CC(N2CC(C(C)(C)C)C2)=O)(OC)CN(C(=O)CCCN(C)C)C1 C1(C(=O)NC(CC2CC2)CO)(CSC)CN(C(=O)C(C)c2cncs2)C1 CC(C)CC(CNC(c1ccc(NC(=O)C(C)N2CCC2)cc1)=O)N(C)C c1(C(=O)NCC2OCCN(C(CCNC(=O)OC)=O)C2)coc2ccccc12 c1cc(NCC2CN(Cc3cccs3)CCCO2)n2nccc2c1 CC1CC(c2ccc(F)cc2)CCN1C(C(=O)NC1CC1)C1CC1(Br)Br C=CC(C)(O)CC(=O)N1CC2(CNC(=O)CCCC3(C)CC3)CC1CO2 N1(C(COc2cn(C)nc2)=O)CCC(=CCNC(C2CC3CCC2C3)=O)CC1 n1(Cc2cccc(CC(=O)N(CC(CN(C)CC)O)C)c2)ccc2ccccc12 c1(OC)ccc(-c2cn(C3CC(C(N4CCSCC4(C)C)=O)C3)nn2)c(F)c1 c1(C(=O)NC(C2CCOCC2)C(=O)OCC)ccc(C(F)(F)F)cn1 Cc1cncc(C(N2CCC(N(CCC(C)C)C(C3CCN(C)C3C)=O)CC2)=O)n1 C1(C2CCN(C(c3cc(CSC(F)(F)F)c[nH]3)=O)CC2)(NC(C=CC)=O)CC1 c1(C(=O)NCC(C)NC(C2COCCN2C)=O)noc2ncccc12 Cc1cncnc1C(N1CC(F)CC1C(=O)NCCN1CCCCC1C)=O c1(C(C)=O)cnc(N2CCCC(NC(c3ccc(Cl)cc3Cl)=O)C2)c(C)c1 N=c1[nH]c2ncc(C(=O)NC3CCC3NC(c3cnn4c3CCCC4)=O)cc2s1 C1(C(c2n(CC=C)nnn2)NC2CC23CC(OCC)C3)C2CCCCCC12 CCC(CC)CCCC(=O)N1CC(CNC(c2nc(Cl)ccc2N)=O)C(SC)C1 Cc1c(Cl)ccc(F)c1C(=O)NCCS(=O)(=O)CC1CC1 CC1(NC(=O)CC2CCC(O)C2)CCN(C(=O)CCc2ccc(O)nc2)C1 C1(NC(N(C2CCSC2)C)=O)C=COCC1.C(CSC)O c1(C(C(=O)O)NC(c2nnc(C3CCCCC3)s2)CC)ccc(C)cc1F CC(C)(CNC(c1c[nH]nc1Br)=O)CCNC(C1CCCC1CF)=O c1(C(N(CCCCN(C(=O)CCC2CC2)C)C)=O)c(F)ccc(F)c1N C(=O)(CCN=[N+]=[N-])NCCSCC(=O)NC(CCC)c1ccco1 c1(CC)cccc(NC(c2cc(C3CCC(=O)N3)ccc2Cl)=O)c1C C1(NC(C2C(C)=C2)=O)CCCCC12CCN(C(=O)C1CCCc3ccnn31)CC2 c1(OC)cc(C)cc(C(=O)NCC2CCCCN(C(=O)Cc3cnsc3)C2)c1C CN1CC(CNC(N2CCN(CCO)C(=O)CC2)=O)CCC(O)C1 c1(C(N(C)CC2CCCCN2C(C2(O)CC2)=O)=O)cccc2c3c([nH]c12)CCC3 C1(COC)(CNC(c2ccc(C3CC3)cc2)=O)CCN(C(=O)CC2(C)CC2(F)Cl)C1 c1(C=O)c[nH]nc1[N+](=O)[O-].N1(N(C(=O)CC(C)(F)F)C)CC(NC)C(F)C1 N1(C(CC(CC)SC)=O)CCN(C(=O)CCc2nnc(O)n2C)CC(O)C1 c1(C(N2CC(CNC(c3ncc(CC)nc3)=O)(OC)C2)=O)ccc(=O)n(CC)n1 C(C(C)(O)C(=O)NC(C)CC(C)NC(=O)C(F)(F)Oc1ccc(F)cc1)OC c1(C(=O)NCC2N(C(C(CCCC)CC)=O)CC2)cccn2c(Br)cnc12 N1(C(Cc2c(C)non2)=O)CCOC(C(=O)NCC(Cl)Cl)C1 c1(CC)noc(CN(C(c2ncnn2C)C(=O)NCCOCC2CC2)C)n1 N1(C(C2=CCC(NC(CSC(C)(C)C)=O)C2)=O)CCn2nccc2C1 C(=O)(C1CCCc2n[nH]cc21)NCC1=CCN(C(c2c(N)c(C)n(C)n2)=O)CC1 N1(C(C(=O)NC)CC2CC2(F)F)CCCCC1CCNC(C)=O c1(C(=O)NC2CCC(CCNC(c3c(C)occ3)=O)C2)cccc(F)c1C C1(C(N(CC(C)CNC(C2(CO)CC(F)(F)C2)=O)C)=O)CCn2nncc2C1 C(=O)(C(F)(F)C(C)(C)O)NCC=C1CCN(C(c2cnc(CC(C)C)s2)=O)CC1 c1(CN(CCc2nnc(C)s2)C)ccc2c(c1)CCOC2 N1(C(=O)Nc2c(OCCCC#C)cccc2)CCNC(=O)CC1C C1(C(=O)NCC(CNC(Cc2c(C)n[nH]c2)=O)(C)O)(C(=O)O)CC12CCC2 Cc1cn(C)nc1C(=O)NC(C)(CNC(C1(c2ccc(Cl)cc2)CCC1)=O)CO C1(C(N(CCOC)C(C)C)=O)CC(=O)N(c2cc(C)no2)C1c1cncn1C N1(C(CCCCSC)=O)CCCC2(C1)CN(C(c1coc(Cl)c1)=O)CCO2 C1(C(=O)NC(CC)C(=O)N2CCC2C)CC2(CCC2=O)C1 Cc1ccc2oc(CNC(=O)NC3CCNC3=O)c(C)c2c1 Cc1sc(S(N)(=O)=O)cc1C(N1CC(C)N(C(=O)CC(C)(C)N(C)C)CC1C)=O C1(C(=O)NC(Cn2cc(CN(CCOC)C)nn2)C)CC2(CO1)CC(F)(F)C2 C1(NC(C(CCSC)(C)C)=O)CCC(O)CN(C(=O)Cc2ncc(C)o2)C1 C(=O)(N1OC2C=CC1CC2)C1CCN(C(c2ccc(C)nn2)=O)C1(C)C Cc1csc(C(C)C(N2CCCC2CCCNC(=O)COC2CCC2)=O)n1 S(=O)(=O)(c1ccc(C(=O)NC2CC(CCNC(C3CCNC3=O)=O)C2)o1)NC C1(C(=O)NCCCN(C(=O)C2=CCCCC2C)C(C)C)CN2CCCN1CC2 C1(C)(C(N(C2CCN(C(c3sccc3Cl)=O)C2)C)=O)CCCS1(=O)=O C1(NC(CNS(CC)(=O)=O)=O)CC2CCCC(C1)N2C(c1ccc(OC)nc1)=O C1(O)(C(N)=O)CCN(C(C2(NC(=O)CCc3ccc[nH]3)CCSC2)=O)C1 CC1Cc2ccccc2N1C(N1CCN(CCF)CC1)=O.c12cccc(c1)NC2=O N1(C(CC=CC=C)=O)CCCC(N(C(=O)CC2CCCOC2)CCO)C1 c1(C(=O)NC2(CNC(Cc3n(C)cnc3)=O)CCOC2)cc(C#N)ccc1Cl c1(C(=O)NCCC(C)N(C)C(c2sccc2CC#N)=O)cncc(F)c1 N(C1CCc2cccnc21)C(CC1(N(C(C(C)C(F)(F)F)=O)C)CC1)=O C1(CNC(c2c(C)cno2)=O)CCCN(C(c2nc(Cl)sc2Cl)=O)CC1 c1(C(N(CC(C)NC(C2(CC)CCOC2)=O)C)=O)ccc(C(C)=O)cn1 c1(OC)ccc(F)cc1C(N1CCC(F)C(NCc2sccc2C(=O)O)C1)=O C(=O)(C1=NN(CCO)C(=O)CC1)NCC1C2CN(c3cc(C)nc(C)n3)CC21 c1(C2CN(CC3N(CC(F)(F)F)CCC3)C2)nnc2n1CCOC2 C(C(=O)NCCc1cn[nH]c1)(C1CN(C(=O)CN(C)C(C)C2CC2)C1)OC C1(NC(N2C(C(C3OCCCO3)=O)CCCC2)=O)C(F)(F)C12CCC2 C1(CNC(C2C(C)C2)=O)CCC(NC(c2ccc(C(F)(F)F)s2)=O)CC1 N1(C(c2cc(C)no2)=O)CCN(C(C2CCC(=O)N2C2CC2)=O)CC1C(C)C c1(C(=O)NC2C(C)CN(C(C3(F)CC3)=O)CC2)cc(Cl)cc([N+](=O)[O-])c1O N1(C(C(C(CC)C)O)=O)CC(C2CN(C(c3cnc4[nH]ccc4c3)=O)C2)C1 C1(C(=O)NCC23C(CN(C(CSCCC#N)=O)C2)C3)Cc2nccn2C1 C(=O)(C(C)(C)C(F)F)NC1C(C(=O)NCc2c(C)ccnc2)COCC1 C1(CC)(CC)CCCN(C(C2CCN(C(=O)CCc3cc(C)[nH]n3)C(C)C2)=O)C1 N1(C(C2(CCCC)CC2)=O)CC2(C(N3CCN(C(=O)C(C)C)CC3)=O)CC1CO2 c1(C(N(CC(O)CNC(C2(C)CCOC2)=O)C)=O)cc2c([nH]1)CCCC2 c1(C(N2C(C(NOCC(=C)Cl)=O)C(CC)CCC2)=O)cccc2occc12 CCN=c1[nH]c(C(=O)N(CCC(C)NC(=O)CC2COCCN2C)C)cs1 C(=O)(C1=CC2(CN(C(c3ccc(C)cc3)=O)C2)OC1)NCC(CCCC)CC C1(CC(=O)NC(C(=O)N(C(C)C)CC2CC2)Cn2cccn2)CC(=O)NC1=O C1(N(CCC)C(c2cscc2Cl)=O)CCN(C(C2(C)CCCN2C)=O)CC1 C1(NC(C2CCCO2)=O)CC2CC(C1)N(C(C1(O)CCCCC1)=O)C2 C(C(C)CN=c1cc(C(F)F)nc[nH]1)NC(c1c(OCC=C)cccc1)=O N1(C(c2nc(COC)oc2)=O)CC2(CC(C(=O)NC3(C(C)O)CC3)CO2)C1 c1(C(=O)NCCC2(NC(=O)CC3CC4CCC3C4)CC2)csc2cc(Cl)ccc12 C(=O)CC(C)P(C)(C)=O.CC(C)C(CNCC(F)(F)F)OCCSCC CC(C)(C)CC(C)(C)C(=O)NC(C)CCCn1ccnc1 c1(C(N2CCN(C(C(C(=O)OC)OC)=O)CC2CCO)=O)ccn2cnnc2c1 N1(C(c2cc(C3CC3)ncn2)=O)CCN(C(=O)CC2CCCC2)C2CC12 Cc1ccc(C(=O)NC2CC2NC(=O)C(c2ccc(Cl)nc2)(F)F)cc1N c1(C(=O)NCC2C=CCN2C(=O)COc2ccc(Cl)cn2)cccc(C2CC2)c1 C(c1ccc(F)c(OC)c1)=CC(=O)NCC(CCCC)NC(c1cc(Cl)no1)=O c1(C(N2C(CN(C(c3c(C)occ3)=O)C3CC3)CCC2)=O)ccnc(CO)c1 CC1CC(CCNC(C2CC3(C2)CC3(F)F)=O)CCN1C(c1snc(O)c1Cl)=O c12cccnc1CSC1C(CCC1)C(=O)NCC(=C)CCNC2=O.SCC C(=O)(CCC(CF)CF)NCC1N(C(c2nc(COC)sc2)=O)CCCC1 c1(-c2nc(Cc3ccccc3)nn2-c2ccncc2)cn2c(n1)COCC2 C1(NC(C(C)=C2CCC2)=O)CCCOC1C1CCN(C(=O)C=C2CCCC2)CC1 N1(C(COCCCN(C)C)=O)CCCC(NC(=O)CC2C=CCCC2)C1 c1(CC)cnc(OC)c(C(N2CC(CO)(NC(C3CCCC(C)CC3)=O)C2)=O)c1 N1(C(c2ccc(C)s2)=O)CC(NC(=O)C#CC(C)C)C(C(F)(F)F)C1 c1(C(N(C2CCN(C(=O)CC3CC(n4cnnc4)C3)C2)C)=O)ccc([N+](=O)[O-])o1 N1(C(CC2CC(NC(c3nc(C)sc3C)=O)C2)=O)CCCC(O)C1C Cc1ccc(N2CCN(C(=O)Nc3ccncc3-c3ccc(N)cc3)CC2)cc1 C1(C(=O)NCC(CC(=O)OC)O)N(C(c2ccc(C#N)s2)=O)CCCC1(C)C C1(CNC(C2(O)CCC(C)CC2)=O)CC2(CO1)CN(C(=O)CC1CCSCC1)C2 C1(OC)CN(C(=O)C(c2c(C)noc2C)C)CC1NC(=O)CN1CCOC1=O CON=Cc1ccc(C(N2CCC(N(C(C3COC(=O)C3)=O)CC)CC2)=O)cc1 N1(C(c2c(C)ccnn2)=O)CCC=C(C(=O)NCC(C)(C)C(C)O)C1 N1(C(c2c(C)con2)=O)CCCCC1CCN(C)C(c1c(Cl)nsc1Cl)=O C1(C(=O)NCC(C#C)OC)CCN(C(=O)c2c(C)cccc2C)O1 c1(C(C)=O)ccc(Br)cc1NC(C1CN(C(c2ccc(C)c(C)c2)=O)C1)=O C1(CNC(c2c(C)nc(C)[nH]2)=O)CCN(C(=O)Cc2cc(Cl)n(C)n2)C12CC2 c1(C(N2CCC(NC(C(CC(=C)C)NC(C)=O)=O)C2C)=O)ccc(C)c(C)c1N C(CCO)(C(=O)NC1CCCN(C(=O)CCc2nc(O)n[nH]2)C1)N(C)C C=CCC(C(=O)NC1(C(=O)NCCN2CC3CC3C2)CCCCC1)NC(C)=O C(CNC(=O)C(C)(O)C1CCC1)(CC(=O)NC1COCCCC1)OC C1(NC(C(C)=C2CCC2)=O)CCC2CN(C(C3CCc4nn[nH]c4C3)=O)CC12 c1(OC)ccc2[nH]c(C(=O)NCC3CCN3C(=O)C(C(C)(C)C)OC)cc2c1 Cc1cnn2cc(C(=O)NCC3(O)CC(NC(C4CCN(C)C4=O)=O)C3)cnc12 c1(C(=O)NCc2cccc(NC(CC(C=C)C)=O)c2)nc2cccnc2s1 C1(CC(=O)NC(CCC)C(=O)N(C)C)N(C(=O)CN2CCNC2=O)CCC1(C)C C1(OC)CC2CC(C(=O)NC(C)(C)CNC(c3cnn4c3OCC4)=O)CC12 C(=O)(C1CCOc2c(F)cccc21)NC(CNC(=O)CN1CCC(O)CC1)(C)C N1(C(C=C(C)C(C)C)=O)CCOC(CCCNC(=O)C2=CCSC2)C1 c1(C(=O)NC(C(C)C)C(=O)N(C2CCC3(CC2)CC3)C)cccc(F)c1F C(C(CC(C)C)C(=O)N1CCC2(CCO2)C1)NC(C=CC(CC)C)=O N1(C(C(C)=C(CC)C)=O)CCN(C(C2(C)CCOCC2)=O)C(C2CCC2)C1 C1(C(N2C(C(=O)NC(c3cccnc3)C3CC3)CC(O)C2)=O)CCC(F)(F)CC1 C1(C(=O)NCCCN(C(c2ccc(C(=O)OC)o2)=O)CC)(C(F)F)CCC(=O)N1 c1(C2(NC(C)(CCI)c3nnnn3-c3ccc(F)cc3)CC2)cc(F)cc(F)c1F C(=O)(C1=CCCOCC1)NC1CC(C)(NC(c2c(C)cc(O)cc2)=O)C1 C12(NC(C3CC=CCC3)=O)CCCC1CN(C(c1ccc(F)s1)=O)C2 C1(NC(=O)NC2CCN(c3cnc4n3CCCC4)C2)CC2(CN1)CC2(F)F c1(CN2CCN(C(C3CCN(C(C)=O)CC3)=O)CC2)cn2cc(Br)ccc2n1 C(C(=O)NC1COCC1NC(=O)CCc1ccc(Cl)nc1)(C(C)C)SC c1(OC)cc(N2CCCCC2)ccc1C(=O)NC(C1OCCOC1(C)C)C N1(C(CC=CCC)=O)CC2(CC(NC(=O)C=CC=C(Cl)Cl)CO2)C1 c1(-c2nn(-c3cn(C)nc3)c(CCOc3ccccc3)n2)ccc2c(c1)OCC2 C1(OC)CC(N(C)C)N(C(=O)NC(c2cncs2)C)C1.N12CCCC1C2 c1(C(N2CCC(O)(CN(C(CC(CC)(F)F)=O)C)C2)=O)ccn2cncc2c1 C1(NC(CC(CNC(C(COC)(C)O)=O)C)=O)CCC12CCCC2 c1(C(N(C)CC2CCCCN2C(c2ncc(F)cn2)=O)=O)cc(O)nc(O)n1 C1(C(=O)NCC(COC)NC(=O)C(c2c(C)noc2C)C)(COC)CCOCC1 C(C(C)(O)C(=O)N(C(C)CNC(c1cc(C(c2ccccc2)C)[nH]n1)=O)C)OC C1(C(=O)NCC#CCNC(c2ccc(O)cn2)=O)CCc2ncncc2C1 c1(C(N2CCCCC(CNC(C(C(=C)Cl)(C)C)=O)C2)=O)ccc2c(c1)NCCC2 N1(C(CCC(C)(C)OC)=O)CC2CCCC2(CNC(c2cncc(O)c2Cl)=O)C1 C12(C(=O)NC(CN(C)C(c3ccc[n+]([O-])c3)=O)(C)C)CC1CCC2(F)F C1(C(=O)NCC(C)N(C(=O)Cc2cc(C3CC3)on2)C)CC12CC(C)(C)C2 CCCC#CC(C)(C)NC(=O)CC(C)(C)NC(=O)CC1CCC(=O)N1C CC1CN(C(c2ccc(O)nc2)=O)CCN1C(c1cccc(N2CCCC2)c1)=O c1(C(=O)NCC(CC)NC(c2ccc3nonc3c2)=O)cccc2oc(=N)[nH]c12 C1(NC(C(C2CCOCC2)C)=O)CCN(C(c2n[nH]cc2Br)=O)C12CC2 c1(C(=O)NCC(CNC(c2c(CC)n[nH]c2)=O)F)cn2cccc(F)c2n1 c1(CC(C)NC(CC2(N(C)C(c3ccc[nH]3)=O)CC2)=O)cnccn1 C1(CNC(c2cn(CCNC(C3CC(OC4CC4)C3)=O)nn2)=O)CC12CCOC2 C1(C(=O)NC(C(=O)NCC)(C)C)(CO)CCN(C(=O)CC2CCOC2)C1 c1(C(=O)NCC2C(NC(C(CCOC)(C)C)=O)CCC2)ccc(Cl)c(F)c1F C(C)(CCC(=O)NC(CNC(=O)CC1CCN(C)C1=O)CO)OCC N1(C(Cc2cc(C)c(O)cc2)=O)CC2(C(N3CCS(=O)(=O)CC3)=O)CCC1CC2 C(=O)(C(O)C(F)(F)F)NCC(C)N(C(=O)C(C1(O)CCC1)Nc1ccncc1)C C(CCCC(=O)N1CC2CC2(CNC(=O)Cc2cncs2)C1)NC(N)=O c1(CC(C)C(C2CC2(F)Cl)=O)nccn1C.C12(CC(O)C1)C(=O)NCC2 c1(C(N2CC(CNC(c3ccc(COC)s3)=O)C2)=O)cnc(OC(F)F)c(C)c1 CC12CC(C1NC(=O)Cc1ccc(F)cc1Br)N(C(=O)CC1(CO)CC1)C2 CN1CCN(C)CC1.N1(C(=O)OC)CCCCC1C1COC1 c1(CC(=O)NCC=C2CCN(c3nnc(C4CC4)s3)CC2)n[nH]c2c1COCC2 C(=O)(C(C1CCCO1)NC(C1CCC1C)=O)NCCN(C(C)C)CC c1(OC)ccc(C)c(NC(=O)CC2(OC)CN(C(c3ccnc(C)c3N)=O)C2)c1 N1(C(C=CC)=O)CCOC(Cn2cc(-c3cnoc3)nn2)C1 c1(OC)ccc(-c2nc(-c3ccc(OC)c(CSC)c3)no2)cc1-c1nnc(C)o1 C1(NC(c2ccn(CC(F)F)n2)=O)COCC1NC(c1cocn1)=O C(CC(C(=O)N(C)CCc1ccncc1)NC(=O)Cn1nccc1C)OC C(=O)(C(C)(CC)CC)N1CCC(CC=C)(C(=O)NCc2cc(CC(C)C)[nH]n2)C1 Cc1cc2c(cc1C)OC(C(=O)NCC1CN(C(c3ccc(Cl)o3)C)CCO1)C2 c1(SCC(N2CCC(C(c3cccs3)N(C)C)C2)=O)ccc(F)cc1 c1(OC)nc(C)ncc1C(N1CCCC(C(C)NC(=O)Cc2cc(C)on2)C1)=O C1(NC(CCC2N(C(C3CNC(=O)N3)=O)CCC2)=O)CCCCC12CCC2 c1(CNC(C2C3CN(C(Cc4c(C)nc(C)s4)=O)CC32)=O)ccc(F)c(C)c1 N1(C(C(CC)Nc2cccnc2Cl)=O)CCCC(C2CN(C(c3cnn[nH]3)=O)C2)C1 C1(C(=O)NC(CNC(CCC#C)=O)C)CS(=O)(=O)CC12CCC2 N1(C(C)=O)CCCC(C2CN(C(=O)C(c3cccnc3)O)C2)C1 c1(C(=O)NCC2CCC(NC(c3cnncc3O)=O)C2)ccc2cnccc2n1 c1(C(N(C(C)CN(C(=O)CC23COC(C)(C2)C3)C)C)=O)cnc2nccnc2c1 C(CC(F)F)(C(=O)Nc1cccc(F)c1)NC(Cn1ccc(C)c1)=O C1(CN(C(=O)CNC(=O)Cn2cncn2)C)CC(F)CN1C(=O)Cc1ccsn1 C#Cc1cc(NC(=O)CC(C)(C)c2ccccc2)cc(C(=O)O)c1 C(=O)(C(CNC(c1ccn(C)n1)=O)N(C)C)NC(C(=O)OCC)C1CC1 C1(NC(C2(C)CCOCC2)=O)CS(=O)(=O)CC1NC(c1ccnn1C(C)(C)C)=O c1(C(=O)NCC2(CNC(=O)CN3CCCCCC3)CC2)n[nH]c2c1C(=O)CCC2 N1(C(C(C)(C)c2ccsc2)=O)CCc2[nH]nc(CNC(C34CC5CC3C4C5)=O)c2C1 CC(C)CC(C(=O)NCCCN(C(C1CCCCC1)=O)C(C)C)NC(N)=O c1(COC)nc(C)cc(=NCCC(C)NC(C2OCCC2(C)C)=O)[nH]1 N1(C(C(SC)SC)=O)CCN(C2CN(C(C3CCC=CCC3)=O)C2)C(=O)C1 C1(C(=O)NCc2c(C)ccs2)CC(F)CN(C(c2nc[nH]n2)=O)C1 Cc1ccsc1CC(=O)NC(C)(C)CC=CC(=O)NC1(C(C)C)CC1 C(=O)(C(C(C)(C)C)NS(C)(=O)=O)NCC1CN(C(c2cnn(CCC)c2Cl)=O)C1 C1(NC(c2ccc(CNC(c3cc(C)c(F)cn3)=O)cc2)=O)CCN2CCCC2C1 C(C)(N=c1ccc(Br)c(S(=O)(=O)NC2(C(C)(C)C)CCC2)[nH]1)c1cn(CC)nn1 c1(CC)ccc(C(CNC(C2CC3CCC2C3)=O)N(C)Cc2cnn(C)c2)cc1 C1(O)(CN(C)C(C2CCC(N(C)C)CC2)=O)CCN(C(=O)CN2CCC(C)(O)C2)C1 c1(C(=O)NCC2C(NC(C(c3ccn(C)n3)(C)C)=O)C2)cc(Cl)cn1C C1(NC(c2c(C)cc(C)s2)=O)CCN(C(=O)C(C)(C)N2CCOCC2)CC1F C1(NC(c2ccc(SC)cc2)=O)CC2CCC(C1)C2NC(c1cccc(=O)o1)=O Cc1cc2ncn(CC(=O)NCC(F)CNC(=O)C(F)(F)C(C)O)c2cc1C C(CC1=CCN(C(c2ncoc2C2CC2)=O)CC1)NC(Cc1cc(CC)no1)=O C1(NC(C(CC)CC)=O)C2CCN(C(c3csc4sccc34)=O)CCC12 c1(C(N2CCC3(C(NC(CCNC(N)=O)=O)C3)C2)=O)ccc2cnnn2c1 C1(NC(C2N(C(CCC)=O)CCC2)=O)CCN(C(c2ccccc2)=O)C1C Cc1noc(C)c1C(C)C(=O)NCC1CCCN(C(c2snnc2C(C)C)=O)C1 c1(C(=O)NCC(C)NC(=O)C(c2ccc(F)cc2)(C)F)ccc(O)nc1Cl c1(C(=O)NC(C)C(C)NC(=O)CCCn2ccnn2)ccc([N+](=O)[O-])[nH]1 c1(C(N(C2CCN(C(=O)Cc3cnc[nH]3)CC2)CC#C)=O)nc(C)oc1C C(=O)(C(C)(C)n1cc(Br)cn1)NC1C(CN(C(C2CN(C)C2)=O)CC2CCC2)C1 C1(C(=O)NCC2N(C(C(C3CCOC3)OCC)=O)CCCC2)CCC(C#N)CC1 O=C(C1=C(Cl)CCC1)NC12CC(C(N3CCC(c4ncco4)C3)=O)(C1)C2 C1(NC(c2ccc(F)cc2F)=O)CC2CC1CN2C(=O)C(F)(F)CC1CCC1 c1(C(=O)NCCC(C(=O)NCC(n2ccnn2)C)OC)cc(O)ncc1F N1(C(N(C(c2ccccc2)C)C)=O)CCC=C(Cl)C1 C(N=c1[nH]c(N(C)Cc2cnn(C)c2C)nc2ccc(Cl)cc12)c1ccc(C)s1 C1(NC(c2n(CC)ncn2)=O)CN(C(=O)CN2CC(C)C2)C2(CCOC2)C1 c1(Cn2ncc(OC)c2)nn(C)c(C(N2C3CCC2C(C(=O)OCC)C3)=O)c1Cl C1(C(=O)NCCN(C(C2(C)CCC(C)CC2)=O)CC2CC2)CCC2C(C1)C2(F)F CC(CN(C(=O)CC(C)(C)C)C)C(=O)NNC(=O)C(C)(C)CCCCOC(C)=O Cc1nc2cncc(-n3cc(C4CCN(C(=O)CN(C)C)C4)nn3)n2n1 N1(C(CCC(=O)Nc2c(OC)cc(Br)cc2)=O)CC2CCCCC2C1 C(=O)(C1=CC(O)C(NC(=O)C(c2ccccc2)F)C1)NC1(C(N)=O)CCC1 C1(NC(C(N2CC(C)CC(CC(=O)O)C2)c2ccco2)=O)CC2CCCCN2C1.CC C1(CNC(CCSCCC)=O)CC2(CCC2)CN1C(c1n[nH]cc1OC)=O C1(C(N2CC(n3cc(CCCCC)nn3)C(C)C2)=O)Cc2ccncc2N1 c1(OC)cc([N+](=O)[O-])c(C(N2CCCCC2C)=O)cc1OC Cc1ccc2nc(C)cc(C(=O)NCCC(C)NC(=O)Cc3cnc(C)s3)c2c1 C1(c2onc(-c3n(C)c4c(n3)cccc4)n2)CC12CCc1ccccc12 N1(C(CC(C2CC2)NC(N)=O)=O)CCC(C2CCN(C(c3ccnnc3)=O)C2)C1 C1(CC(=O)N(CCCC)C)CN(C(=O)C(C)CCN(C)C)CC1C C=CCC(C)C(=O)N1CC2C(CNC(c3nnsc3C(F)F)=O)C2C1 c1(C(=O)NCCN(C(=O)C2=CS(=O)(=O)CCC2)CCC)cnn2ccnc(N)c12 c1(C(N2C(CN(C(C3C(C)OCCO3)=O)C)CCC2)=O)ccc(F)c(Cl)c1 C1(Sc2ccnn2C=C)CC2CCCC(C1)N2CC#C.C1(C)(C)C(=O)N1 CCCCC(O)CC(=O)NC1(CO)CCN(C(c2cn(C(F)F)c(C)n2)=O)C1 C1(NC(C2C(C(C)(C)C)CC2)=O)CCCN(c2ccccc2)C1 c1(-n2ncc(-c3nc(C(C)OCC)nn3CC(F)F)n2)ccc(F)cc1F c1(C(=O)NCC2C(CCC)CCCC2)nc2ccncc2[nH]1 CCCCCCCCCCCC(O)C(=O)N1CC(C2CN(C(=O)C(C)CC)C2)C1 c1(CCCC(N2CCN(Cc3c(C)noc3C)CC2C)=O)ccc2[nH]ccc2c1 Cc1oc(C(=O)NC2C3CCN(C(=O)C=Cc4cnc[nH]4)C23)cc1Br c1(C(=O)NC(C(=O)OCC2N(CC)CC2)COC(C)C)cnn2ccccc12 c1(CC(=O)NC2CCC(CCNC(CC=C=C)=O)C2)coc2c(Cl)c(Cl)ccc12 N1(C(C2(C)CCC(F)(F)CC2)=O)CCC2(CCC2NC(C2CC2C2CC2)=O)CC1 C1(C(N2CC(NC(COCC(=O)NC)=O)C2)=O)COC2CCCCC12 c1(CC(=O)NC2CCN(C(C(C)(C)N3CCCCC3)=O)C2)cncc(C#N)c1 c1(C(N(C(CCNC(CCc2ccc(C)o2)=O)C)C)=O)cncc(P(C)(C)=O)c1 CC1(C)CCC=C(C(=O)NC2C3CN(C(c4nn[nH]c4Cl)=O)CC23)C1 Cc1nn(C)c(N)c1C(N1CC(C2CC2C(=O)NCCc2ccc(F)cc2)C1)=O N1(C(C2CC(=C)C2)=O)CCC(C2CC2NC(=O)Cn2nnc(C)c2C(F)F)CC1 c1(C(=O)NC(C(C)(C)C)CNC(C2CC3(CCOC3)C2)=O)[nH]nc([N+](=O)[O-])c1Cl S(=O)(=O)(c1cc(C#N)ccc1F)N1CCC2(N(S(CC)(=O)=O)CC2)CC1 C12(C(=O)NC3C(NC(c4ccccc4-c4cccnc4)=O)C3)COC(CCO1)C2 N1(C(C(COC(C)=O)C)=O)CC2CC(NC(=O)C(C)Cc3ccncc3)CC2C1 Cc1nocc1C(=O)NCC1(F)CC(NC(=O)CCN(C)CCO)C1 N#Cc1cccc(C(O)C(=O)N2CCC2C(=O)NCC2CC3CC2CC3O)c1 c1(C(N2CCCC(CNC(=O)CC3CCCCO3)CC2)=O)ccc(Br)c(Cl)c1F c1(OC)ccc(Cl)c(C)c1C(=O)N(CCCCNC(c1cc(Cl)no1)=O)C Cc1ccc(O)cc1C(N(C1CCN(C(C2CC2C2CCC2)=O)CC1)CCO)=O C(C(=O)NCC1CCCCN1C(c1cnns1)=O)(C(C)C)SCC Cc1nc2ncccc2cc1C(=O)NC1(C)CC(NC(=O)C(C(C)O)N(C)C)C1 C1(C(=O)NC(C)COCC2CC2)CCC(O)CN1C(c1ccc(C#N)s1)=O CC1(C)CCCC1NC(N1CC(CC(F)(F)F)C1)=O N1(C(CCC(=C)Br)=O)CC(C)CN(C(c2sccc2C)=O)CC1C c1(NC2C(C)(CC)C2)ncc(C)cc1S(=O)(=O)N(C)CCOCCOC C(=O)(CC(O)CNC(=O)CC1(C)OCCO1)NC(CN(CCCC)C)C C12(C(N3CCC(C)(CNC(=O)CCC(N)=O)CC3)=O)CC3CC(C(=O)N1)C2C3 C1(C(=O)NCC(CN(C)C)O)CC12CN(C(=O)Cc1ccccc1C(F)(F)F)C2 C1(C(=O)NCc2cccc(CC)c2)CC(F)(F)CN1C(C1C=CC(=O)N=N1)=O Cc1cc(NC(c2ccnn2CCF)=O)ccc1NCc1cnns1 C12CCCC(C1)OC2.c1(CC(=O)NC(CNC=O)C2CC2)csc(S)n1 CC1(C)C(NC(c2cnc(C(F)(F)F)[nH]2)c2nnnn2CCCF)C2CCOC12 C1(n2ncc(C(C(=O)NC(C)C)N(C(CC)C#N)CC)c2)CCS(=O)(=O)C1 C(C1CCc2ncnn21)N1CCCC(NC(C(C)OC(C)(C)C)=O)C1 Cc1ccc(Br)c(C(N2CCOC(C3CN(C(C4CCN(C)C4)=O)C3)C2)=O)c1 N1(C(C2(F)CCN(C(C(C)OCC(C)C)=O)C2)=O)CCC12CCCOCC2 C=CCC(C)(C)CC(=O)N1CC(NC(C2(C(=O)NCC)CC2)=O)CC1(C)COC N1(C(C(C2CCCN(C(CC=CC)=O)C2)(C)C)=O)CC(F)(F)CCC1C C1(NC(C(c2cc(C)sc2)(F)F)=O)CN(C(c2cccnc2CO)=O)CC1C N1(C(C2=C(C)OCC2)=O)CC(C)(C)OC2(C1)CN(C(c1nncn1C)=O)C2 c1(C(=O)OC)cc(C(=O)NCC2CC(NC(=O)CCOC)C2)c[nH]1 C1(F)(CNC(c2ccc(CN(C)C)o2)=O)CCN(C)C1 c1(C(=O)OCC)cnc(C(C)C)nc1N1CCC(NC(C2CC2(F)F)=O)C(C)C1 c1(NC(C2(NC3CC3)CC3CC3C2)=O)c(-c2ccccc2F)nc2ccccn12 C1(CC)CN(C(=O)C=Cc2nnn(C)n2)CCC1NC(=O)Cn1cc(C#N)cn1 C=CC(CCC)CC(=O)NCC1(C(=O)NC2CC(=O)N(c3cnn(C)c3)C2)CC1 C1(C(=O)NC(C(O)CO)C2CC2)(CO)CCN(C(=O)CC2CC3CC3C2)CC1 Cc1cc(C(=O)NCC(C2CCN(C(=O)CC3(O)CCC3)CC2)C)nc(O)c1 c1(C(N2CC3C(C(=O)NCCC4(C)CCOCC4)C3C2)=O)nc(Cl)ccc1N C12(C(N3CC(N(C)C(=O)NC4CCC45CCC5)C(O)C3)=O)CCC(C(F)F)(CC1)C2 N1(C(CC2(SSC)CC2)=O)CC(CO)C2(CCN(C(=O)C(C)(O)COC)CC2)C1 C(=O)(CCCC(F)(F)Br)N1CC(CC)C(NC(=O)CNC=O)CC1 Cc1nn(C)c(Cl)c1C(=O)N(C(CNC(=O)CN1CCCCCC1)C1CC1)C c1(C(=O)NCCN(C(c2c(C)c[nH]c2CC)=O)CC)ccnc2ncc(C)cc12 C(C(C(C)C)NC(c1cc(C(C)C)[nH]n1)=O)NC(CC1(OC)COC1)=O N1(C(CCCC)=O)CCC(OCCCNC(=O)C(C)n2cccn2)CC1 N1(C(C2(COC)CCC2)=O)CCN(C(=O)C(C)CSC(F)(F)F)CC1C1CC1 C(=O)(C1=COCCC1)N(CC(C)O)CCNC(=O)CC1CCCC1(F)F c1(C(=O)NC(C2CN(C(c3cc(Cl)c(Cl)n3C)=O)CCO2)C)cnn2cc[nH]c12 C1(=CC(=O)NC2CCC2Cc2ccccc2)CN2CCC1CC2 C1(NC(c2c(C)noc2C(F)(F)F)=O)CC2CC1N(C(c1cncn1C)=O)C2 c1(CN)c[nH]nc1C(=O)O.C(C=O)N(CCC)C.C1C(=O)N1C1CCC1 CC1(C(=O)NCC(CC(F)(F)F)NC(c2cnc(Cl)s2)=O)CCCC1(F)F N1(C(C=CCCC(C)C)=O)CCC(F)(C(N2CCCC2C(N)=O)=O)CC1 N1(C(CCSC)=O)CCC(NC(C23CC4CC2C3C4)=O)C(CO)CC1 C1(C(N2CC3(CCCN(C(CCC#N)=O)C3)C2)=O)CC(c2ccccn2)=NO1 c1(C(N2CC(C(=O)NCCNC(C3C(C)OCC3)=O)C2)=O)ccc2nc[nH]c2n1 C12(NC(=O)CSc3nc[nH]n3)CCC(O)(CC1)CC2 CC1CCCC(C)N(C(=O)C=CCC2(NC(=O)C3=COCC3)CCC2)C1 c1(CC)cc(OC)cc(C(=O)NC(c2ccc(C3CC3)cn2)=O)c1.C12CCC1C2 N1(C(C(CC(C)C)F)=O)CC2CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CC12 c1(O)ccc(-c2cnccn2)cn1.N12CCOCC1C2=O.CC(=O)NCCN CC1CN(C(=O)CSCC#N)CCN1C(c1ccsc1Cl)=O c1(C(=O)NC2CN(C(CNC(CNC(C)=O)=O)=O)C(C)C2)cccn2c(C)nnc12 CN1C(=O)NCC1C(=O)NCC1CCC(NC(=O)CCOC2CC2)C1 N1(C(C(C)(C)C)=O)CCN(C2CCCN(C(c3cccnc3C3CC3)=O)C2)CC1 N1(C(C(C)OC)=O)CC(NC(c2ccn(C(C)(C)C)n2)=O)C2(COC2)C1 C(=O)(C(F)C(F)(F)F)N(C)CC1(O)CN(C(C(C)COc2ccccc2)=O)C1 c1(C(N(C2CCN(C(=O)C=Cc3cncs3)CC2)C)=O)cc(O)cc(F)c1 CC1CC(C(=O)NC(C2(O)CN(C(=O)CC3CCCOC3)C2)C)CC(C)C1 C=C(C)CCC(=O)N1CCC(NC(=O)COc2ccccc2CC)C1CC N1(C(C2(CCC)CC2)=O)CC2CCCC2(NC(C2CCCC(C)(C)CC2)=O)C1 C#CC(C)(C)C(=O)NCC1CCC(NC(C2(N3CCOCC3)CCC2)=O)C1 C(=O)(CC1=CCOCC1)NC(C1CCCCC1)C(C)NC(=O)Cn1nnc(=N)[nH]1 C(=O)(C1=CNS(=O)(=O)N=C1C)N1CCC(OC)(CNC(C2(C)CCCOC2)=O)C1 CC1CN(C(=O)CC23CCC(C)(C2)OC3)CC(C)C1NC(=O)CSCCN(C)C CCC(C)C(C)C(=O)NCCCC1(NC(c2cnn(CCC#N)c2)=O)CC1 N1(C(COCCC=C)=O)CCc2sccc2C1C(=O)NCC(CNC(C)=O)OC c1(C(N)=O)cccc(C(=O)Nc2ccc(NC(C34C5CC3C3C4C5C3)=O)nc2)n1 C1(C(N(CCC2CCN(C(CC3CCC(C)O3)=O)CC2)C)=O)COCCC1(F)F c1(C(=O)NCC2C(F)(F)CCN(C(CCNC(C)=O)=O)C2)ccc(F)c2occc12 C12(C(N(CC(C)NC(=O)C=Cc3cncn3C)C)=O)CC(CO)(C1)OC21COC1 N1(C(COCC=C)=O)CCN(C(=O)C(C)C)CC1CCOC c1(N(C(C)=O)CC2CCN2Cc2ccccc2)c(C)cnc(Br)c1F C1(CNC(=O)Nc2nccc(C(C)(C)C)n2)CCc2ccccc2O1 c1(CN2C(CNC(COCCOC)=O)CCC2)cc([N+](=O)[O-])cc(OC)c1O c1(C(CC)C)ccc(C#N)c(N2CCC(C)(NC(C3CC4C=CC3C4)=O)C2)n1 C(C(C)(O)CC(=O)NC1CC2(C1)CC2(F)F)OC N1(C(C(CCC)F)=O)CC2(C=C(C(=O)NC3(CO)CCC4(CC3)CC4)CO2)C1 C1(C)(CSc2c(OC)cccc2)CCC2(CC1)CC2 C(=O)(C(O)CC(=O)OC(C)(C)C)N1CC(=O)N1Cc1nc[nH]n1.CCCC.O(C)OC.O.OC.C C(=O)(CP(C)(C)=O)NC(CC=C)CNC(=O)C(C)OCCC(C)C c1(C(N(CC(C)NC(=O)CCSC)CC)=O)oc(CO)cc1C C1(C)(NC(=O)NCc2cnc(-c3c(OC)cccc3)s2)CC2CCC1C2 C1(C)(C(=O)NCC(CNC(CC(CCC)C)=O)C)CCCCCCC1 c1(C(N2CC(COC)N(C(=O)CCC(C)OC)CC2)=O)cc2sc(C)cc2[nH]1 CC1CN(C(CN(C)C)=O)CC1NC(=O)C(C)(O)Cc1ccccc1 c1(C(=O)Nc2ccc(C(N3CCCC(F)CC3)=O)c(Cl)c2)cc(O)nc(Cl)c1 C#CC1CCCN(C(c2cc(C3CC3)no2)C(=O)NC2CCCC2)C1 Cc1cccc2oc(C(N3CC(NC(=O)CN4CC5CC5C4)CC(C)C3)=O)cc12 c1(C(N2CC(C)(NC(=O)COCC(F)(F)F)C2)=O)c(Br)ccc(F)c1F c1(C(=O)NCCN(C(=O)CCc2cnn(C)c2C)CCC)cc(C)cc(N)c1 N1(C(c2[nH]cc(C)c2)=O)CC(CNC(=O)C(O)CCn2cncn2)OC(C)(C)C1 C1(NC(C(CC)N(C)C)=O)CN(C(=O)CCCC(=O)OC(C)(C)C)CC1(C)C C1(CCNC(c2ccc(OC)cc2)=O)CCCN(C(=O)CCC=CC=C(C)C)CC1 C1(CCNC(C2CC(Cl)(Cl)C2)=O)CCCN(C(c2ccoc2C2CC2)=O)C1 N1(C(c2c(NC)scn2)=O)CCN(CCCNC(C2(CSC)CCC2)=O)CC1 c1(N(C(CCNC(=O)OC)=O)C)n[nH]c(C2CN(C(=O)C(C3CC3)SC)C2)n1.O c1(NC(C)=O)cccc(NC(=O)CC2(C)CN(Cc3cncc(C)n3)C2)n1 C1(N(CCc2c(C)cco2)C)CCCCN(C(C2(NC(N)=O)CC2)=O)C1 C1(C2CCCN(C(=O)CC3CCC=CCC3)C2)(NC(C2CSCC(=O)N2)=O)CC1 c1(N2CCN(C3CCC(NC(C4(C)CC(C)C4)=O)CC3)CC2)cc(=O)n(C)c(O)n1 c1(OC)ccc(C(n2cccn2)NC(N2CC(C#N)C2)=O)cc1OCCO n1(CC)nc(C)c(C(N2CC(O)(C3CCCN3C(=O)CC3CC(=O)C3)C2)=O)c1C c1(CC(=O)NC(C)CC(C)NC(=O)CCc2cccc(F)c2)cc2ccccc2o1 C1(C)(C(=O)NCCN(C(=O)CCNC(=O)CO)CC)C=CCCC1 c1(CC)[nH]nc(C(N2CCC(C(=O)NC3CN(C)CC3C)C2)=O)c1C CCCCCCCCC(F)C(=O)N1CC(O)(CNC(c2coc(CC)n2)=O)C1 Cc1nc(NC(=O)NCC2(CO)CCCC2)c(C)c(O)n1.C12(CCC1)CC(=O)N2 N1(C(CC)=O)CC(F)CC1CNC(C1CC(C(=O)OC)C1)=O CN1CCC(CC(N2CCC(NC(c3cnn(C4CCCC4)c3)=O)C2)=O)C1=O c1(OC)ccc(Cl)c(C(=O)NCC2CC(NC(C3CCCC(C)CC3)=O)C2)c1N Cc1cc(C(=O)NCC(C)CNC(c2n[nH]cc2Cl)=O)n(C)n1 CC(C)CCC(C(=O)NC(C1CCN(C(=O)CC2C=CCC2)C1)C)NC(N)=O c1(OC)cnc(Cl)cc1C(N1CCC(CO)(CNC(C2CC(F)C(=O)N2)=O)C1)=O N1(C(C2C(F)(F)C23CC3)=O)CCC2(CCN(C(c3cc(Cl)cnc3O)=O)C2)C1 CC(C)CC(CNC(=O)CC1CNC(=O)C1)NC(=O)CNC(=O)Cn1cncn1 C1(C(N(CCN(C(C2CC(=C)C2)=O)C)C)=O)CCCN1Cc1ccsc1 C(c1cncnc1O)=CC(=O)NCC(O)CCNC(c1cnoc1C1CC1)=O c1(OCCC)ccc(C(=O)NC2C3CCN(C(=O)C(C)C4CC4)C23)cc1 C1(C(=O)NCC(N(C(=O)C=CS(C)=O)C)C2CC2)CCc2nnc(O)cc2C1 CC(C)CC(C(=O)NCc1ccc(CC(=O)O)cc1)c1cccs1 C=CCCCCC(c1nnnn1-c1ccccc1Cl)NC1(COC)CCOCC1 CCC1=C(C(=O)NC(CNC(C2CCN(C3CC3)CC2)=O)C(C)C)SCCO1 C(=O)(C(C)(O)C(C)C)N(CCCC(N1CCN(C(C2C(=C)C2)=O)CC1)=O)CCC C(=O)(CCCS(C)(=O)=O)N1C(CNC(C(C2CCC2)OCC)=O)C(C)(C)CC1 C=CCCCCC(=O)N1CCC(C(N2CC=C(C)CC2)=O)C1CC C1(C)(CNC(CC2CC(OC)C2)=O)COCCN(C(=O)C=Cc2ncc(C)[nH]2)C1 C=CC(C)(O)C(=O)NC1CCC1NC(c1nnn(-c2ccon2)c1C)=O CC(C)CC(C)CC(=O)NC(CNC(=O)COCCc1ccccc1)CC(C)C N1(C(C(C(=C)Cl)(C)C)=O)CCCC2(NC(c3csc([N+](=O)[O-])c3)=O)CC2C1 c1(CC(=O)NC(C(=O)OC)Cc2ccc(O)cc2Br)c(C)ccc(F)c1Br O(N1CCC(CC(=O)NC(C)CCNC(C2(C3CCCO3)CC2)=O)CC1)CC N1(C(C(CC)C)=O)CCC2C(NC(c3cnn(Cc4cccc(F)c4)c3)=O)C12 C1(NC(C2(CNC(C3C(OC(C)=O)C3)=O)CC3(CC3)C2)=O)CCN(OC)CC1 N1(c2nc(=N)nc(C3CCCCC34CCC4)[nH]2)CCOc2cccc(Br)c2C1 c1(NCC(CC)(C)OC)cc(Nc2cc(-c3cccc(OC)c3)[nH]n2)ncn1 C(=O)(N=c1ccn(CCc2ncncc2F)[nH]1)C12CC(C(=O)OCC)(C1)C2 CCC(CC(=O)NC1CCC1NC(C1(C(F)(F)F)CCCC1)=O)C1CCC1 N1(C(C2C(CC)N(C)CC2)=O)CC(NC(=O)CCCn2ccnc2C)C2(CC2)C1 Cc1cnc2c(C(N3CC(NC(=O)CC4CCC(C)CC4)C(C)C3)=O)cccn12 C=C(Cl)C(C)(C)C(=O)NCC1(C)CN(C(=O)COCC(=C)C)CCO1 CCCC(C)(O)C(=O)NC1CC2(C1)CC(C(=O)N(C1CC(OC)C1)C)C2 n1(CC(C)C)cc(CCCNC(=O)CN(C(=O)OC(C)(C)C)C2CC2)nn1 N1(C(c2c(OCC=C)c(C)ccc2)=O)CCCC2C1CCN2C(c1cc(C)[nH]n1)=O C1(NC(CSc2n(C)nnn2)=O)CCC2(CCN(C(C3(Cl)CC3)=O)CC2)C1 CCC(CCCC(=O)NC(CO)C(=O)OC)NC(=O)C=CC=C(Cl)Cl C=CC1(C(N2CCCC(NC(C3CCC3CF)=O)CC2)=O)CCCCC1 CN1CCN(C(c2nc(Cl)c(Cl)s2)=O)CC1CNC(=O)C#CC1(C(F)(F)F)CC1 N12CCC(C1)n1cc(nn1)CN(C)C(C)C2=O.c1(SC(C2CC2Cl)=O)ccccc1 Cc1cc(=N)[nH]cc1C(N1CC2(CNC(c3snnc3C)=O)CC1CO2)=O Cc1c(C(C)NC(C2CC(O)(C(=O)O)C2)=O)sc2ccccc12 CC1(C)C(NC(C2CCCC2F)=O)CC1CNC(c1cc[nH]c(=N)n1)=O c1(C(N2C(CNC(=O)COCC3(F)CC3)CC(OC)C2)=O)ccnc2ccsc12 CC(C)(CC(F)F)C(=O)NC1CC=C(C(=O)N2CCNC(=O)CC2)C1 C(=O)(C1CCCc2nccn21)N1CC(N(C(c2ccc(C)s2)=O)C)C2(C1)CC2 c1(C(=O)NCCCC(=O)N2CC(C(N(C(C)C(N)=O)C)=O)C2)cc(F)cc(F)c1 N1(C(C2C(COC)(COC)C2)=O)CCC(C2CC2)(CNC(=O)CO)CC1 CC1(C)CC(NC(c2csc(CO)n2)=O)CN(C(c2ncccc2C2CC2)=O)C1 C#CCCCC(C)C(=O)NCC(C)(F)CNC(c1cncc(OCC)c1)=O C1(C(CN(C(CC(C)C(F)F)=O)NC(=O)CO)(C)C)CCCN1C(=O)CCc1nncs1 N1(C(c2c(C)nn(C)c2F)=O)CCC2(CC1)CC(NC(=O)CC1CCCO1)CO2 C(=O)(CC(O)CC(C)(C)C)NCC12OCC(NC(CC(C(N)=O)NC(C)=O)=O)(C1)C2 c1(C(C(=O)NC2CCCC(NC(C(C)=C3CC3)=O)C2)C)ccc(F)cc1F C1(C(N(CCCNC(CC(C)C2CC2)=O)C2CC2)=O)CC(C)(C)OC1 C#Cc1ccc(F)nc1NC(=O)CCc1ccc(OCCNC)c(C(F)(F)F)c1 N1(C(CC(CC)NC(=O)Cn2nccc2C)=O)CCn2ccnc2C1 CCC(CC)C(c1nnnn1C(C)C)NCC1(CC2CCOCC2)CC1 C1(CC(=O)Nc2ccccc2OC2CC2)CCCCN1C(c1cccc(F)n1)=O C(=O)(C(C)(C)C(F)F)NCC1CN(C(C=C(C)C)=O)C(C)C1 C1(S(=O)(=O)c2ccccc2)(C(=O)NC(CNC(CC(=O)NCC)=O)C)CCCC1 C1(n2ncc(C)c2)CCN(C(=NCC(F)(F)C2CCC2)NC2CCS(=O)(=O)C2)C1 c1(CC(=O)NC2CC(CCC(=O)NCCCO)C2)ccc2n[nH]cc2c1 N1(C(C2C(C)CCC2)=O)CCCC12CCN(C(c1cnc(N)c(CO)c1)=O)C2 N1(C(CCCCCC)=O)CC(C)(C)OCC1CNC(=O)CSCC1CCCCO1 N1(C(c2cnn(C)c2F)=O)CCOC2(CCN(C(=O)C=Cc3ccco3)C2)C1 C(=O)(C(CC(C)C)N(C(=O)CCOC(C)C)C)N1CC(F)(CC)C1 c1(C(N2C3CCC(CCNC(c4c(C)c[nH]c4)=O)(C3)C2)=O)nn(C)c2c1CCC2 C=C=CC(C)C(=O)NC1(CC(=O)NC2CSC2)CCCCC1 C1(C(N2CC(CN(C)C(c3c(CO)nnn3C)=O)OCC2)=O)Cc2nccn2C1 N1(CCO)CCN(S(=O)(=O)N(C)C)CC1.N1(C(C2CN(C)C2)=O)CC2(CC2C(=O)N)C1 Cc1cc(CC(=O)NC(C)(C)CNC(=O)C(CO)N(C)C)ccc1Cl c1(CC)ncc(C(=O)NCC(O)CNC(=O)CCCSC(C)(C)C(=O)OC)c(C)n1 C1(CC(=O)NCCC2(O)CN(C(CSCC#C)=O)C2)CCC(C)(O)CC1 c1(C(=O)NC2C(NC(=O)Cc3cccc(Cl)c3)COCC2)cc2n(c1)CCOC2 N1(C(CC2CC(=C)C2)=O)CC(N=[N+]=[N-])CC1C(=O)NC(c1ccn(C)n1)CC c1(C=O)cc2cccnn2c1.N#CC1CN(S(=O)(=O)C(F)(F)F)CC1N c1(CC)cc(NC(=O)NC(c2ccncn2)C)c(C)cc1F C(=O)(C(C1(C)CC1)NC(=O)C(C)C1CCC1)N(CCOCC)CC1CC1 c1(CNCc2ccc(-c3ccc(C(C)(F)F)cc3)nc2)cccc(F)c1[N+](=O)[O-] C(CC(CC)C(=O)NC1CCN(C(=O)Cc2c(Cl)cccc2Cl)CC1)=CC Clc1ccccc1CN(Cc1ccccn1)Cc1ncc(Br)cn1 C(=O)(C1=CC2(CCN(C(c3c(C)nn(C)c3)=O)C2)C1)NC12CC1CNC2=O C1(CCc2cn(CC)nn2)CCCCN1C(c1cnc(Cl)[nH]1)=O C(C(CC1CCCC1)C(=O)Nc1cccc(CO)c1)NC(=O)C=CCn1cncn1 C1(CCOC)(NC(c2c[nH]c(C(F)(F)F)c2)=O)CCN(C(=O)Cc2ccoc2)C1 c1(C(=O)OC(C)=O)ncccc1C(C)(C)C.c1(C)cn(CC2CCC(N)C2)nn1 c1(C(N2CC(NC(=O)C3=CCCC3)CC(C)C2)=O)ccc2c(c1)ncn2C(C)C c1(CNC(CC=C(C)C)=O)c[nH]nc1C(=O)NC(C)CC(C)C c1(C(C(=O)NC(CN(C)Cc2c(C)noc2C)C)O)cccc2c1OCC2 c1(COCC(=O)N(C(C)CNC(CCSC2(C#N)CC2)=O)C)ccccc1 Cc1nnc2n1CCCC2C(=O)N(C(C)CCNC(=O)CN1CCCC1=O)C C=C(C)CCCC(=O)NCC12CC1CN(C(=O)C(C(C)C)N1CCC(C)CC1)C2 n1(C(C)C)cc(C(N2CCC(C)C2CNC(=O)C=CCF)=O)c(O)nc1=O O=C(CCCCCF)NC1(CCNC(c2ccc(C3CC3)cc2)=O)CCOCC1 n1(CC)cc(Cl)cc1C(=O)NC1(CC(N2CC(CCOC)C2)=O)CCCC1 C(C(C)(C)CC(=O)NCC1CCC(NC(=O)CCC2C(=O)ON=C2C)CC1)OC c1(OC)cc(-c2cccnc2)c(OC)cc1CN1CCC(CO)C1 c1(CN2CC(N(C)C)C(C(=O)O)CC2)cccc2c1CNC2=O C1(C(N2CCCC2)=O)CCN(C(N)=O)CC1.C1(=O)C=CC(=O)NCC(C2CC2)N1C C1(CCOC)CN(C(C2CCCCC2C)=O)CCN1C(=O)CCC1CCOCC1 c1(C(=O)NCCC2(OC)CN(C(C3CNC(=O)C3)=O)C2)cc(C)cc(C)c1 C1(NC(c2cc(C)ncc2)=O)CC2CC(NC(C3(c4ccncc4)CC3)=O)CC12 Cc1cncc(CCNC(=O)CN2CCN(C(=O)COC3CCC3)CC2)c1 C1(NC(C(C2CCCN(C(CCSC)=O)C2)C)=O)CCOCC1(C)C c1(CC(N2CCC(OCCNC(C3CCSC3)=O)C2)=O)ccc2ccccc2c1 c1(-c2n(CCCC)ccc2)nnc(N2CCC(CC)CC2)n1Cc1cnn(C)n1 C1(NC(c2cncc(O)c2)=O)CCCCC12CCN(C(=O)Cc1ccsn1)C2 C1(C(N2C(CC(=O)OCC)CCC2)=O)CCCCN1C(c1cnc(C)o1)=O N1(C(C(CCC)OC)=O)CC(CNC(C2(CC(F)F)CCC2)=O)C2(CCOCC2)C1 C1(N(C(C2C(CNC(CC3CC(SC)C3)=O)CC2)=O)C2CC2)CCCC(C)(C)C1 CCC(CC)C(C)C(=O)N1C2CCC1C(CNC(=O)C(C)(C)CC(=O)OCC)C2 C(CCCCCCCO)NC(C1CC12CN(C(c1cccc(F)c1)=O)C2)=O C1(NC(=O)Cn2cc(C3CC3)cn2)CCOC12CCN(C(C1CCOC1)=O)CC2 N12CCC(C)C(C1)NC(=O)c1cc(on1)CSCC2=O.C#CCCOC(F)F O=C1NC(C(N2CC(OCC(=O)NC3CCCCNC3=O)C2)=O)CC1F C1(CC(=O)NC2(CNC(c3c(O)cccc3F)=O)CCC2)CCCCC1(F)F CC1CCOCC1C(=O)NC1CC(NC(c2ncnn2C2CC2)=O)C1 CC#CC1CCN(C(=O)CCC2CC(NC(=O)C(COC(C)=O)OC)C2)C1 c1(C(=O)NCC(CC)NC(CCCC=C)=O)ccc2cnccc2n1 c1(COC2CCN(C(C3CN(C(CC)C)C(=O)C3)=O)C2)ccc(O)c(N(C)C)c1 N1(C(Cc2ccc(SC)cc2)=O)CCC(NC(=O)COCCF)CC1C N1(C(c2cc(F)c(F)cc2O)=O)CC2(CCCN(C(c3cccc(Cl)c3)=O)C2)C1 N1(C(C2(CC)CCCCO2)=O)CCCCC(NC(=O)C(N2CCCCCC2)C)C1 c1(C(N2C(C(c3ccco3)=O)CC2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 CC1(C)CC(CNC(C2(F)CCS(=O)(=O)C2)=O)N(C(c2nocc2Br)=O)C1 CC1CC(NC(=O)CCC(C)(C)F)CCN1C(c1nn(C)c(Cl)c1Cl)=O c1(C(N2CCC(F)(C(=O)NCC(N(OC)C)=O)CC2)=O)[nH]nc2ccncc12 N1(C(CNC2CCCN(OC)C2)=O)CCc2ccc(NC(=O)C(C)S)cc2C1 c1(CC)cc(Cl)ccc1C(=O)NCC(C)(C)NC(C1(C)CCOC1)=O C(=O)(C(F)(F)C(C)O)NC1CCN(C(CO)=O)C1C.Cc1cnc(COC)o1 C1(CC(=O)NC)CN(C(=O)CCOCCN(C)C(C2(F)CC2)=O)C1 C(=O)(CCCC(=O)NCC(F)CNC(c1n[nH]cc1-c1ccncc1)=O)OCC c1(C(N2CC(NC(=O)CCOc3cccc(C#N)c3)C2)=O)cc2scc(Cl)c2[nH]1 C1(NC(c2cc(C(C)=O)n[nH]2)=O)CCC12CCN(C(c1ccn(C)n1)=O)CC2 C1(C)(CNC(c2ccc(CC)cn2)=O)CN(C(c2coc(Cl)n2)=O)CC1C C1(NC(=O)C=CC(F)F)CCCCN(C(C2CCCCS2)=O)C1 c1(C(=O)NC(C)CC(C)NC(=O)CCN2CCCS2(=O)=O)cc2cnn(C)c2s1 c1(C(N(C)C)=O)nc(=NCc2ccc3n[nH]cc3c2F)nc(N2CCOCC2)[nH]1 C1(F)(C(N2CCN(C(Cn3nnc(=N)[nH]3)=O)C(C(F)F)C2)=O)CCC(F)(F)CC1 C(=O)(CC1C(=O)Nc2ccc(F)cc21)NC1CC(NC(C2(CSC)CCC2)=O)C1 Cn1ncc2c(-c3csc(=NCC4CC(O)C45CCC5)[nH]3)cccc12 CN=C(NCc1cccc(CO)c1F)N1CCC(C2CC2)C1 C1(CNC(c2cc(C3(O)COC3)on2)=O)CCCN(C(C2(CCO)CC2)=O)CC1 CS(=O)C1(CNCC2CC3(CCN3)C2)CCC1 C(=O)(C1CCOc2ccccc21)N1CC(C)(C)C(CNC(c2cncnc2)=O)C1 N12Cc3cnc(nc3C1)C2.Cc1ncc(C(=O)NCc2ccccc2)o1 Cc1nc(CC(=O)NC(C)Cc2cnccn2)cs1.C12(CCCO1)C(=O)NC2 C=CCCC(C(=O)NC1(C)CC(NC(C2CC3CCC(C2)O3)=O)C1)c1ccccc1 c1(NC(C2CCCC(NC(c3ccncc3F)=O)C2)=O)c(Cl)ccc2c1OCO2 N1(C(C(CCSC)O)=O)CCC(NC(=O)COCCCF)C12CCC2 CCCCC(C(=O)NCC1CCC(NC(C2CCCC(N(C)C)C2)=O)CC1)OC C1(C(=O)NC(CC#C)CC)CN(C(c2nn(C)cc2Cl)=O)CC12CCC2 C(=O)(CS(=O)(=O)CCOC)NCC1(C(C)NC(COCC)=O)CC1 C1(NC(c2c(CCC)n[nH]c2)=O)CCN(CCn2[nH]cnc2=N)C(C)C1 c1(NC(C2C3(CN(Cc4nc(CCCC)[nH]c4Cl)C3)C2)=O)cc(C)c(Cl)cc1I Nc1cnc(Cl)c(C(N2CCC(CF)(NC(c3cncc(OCF)c3)=O)C2)=O)c1 C(=O)(CCCCC(F)F)NC1C(C)CCN(C(CCC(=O)N(CC)CC)=O)C1 Cc1ccc(Cl)c(OCC(=O)NC(C2CN(C(=O)C(C)C3(O)CCC3)C2)C)c1 C1(C(=O)NC(C2CCN(C(=O)CCc3ccoc3)C2)(C)C)CCC2CC1C2(C)C c1(C(=O)NCC2(C)CN(C(CC(C)C)=O)C(C)(C)C2)cc(F)cc2nccnc12 C#CCC(CC#C)C(=O)NCC(C)CN(C(=O)CSc1ccc2c(c1)CCC2)C N1(C(c2nc(OCC)oc2)=O)CC(CNC(=O)C(F)C(F)(F)F)CC(C)C1 C1(N(C(c2cc(OC)ncc2)=O)C)CN(C(c2ccc(C)nc2O)=O)CCC1C N1(C(C=Cc2ccc(CC)o2)=O)CCCC(CO)(NC(=O)CCC2CCOC2)C1 C1(C2(O)CCN(C(c3c[nH]c(=N)o3)=O)CC2)(NC(CC(C)(C)O)=O)CC1 C1(C(N2C(C(=O)NC(CCC)C3CCC3)C=CCC2)=O)CCCCC(=O)N1 c1(C(=O)NCCCC)cccc(C(=O)N(CCC(C)(C)CO)C)c1F CN(C)S(=O)(=O)N(C)CC(=O)NCC1CCCCC1NC(C1COC(=O)O1)=O N1(C(C2CC(=C)C2)=O)CC2CC(C1)CN(C(=O)C(CCC)CC(C)C)C2 c1(C(=O)NCC=CCNC(C=C(C)c2ccc(F)cc2)=O)ccc(O)c(N=[N+]=[N-])c1 CC(C)C(C)C(=O)NCCN(C(=O)C(C)Oc1cccnc1)C C1CC(C(=O)O)C12CCC2.n1(CCO)cc(C(CC(N)=O)NC(=O)OC(C)(C)C)nn1 CN1CC(C(N2CCCOC(CNC(=O)CCC(F)(F)F)C2)=O)OCCC1=O c1(C(CC)C)ccc(C#N)c(NCC(O)CNC(=O)CCc2nc[nH]n2)n1 C1(NC2CC2)C(C)CN(C(N2C(C(=O)Nc3c(C)cncn3)CCC2)=O)CC1C CC(O)C(C(=O)NC(C1CN(C(C2(n3cnnn3)CC2)=O)CCO1)C)N(C)C C12(NC(C(C3CC(F)(F)C3)OCC)=O)CCN(C(=O)COC3CCC3)CC1C2 Cc1cccc(-n2cc(CN3CCC(C(N4CCCC(CO)C4)=O)C3)nn2)c1 c1(NC(C2(Cc3ccc(F)cc3)CC2)=O)cc(Cl)cnc1F O=C(CCn1cc(C2CCCCC2)nn1)NNC(=O)c1ccsn1 CC(C)CC(C(=O)NCc1cnn[nH]1)N(C(=O)Cc1cccs1)C c1(C(=O)NC(C)Cn2cc(-c3ccc(F)cc3)nn2)cc(N)c(F)c(F)c1Cl CCC(F)(F)C(C)(C)CS(=O)(=O)Nc1ccc(OC(F)F)cc1C CCC(CC)C(=O)NCC(CNC(=O)Cc1ccnn1C)(C)OC c1(C(=O)NCC=CCNC(CC2(CSC)CC2)=O)cc(C)ncc1NC C1(CC(=O)NCCc2nccc(C)n2)C2CCCC2N1C(=O)C1=C(Cl)CCC1 Cc1ccc2[nH]cc(C(N3CCN(C(=O)Cc4cnoc4)C4COCC34)=O)c2c1 c1(NC(NC2c3cnn(C)c3CCC2)=O)c[nH]c2ccc(Br)cc2c1=O C1(CNC(CCOCCOC)=O)CCCC1NC(=O)NCCCCN(C)C C1(C(N(C)CCOCCN(C)C(C2(CO)CCOC2)=O)=O)CCc2cnnn2C1 N1(C(C(CC(C)C)OC)=O)C2CCC1C1CC1(NC(=O)C(C)=CC1CC1)C2 C1(CNC(c2cncc(NC)c2)=O)CCC(C)(C)CN1C(C1CC1F)=O c1(C(=O)NCCCCC(C)NC(c2ccco2)=O)cccn2ncnc12 CCCCC(C)CCC(=O)NCC1(O)CCN(C(c2coc3c2COC3)=O)C1 C1(C(=O)NCC2CN(C(c3cc(CC)nn3C)=O)CC2C)CCN2CCOCC12 c1(C(N2CC(NC(=O)C(C)S(N)(=O)=O)CC(C)C2)=O)cccc2[nH]ncc12 C1(CNC(COCCN(C)C)=O)CN(C(c2cncn2C2CC2)=O)CCC1(F)F C(=O)(C(C)(CSC)NC(C1CC(C)(O)C1)=O)NC(CCC)CC Cc1c(C(=O)NC(C)CN2CCN(C(C3C=CCCC3)=O)CC2)sc2nccn12 C(=O)(C(C)CC(=O)N(CCCN(C(=O)C=Cc1ccncn1)C)C)OC c1(CC(N2CC(C=C)C(NC(=O)CSC(F)F)C2)=O)cnc2cccnn12 C1(C(N2CC(C(C)C)N(C(=O)CCc3cccs3)CC2)=O)CCc2nn[nH]c2C1 CC1CC=CCC1CNC(c1ccc(CNC(C2CCC2C#N)=O)o1)=O C(=O)(CCCCCCCCCO)N(CCCNC(C(C)OCC=C)=O)CCO C1(NC(CC=CC)=O)CN(C(C2(C#N)CC23CCC3)=O)CC1N=[N+]=[N-] c1(OC)cccc(C#N)c1NC(c1c(-c2ccnn2CC2CCC2)cnn1C)=O Cc1ccc(CC(=O)NC2CC(NC(c3cnn(C)n3)=O)C2)o1 c1(C(=O)NCCC(C)NC(=O)C(c2cnccn2)C)cc(NC(N)=O)ccc1Cl C1(c2nnnn2CCCF)(CCc2ccc(C)o2)CCSC1C.C1CC1N c1(C(CC)C)ccc(C(=O)NC2CCC(CNC(C34CCCC3C4)=O)CC2)cc1 N1(C(C(CC)C)=O)CC(NC(c2cc(F)ncc2Br)=O)C(F)(F)C1 c1(CCOC)cccc(NC(=O)NC(C)CCc2ccc(Br)s2)c1 C1(S(C)(=O)=O)(C(N(C(CNC(C2CCC(C)(C)O2)=O)C2CC2)C)=O)CC1 C1(CNC(CCc2c(C)n(C)nc2)=O)CCC(C)CN1C(=O)CS(C)(=O)=O Cn1nc([N+](=O)[O-])cc1C(N1CCCC(CCNC(C2CC3(CSC3)C2)=O)C1)=O C(C1(CO)CCc2ccccc21)NC(C(n1cc(SCC)nn1)C)=O CCC(CC)CCCC(=O)N1CCC(C)(CCNC(=O)CCC2CCC(=O)N2)C1 c1(C(N(CCNC(C2(OC)CCOC2)=O)C2CC2)=O)ccc2[nH]c(=N)oc2c1 C1(O)(CNC(CCC#C)=O)CC2CCC(C1)N2C(c1ccc(SC(F)(F)F)nc1)=O CC(C(=O)N(CC(C)O)CCNC(=O)C(c1ccc(Br)s1)=O)C(C)O C1(NC(C=CC)=O)CCCC1C(=O)NCCCC1(C)CC1 C1(NC(C(CCOCC)NC(=O)C(N2CCOCC2)C)=O)CC(C)CCC1O Nc1c(Cl)cnc(C(=O)NC2CCC(CNC(=O)CCCc3cc[nH]n3)C2)c1Cl c1(C(=O)NC23CC(NC(CC4C(C)(C)CCC4)=O)(C2)C3)cc2c(cn1)CCCC2 C1(NC(c2cncc3n[nH]cc23)=O)CC2CCC(C1F)N2C(=O)C1=CCOC1 Cn1cnc2sc(C(=O)NCC34CCC3CCN4C(c3ccnc(S)c3)=O)cc12 C1(NC(C(CSC)O)=O)CC2CCCC(C1)N2C(c1cccc(C)n1)=O c1(C(=O)OOC(C2C(CNC(=O)C(F)C(F)(F)F)CCC2)=O)ccn2nccc2c1 c1(C(c2n(C(C)C)nnn2)NC2CCC(C)(C)CC2)cc(Cl)ccc1[N+](=O)[O-] c1(C(N2C(COC)CCC2)C(=O)NCC2CCCO2)nn(C)cc1C CC1(C)C2CC1CC(=O)N2.N1(C(=O)Nc2csc(Cl)n2)CC12CCC2 C1(C(=O)NC(CNC(c2cccc(F)c2F)=O)C2CCC2)CC2C=CCC(C1)C2 Cc1cccc(C(O)C(=O)NC(C2CN(C(=O)CSc3cccs3)C2)C)c1 C(=O)(CCCC(C)(C)C)NC(CCC(=O)NC1(CC#C)CC1)CC C1(NC(=O)NC(CC(=O)OC)C)CN(C(=O)CC2CCCOC2)CC12CCC2 C(=O)(CCC(F)F)N(CCN(C(c1cc(-c2cccnc2)no1)=O)CC)CC CC(CC(C)(C)C)C(=O)NCCN1CCN(C(=O)CCC#N)CC1 Cc1cc(C(F)(F)F)nc(N2CCC(CCNC(C3(C(F)F)CCCO3)=O)C2)n1 CCCCCCC(=O)NC1CCC1NC(=O)CCc1cccc(C(F)F)c1 C=CCCCCCCCCC(=O)N1CC(NC(=O)C(C)CC(N)=O)C2(CCC2)C1 N1(C(CCCCN=[N+]=[N-])=O)CCOC(c2cn(C3CCOC3)nn2)C1 CC1(C)C(NC(=O)CN2CC3CC3C2)CCN1C(C1SCCS1)=O C1(NC(C(CCN(C)C)N(C)C)=O)CCN(C(c2ccn(CCF)n2)=O)CC1F c1(C(N2CCC(OCC(N3CCn4nncc4C3)=O)C2)=O)ccccc1[N+](=O)[O-] C(CC1=CCN(C(c2ccns2)=O)CC1)NC(=O)CN1CCCC1CO C=CCC(CC=C)C(=O)NC1CCN(C(c2ccc(OC(F)(F)F)nc2)=O)C1C C1(CNC(C2CN(C3CCC3)C2)=O)(CO)CCN(C(=O)Cc2ccsc2)C1 N1(CC)CCCCC1C(=O)N(CC(C)C(=O)NCC1CS(=O)(=O)C1)C C1(CNC(C2CCC2C(=O)NCC2(O)CCCC2)=O)CNC(=O)O1 Cc1nn(C)c2c(NCC3(C)CC(F)(F)C3)nc(=NCC3OCCC3(C)C)[nH]c12 C(=O)(CC(C(C)OC)NC(=O)C(C)C)NCCC(=O)OC c1(C(CF)NC(c2cc(CS(C)(=O)=O)no2)=O)ccc(F)cc1F c1(NC(c2ccccc2F)=O)ccccc1C(=O)NCCCn1cncn1 C(=O)(C1CCCc2ccccc21)NC1CCCN(C(c2ccc(C#C)cn2)=O)C1 C(=O)(C1=C(C)OCCS1)NC(C1CCN(C(C2C(CC)C2)=O)C1)C C=CCC(CC(F)F)C(=O)NCC(C1CCC1)NC(c1cccc(OC)n1)=O N1(C(Cc2cncc(C)c2)=O)CCC(NC(C2CC2C(=O)N(C)C)=O)C(F)C1 c1(C(=O)NCCC2N(C(CCS(C)=O)=O)CCOC2)cc2ccc(Cl)cc2o1 C1(C(N2C(CC(=O)NCc3c(C)n(C)nc3)CCCC2)=O)CCCCC(=O)N1 C1(C(N2CCC(CC#N)C2)=O)C2Cc3cc(F)ccc3C12 c1(OC)ccc([N+](=O)[O-])c(C(C)OC)c1.C12CC(C1)NC(=O)NC2 C(=O)(CCCCCC#N)N1CCC(OCC(N2CC(C)OCCC2)=O)C1 C1(NC(C(C#N)C2CC2)=O)CC(=O)N(C2CN(C(c3nscc3Br)=O)C2)C1 C(=O)(C1=CCCCO1)N(CCN(C(=O)CC1CCS(=O)(=O)CC1)C(C)C)C Cc1ncsc1C(=O)NCC.c1(C2CNC(=O)OCC(=O)N2C)ccccc1 c1(C(=O)OCC)c[nH]c(=NC(CNC(=O)CSc2nc[nH]n2)C(C)C(C)C)cn1 c1(C(=O)NCC2(NC(C3(CSC)CC3)=O)C(C)CCCC2)c(N)sc2ccccc12 c1(C2(C(=O)NC3CCN(CC(=O)NC)C3)CC2)cccc(F)c1F c1(CC)c(C(=O)NCC(C2(O)CCN(C(c3c[nH]ccc3=N)=O)C2)C)cnn1C C(=O)(C#CC1CCCO1)N1CCCC(n2cc(C(C)(C)NC(C=NOC)=O)nn2)C1 C(=O)(CC(C)C(C)C)N1CCC(N(C(c2ccc(N(CCC)C)nc2)=O)CC)C1 N1(C(=O)NCc2n(C)nc(C(F)(F)F)c2)CCN2C(=O)CCCC2C1 c1(C(=O)NCC2CN(C(C=COCC)=O)C(C)CC2)cc(Cl)c(N)cc1OC c1(N(CC2CCN(C(C(C)OCC=C)=O)CC2)CC)cccc(OC)c1F CC1COCC(O)(CNC(c2cc(CNC(=O)C(CO)NC(N)=O)nn2C)=O)C1 N1(C(C=C(COC)C)=O)CCC2CCCC12CNC(=O)CSc1ccc(C)c(C)c1 C(=O)(C1=CC(O)C(NC(c2coc(C3CC3)n2)=O)C1)N1CC(CC#C)OCC1 c1(CC(=O)NCCNC(C2CC3CC(OC)C3C2)=O)ccc(S(C)(=O)=O)cc1 n1(C(=O)N(O)CN(C2CCC2)C2CCC2)nc(-c2ccccc2)cc1C1CC1 Cc1ncc(C(=O)NCCc2cn(C3CC3)nn2)c(F)c1Br Cc1ccccc1C=CC(=O)NC1CCN(C(C2CCCC2C(F)(F)F)=O)C1 O=C(C(F)C1=CCCCC1)N1CC(F)(F)CC1CNC(C12CCCCC1C2)=O c1(N(CCCCCC=C)C)ccc(S(=O)(=O)N2CCC(CC(C)C)C2)cc1Br CC1c2ccsc2CCN1C(c1ccc(-c2ccncc2)cn1)=O C1(NC(c2cc(CCCCC)[nH]n2)=O)C=CCN(C(C2(P(C)(C)=O)CC2)=O)C1 c1(-n2ccc(C(=O)NC3CCN(C(C4CC5CC5C4)=O)C3)n2)ccc(F)cc1F C1(N(C)C(C2CCC(n3cc(CC4COC4)nn3)CC2)=O)CC(O)C1(C)C c1(NC(C(c2cccc(Cl)c2)N(C)C)=O)ccc2c(c1)C1(CC2)CC1 c1(COC)csc(-n2cc(C(=O)N(CCCCNC(c3ccc[nH]3)=O)C)cn2)n1 C1(C)(NC(C(COC(C)C)NC(=O)CCC2CCCCO2)=O)C(C)(C)C1(C)C c1(C(N2CCN(CCNC(COCCC(C)C)=O)CC2)=O)nc2ncccn2n1 c1(C(=O)NCC=CCNC(c2ccc(CC)s2)=O)cnn(CC)c1-c1ccccc1 c1(C(=O)NCCCN(C(c2onc(Br)c2C)=O)CC)c[nH]c(=N)cc1C C(C(=O)NCC(C)CNC(c1cnc(CCC(F)(F)F)s1)=O)(C(C)C)OC C#Cc1cccc(C(=O)NC(C)CNC(=O)Cn2cnc3c2CCCC3)c1C CON1CCC(NC(N2CCOC(CSc3cccnc3)C2)=O)CC1 c1(C(N2CCC(C(C)NC(C3C(C=C)C3)=O)CC2)=O)cccc(C)c1F CC1CN(C(=O)CN(C)C2CC2)CCN1C(=O)CCC1CCCCC1 CC(CNC(=O)CCN(C)CCO)C(F)C(=O)N1CCC(C)(CCO)CC1 C1(NC(CNC(=O)CC2CCCC2)=O)CN(C(c2cscn2)=O)CCC12CCC2 N1(C(CCC#C)=O)CCC2(CNC(=O)CN=S(C)(C)=O)CCCCC12 CCCCCCC(=O)NCC1(F)CCCN(C(=O)C(=O)NCCC(N)=O)C1 C(=O)(C1CCc2c[nH]nc21)N1CC(CCCCNC(C(CC)C)=O)C1 C1(NC(CC(CC)O)=O)CC2(CCCCN2C(C2(C3CCCO3)CC2)=O)C1 c1(C(CC)NC(=O)CN(C)C(C2CCCNC2)=O)cc(F)cc(Br)c1 c1(OC)cc(C(=O)NC(C)CNC(=O)C(C)N2CC(C)C2)ccc1OCC(N)=O c1(OC)ccc(C(=O)N(CC(C)(C)NC(=O)CN(C2COC(=O)C2)C)C)nc1Cl c1(CNC2C(CNC(CCCC3(C)N=N3)=O)CCC2)cc(Cl)c2n[nH]cc2c1 c1(C(=O)OC)cc(-n2cc(C(C)N(C)C(C34C=CC(CC3)C4)=O)nn2)ccn1 n1(CCNC(C2CC(=C)C2)=O)cc(COCC(N2CCC(OC(C)C)C2)=O)nn1.N c1(CCC(=O)NCCCNC(C(C(CC)C)OC)=O)ccc([N+](=O)[O-])cc1.C(C)(=O)N CC1C(C(=O)N(CCCO)CCOC)CCN1C(=O)Cc1cc[nH]n1 N1(C(C2(NC(C3(C)C(C)OCC3)=O)CCCC2)=O)CC2COCC2(CO)C1 C1(C(N(CCOC)CCNC(=O)C(C)SC2CC2)=O)CC(=O)N(CC(F)(F)F)C1 c1(C(C)NC(CCC2N(C(c3cnc(CC)s3)=O)CCC2)=O)ccc(C)c(C)c1 C(=O)(C(O)P(C)(C)=O)N(C(C)CCNC(=O)Cn1cnc(Br)c1)C NC(=O)CCCC(=O)NCCNC(=O)CCc1ccc(Br)cc1 C=C(C)CC(C(=O)NCCC(C)N1CCC1)NC(=O)COC1CC1(F)F O(NC(=O)C(CCOC)NC(=O)C(C)O)CC(=O)NCC c1(CC(=O)NC(C)CCNC(=O)CCC2(C#N)CCC2)cc(Cl)cc2ccccc12 c1(N2C(C)(CNC(C=Cc3cc(C)cc(C)c3)=O)CCC2)ccc([N+](=O)[O-])cc1Br c1(CC)ccc(N)c(C(N2CC(C)(NC(C3CC3C3CC3C)=O)C2)=O)c1 C#CCCCC(=O)N=c1cc(-c2ccc(C3OCCO3)cc2)[nH][nH]1 c1(CNC(C2C(CNC(=O)CC3C=CCCC3)CC2)=O)ccc(F)cc1 C1(NC(CC)CC(=O)N2CCC(F)(C(=O)SC)C2)CC2(C1)CC(CO)C2 C12(NC(Cc3c(C)noc3)=O)CC(CNC(=O)CC3C=CCC3)(C1)OC2(C)C NS(=O)(=O)CCC(=O)NC1CN(C(=O)COCCF)CC1Cc1cccc(F)c1 C12CC(O)C(O)CC1c1cn(nn1)C1COCC1S2.C1(CC)CCCN(C(C)=O)C1 c1(CCC)ccc(C(=O)NC(CNC(c2cc(CCO)on2)=O)CC)s1 C(=O)(C1=CCN(C(=O)CCC=C(C)C)C1)NCCC(C)N(CCC)CC C(N=c1[nH]c(=NCCCCOC2CCC2)c2sccc2[nH]1)c1cc(C)ncc1 C(=O)(CCC(C)S(C)(=O)=O)N1C2C(CNC(C(CC(=C)C)OC)=O)C(C2)C1 C(=O)(C#CC1CCCO1)NCC(C)CNC(c1occc1Cl)=O C12(C(=O)NC(C(C)NC(Cc3c(C)con3)=O)C)CCC(CC1)C2(C)C C#CCCC(C(=O)N1C(CO)CCC1CO)NC(C1SCC=C1C)=O C1(CC(=O)NCC(c2ccc(OC(C)C)cc2)N(C)C)CCCC2(CC2)C1 N1(C(c2cc(F)ccc2Cl)=O)CC2(CCC(CNC(C34CC(F)C3C4)=O)O2)C1 c1(CN(CCNC(c2nccc(C)n2)=O)CC)cc(O)nc(-c2ccccn2)n1 N1(C(c2ccn(CCC)n2)=O)CCCC(NC(=O)C(F)=CCCF)C1 n1(CCSC)nnnc1C(C1CCC1)NCCSc1cc[nH]n1 c1(CC)nn(C)c(CC)c1C(=O)NCC(C)CNC(=O)C(C)CSC(F)(F)F n1(CC)ccc(CC(N2CC(O)(CC(=O)N(C)C(c3ncc[nH]3)C)C2)=O)n1 c1(OCC)cc(C(=O)N(C)CC2CCCN2C(C2CCCC(C)C2)=O)cc(F)c1 C(=O)(CC(F)(F)CC(=O)N1CCN(C(c2c(C)cc(C)cc2C)=O)CC1C)OC c1(C(=O)NC(CCSC)C(=O)NCC2CSCCO2)cccc(C)c1C c1(OC)ccc(F)c(S(=O)(=O)N2CC3CCCC2C3CNC(=O)OC(C)(C)C)c1 C=CCC(C(=O)OC(=O)C(C)(C)C)N(C(=O)C(N1CCCC(C2CC2)C1)=O)C N(C1CCCc2ccccc21)C(CN1C(=O)NC(C)(CCCCC)C1=O)=O Cc1nn2c(C(=O)NCC3CC4CC4N3C(=O)C=CCBr)c(C)nc2s1 c1(C(=O)NC2C(NC(C(CC#C)O)=O)COC2)ccc2c(c1)nnn2C C1(C(=O)NC2CC(OC)CN(C(C3(C)COCCO3)=O)C2)CC2CCCC(C1)C2 N1(C(c2ncn(CC)n2)=O)CCC(CNC(=O)CCCc2cnn[nH]2)C(O)C1 C(C(O)C(=O)NC1(c2cccnc2)CC1)NC(=O)Cc1nc[nH]n1 c1(C(=O)NC2C(CNC(=O)C(=O)NC3CC3)CC2)cc2cccc(F)c2o1 N1(C(=O)COCCF)CCN(C(C2CC(CF)C2)=O)C(c2ccc(F)cc2)C1 Cc1ccc(NC2CC(C)N(C(C3(C)CC(O)CN3C)=O)C2)c([N+](=O)[O-])c1 N1(C(C(CNC(C(CC)N(C)C)=O)SC)=O)CCC(N(C(C)=O)C)CC1 C=CCCC(F)(F)C(=O)NCc1cc(C(=O)NC2CCCC2SC)co1 C1(NC(C(C(=O)OC)C)=O)CN(C(c2sccc2OC)=O)CCC1CO S(=O)(=O)(c1ccc(CNC(c2cncc(Br)c2)=O)o1)NC Cc1c(Cl)c(C(N2CC3C(NC(C4CCCCC4(C)C)=O)C3C2)=O)nn1C c1(N2CC3(C)C(C)(C2)C(=O)NC3=O)ncnc2c(Cl)cc(Cl)cc12 C(=O)(CCCCCNC(=O)CC(C)(F)F)N(C)CC1CCCS1 c1(C(N(CCC(N2CCCC(CC=C)C2)=O)C2CC2)=O)cc(O)nc(O)n1 N1(C(c2cc3sccc3s2)C(=O)NCCCCCC)CC2C3CCC(C3)C2(C)C1 c1(C(=O)NC(C)CNC(=O)C(F)(F)c2cncs2)nnn2c1CSCC2 C=CC1(C(N2CC(CN(C)C)C2)=O)CCN(C(=O)C(CN(C)C)CC)C1 c12cccc(c1)CNC(C)C1CN(C1)C2=O.C1(C(C)(C)C)CCOC1C1CCC1 c1(C(N2CCCC(C3CCCN3C(c3cnsn3)=O)C2)=O)noc2c1COCC2 C(C(=O)NC1(C)CC(Nc2cc(=O)n(C)cn2)C1)(C(C)(C)C)SC.c1ccccc1 C12(NC(CCCCOC)=O)CCCC(CN(C(=O)CCCN3CCCCC3)C1)C2 c1(C(N2CC(C(=O)NCCC#CCC)(CC)C2)=O)cccc(=O)n1C C1(CNC(C(CC)N(C)C)=O)CC2(CCC2)CN1C(=O)CCCCCN(C)C C(=O)(CCN=c1[nH]ccs1)N1CC(CN(C(c2c(CC)scn2)=O)CC)OCC1 C(CC(C)C)(C(=O)NCC(O)C1(Cl)CC1)NC(c1ccc(CC)o1)=O Cc1[nH]c(=NCC2CN(C(=O)CC3CCC(O)C3)CC2(C)C)ccc1[N+](=O)[O-] N1(C(C(=O)Nc2n(C(CC)C)ncc2)=O)CCC(F)(F)C2(CCOC2)C1 C(=O)(C(CNC(c1cc(F)ccc1C)=O)C(C)(C)C)NC1(C(=O)NCC)CC1 C1(C)(OCC(=O)NC(CC(C)NC(Cc2cc(C)[nH]n2)=O)C)CCOCC1 CC1CCCN(C(c2cnoc2C2CC2)=O)C1CNC(=O)CSS(C)(=O)=O C1(N(C(c2c(CCC)nco2)=O)C)CN(C(C2CCS2(=O)=O)=O)CC12CC2 C=CC(CC)C(=O)NC(CC(=O)NCc1ccsc1)C1CC1 C1(CCOC(C2C(C)CN(C(=O)OC(C)(C)C)C2)=O)(N(C)C)CC2(CCC2)C1 c1(CNC(CC=CC=C)=O)ccc(C(=O)NCCC2(O)CCCC2)s1 c1(OCC(=O)NCCCC(=O)NCC)ccc(C(F)(F)F)cc1S(N)(=O)=O CCC(CC)CCC(=O)NCC1CC(NC(=O)C(C(C)(C)C)N(C)C)C1 C1(CNC(CCCSC)=O)CC(NC(=O)CCc2cc[nH]c(=N)c2)C12CCC2 CCC(C)(COC)C(=O)N1C(C(=O)NC2CN(C)C(C)(C)C2)CC2CC12 C1(C(=O)NC2(CCNC(=O)CCn3cccn3)CC2)(Cn2ccnn2)CC12CCC2 c1(C(=O)NC2CCN(C(C3COCC(C)(C)O3)=O)C2)cnc2c(c1)CNC(=O)N2 c1(OC(CNC(C(CC)(C)c2ccncc2)=O)(C)C)cccc(C=CC(=O)O)c1 CC#CCC(C(=O)NC1CN(C)CC1O)NC(=O)CCCCC=CC C1(C(N2C3CC(CNC(=O)Cc4ccoc4)C2CC3)=O)CCn2nnnc2C1 C1(CNC(C(CC2CCC2)OC)=O)CN(C(C2(C)CCCCC2)=O)CCCO1 N1(C(C(C)=CC2CC2)=O)CC2(CCCCN2C(=O)C(C)OCCN(C)C)C1 Cc1nn(C)c(=O)c(C(N2CC3CCC2C(NC(c2csc(Cl)c2)=O)C3)=O)c1C c1(C(=O)Nc2ccc(N(C)C)nc2)c(Cl)ccc2cccnc12 c1(NC)cnccc1C(=O)NCC1(C)CCCN1C(=O)CCCCC1CC1 N1(C(CC(C(=O)OC)C)=O)CC2CC1CCN2C(c1cc(O)ncn1)=O c1(C(c2ccc(F)cc2)NCC(N2CCc3ccsc3C2)=O)cc(F)c(F)c(F)c1 C1(C)(NC(CC2N(C(C)C)CCC2)=O)CCN(C(=O)Cc2ccc(Br)cc2)C1 Cc1nc(N2CCN(C)C(CNC(c3cncc(Cl)c3)=O)C2)cc2nncn12 C1(OCC)CC2(C1)CC2C(=O)NCC1CCN(C(=O)C(c2cnn(C)c2)C)C1 N12CCC(O)(CC1)CCC2=O.c1(C(N2CCCC2CO)=O)cc(CCCO)on1 N1(C(c2[nH]cc(CC)c2)=O)C2CCC1CN(C(=O)CN1CC=CC1)C2 c1(-c2nc(-c3nccc(SC)c3)nn2C2CCOC2)cc(F)cc2nc[nH]c12 C1(C)(NC(CNC(CN(C)C)=O)=O)CCN(C(=O)CC2CCCN2C)CC1 CC1(C)CC(O)CCN(C(=NCc2nccs2)NC2CCS(=O)(=O)C2)S1 C1(NC(=O)C(CCF)NC(c2sccc2Cl)=O)CCc2n[nH]cc2C1 C1(C(=O)NCCCCCNC(=O)Cc2ccon2)C2CC2C2CC12 C1(OC)CCC(NC(C2CC(O)CN2C(=O)C=C2CCC2)=O)CC1 c1(C(N2CCC(C)(CNC(c3ccc(C#N)o3)=O)C2)=O)cc(O)ncc1Br CC(CCC(=O)NCC(CO)NC(C1(C)CCOCC1)=O)c1ccccc1 N1(C(C(C(C(C)C)O)(F)F)=O)CCC2(CC1)CN(C(=O)CCCCF)CCO2 C(C)(CN=c1[nH]c(Cl)ncc1Br)(C1CC1)NC(C=CCOCCOC)=O N1(C(c2c(C(C)(C)C)c[nH]c2)=O)CC2CC(NC(=O)CCn3ccnn3)CC1C2 CCCCCCCCCC(=O)NC1CN(C(C2CC3CCC(C2)S3)=O)CC1O Cn1nc(CNC(C2CCC2C(=O)O)=O)cc1NCC1CC(F)(F)C1 C=CCCCC(C(=O)N(CC(F)(F)COC)C)NC(=O)C(CCC)N(C)C CC(CCCCNC(c1ccsn1)=O)NC(c1ccc(CN(C)C)nc1)=O c1(C(N(CCCN(C(C(CC)NC(N)=O)=O)C)C)=O)nccc2ccsc12 Cc1ccc(C)c(C(N2CCC(CNC(c3cnn[nH]3)=O)CC2)=O)c1C c1(C(=O)NCCC(CNC(CC=C(C)C)=O)O)ccnc(Oc2ccccc2)c1 C12CC(C1)C(=O)N2CCN(C)C(C)C.C(=O)(C(C)SC(C)C)NCC C(=O)(CCCCC(=O)N1CC2CC(NC(C3CCOC(C)(C)C3)=O)C(C2)C1)OC c1(C(N(CC(C)NC(c2c(Cl)cnn2CC)=O)CC)=O)onc2cc(C)ccc12 c1(C(N(C)CC2COCCN2C(=O)Cc2csc(Cl)c2)=O)ccnn2ccnc12 C1(CC(C)O)CN(C(=O)NC(C)(CCN(C)C)N(C)C)C2(CCC2)CO1 Cc1cc(=O)n(CC(N2CCC(O)(CCNC(=O)C(O)C3CCCC3)C2)=O)cn1 N1(C(C)C)CCCCC1CCCNC(=O)NC(=O)C(C)C(C)n1cccn1 N1(C(C=C(CC)CC)=O)CCCC(CCC(=O)NC(c2ccc(COC)o2)=O)C1 C1(NC(C(CSC)C)=O)CCN(C(c2cn(CCCN(C)C)nn2)=O)C(C)C1 C1(C(NOCCCOC)=O)CC2(CCN1C(=O)C1=NOC(C)C1)CC2 C1(C)(C(=O)NCCCCNC(c2cc(C)c(C)[nH]2)=O)CCC(C)C1(C)C c1(OCCC)cccc(CN2CC3(CC3C(=O)Nc3c(NC=O)nsn3)C2)c1.NCC N1(CC(C)NC(c2cc(CCC)on2)=O)CCN(C(=O)CC2CC2)CC1 CC1(C(N2CC3(NC(C4CCCS4(=O)=O)=O)CC2C3)=O)CCCCNC1=O c1(OC)cnc(C(=O)NC(CCCCO)(C(=O)COCC=CCO)CC)cn1 C=C(F)C(=O)N1CC(NC(=O)C=C(C)C(C)C)C1 N1(CCNC(c2ccc(C)cc2)=O)CCC2CN(C(=O)C(C)SC)CC12.CO S(=O)(=O)(c1cccc(N2CCC(CO)CC2)n1)N1CC(C)C(C)CC1 c1(C(N2CC(C(=O)Nc3c(OC)c(C)ccc3)C2)=O)cn(C)c2ccccc12 N1(C(C2(OC)CCCC2)=O)CC2CC(NC(=O)CN3CCOCC3=O)CC(C2)C1 C1(CCNC(c2cc(C)c(C)s2)=O)CC(F)(F)CN1C(=O)CC1CCCCC1O C1(CNC(C(C=CC)O)=O)COCCN1CCc1nnsc1N Cc1c(C(=O)NC2(C)CCN(C(C3CC3c3nccn3C)=O)C2)n[nH]c1C1CC1 c1(C(N2CCN(C(C(C=C)O)=O)CC2CC(F)F)=O)ccc2[nH]ccc2c1 Cc1c(C=CC(N2CCCN(C(=O)CC3COCC(C)(C)O3)CC2)=O)cnn1C N1(C(C(=O)NC2CC2)=O)CCC(NC(C2(C(F)(F)F)CCCC2)=O)C(CO)C1 C12CC(CCO1)NCCN(C1CC1)C2=O.c1(C(=O)NCC)cn(C(C)C)cn1 Cc1nc(N2CCCC(CO)(NC(=O)Cc3csc(C4CC4)n3)C2)cc(O)n1 Cc1cscc1C(=O)N(CCCCN(C(=O)CCCc1ccccn1)C)C CC(C)C(O)C(F)(F)C(=O)NC1CCCCN(C(c2csc3cnccc23)=O)C1 C1(CC)CCCN(C(=O)CC2(C)CCN(C(=O)CCCNC(=O)OC)C2)C1 N1(C(COCC(C)C)=O)CCOC(C2(NC(c3cc(C(N)=O)[nH]n3)=O)CC2)C1 CC(C)C(C#N)C(=O)N1CC(C(=O)Nc2ccn(NC(c3ccccc3)=O)c2)CC1(C)C C(c1cncc(F)c1)=CC(=O)NC(CC)CNC(=O)CCNC(=O)CO C1(c2ccc[nH]2)C(C2(CNC(C3(COCC)C=CCC3)=O)CC2)C1(C)C.C(=O)NC c1(C(=O)NCCCN(C(c2ccc(CC)nc2C)=O)C)ccn2c1CCCC2 c1(C(N(C)CCOCCNC(=O)C=C(C2CC2)C2CC2)=O)c2c(nn1C)CCC2 C1(C(N(CCCn2ccnc2)C)=O)CCCN1C(=O)CC1CCCC1 CC(C)C(C)CC(=O)N1CC(C)(NC(=O)C(F)C(C)(C)O)C1 C1(CCNC(C2C(F)(F)C23CC3)=O)CCCN(C(c2ccsc2Cl)=O)C1 c1(C(N2CCN(C(CCC=CC)=O)C(C)C2C)=O)cccc(C)c1N=[N+]=[N-] c1(SC)snnc1C(=O)NCCCN(C(=O)CCCn1ccnc1C)C(C)C c1(C(CNOC)OCc2cccc(NC(=O)CCSC)c2)cccc(F)c1 C1(C(=O)NCCNC(C2C3CN(C)CC32)=O)CC12CC(F)(F)C2 c1(CC)cc(C(=O)NC2CC(C)N(C(=O)CCOc3cccc(OC)c3)C2)c(C)o1 c1(N2CCC(NC(CCc3cc(OC)ncc3)=O)CC2)ncnc2c1SCCC2 C1(CNC(=O)C=C2CCOCC2)C(O)C(O)CN1C(C1CCC(O)C1)=O Nc1ccc(C(=O)NC2CC(CCNC(c3cocn3)=O)C2)cc1Br c1(CC)nc(C)c(C(N2CCN(CCNC(=O)C(C)=C3CCCC3)CC2)=O)s1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)NCCSC1CC1.CC1(C)CC(n2cc(C)nn2)CO1 N1(C(c2ccc(C(C)O)cc2)=O)CC=C(CNC(=O)C(N2CCOC2=O)C)CC1 c1(CCNC(C(C2CC2)NC(C(CN(C)C)O)=O)=O)cc2ccccc2[nH]1 C1(C)(C(=O)NC)CCN(C(c2ccsc2-c2cccnc2)=O)C1 CCC(CO)(C(=O)NC1CCCC(C(=O)NCc2cn(C(C)C)nn2)C1)OC N1(C(c2ncc(C)c(Cl)c2)=O)CCC2(CCCN2C(c2nc(=O)cc[nH]2)=O)CC1 N1(C(C(C)(C)OC(C)C)=O)CCCOC(CNC(c2ccnnc2)=O)C1 c1(OC)cc(C(N2CCC3CCN(C(=O)C(C)O)C3C2)=O)c2cccnc2c1 N1(C(Cc2nc(C(C)C)sc2)=O)CCN(C(C2CCC(=O)O2)=O)CC1CF c1(OC)cc(C(=O)NCCC2(NC(c3ccsc3C(F)(F)F)=O)CC2)ccc1C Cc1ccn2ncc(C(=O)NC3CCCCC3NC(=O)C(O)c3ccsc3)c2c1 N1(C(C(C(C)C)SCC)=O)CCCC(O)(CCNC(c2cnc3n2CCC3)=O)C1 N1(C(C2CCCC(C)(C)C2)=O)CC2CN(C(=O)CC3(O)COC(C)(C)C3)CC2C1 N1(C(c2c(CC)scc2)=O)CC2CC(NC(c3cc(F)c[nH]3)=O)C1C2 CCS(=O)(=O)CC(=O)N1CCN(C(c2c[nH]cc(C)c2=O)=O)CC1CC C(C(O)CCNC(c1c[nH]nc1-c1ccsc1)=O)NC(CCOCCOC)=O CC1(C)C(NC(C2(n3cncn3)CC2)=O)CC1CNC(=O)CCc1nccs1 C(=O)(C(F)(F)C1(O)CCC1)NCC(CNC(=O)CCOC1CC1)F N1(C(=O)Nc2cncc3c2CCC3)CCc2nc(Cc3ccc(C)cc3)sc2C1 N1(C(Cc2ccc(C)s2)=O)C2CCC1CC(CNC(=O)CCc1ncco1)C2 CCS(=O)(=O)CC(=O)NC1(CO)CN(C(=O)C=CCN(CC)CC)C1 c1(CN2C(C(=O)NC(c3ccncc3)C)CNCC2)cc(Cl)c(Cl)cc1O c1(C(C)(C)C(=O)NC2CCN(C(C3(C)CC3(F)Cl)=O)C2)cccnc1F Cc1cncc(C(=O)NC2CCN(C(C3CCC(C(N)=O)N3C)=O)C2C)n1 c1(-c2[nH]cc(CC)c2)nc(-c2ccc(C)cc2)nn1C1CCCCC1C C1(C(N(CCOCCN(C(C(C)=C2CC2)=O)C)C)=O)CC2CCC1NC2=O Cc1cc(N)cc(C(N2CC(O)(CNC(=O)C(c3ccccc3)C)C2)=O)c1F CCC(CC1CCC1)N=c1[nH]c2c(c(=NCC3CC(=O)N(CCOC)C3)[nH]1)CCC2 c1(OC)ccc(NC(C2CCN(C(=O)C=Cc3ccc(C)s3)CC2O)=O)cc1Br C(CC(C)(C)CC(=O)N1CC2CC1CCC2NC(c1coc(SC)c1)=O)OC C(=O)(CCN=C(NC1CC2CCC1O2)N1CCC(n2nnnc2C)C1)N(C)C1CC1 CCCCCCC(CC)NC(C1CC(NC(=O)CSC)C1(C)C)=O CCC(O)CC(=O)NC1C2CC(NC(=O)C(C)(C)N3CCCCC3)CC12 C(=O)(C1Cc2c(Cl)cccc21)NCC1CN(C(c2n(OC)cnc2C)=O)C1 c1(C(=O)NC2(C)CN(C(c3c(OC)csc3)=O)C2)ccc2c(c1)C(C)CO2 CC(C)CCCCCCNC(=O)CNC(=O)CNC(c1ccc2cc[nH]c2n1)=O C1(CNC(CCc2ccn(C)c2)=O)CC2CCC(C1)N2C(=O)C(O)CC(F)(F)F c1(OCC)cccc(CN=C(NC(C)C)NC2CCN(C(=O)OC)C2)c1 CC(C)C1(C(=O)NC23CC(NC(=O)COC(C)(C)C)(C2)C3)c2ccccc2N1C C1(C)(CNC(Cc2cc(C)ns2)=O)CCN(C(C2CCCCC2O)=O)C1 N1(C(C2CCN(C(C=Cc3cn(C)nc3)=O)C2(C)C)=O)CC(CO)C2(CCC2)C1 C1(C(c2cn(CC(=O)N(C(C)C)CCF)nn2)N(C)C)CCCS(=O)(=O)C1 C(C(C)C)(C(O)C(=O)N1CC(CNC(C2CN(C)CCO2)=O)CC1(C)C)OC N1(C(C(C)=C(CC)C)=O)CCC(CC)C1CNC(=O)C(C)CC C(=O)(C(C)(C)CC(=O)NCC(CNC(C12CCCCC(F)(C1)C2)=O)CO)OC CCCC(C)(C)CC(=O)N(C1CN(C(=O)C(C2(O)CCCC2)F)CC1(C)C)C C(=O)(C1=NOC2COCC12)N(CCCC)C.O(CP(C)(C)=O)C(=O)C N1(C(CCC(C)SC)=O)CCC2(CC1)CCN(C(c1ccc(O)cc1F)=O)C2 c1(CC=C)ccc(CNC(=O)CNC(=O)Cc2ccn(C)c2)cc1 N1(C(c2c(C)nc(C3CCCOC3)s2)=O)CC2CC(NC(=O)CC(C)(F)F)CC1C2 Nc1cccc(Cl)c1C(N1CCC1CNC(=O)CCCCc1ccccc1)=O C#Cc1cncc(C(=O)NC2CN(C(C3(N(C)C(C)=O)CC3)=O)C2)c1 C1(CC(=O)NCc2n(CC)nnn2)CC2(C1)CN(C(C1CCSC1)=O)C2 CC(CC1CC1)C(=O)N(CCC(=O)NCC(C)(C)n1ccnc1)C1CC1 C1(C(=O)NCC2(C=C)CCC2)C2CN(C(=O)CC(C)F)CC12 N1(C(CCSCCC)=O)CC(C(=O)NC(C)CCCCO)C(C)C1 Cc1ccc(Cl)c(C(N2CCC(O)(C(C)CNC(C3(CO)CC3)=O)C2)=O)c1O N1(C(=O)OCC=C)CCCN(N2CCC(C)(c3cc(C)[nH]n3)C2)CC1 c1(C(=O)NCCN(C(c2c(OC)cccc2)=O)CC)cc(F)cc2nn(C)cc12 C=CCC(C)(CC)C(=O)N1CC(C(=O)NC2C=CC(CO)C2)C(F)(F)C1 C12CCSC3(C1)CC(C3)C(=O)NO2.c1(NC(CN(C)C2CC2)=O)n[nH]c(=N)[nH]1 CC(CC(=O)NC1CC1NC(c1ccn(Cc2ccccc2)n1)=O)N(C)C c1(C(=O)NCC2C(C(NOC(C)(C)C)=O)C2)ccn(C)c1 CCC(C(=O)OC)C(=O)NCCCC(C)NC(C1(O)CCSCC1)=O c1(C(=O)NC(CC)C(=O)N2CCC2(C)C(=O)OC)cc(O)cc(F)c1 C(=O)(C(O)C(F)F)N(CCN(C(=O)CC1C=NNC1=O)CC)CC C(=O)(C(F)(F)C(O)C1CC1)NC1CCC(CNC(c2n(C)ccn2)=O)C1 C(=O)(C(C)(C)Cc1ccccc1)N(C)CC1(O)CN(C(CCCC2C(C)C2)=O)C1 C(=O)(C(O)CC(F)(F)F)N(CCCNC(c1cccc(C(F)(F)F)c1)=O)CCO c1(C(C(=O)NC2CCCCCC2)N(C(CCCC)C)C2CC2)ccc(OC)cc1C C12(CCNC(C(CC=C)C)=O)CCC1CN(C(c1csc(C(F)F)c1)=O)C2 N1(C(CC(=O)NCC)=O)CC(C)CN(C(c2cnc(NC3CC3)s2)=O)C(C)C1 C1(C(=O)NCCC(C(=O)NCC(CC)(F)CC)O)Cc2nccn2C1 c1(SC)nn(C)cc1C(=O)NC(CO)C(C)NC(C1CC(C)C1)=O C1(CN2C(=O)CN(CCCC)C2=O)CC2CC1CC2(F)F N1(C(C(F)=CC)=O)CCC(O)(CC(=O)NC(C23CCC(CC2)C3)C)CC1 C1(NC(C2CNC(=O)N2)=O)CC2CCC1N(C(=O)C(c1ccc(F)cc1)O)C2 C(=O)(C1CCCc2cccnc21)NCCN(C)C(C1(c2cnn(C)c2)CC1)=O c1(CCC(N2CC(CNC(COCCC#C)=O)(COC)C2)=O)ccc(O)cc1 C(CCN=C(NCC1(C)CCC(=O)N1)NC1CCCC(NC(C)=O)C1)OCC CC1=C(C)CN(C(C2CCCC(NC(c3snnc3C)=O)C2)=O)CC1 c1(C(C(=O)N(CCF)CC)NC(=O)CC2CCCCN2C)c(C)cccc1Br c1(NC(=O)C=CC(=O)NCCOCCCNC(=O)CC2CC2(F)F)cccs1 N1(C(C2CCC(C)O2)=O)CCN(Cc2cn(CC3(C)CCC3)nn2)CC1 c1(C(N(C2CC(NC(C3N(C(C)=O)CCC3)=O)C2)C)=O)cc2ccnc(Cl)c2[nH]1 c1(SCC)ccc(NC(=O)Nc2ncc(C(=O)OC)s2)cn1 CCCC(C(=O)OC)C(=O)NCCNC(c1ccc(C(N)=O)cn1)=O c1(C(=O)NCC(c2ccccc2)CNC(C(COC)O)=O)cc(C#N)ccc1Cl C(CO)(CC(O)c1ccccc1)NC(C1(O)CC(N2CCCCC2)C1)=O C1(CC=C)(NC(=O)CCn2ccc(=N)[nH]2)CCCN(C(C2(C)CC2Br)=O)C1 O=S(=O)(c1ccc(NCC2CCCCC2C(F)(F)F)c(Br)c1)NCc1cnsc1 C1(CNC(C2(N(C)C)CCCC2)=O)CN(C(=O)C(C2CCCCC2)F)C(C)(C)C1 N1(C(C(C=CCCC)O)=O)CC(C)(CNC(=O)Cn2ncccc2=O)CC1(C)C C1(O)(CNC(C2(COC(C)C)CC2)=O)CCN(C(=O)C#CC(C)C)CC1 C1(NC(C(NOC)=O)=O)CN(C(=O)C(Cl)=CCl)C(C)(C)C1 Cc1cccc(C)c1CC(=O)NCCC(C)NC(c1cncnc1C1CC1)=O c1(N2CC3N(CCN4CCC(F)C(F)(F)C4)C(CC3)C2)ncc2cc(Br)cnc2n1 C(=O)(C1=NOC2(CCOC2)C1)NC1(CN(C(c2c(C)coc2C(C)C)=O)C)CC1 C1(CNC(=O)NC(c2nncs2)C)CC2(CCC2O)C1 C1(C(C2CCCO2)NC(C(=O)OC(C)(C)C)=O)CCCOC1 c1(CNC(C2(C(N)=O)CC2)=O)ccccc1CN(C(=O)CC1CCCOC1)C1CC1 C1(COC)CC(O)CN1C(C1CC(NC(=O)C(C)C#N)CO1)=O Cc1cc(F)c(N)cc1C(=O)NC(C)C(C)NC(c1ccc2[nH]ccc2c1)=O C1(C(N2CC(C=CC)C(CCC(C)C)C2)=O)CN(C(=O)CCCOC)CC(C)(C)O1 N1(C(CCCCOC)=O)CC(C)CN(C(C2(C3CC3)CCOCC2)=O)CC1C C1(C(=O)NCC(C)Cn2ccnc2)CCN(C(c2sccc2F)=O)C12CCC2 N1(C(CC)=O)CCOC2CN(C(c3ccc(Cl)c(OC)c3N)=O)CC12 Cc1ccsc1C=CC(=O)NC(C1(CNC(=O)CC(C)CF)CC1)C C#CC(C)(C)C(=O)NCc1nc(C2CN(C(c3ncccc3SC)=O)CC2C)n[nH]1 N1(C(C(CC)CC)=O)CCN(c2cc(F)ncn2)C(C(C)C)C1 c1(-c2nc(NC(c3cccc(F)c3I)=O)sc2)cnc2[nH]ncc2c1 Cc1oc(Cl)nc1C(N1CCOCC1CC(=O)NC(C)CC1(O)CCC1)=O N1(C(=O)OC(C)(C)C)CC=C(C(C)(C)C(=O)NCCOCC2CCCOC2)C1 N1(Cc2onc(CC(C)C)n2)C(=O)CCN(Cc2nc(C(F)F)no2)C1=O CC1CN(C(c2cc(-c3ccnc(F)c3)cs2)=O)CCO1 C1(NC(CC(C)F)=O)CCN(C(=O)C=Cc2ccc(C(N)=O)o2)CC1C Cc1nc(NC(C)CNC(c2ncoc2-c2cnn(C)c2)=O)c2c(C)csc2n1 c1(C(N(C2CCN(C(C3C(C)CCS3)=O)CC2)C)=O)cc2nccc(Cl)c2s1 c1(C(=O)NC2C(C)CN(C(C3CC(S(C)(=O)=O)C3)=O)C2)cc2cccnn2c1 c1(CC)ncc(C(=O)NCCC2CCN(C(c3cc(O)cc(O)n3)=O)C2)c(O)n1 C1(NC(C2(COC)CCCO2)=O)CN(C(=O)Cc2cncnc2O)CC1O C1(CC(=O)NC(C(C)C)CO)CCCN(C(C2(C#N)CCOC2)=O)C1 c1(NC(CN(C(c2ccc(F)cc2)C)CC)=O)ccc(C)nc1OCC(F)(F)F S(=O)(=O)(c1c[nH]ccc1=NCc1cc(F)ccc1F)N(C(C1CCC1)C)CCO c1(C(N(C(C)CN(C)C(C2CC2C(F)F)=O)C)=O)cncc2cccnc12 c1(CCC(=O)NC23CC(NC(=O)C(O)CC4CC4)(C2)C3)cnccn1 c1(C(=O)NC(CN(C(C2(OCC)CCOC2)=O)CC)C)ccc(Cl)nc1O N(C1CCCc2ccoc21)C(C(CC(=C)Cl)NC(c1ncccc1N)=O)=O c1(NC(CNC(C2(SC)CC2)=O)C2CC2)ncnc2scc(Br)c12 CC1CC1C1CC1C(=O)NCCN(CCCCN(C)C)C(c1ccc(CO)nc1)=O c1(C(N(C)CCNC(=O)CC2(CN3CCCC3)CC2)=O)ccc(Cl)cc1 C(=O)(C1=CCS(=O)(=O)C1)NCC1CCC(NC(C#CC(C)C)=O)C1 Cc1cc(CCC(=O)NCC2CCN(C(c3cc[nH]c(=N)c3)=O)C2)ccc1Cl CCC(CCC(=O)NCc1ncnn1C)NC(=O)C=C(C)C(C)(C)C C1(CNC(CC(C)(C)F)=O)COCCN(C(=O)CCc2cncc(F)c2)C1 CN1CCOCC1CNC(=O)CC1CCCN(C(C2CC(N(C)C)C2)=O)C1 C(=O)(CCCCC(=O)CN(C)CCNc1cc(C)ccc1F)OC Cc1cc(C)c(CNC(C2(NC(=O)CC3CCSC3)CC2)=O)s1 C(c1ccccc1[N+](=O)[O-])=CC(N1CCCC2C1CCN2C(c1ccsc1)=O)=O CN=c1[nH]c(=NCc2cc(Br)cs2)[nH]c(=NC(C)c2ccnc(C)n2)[nH]1 C(c1ncccc1C)=CC(=O)NC1C(NC(c2cccc(C)n2)=O)CCC1 C(=O)(C(C)(CC)CC)NC.C(CC(=O)OCC)N1CC1CC C1(CCOC)(C(=O)NCC(C)(C)NC(N)=O)CCN(C(=O)CC(C)C(C)C)CC1 C#Cc1ccc(C(N2CCC3(CC3NC(C3CC(OC(C)=O)C3)=O)C2)=O)c(F)c1 C(=O)(C1=CCCN(C(c2nc(-c3cccs3)cs2)=O)C1)Nc1c(C)cc(Br)cc1 c1(N2CC(N3CCC(O)CC3)C2)nc(N2CCCC(F)(F)C2)c2c(F)cccc2n1 c1(SC(C)(C)C)cncc(CNC2(c3nnnn3CC(F)F)CSCCSC2)c1 N1(C(c2cc(OC)ncc2)=O)CCN(C(c2oc(C)cc2C)=O)C(C)C1C N1(C(CC2N(C(CCCNC(C)=O)=O)CC(F)C2)=O)CCCN(C)CC1 c1(-c2cn(CC3CN(C(CC)=O)C3)nn2)ccccc1SC.C12CCCN1C2 C#CC1(COC(C)(C)C)CCN(C(=O)NCc2nc3c(s2)COCC3)C1 N1(C(C(C(CC)CC)C)=O)C2CCCC1CC(NC(C1(O)CCCCCC1)=O)C2 C(=O)(CCC(C)(C)[N+](=O)[O-])NCC12C(CN(C(CCC(=C)Cl)=O)C1)C2 N1(C(c2ccc(OC)cc2)=O)CCC2(CC1)CC(NC(c1ccon1)=O)CCO2 N(C1CCc2cccnc21)C(=O)CC1COCCN1C(=O)C1CC1 Cc1cc(C(=O)NC2CCN(C(c3sc(Br)cc3Br)=O)CC2O)c(F)c(F)c1 C1(NC(=O)CSC2CCS(=O)(=O)C2)CCc2ncccc2C1 C1(NC(CC(CC=C)(C)C)c2nnnn2C2CCCCC2)CCCC2(CC1)CC2 CC(C)(C)C(=O)NCC(=O)NC1C=CC(CC(=O)NCC(c2ccsc2)O)C1 c1(OCCN(C(=O)CC2CCNC(=O)C2)CC)cccc(C)c1 c1(CCC(N2C(COC(C)(C)C)CCC2)=O)ccc(Cn2ccccc2=O)cc1 N1(c2ccc(C#N)nc2)CCC(NC(=O)C(F)(F)CC2CC2)C2(CCC2)C1 c1(CC(N2CC(F)(CNC(CNC(C)=O)=O)C2)=O)ccc(CS(C)(=O)=O)cc1 CCC(C(=O)N1CCC(N(C)C(C2CCOCC2(C)C)=O)CC1)C(C)(C)CC C(=O)(C(F)(F)C(C)(C)O)NC1C(CNC(c2cccc(COC)c2)=O)COC1 N1(C(COCCCOC)=O)CCC(C)(C)C(CNC(c2cnc(C)cc2C)=O)C1 C12CCCC1C(=O)N2.c1(C(=O)NC(c2cn(C)cn2)C)cc(C2CC2)[nH]n1 C1(CNC(c2nc(CCOCC)sc2C)=O)CCCC2(CCOC2)O1 C1(C)(NC(c2ccn(CC)n2)=O)CCCCC1C(N1CCC=C(Cl)C1)=O N1(C(C2COCC(C)O2)=O)CCN(C(=O)Cc2ccccc2Cl)C(CO)C1 c1(C(=O)NC(CNC(C=NOC)=O)(C)CC(C)C)cc2ccccn2n1 C1(CNC(C=C(CCC)C)=O)COCCN1C(=O)CCc1cccc(C(F)F)c1 N1(CC(=O)NCC(=C)CCOC)CCC(c2ccccc2)(Cc2nnc(C)o2)C1 c1(CNC(C2(C)CN(Cc3c(C)cco3)C2)=O)cccc(SC(F)(F)F)c1 O(NC(=O)C(CCC1CC1)NC(=O)Cn1cccc1)CC=C c1(C(=O)NCC2C(C)CN(C(=O)CNS(C)(=O)=O)C2)cnc2nc(O)ccc2c1 Cc1ccc(C(N2CC(=O)CC2C(N2CC(C(N)=O)C2)=O)=O)cc1O CC(CC(F)F)C(=O)NCc1ccc(C(=O)NCC2(CO)CC23CCC3)o1 c1(N2CC(CNC(c3cc4ccccc4o3)=O)OCC2)ccn2ccnc2n1 Cc1nc2cc(O)nn2c(C)c1S(=O)(=O)N(CC(F)(F)F)CC1CCCO1 N1(CC(=O)NCCN(CCC)C(c2cc(Br)co2)=O)OC(C)(C)CC1=O n1(CC(=O)NCCN(C(CC2CC(C)C(C)(C)C2)=O)C2CC2)cc(F)ccc1=O C1(OC(=O)CCOC2CCOC2)CC=CCC1C(F)(F)F C1(CNC(c2c(C)nc(C)[nH]2)=O)CC(NC(c2c(F)cccc2Cl)=O)C12CCC2 N1(C(C(C)OCC2CC2)=O)CCC2CCCC12C(=O)NC1CC2CC1CC2(C)O n1(CC(=C)C)c(N2CCC(c3ccccc3)C2)nnc1CC(CC)CO c1(C(C)C)ncc(C(N2CCCC2CCNC(=O)CN2CCCC2C)=O)o1 N1(C(C2(C(C)(C)OC)CC2)=O)CCC2C(NC(c3ncc(C)cn3)=O)C2C1 N1(C(CC(C)OC)=O)CC(NC(=O)CN(CC(=O)NC(C)C)C)C(O)C1 c1(CN(CCOCCN(C(C(C)NS(C)(=O)=O)=O)C)C)csc(Cl)n1 N1(C(C(=O)NC(C)C)CCC2(C)CCOCC2)CCC(CCO)(CO)CC1 C(=O)(CC(C)C(=O)N(C)C(c1cccnc1SNC)=O)OCC.c1(C)cnccn1 N1(C(CCC=C=C)=O)CCCCC(CNC(=O)COc2ccc(C(C)C)cc2)C1 c1(C(N2CCC(O)(C(C)CNC(=O)C(N)=O)C2)=O)c[nH]c2ccc(F)cc2c1=O c1(C(=O)NC2CC3CN(C(c4scnc4Cl)=O)CC23)nncc2c1CCCC2 n1(CC(=O)NC(C(=O)N(CC(C)(C)C)CCC)CC2CC2)c(O)nnc1O C1(CCNC(Cc2n(C)nnc2)=O)CCCN(C(C2(C#N)CCCO2)=O)C1 CC(CCCCNC(=O)C(C1CC1)CC1CC1)NC(C1COC1)=O C1(CCC)CN(C(=O)C(O)c2ccsc2)CC1NC(=O)Cn1nnnc1C C1(C(=O)Nc2ccc(C3CC3)cc2)CC2(CCN1C(C1CC3CCC3C1)=O)CC2 N1(C(C2(F)CCN(C(CNC=O)=O)C2)=O)CCCC2OCCC12 c1(C(N2CC=CC(NC(C(C)S(N)(=O)=O)=O)C2)=O)cncc2cccnc12 c1(OCC)ccc(CC(=O)NCC2(C)CCCN2C(c2nc(=O)n(C)[nH]2)=O)nc1 C1(CC(=O)NCCNC(C(C=C)c2ccccc2)=O)CC2(CCC2)CCO1 n1(CC(C)C)nc(C2Cc3ccccc32)nc1-c1ccc(-c2nn[nH]n2)nc1 C1(NC(CNC(C)=O)=O)CCN(C(C2CSC2)=O)C12CCC2 C1(C(=O)NC(CNC(C(COCC)(C)C)=O)(C)C)CC12CC(C)(C)C2 C1(CNC(C2(COC)CC=CC2)=O)CCC(C)(C)CN1C(c1oncc1CC)=O C1(NC(CCCCCC)=O)CN(C(C2C(C)C2C)=O)C2(CCC2)C1 CS(=O)(=O)c1cscc1C(N1CC(NC(=O)CCCNS(C)(=O)=O)C2(CC2)C1)=O C(=O)(CCCCCN1CCC(C(=O)O)C1)NC(C1CCCC(C)C1)CC CC(CC(=O)N1CCCC1(C)CCC(=O)N(C)CC1(O)CCCC1)C(F)(F)F N1(C(c2cnn(C)c2Br)=O)CCC(CO)C(NC(c2cc[nH]c2)=O)C1 c1(CC2C(=O)O2)ccc(C#N)cc1.Cc1nc(C)c(C(=O)NC(=O)C(C)C)s1 CCC(C(=O)N(CC(C)NC(=O)CCCN1CCCC1)C)n1cncn1 CCCS(=O)(=O)C(C)C(=O)N1CC(NC(c2cc(C3CC3)on2)=O)C(N=[N+]=[N-])C1 CC(O)C(C)C(=O)NCc1cc(C(=O)NC2CCC(CN(C)C)CC2)ccn1 CCC(CC)C(F)C(=O)NCCC(O)C(=O)N1CC(O)CC1CO C1(NC(c2c(SC)nccn2)=O)CCN(C(=O)Cn2c(C)ccc2C)C12CC2 N1(C(C=CCC)=O)CCC2CCCN(C(=O)CCn3cc(C(=O)OC)nn3)C2C1 c1(NC(=O)NCCC2CC(OC)C2)ncccc1I C(c1ccc(C)cn1)=CC(=O)NCCCOCCN(C(CN(CCC)C)=O)C c1(CNC(CCSCCC)=O)ccc(NC(C2(COC)CC(F)(F)C2)=O)cc1 C1(CNC(C(CC)N(CC)CC)=O)CN(C(c2snc(O)c2Cl)=O)CC1(F)F C1(NC(c2c(CC)onc2C)=O)CC2(C1)CN(C(=O)C(C)=C1CC1)C2 c1(C(=O)NCC2N(C(C(C)OCCOC)=O)CC3(CC3)C2)c[nH]c2nccc-2c1C CCS(=O)(=O)CCCc1nc(C2CN(c3ccc(C)cc3)CCO2)no1 c1(C(=O)NC2CC(NC(C3(CO)CC(C)(C)C3)=O)C2)nnn2c1CCCC2 C1(NC(C2(CC=C)CC=CC2)=O)COCCN(C(=O)C(C)CC(N)=O)C1 C1(N(C(=O)Cn2cnnc2)C)CCC(NC(C2CC2CO)=O)CC1 CCC(C)CCC(O)CC(=O)N1CCCC2(C1)CN(C(=O)CSc1nncs1)C2 c1(C(=O)NCC2C(C)CCN2C(=O)CCC#N)c(Cl)ccc2cccnc12 c1(OC)cc(OC)cc(C(C)N)c1.c1(C2CCN(C(C)=O)C2)cccc(OC)n1 N1(C(CCCCCC)=O)CCN(C(c2nccnc2C)=O)CC12CCC2 C(=O)(C1=COCC1)NCC(C)(C)NC(C(CC)N(CC)CC)=O CCCCC(C)CCC(=O)NCC(c1ccccc1)N(C)C(C1C2COCC12)=O Cn1cc2ccc(C(=O)NCCNC(C3CCCN3c3cnccn3)=O)cc2n1 CC1Cc2ccc(Br)cc2CN1Cc1sc(Cl)nc1Cl N1(C(CCCC(=C)C)=O)CCCC2(CCN(C(c3c(C)oc(C)c3C)=O)C2)C1 c1(CC(=O)NC2C(NC(C3C(C)OCCC3)=O)COC2)cc(Cl)ccc1Cl C1(C(=O)OC)CC(C(N2CC(CO)(NC(=O)CCN3CCCC3)C2)=O)C1(C)C N1(C(C(c2c(C)cccc2)C)=O)CCN(C(=O)CC2CN(C)C2)CC1C(C)C C1(NC(C(c2cccc(Cl)c2)CC)=O)CCC12CN(C(=O)CN1CC=CC1)C2 CCCS(=O)(=O)C(C)C(=O)NC1CN(C(=O)C2=C(C)CCCC2)CC1C C(=O)(N=c1cc(-c2cccc(F)c2)[nH][nH]1)C1(C)CN(C(C2CC3CCC2C3)=O)C1 C1(C(C)NC(c2cnc(C)o2)=O)CCN(C(=O)CC2CCCN2C)CC1 N(C(=NCCCCl)NCc1nc(C(F)(F)F)cs1)C1CC(OC(C)C)C1(C)C CC1CCC(NC(=O)CCC2CC(F)(F)C2)CN1C(=O)CCC[N+](=O)[O-] C1(CNC(=O)C(O)C(F)F)CCCC2CN(C(=O)C=Cc3ncc[nH]3)CC12 c1(C(=O)NC2C(NC(c3nccc(C)n3)=O)CS(=O)(=O)C2)c(F)ccc(O)c1F CC1(C)CC(CC(=O)NC2CC2CN2CCC2)CN1C(C1CC(=O)OC1(C)C)=O c1(C(=O)NC2C(NC(c3ccc(CC)o3)=O)CC2)sc(-c2ncccn2)nc1C N#CC1CNCC12CC(NCCn1cc(N3CCOCC3)c(=O)cc1Cl)C2 C(=O)(C1=C(F)CN(C(C2CC23CCC3)=O)CC1)N1CC(=O)NCCC1 c1(COC)ccnc(N(C)CCN2CCN(C(c3cc(C(C)C)[nH]n3)=O)CC2)n1 Cc1cc(N2CC(C(N3CC(C)(NC(c4cnsc4)=O)C3)=O)CC2=O)cc(C)c1 c1(C(=O)NC2C(NC(C(CC(C)C)O)=O)C2)ccc2c(O)nnc(O)c2c1 C1(NC(CC2C(C(=O)OCC)C2)=O)CCC(NC(c2occ(C)c2C)=O)CC1 N1(C(c2cncc(Cl)c2)=O)CCC2(CNC(C34CCCC3CCC4)=O)CCCC12 N1(C(CCSC)=O)CCC2(CCC2)C(CNC(=O)C(C)CCc2ccccc2)C1 C1(C)(CNC(CSCC=C)=O)CN(C(c2c(-c3ncco3)noc2C)=O)CCO1 c1(C(CC(=O)NC(C)CCCCNC(=O)C(O)CF)C2CC2)cc(F)ccc1F N1(C(c2c(C(C)C)csc2)=O)CC(NC(c2nccn2C)=O)CC(O)C1 N1(CC(=O)N(CCN2CCN(C(=O)Cc3cnsc3)CC2)CC)CC2C=CC1C2 CC1CC(NC(c2ccc(Br)cc2)=O)CN(C(c2ccccc2CC(=O)O)=O)C1 c1(OC)cc(Br)c(C)nc1NC(C1(O)CCN(Cc2cncnc2)C1)=O c1(NC(c2cnc(N(C)C)o2)=O)cnc(Cl)cc1C(=O)Nc1c(Cl)cnnc1Cl N1(C(COC(C)C)=O)CC2(CCC(CNC(c3cc4cccnc4s3)=O)O2)C1 c1(Nc2ncc(C(=O)NCc3cnc(C)[nH]3)nc2)cncc(Cl)c1C C1(CCC)CN(C(c2nc(O)sc2C)=O)CC1NC(=O)CCOC1CCCCC1 c1(C(N(CC(C)NC(c2ccccc2OC(F)F)=O)C)=O)cccn2nccc12 N1(C(Cc2c(C)scc2)=O)CCC(C)C(NC(=O)CC(C)C)C1C CC(C)C(CC(=O)NCC(C(C)(C)C)NC(c1cccc(C(N)=O)c1F)=O)C(C)C c1(CC(=O)NC2CC3CN(c4c(C#N)ccnn4)CC32)ccc2cccnc2c1 Cc1nn(-c2ccccc2)cc1C(N1CCCCC1C)C(=O)NCCN1CCOCC1 C(=O)(C1CCc2c(Cl)cccc21)NCC1(CN(C(CCCC(=O)OC)=O)C)CC1 c1(C(=O)NCC2C(C)CN(C(c3sccc3F)=O)CC2)cnn2ccccc12 Cc1c(Br)c(C(N2CCOCC2CC(=O)NCc2cc(Br)nn2C)=O)nn1C c1(NC(C2C(NC(C3(OCC)CCC3)=O)C2)=O)ccc(Br)cc1Cl C1(C(N(CCCCCNC(c2cccc(SCC)c2)=O)C)=O)CC2COCC2C1 C1(O)(CNC(CSCCC)=O)CCCN(C(=O)C(C)C(F)F)C1 C(CC(=O)N(C)CCN1CC=CC1)N(C)CCO.C1=CNC1=O CC1(C)CC(NC(C2(N3CCOCC3)CC2)=O)CCN(C(=O)CN=S(C)(C)=O)C1 C1(C(N(C)CC2CC(C)C2)=O)C=CCN1C(C1CC1C#N)=O Cc1cnc(Cl)nc1NC1CCC(NC(=O)Cc2csc(C3CC3)n2)CC1 N1(C(Cc2c(C)cccc2)=O)CC(C)(C)CC1C(N1CC(F)(F)C1C1CC1)=O C(=O)(C(O)CC(C)C)NCC(CC)(CC)NC(C1CCN1S(C)(=O)=O)=O C1(NC(=O)Cc2ccccn2)C2CCN(C(c3ccc(=O)oc3)=O)C12 C(=O)(CC(C)C(=O)N1CCC1(C)CC(=O)NCCC(C)C(F)(F)F)OCC c1(C(=O)NC(C(=O)OCC)Cc2ccccc2)cncc(F)c1 C12(C(=O)NC3C(NC(=O)CC=C(Cl)Cl)COCC3)CCCN1CCC2 N1(CC(=O)N(C2CCCC2)CC)CCC(C(=O)NCC(c2ccc(C)o2)=O)CC1 N1(C(CCCc2nnc(C)n2C)=O)C2CCC1C(NC(c1cc(F)c[nH]1)=O)C2 C1(C(=O)NC2CCN(C(COCCC)=O)C2CC)CC2CCC(C1)C2O C(CCCCF)NC(C1(NC(COCC(=C)C)=O)CSC1)=O CCC(C)C(C(=O)NC)N(C(=O)C(c1cnn(C)c1)C)C c1(CC(N2CCN(CC(C)(C)NC(CC(C)(F)F)=O)CC2)=O)ccc(F)cc1F C=CCC(CNC(=O)C(c1cncn1C)OC)NC(c1cc(CCC)[nH]n1)=O Cc1cc(C#N)ccc1C(=O)N(C1(CC(=O)NCC2C=CCCC2)CC1)C Cc1nc(C(=O)NCC2C3CCCOC23)cc(O)n1.C12CCCCC1NC2=O c1(C(=O)NC2CC(C)N(C(=O)C(C)NS(C)(=O)=O)C2)cc(O)cc(C#N)c1 C1(CCNC(C=C(CNC(CCNC(=O)OC)=O)C)=O)CC(F)(F)C1 c1(CC(C(=O)NC(c2noc(CC(F)(F)F)n2)C(=O)OC)=O)ccc(O)cc1 C1(CC(=O)N(CC(=O)NC(c2nc(C)no2)C)CCC)CCN(CC)C1 N1(C(c2nc(C)c(F)cc2)=O)CC2CCC(NC(c3ccc(Br)nc3F)=O)C2C1 C=CC1(C(=O)NC2CCCC2OCC)CCN(C(=O)C(C2CCCCC2)F)C1 CC1CCc2nc(C(N3CCC4CC4(NC(=O)CNC=O)CC3)=O)cn2C1 C1(NC(C(CC)COC)=O)C(C)(C)C(NC(C2CC(OC)(OC)C2)=O)C1(C)C C(CC1=CCN(c2cc(C(F)F)ncn2)CC1)NC(Cc1ccc(C)cc1Br)=O Cc1cc(C2CC2)ccc1C(N1CC2CC(NC(=O)C(C)C(F)(F)F)C1C2)=O n1(CC)nc(C)c(C(=O)NCC(CNC(=O)CCC(=O)OC)OC)c1Cl.OC Cc1coc(C(C)(C)C)c1C(=O)NCC1CCC(NC(c2cnnc(O)c2)=O)C1 C=CC(C)CC(=O)N1CC(CCCCNC(C2C3CCCC23)=O)C1 C1(C)(CNC(COCC=C)=O)CCN(S(=O)(=O)CC(C)C)C1 C#CCCCCCC(=O)N1C2CCC1CN(C(C1CC1(c1ccccc1)C)=O)C2 c1(OC)ccc(OC)c(C(=O)NC(C)CNC(c2ccccn2)=O)c1 C1(CN=[N+]=[N-])COCCN1C(c1ccc(CNC(c2nn(C)cc2Cl)=O)nc1)=O C1(CNC(C(c2ccc(C)cc2)(C)F)=O)CCCCCN1C(=O)C(O)CC(N)=O c1(CC)cc(=NC(=O)c2sccc2CNC(=O)CC2COC(=O)C2)[nH]n1C C(C)(CO)(C(=O)NC1CCN(C(C)C)CC1)NC(c1c(C)cns1)=O C1(C)(COC)CCCC1NC(C12CC1CN(C(C)=O)C2)=O C(C(C(C)C)NC(CC1CC(OC)C1)=O)NC(C1CCCC1)=O.N1(CC=O)CCCC1 C12(CCC)CN(C(c3cnn(C)c3)C(=O)NC3CC3)CC(CO)(C1)C2 N1(C(CC(C)NC(c2cnc3n2CCC3)=O)=O)CCC(O)C1(C)C c1(NC(c2cnn3c2OCC3)=O)c(Br)cc(Cl)cc1Br CC1(C)CC(NC(=O)CC2CCC(=O)C2)CN1C(=O)C(N1CCCC1=O)N N1(C(CCC2(C)CC2)=O)CCC2(CCCN(C(C34CCCC3C4)=O)C2)CC1 CC(C)C(C)(C)C(=O)NCC(C)(C)OCCNC(=O)CCc1ccncc1 C(=O)(C(C)(C)C(N)=O)N1CCC(CN(C)C(c2cnn(CC(F)F)n2)=O)CC1 C12(F)COCCN(C1)C(=O)N2.C(C)(C)(COCCO)OC(C)(C)C C1(F)(CNC(=O)C=CC(F)(F)F)CCCN(C(c2c[nH]c(=S)cn2)=O)C1 C1(C(=O)NC(CNC(=O)CC(C)SC)C2CC2)(OC)CCCC1 C12(C(N(CC(=O)NC(C)C)C)=O)CCC(CC1)N(C(=O)C(F)CC1CCCC1)C2 N1(C(c2c(CC)c[nH]c2)=O)CC2CN(C(c3c(C(F)(F)F)ncn3O)=O)CCC12 N1(CCCOC)CCN(C(=NCCC(C)(C)C)NCC(C)(C)C)CC1 c1(C(N2CC(NC(C3C(CC)OCCC3)=O)C(SC)C2)=O)cc(O)nc(O)n1 c1(OC)cccc2c(=O)c(C(=O)NC(C)C(C)NC(=O)COC(C)C)c[nH]c12 C1(C(=O)NC2CCN(C(c3c(C)[nH]c(C#N)c3)=O)C23CC3)CC2(COCCO2)C1 c1(C(=O)NC(C2CCN(C(CCC)=O)C2)C)ccc(Br)c(F)c1OC C1(CC)CN(C(=O)Cn2cccc(C)c2=O)CCN1C(c1cn(C(C)C)cn1)=O CCC(O)CC(=O)N1CCCCC1CCNC(=O)C(c1ccc(C)o1)C Cc1cc(Cl)ccc1OCC(=O)NCC1(NC(c2onc(C)c2C)=O)CC1 c1(CC(=O)NC(C)CNC(c2ccnc(SC(F)F)c2)=O)ccc(Cl)cc1F N1(C(C#C)C)CCN(N2CCN(C(C)=O)C(C)C2)CC1 C=CCN=C(NCc1csc(Cl)c1)NC1CCC(C#N)C1 N1(C(C(CC)OCC)=O)CC(NC(=O)C2=NOCC2)C2(CCS(=O)(=O)CC2)C1 c1(C(=O)NC(CN(C(c2ccnc(N3CCCC3)c2)=O)CC)C)ccc(O)c(F)c1 C(=O)(C(O)P(C)(C)=O)NCC1CC(NC(c2nn(C)c(Cl)c2)=O)C1 c1(OS(C2CC(CCC)C2)(=O)=O)ccnc2[nH]c(C)nc12 C12(C(N3CC4CC(OC)C4C3)=O)CC(CN(C(C3CC34CCOCC4)=O)C1)C2 N1(C(C2C(C#C)C2)=O)CCC2(CC(NC(=O)C(CC(C)C)N(C)C)C2)C1 c1(OC)ccc(C(N2CSCC2C(=O)NCCSC2COC2)=O)cc1C N1(CC)CCCC(C(=O)N(CC(C)CNC(C2(CC#N)COC2)=O)C)C1 Cc1noc(C)c1CC(=O)NCCOCCN(C)CCC1CC(F)(F)C1 N1(C(C2=C(C)S(=O)(=O)CC2)=O)CCCC(C2CCCN(C(=O)C(O)C(C)C)C2)C1 N1(C(C23N(C(C(CC)=CCCC)=O)CC(CO)(C2)C3)=O)CCCCC(C)(F)C1 CCCCCCC(C)(CC)C(=O)NCCNC(=O)C(C)(Cl)CCl C1(NC(c2c(C)nc(CO)nc2)=O)CC2CN(C(=O)Cc3cocn3)CC2C1 C1(C(N(CCN(C(C2CCC(OC)C2)=O)C(C)C)C)=O)CCN(C)CC1 N1(C(c2c(N)cc(CC)cc2F)=O)CC2CC(C)N(C(c3csc(Cl)c3)=O)C2C1 Cc1ccnc(C(F)(F)C(=O)N(C2CC(c3ccccc3)C2)C)n1 N1(C(C(C)CN(C)C)=O)CCC(NC(=O)Cn2ccc(=N)[nH]2)C(C)(C)C1 C1(C(CC(=O)OCC)OC(C2CC(=C3CC3)C2)=O)COC(C)(C)O1 N1(C(CC(c2ccc(C)cc2)C)=O)CCOCC(NC(C2CCS2(=O)=O)=O)C1 Cc1ccc(C(=O)NCCC2CN(C(C3(C)CC=CCC3)=O)CCO2)c(N)c1F C1(C(NNC(c2nn(C)c(=O)cc2)=O)=O)CCc2ncncc2C1 N1(C(C2(NC(=O)CN3CC=CC3)C(C)(C)C2)=O)CC2(CC=CC2)C1 N1(C(c2c(OC)noc2C)=O)CC(CNC(=O)CC(C)(C)OC)C2(CCC2)C1 N1(C(COC(CC)C)=O)CC(NC(c2cc(SC)n(C)n2)=O)C(C)C1 Cc1ccc(C(F)(F)F)cc1C(=O)Nc1ccsc1C(=O)Nc1cn(C)nc1C N1(C(C=CCOC)=O)CC(C(F)(F)F)CC(C)C1.C1C(C(C)C)CO1 C1(C)(C(=O)NC2(CC=C)CCN(C(=O)CC(C)(C)C3CC3)CC2)COC(C)(C)OC1 c1(NCC2(N(C(C(C)(C)C3CCCC3)=O)C3CC3)CCC2)ncc([N+](=O)[O-])cc1F CC1CCCC(OCC(=O)NCC#CCNC(C2(C(C)(F)F)CCOCC2)=O)C1 c1(C(N2C(CNC(C(CSC)O)=O)CC(O)C2)=O)cc(C)c(C)cc1Cl Cc1cc(F)ccc1S(=O)(=O)N1CC2CCC(C1)C2NC(=O)CCC1CCOC1 C1(CC)CCC(C(=O)NCc2nc(CNC(c3coc(Cl)c3)=O)cs2)C1 c1(C(C(COCC)=O)=O)coc(S)c1.C(CNC(C1CC1C(N)=O)=O)(CO)N C1(CCNC(=O)CSC2CC2)CCCCN1C(=O)CCCCSc1ccccc1 C(C(C)(C)CC(F)(F)F)NC1=NCCN1.C1(NCSC)COC(C)(C)C1 N1(C(CCCSCC)=O)CC(CNC(c2csnc2-c2ccccc2)=O)C(O)C1 C1(OC)CC(NC(=O)NCCn2c(C)ccc2C)CC1NC(=O)OC(C)(C)C c1(C(N2CC(NC(C3N(CCC)CCC3)=O)C(OC)C2)=O)cc(C)c(O)nn1 C1(F)(C(N2C(C(=O)NCc3cc(COC)on3)CC(O)C2)=O)CCC(C)CC1 CCC(C)(C(=O)N1CC(CN2CCN(C(C3CCCN3CC)=O)CC2)C1)C(N)=O C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC(NC(c2c(CC)nc[nH]2)=O)C(C)C1 C(=O)(C1=C(C#N)CCC1)N1C(C(F)(F)F)CC(OC)C1.C1(=O)CCN1 c1(COC)cc(C(=O)NC(C2CCCN2C(c2nocc2Cl)=O)(C)C)cs1 C(CC(C)(C)C#N)(C(=O)NCC1CCC(F)(F)CC1)N(C1CCOC1)C N1(C(c2c(C)nc(C)o2)=O)CCCC2CN(C(C3CC(N=[N+]=[N-])C3)=O)CCC12 C1(NC(C2CN(C(C)C)C(=O)C2)=O)CC2(C1)CC(NC(=O)C1=COCCC1)C2 C12(NC(CN(CC(C)(C)C)C)=O)CCCC1N(C(=O)C=C(Cl)Cl)CC2 c1(OC(CC)CNC(=O)N(c2occc2C)C(C)(CO)C2CCC2)cccnc1 C(=O)(CC(C)(C)N(C(=O)Cc1ccccc1O)C)NCC(=O)NCCOC Cc1ccnc(NC(C)CCNC(c2ncn(C(C)(C)C)n2)=O)n1 C1(NC(c2cccc(NC)n2)=O)CCN(C(c2ccc(O)c(OC)c2)=O)CC1C Cc1cc(C#N)cc(C(=O)NCC2CCN(C(=O)COCCCF)CC2)n1 N1(C(C=CCC)=O)CC(C(=O)Nc2nn(C)c(N)c2C)CCC(O)C1 c1(OCC(=O)NC2C(NC(C(C)NC(C(C)C)=O)=O)C2)cccc(Cl)c1Cl c1(C(N2CCC(NC(CC)=O)CC2)=O)csc(N=S(C)(C)=O)n1 C(CC(=O)N1CC(SC(F)F)C1)(C(C)CC)NC(C(C=CC)O)=O c1(OC)ccc(C(=O)NCC2CC3CN(C(=O)C(O)CC4CC4)CC23)nc1Cl CC(C)C(O)C(C)C(=O)NC1CCCCC1NC(=O)CCCN1C(=O)CNC1=O C(=O)(CCCCCCCCCO)NC1C=CCN(C(c2c[nH]c(=N)o2)=O)C1 NC1CCCN(C(=O)C(=O)NCc2nc(-c3ccccc3O)cs2)C1 c1(C(N(CC(C)CNC(=O)CNC(=O)CN(C)C)C)=O)ccc(Cl)cn1 C12(C(N(C3CN(C(=O)CSCC4CCCCO4)CC3O)C)=O)CCC(C1)C2(C)C C(=O)(C(C(C)(C)OC)OC(=O)C(C(C)N)NC(c1ccccc1)=O)OC CC1=CCC(C(=O)NC2C=CCN(C(c3sc(C(C)(C)C)nc3C)=O)C2)CC1 Cn1c(C(N2CCCC(CNC(C3(CF)CC3)=O)CC2)=O)cc2ccsc12 N1(C(CCN(C(C)=O)C)=O)CCC2(CC(C(=O)NCc3c[nH]nc3C)CO2)C1 N1(CC)CC(COC(CC(C)Cc2nccc(C(F)(F)F)n2)=O)CCC1=O C1(NC(c2cc(OC)ns2)=O)CN(C(c2cccc(Cl)c2F)=O)C2(CCCC2)C1 c1(OC)ncccc1NC(=O)C(C)CCc1ccc(F)cc1.N12CC(C1)NC2=O CCCCCC(=O)N1CC(CC(C)NC(=O)CC(O)CN(C)C)C1 C12(C(=O)NCC(C)(C)O)COCC1CN(C(=O)CC1COCCO1)C2 C1(COC)(NC(=O)C(C)c2ccsc2)CCN(C(=O)C(F)=C(C)C)C1 Cc1nc2ccc(-c3noc(C(N4CCSC(C(=O)NC5CC5)C4)=O)n3)cc2o1 c1(OC)ccccc1C(CNC(=O)C=CC1CCCN1C)NC(=O)C(C)(Cl)Cl c1(C(N2CCN(C(CSc3c(C)nn(C)c3Cl)=O)CC2)=O)ccc2c(n1)CCC2 C1(CNC(C(CC)=CC)=O)CN(C(=O)CSc2ccccc2)CC12CCOCC2 c1(C(N2C(CCNC(CC(C)OC)=O)CCC2)=O)cncc(Cl)c1C C1(C)(C(N(CCC2CCN(C(C(CSC)C)=O)CC2)C)=O)CCN(C)C1=O Cc1cc2c[nH]nc2cc1-n1cc(C(=O)OCC2(C)NC(=O)NC2=O)nn1 c1(C(=O)OC)cncnc1NC(=O)NC(c1ccc(C(F)(F)F)nc1)c1cscn1 C(=O)(C(O)CCCNC(=O)Cc1ccccc1C)NCCC(C(=O)OC)O c1(C(C2CC2)NC)ccc(OC(COC)=O)nc1.C12CCC(C1)C(=O)NC2 Cc1sc(N)c(C(=O)N(CC(C)CNC(C2(N(C)C)CC2)=O)C)c1C c1(C(N(CCCN(C(=O)CC2(O)CCC2)C)C2CCC2)=O)ccnn1CC1CC1 C1(NC(C=CSC)=O)CCC(NC(c2cncc(-c3ccncc3)c2)=O)CC1 C1(CNC(CC(C)SC)=O)CCN(C(=O)CSCc2ccc(C)cc2)C1(C)C C(C)(C(=O)N(C)CC1CC1C)(C1CCC1)NC(C(C)=CC(C)(C)C)=O C1(CNC(C(COC)C)=O)CCN(C(=O)Cn2cc(C#N)cn2)C12CCC2 C1(C#N)(NC(CCSC)=O)CCN(C(=O)NC(c2ccccc2)C)C1 CC(C)(C)S(=O)(=O)CCN=c1[nH]c(=NCC2CC23CCC3)[nH]c2c(F)cccc12 C(CC(C(=O)N(CCC(C)C)CC)NC(C1CC(O)C1)=O)=CC CCC(CC)C(=O)NC1CN(C(=O)C(F)Cc2ccccc2)CC1c1ncc[nH]1 C1(CNC(c2c(COC)nn[nH]2)=O)CC(NC(=O)C=CS(C)=O)CCO1 c1(C(=O)NCC(N2CC(C(=O)Nc3nccs3)C2)=O)ccn(C2CCCCC2)n1 N#Cc1ccc(C(=O)NCc2ccc(C(=O)NCC3(F)CCC3)o2)s1 C12CCC(C1)NCC(=O)NC2.C1(C(=O)OCc2ccccc2)CCCOC1 c1(C(N2C(Cn3cc(COC(C(=O)OCC)CC)nn3)CCC2)=O)ccnnc1C N1(C(c2ccn(C)c2)=O)CCN(C(C2CC2C2CCCO2)=O)C2COCC12 N1(C(c2cccc(C(=O)OCC)c2)=O)CCC(C)(CNC(=O)C#CC(=O)O)CC1 C1(CC(=O)N(C)CC2C(NC(C(Br)=C(C)C)=O)CCC2)CCN(C)C1=O N1(C(c2cc(C)ncn2)=O)CC(C(=O)NCCCCC2CCCC2)CCC1(C)C c1(CC(=O)NC(c2cc(Cl)sc2Cl)CC)ccccc1[N+](=O)[O-] CCC(CC(=O)NCC1CC(C(C)(C)C)CN(C(=O)CN=S(C)(C)=O)C1)C1CC1 C1(C(F)(F)F)(CNC(CN(C(COCC)=O)C)=O)CCN(C)C1 CCC(C)CCCC(=O)N(C)CC1CCCN(C(C2(NC(C)C)CC2)=O)C1 C1(NC(C(CCC)O)=O)CCCC2CN(C(=O)C(F)(F)COC)CC12 CC1(C)C2CCC(C(=O)NC34CCCC3CN(C(=O)C3=CCOC3)C4)C1C2 c1(C(=O)NCC2C(NC(C(C)(C)C3CCOCC3)=O)C2)ccn2nccc2c1 N1(C(c2nc(C)oc2)=O)CCCC(C(C)C(N2CCC(F)(CO)C2)=O)C1 Cc1ccc(O)nc1C(=O)NCC1CSCCN1 C1(NC(C(CCC#C)O)=O)CN(C(C2(CCC)CC2)=O)CCC1(C)C CCCC(O)CC(=O)NCCC1(O)CCN(C(c2ncn(C)c2C)=O)C1 c1(C(=O)NC2C(CNC(CCCC(=C)C)=O)COC2)ccc2nc(O)n(C)c2c1 CN1C(=O)CCC1C(=O)NCCCNC(c1sccc1Br)=O C1(OC(c2c[nH]nc2CCC)=O)CCCCC1CNC(c1nnc(S)n1C)=O C(=O)(CC(CNC(C1(C)CC(F)C1)=O)OC)NC(c1nccs1)CC C(=O)(CC1OCCc2sccc21)NCCC(C)N(C(c1[nH]cc(C)c1)=O)C c1(OC)nc(NC(C2CCC(NC(C3CNC(=O)CO3)=O)C2)=O)cc(O)n1 C1(C)(NC(CCC(C)SC)=O)CCCN(C(c2n[nH]c(C)c2Br)=O)C1 c1(C(=O)NCCC2(NC(c3cc(F)c[nH]3)=O)CC2)ccc(-n2ccnc2)cc1 c1(C(N2CC(CCCCNC(CCC#CC)=O)C2)=O)cc2cc(Br)ccc2[nH]1 C(CNC(=O)CC(=O)NCc1cn(C)nc1C)(CC(=O)NCC1CC1)OC Clc1ccc2c(c1Cl)CCC2NCc1nnnn1Cc1ccccc1 Cc1ccc(CN2CCN(C(c3cccc(C#N)c3C)=O)C(C)C2)c(O)c1 C(CN=c1[nH]c(N2CCC(CC(N)=O)CC2)nc2ccccc12)c1n(C)cnc1 C1(C)(CNC(CN(C(C(C2CCCCC2)C)=O)C)=O)CCC(=O)C1 n1(CC)cc(C(=O)N(C2CCCN(C(=O)C=CC3CCC3)C2)CC)c(C2CC2)n1 Cc1cc(Cl)c(C)c(C(=O)NC2CN(C(=O)C(C)(C)CC(C)C)CC2C)c1N C1(CCN(C(C)=O)C2CC2)CN(C(=O)CC2COC(C)(C)CO2)CCS1(=O)=O N1(S(Cc2ccc(C)cc2)(=O)=O)CCN(C(C2(COC)CCCCC2)=O)C(C)C1 C1(NC(C2CCOC2)=O)CCC(C(=O)NCC(C(=O)NC)C)CC1 N1(C(C23N(C(CC4(C)CCCCC4)=O)CC(C)(C2)C3)=O)CCC(F)(F)C(O)C1 CC1CN(C(=O)CP(C)(C)=O)CCCN1C(=O)CS(=O)CCl C(C(F)(C(=O)NC1(CC(C)C)CC1)C(C)C)NC(c1cn(CC)nc1)=O Cc1cscc1C(=O)NCC(O)C(=O)NCCNS(C)(=O)=O Cc1c(F)cc(-c2ccc(NC(C3(C)CCCN3)=O)c(F)c2)c(F)c1N C1(OCC)(CNC(=O)CC2(C)CC2)CN(C(C2CCCN2C(C)C)=O)C1 N1(SCCOCCN(C)C)CC(NC(c2cccc(Cl)c2)=O)CC1=O c1(C(N2C(CNC(C3CC(N(C)C)C3(C)C)=O)CCC2)=O)cccc(Cl)c1N N1(C(c2ccn(CCOC)n2)C(=O)NCC(F)F)CCCC2CN(C)CC12 S(=O)(=O)(CCC(=O)N1CC2CCC2(CCNC(C2(C#N)CC=CC2)=O)C1)NC CC1(NC(=O)CC=CC(N)=O)CCN(C(c2cccc(C3CNC(=O)C3)c2)=O)C1 C(CC(C)(C)C)(C(=O)NCCCSC(C)(C)C)NC(C(C)S(C)(=O)=O)=O N1(C(CCc2cccc(C)c2)=O)CC(C(=O)NCCc2ccncc2)CC(F)C1 C(C)(C(F)(F)F)(c1ccccc1)Nc1cn(CCNC(=O)OC)nc1 Cc1c(C(=O)NCC2CC2CNC(c2cc(Br)ccc2F)=O)sc2nccn12 c1(C(N2C(C)C(NC(c3n[nH]cc3Br)=O)CCC2)=O)ccc2nnnn2c1 C(=O)(C(C#N)C(C)(C)C)N1CCC(CC)C1C(=O)NC1(CCF)CC1 C(=O)(C#CC1(CO)CC1)NCCN(C(=O)CCN(c1ccncc1)C)CC(C)O C1(C(NOCCC(C)C)=O)(CNC(=O)CC2(C)CC2)CC12CCC2 Cc1ccc(CNc2ccc(NS(=O)(=O)CC3CCOCC3)cc2Cl)c(F)c1 C(C)(C(=O)NC1CC(CC(=O)NCCc2ccsn2)C1)SC C1(C(N2CCC(N(C)CC)C2)=O)CCC(C)N(C(=O)CCc2nncn2C)C1 C1(NC(c2cc(C)n(C(C)C3CC3)n2)=O)CCC(C)N(C(=O)CCF)C1 C1(COC)(CNC(c2csc(C)c2C)=O)CCN(C(=O)CC2(C)CC2)C1 c1(CN(C(C)C)C(c2cnc(N(C)C)nc2)=O)cccc(Br)c1O C1(C(N(CC(C)N(C)C(c2csc([N+](=O)[O-])c2)=O)C)=O)CC2CCC1CC2 c1(C(=O)NCC2(O)CN(C(C3CCC4(CCC4)C3)=O)C2)c(Cl)ccc2c1OCO2 Cn1nc(Br)c2ncnc(NC3CC(NC(C4CCCC(O)C4)=O)C3)c12 CC(C(F)(F)C(F)(F)F)=CC(=O)NCC1CCC1NC(C1CC2CC1C2)=O c1(C(c2n(CCSC)nnn2)NCC2(SC)CC2)sc(Br)nc1Cl C1(C(=O)NCCc2cnn[nH]2)CC=CC(NC(c2sccc2F)=O)C1 C1(CCCOCCOCCC(=O)NC)CCCCN1C(=O)CCc1cncs1 c1(C(N2C(C)(C)CC(NC(=O)COc3ccccn3)C2)=O)cc(F)c(Cl)cc1F c1(C(N2CCCC(C(C)(C)C(=O)NC3(CC4CC4)CC3)C2)=O)cnc(S)nc1 N1(C(c2c(C)nn(C)c2)=O)CCCC12CN(C(=O)C(c1ccc(Cl)cc1)C)C2 C1(C(=O)NCC2C(OCC)CCC2)CCCN(C(=O)C(F)(F)C(F)F)CC1 C(CC(C)(C)CC(=O)N1CC(C(C(=O)NCC2CCSC2)OC)C1)OC N1(Cc2ncc(C)nc2)CCN(S(=O)(=O)N(C)C)CC1 N1(c2ccnc(OC)n2)CCN(C)CC1C(=O)Nc1ncc(-c2ccncc2Br)s1 C1(C(=O)NCCC2(NC(=O)C3=CCOC3)CC2)Cc2cc(F)cc(F)c2O1 c1(OC)ccc(C(N2CC(CNC(=O)C(=Cc3cn(C)cn3)F)C(C)C2)=O)nn1 C1(C(=O)NCC(C)NC(CCNC(COC)=O)=O)CCOCC12CCCCC2 N1(CC(N2C(C(=O)NCc3c(C(C)C)n[nH]c3)C=CC2)=O)CCCNC1=O C=CCCC(F)(F)C(=O)NC1CN(C(=O)C(C)CN2CCCCC2)CC1C=C N1(C(C2C(=C)C2)=O)CCCC(CCNC(=O)Cn2cccc2C(=O)OC)C1 Cc1cc(C(=O)N(C2CCN(C(=O)C(C)(C)C(N)=O)C2)CCO)cc(F)c1C C1(C(=O)NC(CNC(CN(C2(C)CCNC2=O)C)=O)CO)(C(F)F)CC(F)(F)C1 c1(N2CCC(C3CCN(C(=O)CNC)C3)CC2)ccc(C#N)nn1.CS C(c1ccc(OC)c(O)c1)=CC(=O)NCC(CNC(C(C=C)O)=O)OC CC(C)C(C)C(CNC(=O)Cc1c(Cl)cccc1Cl)NC(=O)C=C1CCC1 c1(CCC)cc(C(=O)NC(C)(CNC(=O)C=Cc2nccn2CC)CC)ccn1 C1(OC)(CNC(c2cc(C)nc(C)n2)=O)CCN(C(=O)Cc2cn(C)nn2)CC1 c1(CN(C(c2nc(C)sc2)=O)C)ccc(CNC(c2ccnnc2)=O)cc1 C(c1ccc(F)c(F)c1)=CC(=O)N(CC(C)NC(c1oncc1C)=O)CC n12nnc(n1)C2C.c1(C2(C(=O)NC)CC2)cn(C(C2CCCCO2)C2CC2)nn1 N1(CC=C(C)C)CCC2(CNCC(C)O2)C1.c1(C=O)cc2n(n1)CC1(CC1)C2 C1(NC(C(c2ccccc2)OCC)=O)CCN(C(=O)CC23CCC(CC2)C3)CC1 C1(C(=O)NCC2N(C(Cc3nc(C(C)C)sc3)=O)CCCC2)CCCS(=O)(=O)N1 N1(C(c2c(C)c(F)ccc2)=O)CC2(CCCC2NC(c2cc(=O)cc(Cl)[nH]2)=O)C1 N1(C(c2c(OC)c(=O)cco2)=O)CC2CCC(C1)C2CNC(=O)C(F)(F)C(C)O C1(NC(C2CC(=O)C2C(C)(C)C)=O)CN2CCC1NC(=O)C2=O.C(C(F)F)OCC c1(NC(CC)CNC(=O)C=Cc2cccnc2C)cc(S(C)(=O)=O)ncn1 c1(NC(N(C(C2Cc3ccccc3O2)C)C)=O)ccccc1[N+](=O)[O-] c1(C(=O)OC)cc(S(=O)(=O)N2CC(c3ccc(I)s3)C2)ccc1N CCCCN(CC)N1CCN(C(c2ccccc2)C(N2CCCCC2)=O)CC1 N1(C(C2(C)C=CCCC2)=O)CC2OCCN(C(C3CCCCN3N=O)=O)C2C1 S(=O)(=O)(c1cc(Br)ccc1Cl)N1CCC(CC(=O)Nc2ncccc2Br)C1 CCC(CC)CC(=O)NC1CC(C)N(C(c2ccc(C)cc2)=O)C1 C1(ONC(=O)C)CCn2cncc2C1.C=CC1(c2nocn2)CCCC1 N1(C(CC2CC(=C)C2)=O)CCOC(C(=O)Nc2cccc(CO)c2C)CC1 C12CC(OC)CN1C2=O.N1(C(C2C(=C)C2)=O)CC(C(C)NC(=O)OC(C)(C)C)C1 C=C(CC(F)(F)F)C(=O)NC1(CCO)CCCCC1 C1(C(N2C(C)CC2C(=O)NCC2CCCC2C)=O)C2CN(C)CC12 c1(C(=O)NC2CC3CN(C(=O)CCC4CC4)CC23)cc(=O)c2cc(O)ccc2o1 C1(O)(CC(=O)NCC(C(=O)NCC(=C)F)N(C)C)CCOCC1 Cc1cnn(C)c1C(N1CC(NC(C2(C)CC2(F)F)=O)C(F)C1)=O C(=O)(C(C)(F)C(=O)N(CCC(=O)NC1CC2OCCCC12)C)OC c12cccc(c1)C(=O)NC2.n1(CC(=O)NC2CC(CCC)C2)cc(CC(C)O)nn1 CCC(F)(F)CC(=O)N1CCCC(CC)(NC(=O)CCCc2ccncc2)C1 CC1C=C(C(=O)NCC(C2(O)CCN(C(=O)Cc3ccc(F)cc3)C2)C)C1 C1(C(N2CCC(CCC)C2)=O)C(C)OCCN1C(c1cnnn1CC)=O C1(C(=O)OCC)CN(C(c2nc(CC(F)(F)F)sc2C)=O)CC(C)S1(=O)=O c1(C(N(CCCN(C(C2C(OCC)C2)=O)C)C)=O)ccc(C)nc1OC C(=O)(CC1=CCOCC1)N(C1CCN(C(C(CC(=C)C)C)=O)CC1)CCC Cc1[nH]nc(N(CC(=O)NC2CC2)C(N2CC(c3ccccc3)C2)=O)c1C C1(NC(CN(C2CCC2)C)=O)CCOCC1C(=O)NCc1ccnnc1 N1(C(C2C(CNC(C(CC=C)CC)=O)OCC2)=O)CC(F)(F)C(F)(F)C1 c1(C(=O)NCC(CN(C(C(CCOC)C)=O)C)(C)C)c(C)cc(C)oc1=O C12(CCC(=O)Nc3cc(O)ccc3NC3CC3)CCC(CC1)NC2=O N1(C(CSCCCC)=O)CCC(CCOC)(NC(=O)C(O)C(C)SC)CC1 C1(C(=O)NCCC(C)(C)NC(=O)CCCCCF)Cc2cc(Cl)ccc2C(=O)O1 C12(CCNC(C(C)NC(=O)C(C)(C)C)=O)CCC(CC1)N(C(c1cnsn1)=O)C2 C1(NC(CON(C(C)=O)C)=O)C(O)C(O)CN1C(c1cn(CCO)nn1)=O N1(C(=O)C#CC2CCC2)CCC2(CCN(C(c3cc4cnccc4o3)=O)C2)C1 C1(CNC(C=CC(C)(C)C)=O)COCCN(C(c2csc(C(F)(F)F)n2)=O)C1 c1(C(=O)NCc2cc(C(N3C(C)CCC3)=O)no2)cc(N)cc(F)c1 c1(CC(=O)NC(CNC(c2c(N)ccc(C)c2F)=O)C)noc2cc(F)ccc12 c1(Cn2cc(-c3ccc(F)cc3I)nn2)cn2cccc(F)c2n1 N(C1CCCc2n[nH]cc21)C(C(CCC1CC1)NC(CC(CCCC)O)=O)=O N1(C(c2c(C)c(Cl)ccc2)=O)CCN(C(C2CCc3nccn3C2)=O)C2CCC12 C(CO)(CCCCNC(=O)C(c1c(F)cccc1F)(C)C)NC(C(CC)F)=O c1(C(N2CCC(N3CCN(C(=O)C4CC4)CC3)C2)=O)c(Cl)ccc(Cl)c1Cl C1(NC(C(C=C)(C)C)=O)CCN(C(c2ccc(C(C)=O)c(C)c2)=O)C(C)C1 N1(C(CC2C(C)CCO2)=O)CCCCC(C(=O)NCC(=O)OCC2CC2)C1 C#CC(C)(C)C(=O)N1CCCC(N(C)C(c2cccc(CS(C)=O)c2)=O)C1 N1(C(COC2(C)CCC2)=O)CC2CCCC2(NC(=O)CCOCC(F)F)C1 C(CNC(=O)Cc1cnsc1)(C(C)C(C)C)NC(c1c(C)nc(Br)s1)=O C1(CNC(C=C(C)C)=O)CC2CCC1N2C(c1cccc(C2CC2(F)F)c1)=O CC1(C)CCCC(C)(NC(=O)C=CCN=c2nc(C3CCCCC3)[nH]s2)C1 c1(C(N2CC(CCNC(c3c(C)snc3)=O)C(C)C2)=O)cc2ccccc2s1 C1(C(=O)NCc2c(C(=O)NC(C=C)(C)CC)c[nH]n2)CC(C)(C)CCO1 CC1CCC(Cl)=C(C(=O)NCC2CCCN2C(=O)CCS(=O)(=O)NCCO)C1 c1(C(=O)OC)ccc2n1CCN(C(c1ccccc1I)C(=O)NCCC#N)C2C c1(CN(C2CCN(c3ccncc3)C2)C)cnc(F)c(F)c1 C1(NC(C(CC2CN(C(c3c(C#N)scc3)=O)C2)F)=O)CCN2CCC1C2 C1(NC(CC(CCC)CC)=O)Cc2ccccc2C1NC(c1snnc1C)=O C1(C(=O)NCC2CCN(C(COCC=C)=O)C2)C2CCC1(c1cscn1)C2 C12CCCN(C1)C(=O)c1cnn(c1)CCN2C(C1C(=C)C1)=O.c1(NC)cccnc1 Cc1cn2c(n1)CC(C(=O)NCC1CC3(CC(NC(c4cnsc4)=O)C3)C1)CC2 c1(C(=O)NCCN(CC(=O)NC2CN(C)CC2C)CC)sc(N2CCCC2)nc1Cl N1(C(c2c(C)nc(C)s2)=O)CC2=C(C1)CN(C(C1CC(N3CCCC3)C1)=O)C2 N1(C(Cc2ccn(C)n2)=O)CCCC(C(=O)NCCn2cccn2)CC1 N1(C(c2n(CCC)ncc2)=O)CC2CC(C(N3CC(=O)NC4(CC4)C3)=O)C(C2)C1 C1(C(=O)NCC(C)N(C(c2c(C)nc(CCC)s2)=O)C)CCc2cnnn2C1 C1(C2(O)CCN(C)CC2)(C(=O)NCC2C(CNC(C(C)C(C)(F)F)=O)C2)CC1 C1(C(N2CC(CCNC(=O)CC3CCCC34CC4)C2)=O)CCC2(CCCCC2)C1 N1(C(C(C2(O)CCC2)NC(C=CC2N(C)CCC2)=O)=O)CCC(F)(F)C(F)C1 c1(C(=O)NC2(CNC(Cc3c(C)nsc3)=O)CC(C(=O)O)C2)ccc(F)cc1F Cc1noc(C)c1CC(=O)NC1CCC(NC(=O)C(O)Cc2cnn(C)c2)C1 c1(SCC)nccc(Cl)c1CNC1CCCCC1C(=O)Nc1cc(F)cc(Cl)c1 C=C=CCCC(=O)NCCC1(NC(c2ccnc(Cc3cscn3)c2)=O)CC1 Cc1nn(C)c(C)c1CNC(C1COCCN1Cc1ccc(I)c(F)c1)=O C(=O)(C1=CCCOC1)OCC(N1CCN(CCC(C2CCOC2)C2CC2)CC1)=O c1(C(=O)NC2C(F)CCN(C(C=CS(C)=O)=O)C2)cnc2[nH]cnc2c1 S(=O)(=O)(c1cc2ccccc2s1)NCC1N(Cc2cc(C)cc(Br)c2)CCCC1 C1(NC(C2CC2CF)=O)COCCN(C(c2cccc(C3CC3)c2)=O)C1 c1(C(=O)NCC2N(C(C3(OC)CCC3)=O)CCC2)ccc(C)cc1[N+](=O)[O-] N1(C(C(CCC)O)=O)CCC2(C1)CN(C(c1cc(Cl)cc(Cl)n1)=O)CCO2 C1(CCC(=O)OCC)CCCCN(C(=O)C(C)(C)CO)C1 N1(C(C)=O)CCC(N(c2ccc(F)cc2)C(=O)CCCn2c(O)nnc2O)C12CCC2 c1(NCCSCCOC)nc2cc[nH]c2c(=NCC2CCC3(CCC3)CN2C)[nH]1 C=C(C)CCCC(=O)N1CC(C)CCC1CNC(C12CCC(C1)C2)=O C1(CC(F)(F)F)(CN(C)CC2CCCNC2)CCOCC1 c1(C(=O)Nc2ccc(NC(CCNC(C)=O)=O)nc2)cc(Cl)c(Cl)cc1O C1(NCc2nc(C)cc(OC)n2)CC2CCCCN2C1=O C1(NC(c2cc(OCC)ns2)=O)CCN(CC(=O)O)CC1 C1(CNC(C(C)SC)=O)CN(C(=O)CCOC2CC2)CC1O c1(CNC(COC2(C#C)COC2)=O)cc(C(=O)NCC(O)CCOC)n(C)n1 N1(C(=O)CC2CCCC2(F)F)CC2CC(C1)N2C(C1(F)CC1)=O c1(CC)cc(C(=O)NCC(C(C)C)NC(=O)CN(C)C2CC2)ncn1 C1(OC)CC(CF)N(C(=O)C(C)=C2CCCC2)C1.C123CC(C1)(C2)NC3=O CC1(C)CN(C(=O)C(C#N)C2CC2)CCN(C(c2cccc3ccncc23)=O)C1 c1(N(CCNCCCN2CCC(F)(F)CC2)C)cc(C#N)ccc1F N1(C(=O)Nc2c(F)cc(Cl)cc2F)CCCc2sccc2C1.C1CCN1C N1(C(C2CC(OC)C2)=O)CCN(C(=O)CC(C)c2ccncc2)CC1CC(F)F C1(C(N2CCCCC(NC(c3ccc(Cl)cn3)=O)C2)=O)CCCC12CCOCC2 c1(OC)nc(C)nc(Cl)c1NC(C1CCCN(C(c2occc2Br)=O)C1)=O C1(C(=O)NCCc2cnc(C)o2)CC2C=CC1N(C(=O)CC1=CCCCC1)C2 C1(C(N(C)CCNC(c2csc(C3CCCCC3)n2)=O)=O)CCCS(=O)(=O)C1 c1(C(=O)NCCC(C)NC(CCC(C)OC)=O)ccc(C)c(F)c1Br C1(c2ccccc2)(COC)CN(C(=O)C(C)OC(c2cccc(Br)c2)=O)CCO1 N1(C(C=C2CCC(C)CC2)=O)CCC2(C(=O)NCc3cc(F)ccc3O)CCCC12 c1(C(=O)NCC2CC(NC(C(CCC)CC)=O)C2)cc(C)c(C)nc1C N1(C(COC2CCN(C(=O)OC(C)(C)C)C2)=O)CC2(CC2)CC1CO Cc1nc(C2CC2)oc1C(=O)NCCN1CCN(C(C2NC(=O)CC2C)=O)CC1 c1(CCN(C(=O)NC(C)CCN2CCCC2)CCO)ccc(Br)cc1Br c1(OC)ccc(Cl)cc1C(c1nnnn1C1CCOC1)NCCS(=O)(=O)CC1CC1 CC(CC(=O)N1CC(C2(NC(=O)CCc3ccc(=N)[nH]c3)CC2)C1)P(C)(C)=O c1(CCC)onc(C)c1C(N1CCC(CCNC(=O)Cc2nccn2C)C1)=O Cc1nn2cc(C(N3CCC(CNC(=O)C4=CC(C)CC4)CC3)=O)nc2s1 c1(C(=O)OC)cnccc1C(=O)NCC(O)CNC(C1NC(=O)OC1C)=O c1(OC)ccc(CNC(N2CCC(N3CCCC3=O)C2)=O)c(C(F)F)c1OC CC(C)CC(O)CC(=O)NC1(CNC(C2CCC(C)(C)OC2)=O)CCCCC1 N1(N(C2CCC(O)CC2)C)CCC2CN(C(C3C(C=O)C(C)(C)C3)=O)CC12.C(=O)O N1(C(C#C)=O)CCC12CN(C(c1cnc(OC3CCOCC3)nc1)=O)C2 N1(c2ccc(C(=O)NC3C(OCC)CC3)cn2)CC(C)OC(C)C1 N1(C(c2cc(CCC)ncc2)=O)CCC2C(C(=O)NC3CN(C(=O)CC)C3)C2C1 c1(N(C)C2CC2)nnc(C2CCCCO2)n1CC(CCCS(C)(=O)=O)=O c1(C(=O)NC2C(CNC(C(C)SCCCC)=O)CC2)cc(N)c(Cl)c(O)c1 CCC(C(=O)NC(C)CNC(=O)NC1CC1)NC(c1csnn1)=O N1(C(c2c(CC)ccs2)=O)CC(F)(F)CC1CCNC(C1C(F)(F)C12CCC2)=O N1(c2snc(SC)n2)CCC2(CC1)C(NC(c1[nH]nnc1C1CC1)=O)CS2(=O)=O c1(C(N2CC=C(CNC(C3CC(CC)OCC3)=O)CC2)=O)cc(C#N)ccc1Cl C1(C(CNC(C(C)N(C(C)=O)C)=O)C)CCN(C(=O)Cn2[nH]cnc2=N)CC1 C1(NCCN)CC12CCN(CCSc1ccc(OC)c(O)c1)CC2.C(=O)(C1CC1)OC c1(CCCC(=O)NCC2C(C(=O)NCC(C(=O)OC)OC)C2)ccc(Cl)nc1 c1(C(=O)Nc2cc(-c3ccncc3)n[nH]2)cccc2c1CN(Cc1cc[nH]n1)C2 N1(C(C(C=C)(F)F)=O)CC2(NC(=O)CCNC(=O)OC(C)(C)C)CCC1C2 c1(C(=O)NC2CCC(CNC(C(CCSC)O)=O)C2)ccnn2ccnc12 c1(C(N2C(CN(C(c3c(CC)noc3C)=O)C)CCC2)=O)cc(C)nnc1O O(NC(=O)C(C)(CO)NC(c1ccc(C)o1)=O)C(COC)COC C1(CC)CN(C(c2cnccc2SC)=O)CCC1NC(=O)C(F)(F)c1cscn1 C12(CC=C)CN(C1)C(=O)CCCNC2=O.N1CCCC1CC1CC1.C(C)=O C1(F)(C(=O)NC(CC)C(=O)N(C)C)CCCN(C(=O)CCOCC(F)F)C1 c1(C(=O)NC2(CNC(C3C(C)(C(=O)OC)C3)=O)CCOC2)ccnnc1O C1(CSCC(=O)NC(C2CCOCC2)C#C)CCC(=O)O1 c1(C(CNC(C(c2cscc2Br)N(CC)CC)=O)(C)C)cccc2ccccc12 C1(CNC(C2(C(C)NC(c3ccc(C(N)=O)[nH]3)=O)CC2)=O)(CC)CCN(C)C1 c1(C(=O)NC(C2CN(C(=O)COCCF)C2)C)ccc(N=NC(N)=O)cc1 C1(C(=O)OC2C(CNC(C=COC(C)=O)=O)CCCC2)CC(C)OC(C)C1 Cc1c[nH]c(=NCC2CCCN2Cc2ccc(C(F)(F)F)cc2)c(C)n1 C1(CNC(C2CCC=CCC2)=O)CCCN(C(c2coc(O)n2)=O)CC1 N1(C(CC=C)=O)CCC2(CC(NC(c3cnc(-c4ccccn4)s3)=O)CO2)C1 c1(CC(=O)N(CC(CNC(C2(C#C)CCCC2)=O)O)C)cnc2c(=O)[nH]ccn12 C(=O)(C1=CCN(C(C2CCCC(C#N)C2)=O)C1)NCc1ccn(C(C)C)n1 C1CC(C)C(=O)N1.C1CCCC1C(=O)N(C)CC1(N(C)C)CC1.CN N1(C(c2c(COC)scc2)=O)CC(C)CN(C(c2cncc(OC)c2)=O)C(C)C1 CC1CCN(S(=O)(=O)CC(=O)NCC=CCNC(C2CC=CCC2)=O)CC1 N1(C(c2c(C)scn2)=O)C2CCC1CN(C(C1(C)CC1Br)=O)C2 c1(C(N2CCC(c3nc[nH]n3)C2)=O)ccc2c(c1)oc1ccccc21 c1(C(=O)NC2COCCN(C(C(CN(C)C)(C)C)=O)C2)ccc2nccnc2n1 c1(C(=O)NC2C(F)(F)CCN(C(C3=C(C)OCC3)=O)C2)ccc2nccc(Cl)c2c1 c1(C(=O)NCC2N(C(c3cccc(OC)n3)=O)CC3CC32)cnc2nc(C)oc2c1 C(C1=CCN(C(c2ccc(Br)cc2C)=O)CC1)NC(C1C(OC)CCC1)=O C(=O)(C(C)(C)CS(N)(=O)=O)NCC(CC)NC(c1ccc(CO)c(Cl)c1)=O C(c1cccnc1)=CC(=O)N(C1CCCCC1)CCNC(c1cc(SC)oc1)=O C1(NC(CCCC#C)=O)CN(C(C2CCCO2)=O)CCC1(C)C CC(CC(=O)NCCOCCN(C)C(C1CC(C)(C)CCO1)=O)C(F)(F)F c1(CC(=O)NCCCCCNC(c2c(CC)noc2C)=O)nc2ncccn2n1 c1(C2(C(=O)NC3CC(C(C)C)SCC3)CC2)cc(Cl)ccc1Br C(CNC(=O)C=CCCC(C)C)(CC(=O)N1CC=CC1CN(C)C)OC c1(C2(C(=O)NCC3(NC(C4CCO4)=O)CCOC3)CCC2)ccc(O)nc1 C(=O)(C1=CCCCO1)N1C(C2CCN(C(C(CC)Cc3ccccc3C)=O)CC2)CC1 c1(OCC)ccccc1C(=O)NCC1(C)CCCN1C(=O)CC(C)n1cccc1 c1(C(=O)NCCCOCCNC(c2ccsc2)=O)ccc(-c2ccccc2)[nH]1 c1(C(=O)NC2(C(=O)NCC(C)OCC=C)CC(O)C2)ccc(CO)nc1 c1(NC(=O)NCCCC)cc(CNC(=O)NCCn2cncn2)ccc1C C1(c2onc(-c3c(Cl)ccc(OC)n3)n2)CCNC2(CCC2)C1 O=C(C(O)C1=CCCCC1)N1CCC(C(=O)NC2CCCN(O)C2=O)(CF)C1 Cn1ncc2c1CN(C(=O)CC1CCCCC1(F)F)C2 C(=O)(C(C#N)CC)N(CC(N1CCC1C(=O)NCC#C)=O)CC N1(C(C(C)NC=O)=O)CCC2(CC1)CC2NC(c1cc2ccccn2c1)=O Cn1nnc(C(N2CCC(NC(c3cc(C(C)(C)C)c[nH]3)=O)C2)=O)c1C(F)(F)F C1(C(=O)OC(C(C)(C)F)c2cccnc2)CCC(=O)N(C(=O)Cn2nccn2)C1 c1(C(=O)NC23C(CN(C(CSCC#C)=O)C2)CCC3)c[nH]c2cccc(Cl)c12 Cc1cccc(C)c1C(C)NC(N1CCCCC1c1cnc(=N)[nH]c1)=O c1(C(=O)NC(c2nccc(O)n2)C)coc2c1COC2 N1(C(C2(C(=O)NC)CCC2)=O)CCCOC(CCNC(=O)Cn2cnnc2)C1 N1(C(C(CC=C)(C)C)=O)CCOCC12CCN(C(=O)Nc1ccc(Cl)cc1Br)C2 C(=O)(C(C)C(C)S(C)(=O)=O)N1CCC(NC(CCC(C)(C)OC)=O)C1C S(=O)(=O)(c1ccc(O)c(OC)c1)NCC(=O)OCC.c1(S)ccc(COC)cc1 c1(C(C(=O)NCCCC(C)NC(C(C2CCOC2)OCC)=O)C)cccc(O)c1 c1(C(N2CCC(CNC(C(C=CC)O)=O)C23CC3)=O)[nH]cc2c1CCS2(=O)=O CC(C(=O)NCC1CCN(C(=O)CN2CC3C=CC2C3)CC1)C(F)F Cc1cccc(C)c1N=c1[nH]nc(C2CN(C(=O)Nc3cc(C)sn3)C2)s1 C1(C)(NC(C2(F)CCN(C(COCC(C)C)=O)C2)=O)CCC(=O)NC1=O CC(C)CCCCN(C(=O)C(O)C1CN(C(C2CC2OC(C)(C)C)=O)C1)C N1(C(c2sccc2Cl)=O)CCn2c(-c3cn(C4CCC4F)nn3)nnc2C1 c1(C(=O)NCCC(C(C)C)NC(C(C2CC2)OCC)=O)ccc(O)c2ccccc12 C12(NC(CC=CC=C)=O)CCCCC1N(C(C1CCCCN1C(C)C)=O)CC2 C1(C(=O)NCC=C)CCOC(C(=O)NCCC2CCCN2C)C1 N1(C(C(C=C)(C)O)=O)CC2CCCC(NC(c3ccsc3COC)=O)C2C1 C(C)(CNC(C1CC1C)=O)(CO)NC(C1(C(C)C)CC1)=O N1(C(Cc2c(C#N)nc(Br)cc2)=O)CCC2(CCCOC2)C1 Cc1ccc(Cl)cc1C(=O)NCC1CCN(C(=O)CCCC2CCCC(=O)N2)C1 Cc1cc(C(=O)N(C(C)CNC(c2cnc(C3CC3)nc2C)=O)C)ncc1N C#CCC(C(=O)NC(C)=O)NC(=O)C(C)NC(C)(C)CC C(C)(CCC(=O)NCC=C1CCN(C(c2cc(C(N)=O)nn2C)=O)CC1)OC C1(NC(CCOCCOC)=O)(CNC(c2snnc2C)=O)CCCCCC1 c1(NC(c2nc(C(=O)NCCC3CCCO3)cs2)=O)ccnc(C(F)F)c1 C(c1ccc(O)c(OC)c1)=CC(=O)N(C(CNC(C(CC)(C)O)=O)C)CC N1(C(C(CCC)NC(N)=O)=O)CCN(C(C2(C(C)C)CCCO2)=O)C2(CC2)C1 N1(C(C(CC)n2ccnc2)=O)CCC(C(N2CCC2(C)COCC)=O)C(C)C1 Cc1c(C)c(NC(=O)CN2CC=CCC3(CCCC3)C2)c(C)c(C)c1Br c1(C(N2CCC(N(C)C(C34CCC3C4)=O)C2)=O)cnc2[nH]c(C(F)(F)F)nc2c1 CCCC(C)CC(=O)NC(C)(CNC(c1cncc(OC)c1)=O)CC c1(C(N2CCC(C(C)(C)C)(CNC(C(C)SCC)=O)C2)=O)cc2c([nH]1)CCOC2 C=CC(C)(C)CC(=O)NC(CCSC)C(=O)NCc1csnc1OC c1(C(N(CCCNC(C2CC(OC)C2)=O)C2CC2)=O)cccc(OC(F)F)n1 C1(CNC(C2CC(OC)CN2C(=O)Cc2ccnn2C)=O)CCCN(C)C1=O C1(C(N(CC(=O)N(CC)CC)C)=O)CNC(=O)CN1C(=O)CC1CCCCO1 C(=O)(C1=CCS(=O)(=O)C1)N1CCOCC(CNC(C=Cc2ccc(CC)o2)=O)C1 C(=O)(C(C(C)C)NS(N)(=O)=O)NCC(CC)N(C(CC(=C)C)=O)C N1(C(c2ccc(C(C)O)cc2)=O)CC(N(C(=O)CCc2nc[nH]n2)C)C2(CC2)C1 C(=O)(C(C)(C)C(=O)OC(C)(C)C)N(CC(C)NC(C1CC(F)C(=O)N1C)=O)CC C1(C2(NC(C3C(OC)C3)=O)CC2)CCCCN1C(=O)CCOc1cccc(C)c1 N1(C(Cc2c(C)nc(C)[nH]2)=O)CCC(NC(c2cc(C3CC3)ncn2)=O)C(O)C1 N1(C(CCCCCC)=O)CC2CC(C(=O)NCC3(C(=O)OC)CC3)C(C2)C1 N1(C(CNC(c2cc[nH]n2)=O)=O)CCC2(CCOCC2)C(CNCC2(C)CC2)C1 c1(C(N2CC(CCNC(C=CCCC)=O)OCC2)=O)cc(O)ccc1OC C1(C(N(CC(CC)C)C)=O)CC(O)CN1C(=O)CC(C)COC C1(NC(C(COC)O)=O)CCN(c2ccnc(C#N)n2)CC1O N1(C(CC(N2CCC3(CN(C(c4ccsc4)=O)C3)C2)=O)C)CCc2ccccc2C1 N1(C(CC(CC)C2CCC2)=O)CC(CO)C2(C1)CN(C(c1ccc(O)c(F)c1)=O)C2 C(=O)(C(CO)C(C)(C)C)N1CC(NC(C(=O)N(C(=O)CC2CCCC2)C)C)C1 N1(C(C(C)N(C(C(=O)NCCC)=O)C)=O)CCCC(C)C1CO c1(C(N2CCC(NC(C3(C)C(C)(C)C3)=O)C2C2CC2)=O)cc2c(s1)COCC2 c1(OC)ccc(C(N2CC(NC(C3CNC(=O)C3)=O)C(C#N)C2)=O)c(C)c1C Cc1cc(OC(CC=O)OCC(=O)N(C)C(C)C)no1.C(=O)(C(C)C)N C1(CNC(CSCC#C)=O)CCC(CNC(C23CCC(OC)C2C3)=O)CC1 C1(NC(c2c(OC)nn(C)c2)=O)CCCCCC1C(=O)NCC1(O)CCC1 c1(CN2C(=O)NC(CCSC)C2=O)cc2ccc(F)cc2nc1O C(=O)(C1=NOC(C)C1)NCC1(F)CCN(C(c2c(C)coc2C)=O)C1 C=CC(CC)C(=O)NC1CCCCC1CNC(c1ccc(C(=O)OC)o1)=O c1(C(=O)NCC(C)(CO)NC(CCN(CC)CC)=O)cc(F)c(O)c(Br)c1 C1(C)(C(N(CCC(C)NC(c2cc(OC)ncc2)=O)C)=O)CCCNS1(=O)=O CCCCC(CC)C(=O)N1CCC2(C1)CN(C(=O)CCN1CCN(C)CC1)C2 C1(C(N2CCCC(CC)(NC(c3cnnc(O)c3)=O)C2)=O)CCn2ncnc2C1 C(=O)(N=c1cc[nH]cc1Cl)c1ccc(CCC(=O)NC2CC2C2CC2)[nH]1 C(=O)(C1=C(C)OCCS1(=O)=O)NCC1(O)CC(NC(CCCC(=O)NCC)=O)C1 c1(CC(C)NC(C2(n3cc(C(CC)(C)O)nn3)CC2)=O)ccc2cccnc2c1 N#Cc1cncnc1C(=O)NCCOCCNC(C1C2COCC12)=O N1(C(C(COC)N(C)C)=O)C(N(C)C)CCC1C(=O)NCCOC(C)=O c1(C(C)(C)C)c(C(=O)Nc2nccnc2C(F)(F)F)c(O)nc2[nH]nc(O)c12 C(=O)(CS(=O)(=O)CCO)N1CC(c2ccc(OC)cc2)N(C(C)=O)CC1 C1(CN(C(=O)CC2C(C)(C)C2(C)C)C)CCCCN1C(c1cnn(C2CC2)c1)=O c1(OCCC(N2CCCC(CNC3CCCN(CC)C3)C2)=O)ccc(F)cc1Cl c1(C(N(C2CN(C(c3ccc(F)c(Cl)c3N)=O)C2)C)=O)ccc2oc(S)nc2c1 C1(O)(N(CCOC(=N)O)C(C2C=CCN2)=O)CN2CCC1CC2 N1(C(CCNC(COC)=O)=O)CCN(C(c2ccc(-c3ccncc3)o2)=O)CC1 CC1CCC(CNC(C2(CO)CC(F)(F)C2)=O)CN1C(c1ncncc1N)=O CC(C)C(CCNC(c1cncnc1C(C)(C)C)=O)NC(c1ccns1)=O c1(OC)ccc(CC(=O)NC2CC(N(C(=O)C(C(C)O)N(C)C)C)C2)cc1O c1(C(N2CC(C(=O)NCC3CCN(C)C3)C(O)CC2)=O)[nH]nc2ncccc12 C1(NC(C2(CC)CCC2)=O)COCCN(C(c2cc(=N)[nH]c(Cl)n2)=O)C1 Cc1cc([N+](=O)[O-])ncc1C(N1CCC(NC(=O)CNC(=O)C(F)(F)F)C(C)C1)=O C1(NC(Cc2nc(C)sc2Cl)=O)CC2(C1)CN(C(C1CCCSC1)=O)C2 c1(C(=O)NC2CC(NC(CSC(C)(C)C)=O)C23CCC3)nc2ccccn2c1F C(C1CN(C(=O)C(C)CC(N)=O)CC1C(=O)N(CC(C)C)CC(C)C)=CC C(F)(F)(C(=O)OCCC1CCCO1)C1(OC)CCC1 c1(OC)ccc(C(C)C(=O)NC(C)CN(C)C(C2C=CCC2)=O)cc1 C1(C(=O)C(=O)OC2CC2)(CN(CC(=O)NC2CCC(C(N)=O)C2)C)CC12CCC2 c1(C(=O)NCCCCC2C(C)C2)ccc(CNC(C2(C)CS(=O)(=O)C2)=O)cn1 N1(C(C(C(C)C)C#N)=O)C2CCC1CN(C(c1cc(-c3ccoc3)[nH]n1)=O)C2 CC(C)C(CCNC(=O)CC1CCCC1O)NC(c1cncnc1C1CC1)=O c1(NC(C(c2ccn(C)n2)C)=O)ccc(N2CCC(=O)NC2=O)cc1Cl C1(NC(c2c(CC)scn2)=O)CN(C(c2ccc3c[nH]nc3c2)=O)CC1N=[N+]=[N-] C(=O)(C(C)(F)C(F)(F)F)N1CC(F)(CNC(c2cccc(NC(C3CC3)=O)c2)C)C1 N1(C(c2c(Cl)cnc(OC)c2Cl)=O)CCC2(CCC(NC(=O)CC3(C)CC3)C2)C1 CC1CCC(=CC(=O)NC2(C(=O)NC3CC4(CC4)C3)CCC2)CC1 c1(C(=O)NC2CC(NC(c3c(Br)ccnc3Cl)=O)C2)cc(Cl)ccc1I C1(C(=O)NCC2CC3C=CC2O3)(NC(C(CC)O)=O)CCOCC1 CC(C)C(CC1CCCCC1)C(=O)NCCCN(CCO)C(C1CCSC1)=O N1(c2cc(C)ncn2)CCN(C(=O)CC(C)c2ccncc2)C(C)C1 C1(C(=O)NCC2CC3(CN(C(CSSC)=O)C3)C2)CS(=O)(=O)CC(=O)N1 C=CCC(CC(F)F)NC(C1CC(C)(NC(=O)CCC=C)C1)=O CCC(C#N)C(=O)NCC1CCCC1NC(C1(O)CCOCC1)=O N1(C(CCCC)=O)CCN(C(=O)COc2ccc(C#N)cc2)C(CO)C1 Cc1[nH]c2c(F)cccc2c1CCN(C)Cc1ccccc1OC(F)F N1(C(C(CCC)OC)=O)CC23CCCC2(C1)CN(C(=O)Cn1cncn1)C3 C1(C(C)C)(C(=O)O)CCCO1.C(C(C)O)N(C(=O)CN(C)C(N)=O)C N1(Cc2cccc(OC)c2)CCCC(NC(C2(C)CCC(=O)CC2)=O)CC1 c1(OC)cc(CCC(=O)NC(C2CCN(C(=O)CNS(C)(=O)=O)C2)C)ccc1F c1(CC(=O)N(C2CCN(C(=O)C(C)(C3CC3)N(C)C)C2)CC)c(F)cccc1Cl C(=O)(C(Cn1cccn1)NC(C1C=CCS1)=O)N(C)CC1CC(=C)C1 Cc1ccc(C(=O)NCC2CCCC(NC(=O)CNS(=O)(=O)N(C)C)C2)cc1O C1(CNC(C(CCC2CC2)NC(CN(C(=O)OC)C)=O)=O)CCCOC1(C)C c1(OC)cc(CC(=O)NCC2CCC(NC(=O)CSC3CCCCO3)C2)on1 C(=O)(C1=C(C#N)CCC1)NCC(C(=O)NC1CC(C(F)(F)F)C1)N(C)C Cc1cc2cccc(NC(=O)Nc3ncc(CC4CC(F)(F)C4)s3)c2[nH]1 C(=O)(C(C)(CC)C(N)=O)NC(CC)CN(C(=O)CSCc1ccncc1)CC C1(C(=O)NC23CC(CNC(C4CCCCS4)=O)(C2)C3)CC2CCC(C1)C2 Cc1ccc(N)cc1C(=O)NCC(C1CCC1)NC(c1nc(C(F)(F)F)cs1)=O C(c1c(C)cc(C)cc1C)=CC(=O)NC1C2CN(C(C(C)OC)=O)C(C2)C1 Cc1ccc(C(=O)NC2CN(C(C3CCC(=O)N3C(=O)C(C)C)=O)CC2C)cc1 Cc1oc(C(F)(F)F)c(C(N2CC(O)(CN(C(=O)COCC(F)F)C)C2)=O)c1C c1(C(=O)NCC(C2CCN(C(C3(O)CCC3)=O)CC2)C)ccc2nc(O)oc2c1 C1(C(=O)NC(CC(=O)NC)C)CN(C(c2c(Cl)cccc2Cl)=O)CCC1O CC(C)(C)C(C(=O)NCC12CCC1CN(C(=O)Cc1cn[nH]c1)C2)n1ccnn1 C(C1=CCN(C(=O)C(C)(C)OC(C)=O)CC1)NC(COCCC#C)=O CCCC(C)(O)CNC(c1cn(CCNC(c2scc(C)c2C)=O)cn1)=O C1(NC(c2cn(-c3ccccc3F)nn2)=O)C2CC1N(C(C1CC1F)=O)C2 CCCC(O)CC(=O)NC1CCCN(c2cc(C)nc(CC)n2)C1C N1(C(C2(C(N3CC(c4cccc(Br)c4)(C)C3)=O)CC(=C)C2)=O)CCC(C#N)C1 n1(CCOCC=C)c(N(C)CC2(C)CC(O)C2)nnc1-c1ccc[nH]1 C=Cc1ccc(C(N2CC(C(=O)NC3CCCN(C(C)=O)C3)CC2(C)C)=O)cc1 Cc1cccnc1CCC(N1CCC(CO)(NC(C2CCC(C)CC2)=O)C1)=O N1(C(C2(c3ccccc3)CC2)=O)CCC(C2CCCN2Cc2cnc[nH]2)CC1 NC(=O)CCC(=O)NCc1cn(CCNC(c2cc[nH]c(=N)n2)=O)nn1 C1(CNC(C2CC(SC)C2)=O)CN(C(=O)CCC2NC(=O)NC2=O)CC(C)(C)O1 c1(C(=O)OCC)cc(COC(C2CC3(CCO3)C2)=O)n(C)n1 C(S(=O)(=O)CC(=O)NC(CN)C(F)(F)F)c1ccc(NC(C(C)C)=O)cc1 N1(C(=O)C=CCO)CCCCC2(CCN(C(c3c[nH]c4cccnc34)=O)C2)C1 c1(OC)cc(C(=O)NC2(CN(C)C(C3CCC(C)O3)=O)CC2)ccc1Cl C#Cc1cccc(C2CC2C(N2CC(NC(=O)Cn3cc([N+](=O)[O-])cn3)C2)=O)c1 CC1(C)CN(C(=O)CC23COC(CF)(C2)C3)CC1NC(=O)CC1CCOC1 N1(C(c2cc(C)cc(C)c2)=O)CCC(NC(C2CC3CC3C2)=O)C(C)(C)C1 C1(C(=O)NCC(C(C)C)OC)(OC)CCCC1 N1(Cc2ccc(C(N)=O)cc2)CCc2ncccc2C1.N12CCC3(CC1)CC3C2=O C(=O)(C1CCc2ccccc21)N(CC(=O)NC1COC1)CCCF c1(CNC(C)=O)ccc(C(=O)NCC2(F)CC(C)C2)s1.c1(C(=O)N)nscc1C C1(OC)CC2(C1)CC(C(N1CCOCC(CNC(c3cncnc3)=O)C1)=O)C2 CCC(O)CC(=O)NC1CCC(C(=O)NCc2cnn(C(C)C)c2)C1 C1(N(C(C2CC23CCC3)=O)CC)CCC(NC(=O)C(C)=CCO)CC1 C(=O)(C1=CCCC1(C)C)NCC1(COC)CN(C(C2OCCOC23CCC3)=O)C1 Cc1nc(CNC(=O)CC2CC(F)(F)C2)oc1C(=O)N(C)CC1OCCC1(C)C c1(C(=O)NC2C(OC)CN(C(=O)C(C)CC3CCC3)C2)c[nH]c2cccc(F)c12 c1(C(N2CCC(OCCNC(c3c(C)cc(C)o3)=O)C2)=O)cc(S(C)(=O)=O)co1 c1(NC(C2C3(CN(C(CCOC)=O)C3)C2)=O)cccc2[nH]nc(I)c12 C1(NC(COCCC)=O)CN(C(c2ccccc2N)=O)CCC12CCC2 c1(CCNC(c2cccnc2)=O)cc(C(=O)N(C2CC2)CC2C3COCC23)no1 C1(CNC(c2c(OC)n(C)nc2)=O)CN(C(C2CC2C(C)(C)O)=O)CC1(F)F N1(C(=O)CNc2ccccn2)CCC2CCN(C(=O)CSS(C)(=O)=O)C2C1 C(=O)(CC1OCc2ccccc21)NC(CN(C(c1cn(CCC)nn1)=O)C)(C)C c1(C(=O)NC2C(NC(CCc3cnc(C)o3)=O)C2)cc(F)c(Br)cc1F CCC(C)CCC(O)CC(=O)NCCNC(=O)CS(=O)(=O)C(C)(C)C C(C)(C)(CC(=O)NCCc1cnnn1C)n1cc(CCCOC)nn1 N1(C(c2c(-c3cn(C)nc3)ocn2)=O)CC2CC(C1)C2NC(=O)Cc1csnn1 CC(=O)CCCC(C)C(=O)NC(C)CCN(C(=O)CSc1ccccc1F)C C1(CNC(C2C(C)CC=CC2)=O)CN(C(c2ncoc2C2CC2)=O)CCC1(C)C C(C#CC(=O)NCCNC(=O)NCC)NC(CC=CC=C)=O C1(CNC(CCSCC)=O)CCC2(CCC2)CN1C(c1cccc(N(C)C)c1)=O C(=O)(C1=CCc2ccccc21)N1CCC(NC(C2(C(N)=O)CC2)=O)C(CO)CC1 N1(C(C2(C(=O)NC)CC2)=O)CCC(C)(NC(C2CC(N3CCOCC3)C2)=O)CC1 C1(C(=O)Nc2c(SC)cccc2)CC12CCN(C(=O)OCCC(C)(C)C)CC2 N1(C(CCC2(NC(CC3CCCC(C)O3)=O)CCC2)=O)CCC2(CNC(=O)N2)C1 c1(C(N2C(C)CCC(Cc3ccco3)C2)=O)nccn2nc(Br)c(I)c12 N1(C(CSCc2ccc(C)cc2)=O)CC2CCCC(C1)N2C(C1CC1(Cl)Cl)=O c1(C(=O)NCCC(CNC(C=CC(CC)C)=O)O)cc(Cl)c(C)cc1OC C1(C(=O)NCC2C(C)CCN2C(=O)CCC2CCCC(=O)N2)CC(C2CC2)=NO1 N1(C(c2nc(C)nn2C)=O)CCC2CN(C(=O)CC(C)c3ccncc3)CC2C1 C1(C2CC2)(CNC(c2scc(C)c2C)=O)CCN(C(C2(C(F)F)CC2(F)F)=O)C1 c1(CNC(C(COCC)N=[N+]=[N-])=O)cnn2c1CN(C(=O)Cn1nccn1)CC2 c1(CC(=O)NC(C)C(CO)NC(C2CC2(F)F)=O)cccc(OC(F)(F)F)c1 c1(Cn2cc(CN3C(CC(F)F)CCC3)nn2)ccc(Br)cc1C(F)(F)F N1(C(C2(C#N)CC3CC3C2)=O)CCN(C(=O)Cn2c(C3CC3)nnc2S)C2(CC2)C1 c12cc(ncn1)N1CCCC1C(=O)NC2.C1(C(F)(F)F)(CCOC)CC(C)(C)C1 N1(C(CCc2ccc(C)o2)=O)CCC2CN(C(=O)COCCF)CCC12 CC1(C)CN(C(c2ccccc2CC(F)(F)F)=O)CCC1NC(=O)CC1=CCCC1 Cc1cccc2oc(C(N3CC(O)C(O)C3CNC(c3ncn(C)n3)=O)=O)cc12 N1(C(C(c2c(C)cncc2)C)=O)CCC2CC2(NC(=O)COCCCOC)CC1 C(CCC(C)C)=C(C)C(=O)NCCC(C)NC(C1CCN1S(C)(=O)=O)=O C(=O)(C1=NN(CCO)C(=O)CC1)NC(CNC(C(CCC(C)C)F)=O)CC(C)C c1(-c2nc(-c3ccc(C)o3)nn2CC(C)C)cnn2c1NCC2 c1(CNC(C2CCCN2C2CC2)=O)cccc(-c2ccc(O)nn2)c1 N1(C(c2cc(CC)oc2C)=O)CCC(NC(=O)C2=CCCO2)C(C)C1 c1(C(N2CC3(CN(C(CCS(C)=O)=O)C3)C2)=O)cc2cc(Cl)c(Cl)cc2[nH]1 C1(CNC(Cc2ccc(C)s2)=O)CN(C(C2(N3CCNC3=O)CC2)=O)CC1(F)F C(=O)(C(C)CC(C)CC)N1C(CC)CCC1C(=O)NC1CC(N2CCCC2)C1 C12(C(N(CCCNC(Cn3ccc(C)n3)=O)C(C)C)=O)CC1COC21CCC1 c1(C(N2CC(NC(C(C)C3CC3)=O)C(C)C2)=O)ccn2c(O)nnc2c1 C(CC(C)(C)C(=O)N1CCC(CNC(C23CCC(OC)C2C3)=O)CC1)SC C(=O)(CCC(F)(F)C(F)(F)F)NC(C(C(C)C)NC(c1cc(C(N)=O)c[nH]1)=O)C N1(C(c2c(CCC)n[nH]c2)=O)CCC12CN(C(C1CC3(C1)CC(F)C3)=O)C2 c1(CC(N2C(CNC(CC(C=C)(C)C)=O)CC2)=O)c(Cl)ccc(O)c1Cl Cc1cc(C(N2CCC(NC(c3cccc(C)c3Cl)=O)C2)=O)[nH]c1C#N CCC(C)C(C(=O)NCCc1ccc(O)cc1)N(C(=O)CC(C)C)C CCCCC(CC)C(=O)NCC1(F)CC(NC(C2(C)CC(=O)N(C)C2)=O)C1 c1(-c2ccc(CNC(C=CC)=O)cc2)ccc(OC)cc1-c1nn[nH]n1 c1(C(N(CC(C)N(C(C(C)=CC)=O)C)C)=O)cc(S(=O)(=O)N(C)C)oc1C C1(C(=O)NCC(=O)O)CCCN(c2ccc(C(=O)O)cc2)C1 C1(C(=O)NCC2(O)CN(C(C(C)=C(CC)C)=O)C2)COCC2(CCC2)O1 N1(C(CCSCCC)=O)CCN(C(c2cnc(=N)[nH]c2)=O)C(C)C1C C1(C(N2CCN(C(=O)CN(C(=O)CC(C)O)C)CC2)=O)(CC)CCCCC1 N1(C(C=CCOC)=O)CCS(=O)(=O)C(CCNC(=O)CCN2CCNC(=O)C2)C1 Cc1cccnc1C(=O)NCCC(=O)OCCc1n[nH]cc1NC(C)C C1(COC)(NC(C2CCCC2O)=O)CCN(C(c2cc(C(=O)OC)n(C)n2)=O)CC1 N1(C(C(CC=CC)NC(=O)Cc2cc(C)no2)=O)CCN(C)CC(O)C1 C1(NC(=O)NC(C)(C)C(O)C(F)F)CC12CCOc1ccccc12 N1(C(c2c(CCC)n[nH]c2)=O)CC(NC(C2(CCF)CC2)=O)C2(CCC2)C1 C1(C(N2CC(C=C)C2)=O)(COC)CCN(C(c2oc(C)nc2C)=O)C1 CN1CC(C(=O)NCC2COCCN2C(=O)C(N)=O)CC1=O C1(C(=O)NCC=CCNC(CC2CC(CC)C2)=O)CCCC2CCCN12 C(=O)(C(O)CCCCC)NC(CCC=C)C(=O)N1CC(NC(C)=O)C1 c1(C(=O)NCCN(C(C2(Cl)CC23CCC3)=O)C2CC2)cnc2c(c1)COC2 C(CC(=O)NC(C)(C)C(C)NC(=O)CCC1(C)CC1)(C(F)(F)F)OC C1(C)(C(=O)OC)CCC(N(C(CO)C(O)c2cccnc2)C)CC1 CCC(C)C(C)CNC(c1cn(CCNC(c2cc(OC)ns2)=O)cn1)=O CC(C)(CCC(=O)N1CCC(C)(CC2CC2)CC1)NC(c1cccnc1)=O C(=O)(C1CCCc2nncn21)N(CCCCN(c1nccc(C#N)n1)C)C C1(NCC2(n3ccnc3)CCCC2)CCN(CN(C)C(C2(O)CCCC2)=O)CC1 C(=O)(C(F)CCC(C)C)NCC1CCCN(C(C2CCC(CCC)CC2)=O)CC1 CC1CN(C(c2cc(-c3cccs3)[nH]n2)=O)CC(C)N(C(c2cnco2)=O)C1 C12(NCc3ccc(C(N(C)C4CC4)=O)nc3)CCCCC1NCC2 Cc1ncc(NC(=O)C(Cn2ccnn2)NC(c2cc(CO)[nH]n2)=O)cn1 Cc1nc(Nc2cnc(C(N3CC(O)C(F)C3)=O)s2)c2sccc2n1 C(=O)(CCS(C)(=O)=O)N(C)CC1CCCN(C(c2cc(COC)on2)=O)C1 c1(CC(=O)NCC(CN(C(=O)CCCN(C)C(C)=O)CC)O)cccc(F)c1 Cc1nn(C)c(C)c1CC(C)C(=O)N(CCCNC(C1(O)CCOCC1)=O)C c12cc(ccc1Br)CN2.c1(NC(c2c(C(=O)OC)cccc2)=O)cc(Cl)cc(Cl)c1 C1(CCC)CN(C(=O)CCC2CCCN2C(=O)Cc2scnc2C)CCO1 C(CC(F)F)(C(=O)NCC1(O)CC=CC1)NC(c1cc(=N)[nH]cc1)=O Cc1cc(N)cnc1C(=O)NCCC1CCCN(C(C2CC2c2ccco2)=O)C1 C1(NC(C2CCCC(OC)C2)=O)CCCCN(C(C2(c3cccs3)CC2)=O)C1 C=CCC(CNC(=O)C(C)(C)F)C(=O)NC(C)C(=O)OCC1CC1 Cc1ccc(C(=O)NCCCC(C)NC(=O)CCCc2cccs2)o1 C(C(CNC(C1CCC(F)(F)CC1)=O)CC(F)(F)F)NC(C(C)(C)C#N)=O CC#CC1CCN(C(=O)CC2(NC(C3(N(C)C)CC3)=O)CCC2)C1 c1(C(N2CC(NC(C(Cc3c(C)nc[nH]3)O)=O)(CO)C2)=O)cccc(CO)n1 C(=O)(CCC(c1ccccc1)N(C(=O)C(C)N1CC(C)C1)CCC=C)OCC C1(CC)CC(O)CN1C(C1CCC(CNC(=O)CC2(O)CCC2)O1)=O C(=O)(C1CCc2nnc(C)n21)N1CC(NC(C=C(C)Cl)=O)C(O)CC1 C1(C(=O)NCCC(C)(C)NC(CCOC(C)=O)=O)CN2CC3CC2(CO1)C3 C(=O)(CCCCC(=O)N(C)CC1(NC(c2cn3ccccc3n2)=O)CC1)NC c1(OC)cc(C(N2CCCC(O)(CNC(C3CCS(=O)(=O)C3)=O)C2)=O)cc(F)c1 CCC(C)(CC)C(=O)N1CC(n2cc(C(O)C3CC3)nn2)C(C)C1 c1(OC)cc(NC(C2CN(C(c3ncn(C(C)C)n3)=O)CC2C)=O)cc(OC)n1 C1(NC(C2C(=C)C2)=O)(CNC(=O)CC(=O)NCC)CCCCC1 c1(CNC(CCN(CC#C)C(c2cscc2C)=O)=O)ncoc1C1CC1 N1(C(Cc2n(C)nnc2)=O)CCC(NC(C2CC3CC3C2)=O)C(O)C1 N1(C(C2N(C(c3c(C)cn(C)c3)=O)CCC2)=O)CCC2(CCOC2)CC1 n1(CC(=O)NCCc2ccc(-c3cccs3)cc2)nc(C2CC2)oc1=O c1(C(C(=O)NCCC(C)N2CCCC2)N)cccc(-c2ccc(C)cc2)c1 C(c1ccc(C(N2CC(NC(=O)CCc3ncco3)C2)=O)cc1)=CC(=O)O C(N=c1[nH]c(C(F)F)co1)c1cnc(C(=O)OC)s1 C(=O)(C1=CCCOCC1)NCCCOCCNC(c1nccc(CC)c1)=O C=CC1(NC(c2cnc(CNC(=O)C(C#N)C(C)C)nc2)=O)CCCCC1 C(=O)(CC(C)C(C)C)N1C(C(=O)NCCOCCCOC)C=CCC1 N1(C(c2cncc(C)c2)=O)CC(C(N2CCCC(CO)C2C)=O)C(F)(F)C1 N1(C(c2cc(OC)cc(Br)c2)=O)CC2ON=C(CNC(=O)CCC3CC3)C2C1 N1(C(C(C)NS(C)(=O)=O)=O)CCC2CN(C(=O)CCSc3ccccn3)C2C1 Cc1cccc(C(=O)N(CCCCN(C)C(c2conc2C2CCCO2)=O)C)c1 c1(C(N2C(C(N3CC(c4n(C)ncc4)C3)=O)CCC2)=O)cc(I)ccc1F N1(C(=O)CCc2cccc(Cl)n2)CCCC(Cn2cc(C3CC3)nn2)(CO)C1 c1(NC(C2(C)CCN(C(c3ccc(I)cc3Br)=O)CC2)=O)cccc(Cl)c1C#N CC1COCC(CC(N2CCC(CF)(NC(=O)CC3CCSC3)C2)=O)O1 c1(C(N(C(CNC(c2cn(CCC)nn2)=O)C)CC)=O)cnc(F)c(C)c1 Cc1c(C(N2CC(NC(c3n[nH]c(C4CC4)n3)=O)CC(O)C2)=O)cccc1F N1(C(C(CC(C)(C)C)(C)C)=O)CC(NC(=O)CC2=CCCC2)C2(CCOCC2)C1 c1(C(N2C(CNC(CCc3cc(C)[nH]n3)=O)CC2)=O)n[nH]c2c1NCCC2 C1(CNC(CCC(=C)C)=O)CC2CCC1N2C(c1cccc(O)c1Cl)=O N(C(=NCC(C)F)N1CCC(n2ccccc2=O)CC1)C1CCCC1.CCC N#CC12CCOCC1C(N1CCC(CF)CC1)C2 C1(C2CN(C(C3(C(=O)OCC)CCC3)=O)C2)=NOC(C)=NC=N1 C(=O)(C(C)C(C)NC(=O)NC1CC(N2CCNC2=O)C1)OCC C12(CNC(=O)NCC(N3CCC(O)C3)C)CCC(C(F)(F)F)(CC1)CC2 N1(C(c2ccn(C(C)C)n2)=O)CCCC(CNC(c2cncc(F)c2Cl)=O)CC1 CC12CSCC1CN(C(=O)C=CC(C)(C)NC(C1CC3(CC3)CO1)=O)C2 N1(CCC(=O)NC(CC)CN(C)C(c2ccc(OC)o2)=O)CCOCC1 c1(C(=O)NCCOCOCCNC(CC(=C)C)=O)nccc2[nH]ccc12 C1(NC(C=Cc2ncn(C)c2)=O)COC2C(NC(=O)C(F)C(F)(F)F)COC12 C(c1ccc(-c2ccc(F)cc2)s1)=CC(=O)NC(CC)CNC(c1csnn1)=O C(=O)(N=c1ccn(C(C)(C)C)[nH]1)C1OC(C(=O)O)CN(CC=C(C)C)C1 c1(C(=O)NCC2(C)C(NC(C=CC(C)C)=O)CCC2)ccc(O)nc1Cl c1(N2C(C(=O)Nc3cc(C)c(O)cc3)CC(C)C2)ncc2c(ccn2C(C)C)n1 CCC(F)(F)CC(=O)NCCC1CCN(C(C2CC2(C)C(C)C)=O)CC1 c1(OC)cc(C)c(NC(C2CC2C(=O)NC(c2ccc(F)cc2)C)=O)cc1Br Cn1cc(C(=O)NC2(CCCNC(=O)CN3CCOCC3)CCCC2)nn1 C12(CCC(=O)N(CCCCN(C(c3c(C)con3)=O)C)C)CCC(CC1)C2 c1(CC(=O)NCCC(C)NC(C2CC(OC)C2)=O)ccccc1S(C)=O C=CCCC(C(=O)NC1CC(=O)N(O)C1)NC(=O)CN1CCOCC1 c1(C(N2CCC(CNC(c3cn(CCO)nn3)=O)C2)=O)cn2cc(Cl)cnc2n1 CC(C)(C)C(CN1CCCC(N)C1C(F)(F)F)C(=O)NCc1cscn1 C1(C(=O)NCC(C2CCCC2)NC(c2sccc2F)=O)CCC(C(F)(F)F)CC1 N1(C(CC2CC(=C)C2)=O)CC2CCC(C1)N2C(C12CC(c3ccccc3)C1C2)=O C1(CNC(c2c(C)nns2)=O)CCC(F)(CNC(=O)CC2C=CS(=O)(=O)C2)C1 C(CC(C)C)(C(=O)NCc1ccc(F)cc1C)N(C(C(CCOC)OC)=O)C C1(C(=O)NCCC(C(C)C)OC)COCCN(C(c2ccc(C(F)F)cn2)=O)C1 C(=O)(C(CCC=C)NC(c1ccnc(C)c1C)=O)N(C(C#C)C)C N1(C(CC(C=C)C)=O)CC(NC(C2(CO)CCCCC2)=O)CCC(O)C1 N(C1CCCn2cnnc21)C(=O)C(C1CCN(C(=O)CCCC(F)(F)F)C1)F c1(C(=O)NCC2(C)N(C(CN(C(C)=O)C)=O)CCC2)ccccc1N=[N+]=[N-] CC(C)C(C)(CNC(=O)CN1CCC(C)C1)NC(=O)C(c1ccc(F)cn1)(F)F c1(C(C)NC(COC)=O)ccc(CNC(c2cc(Br)ccn2)=O)cc1 c1(C(=O)NC2CCCC(N(C(=O)Cc3csnn3)C)C2)ccc2[nH]c(=N)[nH]c2c1 c1(C(=O)NC2CCN(CC=C)CC2C)noc2cc(Cl)ccc12 C(=O)(C(CNC(C1CC(O)CN1C)=O)C(C)(C)C)N(CC(C)O)CC(C)O N1(C(C2(OC(C)C)CC2)=O)CCOC(C(C)NC(=O)C(C)NC2CCCC2)C1 N1(C(CC=CCCCCC)=O)CCN(C(C2(O)CC(F)(F)C2)=O)CC(C)(C)C1 c1(C(=O)NC(CC)CNC(=O)CCC2CC2(Cl)Cl)ccncc1F C1(NC(CCC=C=C)=O)COC2CN(C(C3CN(C(=O)C(C)(C)C)C3)=O)CC12 N1(C(C=CC(CC)C)=O)CCCCCC1CNC(c1c(C)oc(C)c1Br)=O c1(C(=O)NCc2ccco2)ccc(C(C(=O)OC)N(CCCC(C)O)C)c(C)c1 CCC(C)C(C(=O)NC1CCN(C(C2SCCCS2)=O)CC1F)NC(N)=O CC(C)CCCC(C)C(=O)N1CCC2CN(C(c3cc(O)c(C)cc3C)=O)C2C1 N1(C(C(CC)N(CC)CC)=O)CCOC(CCC(=O)NC(c2ccc(F)cc2)C)C1 C1(OC)CCCC(CC(N2CC(C(F)(F)F)C(CNC(=O)C#CC3CC3)C2)=O)C1 CCCCCC(O)CC(=O)NCCNC(c1[nH]nc2ncccc12)=O C1(N(C(=O)CN)S(C)(=O)=O)CCN(C(=O)CCc2ccc(OC)cc2)CC1.CCO C12(NC(c3ccc(SC)s3)=O)CC1CN(C(c1cnc(-c3ccccn3)s1)=O)C2 N1(S(CC)(=O)=O)CCCC(C(N2CCC(CNC(C3(CO)CCCC3)=O)C2)=O)C1 C1(CCCC)CN(C(c2ccc(Cl)s2)=O)CCN1C(C1CC1COC)=O N1(C(CC=CC=C)=O)CCCC1(CNC(=O)COC(C)CC)COC C(C)(CS(C)(=O)=O)NC(C(C)N(C(C1CCNC1=O)=O)C1CC1)=O c1(OC)ccc(C(=O)NC2CN(C(=O)C(C)Sc3ccccn3)CC2C)cc1F C(=O)(C(O)C(F)F)N(C1CCN(C(C2CC(F)(CO)C2)=O)CC1)C CN1C(=O)CCCC1C(=O)NC1CCCCC1NC(=O)Cc1cncn1C Cc1nc(C)c(CC(N2CCN(C(C3(N(C)C)CCC3)=O)C(CO)C2)=O)c(O)n1 C(=O)(C(C)C(O)CC)N(CCNC(c1cc(Cc2ccccc2)n(C)n1)=O)CC N1(C(CN2CC(=O)NCC2)=O)CCn2cnc(C3=CCSCC3)c2C1 C(=O)(C(CC(C)C)NC(=O)CC(C)C1CC1)NC1(CCOC)CCC1 C1(C(=O)NC(CN(C(=O)CNS(C)(=O)=O)C)(C)C)CCCOC1c1cn[nH]c1 C=C1CCN(C(c2ccn(CCNC(C3CCC(CC)C3)=O)c2)=O)C1 C1(NC(C(CCC)O)=O)CCN(C(=O)C=CCO)CC(C)(C)C1 C1(NC(C(C=C)(C)C)=O)CCCCCC1C(=O)NCC(O)CC(C)(C)C C1(CC)Oc2cc(CC(=O)NC(C3(CO)CCCC3)=O)ccc2NC1=O c1(C(=O)NC(CNC(c2cccnn2)=O)C2CC2)ccc2cc(Cl)ccc2c1 CC1CN(C(=O)CCSCCNC(=O)CN2CCCC2C)CC1(F)F Cc1ccc2c(c1)CC(C)N(Cc1cn(C(c3ccccn3)C)nn1)C2 C(CCC(O)CO)NC(C(C1CCOC1)NC(c1csc(O)n1)=O)=O C1(C(=O)NCC(=O)NCCN(C(=O)C(C)(C)C)C(C)C)CCc2c[nH]nc2C1 C1(CC(N2C(CCC)COCC2)=O)CCCN(C(C2CC(C)(O)C2)=O)CC1 CCCC(C(O)C(=O)N=c1ccn(CC(N)=O)[nH]1)NC(=O)CCCCCC C(=O)(C(C)CC(F)(F)F)NC1CN(C(CCCCCOC)=O)C(CO)C1 Cc1ccc2[nH]c(C(N3CC(C)N(C(=O)CCCCC4CC4)CC3C)=O)cc2c1Cl C(=O)(CS(=O)(=O)CC)NCCCN(C(c1c(OC)scc1)=O)CCOCCO c1(C(=O)NCC(CC)NC(=O)CN2CSCC2=O)ncc(SC)s1 C(CC)(C(=O)N1CCC(NC(=O)CNC(=O)COCCSC)C1)OCC c1(C(=O)NC(CC)CNC(c2ccn(CCOC)n2)=O)cccc2c1OCC2 C(C(=O)NCC1(CC(=O)NC2C=CCCC2)CC1)(C(C)(C)C)N(C)C N1(C(CCCCCC=C)=O)CC2(C)CN(C(C3C4CC(F)(F)CC34)=O)CC2(C)C1 c1(C(=O)NCC(C)NC(C2CCC(=O)NC2)=O)cccc2nn(C)nc12 c1(OC)cncc(C=CC(=O)NCC(C)NC(=O)CC2CC3C=CC2CC3)c1 C(=O)(C(C)(C1CCC1)NC(=O)CSC(C)C)N(CC(C)OC)C N1(C(CCC(C)(C)O)=O)CCC2CCCC12CNC(=O)C(F)(F)c1cscn1 c1(N(C(C2CC(C)CN2C(=O)CO)=O)CC2CC2)ccc(F)c(F)c1 C=CCCCCC(=O)NC1(CC(N2CCC(COC)C2(C)C)=O)CCOCC1 Cc1ccn(C)c1C(=O)NCC(C(C)(C)C)NC(=O)C=CC(C)C CCC(C)(C)CCCC(=O)N1CCOCC1CN(C(=O)C=Cc1ccnn1C)C Cc1csc(C(C)(C)C(=O)NC2CN(C(=O)C=CBr)C2)n1 c1(OC)ccc(C(=O)N(C)CCOCCN(C(=O)C(F)C2CCC2)C)nc1Cl N1(C(C2COCCN2C(c2ccc(CF)cc2)=O)=O)CC2(CCC1CO)CC2 C(=O)(C(O)CCCNC(C1COCC1(C)C)=O)NCCc1cn(CC)nc1 c1(C(N(CC(CC)NC(C2C=CCCC2)=O)CC)=O)cccnc1-n1ccnc1 CCC(CC)CCCN(C)C(C1CN(C(=O)C(C)SC(C)C)CC1C)=O C1(CC)OCCC1C=O.N1(N2CC(CN(C)C)C2)CC(OCC=O)C1 N1(C(C23CC(C(=O)OC)(C2)C3)=O)CCN(C(=O)CC2CCC(C)(C)O2)C(CCO)C1 C1(C(NOCCC)=O)CCN(C(=O)C(CO)C(F)(F)F)CC1(C)C N1(C(Cc2scc(CC)n2)=O)CC2CCCC2(C(N2CCC(CO)(CO)C2)=O)C1 c1(C(=O)NCC(CC)(C)NC(=O)CSCC(F)F)ccc(C(F)F)cc1 C1(C(=O)NC2CC(OC)CN(C(c3ccccc3F)=O)C2)CCCN2CCCC12 C=CC1(CC(=O)NC(c2cn(C)cn2)C)CN(C(=O)COC(C)CCC)C1 C1(NC(c2ccco2)=O)CN(C(C2CCN(CC(F)(F)F)C2)=O)CC1C(F)(F)F C12(CNC(c3c(SC)snn3)=O)CCC1CN(C(=O)CN(C1CCCC1)C)C2 N1(C(Cc2ccc(C)o2)=O)C2CCC1CN(C(c1ocnc1C)=O)C2 C1(NC(=O)C=Cc2ccco2)CC2(CCC(NC(C34CCC(F)C3CC4)=O)CC2)C1 N1(C(c2c(C)csc2)=O)CCC(C(N2CCCC(Br)C2)=O)C2OCCC12 CC(C)CC(CNC(=O)C(F)=CCCF)NC(c1ccc(C(O)CF)cc1)=O C1(CNC(Cc2nnc(C)s2)=O)CCCC(CNC(c2c[nH]nc2C2CC2)=O)C1 C(=O)(C(C)CC(=O)NCC12CC(C(=O)NC3(C(=O)N(C)C)CC3)(C1)C(C)O2)OC c1(CC)c(F)ccc2c1CN(c1nc(NCCN=[N+]=[N-])c3cnn(C)c3n1)CC2 Cc1ccc(C#N)cc1-c1cn2cnc(C(=O)NC3CC(F)C3)c2s1 Cc1cc(C(=O)NCC2CN(C(c3cc(Cl)n(C)n3)=O)C3CC23)cnc1F N1(NC(C2N(C(C3C=C(C)CS3)=O)CCCCC2)=O)Cc2ccccc2C1 CC1=NOC(C)(C(N2CC(C(C)NC(c3cn(C4CCCC4O)nn3)=O)C2)=O)C1 N1(C(C(CCC)O)=O)CCCC(NC(C2(C(F)(F)F)CCCCC2)=O)CC1 N1(C(c2c(CNC(c3n(CC)nnc3)=O)occ2)=O)CCCOC(C)C1 c1(C(=O)NCC23CC(NC(C(C)OC)=O)(C2)C3)cc2c(F)cccc2[nH]1 N1(C(CC(CC)(C)C)=O)CCC2CN(C(c3csc(C(F)(F)F)c3)=O)CC12 C1(NC(CCC)=O)CN(C(=O)CC2CCC(F)(F)C2)Cc2ccnn2C1 N1(C(COCC=C)=O)CC2(CCOCC2C(=O)N(CCO)CCOC)C1 CN1CC(O)CCC1C(=O)NCCCNC(=O)C(c1ccnn1C)O n1(C(C)C)cc(C(N2CC(C(C)NC(=O)CCc3nncs3)C2)=O)nn1 O=C(C1CCCc2nc[nH]c21)NCC1CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CCO1 c1(-n2c(C3CCC(C(F)(F)F)O3)nc(COC)n2)cc(F)ccc1-n1cncn1 C1(CNC(=NCCc2cccc(C(=O)OC)c2)NCC2CC2)CC2CCC1CC2 C1(c2nnnn2CC(F)F)(NCC2C(C)(C)C2Br)CC2(CC2)C1 c1(NCc2c(C)ccc(C#N)c2)ccc(S(=O)(=O)NC2(C3CC3)CC2)cc1Br c1(C(=O)NC2CCC(NC(c3cccc(C)c3Cl)=O)C2)cc2cc[nH]c2cc1F CC1CN(C(C2(C)CN(C(=O)C(=O)N(C)C)C2)=O)Cc2nncn21 C(=O)(CCCC(F)(F)CO)NCC(CNC(C(C(=O)NCC)(C)C)=O)OC Cc1cc(C(N2CCC(NC(c3cccc4nn[nH]c34)=O)C2)=O)n2nccc2n1 C1(C(=O)NOCCN(C2CCCC2)C)(CC#C)CCN(C(=O)CC2CCN(C)C2)C1 c1(C2CCN(C(C3C(CCCC)CCCC3)C(=O)NC)C2)ccc(Cl)c(Cl)c1 C(=O)(C1=CCC(F)(F)CC1)NC1(CC=C)CN(C(=O)Cc2cnoc2)C1 N1(C(CCc2nc(C)c(C)o2)=O)CCCCCC1CNC(=O)C(C)N(C)C1CC1 N(C(=NCCF)N1CCN(c2ccccc2)C(=O)C1)Cc1n(C)ncc1 c1(C(=O)NC2COCCN(C(=O)NC3CC3)C2)cc(Br)cc2nc[nH]c12 C12(C(N(C3(C(=O)NC=O)CC3)C)=O)C(NC(C3CC4(C3)CC4(F)F)=O)C3CC1C2C3 c1(CCC(N2C(CCNC(=O)CCF)COCC2)=O)ccc(F)cc1Cl N1(C(c2c(C)nco2)=O)CC2CC1C2NC(c1scnc1C1CCCC1)=O C(=O)(C#CC1(C)CCCO1)NCC1N(C(CCOc2cn(C)nc2)=O)CCC1 N1(C(c2ccc(F)cn2)=O)CCC2(CCCN2C(c2cc[n+]([O-])cc2)=O)C1 C(=O)(C1=CC2C=CC(C1)C2)NCC1(OC)CN(C(=O)Cc2cnc(=N)[nH]c2)C1 N1(C(C(C2CC2)OCC)=O)CCCC(N(C)C(c2[nH]nc(C(F)(F)F)c2C)=O)C1 c1(C(=O)NCC2N(C(c3c(C#C)c[nH]n3)=O)CCCC2C)cc(C)cc(Cl)c1N c1(NC2CN(C(C)=O)C2)ccc(S(=O)(=O)NCCC(O)C2CCC2)cc1C#N c1(SC)nc(N(CC(O)CN(C(=O)CCS(C)(=O)=O)C)C)cc(C)n1 n1(CC)cc(SCCSC2C=CCOC2)nn1 C12(CNC(C(CCC)C)=O)CCC(NC(=O)Cc3cncs3)(CO1)C2 Cc1cccc(CNC(=O)CC2C(NC(c3cccnc3S)=O)CC2O)n1 C1(C(=O)NCCCN(CCCOC(=N)O)C)C=CCN(C(c2ccccc2F)=O)C1 c1(C(=O)Nc2c(C(=O)Nc3ccc(Br)nc3Cl)n[nH]c2)cc(Br)cnc1[N+](=O)[O-] N1(C(C=CCNC(CCn2c(C)ncc2)=O)=O)CC(F)CC1CO c1(C(=O)NC(CC)CNC(c2cnn(C3CCOCC3)n2)=O)cc2n(n1)CCO2 C(=O)(CC(C)CC(C)C)N1CC(OCC(=O)NCC(C=C)O)C1 Cc1nc(C(N2CCC(CC(=O)NC(CO)C(C)O)C2)=O)cn1C O=S(=O)(c1ccc2c(c1)OCCCO2)NCC1(SC)CC(c2ccccc2)C1 C(=O)(CCC(C)S(C)(=O)=O)N1CCN(CCNC(c2c(C)n(C)nn2)=O)CC1 c1(C(=O)NCC2(O)CN(C(=O)CC34COCC(C3)C4)C2)cc(F)cc2nccn12 C#Cc1cncc(C(=O)NC(CCOCC)C(N2CCC23CC(CO)C3)=O)c1 Cc1cc(C(N2CC(NC(=O)C=CC3CCCCCC3)C(C)(C)C2)=O)nnc1C c1(CCC)ccc(C(N2CC(CNC(c3coc(C)n3)=O)CC2C)=O)cc1N N1(C(c2c(C)nn(-c3cccc(Cl)c3)n2)=O)CCCN(C(=O)C(N)=O)CCC1 n1(C(C)C)ncc2c(NCc3ncnn3C(C)C)[nH]c(=NC3CC3C3CCC3)nc12 C(C(C)(C)CC(=O)NOCc1cccnc1)NC(C1C(C(C)(C)C)C1)=O Cc1cccc(Br)c1C(C(=O)N1CCC1CN=[N+]=[N-])NC(C1CSC1)=O n1(CC2CCCC2)cnc2c(NC(C34CCCC(OCC)(CC3)C4)=O)ncnc12 C123CC(C1)(C2)CNC3=O.C1(C(=O)NC2CC2CC(=O)OC)(COC)CC1 N#Cc1ncn(CC(=O)NC(CC(=O)NCCCCCF)C2CC2)n1 C(CC(CC)CO)NC(c1nnnn1C1COC1)C.c12ccn(c1)CCOC2 C1(C(N2CC(CNC(c3cccc(C)c3C)=O)C(C)C2)=O)CN2CCC1(C)CC2 C1(CC)CN(C(=O)Nc2ccnn2-c2ccccc2C(F)(F)F)CCN1C CCCC(CCCNC(c1ccc(F)c(CO)c1)=O)NC(C1(CC2CC2)CC1)=O c1(OCC(N2CCOCC(NC(C3(CF)CC3(F)F)=O)C2)=O)cccc([N+](=O)[O-])c1 C1(NC(CSCC=C)=O)COC2(CNC(c3cnc(CC)s3)=O)CC1C2 N1(C(C2CCCN(C(C3(C(C)C)COC3)=O)C2)=O)CC2(CCC2)CC1C CC1(C)CC=C(C(=O)N(CCCC2CCCC2)CCO)CC1 Cc1cnc2c(C(=O)NCC(C3CC3)N(C)C(c3ccc(O)nn3)=O)cnn2c1 Cc1nc(C)c(C(N2CC(O)(CN(C)C(c3cocn3)=O)C2)=O)[nH]1 Cc1cc(C(N2CCC(CC(N3CCOC(C(N)=O)C3)=O)CC2)=O)nn1C1CC1 c1(CNC(CC2(N(C)C(c3cc([N+](=O)[O-])c[nH]3)=O)CC2)=O)cncc(C#N)c1 CCCC(CCC)C(=O)NC1COCCC1NC(c1cccc(O)n1)=O Cn1cc(NC(C2(C)CCCS2)=O)nc1C(=O)NCCCC(O)CO CC1(C(N2CC=CC2CF)=O)CC(O)CN1C(=O)CC1CSCCO1 CC(C)C1=NOC(C(N2CCC(NC(C3CC(F)(F)C3(F)F)=O)CC2)=O)C1 C1(N(C(=O)C=CC(=O)NCc2nc(C)no2)CC=C)CCN(C(C)C2CC2)CC1 N1(C(c2cccc(C)c2)=O)CCN(C(=O)C=CCO)C(c2ccc(F)cc2)C1 C1(NC(CC2(N(C(=O)C(C)c3cc[nH]n3)CC)CC2)=O)COCCC1CO C(=O)(CC(=O)NCCC1CCN(C(c2nc(C3CC3)cs2)=O)C1)OC(C)(C)C C1(SC2(C(N(CCN(C(=O)Cc3cc[nH]n3)C)C)=O)CC2)CCC(F)(F)CC1 n1(CC(=O)NCC(CC)NC(C2COCCC2C)=O)cc(Br)ccc1=O N=c1[nH]ccc(F)c1C(=O)NC1CCOC1c1ccccc1 CC1(C)COc2c(C(=O)NCC(O)CNC(=O)C#CC3CC3)cnn2C1 CCC(C)C(O)C(=O)NC(C)C(CO)NC(C1CCC(N(C)C)C1)=O C1(C(=O)NC2C(NC(C(N)=O)=O)C2)CC2CCC(C1)C2O c1(C(=O)NCCC2N(C(C(P(C)(C)=O)O)=O)CCC2)cnc2c(c1)NC(=O)CO2 C(=O)(CCCS(C)(=O)=O)NC(C(C(C)C)C)CNC(c1cocn1)=O S(=O)(=O)(c1cc(NC(C)=O)c(Cl)cc1F)NC(=O)Nc1cc(OCC)ncc1 C(C(C)C(=O)N1CCC(CN(C)C(c2ccoc2C2CC2)=O)C1)OC C(=O)(C(C)(C)C(C)C)NCCCCCCNC(c1cc(C(=O)OC)sc1)=O C(=O)(C#CC1(C)CCCO1)NCC1(C(=O)NC(CCOC)COC)CC1 c1(C(C)OC(C2(O)CCCN(C(=O)OCC#C)C2)=O)ccc2ncccc2c1 Cc1ccc(Cl)cc1C(=O)NCC(C)N(C(=O)CC1CCC1(C)C)C Cn1cnc2cc(C(=O)NC3C=CCN(C(C4(C#N)CCC4)=O)C3)sc12 c1(C(=O)NC2CCN(C(CCC(=O)N(CC)CC)=O)C2)cc2c(cn1)OCCC2 O(NC(=O)CCC1CCCCN(C(=O)CCOC2CC2)C1)CCC#C C1(NC(C2N(C(C3CCC(=O)NC3)=O)CC(F)(F)C2)=O)CCc2nn[nH]c2C1 C1(c2n(CCOCC)nnn2)(Nc2ccccc2)CC(C)(NCCCC(C)C)C1 C1(CC(=O)N(C)CC2CCCN2C(C2CCC(N(C)C)C2)=O)CCCCCC1 C1(CNC(Cc2cc(C)sc2)=O)(CNC(=O)CN2CCN(C)CC2)CC12CCC2 N1(C(C(C)NC(COC)=O)=O)CC2CCN(C(=O)C3=C(Cl)CCCC3)C2C1C N1(C(c2cnc(Cl)s2)C(=O)Nc2ccc(OC)cc2)CCC2OC(=O)OC2C1 c1(OC)ccc(S(=O)(=O)N2CCN(S(=O)(=O)Cc3cccc(Cl)c3)CC2)cc1F CN1CCN(C(=O)C(N2CCCC(CC(F)(F)F)C2)=O)CC1.C1CCN1C(N)=O N1(C(C2(NC(CCSCC)=O)CC2C)=O)CCC(C)C1 c1(C(=O)NC(C)Cn2cc(C3(O)CCOCC3)nn2)nc2c(cc1Cl)OCCO2 C1(C(F)(F)F)(C(N(C(C)CNC(=O)CC2CSC2)C)=O)CCCC1 c1(NC(c2[nH]cc(C)c(=O)c2)=O)ccc(S(C)=O)cc1 N1(C(C=CC)=O)CCC2(CCCN(c3nc(C)ncc3F)C2)CC1 c1(C(=O)NCCCCCN(C)C(c2cnn(CCF)c2)=O)cc(C(N)=O)cn1C C(C(C)(C(C)C)NC(c1csc(Cc2ccc(F)cc2)n1)=O)NC(C(C)OCC)=O C1(C(=O)OC)CN(c2c(Cl)c(C)nn2C)CCC12CCOCC2 c1(CC)nc(C(=O)NC(CC2CCC2)C(=O)NCC2(CO)CC=CC2)c(C)o1 C1(NC(C)=O)CC=C(C(=O)N2CC3C=CC3C2)C1 c1(CC)cc(C(=O)NCC2CC(O)CN2C(=O)C=CCOC2CCOCC2)n(C)n1 N1(C(C(C)OCC)=O)C2CCC1CC(NC(c1ccccc1-n1cccc1)=O)C2 N1(C(c2cc(C)nnc2O)=O)CC(NC(c2cccc(Cl)c2)=O)C2CCCC12 c1(C(=O)NCC2(C)COCCN(C(C(C)SC)=O)C2)c(O)ncc2c1CCC2 C1(CNC(c2n(CC)c(O)nc2)=O)CN(C(c2ccc(F)c(N)c2)=O)CCCO1 C1(C(=O)OCC(COC)Sc2ccco2)CC(=O)N(CSc2cccc(C)c2)C1 c1(OCC(C)C)ccc(NC(N2CCC2CCCn2nccn2)=O)cn1 N1(C(C(N2C(=O)CCC2=O)C)=O)CC(F)CC1CN(C)C(c1cncc(F)c1)=O Cc1cccc(C)c1CC(C)NC(C1(C)CCN(C(=O)Cn2ccnc2)CC1)=O N1(C(c2c(NC)scn2)=O)CC(C)(C(N2CCSCC2)=O)CC1(C)C C1(OCCCNC(C=C(C)C)=O)CCOC1=O.C1(C)(C)C=CC(=O)N1 CC1=C(C)CC(C(N2CC3CC(NC(=O)CSc4ccc(F)cc4)C2C3)=O)CC1 CC#CCCC(=O)N1CC(C(C)NC(=O)CCc2ccccc2OC(F)(F)F)C1 O=C(CC(C(F)(F)F)NC(c1cscn1)=O)NCc1cccc(F)c1 c1(-c2nc(CN(C(=O)CC3CCC3)C(C)CC3CCCO3)on2)cccc(Br)c1 c1(-c2ccn(-c3ccc(OC)c(F)c3)n2)ccc2nc(C(=O)OC)cn2c1 C1(C(N(C(c2cccc(F)c2)CO)C)=O)CCc2nc(C(F)(F)F)[nH]c2C1 N1(S(Cc2ccc(C)cc2)(=O)=O)CCC(F)(F)C(C(=O)Nc2cc(Br)nn2C)C1 C1(CCN(C)C)CN(C(c2ccc(Cl)o2)C(=O)NCc2ccc(F)cc2)CCO1 c1(CC)cc(C(=O)NCCC(C(C)C)NC(=O)C(C)NC(C)(C)CC)ccc1C N1(CC(=O)NCC=CCNC(C(C)NC(c2ccco2)=O)=O)CCc2sccc2C1 C(CC(C)CCNC(c1ccnn1C1CCCCC1)=O)NC(CNC(=O)NC)=O N1(C(C(N2CSCC2=O)C)=O)CCN(C)C(C(=O)NOCC2CNC(=O)C23CC3)C1 C1(NC(CCCn2ncc(C)c2)=O)CC(CO)N(C(=O)Cc2ccc(O)nc2)C1 Cc1cccc(CC(=O)NCC(C(C)C)NC(C2(Br)CC23CCC3)=O)c1 N1(C(C=CCC#N)=O)CC(CNC(c2cccc(O)n2)=O)C2CC12 C1(C(=O)NCC=CCNC(c2c(C)ncn2C)=O)CCCC(=O)N1C c1(C(N2C(CN(C(C3CCC(OC)C3)=O)CC)CCC2)=O)ccc(OC)cc1F C12(CNC(C3(N(C)C)CC3)=O)CCCCC1N(C(c1snc(O)c1Cl)=O)CC2 N1(C(c2c(C)ccnn2)=O)CCN(C(C2CCCN(C(C)C)C2)=O)CC(C)(F)C1 c1(NCC(c2ncc[nH]2)C)nc(N2CCN(C)C3(CC3)C2)nc2c1COC2 Cc1[nH]c2cnc(Cl)cc2c1C(=O)Nc1nccnc1N(C)C C=C=CC(C)C(=O)NC1CCN(C(=O)NCc2nnc(-c3ccc(F)cc3)s2)C1 CCC(CO)C(=O)NC(C1CN(C(=O)Cc2ccc(O)nc2)C1)C C1(F)(NC(Cc2cc(OC)ncc2)=O)CCCN(C(=O)COC2CCOC2)C1 CN1CCN(C(C2CCOCCN2C(=O)C=CC2CCOC2)=O)CC12CC2 N1(CC)CCOC(C(=O)N(C2CC(NC(=O)COC(C)C)C2)C)C1 C1(F)(CNC(C(CC)Cc2ccccc2)=O)CCN(C(C2COCCOC2)=O)CC1 C1(NC(C2CCN(CCCCC)CC2)=O)C2CC1CN(C(C1CCCCC1)=O)C2 C12(NC(C3ON=C(CC)C3)=O)CCC(CC1)N(C(=O)CC1C=CCC1)C2 C1(NC(CCCCCSC)=O)CCCCC12CCN(C(c1csc(Cl)c1)=O)C2 C1(C2CCC(=O)NC2)(C(N(CCCn2cc(C(C(=O)OC)(C)C)nn2)C)=O)CCC1 C1(CNC(c2ccc(CNC(C)=O)o2)=O)CC2(CC2)CN1C(C1C2CC3C(C2)C13)=O Cc1c(NC2CC3CCCCC23)ncnc1NC1CCC(c2ncc[nH]2)CC1 C1(CNC(C(CC(C)C)(C)O)=O)CN(C(c2ccnn2C(C)C)=O)CCC1(C)C C1(CNC(C=CC=CC)=O)CC2CCC1N(C(=O)C(C1CC1)C1CC1)C2 N(C1CCCc2n[nH]cc21)C(CC)CNC(=O)OC(C)(C)C C1(NC(C(C=CC)O)=O)CCN(C(c2ccc(C)cc2O)=O)C12CC2 C12(C(N3CCC(CCC)(CO)C3)=O)CCCC1CCN2C(=O)CC1COCCO1 CC(C)C(CC(=O)N(CCNC(C1CC(C2CCC2)C1)=O)C(C)C)C(C)C Cc1ccc(CC(CO)NC(=O)C(N2CCC(c3ncccn3)C2)=O)cc1 c1(C(=O)NCC2(C(N)=O)CC2)ccnc(CNC(=O)CCC2CCC2)c1 c1(C(=O)NCCNC(C(c2ccccc2F)OC)=O)cccc(C(C)(F)F)n1 N1(C(C(=Cc2ccco2)C)=O)CCCC(NC(c2ccsn2)=O)CC1 c1(C(N(C2CCCN(C(c3ccn(CC)n3)=O)C2)CC)=O)ccc2n[nH]cc2c1 N1(C(CCC=C)=O)CCN(C(c2scnc2Cl)=O)C(c2ccncc2)C1 c1(CC(=O)NC2COCC2NC(C2(CO)CC2)=O)ccc(Cl)cc1F N1(C(C2NC3C(C2)C3)=O)CCCCC(OC)C1.C(C(=O)NCC)(C1CCC1)OCC c1(NC(C2(F)CCN(C(C(CC)OCC)=O)C2)=O)cccc(Cl)c1O c1(OCCNC(C)COc2nc(OCC)ccc2C)ccccc1[N+](=O)[O-] c1(C(=O)NC2C(NC(C(c3cc(C)sc3)(F)F)=O)COC2)ccc([N+](=O)[O-])cn1 CC(C)CC(C(=O)N1CC(CNC(=O)CC2(O)CCCCC2)CC(O)C1)N(C)C C(=O)(C(F)C(C)CNC(C1CCCC2(CC2)C1)=O)N1CCC(OC(C)C)CC1 N1(C(c2cc(OC)no2)=O)CCCCC(NC(C2CCC(F)(F)C2)=O)C1 C1(OC(C)=O)CC2CC1CN(C(C1(NC(C3(C4CC4)CC3)=O)CC1)=O)C2 C1(C(C)(C)C(=O)NC(=O)CC2CCN(c3nnco3)CC2)NC(=O)NC1=O c1(C(=O)NC2CN(C(C(C)(CO)OC)=O)CC23CC3)ccc(C)c(F)c1N C12(C(N3CC(CC(C)NC(c4cncnc4)=O)C3)=O)CC3CC(C(=O)N1)C2C3 CC(C)(C)C(CO)C(=O)NCC1C(O)C(O)CN1C(c1ncncc1Cl)=O C1(C#N)(C(=O)OC)CCN(C(CC(C(F)(F)F)N2CCOCC2)=O)C1 N1(C(C(C)CC(F)F)=O)CCC2(NC(c3ncoc3-c3cccs3)=O)CCCC12 c1(CC(=O)NCCC2CSCCN2C(=O)CN2CC=CC2)ccc(Cl)c(F)c1F C1(C(=O)OCCC(=O)NC)(CNC(=O)C(C)(C)C)CCCC1O C1(C(N2CC(N(C(=O)COc3ccon3)C)C(O)C2)=O)CCC(C2CC2)CC1 c1(NCCNC(=O)NCC2CCC(CCC)CC2)cc(C)cc(C)n1 C(=O)(CCC1=CCCCC1)NC1CN(C(c2cc(C)n(C)c2C)=O)CC1(C)C c1(CCCNC(C(=O)NCC#C)=O)ccc(C)c(C)c1 N1(C(c2cc(SC)oc2C)=O)CC(NC(=O)C=C2CCC2)CCC1C C1(CNC(C(C)P(C)(C)=O)=O)CC12CCN(C(C1(CN(C)C)CC1)=O)CC2 C=CCC(CC)C(=O)NCc1ccnc(C(=O)NCC2CCCC(C)O2)c1 N1(C(C(C(C)(C)O)F)=O)CCN(C(c2coc3c2COC3)=O)C2CCCC12 N1(C(C(CC)OC)=O)CCC(CC(C)NC(c2cnns2)=O)CC1 Cc1ccc(SCC(=O)NC2CC(N(C)C(c3ccncc3N)=O)C2)cc1 N1(C(CCC=C)=O)CCCC(CNC(=O)Cc2conc2C)CC1 N1(C(CC2CCC(NC(c3c(NC)nccc3)=O)C2)=O)C2CCCC1COC2 c1(CC)nc(C)sc1C(=O)NC1CCC(NC(=O)Nc2sncc2C#N)C1 N1(C(=O)NC(c2nc(CC)[nH]n2)CC)C(CC)CCC1(C)C1CC1 N1(C(N2C(OC(c3onc(CC)n3)=O)CCCC2)=O)CC2(CC)CC1(COC)C2 c1(C(=O)NC(CC)(C)CNC(=O)C(C)Cc2cnc[nH]2)cc(O)n(C)n1 C1(C(N2C(CCN(C(Cc3cnc(C)[nH]3)=O)C)CCCC2)=O)CCCC(C#N)C1 CC1CC=C(C(=O)N2CC3=C(C2)CN(C(C2(CO)CCOCC2)=O)C3)CC1 Cc1cc(=O)n(CCC(N2CCOC(CNC(C3C(C)C3C)=O)C2)=O)cn1 C1(NC(c2n[nH]cc2C2CC2)=O)CCCN(C(=O)Cc2csc(Br)n2)C1 N1(C(C(C)NC(=O)C(O)CC(F)(F)F)=O)CCC2(CCCC2)CC1 c1(N(CC#C)CC2CCCO2)nnc(-c2ccc(O)nc2)n1CC(C)(C)OC N1(C(c2cc(C)[nH]c2C)=O)CC(CNC(=O)CCC2CNC(=O)N2)CC1(C)C N1(CC(=O)NC(CCSC)=O)C(=O)CNC1=O.C1CNCCO1.C1CO1 C(=O)(CCCCC(N)=O)N1CC(COC)(NC(=O)Cc2cc(C)no2)C1 C1(CC)(CNC(=O)C(c2ccco2)NC(=O)Cc2cccc(O)c2)CCC(=O)N1 c1(C(=O)OC(C)C)ccc(S(=O)(=O)N2CC3(CCCN3C(=O)C(C)CN)C2)cc1 Cc1c(Cl)ccnc1CNC(=O)CCC1CCCN1C(=O)C(C(C)C)NC=O CC1CCc2nc(Cl)nc(NC(C3CCN(C(C45CCC(CC4)C5)=O)C3)C)c2C1 N(C(=NCCCCl)N1CCN(Cc2cccs2)CC1)CC1CCS(=O)(=O)C1 CC#CCCCC(=O)N1CCC(C(N2CCOC(C3CC3)C2)=O)O1 c1(SCc2cccc(O)c2)nc(C(F)(F)F)n2ccncc12 C(N=c1[nH]c(=NCC2(Cl)CC2(F)F)c2[nH]ccc2[nH]1)c1cc(C)oc1C C(=O)(C1=CCCN(S(=O)(=O)C2CC2)C1)N(C)C(C1CCCN(CC(F)F)C1)=O C1(C(=O)OC)CCC(C(=O)Nc2nc(C)c(C(=O)NC(C)C=CC3CC3)o2)CC1 Cc1cc(F)ncc1-c1cn(CC2C=CCN2C(=O)Cc2c[nH]c(Br)c2)nn1 c1(C(CC)NC(N(C(C#C)C)C2CC2)=O)ccc(Cl)cc1Cl c1(-c2cc(OCC)cc(C)c2)ccc2c(C(=O)NC(=O)C(C)(C)Br)n[nH]c2c1 C(CC(C)C)(C(=O)C(C(C)NN(C(C)(C)C)C)=O)N(C(C(C=C)C)=O)C C1(F)(CNC(COCC#C)=O)CC(NC(=O)Cc2ccsc2)C1 C(CC(C)(C)C)(C(=O)N1CCC(C)(C)C1C(=O)NCCCc1cncnc1)OC n1(C(C(=O)N(CC(=C)C)CC)C)cc(C(O)C(C)(C)C)nn1 CCC(C(=O)NCC(C)(C1CCC1)NC(=O)CC(=O)Nc1cccnc1)C(C)C C1(NC(CCN(CC=C)C(c2cccc(C)c2)=O)=O)CCCCC1OC c1(OC)ccc(OC)c(C(N2CCC(F)(CNC(=O)CNS(=O)(=O)C3CC3)C2)=O)n1 C1(C(=O)NCC(CC)NC(c2c(Cl)ccc(C)c2N)=O)CCC([N+](=O)[O-])CC1 C1(C(=O)NCC(C)(O)CO)(COC)C=CCN1C(c1csnc1Cl)=O c1(C(=O)NC(C(C(C)C)NC(C=C(C)c2ccco2)=O)C)ccc(C)cc1Cl c1(OC)cc(C(N2CC(NC(c3cc(N)ccc3C)=O)C(C)C2)=O)ccc1Br N#CC1CCCN(C(c2ccc(-c3ccccc3)[nH]2)=O)C1 CC1(C)CCN(C(=O)COCC2CCC2)C1CNC(c1cc(O)nc(C)c1N)=O C1(CNC(C=CC=CC)=O)CN(C(=O)Cc2conc2C)CC1O C1(NC(=O)CC2CC2(Cl)Cl)C(CNC(C2(C(F)(F)F)CC2)=O)CCC12CCC2 C1(CC=C)(NC(C(CO)OC)=O)CCN(C(=O)CCc2ccc(C)o2)C1 N1(C(C2C(CC)C2)=O)CC2CCCC2(CNc2ncc(C)c(O)n2)C1 N1(C(CCN(C(CCCOCC=C)=O)C)=O)CCOCC1CC1CC1 c1(C(=O)NCC2C(C)CCN(C(=O)C#CC3CC3)C2)cc(O)c2ccoc2c1 c1(NC2C(CC)CN(C(c3ccc(OC)cn3)=O)CC2)nc(C)nc2[nH]ccc12 C(=O)(C(CNC(=O)CC1CCC(C)(C)O1)C(C)C)NCCCC=C N1(C(c2ncn(C)c2)=O)CCC(CO)(CNC(c2cc(C(N)=O)c[nH]2)=O)CC1 CCCCCCC(CC)C(=O)N1CCCC1CN(C(=O)C=Cc1nccs1)CC c1(CC(N2C(CCCNC(C(CC)(C)F)=O)CCC2)=O)nn(C)cc1[N+](=O)[O-] C12CCC(CC1)n1cc(nn1)C2.C1(C)(CC)CC(NC(C2CCCCO2)=O)C1 c1(CN2CCN(C(C3CNCCO3)=O)CC2)cc(F)cc(I)c1 c1(OC)ccc(C(=O)NCC(F)CNC(C2CCCN(C(C)=O)C2)=O)cc1N CCC(CNC(=O)C(F)CC(C)(C)C)(CC)C(=O)Nc1cn(CCF)nc1C C1(NC(c2cc(COC)no2)=O)CCN(C(c2cc(Cl)cn2C)=O)C1C CCCCC(CC)C(=O)NCCC(CC)(CC)NC(c1cnc2[nH]cnc2c1)=O C=CCC(CNC(c1ccc(O)nc1)=O)C(=O)N(CCCO)CC NS(=O)(=O)CC(=O)NC(=O)C(CNc1ccccc1)NS(C)(=O)=O.N12CC(C1)C2=O C(=O)(N=c1cc(C2CC2)[nH][nH]1)c1cc(C(N2CC3C(C2)C3(F)F)=O)c(I)cc1 CCC(C)C(O)C(C)C(=O)N(C)CCOCCCNC(=O)CC1CC1C(F)(F)F c1(C(=O)NCC2CCC(NC(c3c(CCC)n(C)nc3)=O)C2)cccc(C)c1O CC1CN2CCN1CC2C(N1CCN(C(=O)C(Cl)=CCl)C(c2ncc[nH]2)C1)=O C1(C#C)(NC(C2N(C(c3cncc(C#C)c3)=O)CC2)=O)CCC(C)(C)C1 N1(C(c2nnc(CC)s2)=O)CC(CNC(=O)CCNc2cccnc2)CC1C N1(C(c2ccn(C)n2)=O)CC2CCC(C1)C2CC(=O)Nc1cnc(Br)c(F)c1 C1(NC(CC(CC)(F)F)=O)COC2(C1)CN(C(c1cncc(C#N)c1)=O)C2 CCC(C)CC(=O)C(=O)NC1CN(C(=O)Cc2cnsc2)CC12CCC2 N1(C(Cc2ncc(C)[nH]2)=O)C2CCCC1CC(NC(C1CCCCO1)=O)C2 c1(NC(C(CC(=C)Cl)NC(c2cc(C3CC3)[nH]n2)=O)=O)cccc2c1CCC2 C(CC(=O)NC1CN(C(c2c(C)cc(C)cc2C)=O)CC12CC2)(C(F)(F)F)OC C(=O)(CC1C(=O)Nc2ccccc21)NCC1CN(C(C2CC2F)=O)CC(C)(C)O1 OCC(CN=c1[nH]c(=NCc2nccn2C2CC2)[nH]c2c1CCC2)C1CC1 c1(-n2cc(C(C)NC(c3ccccc3Cl)=O)nn2)cccc(S(N)(=O)=O)c1 c1(OC2CN(C(N(C(C)C)C)=O)C2)cc(F)c([N+](=O)[O-])cc1F C1(NC(N2CCN(C)CC2)=O)CCCN1N1CCc2ncsc2C1 CC1CN(C(=O)CC2C=CCCC2)CCCN1C(=O)C=CSn1ncnn1 C=C=CCCC(=O)NCCC(CNC(C1(C(N)=O)CCC1)=O)OC c1(COC)ccccc1C(=O)NCC1CN(C(=O)CC2CCS(=O)(=O)C2)CC1C c1(CNC(c2ccn(CCC)n2)=O)cccc2c1CCN(C(=O)C1CC1)C2.C1CC1 N1(C(C2CCC(NC(C(CCC)=CCC)=O)C2)=O)CC(N(C)C)C2(CC2)C1 Cc1ccc(C(N2CC(NC(=O)C(F)CC)C(O)C2)=O)cc1N Cc1cc(C(=O)NCc2cccc(C(=O)NCc3ccnc(Cl)c3)c2)ccc1Cl N1(C(COCCOCC)=O)CC2CC1(CNC(=O)Cc1nocc1C(C)C)C2 c1(CC(C(N2CCc3nocc3C2)=O)NC(CC(C)(F)F)=O)cccc2ccoc12 n1(CC(=O)NC2CN(C(C(C(C)C)n3ccnc3)=O)C2)cc(Br)ccc1=O CC1CCN(C(C2CCOC2(C)C)=O)C(C(=O)NC2CC(CC(C)(C)C)C2)C1 C1(NC(CCOCCOC)=O)CCN(C(=O)CSC(F)(F)F)CC1F CCC(CC)C(C)C(=O)NC1CCCC1(C)NC(=O)C(C)(C)CCCF CC(CC(=O)NCCC1CC2CCC1O2)C(C)(C)NC(C1(C)CC(F)(F)C1)=O C1(C)(NC(C(C)=CCC)=O)CCCCC1C(=O)N(C1CC1)C1CC1 c1(C(=O)NCC(C2CCN(C(=O)C3=CCC3)CC2)C)cc(Cl)cc(F)c1F C=CCC(CC1CCCC1)C(=O)N1CCCC(CO)(NC(C2CC2F)=O)C1 N1(C(CC2(CC)CCC2)=O)CCN(C(=O)C(C)CC(OC)OC)C(CO)C1 c1(C(=O)NCC2(F)CC(CNC(CC3C(C)CCO3)=O)C2)nc(Cl)ccc1N C1(C(=O)NCCC2CC2)(CNC(CN)=O)CC1C.c1(C)cscn1.C(=O)NC c1(C(=O)NC2C(COC(C)C)OCC2)cc(C2CC2)cs1 CC(CN(C)C)N=c1[nH]c(=NCc2ccc(Cl)nc2OC(F)F)c2cc(Cl)ccc2[nH]1 C12(NC(c3occ(C)c3)=O)CCCCCC1N(C(=O)C(O)C1CC1)CC2 N1(C(c2cccc(C#C)c2)=O)CC(C)(C)C(N=c2[nH]nc(CC)o2)C1 c1(C(N(C(CN(C(CCC(CC)OC)=O)C)O)C)=O)cccc2ccnn12 Cc1c(C(=O)N(C)CC2CCCN2C(C2(C3CCC3)CC2)=O)nn(C)c1C1CC1 CCCC(C)C(=O)N1CCC(NC(=O)CCC(=O)c2cc(Cl)sc2Cl)(OC)C1 C(=O)(C(CNC(=O)CCCn1ccnc1)(CC)CC)N1CCC(OC)CC1 C1(C(=O)NC(CNC(c2cc(C)[nH]c2C)=O)C)CCc2nnc(C)n2C1 N1(C(CC2CC(=C)C2)=O)CCC(C2CCN(C(=O)Cc3cnc(C)[nH]3)C2)C1 N1(C(C2C(C)(C(F)F)C2)=O)CC(C2CCN(C(=O)Cc3cnc[nH]3)CC2)C1 CC(C)CC(CNC(C1(S(N)(=O)=O)CC1)=O)NC(C1CC(=O)CO1)=O c1(C(=O)NCC=CCNC(C2(F)CCC2)=O)cnc(-c2ccccn2)nc1 c1(OC)nc(C(=O)N(CCC(C(C)C)NC(=O)CC(C)SC)C)ncc1F c1(C(=O)NC(C)CCN(C)C(C2CC23CC3)=O)csc(C2CCCCC2)c1 c1(C(=O)NC(c2cnn(C)c2)C(=O)N(C)CCn2cccn2)cc(F)ccc1O C#CC1(F)CN(C(=O)C(O)C2CN(C(c3ccsc3Cl)=O)C2)C1 N1(C(Cc2ccn(CC(C)C)n2)=O)CC(NC(c2ccnnc2Cl)=O)C(C)C1 N1(C(C2CC(CCC)C2)=O)CC2CC(N(C(=O)COC3CCCCCC3)C)C1C2 CCCC(C)(CC)C(=O)NCC1CN(C(c2ncccc2OC)=O)CC12CC2 C1(NC(CCCCC)=O)CCCC(C(=O)NCC2CCSCC2)CC1 c1(CC)ccccc1CC(=O)NCC(CNC(=O)CCc1cnoc1)OC CC1CN(C(=O)CC(O)C2CCCC2)CCN1C(C1CN(C(=O)N(C)C)C1)=O c1(NC(CCC=C)c2nnnn2C2CCOC2)ccc(N2CCCC2=O)cc1 C1(C)(C(=O)NCCOC2CCN(C(CNC(=O)OC)=O)C2)CCCCO1 C=CC1(CC(N2CC(O)(COC)C2)=O)CN(C(=O)Oc2cc(C)on2)C1 C1(C(=O)NCCN(CC(C)O)C(c2cnn(C3CCC3)c2)=O)C=CCCC1 c1(CCC)nc(C(=O)NC(C)C=CC(=O)N(C)CC)co1 C=CC1(C(=O)NCCOCCCNC(=O)CC2CCC(C)O2)CCC1 CCC(CCCC(=O)NCC(Cl)Cl)NC(=O)C(O)C(C)(C)CC c1(NC(C2CN(C(c3cnc(O)cc3O)=O)C2)=O)nccn2ccnc12 c1(C2(C(N(CC(C)N(C(=O)CNS(C)(=O)=O)C)C)=O)CC2)cc(Br)ccn1 N1(C(C=CC(C)(C)C)=O)CCC(n2cc(CO)nn2)C1.N12CCC1C2=O c1(C(=O)NCCC(CNC(c2occ(C)c2)=O)O)cc2[nH]ccc2s1 C1(=CC(=O)NC2CC(NC(C3CC4(CCC4)CO3)=O)C2)C2CC3CC(C2)CC1C3 c1(C(N2CCC(N(C(C3CC=C(C)CC3)=O)CC)C2)=O)nc2c(s1)COCC2 N1(C(c2cccc(CCC)c2)=O)CCC(NC(C2CC3(C2)CC3F)=O)C(C)(C)C1 C1(CNC(C(CC=C)(C)C)=O)COC(C)(C)CN1C(c1cnn(C)c1SC)=O C1(CNC(C2(OC)CCC2)=O)CCCN1C(c1cc(C)[nH]n1)=O Cc1ccc(C(N2CCCC2c2nc(C(=O)Nc3[nH]cnc3C(N)=O)cs2)=O)n1C c1(CCC(=O)N(CCNC(Cn2ncc(C)c2)=O)CC2CC2)cccnc1F C1(C(=O)N(C(C)CNC(=O)CCc2ncccn2)C)(CC)CCCC1 C1(CC(=O)N(CCCCC)C)CC(NC(C2SCC=C2C)=O)C1(C)C N1(C(C23CC(C)C2C3)=O)CC2CC1CCC2NC(c1cc2occc2n1C)=O C1(NC(C2CCC(CC)O2)=O)CN(C(=O)C#CC2CCC2)C2(CCC2)C1 C1(CC(=O)NCC(CCC)NC(c2cc(CO)[nH]n2)=O)CCC=CCC1 N1(C(Cc2ccn(CC)n2)=O)CC2CN(C(=O)CC3CC3C(F)(F)F)CC2(C)C1 N1(C(C2(C)C=CCN2C(C2CCC3(CC3)C2)=O)=O)CCOC2COCC2C1 CCC(C(=O)N1CCCC(COC)(NC(c2cc(C)c(N)cn2)=O)C1)C(C)(C)CC c1(OC)cccc(C(=O)NC(C2CCN(C(C3CCCCCC3)=O)C2)C)c1Cl C1(C(N(c2ccsc2)CC)=O)CCCN(C(=O)CCOC(C)=O)C1 c1(CC(=O)N(CC(C)(C)NC(=O)CC2C=CCC2)C)sccc1Br C1CC(=O)NNC(=O)N1.CC1CN(c2ccccc2SC2CC2)CC(C)O1 C1(NC(c2ccc(C=C)cc2)=O)CC(C(=O)NC(CN(C)C)C(C)CC)=CC1O C(=O)(CCCCC(F)F)NC1CCCCN(C(c2c(C)cn(C)n2)=O)C1 Cc1ccccc1CC(N1CCCC(C(C)NC(=O)CSc2nc[nH]n2)C1)=O c1(C(N(CCCOCCN(C(C2C(=C)CC2)=O)C)C)=O)nscc1Br S(=O)(=O)(c1ccc(Br)c(F)c1F)N1Cc2c(N3CCC(C)C3)ncnc2CC1 N1(C(CNC(CNC(N)=O)=O)=O)CC2OCC(NC(=O)CC3(CO)COC3)C2C1 C1(C(N2CC(C(N3CCCOC(CC)C3)=O)(CC)C2)=O)OCC2CCCC12 C1(NC(c2cc(OC)n[nH]2)=O)CN(Cc2csc(-c3ccccc3)n2)CC1Cl N1(C(C(C2CC2)SC)=O)CCC(CNC(c2ccc(C)nc2C)=O)C12CC2 C(c1nc(NC(=O)C(C)CC2CCCCC2)cs1)=CC(C)=O Cc1cc(C(N2CC(NC(=O)CC3CCOC3=O)C(C)(C)C2)=O)cc(Br)c1 c1(CNC(=O)C(=O)NC(c2ccccc2)Cc2ccccc2Br)nc(Cl)sc1Cl C1(C(N2C(C)(CCO)CC2)=O)CCC2CCC1N2C(C1(O)CCCC1)=O c1(C(C)N(C)C)cccc(S(=O)(=O)NC(C2CCCCCC2NCCO)=O)c1 C(=O)(C(C)(O)C(C)C)N(CCCCN(C(CCNc1c(OC)cccc1)=O)C)C C(C(C(=O)NCCCc1ccc(Cl)cc1)N(CCC(C)C)C)(C1CCCC1)OC C1(CNC(=O)C(O)C2CC2)CC2(CCN(C(=O)C=Cc3ccccn3)C2)CO1 C1(CC(N)=O)(NC(c2cc(=O)cc[nH]2)=O)CCN(C(c2cnc(C3CC3)s2)=O)C1 C1(C(C)NC(c2c(OCC)scc2)=O)CCN(C(=O)CCc2cnc[nH]2)CC1.C(=O)O C12(C(=O)NN(C3CCN(CC)C3)C(CN(C(=O)OC)C)=O)CCCC(C)(C1)OC2 Cn1c(N2CCC(c3cccs3)CC2)nc(Cl)c1C#N C(=O)(C1=CNC2=NCCC2=C1)N1CC(OCCNC(c2c(C)cccn2)=O)C1 O=C(N=c1c(F)c[nH]cc1Cl)C1(C(c2ccccc2)=O)CCCCC1 N1(C(C=C(C)Cl)=O)CC(CNC(c2c[nH]cc2C)=O)C(C)C1 C(=O)(C(CO)C(C)(C)C)N1C2C(CNC(c3cc(SC)c(F)cc3)=O)C(CC2)C1 C(N=c1[nH]cnc2cc(F)c(F)cc12)C1(CNC(CN(C)C)=O)CC1 C1(CCNC(CC=CC)=O)CN(C(c2ccc(=N)[nH]c2)=O)CC1C N1(C(C2(C)CCOC2)=O)CCSCC1C(=O)NCC1(C2CCCCC2)CC1 N1(C(=O)Nc2cccc(F)c2)CCC2CN(C(c3ccc([N+](=O)[O-])o3)=O)CCC12 Cc1cccc2cc(C(=O)NC3CCN(c4ncncc4Cl)CC3F)[nH]c12 c1(C(=O)NCC2C(NC(CCCCC)=O)C2)c(F)cccc1[N+](=O)[O-] N1(C(N(C)C)=O)CCCC(C(=O)NCCCN(C(=O)C(C2(O)CCCC2)F)C)C1 C1(c2n[nH]c(=N)o2)CCN(c2cc(NCC3CCC(O)C3)ncn2)CC1 C(=O)(C1CC(=O)Nc2ncccc21)NCCNC(c1[nH]c2ccn(C)c2c1)=O c1(C(N2C(C(=O)NC(C#C)CC3CCC3)C(O)CC2)=O)ccc2c[nH]nc2c1 N1(Cc2onc(CC)n2)CCCC(C2CCCN(C(=O)CSC(C)C)C2)C1 c1(C(N(CC(C)(C)NC(C(C)NC(N)=O)=O)C2CC2)=O)n[nH]cc1F c1(OC)cncnc1C(N1CCC(NC(c2cccc(OC(F)F)c2)=O)C1C)=O N1(C(C2(C(=O)OC)CC2)=O)CCC(C)N(C(=O)Cn2cnc(C#N)n2)CC1 C1(F)(CN)CC(C(=O)NC(C)C(=O)NCCc2[nH]cnc2C)C1 C12(C(=O)NC3C4CN(C(C(CC)CC)=O)C3C4)CCCCC1C2(F)F C1(CNC(Cc2c(C)ccnc2)=O)C2CCC(C2)N1C(c1cnc(O)cc1O)=O c1(OC)ccc(O)c(C(=O)N(C2CN(C(=O)C(c3ccc(F)cc3)F)C2)C)c1 N1(C(C(C=C)O)=O)CCC2C(CCCN2C(c2c[nH]c3nc(Cl)ccc23)=O)C1 c1(CC)cc(C(N2CC3C(CO)C3C2)C(=O)NCCSC)n(C)n1 C(C1c2ccsc2CCN1C(c1ccc(C(C)(C)C)o1)=O)NC(C1C(C)C1)=O N1(C(C(C(C)C)SCC)=O)CC(CNC(=O)CCc2nc(C)c(C)o2)CCC1C c1(OC)cc(C(=O)N(C(c2ccccc2Cl)CO)C)nc(OC)n1 c1(OCC(=O)OC(CC#C)C)c[nH]cc1 CC(C)(CC(=O)N1CC(CCNC(C2(c3ccc(F)c(Cl)c3)CC2)=O)C1)C(F)F c1(CN2CCCC(C(N(CCCN(C)C)C)=O)C2)ccnc(F)c1Cl c1(C(N(CCNC(CC(CCC)(C)O)=O)CCOC)=O)cc2cccc(F)c2o1 C1(CN(C(C(CC)O)=O)CC)CCCN(C(=O)CCOC)C1 N1(CCNC(C2CC(NS(C)(=O)=O)C2)=O)CCN(C(C2CC(C)(C)O2)=O)CC1 N1(C(COCC)=O)CC2CCC(C1)N2C(=O)C(C1CCOCC1)C N(C(=NCCCF)NCc1ccco1)C.C1(SC)CCC(N)C1 C1(OC)CC(NC(=O)C(CC(C)C)NC(=O)OC)CN(C(=O)C(O)CC(N)=O)C1 N1(c2cc(OC)ncn2)CC2CCN(Cc3c(C)nn(C)c3C)C2C1 C12(C(N3C(C(C)(C)NC(C4CC4(F)F)=O)CCC3)=O)CCC(C1)OC2 c1(-c2ccnc(OC)c2F)ccc2c(C(N3CC(O)CC3CO)=O)coc2c1 C(N=c1[nH]c(=NCCC2CC2(Cl)Cl)[nH]c2c1CCCCC2)C1C(CO)CCCC1 N1(C(c2cc(OC)cc(COC)c2)=O)CCC2(CC1)CC2c1nnco1 Cc1cc(O)cc(=O)n1CC(=O)NCC1CCCN(C(=O)C(C)NC(C)(C)C)C1 Cc1ncnc(C(N2CCC(NC(c3[nH]nnc3C)=O)C2)=O)c1C CCCC(CCCNC(=O)C(C)CF)NC(C1CC(n2ccnn2)C1)=O N1(C(c2c(C)nsc2)=O)CCCC2(NC(=O)CSC3CCCCO3)CCCC12 N1(CCNC(c2c(OC)ccs2)=O)CCOCC1NC(=O)CC(C)(C)C1CC1 C(=O)(C=CS(C)(=O)=O)N(C1CCC(NC(c2cnncc2O)=O)CC1)C CC(C)C1=CCC(NC(c2cnn(C)c2)C)CC1 c1(C(C(=O)N)N(CC(C)C)C(C)C)cnc(OC)cc1C.C1(CC)COC1 N1(CC)CCc2cc(N(C)Cc3ccccc3-c3cnccc3C#N)ccc21 C1(C(=O)NCCN(C)CC2CC2)N(C(C2CCC(=O)O2)=O)CCC1(C)C c1(C(N(CC(C)N(C)C(C2CS(=O)(=O)C2)=O)C)=O)ncn2c1CCC2 C1(CNCc2n(CCOC)c(C)nn2)CCCC2(CNC2)O1 N1(C(c2scc(CNC(=O)C=CC3CCC3)c2)=O)CCOCC1CN(C)C c1(C(N2CCC(CNC(C(C)(C)C)=O)CC2)=O)cc(F)c(Br)cc1O Cc1c(C(=O)NCC(C2CCN(C(=O)CC(C)C3CC3)CC2)C)cncc1Cl CCS(=O)(=NC(=O)C1CC12CCN(C(c1ccc[nH]1)=O)C2)c1ccccc1 C1(COC)(NC(C2CC2c2cncn2C)=O)CCN(C(=O)C(F)C(F)(F)F)CC1 N1(C(C(CC(=O)OC)C)=O)C2CC=C(C(=O)N3CCC(F)(F)C3)C1CC2 C1(C(=O)NCC(C2CCC2)NC(c2ccc(CO)s2)=O)(COC)CCCO1 N1(C(CCCCCOC)=O)C2CCC1CC(NC(C13CCCCC1C3)=O)C2 CC1CN(C(c2ccc(C(C)(C)C)cc2)=O)CC1CNC(C1(C#N)CC1)=O N1(C(CC2CN(C)CC2O)=O)CC(NC(=O)Cc2cc[nH]n2)C(C)(C)C1 c1(C(N2CCC(C)(CNC(CCCOC(C)=O)=O)C2)=O)c(C)nn(CCO)c1C C1(NC(CC2(C(=O)NC)CCC2)=O)COCCN(C(C2(COC)CCOC2)=O)C1 CC1CCC=C1C(=O)N1CCC(C(C)(C)C(N2CC3CCC(C2)O3)=O)C1 c1(OC)cc(C(N2CCC(CN(C(=O)C(C)(C)C)C)C2)=O)nc(Br)c1 C(=O)(C1=CCCCC1C)NCCCCCCCn1cc(CC(=O)OCC)nn1 N1(C(C(COC(C)=O)C)=O)CCC(C)CC1C(=O)NCC1CCC(=O)NC1C C1(C(=O)NCC2N(C(C3CCCC(OC)C3)=O)CCCC2)CC2CC1CC2O c1(C(=O)NCCC2CCN(C(C(CC)OC)=O)CC2)cc(C)cc(O)n1 N1(C(c2n[nH]c3c2CCC3)=O)C2CCC1CC(n1cc(C3CC3CO)nn1)C2 c1(OC)cnc(Cl)[nH]c1=NCC1CCCC(NC(=O)Cn2ccc(C(F)F)n2)C1 C1(CCCC)CN(C(c2cc(Cl)no2)=O)CCN1C(=O)CC1CCC2CC12 C1(OC)C(NC(=O)NCc2cc(C#N)cn2C)COC12CCC2 c1(C(C)=O)c[nH]c(C(=O)NOC2CCC2)c1.N12C(CC1C)C2=O Cc1cc(NC(c2cn(C)nc2-c2ccco2)=O)ccc1NC(=O)C(F)C(C)C c12cc(cc(Br)c1)C(=O)NCC2.C1(NC)CCOC1C(c1nnnn1C)OC N1(C(CCN(CCC)C)=O)CC2CCC1CN2C(C12COC(CC)(C1)C2)=O C1(CN(C(c2cn(CCC)nc2)=O)C)CC(F)CN1C(=O)Cc1c(C)noc1Cl CCC(O)C(C)C(=O)NCc1cccc(CNC(c2cc(C)no2)=O)c1 c1(C(C)NC(c2n(CC=C)nnn2)c2csc(C(C)(C)C)c2)c(Cl)cccc1Cl c1(CC2(C(N(C)C)=O)CC2)ccccc1.C(C)(C(=O)NC1(CC(=O)N)CCC1)SC N1(C(C2(CO)CCCO2)=O)CCCCCCN(C(C23CCC(CC2)C3)=O)C1 CCCC(C)CCCC(=O)NCC1CCCN(C(=O)Cc2ccc(C)s2)C1 c1(C(N(C)CC2CCN(C(C3(CC)CC3(F)F)=O)C2)=O)onc2ccccc12 C(=O)(C1=COCCO1)NCCC1N(C(c2cn(CCC=C)nn2)=O)CCCC1 c1(NC(C(CC2CN(C(C(CC=C)C)=O)C2)F)=O)cc(CC2CC2)cc(F)c1 CN1CCN(C(=O)CC2CC2(C)C)CC1C(N1CCCNC(=O)C1)=O CC1CN2CCN1CC2C(=O)N(C)CCOCCNC(=O)C(O)c1ccco1 C1(C(=O)NC(C=C)COC)CCCN1NC(=O)C(O)CSC C1(C(=O)NC(C(C)C)CNC(c2cscc2Cl)=O)CCc2n[nH]cc2C1 C12(CNC(COCC=C)=O)CCCC1N(C(=O)CCC1CCCC(=O)N1)CCC2 Cc1cnc(C(=O)NCC2CC2NC(=O)CCCn2c(C)csc2=O)cn1 C1(C(=O)NCC(CC)NC(C(CC)CC)=O)COCC2(CCC2)O1 C1(C(N2CCC(O)(CCNC(CC(C)(F)F)=O)CC2)=O)C2Cc3ccccc3C12 c1(OCC)ncc(C(=O)NCC=C2CN(C(=O)CCNC(=O)C=CCl)C2)cc1Cl C1(OCC(=O)NC2CCC(n3cccc3)CC2)CCCC(C(=O)O)C1 C(=O)(C(CN(C)C)NC(C1OCCC1C)=O)NCC1(CC)CC1 CC1CCCC(c2nnnn2CCOC2CC2)(NC2CCCC(C3CC3)CC2)C1 CC1=C(C)CC(C)(C(=O)N(C(C)CCNC(=O)C#CC2CCCC2)C)CC1 C1(NC(C2(SC)CC2)=O)COC2(CCN(C(=O)CCc3ccc(F)cc3)C2)C1 c1(CNC(c2nc(C(C)NC(=O)C(C)(C)C#N)oc2)=O)ccc(C)c(Cl)c1 C1(NC(C2C(C)CC3CC3C2)=O)CC2CN(CCCOCC(F)(F)F)CC2C1 N1(C(c2c(C)ncc(N)c2)=O)CCN(C(=O)C(C)Cc2cnc[nH]2)CC(C)(F)C1 N1(C(c2cnn(C(C)C)c2Br)=O)CC2CC1CC2NC(=O)Cc1ccco1 N1(C(c2c(CC)scn2)=O)CC(CN(C(=O)Cn2nc(C)cc2C)C2CC2)CCC1C N(C1c2ccccc2CC1NC(C1(C)CCCCCC1)=O)C(C#CC1(C)CC1)=O N1(C(c2ccncc2)=O)CCC2CCN(C(c3ccc(C(F)F)cc3)=O)C2C1 Cc1cc(F)c(C(N2CCCC(NC(=O)CO)CC2)=O)c(F)c1 C(CC(C)(C)C(c1nnnn1C(C)(C)C)NC(c1ccccc1)CSC)OC Cc1ccc(C(=O)NCC23CC2CN(C(C2CC(C#N)C2)=O)C3)c(=O)n1C c1(C(CNC(c2cnn[nH]2)=O)NC(COCCOC)=O)cccnc1 C1(NC(C(C(C)C)NC(C)=O)=O)CCCCCC1NC(=O)C#CC1CC1 C#Cc1ccc(C(N2CC(NC(=O)CCc3nnc(S)nc3O)C3CC23)=O)cn1 C=CC1(C(N2CCNC(=O)C2C)=O)CCN(C(=O)CCc2ccn(C)n2)CC1 N1(C(C(Cc2c(C)cccc2)C)=O)CC2(CCCN(C(C3CCCCO3)=O)C2)C1 c1(CC(=O)NC(CCCC)CNC(=O)Cc2csnn2)ccc(C#N)nc1 CC1CN(C(=O)COc2ccc(OC3CC3(F)F)cc2)CC1C(=O)NCCF C1(C(N2CC(O)(C(C)NC(c3cc(COC)sc3)=O)C2)=O)CCN(OC)CC1 N1(C(C(CC)CC)=O)CC(C(=O)Nc2csnc2OC)CC1(C)C CC1CC(N=c2ccc(Br)c(S(=O)(=O)N3CCC(CF)CC3)[nH]2)CC(C)(C)C1 c1(N2CCC(CNC(C3CC34CCOCC4)=O)CC2)cc2nncn2cn1 N1(C(CC)=O)CCC2(CC1)CN(C(c1cc(O)c(F)cc1N)=O)CC(C)O2 C1(C(=O)NCC2(CC)N(C(COCCCC)=O)CCC2)CCn2nncc2C1 CC(C)(CC1CCOC1)C(=O)N1CCN(CCNC(C2(O)CCSC2)=O)CC1 C(=O)(C1=CS(=O)CCC1)NC(C1CCCCC1)CNC(c1c(OC)c(C)cs1)=O C1(N(C(=O)Cc2cccc(O)c2)C)CCC2CN(C(=O)CC3CCCN3C)CC12 C(C(=O)NC(C1(O)CCCC1)C)(C(C)CC)N(C(C=C(CCC)C)=O)C N1(C(=O)OC(C)(C)C)CCC(CCC(CC)NC(=O)C(=O)Nc2ncc[nH]2)CC1 c1(OC)cc(C(=O)NCC2CN(C(c3ccc(Cl)cn3)=O)C2)c(O)c(Cl)c1 C1(CCC(=O)NC(c2ccccc2)CNC(CN(C)CC)=O)CCCN1C C1(CCNC(CN(CC)CC)=O)CCCN1C(=O)CC1(C)CCOC1 N1(C(CNC(CC)=O)=O)CC(C(F)(F)F)CC1C(=O)N(CC(F)F)C c1(C(=O)NC(c2cn(-c3ncccc3F)nn2)CCC)ccc(Br)c(Cl)c1C N1(C(C(C)NC(CC)=O)=O)CCCC2(C1)CN(C(C1CC(=O)N(O)C1)=O)C2 C1(C)(NC(CCN(C(c2ccc(C=C)cc2)=O)C(C)C)=O)CCC(C)(C)CC1 N1(C(C2(NC(C3CCNC3=O)=O)CCC2)=O)CCCC(CCCO)C1 C(=O)(C1OCCn2ccnc21)NCCC1(CNC(c2nccc(C)n2)=O)CC1 C=CC1CN(C(c2n[nH]cc2C)=O)CC1NC(=O)C(C)(F)c1ccon1 CC(C)CC(C(=O)NCC1(O)CCCOC1)N(C)C(c1cnn(C)c1)=O C1(NC(CCC=C)=O)CC2CCC(C1C)N2C(=O)C(C)CNCCCC CC1(C)CC(O)CN(C(C2(CNC(c3n[nH]c(O)n3)=O)CC2)=O)C1 C1(NC(C(C)=C(C)C)=O)CC2CN(C(c3cc(C(C)C)n(C)n3)=O)CCN2C1=O C1(n2cc(-c3c(CC)c(C)no3)nn2)CCCN(C(=O)CN(C)C(C)=O)CC1 N1(C(C(CC)(F)F)=O)CC(NC(c2cnc(C(C)(C)C)[nH]2)=O)C(C)(C)C1 CC(CCCCNC(C1CCCNC1=O)=O)NC(C1(n2cccn2)CCC1)=O c1(C(N2CCCC(C)(NC(c3cc(C)sc3)=O)C2)=O)oc2c(Cl)cccc2c1C c1(OC(C)C(=O)NCC2(CNC(C3CCC(=O)O3)=O)CCOC2)ccccn1 C1(NC(c2ccc(C(=O)OC)[nH]2)=O)CN(C(C2CCC=CO2)=O)CC1(C)C N1(C(c2cc(C(=O)OC)sc2C)=O)CCOCC(C(=O)NC2(C3CCC3)CC2)C1 C1(C(=O)NC2CCC(Cn3cc(CN(CC(C)(C)C)C)nn3)C2)CCC2CC2C1 C1(C)(C(=O)NCC2(CCNC(c3c(C)n(C(C)C)cc3)=O)CC2)CCNC(=O)N1 N1(C(c2cc(SC)n(C)n2)=O)CCCCC(Cn2cc(CCOC(=N)O)nn2)C1 n1(CC)[nH]nnc1=NCC=CCNC(=O)Cc1cc(OC)no1 N1(C(c2ccc(CNC(Cc3c(C)cco3)=O)o2)=O)CCC2(CCO2)C1 C1(C(=O)NC2COCC(C)(C)C2)CN(C(=O)CC2CCC(=O)NC2)C2(CCC2)C1 C1(C)(C(=O)NCCC(C)CCNC(=O)CCc2ccc[nH]2)CCC(C)CC1 c1(C(=O)NC2CCCNCC2F)ccc([N+](=O)[O-])cc1Cl C1(C2N(CCNC(C3CCCC3N3CCOCC3)=O)CCC2)CCC(F)(F)CC1 c12cc3cccc(c3[nH]1)C2=O.N1(C(C(C)N(CC)CC)=O)CCOCC(NC)C1 Cc1cc(CN2C(=O)CN(CC(N3CCOCC3)C(C)C)C2=O)c(C)c(C)c1O C(CC(C)(C)C(=O)N1CCC(C(F)(F)F)C(NC(C2(C)CC=CC2)=O)C1)OC CCC(C)C(O)C(C)C(=O)NC(c1nocc1C(N1CC(C)(CCO)C1)=O)C C1(C(N2CCC(CCNC(=O)CCF)C2)=O)CCCN1CCC(F)(F)F c1(CNC2CCC(CC(=O)OC)C2)cccc2c(C)csc12 C(=O)(C(C#N)C(C)C)NC1(CF)CCN(C(CCCOCC=C)=O)C1 C=CCCC(C(=O)NNc1cccc(NC2CCCC2)c1)c1ccccc1 C(=O)(C1=CCCCC1C)NCC1C(CNC(C2(CC=C)CCC2)=O)C1 C(=O)(CCC(=O)N1CCC(CNC(C2COC(=O)N2)=O)(OC)C1)NC C12CCN(CC1C)C(=O)N2.CC1CCC(c2cn(C3C4CC5C(C4)C35)nn2)OC1 C1(C(C)(C)C)CCCC(N=c2[nH]c3c(c(=NCCC4CCCC5CC45)[nH]2)CSC3)C1 c1(C(=O)NCCC2C(C)CCCN2C(=O)CCC2(C)CC2)c(F)ccc(N)c1F C(c1cccc([N+](=O)[O-])c1)=CC(=O)NCCNC(C1(c2ccncc2)CC1)=O C1(C(C)C)CCC(C)CC1OC(=O)C(C1CCC1)SC1CCCC1 C1(C(=O)NCC2CCN(C(C3C(CSC(C)(C)C)CC3)=O)C2)CC12CC(O)C2 C1(C(N2CCCCC2)C(C)C)CCN(c2cccc(C(=O)NC(C)(C)C)n2)CC1 C(=O)(C1=CCCCC1)N1CCC(N2CCC(NC(=O)C(F)n3ccnc3)CC2)C1 C1(C(=O)OC(C)(C)C)COc2ccccc2N(S(=O)(=O)c2cc(C#N)ccc2Cl)C1 C1(NC(C2N(CC(C)C)CCC2)=O)CCCN(C(=O)CSC(F)(F)F)CC1 c1(C(N2CC3CCN(C(CCCCC=C)=O)C3C2)=O)cn2cc(C)ccc2n1 N1(C(C=NOC)=O)CCC2(CCN(C(=O)C(C)n3cccc3)CC2)C(C)C1 c1(C(=O)NC2C(CNC(CCSC)=O)C2)sc2ccccc2c1Br c1(CC)nc(C)[nH]c(=NCC2CCN(C(C3(C(=O)N(C)C)CC3)=O)C2)n1 c1(C(C)=O)ccc(C(=O)NC(C)(C)C(=O)NCC(C)NC(c2nnc(C)s2)=O)[nH]1 Cc1cc(C(N2CCCC(NC(=O)C(C#N)C(C)C)C2C)=O)cc(F)c1 C(CCC(C)(C)c1cn(C2(CC(=O)N(C)CCF)CCOC2)nn1)OC c1(C(N2C(CNC(=O)CCSC3CCCC3)COCC2)=O)cc(O)nc(Cl)c1 C1(F)(CNC(C(CSC)C)=O)CCCN(C(=O)CCNc2ccccn2)CC1 c1(C(=O)NCC(CNC(C(C(=O)NC)(C)C)=O)O)cccc(C=C(F)F)c1 Cc1nc(C(=O)NCCN(C(=O)CC2(O)CCCC2)Cc2ccccc2)co1 C(=O)(N=c1cc(CS(c2ccccc2)(=O)=O)o[nH]1)c1cncc(C#C)c1 c1(C(C2C(C(=O)NC)C2)=O)cnn(CC(F)F)c1.O=C1CSC2(CC2)N1.C1CC1 Cc1cc(CC(=O)NC2CN(C(=O)CCCC(N)=O)CC23CC3)ccc1Cl N1(C(C=CSC)=O)CC2CCCC(C1)N2C1CCN(c2ncc(Br)cn2)CC1 N1(C(c2n(CC)cnc2)=O)CCC(CNC(C2CC3CCC3C2)=O)C(F)(F)CC1 S(=O)(=O)(c1nc(N2CCC(C(C)(C)C)C2)ccc1Br)NC(CC)(C)COC n1(CC)ncc(C(N2CCC(CNC(C3(CF)CC3(F)F)=O)C2)=O)c1C C(=O)(CCCS(C)(=O)=O)NCC(c1cccc(Cl)c1)NC(CCCOC(C)C)=O c1(C(=O)NC2CCCN(C(C3C(CCOC)C3)=O)CC2)c(N)cc(Cl)cc1F c1(CN(C(C(=O)NC)C(C2CCCCC2)OC)CC(C)C)c(C)cc(C)cc1C Cc1cnc2cc(C(N3CCN(C(c4cc(F)ccc4Cl)=O)C(C)C3)=O)ccn12 c1(CNCC(N2C(=O)OCC2)c2ccccc2)cccc2cc(O)ncc12 C1(CCC(=O)Nc2snc(OC)n2)CN(C(C)=O)CC1C C1(NC(C(C(=C)C)(C)O)=O)COc2ccccc2C1 CC(CNC(c1c[nH][nH]c1=N)=O)CC(=O)NCC1CC(=O)N(C)C1 CC1(C(=O)NCCCC2CCN(C(C3CCC4CC34)=O)CC2)CCCOC1 N1(C(C(c2cccc(C#N)c2)C)=O)CCN(C(=O)Cc2ccccc2Cl)C(CO)C1 c1(C(N(CCN(C(=O)C=CSc2ccccc2)C)C)=O)ccc2cnn(C)c2c1 C1(C)(C(=O)NC2(CCNC(c3cn(CC(C)(C)C)nn3)=O)CCC2)CCC(=O)N1 C(=O)(C(CC(C)CC)NC(=O)C(C)COC)N(CCC#C)C c1(CC)ncc(C(=O)NCC(O)CCNC(=O)CC2CS(=O)(=O)C2)[nH]1 O=C1NC2(CC2CN=c2nc(-c3cccs3)o[nH]2)C(=O)c2ccccc2NC1=O Cc1ccc(Cl)c(O)c1C(N1CCC(N(C(=O)C(C)C2CCCC2)C)CC1)=O c1(C(=O)NCC2N(C(CC3CN(C(C)=O)C3)=O)CCC2(C)C)cc2cccn2cn1 N1(C(c2nccc(C)n2)=O)CC2CCCC1(CNC(C1CCC(C)(C)C1)=O)C2 C1(C(N(CCN(CC(F)F)C)C(C)C)=O)CC2(C1)CN(Cc1c[nH]c(C#N)c1)C2 c1(-n2c(C)ccn2)cccc(NC(c2nnnn2CC(F)F)C2CCCO2)c1 N1(C(c2cc(COC)sc2)=O)CC(CNC(c2cccc(OC)n2)=O)C(C)(C)C1 C12(CNC(CN(C)CC)=O)CC(NC(C3CCC(C)(F)CC3)=O)(C1)C(C)O2 C1(CNC(C(C)N(C(C)=O)C)=O)CN(C(=O)CC(C)(C2CCC2)N(C)C)CC1O C1(NC(c2ccc(Cl)[nH]2)=O)(CNC(c2ccnc(OC(F)F)c2)=O)CC2CCC1C2 c1(C(=O)NCCCNC(c2c(C)cc(C)nc2O)=O)c2n(c(=O)n1C)CCCC2 c1(C(N2CCC(N(C(c3cc(OC)no3)=O)C(C)C)C2)=O)cc(CC2CC2)n(C)n1 c1(OC)ccc(C(=O)NCCCCCNC(C2CC(C)(C)CO2)=O)cn1 c1(CC(N2CCC(CN(C(=O)C(F)(F)CC3CCCO3)C)C2)=O)sccc1C#N C(CC(=O)N1CCC1C1CC1)OCCN(C(=O)Cn1cccc1)C S(=O)(=O)(c1cnn2ccc(=NCC3CC=CCC3)[nH]c12)NCC(C1CC1)SC C1(NC(C(c2cccnc2)C)=O)CCCC2CN(C(c3ccc(=N)[nH]c3)=O)CC12 c1(C(=O)NC2CCC(C(N3CC(C=C)C3)=O)C2)nnn(C)c1C c1(C(N2CC3C(NC(C(CC(C)C)O)=O)C(C3)C2)=O)nc[nH]c2ncnc1-2 N1(C(CC(OCC)OC)=O)CCCC(CC(N2CCC(CC)C2)=O)CC1 c1(OC)cc(F)cc(S(=O)(=O)N(C)Cc2ccc(C)c(OC)c2)c1 CC(N=c1[nH]c(N2CCC(C#N)CC2)nc2ncn(C)c12)C1CC2(CCC2)C1 c1(C(N2CCCC3(NC(CC(C)OC)=O)C(C2)C3)=O)cccc2oc(C)cc12 C1(NC(C2C(CC(C)C)C2)=O)CC2C1CCN2C(c1cc(N)ccc1F)=O C12(NC(c3cc(C)[nH]n3)=O)CCCC1N(C(c1ncncc1Cl)=O)CCC2 n1(CC)ccnc1C(c1nnnn1C1CCOC1)NCc1scnc1Cl O=C(C=C1CNCC1)NN1CCCC1C(C1CCOCC1)OC.CCO N1(C(CC(C)CN(C)C)=O)CC(NC(=O)C=CCn2cncn2)CC(F)C1 C12(C(N3CC(NC(C4OC5CCC4CC5)=O)C3)=O)CCC(=O)N1CCS2 C#CCCC(O)C(=O)NCCN(CCC)C(C)=O.c12cc(F)ccc1NC2=O C(=O)C1SCCc2sccc21.C1(C(=O)O)CCC2C1C2(F)F c1(C(=O)NC(C(=O)NC(CC)CCOC)CN(C)C)cc(C)c(O)nn1 c1(C(=O)NCC2C(NC(C(C)(C)N(C)C)=O)CCC2)cnc(=N)[nH]c1 c1(COC)cc(C(=O)N(C)CC2CCN(C(c3coc(C)n3)=O)C2)no1 O=C(C1Cc2cccc(Br)c21)NCC1CC(=C2CC2)C1 c1(C(=O)NC2CCC(C)(CNC(=O)CC(F)F)C2)cc2cc(F)ccc2o1 C1(CC)(NC(c2sccc2CC#N)=O)CCN(C(C2CCC(F)C2)=O)CC1 S(=O)(=O)(c1ccc(NCC2CCOC2)nc1)NCC1(C)CCN(CC)C1 N1(CC(=O)NC(CN(C)C(C2CC2C(C)(F)F)=O)C)CCNC(=O)C1 N1(C(C2C(C(=O)OC)C2)=O)CCC2(C1)CN(C(C1(CC)CC(C)(C)C1)=O)C2 CCC(C(=O)NC1CC(CCNC(=O)C(C)(C)C2(C)CC2(F)F)C1)n1cncn1 c1(CC)nc(O)c(C(N2CC3CCC(N(C(=O)C(=O)N(C)C)C)C3C2)=O)cc1C c1(C(N2CC(C)C(NC(=O)COC3CC3)C2)=O)cc2ccc(Cl)cc2o1 c1(OC)c(-c2cn(CC3CCn4c(cnc4C)C3)nn2)ccc2ccccc12 C=CC(CCC)CC(=O)NCC(CNC(=O)Cn1ncn(C)c1=O)S(C)(=O)=O C1(C(C)(C)NC(C(c2cc(C)ccc2F)CO)=O)(C(=O)OC)CCC(F)(F)CC1 C1(CCC)C(O)CCCN1C(=O)C(=O)N(c1c(Cl)ccnc1Br)CC Cc1cc(O)c(Cl)cc1C(=O)NC1(CNC(C2(C)CC(C)C2)=O)CCOC1 C1(NC2C(CC)CC2)CCN(C(N2CCCCC2C(C)C)=O)CC1 C1(NC(CCN(C2CC2)CC)=O)CCCC1NC(C1(N2CCOC2=O)CC1)=O N(C1CCC(NC(=O)COCC2CCCC2)c2ccccc21)C(CC(C)(C)C)=O CCCC(C(=O)NC(C)(CNC(=O)CCOc1ccccc1)CO)NC(=O)NC CCC(CCCC=O)N.C(=O)(CCC(C)N(C)C)ONC(=O)CCSC Cc1cnc(Oc2ncc(NC(=O)C(O)C(F)(F)F)s2)c(NC(=O)C(C)C)c1 C1(C(N2C3(CN(C(C45CCCC(CO4)C5)=O)C3)CC2)=O)CCCC2CCCCC12 N1(CC)CC(C(N2CC(NC(c3c(Cl)sc(C)c3C)=O)C(C)C2)=O)CCC1=O C1(CNC(C2CCCC(OC)C2)=O)CCN(C(C2CC23CC(C)(C)C3)=O)CC1C C(=O)(C(C)S(N)(=O)=O)N1CCC(O)(CCNC(CCC#C)=O)C1 N1(C(c2cn(C(C)C)nn2)=O)CC(NC(C2COC3(CCC3)C2)=O)C(N=[N+]=[N-])C1 c1(CNC(C2(C)CCCC2)C)ccc2cc(F)ccc2n1 N1(C(CCN(C(CC(COC)C)=O)CC2CC2)=O)CC(=O)NCC1C(C)C c1(SC)nc(N(CC(CNC(=O)CC2=CCCC2)C(F)(F)F)C2CC2)ncc1C N1(CC(=O)NCc2cccc(C)n2)CCCC(N=[N+]=[N-])CC1 C(CC(C(=O)NCC1CC1C(C)C)NC(=O)CC1CCOC1=O)OC c1(SC)ncc(C(=O)NCC(C)NC(c2ccc(C3CCC3)cc2)=O)c(O)n1 C1(CC)CCCN(CC(N2CCCC2CNC(c2cc(Br)c[nH]2)=O)=O)C1 C=C(C)CC(C(=O)N(C(CO)C1CC1)C)NC(=O)C(=Cc1ccco1)C CC1CCOCC1C(N1CCN(C2CCCC2NC(c2cccnc2)=O)CC1)=O N1(C(c2c(C)nc(C(F)(F)F)o2)=O)CCCOC(CNC(=O)CC(C)C2CC2)C1 N1(C2CCC(NC(CCNC(C)=O)=O)C2)CCN(C(c2ccc(Cl)cc2)=O)CC1 N1(c2nc(C)nc(N3CCOCC3)c2)CCCN(C(=O)C2=CCCC2)C(C(C)C)C1 C1(CN(C(CCc2onc(CCC)n2)=O)CC)CCCCN1C(=O)C(C)CSC N1(CCC)CC(C(=O)NCCC(O)CNC(=O)CCNc2ncccn2)CC1=O c1(CC(=O)NC2C(NC(c3c(C)[nH]nc3Br)=O)C2)cn(C)c2ccccc12 CCCC(F)C(=O)NC1(CNC(C2CCN2C2CCCC2)=O)CCOCC1 c1(C(N(C)CC2CCCN(C(=O)C=Cc3cc[nH]n3)C2)=O)cncc(F)c1Cl C1(CNC(COC(C)=O)=O)C=CCN(C(=O)CS(C)(=O)=O)C1 C(CC(C(=O)N=c1ccn(C(C)(C)C)[nH]1)NC(=O)C=Cc1cscn1)SC C(=O)(C(C)NC(=O)CC1(N(C(=O)Cc2csnn2)C2CC2)CCC1)OC N1(C(C(F)=CC)=O)CCN(C(C2CC(=O)N(c3cccc(Cl)c3)C2)=O)C2CCC12 C1(C(N2CCC(CN(C(CCC)=O)C)C2)=O)CC2(C1)CC(CO)C2 N1(C(CN(C(=O)OCC)C)=O)CCC(N(C(=O)CC2CC(C)=NO2)CCO)CC1 C1(C(=O)NCC(CNC(c2nc(CC)sc2)=O)F)CCCC2(CCCCC2)C1 N1(C(C(=O)NCCSC)c2ccco2)CCc2cccc(F)c2C1C Cc1c(C(=O)NC2CCN(C(C3OC4CCC3CC4)=O)C2)nc2sccn12 C1(C(=O)NC(C2(OCC)CCC2)C)CC=CCC1NC(c1ncncc1Cl)=O N1(c2snc(CCC)n2)CCCC(NC(C2CCCOC2CC)=O)C1 N1(C(Cc2nc(C)[nH]n2)=O)CC2CC(NC(=O)C(F)(F)C3CC3)CC2C1 C1(C(C)(C)CNC(N2CC(N)C2)=O)CCN(S(C)(=O)=O)CC1.c1(N)ccccc1SC C(=O)(CC1=CCOCC1)NCC1(C(N)=O)CN(C(c2cnsc2)=O)C1 c1(OC)cccc(NC(=O)CC2CCCN(Cc3cccc(I)c3F)C2)c1OC C(C)(C(C)(C)C(=O)N1CCOC(CCF)C1)NC(C(C)C(F)F)=O C1(C(N2C(C3(NC(C=CC(C)(C)SC)=O)CC3)CCC2)=O)CC=CCC1C c1(OC)ccnc(CN(C)C(=O)NCC2CCOC(=O)N2)c1OC C(=O)(C1=C(Cl)CCOC1)NC1CCN(C(CC(CC#C)C2CC2)=O)C1C C(C)(CCN1CCCCC1)(c1nnnn1CC1CC1)NC1CC(=C)C1 c1(N(CCCNC(c2c(C)ccnc2)=O)C)ncnc(O)c1Br c1(NC(=O)NCC2(S(C)=O)CC2)cnc2c(c1)CCC1(CC2)OCCO1 Cn1ncc([N+](=O)[O-])c1C(=O)NCCC1(CNC(=O)C(C)(C)COCCF)CC1 C=Cc1cncc(C(C(=O)NC2CCOC2)N(CC(C)(Cl)CC)C)c1 C#CC1CN(C(=O)CCC2CCCCO2)CCN1C(=O)COCCOCCO c1(C(C(=O)NC2CC2)N(CCOCC#C)C(C)C)ccc(F)c(Cl)c1F C1(c2cc(CNC(CC=CCC)=O)on2)CCN(C(C2CC2(Cl)Cl)=O)CC1 c1(CN2CC(C)N(C(c3cccnc3Cl)=O)CC2)cc(F)c(Cl)c(F)c1 C1(CN(C)C(c2ccccc2-n2cc(CCCC(=O)O)nn2)=O)CCCS(=O)(=O)C1 C1(NC(C)=O)CN(C(=O)C(O)C2CCC2)CC(C)(C)C1.c12ccc(cc1)c(=O)s2 C(=O)(CC(O)CNC(=O)CC1CC1C1CC1)NCCC1(COC)CCC1 CCC(CC(=O)N1CCC(C(C)C(=O)N(C2CCCCC2)CCO)C1)C(C)(C)C C(C(C)(C)CNC(=O)CC1CC1COC)N(C(C1CC1F)=O)CC c1(C(=O)NCC(C2(O)CN(C(CCC(C)C)=O)C2)(C)C)cc2ncccn2n1 C1(CC)CN(C(=O)CC(C)F)CC1C(N1CC(OC(=O)NC)C1)=O C1(NC(COCCC#C)=O)CC2(C1)CC(C(=O)NC1(CCF)CCC1)C2 C1(C(=O)NCC(=O)OC(C)C)(COC)CCN(C(C2CC(F)(F)CS2)=O)CC1 C1(C(N2CC3C(CNC(c4ncccn4)=O)C3C2)=O)CC2(C1)CC1(CC1)C2 c1(N2CCN(C(c3n(C)cnc3)=O)CC2)cnc(Cl)c2cccnc12 C(=O)(CC(F)(F)C(C)(F)F)NC(CNC(C(CCC)C)=O)CCCC C(C)(C(=O)N1CCC(NC(c2ncccn2)=O)CC1)(C(C)C)OC C12(CNC(c3cn(C4CC4)cn3)=O)CCC1CCN2C(=O)COC(F)(F)F c1(C(=O)NC(C)(C2CCC2)CCO)c(Cl)ccc(O)c1N.C12(C=O)COCC1C2 C1(C(=O)NCc2n(CC)cnn2)CC2(CCC2)CN1C(c1ccc(C)[nH]1)=O CC1(CNC(C2CC3CCC2CC3)=O)CCCN(C(C)Cn2cncn2)C1 CN=c1[nH]cc(C(=O)NCCN(C(=O)CCc2cc(Cl)cs2)C2CC2)s1 C(=O)(CCC(C)(C)[N+](=O)[O-])N(C(C)CCNC(=O)CNc1ccc(F)cc1)C CC1(CCNC(c2cccc(CCO)c2)=O)CCN(C(C2CCC(=O)O2)=O)C1 c1(C(=O)NC2C(NC(CC(CC)OC)=O)CCCC2)nn(C)c(C)c1[N+](=O)[O-] C1(C(N2C(CNC(C3(N(C)C)CCC3)=O)CC(OC)C2)=O)CCOC(C)(C)C1 Cc1ncc(Br)c(C(=O)NC2CCN(C(=O)CC3CCC(C)(O)CC3)C2)n1 N1(C(CCCC=C)=O)CCC2CC2(NC(=O)Cc2cccc(C)c2)CC1 N1(C(C2ON=C(CC)C2)=O)CC2CC(C(=O)N(C(C)C(=O)N(C)C)C)(C2)C1 N1(C(Cc2ccc(OC)cc2OC)=O)CCCN(C(c2cc(C)[nH]n2)=O)CC1C C1(C(=O)NC2CC(C(C(=O)N(C)Cc3ccoc3)F)C2)C2CC3C(C2=O)C13 C1(C(N2CCC(C)(CC)C2)=O)C2CCC(C2)N1C(c1coc(OC)n1)=O N1(C(C2C(=C)C2)=O)CCC(C2CCN(C(C3(OC)CCSCC3)=O)CC2)C1 C1(C(=O)NCCCCC#C)CC2(CCN(C(=O)OC(C)(C)C)C2)CO1 c1(C(=O)NCCN(C2CCCCCC2)C(C(F)OC)=O)c(C(F)F)nn(C)c1C C1(C(=O)NCC(CC)N2CCCC2)C2CCCC12.c12cc(on1)CNC2=O CC1CCN(C(C)(C)CNC(C2CCCN(c3cncc(F)c3)C2)=O)CC1 C(=O)(C1=CCc2ccccc21)N1C(C(C)NC(CC(=O)OCC)=O)CCCC1 N1(C(CCC(C)OC)=O)CC2CN(C(=O)Cn3cnccc3=O)CC2C1 N1(C(CC)=O)CCC(NC(=O)C(C)Oc2cc(Cl)cc(Cl)c2)C(C)(C)C1 C1(C(=O)NC(C)Cc2cc(C)[nH]n2)(SC)CCSCC1 CCCCC(O)CC(=O)N1CC(CC(=O)NOCC(C)C)C2(CCC2)C1 C#Cc1cccc(NC(C2CCCN(C(=O)Nc3ccc(O)cc3)C2)=O)c1 Cc1nc[nH]c(=NCCC2CCCCN2C(=O)C(C)C(C)O)c1F c1(NC(C2C(NC(c3cn(CC)nc3)=O)C2)=O)cc(C)ncn1 C1(N(C)C)CCCN(C(=O)CC2CC(F)CN2C(=O)CC(O)C2CCCC2)C1 CN1CC(C)(C)CC1C(=O)NCCNC(=O)CCCc1ccsc1 c1(NC2CCC(NC(c3c(C)c[nH]c3)=O)CC2)ncnc2c1cc(I)n2C c1(C(=O)NC(Cc2cc[nH]n2)C(=O)NCc2cnn[nH]2)ccccc1Cl C1(C)(NC(C2CCC(C(C)C)N2C(=O)C2=CCCC2C)=O)CCCCC1(C)C c1(CC(=O)N(CC#C)C(c2ccc(Cl)cc2)C)nc(C(F)(F)F)nn1C c1(C(N2C3C(NC(C(C=C=C)C)=O)CC(C3)C2)=O)cc2cc(C)cc(C)c2[nH]1 C1(C(=O)NCC(=O)N(CC)CC2CCCO2)CCCSC1C C1(CNC(C=C(C)C)=O)COCCN(C(c2cc(F)ccc2OC(F)(F)F)=O)C1 C(=O)(CCS(N)(=O)=O)NCc1nc(CNC(CC2(OCC)CC2)=O)sc1 c1(C(=O)NC(C(=O)OC)CN2CCCC2)cc2cc(Cl)ccc2s1 C1(CN(C)C(c2ccccc2C(F)F)=O)CCCCN1C(=O)CC1CCCCC1 Cc1nc(NCCC(F)CN=[N+]=[N-])cc(NC2CC3CCC3C2)n1 C#Cc1ccc(OCC(N2CCCC2CCCNC(=O)C(CO)N(C)C)=O)cc1 c1(C(=O)NC(C)CCNC(=O)CC2(O)CCCOC2)coc2c(F)cc(Cl)cc12 N1(C(CC2(C=C)CC2)=O)CC2(CCC(CNC(=O)C(C)(C)NC(C)=O)O2)C1 c1(CC)cccc(C(=O)NC(CNC(c2cnn(CCF)c2)=O)C(C)C)c1C C#CCCCC(C)C(=O)N(C)CCOCCNC(c1cc2occc2s1)=O Cc1nc(CO)sc1CC(=O)N(C)CC1CCN(C(c2cn(C3CC3)nn2)=O)C1 N1(C(C(c2ccc(C)cc2)C)=O)CC2CC(C1)C2NC(C1C2COCC12)=O C(C(C)(O)CC(=O)NC1CC2(C(=O)NCC(=O)N(C)C)COC1C2)OC Cc1nc(=N)[nH]cc1C(=O)NCCC1CCCN(C(C2CCS2(=O)=O)=O)C1 C1(CNC(c2c(C)nc[nH]2)=O)CCCCN1C(C1(CO)CCCO1)=O N1(C(CC(=O)NCC)=O)CC(NC(=O)Cn2cnccc2=O)C2(CCOCC2)C1 N1(C(CCCN(C(C)C)C)=O)CC(NC(c2cnn(C)c2F)=O)C2CC12 c1(C(N2CCC2C2CCCC2)=O)cncc(Cn2cc(OC(C)(C)C)cn2)c1 C(CNC(=O)C(C1CCCCC1)O)(CC(=O)N1CCCC(CCCO)C1)OC N1(C(C=C(COC)C)=O)CCOCC(NC(c2cccc(C3CC3)c2)=O)C1 N1(C(c2c(C)nsc2)=O)CC(C(=O)NCC2(C)OCCO2)C2(CC2)C1 N1(C(CC2(C)CC2)=O)CCOCC1CNC(C1CCCN1C(c1ccccc1)=O)=O c1(OCC(=O)NC2CN(C(CC=CC)=O)CC2O)cccc(C)c1F C(C)(C)(CCNC(C1CC2CC2C1)=O)NC(CCN(CCC(C)(C)C)C)=O C1(OC)CCCC(C(=O)N(C(C)C(=O)NC2(C(=O)OC)CCC2)C2CC2)C1 N1(C(C2CN(C(c3ccc(F)cc3)=O)C2)=O)CC(CNc2n[nH]c(C)c2O)C(C)C1 c1(SCC(=O)NCCN(C2CCCC2)C(c2c(C)cco2)=O)cccc(F)c1 C1(C(=O)NCc2ncccc2F)C2CCCC2CN1C(=O)CC1CCC2CC12 c1(C(N(CC(C)NC(c2ccnnc2)=O)C)=O)c(F)c(F)c(F)c(F)c1F N1(C(c2c(OC)c([N+](=O)[O-])ccc2)=O)CC(NC(=O)C=CCO)CC12CCCC2 c1(C(C)C(=O)NCC(c2ccccn2)O)ccc(C(F)(F)F)cc1 N1(CC)CCCCC1C(=O)NCC1CCN1C(c1ccc(CO)s1)=O C(=O)(CC1=CCCCC1)N(CC(C)CNC(=O)CC1CC2(CCC2)CO1)C C1(NC(c2ocnc2C2CC2)=O)CN(C(c2cccnn2)=O)C2CCCC12 C1(CNC(C=CC)=O)CN(C(=O)Cc2csc3cc(C)sc23)CC2(CCC2)O1 C1(NC(c2nc(OCC)oc2)=O)C2CC3C(C2)C13C(=O)NCC1CNC(=O)CO1 c1(CCC(=O)NC2(C(=O)NCC3CN(CC)C3)CCC2)ncc(C)[nH]1 C(=O)(CN=c1cc[nH]cc1)NC1(C)CN(C(c2cccc(C)c2C(F)(F)F)=O)C1 c1(CC)ncccc1C(N1CCC1C(=O)NCCCS(C)(=O)=O)=O n1(-c2cccc(C)c2)c(C(N2CCCC(C3(C)CC3)C2)=O)cc2ccccc12 c1(OC)ccc2c(C(N3CC4(CC(NC(C5(F)CC5C)=O)CO4)C3)=O)csc2c1 C(=O)(CN=c1cc[nH]cc1)N1CCCC(F)(C(=O)NC2CCN(C)CC2C#N)C1 c1(C(CC(=O)OCc2c(C(=O)OCC)scn2)C)ccc(Br)cc1 CC(c1ccco1)=CC(=O)NCC(C)(C)CNC(c1coc(CC2CC2)n1)=O C1(N(C(CN2CC(CC)C2)=O)C)CCC(NC(c2cncc(C(C)C)c2)=O)CC1 Cc1noc(C(=O)N(CC(O)CN(C)C(c2nnc(C(F)(F)F)s2)=O)C)n1 CCCCCCC(=O)N1CCCC(F)(CNC(=O)CCC2CCC(C)O2)C1 C1(C(=O)OC(COC(C)C)(C)C(C)C)CC(C)CN(C(=O)OC(C)(C)C)C1 C1(C(N(C2CC2C(F)(F)F)C)=O)CCCN(C(c2c[nH]nc2-c2ccoc2)=O)C1 C1(CC)CN(C(c2cnc(C3CC3)cc2C)=O)CCN1C(=O)C(=O)C(F)(F)F CC1C(C)N(C(=O)C=CCO)CCN1C(=O)CS(N)(=O)=O C1(CNC(c2cnn(CC)c2C)=O)CCN(C(=O)C(C)C(=O)OC)C1(C)C C(=O)(C(C)CC(C)C(C)=O)NC1CCC(C(NOCCCC(=O)OC)=O)C1 C1(C)(C(N(C(c2ccccc2)C)C)=O)CCN(C(c2nccs2)=O)C1 c1(OCC)cccc(C(=O)NCCOCCCNC(C2CC(C)(C)O2)=O)c1N c1(COC)nc(C)c(C(=O)NC(C2CCCN2C(C2CC(CC(F)F)C2)=O)C)s1 N1(C(C2CC(C)OCC2)=O)CCC2(CCN(C(C3CCOC(C)C3)=O)C2)C1 N=c1[nH]c2ncc(C(=O)NCC3CC4CCC(C3)N4C3CC3)cc2s1 C(=O)(CCCCCCCCSC)N(CCN(C(=O)C1=C(C)OCCS1)CC)CC c1(CSC)cc(C(N2CC(CNC(C3CC3(C)C(F)F)=O)C2)=O)ccc1F N1(C(=O)C=CCOc2cccc(F)c2)CCN(C(C2C3COCC23)=O)CC1 CC1CN2CC(C)N1CCC(C)(O)C2=O.N(C)C C(=O)(C(CC(C)C)C(C)C)NC1C2CCN(C(c3c(C)nn(C)c3F)=O)C2C1 C1(CNC(C(C)SC2CCCC2)=O)CN(C(C2CN(C(N)=O)C2)=O)CC12CCC2 C1(C(=O)NC(C)CSC(F)F)C2CCN(C(=O)CC3CCCC(C)O3)CC12 c1(C(C)=O)cc(=NCC2CCN(C(C3CCCN3S(C)(=O)=O)=O)C2)[nH]cn1 C1(CC)CN(C(=O)CSCCC(C)C)CCC1NC(C1(COC)SCCCS1)=O c1(NC(c2sc(C)c(CC)c2C#N)=O)nccc2sccc12 C12(NC(C3C(CN(C)C)CCC3)=O)CCC(NC(=O)CCCC3CCC3)(CC1)C2 C(=O)(C1=Cc2ccccc2OC1)NCC(CNC(C1(OC)CCOC1)=O)CO c1(CC)oc2ccccc2c1C(=O)NC1CCC1CNC(c1csc(Cl)c1)=O CC1CN(C(c2nscc2N)=O)CCC1CNC(=O)C(C)(C)Cc1cnn[nH]1 C#CC1(C(=O)NCC(CC(C)C)OC)CCN(C(=O)CCCCC2CC2)C1 N12CC3(CC(CO3)C1=O)C2.c1(CNC(COC(C)=O)=O)cncc(C(F)(F)F)c1 c1(C(C(=O)N(C2(c3ccc(OCOC)cc3)CCC2)CC)O)ccc(F)c(Cl)c1 c1(C(C2CCCC2)NC2C(NC(C=C(C)C(C)C)=O)CC2)cn(C2CCC2)nn1 N1(C(C(C)(C)F)=O)CCN(C(c2ccc3nccn3n2)=O)CC(CO)C1 C1(CC=C)(NC(c2n[nH]c(C3CC3)c2C)=O)CCN(C(=O)C(C)C(C)O)C1 CC1N(C(=O)CCC(C)(F)F)CCC12CNC2 N1(C(CCCC=C)=O)CCC(C(=O)NCC2C(C)(C)C2(F)F)C12CCC2 c1(CC(N2C(C3(CCC)CC3)CCC2)=O)cccc(OC(=O)CCNC=O)n1 CCN=C(NCC(CO)CC(C)C)N1CCc2cc(Cl)cc(Cl)c2C1 c1(C(N2CC(CNC(C=C(C)C3CC3)=O)C3C2C3)=O)cccc([N+](=O)[O-])c1C C1(C(=O)NC(C)Cc2ccccn2)CCCN(N2CCC(c3ccccc3)C2)CC1 N1(Cc2cc(C)cc(Cl)c2)CCc2ccccc2C(N)C1 Cc1ccc(F)c(C(=O)N(CC(O)CNC(c2csc(C(C)OC)n2)=O)C)c1 N1(C(=O)NCc2ncc(COC)s2)CC2CC(=O)CC1C2 c1(C(=O)NCC2(O)CCN(C(C(n3ncc(C)c3)C)=O)C2)cc2n(c1)CCOC2 C1(C(N(C2COC(C)(C)C2)C)=O)C2CC(O)C(C2)N1C(C1(C)COC1)=O c1(NC(C2(OC)CCC2)=O)cc(N2CCOC(CN(C)C)C2)nc(C)n1 c1(C(N(CCNC(CCC#C)=O)C)=O)c(Cl)ccc(C)c1N C1(CC=C)(NC(c2nc(F)ccc2Cl)=O)CCN(C(C2CCN(C)C2C)=O)CC1 C(C)(CCC(=O)N(CCC(=O)NCCCc1n[nH]c(C)n1)C)OCC CC(c1cccs1)=CC(N1CC(CNC(=O)Cc2ccc(Cl)cc2)C(C)C1)=O N1(C(CCCCN(C(c2c(C)c(F)cnc2)=O)C)=O)CC(O)CC(C)(C)C1 c1(OCC)ccc(C(N2CC(NC(=O)Cc3cncs3)C(O)C2)=O)cc1OCC N1(C(C=CC=CC)=O)CCC(NC(c2coc(Cl)n2)=O)CC(O)C1 c1(C(N(CCC)CCNC(=O)C(C)CN(C)C)=O)cnn2c1C(=O)NCC2 N1(C(=O)NC2CCC(CC)C2)CCC(O)(CCNC(=O)C(F)=C(C)C2CC2)CC1 c1(OC)ccc(C(=O)N(C)CC2CN(C(=O)CCC3(O)CCC3)CCO2)cc1F C1(NC(c2cc(C(=O)OC)no2)=O)CCC(N(C)C(c2cn[nH]c2)=O)CC1 Cc1ccc(C(=O)NC(C)(CNC(=O)C(C)C(F)(F)F)CO)c(O)c1C CC(C)C#CC(=O)NCc1cnn(C)c1C(=O)NCC1CC2CCC2C1 c1(NC(=O)NCCN2C(C(C)O)CC2)cncn1-c1ccccc1 c1(OCc2nn(CC)c(=O)cc2)ccc(Cl)c(C#N)c1 S1(=O)(=O)C2=C(Br)C=CC(=NCCCNN1C)N2.C(C(COC)OC)OCC N1(C(C(C)(C)OCC)=O)CC(CNC(c2cc(-c3ccoc3)[nH]n2)=O)C(C)C1 c1(CNC2CC(C(=O)Nc3cnc(C(=O)OC)nc3)C2)ccc(F)c([N+](=O)[O-])c1 C1(Cc2n(CC=C)c(N3CCCC(C)C3)nn2)CC(C)CCC1OC c1(NC(C2CSCCN2)=O)ccc(Cl)c(Cl)c1.C12CN(CCO1)C(=O)NC2=O c1(OCC)ccc(SCC(=O)NC2CCCC2CNC(c2ccns2)=O)cc1 CC(C)(C(=O)N1CCN(CCNC(=O)COCC2CCCO2)C1=O)C(F)F C(c1cc2ccccc2o1)=CC(N1CCC(NC(C2CC=C(C)CC2)=O)C1C)=O C(=O)(CCCC(C)(C)C#N)C12COCC1CNCCN(C(C)C)C2=O c1(C(C)C)nc(C(=O)NCc2ccoc2C(=O)NCC=C(Cl)Cl)co1 Cc1cccc(F)c1CC(N1CC2CC(N(C(=O)CCC3CC3(F)F)C)C1C2)=O C(=O)(N=c1[nH][nH]c2ncccc12)c1ccc(NC(Cc2c(C)ccc(C)c2)=O)[nH]1 CCCCC(CC)CCCN(C(c1ccc(Br)cc1)C(C)CC)C(=O)NCC#N N1(C(CCC2(C)CCCN2C(C2CC3CCC3C2)=O)=O)CC(C2CCCCC2)C1 N1(CCNc2nnc(CCCOC)n2CCS(C)(=O)=O)CCCC2(CCOC2)C1 CC1CCC(COc2ccccc2)N(C(c2cnc(O)o2)C(=O)NCC2CC2)C1 C12(NC(C=NOC)=O)CCC(CNC(=O)C(F)C3CCOC3)(CC1)OC2 C=CCN=c1[nH]c(N2CCC3(C2)CC(F)(F)C3)nc2cc(OC)ccc12 c1(OCC)cc(C(=O)NCC2CCC(N(C)C(c3ccsn3)=O)CC2)cc(F)c1 C(C1=NOC2CN(C(c3cc4c(ncn4C)[nH]3)=O)CC12)NC(C(COC)(F)F)=O C(=O)(C1=COCCC1)NC(C(=O)N(CCCCO)CC)(C)CSC C1(N(C(=O)C(Cl)(Cl)Cl)CC)CC2CCC(C1)N2.C(C)(C(=O)O)CC c1(C(=O)NCC(CC)NC(=O)CN2CC3CC3C2)ccnn1CC(F)F c1(C(=O)NC2(CF)CCN(C(C(CC(=C)C)C)=O)C2)cnc2ccccn2c1=O C1(CCNC(=O)NC(C)C)COC(CNC(OC(=N)O)=O)C1 c1(C(=O)NC(C2C(C(=O)NC3CCC3N3CCC3)C2(C)C)C)cc(F)ccc1F C1(CNC(C2C(C)C2C)=O)CCC2(CCC2)C1NC(=O)CCCc1ccccn1 C1(NC(C(=O)NC2(C#C)CC2)=O)CC2C=CC1C2 C(C(=O)NCC(=O)NC(C)CO)NC(C)=O.CCF N1(C(C(C2N(C(c3n(CCC)ccc3)=O)CCC2)(C)C)=O)CC(O)C(C)(C)C1 N1(C(CCOc2c(C)cccc2)=O)CC(NC(C23CCC(C2)C3)=O)CC(F)(F)C1 c1(C2CCC(NC(=O)Cn3ccnc3)CC2)cc(F)cc(F)c1 CC1(CNC(C2CCCSC2)=O)CC(F)(F)CN1C(=O)Cn1nc(Cl)ccc1=O N1(C(C23CC2C3)=O)CC2(CCN(C(=O)C=CC3CCCN3C)C2)C1.COCC C1(CC(=O)NC(C(=O)OC)CNC(=O)CSC(F)(F)F)CCC(C)(C)O1 c1(C(=O)NCc2ccc(COC)cc2)nnn2c1C(=O)NCC2 c1(C(=O)NC(C(CO)NC(CC2(CSC)CC2)=O)C)cnc2ccccc2c1 C=CCC(C)(C)CC(=O)NC(C)(C)CNC(c1c[nH]nc1C1CC1)=O c1(OC)ccc(CCC(N2CCCC(NC(=O)C=CC(=O)N(C)C)C2)=O)cc1F C(=O)(CC(C(F)(F)F)c1ccon1)NC1CCN(C(CCCC=C)=O)CC1C C1(NC(=O)CCc2ccccc2)CC2CCC1N(C(c1cn(CCF)nn1)=O)C2 c1(C(=O)NCC(C)N(C)C)cc(F)ccc1OCC1(c2ccccc2)CC1 CC(C)(CCC(=O)NCC1CCCN1C(=O)CC1(C)CCS(=O)(=O)N1)C1CC1 C1(C(N2CCC(CN(C(=O)CCCCC(F)F)C)C2)=O)(OC)CCCC(C)(C)C1 c1(C(N2CC(CNC(CC=C(C)C)=O)C2)=O)cc(C)nc2c(C#N)cnn12 N1(C(CCN(CCC)C)=O)CCN(C(c2cnn(CC)n2)=O)CC1CSC C1(C(=O)OC(CC2(CC(=O)OC)CC2)=O)CCN(C(C2CCCN2C)=O)CC1 C1(O)(C(=O)NCc2c(C(=O)Nc3cc(C)sc3)nco2)CCOC1(C)C C1(N(C(C(C)N(C(=O)CNC=O)CCC)=O)C(CC)CC)CCCC1CCO c1(C(N2C(C(C)NC(C(CC)C)=O)CCC2)=O)ccc(N2CCCCC2)nc1 C1(F)(C(N2CCC(C(=O)NC(C3CC3)C3CC3)C2)=O)CC=CCC1 C1(NC(C(C)N(C)C)=O)CN(C(=O)CC2Cc3ccccc3N2)CC1(C)C C1(NC(C2CNC(=O)N2)=O)CN(C(=O)CSCCC(F)(F)F)CCC1F c1(C(C)=O)cc(C(=O)NCC2CCN(C(=O)C(c3cnn(C)c3)C)CC2)n(C)c1 C1(C(N(C2CN(C(=O)CSC3CC3)C2)CC)=O)CSCCN1C(=O)OC(C)(C)C Cn1[nH]nnc1=NC1CCCN(C(=O)Cc2cc(C3CC3)no2)C1 N1(C(c2cnc(C)nc2)=O)C2CCC1CC(C(N1CC(n3cnnc3)C1)=O)C2 N1(C(c2cn(C)nn2)=O)CCC2(CC(NC(=O)C3=COCCO3)CO2)C1 CCC(CC)CC(C(=O)NCc1cccc(C(=O)OC)c1)N1CCC2CCCC2C1 N1(C(C)=O)CCC(C2CCCN2C(=O)Sc2ccc(N(C)C)cc2)CC1 N1(C(CC(=O)NC2CC2)=O)CCOCC1C(=O)NCc1cccc(F)c1 C1(C(=O)N(CCO)CCO)CC(O)CCN1C(c1ncccc1Cl)=O CN=c1[nH]nc(CC(N2CCC(N(C(=O)C(C)Cn3ccc(C)n3)CCO)C2)=O)s1 c1(C(N2C(C)CCC(NC(=O)CCC3CCOC3)C2)=O)cc2ccsc2n1C C(=O)(CCC(C)(C)NCCC1CCC(C)C1)NC(c1cnn(C2CC2)c1)=O N1(CC)C(=S)NC(c2cc(Cl)c3ccccc3n2)C(C(=O)OC)=C1c1ccnn1C N(C(=NCCC(=O)N(C)C)NCC(C)Cc1cccc(Br)c1)C(C#C)CC1CC1 CC1C(NC(c2nc(Cl)ccc2F)=O)CC2CCC1N2C(=O)CCCC(F)(F)F CC#CCC1C(=O)CC(OC)C(=O)N1.C(CC1CC1)(C(C)CC)NC(C)=O C1(NC(c2cn(C)nn2)=O)C2CC1N(C(C1(CO)CCOCC1)=O)C2 N1(C(c2cnc(C)s2)=O)CCN(CCNC(=O)CCSC(F)(F)F)CC1 C1(NC(C2(NC(CSCC#C)=O)CC2)=O)CCCC1c1nc[nH]n1 c1(C(=O)NCC(CC)NC(=O)CC(C)N(C)C2CC2)cn(C(C)C)cn1 C1(N(CCC)C(c2sncc2C)=O)CCN(C(=O)C(C(C)C)n2cnnn2)CC1 N1(C(C(F)=CCC)=O)CC2CCN(C(=O)COc3cc(C)ccc3F)CC2C1 c1(CN(C(c2cccnc2)(C)C)C)nccc(=NCC2(N(C)C)CC2)[nH]1 N(C1CC2(CCN(C(=O)C(O)C3CCC3)CC2)c2c(C)cccc21)C(CC=C)=O c1(CCNC(=O)NCC2C(CCC)CCC2)ccccc1Br C(=O)(CC(F)(F)C(F)(F)F)NC1C(CNC(CCc2cc(C)no2)=O)C1 c1(N2CC(=O)N(C)C(=O)C2)nc(N2CC3CC3(CO)C2)c2c(n1)CCOC2 n1(CC)ncc(C(=O)NC2CN(C(=O)C(c3ccn(C)n3)C)CC2C)c1Br C(=O)(CC1=Cc2ccccc2C1)NC1C(NC(c2cnn(C(C)C)n2)=O)CCC1 CC(C)CC(C)CS(=O)(=O)Cc1cc(Cl)ccc1Cl N1(C(C)CNC(C2CCC(NC(c3cocn3)=O)C2)=O)CCCC(O)C1 N1(C(C(C)SC)=O)CC(NC(C2CCCN2C(=O)OC(C)C)=O)C(C2CC2)C1 C(=O)(CCC(C)CNC(c1ccccc1OC)C)OC C1(C2(C(=O)NCCN(CC(F)(F)F)C(=O)C3CC3)CC2)CCCCO1 CC1=C(C(=O)N2CCC(C)(NC(=O)C(F)n3ccnc3)C2)CCC(C)(C)C1 C(=O)(C(O)C(C(C)C)OC)NC(CC(=C)Cl)C(=O)NCC1C(C)C1(F)F N(C(=NCc1ccc(NC(CC(C)C)=O)s1)NCC(C)C)CCN1CCCC1 c1(C(N2CC(O)(C(C)NC(C3CN4CCN3CC4)=O)C2)=O)c(F)cc(F)cc1F Cc1cc(C(=O)NC23CCC(CC2NC(=O)CCNC(=O)CO)C3)cnc1O N1(C(C(C)SCc2ccncc2)=O)CCCC(C)(CNC(c2ccccn2)=O)C1 c1(C(C)C)cc(-c2cn(CC(N3CCC(CC#N)C3)=O)nn2)ccn1 C(=O)(CCCN(C)N=O)N1C(CNC(CC(C)CF)=O)CC(F)C1 c1(NS(CCC)(=O)=O)ccc(CNC(C)(CO)CCF)cc1 CC(C)C(=O)C(=O)NC1(c2ccccc2)CCC(C)C1.C(=O)OC N1(C(C2C(C)C2C)=O)CCC(NC(c2cc(=O)c(O)c[nH]2)=O)C(C)(C)C1 C#CCCCCCC(=O)N1CCC(N(C(=O)CCc2ccsc2)CCC)CC1 CC1CC(NC(c2ccc(C(F)F)s2)=O)CN(C(c2ncccc2Br)=O)C1 c1(CC)ncc(C(=O)NCC=CCNC(=O)C(O)C2CCCC2)c(O)n1 N1(C(C=CSC)=O)CCN(C(=O)C(C)(C)c2ccccc2)CC1CC(F)(F)F CCC(C)C(O)C(C)C(=O)NC1CCC(CC(N2CCOC(C=C)C2)=O)C1 CC1CN(C(c2cc(Cl)ccc2C(N)=O)=O)CCCN1C(=O)Cn1nnnc1O N1(C(C(C)OCCOC)=O)CCC2(CC1)CCN(C(=O)Cc1cn(C)nn1)CC2 C(=O)(C#CC1CCCCC1)N1CC(C(=O)NC(C)CC2CCCCCC2)OCC1 C1(C(=O)NCCNC(C(=O)NC(C)C)=O)CCC2(CCCC2)CC1.C1CO1 O=C(CCCC(F)(F)F)NC(C1CCN(C(c2cccnc2)=O)CC1)CCO C(=O)(CS(=O)(=O)C(C)C)NCC1(C)CCC(NC(C=C(COC)C)=O)CC1 Cc1cccc(C(=O)N(c2cc(CNCC3(C)CC3(F)Cl)ccn2)C)c1 c1(C(=O)NC2CCC(c3nn[nH]n3)C2)cc2n(n1)CCOC2 C1(CN(C(COC(CC)CC)=O)C)CCCN(C(C2CC2CF)=O)C1 c1(CC(=O)NCC(C)NC(COC)=O)cccc(Cl)c1.C1(C2CC2)C(=O)N1 C1(C(=O)NCCC2N(C(c3ccc(C(N)=O)[nH]3)=O)CCC2)CCC([N+](=O)[O-])CC1 C1(c2cn(CCN(C)C)nn2)(NC(=O)C(C2CC2)C2CC2)Cc2ccccc2C1 C1(C(=O)NCCC(=O)N(CCC(=O)OC)C2CC2)OCCC1(C)C CCC(F)(F)C(=O)NCC1(NC(=O)C(C)c2cccs2)CCC1 c1(C(N2CC3CCN(C(c4nn(C)c(O)c4)=O)CC32)=O)ccc2cccnc2c1 Cc1cn2cc(C(N3CCC(NC(c4ccnn4C)=O)C3(C)C)=O)nc2s1 C(=O)(C1=CCC2CCC1N2C(C1CCC(N=[N+]=[N-])C1)=O)N1CCOCC(C)(F)C1 C1(CN(C(C2C(CC)CCC2)=O)C)CCCN(C(=O)COCC2CCC2)C1 c1(CN(C(CN(CCC(=O)NCCOC)CCC)CC)C2CC2)cccnc1 Cc1ccc(C(=O)NC(CNC(=O)CC2(C)CCC2)C2CC2)o1 c1(CC(=O)NCC(CC)NC(=O)CCc2ccncn2)ccccc1Br Cc1ccc(C(C)C(=O)NCCOCCNC(c2cc(-c3ccco3)n[nH]2)=O)s1 C1(NC(CC2(C(=O)OC)CC2)=O)C2CCC1N(C(C1CC(O)C1)=O)C2 N1(C(COCCC#C)=O)CCC2(CC1)CC2NC(=O)C(c1cccnc1)OC c1(C(=O)NCC2CN(C(COCC)=O)CC2(C)C)cc(Cl)cc2c1CCC2 c1(CC(=O)NCCCCNC(c2ccc(SC)o2)=O)c[nH]c2ccncc12 N1(C(C(C=C)c2ccccc2)=O)CC2(CC(NC(c3ccnnc3)=O)CO2)C1 C1(C#N)(C(N2C(C)CN(C(=O)CCc3ccccc3F)CC2)=O)CC12CCCC2 N1(C(C2CCC(OC)C2)=O)CC2(CC(NC(=O)Cc3cncc(C)c3)CO2)C1 N1(C(C2(C#N)CC2)=O)CC2CC(NC(C34CC3C4)=O)CC1C2 C1(NC(C2C(CC)CCN2C(c2scnc2C)=O)=O)CCCN(O)C1=O C(=O)(C1CCCc2c[nH]nc21)N1CC(F)CC(NC(=O)CCc2cscn2)C1 Cc1c(Cl)ccc(C(=O)Nc2cccc(C(N3CCn4ncnc4C3)=O)c2)c1F C1(CCCC(=O)NCCOCCN(C)C(C2CC23CCC3)=O)CCCC(=O)N1 c1(C2N(C(=O)NCCCNc3c(Cl)cccc3Cl)CCCC2)cc(Cl)cc(Cl)c1 C1(C(N(CC(C(C)C)C)C(C)(C)C)=O)C=CCN(C(c2cccs2)=O)C1 N1(C(C(C)OCC#C)=O)CC(NC(c2cc(-c3ccco3)cn2C)=O)C(C)C1 C(=O)(C(O)C(C)C)NC1C=CC(C(=O)NC2(c3nc(C)on3)CC2)C1 CC1CN(C(=O)CCC2CCC2)CCCN1C(=O)CC1CCOCC1(C)C c1(C(=O)NC(C)CN(C(=O)CC2C=CCCC2)C)c(Cl)ccc(F)c1N C1(CN(C)Cc2c(C)cc(F)cc2)CN(c2ccc(C3CC3)cc2)CC(F)(F)C1 c12ccc(cc1)C(=O)CC1CC1NC2.C(=O)(CN(CC(=O)OCC)C)NCC CC1CC(CNC(=O)C(Cc2ccccc2)N2CCCC2)CN1C(=O)C=C1CC1 c1(CS(N2C3CN(Cc4cncc(C)n4)CC32)(=O)=O)c(C)cccc1C C1(C(=O)NC2C(NC(c3cc(Cl)c(F)cc3F)=O)C2)CCc2ccccc2C1 C#CCCCCCCCC(=O)N1CC(CCNC(c2cc(CC)on2)=O)C(C)C1 C1(CC)CCN(C(c2c[nH]c(C(N)=O)c2)=O)C(C(=O)Nc2cnc(SC)nc2)C1 N1(C(c2c(C)con2)=O)CC(F)(F)CC1CNC(C1(S(C)(=O)=O)CCC1)=O C(CS(=O)(=O)NOC1CCOCC1)(C(F)(F)F)OC Cc1cccc2c1OCC(NC(=O)NC(C(F)F)C1CCC1)C2 c1(C(=O)NCCC2(NC(c3cccc(C)c3)=O)CCC2)occ2c1CCOC2 C1(CNC(=O)C(=O)Nc2ccc(-c3cnn[nH]3)o2)CCCC12CCOCC2 C1(NC(C2C(COC)C2)=O)C(C)(C)CN(C(=O)Cc2cccnc2)CC1(C)C c1(C(N(CC(=O)NC2(C)CN(C(=O)CSc3cccs3)C2)C)=O)cnn(C)c1N C(=O)(CC(C)(C)O)NC1(CCC(=O)NCC(C2CCC2)OCC)CCCC1 C1(CC(=O)OC(C)(C)C)CCCC(C)(C)O1.C1(=O)C(CCc2ccco2)N1 N1(C(C(c2ccc(C)cc2)(C)C)=O)CC2CCC(C1)C(NS(C)(=O)=O)C2 c1(NC(C(CCC)NC(=O)C(CC)C(C)C)=O)ccc(C(C)=O)c(F)c1 c1(OC)ccc(CN2CCC(C)(C(=O)NC(c3ccccc3)CC(C)(C)O)C2)cc1O C1(C2(O)CCC2)(CNC(C2(OC)CCN(C(c3ccn(C(F)F)n3)=O)C2)=O)CC1 CC(C)CCC(C)N(C(=O)CC1CCCN(C(C2(C(C)C)COC2)=O)C1)C Cc1ccc2sc(C(=O)NCC3(NC(c4cnsc4)=O)CCC3)c(C)c2c1 c1(CC(=O)NC2CCN(C(C3CC3(F)F)=O)C2)c(F)cc(Br)cc1F CC(C)CCCCC(=O)N1CCCC(CNC(=O)CSc2ccc(O)cc2)CC1 n1(CC)ncnc1C(N1CCCC1CCCNC(=O)CC1CCCN1C(C)=O)=O C1(NC(CNC(CC)=O)=O)CCCN(C(c2cc(C(C)(F)F)on2)=O)C1 c1(C(=O)NC(CCCC)CNC(=O)CS(C)(=O)=O)cc2cccc(OC)c2o1 c1(CC)ccc(C(=O)N(CCC(N2CC3CC3(CC)C2)=O)C2CC2)nc1 N1(C(c2scc(C)c2Cl)=O)CCN(C)C(CNC(=O)COc2cccc(Cl)c2)C1 CCC(C)(CO)C(=O)NC(C)CNC(=O)CCSc1cc(C)ccc1C N1(C(COCCOCC#C)=O)CCC(C(=O)Nc2ccccc2Br)CC1C c1(C(=O)NCC2(C)CN(C(C3CCCC(=O)N3)=O)CCO2)n[nH]c2c1COCC2 c1(C(=O)NC(CC)CNC(C2(c3cccs3)CCCCC2)=O)ccc(C)c(Cl)c1 Cc1ccc(C(=O)NC2CCCC2NC(=O)C(O)CC(F)F)nc1C c1(CC(C)NC(c2c(C(C)=O)nccc2)=O)c(F)ccc(Cl)c1F Cn1cnc(N2CCC(O)(Cc3c(F)cccc3F)CC2)cc1=O C1(C(=O)NC(n2cc(C(=O)NC34CCC(C3)OC4C)nn2)C)CC2(C1)OCCO2 C(=O)(C(O)P(C)(C)=O)NC(C)CN1CCN(C(C23CC(CCO2)C3)=O)CC1 C(=O)(C(C)S(N)(=O)=O)NCC1(OC)CCCN(C(=O)C(C#N)C(C)C)C1 C(C(CC(=O)OC)CC(C)C)NC(=O)CC(CC(C)C)NC(C)CNC(=O)OCC N1(C(C2C(C)(C)C2)=O)CCC2CN(C(c3nc4ccc(F)cn4n3)=O)CC2C1 C1(NC(C(C)=CC2CC2)=O)CCC(C)N(C(C2C(Cl)(Cl)C23CC3)=O)C1 CC1CCC(NC(C2CCCC23CCC3)=O)CN1C(=O)COc1cccc(O)c1 c1(OCC)ccc(C)cc1C(N1CCC1CNC(C1(C)CC1(F)F)=O)=O C1(NC(c2c(C)ccnc2)=O)CC=C(C(=O)N2CCC(n3ccnn3)C2)C1 c1(C(N2CCC3CCC23)C(=O)N(CC=C)C2CC2)cc(C(F)(F)F)ccc1Br C=C1CC2(C1)CC(C(=O)NCC1CC(OC)CN1C(=O)C(C)OC(C)(C)C)C2 c1(CC)cccc(C(=O)NCC2CCC2CNC(C2(C3CCC3)CC2)=O)c1N C1(CNC(C2CCCO2)=O)CN(C(c2cnc(S)[nH]2)=O)CC1C(F)(F)F C1(C(=O)NC(C(=O)OC)Cc2cccc(F)c2)CC2OC(=O)OC2C1 C(=O)(C#CC1(CC)COC1)NCC(CC=C)NC(=O)C(C)COC c1(C(c2n(CCCCCC)nnn2)NCC2CSCCS2)cc(C)cc(Cl)c1 CCCC(C)(CC)C(=O)NC(C)CCN(C)C(c1ccccc1NC(=O)NC)=O Cc1cc(CN(CC(C)(C)CO)C(c2cccc(F)c2C)=O)ccc1Cl CCC(CC(=O)N1CCC(C(=O)NCCCc2n[nH]c(C)n2)C1CC)CC(C)C C1(C(N2CCN(C(CCCCCC)=O)C(C)CC2)=O)C2Cc3cc(Cl)ccc3C12 C(C(C)(O)CC(=O)N1CC(CNC(c2cnn3c2OCC3)=O)CC1C)OC c1(C(C)NC2C(C)CC(C)OC2)ccc(Cl)c(Cl)c1Cl C(=O)(C1SCCc2sccc21)NC(C1(O)CN(C(=O)C2CCc3c[nH]nc32)C1)C C1(C(N2C(C(C)NC(C(C)(C3(C)CC3)OC)=O)CCC2)=O)CCc2nnnn2C1 Cn1cc2c(n1)CCC(C(=O)NCC1(NC(=O)CC3CCC4(CCC4)O3)CC1)C2 c1(C(N(C2CCN(S(=O)(=O)C3CC3)CC2)C)=O)cnn2c1CCCC2 CCC(F)(F)CC(=O)N1CCCC(C)(NC(=O)CC2CN(C)CC2O)C1 N1(C(C(C)N2CCC2)=O)CCCC1(C)CNC(c1cn(CC(F)F)cn1)=O C(=O)(C#CC(C)(C)C)NC(C(C)NC(=O)C(c1cnn(C)c1)O)(C)C N1(C(COCCOCCOC)=O)CC(NC(C2C=CCC2)=O)CC12CCOCC2 C(C(=O)NCC(C)=CC(=O)NC(c1cnn[nH]1)C1CC1)(C(C)C)SCC N1(C(c2c(C)cncn2)=O)CC(CCNC(=O)CC2CCN(C)C2=O)OC(C)C1 C(C(=O)NC1C(CNC(=O)OC)CCC1)(C(C)C)NC(C1CC2CCC2C1)=O c1(C(=O)NCC(CC)NC(=O)C2CC2)csc(C2CC2)n1 C1(NC2(c3nnnn3C3CCCCC3)CCSC2)CCN(NC(=O)OC)CC1 c1(C(C)C)ncc(C(N2CC(NC(c3cnco3)=O)C2)=O)[nH]1.C(CCOC)O N1(C(CCOC(CC(C)C)C)=O)CC2CC(NC(c3ccc(F)s3)=O)C(C2)C1 c1(SCC)cc(C(=O)NCC(C)CNC(C2C=CCC2)=O)ccn1 CC(CCC(C)(C)C)C(=O)N1CCC(C)C(NC(=O)CC2COC(=O)C2)C1 c1(C(=O)NCC2OCCN(C(C(CC)C(=O)OC)=O)C2)n[nH]c2cc(C)ccc12 N12CCCCC1C(C)(C)CC(=O)OC2=O.C1(C(C)O)CCCN1NC(C)(C)C c1(OC)ccc(C#N)c(C(F)(F)F)c1.c1(N2C(=O)N3C(CC3)C2)ncc(C)s1 N1(C(CCOCCCN(C(CN(C(C)=O)C)=O)CO)=O)CCCC(n2ccnn2)C1 N1(C(C(c2cccc(F)c2)C)=O)CCC(CNC(c2n[nH]c(=N)[nH]2)=O)C(C)C1 Cc1cc(F)cnc1C(=O)N(C)CCOCCCNC(C1CC(C)(O)C1)=O C=CC(CC)C(=O)N1CC(=C(CNC(C(c2cccnc2)N)=O)F)C1 C1(C(=O)C)CC2(CC2)CN1C.c1(C(=O)OC)ccon1.C12(CCC1)C(=O)NC2 c1(C(=O)NC2(CO)CCN(C(C3C(C)(C(F)(F)F)C3)=O)C2)coc2c1CCCC2 Cc1cc(C(=O)NC2CC(C)N(C(=O)Cn3cc(CO)nn3)C2)nnc1O c1(C2OCCN(Cc3c(C)csn3)C2)ccc(F)c(F)c1 N1(C(c2c(CC)noc2C)=O)CCC(NC(c2ncnc(OC)c2F)=O)C(F)C1 C(=O)(C1=CCC(C)CC1)N1CCC(CNC(C2(C(=O)NC)CC2)=O)C12CC2 c1(C(=O)NCC2C(N(C)C)CN(C(=O)C(O)C3CCC3)C2)n[nH]c2c1CCCC2 c1(C(C)N)ccc(Cl)cn1.c1(N2CCCNC2=O)cccc(Br)n1.CO N1(c2cc(CC)ncn2)CC2CCCC(NC(=O)CCCc3ccccc3)C2C1 C1(CNC(C2(C)CCN(C(C)=O)C2)=O)CCC2(CN(c3nnco3)C2)O1 c1(OCC(N2C(C(=O)NCC(=O)OCC)CCC2)=O)ccccc1Cl Cc1nsc2ncc(C(=O)NC3COCCC3NC(=O)C(C)C#N)cc12 c1(C(=O)OC)cnc(Cl)c(C(=O)NCC2CC2CNC(C23CC(CO2)C3)=O)c1 C#Cc1cc(C(C)N(CCC(=C)C)CC2CCCCCC2)cc(Br)c1 c1(C(=O)NCCOCCOCCNC(=O)C=CCO)c(Cl)cccc1Cl n12c3c(cc(cc3)c1=O)NC(=O)C2.C1(CC)(CO)CCCN(C(=O)C2=CCC2)C1 c1(CC2CCN(Cc3c(OC)cccn3)C2)ccc(F)c(Cl)c1 CC1(C(=O)N2CC3CC(NC(C4CC(F)(F)C4)=O)C2C3)CCOc2ccccc21 CC(C)(C)C(CNC(=O)COCC1CCCCO1)NC(=O)C=C1CCCC1 C(=O)(CCCC(=O)NCCOC)NC1CCN(C(C2C(OCC)C2C)=O)C1C C(=O)(C(O)CC(=O)NC1(C2CCCN2C(=O)C(C)c2cc[nH]n2)CC1)NC N1(C(CN(C(=O)COC)CC)=O)CCCC(CC)C1 Cc1cc(C)c(C(=O)NC2CCC(NC(C3CC3(F)Cl)=O)CC2)cn1 N1(CCCC)c2ccccc2CCC1C.c12c(cc(C(C)(C)C)cc1Cl)C(=O)N2 c1(NC(=O)NCC(C2(C)CC2)OCC)cc(Cc2ccccc2)sn1 N1(C(c2c(N)ccc(C)c2)=O)CCOC2(CCCN(C(c3ccc(F)o3)=O)C2)C1 N1(C(c2ccc(C)c(C)c2)=O)CCC2C1CCN2C(c1ccn(C)c1)=O C(CC1=CCN(C(C2CC(CC)(CC)C2)=O)CC1)NC(C1C(CC)C1)=O C1(S(N)(=O)=O)(C(=O)NCC2(C)CC(NC(c3c(C)csc3)=O)C2)CCC1 C1(NC(C=CCC2(NC(C(CCC)O)=O)CCC2)=O)CCOC(C)(CC)C1 c1(C(=O)NCC2C(NC(C(C)OCCC=C)=O)C2)ccc(P(C)(C)=O)o1 C1(C(=O)NC(C2N(C(C(C)OCC=C)=O)CCC2)C)Cc2nccnc2C1 N1(C(CCNS(CC)(=O)=O)=O)CCOCC(CNC(=O)C(C)C2CC2)C1 c1(C(N2CCOC(CNCC3(n4cccn4)CC3)C2)=O)ccnc([N+](=O)[O-])c1 Cc1cc(C)n(CC(=O)N(CCCCCCNC(=O)CC2CCSCC2)C)n1 c1(CNC=O)cc(C)ccc1F.c1(C(N(C)C)=O)cccc(C(=O)O)c1 N1(C(C2CC2NC(C2ON=C(CC)C2)=O)=O)CC2CN(C(C)=O)CC2C1 c1(C(=O)NC(COC)C)cn2c(n1)CN(Cc1ccc(C)nn1)CC2 C1(NC(CC2CC(C)(C)C2)=O)CC2CCC1(NC(=O)CCc1ccc[nH]1)C2 C1(CC(=O)N(CCCCC=C)C)CN(C(=O)C(O)CC(C)C)CCC1C c1(C(C)C)ccccc1OC(C1(C)CCN(C(=O)NC(C)(C)C)C1)=O C1(NC(=O)NCCCCC2CC2)C(CO)C2CCCCC12 c1(C(=O)NC(C(C(C)C)NC(=O)CCc2ncc(F)cn2)C)cnc2n1CCC2 c1(CC=C)nnc(Cn2cc(C3CCCN3C(c3cnoc3CC)=O)nn2)o1 CCCC(C(=O)N1CCCN(C(=O)C=C(C)c2cnn(C)c2)CC1CO)C(C)C c1(C(N(C2CCN(C(C3CCCC3OC)=O)C2)CC)=O)nc(=O)n(C)[nH]1 [N-]=[N+]=NC1CC(C(=O)NCC2=NOCC2)N(C(c2cnn(CCF)c2)=O)C1 C1(OC)(CNC(=O)C(F)=CC2CC2)CCN(C(=O)CC(N2CCCCC2=O)C)C1 C(=O)(C(C)CC(C)(C)C)N(CCCCN(C(COc1cncc(C)n1)=O)C)C c1(NCc2ccc(COC(C)=O)o2)ccc(O)c(F)c1.N12CCNCC1C2=O c1(NCC2(C)CCCC2(F)F)cccc(S(=O)(=O)NCC2CC3CCCCC23)n1 C1(C)(NC(C(CC=C)N(C)C)=O)CCC(NC(C2CCC(C)(C)C2)=O)CC1 N1(C(C2CC3CN(C(c4nc(CC)oc4)=O)CC2C3)=O)CC2(COC(C)(C)C2)C1 C1(C(=O)Nc2ccc(-c3cc(O)n[nH]3)cc2)Cc2cccc(F)c2O1 c1(C(=O)NCCC(C)NC(=O)C(=O)N(C)C)cnc(C(N)=O)cn1 C(=O)(CC(O)CC(C)(C)C)NCCN(C(Cc1c(C)cc(Cl)cc1)=O)C(C)C CCC(CC)C(F)C(=O)N(C(C)C(N1CCCC(C)C1CO)=O)C N1(C(c2n(C)ccc2)=O)CCC2(CCOC2)C(CNC(=O)Cc2ncc(Cl)s2)C1 C(C(=O)NOCC=CCl)(c1cn(C)nn1)NC(C1CCSC1)=O N(C1COc2ccc(Br)cc21)C(C(N1C(C)(C)CC(CO)C1)=O)=O CC(C)CC(C)(C)C(=O)NCC1C=CC(NC(=O)CC2SC(=N)NC2=O)C1 N1(C(CC=CCC)=O)CCN(C(=O)C(O)Cn2cncn2)C(CCOC)C1 c1(N(C)C)nc2c(C(=O)NCC#CCNC(=O)C(O)C3CC3)cccc2o1 S(=O)(=O)(c1c[nH]ccc1=NCCCCC1CCCC1)NC1C(C)N(C)CC1 c1(OC)cccc(F)c1CN1CCC(C)(NC(C2CCC2)=O)C1 C(c1nc2ccccc2[nH]1)=CC(=O)N(CCCNC(C1C2CC2C2CC12)=O)C c1(CCC(=O)NC2CCN(C(C(C)(CO)OC)=O)C2C2CC2)c(F)cccc1Cl c1(OC)c(F)cc(NC(C2CN(Cc3ccnc(Cl)c3Cl)CCO2)=O)cc1F c1(C(N2CC3CC(NC(C(COC)(F)F)=O)C3C2)=O)cc2c(cc1Cl)NC(=O)C2 c1(C(=O)NC(CC(C)C)Cn2cc(Cn3ccnc3)nn2)ccccc1C#N N1(C(C(C)(C)OC)=O)CCCC(CC(N)=O)(NC(C2COCC(C)(C)O2)=O)C1 CCCCCCCCNC(CC1(CN)CCN(C(=O)C=CBr)C1)=O C1(SCCn2c(C(C(CC)C)NCCC3(C)CC3)nnn2)CCCC12CC2 C1(C(N(CC(=O)NC2(COC)CC2)CCOC)=O)C2CCC(=O)C12 N1(C(CCN(C)CC)=O)CCC2(CC1)COC(CNC(c1n[nH]c(O)n1)=O)C2 c1(C(C(=O)NCc2cccs2)N(C2CCCC2)CC)nn(C)c(C2CC2)c1Cl NC1(C(=O)NC2CC3CCCCN3C2)CCCCCC1 C(=O)(C1CCCc2nncn21)N1CC(CNC(c2c(C(=O)OC)cncc2)=O)C1 N1(C(C2CCC(=CC)O2)=O)CCC(O)CC1C(N1CC(C=CC(C)(C)C)C1)=O C1(C2CCC2)(C(=O)OC)CCN(S(=O)(=O)Cc2ccc(Cl)c(Cl)c2)C1 CON1CC(C(=O)N(C)CC2(CNC(C3CCOC3C(F)(F)F)=O)CC2)CC1=O c1(SC)cc(Br)ccc1CNc1cc(N2CCC(F)CC2)ncn1 N1(C(CCCOC)=O)CC2CC(NC(c3c(C)ccc(Cl)c3F)=O)CC1C2 Cc1nsc(N)c1C(=O)NCC1N(C(=O)C(C)(C)CCl)CCC1 c1(C(=O)NCCCOCCNC(C=CSC)=O)cc2c(o1)C(C)(C)CCNC2=O C1(C(N2CCC(N(C)C(c3cnn(-c4nccs4)c3)=O)C2)=O)(CC)CCCC1 C1(O)(CNC(C(C2CCOCC2)OC)=O)CCCN(C(c2cc(OC)ns2)=O)C1 CC1CC2(CCCCC2)CN1CC(C1(CO)CCCCC1)O N1(C(c2ccn(CCC)n2)=O)CCCC2(CCCN2C(C2CC=CCO2)=O)C1 c1(C(N(C(C)C)CCN(C)C(C2(C)CC2F)=O)=O)cc2c(O)ccc(F)c2[nH]1 C(CCC(=O)N1CCC(CN(C(=O)CC2CC(C)(C)C2)C)C1)SC C1(NC(C2C(C)(C)OCCO2)=O)CCC2CCN(C(=O)C=CC3CC3)C12 C1(c2ccc(N(CC(C)O)C(C)C)s2)CCCCC1=O C1(CNC(c2c(OC)n[nH]c2)=O)C2CN(C(C)C)CC12.c12ncccc1O2 Cc1cc2n(n1)CCN2Cc1ncnn1C(C)(C)C c1(C(=O)NCC2CN(C(c3cccc[n+]3[O-])=O)CCCO2)ccc2cccnn12 c1(C(C(=O)NC2CC(C(=O)NCc3c(C)ncs3)C2)O)ccc(F)cc1 Cc1cc(C)n2nc(C(=O)Nc3ccc(C(F)(F)F)c(C)n3)cc2n1 NCCC(CC(=O)Nc1ccccc1)NC(=O)C(C1(O)CCCC1)O c12nc(C)c(Br)cc1S(=O)(=O)N2C.c1(COCC)ccccc1SC(C)C CC1(C)CC=C(C(=O)N2CC=CC2CNC(C2NC(=O)C3CCC23)=O)CC1 N1(CC)CCCN(C(=O)C=Cc2ccc(C)cc2)CC1.n12cc(nn1)C1CC1C2 N1(C(C(CC=C)CC)=O)CCC2C(C1)CN2C(c1cc(C(c2ccco2)=O)c[nH]1)=O N1(C(C(=O)NCC2(C(=O)NC)CCC2)=O)CCC(c2cnn(C)c2N)CC1 CCC(CC(=O)NC1C2CN(Cc3scnc3C)CC12)c1ccccc1 C1(C(N2CCC(NC(C3CC4CC4C3)=O)C2)=O)C2CCC1(c1ccc(O)cc1)C2 C1(S(C)(=O)=O)(C(N(CCN(C)C(c2cnn(CC(F)F)c2)=O)C)=O)CCOCC1 CC1(C)C(C(=O)NCCCN(C(N)=O)Cc2cccc(C#N)c2)CCS(=O)(=O)N1 c1(C2CC2)cnccc1C(=O)NC1CCC1NC(C1(SCC)CC1)=O C(=O)(CC1=CCOCC1)N1C(C2(NC(C(CCC)OC)=O)CC2)CCCC1 Cc1ccc(Cl)c(C(N2CCC(NC(=O)CSc3n[nH]c(O)n3)C(O)C2)=O)c1 c1(C(N2CCC(CN(C)C(c3cc(Cl)ns3)=O)C2)=O)ccc2c(c1)C(=O)C(=O)N2 N1(C(C(COC)(F)F)=O)CC2CC(CNC(=O)CN3CCSCC3)CC1C2 N1(Cc2nc(C)[nH]n2)CCC(N(C(=O)C2=CCCC2)C)CC1.C1CC(=O)N1 C(=O)(C1=NOC2(CCOC2)C1)NC(CCN(C(C)=O)C)C(C)C CCCCCCCCCCCCNC(C1(C)CCNC1=O)=O N1(C(C=CC=CCC)=O)CCCC1C=CC(N1CCOCC1C(C)C)=O CC1CCC(C(N2CC3C(CNC(C4(c5ccncc5)CC4)=O)C3C2)=O)CC1C c1(C(=O)NC2CC(C(C)NC(C3C(OC)CCC3)=O)C2)cccc2ncnn12 C(C(C)CC(=O)NC(c1ccccc1)CO)NC(c1c(CC)con1)=O C(CCCC(F)(F)F)Nc1cc(N2CCCC(CCC(=O)O)C2)ncn1 C=CCCCC(C)(C)C(=O)N1CC2(C1)CN(C(c1nccnc1SC)=O)C2 C1(C(=O)NC2CC(CCC(=O)NCC(C(C)C)(C)F)C2)CCC=CCCC1 C1(C(=O)NC2(CNC(COCCC)=O)CCC2)CCCN(CC(F)(F)F)NC1=O c1(C(N2CCC(CC(C)NC(C)=O)CC2)=O)cc(O)cc(C#N)c1 N1(C(c2ccc(CN(C)C)[nH]2)=O)CCC2C(C1)CN2C(c1cnc(C(F)F)s1)=O CC1CC2(CCN(C(=O)CN3CCOC3=O)CC2)CN1C(c1csc(Cl)c1)=O CCC(C(=O)N(CCN(C(=O)C(c1ccccc1Cl)OC)C)C(C)C)C(C)(F)F C1(NC(CN(C(=O)OCC)C)=O)CC(O)CN(C(=O)CCc2ccsc2)C1 N1(C(C=NC(=O)Cn2ncnn2)=O)CC(CCOCCOC(C)(C)C)C1 C12(NC(CCCOCCC)=O)CCCN(C(c3c[nH]c(=N)o3)=O)CC1C2 c1(CC)cnc(CCN(CCCCN(C)Cc2ccccc2)C)[nH]1 N1(C(c2ccc(COC)o2)=O)CCCN(C(=O)CC2CCCC2)C(C)C1 CC1CCCc2nc(C(=O)NCCNC(C3(C#N)CC34CCC4)=O)cn21 CC1CC(NC(c2cc[nH]c2)=O)CCN1C(c1cn(CC(F)(F)F)nn1)=O C1(NC(c2n(C)cnc2)=O)CCN(C(=O)CCc2cccnc2)CC1F c1(N(C)C(C2CCN2C(c2cscn2)=O)=O)ccccn1 C(C(C(=O)N=S(C)(=O)CCNC(=O)OC(C)(C)C)c1ccccc1)N(C)C Cn1nnc2c1CC(C(N1CCCC(c3cn(CC(F)(F)F)nn3)C1)=O)CC2 N1(C(C)=O)CCC(C(=O)NC(=O)COCCCCCC)CC1 CC1(C)C2CCC(NC(C3CCC4(CN(c5cc(O)nc(O)n5)C4)O3)=O)C1C2 C(=O)(C1CCCc2ccnn21)N1CC(NC(CNC(=O)NC2C(C)C2)=O)(CO)C1 C1(CNC(CC(=O)NC)=O)CCCN(C(c2cc3n(n2)CCO3)=O)CC1 C1(NC(CCOC2CN(C(C3N(C)CC(C)(C)C3)=O)C2)=O)CC2CCC(C1)N2C c1(C(=O)NCC(C)(CO)NC(C2CCC(=O)N2)=O)c[nH]c2ccc(F)cc2c1=O C1(CC(=O)N(CCOCCC)C)CCCN(C(c2cnn(C)c2)=O)CC1 C1(NC(Cc2cc(C(C)=O)[nH]c2)=O)CN(C(=O)CCc2ccn(C)n2)CC12CC2 C1(C(=O)NC2CCCN(C(c3c(C)occ3)=O)C2)C2CCC1(C)C2(C)C N1(C(C2(c3cc(C)on3)CC2)=O)C2CCC1CN(c1ncnc(C)c1C#N)CC2 N1(C(C(C)N(C)C)=O)CCC(N=[N+]=[N-])(C(N2CCC(c3nn[nH]n3)C2)=O)C1 C(=O)(C1COc2ccccc21)NC1CN(C(CN(C2CCC2)C)=O)CC2(C1)CC2 CC1OCC2(CCN(C(=O)CCc3n[nH]c(=N)s3)CC2)C1N1CCCC(O)C1 n1(CCNc2n(CC#C)c(N(CCC=C)C)nn2)cnc2ccccc12.C1CC1 c1(C(N2CC3C(CNC(c4ccc(C)cc4C)=O)C3C2)=O)c(N)cc(F)cc1F C1(CNC(c2cnc(C3CCCO3)s2)=O)CCC2(CN(C(=O)CO)C2)O1 c1(SCC)cnc(O)c(C(N2CCC(N(C)C(c3scnc3C(C)C)=O)C2)=O)c1 c1(C(=O)NCC(CO)NC(C2N(C(C)(C)C)CC2)=O)c[nH]nc1-c1ccco1 c1(C(N2CC(N(C)C(c3cnc(-c4ccco4)s3)=O)C2)=O)[nH]cc2c1CCCC2 C1(NC(C=CSC)=O)CN(C(=O)C(F)(F)Sc2ccc(F)cc2)CC1C C1(C(=O)NCC(CC#C)(C)C)CC12CCN(C(=O)CC1CCOC1=O)C2 N1(CC(=O)N(CCOCCNC(C2CC(=C)C2)=O)C(C)C)CC2CC2C1 Cc1ccc(CNC(=O)C(Cc2cn[nH]c2)N2CCC(CS(N)(=O)=O)C2)cc1 C#Cc1cnn(CC(=O)NC2CCCC2NC(=O)C(C2CCCCC2)O)c1 Cc1cc(NC(=O)C(F)OC(F)(F)F)ccc1NC(C1CC1CC(F)(F)F)=O CCC(CC)C(C)C(=O)N1CCCC1C1(NC(c2cc[nH]c2C2CC2)=O)CC1 CC1CCCC=C1C(=O)NC1C=CCN(C(C2CC(=O)C2C)=O)C1 c1(C(C(=O)NC(C)C(=O)NC(C)(C)C)NC(CC=CCC)=O)ccccc1 C1(C(=O)NC2(C3N(C(C(CC)CC)=O)CCCC3)CC2)CC12CC(F)(F)C2 C(=O)(C1=C(Cl)CCC1)N1CCC(CN(C)C(C2(C)CCCN2C)=O)C1 c1(CCC)cc(C(=O)NCC2CCCN(C(c3cn(C4CC4)cn3)=O)C2)n(C)n1 C(CCC(=O)N1CC(C(N)=O)(CNC(=O)C(C)NC(N)=O)C1)NC(C)=O CC(C)CCC(C(=O)N(C)Cc1cnn[nH]1)NC(=O)CC1CCOC1=O N1(C(CN(C)C)=O)CCC(C(N2CCC2CC2CC2)=O)(CO)C1 C=CC(C)(C)CC(=O)NCC1CN(C(c2cnccn2)=O)C2CC12 c1(C(N(CCCCNC(c2c[nH]cc(C)c2=O)=O)C)=O)n[nH]c2c1CCCC2 c1(CNC(CN(CCCNC(C2C(OC)COCC2)=O)C)=O)ccc(Cl)c(Cl)c1 Cc1cc(F)ccc1C(=O)NC1CC(C)N(C(=O)C(O)CC2CCCC2)C1 Cc1cc(=NCc2sc(C)cc2Br)[nH]c(=NCC2NCc3ccccc32)[nH]1 CCCCS(=O)(=O)N1CCCC1C(=O)NC1CC1C(=O)Nc1sccc1C(N)=O N1(C(C(c2n(CC)nnn2)C)=O)CCc2[nH]nc(O)c2C1 N1(C(=O)COC)CCN(C(C)CN(C(C(C=CCCC)O)=O)OCC(C)C)CC1.OC Cc1cccc(C(N(CCN(C(=O)C(O)CF)C2CCCC2)CC)=O)c1 C1(CC)C(NC(=O)CCc2ccoc2)CCCN1C(=O)CCn1cncn1 C=C1CCC(C(=O)NCC(C23CCC(CC2)C3)NC(=O)Cc2ccc(C)o2)CC1 N1(C(c2cncc(C(F)F)c2)=O)CCC2(CCNC2)CC1 N1(C(C(N2C(C)C(c3ccccc3)CCC2)=O)CN(C)C)CCc2sccc2C1 C1(NC(c2n(C(C)C)ccc2)=O)CC2CCC1N2C(=O)CCC1(C)CC1 C(C(C(C)(C)C)NC(=O)CCCSc1ccccc1)NC(CC1N(C)CCC1)=O N1(C(CNC2C(C)N(C)CCC2)=O)CCc2nc(-c3ccccc3)ncc2C1 C1(C(=O)NC23C(CN(C(C4CN(C(C)C)C4)=O)C2)C3)CCn2ccnc2C1 C1(NC(C#C)C(C)OC)C2CCC(C(=O)O)CC12 C1(CC)CN(C(c2cnn(C3CCCC3)c2C)=O)CCN1Cc1scnc1C c1(CN2C(C(=O)Nc3cncnc3Cl)CC(OC)C2)ccc(F)cc1O C1(NC(CN(C(C(C)C)=O)C)=O)CCC(NC(C2CCC3(CC3)C2)=O)CC1 c1(OCC(=O)N(CCCNC(=O)C(C)(C)C(N)=O)C)nn(C)cc1[N+](=O)[O-] N1(C(C2(C(=O)OC)C=CCC2)=O)CCCC2(CCCN2C(=O)C2=CCCSC2)C1 CC(C(=O)NC(C1CCCCC1)C(=O)NCCOCc1ccnn1C)S(C)(=O)=O c1(C(N(C2CCN(C(=O)C(F)CC3CC3)C2)CC)=O)cc(C(=O)OC)ccn1 C1(NC(CCCCN(C)C)=O)COC2C(NC(c3ncn(C)n3)=O)COC12 C1(OC)CC(CNC(=O)Cn2nnc(C3CC3)n2)N(C(=O)CCc2cn[nH]c2)C1 CCCC(C)CCCC(=O)N(CCNC(=O)CN1CCC(C)CC1)CC1CC1 n1(CC(N2C(CNC(C(C)SCC)=O)CC(C)CC2)=O)ncc2cc(C)cnc12 c1(CC2(C(=O)NC3(CF)CCN(C(CC(=O)OC)=O)C3)CC2)cccc([N+](=O)[O-])c1 C1(C)(C(=O)NCC(C)(C)CCNC(=O)CCc2cn[nH]c2)CCCCNC1=O Cc1ncc(C#N)cc1NC(C1CC(O)CCN1C(c1ccccc1CO)=O)=O C1(C(=O)NC(CC)C)COc2ccc(-c3cnn(C(C)C)c3)cc2C1 Cc1coc(C)c1C=CC(N1CC(C)N(C(=O)Cc2ccc(F)c(F)c2)CC1)=O N1(C(C=Cc2nc(C)sc2)=O)CC2CCC1C(NC(c1cccn(C)c1=O)=O)C2 C12(NC(C(C)OCCC=C)=O)CC3CCC(C1C2)N3C(=O)CSC(C)C c1(CC(C(=O)NC)NC(CC(=O)NCC(c2ccc(F)cc2)C)C)ccccc1Br C(CCN=C(NCc1cnco1)NC1CCC1)C1CCC(C(N)=O)O1 C1(NC(C2CCC(F)CC2)=O)CC2CC1CN(C(c1cn3ccccc3n1)=O)C2 C1(C(=O)OCC2CC3C=CC2C3)CC2(CCC(F)(F)CC2)CO1.O=c1c(=O)[nH]1 C1(C(N(C2(C(=O)OC)CC2)C)=O)CN(C(=O)COCCF)CC1(F)F C1(NC(C(CNC(C2CCCN2C2CC2)=O)N(C)C)=O)CC(O)C(O)C1 n1(CC)nc(C)c(C(=O)NCC(F)CNC(=O)CCC2(C)CC2)c1C c1(C(=O)OCC)cc(NC(N2CC3(CO)C(C2)CCO3)=O)cc(S(C)(=O)=O)c1 C(=O)(C(F)(F)C(C)(C)O)N1CCC(CCNC(C(COC)O)=O)(OC)C1 Cc1cnc(C(=O)NCCNC(C2CC(NS(=O)(=O)C(F)F)C2(C)C)=O)c(F)c1 C(=O)(C(CO)C(=O)OC(C)(C)C)N(C(C)CCNC(c1coc(C(=O)OC)n1)=O)C N1(CC(N2C(CN(C)C(c3cc(F)ccc3F)=O)CCC2)=O)C(=O)CCCC1=O CN1N=CC(CC(N2CCC(CNC(=O)C#CC(=O)O)CC2)=O)C1=O C1(NC(c2cc(C)ncc2)=O)CCOC12CCN(C(c1ccccc1)=O)CC2 C(CC(C)C)(C(=O)N1CCCC1CNC(C1CC2(C1)CC(O)C2)=O)NC(C)=O N1(C(C=C(CCC)CCC)=O)CCCC(NC(=O)C(C)(C)C2CC2)CC1 C(c1cnccc1C)=C(CC)C.C(C)(CN)(Cn1cccn1)NC(=O)CC1CCC1 c1(C(N2CC(C(=O)Nc3cc(C)c(O)cc3)OCC2)=O)ccc2c(c1)C(=O)OC2 c1(C(N2CC(NC(C3(C)COC3)=O)C(F)C2)=O)cc2cc(Cl)cnc2o1 Cc1ccc(SCC(N2CC(CC(C)NC(c3ccoc3Cl)=O)C2)=O)c(C)c1 c1(C(=O)NC2CCN(C(=O)CCSC)CCC2CO)cc(=O)c2ccccc2[nH]1 c1(COC)cccc(O)c1O.c12nc(sc1C)-c1cn(nn1)CC1CCN(C1)C2=O.O=C.N.C C(CN=c1cc[nH]cc1S(=O)(=O)N(CCCOC1CCOC1)C1CC1)c1cn(C)nc1 C1(CCC(=O)N(c2ccsc2)CC)CCCN(C(c2cscc2Cl)=O)C1 CCCC(C(O)C(=O)NC1CCCCC12CC2)NC(c1ccnnc1O)=O c1(C(=O)NCC2CCCCN(C(C3OCCO3)=O)C2)cc(O)nc2c1CCCC2 CC1CC2(CC(C(=O)NCC3(F)CC(NC(C45CSCC4C5(F)F)=O)C3)C2)C1 C1(C(=O)NC(CN(C(CNC(=O)OCC=C)=O)C)C)(CF)CC1(F)F c1(C(=O)NC2(CO)CC3CCC2C3)cnn2c1NCCC2 C(CC(=O)N(C(C)CO)CC)(C(C)OC)NC(c1cnc(CC)nc1)=O C1(CNC(C(C)OCCOC)=O)CC2(CC2)CN1C(=O)CCC1OCCO1 CCS(=O)CC(=O)NC(CNC(c1ccc(C(N)=O)[nH]1)=O)C(C)C C1(NC(C(C)OC)=O)C2CCCN(C(c3cncc(C4CC4)c3)=O)C2C1(C)C C1C(CC(=O)N2CCC(C3CCN(C)CC3)C2)OC1=O.C(C)(C)(C)OC c1(OC)cccc(C(N2CCC(F)(CNC(C3CCC3C(N)=O)=O)C2)=O)c1N C(CC(F)F)(C(=O)N1CC(C)(C)C1CO)N(C)C(c1ccn(CCF)n1)=O C=CC(C)CC(=O)NC(CCC1CCC1)C(=O)N1CCC1CC1CCCC1 C(CN=c1[nH]c(N2CCCCCCCCC2)nc2c1SCC2)c1ccn(C)n1 C(CC(O)CNC(c1ccsc1Cl)=O)NC(C1(C(=O)NC)CC1)=O C12(n3cc(C(C)OC)nn3)CCC(NC(=O)CC(=O)N(C)C)(CC1)C2 CCCC(O)CC(=O)NCC1CCCCCN1C(=O)CSCc1csc(=N)[nH]1 CCCC(C)(CC)C(=O)NCC1(C(N2CC(C3CCCOC3)C2)=O)CC2(CC2)C1 O(NC(=O)C(CNC(=O)C(C1CCOCC1)O)C(C)C)C(CCOC)C1CC1 N1(C(C=CC(=O)NC)=O)CCN(C(C2CCCCC2OC)=O)C(CC(F)(F)F)C1 CCCC(C(=O)N(CC)CC1CCCN1C(=O)CNC(C)=O)OC C1(NC(C2C(CC)CCCN2C(=O)Cc2csnn2)=O)CC(C)(C)OC1=O Cc1ccccc1CC(=O)Nc1ccc(C(=O)NCCCCO)nc1 C12(C(N(CC(C)(C)C)CC#C)=O)COCC1CN(C(=O)C(SC)SC)C2 C1(C(C)C)CN(C(c2cc(Cl)no2)=O)CCN1C(=O)CCc1cnn(C)c1 c1(C(=O)NCC(C)NC(=O)CCC2CCC(=O)NC2)cn2cc[nH]c(=O)c2n1 c1(C(N(C)CCN(C)C(C2CC23CCCCC3)=O)=O)cnc2ccoc2c1 C(=O)(CCC(C)S(C)(=O)=O)N(CCNC(C1(COC)CCCCO1)=O)C1CC1 Cc1cc(C(N2CCN(c3ncncc3C#N)CC2)=O)cc(C)c1O C(=O)(C(C)(C)C(=O)N1CCCCC1CNC(=O)COc1cc(C)ccc1F)OC c1(CNC(C2N(C=O)CCC2)=O)nc2c(s1)CN(C(=O)CC1CC1)CC2 c1(C(N2CC3C(NC(C4(C)C(C)(C)C4)=O)C3C2)=O)cnc(O)n(C2CC2)c1=O O(NC(=O)C(C)(C1CCC1)NC(c1cc(C(N)=O)c[nH]1)=O)C(C)(C)C C1(CC(=O)N(C2CC(NC(=O)CN3C(=O)CNC3=O)C2)C)CC2(CCC2)C1 C1(C(=O)NCC(=C)CCNC(=O)CC2(O)CCCCC2)CCN(C)C(=O)C1 c1(CC)cccc(F)c1C(=O)NC1CCN(C(c2cnc(C)nc2)=O)CC1O c1(C(N(C2CCCN(C(c3oncc3C)=O)C2)CC)=O)cccc2c1SCCC2 C(CN=c1[nH]c(=NCCc2c[nH]nc2O)[nH]c2c1COC2)c1cccc(F)n1 CC1OC2(CO)CC1(C(N1CCC(F)(CNC(c3cc(Cl)c[nH]3)=O)C1)=O)C2 C1(NC(CC2CN(C(c3n(CC#C)cnn3)=O)CC23CC3)=O)CCn2nnnc2C1 c1(N2CC(CNC(CC(CCOC)(C)C)=O)OCC2)cc2c(cn1)C(=O)CCC2 C1(CCC(=O)N(CC(CCC)OC)CC)CCCN(C(c2ccncc2N)=O)C1 C1(C)(CNC(C(CSCC)NC(c2ccco2)=O)=O)C=CCCC1 c1(C(=O)NCC2C3CN(C(COc4cccc(OC)c4)=O)CC32)cnc(O)c(C)c1 C1(NC(=O)Cc2cc(Br)cs2)CCCC(NC(c2cc(C(F)F)no2)=O)C1 N1(C(C(C)SCc2ccccn2)=O)CCC2(CCCN2c2nc(Cl)c(C#N)s2)C1 C(=O)(C(C)C(O)C(C)C)NC(CC(=O)NC(CSC)CO)C1CC1 c1(NC(=O)NCC2C(P(C)(C)=O)C2)ccc2cnn(-c3ccc(F)cc3)c2c1 C1(OC(C(c2ccc(Cl)cc2)C)=O)CCCCC1CC(N1CCOCC1)=O CN1CCCN(C(c2cc(-c3ccc(O)cc3)on2)=O)c2cc(F)ccc21 n1(CC)ncc([N+](=O)[O-])c1C(=O)NCCC(C)(C)NC(C1C2COCC12)=O C(=O)(CC(CN(C)C)C(F)F)Nc1cccc(NC(C=C(C)C(C)C)=O)c1 C1(NC(C=CCC)=O)CCN(Cc2ccc(CCCCCC)s2)CC1O C1(NC(c2n(CCOC)nnn2)CCSC)C(=O)NCCC1C C1(CN(C(C2C(COC)C2)=O)C)CN(C(=O)CCNc2ccccn2)CCO1 c1(C(C)(C)C)ccc(CNC(=O)NC2COCCN2CC(F)F)nc1 c1(C(N(CCCN(C(c2nnc(C)s2)=O)C)C)=O)cc(S(N)(=O)=O)c(C)s1 Cc1c(F)cccc1S(=O)(=O)N1CC2CC2(C(N2CCCC(CO)C2)=O)C1 N1(C(c2cnc(SC)[nH]2)=O)CCOCC1CN(C(=O)CCc1ccc(F)cc1)C N12CCOC(C1=O)C2.Cc1n[nH]c(C)c1-c1cn(CC(N2CCC(O)CC2)=O)nn1 N1(C(c2ccc(C)c(C)c2O)=O)CC2CN(C(c3cc[nH]c3)=O)CCC2(CO)C1 N1(C(C(C(C)NC(CC=CC=C)=O)C)=O)CC2(CCC1CO)CC2 N1(C(C2ON=C(C)C2)=O)C(C)C2CC1C2CNC(=O)CCN(S(C)(=O)=O)C C(CC(O)CNC(C1CC(N2CC(O)C2)C1)=O)NC(=O)CNC(=O)C1CC1 c1(C(N(CC(C)NC(CC2(C(=O)OC)CCC2)=O)CC)=O)cc2ccncc2s1 N1(C(c2c(N)ccc(Cl)n2)=O)CCC2(CCCN2C(C2CCC3(CCC3)C2)=O)C1 c1(COC)nccc(C(N2CC(NC(=O)C(C)(C)C3CCC3)CC2CO)=O)n1 c1(C(N2CCC(Br)C2)=O)ccccc1Cc1noc(-c2cnccn2)n1 c1(NC(C2C(NC(c3ccc(C)c(Br)c3)=O)C2)=O)cc(Cl)c(O)c(Cl)c1 C(=O)(CC(C)(O)COC)N1C(C(=O)NC(C(=O)N(C)CC)C)CC1 Cc1ccn2ncc(C(N3CCCC3(C)CNC(=O)C(=O)NCC(F)F)=O)c2c1 c1(C(N2C(CNC(c3nsnc3O)=O)CC(O)C2)=O)ccnc2cc[nH]c12 CC(C(=O)N1CCCCC(C(=O)NCC2CN(S(C)(=O)=O)C2)C1)C(C)(C)C C1(OC(c2cn(CCOC)nc2)=O)CCOC2(CCOCC2)C1 CC1(C(=O)NCC2(F)CC(NC(=O)CCCc3cc[nH]n3)C2)CCCCO1 C1(c2ccccc2)(CN2CC3CCC2CC3)CC2CCC(C1)N2 c1(CCOC(c2cnnc(C3CC3)c2)=O)ccc(F)cn1 CC1(C)CCC(n2cc(C3COCC3O)nn2)CN1C(=O)C(=O)C(F)(F)F C1(COC)CC12CCN(C(C(=O)NCC1CCOC1)C(C)C1CC1)CC2 C1(C)(C(=O)NCC2(F)CCC(NC(C(CCOC)C)=O)C2)C(C)(C)C1(C)C c1(C(C)C)nc(C(=O)NC(C)(CNC(c2ccoc2)=O)CO)co1 C12(C(=O)NCC3N(C(c4sccc4Cl)=O)CC3)CC=CC(C1)OC2 CCC(F)(F)C(=O)NC(CC(=O)NCCN1CCC1)C1CC1 c1(NC(c2onc(C)n2)C2CCCC2)cc(N2CCC(SC(F)F)C2)ncn1 CN1CCOC(C(=O)NCC2(C)CCCN2C(c2ccc(Br)cc2)=O)C1 N1(c2nc(OC)nc(C)c2)CC2CCC1C1CN(C(=O)C3=CS(=O)CCC3)CC21 C(c1cccnc1)=C(C(=O)NC1CC(CNC(c2c(OC)csc2)=O)C1)C#N c1(C(C(=O)NC(c2ccccc2Br)C)N(C2CC2)CC)cc(C#N)n(C)c1 N1(C(=O)C2=C(Cl)CC2)CCC2CCN(C(=O)Cc3csc(Br)c3)C2C1 Cc1cccc(SC(C)C(N2CCC(CF)(NC(c3cccnc3)=O)C2)=O)c1 Cc1cc(C(=O)NCCOCCCN(C(=O)CSCc2cc(C)[nH]n2)C)ncn1 c1(C2N(C3C4(CC(CS(=O)(=O)NC)C4)C3)CCC2)nc2ccccc2[nH]1 N1(C(C(CC(=C)C)C)=O)CC2CC(N=c3cc(C)[nH]c(C)c3C(=O)OC)C(C2)C1 CCC(C)(C)CC(=O)N(C)CCNC(C1CCOC(c2ccc(F)cc2)C1)=O Cc1ccc(C(=O)NCC(c2cccc(O)c2)O)c(O)c1 c1(C(N(C(C(=O)Nc2ccc(OC)cc2)C)C)=O)cc(=O)cc(Cl)[nH]1 Cn1nnc(CNC(C2CCS(=O)CC2)=O)c1C(=O)NCCCSC c1(C(=O)OC(C)(C)C)ccccc1OC1CC(NC(C(CC)NC(=O)OC)=O)C1 S(=O)(=O)(c1c(C)ccc2ccccc12)N(CC(CCCC)CC)C C(=O)(C1=CS(=O)(=O)CCC1)NC1CN(C(C(C)Cc2cnn(C)c2)=O)CC(O)C1 N1(C(Cc2cnn(C)n2)=O)C2CCC1CN(C(=O)CC1CCOC(C)(C)C1)C2 c1(NC2CCCCN(C(=O)COc3ccc(Cl)cn3)C2)ccccc1[N+](=O)[O-] C(CC(C(=O)NCC(C)(O)CCO)NC(c1cc(OC)no1)=O)=CC N1(C(C2(C#C)CC(=O)C2)=O)CC2CCC(CNC(=O)C(F)(F)COC)(C2)C1 C1(NC(CC=C)=O)(CNC(c2sc(-c3cccc(F)c3)nc2C)=O)CCOCC1 c1(SC)cc(F)ccc1C(=O)NCCC1COCCN1C(C1CC1C(F)(F)F)=O C1(C(=O)NCc2c(CNC(C3CCCC3)=O)cccc2)CC2(CCCC2)CO1 N1(C(c2nnc3ccccc3n2)=O)CCC2(C1)CN(C(c1cccs1)=O)CCO2 C(=O)(CC(C(F)(F)F)NC(=O)CCC1CCN(Cc2cccc(F)c2C)C1)OC c1(C(=O)NCC2C(NC(CC(=C=C)C)=O)C2)ccc2cccc(O)c2c1 c1(C(N(CC(CN(C)C(c2ccoc2)=O)O)C)=O)coc(C2CCOCC2)n1 C12(NC(CC3C(OCC)COCC3)=O)CCCN(C(c3ccno3)=O)CC1C2 N1(C(c2cn(C)nc2Cl)=O)CC2CC3CC2C1C3NC(=O)CCCn1cncn1 C1(NC(c2n(C)cc(Cl)c2)=O)CC1C1CCCN(C(C2CC3C(C2)C3(C)C)=O)C1 N1(C(CSc2ccc(C)cc2)=O)CC(CN)C2(C1)CN(C(C13CC1C3)=O)C2.CO C1(N(C(C(C)NC(CC)=O)=O)C)CN(C(c2occc2C)=O)CC1(C)C C1(F)(CNC(=O)CCc2nnc(S)nc2O)CCN(C(c2cnc[nH]2)=O)CC1 c1(C(=O)NC(C2CC(NC(C3C(CC)OCC3)=O)C2)C)c(C)[nH]c2ncccc12 C1(CNC(Cc2nc(C)[nH]n2)=O)CC2CCC1N2C(C1CCCCC1O)=O C1(OC)CCC2C(NC(=O)OC(C)(C)C)CCC1N2N1CCCC(C)=C(C)C1 N1(C(C(C)(F)F)=O)CCCCC1CNC(c1ccn(Cc2ccccc2)c1)=O c1(C(N2CC(CNC(CCSC)=O)OCC2)=O)cnn2c1NCC(C)C2 CCCS(=O)(=O)C(C)C(=O)N1CCCC(N(C)C(c2cc(CC)sn2)=O)CC1 C1(C(N(CCN(C(c2c(C(C)C)c[nH]n2)=O)C)C(C)C)=O)CCCOC1C c1(C(C)C)cc(C(N2CC(NC(c3ccc[nH]3)=O)C(O)C2)=O)sc1-c1ccccc1 c1(C(N2CC(OC)C(NC(C3(CC(F)F)CCC3)=O)C2)=O)nccc(N)c1Cl c1(C(N2C(CNC(C3(CC)COC3)=O)COCC2)=O)cc(Cl)c(Cl)n1C c1(OC)cnc(Cl)cc1C(N1CC(NC(=O)Cc2cncc(F)c2)CC1C)=O N1(C(c2c(C)oc(Cl)n2)=O)CC(=O)N2CCOCC2(CNC(C2CCO2)=O)C1 CC1CCN(C(=O)CN2CCC(OC(=O)CCC(C)(F)F)C2)CC(C)O1 C(=O)(CN1C(=O)Cc2ccccc21)N1C2CC(NC(CSC(=N)N)=O)(C2)C1 CC1CN(S(=O)(=O)Cc2ccc3c(c2)OCO3)CCc2ccc(O)cc21 C1(C(N(CCCO)C)=O)COC2(CCN(C(=O)C=CC(F)F)CC2)C1 c1(CNC(C(COC)NC(C2CCCC2O)=O)=O)cccc(F)n1 c12cccc(c1)OC(C)C(=O)N2.c1(CC)cc(CC(=O)OCCN(C)C)on1 C1(CC(=O)NC(C#C)CC2CCC2)CN(C(c2cc(C)c(C)o2)=O)C(C)(C)C1 CC1NC(=O)CCC1NC(=O)CC1C(C)CCN1C(c1ccc(Cl)cc1)=O C1(C)(CC)CC(NC(c2ccc(Cl)o2)=O)CN1C(=O)CC(C)(C)COC N1(c2nc(SC)nc(C)c2)CCC2(CCCN(C(c3ccncc3N)=O)C2)C1 CCCCC(CNC(=O)C(C)(C)c1ccns1)NC(=O)CCC1CCCOC1 c1(OC)cc(C(=O)NCC2CC2CNC(c2c(C)non2)=O)n(C)n1 N1(C(C=NOC)=O)CCCCCC1C(N1CCC(O)(CN(C)C)CC1)=O c1(CC(C)C)cc(C(N2CC(O)(C(C)NC(=O)C(C)N(C)C)C2)=O)n(C)n1 c1(C(=O)NC(C(=O)NC(C)Cc2cccs2)C(C)O)ccnc(O)c1F C#CC(CNC(=O)CC1CCCN1C(=O)CN1CCCC1=O)CC(C)(C)C C1(c2nc(COC)sc2)CCS(=O)(=O)C1.C1CCCOC(=O)C12CC2 c1(C(N)=O)ccc(F)c(C(N2CCN(C(=O)CC3CCCOC3)CC2)=O)c1 C1(C(=O)NC2C(C)CN(C(c3ccc(=O)oc3)=O)C2)CCC(C)(C)CO1 N12CCC(C1)C(=O)N(C)CC1(CC1)C2=O.C1(CC(=O)NC)CN(C)C1.CCO Cc1cccc(OCC(=O)NC2(CCNC(C3CC4CC4C3)=O)CCC2)c1 C1(CC)CCCN(C(c2cc(C)[nH]c2C)=O)C1C(=O)NCCN(C)C(N)=O CC(c1cnn(C)c1)=CC(N1CC(CNC(c2cnc3sccn23)=O)C(O)C1)=O C(C(CCCOC)NC(=O)NC(C)(C)C)OCC=C.C(C(C)C)NC c1(C(N2CCCC(N(C(C(C)SCCCC)=O)CC)C2)=O)c(C)ccnc1C C(C(C(=O)NC1CN(C(=O)C(C)(O)C2CCC2)CC12CCC2)C(F)(F)F)OC CCC(C)(C)CC(c1nnnn1C1(C)CC1)Nc1ccc(F)c(Br)c1 CC(C)(C#CC(=O)N1CCCC(O)(C(N)=O)C1)CNC(=O)CC1CCCC(=O)C1 N1(C(C(C)N(C(C)=O)C)=O)CC2(CCN(C(C3CCN(C)C(=O)C3)=O)C2)C1 Cc1ccc(NCC(=O)NCCOCCN(C(C)C(=O)N(C)C)C)cc1 N1(C(CC=CC=C)=O)CCC(CNC(c2ccc(-c3nc[nH]n3)cc2)=O)C(C)C1 N1(C(C=Cc2cn(C)nc2)=O)CCCC2C1CCN2C(c1nocc1Br)=O C1(NC(C(CC)SC)=O)C(C)(C)CN(C(C2(OC)CCS(=O)(=O)C2)=O)CC1(C)C Cn1cc(C(N)=O)cc1C(=O)NCC1CCCN(C(=O)Cn2cnc(=N)[nH]2)C1 C1(NC(=O)C#CC2CC2)CC2CC1CN2C(c1cc2[nH]ccc2s1)=O c1(NC)cc(Cl)ccc1C(N1CC(CNC(c2scnc2C(C)C)=O)C(O)C1)=O N1(C(COCCCC)=O)CCC(C)(C)C1CC(=O)N(C(COCC)CC)C C1(C)(C(=O)NC2(CN(C(c3c(OC)c(C)ccc3)=O)C)CC2)CC(C2CC2)=NO1 CC(CN(C)C)CCC(=O)N(C)CCC1CCCCN1C(c1cnn[nH]1)=O CC1(C)CN(C(c2ccoc2Cl)=O)CCC1C(=O)NC1CC(C(F)(F)F)C1 c1(SCCC(=O)NC(C23CCC(CC2)C3)=O)ccc2ncccc2c1 c1(NC(c2c(SC)scc2)=O)cccc(NC(C2CC23CCCC3)=O)c1 C#CC1CN(C(=O)CCCCNC(=O)CC2CCCCC2O)CC1O C1(N(C(C)CO)C(c2ccccc2)=O)CCCN(Cc2cccc(Cl)c2Br)CC1 c1(C(=O)NCC2(NC(c3ccnc(C)n3)=O)CCCC2)c(C)nn(C)c1C N1(C(C#CC(C)(C)C)=O)CCc2[nH]nc(CNC(C3CC3F)=O)c2C1 Cc1cc(Cl)c(C(N2CC(NC(C3(C)CC(C#N)C3)=O)CCC2C)=O)cc1F N1(CCOCC=CC(N2CCC2(C)CC=O)=O)CCCC1(C)CN(C)C.CO c1(NC(CC=C)=O)ccc(NC(=O)C(C)Cc2cccc(F)c2)c(C)c1 c1(CNC(CN(C(=O)CCn2cnnn2)CC#C)=O)cnc(C(C)C)[nH]1 CC1(C)CC(NC(=O)C2=CSCCO2)CN1C(=O)CCCN1CCOCC1 N12CCC(O)(C1)C2=O.CCCC(C)N(CC(N)=O)C(=O)CC1CC=CC1 C=C1CCC(C(=O)NCc2occc2C(=O)NC(C)(CO)C(C)C)CC1 c1(C(N2C(CCNC(C(=O)NC(C)C)=O)CCC2)=O)cccc(C(F)(F)F)c1 C1(NC(c2c(C)nc(C3CCCOC3)s2)=O)CNCCS(=O)(=O)C1 C1(C(=O)NC2(CC=C)CCN(C(=O)C=CCN3CCCC3)C2)CCC2(CC1)N=N2 c1(C(C(N2CC3(CCN(C(CSC(C)C)=O)C3)C2)=O)C)ccc([N+](=O)[O-])cc1F CC1CCC(NC(=O)CCC2NC(=O)NC2=O)CN1C(=O)C(Cl)=CCl c1(C(=O)NC(C(C)C)CNC(c2cncc(C(=O)N(C)C)c2)=O)cc(=N)[nH]c(=N)[nH]1 Cc1cc(F)ncc1C(=O)NCCC1CCN(CC(C)O)CC1 N1(C(=O)NC)CCCC(CCCC(=O)NC2(C(=O)N(C)CCn3cncn3)CC2)C1 CC(CCC(=O)N(CC(C)C(=O)NCc1ccccn1)C)N1CCCCC1 C(=O)(CS(=O)(=O)C1CCCC1)N1CC(CNC(c2ncc(Cl)cc2O)=O)C1 Cc1nnc2n1CCN(C(C1CC=CCN1C(=O)COC1CCCC1)=O)C2 C1(C(N(CC(CO)(CO)NC(CCC=C)=O)C)=O)CCn2c(O)nnc2C1 N1(C(c2c(CC)nn[nH]2)=O)CCOCC12COCCN(C(C1CC(C)(C)C1)=O)C2 FC(F)(F)CC(CN)Cc1noc(-c2ccc(Cl)c(Cl)c2)n1 N1(C(Cn2cc(C(C)O)nn2)=O)CCCN(C(c2cn(C)nn2)=O)CC1 c1(C(=O)NC2C(CNC(C(CC)CC)=O)COC2)ccc(F)c(C)c1 C1(C(C(=O)OCC)NCc2cnc(-c3cccs3)s2)CC=CCC1 CC(C)C(CNC(=O)Cc1cc[nH]c1)NC(C1CC1c1ccccc1)=O Cc1nc2cc(C(=O)NCC3CCC(NC(=O)C4=NNC(=O)C4)C3)cnc2[nH]1 c1(C(=O)NCC2C(NC(C(CC#C)O)=O)CC2)cc(Cl)ccc1[N+](=O)[O-] c1(CC)ccc(F)cc1CC(=O)NCCCOCCNC(C)=O C1(CNC(c2c(C(C)C)[nH]cc2)=O)CCCCC1NC(c1c[nH]nc1F)=O c1(CN2C(CNC(c3cnon3)=O)C=CC2)ccc(OC(F)(F)F)cc1Cl N1(C(C2(CC#C)CCCCO2)=O)CCCC(C2CCN(C(=O)C(C)=C(C)C)C2)C1 c1(CN(C)C(=O)NCCC2CCC3(CC2)COC3)ccc2occc2c1 CC1CC(CO)(C(=O)NCC2CCCCC2O)c2ccccc2O1 c1(NC(C2N(Cc3cccc(OC)c3F)CCC2)=O)nc(O)c([N+](=O)[O-])c(O)n1 Cc1c(C(=O)NCC#CCNC(C2C=CC=CC=C2)=O)sc(Cl)c1Cl Cc1ccc(F)c(Br)c1C(=O)NCCN(C(=O)Cc1ccon1)CCOCCO Nc1cccc(C(N2CCOCC(NC(C3CC3C3CCCC3)=O)C2)=O)c1O Nc1cncc(C(N2CCCCC2CCNC(=O)C(F)(F)c2cccnc2)=O)n1 N1(C(C(C)O)=O)CC=C(C(=O)NCC(C)OCCF)CC1 N1(C(Cc2ccc(CC(C)C)cc2)=O)CCC2(CC1)CC2NC(c1ccco1)=O c1(C(=O)NC2C(CNC(C(C)(C)CC3CC3)=O)CCC2)ccc2nnn(O)c2c1 CC#CCCCC(=O)NC(CC)CC(N1CCN(CC)C(=O)C1)=O N1(C(C2C(C)OCC2)=O)CC(NC(=O)CC2CC(C(N)=O)C2)CC12CCC2 C12COCCC1N(CCC)C(=O)C(C)OCc1cn(nn1)C2.C(C(=O)NC)OC.CCC c1(OC)cnc(C(N2CCC(N(C(C3CCCCS3)=O)CC3CC3)C2)=O)cn1 c1(NC(C2CCN(C3CCN(C(CC=C=C)=O)CC3)C2)=O)ccn2cncc2c1 C(C(=O)Nc1cccc(C(=O)C(F)(F)F)c1)(C(F)(F)F)(c1ccccc1)OCC CC1CN(C(c2ncc(C3CC3)s2)=O)CCC1NC(c1ccnc(N(C)C)c1)=O C1(NC(C(COC)N(C)C)=O)(CNC(=O)CCN2CCOC2=O)CCCCC1C Cc1c(C(=O)NC2CN(C(c3ccc(C4CC4)o3)=O)CC2C)ccn1C1CC1 C(=O)(CCCCCC(C)C)N1CC(CN(C(COCCC=C)=O)C)OCC1 C(=O)(C(F)(F)C(F)F)N1C2C(C(N(C3(C#C)CC3)C)=O)C(C2)C1 CCCC(C(=O)NC1CN(C(c2c(C)ccnc2C)=O)CC1O)S(N)(=O)=O c12ccn(c1)CCNC2=O.C(=O)(CCCc1cnn[nH]1)N(C)CC1(F)CCC1 C(=O)(C(O)CC(F)(F)F)N(C)CC1COCCN1C(=O)CC1CCC(C)(C)CO1 c1(C(=O)OC(=O)C(C)(C)C)ccc(NC(=O)NCC=C)cc1 n1(CC)cc(C(N2CC3(CC3C(=O)Nc3ncccc3Cl)C2)=O)c(C(F)(F)F)n1 c1(C(N(C2CCN(C(=O)C(C)C(C)(F)F)C2)CCC)=O)cc(C)sc1S(N)(=O)=O CCC(COC)(CC)C(=O)NC(CNC(c1c(SC)cnn1C)=O)C1CC1 N1(C(C(C=C)O)=O)CCN(C2CCN(C(=O)CCC3CCC3)C2)CC1 C1(C(F)F)CCCCCN1c1nc(-c2ccccn2)cs1 N1(C(C2(CC#C)CC2)=O)CC2=C(C1)CN(C(c1cc(F)ccc1C)=O)C2 CCN(OC)C(=O)CNC(=O)CC1(CNC(=O)C(C)n2ccnc2)CC1 O=C(C1=COCC1)N1CCCC(CCCC(=O)N2CCC(c3nc[nH]n3)C2)C1 C(=O)(C(C)(F)C(=O)NC(CNC(c1ccc(OC)nn1)=O)C1CCC1)OC N1(C(C(N2CCC(CNC(C(c3cccc(Cl)c3)C)=O)C2)=O)=O)CCCC(C)C1 C1(CCNC(CCOCCOCC)=O)CN(C(c2occc2F)=O)CC1C N1(c2ncnc3scc(C)c32)CC2CCC(NC(=O)CC3CCOC3)CC2C1 Cc1ccc(C(=O)N(C)C(c2ccccc2)C)c(-c2ccccc2C)c1 c1(C(N2CCN(c3ncc(Cl)s3)CC2)=O)cncnc1-c1ccccc1 CCC(CC(=O)N(CC(C)(C)CNC(c1[nH]c(C)cc1C)=O)CC)SC CC(=O)CC(C)(C)C(=O)N1CC2CCC(NC(c3ccc(C)cc3O)=O)C2C1 c1(CC(=O)NCC(CNC(C(C=CC)O)=O)C)ccc(Cl)c(Cl)c1C C12(C(N(CC(=O)NC(C)C(C)(C)CN(C)C)C3CC3)=O)CCCN(CC1)C2 C1(C(=O)NC2CC(O)(c3ccccc3)C2)C2Cc3c(Br)cccc3C12 c1(C(=O)NCCC23CCC2CN(C(=O)C(F)F)C3)cnc2[nH]c(O)nc2c1 c1(C(=O)OC)cc(CN2C(C(=O)Nc3cnnc(Cl)c3)CC3CC23)ccn1 C1(C(=O)NC(CC(=O)OC)(C)C)CN(C(=O)CC2(C)CCOCC2)C2(CCC2)C1 N1(C(C=C(C)C)=O)CCOCC1C(=O)NCCC(C)C.CCOC(C)=O CN1CC2CN(C(=O)C(=O)NCCC3CCCC3O)CC2C1 c1(-c2scc(C)n2)ccc(C(=O)NC2CC(NC(=O)C(C)(C)N(C)C)C2)cc1 c1(CN2CCCC(NC(c3cc(O)ccc3Br)=O)C2)ccc(F)c(CO)c1 C(=O)(C1=NOC(C(C)(C)C)C1)NCC1(NC(C2C3CC(=O)CC23)=O)C(C)(C)C1 C1(C(=O)NCC2(C(N)=O)CN(C(CCCCOC)=O)C2)CCn2nncc2C1 Cc1noc(C)c1C(C)(C)C(=O)N1CCCC1CNC(=O)CNC(=O)C(F)(F)F c1(C(=O)NCC(C)(C)NC(C(CC)SC)=O)cnc2c(C)cccn12 c1(C(=O)NCC(CCCC)NC(=O)CNc2ccc(F)cc2)cccc(F)c1F C(=O)(C1=CCCCCC1)NCC1(C(C)NC(c2c(C)nc(C(C)C)o2)=O)CC1 c1(C(=O)NCCC(C)NC(c2c(CC)ocn2)=O)cnc(OC)c(C(F)(F)F)c1 c1(CNC(C23CC(NC(C=C(C)C)=O)(C2)C3)=O)ccc(N(C)C)c(Br)c1 c1(C(=O)NC(CN(C(C(C(=C)Cl)(C)C)=O)C)CC)ccc(OC)c(N)c1F C(=O)(CC1=CCCCC1)NCC(C)N(C(C1CC2(C1)CC(F)C2)=O)CC N1(C(CC2(COC)CC2)=O)CC(C2CC2)(C(=O)NCC2CCC(=O)N2)C1 N1(C(C2CCC(C)C2)=O)CCCC(C2CCCN2CCNc2ccc(Cl)cn2)C1 c1(C(N(C2C(O)CCN(C(Cc3cc(C)on3)=O)C2)C)=O)c(C)cc(Cl)cc1C C1(NC(c2c(NC)scn2)=O)CCCCN(C(c2cnc(C)nc2C)=O)CC1 c1(C(=O)NC2C(CC)N(C(C3CSCC(=O)N3)=O)CC2)cc(F)c(O)c(Cl)c1 O=C1NCCN2CCN(c3nnc(-c4cc5cc(Br)sc5[nH]4)n3C)CC12 CCCCCC(F)C(=O)NCC1CCC(C)CN1C(c1ccn(C)c1)=O N1(C(C(C)NC(C)(C)C)=O)CCC2(CC1)CCN(C(c1cccc(F)c1F)=O)C2 C1(CC)COCCN(C(C2(COC)CCOCC2)=O)C1.C(CCC(N)=O)N Cc1coc(C(C)(C)C)c1C(=O)N(C)CC1CCN(C(=O)CCC=CBr)C1 C12(NC(c3cnc[nH]3)=O)CCN(C(=O)Cc3nc(F)c(F)cc3F)CCC1C2 N1(C(c2c(CC)nco2)=O)CC(NC(=O)CC(c2cccc(Cl)c2)O)C(O)C1 c1(-c2c(C)c3c([nH]2)CCCC3=O)nc(C2CCC2)nn1C1CCCc2ccccc21 c1(C(N)=O)cccc(C(=O)NCC2CCCCC2NC(C2CC3CCC2O3)=O)n1 c1(CC(=O)NC2C3CN(C(c4ccc(C(F)F)o4)=O)CC23)cc(F)ccc1F Cc1ncc(CNC(C2CCCC2NC(C2(Cl)CC2(F)F)=O)=O)o1 CC1CC(C)(C(=O)NCC2(C(N)=O)CN(C(=O)COc3ccon3)C2)C1 C1(NC(C(C)NC(CC)(C)C)=O)COCCC1C(=O)NC(CC)(CC)CO c1(-c2cc(CC(=O)Nc3cccc(C=C)c3)ncc2)cc(S(C)(=O)=O)ccc1F CCC(CC)C(C(=O)NCCn1cc(C(=O)N(C2COC(C)(C)C2)C)cn1)OC C(C(C)(C(C)C)NC(=O)CSc1nncn1C)NC(c1cc(C)oc1)=O c1(SC)cc(C(=O)NCCCCNC(=O)CCN2CCCC2)ccc1F N1(C(c2c(C(C)(C)C)ncs2)=O)CCCC(C)(CNC(=O)Cn2cc(Cl)cn2)C1 c1(C(=O)NCC2(C(=O)NC(C3CCOC3)CC)CCC2)cncc(C#N)c1 C1(C(=O)NCC(CN(C(C(CC2CCC2)OC)=O)C)(C)C)CC(N=[N+]=[N-])C1 Cc1cc(C(N2CCC(NC(=O)CN(C3CCCC3)C)C(O)C2)=O)c(C)n1C N1(S(CCC)(=O)=O)CCCCC1C(=O)N(CC(C)N(C)C(c1nocc1C)=O)C C1(NC(c2ccc(OC)c(Cl)n2)=O)C2COCC1CN(C(=O)CC1CC(C)C1)C2 c1(C(N(CC(C)NC(c2csc(C3CCCO3)n2)=O)C)=O)c(F)cc(F)cc1Cl c1(OC)cc(CCCC(=O)N)cc(F)c1.c1(CCO)sccc1CO C1(NC(c2cc(Cl)cc(I)c2)=O)CN(Cc2nccnc2Cl)CCC1(F)F C1(CC)CCC(C(=O)N(CCCN(C(=O)CCc2c[nH]c(=N)[nH]2)C)C)C1 N1(C(CNC(CC)=O)=O)CCC2(CCC2NC(=O)CC(C)C2CCCCC2)CC1 C(N=c1[nH]cnc2c(Br)c[nH]c12)C1N(C(=O)C(C2(O)CCCC2)F)CCCC1 C(=O)(CC(C)CC(C)C)N1C(CN(C(c2[nH]cc(CC(C)C)c2)=O)C)COCC1 CC(O)C(F)(F)C(=O)NC(C1CCCC1)CNC(=O)C(c1cccc(Cl)c1)O S(=O)(=O)(c1cccc(S(=O)(=O)NC2CC2(F)F)c1)Nc1cc(C)nc(C)c1 Cc1nc(C)c(CNC(C2CC2C2CN(C(=O)CCn3cccc3)C2)=O)[nH]1 C(=O)(C(F)(F)CCn1ccnn1)NCC1C=CC(NC(C(CCOC)C)=O)C1 c1(NC(=O)NCC2(C(=O)OC)CC=CC2)nc(Cl)c2ncnc-2[nH]1 c1(C(=O)NCC(C)CN(C(=O)C2=CCCCC2)C)n[nH]c2c1C(=O)CCC2 N(C(=NCCC(=O)N1CCCC1)NCC(C)(C)C1CC1)C1CC(OC)C1 C(F)(F)(C(F)(F)F)OCC(=O)NCC1(O)CN(C(C(C2CCCCCC2)C)=O)C1 C1(C(N(C2CCCN(C(=O)COc3ccccc3Cl)C2)CC)=O)CCCC1(C)C C(N=c1cc[nH]c(=NCCCCCC2CCCC2)[nH]1)c1c([N+](=O)[O-])cn(C)n1 c1(C(=O)NC(C)C(=O)NC2CC2C(=O)O)cc(F)cc(F)c1 c1(-n2cc(C(C3CC3CN)=O)nn2)cc(C)cc(F)c1.CCC(O)(C(=O)N)c1ccccc1 CCCC(C(=O)NCC(CC)NC(=O)C(O)CN(C)C)OC N1(Cc2cc(C)no2)CCC(C(C)NC(=O)C2=C(Cl)CC2)CC1 C1(C2CN(C(C3CC4(CC4)CO3)=O)C2)(NC(C(CC#C)O)=O)CC1 N1(C(c2cc(C)n(C)c2)=O)CCCN(C(c2cc(C)n(C(F)F)n2)=O)CC1CO CC(C)CC(C)C(=O)N1CC(NC(=O)CC(O)CN(C)C)C(C)C1 C(CCCC(C(=O)NCCCC1CC1)N1CCCC(C(N)=O)CC1)OC C1(CNC(CCOC)=O)(CNC(C2COCCC2C)=O)CC12CCC2 c1(C(N2CCC3CN(C(CC4CC(=O)NC4=O)=O)C3C2)=O)cncc2cnccc12 c1(C(=O)NCCC2OCCN(C(C(C)=O)=O)C2)ccc(O)c(C)c1C C(=O)(C1CCCn2nccc21)N1CCC(CNC(c2cc(Cl)cc(C)c2N)=O)C1 C(=O)(CC(C)(O)COC)NC(C(C(=O)C(C)(C)OC(C)C)=O)COC.N(CC)CC C1(CCNC(C=CC(C)NC(C2COC(=O)N2)=O)=O)CCCN1C Cc1cn(C=CC(=O)NC2CCC(N(C)C(c3conc3C)=O)C2)s1 c1(CC)cc(C(N2CCC(C)(NC(=O)CCC(=O)c3ccsc3)C2)=O)oc1C c1(C(N2CC(CNC(C3CCC3)=O)C3C2C3)=O)c(F)cc(Br)cc1F c12ccc(nc1)N1CC(C1)CCN2.C(=O)(C=CC(=O)N(C)C)NC Cc1nn(C)cc1CC(=O)NCC#CC(=O)NCC1(C#N)CCCC1 Cn1cnc2c1CCCC2C(=O)NC1CC(CNC(c2sc(C#N)cc2Cl)=O)C1 N1(C(CC(C)OC)=O)CCC(NC(c2ccccc2F)C)C(C)C1 N1(C(COCCCCC#C)=O)CCN(C(=O)C=CC(F)(F)F)CC1c1ccccc1 C=Cn1nncc1C(=O)N(CCC(=O)NC(C)(CC)CC)CC CC1CN(C(=O)CCn2ccccc2=O)CCC1NC(c1cnco1)=O n1(CC(CN2C(C3CCN(C(COC)=O)C3)CC2)O)ccc2cccnc12 C1(NC(c2nnnn2Cc2ccccc2)=O)CCC2CCCC1C2 c1(CC)[nH]ccc1C(=O)N(CCCNC(C1(Cl)CC1(F)F)=O)C(C)C N1(C(COC(CC)C)=O)CCC(C(C)NC(c2csc(Cl)n2)=O)CC1 Nc1cc(C(=O)NC2CCC2CNC(=O)C(C2(O)CCCC2)F)cc(Cl)n1 C(CC(=O)N1CCC(CNC(=O)CC(C)(F)F)C1)(C(N)=O)NC(C)=O N1(C(CN(C(C)C)C)=O)CC(NC(c2ccn3ccnc3n2)=O)C(C2CC2)C1 C1(CC)CN(C(=O)C=Cc2ccco2)CCN1C(=O)CCc1ccc(F)cc1 C1(CNC(CC(C)=C(C)C)=O)CC(C)CCN1C(=O)CC1CCCCO1 c1(NC(CC)CNC(c2ccc(C)c(C#N)c2)=O)cc(C)nc2ncnn12 Cc1ccccc1C(=O)NC1(CNC(=O)CCC(C)N2CCCC2)CCC1 C(C)(C)(CC(F)C(=O)Nc1ccc(CO)cc1C)NC(c1cc(C)cc(C)c1)=O N1(C(c2n(C)ncc2Cl)=O)CCC2(CCC2)C(CNC(=O)C=CCO)C1 CCCCC(CC)CN=c1nc2ncn(C)c2c(N2CCC(CC(N)=O)CC2)[nH]1 CC1CCCN(C(=O)COc2ccc(Cl)cc2)C1CCNCCO C1(C(=O)NCC(C)CNC(=O)CN2CCC(=O)NC2=O)(CC)CCC(F)(F)CC1 C(=O)(CCN=c1[nH]c(=NCC2CCCCC2)c2ncccc2[nH]1)N(C)CC1CC1 C(=O)(C1CCCc2n[nH]cc21)NC(CC)CN(C)C(c1cnoc1C)=O C1(C(=O)NC2C(CNC(c3ccn(C)c3)=O)C2)CNC(=O)CC1(C)C c1(C(=O)NCC23C(CN(C(CC4(C(=C)F)CCC4)=O)C2)C3)nnc2ccccc2n1 c1(C(C)C)nocc1C(=O)N(CC(C)O)CCNC(C1CCC(=O)O1)=O c1(C(N2CCC(C(C)NC(Cc3c(C)scc3)=O)C2)=O)cnc2sccn12 c1(C(=O)NC2CC3N(C(C(CC)C#N)=O)C(CC3)C2)nc2ccccc2cc1Cl c1(OCC)ccc(C(C)C(N2CCCC2C(C)NC(c2coc(O)n2)=O)=O)cc1 c1(CCC(N2C(C(=O)Nc3cc(C)ncc3)CCCC2)=O)cccc([N+](=O)[O-])c1 c1(C(N(C)CC2CCCN(C(C(F)OC)=O)C2)=O)c(C)nn(C)c1F C(c1cccc(F)c1Cl)=CC(N1CC(NC(c2cc(C)oc2)=O)C2C1C2)=O C1(NC(c2n(C=C)nnc2)=O)CCN(Cc2ccc(CF)cc2)CC1C CCS(=O)(=O)C=CC(=O)N1CCOCC1Cc1cn(CC(C)C)nn1 C1(CCNC(c2c(CC)occ2)=O)CCCN(C(=O)C(c2ccccc2)O)C1 C1(NCC2CC2)CCCCC1.O=C1CN1C1CC1.C1CCN1 CC12CCC1CN(C(=O)CCC1CCCCN1C(=O)CC1CC(=O)C1)C2 C1CCN(C(=O)CCn2cc(CN)nn2)C1.C1(C(=O)NC)CCC1 c1(NCC(=O)N(CC#CCSC2COCC2N=[N+]=[N-])CC)ccccc1[N+](=O)[O-] CC1CN(C(=O)Cc2cnn(C)n2)CCN1C(C1CC2OC1C1CC21)=O C(C)(C)(C(C)CC(=O)c1nc(C(=O)O)c(Br)s1)NC(C1C(C(=O)OC)C1)=O C1(CCO)(NC(C(C)=CC)=O)CN(C(=O)C(c2cnn(C)c2)C)C1 N1(C(COCCN(C)C)=O)C2CCC(C2)C1CC(N1CC=CC1CF)=O C=CCN(OC)C(=O)CC1CCCN(C(=O)C(C)OCC2CC2)C1 C1(C(=O)NC(CC2CC2)CO)CC2(CCC2)CN1C(=O)CCOCC1CCC1 C=CC1CCCN(C(=O)C(c2ccco2)NC(=O)C=Cc2ccncn2)C1 N1(C(CN(C(=O)C(F)C2CCCC2)CC#C)=O)CC(O)(C2CC2)C1 Cc1n[nH]c(C)c1CC(=O)NCC1C(C)CCN1C(c1ccn(C(F)F)n1)=O C(C1=CCN(C(=O)C=CCOC)CC1)NC(c1c(CC=C)cccc1)=O C#CC1(C(=O)NOCCCCC)CCN(C(=O)C(F)C(C)(C)O)CC1 C1(C(N(CCOCCCN(C(=O)Cn2ccnn2)C)C)=O)CCC=CCCC1 C1(C2CCN(C(C3CCCC(C)(C)O3)=O)CC2)(NC(CSCC#C)=O)CCC1 CC(CCCNC(=O)CC(O)c1ccccc1)NC(C1(CC(F)F)CCC1)=O CCCCCC(C)CC(=O)NCC1(C(=O)NC2CCCC2CN(C)C)CC(=C)C1 N1(C(C(C2CCCN(C(c3c(CC)csc3)=O)C2)C)=O)CC(=O)N2CCCC2C1 C(CCC(C)C)(C(=O)NCC(C)(C1CC1)SC)NC(CN(CCC)C)=O c1(C(=O)NC(C2CCOC2)CNC(c2c(C)ocn2)=O)cc(O)ccc1F CN(CC1CCCc2n[nH]cc21)N1CCCCC1CCN(C)C c1(CC(=O)NCC(C2CCC2)NC(C2CC(=C)C2)=O)cc(OC)ccc1[N+](=O)[O-] C1(C)(CNC(c2[nH]cc(C)c2)=O)CCCN(C(c2cnc(C(F)(F)F)nc2)=O)C1 c1(C(=O)NC(CNC(c2cnc(OCC)s2)=O)CO)cc(CO)ccn1 CC(C)C(C(=O)NC(C)CCCNC(=O)Cc1ccno1)C(C)C C1(F)(C(=O)NCCCCNC(C(CCC)C)=O)CS(=O)(=O)CC12COC2 C(=O)(C(C)(C)COC=CC)NCCN1CCC(NC(C2(C(F)F)CC(=C)C2)=O)CC1 C(=O)(C1COc2ccccc21)N1CC(NC(CCC)=O)CC2(C1)CC2 N1(C(c2c(C)nc(C)s2)=O)CCCCC(CCC(=O)Nc2ccccc2)C1 C(=O)(CC(C)(O)CCCC)N1CCC(CC=C)(NC(c2ccsn2)=O)C1 C(=O)(C(O)P(C)(C)=O)NC1CCC(CNC(C2(NS(C)(=O)=O)CCCCC2)=O)C1 C(C(C)(O)C(F)(F)F)N(CCOC)C(=O)Nc1ccc(OC)nc1 Cc1ccc(NC(C23CCC2CN(C(c2ccc(Cl)o2)=O)C3)=O)cc1O c1(C(=O)NCC(CN(C)C(C23CCC(CO)(CC2)C3)=O)O)ccc(CO)c(F)c1 c1(C(N2C(C(N)=O)CC2C(N2CCC(O)(CO)CC2)=O)=O)cc(O)ncc1F Cc1cc(C)c(C(N2CC(C(C)NC(=O)C(c3cn(C)nc3C)C)C2)=O)c(S)n1 Cc1ccnc(O)c1C(=O)NCCCCC1CN(C(C2CCOC(C)C2)=O)C1 CC1(NC(c2cc(C(N)=O)c[nH]2)=O)CCN(C(=O)CCn2cc(Br)cn2)C1 N1(C(Cn2nnc(=N)[nH]2)=O)CCC2CCN(C(c3cccc(F)c3)=O)CC12 C1(C(C)C)CCc2sc(C(=O)N(C)CCN(C)C(C3(C4CCC4)CC3)=O)cc2C1 c1(C2CC(C(=O)NC3CN(C(c4ncsc4C4CC4)=O)CC3F)C2)ccc(F)cc1 c1(NC(c2cc(CNC(c3ncn(C)c3)=O)on2)=O)ccc(I)c(F)c1F C(=O)(CCCC(C)(C)C)N(C)CC1CCN(C(C=CCCC(C)C)=O)C1 c1(C(=O)NC(C2CCN(C(c3csc(=N)[nH]3)=O)C2)(C)C)ccc(C(F)(F)F)nc1 CCCCC(O)C(=O)NCC(C(C)C)NC(C1CC1(C)C(=O)OC)=O C1(NC(c2scc(C(=O)OC)c2)=O)CCCCN(C(=O)C(C)(C)CC2CC2)C1 N1(C(c2c(OC)cccc2O)=O)CCC(C2CCN(C(=O)C3=CSCCO3)C2)C1 C(CCCCC(=O)N1CC(CO)C(O)C1)N(C)C(C1(C)CC1(F)F)=O CC1CS(=O)CCN1C(=O)CC1(C)CCN(C(C2CC3C=CC2O3)=O)C1 CC1(C)C(C(=O)NCc2nccs2)CCN1C(C1C=CCS1)=O C(CCCC(CO)NC(c1cccc(-c2cscn2)c1)=O)NC(=O)C1=CCCC1 c1(OCC(N2CC(CNC(c3n(CC)ncc3)=O)C2)=O)c(C)cccc1C S(=O)(=O)(c1ccc(N2CCCC(CSC)C2)c(Br)c1)NCC(C)OCC=C C(=O)(C(F)(F)CO)NCC(c1ccc(F)cc1)NC(C1(CCOC)CCC1)=O C1(C(C)C)CN(C(c2nccc(C(F)F)n2)=O)CCN1C(C1(C)COC1)=O Cc1c(F)ccc(Cl)c1C(=O)NCC=CCNC(C1(CS(C)(=O)=O)COC1)=O c1(C(=O)NC2CCN(C(CCCC(C)=O)=O)CC2CO)cnc2sc(C)cn12 c1(OC)noc(C)c1NC(=O)CCCNC(=O)CC1CC1(C)C C1(C(=O)NCC2(CNC(CCC(NN(C)C)=O)=O)CC2)CC2(C1)CC1(CCC1)C2 c1(CN2CC3C(NCC(=O)NC(C)(C)C)C3C2)ccc2c(c1)Cc1ccccc1-2 C1(C(=O)N(CCCCCNC(=O)C(=O)NC2CC2)C)(CC)CC(C)(C)C1 c1(C(=O)NCC(CO)NC(C2(CCCC)CCC2)=O)cccc2ccccc12 C1(C(=O)NCC2C(C(=O)NCC[Si](C)(C)C)OCC2)CC(F)C(=O)N1 N1(C(c2occ(C)c2)=O)CCC(C(=O)NCc2ccc(C)c(O)c2)=C(F)C1 c1(C(=O)NCCOC2CCN(C(C3C(C)=C3)=O)CC2)cc(F)cc(C)c1N c1(N2CCCCC(NC(CCC(=O)N(C)C)=O)C2)ccc2c(n1)CCC2=O C1(CN(C(=O)C=C(Cl)Cl)CC)CCCN1C(=O)CC(C)c1cccs1 n1(CCC(N2C3(CNC(COC(C)=O)=O)CCC3CC2)=O)cnc2sccc2c1=O N(C(=NCC1CCC1)NC1CCOc2ccccc21)CNC1(C2CC2)CCS(=O)(=O)C1 C1(C(=O)NCc2c(CC)nccn2)CC(C)(C)CN1C(=O)C(C)NC=O c1(COC)ccc(CC(C(=O)N(C)NC(C2(C(F)F)CC2)=O)C2CC2)cc1 CCC(CCC(=O)NOCC1(F)CCC1)NC(C1CC(C)(O)C1)=O c1(CN(C2(CCC)CCC2)C2CC2)nnnn1C(C(=O)NC(C)(C)C)C1COC1 N1(C(c2cc(C3CC3)no2)C(=O)NC2CC2)CCC(F)(F)CC1 c1(C(N2CC(OCCNC(C3C(CC)CCO3)=O)C2)=O)scc(C)c1C N1(C(C(C)c2cccs2)=O)CCCC12CCN(C(c1ccc(N=[N+]=[N-])cc1)=O)C2 CN1CCN(C(=O)CCCC2OCCO2)C(CNC(=O)CC2CC23CC3)C1 Cc1ccc(C(N2CCC(C)(CC(=O)NCCc3cc[nH]n3)C2)=O)nc1O c1(N2CC=CC(NC(CC(C(C)C)O)=O)C2)ncnc2[nH]c3ccccc3c12 N1(C(CC2C(C)(C)C2)=O)CCCC2C1CCN2C(c1ccc(Cl)c(C(F)F)c1)=O N1(CCC(=O)NC(c2ccccc2)C)CCCC1P(C)(C)=O c1(N2CCCC(COC)(NC(c3cc4c(s3)CCC4)=O)C2)nc2cccnc2s1 C(=O)(CCCCCC(C)O)NC1(CNC(c2ccc(C)c(Cl)c2)=O)CCC1 Cc1ccncc1C=CC(=O)NC1CN(C(c2nnc(O)nc2O)=O)CC1C C1(NC(CC)=O)CCCCN(C(C2(c3cccc(C#N)c3)CCC2)=O)C1 CC1(C)OCC2CC12C(=O)NCC#CCNC(c1ccc(C(N)=O)c(Cl)c1)=O C1(c2ccc(OC)cc2)C(C(=O)Nc2cnn(C3COC3)c2)CCC(=O)N1C c1(C(N2CC(CNC(c3cc4cccnc4[nH]3)=O)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 C(CN=C(NCC(C)C)N1CCC2(C1)CC2(F)F)OCCCC CCCC(CCCNC(=O)C(OC)OC)NC(=O)C(C1CN(C(C)=O)C1)NC1CC1 C(=O)(CC(F)(F)C(F)F)NC1CCN(C(CCOCCC2(C)OCCO2)=O)CC1 C1(N(C(c2c(CC)nn[nH]2)=O)C)CCCN(C(C2C(C)C2C)=O)CC1 C12(OC)CCCC(C(=O)NCC3CCN3C(C34CC(F)(C3)C4)=O)(CC1)C2 C1(CC(=O)O)CC(F)(F)CN1C(=O)CC12CCC1CCN2 C(=O)(C(C)(C)CCC#N)NC1CCC(C)(CNC(c2n(C)c(S)nc2)=O)C1 Cc1c(C(N2CCC(NC(=O)OCC3CN(C)C3)CC2)=O)ccc2c1OCCO2 CCC(F)(F)CC(=O)NC(C(=O)N1CCCCC1)C(C)C c1(C(N2CCCC(C(N(C(C)C)CC)=O)C2)C(=O)OC)ccc(Br)cc1C C12(C(N3CC4C(NC(c5n[nH]c(C6CC6)n5)=O)(C4)C3)=O)CCC(C1)S(=O)(=O)CC2 C1(NC(c2cn(CCC)nn2)=O)CN(C(c2ccc(Br)o2)=O)CC(C)(C)C1 CC1CN(CS(=O)(=O)Nc2cccc(Cl)c2)Cc2c(Br)ccc(F)c21 c1(C(=O)NCC(CN(C(C=CCC)=O)C)C)cccc(COC)c1 CC1(C)CC(C(=O)NC(C2CCCC2)CNC(c2c[nH]nc2Br)=O)C1 C1(OCC)COCCC1C(=O)NCC1CN(C(=O)CSc2ccccc2F)C1 N1(C(C(C)C2CCC2)=O)CCC2(CCC2)C(CNC(c2cnn3c2CCC3)=O)C1 c1(-c2c(C)nccc2)ccc2sc(C(N3CCNC(=O)CC3)=O)cc2c1 c1(SC)cccc(C(=O)NC(CNC(c2cn(C)nc2C2CCC2)=O)CO)c1 c1(C(N2CCC(NC(CCC3C(C)(C)C3)=O)C2)=O)cc(Cl)ccc1O c1(C(N(CC)CC2CCCN2C(c2ccoc2C)=O)=O)cc(C)c(C)cc1C c1(CC(=O)OCC)nc(=N)[nH]c(C)c1-c1cccc(-c2ccc(C(F)(F)F)s2)c1 c1(C(C)NC(N(CC(COCC)C)C)=O)cc(OC(C)(C)C)cc(Cl)c1F Cc1cnc(F)c(-c2cn(CC3CN(C(C4CCCC(C5CC5)O4)=O)C3)nn2)c1 C#CC1CN(C(=O)C(C)OC)CCN1C(c1ccc(C(C)=O)cn1)=O C1(NC(=O)C2=CCSC2)CC(F)CN(C(=O)C(=Cc2cccc(F)c2)F)C1 C(c1cccnc1)=C(C)C(=O)NC1C2CN(C(=O)CSC3CCCCCC3)CC12 N1(C(c2cc(C(=O)O)sn2)=O)CC(Cn2cc(CC(=O)O)nn2)C(C(F)(F)F)C1 Cc1ncncc1NC(c1ccc(-c2cnn(C(C)C)c2)cn1)=O S(=O)(=O)(c1c[nH]ccc1=NC(C)c1nc2c(s1)CCCC2)NC1C(OC)COC1 CCC(C)(C)CC(=O)NCCC1CCCN(C(C2(c3ccncc3)CCC2)=O)C1 Fc1cc(CCCNC(C2CCOC2)CC2CC2)cc(Br)c1 C#CC1(C(NOCC2CC(=O)N(C)C2=O)=O)CCN(C(=O)Cc2ccn(C)c2)CC1 c1(CNC(C2CC=CC(NC(c3cc(Cl)no3)=O)C2)=O)cccc2[nH]ccc12 C1(c2n(C)ccn2)CCCN(C(C2C=CCCC2)=O)C1 Cc1[nH]cc(C(N2CCC3(NC(c4cccc(CO)n4)=O)CC3C2)=O)c(=O)c1Cl C1(CC(=O)N(CCCNC(c2ccnnc2)=O)CC2CC2)CCCC1O C1(CCC(=O)OC)CN(C(C)=O)CCN1Cc1oc(C(=O)OC)nc1C c1(C(=O)NC2CC(C)(C)N(C(=O)CCCNC(N)=O)C2)[nH]cc2c1CCS2(=O)=O CC(C(C)(C)C(=O)NCC1CCCCS1)NC(=O)CSc1cn[nH]c1 c1(N2C3CC(=C)C(C3)C2)[nH]c(=NC(C)CF)nc2c1ncn2C(C)C C1(N(C(CNC(=O)OC)=O)CCO)CCCN(C(=O)CCc2ncco2)C1 N1(C(c2c(C)nn(C)c2)=O)CCN(C(=O)C(C)CN2CCOCC2)CC1CCO CC1CC(O)CN1CC(=O)NCCC1CCN(c2ccccc2)CC1 C1(NC(CC(CC)C2CC2)=O)C(C)CCN(C(=O)C=C2CN3CCC2CC3)C1C CCC(C(=O)NCC1CCN1C(c1nc(C)ccc1OCC)=O)C(C)(C)CC CC1CCC(C(N2CC(C)(C)CC2CNC(c2cc(O)n(C)n2)=O)=O)CC1C C1(NC(CCNS(CC)(=O)=O)=O)CCCCCC1NC(c1cc(C(N)=O)cs1)=O C1(C)(NC(C#CC(OCC)OCC)=O)CCCN(C(c2ncnc(O)c2F)=O)C1 Cc1cc(CNC(c2[nH]cc(C)c2C)=O)oc1C(=O)N(C1CCN(C(C)C)C1)C n1(C(CC2(N(CC(N3CCCC3)=O)C3CC3)CCCC2)=O)nc(O)ccc1=O.NC N1(CC2CCC(NCC)CC2)CCCC(C(=O)NCCSCCO)C1 C1(CCNC(C2CCN(C(C)=O)C2)=O)CN(C(c2cnc(N(C)C)nc2)=O)CCO1 N1(C(c2c(C)nn(C)c2)=O)CC2CCN(C(C3(S(N)(=O)=O)CC3)=O)CCC2C1 C1(C(=O)NC(CCOC(C)C)C(=O)O)CC2(C1)CC21CC1 CC(C)CCCC(C)C(=O)N1CCC(CC(N2CCn3cnnc3C2)=O)C1(C)C c1(NC(C(=O)O)=O)cc(Br)cnc1Cl.CN(C1CC1)CC1CC1 C(=O)(C(C(C)CC)N(C)C)NCCCN(C(=O)Cc1cncnc1O)CC CC1(C(=O)NC2C3CN(C(=O)C=CC4CCCCC4)CC23)CCC(=O)N1 CCC(C(O)C(F)(F)F)NC(c1ccc(C2CNC(=O)C2)cc1)=O C1(C(=O)NCCOCCC(=O)OC)(CO)CC12CCC2.C12CC(C1)C(=O)N2 CC1=NOC(CC(=O)NC(C(=O)N(C)Cc2ccncc2)C2(O)CCC2)C1 CC(C(=O)N1CCN(CCN(C)C(C2(N3CCCC3)CC2)=O)CC1)C(F)(F)F CCCC(C(=O)N(C1CCN(C(=O)CC2C(=O)ON=C2C)CC1)CC1CC1)OC N1(C(C(N2CCOCC2)C)=O)CC(C(=O)NC2CCCC2)OC(C(F)(F)F)C1 c1(C(=O)NC2CCCN(c3cc(C4CC4)nc(Cl)n3)C2)ccc2nn[nH]c2n1 C(=O)(CCCc1nc(C2CC2)no1)N(CCOC)C(=O)C1CC1 N1(C(C23N(C(c4csc(C)c4C)=O)CCC2C3)=O)CC(C2=NOCC2)C1 C1(C(=O)NCC(C)C)CC(NC(c2ccc(O)cn2)=O)C1(C)C N1(C(C(C)(C2CC2)OC)=O)CCC2(CC1)CN(C(c1cc(C)c(C)s1)=O)C2 c1(CC)nc(C)c(C(N2CCC(COC)(NC(=O)CCc3ncnn3C)C2)=O)o1 c1(NC2CN(C(CN(CCCC)C(C3CCC3)=O)=O)C2)csc(C2CCC2)n1 C1(N(C(COCCOCC#C)=O)C)CC2CC1N(C(C1CCCCC1O)=O)C2 C(C(O)C(=O)NCc1ccc(C(=O)NCc2nnc(C)s2)s1)=CC CCC(C)CC(=O)NC1C2CC1N(C(c1c[nH]c(=NC)o1)=O)C2 N1(C(CC(C)(C)OC)=O)CC(NC(=O)C(C)(C)c2cccs2)C(C)(C)C1 c1(C(N2CCC(O)(CNC(C3(F)CCCOC3)=O)C2)=O)cc(F)cnc1O C1(C(N2CCCC(N(C(C(C)c3ccsc3)=O)CCO)C2)=O)CN2CCC1CC2 c1(C(=O)N)cc(C)ccc1F.C1(C(=O)NCc2c(C)ocn2)C(C)CCN1OC N1(C(C(N2CCC(C)C2)=O)=O)CCN(C(c2ccc(C#N)o2)=O)CC1C1CC1 C1(CC(=O)NCCC#C)CCN1C(=O)CC1CC1(C)C C1(CNC(C2CC3(CCC3)C2)(C)C2CC2)CC(=O)N(c2cccc(C3CC3)c2)C1 Cc1cc(C(N2CC(CO)C3(CC3)C2)C(=O)NCC2CCOCC2)cc(C)n1 CC1(C)CN(C(=O)Cn2ccc3ccccc23)CCC1NC(=O)Cc1cnsc1 C1(N(C)C)CCCN(CC(=O)NCC2CCCN(C(=O)C=CCF)C2)C1 N12CCC(C(O)C1)C2=O.c1(C(c2n(CCCC)nnn2)NC)c(Br)n[nH]c1C N1(C(C2(CC)CCC2)=O)CC2CCCC(NC(c3cn4cccnc4n3)=O)C2C1 CCC(CC)(CC(=O)OC)C(=O)NCC(CC)(CC)NC(C1C(C=CC)C1(C)C)=O c1(C(=O)NC(C(N2CCC(c3n[nH]cc3CO)C2)=O)C2CC2)ncccc1F N1(C(C(C)OC)=O)CCC(C(C)C(=O)N(CC(C)O)C(C)C)C1 C=C1Cn2c(C(=O)N(C3CCC(NC(=O)CNC(C)=O)C3)C)nnc2S1 N1(C(c2c(OCC)ccs2)=O)CCC2(CCCN(C(=O)C3=COCC3)C2)C1 CC1(CNC(C23CCCC2OCC3)=O)CN(C(c2cc[n+]([O-])cc2)=O)CCO1 c1(C(N2CC(C)(NC(C3CC(N4CCCC4)C3)=O)C2)=O)cccc(C2CCC2)c1 O=C1CC2(CO1)CN(C(C1CN(C(=O)Cc3ccon3)CCO1)=O)C2 c1(C(=O)NC2(C3CCCN3C(=O)C(c3ccccc3)=O)CC2)cc2ccccn2c1 CC(C)(CCN(C(=O)CCC1CCC(=O)N1)C)NC(=O)COCc1cccnc1 Cc1cc(C(=O)NC(C2CN(C(=O)C=CC(C)C)C2)C)cc(C)c1F C1(C(N2C(CN(C(COCC=C)=O)C)CCC2)=O)CCC(C(C)C)NC1=O c1(CNC(=O)C(NC2CCc3ccccc32)=O)ccc2c(n1)CCCC2 C(C)(CC1=CCCCC1)NC(C1(NC(CC)=O)CC1(C)C)=O N1(C(C=C(C)c2cccs2)=O)CCC(NC(=O)Cc2ccc(C)nc2)C(CO)C1 CCCC(C)CC(=O)N1CCCC1CN(C(C1CC12CCC2)=O)CC C(=O)(CCCCCC(C)(C)C)NCCN(C(c1cc(C)ncc1C)=O)CC C(=O)(C(F)C1=CCCCC1)NC1C(C)CCN(C(c2cc3ccsc3[nH]2)=O)C1 C(=O)(C(C)(C)C(F)F)N1CCC(C(N(C)CC23CCC(CO2)C3)=O)C1 CC1=CC(C)CN(CCNCc2ccc(N3CCOCC3)cc2)C1 C1(CC(=O)N(CC(C)NC(=O)C(=O)NCC(F)(F)F)CC)C(=O)ON=C1C c1(OC)cc(C(N2CCC(C(C)NC(=O)C(C)(C)C(N)=O)C2)=O)c(Cl)cc1Cl C1(CC)CN(C(=O)Cn2cncn2)CCC1NC(=O)C(C1CCCCCC1)(C)C CCC(C(=O)NC1CN(C(=O)C(c2ccc(Cl)cc2)=O)CC1(C)C)C(C)C N(C1CCCc2occc21)c1nccc(=NCC2(COC)CCOCC2)[nH]1 C(C1=NOC(C)C1)N(C(=O)COCCCN=[N+]=[N-])C.C(CC(=O)NCC)NC(C)=O.O N1(C(c2ccc(OC)nc2)=O)C2CCC1CN(C(=O)C(C)CC(C)C)C2 Cc1cn(-c2ccccc2)nc1NC(=O)NC(C)(CO)c1cccs1 C(C)(C)(CCOC(C)=O)NCCCN(C)CC n1(CC(=O)NC(C)(C)CCNC(C2(CO)CCCO2)=O)cc(S(C)(=O)=O)cn1 c1(C(=O)NCC(c2ccc(F)cc2)NC(C(C)(C)C2CC2)=O)cc2scnc2[nH]1 Cc1cccc2c1CCN(N1CCCC(c3nc4cccc(Br)c4[nH]3)C1)C2 C(=O)(CC(C(C)OC)NC(C1CCCCO1)=O)N1C(C)(CC)CC1 C1(C(C)C)CCCCC1CNC(=O)N(CCN(C)C)Cc1ccccc1 C(C(CCC(F)(F)F)N=c1cccc(S(=O)(=O)NCc2csnc2C)[nH]1)OC C1(CNC(=O)Nc2ccnc(C)n2)CCC2(C1)OCCO2 C1(CCN(C)C)CCCCN1C(C1CC(CNC(c2cnnn2C2CC2)=O)C1)=O CC1CCC=C1C(=O)N1CCN(C(c2cc3c(s2)CCC3)=O)C2CC12 CC1CN(C(=O)CN2CCC(CO)CC2)CC1NC(c1cn(C(C)(C)C)nn1)=O N1(C(C(C)(C)OC(C)C)=O)CCC(NC(=O)C#CC2(C)CCCO2)CC(C)(C)C1 Cn1ncc(C(N2CC(O)(CNC(c3cnoc3-c3ccoc3)=O)C2)=O)c1C#N Nc1ncc(C(F)(F)F)cc1C(=O)NC1CC(NC(=O)C#CC(=O)N(C)C)C1 Cc1c(C(=O)N(C(c2c[nH]c(Br)c2)=O)CC2CCN2)cccc1-c1ccccn1 C1(CNC(c2c(CC)ccs2)=O)CN(C(=O)C(C)(C(C)C)OC)CCC12CCC2 C1(N(C)C)C2CN(CC(C3CCCC3C(F)(F)F)=O)CC12 C12(C(=O)NC(C)CNC(=O)C(=O)NCCC(F)F)COC(CF)(C1)C2 C1(COC)(CNC(=O)C(C)COC)CCCN1C(c1cn(CCO)nc1C)=O C(=O)(C1=CC2CCCCCCC12)NC1(CC)CCCN(C(c2[nH]nnc2C)=O)C1 C1(C(=O)N(C)CCC2CCCO2)(CC)CCCN(C(=O)CC#N)C1 C12(CC(=O)NCC(C(C)(C)C)NC(CC)=O)CCCCC1C2(F)F c1(OCC)cccc2[nH]cc(CN=c3[nH]c(C(=O)Nc4sccc4C#N)cs3)c12 N1(C(=O)C2=COCC2)CC2CC(N=c3[nH]nc(-c4ccon4)s3)CC1C2 Cc1ccccc1NC(=O)C(c1csc(Br)c1)NC(=O)C(C)C c1(Nc2ccc(C(N(CCC#N)C)=O)cc2)cc(=NC2CCOCC2)cc[nH]1 Cc1ccc(Cl)c(C(N2CC(NC(=O)CC3CCCS3(=O)=O)CC(F)C2)=O)c1O N1(C(c2nc(C)sc2)=O)CCC(NC(c2cc(Cl)nnc2Cl)=O)CC1C N1(C(c2occc2C2CC2)=O)CCC2(CC1)CN(C(C1(C3CC3)CCC1)=O)C2 C#CCCN=C(NCCC1COC1)NC1CCC1C N1(C(c2c(CC)ocn2)=O)CC(C2CCCN(C(c3cc(C4CC4)ns3)=O)C2)C1 c1(C(=O)NCCC2N(C(CNC(C)=O)=O)CCCC2)ccc(Cl)nc1N C(=O)(C(C)(C)CC(F)F)N1C(CCNC(C(CC(C)C)NC(C)=O)=O)CSCC1 C#CCCCC(=O)NOC(CC(C)C)C(=O)NC(C)CCC(F)(F)F C#Cc1ccc(C(=O)NC2CCC(N(C)C(c3cn(C4CC4)nc3C)=O)C2)nc1 C1(O)(C(=O)NCCN(C(C(Cc2ccccc2)OC)=O)C(C)C)CCCCCC1 Cc1cc(C(=O)NC2CN(C(c3ccon3)=O)CCC2F)nnc1C C1(NC(CC(C)(C)C)=O)CC2CCC(C1)N2C(c1ccc(I)c(O)c1)=O C(=O)(C(C)C(O)C(C)C)NC1(CNC(C=Cc2cccc(C)c2)=O)CC1 CC1CCCN1CC(=O)NCc1occc1C(=O)NC1CCCC1O c1(C(=O)NCC(CC2CN(C(COCC(=O)NC)=O)C2)(C)C)cc2n(n1)CCO2 N1(C(c2ccn(C)c2)=O)CCN(C2CCC(NC(C3OCCO3)=O)C2)CC1 C12(C(N3C4C(CNC(C)=O)CC(CC4)C3)=O)CCCCCC1OCC2 CCC(CC)CCC(=O)NCC=C1CCN(C(=O)CCNC(C2CC2C)=O)CC1 c1(CC)cc(NC(c2ccccc2NC(C)=O)=O)c(OC)s1 CC1CCN(C(=O)CCc2ccc(Cl)cc2)C(CNC(=O)CN(S(C)(=O)=O)C)C1 Cc1ccncc1CC(=O)NC(CC1CC1)CC(=O)NC1(C(O)CO)CC1 C1(C(N2CC(C)(CCC(=O)NC3CC=CC(O)C3)C2)=O)C2CC(=O)CC12 C12(C(=O)OC)COCC1CN(CC1CCCN1C1CCCCC1)C2 CC1CN(C(c2ncsc2C2CC2)=O)CCN1C(=O)CC(C)n1ccnc1 Cc1cc(=NC(=O)CN2CCN(S(=O)(=O)Cc3ccc(F)cc3)CC2=O)[nH]n1C C1(C(=O)NCCC2(O)CCN(C(C(CCCC)O)=O)CC2)CCc2cncn2C1 S(=O)(=O)(c1sc(O)nc1C)NC1CN(CC(=O)OC)CC1C C1(NC2(CNC(=O)CNC(c3cnccn3)=O)CC(O)C2)CCC2(CCC2)O1 CN1CCN(C(=O)COC2CCOCC2)C(CNC(=O)CC2CC(N(C)C)C2)C1 CC(C)(C)CCCC(=O)NC1(O)CCN(CCNC(C23COC(CF)(C2)C3)=O)C1 C(CCCCCOC)(C(=O)NC1COC1)N(CCCCCCCC)C C1(OC)CC(CNC(=O)CO)N(C(=O)CCc2ncc(C)[nH]2)C1.C(C(C)(C)C)N Cc1cc(C(=O)NCC(C(C)C)NC(c2cccc(NS(N)(=O)=O)n2)=O)nc(C)c1 N1(C(C=CC(=O)OCC)=O)CC(C2(NC(=O)C(O)CC(N)=O)CC2)C1 C(=O)(C(C)(C)CO)NC(C)CCNC(=O)COCC1CCCO1 c1(C(N2CC(CNC(C3(OC)CCSC3)=O)OCC2)=O)ncc(C)cc1F C1(NC(C2(CO)CC(C(F)(F)F)C2)=O)CC2CCC1N(C(=O)COCC(F)(F)F)C2 N1(CC#N)CCN(N2CCCC(Nc3ncccn3)C2)CC1 CCCCC(CNC(C1(CC)CC1)=O)NC(=O)CCCc1nc(C(C)(C)C)no1 N1(C(C2N(CCC)C(=O)CC2)=O)CC2(CCC2)CCC1CNC(=O)C(C)SC N1(C(C=CC(C)NC(=O)CCC2CCCN2C)=O)CCCC(C)(C)C1C C=CC(C)(C)CC(=O)N(C)CCN(C(=O)CNC(c1cccc(OC)c1)=O)C CC(C)CS(=O)(=O)CCC(=O)NCC(C)(F)CNC(=O)CC1CC(=O)NC(=O)C1 c1(C(=O)NCC2(C)CCN(c3cnc(F)cn3)CC2)ccc2n[nH]cc2c1Cl C1(CC(=O)NC(CC2CN(C(c3cnc(C(C)C)[nH]3)=O)C2)C)CCC(C)CO1 C12(CC(=O)NC3CCN(C(CC=C(C)C)=O)C3C3CC3)CCC(CC1)OC2 C1(NC(NC(COC)C)=NCCCc2cc(C)no2)CCOC2(CCCC2)C1 c1(CSC)cc(C(=O)N(C2CN(C(c3csc(O)n3)=O)CC2O)C)ccc1F N1(C(CC2N(C(Cc3nc(C)[nH]n3)=O)CC(F)(F)C2)=O)CC2CCCCC2C1 c1(C(N2CCC(O)(C(CNC(CCCCCC)=O)C)C2)=O)nc(O)nc(O)c1N C(=O)(CC(C1CC1)NC(C12CC(F)(C1)C2)=O)N(c1ccccc1)CC#C C1(NC(CC(CC)(F)F)=O)CC2CN(C(c3cc(COC)on3)=O)CC2C1 CC(C)N=c1[nH]c(N2CCN(c3nnc(C(F)F)s3)CC2)nc2c1COC2 C1(CC(=O)NCCc2ncc(C)o2)(NC(=O)Nc2ccccc2)COC(C)C1 CC1CN(C(=O)Cc2cccc(F)c2Cl)CC1(C)CNC(C1CCOC1=O)=O C1(C(=O)NCC2(O)CN(C(=O)CCCn3ccnn3)C2)CC2CCC1CC2(F)F c1(N2CCC(C(=O)NC(Cc3cccc(C)c3)C)CC2)nc(=N)[nH]c2[nH]ccc12 c1(C(=O)NC2CCC(C)(OC)C2)c(C)[nH]c(-c2cccs2)nc1=O C1(CC)CN(C(c2ccc(Cl)cc2O)=O)CCN1Cc1sc(Cl)nc1Cl c1(CN2CC3(C(C(=O)Nc4cc(OCC)c(C)cc4)C3)C2)c(F)ccc(F)c1C C1(C(CNC(c2cc(CCC)on2)=O)C)CCN(C(=O)C(C)CCN(C)C)CC1 C1(=O)CCN=C(NCS(C)(=O)=O)N2CCC(C2)N1C.C1(CC(C)C)CCOCC1 C1(CC)CN2CCCC2CN1C(=O)NC1COC2(CCCC2)CN1CC CCCCCC(CC)C(=O)N(CC(C)NC(c1cccc(C(C)(C)C)c1N)=O)CC C1(CC)CN(C(c2cc(C(C)C)cnc2O)=O)CCN1C(=O)CN1CSCC1=O C#CC1CC2(CC2)CN1C(=O)C(C1CCOC1)NC(=O)COCC(C)C C1(CCNC(C2(C(=O)NC)CCC2)=O)CN(C(=O)CCC2CC2(Cl)Cl)CCCO1 N12CCCC(C)(C1)CC2=O.c1(CC)nn(C)cc1C(=O)NC1COC(CC)C1 C(=O)(CC(C)CNC(=O)Cc1cc(-c2ccc(Cl)cc2)on1)OCC N1(C(C2CNC(=O)N2)=O)Cc2n[nH]cc2C1C(=O)NC1CCn2nnnc2C1 N1(C(C(=Cc2cccs2)C)=O)CC2CCC2(CNC(=O)CC2OCCC2(C)C)C1 CC(O)(Cc1ccccc1)CC(=O)NCCCN(C(=O)CCC(N)=O)CCO C12(C(F)F)CCN(C1)C(=O)C1CC(C1)OC2.C1(C(=O)NC2CC2)CC1Cl c1(C(=O)NCC2CCCN2C(=O)C(F)=C2CCCO2)cccc(C(F)F)n1 C(=O)(CC(C)(C)CNC(=O)CC1CCCC(C)(C)O1)NCCC(C)CCO C1(NC(c2cc(C)c(O)nc2)=O)C(CNC(=O)CCC2(C)CC2)CCC12CCC2 c1(C(=O)NC(CCCC)CNC(=O)C(C)O)c[nH]c2c(OC)nccc12 C1(NC(=O)CC2(O)CC2)CCC(NC(c2cnc(C(F)(F)F)s2)=O)C1 c1(CC)c(C(=O)NCC2CCCN(C(=O)CNS(=O)(=O)CC)C2)csc1C C1(CC)CCOC1C(N1CCC(CC(=O)NCCC(C)CO)C1)=O C1(CC)CN(C(c2cnn3cc[nH]c23)=O)CCN1C(c1ncccc1F)=O N1(C(CC=C=C)=O)CCN(C(c2ccc(C3CCCO3)[nH]2)=O)C(CS(C)(=O)=O)C1 CCC(CC(=O)N(C1(CC(=O)NC(C2CSC2)C)CC1)C)C1CC1 c1(C(=O)NCC(C)NC(=O)CC2CCOC2(C)C)ccc2cnnn2c1 N1(C(COCCCCC)=O)CC(NC(C2CC3(C2)CC3F)=O)CC2(CCC2)C1 N1(C(CCCNC(C)=O)=O)CC(C)C(C)(C(N2CCC(O)C(C)C2)=O)C1 C1(C(=O)NC(CNC(c2ccn(CCOC)n2)=O)C)Oc2ccccc2OC1C c1(NC)cc(C(=O)N(C2CCN(C(c3cnccc3OC)=O)C2)CC)cc(Cl)n1 n1(CC(N2CC3C(CNC(C(c4cccnc4)C)=O)C3C2)=O)cc([N+](=O)[O-])cn1 c1(C(N2C(C)C3CC2C3NC(=O)C=CCO)=O)ccc([N+](=O)[O-])c(O)c1 C(CCC(=O)NCC1CCN1C(=O)CC1CC(F)C1)NC(=O)CO c1(C(N2CCN(C(C(CC=C)C)=O)CC2c2cn[nH]c2)=O)snc2ccccc12 C1(C(=O)NCc2cccc(SC)c2)CCC2C(C1)C2(F)F.C12(CC1)C(=O)NC2 CCC(CC(=O)NC(C)CC1CN(CCOC)CC1C)c1ccccc1 C#CCCCCC(=O)NCC1C2CN(C(=O)CCN3CCC(CO)CC3)CC12 CC(F)(F)CCC(=O)OCC1CCC(=O)N1C(=O)C(C1CCCCC1)O N1(C(c2ccc(C)c(O)c2)=O)CC2(C1)CN(C(c1c[nH]ccc1=N)=O)CCC2O C1(c2n(CCC)nnn2)(NC(C(C)NCC)C)CCCCC1CS(N)(=O)=O C=C(C)C1OCCC1C(=O)NCC1CCN1C(c1ccc(NS(=O)(=O)CC)cc1)=O n1(CCCC)nnnc1C(C)(CCc1nccs1)NCC1CC1C(F)(F)F CONC(=O)C(=O)N1CCOC(C(=O)N(C)Cc2nnc(C)o2)C1 C1(C(N(CC(COC)O)C)=O)CCCCCN1C(=O)Cn1nccc1C CC1(C#CC(=O)NC2COCC2C(N2CCC3(CC2)CC3CO)=O)CCCO1 N1(C(CCn2c(C(C)C)ncc2)=O)CCC2CN(C(c3cnc(S)n3C)=O)C2C1 c1(CC)ccc(OC)c(C(=O)NC2CN(C(C3(N(C)C)CCCSC3)=O)C2)c1 Cc1cc(C=CC(N2CC3(CNC(C4(F)CCOC4)=O)CC2CO3)=O)c[nH]c1=N c1(C(=O)NCC2N(C)CCN(C(c3c(C)con3)=O)C2)cc(C)nc2ncnn12 C(=O)(C1=NN(C(C)C)C(=O)CC1)N1CCCC(O)(CNC(C(C)C)=O)C1 c1(CCC(=O)NC(C)CNC(c2ccnn2C)=O)ccc2c(c1)OCCO2 C1(C(N2CC(COC)(CO)C2)=O)CN(C(C2CC23CC3)=O)CC1F c1(C(=O)NC2CN(C(c3ccn(C4CC4)n3)=O)CC2F)cn2c(n1)SCC2 C#CC1(C)CCCN(C(=O)CC2CN(C(=O)C(c3cncnc3)C)CC23CC3)C1 C(=O)(C1=NNC(=O)C1)N1CC2C(C(=O)NCc3ncn(C)c3)(C2)C1 c1(C2(C(=O)NCCN(C(c3cncc(OC)n3)=O)C)CC2)cc(C)ccc1F N(C1CCc2ccc(F)cc21)C(=O)NC(c1ccc(OC)cc1)C N1(C(c2c(CC)ncs2)=O)CCCC(NC(=O)COC2CC=CC2)CC1C Cc1cc(C(N2CCNC(C(N3CCCC(C)(O)C3)=O)C2)=O)ccc1F Cc1ncnc(O)c1C(=O)NCCC1CSCCN1C(C12CCC(C)(C1)OC2)=O c1(C(N2C(C(N3CC(C)(C(F)(F)F)C3)=O)CC2)=O)ccc(F)cn1 c1(C(CNC(c2cnnc(O)c2)=O)NC(=O)CC2CC2CC2CC2)ccccc1F N1(C(c2n[nH]c(=N)[nH]2)=O)CC2(CC2)CC1C(=O)NC1CCC2CCC12 C1(NC(c2n(CC)nc(C)c2)=O)CCN(C(=O)Cn2ccnc2)CC1F C(=O)(CC1OCc2ncccc21)N(C)CC1N(C(CCC(=O)OC)=O)CCC1 CCCCCC(C)CCN(C(=O)CCCn1cc(C2CCC3(CC3)CO2)nn1)CC N1(CC(=O)N(CCOC)CCNC(=O)CCCSC(C)C)C(=O)C(C)C(C)C1=O C(=O)(C(C)(C)C)N1CC(C(C(=O)NC(c2nccn2C)C)OCC)C1 C(=O)(CCCCCC#N)N1CCC(O)(C(C)C(=O)NC2CCCN(O)C2=O)C1 C(CC(O)CC(=O)NCC1(NC(c2cccc(N3CCCC3=O)c2)=O)CC1)SC C(S(=O)C1CCCCC1)c1ccc(COCC(C)C)o1 N1(Cc2ccn(C)c2)CCC2CN(C3CCC3)CC12.c12ccccc1SC2=O N1(CC(=O)N(C(C)C)C)CCN(c2cc(C3CCCCC3)ncn2)CC1 Cc1nc2ncnn2c(C)c1C(=O)NC(CNC(=O)C(C)(C)C#N)CC(F)(F)F N1(C(C(CCC)CC(=O)NC2CN(C3CCC3)C2)=O)CC2(CCC2)CC1C CCC(C)CC(=O)C(=O)NCC1CC(NC(c2ccoc2CC(N)=O)=O)C1 C1(CC=C)(C(N2CC(C(C)NC(=O)CN(C)C(=O)OCC)C2)=O)CCOC1 c1(C(N2CC3C(NC(C(C)OCCC=C)=O)C(C3)C2)=O)nc2cccnc2s1 C#Cc1ccc(C(N2CC(NC(=O)C(c3cc(F)cc(F)c3)C)C2)=O)nc1 N1(C(CCCN=[N+]=[N-])=O)C2CC=C(C(=O)NCCN3CCCOC3=O)C1CC2 C1(C)(C(=O)NC(C2(O)CN(C(=O)C=Cc3cn[nH]c3)C2)C)CNC(=O)C1 C1(CNC(c2cc(=O)cc(O)[nH]2)=O)CC2(CCCC2)CO1 C(C(=O)N1CC2(C=CCO2)C1)(C(C)CC)N(C(c1c(CC)con1)=O)C C1(C(=O)NCC2C(NC(c3ccc(CN(C)C)cc3)=O)C2)CC2(C1)CC1(CC1)C2 C1(CNC(c2c(C)cco2)=O)CC(C(C)C)CCN1C(=O)CN1C(=O)CNC1=O N1(C(C=C2CCC(C)C2)=O)CC2CC(NC(c3cn(C(C)(C)C)nn3)=O)C(C2)C1 C(CC(N)=O)(C(=O)NOCC1CCOC1)NC(C(n1c(C)ccn1)C)=O N1(C(CCCC(=C)C)=O)CC2CC(C(N3CCCC(CCCC)C3)=O)CC2C1 CCCC(C(=O)NCC12CN(C(=O)CCNC(=O)COC)CC1CCO2)C(C)C N1(C(C(C)(C)NC(=O)NCC)=O)CC(OC)CC(NC(=O)C(C)N2CCCC2)C1 N1(C(C(C(CC)O)C)=O)CC(C)N(C(c2cnncc2C(F)(F)F)=O)CC1C c1(CCC(=O)N(CCNC(C2C(=C)CC2)=O)CCc2ccccc2)c[nH]c(=N)[nH]1 C1(C)(CCCC(=O)NCCN(C(c2cncc(C)c2)=O)C2CC2)NC(=O)NC1=O c1(C(N2CCCC(F)(CNC(C3CCCC3)=O)C2)=O)cc(F)c2ccccc2c1 N1(C(c2cc(C)c(F)nc2)=O)CC2(C1)SCCC2NC(=O)C=C1CCCC1 C(CCCC(=O)NCC(C)(C)OCCNC(=O)CCc1ccccc1O)OCC Cc1nc2ccc(C(=O)NCC(F)CNC(c3ncnc(C)c3C)=O)cc2[nH]1 C1(CC=C)(C(=O)NC2CCC2CNC(=O)COC2CC=CC2)CCOC1 c1(CCC)cnnc(C(N2CCC(C3CCCN3C(C3CC3OC)=O)CC2)=O)c1 c1(C(=O)Nc2cnc(I)c(Cl)n2)nnc2ccc(-c3cccc(I)c3F)cn12 C1(C(C)(C)C)COCC1C(=O)NCC=CCNC(=O)C(O)CC1CCCC1 N1(C(C(C(C)C)OC)=O)CC2OCCN(C(c3cc4cc(Cl)sc4[nH]3)=O)C2C1 CC(O)C(C)(C)C(=O)NCC1(CNC(C2(CN(C)C)CCC2)=O)CC(F)(F)C1 C12(NC(C3(c4ccon4)CC3)=O)CC1CN(C(=O)CN1CCC(O)CC1)C2 C(C)(C)(C(C)CC(=O)NC)NC(C1(CC(=O)Nc2nc[nH]n2)CC1)=O.COC CC(CCC(C)(C)C)C(=O)N1CC2(CC(NC(=O)CCN(S(C)(=O)=O)C)C2)C1 c1(CC)nnc(CNC(c2n[nH]c(O)n2)=O)n1C CC(C)C(CCNC(C1(C)CNC(=O)C1)=O)NC(=O)CCn1cccn1 C1(CNC(N(C)CC2CC(OC)C2)=O)CCCN1CC(F)(F)F C1(O)(CCNC(c2cc(OCC)no2)=O)CCCN(C(C2CCCC23CC3)=O)C1 C1(NC(c2cn(C(C)C)nc2)=O)C=CCN(C(c2cc(C3CC3)nn2C)=O)C1 C1(C(N(CCOCCCN(C(C(C)OCC#C)=O)C)C)=O)CCCN(C)C1 c1(C(N(CCNC(C2CC(OCC)C2)=O)CC)=O)ccc(C2CC2)nc1 c1(CNC(c2nc(C)oc2)=O)ccc(CC(CO)NC(C23COCC2C3)=O)cc1 c1(OC)c(F)ccc(F)c1C(=O)NC1COCC1CNC(C12CC1C2)=O C=CC1(CO)CCN(C(=O)C(CCOC)NC(c2cccn2C)=O)CC1 c1(CNC(C2(F)CCCC2)=O)ccc(SC(F)(F)F)cc1 C1(CC(=O)NC(c2ncnn2C)C)CC2(C1)CN(C(C1CCCC1)=O)C2 C1(C(N2CC(CC=C)(NC(=O)C(F)=CC(C)(C)C)C2)=O)CC2(COCCO2)C1 Cc1cc(C(=O)NC2(C)CC(NC(c3cc(=O)n(C)cn3)=O)C2)c(Cl)cc1F Cc1cnn(C)c1CC(N1CC2C(CC(=O)NC3COCC3C)C2C1)=O CCC(C)(C)C(=O)N1CC(NC(C2CCC(C)(CC)O2)=O)C(CC2CC2)C1 C1(CC(=O)NCCN(CC(C)O)C(C23COCC2C3)=O)CC2(CC2)CO1 c1cnc(O)c(Cl)c1.N1(CC)CCN(C(N)C2CC2)CC1 C1(CC)CN(C(=O)C(Cc2ccsc2)NC=O)CCC1NC(=O)C(C)(C)SC c1(NC(=O)NCc2cccnc2Br)csc2ccncc12 c1(C(C)C)occc1C(=O)NC1CCCC1NC(=O)CCCc1ccccc1 CC1CCc2[nH]c(=NCc3cc(C#N)cs3)[nH]c(=NCCCC(N)=O)c2C1 N1(C(C2CCC(OC)CC2)=O)C2CCC1C(C)C(NC(C1CCCO1)=O)C2 N1(C(c2cnn(C)c2Cl)=O)CC(NC(=O)CC2(CN(C)C)CCC2)C2(CC2)C1 CCCCCCNC(=O)C(c1cc(C)co1)N1CCC(C(N)=O)C1 C1(C(N2C(CC(C)(C)C)CC2)=O)CCN(C(c2cnc(N)cn2)=O)C1(C)C C1(C(N(C)CC2(O)CCN(C(=O)CC3(O)CCOCC3)C2)=O)CC(=O)NC(C)C1 C(CCSC)(C(=O)NCC(n1cc(CC2CC2)nn1)C)NS(CC)(=O)=O.C1(C)CC1 C1(NC(C2N(C(C)=O)CCC2)=O)CCN(C(=O)CC2CCCCC2O)C1(C)C C1(CCNC(C(C)OC)=O)CCCN1Cc1ccn(C2CCCCC2)n1 CC1CN(C(C2CN(S(C)(=O)=O)C2)=O)CCCN1C(c1ccc(C(F)(F)F)[nH]1)=O c1(C(=O)NC(C2(O)CN(C(C3CC4C=CC3C4)=O)C2)C)c(F)ccc2[nH]ccc12 Cc1ccc(CNc2ccc(C(N3CCCC3(C)C)=O)nc2)cn1 n1(CC(=C)C)c(N2CCC(O)(CN(C)C)C2)nnc1-c1cccc(C)c1 CCC(CCC(=O)NCc1ncccc1C)NC(=O)C(OC)OC C1(CNC(CCOCCC)=O)CC(O)CN1C(=O)C(O)C1CC1 C(=O)(CCCCOCCC)N(CCC(=O)N1CC(CCC)C1)CC=C N1(CCC)CCC(C(N2CC=CC(NC(c3nccc(C)n3)=O)C2)=O)CC1 CCC(C(=O)OC)C(=O)NCC(O)CN(C)C(C1C=CC=CC=C1)=O C1(C(=O)NCCN(C(=O)CC2CCC(C)(C)C2)C)CCn2cncc2C1 Cc1c(CC(=O)NCC2(O)CC(NC(C3(C)CC4CC4C3)=O)C2)cnn1C C1(NC)CCCC2(CCCC2)C1.C1C(C)NC(=O)N1CCO.CC c1(C(=O)NCC2CC(NC(C3C(CC)C3)=O)C23CCC3)nc2c(s1)COCC2 c1(OC(C)C)cc(C(N)=O)c(-c2cn(C)nc2C(=O)Nc2cccc(O)n2)cn1 CCC(CC)C(CN1CCCC1)N1CCC(c2ccc(C(=O)NC)cc2)CC1 CC1(C)CCC=C(C(=O)N2CCC(Cn3cnc4ccccc34)C2)C1 c1(CN(CCN(C(CN(CCC#C)C)=O)C)CC)cc(N(CC)CC)nc(Cl)c1 C1(CNC(C(CCC)NC(c2ccc(Cl)s2)=O)=O)CC2CC1CC2O N1(C(C(C)(O)C2CC2)=O)CCC2(CCCCN(C(=O)CCS(=O)(=O)C(F)(F)F)C2)C1 C(=O)(CC(CC(C)C)NC(c1[nH]cc(C)c1C)=O)NCc1ncc(C)nc1 C1(NC(C(C2CCCC2)NC(C)=O)=O)CC2(NC(=O)C(C)OC(C)C)COC1C2 C1(CC)CCCCC1C(=O)NCCN(CC(C)O)C(c1cc(C)sc1N)=O Cc1nn(C(C)(C)C)c(C)c1C(=O)NCCCN(C(=O)C(C)P(C)(C)=O)CCO c1(OC)ccc(C2(C(=O)NC3CCC3NC(C3CCCSC3C)=O)CC2)cn1 C1(NC(C=C(C)C(F)F)=O)C=CCCC1C(=O)N(C1CCC1)CCC1CC1 C1(C(=O)NCC2COCCN(C(C3N(C)CCCC3)=O)C2)Cc2ccccc2C1 c1(C(C)C)cc(F)cc(F)c1.c12nc(n(CC3CC3C)n1)-c1cnn(c1)C2 c1(CC(N2C(CNC(C(C)CO)=O)C(C)(C)CC2)=O)cccc2c1OCO2 n1(CC)nc(C)c([N+](=O)[O-])c1NC12CCC(CC1NC(=O)CC1CC3CC3C1)C2 C(=O)(C(O)C(C)(C)C)NCCC(=O)NCC(C)(C)CNC(=O)OC1CCC1 c1(C(N(CCC(C)(C)NC(C=CC=CCC)=O)C)=O)cc(Cl)ccc1OCCC c1(OC)ccc(Br)c(N)c1C(=O)NCC(C)NC(c1cccnc1OC)=O c1(CNC(C2CN(C(c3ccncc3)=O)CC2O)=O)c[nH]c2cc(Cl)ccc12 N1(C(C(C)OC)=O)CCCC2(C1)CN(C(c1n[nH]c3c1C(=O)CCC3)=O)CCO2 c1(CC2(C)N(C(C(C(=O)OC)C)=O)CCC2)ccc([N+](=O)[O-])cc1 C(=O)(C1=CCCC1)NC(c1ccc(F)cc1)C(=O)NC1(C)CSC1 C1(CC(=O)NCC(=CC(N2C(COC)C=CC2)=O)C)CCOC1(C)C C(CS(=O)(=O)CC(=O)NC1COC2(C1)CN(C(C1CCSCC1)=O)C2)OC c1(CC(N2C(C(N3CCOC(CO)C3)=O)CSCC2)=O)c(F)cccc1F N1(C(C2(CC)CCC2)=O)CCC2(COC(CNC(c3nc(C)sc3C)=O)C2)C1 c1(CC2C(=O)N2)cccc(N)c1.c1(C2N(C(C)(C)C)CC2)ccccc1 C1(CNC(C2(NC(CC(=C)C)=O)CC2)=O)CCCCN(C)C1 N1(C(c2n[nH]c(CC)c2C)=O)CCCC(F)(CNC(C2C3COCC23)=O)C1 c1(C(N2CCC(C(C)NC(c3c(C)coc3C)=O)C2)=O)ccc2cnsc2c1 CC(C)C(C(=O)N1CC(CNC(=O)C(C2CC2)C2CC2)C1)N1CCCS1(=O)=O c1(C(=O)NCC2C(NC(=O)C=CCF)CCCC2)ncn2ccccc12 C1(C(=O)NC(CC2CCN(c3snc(CC)n3)CC2)C)CCc2ccccc2C1 c1(C(=O)NCCc2cnc(NS(=O)(=O)c3nccs3)s2)cc(Cl)ccc1O Cc1cc(NC(C2CC(C)N2C(=O)C(c2cncnc2)C)=O)cc(C)c1 CCC(CC(=O)N(CCCNC(C1CCN(c2ccn(C)n2)C1=O)=O)CC)SC CC(C(=O)NCC(O)CNC(c1cnc(C(F)(F)F)nc1)=O)P(C)(C)=O CC(C)C(C#N)C(=O)N1CCC(C(=O)NCCc2ncon2)C1(C)C c1(C(=O)NC2(CO)CN(C(C(C)OCC#C)=O)C2)cnc2[nH]cnc2c1 N1(C(CC2(N(C)C)CCC2)=O)CC(C(=O)NC2CC(O)C23CCC3)C2(CCC2)C1 c1(CNC(COC)CS(=O)(=O)N2CCNCC2)ccc2nc(Br)nn2c1 c1(-c2cc(C#N)c(F)cc2)ccc2cc(C(N3CC4(COC4)C3)=O)[nH]c2c1 C1(C(N2CCC(CC(=O)NC(c3cscn3)C)CC2)=O)CC(=O)OC1(C)C C(=O)(C(O)CC(N)=O)N1CC2C(CNC(CN(C3CC3)CC)=O)(C2)C1 c1(CC)cn2c(C(=O)NC3CC(NC(=O)N(C)C)C3(C)C)cccc2n1 N1(C(C(C2CCOCC2)C)=O)CCC(C)N(C(c2ncnn2C)=O)CC1 C12(C(=O)NC(CC#C)C(=O)NCc3csc(C)n3)CC(C)(CCO1)C2 C1(C(=O)NC2CN(C(c3ccn(CCC)n3)=O)CC2C)CCn2nnnc2C1 S(=O)(=O)(c1ccc(N(C)Cc2ccco2)cc1Cl)NC(C1CCCO1)COCC n1(CCSc2nnc(C)n2-c2ccccc2)c(C)c(C)n(C(C#N)C(C)(C)C)c1=S C1(CNC(=O)NCc2cnn(CCc3ccccc3)c2)CC(Cl)=NO1 CCCC(CC(=O)NC1CC(C2CCC2)C1)NC(=O)CC1(O)CCC1 Cc1cc(CCC(=O)NC2CCCC2NC(=O)C=C2CCCC2)cc(C)c1 C1(NC(c2cc(CC)no2)=O)CCN(C(=O)CC2(C)CC2)CC1F C1(=CNN2CC3CN(c4ncc(Br)c(C)n4)CC3C2)CC2(CCOCC2)CO1 C(C(C)(C)CC(=O)N1CCC(CCNC(C23CCC2C3)=O)C1)N(C)C N1(C(C2(COC)CN(C(=O)C(F)(F)C(C)O)C2)=O)C2C=CCC1CCC2 N1(C(Cc2c(C)non2)=O)CC(O)CC1(C)C(=O)NCc1ccc(C2CC2)o1 CCCCCC(O)CC(=O)NC1(C)CC(C(=O)N(C2(CO)CC2)C)C1 N1(C(CCC(C)=O)=O)CCCC2(NC(c3ccoc3C)=O)CC2C1 Cn1cnc2[nH]c(=NCCNC(c3ccccc3N3CCCC3)=O)nc(O)c12 c1(C(=O)NC(CC=C)CNC(c2cc(C)c(Cl)c(C)c2)=O)ccc2nncn2c1 c1(OC)cc(C(=O)NCC(C)CNC(=O)C(O)Cc2ccccc2)ccc1F C1(CC(=O)NC2(C(=O)N(C)CC3CCCCC3O)C(C)C2)CCCC(C#N)C1 Cn1nnc(CNC(C2CCCC2F)=O)c1C(=O)N(C1CC(C)(C(C)(C)C)C1)C1CC1 N1(C(COCCCC(C)C)=O)CCOC(C(=O)NCC2CCC(=O)N2)C1 C(CC(O)C(=O)NCCC1CCCCN1C(C1CSCC(=O)N1)=O)SC c1(C(=O)NC(C(C)NC(CC=CCC)=O)C)ccccc1COC C1(F)(CNC(C2CCCC2C(F)F)=O)CCN(C(C2SCCS2)=O)C1 c1(NC(=O)NC2CCC(=O)NC2=O)nccc2c(Br)cccc12 C1(NC(CCNC(C)=O)=O)CCCC1CC(=O)NCCC1C=CCC1 N1(C(C(C)OCCOCC)=O)CC(F)CC1CNC(c1c[nH]c(=O)cn1)=O C(=O)(CC(O)CNC(=O)Cc1cccc(O)c1)N(C(C#C)C)CCCC c1(C2(NC(C)C(C)(C)F)CC2)c(F)cccc1F C(=O)(C(=O)C(C)(C)C)N1CC(NC(C(c2c(OC)cccc2)C)=O)C(C)C1 N1(C(CSC)=O)CCC(NC(c2cc(C)ccc2Br)=O)CC1C N1(C(=O)COc2ccccc2)CCC2CCCN(C(=O)Cn3nnc(=O)[nH]3)C2C1 Cc1cc(C)c(C(=O)NCC2CC(NC(=O)C(C)Oc3ccccn3)C2)[nH]1 Cc1cc(=NC(=O)C(=O)N2CC3CCC2C(NC(=O)CN2CCCC2=O)C3)[nH]o1 Cn1ncc([N+](=O)[O-])c1N1CCOC(C)(CNC(=O)CSCC2CCCCO2)C1 c1(OC)ccc(OC)c(CC(=O)NC2CCC(C(=O)Nc3cc(Cl)cc(Cl)n3)C2)c1 Cc1cc(Br)ccc1C(=O)NCC12CC1CN(C(c1cnc(O)nc1O)=O)C2 C1(NC(CC2CC(NC(C3CC(=C)C3)=O)C2)=O)CCC(C)(COCC)C1 c1(NC(=O)CN2CCCC2)cccc(NS(=O)(=O)CCc2ccccc2)c1 Cc1cc(C(N2CCN(C(C3CC4(C3)CC4F)=O)CC2C(F)F)=O)cc(=O)n1C C(CC(C(=O)N1CC(NC(c2csnc2Cl)=O)C(F)C1)NC=O)SC c1(-c2nc(-c3c4ccc(OC)cc4oc3)sn2)ccc2c(c1)CCN(C(C)=O)C2 S(=O)(=O)(c1ccc2oc(O)nc2c1)NC(c1cc(Cl)ccc1Br)C C1(C(=O)NCC2N(C(C3CN(S(C)(=O)=O)C3)=O)CC2)CC2(CCCC2)C1 C1(C(N(CCN(C(=O)C(C)OCOC)CC)CC)=O)CC2(CC2)CN1C C1(C(=O)NC2CCCN(C(CCn3c(C)cc(C)n3)=O)C2)CCOCC12CCC2 CC1CN(C(=O)CCC2CCCCN2C(c2sc(Cl)nc2Cl)=O)CC(=O)N1 N1(C(C(COCC)(C)C)=O)CCC(NC(c2ccc(C)nc2C)=O)C(F)C1 C1(NC(C(C)O)=O)CC2(C1)CC(CNC(c1cn3c(n1)SCC3)=O)C2 C1(C(N(C(CN(C(c2cn(CCOCC)nn2)=O)C)C)C)=O)CCCC(=O)N1C Cc1nc2cc(C(=O)NC(C)CCNC(c3cc(C(F)(F)F)ns3)=O)cnc2s1 C1(NC(C(F)=C(C)C)=O)CCN(C(=O)C(CO)c2ccccc2)C1(C)C C1(C(=O)OCC)CC2CC(C(N3CCC(Br)CC3)C)CC2C1 O=[N+]([O-])c1cc(C(F)F)c(Cl)cc1N1CCOC(Cc2nc3cnccc3s2)C1 C1(C(N(CCC(=O)NCCC2CC(C)C2)CC2CC2)=O)CCN(C)C1 C(=O)(C(C)(C)C1=CCSCC1)N1C(CN(C(CC=CC)=O)C)CCC1 c1(C(=O)NC(C(C)C)C(C)NC(c2c[nH]c(Br)c2)=O)nnc2n1CCCC2 c1(CC(C(=O)OC)NC(c2cc(Cl)cnn2)=O)c(C)nc2n(c1=O)CCCC2 N1(C(c2c(CC)[nH]cc2)=O)CCCC(NC(C2(C)CC(C3CC3)=NO2)=O)CC1 C1(CCN(C)C)C2CC1CN(C(=O)CCC(N)=O)C2.c1ccc(C=O)cc1 Cn1c(NC(C2CC2c2ccc(Br)s2)=O)cc2ccsc12 CC1(C)CN(C(=O)CC2(C#N)CC2)CCC1C(=O)Nc1ccc2nonc2c1 C1(NC(C(CN(C)C)N(C)C)=O)CCCCN(C(=O)CN)C1 c1(CN2CCC(N(C(C(CC3CCC3)OC)=O)C)CC2)c[nH]c2ncc(C)cc12 c1(C(=O)NC2(CCNC(C3CC(C)OCC3)=O)CCCC2)cc2c(nn1)CCC2 C(C(CC(F)(F)F)NC(=O)C=C(C)C1CC1)NC(c1c(CC)occ1)=O Cc1oc(C(C)(C)C)cc1C(=O)NC1CCN(C(=O)CC2CN(C)C2)CC1 n1(CC(=O)NCC2CN(C(C(CC)OCC)=O)CC2C)cccc(N)c1=O c1(CC)noc(C)c1CC.C1C(CO)CNC(=O)C2CC(C2)CC(=O)N1 Cc1c(C(=O)NC2CC2NC(C2CC(=O)N(CC3CC3)C2)=O)cncc1Cl CC1(C)CC(=O)OC1CNC(C1CC(CNC(=O)CC2(N(C)C)CCC2)C1)=O CC(CN=c1nc(N2CCN3CC(O)CC3C2)c2c(ncn2C)[nH]1)C(C)(F)F c1(CC)cnc(CNC(C2CCN(C(=O)Cn3nnnc3-c3ccsc3)C2)=O)s1 C1(CNC(C(CCC)N(C)C)=O)COC(C)(C)CN1C(c1cncnc1)=O n1(CC(=O)NCC2(F)CC(NC(Cc3n(C)cnc3)=O)C2)cc(Br)ccc1=O c1(C(=O)NC2CC23CCN(C(c2cncs2)=O)CC3)ccc(Br)c([N+](=O)[O-])c1 C(=O)(C1Cc2ccccc21)N1C(CNC(c2cc(-c3ccccn3)ns2)=O)CCC1 C(=O)(C(COC)CC(C)C)NCCCOCCN(C(c1c(OC)cccn1)=O)C C1(SC)CCC1C(=O)N(CC(C)NC(=O)CC=CC(C)(C)C)C C1(CNC(c2cc(OC)ncn2)=O)CC(C)(C)CN1C(C1CC(C)OC1C)=O C1(NC(C(C2(O)CN(C(CC3(C)CCCCC3)=O)C2)F)=O)CCCCC12CC2 C1(OC)CN(C(C2CC2(C)Br)=O)CCC1NC(=O)CCC(C)(F)F C1(CNC(=O)CC2CCC(O)C2)CC2(CC(C(=O)NCC3CC34CCOC4)C2)C1 c1(CC(C)C)ccc(CC(N2CCC(C)(NC(C3CC=CC3)=O)C2)=O)cc1 C1(F)(CNC(C2CCCS2)=O)CN(C(c2occc2C2CC2)=O)C1 CC(C)CC(C(=O)NCC(C)(C)CCNC(c1ccoc1Br)=O)C(C)C c1(C(N2CCC(NC(c3ncn(CC)c3)=O)C(F)C2)=O)cc(=O)c(OC)cn1C Cc1c(Cl)nc(C2CC2)[nH]c1=NCC(O)CNC(c1cc(CC(=O)O)ccc1Cl)=O N1(C(CCOc2cncc(C)n2)=O)CCCCCC1C(=O)NC(C)C C1(C)(NC(C(c2ccc(OC(F)(F)F)c(Cl)c2)C)=O)CCCCC1(C)C CC(C(=O)OC=CC(=O)N1CC(n2cc(COCCO)nn2)C1)S(N)(=O)=O Cc1oc(S(N)(=O)=O)cc1C(=O)NC1CCC2COC1O2 c1(COC)cc(C(=O)NCc2ccoc2C(=O)NC2CC2C(C)(F)F)on1 C1(CCNC(C2(C)CCC(C)C2)=O)CN(C2CCc3cc(Cl)ccc32)C1 CCCCC(CC)C(=O)N1CC(OCCCNC(=O)C#CC2CCC2)C1.C1CO1 N1(C(c2ccc(CC3CCC3)cc2)C(=O)NCC)CCOC2CCN(C)CC12 CC(C)(C)C(C#N)C(=O)N1CCCC1C1(C(N2CC3(CCNC3=O)C2)=O)CC1 c1(OCC)nc(CN(CC)CC2CC3OC2C2CC32)cc(O)n1 Cc1cc2scc(C(=O)NC34CCC(CC3NC(c3c[nH]nc3N(C)C)=O)C4)c2s1 c1(-c2cc(C(=O)NC(CC#CC)CO)n[nH]2)ccc(OC)c2cccnc12 Cc1cc(Cl)ccc1OCC(N1CCCCC1c1cn(-c2nc(C)c(C)s2)nn1)=O c1(NC(C2N(C(CC(C)(C)N)=O)CC2)=O)c(F)ccc(F)c1[N+](=O)[O-] S(=O)(=O)(c1cccnc1)NCC(N1CCC(CN(CCC(C)C)CC(C)C)C1)=O c1(N(C)C(c2nnnn2C2CCCC2)CC2CCOC2)cccc(CCC(=O)NC)c1 N1(C(=O)CCOCCCO)CCC(N(C(C2(O)CC2)=O)CC2CC2)C1 CC(C(=O)N(C1CCCCCC1)CCNC(C1CC(CC2CC2)C1)=O)C1=CCCC1 C(CNC(C1(C)CC1C)=O)(CCNC(C1CCCOC1)=O)OC C(=O)(C#CC1CCCOC1)N1CCN(C(CCc2nc(=N)[nH][nH]2)=O)C(C2CC2)C1 C1(NC(C2OCC(C)(C)C2)=O)C2CCC1N(C(=O)C(C)(C)OCC(F)(F)F)C2 c1(C(=O)NCC2CN(C(C(CC)F)=O)C(C)(C)C2)c[nH]c2cccc(C)c12 c1(CC(=O)NCC(CNC(CC2N(CC)CCC2)=O)OC)ccc(F)cn1.SCC c1(-c2cn(CC)c(=O)cc2)cc(C(=O)NCCCSC)c2[nH]ccc2c1 c1(C(=O)NCCNC(C(C)NC(c2ccc(C)cc2)=O)=O)ccnc2[nH]nnc12 N1(C(C2CCC(CC)CC2)=O)CCC(NC(C2(n3cccn3)CC2)=O)CC1C c1(C(N2CCCC(CNC(CC(CCC)CC)=O)C2)=O)c(F)ccc2c1OCO2 C(=O)(C1CCc2ccccc21)Nc1scc(C(=O)NC2(COC)COC2)n1 C1(C(C)(C)NC(C(CC)=CC)=O)CCN(C(c2ccc(SC)cc2)=O)CC1 CC(C)CC(CCO)NC(=O)C(CNC(c1cc(Cl)ns1)=O)C(C)C Cn1nc(Br)cc1CC(=O)NC1(C)CC(NC(=O)CN2CCCC2=O)C1 C1(C(N(CCC#C)CCO)=O)CCN(C(=O)C(=O)C(C)C)C(CC)C1 Cc1nc(CCCC(=O)NCCC(C)N(C)C(c2coc(Cl)n2)=O)cs1 C=CC1(C(N2CCC(NC(=O)C(C)CCOC)C(F)C2)=O)CCOCC1 C(=O)(C(C)(C)CCNC(=O)CC1COC(=O)C1)NCCC1N(C)CCC1 C1(COC)(NC(C2CCN(C)C2)=O)CCCN(C(c2snnc2C(C)C)=O)C1 N1(C(CC2N(C(c3cn(CC=C)nc3)=O)CCC2)=O)CCC(C2CCCC2)C1 C(=O)(CC(C)c1ccco1)NCC1CC(NC(C(C)=CC2CC2)=O)C1 N1(C(C(N2CCCC2=O)C)=O)CC2CC(C1)CN(C(=O)Cc1ccc(F)cc1F)C2 N1(C(C(C)(C)SC)=O)C(CNC(=O)CC2CCCO2)CC2COCC12 CCC(C)C(CC(=O)N1CCC(CO)C(C)C1)NC(C1(COC(C)C)CC1)=O C1(C(=O)Nc2c(C(=O)OC)scc2)CCCCN1C(=O)Nc1cc(CO)ccn1 C(=O)(C(C)(COC)NC(C1CC1CCNc1ccc(NS(C)(=O)=O)cc1)=O)OC CC1(C)C2CCC1(OCC1CCSC1(C)C)CC2.c12cn(nn1)C1CN(C1)C2=O C1(NC(c2cnc3ncccn23)=O)CCCC12CN(C(c1ncccc1F)=O)C2 N1(C(c2cccc(C)c2F)=O)CC(CNC(=O)CC(F)F)CC12CCC2 C(CC(C)(C)CC(=O)NCC(C)CN(C(=O)Cn1nc(C)n(CC)c1=O)C)OC C(=O)(C#CC1CCCO1)N1CCC(CCNC(CCNC(c2cccs2)=O)=O)C1 N1(C(C2C(O)CCN(C(c3nc(C(C)C)oc3)=O)C2)=O)Cc2cccc(F)c2C1 C=CCCCCCCCC(=O)NC1CN(C(=O)C(C)(CC)C(N)=O)CC(F)(F)C1 C1(NC(C2(OCC)CCOC2)=O)CN(C(C2(C)CC(F)(F)C2)=O)C2(CCCC2)C1 Cc1ncnc(O)c1CC(N1CC(NC(=O)Cc2cncnc2)C(F)C1)=O C1(C(=O)Nc2c(CNC(C(C)P(C)(C)=O)=O)cccc2)CCn2cncc2C1 Cc1cc(C(=O)NC2CC(C(=O)Nc3ccc(C(F)F)nc3)C2)nn1CCO C1(N(C(C(C)(C)O)CO)C(c2ccoc2Cl)=O)CCC2(CCNC2)CC1 C12(CC(=O)OC)CC(C1)C(NC(c1ccc(OC(C)(C)C)o1)=O)CO2 N1(C(C2(CNC(c3c(C)n(C)nc3)=O)CCCCC2)=O)CCC(O)C(F)C1 C1(OC)CC(CCNC(c2ccnc(S)c2)=O)N(C(c2ccnc(C)c2)=O)C1 C1(C(=O)NCC2N(C(c3nn(C)c(CO)c3)=O)CCOC2)CCC2CC2CC1 C#CC1CC2CCC1N(C(=O)C=CCNC(C1CCC(OCC)CC1)=O)C2 C(=O)(CC(O)CC(C)(C)C)NCCCC(C)NC(COc1c(CC)cccc1)=O N(C1c2ccccc2CC1NC(=O)C(O)CF)C(Cc1cn(C(C)C)nc1)=O C(=O)(C1=NNC(=O)CC1)NC1(CCCCNC(C#CC(C)C)=O)CC1 CC1C(NC(c2cnc(C(C)(C)C)s2)=O)CCCN1C(=O)Cc1cn[nH]c1 N1(C(c2cn(CCOC)nc2)=O)CCN(C(=O)CN(CCCF)C(C)C)CC1 C1(NC(C2(C(N3CCC(CC)C3)=O)CC2)=O)CC(F)(F)CS1.N(C)C CC1CCCC1(C)C(=O)N(CC(C)NC(=O)Cc1ccsc1Cl)C C12(CNC(C(C)Nc3nccs3)=O)CCCCC1N(C(c1cnsc1)=O)CC2 CCCC(C(=O)NC1COCCC1NC(=O)C=CC(C)(C)SC)NC(C)=O c1(C(C)=O)ccc(C(=O)NCC2CCCC2NC(c2snc(O)c2Cl)=O)cc1F Cc1cc(C2CCC2)ncc1C(=O)NC(CNC(=O)C(C)c1cccs1)C1CC1 Cc1cc([N+](=O)[O-])cc([N+](=O)[O-])c1N1CCCC(NC(c2cocc2C)=O)C1 C=CC12CC(CCN1C(=O)Cc1c(C)n[nH]c1C)C2 Cc1nc(C(N2CCC(CCCCCNC(=O)C(C)NC(N)=O)CC2)=O)cn1C CCCCCCCCC(C)C(=O)N1CCC(NC(=O)Cc2nc[nH]n2)C(C)(C)C1 C12CCC(=O)N1CNC(=O)C2.C=C(CN)CCNC(c1n[nH]c(CCC)n1)=O c1(C(C)C)cc(C(N2CCCCC2CN(C)C(C2(O)CC2)=O)=O)nc2ncnn12 CCCCC(C(=O)N(C(C)CNC(=O)CCF)C)N(C)C c1(OC)ccc(C(=O)NC(C2(CNC(=O)C(C(C)O)N(C)C)CC2)C)c(F)n1 C(=O)(N1OC2CC1C(O)C2O)C1(CF)CCN(C(c2c(OC)nccc2)=O)C1 c1(N(C2CCN(C(Cc3c(C)noc3)=O)C2)C)ncnc(O)c1Br N1(C(C23N(C(C(C)NC=O)=O)CCC2CCC3)=O)CCCC(C2CCC2)C1 Cc1c(C(N2CC3(CC(NC(c4ccco4)=O)C3)C2)=O)cnc2ncnn12 N1(C(c2c(CC)onc2C)=O)CCC(F)(C(=O)Nc2ccc(C)nc2)CC1 n1(CC(=O)NC2CCC(F)(CNC(c3c(C)ncnc3)=O)C2)cnc([N+](=O)[O-])n1 CC(CC(F)F)C(=O)NCC1CCCCCN1C(c1ccnc(C(C)(F)F)c1)=O C(C)(C(C)(C)NC(=O)Cc1csnc1C)NC(CC)=O C1(CNC(C(=O)Nc2c(C(=O)OC)cccc2)=O)CCNC2(CCCC2)C1 CCC(C(N)=O)NC(=O)CNC(=O)C(C)(C1(C)CC1)OC C(=O)(C(=O)N=c1cc(C)n(-c2ccc(C)cc2)[nH]1)Nc1cnc(C(=O)NC)nc1 N1(CC(N2CCC(O)(CCNC(C3N(C)CCOC3)=O)C2)=O)CCC(=O)NC1=O c1(NC(C2N(CC)CC3C2C3(C)C)=O)cc([N+](=O)[O-])cc(C(=O)OC)c1O C(=O)(C1=C(C#N)CCC1)NCC1CCCN(C(c2ccc(CSC)o2)=O)CC1 N1(C(c2cn(CC=C)nc2)=O)CC2(CCN(C(=O)CC3CC(C)=NO3)CC2)C1 C(C#Cc1ccccc1Cl)N(C1(C#N)CCCOC1)CC=C N1(C(C(C=C)(C)C)=O)CC(NC(=O)C(C)OCc2ccccc2Cl)CC2(CC2)C1 c1(CNC2(c3nnnn3C3CCCCC3)C(C)CSC2)ccc2nonc2c1 Cc1cc(=NCC2CN(C)C2)[nH]c(=NCCOCC2CC2)[nH]1 C=CC(CC)CC(=O)N1CCCCC1CN(C(=O)C(C)(C)C(F)F)C C1(NC(C(C)CO)=O)CCCC12CN(C(c1cc(C(F)F)ccn1)=O)C2 N1(C(c2c(C)cn(C)c2)=O)CC2CC(NC(c3cnn(CC(C)C)c3C)=O)C1C2 c1(CC)sc(C(=O)N(CCN(CC(C)O)C(c2cccc(F)c2)=O)C(C)C)cc1C C1(C(N2CC=CC(NC(C(C)(C)C)=O)C2)=O)CCc2nncn2C1 C(C)(C(=O)NC1CCCN(C(=O)Cn2nc(C)n(C)c2=O)C1)(C(C)C)OC c1(C(=O)NCC2CN(C(C=NOC)=O)CC2(C)C)cccc2nc(S)oc12 C1(C(N(CC(N2CC(N(C)CCO)C2)=O)CC2CC2)=O)CCN(C)C1 C1(C(=O)CC=CCN(c2ccccc2F)C(C2(C(C)(F)F)CC2)=O)C(Cl)(Cl)C12CC2 C1(C(=O)NCC(CC(C)C)OC)(CNC(C(C)NC(CC)(C)C)=O)CCCCC1 c12cc(ccc1[N+](=O)[O-])NCCN(C(C)Cc1cccn1C)C2=O.C(CO)OC C1(CNC(C2(CC=C)CCC2)=O)C2CCC(C2)N1C(C1CCCCN1C)=O C1(CC#C)(C(N2CC(OCCNC(C3CCS3(=O)=O)=O)C2)=O)CCOCC1 C1(NC(CC(C)O)=O)CCC2(CCN(C(=O)CCNC(=O)OC(C)(C)C)CC2)C1 Cn1ccc2c(NC(C3CCN(Cc4cccc5ccncc45)C3)=O)ncnc12 C1(CNC(C(COC)(F)F)=O)Cc2ccccc2CN1C(c1ccc(Cl)cn1)=O c1(C(=O)NC(C2CCCCN2C(c2ccc[n+]([O-])c2)=O)C)c(F)cc(Cl)cc1F CC(C)CC(O)C(=O)N1CC=CC(C(=O)N(C2CCCC2C#N)C)C1 C1(C2CCCN(C(c3cnc(Cl)c(F)c3N)=O)C2)(NC(c2c(C)con2)=O)CC1 c1(NC(N(C(C)C)Cc2cnn(C)c2)=O)nnc2n1CCCCC2 c1(CN(CCCNC(c2cn(C)nc2)=O)C(=O)COCCCO)ccccc1Cl c1(C(N2CC(=C(CNC(c3nc(CC)oc3)=O)F)C2)=O)onc2cc(C)ccc12 C(=O)(C1CCCc2n[nH]cc21)N(CCCNC(c1c(C)oc(C2CC2)n1)=O)C1CC1 C1(CNC(C2N(C)C(=O)CC2)=O)CCC2(CCC2)CN1 C1(C#N)(N(CCCCCO)C(C23C(CN(C(C)=O)C2)C3)=O)CCOCC1 C1(NC(c2nc(SC)sc2)=O)CN(C(C2CCCOC2C)=O)C(C)(C)C1 N1(CCC(=O)NCC2(NC(c3cc(OC)n[nH]3)=O)CCC2)CCCS1(=O)=O C1(CCC)CN(C(C2(C)CC(C)=NO2)=O)CCN1C(c1csc(Br)c1)=O CC(C)CC(O)C(=O)N1CCCN(C(c2cccc(Cl)c2)=O)CC1 C1(NC(c2ccc(C(C)C)o2)=O)CCN(C(C2(C)CCC2)=O)CCC1CO C(=O)(C#CC1CCCCC1)N1CC2(OCC(NC(CCCC3C(C)C3)=O)C2)C1 C1(NC(C23CC(COC)(OC2)C3)=O)C2CCC1N(C(=O)C(C)(C)F)C2 C(CC)(CC(C)CO)NC(c1ccc(CNC(C2(CC=C)CC=CC2)=O)cn1)=O N1(C(C2(C)CC2(F)Cl)=O)CC2(CCCC(CNC(c3ccsc3C(N)=O)=O)O2)C1 C1(CCOC)(NC(C2CCSC(C)C2)=O)CCN(C(=O)Cn2nc(C)oc2=O)C1 Cc1cc(Cl)ccc1OCC(=O)NCC1(CCNC(C2CCS(=O)CC2)=O)CC1 C1(C)(NC(C(C)(Cl)Cl)=O)CCCN(C(c2ccc(CCO)cc2)=O)C1 N1(C(C2N(C(C)=O)CCCC2)=O)C2CCC1C(CNC(=O)CN1CCCC1=O)C2 N1(CCOCC=C)CCCC(C)(COC(=O)COCCOC)C1 C=C(Cl)CCC(=O)N1CC(OC)CC1CNC(=O)C(C(C)C)c1cc(C)no1 N1(C(C2CC(N(C)C)C2)=O)CCN(C(=O)C(F)CC2CC2)C(CC(F)F)C1 N1(C(CN(C)CC)=O)CCC(C2(O)CN(C(c3cnn(C)c3N)=O)C2)CC1 C(c1cccc(Cl)c1Cl)=CC(N1CC2C(CNC(c3nc(C)[nH]n3)=O)C(C2)C1)=O CC1(CNC(=O)Cn2ccc(Br)n2)CCCN(C(=O)Cn2nnc(=O)[nH]2)C1 c1(C(=O)NC2CN(C(c3cncc(C)c3)=O)C(CO)C2)cc(Br)c(Cl)cn1 c1(N2CC(c3ccc(C)o3)C2)ccc(S(=O)(=O)N2CC=CC2CNC2CC2)c(Br)c1 C(=O)(CCCC(=O)N(CCNC(=O)CC1CC1(C)C(F)F)C)N(CC)CC C1(CNC(C2(CS(C)(=O)=O)COC2)=O)CCC(NC(C2CC3(CCC3)C2)=O)CC1 c1(C(=O)NC2CC3CCC2O3)nnc(O)nc1O.C12(CC13CCC3)C(=O)NC2 c1(C(N2CCC(N(C(=O)CCC(=O)NC)CC)C2)=O)n[nH]c2c1CCCC2.CCN c1(SCC(=O)OC2CCCN(C(CC)=O)C2)ccc(C)cc1C N(C(=NCc1ccc(Cl)nn1)N1CCC(CCOC)C1)C(CC)CC C1(C(=O)NC(CC)CNC(=O)Cc2nc(C)cs2)C2C3CC4C1C1C2CC3C41 C12(CNC(C3CC(OC)C3)=O)CC1CN(C(c1cncc(C(F)F)c1)=O)C2 N1(CC=C(C)C(C)(C)C)CCCCC1CNC(=O)C1CC1 c1(CC)c(C(=O)NCCN(C)C(C2CCCN2C=O)=O)[nH]c(C)c1C(N)=O C1(CCNC(COC)=O)CC(F)(F)CN1C(C1CC1CC(C)C)=O CC1CC(NC(=O)CSCC(N2CCOCC2)=O)CN1C(=O)CC1CNC(=O)O1 n1(C(C2CCCOC2)C)[nH]cnc1=NCc1ncco1 CC1CCN(C(C2CCC=CCC2)=O)CCN1C(c1cnc2c(c1)COC2)=O C1(C(N2CC(CNC(c3cc(CC)nn3C)=O)C2)=O)CC(c2cnn(C)c2)=NO1 c1(OC)cccc(C(=O)N(C)CCN(C(=O)CC2(c3ccon3)CC2)C)n1 N1(C(C(C)=CC)=O)CCN(C(C2C(OCC)C2C)=O)CC1c1ccccc1 C1(C(=O)NCCCN(c2ncc([N+](=O)[O-])cc2Cl)CC)CCc2ccc(F)cc2O1 C1(COC)CN(C(c2cc(Cl)ns2)=O)CCN1C(=O)CC1CC2(CCC2)CO1 C=CCC(C(=O)NC1(C)CC(NC(=O)CC2CCCC2)C1)C(C)(C)C C1(C#CC(=O)NCC2(C)CCCN(C(=O)C(C(C)C)SC)C2)(CC)COC1 C(=O)(CCCCCCNC(=O)CC1COCC1O)NC(C)CSC(F)F C1(CC(=O)NC(C2CCCC2)(C)C)CCN(C(C2CCCN2C2CC2)=O)C1 CC(CC(=O)NCCCC(N1CCC(O)C(F)(F)C1)=O)C(C)(C)C N1(C(C2=CC(O)C(NC(Cc3cn(CC)nn3)=O)C2)=O)CCN2C(=O)CCC2C1 C1(NC(c2n(C)nc(C)c2Cl)=O)CC2CC(C1)N(C(=O)CSc1cnn(C)c1)C2 C1(CC(=O)OCC)CCCC2(CN(C(=O)Nc3ccc4cnnc(O)c4c3)C2)O1 CCN=c1[nH]c(C)c(C(N2CCCN(C(=O)CC3CCC34CCC4)C(C)C2)=O)s1 c1(C(=O)NCC(CNC(=O)CCc2nc[nH]n2)OC)sc(O)nc1C c1(N2CCC(CNC(C3CCS(=O)(=O)CC3)=O)C23CC3)nc(Cl)nc2sccc12 CC1(C(=O)NC2CCN(C(C3CC(N4CCOCC4)C3)=O)C2)CC=CCO1 C12(C(C(=O)COCC(=O)NC3CCC(COC)C3)=O)CCCC1C2(F)F c1(OC)cnc(C(=O)N(C2CCOCC2)C2CC2)cn1.C1(C(=O)ON)CC1CC(C)C n1(CC(N2CCC(NC(c3cn(C4CCC4O)nn3)=O)C2)=O)cc(CO)nn1 N1(C(c2ccc(CO)cc2)=O)CC2(CCC(C(N3CCS(=O)CC3)=O)O2)C1 c1(OC)c(-c2noc(C3CCC(C)C3)n2)cc(F)cc1F N1(C(C2N(C(C(CCCC)O)=O)CC(C)(C)C2)=O)CC2CCN(C)CC2C1 c1(C(N2CCC(O)(CNC(=O)C(F)C3CC3)C2)=O)cc2ccnc(Cl)c2[nH]1 c1(CC(C)C)ccc(C#N)c(NCCNC2CCS2(=O)=O)n1 c1(C(N2CCC(N(C(c3ccco3)=O)CC)C2)=O)ccc(C(=O)NC)c(F)c1 C(CCCCC(=O)N(C)Cc1ccccc1)NC(C12CCC(OC)C1C2)=O Cc1c(N)ccc(C(=O)NC2CCN(C(C3C4CCCCC34)=O)CC2)c1F C(CC(=O)N1CCC(C)(CN(C)C)C1)(C(F)(F)F)NC(c1c(C)nc(C)s1)=O c1(C(N2CC(NC(CC(C=C)(C)O)=O)CC2(C)C)=O)ccc(Cl)c(S(C)(=O)=O)c1 C(N=c1[nH]c(=NCCC(=O)N(C)C)c2sccc2[nH]1)c1cc(OCC)ncc1 C1(C(N2CC(F)(F)C2)=O)CC2C=CC1N(C(c1cnsc1)=O)C2 c1(N2CCCC(NC(c3c(C)ocn3)=O)(CO)C2)c([N+](=O)[O-])cccc1[N+](=O)[O-] C1(NC(C2CCC(F)(F)C2O)=O)CC12CCN(C(C1CC1c1ccco1)=O)CC2 C1(C(=O)NCC(CC#C)(C)CO)CC2(CCN1C(C1CC3(CC3)CO1)=O)CC2 N1(C(c2ccc(-c3cn(CCCN)nn3)o2)=O)CCC2CCCC2CC1 C1(C(C)(C)C)(CNC(C2CC2(C)C)=O)CCN(C(C2CCN2C)=O)C1 c1(C(=O)NCC2CN(C(C3=C(C)OCC3)=O)C2)cc(C(C)C)nc2onc(C)c12 C#Cc1ccc(C(N2CC(NC(=O)C(C)N3CCC3)CC(F)C2)=O)cc1 c1(N(C(CNC(CCc2onc(COC)n2)=O)C)C)nc(C)ccc1C(C)=O c1(OC)ccccc1C(=O)NCC1CN(C(c2cnns2)=O)C2CC12 Cc1ncn(C)c(=O)c1C(=O)NC(Cn1cccn1)CCNC(=O)C(O)C1CC1 c1(C(=O)NCC(CC)(C)NC(=O)CC(C)O)cn2cc(C)c(C)cc2n1 O=C(C1=CCSC1)NCC#CCNC(c1nccc(C(F)(F)F)n1)=O C12(C(=O)NC(C3C(Cn4cc(CNC)nn4)CCC3)=O)COCC(C1)OC2 N1(C(CSCCC)=O)CCCCC(NC(c2cn(CC3CC3)nn2)=O)CC1 C1(O)(CNC(CCN(CCCCC)C)=O)CN(C(c2cc(C3CC3C)on2)=O)C1 CCC(C)C(O)C(C)C(=O)NCC1(NC(c2ccc([N+](=O)[O-])s2)=O)CCCCN1 CC1CCC=C1C(=O)N1CC(O)CCC1C(=O)NC1CCC=CCCC1 N1(C(c2c(C)con2)=O)C2CCC(C2)C1C(N1CCC(C(C)C#N)CC1)=O C1(C(N2CCCCC(NC(c3c(C)nn[nH]3)=O)C2)=O)CCC2C(CC1)C2(F)F Cn1cc2cc(C(=O)NCC3CC3NC(c3cc(Br)n(C)c3)=O)ccc2n1 c1(CNC(=NCC)NCC(C)SC)c(F)c(F)c(F)c(F)c1F CC1CCN(CC(=O)N(CCCn2cc(-c3cnccc3Cl)nn2)C)CC1 N1(c2n(Cc3cc(C)on3)c(CC3CCC(=O)CC3)nn2)CCCC2(COC2)C1 C1(NC(CC2(NC(C)=O)CC2)=O)CC(CNC(c2ccc(F)cn2)=O)CC1O Cc1cc(=NC(=O)C(C(C)C)Sc2nc(-c3ccc4ccccc4n3)no2)[nH]o1 Cc1cc(C(=O)N(C(CC(F)F)C(=O)NCCP(C)(C)=O)C)nnc1O C(=O)(CC(O)C(C)CC)N1CCC(C=C)(C(=O)NC(c2nc[nH]n2)CC)C1 N1(C(c2nc(C)n(C)n2)=O)CC2=C(C1)CN(C(C1CN3CCCC1C3)=O)C2 N1(C(C2CNC(=O)N2)=O)CCOC2(CCN(C(c3ncsc3C(F)(F)F)=O)C2)C1 N1(C(c2coc(C3CC3)n2)=O)CCC(NC(C2(OCC)CC(C)(C)C2)=O)C(O)C1 c1(C(N(C(CNC(C2(F)CCCC2)=O)C2CC2)C)=O)ccc2nnnn2c1 C1(CC(=O)NC(CCNC(c2c(C)cnnc2)=O)C)NC(=O)CN(C)C1=O C(=O)(CC(CC(C)C)NC(=O)C(F)C(CC)CC)N(C(CCCCC)C)C1CC1 c1(C=O)cc(N(N2CCN(C(=O)CC(C)(F)F)C(CCO)C2)C)cc(C#N)c1 c1(C(C)C(=O)Nn2cc(-c3cnc(OCCN(C)C)o3)nn2)cncc(F)c1 N1(C(CCOC)=O)CCC2C1CCN2C(=O)CCn1ccccc1=O C(=O)(CC(C)C(C)(C)NC(=O)CCc1cnco1)NC(c1c(C)nc(C)[nH]1)C N1(CC(=O)Nc2cc(C(=O)OCC)sc2Cl)CCC(C(N)=O)(CC)CC1 C(=O)(C1CCCc2cncn21)N1C2CC(C(NC(c3cc(=N)[nH]cc3)=O)C2)C1 C1(C(C)C)CCNCC1.c1(NCc2cccs2)cc(O)ncn1 C1(OC)CN(C(=O)CCOc2ccccc2Br)CC1NC(c1ccsn1)=O c1(Cc2scc(C(N(C)CCNC(=O)CC3(C)CC3(Cl)Cl)=O)n2)ccccc1 C1(F)(CNC(CC2(C)CC2)=O)CCN(C(=O)Cc2cc(Cl)cc(Cl)c2)CC1 CC1(C)CCCC(NC(=O)C(C2CCCO2)NC(C2CCC(=O)CC2)=O)C1 N1(C(CSCCN(C)C)=O)CCCC(N2CCN(C(C3(C)CCCOC3)=O)CC2)C1 C(=O)(N=c1cncc[nH]1)C1N(C(c2cc(OCC)nc(Cl)c2)=O)CCC1 C(C(CCC(F)(F)F)C(=O)O)N(C(C(=O)NC(C1CCCC1O)C)=O)CCO CC1=C(C(=O)N2C(C(N3CCC3CO)=O)CCC2C(C)(C)C)CCO1 C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)NC1C2C(C)N(C(C3C(=C)C3)=O)C1C2 S1(=O)(=O)c2ccc(c(Br)c2)N(N(C)CCOCC)CC(C)N(C)CCN1.CC c1(C(N2CCN(C(C34CCC(C3)C4(C)C)=O)C3CC23)=O)ccc(C)c(O)n1.CN C1(CC(c2nnnn2C2CCC2)NC2(C(N(C)C)=O)CCCC2)CCCCCC1 c1(OCC)cc(C(=O)NC2CCN3CCC2C3)ccc1OCC1CCC1 c1(COC)cccc(C(=O)NC(C(=O)NC2(C)CCOC2)Cc2cnc[nH]2)c1 C(=O)(C(C)(O)C(C)(C)C)NC1CC(F)(CNC(c2ncc(C)cn2)=O)C1 C12(NC(CS(CC)=O)=O)CC3CC(C1)CC(NC(=O)C(C)CN1CCCC1)(C3)C2 C(=O)(C(CNC(c1cnncn1)=O)C(C)C)N(CCC(N)=O)CC N1(C(C(C=CCCC)O)=O)CCN(C(=O)COCc2cccc(C)c2)C2(CC2)C1 c1(OC)ccc(Br)c(C(=O)NC(C)(CNC(=O)CCc2ccoc2)C2CC2)c1 C1(NC(c2cc(F)c(Cl)cc2I)=O)CC2CCC(C1)N2C(c1ccc(Br)s1)=O c1(OCc2nc(CCOC)nn2-c2cc(C)ccn2)ccc(Cl)c(Cl)c1 CC12CN(C(C3CC3(F)Cl)=O)C(C(=O)NC3(C4CCC4)CC3)(C1)C2 CC1CCN(C(=O)CCn2ccccc2=O)C(CNC(C2CC2C#N)=O)C1 C1(C(=O)NCC(CO)NC(c2cc(C)n(C)n2)=O)(CC)CCC(O)CC1 N12CCN(CC1)C2=O.c1cnn(C)c1-c1ccccn1.Cn1nncc1CN1CC1 CS(=O)(=O)CCCC(=O)N1CCN(C(c2cccc(O)c2)=O)C(CO)C1 C(=O)(C(C(C)C)C(C)C)N1CCC(CC(N)=O)(NC(CCc2onc(C)n2)=O)C1 Cc1nnc2ccc(C(N3CCOCC(CNC(=O)C4=CC(C)CC4)C3)=O)cn12 c1(OCC(=O)NCC(CNC(=O)C(C)S(N)(=O)=O)OC)ccc2c(c1)CCC2 C1(C(N(CCOC)C)=O)CCCC(NC(c2nnccc2C)=O)C1 c1(CCCn2cc(CC3OCCN(C(=O)CSC(F)F)C3)nn2)cc(Cl)ccc1Cl C(N=c1nc(NC2(C)CC3CC3C2)c2c([nH]1)c(C)nn2C)c1c(C)nn(C)c1 C(C(O)C(=O)N(C(CNC(=O)CSC1CC1)Cc1ccccc1)C)SC c1(N2CCC(NC(C3CC3c3ccco3)=O)CC2)ccc([N+](=O)[O-])cc1Cl c1(C(N(C2CCCN(C(C3C=CCC3)=O)C2)CC)=O)cc(Cl)cc(Cl)c1F CC1CC(=O)NCC1C(N1CCC(CO)(CNC(=O)CSc2nc[nH]n2)CC1)=O C1(COC)(CNC(=O)COC)CCN(C2CCC2)CC1.C1(C=O)CCC=CCCC1 C(C1CCOCC1)=NC(N1CC2C(NC(=O)Nc3cccc(OC)c3)C2C1)=O c1(OC)ccc(F)cc1C(N1CCOC(CC(=O)NCc2cncn2C)C1)=O CC(=O)CCCC(=O)N1CC(O)(CNC(=O)CCOc2ccc(F)c(F)c2)C1 N1(C(c2c(C)cn(C)c2)=O)CCCCCCC1C(=O)NC(c1cccnc1O)C c1(CC(=O)NCCC(C)NC(=O)Cc2csnn2)ccc2ccccc2c1 CC1CCc2[nH]c(=NC3C=C(c4ccccc4)C3)[nH]c(=NCCOCC(F)F)c2C1 N1(C(c2snc(C)c2N)=O)CCC(NC(=O)C=CC=C(Cl)Cl)C(CO)CC1 C1(C(N(CC(CC)NC(=O)CN(C)CCOC)C)=O)CCc2ccc(F)cc2C1 N1(C(C(C)OC)=O)CCC2CN(C(C3(C(F)(F)F)CCCCC3)=O)CC2C1 N1(C(C2CC3(CC(=O)C3)C2)=O)CCN(C(C2CC=CC2)=O)CC(O)C1 C1(C(=O)NCCN(C(=O)CC2CS(=O)(=O)C2)CCC)(C(F)F)CCOCC1 N1(C(CSC(C)(C)C)=O)CCC2CN(C(c3c[nH]ccc3=O)=O)CCC2C1 N1(C(c2c(NC)cccc2)=O)CCC2(CC1)CC(C)N(C(=O)C=CC(F)(F)F)C2 C1(C(=O)NCC2OCC(CNC(CCC#CC)=O)C2)CCOCC12CCCC2 c1(C(C)NC(c2ccc(C)s2)c2nnnn2CC(F)F)cc(Br)ccc1C c1(C(=O)NC2CCC(NC(COCCCC)=O)CC2)cc(SCC)ccc1Cl c1(CNCC2N(C(CCCC#C)=O)CCOC2)cccc2c1CCC2 N1(Cc2c(C(F)(F)F)csc2)CCC(C2(O)CCOC2)CC1 C1(C(=O)NC2CCSC2C)(OC)CCN(CCn2nc(C)cc2C)CC1 C1(C(N(C)CCOCCC(=O)NCC=CC2CCOC2)=O)CCOC1(C)C C#CCCCCCCC(=O)N1CCCCC1CNC(c1cc(N)c(O)c(F)c1)=O C1(C(=O)NCC(CN(C(C(CC(=O)OC)C2CC2)=O)C)C)CC2(CCCCC2)C1 n1(CC(=O)NC(N(CCCCC)C(C2CCN(C(C)=O)C2)=O)=O)cc(Cl)c(C)n1 c1(CC)ccc(C)nc1NC(C1CCCN(C(=O)CCc2nc(O)n[nH]2)C1C)=O C1(CC(=O)NCC2C3CN(C(C(C=CC)O)=O)CC32)CCCS(=O)(=O)C1 CCC(CC)C(=O)NC1(CNC(C2CC3(CSC3)C2)=O)CC(OC2CC2)C1 N1(C(C2=CC(C)(CC)CC2)=O)CC2CCC(N=c3nn[nH]n3-c3cc(OC)ns3)C2C1 C1(NC(C2CCN(C(=O)CNc3ncccn3)C2)=O)C2CCC1CC2 C(C1(C)CCOCC1)=CC(=O)NC(C)C(=O)NO.C12CCCCN1C2 N1(C(CSCCCC)=O)CC(O)(C2CCCN2C(=O)CCOCC)C1 c1(OCC(=O)NCC2N(C(C(C(C)C)F)=O)CC(O)C2)ccc2c(c1)CCC2 C12(CNC(C#N)=O)CCCC1N(C(c1nnn3c1CCC3)=O)CCC2 N1(C(CC(C)NCc2ccccn2)=O)C2CCC1CC(NC(C1CC1(C)C)=O)C2 Cn1cnc2ccc(C(=O)OC(N3CC3)OCc3ccc4ncnn4n3)cc12.C1CN1 C1(C(=O)NC(C2(C(=O)NC(CCC)C(=O)NC)CC2)C)C2CC2CC(=O)C1C C1(NC(C2C3CN(C(CC(C)F)=O)C2C3)=O)CC2(CCOC2)C1 CC(C)CC(C(=O)NC1(CC(=O)NC2CCN(CCF)C2)CC1)N(C)C C1(NC(CC(CC)(F)F)=O)C(C)CCN(C(c2ccc(SC)cc2)=O)C1C Cc1cc(C)c(C(=O)N(CC(C)CNC(=O)Cn2nnnc2C(C)C)C)[nH]1 CC1(C)CC(C(=O)NC2CCN(C(=O)CN3CCOC3=O)CC2)C(C)(C)O1 N1(C(CCOCC#C)=O)C2COCC1CC(NC(=O)Cc1cn(CCC)nn1)C2 CC1OCC2(CCNCC2)C1N(CCC(C)O)C(c1ncccc1[N+](=O)[O-])=O C1(O)(CNC(C2CN(C)C(=O)C2)=O)CC(N=c2cc(Cl)nc(C(F)(F)F)[nH]2)C1 c1(C(C(=O)NCC(C)CN2CCC2)NC(=O)CCn2cccn2)cccnc1 c1(NC2C3CN(C(C(C=CCCC)O)=O)CC32)cc(=O)n2cc(Cl)ccc2n1 C1(C(N(CCCCCNC(CS(CC)=O)=O)C)=O)CC2CCC(C1)S2(=O)=O C(=O)(CCCCCN=[N+]=[N-])NC(c1cn(C)nc1)C(N1CC(CO)C2(CC2)C1)=O O=C1CC(CC(=O)N2CCC(CNC(c3c[nH]c(C(F)(F)F)c3)=O)CC2)=NN1 C(=O)(N=c1ccn(-c2ccc([N+](=O)[O-])cc2)[nH]1)N(C)CCc1ccccn1 c1(C(=O)NCC23CC2CN(C(c2ccsc2Cl)=O)C3)cnn2c1OCC(F)C2 c1(OCC)cc(N(C)CCCC(C)(C)C)ccc1-c1ccc(O)cc1 N1(C(CSCC=C)=O)CCC2CN(C(c3cccc(C4CC4)c3)=O)CCC2C1 C1(CNC)CCCCN1C(=O)NCc1conc1CCCCN C1(CNC(c2noc(C3CC3)c2C)=O)CN(C=O)CCC12CCC2.C(C(F)(F)F)=C C1(N)CCC(C)(C)CC1.C1C(C)(COC)NC(=O)C2CC(C2)CC(=O)N1.CC c1(COC)ncc(C#N)c(NC2CC(NC(=O)CC(=O)Nc3cccc(C)c3)C2)n1 c1(C(=O)NC(CC)CN(C(=O)CN2CCCC2CO)C)cnc(-c2ccco2)s1 CC1=C(C)CC(C)(C(N2C3CCC2C(CNC(c2ccc(=O)oc2)=O)C3)=O)CC1 C(=O)(CCCCSC1CCCCC1)NC(CN(C)Cc1onc(COC)n1)=O c1(C(=O)OCc2ccccc2)csc(=NCCc2ccsc2Br)[nH]1 C(=O)(C(=O)C(C)(C)C)NCC1CC(O)(CNC(C2C(c3ccc(C)s3)C2)=O)C1 c1(C(=O)NCC2CN(C(C(CC=CC)CC)=O)C2)cc(F)cc(F)c1N c1(CC(C)Nc2cc(NCC(C)CC(F)(F)F)ncn2)ccc2c(c1)OCCO2 CC(O)C(C(=O)N1CCC(OCCNC(c2ncn(C)n2)=O)CC1)N(C)C C1(c2n(CC)nnn2)(Nc2cnnn2C)CCCN(C2CCCC2)C1 c1(C(=O)NC2CC(C(=O)Nc3ccc(C(O)CF)cc3)C2)cc2ncccc2[nH]1 C1(NC(C=CCCC=C(C)C)=O)CCN(C(c2ccnnc2C)=O)CC1(C)C C1(CC(=O)N(CCNC(c2c[nH]c(=NC)s2)=O)CC2CC2)OCCOC1(C)C CCCCCC(F)C(=O)NC(CC(=O)N1CC(OC)CC(C)C1)C(F)F c1(C(=O)NCC2(C(=O)NCc3cc(=O)cc[nH]3)CC3(CC3)C2)cnc(O)c(F)c1 N1(C(C2=CC(C)(C)C2)=O)CC2(CCCN(C(C3Cc4ccncc4C3)=O)C2)C1 C1(NC(CC2CCCN(C(C)C)C2)=O)CCCCCN(C(C2(C)CCCC2)=O)C1 c1(CC)ccc(C=CC(=O)NCCC(C)N(C)C(C2CC2CC)=O)cc1 C1(C)(NC(C2C(C(=O)OCC)C2)=O)CCN(C(=O)Cn2cc(Br)c(C)n2)C1 C(C)(N=c1cc[nH]c(-c2nccs2)n1)C1CCN(C(C(C=C)O)=O)C1 C1(CC(N2CC(O)(CCNC(C=C(C)C(C)(C)C)=O)C2)=O)CCCCC12CC2 N1(C(c2c(CC)csc2)=O)CCOC(C(=O)N(C)CCc2cnc[nH]2)C1 Cc1cc(C)c(OCCCC(=O)NCC(=O)NC(C)CCCC(C)C)c(C)c1 CC(=O)CCC(=O)N(C1CCN(C(c2conc2C)=O)C1)CC1CCCO1 C1(C(=O)NCC(CC)NC(=O)C(CSC)OC)CCC(C(C)C)CC1 CCCC(C)(O)CC(=O)NC1CCN(C(c2ocnc2C)=O)CC1(C)C N1(C(CN(CCCO)C(c2c(C#N)ccs2)=O)=O)CC2COC(=O)C2C1 c1(C(N2CC3C(CNC(CC(C=C)CC)=O)(CC3)C2)=O)ccc(C)c(OC)c1F CC1CC(C2CN(c3nc(C(F)(F)F)ccc3C(F)(F)F)C2)=NO1 N12CC(O)CC1C2=O.c1(CC(=O)NCC(CCNC(COC)=O)O)cccc(C)c1 CCCCCCCC(=O)NCC1(OC)CN(C(c2c[nH]cc(Br)c2=N)=O)C1 C(=O)(C1CCCc2ccnn21)NC(=O)CN1CCCS1(=O)=O.C12CC1C(O)C2 c1(C(N(C(C)CCN)C(C2COC(=O)N2)=O)=O)ccccc1S(C)(=O)=O.N(C)C C1(NC(C2COC3COCC23)=O)COCCN(c2nc(CC3CC3)ns2)C1 C1(CNC(CC=CC=C)=O)CCCN1C(c1cnc(F)s1)=O c1(C(=O)NCCCCCNC(CCC(=C)Cl)=O)cccc(Cl)c1OC(F)(F)F C1(NC(COCc2cc(C)no2)=O)CN(C(=O)CC2CCCC(=O)N2)CC12CC2 c1(C(=O)NCC2N(C(C=CCOC)=O)CC(F)(F)C2)cncc2cnccc12 C(=O)(C(C)CNC(=O)CC1CCC(=O)N1)N(CC(C)OC)CC c1(OC)cc(C(=O)NCC(C)NC(c2cnn3c2OCCC3)=O)c(F)c(Cl)c1 C(=O)(CCCC(=O)c1ccccc1N)N1CC(CNC(Cn2ncc(C)c2)=O)C1 C1(N(C(c2ccc(C(C)C)o2)=O)C)CCCCN(C(=O)CCn2cnnn2)C1 c1(CC)ccc(C(=O)NCC2(NC(C3CC(F)(CO)C3)=O)CC2)[nH]1 C(C1=CCCC1)(c1nnnn1CCCF)NC(c1onc(COC)n1)C CCC(CO)C(=O)N(CCCCN(C)C(c1ccc(SC)o1)=O)C C1(CC=C)(NC(C2OCC2(C)C)=O)CCN(C(=O)COC2CCCOC2)CC1 C=CC(CCC)CC(=O)N(CCC(N1CCCC(CC)(CC)C1)=O)CCO N1(C(c2cccc(CC)n2)=O)CCCC(CO)(CNC(C2(C)C=CCC2)=O)C1 c1(CCC(N2CCC3C(NC(C(C)OCCC#C)=O)C32)=O)n[nH]c2c1CCCC2 C1(NC(C2CCS(=O)(=O)C2)=O)CN(S(=O)(=O)CCBr)CC1O c1(C(=O)NCC(CO)NC(COc2cccc(C)c2)=O)cnc2scnc2c1 c1(NC(C=CC(CC)C)=O)cccc(CO)c1.C1CC(=O)N1 C1(CN(C(C(CO)OC)=O)C)CCCN(C(c2ncccc2N)=O)C1 Cc1[nH]c(=N)nc(O)c1N(C1(CO)CCC1)Cc1ccc(OCc2cnn[nH]2)cc1 c1(CNC2CC(C(N3C(COC)CCCC3)=O)C2)c(F)cncc1F CCC(N)(C)C(=O)N(C)Cc1ccc(SC)o1 C1(CCNC(=O)Nc2cccnc2-c2ccco2)CCC2(CC1)COC2 C(=O)(C1OCCc2ccccc21)N1CC2(CCN(C(=O)CCSC(F)(F)F)C2)C1 C1(CCO)(NC(C(C)SC(C)C)=O)CN(C(C2(c3ccncc3)CC2)=O)C1 c1(NC(C2N(C(c3cc(C)[nH]c3)=O)CC2)=O)c(Br)cc(Cl)cc1C#N C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CCCC(NC(c2cc(CC)[nH]n2)=O)CC1 CC(C)(O)CC(=O)NCC1CC1CNC(c1cnoc1-c1ccccc1)=O C12(C(=O)NCCN(C)CCO)C3CC1C1C(C(=O)Nc4ccc(O)nc4)C3C21 C(=O)(C(O)(C(F)(F)F)c1cn[nH]c1)N1C(C(N2CCC(CO)C2)=O)C2CCC1C2 N#Cc1c[nH]c2c(F)ccc(Cl)c2c1=NCC1CCCN(C(=O)CCC2CC2)C1 CC(CCCC(=O)N1CCCC1CC1CC1)NC(=O)CCC1CC1(F)F N1(C(c2cc(CO)[nH]n2)=O)CCCC1C=CC(=O)NCC(O)C(F)F C(=O)(C(CO)C(C)(C)C)NCC(C(N1CCC2(CCOC2)C1)=O)N(C)C C1(C(c2nc(CCCCl)n[nH]2)C)NCCC1C(=O)O.NC N12CC(C(c3ccc(F)cc3)C1)NC2=O.C(C(C(=O)OC)c1ccccc1)CC c1(COC)cc(C(=O)NC(C(=O)N(CCN(C)C)CC)C2CCCO2)no1 Cc1ccc(NC(C2CCC2CNC(=O)Cc2cccc(CNC(N)=O)c2)=O)cc1 c1(C(N2C(CNC(C(CCC)OC)=O)CC(C)(C)C2)=O)snc2ccccc12 C1(NC(COCCC(C)C)=O)(CO)CCN(C(=O)C(O)Cc2cccc(Cl)c2)C1 CC1CN(C(=O)Cn2ccc([N+](=O)[O-])n2)CCCN1C(=O)CC1C=NN(C)C1=O CC1(C)CC1(c1ccccc1)CC(=O)NCCC(O)CNC(=O)Cn1cccn1 C1(C(=O)NC(CC#C)CC#C)CN(C(=O)CC2CCCCC2O)C(C)(C)C1 N1(C(c2scc(C(N3CC(OC)NC(=O)C3)=O)n2)=O)CCN2C(=O)OCC2C1 C(=O)(CCC(CF)CF)NC1CC=C(C(=O)N(C2CC(C)CC(C)C2)C)C1 C1(NC(c2cc(C)oc2)=O)CCC(C)(NC(=O)CN2CCCOC2=O)CC1 O=C1CCCC(C(=O)N2CC3(C2)CN(C(C2(O)CCSC2)=O)C3)c2ccccc21 Cc1cc(CNC2CC(C(=O)Nc3cnc(O)c(C)c3)C2)c(O)c(C)c1 c1(OCC)ccccc1C(=O)NC1C2CN(C(c3ccc(C(F)(F)F)o3)=O)CC12 c1(C2C(NC(=O)NCC(=O)NC3CC3)CCOC2)ccc(F)c(F)c1 c1(-n2c(Cn3ncc(C)c3)nc(-c3ccc(Cl)s3)n2)cc(Cl)cc(Cl)c1 C1(CC(=O)N(C2(CC(=O)NC3(C)CC(C(=O)OCC)C3)CC2)C)CCC(=O)CC1 n1(CC)cnc2c(NCCC3CCCO3)[nH]c(=NC(C)C3CCCC3)nc12 C(C(C)C(F)C(=O)NCc1cc(C)sc1C)NC(C1(CC)CCCCC1)=O C(=O)(C1=NOC2(CCC2)C1)NCCC1CC(NC(CC(CC)O)=O)C1 N1(C(CC2(OC)CCC2)=O)CCC(C)(NC(=O)C(OC)OC)C1 c1(OC)ccc(N(C(c2cnn(C)c2Br)C(=O)NCC(C)OC)C2CC2)cc1 N1(C(c2c(SC)snn2)=O)CCN(C(C2CC2COC)=O)C(C2CC2)C1 CC1CN(C(=O)C(O)CN2CCCC2)CC1(C)C(=O)NCc1ccno1 C1(CNC(c2ccc(O)cc2O)=O)CN(c2ccnc(CO)n2)CCC1(F)F C(CC(O)C(=O)N1CCC(F)(CNC(=O)CSC2CCCO2)C1)SC C1(C(=O)NCC2CCC(CNC(c3cnc(Cl)s3)=O)CC2)CCCCC(=O)N1 c1(C(=O)OCCC(N(CCC(=O)NC(C)C)CC=C)=O)ccn(COC)n1 N1(C(CC(C=C)c2ccccc2)=O)CCC(F)(CNC(c2cc(=O)cc[nH]2)=O)CC1 C(CCN=[N+]=[N-])N(C)C(C1OCCC1CNC(C1(CCCF)CC1)=O)=O N1(CC(=O)NCC(CC)NC(=O)C(C(C)C)c2cccnc2)CCC(=O)NC1=O c1(C(=O)NC2CN(C(c3cc(C(C)=O)sc3)=O)CC2C)ccn2nncc2c1 C1(C(=O)NCc2cn(C(C(=O)NC(C)C)C)nn2)CCCOC1C C1(NC(CCCCOC)=O)COC2(CCN(C(=O)Cc3cnn(C4CC4)c3)C2)C1 CN1CC(F)CC1C(=O)NCCC1COCCN1C(c1cnc(Cl)s1)=O n1(CC(=O)NC2CC(NC(C3CCC(C)S3)=O)C2)ncc2ncccc12 N1(C(C2(CC)CC2)=O)CCC(NC(=O)C(c2cnn(C)c2)C)C1 C(C(=O)N1CCC(C(=O)N(C)CCc2cnn(C)c2)O1)OC(CC)(C)C c1(CN(C)C)ccc(NC(c2nnnn2CCC2CC2)c2ccns2)cc1 c1(C(=O)OC(C(=O)OC)Cc2ccccc2)cc(C)nn1C(C)(C)C C1(CC(N2CCC3CCCC23)=O)CC2(C1)CN(C(=O)Cc1cnsc1)C2 C1(N(C(=O)NCc2ccccn2)CC2C3CNCC23)CCC2(CCNCC2)CC1 C=CCCC(C(=O)OC(C)(C)C)C(=O)OC(C1CCCCCC1)c1nnnn1C CC#CCCCC(=O)NCCOC1CCN(C(=O)CN2CC(C)(OC)C2)C1 CC(C(F)(F)F)NC(=O)C(c1ccco1)NC(=O)CCC1CCCC1 C(=O)(CCN=C(NCCSCc1ccccc1)N1CCC(F)(CF)CC1)N(C)C c1(C(N(CCN(C(CCCO)=O)C)C(C)C)=O)cc(Br)nn1C.C(C)(=O)OCC N1(C(C(C)(C)NC(=O)OC)=O)CCCC(C)(C(=O)NC2(C)CC(O)C2)C1 c1(C(N)=O)nc(Br)cnc1NC(=O)C=C1CCN(C(C2(CC#N)CCC2)=O)CC1 N1(C(c2sccc2-n2ccnn2)=O)CC(NC(C2CC(O)C2)=O)C2(CCOCC2)C1 Cn1ccc(C(=O)NC2(C)CCCN(C(C3CC4CC4C3)=O)C2)cc1=O c1(C(N2CC(C(C)NC(Cc3cc(OC)ncc3)=O)C2)=O)nc(O)[nH]c(=O)n1 CCCC(CCCNC(c1cnc(SC)[nH]1)=O)NC(=O)C(c1cccc(C)c1)O Cc1nn(CC(N2CC(NC(c3[nH]cnc3C#N)=O)CC2C)=O)c(C)c1C#N N1(C(C(C)(C)C2CC2)=O)C2CCCC1CC(N=c1cc(Cl)nc(C3CC3)[nH]1)C2 C#CC1CN(C(=O)C=CCN(C)C(C2(C)COC(=O)N2)=O)CC1O CCC(O)(CN(C)C(C12CC1CN(C(=O)CCSC(F)(F)F)C2)=O)CC c1(OC)ccc(Cl)c(CC(N2CC(O)(CCNC(=O)C(F)=CC3CC3)C2)=O)c1 NC(=O)CCCC(=O)NCCCCC1(NC(C23CCCN(CC2)C3)=O)CC1 CCCC(CNC(=O)CN1C(=O)CCCC1=O)C(=O)Nc1cnc(C(C)C)nc1 C1(C(N(CCCCNC(C23CC(CC)(C2)C3)=O)C)=O)CCCCN1S(C)(=O)=O c1(C(=O)NC2CCN(C(C(C)CCN(C)C)=O)CC2)cc(N)c(F)cn1 c1(C2C(CC(N3CC(NC(=O)C(F)(F)C4CCOC4)C3)=O)C2)ccccc1 c1(NC(=O)NC2CN(C(C(C)(C(C)C)NC(C)=O)=O)C2)cc(Cl)cc2c1OCC2 N1(C(c2c(C)cns2)=O)CC2CN(C(c3nccn3C)=O)CC2(C)C1 CC1(C)CCC(C)(NC(C2CN(C(C3CC4CCC4C3)=O)CCO2)=O)C1 c1(NC(C#C)=O)ccc(C(N2CC(COC)C2)=O)cc1C CC1C(NC(=O)C(=O)NCC2CC2(C)C(F)F)CCN1Cc1ccccc1 C1(NC(c2cn(CC3CC3)nn2)=O)(CO)CCCN(C(C23CCCC2C3)=O)C1 c1(CC(=O)NCC(CC)N(C)C(c2cnsn2)=O)cc(F)cc2c1OCOC2 N1(C)Cc2ccncc2C1.C1(C(=O)NC2(c3nc(C)cs3)CC2(F)F)CCC(C2CC2)C1 c1(C(=O)NCCC2CCC(NC(c3c(CC)cno3)=O)C2)cc(F)cc(F)c1O N1(C(C(C)OC)=O)CCC2(CC1)COCC(COC(c1ccccc1F)=O)O2 N1(C(C2CCC(CC)C2)=O)CCC(C(C)(C)NC(C23CC(C)C2C3)=O)CC1 N(C(=NCCn1ncnn1)N1CCCC(C(F)(F)F)C1)C(COC)C C1(NC(C)C(=O)N(CCCc2ccccc2)C)CCn2ccnc2C1 c1(C(=O)NC(C2(O)CCN(C(c3ncccc3Cl)=O)C2)C)cc(F)c(F)cc1N N1(C(C(=O)OC)C)CCC(N(CCCc2nnc(C3CCCC3)o2)C)C1=O C(c1cccc(Cl)c1)=CC(=O)NCC(C1CCCC1)NC(CSC)=O C1(SC)CN(C(=O)NCc2ccc(F)cc2)CC1n1cc(CC(O)C(C)(C)C)nn1 N1(C(CC(CC)NC(=O)CCc2nccn2C)=O)CCOCC(O)C1 c1(C(=O)NCCC2=CCN(C(c3cc(C)[nH]n3)=O)CC2)cnn2c1CC(C)CC2 C1(CC(=O)NCCCOCC)CCCN1Cc1cnc(C)o1 c1(SC)ccc(CNC(N2CCN(c3nc(C)c(Cl)s3)CC2)=O)nc1 CC1(C)CC(C(=O)NC23CC(C2)N(C(c2csc(Br)c2)=O)C3)CCO1 N1(c2nccc(C)n2)CC2CCN(C(c3cc4cccnc4s3)=O)C2C1 c1(-c2n(CC=C)ccn2)cccc(NC2(CC=C)CCC(C(F)(F)F)C2)c1C N1(S(C)(=O)=O)CCC(C(=O)NC2CC3(C2)CC3NC(c2cccnn2)=O)CC1 N1(C(C2C(C(C)O)C2)=O)CCCC(C)(C)C1CNC(c1ncnc2ccsc12)=O C=CC(C)(C)CC(=O)N1CCN(C(=O)CCS(C)=O)C(C2CCC2)C1 C1(n2cc(COC)nn2)CC(NC(C)=O)N(C(c2ccn(C)c2)=O)C1 CC1CCN(CC(=O)NCc2cc(C(=O)NCC3(O)CC=CC3)on2)C1 C1(C(=O)NCC2C3CN(C(CC4(C)CCC4)=O)CC32)Cc2nccn2C1 C1(C(N(CC(CC)NC(c2cc(C(C)C)on2)=O)CC)=O)CC(=O)N(C(C)C)C1 S(=O)(=O)(c1cccnc1)NCC(=O)N(C)CC1CN(C(C(CCC)O)=O)C1 N1(C(=O)C(O)CC(F)(F)F)CC2CCC(C1CO)N2C(c1ncc(F)cn1)=O Cc1cccc2nc(C(N3CC4CN(C(=O)C(=O)CCS(C)=O)CCC34)=O)cn12 CC1CCC(C(N2CCSCC2CCNC(=O)CCc2nccn2C)=O)CC1 c1(NC(c2c(OC)cccc2)CC(N)=O)nccc(=NC2CC(Cl)(Cl)C2)[nH]1 [N-]=[N+]=NCCCC(=O)N1CCCOC(CNC(=O)CCc2ccsc2)C1 C(=O)(C1=C(C)CCCC1(C)C)N1CC(C)CC(NC(C(COC)COC)=O)C1 c1(C(N(C(C)CNC(C2CCCC(N(C)C)C2)=O)C)=O)ccc(Cl)c(O)c1 N1(C(C(c2cncnc2)C)=O)CC(N(C(=O)C2=CC(C)C2)C)C2(CC2)C1 N1(C(CC2(OC)CCC2)=O)CCOC2(CCN(C(c3ccc(Cl)c(Cl)c3Cl)=O)C2)C1 c1(OC)ccc(Cl)c(CN2CCN(C(C3Cc4nccn4C3)=O)CC2)c1F N1(C(C(C)OC)=O)CCC2(CCCC2C(=O)Nc2ccc(F)c(Br)c2F)C1 c1(NC(C2CCC(NCc3ccc(C=O)s3)CO2)=O)cc(Br)c([N+](=O)[O-])cn1 N1(C(Cn2nnc(C)n2)=O)CCCC2(CCN(c3nnc(C(C)(C)C)o3)C2)C1 C1(CNC(C(CC=CCC)C)=O)(CO)CCN(C(=O)COCc2nc[nH]n2)CC1 c1(CC)cc(C(=O)NCC2CN(C)CCN2C(c2cocc2C)=O)c(C)nn1 C(CC(C)C(=O)N1CC(C(N)=O)(CNC(=O)CCN(C)CC)C1)=CC N1(C(c2c(OC)scc2)=O)CCCCCC1C(=O)NCc1cnc[nH]1 c1(CCC)ccc(N)c(C(N2CCN(C(C3C(C)CC3C)=O)CC2)=O)c1 c1(-n2cc(C(C3N(C(C(=O)N(C)C)=O)CCC3)C3CC3)nn2)c(F)cncc1F S(=O)(=O)(c1cc(Br)ccc1F)N1CC2(N(C(C3C(C(=O)OC)CC=CC3)=O)CC2)C1 N1(c2ncnc(C(C)(C)C)n2)CCC2(CC1)C(NC(=O)C1=CCCS1)CS2(=O)=O Cn1ncc(Cl)c1C(c1nnnn1-c1ccccc1Cl)NCC1COC1 c1(C(=O)OC)ccc(N=c2scc(-c3ccc(Br)o3)n2CC2CC2)cc1C C(CC)(CCCC(=O)NC(c1ccccc1)C)NC(c1c(CC)n(C)nc1)=O c1(NCCCOCC)[nH]c(=NCC2(CO)CC(C)(C)C2)nc2scnc12 CC1(C(=O)Nc2csc(Cl)c2)CC(O)CN1C(c1cccnc1S)=O Cc1nn(C)c(C)c1C(=O)NCC1CN(C(=O)CCc2cncnc2)CCN1C N1(C(CC2(COC)CC2)=O)CCN(C(=O)CC(C2CCC2)C2CCC2)C(C)C1 C(CS(=O)(=O)CC(=O)N1C(C(N2CCC(F)C2)=O)CCC12CC2)OC N1(C(c2c(C(C)C)ocn2)=O)CCCCCC(NC(c2ccc(Cl)c(Cl)c2)=O)C1 N1(C(c2cnc(C(c3ccncc3C)C)[nH]2)=O)CCC2(CCN(C3CC3)C2)C1 C(=O)(C(C(=O)NC(CNC(c1ccccc1C)=O)C1CCC1)OC)OC C1(NC(=O)Cc2cnns2)CC2(CCN(C(c3ccc(Cl)c(F)c3)=O)CC2)C1 C1(C(N(C2(C(N)=O)CC2)C)=O)CC(F)CN1C(C1CCC2(CC2)C1)=O C1(C)(C(=O)NC(CNC(C(C)(C)F)=O)CC(F)(F)F)CCCCC1(F)F c1(C(N2CCC3CC23C(=O)NCc2ccncn2)=O)ccc2cc[nH]c2n1 C1(NC(c2nc(COC)cs2)=O)CC2CCC1N2C(C1CCCCC(=O)N1)=O Nc1ccc(C(N2C3CCC2C(NC(=O)Cc2ccc(F)c(F)c2)C3)=O)nc1N N1(C(COC(CC)CC)=O)CC(NC(C2(C)CCN(C)CC2)=O)CC(C)(C)C1 N1(C(C2C(C)C2)=O)CCN(C2CCCN(C(c3ccccc3)=O)C2)C(=O)C1 C1(C(=O)NC(CC)CC(=O)NC2CC(C)(CC)C2)CCC2(CC1)CC2 C(=O)(C(C)(C)C(F)(F)F)N(C(C)C)CCN(C)C(c1c[nH]nc1[N+](=O)[O-])=O N1(C(C(CC)C)=O)CC(NC(c2cc(F)c[nH]2)=O)C(O)C1 c1(OC)ccncc1C(=O)NCC(CNC(=O)C(C)=CC1CC1)OC c1(C(=O)NCC2C(C)CN(C(c3cscn3)=O)C2)cc(O)nc2[nH]c(=N)ccc12 n1(CC#C)cccc1C(=O)N(CCCNC(=O)C(F)(F)C1CC1)C(C)C C1(CNC(C(CN(C)C)(F)F)=O)CC2(CO1)CN(C(C1CC3(CC3)C1)=O)C2 C(=O)(C(C(=O)N1CC(CNC(=O)CCCn2ccnc2)C(O)C1)C(C)C)OCC C(C(C(=O)N1CCC(CNC(=O)C(C)(C)c2ccnn2C)C1)C(C)(C)C)OCC S(=O)(=O)(c1c[nH]c(=N)c(C)c1)N1CC(c2c(C)[nH]nc2O)C(C(=O)O)C1 C(=O)(C#CC1CCCO1)NCC1CCN(C(Cc2cccc(OC)c2)=O)C12CC2 C(N=c1nc2c(ncn2C)c(NC2CCC2C(N)=O)[nH]1)C1(C)N(C)S(=O)(=O)CC1 c1(-n2c(N3CCC(C(=O)OCC)C3C)nnn2)ccc(C)c(C)c1 c1(CNc2cc(C(=O)Nc3cc(OC)cc(O)c3)n(C)c2)cc(F)cc(C)c1O Nc1cc(C(=O)NCC2CCCN(C(c3cc4sccc4[nH]3)=O)C2)nc(O)c1 C1(CCC)(CO)CCCN(C2=NCc3ccccc3CN2)C1.C1(SC)CCCO1 c1(C(N(CCN(C(=O)CC2CCC(F)(F)CC2)C)C)=O)ccc2c(n1)CCC2 c1(C(C(=O)NC(C)CC)N(CCC#N)CC=C)cc(OC)ns1 c1(CNC(c2cn(C3CCC3)nn2)=O)ccc2c(c1)CN(C(C1CC1F)=O)C2 c1(OC)cccc(C(N2CCC(N(C(=O)CCN3CCCC3)C)CC2)=O)c1 N1(CC)CCCC2(CCCN2C(=O)CC(C)C)C1.c12cc(Cl)ccc1C(=O)S2 c1(CNC(CC(C)n2cccc2)=O)cccc(CN(C)C(C23CSCC2C3)=O)c1 N1(C(c2ocnc2C(F)F)=O)CCC2CN(C(=O)CN3CC4CC4C3)CCC2C1 c1(C(N(C)CC2(n3cc(Br)cn3)CC2)=O)cc(F)c2cc[nH]c2c1 c1(OC)ccc(C(N2CC(NC(c3scnc3C)=O)CC2C)=O)c(Cl)c1 CCCCC(O)CC(=O)NC(CO)C(C)NC(=O)C(c1ccccc1)=CC(C)(C)C CC1CCCC(C(=O)N(C2CCCCC2)CCN(C(C2CC(F)C2)=O)C2CC2)C1 N1(C(C)=O)CCC(NC(C2C(NC(=O)C(O)CN(C)C)C2(C)C)=O)C1 C(=O)(C(F)C(C)C(F)(F)F)NCCN(CCC)C(c1c(O)cccc1O)=O CC1(C)CN(C(c2ccc(Cl)cc2)=O)CCN1C(c1cnc(O)c(Br)c1)=O c1(CNC(c2cnc(CCC)s2)=O)ncccc1CNC(C1CC(OC)C1)=O N1(C(C=C(C)C(C)(C)C)=O)CC2CCCC(Nc3ncccc3[N+](=O)[O-])C2C1 CC1(C)CCC(O)C(NC(=O)NCCOc2ccc(C(F)(F)F)cc2)C1 c1(C(N2CC(O)CC2c2cccc(F)c2)C(=O)NCC)cc(C(F)(F)F)ccc1Br c1(C(=O)NC(C2CCCN2C(c2ccc(C(N)=O)o2)=O)C)ccc([N+](=O)[O-])nc1 CC1(C#CC(=O)NCC2CCCCN2C(=O)C(c2cccc(Cl)c2)O)CCCO1 C1(C(N2C(C)CC(CNC(=O)C(F)(F)C(C)(C)O)C2)=O)CCCC2CCCCC12 Cc1cc(C(=O)N(C2(CC(N3CC(C)CC3C)=O)CC2)C)cc(F)c1 c1(N(C(C2(C)CCN(C(C(C)Sc3cccc(Cl)c3)=O)C2)=O)CCO)ccc(Cl)nc1 c1(C(C)C)ccc(N)c(C(=O)NCCC(C)(C)NC(=O)Cc2cnccn2)c1 c1(C(=O)NC2CN(C(C3CC(OC)C3)=O)CC2(C)C)ccc2occc2n1 c1(C(C(=O)N(CCOC)CCNC(=O)C=CCN(C)C)C)c(C)n[nH]c1C C1(CC(=O)OC)C2CCC(C2)N1C(C1CCCCC1)C(=O)NCCC(=O)N(C)C N1(CCNC(C(C)C)=O)CCCC1C(c1ncnn1C)=O N1(C(C(C)Sc2ccccc2)=O)CCC(F)(C(=O)NCC2CC23CC3(F)F)CC1 C(=O)(C1=CC2CCCCC12)NCC1(NC(Cc2nc(COC)sc2)=O)CCCC1 C1(C(N2CC(O)(CN(C(C(CCC)OC)=O)C)C2)=O)CCOCC1(C)C C1(C(=O)NCC2N(C(C(C)OC(C)(C)C)=O)CC2)(CC)CCOCC1.C#CCC(=O)O S(=O)(=O)(c1cnc(NC2CCC3(CCC3)CC2)cc1C)NCC(CC)(C)OC C(C(CO)(CO)NC(=O)CC1CCCCN1C)N(C)C(c1cccc(CO)c1)=O C1(NC(c2ccc(C)cc2Cl)=O)COC2CN(C(=O)CN(C)C3CC3)CC12 c1(NC(C2(C)CCCN(C(=O)Cc3ccc(F)cc3)C2)=O)cc(Cl)c(Cl)cc1Br C(=O)(C(CCF)NC(c1c[nH]c(C#N)c1)=O)N(C(C)C)C CCCCCCC(C)C(=O)NCC(C)(O)CNC(c1coc(CCC)n1)=O C(CCC(C)C)(C(=O)NCc1cncn1C(=O)OCC)N1CCC(CC=C)C1 C1(C(=O)NCCO)COCCN(C(=O)C2CC2)C1.C(=O)(CCOC)SCCC=C CN1CCCN(C(C2CN(C(c3cc(Cl)cnc3Cl)=O)CCS2)=O)CC1 Cc1ccc(COCC(N2CC(NC(=O)CC3CC3)C(C)C2)=O)cc1 C1(C(=O)OC)CCC2CN(C(=O)C(C3CC(F)(F)C(=O)N3)N)CC12 C#CCC(O)C(=O)NCC1(C)CCCN1C(c1nn(CC(F)(F)F)cc1Br)=O CCC(CC)CCCC(=O)N1CCC(C(C)(C)NC(c2nn(C)c(Cl)c2Cl)=O)C1 N=C1NC(=O)C(NCC(=O)NCC2CCCCN2C(=O)CC2(F)CCCCC2)S1 c1(OC)cc(F)ccc1C(N1CCCC(N(C(=O)CCCCF)C)C1)=O N1(C(c2nnn(CC)c2C(F)(F)F)=O)CC(C)C(C2CCCCC2)C1 Cc1ccnc(-n2cc(C(N3CCCC3CNC(=O)CC3CC=CC3)=O)cn2)c1 c1(C(=O)OCC)cc(N(CC(=O)OC(C)(C)C)CC)ccc1[N+](=O)[O-] C1(NC(C(C2CCCC2)OC)=O)CC2CC(NC(C3(CF)CCC3)=O)C2C1 c1(CC(C)C(=O)NCC2CCN2C(=O)CCc2ccoc2)ccc(Cl)c(Cl)c1 c1(C(=O)NC2CC(F)(CNC(c3cncc(CO)c3)=O)C2)ccc2occc2n1 c1(C(N(C)CCNC(c2ccc(F)c(O)c2F)=O)=O)c2c(nn1C)CCSC2 Cc1ccc(N)c(C(=O)N(CC(C)NC(C2(C3CCOCC3)CC2)=O)C)c1F C(=O)(C1=CC2CCC(C1)C2)N(CC)CC1CCCN1C(=O)Cn1cc(CO)nn1 C(=O)(C(CCCC=C)NC(C1CCCCCN1C)=O)NCCCCC#C C1(CNC(C2CCC(C)C2)=O)CCN(C(=O)C(c2ccc(O)cc2)=O)C12CC2 CCCC(CC)C(=O)N1CCN(C(c2ccc(Br)cn2)=O)C2CC12 C1(CC)C(=O)N1.C(C)(C=CC(=O)NCCF)NC(COCCC)=O N1(C(C(C)(C)OCC)=O)CCC(C2CCN(C(=O)COCc3ccccc3)C2)C1 Cc1nc(C(=O)NCCC2(CNC(c3cc(F)c[nH]3)=O)CC2)ccc1[N+](=O)[O-] Cc1c(C(=O)NCCc2ccc(CNC(C3C(C)C3C)=O)cc2)cccc1F C(=O)(C1=C(C)CCC1)N(C1CCN(C(c2cc(C)nn2C(C)(C)C)=O)CC1)CC c1(CC(N2CCN(CCN(C)C(C3(O)CCOC3)=O)CC2)=O)cccc(Cl)c1Cl CCCCS(=O)(=O)CC(=O)NC1CCCC1NC(C1CCc2nn[nH]c2C1)=O c1(CNCC2CC(CC(=O)O)C2)ccc2c(c1)OC(F)(F)C(F)(F)O2 C1(CNC(c2cn[nH]c2)=O)CN(C(c2ncncc2Cl)=O)C2(CCC2)C1 N1(C(c2ccc(OC)s2)=O)CCC2(CC(C(=O)Nc3cnn4c3CCC4)=NO2)C1 c1(C(=O)NC(C2CC3(CCC3)C2)C)ccn2nnnc2c1 N(C1CCc2c(Cl)cccc21)C(=O)Nc1cccc(C)c1[N+](=O)[O-] S(=O)(=O)(c1cccc(N(C)Cc2cn3cc(C)sc3n2)n1)NC1CC(CC)C1 c1(C(N2CC(CNC(c3ccc(C#C)o3)=O)OCC2)=O)ccc(Cl)cc1C(C)=O N1(C(c2c(C)cc(N)cn2)=O)CCCN(C(=O)C(C)Sc2ccccc2)CC1C c1(C(N2CC(CCNC(C34CC3CNC4=O)=O)OC(C)C2)=O)cc2sccc2[nH]1 c1(CC)ncc(C(N2CC(O)(C(F)C(=O)N(CC)CC3CCC3)C2)=O)cn1 n1(CC(=O)NC2CCN(C(COCCC)=O)C2)c(C)cc(O)cc1=O N1(C(c2n(C)c(Cl)nc2)=O)CC(NC(=O)CCN2CCOCC2)C(C2CC2)C1 CC1(C)CC(C(=O)OC)C1C(F)(F)F.n1(CC)cc(C2(O)CCCC2)nn1.C1CO1 c1(C(=O)NCC(C)N(C)C(C2C(C)C2(F)F)=O)ccc2nnn(C)c2c1 C=CC1(C2(C(=O)NC(CNC(=O)CCCCC(C)C)C3CC3)CCC2)CCC1 c1(CC(=O)OC)cnc(N2CCOC(CNC(c3cccc(F)n3)=O)C2)nc1 Cc1nnc(C(CC(C)C)NC(=O)NC(C)C(C)C2CC2)o1 c1(C(N2C(CNC(CSC)=O)C(C)CC2)=O)ccc(-c2ccccn2)nc1O C(=O)(CC1=CCN(C)CC1)NC(C(N1C(C(C)O)COCC1)=O)(C)C1CCC1 c1(NC(C)=O)cc(S(=O)(=O)C(F)(F)F)ccc1F.c12ccc(cc1O)oc2=O C=CCCCC(=O)NCCc1cc(C(=O)NC(CCC=C)C2CC2)no1 Cc1cnc(C(N2CCOCC2CNC(=O)CCc2ccc(F)cc2F)=O)cc1Cl c1(N2C3CC(=C)CC2CCC3)nc2c(c(=NCC3CCc4ccccc43)[nH]1)CSC2 c1(NC(C)=O)cccc(NC(N2CC(NC(c3ccnc(C)c3)=O)C2)=O)c1C C1(CC(=O)N(CCNC(C(C)NC(C)=O)=O)CC2CC2)CCCOC1 c1(C(C(=O)N(CCC(C)NC(=O)CC2CC(=O)C2)C)OC)cc(F)cc(F)c1 Cc1cc(N2CC(NC(c3cc(C)c(Br)s3)=O)C(F)C2)ncn1 C(=O)(C#CC1CCOCC1)N1CC(CNC(C2(C)CCC2)=O)C1.c1(OC)ccccc1 N1(C(C=C(COC)C)=O)CC2CC(NC(c3c(C)cc(C)nc3C)=O)CC1C2 Cc1cc(C(=O)NC2C3CN(C(=O)Cc4cccs4)CC23)cc(C)n1 S(=O)(=O)(CC(=O)N1CCC(O)(CNC(=O)C=CS(C)=O)C1)NC(C)(C)C CC1(C)CN(C(c2cccc(Cl)n2)=O)CC(CNC(=O)CNC(=O)C(F)(F)F)O1 c1(C(=O)NC(CN2CCCCC(N(C)C)C2)=O)ccc(C(=O)O)n2nc(C)c(I)c12 c1(C(=O)NCCC(CCNC(C(C)SC)=O)C)ccn2ncccc12 C1(C(=O)NC2CC(C)(C)N(c3cc(C4CC4)ncn3)C2)CCCC2CCCCC12 CCC(C)(C)C(O)C(=O)NC1CC2CC(NC(=O)COC(C)(C)CC)CC12 C1(NC(c2c(C(C)C)nns2)=O)CN(C(C2(O)CCC2)=O)CCC1CO C1(CNC(CCOCC(C)C)=O)CN(CC2CCCO2)CCCO1 N1(C(COC)=O)CCCC(O)(CNC(c2cccc(CSC)n2)=O)C1.C1(C)C(=O)N1 c1(C(=O)NCC2CC(C)(C)N(C(c3cccnc3)=O)C2)cccc2cnccc12 c1(C(=O)NC(C)C(C)NC(c2ccc(-c3ccco3)o2)=O)noc2c1CCCC2 N1(C(c2n(C)[nH]c(=N)c2)=O)CCCCC(C2CN(C(=O)CSc3nncs3)C2)C1 N1(C(CC(=C)Br)=O)CCC(CNC(c2csc(C)n2)=O)(OC)CC1 C1(C)(CNC(C)=O)CCN(C(=O)COCC2CCCCO2)CC1.c1(N)ccc(F)nc1 N#Cc1cnc(N2C3CCC2CN(C(=O)CC2CCOCC2)CC3)c2sccc12 C1(CNC(C2CC(C(C)=O)C2(C)C)=O)CN(C(C2C3CCN2CC3)=O)CCCO1 N1(C(C2CN(C)C2)=O)CCC12CCN(Cc1cc(S(C)(=O)=O)cs1)CC2 C1(NC(C(=O)NCCCCCC)=O)CCN(C(=O)COC2CC2)CC1O CC1CCC(NC(=O)Cn2cc(Cl)cn2)CN1C(c1ccn(C(F)F)n1)=O c1(OC)c(C(=O)NC2CC(n3cc(C4CCCC4)nn3)C2)cccc1Cl C1(CC(C)C)CCCCN1C(=O)C(CN(C)C)NC(C1CCCN1C)=O c1(CNC(C)Cc2nccs2)noc(C(C)(F)F)n1 C1(NC(C2C(C=C)CC2)=O)CCCCN(C(=O)COc2ccc(C(N)=O)cc2)C1 CC(C)C(C#N)C(=O)N1CCC(NC(c2ccc(C3CC3)c(F)c2)=O)C1C Cc1c(C(=O)NC(CNC(=O)C2=CCCS2)C(C)(C)C)ccn1C(C)C c1(C(=O)NC(CC)(C)CNC(=O)C=CC(F)(F)F)ccc(Cl)cc1O C1(C2CCN(C(c3ccn(C(C)(C)C)n3)=O)C2)(NC(CCC(C)(F)F)=O)CC1 C12(SC(C)C(=O)NC3(C(=O)O)CC3C)CC3CC(CC(C3)C1)C2 C(=O)(CCCCCCS(N)(=O)=O)NC(CC)CNC(c1ccc2ocnc2n1)=O Cc1cc(NC(C2CCCC(NC(=O)C(=O)N(C)C)C2)=O)c(C)cn1 Cc1cc(C(=O)N(C2CCN(C(C3CC(Cl)(Cl)C3)=O)C2)CCO)c2c(c1)CCO2 C1(NC(C(CC(=O)OC)C)=O)CC(O)(C2CCN(C(=O)CC3CC(C)C3)CC2)C1 CC(CCNC1CC(C(F)(F)F)C1)N=c1ccnc(NC(=O)OC(C)(C)C)[nH]1 Cn1cc2cc(C(N3CC4CCC3C(NC(C3CCCSS3)=O)C4)=O)ccc2n1 N1(C(=O)C(C2CCN(C(c3csc(O)n3)=O)C2)F)CC2CC(O)CC1C2 c1(C(N(C)CC2N(C(Cc3ccc(C)s3)=O)CC(F)C2)=O)cnn2c1NCCC2 c1(-c2nc(C(CC)C)nn2-c2nccn2C)ccnc2[nH]cnc12 Cc1cc(Cl)ccc1C(=O)OCC(C1CC2CCC1C2)=O N1(C(C(CC)=CC)=O)CCC2(CCCN(C(c3cnn(C4CC4)c3)=O)C2)C1 c1(C(N(C2CCCCC2NC(c2cnc(C(F)F)cn2)=O)C)=O)ccnnc1O C1(NC(C=CC(C)NC(C2CC3(C2)CC(C)C3)=O)=O)CCc2nn[nH]c2C1 c1(NC(=O)NC(CC)COC(F)(F)F)scc(-c2ccccc2)c1CC CCCCC(=O)NCCCC(=O)NC(c1cscn1)CO N1(C(N(c2ccn(C)c2)C)=O)CCC2(CC1)C(O)CC2O C1(C(N(C)CC2N(C(C(c3scc(C)n3)C)=O)CCCC2)=O)COCCN1C=O C1(NC(C2C(Br)(C(=O)OC)C2)=O)CC(F)(CNC(C2CC(OC)C2)=O)C1 C1(O)(C(C)NC(c2nc(CCCC)sc2)=O)CCN(C(=O)CCC(F)F)C1 N1(C(Cn2ncc(C#N)c2)=O)CC2CCCC1CN(C(c1cc(CO)[nH]n1)=O)C2 Cc1cccc2cc(C(=O)NC(C3CCN(C(=O)C#CC(C)C)CC3)(C)C)nn12 c1(C(=O)NCC2CC(NC(C3(COC)CCOC3)=O)C2)cc(C2CC2)cnc1F C(=O)(C(CCC(N)=O)n1cc(C2CC3(C2)CC(O)C3)nn1)OC N1(C(C2CCCC(C)C2)=O)CC2(CCCN(C(C3(C)CS(=O)(=O)C3)=O)C2)C1 CC1CCCCC1(CNC(C1CCC2(CCC2)O1)=O)NC(=O)CSCC#N C1(C(N(CCCCN(C(=O)CCNC(C2CCCO2)=O)C)C)=O)CCC(=O)NC1 Cn1cnc(Cl)c1C(N1CCCC(C(N)=O)C1)C(=O)NC1CCOC1 C#CCCCCCC(=O)NC(C(=O)NC1(CN(C)C)CCCC1)C1CCOC1 N1(CC(=O)NC(C)CC(=O)NCCC2CC(C)(C)C2)C(=O)CNC1=O Cc1cc(C(N2CCC(C)(CC(=O)N(C)CC3CCCS3)C2)=O)c(C)cn1 c1(COC)cc([N+](=O)[O-])c(O)cc1NCC1=CCN(C(=O)OC(C)(C)C)CC1 CC1(C)CCCC1(N)C(=O)Nc1ccc(Cc2cccc(F)c2)cc1 N1(C(C2=C(C)OCC2)=O)CCC2CC2(C(=O)NCCCCCC(C)C)CC1 N1(C(C(C)SC(c2ccccc2)CO)=O)CCC2CN(C(=O)CC3(C#N)CC3)C2C1 c1(CC(=O)NCC(CNC(c2cnc(COC)s2)=O)C)ccc(C(F)(F)F)nc1 N1(C(CCC)=O)CCN(C(c2cnc(OC)nc2)=O)CC1c1cn[nH]c1 C12(C(=O)NC3CCCCC3)CCC(N(CCO)CC3(C)COC3)(CC1)CC2 CC1(C2CC2)CCN(C(C2(C)CCN(C(c3cccc(O)c3)=O)C2)=O)C1 C1(C(=O)Nc2cc(CC(N3CCC(OCCOC)C3)=O)on2)CC2(C1)CC2(F)F C=CCC(C(=O)NC(CC=CC)C(=O)NCCCCC#CC)C(C)C N1(c2cc(C(C)(C)C)ncn2)CCN(C(=O)C(CO)c2ccccc2)CC(O)C1 N1(C(C(CC)(F)F)=O)CCC2(CCC2)C(CNC(C2(OC(C)=O)CCCOC2)=O)C1 O=C1Cc2cc(C(N3CCC4CCC34CNC(c3ccoc3)=O)=O)c(Cl)cc2N1 C12(C(N(CCNC(C(C)OC)=O)CCOC)=O)CCC1CC2 N1(C(C(C)NC(C)=O)=O)CCC(C)C(NC(c2cccn2C)=O)C1C C(C(=O)N1CC(n2ccnn2)C1)(C1CC1)SC.C1(c2cccs2)C(=O)N1 C(=O)(C(C)(C)CC(C)(C)C)N1CCC(CNC(C(C(CC)CC)F)=O)C(C)(C)C1 CCCCCCCC(=O)N1CCCC(NC(=O)COC2CC=CC2)C1C N1(C(C(C)=CC)=O)CCCC(N(c2cc(C)ncn2)C)C1 C1(C(=O)NC(CCOC)C(N2CCNC(=O)C2C)=O)CCCCC(=O)C1 c1(-c2cn(C(CNC(CCSC)=O)C)nn2)ccc(OCCN(C)C)cn1 c1(CC)nc(C)ncc1C(=O)NC(C1CCN(C(=O)C(C2CCOCC2)=O)C1)C C1(CN(C)C(C2CCC(F)(F)C2)=O)CCN(C(=O)CCC2CC2(Cl)Cl)CC1 C1(NC(C(COC)C)=O)CCC(C)(CNC(=O)CSCC#N)CC1 C(c1cncc2ccccc12)=CC(=O)NC(CNC(c1ccc(C)nc1)=O)CO CC1=C(C(=O)NCC2(CNC(C3(C)CC4CC4C3)=O)CCCC2)CCO1 N1(CCCC=C)CCC(C)C(NC(c2coc(C(F)F)c2)=O)C1 N1(C(CCCC=C)=O)CC(NC(c2cc(CCCC)oc2C)=O)CC1(C)COC C1(OC)(CNC(c2ncccn2)=O)CCN(C(=O)CCSC2CCCC2)C1 c1(C(N(CCN(C(c2cnc(SC)s2)=O)C)C)=O)cnc2onc(C)c2c1 c1(C(N2CCCC2N2CCCC2=O)=O)cccc(-c2cnc[nH]2)c1 C1(CNC(CC)=O)CC2(CCN(C(C3CCCC3c3ccc(F)cc3)=O)C2)CO1 c1(C(N(CC(CC)NC(c2[nH]c(O)nc2C)=O)C)=O)sc(F)cc1Cl n1(CC(=O)NCC(C)N(C(=O)CCN2CCCCC2)C)cc(C2CC2)cn1 N1(C(CCC2CCC(C)O2)=O)CC2CCC1CN2C(=O)Cc1cccc(F)c1 C1(NC(CC)=O)CN(C(=O)CCC2CC(F)(F)C2)C2(CCCOC2)C1 c1(C=O)cc2ccccc2n1C.C=C=C(C)CC(=O)N1CCC1CC1CC1 CC1C(=O)NC(=O)CN1C(=O)C(C(C)(C)C)NC(c1cc(=N)[nH][nH]1)=O N1(C(c2cnn(CC)c2Cl)=O)CCCC2C(CCCN2C(c2nocc2C)=O)C1 c1(C(N2CCC(F)(CNC(C(C)SCC)=O)C2)=O)nc(Cl)ccc1OC(C)C C(=O)(C(O)CC(C)(C)C)N(C1CCCN(C(C=C(C)c2cccs2)=O)CC1)C c1(OCC)ccc(Cl)c(C(=O)NCC#CCNC(c2ccc(OC)c(N)c2)=O)n1 CCCCC(O)C(=O)NC1CC=CCC1C(=O)N(C)CCN1CCCC1=O Cc1oc(Cl)nc1C(=O)NCC1CCCC(CNC(=O)CCCn2cccn2)C1 C1(C#N)(CNC(C(CC=C)NC(=O)CN2CCCC2)=O)CCCCC1 C(=O)(C(CC1CC1)NC(c1ccsc1)=O)N(CC(C)OC)C C(=O)(C1CCCn2nccc21)NC(C1N(C(CCC(C)(F)F)=O)CCC1)(C)C C(=O)(C1=CCCN(C(c2ccc([N+](=O)[O-])o2)=O)C1)NC(C1CCCCC1)C#C C1(NC(COc2cn(C)nc2)=O)CCCN(C(=O)CN2CCOCC2=O)CC1 N1(C(C(C2CCOC2)NC(c2ncoc2C(F)(F)F)=O)=O)CCN(CCSC)CC1 CCC(CC(=O)N(CC(C1CCC1)OC)C)NC(=O)C1CC1 C(=O)(C(C)(C)CF)NCc1ccc(C(C)NC(=O)CSC2CCOC2=O)cc1 C(N=c1[nH]c(=NCC(C)C(C)(F)F)[nH]c2c1CCCC2)c1cccc(OCC)n1 N1(C(C(CC2CN(C(C3C(C)(C)C3(C)C)=O)C2)F)=O)CCC12CCCSC2 C1(NC(C2(CCOC)CC2)=O)C2CC3C1C3C2C(N1CCS(=O)CC1C)=O C(c1nnn(C)n1)=CC(N1CC(CNC(c2c(CC)nn[nH]2)=O)C1)=O C1(O)(Cn2cc(C(C)O)nn2)CCCN(C(c2csc(C3CCCO3)n2)=O)CC1 N1(C(c2n[nH]cc2Br)=O)CCCC(C2CCCN(Cc3cncs3)C2)C1 C1(C(C)CNC(C2CCCS2)=O)CCN(C(=O)C(C)CC2CCC2)CC1 C1(CNC(CC(=O)OC)=O)CC(C)N(C(C2CC(=O)N(C)C2)=O)C1 c1(C(N2C(CNC(C(CC)NC(N)=O)=O)C=CC2)=O)sc(COC)nc1C C1(NC(C2C(CNC(c3c(C)n[nH]c3C)=O)OCC2)=O)CCCN(C)C1C C1(CC=C)(NC(=O)C=Cc2ncc[nH]2)CCN(C(C2COC(=O)N2C)=O)C1 Cc1ccc(OCC(O)CNCC(=O)Nc2cnn(-c3ccncc3)c2)cc1 N(C(=NCCc1ccc(OCC)nc1)NCc1nc(C(F)(F)F)cs1)C(CC)C C(CCCCN(C)C(C1CCCN1c1ncccn1)=O)NC(C(F)=CCC)=O C(=O)(C(C)(O)C(C)(C)C)NC1C(NC(CS(CC)(=O)=O)=O)CCCC1 c1(C(N2CC(COC)(CNC(=O)C(F)(F)C3CCCC3)C2)=O)ccnc(O)c1 C1(CNC(C2N(CC#C)CCC2)=O)CCC(C)(C)CN1C(=O)CNC(C)=O C1(NC(Cn2c(C)csc2=O)=O)CC(C)CN(C(=O)CSc2nncn2C)C1 N1(C(C(C)Sc2ccccc2)=O)CC2(NC(=O)CSc3ccccn3)CC1C2 Cc1ccc(C(N2CCOC(C(=O)NC3CNCC(OC(F)F)C3)C2)=O)c(O)c1 c1(C(N(C2CCN(C(C3(C)CC3F)=O)CC2)CC)=O)cc(OC)cc(Cl)c1O c1(OC(C)C(=O)NCC2CCCN(CCC(F)(F)F)C2)ccc(O)cc1 c1(C(=O)NCCC2OCCN(C(CC3CCCN(C)C3)=O)C2)csc([N+](=O)[O-])c1 N1(C(C)=O)CCN(C(C2CSCCN2C(=O)CC=C(Cl)Cl)=O)C(C)C1 C(=O)(C(C)C1=CCCC1)N1CC(CNC(c2c(OC)cccn2)=O)OCC1 C1(C(=O)NCC(C(=O)NC(C(=O)OC)Cc2ccoc2)N(C)C)CCCC(=O)N1C C12(NC(C(CCC)OCC)=O)CCCC1N(c1ncc3ncnc-3[nH]1)CCC2 C1(CNC(CNC(CNC(C)=O)=O)=O)CCC(NC(=O)CS(N)(=O)=O)CC1 C1(NC(C2(C=C)CC2)=O)CCCC(NC(c2ccnc(OC(F)F)c2)=O)CC1 N1(C(=O)NCCC(=O)NC2(C)CCCS2)CCc2nc[nH]c2C1c1ccc(Br)cn1 C12(NC(C3(C=C)CCOCC3)=O)CC3CCC(C1C2)N3C(c1cccc(Cl)c1)=O C1(CC)(NC(C2COCC2(C)C)=O)CCN(C(C2CCCC3(CC3)C2)=O)CC1 C1(C(=O)NCCC(C)(C)N(C)C)CCCCC1NC(=O)Cn1ncn(C)c1=O CCCCCCCC(=O)NCC1(F)CC(NC(=O)C=Cc2ccc(OC)cc2)C1 c1(C(=O)NCC2C(OCC)CN(C(CC=C=C)=O)C2)cnn2c1OCC(C)C2 N1(C(c2c(C)cc(CNC(c3c(COC)c[nH]c3)=O)o2)=O)CCC(F)(F)CC1C c1(C(=O)NCCCCNC(C(C=CCCC)O)=O)cc(C)ncc1Cl Cc1cc(NC(c2nnnn2C2CCOCC2)C2CC2(C)C)cc(C)c1Br c1(CC#N)ccccc1NC(=O)C(=O)Nc1ccc(C(F)(F)F)cc1 C1(c2nnnn2CCC2(C)CC2)(NCc2c(C)ocn2)CC(C)N(C)C(C)C1 CC1(CNC(c2cc[nH]n2)=O)CCC(NC(=O)CCc2ccon2)C1 N1(CC2CCC(C)(C)CO2)CC2(CC(=O)O)CCC1CC2 c1(CC(N2CCC(N(C(C=NOC)=O)CCO)CC2)=O)c(C)nn(CC(C)C)c1C C1(CNC(CCCCCOC)=O)CN(C(C2CC2C(=O)OC)=O)CC(C)(C)C1 O(NC(=O)C(F)C1CCC1)CC(=O)N(CCCC)CC(C)C c1(C(N(CC(CC)NC(=O)COc2cccc(C)c2C)C)=O)cc(N)c(F)cn1 N1(CC(N2CCC(N(C(=O)CSC(F)F)CCC)CC2)=O)CCCCS1(=O)=O c1(C(N2CC3C(CNC(c4cc(C)sc4C)=O)(C3)C2)=O)ccc(O)cc1O c1(NC(C2C3CN(Cc4ccc(C(C)C)cc4)C2C3)=O)nc(O)nc(O)c1[N+](=O)[O-] C(=O)(CCC(F)(F)C(F)F)N(CCN(C(c1c(C=C)cnn1C)=O)C)C(C)C c1(CC)ncccc1C(N1CCOC(C(=O)NC(c2cccc(C)n2)C)C1)=O N1(C(CCc2cc(C)nc(C)c2)=O)CC2CCC1CN2CCO Cc1nc(CCC(=O)NCCOCCCNC(c2n[nH]c(C3CC3)n2)=O)oc1C C1(C(=O)NCCC2CN(C(=O)Cn3cncn3)C2)CCc2nncn2CC1 c1(C(=O)NC(CC2CN(C(C(C(C)C)O)=O)C2)C)c(C)nn2cccnc12 C1(NC(c2ccc3[nH]ccc3n2)=O)CN(C(=O)Cn2ccnn2)C2CCCCC12 N1(C(c2occ(C)c2)=O)CC(N(C)C(c2coc(CO)c2)=O)C2(CC2)C1 Nc1ccc(F)c(C(N2CCCCC(NC(=O)CCCc3nccs3)C2)=O)c1F C1(NC(C2(C#C)CCC2)=O)CN(C(c2cccc(Cl)c2OC)=O)C2(CCOC2)C1 CS(=O)(=NCC(=O)OC1CCCOC1)c1ccc(Cl)cc1 N1(C(Cc2ccc(C)cc2)=O)CCC(O)(C(=O)NCc2nccs2)CC1 C1(NC(c2c(C)occ2)=O)CCC2(CC1)CN(C(=O)C1=NOC(C)C1)CCO2 C(=O)(C(F)C(C)CNCc1nn(C)c(=O)n1C)Nc1ccc(OC)nc1 CCC(CC(=O)NC12CC(CNC(=O)C(F)C3CCOC3)(C1)OC2(C)C)C(C)C N1(C(CC(C)C)=O)CCC2CC(NC(=O)CCCF)CCC2C1 N1(CC)CC(NC(=O)C(CC2CC2)NC(c2cncc(OCC3CC3)c2)=O)CC1=O N1(C(C=CCOC)=O)CCCCC1CCNC(C1CCCN1CC(F)(F)F)=O C12(CNC(=O)C3=CCC3)CCC(CN1C(c1ccccc1OCc1cscn1)=O)C2 CC1(C(=O)O)CCC(=O)N1.C1CCCC(=O)NC2(c3cn1nn3)CCC2 N1(C(C(C=C)(C)C)=O)CCCC(NC(=O)C(CC2CCCC2)CC)CC1 c1(OC)ccc(F)cc1C(=O)N(C)CC1CCCCN1C(C1CC2(CCC2)C1)=O CCCCC(O)C(=O)NCC(C1(O)CN(C(=O)Cn2nc(C)c(C)c2C)C1)(C)C c1(C(C)OC)nc(C)c(C(=O)NCC(CNC(c2coc(Cl)n2)=O)OC)s1 CC1(C)OCC2CC12C(=O)NC1COCC1NC(C1SC2C=CC1CC2)=O Cc1ccc2c(c1)SCC2(C)C.N1(C(=O)C2CC2)C(C(N)=O)CCC1C c1(C(=O)NCC(C)NC(CC(CCCC)O)=O)cc(C)nc2c1c(O)nn2C CC(C(=O)NCCC1(C(N2CCN(C3CC3)CC2)=O)CCCC1)S(N)(=O)=O C(=O)(N=c1cnn(-c2ccc(Br)cc2)[nH]1)NC1(C)C(C)OCC1 C(=O)(C(CC(C)C)NC(=O)C(CO)NC(=O)C(F)(F)F)NCC(C)N CCN=c1cccn[nH]1.C1(C(c2cn(C)nc2)=O)C2(CC2)C12CC2 c1(OCC)cc(Cl)ccc1C(=O)N(C1CCN(C(C2CC2F)=O)CC1)CCO c1(C(N(CCC(C)NC(C2(C)CC2C(F)(F)F)=O)C)=O)ccc(F)cc1Cl c1(OC)cccc(C(=O)NCC2(C)CN(C(C3CCCN3N=O)=O)CC2C)c1F N1(C(C(C2CCC2)OC)=O)CCC(C(F)(F)F)C(CNC(c2cnn(C)n2)=O)C1 C(=O)(C1CC(=O)c2c(F)cccc21)N1C(CNC(c2ncccc2F)=O)CCC1 c1(C(N(C)CCNC(C2CCC3C(CC2)C3(F)F)=O)=O)ccc2c(c1)C(=O)CCS2 C(C(C)(CC(C)C)NC(=O)CC1C(CC)C1(F)F)NC(c1c(CC)nccc1)=O c1(C(N2CCCC(NC(C(C)OCC)=O)(CC)C2)=O)ccc2c(c1C)CCC2 C1(NC(C2C(=C)C2)=O)CC(F)(F)CN(C(=O)CN(CC)CC)C1 N1(C(CC2OCCN(C(CCCN(C(C)C)C)=O)C2)=O)CC(O)(C2CC2)C1 C1(=O)CCCN1.C1(=O)C(C2(O)CCC2)N(CC)CCN1.C(=O)(OC)NC c1(C(=O)NC2CC3(CN(C(c4c(C)ccn4C)=O)C3)C2)nc2ccccc2[nH]1 N1(C(C2C(C=C)C2)=O)CCC2(CCCN2C(c2nnc(O)nc2O)=O)C1 c1(OC)nc(Cl)ccc1CN1CCC(NC(c2cccnc2C)=O)C(F)C1 CC1(C(N2CCC(CCCNC(c3cc(C#N)on3)=O)CC2)=O)CCC(=O)NC1 c1(C(N2CCC(NC(c3c(=N)cc[nH]c3)=O)CC2)=O)cc2cnccc2cc1F c1(C(=O)NCC2C(NC(CC(=O)OCC)=O)CCC2)ccc(CC)c([N+](=O)[O-])c1 C1(C(C)(C)C)CC(C(=O)N2CC(F)CC2C2(NC(=O)Cn3nccn3)CC2)=NO1 C(=O)(CCC(C)(C)C#N)N(CC)CC1CCCN1C(c1coc(Br)c1)=O CCC(C)(C)CCCC(=O)NCC(CNC(=O)C(C)(C(C)C)NC(C)=O)OC N1(C(CN(C(=O)CC(=O)O)CCOC)=O)CCC(CC#N)C1 c1(CCC(=O)NC2CC(NC(c3cc(-c4ccccn4)no3)=O)C2)cnc(O)[nH]1 O(NC(=O)C(Cc1ccco1)NC(c1sccc1C#N)=O)C(C=C)C C1(CC)(NC(=O)CC2CCCC(=O)N2)CCN(C(c2ocnc2C)=O)CC1 C=CCC(C(=O)NC(c1cccs1)CC)NC(c1nnsc1N)=O CC(C)C(F)C(=O)N1CCC(C(C)NC(=O)C(C)CC2CC2)C1 CC1(C(N2CCC(NC(c3ncoc3C3CCC3)=O)C2)=O)CCCS1(=O)=O CCC(CC)(CN=c1[nH]c(OCC)ncc1F)NC(=O)CCn1cnc(C)cc1=O CSC1=C(C(=O)NCC2CCCN2C(=O)C=CC=C(Cl)Cl)CCCC1 C1(NC(c2cn(C)[nH]c2=N)=O)CCN(C(=O)Cn2nccn2)CC(C)(C)C1 C1(C(=O)NCC=C=C)CCCN(C(c2ccc(CO)nc2)=O)CC1 N1(C(CNC(CC)=O)=O)C2CCC1C(C(=O)N(C1CN(C)CC1O)C)C2 C1(CNC(CCC#C)=O)CN(C(=O)C(C)(O)C=C)CC1(C)C C12(CC(=O)NC(c3ccc(C)o3)CCC)CCC1CN(C(=O)C(O)C(C)C)C2 C(=O)(C1=C(C)OCC1)N1CC(COCC)(NC(c2ccncc2CC)=O)C1 N1(C(CC(=O)NC)=O)CCCC(NC(c2ccn(CCN(C)C)n2)=O)CC1 C(=O)(C1Cc2c(Cl)cccc21)NC1(C)CN(C(c2cnc(F)c(Cl)c2)=O)C1 N1(C(CC2CCC(C(=O)Nc3c(C)nn[nH]3)C2)=O)CC[Si](C)(C)C1 c1(C(=O)NC2C(CNC(C(C)(C)OC(C)=O)=O)CC2)cc2cccc(C)n2n1 c1(C(=O)NCC(C)(C2CCC2)NC(C(C2CC2)OC)=O)csc(CS(C)(=O)=O)n1 c1(C(N2CCC(C(N)=O)C2)c2ccccc2)ccc(Cl)cc1 c1(C(=O)NC(CNC(c2cc(CC)c(F)cc2)=O)CCOC)cnc2n1CCCC2 N1(C(c2cc(C(C)C)n(CCO)n2)=O)CC2CC(NC(=O)C=CCO)C1C2 c1(C(=O)NCCN(C(CCCCC=C)=O)C2CC2)ccc2nc(C)oc2c1 CC1CC(NC(=O)N(C(C)C(F)F)C)CCCN1C(=O)OCc1ccccc1 c1(C(=O)NCCCOC(=C=C)C)n[nH]c2c(C)cc(Br)cc12 c1(CNc2cc(OC)cc(Cl)c2Br)cc(Cl)cc(S(C)(=O)=O)c1 N1(C(CCCOCCC)=O)CCC(O)(CNC(c2ccn(C)n2)=O)C1 C(=O)(C1CCc2scnc21)NC1(C)CN(C(=O)Cc2ccc(Cl)cc2Cl)C1 N1(C(c2cc3ccsc3n2C)C(=O)NCCCC)CCCCC1C1(C)CCCO1 C1(O)(CN(C(=O)COC2CC(F)(F)C2)C)CCCN(C(=O)C2=CCN(C)C2)C1 c1(SC)ccnc(C(=O)NC2CN(C(=O)C(F)CC3CCCCC3)C2)c1 C(=O)(C(C)CC(F)(F)F)NC(N(CCC(C(C(C)=O)CC)NCCSC)C)=O C#CCC1C(=O)N1.C(c1cocn1)=CC(N1CC(NC(=O)COCC)C1)=O N1(C(C2C(C)C2)=O)CCCC(N(C(=O)C=C2CCC2)C)CC1 c1(C(N2CCCCC(CNC(=O)C3=CCCSC3)C2)=O)ccc2nccn2c1 C1(CC=C)(NC(CCC#C)=O)CN(C(=O)C(C)OC(C)C(=O)NCC)C1.C1(O)CCCC1 n1(CCC(N2CC(O)(CNC(C(C)NC(=O)OC)=O)C2)=O)c(C)csc1=O C(=O)(C1=C(C)CCCC1)NN(C(c1ccc(NC(=S)NC2CCC2)cc1)=O)CC c1(CN)cn(CC2C=CCN2C(=O)CC2(CNC(c3ccco3)=O)CC2)nn1 c1(C(C(N2CC(N(C)C(C3CC3C(F)(F)F)=O)C2)=O)O)cccc2c1OCC2 C12CCCN(C1)C(=O)C(c1ccc(F)cc1)NC2=O.C(C(=O)OC)OC n12cc(cn1)C(=O)NC2C.C(=O)(CC(O)C1CCCC1)NCCOC1CCCC1 N1(C(c2cc(CC)no2)=O)CC2CC(CNC(=O)CCn3ccnc3)C2C1 C(C(C)(CC(C)C)NC(=O)C(c1cnn(C)c1)C)NC(C(C)OCC#C)=O N1(C(CC(CCCCC)O)=O)CCC2(NC(c3ccncc3)=O)CCCCCC12 CC(C)(C(=O)N1CCC2(CC2C(N2CCC(c3ccccc3F)C2)=O)C1)C(F)F C(CC(C)C)(C(=O)N1CC(OC)CC1CSC)N(C(C=CC=CCC)=O)C N1(C(C(=O)NC2CCCC(C(C)C)CC2)=O)CCC(F)(F)C(C)C1 Cc1ccnnc1-c1ccc(CCNC(N2CCCCC2CC(C)O)=O)cc1 C1(C(=O)NC(c2ccccc2Cl)CO)CC(O)CN1C(=O)Cc1ccc(O)cn1 Cc1c(C(=O)NC2(C)CCCN(C(C3CCCCS3)=O)C2)[nH]c2c(Cl)cccc12 N1(C(C(CC)(C)OC)=O)CC=C(C(=O)N2CCC=C(Cl)C2)CC1 C(CCC(C)C(=O)NCC(C)(C)CN(C(=O)CN1CCCCC1)C)OC N1(C(c2c(NC)nccc2)=O)CC2CC(NC(=O)CC3CCCCCC3)CC1C2 Cc1[nH]nc2ncc(C(N3CCC(F)(CNC(C4CC4(F)Cl)=O)CC3)=O)cc12 Cc1c(F)ccc(Cl)c1C(N1CC=CC(NC(c2cc(Cl)n(C)n2)=O)C1)=O c1(N(C)CC2CC2)ccc(C(N2CCC(C)(NC(=O)COC3CC3)C2)=O)cc1 c1(C(=O)NCC(C2CCOC2)NC(=O)COC2CC2)cccc(-n2cccn2)n1 c1(C(=O)NC(C(C)C)CCN(C(=O)C(C)(C)CN(C)C)C)cc2c(ccn2C)[nH]1 c1(C(=O)NC(C2(CNC(CN3CC(C)C3)=O)CC2)C)c2c(nn1C)CCOC2 c1(C(N2CC(NC(c3c(CC)c[nH]c3)=O)C(C)C2)=O)cccc(F)c1OC(F)(F)F c1(OC)cc(C(N2CC3CC(NC(c4ccc(C)c(F)c4)=O)C2C3)=O)ccc1C c1(N2CCC(O)(CCNC(=O)CCCN3CCCC3)CC2)ncc([N+](=O)[O-])cn1 N1(S(CC)(=O)=O)CCCC(C(=O)NC2CC(CNC(C3(CO)CC3(F)F)=O)C2)C1 N#Cc1cccc(CNC(=O)CC2CCCN2C(=O)COc2cccc(I)c2)c1 c1(CC)c(C(N2CCN(C(C)=O)CC2C(F)(F)F)=O)ccc(Br)c1F N1(C(CC(COC)C)=O)CCC2C1CCCN2C(=O)CN(c1ccccc1)C C1(NC(CC2(C(=O)NC3(C(=O)OC)CC3)CC2)=O)CC2C=CC1C2 c1(OC)cc(C(=O)N(CC(C)CNC(c2ccc(CO)s2)=O)C)cc(C)n1 N1(C(C(CC#C)CC#C)=O)CC(NC(=O)CCC(=O)NC)CC12CCOC2 C1(OC)CN(C(n2ccnc2C)=O)CCC1NC(=O)CC1CCCCO1 C(=O)(C(F)(F)CCn1ccnn1)NC(c1nc(C)[nH]n1)CC.C1(=O)CCN1 c1(OCCN2CCCCCC2)cccc(C(=O)NCC)c1 c1(C(=O)NCCC2COCCN2C(C2(c3cc[nH]n3)CC2)=O)cnc(O)nc1O Cc1cccc2c(CC(C3CC3)NC(=O)CCNc3cnn(C)c3)c[nH]c12 N1(C(C2N(C(CCN(C)C)=O)C3C(C2)C3)=O)CCCC(F)(F)C(F)C1 c1(OC)c(C(=O)NCC23CC(NC(=O)C(n4cc(Cl)cn4)C)(C2)C3)c(C)nn1C N1(C(c2ncn(C)c(=O)c2)=O)CCC(C2(O)CCN(C(=O)CSCC(N)=O)C2)CC1 c1(NC(C2CCC3CCC2N3C(=O)Nc2cn[nH]c2)=O)ccc2nccn2c1 C12CC3(CCN(C3)C1=O)CO2.c1(CNC(CCOCCCOC)=O)ncn(C)n1 C1(C2CN(C(=O)CC3CCC(NC(C)=O)CC3)C2)(NC(C(C=C)O)=O)CC1 C1(CC(=O)NC2CCCC(NC(C3(SC)CCC3)=O)C2)CCCNC(=O)C1 c1(N2Cc3c(ccc(OC)c3)C2)cc([N+](=O)[O-])c(C(F)(F)F)cc1OCCC(C)C c1(C(N2CC(NC(C3(OC)CCCC3)=O)C2)=O)cnn2ccc(C#N)cc12 N1(C(c2n(C)ncc2C#N)=O)CCC(F)(F)C(CNC(=O)CC2C=CCC2)C1 c1(C(N2CCC3(CCSC3)C2)C(=O)NC(CC)(C)C)ncc(C#N)cc1C C(CC(C(=O)NCC(C)(C)C1CCC1)NC(=O)CCc1cc(C)no1)OC n12cc(nn1)C=CC(=O)N1CC(CC)(C1)C2.c1(C)ccccc1.C(C)(C)(C)NC(=O)O C1(C(=O)NCC2C(NC(C=CCCC(C)C)=O)C2)C2CCC1(C)C2(C)C C1(C(=O)NCC2CCCC2NC(C2(C(F)F)CC2)=O)COc2ccccc2O1 N1(C(CCCn2cc(C(CC)CCC)nn2)=O)CCn2cc(C)nc2C1COC c1(C(=O)NC2CC(NC(C3(C=C)CCCCC3)=O)C2)cccc2[nH]c(C)cc12 C1(NC(=NC)NCC(N2CC=CCC2)=O)CCc2nnc(C(F)F)n2C1 C#Cc1cc(NC2CCC(S(C)(=O)=O)C2)ccc1Cl C(=O)(C(O)CC[S+](C)C)N(C1CC(NC(c2ccc(C#N)s2)=O)C1)C C1(CNC(CC(CC)OC)=O)CCCCN(C(=O)COCC(F)(F)F)C1 C1(C(=O)NCC2(OC)CCN(C(=O)C(F)=C(C)C)CC2)CCc2ccccc2C1 N1(C(COCCC)=O)CCC(CNC(=O)CC2C(C)(C)C2(C)C)(COC)C1 c1(SC)ncc(C#N)c(N2CC3C(NC(=O)Cc4cc(F)cc(F)c4)C3C2)n1 c1(C(=O)NCCC2(NC(C(C3CCCC3)OC)=O)CCC2)cc(C)c(=O)n(C)c1 C(=O)(C1SCc2cccnc21)NCCN(C(=O)Cc1cn2ccsc2n1)C(C)C c1(C(N2CCCCC(NC(c3c(C)nc(C)s3)=O)C2)=O)ccc2sccc2c1 CCCCS(=O)(=O)NC(CC1CCC1)C(N1CCC(SCc2ccccc2)CC1)=O c1(C(CNC(C2C(C)C2)=O)NC(=O)CCc2cncn2C)ccccc1F N1(C(c2n(C)ccn2)=O)CC2(CC(C(N3CCC3CO)=O)CO2)C1 C1(C(N2CCC(CC(C=C)O)CC2)=O)CC2OC1C1CC21.CC(C)C(=O)C=O c1(C(N2CCC(C(C)(C)NC(c3cn(CC=C)nn3)=O)C2)=O)cc([N+](=O)[O-])n[nH]1 c1(OCC)ncc(NC(C2CC(O)CN2C(c2cc(C)on2)=O)=O)cn1 CC1CC(NC(C2C3CCCOC23)=O)CN(C(=O)CCC2CCCC2)C1 CC1=C(C)CC(C(=O)N(C(C)CCNC(C2C=CCCC2)=O)C)CC1 C1(CNC(=O)C(F)n2cccn2)CC2COCC2N1C(c1cccc(Cl)c1)=O C12(NC(CCCC=C)=O)CCCC1CN(C(c1cnccc1COC)=O)C2 c1(CC)ncc(C(=O)NCCC2(OC)CN(C(C3(O)CCSC3)=O)C2)c(C)n1 c1(C(=O)NCCC(CNC(c2nc(CCC)oc2)=O)O)cn(C)[nH]c1=N c1(C(=O)NCCOC2CCN(C(C(C)NC(C)=O)=O)C2)cccn(CCNC)c1=O c1(C(=O)NCCOCCN(C(c2c(C)noc2)=O)C)cc(C#N)c(N)cc1O N1(C(CCN(C(c2cc(F)cnc2O)=O)CC)=O)CCC(C2CCOC2)C1 N1(C(C=C(C)C(F)(F)C(F)(F)F)=O)CCCC2(CCN2C(C2C3CC4C(C3)C24)=O)C1 c1(NC)ccc(C(=O)NCC2CN(C(=O)CCC3CCOC3)C(C)(C)C2)cc1F N1(C(c2cn(C)nc2)=O)CCC(F)C(NC(=O)CNC(c2cccc(F)c2)=O)C1 c1(C(=O)NC(CC)(C)CNC(C2CNC(=O)C2)=O)occ(C)c1C N(C1C(=O)Nc2cc(Cl)ccc21)C(c1ccc(C)cc1C(F)F)=O c1(C(=O)NC(C)CCCNC(c2cnc(C(F)(F)F)nc2)=O)cccn(C)c1=O C(c1sccc1Br)=CC(=O)NCC(C)NC(C1(F)C2CCCC12)=O CC(C)(C)C(CNC(C1CCC12CCC2)=O)NC(=O)CCc1ccccc1 C#CCC(C)(C)C(c1nnnn1Cc1ccco1)NCc1cnc(F)c(C)c1 Cc1cc(Br)c2oc(C(N3CC=CC3CNC(=O)C3=CCCOC3)=O)cc2c1 C1(N(C(c2nc(C)sc2)=O)C)C2CN(C(C3CNC(=O)N3)=O)CC12 N1(C(c2c(C)oc(C)c2C)=O)CC2CCC(C1)C(NC(C1C=CCC1)=O)C2 C(=O)(C(C)C(C)(C)C)NCC(CCNC(c1ccc(CC(C)C)s1)=O)O CC(CC(=O)NCC1(NC(=O)Cc2ccsn2)CCCC1)n1cc(Br)cn1 Cc1cc(NNC(=O)N2CCC2CC(=O)N(C)C)nc(=N)[nH]1 N1(C(C(C)=O)=O)CC(C)C(C)(CNC(c2ccc(F)c(CO)c2)=O)C1 N1(C(C2C(C)CC2)=O)CCC2(CCC2NC(=O)Cc2ccc(F)cc2Cl)CC1 O=[N+]([O-])c1cc(-c2cccc(C(C(Cc3ccccc3)N)O)c2)nc(Cl)c1.C1(CO)CC1 C1(COC)COCCN1C(=O)C(CCC1CCC1)NC(=O)Cc1cn(C)nn1 c1(C(=O)NC2C(C)(C)C2c2nc[nH]n2)ccc(F)cc1Nc1ncccn1 C1(NC(CCc2nc(C)c(C)[nH]2)=O)CCCN(C(=O)C(CO)C(C)C)CC1 CCC(CC(=O)NCC1CCC(C(=O)NC(c2nccn2C)C)CC1)C(C)C C1(C(=O)O)(NCc2cccnc2F)CCOCC1 C(C(C(C)(C)C)NC(C1CC1NC(C)=O)=O)NC(C1(CCC)CC1)=O c12nc(c3ccccc3n1)n2C.c1(COCC)ccc(CNC2(OC)CC2)o1 c1(C(=O)NC2(CNC(c3coc(Br)n3)=O)CC2)cnc2[nH]ncc2c1 C1(NC(=O)CC2(O)CC2)CCC(NC(C2(C(F)(F)F)CCOCC2)=O)CC1 N1(C(c2nc(C(C)NC(C3CC=CC3)=O)oc2)=O)C2COCC1C2 CC1=C(C(=O)N2CCCC(N(C(=O)CCNC(c3ccoc3)=O)C)C2)CCC1 C12CN(CCC13CCC3)c1ccc2cc1.c1(C(N)=O)cnc(C2CC2)o1 CCC(CC)CCC(=O)NC(C)(C)CCNC(C1CC(C)CO1)=O N1(C(c2cnc[nH]2)=O)CCC2(CCCN2C(=O)CN2CCS(=O)(=O)CC2)C1 c12cc(nc(OC)n1)N2.C(CCNC(=O)OCC)N(C(C)C)C(C)C N1(C(C(CCOC)NC(=O)C(c2ccn(C)n2)C)=O)CCCC(CCO)CC1 N1(C(C2(OC(C)=O)CC2)=O)C2CCC1CC(O)(CNC(=O)C(O)c1ccsc1)C2 N1(C(c2n[nH]c(C)c2C)=O)CCN(C(c2cc(Cl)cn2C)=O)C(C(C)C)C1 C1(C(=O)NC(C(N2CC(C)OCC2)=O)(C)C2CCC2)CCC=CCCC1 c1(C(=O)NC2CCC(NC(c3cc(C)cc(O)c3)=O)C2)ccc2c(c1)OCCO2 N1(C(C=C(C)c2ccc(F)cc2)=O)C2CCCC1CN(C(=O)C(=O)C(C)(C)C)C2 CC1CC(C)OC1CNC(=O)CCCNC(N)=O N1(C(CCC(C)OCC)=O)C2CC1CN(C(=O)CC1OCCC1(C)C)C2 N1(C(COCC(=C)C)=O)CC(NC(=O)CC2CCCNC(=O)C2)CC(C)(C)C1 c1(C(C)NCC#CCN(C)C)c(F)cccc1F CC1OCCN(C(=O)CC2CC(=O)NC2=O)C1C(=O)NC1COCC1CO C(=O)(C(F)C(F)(F)C(F)(F)F)NCC1(F)CCN(C(C(C)(C)F)=O)C1 C1(C(=O)NCCc2onc(CC)n2)CC(F)CN1C(=O)CCc1nncs1 c1(CNC(C(C)=C2CC2)=O)nc(C(N2CCC(F)(CF)C2)=O)c(C)o1 C(=O)(C(C(C)(C)C)SC)NCC1CN(C(c2n[nH]c(CC)c2Cl)=O)C(C)C1 c1(OC)c(C(N2CCC(C)C2C(=O)N(C)Cc2cc(C)n(C)n2)=O)cnn1C c1(CNCC2N(C(c3n(C)ncc3Br)=O)CCCC2)ccc(F)nc1F CN1CCC(C2(C(=O)NCC3CC(C)(C)CN3C(=O)C3CC3)CC2)CC1 c1(NCC)cc(Cl)ccc1C(N1CCCC(C(=O)NC2CC2C2CC2)(OC)C1)=O CC(C(O)C(=O)N(Cc1ccco1)CC1(n2cc(Br)nn2)CC1)c1ccccc1 CNS(=O)(=O)NCC(=O)NCC1COCC1NC(=O)C(c1cnn(C)c1)O N1(C(C(C2CCC2)OC)=O)CC2CCC2(CNC(=O)Cc2nncn2C(C)C)C1 C1(CC)OCCC1C(=O)NCc1csc(C(=O)N(c2cnn(C)c2)CC)c1 C(C(C)(F)C(C)(C)F)NC(CC1(C)N(C(CCCN(C)C)=O)CC1)=O N1(C(=O)CCF)CCC(CC2COCCN2C(C2CCSCC2)=O)CC1 Cc1ccnc(C#N)c1NC(C12CC(NC(c3cnn(C(C)C)c3)=O)(C1)C2)=O C1(C)(C(N2C3C(CNC(CN(C(C)=O)C)=O)C(C3)C2)=O)CC2C=CC1C2 Nc1cc(C(N2CC(CNC(=O)CC3CCC(=O)NC3=O)C(O)C2)=O)cc(Cl)n1 C1(CNC(c2c(C)coc2C(C)C)=O)CC(C)(C)CN1C(C1CCCS1)=O S(=O)(=O)(c1c[nH]c2ncccc12)NC(=O)C1=CCCS1 C1(O)(C(C)NC(=O)Cc2cnoc2)CN(C(=O)Cc2ccn(C)n2)C1 C(=O)(C(CC(C)C)OC=CC=C)N(CCC)CCNC(CC1CCCCC1)=O Cc1cc(C(F)F)ncc1C(N1CCN(C(C2CCC3(CCC3)O2)=O)CC1C)=O C12(C)CCCN1C(=O)CC2.C1(C(=O)NCCOC(CC)CC)CC2(CCC2)C1 N1(C(Cc2ncc(CC)[nH]2)=O)CCC2(CC1)CN(C(=O)CC(C)C1CCCC1)C2 C1(NC(C2(C3CC3)CN(C(=O)C=CC3CCCCC3)C2)=O)C2CCC3C(C2)CC13 C1(NC(CCCC=C)=O)CN(C(=O)CC2CCCC(C)(C)O2)Cc2nccn2C1 c1(C(=O)NCCN(C(=O)CCc2ccsc2Cl)CC(C)O)occc1F c1(CNC(C2CC23CC3)=O)cncc(C(N2CC(c3ncc[nH]3)C2)=O)c1 c1(C(N2CCC(N(C(C=C(CCC)C)=O)C)C2)=O)cnc(O)cc1OC c1(-c2c(C)cc(C(N3CC(N(C)C)C(O)C3)=O)cc2)ccccc1S(C)(=O)=O Cc1nn(C)cc1C(O)C(=O)NCCCC(C)(C)NC(c1ccncc1)=O C(=O)(C(CC(F)F)C(C)(C)C)NCC(CNC(c1c(C)nc(N(C)C)s1)=O)(C)C c1(C(=O)NCCC(C)NC(=O)CNc2ccccn2)coc(C2CC2)c1 C1(CNC(CNS(CCCC)(=O)=O)=O)CCC12CCN(C(=O)C(C)(C)CF)CC2 C(=O)(C1CCCc2c[nH]nc21)N1CC(O)CC(NC(Cn2c(C)ccn2)=O)C1 C(=O)(NNC(=O)NCc1ncon1)c1snc(C)n1 c1(OC)cc(Cl)ncc1C(N1CCC(O)(C(=O)Nc2cccc(Cl)n2)C1)=O C1(CC)C(C(=O)N(CCCC2CC2)C2CC2)CCCN1C(C1CC1c1ccco1)=O c1(OC)nn(C)cc1C(N1CCC(CC(=O)NCCc2cccs2)C1)=O N1(C(C(C)=O)=O)CC2(C(=O)N=c3ccn(CC(N)=O)[nH]3)CC1CCO2 Cc1nc2ncnn2c(NCCCCC(C)NC(=O)CC2CC3(CC3)CO2)c1C c1(OCC)nccc(C)c1C(=O)NCC1=CCCOC1 C(C(F)(F)C(=O)N(C1CCN(C(C2COCC(C)O2)=O)CC1)CC1CC1)OC Cc1cc(N2CCCC(CNC(=O)CCSCc3csc(C)n3)C2)nc(C)n1 C(=O)(CCCC(C)(C)NC(=O)C(c1ccn(C)c1)C)NCC1N(CC)CC1 C1(CCCC)CN(C(=O)C(C)C(C)(C)C)CCN1C(=O)CCCOCN(C)C N1(C(C2N(C(COCCC#C)=O)CC=C2)=O)CCC2(COC(C)C2)C1 N1(C(C2(C)CCCS2)=O)CCCC2CN(C(C3CCCC4(CC4)C3)=O)CCC12 C(C(C)C(C)C(=O)NC1(CNC(c2ccnc(O)c2Br)=O)CCC1)OC C(=O)(C(=O)N=S(C)(C)=O)NC1CCCC(NC(c2cccc(C(=O)OC)c2Cl)=O)C1 C1(NC(c2cnn(C(F)F)c2)=O)CC2CC1N(C(=O)Cc1csc(C3CC3)n1)C2 Cc1cn(CC(=O)NC2CC(F)(CNC(C3CCC3)=O)C2)c(=O)nc1O N12CCN(C(=O)CC1)C2=O.CC1(C2(c3nc(-c4cccnc4)no3)CC2)CC1 C(CC(F)(F)Cn1cc(CO)nn1)NC(c1ccn(-c2ccccc2)n1)=O N1(CC)CCCC(CNC(C2C3CN(C(c4sccc4Cl)=O)CC23)=O)C1 CCC(C)C(=O)C(=O)OCc1cc(F)ccc1F c1(N2CCCC(C(N3CC(C(C)C)N(C)CC3)=O)C2)ncc2ccc(F)cc2n1 C1(NC(C2(C)CCSCC2)=O)CC(F)CN(C(C2CC3C=CC2CC3)=O)C1 C1(CC(=O)NCCOCCC(=O)NCCC2CCCOC2)CCCOCC1 c1(CC(N2C(C(=O)NCc3sccc3Cl)CC2)=O)ccc(F)nc1 Cc1[nH]c2ccccc2c1C(N1CCOC(C(C)NC(=O)C(=O)NC2CC2)C1)=O Cc1sc(Cl)nc1C(N1CC(=C(F)CNC(C2CC(=O)N(C(C)C3CC3)C2)=O)C1)=O C(=O)(C(O)C(C)(C)CC)N1CCC(O)(C(C)NC(CC(=O)NCC)=O)CC1 c12cc(on1)CC(=O)NCCN(C)C2=O.C1(COC)CC(CC(=O)OC)C1 C1(C(=O)NCCCCN(C)C2CC2)CCN(C(C2CC3(CC(=O)C3)C2)=O)C1(C)C N1(CC(C=C)N(C)C)c2ccccc2CC1C C1(NC(C(C)CC2CCC2)=O)CC(F)CN(C(c2cc(C(=O)OC)cs2)=O)C1 c1(C(=O)NCC(C2CCOC2)OCC)ccc(OCC(F)(F)F)nn1 C1(C)(CNC(C2(CC=C)CCC2)=O)CCCC1NC(=O)CCN1CCCCCC1 N1(C(c2cn(C)nc2)=O)CCCCC1CNC(C1CC1(c1ccccc1)C)=O C(=O)(CN=S(C)(C)=O)NCCC1N(C(c2c(SCC)nccn2)=O)CCSC1 CC1CCC(CNC(c2cccc(CO)n2)=O)CN1C(c1ncn(C)n1)=O N1(C(CCOCC)=O)CCC(CF)(NC(=O)Cc2cc(C)n(C)n2)C1.C1CS1 c1(OC)cc(C(N2CC(NC(=O)COCCSc3cccs3)C2)=O)c(Cl)cc1Cl C1(C)(CNC(CNC(C(CC)C)=O)=O)CN(C(=O)CC2(C#N)CC2)CC1C c1(C(=O)NCC23C(CN(C(CC4(C(=O)OC)CC4)=O)C2)C3)cccc(P(C)(C)=O)c1 C1(CNC(=O)CCOCCCNC(C23CCC(C2)C3)=O)CC2CCC2C1 Cc1csc2ncc(C(=O)N(C3CN(C(C4CCCCS4)=O)C3)C)n12 c1(SCC(=O)NC2CCN(C(C(C)OCC)=O)CC2)nc2ccccc2o1 c1(OC)cc(F)cnc1-n1cc(CN(O)C(c2ccc(C(=O)O)c(Cl)c2)=O)nn1 c1(-c2cccc(OC)c2)ccc(S(=O)(=O)NNC(=O)C2CCC(=O)N2C)cc1 c1(CNC(c2nc(NC(C)=O)sc2)=O)cc(C(=O)NC(C)CN(C)C)ccc1F C(=O)(C(C#N)CC)N1CCN(CC(C)(C)NC(c2c(CC)ccs2)=O)CC1 Cc1ccncc1CNC(c1csc(-c2ccccc2)n1)=O CC1CCCN(C(=O)Cc2csc(-n3cc(-c4cccnc4)nn3)n2)C1C(=O)O c1(C(=O)NCC(C(C)C)NC(C2CCCN(C(N)=O)C2)=O)cc2nc[nH]c2cn1 N1(Cc2c(C)nc(-c3ccc(Br)cc3)o2)c2ccccc2CC1C C(=O)C(C)(C)CC(=O)N(C)CCN(C(=O)C(O)CN(C)C)C.CCOC c1(C(N2CCC(N(C(C(C)C)=O)C)C(C)C2)=O)c(O)cc(Cl)cc1F c1(CC2C(NC(c3ncc(CN)s3)=O)C2)cccc(Br)c1 C(=O)(CCCCCNCCC1(C(=O)NC)CCCO1)N(CCOC)CC1CC1 N1(C(C(C)OCC=C)=O)CCC(CN(C(=O)CN(C)CCC)C)C1 c1(CC(C)CNC2(C3CCCO3)CC2)ccc(CCC(=O)N)cc1.C(=O)O CCC(C)(C)C(=O)C(=O)NC(C)(C)CCNC(C1CC2(CCOC2)C1)=O C1(C(=O)NCCOCC#C)(NC(=O)C(C2CCOC2)SC)CCN(C)C1 n1(CC)nc(C)cc1C(=O)NCc1nc(C(=O)NC(C)(CO)CCF)c(C)o1 C1(C(=O)NCc2c(CN(C(C(F)OC)=O)C)cccc2)CC2(CCC2)CO1 N1(CC(=C)C)CCN(C(=O)COC2CCN(C(c3ccsc3)=O)C2)CC1 N1(C(C2(C)CN3C2c2cc(no2)C3=O)=O)CCC2(CC(OC)C2)C1.CO.OC C1(NC(C2(CC=C)CCN(C(=O)C(C3CCOCC3)C)C2)=O)CC2(C1)CN(C)C2 C=CC1(CC(=O)NCC2C=CCN2C(C2CC23CC3)=O)CCOCC1 C(=O)(CC(F)(F)c1ccccc1)N1CCC(N(CC2C(C)CCO2)C)C1 N1(C(CCc2ccc(C)s2)=O)CC(C(=O)Nc2ccnc(O)c2)CC(F)C1 N1(C(CN(S(C)(=O)=O)C)=O)CCCCC(NC(c2nc(C(F)(F)F)no2)=O)C1 C12(C(=O)NC3C(CNC(C4(C)CCC4)=O)CCC3)CC3CC1C2C3O CC1CNc2ccccc2C1N(C=O)Cc1cccc(C(C)(C)C)n1 c12cn(nn1)C1CC(C1)C(=O)NCC2.C1(CC)CC1C(=O)OC(C)(C)C C1(NC(=O)NC(CC)S(C)(=O)=O)CCC2(CC1)CC(CC(=O)OC(C)(C)C)C2 C1(NC(C(CC)N(CC)CC)=O)CC2C1CCN2C(c1cc(F)ccc1O)=O C1(C(C)NS(=O)(=O)CC2(NC(c3cocn3)=O)CCC2)CCC(C(N)=O)CC1 c1(OCCNC(C2CCCN(CCO)C2)=O)ccc(-n2cc(Cl)cn2)cc1 c1(CC(=O)NC(C2(O)CN(C(C3CCC4CC34)=O)C2)C)ccc(C(F)(F)F)nc1 N1(C(=O)NC(C(=O)OC)C(C)(C)C)CCC(C2CC2)(NC(C)(C)C)C1 c1(C(=O)NC2CCN(C(CCC(C)OCC)=O)C2CC)cccc2nc(C)nn12 N1(C(N=c2cc(C3CCCN(C(C)=O)C3)[nH][nH]2)=O)CC2CCCC(CO)C2C1 N1(C(C2N(C)CCC2)=O)CCC2(C(=O)NCCCc3cnccn3)CCCC12 N1(C(CSC(C)=O)=O)CCC(Nc2ccc(C(F)(F)F)c(Cl)c2)C(C)(C)C1 N1(C(c2cnn(C)c2C(N)=O)=O)CCC(F)C(NC(=O)OC(C)(C)C)C1 C1(N(C(C(C)C2CC2)=O)C)CCN(C(=O)Cc2cn(C)nn2)C1 C1(C(C)OC(N2CCC(C(=O)OCC)(OC)C2)=O)CC2(C1)CC1(CC(F)(F)C1)C2 c1(CNCC2(C)C(C)(C)C2c2nc(N)n[nH]2)ccccc1COc1ccccc1 c1(C(=O)OC(C2(C(=O)OCC)CC2)C)ccc(O)c([N+](=O)[O-])c1 CCCC(C)C(C)(c1nnnn1Cc1cccs1)NCCSc1cccc(Br)c1 c1(CC)onc(C(=O)NCC(C)(CNC(c2scnc2C(C)(C)C)=O)OC)c1C C(=O)(C(CC=C)CC(C)C)N1CC(c2n(CC)c(S)nn2)C12CCC2.C1C(=O)N1 N1(C(CCc2ccc(C)nc2)=O)CC2COCC(C1)N2C(=O)C=CC1CCCC1 c1(C2(C(N3CCC(C)(CNC(COCC)=O)C3)=O)CC2)ccc(Cl)cc1F N1(C(c2cc(OCC)no2)=O)CC(O)CCC1C(N1CCC(C(N)=O)CC1)=O c1(C(=O)NCC2CC(NC(C3CCS3(=O)=O)=O)C2)cscc1CC1CCC1 CCCCS(=O)(=O)NC(C)C(=O)N(C)CC.C1(=O)C(C2CC2)N1 CC1(C)CCC(N=c2[nH]c(N3CCC(C(F)F)CC3)nc3c(F)cccc23)CC1 C=CC(O)C(=O)NC1CCN(C(C2CCCN2C2CC2)=O)C1 CCCC(F)C(=O)NCCN(C(=O)CSC(F)(F)F)C1CC1 C(=O)(C(C)(C)CCCO)NCC1CC(C)N(C(=O)CC2CCOC2)CC1 c1(C(N2CCC(N(C(C(CC)C)=O)CCO)C2)=O)cncc(Br)c1 c1(C(N2CC(CCC)N(C(=O)CSS(C)(=O)=O)CC2)=O)cccc2c1OCCO2 N1(C(C(C(C=C)C)C)=O)CC(CNC(c2cnc(C)[nH]2)=O)OC(C)(C)C1 c1(CNCC(CC)(CC)CO)ccc(S(=O)(=O)NCc2ccccc2)s1 Cc1cccc(OCC(=O)NCC(C2CCCC2)NC(C2CCO2)=O)c1C C(=O)(CCC(C)(F)F)NCC(C1CCN(C(c2c(C)cc[nH]2)=O)CC1)(C)O C1(O)(CNC(CN(C)CC)=O)CCCN(C(=O)CN2CCCCC2=O)CC1 c1(C(N2CCC(COC)(NC(=O)Cc3cnc[nH]3)CC2)=O)cc2ccccc2[nH]1 Cc1ccc(-c2nc(C(C(F)(F)F)NC(=O)Cc3ccccc3)n[nH]2)cc1C(=O)O N1(C(C2(C=C)CCN(C(=O)CCC3CC(OC)C3)C2)=O)CC(O)CC12CCC2 CCC(C)(CO)C(=O)NCC(C)(O)CNC(c1cc2n(n1)CCO2)=O C(C)(CO)(C(=O)NC1CN(C(=O)CSCc2ccncc2)CC1SC)SC N1(C(CC(=C=C)C)=O)CCC(C2CCOCC2)(CNC(=O)C(C)CN(C)C)C1 C#Cc1cncc(C(N2CCC(F)CC2C(=O)NCC(C)C(C)(C)C)=O)c1 C1(OCCCCC#C)CC2COCC(C1)N2C(=O)OC(C)(C)C C1(C(=O)NC2C(CNC(c3nc(COCC)sc3)=O)CC2)COCCN1C CS(=O)(=O)CCCC(=O)N1CCC(O)(CNC(C2CCc3[nH]nc(O)c3C2)=O)C1 C1(O)(CC)CCN(C(C2(CC)CCN(C(=O)CCOC(C)=O)C2)=O)C1 c1(OC)cc(C)sc1C(=O)NC(C1CCN1C(=O)C(O)Cn1cncn1)C1CC1 c1(CCC)cc(N(CCC)CC2CCN(C(C3C4CCCC34)=O)CC2)nc(Cl)n1 c1(OC)cc(NCc2cccnc2O)c(OC)cc1Br c1(CC(=O)NCc2cn(CCNC(=O)COC3CCC3)nn2)csc(Cl)n1 Cc1oc(C(C)(C)C)cc1C(=O)N(CC(C)NC(C1(O)CC1)=O)C c1(CC(=O)NCCN(C(=O)Cn2nccn2)C2CC2)ccc(Cl)cc1Br c1(CNC(N(C)Cc2onc(CC)n2)=O)c(C)cccc1C CN1CC(O)CCC1C(=O)NCCC1(NC(=O)CNC(c2cccs2)=O)CC1 CN1CCC(CC(=O)NCC(C)(C)CN(C)C(c2cnc(C3CC3)s2)=O)C1 C1(S)CCS(=O)(=O)C1.C1(CC(=O)NCC#CCNC(=O)CC2CC2)CCCOC1 c1(CC(=O)Oc2ccc(C)cc2)ccccc1NC(N1CCC2CC12)=O c1(CC)cc(C(N2CCC(NC(=O)Cc3cscn3)C(C)C2)=O)ccc1C N1(C(CCNC(C)=O)=O)CCCCC(NC(C2CCC(=O)C2)=O)C1 C1(C(N(CCNC(c2cnsn2)=O)CC2CC2)=O)CC12CC(F)(F)C2 C(=O)(C(C)C(C)(C)C)NC1CN(C(c2nc(C)c(C)[nH]2)=O)CC1C c1(C(N2CCC(OCCNC(C(CCCOC)C)=O)C2)=O)cccc2c1CCC2=O c1(CCC(c2cncn2C)NCc2cccc(N(C)C)c2)c[nH]c2ccccc12 N1(C(C2C(C(=O)OCC)C2)=O)CCC2(CC2NC(C2(OC)CN(C)C2)=O)C1 N1(C(C(CC2CC2)NC(CCCC=C)=O)=O)CCC2(CCCOC2)C1 N1(C(C(C)NC(CNC(=O)NC)=O)=O)CCC(C)(OC)CC1 C1(C(N2C3CC(=C)C(C3)C2)=O)CCN(C(=O)CN(CC)CC)O1 C(=O)(C(F)C(C)CNC(c1cccnc1OC)=O)NC1(CCCC)CC1 C1(C(N2C(CNC(CCCN(C)N=O)=O)CC2)=O)CSC(c2ccccc2O)=N1 c1(NC(c2ccc(NC(C3CC(=C)C3)=O)cc2)C)ncnc(Cl)c1C(C)=O N1(CC(C)NC(=O)CC2CC(N(C)C)C2)CCN(C(C2CC(=O)N(C)C2)=O)CC1 c1(C(N(C(C#C)C)CCCC)=O)n[nH]c2c1CN(C(=O)CC1CCCC(=O)C1)C2 C12CCN(CC1)C(=O)OC(=O)C2.c1(CN(CC(F)F)CC)ccccn1 C(=O)(C1=CS(=O)(=O)CCC1)N1CCN(C(C(C)=CC)=O)C(C)C1C CCCCCCN1CCC(CC(=O)NC2CCC(C(N)=O)C2)C1 Cc1cc2cc(C(=O)NC3(CNC(=O)C(C)C4CCC4)CCOC3)oc2cc1C C1(C)(NC(CC2CCC(C)(C)O2)=O)CCN(CC2CC2)CC1 CCCCC(=O)NC(COC)C(=O)N(C1(C2CC2)CC1)C c1(C(N2CC(CCNC(=O)CN3CC4CC4C3)(OC)C2)=O)cc(C)sc1C N1(C(CNC(=O)OC)=O)CCC2(CC1)CC2NC(c1ccn(C2CC2)c1C)=O Cc1ccc(C)c(CSCC(N2CC3(C2)CN(C(=O)C(C)CF)C3)=O)c1 C#Cc1cc(CN2CCCC(C(=O)OC)CC2)c(N2CCC(CO)C2)cc1F N1(C(c2c(C)cc(C)nc2)=O)CCC2CCC(C1)N2C(c1cc(CO)ccn1)=O C1(C(N2CC(NC(C3(SC)CC3)=O)C(C)C2)=O)CS(=O)(=O)CCO1 C(=O)(C(C)CC(C)(F)F)N1CC(OCCNC(c2c(CC)n(CC)nn2)=O)C1 C1(C(N(C)CC2(CNC(=O)C=CBr)CC2)=O)CC(C2CC2)=NO1 N1(C(C(CN(C)C)N(C)C)=O)CCC(F)(CNC(=O)CC2CCC(C)(C)CO2)CC1 c1(-c2nc(CN3C(C(=O)OC)CCOCC3)on2)c[nH]c2nccc(Cl)c12 c1(CNC(CC2N(C(c3cn(CC)nc3)=O)CCC2)=O)ccccc1CO CCCCC(C)(F)C(=O)N1CCC(O)(CN(C)C(c2ccc(C#N)s2)=O)C1 CN1CC(CC(=O)NC(C)(C)CCNC(C2COCCO2)=O)c2ccccc21 C(N=c1[nH]c2cc(F)ccc2o1)C1(C)CCCN(C(c2ccc(C(C)C)s2)=O)C1 C(=O)(CC(C(F)F)NC(C1CCCSC1)=O)NCC1(C)C=CCCC1 C(CCCC(=O)NC1(CNC(C2C3CC(=O)CC23)=O)CCCC1)SC c1(C(=O)OC)cnc(Cn2cc(C(C)NC(C3CCC(CO)CC3)=O)nn2)n1C c1(Nc2ccc(C(=O)OC)c(C(C)C)c2)cc(Br)cc2[nH]ncc12 c1(COCC)cc(C(N2CCCC2CNC(C2CCOC2)=O)=O)on1 C12(C(=O)NCCCNC(=O)Cc3ccc(F)c(F)c3)CCCCC1CCC2 C=CCCCCCCCCC(=O)N1CCN(Cc2cc(O)ccc2Cl)C(C#N)C1 c1(C(N(CCCC(=O)NCC(F)C2CCC2)C)=O)cc(F)ccc1F C12CC=CCC1C(=O)N1CCC(CC1)CN(C)C2=O.C1(=O)C(C2CC2)N1.C=C.NC C123CCCC1N(CCC2)C(=O)CN(C(=O)OC)C3.C(C)(C)(C)OC(=O)NC1CC1 N1(C(C23CN(C(C(N4CCOCC4)C)=O)C(C2)CO3)=O)CCC2(CC(F)C2)C1 c1(C(C(=O)NC(C)C)N(CC)Cc2ccnn2C)cccc(C(C)C)c1 c1(CCCNC(C(=O)NCC(C(C)C)C(C)C)=O)nc2c([nH]1)CCCC2 C1(NC(CCCC=C)=O)COCCN(C(c2coc(C(N)=O)c2)=O)C1 Cn1cc(C#N)cc1C(N1CCC1CC(N1CC(Cc2ccoc2)C1)=O)=O CC1(C(=O)O)CCN(C(=O)NC(=O)CN2CCN(S(C)(=O)=O)CC2)CC1O N1(C(C(=O)NC)c2ccoc2)CCC(C(F)(F)F)C1C c1(COC)ncc(C(N2CCC(CNC(C3CC4(CC4)C3)=O)C2)=O)s1 C1(NC(c2cc(OC)no2)=O)COCCN1C(C1(c2sc(C)nc2C)CC1)=O C(C(=O)N1CC(O)CC1CNC(=O)C(F)(F)c1csc(=N)[nH]1)(C(C)C)OC C(=O)(C(C)(C)C(F)F)N1C(CCN(C(c2c(C)nc(CCC)o2)=O)C)CCCC1 C(=O)(CC1=CCCC1)N(C1CCN(C(C2CCC(OC)C2)=O)CC1)C c1(COC)ccc(C(N2CC(C(N)=O)(CNC(c3csc(C)c3)=O)C2)=O)o1 C1(C(N2CC(CC(C)NC(c3ccc(SC)s3)=O)C2)=O)CCOC(C)(C)C1 Cc1cccc(C(=O)NCC2CCCN(C(C3(O)CCOC3)=O)CC2)c1F C=C1CCC(C(N2CCC(OCCNC(CCn3c(C)ncc3)=O)C2)=O)CC1 C1(NC(c2c(CC)onc2)=O)CC(C2CCN(C(C3(C(C)C)COC3)=O)C2)C1 c1(Cc2onc(-c3c(C(=O)OCC)nn(C)c3)n2)nnc2n1CCCC2 c1(C(N(C)CC2N(C(C(n3ccc(C)n3)C)=O)CCC2)=O)cc(F)c(O)c(Cl)c1 C(=O)(CC1OCc2cc(Cl)ccc21)N1CCN(C(c2c(SC)nn(C)c2)=O)CC1 Cn1ccc2cc(NC(C3CCCN(S(=O)(=O)c4cccs4)C3)=O)cnc12 C(c1ccc(C)c(C)c1)=CC(=O)NCC=CCNC(C1CC=C(C)CC1)=O c1(CNC(C(N2CC3CCCC2C3)c2ccn(C)n2)=O)ccc(Cl)c(Cl)c1 c1(C(=O)NCCC(=C)CNC(=O)C(C)=C2CCC2)nn(C)c(Cl)c1Br CCCCCC(=O)N1CCCCC1C1(NC(=O)CCN2CCC(F)C2)CC1 N1(C(=O)NC(C(CC)(C)C)c2ccccc2)CCCN2C(=O)CCC12C C(=O)(C1=CC2CCC=CCCC12)NCCCNC(c1cc(C)c2c(c1)CCC2)=O C1(C)(NC(C2C(C)OCC2)=O)CCN(c2ccnc(C3CC3)n2)C1 C1(C)(CN(C(c2cc(OC)ns2)=O)C)CCCC1NC(c1cnc(Cl)n1C)=O C1(C(=O)NCC2CC(NC(=O)C(F)(F)C3CCCC3)C2)CN2CCCCC2CO1 C1(CNC(C(c2ccc(C)s2)C)=O)(NC(=O)CC2CC(C)(C)CO2)CC(F)(F)C1 Cc1coc(C)c1C(N1CCC(C)(NC(=O)CSc2nnnn2C2CCC2)C1)=O c1(C(N2CC=CC(NC(C)=O)C2)=O)cc2ccnn2cn1 C1(CNC(c2ncc(OC)nc2OC)=O)CC2(CO1)CN(C(=O)C=CCOC)C2 C1(C(N2CCN(C(C#C)C)CC2)=O)CN(C(C2CCSCC2)=O)CC12CCC2 c1(C(N2CCC(CCNC(c3ncn(C)c3)=O)C2)=O)ccc2cccc(O)c2c1 C1(OC)(CNC(=O)CC2CC(C)C2)CCN(C(C2CC(O)C2)=O)CC1 CCC(C)(CNC(c1cc(C)n(C)c1)=O)C(=O)NCC(c1ccncc1)O N1(C(C2C(CC)CCCC2)=O)CCN(C(=O)C(C)(C)OC(C)=O)CC2(CC2)C1 N1(C(c2ccc(OCC)cc2)=O)CCOC(C(=O)NCC(C)(O)CO)CC1 N1(C(CC(C(C)C)OCC)=O)CC2CCN(C(=O)C(F)(F)CO)CC2C1 CCC1=C(C(=O)N2CC3CCC(C2)C3NC(=O)CCC(C)N(C)C)CCCO1 CC1(C)C=CC(NC(=O)C(C)(C)C2CCCN2C(C2CCC(=O)C2)=O)CC1 c1(C2CC(CC(=O)N(CC(C)NC(c3nncn3C3CC3)=O)C)C2)ccccc1 C=CCCC(F)(F)C(=O)N1C2CCC(C2)C1CC(=O)N(CC(O)CF)C CC1CC(C(=O)NC2CC(OCC(=O)NCCc3cccc(F)n3)C2)=NO1 C=CC1(C(=O)NCC2OCCC2C(=O)NCCN(C)C2CC2)CCOCC1 C12CN(C3CC13)C2=O.c1(SCC(=O)Nc2ccc(-c3cc[nH]n3)s2)ccccn1 N1(C(c2cc(OCC)ncn2)=O)CC(NC(=O)OC(C)(C)C)CC2(CCC2)C1 C=CCCCCCCCCC(=O)NCCC(C)NC(C1CNC(=O)C1)=O N1(C(C=NOC)=O)CC2ON=C(CNC(c3ccc4nnc(C)c(C)c4c3)=O)C2C1 C=C=CC(C)C(=O)NCc1cccc(NC(=O)C(C)NC(N)=O)c1 c1(C(=O)NC2CC(NC(=O)C=Cc3cn[nH]c3)C2)ccc2nc[nH]c2c1 c1(C2(C(N3CC(N(C)C(C4CC5(CC5)C4)=O)C3)=O)CC2)ccnc(Cl)c1 c1(CSCCNC(=O)CCOCC(N2CC(CF)C2)=O)cccnc1 N(C)(C(=NCC1(OC)CCOC1)NC(c1ncn(C)n1)C)CCCCC=C Cc1cc(C(=O)NCC(C)NC(=O)CC2CCC=CCC2)c(C)n1NC(N)=O N1(C(C=CCCC)=O)CCN(C(=O)CCc2nc3ccccc3o2)C2CCCC12 c1(C(N(CC(=O)NCC(=O)NC(C)C)CC2CC2)=O)cn(CCO)nn1 c1(C(=O)NC2CC(NC(C3CCCNC3=O)=O)CC2O)csc2nccn12 c1(OC)ccc(C(=O)NCC2(O)CN(C(c3cn(C)cn3)=O)C2)cn1 C1(C(=O)OC)(C(=O)NCC2CC(NC(c3conc3C(F)(F)F)=O)C2)CCOCC1 C(CCCCCC(=O)NCCC1CN(C(C2C(C)(C)C2(C)C)=O)C1)SC N1(C(c2ncc(CC)s2)C(=O)NC2CCOCC2)CCC2(CCNC(=O)O2)CC1 c1nc(NC2(C3CC3)CC2)cc(N2CCCC(CC3CC3)C2)n1 C(=O)(CCC1=NNC(=O)CC1)NCCC(=O)NCCC(CCC)O C(c1ccc(O)cc1)=CC(=O)NC(C)(C)CCNC(=O)CCCC(F)F C(=O)(C(CC)C(C)(F)F)NC12C(CN(C(c3c(OCC)cccc3Cl)=O)C1)CC2 n1(CC)c(C(=O)NCC(C)C(=O)NC(c2ncco2)(C)C)cnc1O CC(CN(C)C)CCC(=O)NC1CCN(C(=O)Cc2cn(C)nn2)C12CC2 Cc1cc(=NCC2CCNC(=O)C2)[nH]c(=NCC2CCN(C(C)C)CC2)[nH]1 c1(C(=O)NC(CC)CNC=O)ccc(CN)cn1.c1(COC)cnoc1CC(C)C c1(C(N(C(=O)CCNC(=O)N(C)C(C)C)C(C)C)=O)cccc(S(C)(=O)=O)c1 c1(NC(C(CNC(C(C)N(CC)CC)=O)N(C)C)=O)cc(C)ncn1 C1(NC(C=CCC)=O)CCCC1CNC(=O)CNC(=O)OC(C)(C)C C(=O)(C(C)S(N)(=O)=O)N1CC2C(CNC(C3(CC(C)C)CCOC3)=O)C2C1 Cc1cc(C(N2CCC(NC(C3CCCN3N=O)=O)CC2C)=O)c(O)nn1 N1(C(CCNC(COC)=O)=O)CC2(CCC2C(=O)NCCN(C)OC)C1 CC1CCCCC1n1nc(C(F)F)nc1C1CC1C(F)F CC#CCCCC(=O)NCC1CC(NC(=O)C(CC)Oc2ccccc2F)C1 c1(OC(C(=O)N(CCCCN(C(C2C(C)C2)=O)C)C)C)ccc(F)cc1 N1(C(CCN(CC=C)C(C2CCCCN(C)C2=O)=O)=O)CC2CC1C(F)(F)C2 c1(C(C(N2CC(c3cn(C(CC)C)nn3)(C)C2)=O)F)ccc(Br)cc1 c1(C(=O)NCCC(C)NC(=O)C(CO)N(C)C)cccc(Br)c1Cl c1(-n2ccc(C)n2)cn(C)nc1NCC1(c2ccc(C(=O)O)cc2)CCOCC1 CCS(=O)(=O)c1ccccc1NNC(=O)c1cc2c(s1)CCOC2 c1(OC)c(C(=O)NC2CCN(C(c3onc(C)c3C)=O)C2(C)C)cc(F)cc1F C1(C(N2CCC(CNC(C(CC)NC(C)=O)=O)C2)=O)CC2(C1)CS(=O)(=O)C2 c1(OCC)cccc(CCC(N2CC(CNC(=O)Cn3cnnc3)C(C)C2)=O)c1 c1(NC(N(CC)CC2CCOC2)=O)ccc(C(=O)OC(C)(C)C)n1C C(=O)(C1CCCc2ncccc21)N1C(C)CC(CNC(C2CNC(=O)O2)=O)C1 C1(NC(CCC)=O)CN(C(=O)C=CCOCC(F)(F)F)C2(CCCCC2)C1 C1(CN(C(CC)C#N)C(=O)CCC)CCCC(C(=O)OC)C1 N1(C(CC2CC(C)(C)C2)=O)CCCCCC(NC(=O)C(O)CC(C)(C)C)C1 CCC(O)C(F)(F)C(=O)NC1CC=C(C(=O)NC(C)CCn2cncn2)C1 c1(SC(C(=O)N(CC(C)NC(CCOCC(C)C)=O)C)C)cccc(Cl)c1 Cc1ccncc1NC(=O)N(C1CCCCC1)CCCN(C)C.C(=O)N c1(C(N2CC(C)C(NC(c3nc(Cl)cs3)=O)CC2)=O)cccc2c1OCCCO2 C12(NC(C(CC)C(C)C)=O)CCC(CN(C(=O)C(F)(F)C(N)=O)C1)C2 C1(NC(CCc2ccc(C)s2)=O)CN(C(c2csc(C3CC3)n2)=O)CCC1(C)C N1(C(C(=O)NCC)=O)CCC2C(C1)CN2C(=O)Cc1cccc(OC(F)(F)F)c1 C1(CC(=O)NC2CC(n3cc(CNC(CCC=C)=O)nn3)C2)C(=O)NN=C1C C1(CNC(C2CC(C)(CC)C2)=O)CCN(C(=O)C(F)=CCCF)CC1 N1(C(c2c(CC)cco2)=O)CC(CNC(=O)CN2CC(C)(OC)C2)CCC1C N1(C(CC2ON=C(C)C2)=O)CC(CCNC(c2scc(C)c2Cl)=O)C(C)C1 c1(OS(CC2CC(C)OCC2)(=O)=O)ccc(OCC(F)(F)F)c(S(=O)(=O)N(C)C)c1 c1(C(N2C(CNC(CSCCOC)=O)CCC2)=O)nc(Cl)c(C(F)(F)F)[nH]1 Cc1c(N)ccc(C(=O)OCCCCC2CCN(C(=O)OC(C)(C)C)CC2)c1Cl CC(C)CS(=O)(=O)CC(=O)N1C(C)C2CC1C2NC(=O)CCc1cnoc1 Cc1coc(C(=O)NC2CC3(C2)CC3NC(c2cc(C)n(C(C)C)n2)=O)c1C N1(C(C2C3C4CCC(C4)C23)=O)CCC2(CCN(C(c3cc(Br)ccn3)=O)C2)C1 N1(C(CC#N)=O)CCN(C(c2csc(C(F)(F)F)n2)=O)C2CCCCC12 C1(CC(=O)NCCCN(CCCNC(CCC2CC(C)C2)=O)C)CCCC1O N1(C(c2nc(C)c(Br)cc2)=O)CCC(F)(F)C(NCc2cc(Br)c(O)c(Br)c2)C1 C1(NC(CSCCOC)=O)CCC(CNC(=O)CC23CCCC2C3)CC1 Cc1cc(C)n(CCC(=O)NCC2CC2CNC(=O)C(O)C2CC2)n1 c1(C2CC(C(=O)NC(CCNC(CCC=C)=O)(C)C)C2)ccc(OC)c(OC)c1 c1(OC)cc(C(=O)N(C)CC2CCN(C(=O)C3=CCSC3)CC2)cc2c1OCC2 Cc1nc(C(C)C)ccc1C(N1CC(C)CN(C(=O)COC2(C)CCCC2)C1)=O c1(C(COC)COC)nc(-c2ccc(SC)nc2)nn1Cc1ccc(C)cc1.CSC C(=O)(C(C)(C)CC(F)(F)F)N1CC(n2cc(CNC(c3occ(C)c3)=O)nn2)C1 N1(C(C2C(NC(c3cc4cccnn4c3)=O)COCC2)=O)CCN2CCCCC2C1 c1(C(N(CCCNC(C2CCCSC2)=O)C2CC2)=O)nccc2[nH]ccc12 C(N=c1nc2c(cnn2C)c(NCCn2ncnn2)[nH]1)c1[nH]nc(CC)n1 C(C(=O)OC)(C(C)CC1CCOCC1)N(CC(=O)NCCSC)CCC c1(C(N(CC(C)N(C(CCC#C)=O)C)C)=O)cc(C(F)(F)F)cnc1OCC C(=O)(CC1OCc2ncccc21)NC1(CCCNC(C2CC=C(C)CC2)=O)CC1 c1(NC2CCCNC2)cc(Cl)ccc1Cl.N12CCN(CC1)CCNC(=O)C2=O C(=O)(CC(F)(F)F)NC1C(NC(CCCc2ncc(C)o2)=O)C1 C1(C(N2C(CNC(c3cc(C)nn3C)=O)CC(F)C2)=O)CCN(C2CC2)S1(=O)=O C1(CC(=O)NCCN(C(CC2(C(=C)F)CCC2)=O)CCC)CCCC(C#N)C1 c1(CNC(C2(COC)CC2)=O)cc(C(=O)NC(c2ccns2)C)on1 N1(C(C=CC(CC)C)=O)CCC2(CC1)CN(C(=O)C(C(C)OC)N(C)C)CCO2 C(C(F)(F)C(=O)NCCCC(c1ccccc1)NC(C1(C)C=CCCC1)=O)OC C1(NC(N(C(C)(C)CCc2ccccc2)C)=O)COC2COCC12 CC(CC(=O)NCC1CN(C(c2cccc(C3CCOC3C)c2)=O)C1)C(F)F c1(NC(=O)C2CC2)ccn(CC(F)(F)F)n1.C12(CCC1)CC(=O)N2C C1(C(=O)NC2(CCNC(Cc3n(C)cnc3)=O)CCCC2)CC(F)C(=O)N1 c1(OCC(=O)NC2CC(N(C(c3c(COC)ccs3)=O)C)C2)c(F)cccc1F C1(CNC(C2CCC(=O)N2)=O)C2CN(C(c3cnnc(O)c3)=O)CC12 c1(CC(C(=O)C(C)(C)C)COC(=O)NCCNc2cccc(F)n2)ccc(F)cc1 C1(C(N2C(C)CCN(C(CCC(C)OCC)=O)CC2)=O)CCCC2(C1)CC2(F)F C(=O)(C(C)(O)C(F)(F)F)N1CCC(CN(C(=O)CC2CCCC(OC)C2)CC)CC1 C(=O)(C1=CCCN(C(=O)CCCN(C)C)C1)N1CCC(C(C)O)C1 N1(C(C(N2CCCCCC2)C)=O)CC2CN(C(=O)C(C)(C)c3ccnn3C)CCC12 C(=O)(C1CCCn2ccnc21)NC1CCC(NC(C(C(C)C)(C)O)=O)CC1 N1(C(c2c(C)n[nH]c2C)=O)CCC2(COC(CNC(c3nnn(C)n3)=O)C2)C1 C#CCC(C)(C(=O)NCc1ccsc1C)NC(=O)Cn1ncn(C)c1=O N1(C(CSCC(=O)NC)=O)CCN(C(=O)C(=O)NCCNc2nnc(C)s2)CC1 c1(OC)ccc(C(N2CCCC2C2(NC(C3CC3(F)F)=O)CC2)=O)cc1Cl N1(CC(=O)NCc2ccc(C(F)F)cc2)CCOC(CC2CC2)C1 O=[N+]([O-])c1cc(-c2ncccn2)ccc1NCC1CCNC12CC2 C1(NC(CC=C)=O)CCN(C(=O)C(C)(C)SC)CC1O c1(CSC)csc(COC(=O)Cc2ccn(C(C)C)n2)n1 C1(O)(C(CNC(C(=O)NCC)=O)C)CCN(C(=O)CCC2CCCC2)C1 C(CCCCC(=O)NCCC1COCCN1C(=O)C(O)C=CC)=CCC=C N1(C(Cc2c(C)nc(C3CC3)s2)=O)CCC2CN(C(=O)CCC(C)(C)C)CC2C1 CC1c2ccccc2OC1CC(N1CC(NC(=O)CCCF)C(O)C1)=O N1(C(C(CC)C)=O)CCCCC(CNC(c2ccc(C(=O)NC)nc2)=O)CC1 Cc1[nH]nc(C(=O)NCC2CC(NC(C3(n4cccn4)CCC3)=O)C2)c1F CC(CS(C)(=O)=O)C(=O)NCC1COCCN1C(=O)Cc1ccnc(O)c1 CCCCCC(O)C(=O)N1CCC2CN(C(=O)CN3C(=O)CCC3=O)CC12 C12(NC(C(=Cc3ccco3)C)=O)CCCC1N(C(=O)C(F)(F)CO)CC2 N1(C(c2ccc(OC(CC)C)cc2)=O)CCC(NC(=O)CSC(=N)N)C(F)C1 C#Cc1ccc(C(=O)NC2CCC2NC(c2cn(C)nc2C(C)C)=O)cc1C c1(OC)cccc2c(C(N3CCCC(C)(NC(=O)C=C(C)C)C3)=O)n[nH]c12 N1(C(CNC(=O)NC)=O)CCC(CCOC)(CO)C1.C(C)(CF)C=O Cc1ccc2c(=NCc3cc(C(C)C)no3)[nH]c(=NCC(C)C(C)C)[nH]c2c1 Cc1cc(Cl)c(C(=O)NC(C)CNC(c2cnsn2)=O)cc1C C(C(C)NC(c1cccn1C1CCCC1)=O)(C(C)C)NC(C=CC(CC)=CC)=O C=CCC(CC)C(=O)NCC1CC(NC(c2cncc(OCC)c2)=O)CCO1 C1(NC(CNC(C=C)=O)=O)CC2(C1)CC(CNC(=O)Cc1cccnc1)C2 C1(C(N(CC)CC2CCCC2)=O)CC12CCN(C(=O)Cc1cncnc1)C2 CCCC(CC)C(C(=O)NCc1cccs1)N(CCCC(CC)OC)C C1(CNC(C=NOC)=O)CCN(C(=O)CC2CCN(S(C)(=O)=O)CC2)C(C)C1 S(=O)(=O)(c1ccc(SCC(C2CC2(Br)Br)=O)cc1)NCC=C c1(C(N2CC3C(NC(C(C=CCCC)O)=O)C3C2)=O)ccc(O)c(Cl)c1 CC(C(=O)N1CC(C)(NC(=O)CCCNC(c2ccco2)=O)C1)C(F)F N1(C(C(CC)C)=O)CC(NC(=O)CNC(=O)C(c2cccnc2)O)C(C)C1 c1(C(N2CCC(CCOC)(NC(C3CC4(CC4)C3)=O)C2)=O)cc(Cl)ccc1C(C)C c1(C(N(C2CCC(NC(C3(SC)CCC3)=O)C2)C)=O)c(C)cnc2ccccc12 C1(C(N2CC(CC#C)OCC2)=O)CCC(C)N(c2nnco2)C1 CC1CCC(CC(=O)NC2(C)CN(C(=O)Cn3cc(C#N)cn3)C2)OC1 N1(C(C2OCC(C)NC2)=O)Cc2cccc(Cl)c2C1 C(=O)(C1=C(Cl)CCCC1)N1CCN(C(C(COCC)C)=O)CC1CC c1(C(=O)NC2CCN(C(C=Cc3c(C)ncs3)=O)C2C)cc2cccnc2[nH]1 c1(-c2nc(C(C)(C)C)nn2CCOc2ccc(Br)cc2F)cccc2ccncc12 C1(C)(CNC(CCn2ncc(C)c2)=O)CN(C(c2cnncc2O)=O)CC1C c1(C(=O)NC(C)CN)c(Cl)ccc(I)c1F Cc1cccc2oc(N3CCOC(C(C)NC(=O)C(C)S(C)(=O)=O)C3)nc12 C(C(=O)NCc1ccnc(N2CCOCC2)c1)(C(C)C)OCC C1(CNC(CCC#C)=O)(NC(C2CCC2C(=O)OC)=O)CC2CCC1CC2 CC1=C(C)CC(C(=O)NOCc2cn(CC3CC(=O)C34CCC4)nn2)CC1 N1(C(C(C)(CO)NC(C)=O)=O)CCC12CN(C(c1cccc(C(N)=O)c1C)=O)C2 C(=O)(C(F)(F)C(O)C(C)C)NC1C(NC(c2cc(CC)on2)=O)COCC1 N1(C(C(CCCC)O)=O)CCC2(NC(=O)CS(=O)(=O)CCC)CCCC12 C(C(C)(C)CCC#N)NCC(C)OC(C)C C1(C(N(CC(=O)N(C2CCC(CO)CC2)C)CC#C)=O)CC(O)C(F)C1 c1(NC2CCC(C(=O)NC(c3c(F)cncc3F)CC)OC2)c(C)ccnc1Br C(=O)(C(CCS(C)(=O)=O)N(C)C)N1CCC(C(C(=O)OC)NC)CC1 C1(CNC2(OCC#C)CCOCC2)CCCCN(C)C1=O C1(C(=O)NC2C(OC)CCC2)CN(C(c2[nH]ccc2C2CC2)=O)CCC1(C)C c1(C(=O)NCCCCN(C(C(COC)N(C)C)=O)C)ccc(P(C)(C)=O)nc1 N1(C(C2C(OC)COCC2)=O)CCC2(CCCC2NC(=O)C(C)(F)C(C)(C)F)CC1 c1(CNC(=O)CC2CC2CNC(=O)CC23CCCC2C3)ccnc(O)c1 C1(NC(CCOC)=O)C(C)(C)C(NC(=O)C=Cc2ccnn2CC)C1(C)C c1(OC)ncc(C(=O)NCC(C)CNC(C2CCOC2C)=O)nc1C N1(C(C2(OC)CC2)=O)CC2CC(C1)C(CO)C2NC(C1CCCCC(=O)N1)=O O=S(=O)(c1cnn2ccccc12)N1CCC2(CCCC(CO)O2)C1 C1(NC(C2CCC(N(C)C)CC2)=O)CCC(C(N2CC3CC3C2C#N)=O)OC1 N1(C(C(c2ccc(C)cc2)C)=O)CCN(C)CC1CNC(c1cccn1C)=O N1(c2cc(CC(C)C)ncn2)CCCC12CN(N1CCOC3(CCC3)C1)C2 c1(C(=O)NCCCCN(C(c2cn(CCC)nn2)=O)C)cccc(OC)n1 C1(NC(c2csc(C(F)F)n2)=O)C2COCC1CN(C(C1CC13CCCC3)=O)C2 c1(CNC(Cc2c(C)con2)=O)cnn(C)c1C(=O)NCC1CCCC12CC2 CC1(C)NC(=O)CC1C(=O)NC1CCOC1C(=O)NC1C(O)CC1O C1(CNC(c2sccc2F)=O)C2CN(C(c3cc(-c4ccccc4)co3)=O)CC12 CCCC(CC)C(=O)NC1CN(C(c2sccc2Cl)=O)CC1F Cc1oc2ccc(C(=O)NCC(C)(C)Cn3cc(CO)nn3)cc2c1C N1(C(C2CCN(CC)C2)=O)CCC(NC(c2cc(F)ccc2OC)=O)C(C)C1 CC(C(=O)NCCOCC(C)(C)NC(=O)Cc1cnccn1)C(C)S(C)(=O)=O Cc1cc(CNC(C23CC(C(=O)Nc4ccnn4C(C)C)(C2)C3)=O)c(F)cc1Br Cc1cc(C(N2CCCC3(NC(=O)CS(=O)(=O)N(C)C)CC3C2)=O)cc(=O)n1C CCCC(CNC(c1cccc(OC)c1)=O)C(=O)NCCN1CCCOCC1 Cc1cc(CC(=O)NCc2ccoc2C(=O)Nc2ccsc2)cs1 C(=O)(C(C)C(C)C)N(C1CCN(C(=O)C(O)CCN(C)C)C1)CC#C C=CCCC(C)(C)CNC(=O)C(O)C1CN(C(c2nc(C)c(C)s2)=O)C1 c1(C(=O)NC(CCNC(c2cc(C)nnc2)=O)C)cc(Cl)ccc1C(C)C CCC(C)(CO)C(=O)NC1CC(C)(NC(c2cnn(C3CCC3)n2)=O)C1 C1(CCOC)(C(=O)NC2CC(CNC(=O)CC3(COC)CCCC3)C2)CCCC1 C1(C(N2CCC(C(F)(F)F)C2)=O)Cc2ccccc2CN1Cc1cccc(Cl)c1 N1(C(CC(CC)C2CCC2)=O)CCC2(CC1)CC2NC(c1nsnc1O)=O Cn1nc(Br)c2ncnc(NC(C)(C)CNC(C3(C)CC4CCC3C4)=O)c12 Cc1ccc2nc(C(=O)NCC3CC(CC(F)F)C3)cn2c1.C1C(O)CC(=O)N1 C=CCC(C)C(=O)N(CCNC(C1CCCN1C(C)=O)=O)CCOCCO c1(NC(C23C(C)(C)OCC2C3)=O)cc(Br)cn(-c2ccc(F)cc2)c1=O C1(NC(c2ccc(C)s2)=O)C2CC3CN(C(c4cc(C)c(Cl)s4)=O)C1C3C2 c1(C(CNC(C=CSC)=O)O)cc(Cl)cc(Cl)c1 C1(CC(=O)NCCC2CCC(NC(C3SCCS3)=O)C2)CCS(=O)(=O)CC1 N1(CC)CCC(NC(=O)CCCNC(=O)CC2CCCSC2)CC1 CC(C)CCCC(C)NCC1CC2(C1)CC2(F)F N1(Cc2c(Cl)cnc(CC(=O)OC)n2)CCCc2[nH]ccc(=O)c21 C1(O)(CNC(C2(C)CCC2)=O)CCCN(C(c2ccccc2F)=O)C1 N1(C(COCCC)=O)CC(N(C)C(c2cc(F)ccc2Cl)=O)C(C)(C)C1 C(=O)(N=c1ccc(C#N)c[nH]1)Nc1nccc(C)c1.N12CC3C(C3C1)C2=O C(CC(=O)OC)(N=c1ccn(Cc2ccccc2)[nH]1)c1ccn(CC)n1 N1(C(C2(CCC)CCC2)=O)CCC2(CCCN2C(c2ncn3ccccc23)=O)C1 C1(C(N(CC(CO)(CO)NC(COCC(=O)NC)=O)C)=O)CCC(C)NC1=O C12(C(=O)NCc3c(C)ccnc3C)CCCC1N(C(=O)C(=O)NC1CC1)CC2 C12(CNC(c3cc(C)n(C)c3)=O)COCCN1CCN(C(=O)C=CC(F)(F)F)C2 N#Cc1c[nH]c(=NCc2c(F)ccc(Cl)c2F)c2c1NCCC2 c1(C(=O)NCCOCCN(C)Cc2cnc(C(C)(C)C)s2)ccc(Cl)cc1 Cc1ncc(C(=O)NC(C(=O)N2CC3C(C2)C3(C)C)C(C)(C)O)c(=N)[nH]1 N1(CC(=O)NCC2N(C(CCCN(C(=O)OCC)C)=O)CC2)CCOCC1=O N1(C(C2(NC(C3CCC4(CCC4)C3)=O)CCSC2)=O)CCC(F)C(F)C1 C1(CC=C)(NC(=O)CC2C=CCC2)CCCN(C(=O)CC=C(C)C)C1 c1(C(N2C(C(=O)OC)CC(CNCc3cc[nH]c3OC)C2)=O)cc(O)ccc1F C1(C(N2CCC(CNC(C(c3c(C)cccc3)(C)C)=O)C2)=O)CCC(C)(C)OC1 C(=O)(C1=C(Cl)CCCC1)NCC1N(C(CC(C)C(=O)c2cccc(F)c2)=O)CC1 N1(C(c2cnn(C)n2)=O)CCC(N2CCN(CC(=O)NC3CCC3)CC2)CC1 CC1CCC(C)(C(=O)NC2CC3CCC2N3C(C2CCCN2C)=O)CC1 C1(C(=O)NC(C2CCCO2)CC)CC=CCN1C(=O)CCC1CC1 CC1(C)CCCC(C(N2CCN(C(=O)CCc3cncc(O)c3)C3CC23)=O)O1 c1(CN2CCC(C(=O)NCCC(=O)Nc3ccccc3)C2)ccccc1[N+](=O)[O-] N1(C(C(C)OC)=O)CCN(C(c2ccc(C(F)(F)F)cc2I)=O)C(C#N)C1 N1(C(C(CC2CCCCC2)OC)=O)CCC(C)(NC(=O)CCc2cnoc2)C1 N1(C(C2CCCCN(C(C(c3cncnc3)C)=O)C2)=O)CC(C)c2ncccc21 C=CC1CN(C(=O)C(C)(C2CCC2)NC(c2ccc(C)c(C)c2)=O)CCO1 c1ccc(Br)cc1.c1(Sc2nnco2)cnn(CC2CCCC2)c1.C12(CC1)C(=O)N2 N1(CC(C)C)CCCC(CN(C(=O)COCC)C2CC2)C1.C1(=O)CN1 C12(C(=O)NC3CC(N(C)C(c4cccc(CCO)c4)=O)C3)CCCN(CC1)C2 [N-]=[N+]=NC1CCC(C(=O)NCC2(CCNC(C3CCCC(=O)N3)=O)CC2)CC1 C(c1cscn1)=CC(=O)NCC(C1CCOC1)NC(C1(COC)CC1)=O C1(=O)C(C)(C)CCNC2(CC2)C(=O)NCCCCN1.CCOC.OC c1(OC(C(=O)NCC(N(C(C2CC(=C)C2)=O)C)C2CC2)C)ccc(Cl)cc1Cl c1(C(=O)NC2CC(C)N(C(=O)Cn3cnc(=N)[nH]3)CC2)cc2cccnc2[nH]1 C1(NC(c2csc(O)n2)=O)CCCCC1CNC(C1(N2CCCC2)CCC1)=O c1(C(N2C(CCN(C)C(C3CCCO3)=O)CCCC2)=O)ccnc(Cl)c1N c1(C(=O)NC2(C)CC(NC(C3N(C)CCOC3)=O)C2)nc(O)nc(O)c1N N1(C(CNC(=O)NC)=O)CC(C2CCCN(C(C3CCC4(CCC4)C3)=O)C2)C1 C12CN(C(C)(C)C1)C(=O)CNC2=O.CCC(C)CC(=O)NC(=O)Cn1cncn1 C1(CNC(CN(C(C(C)C)=O)C)=O)CN(C(C2(C)CC2C)=O)CC12CCC2 C(=O)(CS(C)(=O)=O)N1C(C(C)(C)NC(=O)C=CC2CCCC2)CCC1 c1(C(N(CCNC(C(CC)COC)=O)C2CC2)=O)cccn2nnnc12 CN(C(=NCC1CC1)NCC(c1cn[nH]c1)(C)C)CC1CCCCC1 N1(C(C(C)OCC=C)=O)CCC2(CCN(C(=O)NC(=O)CCCCO)C2)C1 C#CC1CC2(CC(C(=O)NCCC3(O)CCCN(C(=O)C=CC(C)C)C3)C2)C1 N1(C(c2cc(OC)n[nH]2)=O)CCN(C(=O)CC2CCC(O)C2)C(CO)C1 CON1CCC(C(=O)NC2CCCC(N(C)C(C3CC(C)(F)C3)=O)C2)CC1 C(=O)(C(CCC(C)C)NC(=O)Cc1ccc(O)cc1)N(CC(C)C)C N1(C(c2nc(C(C)NC(C3(C)CC(=C)C3)=O)oc2)=O)CCC(F)(C(N)=O)C1 c1(C(C)Nc2cc(N(CCCSC)C)nc(C)n2)nnc2n1CCCC2 C1(N)C(=O)NCC12CCCO2.c1(CC(CC2CC2)N(CCC)C(C)=O)nnc(C)n1C c1(CC(=O)NCC(C)N(C(=O)C(F)F)C)ccoc1 C(N=c1[nH]c(=NC2CCSC2)c2[nH]ccc2[nH]1)c1cc(CC)c(C)cc1 c1(C(=O)NCCCN(C)C(C2CCO2)=O)cnc(N2CCCCC2)s1 N1(C(c2c(C)cc[nH]2)=O)CCC2(CC(NC(=O)Cc3ccc(F)c(Cl)c3)CO2)C1 Cc1cc(O)c(C(=O)Oc2cccc(-c3cc[nH]n3)c2)cc1Br Cc1cc(CNc2cccc(OCC3CCOCC3)c2)cnc1Cl.OC(O)C c1(OC)ccc(S(=O)(=O)N2CC3CCCN(C(C)C)C3C2)cc1NC(=O)COC C12(NC(CSC(C)(C)C)=O)CCCN(C(=O)Cc3nccs3)CC1C2 c1(CNC2CC(C(N3CCC(O)C(O)C3)=O)C2)cc(F)c(F)cc1Cl N1(C(C2C3(CC(NC(C(C(C)(C)O)F)=O)C3)C2)=O)Cc2cccc(C#N)c2C1 N1(C(C(C)CNC(=O)CCc2ccco2)=O)CC2CCCC(O)C2C1 c1(OC)ccnc(C(c2nnnn2C2CCCC2)NCc2ccc(Br)cc2)c1C c1(C(=O)OC)c[nH]c2ncc(-c3cncc(-c4ncc(C#N)cc4O)c3)cc12 CC(C)CC(C)C(=O)N1CCCC1CN(C)C(c1cnnc(C)c1)=O C1(C(=O)NC2CN(C(c3ccc(C(N)=O)[nH]3)=O)C2)CCCN(c2ncccn2)C1 C1(NC(c2cncc(OC(C)C)c2)=O)CC(N=c2nc3[nH][nH]cc-3c(O)n2)C1 O=C(OC1CCCC1)C(F)(F)CCNC(=O)Cc1cncs1 CCC(F)(F)CC(=O)NCC(CC)(CC)NC(=O)CCOc1ccc(OC)cc1 Cc1cc(=NC(C)CC#N)[nH]c(N2CCN(C(c3nccs3)C)CC2)n1 Cc1c[nH]cc(Br)c1=NC(=O)C1CC1NC(c1cc(S(C)(=O)=O)ccc1O)=O Cc1noc(C)c1CCC(N1CCOC(c2cn(-c3ncccc3O)nn2)C1)=O C(=O)(C1=NNC(=O)CC1)N1CC(CC)C(NC(c2ccc(C)c(Cl)c2N)=O)CC1 C1(C)(OC)CCCN(C(c2cccc(C)n2)C(=O)NCC(C)C)C1 C1(C(=O)NC2CC(CNC(c3c(C)coc3)=O)C2)CC(C)CCC1C(C)C Cc1c(F)ccc(Br)c1C(=O)NC1CC2CCC(C1)N2C(C1CCCCC1)=O C1(C(=O)NC(CN(C(C=C(C)C(C)(C)C)=O)C)C)CCS(=O)(=O)C(C)C1 C(=O)(N=S(C)(=O)CC1CC(=O)N(C)C1=O)NC(c1ccccc1Cl)C C(=O)(C(CNC(c1ccc(O)c(F)c1)=O)CC(C)C)NC(C=C)C(F)(F)F C1(NC(CC2CCN(C(c3scc(COC)c3)=O)C2)=O)CC(CO)C1(C)C c1(C(N2CCC(NC(C(C)CO)=O)C2c2ccccc2)=O)nc2cnccc2s1 Cc1onc(C(N2CCCCC2C(C)NC(=O)Cc2cnn(C)c2)=O)c1Br Cc1cc(C#N)nc(N2CCN(CCCCCNC(=O)Cc3cnns3)CC2)n1 N1(C(CS(C)(=O)=O)=O)CCC2(CCN(S(=O)(=O)c3ccc(F)cc3)CC2)C1 c1(NC(c2ccc(-c3cnn(C4CC4)c3)nc2F)=O)cc(F)ccc1C(F)(F)F CCCCC(CCC)NC(=O)CCC(C)NC(C1(COC(C)C)CC1)=O C(=O)(C1=CCCOC1)NCC=C1CCN(C(C(CN(C)C)N(C)C)=O)CC1 Cc1[nH]c2ncccc2c1C(=O)NCC(C)NC(C1CCCN1C(N)=O)=O Cn1ccc2cccc(C(N3CCC(F)(CNC(C4CCC(F)(F)C4)=O)C3)=O)c12 C1(C(=O)NCc2ccco2)CC12CCN(C(=O)Cc1cccnc1F)CC2 c1(C(=O)NC(C)C(=O)NC2C(CNC(CC)=O)C2)ccnc(C(F)(F)F)c1 N1(C(Cc2c(C)nc(SCC)s2)=O)CC2CCC(C(N3CCC(OC)C3)=O)(C2)C1 C=C=CCC(=O)N1CC(O)(C2CCCN2C(c2cnn(CCOCC)c2)=O)C1 C12(C(=O)NCC3N(C(C4C(CC)OCC4)=O)CCOC3)CC1COC2(C)C C1(CNC(c2cnc(C)[nH]2)=O)CN(C)CCN1C(c1n[nH]c(C2CC2)c1Cl)=O C(c1cccc(C#N)c1)=CC(=O)NC1(C)CN(C(=O)CCN2CCNC(=O)C2)C1 c1(C(=O)NCC2(CC)CC2)ccc(F)c(S(=O)(=O)NC=O)c1.C1(N)CCC(O)CC1 N1(C(c2cc(C)no2)=O)CCC(NC(=O)Cn2ncc(Br)n2)C12CC2 c1(C(=O)NCC2CN(C(c3ccc(C#C)cc3)=O)C(C)C2)cncc2n[nH]cc12 Cc1nn(C)c(C)c1-c1cc(C(N2CCCC2CC(c2ccncc2)O)=O)n[nH]1 C1(C(N(C(C)C)C)=O)C2CCCC2CN1C(C1CC1(C)C(F)F)=O C1(CC)C2CCCN1C(=O)C1(CC1)CNC2=O.C1(C(N)=O)C=CCCC1 C1(CC(N2CC(OCCNC(C3COC(=O)O3)=O)C2)=O)COCCOC1 N1(C(C2CC(SC)C2)=O)CCC(CNC(=O)Cc2ccc(Br)nc2)C(O)C1 C1(OC)CN(C(=O)C(n2cc(C)cn2)C)CC1NC(c1cc(C2CC2)nn1C)=O CCC(C)C(=O)C(=O)N(C)CCOCCNC(=O)C(COC(C)C)C1CC1 c1(C(C)C)ncc(C(=O)N(C)CC2(CNC(C3(C#N)CC3C)=O)CC2)[nH]1 Cc1cc(C)c(C(N2CC(NC(c3n[nH]c4c3CSCC4)=O)C(F)C2)=O)cc1C Cc1cc(C)n(CC(=O)NCCC(O)CNC(=O)C(C)(C)c2ccc(Cl)s2)n1 c1(C(N(CC(C)NC(=O)C(C)Oc2cccc(F)n2)CC)=O)ccn2c1CCC2 CC(C)CC(CN1CCCC1)NC(=O)C(n1cc(CN(C)C2CC2)nn1)C Cc1nc2cc(C(N3CC4(CCCC4NC(=O)CN4CCOCC4)C3)=O)ccc2s1 C1(NC(c2n(CCC)ccc2)=O)CCCC(NC(c2cccn2CCC)=O)C1 C1(NC(C(CC(=C)C)C)=O)CCCC12CN(C(C1CN3CCCN1CC3)=O)C2 c1(C(=O)NC2CC(C)N(C(=O)CC3CC(F)C3)C2)cnc2c(c1)CCCO2 Cc1nc(N(C(C)CCNC(=O)CCc2ccnn2C)C)[nH]c(=N)n1 C(=O)(C1Cc2ccc(Cl)cc21)N(C)CC1CCN(C(=O)Cc2csc(NC=O)n2)C1 N1(CCC(CCC)C)CCC2(CC1)CC2NC(=O)C(C)N(C1CC1)CC c1(Cc2ccc(C(=O)NCCc3nn[nH]n3)s2)ccncn1 Cc1cnn(C(C)C(=O)NC(C)CC(=O)N(C)C(C)C2CC2)c1 c1(NC(=O)NC2(C)CCCC2O)cc(C2(C(=O)OC(C)(C)C)CC2)cc(O)c1 c1(C(N2CCN(C(c3c(OC)nccc3)=O)C(C)C2)=O)[nH]nc2ncnc(O)c12 C1(C(N(CCCCCCNC(c2csc(CO)n2)=O)C)=O)CN2CCC1CC2 [N-]=[N+]=NC1(C(N2CCC(N3CCCC3)C2)=O)CCN(C(C2CCCC3(CC3)C2)=O)C1 N1(C(COC)=O)CCC(NC(=O)CC2(C#N)CC2)C(CO)C1 c1(C(N(c2ccc(I)cc2)C)=O)cc(S(=O)(=O)N2CC(C)(C#N)C2)ccc1F C(=O)(C1=C(Cl)CCC1)NCC1OCCN(C(C2C(c3c(C)cccc3)C2)=O)C1 C1(C(=O)NC(c2c(C)cc(Br)cn2)C)C2CCCC(F)(F)C12 N1(C(C(C)(C)OCCC)=O)CCCC(NC(c2cnoc2C)=O)CC1 CCCC(CC)CC(=O)NCC1(C)CN(C(c2ccccc2C#N)=O)CCO1 C12(C(=O)NCCCC3CCC(=O)C3)CC1CN(C(=O)CCC1CCCCO1)C2 C1(CCNC(=O)CCC2CCOC2)CCCN(C(C2SCCS2)=O)CC1 CCC(CO)C(=O)NC(C)CC1CCCN(C(=O)COCCCOC)C1 c1(NC(c2n(CCCSCC)nnn2)c2cn(C)cn2)cccc(CCF)c1 C1(C(=O)NCc2ncc[nH]2)CC2(CCC2)CN1C(C12CCCC1C2(F)F)=O C1(NC(c2n(CC)nnc2C)=O)CN(C(c2cnc3n2CCC3)=O)CC1C1CC1 c1(CNC(C2C(=C)C2)=O)csc(C(=O)NC2CCNC2=O)c1 C1(F)(C(=O)NC(C=C)C2CCC2)CN(C(c2ccn(C3CCCC3)n2)=O)C1 O=C(C1=CC2(CN(C(=O)C(F)C(F)(F)F)C2)OC1)NCCCc1nccs1 CC(CC(C)C(F)F)NC(=O)C(C)(C)CNC(c1ccc(CC#N)cc1)=O N1(C(COCCC=C)=O)CCCC(N(C(=O)C(C)(C)Sc2ccoc2)C)CC1 C(=O)(CN=S(C)(C)=O)N(C(C)C)CCN(C)C(c1ncsc1C(F)(F)F)=O c1(NC(C2CCC(NC(C3N(C)CCC3)=O)C2)=O)cncc(Cl)c1 c1(C(=O)NCCCCCNC(CC2C(C)CCC2)=O)ccc(O)cc1F c1(Nc2nc(C)cc(NCC3C(C(=O)OCC)C3)n2)c(Br)ccc2ncccc12 C(=O)(CC(O)CCC)NC1CC(NC(CNC(CCCCC)=O)=O)CC1O C12(C(=O)OC)CCCCC1N(C(C1(C)CCOC1C)=O)CCC2 Cc1nc(C)c(C(=O)NCC23CC(CO2)N(C(C2CCCSS2)=O)C3)nc1C CC1=C(C(=O)NCC2CCC(C)CN2C(=O)CCCCN2CCCC2)COCC1 CC(CC(F)F)C(=O)NCC1CN(C(c2cnc(-c3cnccn3)s2)=O)CCO1 C1(NC(C(c2ccc(Cl)s2)C)=O)CC2(C1)CC(NC(C1CC3C=CC1CC3)=O)C2 C1(C(=O)NCC2N(C(c3c(F)ncc(C)c3)=O)CCC2)CC2(C1)CC21CCCC1 O=C(C1=CCCN(C(=O)C=C2CCOCC2)C1)N1CCC2C(O)CC12 C=Cn1nncc1C(=O)NCC(c1cccc(C)c1)NC(=O)C=C(CC)CC.C1(C)CC1 Cc1cc(Cl)cc(N)c1C(=O)NCC1CCN(C(=O)CCc2cncnc2)CC1 N1(C(c2c(C)noc2C)=O)CCOC2(CCN(C(c3cc[nH]c3C)=O)C2)C1 C(=O)(C1=CCC(C)(C)CC1)N1CC(N(C(c2occ(C)c2)=O)C)C(O)C1 C1(CNC(=O)C(=O)NC2(c3ccccc3)CCCO2)CC(O)C12CCC2 N1(C(c2c(C)n(C(F)(F)F)nc2)=O)CCSC(C)CC1 Cc1ccc(COC(C)C(N2CC(NC(C3CC(N(C)C)C3)=O)C(F)C2)=O)cc1 C(=O)(CC1=NNC(=O)C1)NCCN(C(c1cncc(C)c1Cl)=O)C1CC1 CCCC(CNC(=O)CCCCCN(C)C)C(=O)NC(C)CCO C1(C(=O)NCCCC)CC=CCN1C(=O)C(C)c1cc[nH]n1 CP(C)(=O)c1ccc(CN=c2ccnc(NCC3(CCO)CCOC3)[nH]2)cc1 c1(C(=O)NC(CC(C)NC(=O)C=CSc2nc[nH]n2)C)cnn2c1NCCC2 N1(C(c2c(C)nn(C3CCOC3)c2)=O)CC(NC(c2scnc2Cl)=O)C(C)(C)C1 C(=O)(CC(C(F)F)NC(c1cnn(C)c(=O)c1)=O)NC(c1cncs1)C c1(C(=O)NC2(C)CC(NC(c3c(Cl)cn(CCC)n3)=O)C2)[nH]cc2c1CCC2 c1(OC)c(NC(C2CCCC2NC(C23CC(F)(C2)C3)=O)=O)cccc1F c1(C(N2CCC(C)(NC(C3C(C)C3)=O)C2)=O)ccnc2ncccc12 C1(NC(=O)CCC2CC(F)(F)C2)CCCCC12CCN(C(=O)C(F)C1CCC1)C2 c1(C(=O)NC2CCN(C(C(c3ccccn3)N)=O)CC2O)ccc2nonc2c1 Cc1cc2c(CC(=O)NCC3CC3NC(c3c[nH]c4ccccc34)=O)csc2s1 Cc1ccc(C(C)NC(=O)NCC2(c3c(C)cccc3C)CC2)c(Br)c1 C1(CC(=O)N(CCC(C)NC(COCCC#C)=O)C)CCC(=O)N1 c1(C(N(C2CC3CN(C(C(C)OC)=O)C2C3)C)=O)c[nH]c2cccc(F)c12 CC1CCC(C(=O)NCCCN(C(=O)C(=O)Nc2ccccc2)C(C)C)C1 C(C)(CC(C)(C)OC)NC(CCOCCN)=O.N1(C(C)=O)CC(C(=O)N(C)C)C1 N1(Cc2cc(C(C)(F)F)on2)CCC(=O)N(CC(C)(O)c2cccs2)C1=O CC1(C)CCC=C1C(=O)N1CC(NC(c2ncccc2Br)=O)C(O)C1 C1(CC(=O)NCC2C(CNC(c3nc(C)sc3)=O)C2)(OC(C)C)CCCSC1 C#CC1CCCN(C(=O)C(CNC(=O)C(CC2CC2)OC)OC)C1 c1(OC)cc(OC)cc(CCC(N2CCCC2CNC(C2CN(C(N)=O)C2)=O)=O)c1 c1(C(NOCCC)=O)cc(Oc2ccccc2)c2c(c1)CCCO2 N12CC(C3(CC3)C1)CC2=O.CC(C(=O)N(C1CCSC1)C1CC1)=CC(C)(C)C CC(Cn1cccn1)C(=O)NC1C=CC(CC(=O)NCCC(F)(F)Cl)C1 N1(C(C=CCC)=O)CCC(C)(CC(=O)NCC2=NOCC2)C1 C=C=C(C)CC(=O)N1CC(NC(c2nccnc2C(=O)OC)=O)C(C)C1 C1(CNC(c2onc(C)n2)=O)CCCCC1NC(c1cc(C)ncn1)=O N1(C(C2(COC)CCOC2)=O)CCN(C(=O)Cc2ccns2)CC12CCC2 CCCCCCCCOCC(=O)NC1CCN(C(C2COC(=O)C2)=O)C1(C)C c1(C(N(CC(C)(C)CNC(=O)C=C2CCC2)C)=O)cc(Cl)ccc1-n1cccc1 C(C)(C(C(=O)NC1CCC(F)CC1)C(C)C)NC(c1c(O)ccc(C)c1)=O c1(C(=O)NCC(CNC(C(C)(C)C(F)(F)F)=O)F)ccc2c(c1)NC(=O)CN2 c1(C(=O)NC2CCCC(NC(C3N(C)CC3)=O)C2)nccc2c1[nH]c1ccccc21 N1(CCC(=O)N(CC(CC)NC(c2ncc(F)cn2)=O)C)CCCC(N(C)C)C1 Cc1nc(O)[nH]c1C(=O)NC1(CO)CCN(C(=O)C(C)(C)C2CCCCO2)C1 CC1(C)C(CO)CN1C(=O)C(CC1CC1)NC(=O)Cc1cn[nH]c1 c1(OCC)ccc(C(C)OC)nc1C.N12CCC=CC1CNC2=O N1(C(C(C)OCC#C)=O)CCN(C2CCN(C(C3(CC#C)COC3)=O)CC2)CC1 C1(Cn2cccn2)COc2cscc2O1.Cc1cccc(C(=O)OCC)c1C C1(C(=O)NCCCNC(CSCCCC)=O)CCc2n[nH]cc2C1C CCCCC(C)(F)C(=O)NC(CNC(C12CCC(CC1)C(C)O2)=O)C(C)C N1(C(c2c(C)nco2)=O)CCC(CNC(C2CC3OC2C2CC32)=O)C(O)C1 C12(NC(C3C(OC)CC3)=O)COC(CNC(=O)CCn3cccnc3=O)(C1)C2 c1(C(=O)NC)cc(N(CCO)CCc2cnc(C)s2)ccc1F C(=O)(C(F)C(F)(F)F)NCC1(C(N2CC3(C(C(=O)OC)C3)C2)=O)CCCC1O c1(NC(C(C)OC)=O)ccc(NC(=O)CC2CC=CCC2)cc1C Cc1nn(CCNC(=O)NC2(C(=O)N(C)C)CCCSC2)c(C)c1I Cc1cnc(Br)c(NC(C2CC23CN(Cc2cncc(Cl)c2)C3)=O)c1 n1(CC)nc(C(=O)NC(C)CNC(c2nn[nH]c2Cl)=O)c(C)n1 CCCCCC(F)C(=O)N1CCC(C=CC(N2CC(C)(C)CC2C)=O)CC1 C(=O)(C(C)(C)CO)NCCOCCN.C1CCC(=O)N1C(C)C.CC=O c1(C(N(C(c2ccccc2)CNC(C23CC(C)C2C3)=O)C)=O)ccc2c(n1)CCC2 N1(CCNC(CCN(C(C)C)C(C2CCSC(C)C2)=O)=O)C(=O)CCC1=O N1(C(C2(COC)COC2)=O)CC2CCC2(CC(=O)N(C2CCOCC2)C)C1 O(NC(=O)C(C(C)C)C(C)C)CC(N1C(CCc2nc(C)on2)CC1C)=O C1(C(N2CC(N(C(=O)COC3CCC(F)(F)CC3)C)C2)=O)COCC2(CCC2)O1 N1(C(C)=O)C(=O)CCC1C(=O)N(C)CCN(C)C(C1(C)CC(C)C1)=O N1(C(N(CC(F)(F)F)C)=O)CCC(N(C2CCCSC2)C)CC1 C(C)(C)(CCCCC(=O)N1CCC2CN(C(c3cccnn3)=O)CCC12)OC N1(C(c2c(C#N)scc2)=O)CCC2(C(N3CCC(n4ccnc4)C3)=O)CCCC12 C1(C(C2CCC2)=O)CC2CC(C1)N(C(=O)C(CC(N)=O)OC)C2.C(=O)N C=CC(C)(C)CCN=C(NCCC1CCCN1C)N1CCC(CC(N)=O)C1 N1(C(COC)=O)CC2CC(C1)N(C(C1COCC(=O)N1C(C)C)=O)C2 N1(C(c2ccc(C)cc2C)=O)CCC2(CC(NC(=O)CNS(N)(=O)=O)CO2)C1 N1(C(C(=O)NC2CCOC2)=O)CCC(F)(c2cccnc2)CC1 C(C(C)(COC)CO)NC(C(CC)NC(C)=O)=O.C(CC=O)=C(C)C c1(N2CC(CCN(C(C)(C)C)C3CC3)C2)nnc([N+](=O)[O-])n1C.C(=O)O C(=O)(C1=NNC(C(F)(F)F)C1)N1CC(C(C)NC(C2CC(Cl)(Cl)C2)=O)C1 c1(C(N2CC(C3CN(C(C4C(C)=C4)=O)C3)C2)=O)cc(C)n(NC(N)=O)c1C c1(SC)nc(NCC2CCCN2C(=O)CCc2cccc(Cl)c2)cc(C(F)F)n1 c1(C(N(CC(C)N(C)C(c2n[nH]cc2Cl)=O)C)=O)cc(F)cc2nc[nH]c12 n1(CC=C)c(N2CCC(OCC3CCC3)CC2)nnc1-c1c(C)noc1C C1(C(=O)OC)C(=O)N(C)CCN1C(=O)C(N1CCN(CC(=O)NC2CC2)CC1)=O c1(CC(=O)NCC(CCCC)NC(c2csnn2)=O)c(F)cncc1Cl C(=O)(C(C(C)N)c1ccccc1)NC(CSC)Cc1ccccc1 C(=O)(C1=CS(=O)CCC1)NCCCC(C)NC(=O)Cc1cn2ccccc2n1 Cc1cc(F)cnc1C(=O)NC1CC(CC(=O)Nc2ccc(Cl)c(C)c2)C1(C)C CC(C)(CC(F)(F)F)C(=O)NCC1(C)CC(F)(F)CN1C(=O)CSCC1CCCO1 N1(C(CC(C)C(F)(F)F)=O)CCC2(CCN(C(C3COC(=O)C3)=O)C2)C1 C1(CCC(=O)NCCCCNC(=O)CCOC2CCCC2)CCCCO1.C(CC)N c1(C(=O)NCCNC(C2N(CCC)C(=O)CCC2)=O)cccc2c1CC(=O)N2 c1(CC(=O)NC(C(=O)NC(CC)CN(C(=O)CC2(O)CC2)C)C)ccccc1 N1(CCCNC(c2cc(C)[nH]n2)=O)CCN(C(=O)CC23CCCC2C3)CC1 C1(C(=O)NCC2(C)CCC(=O)N2)CCN(C(c2ccc(F)c(O)c2)=O)CCO1 N1(C(C2N(C)CCCC2)=O)CC(C(N2CCCC(N3CCC3)C2)=O)CCC1(C)C c1(C(=O)OC)cc(C(N2CC3CC3(CNC(C3CC(O)C3)=O)C2)=O)ccc1C C1(NC(c2cc(CC)nnc2C)=O)CCCCCN(C(=O)Cc2c[nH]nc2O)C1 N1(C(C2CC(CC)C2)=O)CCC(F)C(NC(c2cnn(CCOCC)c2C)=O)C1 C(=O)(C1CCCc2nccn21)NCCCCn1cc(-c2c(C#N)nccc2)nn1 C(=O)(CCCCN=[N+]=[N-])NC1CCN(CC(=O)NCc2c(OCC)cncc2)C1 Nc1c(C(=O)NCCN(C(C2C3CCCCCC23)=O)CC2CC2)nc(O)nc1O c1(CC)cnccc1C(=O)N(C)CC1CCCN1C(C1CC=CCC1)=O CC(Cc1cnc[nH]1)C(=O)NCC=CCNC(c1cc(Cn2cccn2)on1)=O c1(NC(C2CN(C(c3cnccc3Cl)=O)CCN2)=O)nc(Cl)ccc1F S(=O)(=O)(c1cc([N+](=O)[O-])ccc1Cl)Nc1ccc(OC(C)C)cc1Cl C#CCCN=C(NCC(CC(C)C)C(F)(F)F)N1CCN(CCOC)C(=O)C1 N1(C(C2(C)CN(C(c3nc(CC)oc3C)=O)C2)=O)CC2CCC=CC12 N1(C(C=CC=CCC)=O)CC2CC1CN2C(=O)CN(C)C(c1cccs1)=O N1(C(C(CCCC)(C)F)=O)CCCC2(CCN(C(c3nc(C)ccc3F)=O)C2)C1 N#CC1(C(=O)NNC(=O)NCCCC2CC2)CC2CC2C1 C1CCC2(CC2)C1.n1(CNC(CCNC(=O)NCCO)=O)cc(SC)nn1 N1(C(COC(C)C)=O)CCC(=O)NC2CN(C(=O)C(C)(C)C(F)F)CCC12 c1(C(=O)NC2(CC=C)CCCC2)ccccc1OC(C)(C)C.C1(=O)C(C)O1 CC1C(C)N(C(=O)C=CC2CCN(C(=O)C=C3CCOCC3)CC2)CCN1C c1(CN2C(C(=O)Nc3cnnc(Cl)c3)CC3CC32)cccc(F)c1F C1(C(=O)NCCc2onc(C)n2)C(C2CC2)CCN1C(c1c[nH]c(=O)cn1)=O CC(C)(CCNC(=O)C(C)(C)F)NC(C1CC1C(=O)OC(C)(C)C)=O N1(C(c2c(CCC)n[nH]c2)=O)CCCC12CCN(C(c1cnc(C)cc1C)=O)C2 C(=O)(C(CC(C)C)ONC(C1(C)CC(=O)N(C)C1)=O)N(CCC1CC1)CC C12(CNC(C(C)(C)OC)=O)CCCCC1N(C(=O)CSCc1cccs1)CC2 C1(SCC(=O)NCCCN2CCN(C(CS(CC)=O)=O)CC2)CCOC(C)(C)C1 Cc1ccc(OC(C2C(C(=O)NCC3(CNC(=O)CN)CCC3)C2)=O)cc1F CCC(C)C(N)C(=O)N1CCN(Cc2ccc(NC)cc2)C(c2ccccc2)C1 Cc1nn(C)c(N2CCOCC2)c1NC(=O)NCC1COC(C)C1 C1(C(=O)NC(C(=O)NCC2OCCN(C)C2)C2(C)CC2)CC(=O)OC1(C)C C12(CCCC1)CC(=O)N2.C(=O)(C(C1CCCO1)C1CC1)NCC1(NC(C)=O)CC1 CC(CS(C)(=O)=O)C(=O)NCC1CCCN(C(c2cc(-c3ccco3)no2)=O)C1 C=CCC(CC)C(=O)NCC1(F)CN(C(C2CCCN2C)=O)C1 N1(C(C)=O)CCN(CCC2CSCCN2C(=O)OC(C)(C)C)CC1 c1(C(N2C3(CN(C(Cn4cc(C(C)=O)nn4)=O)C3)CC2)=O)cc2c([nH]1)CCOC2 c1(OCCC(=O)NC2CCC(CNC(CCCOC)=O)C2)ccc(F)c(F)c1 C(C(=O)C1CCc2ccccc21)OC(C(n1cc(-c2c(C)cccc2)nn1)C)=O N1(C(C(c2cccc(C(F)(F)F)c2)C)=O)CC(NC(=O)CNC(N)=O)C(C)(C)C1 C1(c2n(CC)nnn2)(NCCOc2ccc(Cl)cc2C)CCCC(C(C)C)CC1 N1(C(C2C(C(=O)OC)C2)=O)C2COCC1CC(NC(C1(n3ccnn3)CC1)=O)C2 C(C)(C(CC(=O)NCC1C=CCC1)NC(c1ccc(C)c(C)n1)=O)OC c1(SC)cscc1CC(=O)NC(CN(C)C)CC Cc1cc(=NCCc2c[nH]c(=N)s2)[nH]c(N2CCCC(C(F)F)C2)n1 c1(OCC)ccc(CN2CC3CN(C(=O)CCSC)CC23)cc1C C1(NC(C2CC(C(F)(F)F)(OC)C2)=O)CN(C(=O)CCCC2CCC2)CC2CC12 N1(C(C(CSC)(C)C)=O)CCC(C2CC2)(NC(=O)CCc2ccc(C)cc2)C1 CN1CC2(CCN(C(COc3ccccc3C(F)(F)F)=O)CC2)OCC1=O CC(CSCc1cccnc1)C(=O)NCC#CCN(C(=O)COC(F)F)C1CC1 Cc1ccnc(C(=O)N(C(C)C(=O)NC2CC=CCC2C)C2CC2)c1F CCS(=O)(=O)CC(=O)N1CCC(C(C)NC(=O)CCCCO)C1 c1(CN(C)C(=O)Nc2csc(Cl)c2Cl)ccc2cccnc2n1 CCCCC(C)CCC(=O)N1CC2CC(C(=O)Nc3cscc3C)C(C2)C1 C1(C)(C(=O)NCCC2CCN(C(CCN3CCC(C)CC3)=O)C2)CCCN(C)C1 CN1C(=O)C(F)CC1C(=O)NCC1CC(NC(=O)C=CI)C1 c1(C(=O)NC(CNC(C(C(C)C)C)=O)C(C)(C)C)cccc(S(=O)(=O)CF)c1 N1(C(c2c(CC)ncs2)=O)CCN(C(=O)Cc2ccn(CC)n2)C(C2CCC2)C1 c1(C(=O)NC2CC(NC(c3cc(CC)c(C)s3)=O)C(O)C2)cc(F)c(O)c(F)c1 c1(C(=O)NCC(c2cccc(Cl)c2)NC(C2C(OC)C2)=O)cccc(Br)c1F C1(OC)CCC(C(N2CCCC(CCNC(=O)CC(C)SC(F)(F)F)C2)=O)CC1 N1(c2c(C)c(NCC3CC(=O)NC(C)C3)ncn2)CCOC2CCCC12 N1(C(c2ccc(C(=O)OC)[nH]2)=O)CCC2(NC(C3(F)CC(O)C3)=O)CCCC12 C(=O)(CCCCCC(C)O)N(CCNC(=O)CCc1nnc(C(F)F)o1)CC C=CC(C)(CCOCC)C(=O)N1CC2CC2(CNC(C2(COC)CC2)=O)C1 C=CC(CCC)CC(=O)NCCCOc1ccc(O)cc1 C1(NC(=O)COCC2CCC2)(CNC(=O)CC2CCCCC2O)CC(F)(F)C1 c1(OC)conc1C(=O)NC1(CC(=O)N(CCC(N)=O)CCO)CCC1 c1(CC(C)C)nc(C(=O)N(CC(CC)NC(=O)C(C)c2cccs2)C)cs1 c1(OC(=O)NC2CC2)cnc(OC(F)F)nc1O.n12cc(nn1)C(=O)C1CC2C1.OC(F)F C1(n2cc(-c3cc(=NC)[nH]cc3)nn2)=C(F)C(F)=C(Br)C1(F)C(=O)OC O=C(C#CC1(C(F)(F)F)CC1)NC(c1ccc(F)cc1)CNC(C1(F)CCC1)=O CC1CCC(C(N2CC(CCNC(=O)Cn3cc(Cl)cn3)OC(C)C2)=O)CC1C N1(C(c2c(C)nn(C)c2)=O)CC2CCC(C1)N2C(=O)C(C(C)(C)C)NS(C)(=O)=O c1(C(C)NCC2CCN(C(=O)OC(C)(C)C)C2C)cn2c(n1)CCCC2 CC(CNC(=O)C(F)CC1CN(C(C2CCCN2C)=O)C1)S(N)(=O)=O N1(C(C(=O)NCC(CNC(c2cc[nH]c(=N)n2)=O)OC)C)C(=O)CCC1=O CCCCC(C(=O)NC1CCCC1NC(c1c(NC(C)=O)c[nH]c1C)=O)C(C)C C1(CNC(COCCCC)=O)C2CCCC1N(C(=O)C=Cc1csc(C)n1)C2 CC(C)C(C)(O)C(=O)N(C)CCNC(c1ccc(C(F)F)nc1O)=O n1(CC(=O)NC2C(CC)CN(C(=O)CCCCSC)C2)ccc(=O)n(C)c1=O C(CCCCC(=O)N1CCCCC1C(=O)NCCC(C)CCO)OC N1(C(c2ccc(C)c(C3CC3)c2)C(=O)NCC)CC(C)C12CCOCC2 C(=O)(C(F)C(C)C(F)(F)F)N1CC(O)(CN(C(c2c(C)cn(C)n2)=O)C)C1 c1(C(=O)NCC(CC)(CC)NC(=O)C(C)=CC(C)(C)C)cc(Cl)ccc1O N1(C(c2cccc(C)n2)=O)CCN(C)CC1C(=O)NCC1CCOC1 C1(N(C(Cc2c(C)n[nH]c2)=O)C)CCN(C(=O)CNC(C2CCC2)=O)CC12CC2 C1(CC)CCN(C(C2CCN(CC)CC2)=O)C1CNC(c1ccoc1)=O N1(C(C(C)NC(C)=O)=O)CC(NC(=O)C=Cc2ccccn2)C2(CCOCC2)C1 c1(C(N2CCC(NC(c3cnn(CCS)c3)=O)C2)=O)cc2c(nn1)CCCC2 c1(C(C(=O)NCC(CN(C(C=CCN(C)CC)=O)C)C)SC)ccccc1 c1(CNC)cnc(C(C)C)nc1N(C)CC1CCCCN1C(C1C2COCC12)=O Cc1cc(C(=O)NCC(C)NC(c2cccn2CC(F)(F)F)=O)n(C2CCC2)n1 C1(NC(C2N(CC)CCOC2)=O)C2CC1N(C(c1ncn(CC)n1)=O)C2C c1(OC(C(=O)OC)COC(C)(C)C)ccc(SC)cn1 CC(C)C(C(=O)NC1COCCC1NC(=O)C1CC1)N1CCCCC1 C1(C(=O)NC(CCC)C2CCCC2)C=CCCN1C(=O)CCCCNC(N)=O c1(OC(C)C(=O)NCC(=O)CC2CC2C)cc(F)ccc1F CCC(CNC(=O)C(O)c1ccsc1)(CC)C(=O)N1CCC(CO)(CF)C1 c1(OC(C2CCCC(C)N2C(=O)OC(C)(C)C)=O)ccc2occc2c1 C(CC(F)F)(C(=O)NCC1CS(=O)(=O)C1)NC(C1C(C)=CCS1)=O Cn1cc(C(N2CCC3CCCC23CNC(=O)C2=CCCSC2)=O)c(O)nc1=O N1(C(CCSCC)=O)CCCC(NC(C2CC(C(C)C)C2)=O)C(F)C1 c1(N(CC(C(C)(C)C)NC(C2CC(=O)NC(=O)N2)=O)C2CC2)ncnc2scnc12 c1(C(=O)NC(CCC)CC(=O)NC(C)C)ccc2c(n1)CCC2 N1(C(C(c2n(C)ccc2)=O)=O)C(C(=O)NCCC(F)CN=[N+]=[N-])CCC12CC2 c1(C(=O)NCCN(C(C2CC(C)C2)=O)CCOCCO)ccn2ccnc2n1 c1(CN2CCC(CNC(c3occc3Br)=O)C2)cn2cccnc2n1 c1(C(=O)NC(C)CCCNC(C2(CCO)CC2)=O)ccc(CN(C)C)cc1 Cc1cc(C(N2CC(CO)(NC(=O)CC3CC4CCC3O4)C2)=O)c(F)cc1Cl N1(CC)CC2CC1CN2C(=O)CC1CCCCC1NC(C1CCOCC1(C)C)=O c1(C(=O)NC(C(C)NC(C2CCN(C3CC3)C2=O)=O)(C)C)cn2c(n1)CCCC2 C(=O)(C1CCCn2c(Br)cnc21)N1CCC(NC(CCOC)=O)(CF)C1 c1(C(=O)NCC2N(C)CCN(C(=O)CNS(N)(=O)=O)C2)ccc2ncccc2c1 Cc1cn(CC(=O)NCC2(C)CCN(C(=O)CCCC(C)O)C2)c(=O)nc1O c1(CC(=O)N(CC(C)NC(C2N(C(=O)OC)CCC2)=O)C)c(C)nn(C)c1Cl Cn1cncc(CNC(=O)NCc2ccc(=O)oc2)c1=O c1(C(CNC(=O)Cc2ccoc2)NC(CC2C(C)C2)=O)ccccc1C(F)(F)F c1(C(CNC(C2COCCO2)=O)NC(c2ccc(CC)[nH]2)=O)ccccc1CC c1(C(C)(C)C)nc(C#N)c(NNC(=O)c2ccc(F)c(Br)c2)o1 C1(C2CCN(C(c3ccn4ccnc4n3)=O)CC2)(NC(C(CSC)C)=O)CC1 O=C(NNc1cccc2ncccc12)NC1CN(Cc2ccccc2)CCC1(F)F C=C=C(C)CC(=O)C(=O)C(C)(C)O.c1(CCC(=O)N(CCN)C)ccccc1 c1(Nc2ncnc(C(F)F)c2Br)ccc(Cl)c(C#N)c1.CC1CN2CC12 Cc1ncc(Cl)cc1CCN(C=O)CC1CC12CCC2 N1(C(CC=C(C)C)=O)CC(CNC(C2(C)CCNC2=O)=O)OC(C)(C)C1 Cc1cc(C(=O)NCC(C)NC(c2cccc(-n3cccn3)n2)=O)c(C)cn1 Cc1csc(C(=O)NCC(O)CCNC(c2nocc2Cl)=O)c1C c1(OC)c(C(=O)N(C(CNC(=O)C(F)(F)CN(C)C)C2CC2)C)cccc1Cl n1(CCC(N2C(CNC(C3C(=C)C3)=O)C=CC2)=O)nc(C)c(C)c1C CC1CC(C(=O)NC23CCC(NC(c4c[nH]ccc4=O)=O)(CC2)C3)CC(C)C1 c1(C(C)=O)cccc(N(c2ncncc2F)C(=O)CN2CCCCCC2)c1 CCCC(CCCNC(c1cc(N)cc(O)c1)=O)NC(c1c(C)cncc1F)=O N1(C(C2(C)CCC(=O)C2)=O)CC(CO)C2(C1)CN(C(c1ccc(C3CC3)s1)=O)C2 CC1(C)CC(C)(C(=O)NC2CN(C3CC3)C2)CN1C(=O)CC=Cc1ccccc1 CC1C(NC(c2cnc(C(F)(F)F)s2)=O)CCN1C(=O)Cc1csc(S)n1 C1(CNC(C(C)CF)=O)CN(C(=O)COc2ccccc2F)CCC1(C)C C(CC1CCC1)(C(=O)N1CC(O)(CNC(c2cc(C(N)=O)co2)=O)C1)NC(C)=O CCCCCC=CCC(=O)NCCC(N1CCC(CC(N)=O)C1)=O C1(NC(CCCCNC(N)=O)=O)CCN(C(=O)C2=NNC(=O)CC2)CC(O)C1 C(=O)(C(F)C(C)CNC(c1cc(OC)ns1)=O)N1CC(O)(CCC)C1 N(C(=NCc1sccc1Cl)NCC1CCCCO1)CC1(C#C)CC1 Cc1c(C(N2CCC(F)(C(=O)NC3CN(C)NC3=O)C2)=O)nnn1C C1(CN(C(=O)CCn2cnc(=N)[nH]2)C)CCCCN1C(c1nsnc1O)=O C(=O)(CC(C)C(=O)NCC#CC(=O)NCC1(C)CCC(=O)N1)OCC C1(NC(c2ccn3nnnc3c2)=O)CN(C(C2CC2Cl)=O)CC(F)(F)C1 N1(C(c2ccc(CNC(c3c(CCC)[nH]cc3)=O)cn2)=O)CCC(F)(F)C(O)C1 N1(C(c2c(C#N)ccs2)=O)CCN(C(c2csc(Cl)c2)=O)CC(O)C1 C1(C(=O)NCC(CC=C)NC(c2ccc(C(F)F)cc2)=O)CC(C2CC2)=NO1 Cn1cc(C(=O)NCCOCC(=O)NCc2[nH]nnc2C2CC2)ccc1=O c1(OC)ccc(CN2CCN(C(=O)Cc3ccccc3O)CC2)cc1Cl c1(C(N(C(CNC(=O)CNC=O)C2CC2)C)=O)cccc(SC(F)(F)F)c1 C1(CCC)CN(C(c2conc2COC)=O)CC1CNC(=O)CN(C)C c1(C(C(=O)NCCC(C)N(C(C(C)NC(=O)NC)=O)C)SC)ccccc1 N1(C(C2C(C)CC2)=O)CC(CCNC(C2(CO)CC(F)(F)C2)=O)C2(CC2)C1 c1(NCC(C)NC(C(CC)OC2CCCCC2)=O)cc2nnc(C)n2cn1 CCCC(C(=O)NCC(C1CC1)N(C(=O)Cn1nc(C)oc1=O)C)S(N)(=O)=O C(CC(C(=O)NC(C12CCC(CC1)C2)C)OC)NC(C1(SC)CCC1)=O N1(C(CCC(C)OCC)=O)CC(NC(=O)CCSc2ccccc2)CC1(C)C c1(CNC(C(N2CCC(C)(C(=O)NC)C2)=O)=O)nc2ccc(C)cc2[nH]1 c1(C(=O)NC2CC(NC(c3nnn(C)c3N)=O)C2)cc(C(C)(C)C)ccc1O N1(C(C(C)NC(c2ccncc2)=O)=O)CCOCC(CNC(=O)CC(C)(C)O)C1 C1(NC(CCC(C)NCC)=O)CCN(CCOC)CCC1(F)F.S(=O)(=O)(CCOC)N N1(C(C(C(C)(C)C)NC(c2c(C#C)c[nH]n2)=O)=O)CC2CC(CO)C(C2)C1 C1(NC(C(C)NC(=O)NC)=O)CCN(C(c2n[nH]c(C)n2)=O)CCC1(F)F c1(C(N2CC(N(C)CC)C2)=O)ccnc(CNC(=O)C=CC2CCC2)c1 C1(C(N(C2CCCN(C(c3c(C)ccc(C)c3)=O)C2)C)=O)CC2(C1)CC1(CC1)C2 Cc1c(C(=O)NCC=C2CCN(C(=O)CC3CCCCN3C)CC2)cnn1C CC1CCCC1(C)C(=O)N(CCCN(C(=O)CCc1cccc(O)c1)C)C C1(NC(CC(C)C)=O)C2C=CC(C2)C1C(=O)NCCCNC(c1cc(Br)n[nH]1)=O c1(C(=O)NC2(CNC(=O)COc3ccon3)CCCC2)cc2ncccc2[nH]1 N1(C(CCN(CCC)C)=O)CCCOC(CNC(c2cc(COC)oc2C)=O)C1 C(=O)(CCCC1CCCO1)NC(C(=O)NC(C(=O)OC)C1CCC1)c1cccs1 c1(CN2CCC(O)(CC(=O)NC(=O)Cc3cnco3)CC2)csc2ccccc12 N1(C(c2c(CCC)occ2)=O)CCC(NC(=O)Cc2cnn(C)c2)C(C)C1 c1(C(N2C(C)CCN(C(CSCC(C)=O)=O)CC2)=O)n[nH]c2c1CC(C)CC2 c1(OC)ccc(CCN(C)C(C)=O)cc1F.c12cc(no1)CN2 c1(NC(C(CC)C)=O)cccc(Cl)c1OC(F)(F)F.C12CCN(CC1)C(=O)CO2 c1(C(=O)NC(C(c2ccccc2)NC(C=CSC)=O)C)sc2nnc(S)n2c1C c1(C(=O)NC2(C3CCCN3C(C3CCSC3)=O)CC2)ccc(O)c(F)c1F Cc1csc2c(N3CC4CC(NC(c5nc(Cl)cs5)=O)C4C3)ncnc12 c1(C(=O)NCCCCC2CN(C(N)=O)C2)ccc(-n2cccc2)nc1.C12CN(C1)C2 N1(C(c2nc(COC)oc2)=O)CC(NC(C2(CF)CCOCC2)=O)CCC1C N1(C(C2C(C)C2C)=O)CC(O)(CNC(c2cc[nH]n2)=O)C1 C1(C(=O)NC(C(=O)N(CC(C(C)C)C)C)C)CCC2(CC2)C1 C123CC1CN(C2)C3=O.C12(NC(C3C4CCC34)=O)CC(CNc3ccccc3)C1C2 C1(O)(C(=O)NCC(C)CC(=O)NC2CN(c3ncco3)C2)CCOC1(C)C c1(C(C23COCC2C3)N(C(C)CC(=O)OC)C(=O)CC2CCCCC2)ccccc1 S(=O)(=O)(CC(=O)NC1(CNC(C2CC2C2CCCO2)=O)CC1)N(CC)CC c1(OC)cc(CN2CCC(C(N3CCC4(CC4)C3)=O)C(O)C2)cc([N+](=O)[O-])c1O c1(NC(C2CC(O)CCN2C(c2scc(Br)c2Br)=O)=O)cc(Br)c(F)cc1I C1(NC(CCS(=O)(=O)NC)=O)CCSC12CN(C(=O)CSCc1ccccn1)C2 c1(C(=O)NC2COCCN(C(CC(C)n3cccc3)=O)C2)cc2ccccn2n1 n1(C(C)C)ccc(C(=O)NCC2(NC(=O)C(C)n3ccnn3)CCC2)cc1=O c1(N2CCC(CC(C)NC(=O)CC3CCC(=O)N3)CC2)ccnc2ncnn12 C1(C(=O)NC(C(=O)OCC)CO)CCCCC1CNC(c1sccc1Cl)=O C1(NC(c2c(SCC)cncc2)=O)CCCN(C(=O)CC2CC2C)C1C C1(CC=C)(C(=O)N(C)CC2C(C)(C)C2(C)C)CCCN1C(C1CC(=O)N(C)C1)=O c1(C2(F)CC(C(=O)NCC3(O)CN(C(c4cnc(O)o4)=O)C3)C2)cccc(F)c1 N1(C(C(CSC)C)=O)CC(C)OC2(CCN(C(c3cc[nH]c(=N)c3)=O)CC2)C1 C(C(COC)CC(=O)NC1CCCCC1N(C(=O)CCCn1cccc1)C)OC C12(C(=O)NCC3C(C)CCN3C(=O)CN3CCCNC3=O)CCOC(C)(C1)C2 Cc1nc(NC2CCOCC2F)c2cccnc2n1 Cc1cc(N)c(C)nc1C(=O)NCC1CN(C(C2OCC3CCCC23)=O)CC1C C12(C(=O)NCC(C)N(C(CC3C(C)CCO3)=O)C)CCC(F)(CC1)CC2 N1(C(c2c(-c3ccc(C)s3)c[nH]c2)=O)CCC(C2(N)COC2)CC1 C1(C(=O)NC(C)CC(O)CO)N(C(=O)CCOCC2CCC2)CC12CCCC2 c1(C(N2CC3C(CNC(C(CNC(C)=O)(C)C)=O)C3C2)=O)cnn2c1N(C)CC2 C1(CNC(CC2(OC)CCCC2)=O)CCN(C(=O)C(=O)C(C)C)C1(C)C Cc1ccc(CNC(N2CCC(NCC(F)(F)F)CC2C)=O)c(C)c1 C(=O)(C(CC)(CO)OC)NCCN1CCCN(C(C(CC#C)C)=O)CC1 C1(C(N(CC(CO)(CO)NC(C2CCC2(C)C)=O)C)=O)CCCCC(C)(C)C1 N1(C(c2c(C)cncn2)=O)CC2CC(NC(c3ccccc3O)=O)C(C2)C1 C1(C(C2CCC2c2cccnc2)=O)CC(COC(c2ccccc2)=O)CCN1 CCC(C)(C)C(=O)C(=O)NCC1OCCC1C(N1CC(F)(COC)C1)=O N1(C(C2C(OC)C2)=O)CC2C(NC(=O)CCCC3CCC3)C2C1 CC(C)C(O)C(C)(C)C(=O)NC(C)C(N1CC2(CCC1CO)CC2)=O C(=O)(N=c1cc(C(N)=O)n(C)[nH]1)C1C2CCN(C(CC=CC)=O)CC21 C1(CC(=O)NC(C)CC2CN(C(C3(CCF)CCC3)=O)C2)CCNC(=O)C1 c1(NC(C(c2ccc(OC)c(Br)c2)NC(CC)(CO)CC)=O)c(C)cc(C)cc1C c1(C(N2C(CNC(CC(=O)NCC)=O)CCC2)=O)cc2c(cc1Cl)OCCO2 c1(CNC(C(=O)N(CC(C2CCC(F)(F)C2)O)C)=O)cnccc1Cl C=CCC(C)(C)CC(=O)NCC1CC(NC(=O)COCCOC)C1 c1(CC(N2C(CNC(c3ccc(F)nc3)=O)CC3CC32)=O)ccn2cncc2c1 CC1(C(N2CCC2Cc2ccccc2)=O)CCN(C(c2cscn2)=O)CC1 C(=O)(C(C)(C)C(C)(C)O)NCC1CC(OC)CN1C(=O)CNC(c1ccoc1)=O C1(C(C)C)CN(C(=O)C(C2CC2)N(C(=O)CCC2(C)CC2)C)CCCO1 C1(NC(CN(CC)CC)=O)CC(CNC(c2cccc(N)n2)=O)C1(C)C Cc1cc(I)ccc1C(N1CCC(CC(=O)Nc2ccc(Cl)cc2F)C1)=O C(=O)(CC(C)C(F)F)N1CCC(CN(C(CCC2CC(C)C2)=O)C)C1 C1(NC(c2ccc(C(C)(C)C)o2)=O)CCCC(C(=O)NCc2ccc(Br)nc2)C1 C(=O)(C(CC(C)C)NC(C)=O)N1CC(CC(C)NC(C2(C#C)CCC2)=O)C1 c1(C(=O)NCCC2(O)CCN(C(CC(=O)NCC)=O)CC2)cc(C)cc(C)c1N C#Cc1ccnc(C(N2CCC(C(=O)N(C3CC(CC)C3)C)(CO)CC2)=O)c1 C1(NC(CN(CC)CC)=O)CC=C(C(=O)NCC)C1.N1(CC)CC(OC)C1 c1(COC)nocc1CNC(c1cc(C(C)(C)C)n[nH]1)c1nnnn1C S(=O)(=O)(c1ccc(C#N)c(NCc2c[nH]c(=N)s2)c1)NCC1CCN(CC)CC1 c1(C(c2nnnn2CC)NCc2c(CC)nc(C)s2)cc(Cl)cc2c1CCC2 c1(OC)ccc2c(=NCC3CCCC(C)C3)[nH]c(=NCC3(CF)CCC3)[nH]c2c1 C1(C(=O)NC2CCN(OCC)CC2)CCN(C(C2C3C4CCC(C4)C23)=O)C12CC2 C1(OCC#C)CCN(C(=O)CCNC(=O)CC2CNC(CC)C2)C1 c1(C(=O)NC(C(C(C)C)NC(=O)Cc2cncn2C)C)ccc(Cl)c(C(F)F)c1 C1(NC(C(C=CCCC)O)=O)CC2CCC1CC2NC(=O)CN(C)C(C)=O C(CCCCC(=O)N1CCC(CCNC(c2cc([N+](=O)[O-])c[nH]2)=O)C1)NC(C)=O c1(C(=O)NCC2(C)CC(NC(Cc3c(C)ccs3)=O)C2)nc2ccccn2n1 C1(NC(c2nccc(CNC(C(C)n3ccnc3)=O)c2)=O)COCC1N=[N+]=[N-] c1(CCC)nc(C)ccc1C(=O)NCCn1cc(CNC(=O)CC2CCC2)nn1 C(CC(=O)N(CC(C)O)CCNC(=O)CCCn1cccn1)(C(F)(F)F)SC N1(C(C(N2CCCCC2=O)C)=O)CCC2(CC(NC(=O)CSC3CC3)C2)C1 Cc1cn(C)cc1C(=O)NCC1CC(CNC(C2(CO)CC2)=O)CO1 CC1C(NC(c2cccs2)=O)CCCN1C(c1scnc1C(C)(C)C)=O CC1CC2CN1C(=O)Nc1csc2n1.C1(O)(C(C2CCC2)NC)CCCCC1 C1(CC)CN2CCCC2CN1C(=O)C(C1CC2(CCC2)C1)F c1(C(=O)NCCN(C(=O)C(C)=C2CCC2)CCC)ncn2c1COCC2 CC(C)C(C)C(=O)NCC1CN(C(c2conc2C2CCCC2)=O)CCO1 N1(C(CCNC(CCCCC)=O)=O)CCN(C(=O)CC(C)N(C)C)CC2(CC2)C1 C1(C(N2CC(CC(C)NC(C3CC(C)(C)O3)=O)C2)=O)CCNC1=O CC1(C)C(=O)CC1C(=O)NC1CCC(C(=O)NCC2CCNC(=O)C2)C1 c1(C(=O)NC2C(NC(C3C(C)(C)CCC3)=O)CC2)ccc(Br)cc1O c1(N(C(=O)C=C2CCN(C(=O)Cc3cncnc3)C2)CC=C(C)C)ccccc1 CCCC(C(=O)NC1CCC(NC(=O)CCCOc2ccccc2)C1)N(C)C N1(C(C=CC(C)(C)C)=O)CC2CC(NC(C3CC3c3cccc(F)c3)=O)C1C2 C(C(C)C(=O)NCCCC1(NC(=O)Cc2nncn2C)CC1)SC.C(=O)CO C1(CNC(c2cc(Oc3ccc(C(=O)C(F)(F)F)cc3)ccn2)=O)CC2CCC1O2 C1(C(F)(F)F)(C(=O)NC(C2CCOC2)CNC(C2CCCC2)=O)CCCCC1 C1(C(=O)NC(C(C)O)(C)C)CCN(C(=O)C(=O)NCC2CC2)CC1O C1(CNC(c2cc(C)nn2C)=O)CC2CCCCC2N1C(C12CC(C)(C1)C2)=O Cc1ccc(C=CC(=O)NC2CC(NC(=O)C(C(C)O)N(C)C)C2)cc1.C1(=O)CN1 c1(C(=O)NC)cccc(C(N2CC(NC(=O)CC3(C)CCCC3)C3CC23)=O)n1 CC(Cn1ccnc1)C(=O)NC(C)CC(C)NC(=O)C(F)(F)c1cscn1 N1(CC(c2ccc([N+](=O)[O-])cc2)n2cnnn2)Cc2nccn2CC(CO)C1 N1(C(c2cc(OC)ns2)=O)CCCC(N(C)C(c2cc[nH]c2C(C)C)=O)CC1 C1(C(N(CCOC)CCOC)=O)CCC(CNC(=O)C=CC(F)(F)F)C1 N1(c2nc(C)nc(O)c2)CC2CCCC(NC(c3c(C)cc(Cl)cc3Cl)=O)C2C1 c1(OCC)ccc(Cl)cc1C(C(=O)NCCC#N)N(C)C(C1CCCCC1)C C1(C(C(N2CCC(N(C(CN(CC)CC)=O)CC)C2)=O)OC)CCCOC1 Cc1cc(F)cc(C(N2CC(CNC(C3OCCOC3(C)C)=O)C(C)C2)=O)c1N c1(SCC(=O)NC2(C)CC(NC(c3n(CC)ccn3)=O)C2)ccc([N+](=O)[O-])cc1 N1(C(C=CC(C)NC(=O)C(C)c2ncco2)=O)CCCN(C)C(=O)C1 C1(NCc2cc(F)c3c(c2)OCCO3)CCC2(CC1)CNCCO2 C1(F)(C(N2C(C(C)(C)C)C=CC2)=O)CCN(C(C2CC(F)(CF)C2)=O)C1 N1(C(C(C)OCC2(c3ccccc3)CC2)=O)CCN(C(CC#C)=O)CC1 C(=O)(CCC(=O)c1cccnc1)NC(C)C(c1cccc(O)c1)C c1(C(=O)NC(C)C(CO)NC(c2ccc(N)cn2)=O)cc2nc(F)ccc2o1 C(=O)(C1CCc2c[nH]nc21)NCC(C)NC12CC3CC(CC(C3)C1)C2 C#CC1CCCC(c2nnnn2C2COC2)(NCC2COC(CCSC)C2)C1 N1(C(CC2C(C)=NOC2=O)=O)CC(NC(c2ccc(CO)nc2)=O)CC(C)(C)C1 N1(C(C(CCC)CC)=O)CCCC2C(NC(C3CSCC(=O)N3)=O)C(C)(C)C12 N1(C(C(C(C)(C)C)O)=O)CC(CO)C2(C1)CN(C(=O)CC1CCC(=O)N1)C2 c1(OCC)cc(Cl)c(C(N2CC(NC(C3CCCO3)=O)C(F)(F)C2)=O)cc1Cl C1(NC(=O)C2=COCC2)CCCCN(C(=O)CCc2ccc(Cl)cc2)C1 c1(C(=O)NC(CNC(C(C(C)C)NC(N)=O)=O)(C)C)ccc2c(O)nncc2c1 C1(N(C(C=C(C)Cl)=O)C)CCCC2CN(C(c3c[nH]cc3Br)=O)CC12 c1(C(=O)NC2COCCN(C(c3c(C)cno3)=O)C2)nc2c(cc1Cl)OCCO2 c1(C(N2CCC(C(C)NC(C3(C#N)CC=CC3)=O)C2)=O)cc(F)cc(F)c1 C1(NC(c2ccnc(C)c2N)=O)C2CC(O)C1N(C(c1cc(=O)n(C)o1)=O)C2 N1(C(C2N(CCC)CCCC2)=O)CCN(C(c2snc(O)c2Cl)=O)CC1CCC Cc1cncc(C(N2CCN(CCN(C)C(c3cc(O)nn3C)=O)CC2)=O)c1Cl N1(C(C2C(NC(c3cn(C)c(=O)cn3)=O)CCOC2)=O)CC2CCCC(O)C2C1 Cc1cc(C(=O)NC2(CF)CCN(C(=O)C=Cc3cc[nH]n3)C2)cc(C)c1O c1(C(=O)NC2C(NCC)CCC2)ccc(C(=O)N)cc1.C(=O)(C(C)OC)NCC1CC1 C(CCOCCO)(C(=O)NCC(C1CC1)N(C)C)NC(C=NOC)=O CC1(C)OCCC1(O)C(=O)NC1C2CC3C1C3C2C(=O)N(C1CC1)CC1CCCO1 C1(C(=O)NC2(C)CC(NC(=O)C3CC3)C2)CC2C=CC1O2 C12(CNC(=O)C=Cc3cc[nH]n3)CCC(CNC(=O)C3=CCCSC3)(CC1)CO2 c1(C(=O)NC(C(C)NC(C(C)c2ccco2)=O)CO)cc(=O)c2ccccc2o1 c1(C2CC(OCC)C2)nc(-c2cn[nH]c2)nn1Cc1cncc(F)c1.C1(C)CCCO1 CC(C)(C)C(O)CCC(=O)N1CCCC1C(=O)N(C)CC1CC1 CC(C)(CNC(c1c[nH]nc1CNC(=O)Cc1cnoc1)=O)CCO CN1CC2(CCCN(c3nc(N4CCCC(F)C4)nc4c3SCC4)C2)CC1=O Cc1nn(CCC(=O)NCC(CO)NC(C2CC23CCCC3)=O)c(C)c1[N+](=O)[O-] CCCC(C)(O)CC(=O)N1CCCC(CO)(NC(c2[nH]nc(OC)c2Cl)=O)C1 Cc1cc(NC(C2(C(C)NC(C3CC(C)CCO3)=O)CC2)=O)c(F)cc1F C1(C(=O)NCCC2(O)CN(C(CN(CCOC)C)=O)C2)CC2(CCCC2)CO1 c1(CC(=O)NC(C(C)C)CNC(C2CC(F)C2)=O)ccc2ncccc2c1 C1(C2CCCN(c3ccnc(C(F)(F)F)n3)C2)(NC(c2csc(Cl)n2)=O)CC1 Cc1cc(C)c(C(=O)Nc2cc(C)nc(-c3ccccc3)n2)c(C)c1 c1(CC(=O)NCC(CCCC)NC(c2c(C)coc2CC)=O)cccc(C)c1Cl C#Cc1c[nH]nc1C(=O)N(C1CCN(C(c2ccc(F)nc2)=O)CC1)CC(C)C CCC(CC(=O)N(CC(Cc1ccccc1)NC(c1cnsc1)=O)C)C(F)F CCC(F)(F)C(C)(C)C(=O)NCC1CCC1NC(=O)CSc1ccccc1O C1(C2CC2)(CNC(c2c(CC)cccn2)=O)CCN(C(c2csnc2Cl)=O)C1 c1(C(=O)NCC2CN(C(c3ccc(OC)cc3F)=O)C2)ccc2c(c1)COC2 C(CNC(=O)C(c1cccc(OC)c1)C)(CC(C)C)NC(c1ccn(CC)n1)=O C1(=O)C(CC(F)F)N1.Cc1ncc(CN(C(=O)C(F)OC(F)(F)F)C)o1 C1(CCNC(C=C(CCC)CCC)=O)CCN(C(c2cnc(S)nc2)=O)C(C)C1 c1(C(N2CC(NC(c3ccc(C)s3)=O)C(C)CC2)=O)ccc(C2=CCCC2)cc1 c1(CN(C(CCCOC)=O)C)cccc(CNC(c2coc(Cl)c2)=O)c1 C(=O)(C(C)CC(=O)N1CC=CC(C(=O)NC(c2nn(C)cc2O)C)C1)OC C(C(C)(C)CC(C)O)NC(C(CN(C(C1C(C(C)C)OCC1)=O)C)(C)C)=O n1(CC(N2C(C)CN(C(C3CC3C(F)F)=O)CC2)=O)ccc2ccc(F)cc12 C(=O)(CCCCC(F)(F)F)NCCCN(C(CC(C)CF)=O)CC1CCCC1 c1(C(=O)NC(CNC(C2(CC)CCNC2=O)=O)C(C)C)cccc(C)c1N Cc1nnsc1C(=O)NCC1CCC(C(=O)NCC2CCCC2C(=O)NC)O1 Cc1ccc(C)c(C(N2CCC(F)(CNCCCCCn3ccnc3)CC2)=O)c1 C(=O)(CCC(C)(F)F)N1CC(CCC)C(NC(=O)CCCOc2cccnc2)C1 c1(CNC(c2cc(C(C)C)[nH]n2)=O)cnn(C)c1C(=O)NCC1(S(C)=O)CC1 c1(C(c2n(C3(C)CC3)nnn2)NCC2C(F)(F)C23CC3)nnn2ccccc12 c1(CN(C(=O)C(CCC2CCC2)NC(=O)CCOC2CCC2)C)ccnc(F)c1 C(=O)(C1=CCCC1C)NCC(CC(=O)N(CC(F)F)CC)C Cc1c(C(=O)NC2CC(NC(c3cnc(O)c(F)c3)=O)C2)nn(C)c1Br N1(C(C=C(CCC)C)=O)CCC2(NC(c3ocnc3C3CC3)=O)CC2C1 N1(C(C(C)CC2CCCO2)=O)CCC(N(C)Cc2ccccn2)CC1 N1(C(CC=C)=O)CCN(CCCCCC2CCCC(C(=O)OCC)O2)CC1 c1(OC)ccc(C(=O)N(C)CCN(C(=O)CC(C)c2ccco2)C)c(F)c1Cl C1(OC(c2ccc(OC(=O)CCOC(C)C)cc2)COC)CCN2CCOCC12 Cc1cc(C(=O)N(C2CCCCC2NC(C2CC(O)CN2C)=O)C)cc(F)c1 N1(C(=O)C(C)O)CC2CCC(NC(C(C)(C)OC(C)C)=O)(C2)C1 c1(C(N(c2ccccc2Cl)CC2N(CCOC)CCCC2)=O)cc(C#N)cn1C C1(NC(c2cnoc2C2CCC2)=O)(CO)CCCN(C(=O)Cc2csc(S)n2)C1 C1(C(=O)NC2CC(OC)C2)COC2(C1)CN(C(=O)COc1ccc(C)cc1C)C2 N1(C(c2c(C)scc2)=O)CCN(C(=O)CCc2cccnc2)C(C)C1 N1(C(C2CC(C#C)(O)C2)=O)CCC=CC1C(=O)NCc1ccc(Cl)nc1 c1(CCNC(N(C(c2ccccn2)C)C)=O)cc(O)cc(Br)c1 N1(C(C#C)=O)CCC2(CC1)CCN2Cc1ccccc1CC N1(Cc2cc(C)c(Br)cc2)CCC2(CCCN(C(C3(CS(C)(=O)=O)COC3)=O)C2)C1 N1(C(c2cnc(NC(C3(CF)CC3(F)F)=O)s2)=O)CCOC(CCOC)C1.CO CC1CN(C)CC1(c1nnnn1CC1CC1)Nc1ccc(N2CCCC2)c(Cl)c1 c1(C(=O)NCC(CNC(CCn2c(=O)cc(C)nc2)=O)F)cc(C)c(C)c(F)c1 c1(C(=O)NCC2CCCN(C(CC3CC(C)C3)=O)C2)cc(O)nc(Cl)c1 C(CN=c1nn[nH]n1-c1ccccc1)N1CCN(C(=O)CCC2CCCCC2)CC1 c1(C(=O)NCC(=O)NC2CN(C(C(C)C3CCC3)=O)CC2C)ccc(C#N)cc1 N1(C(CC)=O)CCCC(C(=O)NC2(C)CN(C(C3(c4cccc(C)c4)CC3)=O)C2)C1 c1(N2CC=C(C)CC2)nc(=N)[nH]c(=NCC(C)(C)N2CCOCC2)[nH]1 c1(COC(c2ccccc2-c2cccc(Cl)c2F)=O)cc(F)cc(Br)c1F c1(C(=O)NC2C(NC(C(CC)OCC)=O)CCC2)c(OC)ccc(F)c1OC c1(C(N2C3C(N(C)C(C4CCCCC4)=O)CC(C3)C2)=O)c(N)cccc1[N+](=O)[O-] CC1c2nccn2CCN1C(C1CCC(NC(=O)CCc2cncnc2)C1)=O CC1CC(C)(C(=O)NCCCC2(NC(c3cnc(C4CC4)s3)=O)CC2)C1 C=CC(O)(C(=O)N1CC2CCCC(NC(C3SCCCS3)=O)C2C1)C(F)(F)F C(=O)(CC1=CCN(C)CC1)N1C(C)CC(NC(C2CC(=O)NC(=O)C2)=O)CC1 Cc1nn(C)cc1NC(C1CC(NC(=O)COCCCF)CC1O)=O C1(C(=O)NC(C(C)C)CNC(=O)Cc2ncc(Cl)s2)CC1C1CCOCC1 C(=O)(C(CN(C)C)C(C)C)N(CCNC(CC)=O)Cc1cc(C)n(C)n1 N(C(=NCC(C)c1ccc(Cl)cc1)N1CCC(CC2CCC2)C1)C(C)C c1(C(N2CC=C(CNC(CC3C(C)OCC3)=O)CC2)=O)occ2c1CCCC2 CC(C)(C)C(CO)C(=O)NCc1cc(C(=O)NCCc2cccc(O)c2)n[nH]1 c1(C(=O)NCC2CN(C(CCN(C(CCC)C)C)=O)C2)csc(C2CCCO2)n1 N1(C(C(C(C)C)O)=O)CCC(C2(NC(=O)Cn3cc(C(C)O)nn3)CC2)C1 C1(N(C(=O)CCCn2cncn2)C)CCC(NC(c2cccc(C(N)=O)c2)=O)CC1 c1(C(=O)NC(CC=C)CNC(c2nccnc2N)=O)ccc(C(C)=O)c(F)c1 c1(OC)ccccc1CN(C)C(C1CC=CC(n2cc(CC3CC3)nn2)C1)=O c1(C(N2CCC(NC(CCc3n(CC)ccn3)=O)CC2)=O)nn(C)c(C)c1Cl C1(NC(=O)C2=CCCCC2)CCCC12CN(C(c1ccoc1Br)=O)C2 C1(CC)CNC(=O)CN1C(c1coc(CCCNC(=O)COC(C)C)n1)=O CC1(C)CC(C(=O)NC2(CO)CC2)CN1C(=O)C(O)CC1CCCC1 c1(C(N2CCC(NC(C)=O)C2)C(=O)NCCOCC2CC2)nnc(O)nc1O N1(C(CCC#C)=O)CCCCC1C1CCCN1C(c1ccc2nc(O)oc2c1)=O N1(C(c2cc(CNC(c3nc(C)oc3)=O)on2)=O)CC2CC1CS2=O Cc1cc(N)c(C(N2CCCC(C)(CNC(C3(C)CC(F)(F)C3)=O)C2)=O)c(F)c1 c1(CCC)cc(C(=O)N(CC(C)(C)C(=O)OCC)C)c(C)o1 CC1CCCCC1(C)C(=O)NCC1(C(=O)NCC2NC(=O)NC2=O)CC2(CC2)C1 C1(CC)CN(C(c2c(CO)noc2C)=O)CCC1NC(=O)CC1CSCCS1 c1(OC)ncnc(N2CCC(NC(c3c(NC(C)=O)cccc3F)=O)C2)c1C C1(C(N2CCCC(C(=O)NCc3nc[nH]n3)C2)=O)(COC)CCCOC1 C1(C(=O)Nn2c(O)cc(N3CC(CCn4cc(CC)nn4)C3)n2)CC2CCC1CC2 C1(NC(CC=CC)=O)CC2CC1CN(C(=O)C(C)=C(C)CC)C2 C(CNC(c1cc(C#N)cs1)=O)(C(C)(C)C)NC(Cc1cn(CC)nc1)=O N1(C(C2(OC)CCSC2)=O)CC2(CCN(C(C3(COC)CCCCO3)=O)C2)C1 N1(C(c2c(CC)ncnc2)=O)CCCCC(NC(C2CC2Br)=O)C1 c1(C2(NC3C(C)(N(C(N4CCCC4C(F)(F)F)=O)C4CC4)C3)CC2)ccncc1F C(=O)(CC(C)(C)C(=O)N(C1CN(C(c2ccc([N+](=O)[O-])o2)=O)CC1(C)C)C)OC N1(C(c2cc(C(F)F)[nH]n2)=O)CCCC2(CCN(C(C3CCCSS3)=O)C2)C1 C#Cc1ccc(F)c(C(=O)NC2CN(C(c3cc(C)nn3C)=O)CCC2F)c1 C1(O)(CN(C)C(c2nc[nH]n2)=O)CN(C(=O)CN2CCCC2)C1 N1(C(CC2C(C)=NOC2=O)=O)CCCC2C1CCN2Cc1ccc(F)c(F)c1 Cc1cc(C(N2CC(CC(=O)NCCCc3ccsc3)CC2(C)C)=O)ccc1F c1(CNC(CC2C(C)=NNC2=O)=O)nc2c(s1)CCN(C(=O)C(C)N1CCC1)C2 c1(C(=O)OCc2ccc(OC)cn2)cc2nc(-c3ccoc3)ccc2[nH]1 c1(C(=O)OC)ccc2nc(NOCC3COCCO3)[nH]c2c1 C1(NC(C(c2ccc(Cl)cc2)OC)=O)C=CCN(C(=O)C(C)(C)CC2CC2)C1 C#CC1CCCCN(C(C23C(N)C(O)C2OC3)=O)C1.C123CCC(CC1)(C2)C3=O N1(C(c2cc(C)nnc2)=O)CCOC2CCN(C(C3CNC(=O)CC3C)=O)CC12 c1(CC)ccc(C=CC(=O)NCC2CCC(CNC(=O)CO)C2)cc1 C(=O)(CCCCCCNC(C1(C(F)(F)F)CCC(N)C1)=O)OC C1(CCCC)CN(C(C2CC2c2ccncc2)=O)CCN1C(c1nn[nH]c1Cl)=O CCCC(C(=O)NCCCNC(c1sccc1NS(C)(=O)=O)=O)OCC N#CC1(CNC(=O)C(CO)NC(=O)CC(O)C2CCCC2)CCCC1 N1(CCCCC)CCC(c2nnnn2C)(NCCc2ccc(N(C)C)nc2)CC1 c1(CCCC(=O)NCCCN(C(=O)CC2C=CCC2)C2CC2)ccc(Cl)cc1 CC(C)C(C)CC(=O)N1CCN(C(=O)Cc2cncn2C2CC2)CC1C C(=O)(C#CC1CCCC1)N1CCN(C(c2c(C(=O)OC)c[nH]n2)=O)C(CC2CC2)C1 c1(N(CC(C)C(F)F)C)ccncc1S(=O)(=O)NC1CCN(c2ccccn2)C1 C(=O)(C1CCCn2cnnc21)NCCCC(C)NC(c1cnns1)=O C(=O)(C(C)(C)S(C)(=O)=O)NCC1(C)CCCN(C(C2C(OC)(OC)CCC2)=O)C1 c1(CC(N2C(C)CCCC2CN)=O)ccccc1S(C)(=O)=O c1(CC(=O)NCC2C(C)CN(C(=O)CC3CC3)C2)ccccc1S(C)(=O)=O C1(C(C)NC(=O)CCc2cnc(C)s2)C(C)CCN1C(=O)COC(C)=O.C(CC(C)C)S N12CCCC(C1)N(CC)CCC2=O.c1(C(C(=O)NC)O)ccc(F)cc1 c1(CC(=O)NCCSC)ccc(C(C)(C)C)cc1.N12CCC(C1)N(C)C(=O)C2 Cc1cncc(CCC(=O)NCC23CC(CNC(c4ncn(C)n4)=O)(CO2)C3)c1 c1(C(N(C(C)CN(C(=O)CCS(N)(=O)=O)C)C)=O)cccc2occc12 c1(CC)cc(CNC2CN(C(=O)OC(C)(C)C)C(C)CO2)ccc1C#N c1(C(=O)NCCOC(COCC2CCCC2)OC)ccc(OC)c(OC)c1 c1(C(N2C(C(=O)Nc3ccc(C)cc3C)CC2C)=O)ccn2cncc2c1 C1(C(N2CC(N(C(COC)=O)C)C2)=O)CCN(C(C2CCC(C)(C)O2)=O)CC1 C#CCCCC(C)C(=O)NCC1CN(C(=O)C=C2CCC(C)CC2)CCC1(C)C Cc1n[nH]c(C)c1CC(C)C(=O)N(CC(C)N(C(=O)Cc1cnoc1)C)C c1(OCC)cc(N2CCOC(CNC(c3cnnn3CC)=O)C2)ncn1 Cc1nnc(SC(=O)CCCNc2cccc(F)c2)n1C1CCCCC1 C1(CNC(c2cccc(CC)n2)=O)CCN(C(c2sccc2C#N)=O)C12CCC2 C(C(=O)N1CC(O)CCO1)N(C(=O)C(C)CC1CCCC1)CCOC c1(N2CC3CN(C(c4c(C)ccnc4)=O)C3C2)ncnc2c1ncn2C(C)CO c1(C(=O)NCC(CO)NC(c2nccc(Cl)c2O)=O)ccc2oc(O)nc2c1 C(C)(C)(CC(C)N=c1[nH]c(=N)[nH]c(=NCCC2OCCC2(C)C)[nH]1)OC C(C(C(=O)NCCN(C)C)NC(=O)CCOCc1cc(C)no1)OC c1(N(C(C(=O)NC(CC(C)C)c2ccccc2)=O)C)cccc(N)c1 CC(C)(O)C(F)C(=O)NCC(C1CCCCC1)NC(c1c[nH]cc1Br)=O C1(NC(c2c(COC)scc2)=O)C=CCN(C(c2sc(NC3CC3)nc2C)=O)C1 C1(NC(c2ccnc(Cl)c2Cl)=O)CCC2CN(C(=O)CC3OCCCO3)CC2C1 c1(C(=O)NC(CCCNC(c2cccc(C)n2)=O)(C)C)ccnc2[nH]c(C)nc12 C(=O)(C(=O)N(CCCN(C)C)C)N(C1CC1)CC c1(C(C(=O)NC2CCCC2)N(N2CCCC2)CC=C)cc(OC)cc(OC)c1Br N1(C(C(C)OCCCC)=O)CCCCC(NC(c2ccoc2C)=O)C1 C1(C(N2C(C(C)(C)C(N3CC4CSCC4C3)=O)CCC2)=O)CCCCNC1=O Cc1cccc2cc(C(=O)NC3CCCCC3NC(c3ccnc(O)c3)=O)[nH]c12 Cc1ncc([N+](=O)[O-])cc1-c1ccccc1C1CC1C(=O)NCC1(N(C)C)CC1 C12(NC(CC(C)SC)=O)CCC(C1)N(C(C1CC(C)(O)C1)=O)C2 C(c1csc2ccccc12)=CC(=O)NCC(C1CC1)NC(CC(C)F)=O C1(CC(=O)NCCN(C(c2ccc(C(F)(F)F)nc2N)=O)CC)CCCCC(=O)N1 C(C(CC(C)C)NC(C1(CO)COC1)=O)NC(C1CC(C)(C(=O)OC)C1)=O C(c1cncc(C)c1)=CC(N(C1CCN(C(C(CC=C)C)=O)C1)CCC)=O c1(Nc2ncc(-c3ccc(CCCC)s3)cc2Cl)cnc(Br)c(Cl)n1 C(=O)(C(C)CC(=O)N1CCC(NC(c2ncccc2OC(C)C)=O)CC1C)OC c1(C(COC(C)C)C)cn(CCCC(=O)NCC2CCC(F)C2)nn1 C1(C#N)(C(=O)NC2CCC(CC(N3CC(N(CC)CC)C3)=O)C2)CCCO1 C(N=C(NC1CCCC1)N1CCN2C(=O)NCC2C1)c1c(C)occ1 N1(C(C2CC(C)OCC2)=O)CC2CC(NC(c3cc(C(F)F)[nH]n3)=O)CC2C1 Cc1nc(C(N2CCC(NC(c3cc[nH]c3C3CC3)=O)C2)=O)cc(O)n1 c1(NC(c2ncccn2)CC)cc(NC2CCOC2C2CC2)ncn1 C1(OC)CC(CCNC(C2CCCS2)=O)N(C(=O)COc2ccccc2F)C1 C1(CNC(CC2C(CC)C2)=O)CCC2CCC1N2C(=O)C(F)=C(C)C1CC1 C1(CC(=O)NCC(C)NC(c2nc(C(C)OC)sc2)=O)CC2(CCC2)C1 C12(C(=O)NCCC=C)CCC(C(=O)Nc3c(C)nn(CC)c3C)(CC1)CC2 N1(C(COc2cccc(CC)c2)=O)CCC(C)(NC(c2ccc(SC)o2)=O)CC1 C(CCCCCC(=O)NC1CCC(Cn2cc(-c3cnc(CC)o3)nn2)C1)SC C(=O)(CCCCC(=O)NOCCO)OC(C)(C)C.C(C(C)CO)N(C)C=O Cc1cc(C2=NNC(=O)CC2)nc(N2CC(C(N)=O)CC(C)C2)n1 CC1(C#N)CCCN(C(C23C(NC(C4CCCO4)=O)C4CC2C3C4)=O)C1 N1(C(C2CCN(C)CC2)=O)CCN(C(=O)CC2C=CCC2)CC1CC(C)(C)C c1(C(C)=O)cc(CN2CCCC2(C)C(=O)NCC(F)(F)F)ccc1O C(=O)(C(C)(C)C(C)O)NCC(CC)NC(c1snc(C)c1N)=O C1(CC=C)(NC(C2COCCN2C)=O)CCN(C(=O)CCc2nc(O)n[nH]2)C1 CCCCCC(O)C(=O)N1CC(NC(c2cnc(C)s2)=O)CC1(C)C C1(C(N2CCOC(c3ccccn3)C2)C(=O)NCCCF)CCC2(CCC2)CC1 C(CCCCC(=O)NC1CC(C)CN(C(c2cnco2)=O)C1)NC(C)=O Cc1nc(C)c(CNC(=O)C(C)(C2CCC2)NC(C23CC2CNC3=O)=O)s1 C1(C(=O)NC2(C)CCN(C(Cn3c(C(C)C)ncc3)=O)C2)CCCC12CCC2 CC1CC(C(N2CC(CO)C(C)C2)=O)CN(C(c2ccn(C3CC3)n2)=O)C1 c1(C(C(=O)NCCCOC)N(CC(C)CN(C)C)C)ccc(-c2ccccc2)s1 C(C(=O)N=c1ccn(Cc2cccs2)[nH]1)c1cn(C)nn1 C1(C(=O)NCc2c(OCC#C)cccc2OC)CC(O)CC(C)(C)C1 c1(C(=O)NC(C)(C)CCCNC(=O)COCC2CC2)cc(F)cc2c1NCCC2 c1(CCN2CCN(C(c3n[nH]c(C4CC4)n3)=O)CC2)cc2ccncc2o1 N1(C(C2ON=C(C)C2C)=O)CC2CN(C(c3ccc4c(c3)OCO4)=O)CCC12 Cc1cc(C(N2CC3CC3(C(=O)NC(C)CC3CCOC3)C2)=O)c(C)n1C c1(N(CCC(=O)NCCNC(CCC)=O)C)nc2c(C(F)(F)F)cccc2s1 N1(C(=O)CC2CCCC2)CCC(C(=O)NCCc2ccccc2F)(CO)C1 N1(C(c2c[nH]c(=NC)s2)=O)CCN(C(=O)CC2CCCCC23CC3)CC1C1CC1 C(=O)(CCCN1CCOC1=O)N(C(CC(N)=O)c1cccnc1)C c1(CC(=O)NCC(C(=O)N2CC(OCC(N)=O)C2)N(C)C)cccnc1F n1(CC(N2CCC(C)(CNC(C3(C#C)CCC3)=O)C2)=O)cc([N+](=O)[O-])ccc1=O c1(C(=O)NC2C(c3ccc(C)cc3)C2)ccc(Br)cc1Cl c1(C(C)C)cccc(C(=O)N(CC(C)(C)NC(C2CC2c2cncnc2)=O)C)n1 CN1CCn2nc(C(N3CC4CCC3C(CNC(c3cnsn3)=O)C4)=O)cc2C1 c1(C(N2CC3(CN(C(C(C)CC(F)(F)F)=O)C3)C2)=O)cc(Cl)c2c(c1)OCCCO2 CCCC(C)(C)CC(=O)N1CCCC(CN(C(=O)COCc2nc[nH]n2)C)C1 c1(C(=O)NCC(C2CC2)NC(C(CN(C)C)N(C)C)=O)ccc(F)c(C(F)(F)F)n1 N(C)(S(=O)(=O)N1CCN(S(=O)(=O)CC2CN(CC(C)(C)C)C2)CC12CCC2)CC c1(C(=O)NCC2(C)N(C(C3C(C=C)OCC3)=O)CCC2)c(C)nn(C)c1Br C1(OC)CC(CCN(C(=O)Cc2ccc(C)cc2)CC)N(C(=O)CCC(C)OC)C1 c1(OCCC(=O)NC2C(NC(C3(C)CCCO3)=O)C2)ccc(S(N)(=O)=O)cc1 c1(C(=O)NCCN(c2nc(C3CC3)ncc2Br)CC)cc(C)nc(Cl)c1 Cn1cc(N2CCC(OCCCNC(=O)CCCOc3cccnc3)C2)cn1 C12(C(N3CC4C(NC(c5c(CC)cco5)=O)(C4)C3)=O)CC3CC(C(=O)N1)C2C3 C(=O)(N1CC(O)CO1)C1C(NC(=O)CC(C2CC2)C2CC2)OCC1 N1(C(c2c(C)nc(C)s2)=O)CC(C(N2CC3(C2)CN(C)C3)=O)OC(C)C1 C(c1cc(Br)cs1)=CC(=O)NCC1N(C(C(c2cccnc2)OC)=O)CC1 N1(C(CNC(CN(C)C(c2ncc[nH]c2=O)=O)=O)=O)CCCCCC1C(=O)N(C)C N12CCN(CC1)CC2.c12cc(cs1)C(=O)N2.C1(C2(C(C)(F)F)CC2)CSCCS1 N1(C(CCC)=O)CCCC(C2CC2C(C2(N3CCCC3)CC2)=O)C1 O=C1OC2CC(C(N3CCC(NC(=O)CCn4cc(Cl)cn4)C34CC4)=O)CC2O1 C1(C(=O)NC2C(CN(C)C)CCC2)CC2CCCC2N1C(c1ccc(O)c(F)c1)=O c1(OCC(=O)N(CCCNC(=O)CC(O)C2CCCC2)C)ccc(C(C)(C)C)cn1 Cc1nccc(C(=O)NCC(O)C(=O)N2CCC(c3cnn[nH]3)C2)n1 C1(OC)(CNC(C2CCCC2C)=O)CN(C(=O)CN(c2cncn2C)C)C1 c1(C(=O)NCC2CN(C(CCCCCC)=O)CC2(C)C)cc(C#N)c(F)cc1F C1(CC(=O)OC)CCCN1C(C1CC(C)N1C(=O)C(N1CCOCC1)C)=O O=C(C#CC1CCCOC1)N1CCCC(CCNC(C2(c3nccs3)CC2)=O)C1 Cn1cc2c(n1)CCCC2C(=O)NC1CC1NC(=O)CN1CC(=O)NC1=O N1(CCCC)CCCCC1C(=O)NC(c1nnc(C)s1)C(=O)OCC C(=O)(CCCCC(C)CC)N1C(CNC(CCCOCC)=O)C(C)CCC1 C1(CN(C(C2(C(=O)NC)CCC2)=O)C)CCCCN1C(c1sc(CO)nc1C)=O CN1C(C)(C)C(CNC(N2CC(CO)C2(C)C)=O)CS1(=O)=O CC(C)C#CC(=O)NCCC1CCN(C(=O)CCCONC(=O)OC(C)(C)C)C1 C(=O)(C(C(C)C)C(C)C)NCC(CCC)C(N1CC(C2CC2(F)F)C1)=O c1(SC)ccc(C)cc1C(=O)NCCC1CN(C(C)=O)C1 C1(NC(=O)CCCN2CCCCC2)CC2CC(NC(C3CC=CCO3)=O)CC12 c1(C(=O)OC)ccc(NC(C2CC2NC(c2ccccc2[N+](=O)[O-])=O)=O)cc1O C1(NC(CC=CC(C)(C)C)=O)C2CC3C1C3C2C(=O)NCc1nc(COC)n[nH]1 N1(CC(=O)NC2CC(CO)N(C(c3cnn[nH]3)=O)C2)C(=O)CCC1=O N1(C(C2(C)CCC(=O)N2)=O)C2CCC1CC(NC(c1ccc(Br)o1)=O)C2 C1(CNC(CSCCOC)=O)(NC(C2(n3ccnn3)CC2)=O)CCOC1 N1(C(c2c(CC)nns2)=O)CC2CCC(C1)C2NC(c1conc1CN(C)C)=O C1(C(=O)NC(c2nnc(O)o2)C)CN(C)CCN1C(c1ccncc1Cl)=O CCCC(CC(C)C)C(=O)NCc1ccsc1C(=O)NCC1(C)COCCO1 c1(C(=O)NCC2CC(NC(=O)C(F)CC3CC3)C2)ccc2ncncc2c1 c1(OC)cc([N+](=O)[O-])ccc1C(=O)NC(C)CNC(c1oc(C(F)F)cc1C)=O c1(CC)ccc(C(=O)NC2CN(C(C3CCC3OC)=O)C2)c(Cl)c1 C1(C(N(C2CCCC2(C)O)C)=O)COC2(C1)CN(C(C1CCCSC1)=O)C2 C(c1ccccc1)=C(CC)C(=O)NC1(C2CCCCN2C(c2c[nH][nH]c2=N)=O)CC1 Cn1cc2cc(-c3ncc(Cl)cc3C(=O)N(CCO)CC3CC3)ccc2n1 c1(C(=O)NCC(CCOC)NC(C2CCC(=O)NC2)=O)cccc2c(C)[nH]nc12 CN1CCCCCC1C(N1CCCC(CCC(=O)NC2(CO)CCSC2)C1)=O c1(CC(=O)NCC2CCC(F)(CNC(C3CN(C)C3)=O)C2)ccc2c(n1)CCC2 C1(C(N2CCCC(C(C)NC(C=C(C)C)=O)C2)=O)CC12CCOCC2 c1(C(=O)NC(CNC(C2(OC)CC2)=O)C)oc(C(C)C)nc1C c1(C(=O)NCC2C(NC(C3N(C)CCOC3)=O)CCC2)cc2sccc2s1 CCCC(C)(O)C(=O)NCC1CC(F)(CNC(=O)CN2CCCC2)C1 C(CCC(C)C(=O)N1C(C(N2CCC(C#N)CC2)=O)CCC1C1CC1)OC CC(C)C(N=[N+]=[N-])C(=O)N1CCC(C)(CC(=O)NC2(CF)CC2)C1 C12(CNC(C3(CC#C)CC3)=O)CN(C(=O)C(c3ccccc3F)C)CC(F)(C1)C2 c1(OC)ccc(C(=O)NC2CC(C(=O)N(C(C)CC)CCO)C2)cc1OC C(=O)(CCCCC(N)=O)NC(CC)CCC(=O)N(C1CC(C)(C)C1)C C1(NC(Cc2cccc(OC)c2)=O)CC12CCN(C(c1cc(Cl)ncc1N)=O)C2 c1(C(=O)NCC(Cn2cc(-c3cccc(C)c3)nn2)(C)C)ccc(O)cc1Cl C(=O)(CCCSC)N(C1CCN(C(C2(F)CC2)=O)C1)CC c1(C(N2CC(C)(c3cn(C4CCCC4)nn3)C2)=O)ccc2c(c1)CCC2 Cc1cc(N)c(C(N2CCCC(NC(C3C=CC=CC=C3)=O)C2)=O)cc1C c1(N(C)C)ccc(Br)c(C(=O)NC2(C)CCN(C(=O)Cc3nc[nH]n3)C2)c1 N1(C(C)=O)CC2(C1)OC1(CO)CC2(NC(=O)Cc2ccnc(F)c2F)C1 C#Cc1ccc(C(=O)NCC(C)CNC(=O)C(C)Cc2ccncc2)cc1 N1(C(CSC)=O)CC2COCCC2(NC(c2cc(NC(C)=O)ccc2Cl)=O)C1 C(N=c1[nH]c(N2CCCC(CCF)C2)nc2c1SCC2)c1cccc2c1scc2 C1(NC(C=Cc2nnc(C(C)C)o2)=O)CCCC12CN(C(=O)Cc1cscn1)C2 c1(NC(C(=O)NC(c2c(C)c(Cl)ccc2)C)=O)cc(F)c(F)cc1F c1(C(=O)NCCCN(C(C2(CS(C)(=O)=O)CC2)=O)C2CC2)ccc(S(C)(=O)=O)s1 N1(C(C(C)Cc2cnn(C)c2)=O)CC(NC(=O)C(C)(C)NS(C)(=O)=O)CCC1C C1(NC(C(C=CC)O)=O)CC2CCC1N(C(=O)CC1(CS(C)(=O)=O)CC1)C2 C(c1ccc(C)cc1)=CC(=O)NC1C(NC(c2c(CC)noc2C)=O)CC1 c1(NC(C)=O)ccc(C(N2CCC(NC(c3ccc(C)cc3C)=O)C2)=O)c(C)c1 C1(NC(CC=CCC)=O)CCCN(C(C2CCCCCN2C)=O)CC1 C1(C)(NC(c2ccc(CC(=O)OC)cc2)=O)CCCN(C(C2CC2CF)=O)C1 N1(C(C2(C(=O)OCC)CC2C)=O)CC(C2CCN(C(=O)CN(C3CCC3)C)CC2)C1 CC1OCCC1C(=O)NCC1CCN1Cc1ncsc1Br CC1(C(=O)NC2CC(CNC(C3CCCCC3(C)C)=O)C2)CCCC(F)(F)C1 C(=O)(CCCS(N)(=O)=O)NC1C(N2CCN(C(CC(C=C)CC)=O)CC2)COC1 CCC(CC)CC(=O)NCCCN(C(=O)C(C)n1cncn1)CCO C1(C=O)(C)CCC(F)(F)CC1.c1(OC2CN(C(C(C3CC3)OC)=O)C2)cncnc1 C1(C)(C(N(CCN(C(=O)C(c2ccccc2F)(C)F)C)C)=O)CCCCNC1=O C1(C(=O)NCCCCCNC(c2c(C)cnn2C)=O)CCn2c(O)nnc2C1 N1(C(C=CC=CCC)=O)CCCN(C(C23COC(CO)(C2)C3)=O)CC1 C1(NC(c2cccc(C)n2)=O)(CNC(=O)CSCc2ncc[nH]2)CCCCCC1 CC(C)(CCCC(=O)NC1CCC2CCC12)NC(c1nc(Cl)c[nH]1)=O c1(C(=O)NCC(CNC(C2N(C(C)=O)CCC2)=O)O)cc(Br)cn1C(C)C c1(C(=O)NC(CC)CNC(=O)C(C)(C)CSC)c(C)nn(CC)c1C(F)(F)F C(=O)(C1=NOC(CF)C1)NCC1CC(COC)CN1C(=O)CN1CCC(=O)CC1 n1(CCCSC)nnnc1C(c1ncsc1C)NCC1CC1(C)C c1(C(=O)NCCCCCCN(C)C(C2(F)CCCC2)=O)ncn2ccccc12 c1(C(=O)NC2C(NC(Cc3n(C(C)C)ncc3)=O)CCCC2)c(C#N)cnn1C Nc1cccc(F)c1C(=O)NC1COCC1NC(C1CC(F)C1)=O N1(C(C(CNC(C2(CC#C)CCCC2)=O)OC)=O)CCC2(CC1)CC2CSC C(C1CCN(C(=O)CC#N)CC1)=CC(N1C(CC)C(C)CC1)=O N1(C(CCC(=O)OCC)=O)CC(C(=O)NCC2CCC=CCC2)C2CCCCC12 C(=O)(C1=C(CC)OCCS1)NCCC(CNC(c1ccc(CC)cc1O)=O)(C)C n1(CCC(N2C(CN(c3nnc(CCOCC)s3)C)CCC2)=O)nc(C)cc1C C1(C(=O)NCC(C(C)C)NC(c2cc(CC)nnc2C)=O)CCCC2(CCC2)O1 C1(N2CCOCC2)(CC)CCN(CCCn2ccnc2)CC1 c1(CNC(CSCCNC(C(COC(C)=O)C)=O)=O)oc(C)nc1C C1(C2CCCC2)(C(N(c2ccsc2)OC2CCN(C(CCNC=O)=O)C2)=O)CCC1.N C1(C(=O)NC2C(NC(CNC(CCCCC)=O)=O)COC2)COC2COCC12 C(=O)(CC1C(=O)Nc2ccc(Cl)cc21)NCCNC(c1c(N)cc(Cl)c(Cl)c1)=O N1(C(C2(CC3CC3)CC2)=O)CC(CC(C)NC2CC(NC(C)=O)C2)C1 C(C(=C)CCNC(=O)COC(F)F)NC(C(Br)=CC)=O N1(CCCN2CCC(C(=O)OC)CC2)CCC(F)(C#N)CC1.CO c1(CC(=O)NC2CCC(CNCc3nccc(C#N)c3)C2)cnc2[nH]ccc2c1 C1(C(=O)NCC(C)CN(C(=O)C=CBr)C)OCC2CCCCC12 C12(C(=O)NC3CCC(CNC(c4nn(C)c(F)c4)=O)C3)CCC(CF)(C1)OC2 C1(CNC(=O)Cc2cnsc2)CN(C(c2cnc(C(F)(F)F)s2)=O)CC12CC2 Cc1ccc(C(=O)C=CC(=O)NCC2CC2NC(=O)CC2CCCOC2)cc1 c1(C(N(CCCNC(C2(C)CCCC2)=O)CCO)=O)ccnc2[nH]c(O)nc12 c1(OC)ccccc1C(=O)NCC1CCC(C(N2CCCCC2CO)=O)CC1 CCC(Cc1cccc(C)c1)C(=O)N1CCC(NC(=O)C(C)NC(=O)NC)C1C C1(C(=O)NC(C(=O)OCC)Cc2n[nH]c(CC)c2F)OCC2CCCCC12 N1(C(C(C)=C(C)C)=O)CCN(C(=O)CC2CCC(C)(C)O2)CC1c1ncc[nH]1 CC1CN(C(c2cnc(Cl)s2)=O)CCC1NCCNS(C)(=O)=O C(=O)(CC1CCC(=O)c2ccccc21)N1CCC(CCNC(=O)COCC2CC2)C1 C#CCC(C)(CC)C(=O)N1CCCC(CCC)(NC(=O)COC(F)(F)F)C1 N1(C(c2n(CC#C)cnn2)=O)CC(C(N2CCC2CC2CC2)=O)C2(CCC2)C1 Cc1ccc(C)c(S(=O)(=O)NC2CC(F)CN(S(=O)(=O)c3cccnc3)C2)c1 Cc1nc(C)c(CC(=O)NC(CNC(=O)C(c2ccc(F)cn2)(F)F)C(C)C)s1 N1(C(C(C=CC)O)=O)CC2CCC(C1)C(NC(C1Cc3cccc(C)c3O1)=O)C2 N1(C(Cc2cc(C)nn2C)=O)CCC(C(=O)NCCN(C)C(C)C)C12CCC2 C(=O)(C1=CCC(C)(C)CC1)N1CCC(CC(=O)N(C2CS(=O)(=O)C2)C)CC1 N1(C(c2cnncc2O)=O)CCC2CCC(C1)N2C(c1cc2nc[nH]c2cn1)=O C(=O)(CC(F)(F)c1ccccc1)NC(CC)CNC(c1ncncc1OC)=O c1(C(=O)NC2CN(C(CCC=C=C)=O)CC(C)C2)cccc2ncsc12 C1(NC(CCc2n(C)cnc2)=O)CN(C(c2nccnc2Br)=O)CC1F CS(=O)c1cccc(-c2cnc(C(=O)Nc3nccnc3Cl)cn2)c1 c1(C(N2C(CC)CN(C(C3CCSC3)=O)CC2)=O)cnc2c(F)ccc(F)c2c1 c1(C(=O)NC(C(C)NC(CC(CC)CC)=O)C)ccn2ccnc2n1 N1(C(c2cnc(C(C)(F)F)s2)=O)CCC2(C1)CN(C(C1CCC3C1C3(F)F)=O)C2 C1(CNC(Cc2c(C)cnn2C)=O)CC(C(=O)N2CCNC(=O)C2C)=NO1 c1(-c2cn(CCCC(=O)NCc3ccc(C4CC4)s3)nn2)ccc(F)cn1 c1(C(N2C(C(=O)Nc3cncc(CO)c3)CC2)=O)cc(F)c(F)cc1F c1(C(=O)Nc2c(C)nccc2)cnn2c1CN(C(=O)CCc1cncnc1)CC2 c1(C(=O)NCC2(NC(CC3(C)CC3)=O)CCC2)ccc(F)c(C2CC2)c1 C1(C(NOc2c(OC)cc(F)cc2)=O)CN(C(=O)C(C)CCN(C)C)C2(CCC2)C1 N1(C(c2ccncn2)=O)CC2CCN(Cc3cc(Br)co3)C2C1 c1(OC)ccc2[nH]cc(C(=O)NCCCNC(c3ncnc(C)c3C)=O)c2c1 O=C1NC(=O)C2(CCN(C(=O)N(C(CC3CC3)CO)c3ccco3)C2)N1 N1(C(C2=C(C)CC2)=O)CCN(C(=O)CN(C)C(N)=O)CC1c1nccn1C CCCC(C(=O)OC)C(=O)NCC(F)(C(=O)NCCn1ncnn1)C(C)C N1(CCC)C(=O)CCC1C(=O)NCC(C)NC(=O)C(CO)NC(=O)C(F)(F)F C#CC1(C(N2CCCC(CC(=O)NC3CC3)C2)=O)CCCCC1 c1(C(=O)NCC(C)(C2CC2)NC(CC(CC)SC)=O)cc2n(n1)CCCCC2=O c1(SCC#C)cccc(C(=O)N(C)C(C2CC2COC)=O)c1 C(=O)(C(C1CC1)NC(=O)Cc1cnoc1)NCCN(CCC)CCC c1(C(=O)NC(CN(C)C)CCO)ccc2c(n1)CN(C(C1(O)CC1)=O)CC2 C(=O)(CC(C)(C)C(F)(F)F)N1C(N(C(c2ccn(CCOC)n2)=O)C2CC2)CCC1 c1(C(=O)NC)cc([N+](=O)[O-])ccc1N(CC(C)NC(=O)C(c1ccccc1)C)C Cn1nccc1C1=CC2CCC(C1)N2C(C1CCCC(C(F)(F)F)C1)=O C1(CC)CN(C(c2cnc(C)nc2C)=O)CCN1C(C1CC1c1cccs1)=O N1(C(C(CCNC(C2(CCC)CC(=O)C2)=O)OC)=O)CCN2CCC1CC2 c1(CC)ncc(C(=O)NCCC2(C(N3CC(O)(C(C)C)C3)=O)CC2)cn1 c1(CCC)cccc(NC(C2CCCC2CNC(=O)Cn2ccc(C)c2)=O)c1 C(C(CC(F)(F)F)NC(=O)CSc1nnnn1C)N(C(C=CC(=O)N(C)C)=O)CC C=Cc1cncc(C(=O)NC(CNC(=O)CCc2ncccn2)C(C)(C)C)c1 N1(C(C(c2cc(C)sc2)(F)F)=O)CCN(C(c2cnc[nH]2)=O)C(CCO)C1 C1(C(N2C(C(C)C)C(NC(=O)CC3(C)CCOCC3)CC2)=O)COC2(CCC2)C1 c1(C(=O)NC2CN(C(Cc3c(C)con3)=O)C(C)C2)cc(S(N)(=O)=O)n(C)c1 C1(C(N(CCNC(c2cncc(C(F)F)c2)=O)CC)=O)CC12CCCOC2 C1(NC(c2c(OC)cccn2)=O)COC2C(NC(c3n[nH]c(C)c3F)=O)COC12 C1(NC(=O)C(C2CC2)CNC(C2CC(C3CCOCC3)C2)=O)CCCN1C1CC1 Cc1oc(C(=O)NC(C)CCN(C)C(C2CN3CCC2CC3)=O)cc1S(N)(=O)=O c1(NC(c2ncccc2O)C)nccnc1-c1ccco1 CCC(C)C(C(=O)NC1CCC(C(=O)N(CC(C2CCCC2)O)C)CC1)OC C1(CC(=O)NC(C2C(C)CCN2C(=O)CC2(C)CCOC2)C)CCC(=O)C1C n1(CC#C)cc(CNC(c2cncnc2C(C)C)=O)c2ccccc12 CC1CCC(NC(=O)NC2CCC(CO)CC2)(CNC(=O)OC(C)(C)C)CC1 CC(=O)CCC(=O)NCc1nocc1C(=O)NCCC1CCCN1C C(C)(C)(CC(=O)NC1CN(C)CC1C)N(C(C=CC(C)C)=O)C CCCC(C)(O)C(=O)NCCN(C(=O)C(C)Oc1ccc(F)nc1)CCOC C(c1ccco1)=C(C)C(=O)NC(CC(=O)NCC(C)C(C)C)C1CC1 C=CCC(CC(C)C)C(=O)NCc1ccccc1-n1cc(C2CC2OC)nn1 C1(=O)C(C(C)C)CN1.C1(C(=O)NCCCNC(=O)NC)CCCO1 n12nnnc1C(C1(F)CC(CO)C1)NCC2.C1(COCC)CC(F)(F)C1 C(=O)(C(CO)C(C)(C)C)N1C(C(C)NC(Cn2c(C)ncc2)=O)CCC1 CC(CCC(=O)N1CCC(CCC(=O)N(C)Cc2nnc(O)o2)CC1)N(C)C C(=O)(CCCCCF)NC(CC(N1CCN(C(C)C)CC1=O)=O)C(F)F c1(C(N(CC(=O)C(C)(C)C)C)=O)ccc(O)c2ccccc12 Cn1ccnc1NCC(=O)NCCCOCCNC(=O)CCN1CCCC1 C(=O)(CC(C)(C)C(=O)NCC(O)CN(C)C(c1nc(C)n(C)n1)=O)OCC c1(OC)c(C)csc1C(N1CCSCC1CCNC(C1(SC)CCC1)=O)=O CCC(C#N)(CC)C(=O)NC1CCC(CCNC(c2ccc(C)c(C)c2)=O)C1 C1(OC)CC2CC1CN(C(=O)CC(C)(C)CNC(C1CCCC(C)(C)C1)=O)C2 C1(C(=O)NC2C(NC(CC3CC(=O)C3)=O)CCOC2)Cc2ccccc2C(=O)O1 C1(C(=O)NCC(C)(C)NC(c2c(COC)noc2)=O)CN2CCCN1CC2 C1(COC)(CNC(=O)C(C)(C)n2cc(CO)nn2)CCCN1c1cc(F)ncn1 C1(C(N(CCCCC)CC#C)=O)(C(C)C)CCN(C(=O)CCC=C(C)C)C1 Cc1cccc(CC(N2CCC(F)(CNC(c3cnc(C)c(C)c3)=O)C2)=O)c1F c1(C(=O)NC2(CNC(C3C(C)C3)=O)CCCC2)ccc2[nH]ccc2c1F c1(C(CNC(=O)NC(c2nnnn2C)C)(OC)OC)cc(F)c(Cl)cc1F CCCCCC(C)NC(C1CC(C)CN1C(c1nc(C)oc1C)=O)=O Cc1nn(C)c(C)c1OCC(=O)NC(CNC(=O)C=C1CCOCC1)CO N1(C(C)=O)CCC2C1CCCN2C(=O)CC1CCCCC1S(C)(=O)=O C1(CC(N2CCC(NC(CN(C(C)=O)C)=O)(CO)C2)=O)CCCC(C)(C)O1 CC(C)(C(=O)NC1CCN(C(c2ocnc2C2CCC2)=O)C1)c1ccccc1 CC(C)CC(C(=O)NCC(F)CNC(c1cc[nH]n1)=O)N(C)C(=O)OC(C)(C)C c1(C(=O)NCC2CCCN(C(C=CSC)=O)C2)[nH]nc2ncc(Br)cc12 c1(OC)cccc(S(=O)(=O)CC(=O)NC2CCOCC2NC(c2cnsc2)=O)c1 c1(C(N2CCC(C(C(=O)NCc3n(CC)cnn3)C)C2)=O)ccncc1N C(=O)(C(C(C)C1CCCC1)N1CCOC(C(C)(C)O)C1)NC(C)C c1(C(CC)NC(=O)NC(c2nc[nH]n2)C)ccc(Cl)s1 C1(C(=O)NCC2CCC(C)N(C(=O)CC3(C)CCOC3)C2)CN2CCCN1CC2 C1(COC)CC(CNC(=O)COC2CCC2)N(C(=O)C=Cc2ccoc2)C1 c1(CCC(c2n(CC)nnn2)(C)NC(C)CCSC)ccccc1F c1(C(=O)NC(CCCNC(CCC(C)OCC)=O)C)ccn2c1CCCC2 c1(CSCC(=O)NC2CCN(C(C3CC(O)(C(F)F)C3)=O)C2)ccc(F)cc1 C(C)(C(C)(C)C(=O)N=CC(=O)N(C1CCC1)C)NC(C=CC(CC)C)=O C1(NC(COC(CC)CC)=O)CCC12CN(C(=O)COC(C)=O)C2 C(CC(=O)N1CC(CCN(CCO)C)C1)N(C(=O)COC(CC)CC)CC#C.CC C(C(=O)N(CCC(C(C)C)NC(=O)C1=CCOC1)C)(C(C)C)(C(C)C)NC(C)=O N(C1CN(C(=O)C=CCN(C)CC)Cc2ccccc21)C(C1(C=C)CCC1)=O C(=O)(CC(O)c1cc(C)cs1)NCCCN(C(C(C)OC)=O)C Cc1nc(C(C)(C)C)sc1C(N1CCC(C(C)NC(C2CNC(=O)C2)=O)CC1)=O N1(C(=O)OC(C)(C)C)CCN(C(=O)CCNC(=O)NC2CCC2)C2CCC12 Nc1ccc2c(c1)CCC2NC(=O)NC(c1cccc(Cl)c1)C1CC1 c1(CN(C)C)ccc(CN=C(NCc2ccnn2C)NC2CCCC2(F)F)cc1 c1(COC(C(N2CCCC(O)C2)C)=O)ccc(C#N)cc1 C(C(C)C(F)F)NC(C(C1CN(C(CC=CCC)=O)C1)OC)=O Cc1ccc(CC(=O)NCCN(C(=O)CCn2cnnn2)CC2CC2)c(C)c1 c1(C(N2CCC(CCNC(C(CC)c3ccccc3)=O)C2)=O)sc(SC)nc1C N1(C(C(CC=C)OC)=O)CCOCC(CNC(C2(C)CCN(C)C2=O)=O)C1 C(CCCCC(=O)N1CCCC2(CNC(=O)CNS(C)(=O)=O)CC12)=CC c1(N2CCSCC(C)C2)nc(N2CCC3(C2)CN(C)C3)nc2ccsc12 Cc1cc(C(=O)NC2(C(=O)NC3CCCC3CN(C)C)CCOC2)c(C)cn1 c1(N2C(C)CC(CNC(C3COCCN3C)=O)C2)ccc2nnnn2n1 C1(CNC(C(COC)NC(C)=O)=O)CCC(NC(c2cn(CCF)nn2)=O)C1 c1(C(N(CCN(C(c2sc(C)nc2C)=O)CC)CC)=O)cc2c(ccn2C)s1 c1(OC)ccc(CC(=O)NCC2(F)CN(C(C3C(Cl)(Cl)C34CC4)=O)C2)c(F)c1 c1(C(N2CC(COC)(CNC(c3ccccc3C)=O)C2)=O)cccc2c1COC2 CC1CN(c2ccc(C(=O)NC3CC3c3ccc(F)cc3F)cc2)CC(C)O1 C(CC1(C#N)CCC1)(C(=O)NCCSC)NC(C=C)C1CC1 C(CC(=O)NC1CC(OC)(OC)C1)(CC(C)C)NC(C1(C)NC(=O)NC1=O)=O c1(CNCC(c2scc(C)n2)C)cc(C#N)n(C)n1.N12CCC(CC1)OC2=O C=C=C(C)CC(=O)NCC1(NC(=O)C(c2ccccc2Cl)O)CCC1 Cc1ccc(C(N2CCC(NC(C3CCCO3)=O)C23CC3)=O)cc1Cl c1(C(C(=O)NCC(O)C2CC2)NC(c2ccc(Cl)o2)=O)cccnc1 C(=O)(C(CC(C)C)N(C(=O)CC(C)(C)C=C)C)NC1(CC#C)CC1 C1(N(C=O)CC)CCCN(C(=O)NCCCC2CCCN2CCOC)C1.OC c1(C(=O)NC2(C)CN(C(C(C(C)C)SC)=O)C2)cnn2c(=O)cc[nH]c12 CCCCC(C(=O)NC)NC(C1CCCN(C(=O)CC2CCCCO2)C1)=O N1(C(Cc2c(C)occ2)=O)CC2COCC2(C(N2CCOCC(C)C2)=O)C1 N1(C(CCCC(=C)C)=O)CCN(C(=O)C#CC2CC2)CC(O)C1 C#Cc1cc(C(N2CCC(CC)C2C(=O)N(C2(CC)CC2)C)=O)ccc1C C(=O)(CC(C)(C)C)OC.C12CCN(CC1)Cc1[nH]cc(c1)C(=O)N2CC#C N1(C(C2C(C(N)=O)COC2)=O)CCC(C(=O)NC2CCCN(C)C2)(CF)C1 C(=O)(CCCC(C)(C)NC(=O)CN1CCOCC1)N1CC(C)(F)C1 C1(CCNC(c2ccc(-c3cnn(C)c3)o2)=O)(NC(C(C)OC)=O)CCCC1 c1(SCC)nnc2ncnn2c1NCC(C)(C(C)C)NC(=O)C(C1CCC1)OC CC1C(C(=O)NCC2(CC3CC3)CC2)CCCN1C(C1CC2(CC2)CO1)=O CC(C)CC(CNC(=O)C(C(C)C)NS(C)(=O)=O)NC(=O)CC(C)(F)F C(=O)(C(F)(F)CCn1cc(CN2CCCC2)nn1)N(CC)CC12CC(C1)C(C)O2 c1(C(=O)NCCCCNC(c2c(C)nc[nH]2)=O)ccc(N2CCOCC2)cc1C c1(C(=O)NC(CC)CNC(=O)C(C)OC2CCCC2)cnn(CCF)c1 Cc1cnc(C)c(C(N2CC(NC(C3CN(C(N)=O)C3)=O)CC2CO)=O)c1 CC1CCC(C(=O)NCC=CC(=O)NC(c2cncs2)C)O1 N1(C(C(C)NC=O)=O)CCC(n2cc(NC(c3ccnc(Br)c3)=O)cn2)CC1 C=CCCCCCC(=O)NCCCc1ccn(C)n1.C12(CC)CN(C1)C2=O CC1CN(C(c2cn(C(F)F)cn2)=O)CC1NC(=O)C=Cc1ccco1 c1(C(C)C)ccc(C(=O)NC2CC2NC(=O)C(O)Cc2ccccn2)cc1Cl c1(OC)ccc(C(=O)CCC(=O)OCCC2CCCC(O)C2)cc1 c1(N(C2CC(c3cccc(C(F)(F)F)c3)C2)C(=O)CO)ncnc2c1CCS2 c1(CCC(N2CCCC(N(C(C3C(C(C)C)C3)=O)CCO)C2)=O)ccc(Cl)c(F)c1 N1(Cc2cnc(CC)s2)CCCCC1NC(=O)Nc1ccc(F)cn1 CC1(C(=O)NC2CCC(CNC(C3C=CCC3)=O)C2)CC2(C1)CC(F)(F)C2 C(CCCCC(=O)NC(C(N1CC2(C1)CC2(F)F)=O)C1CCOC1)N(C)C N1(C(C(CCC)N(C)C)=O)CCC(C)(C)C1CC(=O)NC1CC1C1CCC1 c1(C(=O)NCCC2(NC(C(OC)OC)=O)CC2)ccncc1NC(C)=O N1(C(c2cc(CC)on2)=O)CC2(CCN(C(C3CCOC3(C)C)=O)C2)C1C(C)C C(C(C)(CC(C)C)NC(=O)CC1CCCC1)NC(C1(C(=O)OCC)CC1C)=O C(=O)(Nn1cnc2ccccc2c1=O)c1c(CN)cn(C)n1 C1(NC(C(F)OC)=O)CC(O)CN(C(=O)Cc2scnc2-c2cccs2)C1 c1(C(N2CC(CN(C)C(C3CCC(C)(C)O3)=O)OCC2)=O)cnc2c(c1)CCOC2 C(N=c1ccn(CCO)[nH]1)(c1c(Br)c(C)nn1C)c1n(CCOC)nnn1 N1(C(c2n(C)c(S)nn2)=O)CCC(NC(=O)CC2(C3CC3)CC2)C(CO)C1 c1(C(N2CC=CC(NC(C(C)NC(C)=O)=O)C2)=O)ccn2cc(C(F)(F)F)nc2c1 CCCCN(OC)C(=O)C1CCCCCC1Nc1ccc(Cl)cc1 c1(C(=O)NC(CNC(COCCC=C)=O)CCOC)ccc2c(c1)C1CCC2O1 C1(NC(C2CN(CCN(CC)CC)C2)=O)C2CC3C(C2)C13 N1(C(C2C(OC)CN(CC)C2)=O)CCN(C(=O)Cn2cncn2)CC1C1CC1 C(=O)(CCCCCF)N1CCCC(NC(C(C)OCC2CC2)=O)C1 C(C#C)(CCC)N(C(CCC1(NC(C(C)OCCC#C)=O)CCC1)=O)CC C(=O)(C1=CC2CCC(C1)C2)NC(CNC(CC(CCC)C)=O)C1CCC1 c1(C(=O)NCCNC(C(CCSC)O)=O)cnc(NC2CC2)c(Cl)c1 c1(SCC(=O)NCC(CCOC)NC(=O)CCn2ccnc2)ccccc1F C1(NC(c2cn(C)nc2Br)=O)CCN(C(=O)C(O)C2CCCC2)CC1(C)C c1(C(=O)NC(C)C(C)NC(=O)CC23CCC(CC2)CC3)cnn2cccnc12 C1(C(N2CCCC(C(C)C)C2)=O)CC12CCN(CCOC(C)(C)C)CC2 C1(CC=C)(NC(c2nccc(SC)n2)=O)CCN(C(c2nc(CO)oc2C)=O)C1 c1(NC(C2C=CCN2C(c2cccc(-n3ccnc3)c2)=O)=O)cc(F)cnc1Cl C(CCC(O)C(=O)N1CCCC(F)(CO)C1)NC(C(COC)COC)=O C(C(C)(CC(C)C)NC(=O)C(C)Oc1ccccc1F)NC(c1c(C)onc1)=O CC(C)C1=NOC(C(=O)NCC2CCN(C(=O)CC(=O)OCCC(C)C)CC2)C1 N1(C(C(C2CCC(=O)N2)C)=O)CCC(C(=O)NCCC2CCCCC2)(CF)C1 C1(C(N2CC3(CC(NC(C(CN(C)C)O)=O)C3)C2)=O)CCc2nncn2CC1 c1(C(=O)NCCOC2CN(c3snc(C(=O)OC)n3)C2)cc2cnc(Cl)cc2s1 c1(C(N(CCC)CCNC(=O)CC2CCC(O)C2)=O)ccc(OC(C)C)cn1 C1(C(=O)NC(CNC(Cn2ncc(C)c2)=O)C)CN(C)CC(C)O1 CCCC(O)(CCC)CC(=O)NCCCCC(C)NC(=O)C(C)=CC CC1(C)CCC(O)(C(=O)NCCC2CCN(C(=O)CN3CC4CCC3C4)C2)CC1 c1(NC(N2C(C)(C)CC(C)(CO)C2)=O)cncc2ccc(F)cc12 C1(C(N2C(C(CNC(c3onc(C)n3)=O)(C)C)CCC2)=O)CC(=O)NC1(C)C Cc1cccc(C2(C(=O)N(CCO)Cc3cn(C(F)(F)C(F)(F)F)nn3)CC2)c1 c1(C(CC)C)nccc(N(C2CC23CC(NC(c2ccc(COC)o2)=O)C3)C)n1 c1(C(=O)NCC(c2ccccc2F)(F)F)cc2cc(Br)cnc2o1 c1(C(=O)NCC(C)(CNC(=O)Cc2csc(C)n2)OC)cc(C#N)ccc1C n1(CC)c(C(=O)NC2CC(O)C2CC(=O)NC2CC(=O)N(O)C2)cnc1O CC1(F)CCCCN(c2ncnc(SC3CC34CCOCCC4)c2C(N)=O)C1 c1(C2(C(=O)NCC3(CNC(C4(F)CC4)=O)CC3)CCC2)c(F)cccc1F c1(NC(C(c2cccc(Cl)c2)C)=O)cccc(C(=O)NCC2CCCO2)c1 C(=O)(C1=C(F)CN(C(c2csc(CO)n2)=O)CC1)Nc1c(C)ccc(C)c1 C#CC(CC(C)(C)C)NC(C1(C)CCN(C(c2cc(C)ncc2C)=O)C1)=O c1(OC)c(CN2CCCC2C(=O)NCc2cccc(OC)c2Br)ccc(F)c1F N1(C(c2cc(-c3cn(C)nc3)[nH]n2)=O)CC2CC2(NC(=O)CSC(F)F)C1 c1(NC(C2CCN(CCc3ccc(CO)cc3)CC2)=O)cccc(C(F)F)c1Cl C(=O)(C1CCc2cc(Cl)ccc21)N(C1CCN(C(=O)CSSC)CC1)CC#C C1(C(N(CCC)C(C)C)=O)CCCCC1NC(=O)CC1OCCO1 CCC(C)CC(=O)N1CCC(OCCCNC(C2(C3CCCO3)CC2)=O)CC1 CC1(C(=O)NC23CC(NC(C4C=CCCC4)=O)(C2)C3)CNC(=O)C1 CCC(C#N)(CC)C(=O)N1CC(NC(c2ccc(-c3cccs3)o2)=O)CC(O)C1 C1(c2n(-c3c(CC)cccc3)nnn2)(NC(C2CSC2)C)CC2(C1)CC(C)(C#N)C2 C1(OCCNC(COCCCC)=O)CCN(C(c2cnc(SC)s2)=O)C1 O=C(CC(c1ccon1)C1CC1)NCCc1cccnc1 c1(CNC(CC2(CCC(=O)N(C)CCN(C)C)CCC2)=O)cnc(C2CC2)s1 O=C(C1CCCn2cnnc21)NCCC1CCCN(C(=O)Cc2cccs2)C1 c1(C(N(CC(CC)NC(=O)C(C)(O)COC)C)=O)cc(Br)cc(Cl)c1C C=Cn1nncc1C(N1CCCC(CNC(=O)C(C2CCCCC2)F)C1)=O C1(C)(C(=O)OC)CN(C(C2C=CCN2C(=O)C(O)C2CC2)=O)C1 CCCC(C)CC(C(=O)Nc1ccc(F)cc1)N1CC(OC)C(CCC(=O)O)C1 c1(C(=O)OC)cc(Br)ccc1NC(C1C=CC(NC(=O)CN(C)C(C)C)C1)=O N1(C(c2cc3n(c2)CCOC3)=O)CCC2OCCN(C(=O)Cc3cn[nH]c3)C2C1 C=C1CCN(C(=O)C(C#N)C(C)C)C(C(=O)NC2CC(C(=O)NC)C2(C)C)C1 C1(C)(OC2CN(C(CNC(C(CC)C)=O)=O)C2)CCN(C(C2CCNC2=O)=O)C1 c1(C(=O)NCCC(CNC(c2c(CC)[nH]cc2)=O)O)cnc(C(N)=O)cn1 N1(CC)C(=O)CCC1CC(N1CCC(CF)(NC(=O)COc2ccon2)C1)=O C1(C(=O)NCC(CC(C)C)NC(c2ccc(C(C)C)o2)=O)CC2CCCC(C1)C2 N(C1COCc2ccccc21)C(=O)Cn1cc(-c2ccnc(C(F)(F)F)c2)nn1 c1(C(=O)NC2CN(C(CCCC)=O)CC(O)C2)sc2ncccc2c1N c1(OCC(=O)N(CCC(C)S(C)=O)C)ccc(Cl)cc1F c1(C(=O)NC(CC)CNC(=O)C(F)OCCCC(C)C)ccccc1C Cc1cc(=NCC2OCCc3ccccc32)[nH]c(N2CC3CCC(C2)C3O)n1 N1(C(C(C)NC(=O)OC)=O)CCN(C(=O)C=Cc2ccc(C)s2)C2(CCC2)C1 c1(C(N2CC(CC)N(C(=O)CC3CCOC3=O)CC2)=O)cnc2c(c1)COC2 c1(C(=O)NCCN(C(=O)CC2COCC2O)CCOC)cnc2c(c1)CCCO2 N1(C(C)=O)CCc2ccccc2C1CC(=O)Nc1cc2ccsc2c(O)n1 c1(C(=O)NCC2C(NC(CC(=C)Br)=O)C2)cc(F)c(N)cc1F N1(C(C2C3C(=O)C4C(C3)C42)=O)CCN(C(c2ccc(O)nn2)=O)CC(O)C1 N1(C(CC(CC)C)=O)CC2(CC2)CC1CC(=O)NCC1CCN(C(N)=O)C1 C(CC1=CCN(C(C2CCN2C(C)(C)C)=O)CC1)NC(C(C=C)(C)CC)=O C(N=c1[nH]c(=NCCCC2CC3CCC2C3)c2sccc2[nH]1)c1cn(C)cn1 N1(Cc2nc(CCC)sc2)CCC(NC(=O)CC(F)(F)F)C(F)C1 c1(OC)ccc(Cl)c(C(=O)NC2C3CN(C(c4nc[nH]c4C(C)(C)C)=O)CC23)c1Cl CCC(CC(=O)N1CC(F)CC1CC(=O)NCCC[Si](C)(C)C)C(C)(C)C N1(C(CSCC)=O)CCC(C(F)(F)F)C(CNC(=O)CCCOCC)C1 c1(-n2cc(CC(CC)CN(C)C)nn2)ccc(C)c(OC(C)(C)C)c1 C12CCC(O1)NC2=O.C1(CNC(CCC2(C)CC2)=O)(CF)CC1(F)F N1(C(CC(C)OC)=O)CC2CC1CN2C(C12CC(CO1)C2)=O CC(=Cn1ccnn1)C(=O)N1CCC1CNC(=O)CCSc1nnnn1C C(=O)(C1CNC(=O)c2ccccc21)NC1CC(CNC(CCCC#C)=O)CC1O C1(C)(C(N(CCCC(=O)NCC(C(C)C)OCC)C)=O)CC=CCC1 N1(C(CN(C(C(CC)OCC)=O)CCN(C)C(C)=O)=O)CCOC(CC)C1 c1(C(N2C(CNC(CC(=C)C)=O)C(CC)CC2)=O)ccc(=O)n(C)n1 C1(C(=O)NC(C#C)C)CC=CCN1C(=O)CCNC(N)=O c1(CC)c(C(=O)NCCOC2CN(C(=O)C(F)=CC3CC3)C2)cnn1C C1(O)(CNC(C(C)c2ccco2)=O)CCN(C(=O)Cn2ccnn2)C1 N1(C(C2(C=C)CCC2)=O)CC(NC(=O)C(C)N(C)C)C(c2nccn2C)C1 C1(N)(C(N(C)CCc2cnccn2)=O)CCCCC1 C1(CNC(=O)C=CC2CCC2)CN(C(C2CCn3nncc3C2)=O)CC12CCC2 Cc1c(C(=O)NCC2CC2CNC(c2cnncc2C)=O)cccc1Br N1(C(c2n(CC)nnc2)=O)CCCC2CN(C(=O)CC3CCOC3)CCC12 c1(CC)ccc(F)cc1NC(C1CCN(C(=O)C(Br)=C(C)C)C1)=O C=C1CC(C)(C(=O)NCCC(=O)OC(C)(C)C)C1.C1(=O)C(Cc2ccc[nH]2)N1 C1(COC)CCCCCC1.c12cnn(c1)CCn1cc(nn1)C1CCN(C1)C2=O Cc1cc2cc(c1)CNC2=O.C1(C(N)=O)CN(C)CCN1C(=O)C(C)CC1CC1 CC1(C)CN(C(c2ccccc2SC2CCC2)=O)CC1NC(c1ccncc1)=O c1(C(=O)NCC2CC(CNC(C3(C)C=CCC3)=O)C2)cnn2ncccc12 c1(C(C(=O)NC2C3CN(C(C(C(C)C)C)=O)CC32)(F)F)ccc(Cl)c(Cl)c1 C1(c2n(CC)cnn2)CN(C(c2cnc(C)o2)=O)CCO1 O=C(CCC(=O)N1CCCC1)NCC1CC(F)CN1C(c1cnc(O)s1)=O N1(C(C(CCC)C)=O)CCN(C(C2CCCCN2C(C)=O)=O)C(C)C1 c1(NC(CCCC=C)C)cc(C)c(S(=O)(=O)NC2CCN(CCC)CC2)cn1 C(CCC(O)C(=O)NC1CCC1(C)C)NC(c1n(CC)ncc1)=O c1(C(N2CC(C(=O)OC)NC(=O)C2)C(=O)NCCCC2CC2)c(Cl)cc(Br)cc1Cl C(=O)(C1c2ccccc2OCC1(C)C)NC(CC)CNC(C1CC1CC(C)C)=O c1(C(=O)NC2CCN(C(C3C(C(=O)OC)C3)=O)CC2)cc2ccccc2cc1Cl CC1C(NC(C2CC2C#N)=O)CCCN1C(=O)Cc1cc(-c2ccccc2)n[nH]1 C12(CNC(=O)CCCF)CCCCC1N(C(=O)CCn1cccnc1=O)CCC2 N1(C(CC2CC(OC)C2)=O)CC=CCC1C(=O)NCCC1CCCC2CC12 c1(C(=O)NC2CC(C)N(C(=O)CC3CS(=O)(=O)C3)C2)cnc(F)c(Cl)c1 C1(CCC)CN(C(=O)COCC)CC1C(=O)N(CCCO)C C(=O)(CCCCCCNC(C1(C)CCN1C(=O)COC(=O)NC(C)=O)=O)OC C(c1cccc(Br)c1)=CC(=O)NCC#CCNC(=O)COCC1(F)CC1 CCCCCC(F)C(=O)N1CCC(C)(CCNC(=O)COC(C)CC)C1 C(CC(C(=O)NCCCCCCO)NC(=O)CC1C=CCC1)SC N1(C(C2(C(C)(F)F)CCC2)=O)CCC(N(C(=O)CSS(C)(=O)=O)CCO)C(C)C1 c1(N(C)C)cc(C(N2CCCN(C(=O)CC3(C)CC3F)CC2)=O)cc(Cl)n1 C1(C(=O)NCC(C=C)(C)C)CCN(C(=O)C2C3CCC(F)(F)C23)O1 c1(C(N(CC(C)(C)NC(C2CCCO2)=O)C)=O)cc(C(=O)NC2CC2)n(C)n1 N1(C(c2ncc(OC)nc2)=O)CC(NC(C2CCCC(=O)N2)=O)CCC1C Cc1c(Br)cccc1S(=O)(=O)N1CCCC(CN2C(=O)CNC2=O)C1 C1(CNC(C2CC(SC)C2)=O)CC(C)N(C(C2CC2(C)C(C)C)=O)C1 S(=O)(=O)(c1ccc(=NCCCSC(F)(F)F)[nH]c1)NCC1CC(C)(C)OC1(C)C N1(c2c(C)cnc(Cl)n2)CCC2(CCOC2)C(NC(=O)CCC(C)N(C)C)C1 C1(NC(Cc2cn(CC)nn2)=O)C2CC(O)C(C2)N1C(c1cnnn1C(C)C)=O C(=O)(C(C)(C)CCCNC(=O)C=CC(F)(F)F)NC1CCC(CCCC)C1 CC1CC(NC(=O)CC2(O)CCN(C)CC2)CCN1C(=O)C1=COCCO1 Cc1ccc(F)c2c1CCN(c1nc3c(c(=NCC4(CCO)CC4)[nH]1)COC3)C2 CC1CN(C(=O)CC(C)C(F)(F)F)CC(C)N(C(=O)CCCN(C)C)C1 c1(CNCC2N(C(c3cc4ccccc4o3)=O)CCC2)noc2c1CCCCC2 CC1(CC(=O)NCC2(C3CC3)CCCO2)CCN(C(c2ccc(F)s2)=O)C1 c1(NC)cccc(C(N2CCCC(CC(=O)NC(C3CC4CCC3C4)C)C2)=O)n1 c1(C(=O)OC)cc(Br)c(CC(N2CC(CO)(NC(=O)C=C(C)Cl)C2)=O)cc1OC C(CC(=O)NCCCCC1CCN(C(C2CCN(C)C2)=O)CC1)(C(N)=O)NC(C)=O C(CCCCC(=O)NCC1C=CC(NC(C2CCCCCN2C)=O)C1)OC Cc1ncnc(O)c1C(=O)NC(CNC(c1ccc(C#N)cc1)=O)CO c1(NC2(CC=C)CCCN(c3nnnn3C)C2)ccc2c(c1)NC(=O)C2(C)C n1(CC)nnc2cc(C(N3CCCC(NC(C4CC5(CC5)C4)=O)CC3)=O)ccc12 c1(OC)cnc(C(=O)N(CC(CO)(CO)NC(c2ccc(C)o2)=O)C)c(F)c1 c1(C(N2CCCC2c2noc(C)n2)C(=O)NCC=C)noc2ccc(F)cc12 c1(C(=O)NC2(CO)CN(C(c3cc(C)nnc3)=O)C2)cc(Cl)c(Cl)n1C Cc1c(Br)c(C(=O)N(CCCNC(=O)CC2(C)CC2F)C)nn1C c1(C(N(C2CCN(C(C3CCOCC3)=O)CC2)CC(C)C)=O)cnn2ccsc12 C(=O)(C(CC)C(=O)N1CCCCC1CNC(c1cnn(C(C)C)c1F)=O)OCC c1(C(=O)NC2CCN(C(C34CC3CCC4(F)F)=O)C2)c(Cl)cccc1Cl N1(C(=O)C=Cc2ccoc2)CCN(C(=O)CCCF)CC1CO c1(C(=O)NC2(CN(C(=O)CC3CC(O)C34CCC4)C)CC2)cccc([N+](=O)[O-])c1O O(NC(=O)C1=C(F)CN(C(c2cn(C)ccc2=O)=O)CC1)CC(C(C)C)O c1(C(=O)NC(C)C(C)(C)NC(=O)CCN2CCC2)cc2ncn(C)c2cn1 N1(C(C(CC=C)c2ccccc2)=O)CCC(NC(=O)CC(C)(C)O)C(C)C1 CC1(C(=O)NC2CC3(CCC3)C2)CC(O)CN1C(c1ccc(F)s1)=O c1(C(=O)NCC23C(CN(C(c4ccc(CCC)[nH]4)=O)C2)C3)cn2c(n1)COCC2 CCCC(C(O)C(=O)N1CCC=C(F)C1)NC(c1nnc(O)nc1O)=O CC(C)CC(C(=O)N1CC(C)(C)CC1CNC(=O)CC(C)(C)CN(C)C)N(C)C n1(CC(C)C)nncc1C(=O)OC(C)(C)C(C)NC(C1CC1OC(C)(C)C)=O N1(C(c2cnn(CC)c2Cl)=O)CC2(CC(NC(c3c[nH]cc3Br)=O)C2)C1 C1(NC(c2nnnn2CC2CC2)C(c2ccccc2)C)CC2CCC1C(O)C2O c1(C(N2CCN(C(c3c(O)ccc(C)n3)=O)C(C)C2)=O)cnn2ccc(O)nc12 CCC(C)(C)CC(=O)NC(C1CCN(C(C2(C)COC(=O)OC2)=O)C1)(C)C CC(CCCO)NC(=O)COC(=O)C(CC1CCCOC1)c1ccccc1 CCCC(O)CC(=O)N1CC2CC(COC)C2C1.C1(=O)CC2(CC2)CN1 c1(CC(=O)NC23CC(CNC(c4c(C)nnn4C)=O)(OC2)C3)ccc(C#N)cc1 c1(C(N(CCCCC(=O)NC(c2nc(C)on2)C)C)=O)cccc2cncn12 CN1CCCCC1CNC(=O)C(=O)NC(C1CCCO1)(C)C C(=O)(C(C)(C)C(=O)N1CCC(CC(C)NC(C2CC2C#N)=O)CC1)NC c1(C(N2C(C3CCCN(C(C(N)=O)=O)C3)CCC2)=O)ccc(Cl)cc1Cl c1(C(N2CC(NC(c3nc(CCC)sc3)=O)(CO)C2)=O)cn(C)c(C(F)F)n1 CCC(C)C(C(=O)N1CC(O)CC1Cn1cc(COC)nn1)N(C)C N1(C(CCC2C(C)C2)=O)CCCCC(NC(c2ccnn2CC(F)(F)F)=O)C1 c1(C(=O)NC23CCN(C(C(F)=CC)=O)CC2C3)oc2ccc(Cl)cc2c1C c1(OC)ccc(N2CCC(NC(=O)Nc3cncc(Cl)n3)CC2)nc1NC1CC1Cl C(=O)(C1CCCn2nccc21)NCCCN(C)C(c1nccc(Cl)c1F)=O CC(C)C(C(=O)NCC1(CNC(=O)CCc2ccoc2)CC1(F)F)C1CCC1 c1(OC)cc(C)c(C(N2CCC(O)C(C(N3CCCC3CO)=O)C2)=O)cn1 C1(C(=O)NC(C(=O)NC2C(C#N)CCC2)CCC2CCC2)CCCC12CCC2 C(=O)(CS(=O)C(F)(F)F)N1CCC(C2N(C(C(CC)=CC)=O)CCCC2)CC1 c1(OCC)cccc(CC(N2CC=CC2CNC(=O)C(C2CC(F)(F)C2)O)=O)c1 C1(CCC(=O)NCCCO)CCC(=O)C1.C(C(C)(C)N)N(C(=O)CCOCCF)C n1(CC(=O)N(C(C)CCNC(c2nccc(Cl)c2F)=O)C)nnc2ccccc12 c1(Cn2ncc(-c3cc(CC(C(=O)NC)NC(C)=O)ncc3)c2)ccc(Cl)c(Cl)c1 CC1(C)CCC(CNC(=O)COc2cccc(O)c2)N(C(=O)CSC(F)F)C1 N1(C(c2ccc(CC)[nH]2)=O)CC=C(CNC(=O)CC(C)C(F)F)CC1 c1(CC(=O)NCC(CNC(C23OC(C)C(C2)C3)=O)(C)O)cnc2ccccc2c1 c1(C(=O)Nc2cnc(N(C)C)nc2)ccc2c(n1)CN(C(=O)C(C)(C)F)CC2 Cc1nn(C)c(=O)c(C(N2CCCC2C(C)(C)NC(C2CCCCO2)=O)=O)c1C C1(NC(C2(CCC=C)CC2)=O)CC2(C1)CC2C(=O)NCC1CCCC(=O)N1 c1(CC)ccc(N(C)CC)c(C(N2CC=CC(NC(=O)C(C)C(O)CC)C2)=O)c1 c1(CNC(C(C)OC)=O)cccc(CNC(=O)C(c2cnccn2)C)c1 CONCC(O)C(=O)NCC(c1ccc(-c2nn[nH]n2)cc1)C Cc1cnn(C)c1CC(=O)NCCC1CN(C(C2OCC2(C)C)=O)CCO1 C(C(C)(C)C#CC(=O)N1CC(O)(C(N)=O)C1)NC(C1COCC(C)O1)=O N1(CCN(C)C)CCN(N2CCN(C)C(C(F)(F)F)C2)CC1 c1(C(C(C)C)NC(c2ccccn2)C2CCCC2)nnnn1C1CC1 C1(NC(=O)NC2(C)CN(C(C=C(CC)C)=O)C2)COc2c(Br)cccc2C1 c1(C=O)ccc(CO)cn1.CCC(CNC(C1CCCN1)(C)C)C1CCC1 Cc1nn(C)cc1C(C)NC(=O)CCC1CCC(NC(=O)C(C)C(C)C)C1 c1(C(=O)NCC(C)NC(=O)COCC2CC2)cccnc1NCC1CC1 c1(OC)ccc(CC(C)=CC(N2CCN(C(C3COCC(C)O3)=O)CC2)=O)cc1 c1(C(=O)NC(CC)CNC(c2sccc2Br)=O)cc2c(s1)CCC2 c1(C(N(C(C)CNC(=O)C(C)OCCN(C)C)CC)=O)cc(O)cc(C#N)c1 CCS(=O)(=O)c1ccc(Nc2ncc(CC(=O)OC(c3ccoc3)C)o2)cc1 C(C(C)(CO)NC(=O)CCC1(C)CC1(F)F)NC(COCC)=O N1(C(c2ccc(C)[nH]2)=O)CCC(NC(=O)C(c2cnn(C)c2)O)C(C)C1 c1(C(=O)NCC23C(CN(C(CC4CC(=C)C4)=O)C2)CC3)ccc(S(C)(=O)=O)cc1 c1(CC(=O)NC2CCN(CC(=O)OC)C2)sc(C2CCC2)nc1C O=C(C1CCCCc2ccccc21)NC1CCCC1NC(=O)COCCCF N1(C(c2cnc(CC)nc2O)=O)CCN(C(=O)C(O)C(C)(C)C)C(CC2CC2)C1 C(=O)(C1=CCc2ccccc21)N1CC(O)(CNC(C2CCC3CCC(=O)N23)=O)C1 C(=O)(C1CCc2nnc(C)n21)NC1CCN(C(C2CCC(SCC)CC2)=O)CC1 c1(C(=O)NC2(CNC(C(C)SCC)=O)CCCCCC2)ccc2nc[nH]c2n1 C1(NC(C(C)C2CC2)=O)CCC2(CCN(C(=O)CNC(=O)C(C)(C)C)CC2)C1 N1(C(CCCC2(NC(=O)OC)CC2)=O)CCC(C2(NC(C3CCCO3)=O)CC2)C1 c1(C(=O)NCC2C(CNC(CCCC#CC)=O)C2)cc(CC)c2n[nH]cc2c1 Cc1cnc2nc(C(N3CCC(C)N(C)CC3)=O)nn2c1 C1(CC(=O)N(C)CC2CCCO2)CCCN(C(=O)CC#N)CC1 C1(CNC(c2cc(OC)ncc2)=O)CC2CN(C(C3CCCN3C3CC3)=O)CC12 N1(C(C(C)CC(N)=O)=O)Cc2ccccc2C(NC(c2c(Cl)nsc2Cl)=O)C1 C(=O)(CCCc1n[nH]c(=N)s1)N(CCC#N)CCNC(C)=O c1(C(C(=O)NCCCC)N(C)Cc2cc(C)n(C)n2)ccc(F)cc1C C(CCC1CCCO1)(C(=O)NCC(C)(C)C1CC1)N(C)CCc1ccccc1 C(=O)(C1=C(C)CCOC1)N1CC(CC=C)(C(N2CC(C(N)=O)C3(CC3)C2)=O)C1 CCCC(O)CC(=O)NCC1C=CC(NC(=O)C(C)CSC)C1 C(=O)(CN=c1[nH]c(=NCCc2nnc(C)s2)[nH]c2c1CSC2)NCC=C Cc1nn(C)c2[nH]c(=NC(C)C3COCCO3)cc(N3CCOCC3)c12 O=C(NNc1nccnc1Cl)Nc1nccc2cccnc12 CC(CC(=O)N1CCC(CF)(NC(c2cccc(N)n2)=O)C1)C(C)(C)C C1(C2CC2)(CNC(C(C=C)C)=O)CCN(C(c2cccc3c2OCO3)=O)C1 c1(CC(=O)NCC2CN(C(c3c(Cl)ccc(C)c3)=O)C2)cnc2n1CCOC2 c1(C(N(C)CC2N(C(C(CSC)C)=O)CCCC2)=O)cc(Cl)cc(Cl)c1 C12(C(=O)NCC3N(C(C4CCN(C)C4)=O)CC3)C3CC(CC13)C2(F)F C(C)(C)(CC(=O)N1CCCCCO1)N(C(=O)CC1CCCCO1)C n1(CC#C)c(N2CCCC(CC(C)C)C2)nnc1C(C1CCCCO1)C CCCCC(C(=O)N(C1CN(C)CC1O)C)NC(=O)C(C)CC1CCC1 N1(C(c2c(C)nn[nH]2)=O)CC2(C=C(C(=O)N3CCC(O)C3)CO2)C1 c1(C(N2CC3C(CN(C(c4c(CCC)n[nH]c4)=O)C)C3C2)=O)cccc(Cl)c1O CC1=NOC(C)(CNC(=O)COC2CN(C(C3CN4CCC3C4)=O)C2)C1 n1(CCOCC)nnnc1C(c1ccoc1C1CCC1)NC(C)C C1(NC(C2CCN(C(=O)NC)CC2)=O)CC(O)CN(C(=O)Cn2cc(Cl)cn2)C1 CC1(C(N2CCC3(CC3NC(c3cnsn3)=O)C2)=O)CCNC(=O)C1 C1(COC)CC(O)CN(C(=O)CCCCc2cn(C3CCC3C(=O)O)nn2)C1 C#CCC(O)C(=O)N(C)CC1(O)CN(C(c2ocnc2C2CC2)=O)C1 c1(OC)noc(C(=O)NC2(CNC(c3cccnc3)=O)CCC2)c1Br C1(NC(CCOCCOC)=O)CN(C(=O)Nc2ccnc(O)c2)CC1F C12(C(=O)NCc3c(C)nsn3)CCC(NC(C3C4CCCC34)=O)(CC1)C2 N1(C(C2(C)COC2)=O)CCC2(CC1)CN(C(c1cc(-c3ccco3)c[nH]1)=O)C2 C1(CNC(C2N(C(c3cc(C)[nH]n3)=O)CC(O)C2)=O)CCCCC1(C)C N1(C(c2c(Cl)cnc(C)n2)=O)CCC(C)N(C(c2cnc3[nH]ncc3c2)=O)CC1 c1(C(N(CC(C)NC(C2(C)CC(F)(F)C2)=O)C)=O)cc(Cl)ccc1Br c1(NC(C(c2ccnn2C)NC(CCCSC)=O)=O)cnn2c1OCCC2 C12(C(C(=O)NC)N(CCC#N)CCN(C)CCOC)CCC(CC1)C2 N1(C(C2C(C)(C)CN(C(=O)C(C3CCOCC3)=O)C2)=O)CCCCC2(CCC2)C1 C(C)(C)(CC(F)C(=O)NC(C)CCN(CC)CC)NC(CNC(C(CC)C)=O)=O C(=O)(CC(O)CN(C(=O)CCNC(C)=O)CC)NCC c1(NC(C2N(C(c3cc(C#N)c[nH]3)=O)CCC(C)C2)=O)cccc2[nH]ccc12 CC(C)(C)C(O)CC(=O)NCCOCCCNC(C1(CF)CC1)=O C1(C(=O)NCC2CN(C(C(C)OCCN(C)C)=O)C2)CCCOCC1 C1(C(=O)OCC2CC2)CCCN(C(c2ccccc2)=O)C1 C#CC1(NCC(=O)Nc2cc(C(F)(F)F)ccc2C)CCCOC1 CC1CC(C)C(C(N2CCC(=CCNC(c3c[nH]c(Br)c3)=O)CC2)=O)O1 N1(C(CCC(C)(C)F)=O)Cc2nccn2CC(NC(=O)CCC2CCOC2)C1 CC1OC2(CO)CC1(C(=O)N(CC(C)NC(c1ccc([N+](=O)[O-])o1)=O)C)C2 C12(CC(=O)NC34CCC(CC3)N(C(=O)C(=O)NC3CC3)C4)CCCCC1C2(F)F c1(C(N2CCCC(C(C)(O)CNC(=O)CNC=O)C2)=O)ccc2ccncc2c1 C1(OCC(=O)NCCn2cc(CCOC)nn2)CC12CCC(F)(F)CC2 C1(CCC)CCCN(C(C2(CSC)CN(C(=O)COCCC)C2)=O)C1 C#CCCCCC(=O)NCC(C(C)C)NC(C1(c2ccnn2C)CC1)=O Cc1ccc(C(N2CCC(NC(=O)Cc3cnc(C)s3)C2(C)C)=O)c(C)n1 C1(C(=O)NCCCN(C(=O)CSC(F)F)CCO)CCC(O)C1 c1(C(=O)NC2CC(NC(CC(=O)OCC)=O)C2)ccc(OC)nc1Cl S(=O)(=O)(c1c(C)cccc1C)N(c1cccc(Cl)c1)CCCCCC C#CCCCCCCC(=O)NCC(C1CCC1)NC(C1CNC(=O)N1C)=O N1(C(C(C2CN(C(=O)CC3CCC(F)(F)C3)C2)OC)=O)CC2CCC1CC2 N1(C(Cn2c(C)ccc2C)=O)CC2CCCCC2(CNC(C2CC(C)(C)C2)=O)C1 CC1C(NC(=O)C(C)OCCc2ccccc2)CCCN1C(c1cnc[nH]1)=O Cc1cc(C(=O)N(C)CC2CCN(C(=O)C=Cc3cnn(C)c3)C2)cc(C)c1 Cc1cc(C)nc(NCC2N(C(C3CCC(=O)N3)=O)CCC2)n1 CCC(F)(F)C(=O)NC1CN(C(=O)CN(C)C(N)=O)CC1C(F)F C1(C(=O)NCCCCN(C(=O)CN(C2CCC2)C)CC)CCOCC1(C)C c1(CC)nc(N2CCCC2CN(C)C(c2ccsc2SC)=O)c2ccsc2n1 C1(C(=O)NCCCC(C)(C)NC(c2n(CC(C)C)ncc2)=O)CCCC(F)(F)C1 c1(C(C(=O)Nc2cccc(OC)c2)N2CCC2C2CCC2)cc(C)cc(C)n1 N1(C(C(C)OCc2cnc(S)n2C)=O)CCCCC1C1(C(=O)N)CC1.C1CC1 C1(CC)C(C(=O)NCC2CCCC23CC3)CCN1C(c1cc(C#N)c[nH]1)=O C(=O)(C(C(C)(C)C)n1ccnn1)NC1CC(CNC(CC(C)F)=O)C1 C(=O)(C1CCCn2ccnc21)N1C2CC(NC(c3ccc(C)cc3C)=O)C2CC1 S(=O)(=O)(c1ccc(C#N)c(NC(C2(CSC)CC2)C)c1)NCc1c(CC)nns1 N1(C(c2ccc(C#C)cc2)=O)CC(C)CN(C(C2CCN2C2CCCC2)=O)CC1C C(c1ccc(F)cc1F)=CC(=O)NCC1C(NC(CN(S(C)(=O)=O)C)=O)C1 N1(C(c2cncc(OCC)c2)=O)CCCC(CNC(=O)CCC(F)F)CC1 c1(OC)cc(C(c2nnnn2C2CC2)NCC2CC2(C)C)ccn1 C12CCCCN(C1)C2=O.c1(COC)cn(CC(C)NC(C2(O)CC2)=O)nn1.C1CC1 CCC(C)CCC(O)CC(=O)NC(CO)C(C)NC(c1sc(C)nc1C)=O Cc1oc(C(C)(C)C)cc1C(=O)NC(C1CCCN1C(C1CC(Cl)(Cl)C1)=O)C c1(C(N(CCNC(C(C)CS(C)=O)=O)C2CC2)=O)cc(Cl)c(N)c(Cl)c1 c1(CC)cccc(C(=O)NCCN2CCN(C(=O)COc3cnn(C)c3)CC2)n1 C(C(C)C)(C(O)C(=O)NCC1CC(F)CN1C(c1cc2n(n1)CCCO2)=O)OC C(c1ccc(OC)cc1C)=CC(=O)NCCC1CC(NC(CNC(C)=O)=O)C1 CCCCCCC(=O)NC1CCC(NC(=O)C(F)=CCCF)C1 n1(CC(=O)NC(CNC(C2(COC)CCCCC2)=O)C(C)C)nc(C)c(C)c1C c1(COCC(=O)NCCCNC(C2CCCOCC2)=O)ccc(Cl)cc1 c1(C(C(=O)NC)NC(C)=O)ccc(N(C(C)C)C(C)C)cc1 C1(N(C(C(C)OC)=O)C)CCCN(C(C2(c3cccc(O)c3)CCCC2)=O)CC1 C12(CC)CN(C(=O)CC3CSCCS3)C(CNC(c3ccc(C)c(F)c3)=O)(C1)C2 Cc1noc(C)c1C(C)CC(=O)OC1CCN(c2ncccn2)C1 N1(C(C2OCCC(NC(c3cncc(C)n3)=O)C2)=O)CCCc2occc2C1 c1(C(N2CCCC(C(=O)OC)C2)=O)n[nH]c2c1CN(C(c1cncs1)=O)C2 C(=O)(C1CCCc2nccn21)N1CCC2CCN(C(CCCOC)=O)CC21 Cc1cc(C(c2nnnn2CCOCC2CC2)NC2(CO)CCC(C)CC2)ccc1F Cc1ccc(C#N)cc1C(=O)NC(CN(C)C)C(=O)NCc1ccc(Cl)o1 N1(C(C(c2cccnc2)OC)=O)CC2CCC1C(NC(C1CCCCCC1)=O)C2 Cc1c(NC(=O)CCC2CCOC2)cnn1-c1ccc(C(C)(C)C)cc1 c1(CC(C)C)c[nH]c(C(N2CC(CNC(c3cc(-c4ccco4)c[nH]3)=O)C2)=O)c1 c1(C(=O)NC2CN(C(c3coc4c3C(=O)NCC4)=O)C2)cnc(O)c([N+](=O)[O-])c1 CC1(C)C(CNC(=O)CNC(=O)CCc2cccnc2Cl)CCN1C(=O)CCF c1(OC)ccc(CN2CCC(C(C)C(=O)Nc3ncc(O)cc3C)CC2)cc1F c1(C(=O)NC2C(O)CCN(C(C(C)(C)c3nccs3)=O)C2)ccc2scnc2c1 C#CC1CCCN(C(=O)C(CCCOC)NC(c2cc(COC)no2)=O)C1 CC(CC(=O)NCCCCC1(NC(=O)C=Cc2ccc[nH]2)CC1)C1CC1 C(c1ccc(F)cc1)=CC(N1C(C)(C(=O)Nc2cccc(COC)c2)C=CC1)=O Cc1nn(-c2ccccn2)c2sc(C(=O)NCc3ccc(F)c(F)c3Br)cc12 Cc1[nH][nH]c(=NC(=O)C2CCC2C(C)(C)C)c1C CC(C)CC(C)(O)C(=O)NC1CC(CNC(C2CNC(=O)C(C)(C)C2)=O)C(O)C1 Cc1cncc(OCC(=O)NCC2(C(N)=O)CN(C(C3COC(=O)N3C)=O)C2)n1 N1(C(C2C(CCC)C2)=O)CCN(C(c2noc(C)c2Br)=O)C(CC)C1 Cc1nc(C(=O)NCC(n2cc(CN3CC4CC4C3)nn2)C)c(Br)s1 c1(C(NNC(=O)CC2(NS(C)(=O)=O)CCSC2)=O)cccc2c3c([nH]c12)CCCC3 Cc1cc(NC(=O)C(N2CCC(C)(C(=O)NC3(CCO)CC3)CC2)C)cc(C)c1 CC1CCN(C(=O)CCCC(=O)N(C)C)CC1NC(c1cc([N+](=O)[O-])c[nH]1)=O N1(C(C(CC#C)O)=O)CC2(CCCC2)C1C(=O)NC(CCC=C)C(=O)OC N1(C(C(COC)(F)F)=O)CC23CCCC2(C1)CN(C(=O)CC(C)(O)CC(=O)O)C3 N1(C(C(C)OCC=C)=O)CCN(C(=O)Cc2c(C)cccc2F)C(C(C)C)C1 O=C(C1=CCC(NC(C2CCCCC2O)=O)C1)NCC1CCCC2(CC2)C1 c1(CC(=O)N(C)CC2CN(C(c3ccn(C)n3)=O)CCO2)c(F)cccc1Cl C(C(C)(C)C(=O)NC(CC1CCCC1)CO)N(C(=O)COC1CCCOC1)C Cc1cccc(-c2nccn2Cc2csc(-c3ccn(C)n3)n2)c1C C1(CNC(C2CCS(=O)(=O)CC2)=O)C2CCC(C2)N1C(C1(O)CCSC1)=O C1(CNC(c2c(CC)cncc2)=O)CN(C(c2ncsc2C)=O)CC1(F)CO N1(C(C2CCN(CC(C)C)C2)=O)CC(NC(=O)Cc2c(Cl)cnn2C)C(C)C1 c1(C(=O)NC(C(C)C)CNC(=O)CCc2cccc(Cl)c2)c(F)ccc(O)c1O c1(C(N(CCNC(c2ccc(C(F)F)o2)=O)CC)=O)c(C(F)(F)F)nn(C)c1C Cc1cc(C(=O)NC(C)(CNC(c2c(C)noc2C(C)C)=O)CO)nc(C)n1 c1(C(c2n(CCOCC)nnn2)NCCc2ccccn2)c(Br)cnc(Cl)c1F CCC(C)(C)C(C)CC(=O)N1CCC(CNC(c2cncc(Cl)c2Cl)=O)(OC)C1 C1(CC=C)(NC(=O)C(C)OCCOC)N(C(=O)C(N)=O)C1 C1(C(N2CC(CCNC(C3(OCc4ccccc4)CC3)=O)C2)=O)CC2CC1CC2O Cc1cccc(OCCCC(=O)NCC2(O)CCN(C(=O)Cc3cn[nH]c3)C2)c1 C(C(CNC(c1ncoc1Br)=O)C(F)(F)F)NC(C(CC)=CC)=O C12(C(=O)NC(CN(C(c3c(C)nc(CO)s3)=O)C)C)CC=CCN1CCC2 CN1CCC(CCC(=O)NCC2(C(=O)NC3(C(N)=O)CCC3)CCOCC2)CC1 N1(C(CCCCCOC)=O)CCCCC2(C1)CN(C(c1cnsc1)=O)C2 N1(C(c2cc(C)[nH]c2)=O)CC(CC(=O)NC(CO)CC(C)(C)C)CC1(C)C c1(NC(c2n(CCCCOC)nnn2)C2CC2)ccccc1C(=O)NC1CC(O)C1 N#Cc1ccc(C(=O)NCC2CC(NC(C3CCS(=O)(=O)N3)=O)C(O)C2)cc1F c1(NC(C2COCC(C)O2)=O)cn(C2CCC2)c(=O)nc1O N1(C(C(CC)(C)O)=O)CC(C(=O)NC2CC3(C2)CC(C)C3)CC(C)(C)C1 C1(NC(C=CC(=O)N(C)C)=O)CC2CN(C(c3ccc(C#N)o3)=O)CC12 C=C(C)CC(C(=O)NC1CN(C(=O)Cc2ccccc2C)CC1C)NC(C)=O c1(CC(=O)NCC2OCCN(C(c3n(CC)nnc3)=O)C2)ccc2sccc2c1 C(=O)(C1Cc2ccccc21)NC1CCN(C(c2c(OC)nccn2)=O)C1 Cc1nn(C)c(C(N2CCC3CN(c4[nH]cnc5nc(Cl)cc4-5)C3C2)=O)c1[N+](=O)[O-] C=CCC(CC(C)C)C(=O)N(CC(CO)(CO)NC(=O)CCn1ccnn1)C C1(CC=C)(C(=O)NCCC(C)F)CCN(C(C23CCC2C3)=O)C1 c1(C(N2CC3C(C(=O)Nc4ncc(CC)cn4)C3C2)=O)ccc([N+](=O)[O-])cc1 CCCCCCCC(=O)NCCn1cc(CNC(=O)C(C)CSC)nn1 c1(NC(c2ccon2)C)cc(Br)ccc1S(=O)(=O)NC1(OC(F)F)CCOC1 CCC(F)(F)CC(=O)NC1CC(F)(F)CC1NC(=O)COCCCC(C)C C(=O)(CC(C)(C)CC(F)F)NC(CC(C)NC(=O)CSc1n[nH]c(O)n1)C CCCCC(C(=O)N(C(C)(C)C)Cc1cn(CCCO)nn1)N1CCCCC1 Cc1cnn(C)c1CC(N1CCC(NC(c2nn(C(C)(C)C)cc2Cl)=O)C1C)=O C1(CN(C)Cc2cnc(CCC)s2)CCCN(C(=O)CC2(CO)CCC2)C1 c1(CC)ccc(C(=O)NC(Cc2cc[nH]n2)C(=O)NCc2nnc(O)n2C)nc1 N1(C(c2ccc(C(N)=O)o2)=O)CC2(CCCN(C(C34CC5CC3C4C5)=O)C2)C1 C1(NC(C2CC2C(F)F)=O)CC12CCN(C(c1ccc3c(c1)OCC3)=O)CC2 c1(C(=O)NC2CCN(C(CCCOC)=O)C2)ccc(C(C)(F)F)nc1 C(=O)(C1=CCCCC1)N1C(CO)CC(NC(COC)=O)C1.c12cccnc1OCC2 C(=O)(CCC(C)(C)F)N1C(C)CC(NC(C)=O)C1.c12ccc(cc1)[nH]c2=O N1(C(C(C)(C)F)=O)CCC2C(C1)CN2C(C1C=CCCC1)=O Cc1nc2cc(C(=O)N(c3cc(Br)ncc3Cl)C3CC4CNC3C4)ccc2s1 N1(C(C2(OC)CCCOC2)=O)CCCC(O)(CC(=O)NCC=CCC2CCC2)C1 C1(C(N2C(CNC(C(C)C)=O)CC(C(F)(F)F)C2)=O)CCn2c(O)nnc2C1 N#Cc1ccc(OCC(=O)NCC2CCC2CCc2ccccc2)c([N+](=O)[O-])c1 c1(CC(C)(C)OCC)cn(CC(F)CCNC(=O)COC(C)=O)nn1 C1(C(=O)NC2CC(C(C)C)OC2)CNC(=O)CN1C(C1CCC2CC12)=O N1(C(c2c(C(N)=O)nccc2)=O)CCC2(CC2C(N2CC(F)(F)CC2CO)=O)C1 c12cc3c(cc1CNC(=O)N2)OCCO3.N1(CC)Cc2cccc(O)c2C1 c1(CC)cc(C#N)c(C(N2CC(C(=O)OCCC)CC(CO)C2)=O)s1.OC C1(CNC(C2(O)CC(C)(C)C2)=O)CC2CCC(C1)N2C(C1CCCC12CC2)=O c1(C(=O)NC(CC(C)C)Cn2cc(CCC3CCCC3)nn2)c(O)cccc1F C(=O)(C(C)S(N)(=O)=O)NCC1CN(C(c2oc(CC)c(C)c2)=O)CC1O CC1(C)CN(C(C2CC(=O)CO2)=O)C1c1nccn1C1CC1 N1(C(C2(C=C)CCN(C(=O)C(C)OCOC)CC2)=O)CC(C)(C)OC(C)(C)C1 C1(NCC(CC)C)CCC(C)N(C(c2cccc(Cl)c2C(F)(F)F)=O)C1 CCCC(C#N)C(=O)NC(CC1CC1)CC(=O)NCc1ccc(C)cn1 C1(CNC(C(c2c(C)noc2C)C)=O)CCN(C(c2coc(C#N)c2)=O)CC1C c1(SC)cc(C(=O)NCC(O)CNC(C2CC2(F)F)=O)ccn1 Cc1nccc(C(N2CCCCC2c2cn(CCCc3cccnc3)nn2)=O)n1 C1(NC(c2nc(C)sc2)=O)COCCN(C(=O)CSC(C)(C)C)C1 CCCN(OC)C(=O)CC(C(C)OC)NC(=O)CC1CCCSC1 C1(N(C(COCC(=O)NC)=O)C)CN(C(=O)C=C(C)c2ccsc2)CC1F C1(O)(C(C)NC(c2c(C)nc(C)[nH]2)=O)CCN(C(C23CCCC2C3)=O)CC1 N1(C)CCC(C(=O)OC)CC1.C1(C)CN(NC(CC2CCN(CC)C2)=O)CCO1 N1(C(=O)Nc2cccnc2)CCCC(CO)(Cc2cn(C3C=CCCC3)nn2)C1 c1(OC)ncc(C(=O)NC(C)(C)C(C)NC(=O)CCc2ccccc2F)cn1 CC(C)C(F)(F)CC(=O)N(C)CCOCCNC(c1ccc(N)cn1)=O c1(CC)cc(C(=O)NC2COCC2C(N2CCCC2CC(C)(C)C)=O)nn1C c1(C(N2CC(C)C(n3cc(-c4ccccc4O)nn3)C2)=O)cnn(C)c(=O)c1 c1(NC(N2C(CNC(c3cc(F)cnc3Cl)=O)CCCC2)=O)ccc(Cl)c(F)c1 C1(F)(C(=O)NCC(C)NC(c2cc3n(n2)CCC3)=O)CCS(=O)(=O)C1 C1(n2cc(C(=O)OCC)nn2)CCCC2(CN(C3CCCc4ccccc43)C2)O1 c1(C(=O)NC(CNC(c2c(C)n(C)cn2)=O)C)cc2c(s1)CCC(C)C2 c1(CC(N2C(CNC(CCCCC)=O)C(C)CC2)=O)c(F)cccc1F S(=O)(=O)(c1ccc(NC(CC)C2CCC2)nc1)NC(c1ncn(C)n1)CC Cn1ccc(CC(N2CC(C)(F)C2)=O)n1.N12CCC(C1)CCC2=O N1(C(C(CNC(C)=O)(F)F)=O)CC(C(=O)NC23CC(C)(C2)C3)CC(C)C1 c1(C(=O)NCC2C(NC(C3(CC)CCOCC3)=O)COC2)cc(Cl)ccc1Cl c1(C(=O)NCC2N(C(c3c(OC)nccc3)=O)CCCC2)ccc2ccncc2c1 N1(C(CCCC)=O)CCC(C(=O)NCCC2=CCOCC2)CC1CC O=C(CC1CCCc2ccc(OC(F)F)cc21)OCc1ccc(Br)c(OC(F)F)c1 c1(C(=O)NCCCCOC)ncc(C(F)(F)F)cc1N N1(C(COc2cc(C)cc(C)c2)=O)CCCC2(CC(NC(C3CCCO3)=O)C2)C1 c1(OC(C)C)cnc(NCC(CC(C)C)NC(=O)C(C)Cn2ccnc2)nc1 n1(CCC)cc(C(=O)NC2CCC(C)(CNC(c3cc(C#N)cs3)=O)C2)c(C)n1 C(=O)(C(CC)CCOC)N1CCC(C(N2CC(C#C)C2)=O)C1 Nc1cccc(Cl)c1C(=O)NCC1(NC(=O)CC2CCC3CC3C2)CC1 c1(OC)ccc2cc(NC(c3noc(C)n3)c3nnnn3C3CCCCC3)oc2c1 c1(C2(C(=O)NC3CC(N(C(CC(CC)C4CC4)=O)C)C3)CC2)ccc(F)c(F)c1 c1(N2CC(C(C)NC(C3C(C=C)C3)=O)C2)nc(C)ncc1C(=O)OCC n1(CCCCN2CC(C(C(=O)OCC)C)C2)ccc(C)n1 CC1(C(=O)NOCC2C=CCCC2)CC(O)CN1C(c1cc(CO)on1)=O CC(O)C(F)(F)C(=O)N1C2CCC1C(NC(c1ncccc1Br)=O)C2 c1(N2CCC(NC(C#CC)=O)C(F)C2)ncnc2cc(Br)sc12 C1(NC(CCNC(=O)OCC)=O)C2CC1N(C(=O)CCc1cc(C)n(C)n1)C2 C1(C(C)C)CCC(C(=O)NC2CCCC2NC(=O)CC2CCCN2C(C)C)CC1 C1(NC(c2n(CCCF)nnn2)c2cscn2)C2CCC1CC2 O=[N+]([O-])C1CCCCCC(NCC2CCN(Cc3ccccc3)CC2)C1 c1(-n2c(C(c3ccccc3Cl)NCC3CC(C)(C)OC3)nnn2)ccc(F)c(F)c1 C(=O)(C1=CCCOC1)NC1(C)CCN(C(Cc2c(CC)n[nH]c2CC)=O)C1 N1(C(C(=Cc2ccncc2)C)=O)CCC(C)C(CNC(c2c[nH]nc2C(F)F)=O)C1 c1(C(C)C)ccc(C(N2CCC(C(C)NC(=O)C(N)=O)C2)=O)o1 c1(C(N2CC(=C)C2)=O)ncccc1OC(C1CCCC1)=O N1(C(CC2OCC(C)(C)C2)=O)CCN(C(C2(C(F)(F)F)CCC2)=O)CC12CCC2 CC(C)C(O)CC(=O)NCC1CCCCC1C(=O)NC(C)CCC1CC1 C(C(C(=O)N1Cc2cccnc2C1)C(C)(C)C)NC(C(C(CC)C)=O)=O N1(C(C=C(COC)C)=O)CCC(C)C1C(=O)N(C(C)CN(C)C)CC Cc1ccnc(-c2cn(CCCC(=O)C(C)(C)c3ccccc3)nn2)n1 c1(NC)cnc(Cl)cc1C(=O)OCC1CNC1 C1(C2N(C(C(C)O)=O)CCC2)CCN(C(=O)CN2CCCNC2=O)CC1 c1(-c2nc(NC(CN(C3CC3)CC)=O)sc2)ccc2ccccc2n1 CC(C)CC(C)C(=O)NCC(C)(CO)NC(=O)COCC(C)(C)C c1(CC(=O)NC(C)CCNC(C2(N(C)C)CC2)=O)c(Br)cnn1C C1(NC(c2[nH]n(C)c(=O)n2)=O)CN(C(c2csc(CC(F)(F)F)n2)=O)C(C)(C)C1 C1(CC(=O)NC(CN(C(=O)C(C)C#N)CC)C)(N(C)C)CCCC1 CC1(C(N2CCCC(CNC(=O)CCCC3CCCC(=O)N3)C2)=O)CC=CCO1 C(CCC(=O)NCCCCCF)N(C)C(c1ccsc1Cl)=O C1(C(=O)NC2(CC)CCC2)CC2CN(C(c3cccc(=O)o3)=O)CC2C1 Cc1ccc(Cl)cc1NC(C1CCN1C(=O)NC1CC=CCC1)=O C=C(C)CC(C(=O)NCC(CC)n1cccn1)NC(c1coc(C(N)=O)c1)=O N1(C(c2ccc(-c3ccccc3Cl)o2)=O)CCN(C(=O)CC2CCC2)C(CO)C1 c1(NC(CC)CNC(=O)CCCN(C)C)cc(C)nc2c(C)cnn12 c1(C(=O)NC2CCC3(C(NC(C(COC)C)=O)C3)CC2)ccc2nc(S)[nH]c2c1 c1(C(=O)C(=O)CC)ccc(O)cc1.n1(C(CC)(C)C2CC2)cc(C2(CCOC)CC2)nn1 N1(C(c2ccc(OC)cc2C)=O)CCC(C)(C)C(NC(C2CCC3(CC3)C2)=O)C1 N1(c2ccnc(-c3cn(C4CN(C(C)(C)C)CC4O)nn3)n2)CC(=O)CCC1=O CC1C(C(=O)NC(C)(CNC(c2coc(O)n2)=O)C2CC2)C1(F)F c1(CC(=O)NCC23CN(C(C(CC)(F)F)=O)C(C2)CO3)c(C)nc2ncnn2c1C C1(C(=O)NC(COC)C2CC2)(C(=O)OC)CN(C(=O)CC2CCN(C)C2)C1 C(=O)(C1=CS(=O)CCC1)NCC12C(CN(C(CCc3ccn(C)n3)=O)C1)CC2 C1(NC(C2CC23CCCCC3)=O)CC2CCC1CN(C(=O)C=CC1CCC1)C2 c1(SC(c2c[nH]c(C(N3CCCC3COC)=O)c2)(C)C)cncc(F)c1 C(=O)(N=c1ccnc2[nH][nH]cc1-2)C12CC(NC(c3c(OC)ccc(C)c3)=O)(C1)C2 CCC(CO)C(=O)NCC1(F)CN(C(=O)C(C)Cc2ccc(C(F)(F)F)cc2)C1 c1(NC(C2N(C(COCC=C)=O)CCC2)=O)cc(CO)ccc1OC c1(NC(C2CC(NC(=O)Cc3ccc(F)cc3F)C2)=O)cc2ccc(Br)cc2s1 c1(C(C(=O)OC)NC(C2(CC)C=CCC2)=O)ccc(F)cc1 c1(C(N2C3C(N(C(c4c(C)nco4)=O)C)CC(C3)C2)=O)noc2cc(Cl)ccc12 c12cccc(c1[N+](=O)[O-])N2.C1(CCC)CCOCC1(c1nnnn1CC)OCC N1(C(c2ccc(F)c(C)c2N)=O)C(CNC(=O)CCS(C)(=O)=O)CC2CCCC12 C1(NC(C2OCCN(C(c3[nH]cc(C)c3)=O)C2)=O)CC2(CCOC2)C1 c1(C(=O)NCC2(O)CCCN(C(CCN(C(C)=O)C)=O)C2)cc2n(c1)CCOC2 c1(C(=O)NCC(CNC(C2CCOCC2C)=O)OC)ccc(CCF)cc1 c1(C(N2CCN(C(COCc3ccc(C)s3)=O)C(C)C2)=O)cc(O)c(F)cc1N CC1C(NC(c2cc(C#N)c[nH]2)=O)C(C)CCN1C(c1cc(C2CC2)on1)=O C1(C(=O)NC(C)CN(C(=O)CC2CC2)CC2(C)OCCO2)CCc2cc(C)ccc2O1 C(=O)(C1=C(C)CCCC1)NC(CCOC)CNC(=O)CCc1cncs1 n1(C(C2CCCCC2)C)nc(Cc2cccs2)nc1-c1coc(C(F)(F)F)c1 N1(C(c2cncc(NC)c2)=O)CC(NC(c2cc(Cl)cn2C)=O)CC(C)C1 c1(N(C(=O)C(c2ccco2)NCCO)C(=Cc2ccco2)C)ccccc1F c1(C(N2C(CC(=O)NC(C#C)CCC)COCC2)=O)cc(C)c(C)cn1 c1(C(N(C(C)(C)CC(=O)OC)CC)=O)ccc(OC(F)F)c2c1CCN(C(C)=O)C2 C(=O)(CC(F)(F)C(F)(F)F)N(C1C(NC(c2nc(C(C)C)oc2)=O)CCCC1)C Cc1cc(C(=O)N(C2CN(C(c3cccnc3O)=O)CC23CC3)C)ncc1Br c1(C(N2CCOC(c3nn[nH]n3)C2)=O)ncnc2ncccc12 c1(OCC#C)cccc(CN(C(c2ncsc2C)C(=O)O)C)c1 N1(C(=O)Cc2cncc(F)c2)CC2(C1)CN(C(=O)C(O)Cc1cccc(Cl)c1)C2 N1(C(CSCC(=O)OC)=O)CCC(O)(C(C)CNC(=O)CC(C)(C)O)C1 C1(F)(CCC)CCN(CC(OCc2ccccc2)OC)C1 CCCC(CC)C(=O)N1CCCC1(C)CNC(C1(C(F)F)CCOCC1)=O C1(CNC(c2cnc(O)s2)=O)CN(C(=O)CN2CSCC2=O)CC12CC2 CCCC(CCC)CC(=O)NCC1CN(C(=O)C(O)C(F)F)CC1SC Cc1ccc(C=CC(N2CCC(C(C)CNC(=O)CC3(C)CC3(F)F)CC2)=O)o1 C(c1ccc([N+](=O)[O-])cc1)=CC(N1C2CC(NC(c3cn[nH]c3)=O)(C2)C1)=O CC1=C(C)CC(C(=O)NCC2CCN(C(c3cncc(Cl)c3Cl)=O)C23CC3)CC1 N1(C(CCC=CCC=C)=O)C2CCC1CC(CNC(=O)Cc1cc(Cl)n(C)n1)C2 C(CCCCC(=O)NC(C1CCN(C(c2ccc(F)cc2F)=O)C1)C)OC O=C(C#CC1CCCC1)NC1CC(CCNC(c2ccc(Br)c(F)c2)=O)C1 C(c1ccc(F)nc1)=CC(=O)NC1CCN(C(c2n(C(CC)CC)ncc2)=O)C1C c1(C(=O)NC(CCN(C(C(C)OCCOC)=O)C)C)c(C)cnnc1O C(CCC(=O)NCC(O)C1CCC1)(C(C)C)NC(c1cc(C)sc1N)=O Cc1ccc(NC(=O)CC(Cc2cccs2)NC(=O)CCCCBr)cc1C#N N1(CC)CCN(C(=O)C(C2CCC2)NC(=O)CC=C(Cl)Cl)CC1C N1(C(c2cccc(C(C)C)c2)=O)CC2CCC(C1)N2C(C1CCCCN1N=O)=O C1(NC(c2c(C)nc(CC)o2)=O)CCN(C(=O)CCNc2ccccc2)CC1C C#CC1(O)CCCN(C(=O)C(C(C)(C)O)NC(C2COCCO2)=O)C1 c1(C(=O)NCCC2C(C)CCCN2C(=O)CC(C)(C)O)ccc2c(c1)COCC2 C(C)(CC(C)C#N)(c1n(CC=C)nnn1)N.n1(CCCC2CC2)ccnc1 C(=O)(C(=O)NNc1cc(Cl)ccn1)NCc1ccc(OC)c(Br)c1 N1(C(C(CC)C)=O)CCCC1(C)CNC(=O)CCc1cncc(C)c1 c1(OC)cc(C(=O)N(CCC(C)NC(c2ccccc2Br)=O)C)cc(F)c1 C1(C(=O)NC(CNC(c2ccc(Cn3cc(Cl)cn3)o2)=O)C2CC2)CC12CCC2 CC1CN(C(c2cn(CCO)nn2)=O)CC(C)CN1C(c1cc(F)cnc1O)=O CC(C)C(CCO)N=c1[nH]c(=N)[nH]c(=NCc2cnc[nH]2)[nH]1 N1(C(c2cncc(C)c2)C(=O)NC2CCOCC2)CCC2(C)C(F)(F)C2(C)C1 C1(NC(=O)COc2cc(F)ccc2F)CC(O)CN(C(C2CC(CCO)C2)=O)C1 C1(SCc2cc(Br)ccn2)CCCN(C(C2C(C(C)(C)C)C2)=O)C1 C1(CC(=O)NCC2CN(C(c3c(C(C)C)c[nH]n3)=O)C2)CC(F)(F)C1(F)F N1(C(C(C)OC)=O)CCCC(CNC(=O)C(C)COC(C)=O)C1 N1(C(C2(C=C)CCN(C(c3cccc(SC)c3)=O)C2)=O)CCC2CN(C)CC2C1 N1(C(C(N)=O)=O)CC=CC(C(=O)NC(c2ccccc2)C(N)=O)C1 N1(C(c2nocc2Br)=O)CCCC12CCN(C(=O)C(F)(F)C1CC1)CC2 C1(C(=O)NC2CC(NC(C(COCC)C)=O)C2)CCOC(C(=O)OC)C1 CC1=C(C)CC(C(N2CCC(OCCNC(=O)C(C)n3cccn3)CC2)=O)CC1 CC(C)(C)C(C(=O)Nc1c(O)cccc1F)ONC(=O)NC1CCCCN(C(N)=O)C1 c1(CCOCC(=O)NC)ccccc1.C(=O)(CC(=O)N)N(CC(O)CN(C)C(N)=O)C C(=O)(C1=NN2CCC(C)N=C2N1)NC1C(CNC(Cn2ncc(C)c2)=O)CCCC1 C1(C#N)(C(=O)NC(C=CC(=O)NCC(c2ccncc2)C)C)CCCOC1 c1(C(=O)NCC(CNC(CCCN(C)C)=O)(C)F)ccc(N)c(C(N)=O)c1 c1(COC)c(C2CN(C(=O)NC(C(=O)OC3CC3)C3CC3(Br)Br)C2)ncn1C C(c1cccc(F)c1)=CC(=O)NC(C)C(C)NC(c1ccc(CS(C)(=O)=O)o1)=O c1(CC(=O)NC2C(N(C(C(C)=CC)=O)C)CCCC2)cc(C)ccc1C C(CC(CNC(c1sccc1F)=O)NC(c1ccsc1C)=O)OC N#Cc1cc(NC(C2COCCN2C(c2c(Cl)cnn2C)=O)=O)c(F)cc1Cl c1(CNC(C(N2CCN(C)CC2)C)=O)cnn2c1CN(CC(C)(C)CC#N)CC2 N1(C(=O)NC(C)CCC2CCOCC2)CC(CO)C1(C)C c1(CC)ccc(CNC(c2ccc(CNC(C3(C)CC(C)C3)=O)nc2)=O)nc1 N1(C(CC(C=C)(C)O)=O)CCc2nc(O)cc(C(=O)N(C3CC(O)C3)C)c2C1 c1(CC)c(C(=O)NC(C2CN(C(c3nn(C)cc3N)=O)C2)C)csc1C c1(OC)cnc(C(N2CCCC2CC(=O)NCc2ccc[nH]2)=O)c(F)c1 N1(C(C(C=C)(F)F)=O)CC(NC(c2c(C(C)C)cccc2F)=O)C2CCCC2C1 CC1CCOC(C(=O)NC2CCCN(C(=O)Cc3ccccc3Br)C2)C1 C1(C(N2CCC3CN(C(c4ccsc4)=O)C3C2)=O)CCc2nncn2C1 n1(CC)ncc(Cl)c1C(=O)NCC1CCN1C(=O)CCc1ccc(C)nc1 C(=O)(C1=CC(O)CCC1)NC1CC(NC(c2cccc(C)c2N)=O)C1 C1(NC(=O)C=Cc2ccoc2)CC(CNC(=O)CC2CCCC2)C12CCC2 c1(N2CCC(CNC(=O)CC3CC4(CCC4)CO3)C23CC3)nc2ccc(Cl)cc2s1 c1(SC)cc(=NC(=O)CC2CN(C(c3cc[nH]c3C)=O)C2)[nH]n1C c1(CC)[nH]nc(C(N2CCCC(CNC(c3csc(C(C)C)n3)=O)C2)=O)c1Cl C(=O)(C(C(C)C)c1ccncc1)NCCC1(NC(COCCC=C)=O)CC1 c1(C(=O)NCC(c2ccc(C)cc2)NC(C23CC(C2)C3)=O)cc(F)c(N)cc1F C12(OC3CC3)CCCC1N(C(=O)C(O)NC(C1(N(C)C)CC1)=O)CC2 C1(CNC(CCSCC)=O)C2CN(C(c3cnn(C)c3Cl)=O)CC12 c1(SC)nc(NCC2CC(C)CO2)cc(=NCC2OCc3ccccc32)[nH]1 C1(CCN(C)C)(C(=O)NCC(O)CNC(=O)CCc2ccncn2)CCCC1 CC(C)CCCCC(=O)NC1CCN(C(=O)C(C)C(C)n2cccn2)CC1 C1(CCC(=O)NCC=CCNC(=O)CCCc2ccc(Cl)cc2)CCC(O)CC1 C1(NC(C2CCN(C(C)=O)C2)=O)CCN(C(=O)COCCC2CCC2)CCO1 CCC(C)(C(=O)N1CC(NC(=O)C=CC2CCCC2)C(C(F)F)C1)C(N)=O C12(C(=O)Nc3c(Cl)ccc(C)c3)CCC(C(=O)NC3COC(=O)N3)(CC1)CC2 C1(C(=O)NC(C)Cc2cnccn2)CN(C(=O)CN=[N+]=[N-])CC1C1CC1 C1(C(=O)Nc2cccc(Cl)c2)COC2(CCN(C(=O)C(F)Cl)CC2)C1 c1(OC)cc(C(N2CCC(C)(C(=O)NC3CCC(C#N)CC3)C2)=O)cc(Br)c1O c1(NC(C)=O)nc(C(=O)NCC2CC23CCC3)cs1 C(=O)(C(C)(C)C(C)(C)O)NCCCCN(C)C(C1CNC(=O)C1)=O CC1(CC(=O)NC2(CF)CCCC2)CCN1C(=O)CCCn1ccnn1 C(=O)(N=c1cnn(CC(F)F)[nH]1)c1[nH]cc(COC)c1C C1(C(=O)NC2C(CC)CN(C(=O)CCC(=O)N(C)C)CC2)CN2CCCN1CC2 c1(C(N2C(CN(C)C(C3CC(F)(CO)C3)=O)COCC2)=O)cc2sccc2n1C c1(OC)ncc(Cl)cc1C(N1CCC(N(C)C(C2C=CCCC2)=O)CC1)=O C1(C(=O)NC(C2(CNC(C(C)(C)OC)=O)CC2)C)OCCC1C c1(N(C)Cc2cccc(C(=O)NC)c2)ccnc2c(I)cccc12 C(=O)(CC(C(F)(F)F)NC(=O)C(C)(C)OCC)NC(C#C)C(C)OC C1(C(=O)NC(CC)CN(C(=O)Cn2cnnn2)CC)CCCC1CC(C)C c1(C(N2CC(N(C(=O)CC3CCNC3=O)C)C2)=O)ccc(C(C)(C)C)nc1 N1(C(c2cc(OC)ncc2F)C(=O)NCCC2CC2)CCCC2(CNC(=O)C2)C1 n1(CC)ncn(NC(=O)C2(F)CCN(C(=O)Cn3cccn3)C2)c1=O c1(C(c2nnnn2C2CCCC2)NC(C2CCCO2)C(C)C)csc(Br)c1 c1(NC2CC(C(C)C)C2)cc2ccccc2cc1I C1(C(=O)NCC(C(C)(C)C)NC(C(COC)O)=O)CCCC2(CC2)C1 C=CC1CN(C(=O)CC2CCCC(NC(C3CNC(=O)C3)=O)C2)CCO1 O=C(C1=C(Cl)CCOC1)NC1(CF)CCN(C(C2C3CC(=O)CC23)=O)C1 C1(C)(NC(C2CCCC(C(=O)OC)C2)=O)CCN(C(c2ccncc2O)=O)CC1 Cc1ccc(CCC(N2CC(O)(C(F)C(=O)N(C3CCN(C4CC4)C3)C)C2)=O)o1 C(=O)(C1=CC(C)(C)C1)NC(C(=O)N(CC#C)CC)COC(C)C c1(C2N(C(C(C)(O)C3CCC3)=O)CCC2)ccc2[nH]ccc2c1 C1(NC(C(CSC)OC)=O)CC2CC(NC(=O)CCCN=[N+]=[N-])C2C1 c1(C(=O)NCC2C(C)CCN(C(C=C(C)C)=O)C2)cc(O)nc2ncn(C)c12 S(=O)(=O)(c1c(C)noc1C)N1CCCC(C(N2CCC(Br)CC2)C)C1 c1(C(N2C(COC)(CNC(c3cnncc3C)=O)CCC2)=O)cc2scnc2[nH]1 N1(C(c2cc(C3CCC3)[nH]n2)C(=O)NCCCOC)CC=CC(O)C1 c1(NC(C2C=CC(NC(C3CC=CCO3)=O)C2)=O)ncc2c(Cl)cccc2n1 C1(CC(=O)Nc2ncccn2)CCCN(C(=O)CC2CCCOC2)CC1 c1(C(=O)NCCC(CC)(CC)NC(=O)CN(C)C(N)=O)nnc2n1CCCCC2 CCCCC(CCCC)C(=O)N1CC(CNC(C2CCC(C)(C)O2)=O)(OC)C1 c1(C(N(C2CCCN(C(c3csc(O)n3)=O)C2)C)=O)cc2cccn2c(O)n1 Cc1ncc(C=CC(=O)N(C2C3CN(C(=O)CC4(O)CCCOC4)CC23)C)s1 c1(C(=O)OCC)cc(Br)c(CCNC(N2CCC2c2ccncn2)=O)s1 N1(C(C2CC2Cl)=O)CCC(N(C)Cc2c(C)ccs2)CC1 N1(C(c2scc(OC)c2)=O)CC2CCCC(N(C)C(c3cc[n+]([O-])cc3)=O)C2C1 C1(CC)CCCC1(C)C(N1CCOC(CCNC(=O)COCCC(C)C)C1)=O C1(N(C)C(C2Cc3nccn3C2)=O)CCC2CN(C(=O)COc3ccsn3)CC12 c1(C(C)=O)cccc(C(N2CC(N(C(=O)CC(C)C(F)F)C)CC23CC3)=O)c1C c1(CC)cc(NC(C2C=CC(NC(=O)Cc3ccsn3)C2)=O)ccc1C N1(C(C2CCC(CC)C2)=O)CC2(C)CN(C(=O)C(C)(C)CF)CC2(C)C1 C#CCCCCC(C(=O)NC1(C)CC1)N1CCOC2CCN(C)CC12 C1(NC(C2CCC(O)CN2C(=O)Cc2ccns2)=O)C2CCCC1COC2 c1(C(=O)NCC2CN(C(CC(C)(C)C#N)=O)C3C2C3)nc2ccccc2nc1O C(=O)(CCC1CCc2ccccc21)N1CC2CN(C(C3CC(=C)C3)=O)CC2(C)C1 c1(C(=O)NCC(CCOC)NC(C(CC=CC)CC)=O)ccc2c(C)noc2n1 N1(CC(=O)NC2C(NC(C3ON=C(C)C3)=O)CC2)CCC(N(C)C)CC1 c1(C(N2CCN(C(C3CC(C)C(C)CC3)=O)C(C)C2)=O)cccn2nccc12 C(=O)(C(C)C1=CCCC1)N1CC(OCCC(N2CC(CN(C)CC)C2)=O)C1 c1(CNCC(CCCCC)O)cccc2ncoc12 C(=O)(CC(C)C(C)(C)NC(c1cccn1C)=O)N1CC(C(CC)C)C1 CC1(C)COC(C(=O)NC2(CNC(=O)C(F)CC3=CC=CC=CC=N3)CCCCC2)C1 C1(N(C(CNC(=O)OC)=O)C2CC2)C2CC1CN(C(=O)C=CSc1ccccc1)C2 c1(C(N2C(C(=O)NCCC#C)CC(C)C2)=O)cc([N+](=O)[O-])ccc1O c1(C(N(CCC)CCNC(=O)CC2CC(CC)C2)=O)ccc(O)cc1 CCCC(C)(C)C(=O)N(C1CCCN(C(=O)C(C2CCC2)C2CCC2)C1)CC c1(C(=O)NCC(CO)NC(C2(COC)C=CCC2)=O)cc(C)nc2[nH]nc(C)c12 N1(C(c2ccnc(OC)c2F)=O)CC2COCC(C1)C2NC(=O)C(O)CSC C1(C(=O)NCCOCCN(C)C(C2C=CC=CC=C2)=O)CCCCN1S(N)(=O)=O C(=O)(C(O)CF)N(C1CCCCC1)CCNC(=O)Cn1cccn1 c1(C(=O)NC2CC(OC)C2)ccc2cnoc2c1.C12CCC(C1)C(=O)N1CC2C1 c1(CCC(=O)NCCCN(C(=O)C(F)C(C)(C)O)C(C)C)nnc(O)nc1O C(=O)(C(C1=[SH]CCCC1)N1CC(=O)NCC1C(C)C)NCC(=C)C CC1C(C(=O)NC(C)(CNC(=O)CC2CC(C)(C)C2)C(C)C)CCN1C N1(C(c2c(O)cc(F)cc2F)=O)CCC2CN(C(C3CCOC3)=O)CC2CC1 N1(C(C2C(NC(C(n3ncc(C)c3)C)=O)CCC2)=O)CC2(CCC(C(N)=O)O2)C1 Cn1cc(C(=O)NCC(C)(C)C)c(=NC(=O)OCc2ccc(F)cc2)[nH]1 Cc1ncc(Cl)c(C(N2CC3CC(NC(=O)Cc4ccnn4C)C2C3)=O)n1 c1(C(N2Cc3c(-c4ccc(SC)nc4C)n[nH]c3C2)=O)cc(Br)cc2[nH]ncc12 N1(c2n(CC(=O)NC(CC)C)nnn2)CCOC(C(=O)OC)C1C C1(CCOC)CN(C(C2(OC)CCOC2)=O)CCN1C(c1n[nH]cc1Cl)=O c1(C(N(C2CCN(C(=O)CC3C=CCC3)C2)CCO)=O)cnc(O)n(C2CC2)c1=O c1(OC)ccc(Br)c(N)c1C(N1CC(CNC(=O)C=CC(C)(C)SC2CC2)C1)=O c1(C(N2CCCN(C(C(CC)COC)=O)CC2)=O)cc(S(N)(=O)=O)ccc1C C(CNC(c1cn(C(F)F)cn1)=O)(C(=O)NC1(C(O)CO)CC1)N(C)C C#CC1(O)CC(NC)C1.c1(-c2cn(CC(=O)N3C(CC)C3)nn2)c(C)noc1C C1(C(=O)NC(CC(=O)NCCc2c(C)n[nH]c2C)(C)C)CCCCCN1C O(NC(=O)C(C)CCCC(C)(C)N)c1nccc(=NCCC2CCC(CC)CC2)[nH]1 c1(C(C)C(F)(F)F)ccc(C(=O)NC(C)(C)C(C)NC(c2ccc(Cl)[nH]2)=O)cc1 C1(CNC(CC2(N(C)C(c3cc(C#N)cs3)=O)CC2)=O)CC2(CCC2)C1 C=CC(C)C(=O)NC1(C)CC(C(=O)NCC)C1.C12(CC1)C(=O)N2 N1(C(C2CCC(CCC)CC2)=O)CC2CCC1C2NC(=O)CCC(N)=O C1(F)(CNC(CCCCCO)=O)CC(CNC(COC(CC)(C)C)=O)C1.OC c1(COC(c2c(SC)cc(Cl)cc2)=O)cccc2c1ccn2C C(=O)(CCCCc1ccc(Cl)cc1)N1CC(OCCNC(c2cnc(C)s2)=O)C1 CC1CCCC(OCC(=O)NCCC(C)(C)NC(=O)CC(C2CCC2)C2CC2)C1 c1(C(=O)NC(CNC(C(CC)(C)OC)=O)C)cc2sccc2cn1 N1(C(Cn2ccc(=N)[nH]2)=O)CC(NC(C2CC2F)=O)CC2(CC2)C1 c1(NC(=O)N(C2CC2)CC2(CC)CC(C)(C)C2)ccc2ccccc2n1 O=C(CCC(F)F)NC1CCN(C(c2cccn2Cc2cccs2)=O)C1 N1(C(C=CCC)=O)CCOC(CNC(C2CC(F)C(=O)N2)=O)C1 C1(C2CCN(C(c3cn[nH]c3)=O)C2)(NC(C2(OC)CCSC2)=O)CC1 C(C(=O)NCCC(C)(C)CNC(=O)CC1CCOC1)(C(C)C)NC(C)=O C(=O)(CC(N)COC)NC(CC#C)(C)c1ccccc1 N1(C(C(C)N(C(c2ncccc2C)=O)CC)=O)CCC(C)C1(C)C N1(C(C(C)CO)=O)CCC2(CCN(C(c3cn(C)nc3O)=O)CC2)C(C)C1 CC(C)C(F)(CNC(C1CCCC(=O)N1)=O)C(=O)N1CCOC2(CC2)C1 c1(C(N2CC(C(C(N3CCC4CCC4C3)=O)OC)C2)=O)cc(C)nc(C)c1 CCCCS(=O)(=O)NCC1CCCN1c1cc(OCC)ncn1 Cc1cn2c(C(N3CCC(CCNC(c4cscn4)=O)C3)=O)c(Cl)nc2s1 C1(N(C(C(C)NC(=O)OC)=O)C)CN(C(C2CCCOCC2)=O)CC12CC2 c1(C(=O)NCC2(F)CN(C(CC3(C)CC3(F)Cl)=O)C2)cc(Cl)ccc1F c1(C(C(=O)NCCSC)N(CCC(C)C)C)oc2ccc(F)cc2c1C c1(N2CC3CCCN(C(C4CN(C)C(=O)N4)=O)C3C2)ccc([N+](=O)[O-])cc1C#N N1(C(c2c(C)nc(CC)s2)=O)CCC(CNC(C2(COC)C=CCC2)=O)C(C)C1 N1(C(C2N(C(C(C=C)CC)=O)CSC2)=O)CCCC(C)(C#N)C1 C=C(C)C1CN(C(C2(CNC(c3ccn4cncc4c3)=O)CCCCC2)=O)CCO1 c1(C(N(C2CCN(C(c3c(C)ccnc3C)=O)C2)C)=O)cc(F)cc2c1CCC2 C1(NC(c2cn(CC)nc2)=O)CCCC12CN(C(=O)CCNC(=O)CO)C2 C(=O)(C(CNC(=O)CCn1ccnn1)C(C)C)NC(C)Cn1cnnc1 C1(NC(C=COCC)=O)CCC(N2CCN(C(c3oc(C)nc3C)=O)CC2)CC1 C(=O)(C(C)(C)S(C)(=O)=O)N1CC(CNC(c2c(OCC)ccs2)=O)OCCC1 N1(C(=O)COC2CCC2)CCC(C(N2CCCCCC2)=O)C2(CCC2)C1 Cc1nnc2cc(N(C3CCCN(C(=O)COCCCCC(C)C)C3)C)ncn12 Cc1cc(CN2CCCC(CCC(=O)Nc3cnoc3)C2)cnc1Cl CC(C)C(F)(CNC(C1(CCO)CC1)=O)C(=O)NOCC1CCOC1 c1(CC)nc(C(c2nnnn2C2CCCCC2)NC(c2cc(C)on2)C)co1 CCC(CC)C(F)C(=O)N1CCC1OC.C12CC1C(=O)NC2C.C(COC)S N1(C(Cc2c(C)nc[nH]2)=O)CCN(C)C(CNC(c2ccc(C(F)F)cn2)=O)C1 C1(C)(C(N2CC(N(C)C(C3CC3C3CCCO3)=O)C2)=O)CC2(C1)CC(F)(F)C2 c1(C(N2CCCC(CCF)C2)C(=O)Nc2c(C)cccc2)ccnc(S(C)(=O)=O)c1 C(C(CC)(CC)C(=O)N(C)Cc1ccnn1C)NC(C(COCC)N=[N+]=[N-])=O C(=O)(CCCC(=O)N1CC(C)C1C(=O)NCC(C)(O)CSC)OCC C(=O)(CCCCCC(C)(C)C)NC1CCC(NC(C(C(C)O)N(C)C)=O)C1 c1(C(N2C3CC(CNC(C(CC)=CC)=O)CC2CC3)=O)c([N+](=O)[O-])c(C)nn1C c1(OC)nc(N2CCC(O)(CNC(c3ccc(F)c(O)c3)=O)C2)ncc1C C1(C(=O)NCCOC2CN(C(c3cn(CCOC)nc3)=O)C2)CCCCC1C Cc1cnc(C(N2CCN(CC(C)NC(=O)CC3(O)CCOCC3)CC2)=O)cn1 N1(C(CCC(=O)OC)=O)CCC2(CCC2NC(=O)COC2CCN(C)CC2)CC1 C=CCCC(CCC)(c1nnnn1CCOC)NCC1(CSC)CC(F)(F)C1 c1(C(=O)NCC(CNC(CC(CC)CC)=O)O)ccc(F)c(C)c1N c1(C(=O)NCC2CC(NC(=O)C(F)=CC3CC3)C2)ccc(N2CCOC2=O)cc1 N1(C(CCOCC(C)C)=O)CC2CCC(CNC(=O)Cn3ccccc3=O)C2C1 c1(C(N2CC(CNC(C(C(C)C)O)=O)C3(C2)CC3)=O)cc2occ(Br)c2[nH]1 c1(OC)nccc(CC(=O)NC2CC(CNC(c3ccc(C)nc3)=O)C2(C)C)n1 S(=O)(=O)(c1ccc(NCc2nnnn2C2CCC2)cc1Cl)NC(C)C C(C)(C(C(=O)N1CC(C2CCCC3CC23)C1)C(C)C)NC(C1C(OCC)CC1)=O C1(O)(CN(C)C(C2CCCCO2)=O)CCN(C(=O)Cc2cn(C)cn2)C1 C1(C)(C(=O)OC)COC(CNC(c2c(-n3cccn3)cccc2F)=O)C1(C)C CC(C)C(CC(=O)N1CC2(CSC2)C1)NC(C1CCC(O)C1)=O c1(OC(C)C(=O)N(CCC(C(C)C)NC(=O)CC(F)F)C)ccc(Cl)c(Cl)c1 C1(CC=C)(NC(=O)C(C)C(C)O)CCCN(C(=O)C(C)(C)F)C1 C1(C=O)CC=CC(O)C1.n1(CC(=O)N(C)C(C2CC2)C2CC2)cc(CNC(C)=O)nn1 C(=O)(C1=CCc2ccccc21)N1CCN(C(C(C)OCCCC)=O)CC(O)C1 CCC(O)C(C)C(=O)NCCOCC(N1CCC(C)(C(C)C)CC1)=O N1(C(C2C(C)(C)COCC2)=O)CCC2(NC(c3cc4sccc4[nH]3)=O)CCCC12 c1(OC)cc(C)c(C(N2CCC(F)C(NC(c3nc(=N)cc[nH]3)=O)C2)=O)c(C)c1 C(=O)(C1=CCCOC1)N1C(C(=O)NC(c2nn[nH]n2)CC)CCC1C1CC1 C1(NC(c2cnc(CCC)s2)=O)CN(C(c2cnc(C(C)C)[nH]2)=O)CCC1CO C1(C(=O)NCCCCN(C)C(c2ccc(Cl)cc2C(F)F)=O)CC(=O)NC(=O)C1 c1(C2C(C(=O)NC3CCC(NC(C4C5CCOCC45)=O)C3)C2)ccc(Cl)cc1 C1(O)(C(=O)NC2CC(C)(NC(=O)Cc3cccnc3)C2)CCCCC1 CCCC(CC(=O)NC(CCF)COC)NC(=O)CC(O)C(C)C Cc1cnncc1C(=O)N(C)CC1CCCN(C(c2sc(C)cc2Cl)=O)C1 c1(C(=O)NCCOCCNC(CC2N(C)CCOC2)=O)cc2ccccc2cc1Cl c1(OC)cc(CC(C)NC(c2cc(C(=O)OC)c[nH]2)=O)cc(OC)c1C(C)C N1(C(C=CC(CC)=CC)=O)CC2CCN(C(c3cc(C4CC4)nn3C)=O)C2C1 C(=O)(C(CCSC)OC)N(C1CCN(C(c2cccc(F)c2)=O)CC1)CC c1(NC(CC(CC=C)NC(=O)CN(C2CCC2)C)=O)cnc2ccnn2c1 c1(N2C(C)(C)C(NC(=O)C3=CCC3)CC2)ccn2ccnc2n1 C#CCCC(O)C(=O)N(CC(C)NC(=O)CCC(C)(C)c1ccccc1)CC C1(NC(=O)Cc2ccoc2)CN(C(c2cc3[nH]ccc3s2)=O)CC2(CC2)C1 CCC1=NOC(CC(=O)NC(C(=O)NC(C)C(F)F)C(C)C)C1 c1(CC(=O)NCC(C)CNC(c2cn(C3CC3)cn2)=O)sc(O)nc1O N1(C(CC(C)N(CC=C)CCC)=O)CCCCC(C(=O)NC)C1 N1(C(C=CCCC)=O)CCC2(CC2)CC1C(=O)NCc1nc(C)ns1 C(=O)(C(O)(CO)C(F)(F)F)N(CCNC(c1csnc1OC)=O)CC c1(NC(C2C(C(N)=O)CC=CC2)=O)cc([N+](=O)[O-])ccc1F.C12CN(C1)C2=O CCC(C)(C)CC(=O)N1CC2CC2(CNC(=O)Cc2cncs2)C1 C1(C(N2CCCC2c2ccco2)C(=O)NC2COC2)CCCCC1 N1(C(C(n2cc(C#N)cn2)C)=O)CC(C(=O)NC2CN(C)NC2=O)CC1(C)C C1(COC)(NC(=O)C(F)(F)c2ncccn2)CCN(C(C2CCCS2)=O)C1 c1(C(N2CC(C(=O)Nc3ccc(F)c(Cl)c3F)NCC2)=O)ccc2ncnn2c1 c1(C(N2C(CNC(CC(CC)OC)=O)C(C)CC2)=O)cc(F)cc(Br)c1 c1(C(N(C2CCOC2)CC(=O)OC)=O)ccccc1N1CC(C(F)(F)F)OC1=O Nc1c(C(=O)NNC(=O)C2CSCCS2)cc(Cl)nc1F Cc1cc(C)c(-n2nnnc2C(c2nocc2C)NCc2ccncc2)c(C)c1 C1(CNC(C)=O)CCCCC1NC(=O)Cc1cccnc1.C1(C2CCCC2)C(=O)N1 c1(C(=O)NC2(CNC(C(C=C=C)C)=O)CCCCC2)cc(C)nc2c1cnn2C CCC(C)C(O)CC(=O)NC1(C(N2CC(C)S(=O)C(C)C2)=O)CSC1 N1(C(CCC(=O)NCCN(CCCC=C)C)=O)CCc2sccc2C1 C(=O)(C(C)(C)C(F)F)NCC1CCC(CN(C(C2C(COC)C2)=O)C)CC1 C(=O)(C(C)(O)CCN(C)C)NC1CC(CCNC(=O)CC=CCN(C)C)C1 C1(C)(C(=O)NC(CC)CCCO)CCCN(C(c2ccc(Cl)cc2)=O)C1 N1(C(C=C(C)C)=O)CC(CNC(c2n[nH]cc2C)=O)CC(C)C1 C1(C(=O)NCCOCCNC(c2snc(O)c2Cl)=O)C2CCC1(c1cncs1)C2 n1(CC)ncnc1C(=O)NCC1C=CCN1C(=O)CCc1cc(C)on1 N1(C(CCc2nc(C)c(C)o2)=O)CCC(NC(=O)C(C)C(C)(F)F)C(C(N)=O)C1 c1(C(=O)NC(C)CCCCNC(c2n[nH]cc2Cl)=O)c(C2CC2)cccc1F Cc1c(C(N2CC(O)(CNC(=O)Cn3ccsc3=N)C2)=O)oc2c(C)cccc12 C(=O)(CCCC(C)(F)F)NC(CCOC)CNC(=O)CCc1cc(C)sc1C c1(COC)ccsc1C(=O)NC1CCCC1NC(=O)CNC(=O)C1CC1 CC(C1OCCc2ccccc21)NC(=NCC1CC1)NCC1CCCS1 C1(CNC(CCCOC(C)C)=O)N(C(C2OCCN(C)C2=O)=O)CCC1(C)C C1(C(N(C2CCN(C(C)=O)C2)C)=O)C2CCCC2CN1C(=O)CCc1csnn1 c1(NS(Cc2cc(C#N)cc(Br)c2)(=O)=O)ccc2c(n1)OCCO2 c1(C(=O)NC2C(C)(C)CN(C(=O)CC3CC(CF)C3)C2)ccc(F)c2c1OCC2 C(CCC(C)C(=O)N(CC(C)CNC(c1cccc(C)c1N)=O)C)OC CCCS(=O)(=O)C(C)C(=O)NC1CC2CC1N(C(c1cnn(C(C)C)c1)=O)C2 N1(C(CCN(CCC)C)=O)CCN(C(C23CCN(CC2)C3)=O)CC1C C12(CNC(c3c(C)nsc3)=O)CC(CO1)N(C(c1ccccc1O)=O)C2 Cc1cnc(S(C)(=O)=O)nc1N1CC2C(C1)N2C(C1CCc2ccccc2O1)=O c1(C(N2CC3CN(C(C(CCC)O)=O)CC32)=O)ccn2cnnc2c1 C1(NC(C(C)=C2CCC2)=O)CCN(c2nccc(-n3nc(C)cc3C)n2)C12CC2 N1(c2cc(COC)nc(C)n2)CCCC(C2CC2NC(c2ncsc2CC)=O)C1 Cc1cc(N)cnc1C(=O)NC1CCC1NC(=O)C(c1ccc(Cl)cc1F)O C1(C(C(=O)NCC(=C)Br)(C)C)CCCN(C(C2CCC(C)O2)=O)C1 C1(=O)N=C2C=C(N(C)N2)Cn2cc1c(O)nc2=O.c1(COC)noc(C2CC2)n1 C1(CN2CCC(C(N(C(C)CC)CC#C)=O)CC2)CCC2(CCC2)C1 C1(NC(C2COC3COCC23)=O)COC2(CCN(C(=O)C(F)C(F)(F)F)CC2)C1 c1(N(C)C)ccc(C(=O)NCC(C)=CC(=O)NCC2CCNC(=O)C2)nn1 C(C1CCCc2cccnc21)Sc1cnc(NC(N2CCC23CCCCC3)=O)s1 CC1(C(=O)NCc2cc(C(=O)NCC3CCC3(F)F)n[nH]2)CNC(=O)N1 C12CCCCCC1C(=O)N2C.c1(C(=O)O)ncccc1-c1nn[nH]n1.n1(C)cccn1 C#Cc1nc(C(N2CC(NC(c3scnc3C)=O)CC2C)=O)cs1 C=CCCC(C)(C)C(=O)N1CCC(NC(C2CN(C3COC3)C2)=O)C(F)C1 Cc1nc(NCc2nc(C)cn2C)cc(N2CCC(CC(F)F)CC2)n1 C(=O)(C(O)C(C)(C)C)NCC(Cc1ccccc1)NC(c1oc(C)c(CO)c1)=O c1(C(=O)NCCC(=O)OC)cn(C(C(=O)OC)CCN2CC=CCC2)nn1 Cc1noc(-c2ccccc2)c1NC(C1CCCOCC1)=O C(C)(C)(CCC(=O)N1CC(C(=O)NCC2C(C)(C)C2(C)C)C(F)C1)N(C)C C(=O)(CC1=CCCCC1)N1CCC(C(CO)NC(C2(OC)CCC2)=O)CC1 N1(C(c2ccc(CC)cn2)=O)CCC(CNC(=O)C(F)(F)CF)C(F)(F)C1 C1(CNC(C(c2ccc(Cl)cc2)OC)=O)CC(C)(C)CN1C(=O)COCC1CC1 C12(C(N3CC(NC(CCCOCCC)=O)C(F)CC3)=O)CCC(OC)(CC1)CC2 c1(C(=O)NC23CC(CNC(c4ccc(NC)cn4)=O)(OC2)C3)cn(C)ccc1=O c1(CC)sc(C(=O)NC2CN(c3nnc(CCOC)s3)CCO2)cc1C CC1CCCC1(C(=O)NCC1(C2CC2)CCC1)NC(=O)C(c1ccn(C)c1)C C1(NC(c2cnc(C(C)C)s2)=O)CN(C(=O)C(=O)N=S(C)(C)=O)CCC12CCC2 N1(C(C(C)O)=O)CCC2(CCCCC2NC(=O)C(c2cncnc2)C)C1 C(=O)(CCCCCNC(=O)CCn1cccc1)NCCC(CC)CO Cc1cccc2cc(C(=O)NC3CC3CNC(=O)CNC=O)[nH]c12 c1(C(C(=O)NCCSC)N2CCC2c2ccccc2C)cc2ncccc2s1 Cc1cc2ccc(C(N3CC4CCN(C(c5ccc(C)n5C)=O)CC34)=O)cn2c1 N1(c2cc(CN3CC(CC(=O)NC4CC(=O)N4)C3)sc2)CCCS1(=O)=O Cc1nccc(C(N2CC=CC2C(N2CC(N3CCCCC3)C2)=O)=O)c1N CN1CC=C(C(=O)NCC(O)CNC(=O)COc2cc(Cl)ccc2Cl)C1 C1(CCC(=O)NC(C2CN(C(c3ncc(C)o3)=O)C2)C)CCC(=O)NC1 c1(OC)ccc(C2(C(=O)NC3CCCN(C(=O)COC(F)(F)F)C3)CC(O)C2)cc1 CC1(C)OCCC1C(=O)NCC(CO)NC(=O)CNS(C)(=O)=O CCC(C)CC(C)C(=O)N1CCC(CCC2CC2)(C(=O)NC(CO)C(=O)OC)CC1 N1(C(c2c(C(C)C)nccc2)=O)CCC(F)C(NC(C2(C(N)=O)CC2)=O)C1 CC1CCCn2ncc(C(=O)NC(CNC(=O)C=Cc3ccnn3C)C(C)(C)C)c21 CC1CCC(F)(C(N2CC(NC(=O)COc3cc(F)cc(Cl)c3)C(C)C2)=O)CC1 C1(CC(=O)N(CCC)CCNC(=O)CCOCCS)CCCCC1C.C(C)(C)C C(=O)(CC1=CCCCC1)N1CCCC(C(C(=O)NC(C(C)C)(C)C)C)C1 CC1(C)CC(C(=O)NCC2CC3CCC3C2)CN(C(=O)C=Cc2cncs2)C1 c1(C(CNC(c2ccc(COC)cc2)=O)NC(=O)CSC)ccc(F)cc1F C1(F)(C(N2CC3CN(C(Cc4ccc(C)c(C)c4)=O)CC32)=O)CCCCC1(F)F c1(C(N(CCCNC(c2cccc(F)c2)=O)CC)=O)cnn2cccc(C)c12 CC1CN(c2ncnc(Cl)c2CO)CCC1NC(c1cc(C2CC2)n(C)n1)=O c1(C(=O)OC)n[nH]cc1COC(C1CCC(c2ccccc2)C1)=O c1(CCC)nnsc1C(=O)NC(C)CCNC(C1(C2CC2)CCCO1)=O CC(C)(C(=O)NCC1(F)CC(NC(C2OCC2(C)C)=O)C1)C(F)F N1(C(c2c(CC)scn2)=O)CCC(CNC(C2CC23CC(O)C3)=O)C1(C)C Cc1c(C(=O)NCC2CN(C(C3CC4CCCN(C3)C4)=O)C2)ccc2cncn12 c1(OC)cc(C(=O)NC2CCN(C(=O)C=CC3CC3)C2)cnc1Cl C1(c2n(CCCSCC)nnn2)C(C)CCC(=O)O1.C1C(=O)N1C.C(C)(C)OC c1(C(C)(C)C(=O)NCCCCCCNC(=O)CC2(C)CC2F)cc(F)cc(Cl)c1 CCCC(CCNC(C1C2CN(Cc3cccc(OC)c3)CC12)=O)CCC c1(C(=O)NCC2N(C(C3CC(C)OC3C)=O)CCCC2)cc(O)cnc1N C1(CC(=O)NC(C)(COCc2ccccc2)CO)Cn2ccnc2NC1=O N1(C(N(c2c(C)c(Cl)ccc2)C23C(=O)C4CC2C3C4)=O)CCN2C(=O)C(C)CC2C1 C(=O)(C(CC(C)C)NC(=O)COC1CCCOC1)NCc1cc(C)sc1 CC1(C(=O)N(CCCNC(=O)CCC2CCCOC2)C2CC2)C=CCCC1 C(=O)(C1=CCc2ccccc21)NCc1nnc(C(=O)OCC)s1 c1(C(=O)NC(CCNC(c2cn(C)c(Br)c2)=O)(C)C)ccc(=O)n(C)c1 C(=O)(CC(P(C)(C)=O)P(C)(C)=O)N(C)CC1(O)CN(C(C2C(C)OCCC2)=O)C1 C12(CN)CCC(CNC(=O)CCCc3nncn3Cc3ccccc3)(CC1)OC2 C1(CC(=O)N(C(CSC)C)C)COCCN1C(c1ccsc1C)=O n1(CC)nc(C(=O)NC(C2CN(C(=O)CC3CCCCN3C)C2)C)c(Br)n1 O=C1CCCC(C(=O)NCCC2(O)CN(C(c3cscc3C(F)F)=O)C2)N1 C(=O)(CC(C)(C)CC(=O)OCc1nsc(OC)n1)OC(C12CC1CN(CC)C2)=O c1(NCCCOc2c(C)cccc2)ccc(S(=O)(=O)NC(CO)C(C)C)c(Cl)c1 C(N=c1ccnc(N2CCC(c3ccc(F)c(Cl)c3)CC2)[nH]1)N1C(=O)NC(=O)C1 N1(C(COCCOCC)=O)CC(C(=O)NCC2CC2(C)C)C(C)(C)C1 C1(C(=O)NCCCN(C)C(c2c(C(F)(F)F)cnn2C)=O)C2CCCCCCC12 Cc1cccc2c(CC(=O)NC(C)CC(C)NC(=O)Cn3ccnc3C)c[nH]c12 c1(SC)c(C(N2CC(NC(C3(S(C)(=O)=O)CC3)=O)C(C(F)F)C2)=O)cccc1F Cc1[nH]nc2cc(CNc3nnn(CC4CCCO4)c3C)ccc12 C1(CN(C(C2CC2(F)Br)=O)CC)CC(NC(=O)OC(C)(C)C)CCO1 C=CC1CN(C(=O)CCN(C(=O)CCn2cnc(=N)[nH]2)C2CC2)C1 C1(CN(C(=O)CC2CC(NC(c3ccccc3C3CC3)=O)C2)C)NC(=O)NC1=O c1(OCC)ccnc(C(=O)NCCSCc2nnnn2-c2ccccc2)c1O C(C(C)(CNC(CC(F)(F)Cl)=O)OC)NC(C(C)OCCCC)=O N#Cc1ccc(C(N2CC3CC3(CNC(c3ccc(F)cc3O)=O)C2)=O)c(F)c1F N1(C(c2[nH]cc(CC)c2)=O)CCC(CC)(NC(C2CCOC(C)C2)=O)CC1 C1(CN(C(C(C)OCCCC)=O)C2CC2)CCCN1C(C1CCC(CCC)C1)=O c1(C(N2CCN(C(C3C(C(=O)OC)C3)=O)CC2CO)=O)nc2ncc(C)cn2n1 CC(CC1CC1)C(=O)N1CCCC1C1CCN(C(C2(c3ccncc3)CC2)=O)C1 C1(CC=C)(NC(=O)C(N2CCCC2C(=O)NC)=O)CCN(C(C2C=C2C)=O)C1 C#CC1(NC(C2(C(C)NC(c3coc4c3COC4)=O)CC2)=O)CC(F)(F)C1 N1(C(COCCC#C)=O)CC(CNC(=O)C(CC)NC(N)=O)C(C)C1 CC(CC(=O)N1CC2CC2(CNC(c2cccc3cc[nH]c23)=O)C1)CC(C)(C)C C1(N(C(C(CC)N(C(=O)CSC)C)=O)CC)CCCCCC1 C1(OC)CN(C(=O)COC2CCC2)CC1NC(C1CC1c1nccn1C)=O C(=O)(C1=CNC2=NCCCN12)NC(C1CN(C(C2CCCN2C)=O)CCO1)C C12(COC)CN(C(=O)Cc3cc(C)no3)C(CNC(=O)C=CS(C)=O)(C1)C2 c1(C(=O)NC2CCC(C)N(C(c3ccncc3Cl)=O)C2)cc2n(n1)CCNC2=O C=C=C(C)CC(=O)N1CCCC(N(C(=O)CCCCc2ccccc2OC)C)C1 N1(C(c2ccc(CC)s2)=O)CC2CCC1C1CN(C(C3CCC(=O)NC3)=O)CC21 N1(C(C2CC=CN(C(C(C)n3cccn3)=O)C2)=O)CCC2COCC2C1 C1(CNC(c2c(OC)cc(F)cc2)=O)(CNC(=O)CC(C)C)CC2CCCC2C1 C1(CCC)(C(N2CCC2COCCNC(=O)C(C)C2CCCO2)=O)CCNC1=O C(C)(C)(C#Cc1cn(Cc2nsc3c(F)cccc23)nn1)C(C(C(CC)C)=O)=O N1(C(C(C)=CC=O)=O)CCCC(NC(=O)CC2(n3ccnc3)CC2)CC1.C(C)C c1(CC(N2CCCC(COC)C2)=O)cccc(C(=O)O)c1 N1(C(C=CC(C)NC(=O)C2=NOC(C)C2)=O)CCn2nncc2C1 CC1=C(C(=O)NCC2C=CCN2C(=O)CCNC(N)=O)CCCC1 C1(CCNC(CC2N(C(C(C=C)OC)=O)CC2)=O)CCC2(CC2)CO1 N1(C(c2c(CC)[nH]cc2)=O)CC2CCN(C(=O)CC(O)C(Cl)(Cl)Cl)C2C1 C1(C2CN(C(=O)Cn3cnc(=N)[nH]3)C2)(OC)CC1.c12nc(co1)C(=O)NC2 C1(CNC(C2C(C#C)C2)=O)C2CC1N(C(=O)C(c1cccc(Cl)c1)(C)C)C2 C1(NC(c2c(OC)n[nH]c2)=O)CC(C(=O)N(CCO)CCc2ccccc2)C1(C)C c1(CNC(C2CC(NCc3cc(Br)c[nH]3)C2)=O)cc(Br)cc(I)c1 c1(C(N2C3C(NC(c4cn5c(n4)CCOC5)=O)C(C3)C2)=O)cc2ncccc2[nH]1 c1(CC)cc(C(=O)NCC2(NC(c3cnn(C)n3)=O)CCOC2)c(C)nn1 c1(NC(C2C3CN(c4ncc(Br)cn4)CC23)=O)cc(F)cc2[nH]ccc12 C(=O)(C(CC(C)C)N(C)C(C12CCC(C1)C2)=O)NCC(CC)C(C)C CC1=C(F)CN(C(C2CCCC2CNC(c2ccc(O)cc2)=O)=O)CC1 c1(CC(=O)NC2CCC(NC(COCC(C)(C)C)=O)CC2)cnn2c1CCCC2 C(=O)(CCCC(C)CC)NC1(CCC)CCCN(C(C2(C)CCOCC2)=O)C1 C1(NC(c2cc(Cl)cs2)=O)CCN(C(c2cc(C(F)F)ncn2)=O)C12CC2 N1(C(C2(CC)COC2)=O)C2CCC1CN(C(c1ccc(SC)c(Br)c1)=O)C2 CCCCC(CC(=O)NCCCC1C=NNC1=O)NC(C1CN(C)C1)=O N1(C(NOCC=C)=O)CC(O)CCC1CNS(C)(=O)=O C12CC3(C1)CN(C3)C2=O.O=C(C(Cl)=CCl)Nc1cc(CN2CCCC2)on1 c1(OC)nc(=NCC(C2CCCCC2)NC(=O)CC(C)SC)[nH]c2[nH]cnc12 c1(C(=O)NCC2CCN(C(C3(C)N(C(C)=O)CCC3)=O)C2)cnn2ccsc12 CC1CC=C(C(=O)N2CCN(S(=O)(=O)Cc3ccc(F)cc3)C(C)C2)CC1 c1(C(N2CCCC(CN(C(CCC#CC)=O)C)C2)=O)nccc2occc12 CC1(CNC(c2ccc(F)c(F)c2)=O)CCCC(NC(C2CC(=C3CC3)C2)=O)C1 C(=O)(CC(C)C(=O)OC)N1CCC(C(C)(C)C)(CNC(CCN(C)CC)=O)C1 Cc1noc(NC(=O)CC2CN(C(c3ccc(N4CCCC4)cc3)=O)C2)c1Br C(=O)(CCCC(C)(C)C)NC1CCCN(C(COc2n(C)nc(C(F)F)c2)=O)CC1 c1(C(=O)OC)cc(C(N2CCCC2C(C)NC(=O)C(C(C)C)OC)=O)ccn1 C1(C(NOCCOCC)=O)CCCN(C(c2ncncc2OCC)=O)C1 C1(CNC(C2(C)CC2)=O)CCCN(C(C2CCOC2(C)C)=O)C1 C1(CNC(C23CC(C)C2C3)=O)CCC2CN(C(c3cccc(Cl)c3Cl)=O)CCC12 C1(C(=O)NCC(CC)N(C)C)CCNC(=O)C1.C1(=O)CC(CC)N1 CC1CC(NC(=O)CS(N)(=O)=O)CN(C(=O)C=Cc2cccs2)C1 S(=O)(=O)(c1cccc(Cl)c1Cl)N1CC2CN(S(CCOC)(=O)=O)C2C1 CC(=O)CC(C)(C)CC(=O)NC1CCCC2CN(c3nc(C(C)C)ns3)CC12 CC1(C)CCCC(c2ccc(Br)cc2C(N2CCOCC(C(C)(C)C)C2)=O)C1 N1(C(C(CC=C)NC(C)=O)=O)CCC2(C1)CN(C(c1c(Cl)cncc1Cl)=O)C2 CCC(c1ccc(C)cc1)=CC(N1CC(NC(=O)C(C)(CC)OC)CC(F)C1)=O CCCC(CCCNC(=O)Cc1csc(C)n1)NC(c1cscc1Cl)=O C1(CC(=O)NCc2cc(OCC#C)n[nH]2)CCCCN1C(c1ccccc1)=O CC1CCC=C1C(=O)NC1C2CC3C(C2)C13C(=O)NCc1nccc(O)n1 c1(NC(=O)CC2(CO)CCCN(C(C3CC3F)=O)C2)ccc([N+](=O)[O-])cc1Cl c1(COC)cc(-c2cnc(NC(=O)Cc3ccc(F)cc3Br)c(O)c2)ccc1O C(=O)(C(CC(C)C)NC(=O)C1C2CCCN2N1)OC.c1(CO)ccn(C(C)C)n1 c1(C(=O)NCC2C(C(N3C(C)CC3(C)C)=O)CCC2)cccc2ccoc12 C1(C(=O)NC(C)(CNC(=O)CO)C2CCC2)CCCC1(F)F C(=O)(C1=NNC(C(F)(F)F)C1)N1CCC(CNC(C2N(C)CC(F)C2)=O)(CO)C1 C1(CC)(NC(C2CC(O)CN2C(C)=O)=O)CCCN(C(=O)CCC=CC(C)C)C1 CC1ON=C(C(=O)N2CCC(N3CCN(c4ccccc4)C3=O)CC2)C1C CN1CCC(C)(C(=O)NCCC2CCCN2C(C2(C)COC2)=O)CC1 C1(C(=O)NCc2ccc(C)cn2)C(C)OCCN1C(c1ncoc1C)=O C(CC(C)OC)(C(=O)NC1CC1F)NC(c1c(CC)c[nH]n1)=O c1(CCC(=O)N(C2CCN(C(=O)CCCCC3CC3)C2)C)n[nH]c2ccccc12 C(CCO)(C(=O)NCC(C)(O)CNC(=O)COCCF)N(C)C.C(=O)(C1CC1)N n1(CC(C)C)nccc1C(=O)N(C)CCNC(=O)CC1CC12CC2 c1(NC(C2CCCN2Cc2sc(Cl)nc2Cl)=O)cccc2nc[nH]c12 Cc1[nH]c(C#N)cc1C(=O)NC1CCC(CNC(C2CCC(N=[N+]=[N-])C2)=O)C1 C=CCCCC(C(=O)NCc1cc(O)ccc1F)NC(c1cncc(O)c1)=O C1(C(=O)NCc2cccc(C#N)n2)CC2(CCC2)CN1C(c1cc(O)ns1)=O Cc1nc(C)c(CN2CCC(COC(F)(F)F)CC2)s1 C1(NC(CCCCN(C(C)C)C)=O)CCCCCC1NC(c1ccnnc1O)=O C(=O)(CC(O)CNC(=O)C(C(C)C)N(C)C)N(CC#C)Cc1ccco1 Cc1nn(C)c(C)c1C(=O)NC(C)CCc1ccccn1.C1(=O)CO1 C(C)(C)(CCNC(=O)C(CC1CCC1)NC(C1C=C(C)CS1)=O)OC N1(C(c2c(C)nco2)=O)CCc2nc(O)cc(C(=O)NC3(CO)CC(C)C3)c2C1 C1(O)(CNC(C(C(C)C)C)=O)CCCN(C(=O)CSc2cn[nH]c2)CC1 Cc1ccc(C2CC2C(=O)NCC(CO)NC(C2C3CCCOC23)=O)cc1Cl C1(NC(c2c(OC)csc2)=O)CCCCCC1NC(C1(C2CC2)CCCO1)=O C1(C2CCCCC2)(NC(COC2CCN(C(CN(C3CCC3)C)=O)C2)=O)CC1 C(=O)(C(F)CC(C)(C)NC(c1cccnc1CC)=O)NCc1c(CC)nco1 N1(C(CCC=C(C)C)=O)CC(CNC(c2cc3c[nH]cnc-3n2)=O)OC(C)(C)C1 CC(F)(F)C(F)(F)CC(=O)OCCCC1(C)CCCC1 C1(CC(=O)N(CC(C(=O)NC)C)C)CN(C(C2COCCO2)=O)CC1C c1(C(=O)NC2C(C)(C)C(C(N3CCC4(C=C4)CC3)=O)C2)c(O)ccc(F)c1F N1(C(c2ccn(C)n2)=O)C2CCC(C2)C1C(=O)NC(CO)C(N)=O Cc1cc(Br)c(F)cc1C(=O)NC1CC(C(=O)Nc2cnc(Cl)cc2C#N)C1 C(=O)(C(C)CC(=O)N(C(C)CNC(=O)Cc1ccsn1)C)OC N1(C(C)=O)CCC(NC(=O)CCC2CCCN2C(=O)Cc2cnsc2)C1 C(=O)(C(C(C)(C)O)NC(C1CCN(CC)C1)=O)NC1(C#C)CC1 CC1(C)CCN(C(=O)CN2C(=O)CCC2=O)C1C(=O)NCC1CC2CC2C1 c1(C(N2CCCC(C)C2CNC(=O)C2=CCCS2)=O)cn2cc(F)ccc2n1 C(=O)(CCCCC(C)C)N1CCC(CNC(C2(C(COC)C)CC2)=O)C1 CC(C(=O)NCC(C1CCCCC1)NC(=O)COC1CCC1)P(C)(C)=O C1(C(=O)NCCC2N(c3nnn(C)n3)CCSC2)CCOC2(CCCC2)C1 N1(C(C2CCC(CCC)CC2)=O)CCC(NC(=O)Cc2nncs2)C(F)C1 N1(C(Cc2c(C)noc2Cl)=O)CCC(C2CC2)(CNC(=O)C(C)NC(C)(C)C)C1 N1(C(c2cn(CC(N)=O)nn2)=O)CC2CCC1C2NC(c1c(F)cccc1F)=O C1(C(=O)NC2C(c3ccccc3)C2(F)F)CCn2c(cnc2C2CCC2)C1 c1(OC)cc(F)c(F)cc1C(=O)NC1(C)CN(C(=O)C(C)(C)CSC)C1 C1(CNC(C=CC(C)C)=O)CC(NC(c2nccnc2N)=O)C1(C)C CC(N=c1[nH]c(N2CC3CC2C2CC32)nc2c1CCC2)C(F)F C=CCC(C)(C)CN(C(=O)C(Cc1cnc[nH]1)C1CC1)C c1(C(=O)NC(CNC(COC(C)(C)C)=O)CO)cnc2nccn2c1 Cc1nn(C)c(Br)c1C(=O)NC1CC1NC(C1CC2C(C1)C2(F)F)=O C1(C(N)=O)CCC(C)CC1.CC1=NC(C(N2CC3(C2)C(=O)NC3)=O)CS1 CC1CCN(CC(=O)NCC(C)(C)NC(c2coc(NS(C)(=O)=O)c2)=O)C1 N1(C(Cc2onc(C)n2)=O)CCCC(CC(N2CCCC(CC(N)=O)C2)=O)CC1 CCCC(C)(O)CC(=O)NCCCNC(=O)CCSCc1csc(C)n1 C1(C(N2CC(SCC)C2)=O)CCN(C(=O)C(CC)CCC(C)C)O1 Cc1cccc2c1CN(C(=O)NCCOc1cc(Cl)ccc1Cl)C2 N1(C(COC(C)C)=O)CC(NC(c2ccccc2C(C)(C)C)=O)C(O)C1 c1(C(N2CCC(c3cn(-c4cscn4)nn3)C2)=O)cc(OC2CC2)ccc1Cl C1(OC)CC(NC(=O)CS(=O)(=O)CCC(C)C)C12CCN(C(=O)CCF)CC2 c1(NC(=O)NCC#CCNC(C2(CC)CC2)=O)c[nH]c2ccccc12 C1(C)(CNC(CCCOC(C)C)=O)CCN(C(=O)CC2(C#N)CCC2)CC1 CCC(C)CC(=O)NC(c1nc(C(=O)NCc2cccnc2F)co1)C N1(C(c2ccn3c2CCC3)=O)CCC2(CCCN(C(=O)COC3CC=CC3)C2)C1 C1(CNC(C2CSCC(=O)N2)=O)CC(C(=O)NC2CN(C3CCC3)C2)=NO1 Cc1cccc(Br)c1C(C(=O)N(C)C)NC(=O)CSCC(N)=O N1(C(c2cn(CCC)nc2)=O)CCN(C)CC1CNC(C1(C#N)CCOC1)=O c1(N2CC(C)(CC(=O)Nc3ncc(C4CC4)s3)C2)ncc2cc(Br)cnc2n1 c1(C(=O)NCCOCCNC(c2cnn(CC)n2)=O)cccc2c1OC(C)C2 Cc1ccc(C23CC(CCN2C(c2ccc4c(c2)CCC4)=O)C3)cc1 N1(C(=O)CC2(CO)CC2)CCOC2(C1)CN(C(C1CCCC13CC3)=O)C2 C#CC1CCN(C(c2ccc(CNC(c3cc(OC)no3)=O)s2)=O)C1 Cc1cc(Br)ccc1N(c1ccc(F)cn1)C(N1CC(Oc2cscc2Br)C1)=O C1(C(=O)NC2CC3CN(C(Cc4[nH]c(=N)sc4)=O)CC32)CCC2(CCC2)CC1 c1(OC)cc(S(=O)(=O)N2CC3CCNCC23)c(Cl)cn1 CCC(CCCC(=O)Nc1cccc(Cl)c1C)NC(=O)CC1CSC1 N12CCCC(C1)C2=O.N1(CCC(C)(C)OC)CCN(C(=O)CCCN(C)C)CC1 C1(CC(F)(F)F)CCN(Cc2cccc(F)c2Cl)C2(CC2)C1 N1(C(C2(SC)CC2)=O)CCC(CC(C(F)F)NC(c2ccc(F)cn2)=O)CC1 CC1CN(C(=O)CC2COCC(C)O2)CC(C(=O)NC(C23CCC(CC2)C3)C)O1 CN1CCN(C(c2ccc(Cl)nc2)=O)CC1CNC(=O)C(F)(F)C1CC1 C1(NC(C=CCN(CC#C)C)=O)CC2CC1N(C(=O)CN1CCCC1=O)C2 N(C(=NCc1cccc(OC)n1)N1CCC2NC(=O)OCC2C1)CC(CC)SC C1(CNC(C2(C(=O)NC)CC2)=O)CC2(C1)CN(C(=O)Cc1cnccc1Cl)C2 C1(C(N2CC(N(C(C3ON=C(C(C)C)C3)=O)C)C2)=O)CCc2c(cnn2C)C1 c1(C(N2CC(O)CC(NC(c3c(CC)ocn3)=O)C2)=O)ncn2ccccc12 Cc1ccc(F)c(C(N2CCC(NC(=O)CC3C=CCC3)C(C(N)=O)C2)=O)n1 N1(C(CC(CC)C2CCCN2C(=O)CC(C)(C)C)=O)CC2ON=C(CCOC)C2C1 N1(C(CN(CCC)C)=O)CCC2C(CCCN2C(c2cc(N)cc(O)c2C)=O)C1 Cc1cc(C)n(-c2cc(NC(c3ccccn3)C(C)C)ncn2)n1 C(CC(C)(C)CC(=O)N1CCC(C2CCCN2C(=O)Cc2cnn(C)n2)C1)OC c1(C(C(=O)NC2CN(C(CC=CC)=O)CC(O)C2)=O)cc(F)c(F)cc1F c1(NC(C2C=CC(NCc3c(C)cc(OC)nc3)C2)=O)ncc([N+](=O)[O-])cc1O C(c1cnc[nH]1)=C(C)C(=O)NCC(C)NC(=O)CCc1nc(C2CC2)no1 C1(OC)CC2(C1)CC(C(=O)NCC(C1CC1)NC(C1CCOC1C)=O)C2 CCCC(CNC(=O)CC1(NC(c2ccn(C)c2)=O)CCC1)CCO Cc1cc(C(=O)NCC(CO)NC(=O)CC(O)C(C)C)c(C)n1-c1ccccc1 N1(C(C2CCCC(=O)N2)=O)CCC2(CCCCN(C(=O)C(O)C(F)F)C2)C1 CCC(C(=O)N1CC(C)(C)OCC1CNC(=O)Cn1ccnc1C)C(C)(C)CC N1(C(C(CC2C(C)C2)(C)C)=O)CC2CCCC(NC(C3(CO)COC3)=O)C2C1 Cc1sc(O)nc1C(=O)NCC(C)(CO)NC(=O)Cc1csc(-c2ccsc2)n1 c1(C(N(CCOCCNC(CCSCC(C)C)=O)C)=O)cccc2c1SCCC2 Cn1cncc1C=CC(=O)NCc1ncccc1C(=O)NC(CO)C(C)(C)C c1(SC)cc(C(=O)N(C2CCNC2=O)Cc2cn(CC3CC3)nn2)co1 CCCC(O)CC(=O)NCCCCC1CN(C(=O)C(C)(C)C(C)O)C1 C12(CCNC(CCC3CNC(=O)N3)=O)CCC(CC1)N(C(C1CC(O)C1)=O)C2 N1(C(CN(CC)CC)=O)CCC2(CCCCN(C(=O)C(C3CC3)SC)C2)C1.C1CC1 CC(C)C(CCN(C)C(C1CC(=O)N(C(C)C)C1)=O)NC(c1nncs1)=O C12(C(CCC)=O)C3C(=O)C4C5CC(C14)C2C35.C1(NCC(=O)N(CC)C=O)CCSC1.N C1(C(=O)NCCOC2CCN(C(c3c(C)n[nH]c3)=O)C2)CN2CCN1CC2C N1(C(C(c2cccc(Cl)c2)N(C)C)=O)CC2CC(NC(=O)CN3CCCC3)C1C2 C12(COC(c3ccnn3C3CC3)=O)CCC1CCN2 c1(C(N2CCCN(C(CC(C)OC)=O)CC2)=O)cnc2c(ccn2C)c1 c1(C(N(CC(CN(C)C(c2cnc(S)[nH]2)=O)O)C)=O)cccnc1O C(c1ccc(C(F)F)o1)=CC(=O)N(C1CN(C(c2ccc(F)s2)=O)CC1F)C Cc1cc(C)c(C(=O)NC2CCCN(C(=O)C(C)(C)COC(C)C)CC2)cc1C N1(C(C(CCOC)C)=O)CCCN(C(c2cn(CC3CC3)nn2)=O)CC1 N1(C(c2c(CC)c[nH]n2)=O)CC2CC1CC2NC(C1CCCN1C(C)=O)=O CCCC(C)(C)C(=O)NC1C=CC(C(=O)Nc2ncc(CC)cc2C)C1 c1(C(N2CC(C(C)(C)C(=O)NCCC3=CCOCC3)(O)C2)=O)ccc2cncn2c1 C(=O)(C(=O)C(C)(C)C)NCC(C(=O)N(CC(C1CC1)OC)C)C N1(C(CCC=C)=O)CCN(C(C2CCC2C(C)(C)C)=O)C(c2cccc(F)c2)C1 c1(C(=O)NCCCNC(CCC2CCC(C)O2)=O)ccc2c(O)n[nH]c2c1 c1(C(N2C(c3n(CC)c4c(n3)cccc4)CCC2)=O)ccc(F)cc1C#N Cc1ccc(C(=O)N(CCC(=O)NCC(C)O)CCOOCC2CC2)cn1.C CC(CCC(=O)NC1CC(CCNC(=O)Cc2c[nH]nc2O)C1)N(C)C CC1(C)CC(NC(c2n[nH]c(O)n2)=O)CN(C(C2CC3CC3C2)=O)C1 N(C(=NCCc1ccc(Cl)cc1Cl)N(C)Cc1ccn(C)n1)CC(=C)C c1(CC(=O)NC(CC)CNC(C2CCN(CC)C2)=O)ccc(C(N)=O)nc1 CC(C)CC(O)C(=O)NCCC1(NC(c2coc(C3CCCC3)n2)=O)CCC1 C1(C(=O)NCCCC2N(C(C(C)n3cncn3)=O)CCC2)CCC(=O)N1C n1(CC(C)(C)C)nc(-c2cncc(Br)c2)nc1C1CCC(F)C1 C1(C(=O)NCc2cn(CC(=O)NCc3cc(COC)no3)nn2)C2CCC(C2)C1C c1(C(=O)OCC)cc(C(=O)NC2(COC)CC2)cc([N+](=O)[O-])c1 N1(C(c2c(C(=O)OC)ccs2)=O)CC(c2cn(CC3CC4CC4C3)nn2)C(O)C1 c1(CCC)c(C(=O)NC2CCCC(NC(=O)C(C3CCC3)OC)C2)nnn1CC c1(CC(=O)Nc2ccnn2C(F)(F)F)ccc(CO)cc1.C12CCCN(C1)C2=O Cc1ccc(C(=O)NCCC2(NC(C3C(C)C3C)=O)CCCC2)c(O)c1 c1(SC)cccc(C(=O)N(C2CCCC2)CCNC(=O)CN2CCC(C)CC2)n1 c1(SCC(c2n(CCC)nnn2)(C)NC(c2ccsc2)C)cccc(Cl)c1 c1(CNC(C2C(=C)C2)=O)nonc1CC.C1(=O)C(C)(C)C2CCCN12 c1(CC)ccccc1NC(=O)CC1CN(C(=O)CCOC2CCOCC2)C2CC12 N1(C(c2c(NCC)cccn2)=O)CCC2CCN(C(=O)CCCCSC)C2C1 C1(NC(C2C(C)(C)CCCC2)=O)COC2(C1)CN(C(C1CC=CCC1)=O)C2 C1(CCC)CN(C(C2CCC3(CC3)C2)=O)CC1NC(c1ccc(CO)o1)=O C1(CCNC(C2(CCCC)CCC2)=O)CSCCN1C(=O)C(C)OC1CCCC1 N1(C(c2n(CC)nc(C)c2)=O)CC2CC(O)C1C2NC(=O)C=CS(C)=O C(=O)(NNc1cc(F)cc(Cl)c1)c1c(-c2c(Br)ccc(C#N)c2)n[nH]c1 N1(C(CN(C(C)=O)C)=O)CCC(CNC(=O)CSc2nnnn2C)C(C)C1 c1(C(N2CC(C)CC(NC(COC(CC)(C)C)=O)C2)=O)ccsc1S(N)(=O)=O C1(NC(c2cc(C(C)=O)oc2)=O)CN(C(C2CC2Br)=O)CC2(CC2)C1 CCCCN=C(NCC(N1CCOC(C)(C)C1)CSC)NC1CCCCC1C Nc1cncc(C(=O)NC2CC2NC(c2c[nH]c(-c3ccc(Cl)cc3)n2)=O)c1 CC(C(C)C(=O)NOCC1CCOCC1)NC(c1cn(C)c(=O)cn1)=O C1(N(C(=O)C(F)C2CCOC2)C)CCN(C(c2cc(Cl)c[nH]2)=O)CC1 C(=O)(C1=Cc2cc(F)ccc2OC1)NC1CC(CNC(c2snc(C)c2N)=O)C1 C1(CC)CCN(C(=O)C2=CCCS2)C1CNC(=O)CCN(S(C)(=O)=O)C N1(C(CCc2cc(C)no2)=O)CC2CCC2(CCNC(=O)CCC(N)=O)C1 C1(SC)CCCN(C(c2cccc(F)c2)C(=O)NCC(F)F)C1 CC1CC(NC(c2csc3nnsc23)=O)CCN1C(c1cnns1)=O CC(CC(=O)N1CC2CN(C(=O)Cc3cnc4cccnn34)CCC12)C(F)(F)F C12(CNC(c3cn(C4CCC4)nn3)=O)CCCCC1C2.C12CC(C1)CCNC2=O CC1CC(NC(C2CCN(CCO)C(=O)C2)=O)CCN1C(=O)C=C(Cl)Cl C(=O)(C(CC1CC1)NC(c1cncs1)=O)N(CCC)CCC c1(CNC(C2CCC(NC(CCCCC)=O)C2)=O)ccnc(NC(=O)COC)c1 C#Cc1cccc(CC(=O)NCC(C)C(N2CCCC(O)(C(C)C)C2)=O)c1 C12(NC(C(C)OC)=O)CCCC1N(C(=O)C=C(C)c1cccs1)CCC2 CC1CC(NC(C2CN(C(N)=O)C2)=O)CCC1C CC1CCN(C(=O)CCN2CCC2)CC1NC(C1C2(CC2)C12CC2)=O CCCC(CNC(C1CCCCN1C(=O)C(C)(C)C)=O)CCC C1(c2c(C)cc(C3CC3)c(Cl)c2)COC2(CCN(C(=O)CCCC(C)C)CC2)C1 C1(C(=O)NCC2N(C(CCCC(N)=O)=O)CC3(CCC3)C2)Cc2nccnc2C1 c1(C(=O)NCC(C(=O)N(CC(O)CO)CC)CC2CCCC2)ncccc1Cl C1(NC(=O)C=CC2CCC2)CN(C(=O)C(c2ccc(F)cc2)(F)F)CC12CC2 C(CC(=O)N1CCCC(C#N)C1)(C(N)=O)n1cc(-c2nc(C)sc2C)nn1 c1(CC(CO)NC(c2ccc(C(=O)OC)nc2)=O)ccc(Cl)cc1Cl C1(C(=O)NC2(CNC(c3ccc(-c4ccsc4)nc3)=O)CC2)CC2CCCC2C1 C=C(C)CCCC(=O)N1CC2CC1(C(=O)Nc1ccc(O)cc1)C2 C(c1ccccc1)=CC(=O)NCCN.CCC(CSC)NC(=O)CSC c1(OCC)cc(C(=O)NC2CC2NC(=O)CC2COCC(C)(C)O2)oc(=O)c1 C1(NC(C(C)(C2CC2)OC)=O)COCCN(C(=O)Cn2cccc(C)c2=O)C1 N1(CC)CCOC(C(=O)NCCC2(O)CCN(C(c3cccc(OC)c3)=O)C2)C1 C1(NC(N)=O)CCN(C(=O)CNC(N)=O)CC1.C1CCC(=O)N2CCC(C2)O1 Cc1cc(C#N)ccc1S(=O)(=O)NC1CCN(C2CCC3CC23)CC1 C1(NC(CSCC#C)=O)CN(C(=O)C(c2ccc(F)cc2F)C)CC1(C)C Cc1ccnc(CC(=O)N(C)CC2CCCN2C(=O)C(C)Cc2cnc[nH]2)c1 N1(C(C(C)SCCCC)=O)CCOC2(C1)CN(C(=O)C#CC1(CC)COC1)C2 CC1C(NC(=O)CNc2cccc(Cl)c2)CCCN1C(C1CCCCN1C)=O N1(C(C(C)CC2CCCC2)=O)CC(NC(=O)CC(C)C2CC2)CC(C)(C)C1 C12(CNC(C(C)CC3CCC3)=O)CCC(CC1)N2C(C1COC(=O)C1)=O C(N=C(NCC(C)(C)C)N1CC(O)C(C)(C)C1)C1CCCN(C(COC)=O)C1 S(=O)(=O)(c1ccc(C)c(NC(C2CCCC(N)C2)=O)c1)NC(CC)C C=C1CCC(C(=O)NC(C)(C)C(=O)NCC2=CCCOC2)CC1 CCC(CC(C)C)C(=O)NC(CNC(C1(C(C)C)CC1)=O)CC(F)(F)F C1(CN(C(=O)C(N2CCCCC2)C)CC)CCN(C(=O)COCC2CC2)CC1 C(=O)(C1CCCc2ccccc21)NCC1CC(NC(C(C(C)O)N(C)C)=O)C1 c1(C(N2CC(CCC=C)(C(=O)NCC(F)Br)C2)=O)cncc(C)n1 N1(C(C(CCCC)F)=O)CCC(C(=O)Nc2cccc(C(C)C)c2)C12CCC2 C(=O)(CCCCCF)N(C(CCCC=C)=O)C(CNC(C)=O)CCCC C1(C(=O)NCC(C)N=[N+]=[N-])CN(C(=O)CN2C(=O)CCC2=O)C2(CCC2)C1 CC(C)CC(O)C(=O)NCC1C(C)CCCN1C(=O)CN1C(=O)CN(C)C1=O c1(C(=O)NC2CCC(N(C(=O)C=CC3CCC3)C)C2)cccc2c1NCCC2 C(C)(N=c1[nH]c(N(CCCC(C)O)C)nc2cccc(F)c12)c1c(OC)nccc1 C(=O)(CC1CC(=O)c2ccccc21)NCC(C(C)C)NC(C1(C)SCCCS1)=O c1(C(=O)NC2(C)CCN(C(C3CC(CC)C3)=O)C2)cc2cc([N+](=O)[O-])ccc2o1 c1(-n2c(CSC3CCOC3=O)nc(-c3cc(OC)ncc3)n2)ccc(C)c(Cl)c1 O([Si](C)(C)C(C)(C)C)CC(C)NC1(CC2CC(OC)C2)CC1 c1(N2CC(CC(C)NC(C3(F)CC3)=O)C2)cc(=O)n(C)c(=O)n1C C1(C(=O)NCC(C)CNC(=O)C(C)OCCN(C)C)CCCCC1 C(=O)(C1=C(F)CN(C(C2CCCCC2O)=O)CC1)NC1(C#C)CCCOC1 Cc1nc(C)c(CC(=O)NCCC2CCCN(C(c3c(N)cnn3C)=O)C2)s1 N1(C(C2CC(NC(c3ccc(C#C)cn3)=O)C2)=O)CC2(CCCCC2)C1 C#CCC(C(=O)NCCC(O)C(C)C)NC(C1CCOC1(C)C)=O C1(C(=O)NC2CC(NC(C3CS(=O)(=O)CCO3)=O)C2)CC(C2CCCC2)C1 N1(C(C)=O)C2CCC1CC(CNC(=O)CCCN1CCc3ccccc31)C2 c1(NC(=O)OC)cnnc(=NC(=O)N(CCO)C(c2ccccc2)C)[nH]1 C1(OC)CCCCC1C(=O)NC(CNC(=O)CCSc1ccc(F)cc1)C(C)C N1(CCNC(C2C(C(C)(C)C)C2)=O)CC(=O)Nc2ccccc2C1.C(COCCO)O C1(CNC(C=CCCC)=O)CCCC(NC(=O)C=Cc2ccncn2)C1 C1(CCNC(C=CCN(C)CC)=O)CN(C(C2CCS(=O)CC2)=O)CC1C c1(OC)cc(C)c(C(N2CCN(C(c3ccc(CCC#N)cc3)=O)CC2)=O)cn1 c1(OC)c(C(N2CC(C(C)NC(=O)CCC3CCC3)C2)=O)cnn1C c1(C(=O)NC2CC3CC2CN3C(=O)C=Cc2ccoc2)c[nH]c2nccc-2c1 C1(CNC(=O)NC(c2onc(C(C)C)n2)C)COc2ccc(F)cc2C1 C(=O)(C1=C(F)CN(C(c2cnc(C)cc2C)=O)CC1)NC(C=C)COC C(=O)(C(CCC1CCC1)N(C)C)NCCC(CNC(=O)C=CSC)OC c1(C(=O)NCC2(C)CCC(NC(C=C(C)C(F)F)=O)CC2)cn2ccnc2cn1 C(=O)(C(C#N)CCC)NC1CC(C(N2CC(OCCCC#C)C2)=O)OCC1 C1(Sc2ncc(C)cc2O)CC1N=c1nc(C2CC2)s[nH]1 CCC(CCC(=O)NCCC(C)NC(c1cccc(F)c1OC)=O)OC(F)(F)F C(=O)(CC1OCc2ccccc21)N1CC(C)(CCC(N2CCCCCC2)=O)C1 N1(C(C2CCC(CNC(C3(C=C)CCC3)=O)O2)=O)CC=C(C)CC1 C12(CNC(=O)OC(C)(C)C)CC(CO)(CO1)C2.C1(C=O)CCN(CCF)CC1 c1(C(=O)NC2C(CCN(C)C)C2)occc1CNC(=O)COC1CCC1 c1(CCC(=O)NC2(CC)CN(C(c3cncc(N(C)C)c3)=O)C2)cncc(C)c1 c1(C(N2CC3CN(Cc4ccc(NC)cc4)C3C2)=O)ccc2cc(O)ccc2n1 N1(C(C(C(=O)NC)(C)C)=O)CC2CCN(C(C3(CC4CC4)CCCO3)=O)CC2C1 Cc1cc(C#N)sc1C(=O)NC1CC(F)CN(C(C2CC2c2ccncc2)=O)C1 C#CCCN=C(NCC(CC)(CC)CC)NC1CCCCCC(N)C1 CCCCCCCCCCC(=O)N1CC(O)(CNC(C2CCC(CC)CC2)=O)C1 c1(C(=O)NC(C(=O)N(CCCO)CC)c2cccs2)ncn(C)c1C C1(C(=O)NCC2(F)CC(NC(C(CCSC)O)=O)C2)COC2CCCCC12 S(=O)(=O)(CC(=O)NC(C)CCCCNC(=O)CC1NC(=O)NC1=O)NC N1(C(C=CC=CCC)=O)CC2(CNC(c3ccccc3OC)=O)CC(F)(C1)C2 Cc1cccc2[nH]c(=NCC3CN(C(c4ccc(C(N)=O)o4)=O)CC3(C)C)sc12 N1(C(C(CC)N(CC)CCOC)=O)CCC(O)C(C(N2CCC(C(C)C)CC2)=O)C1 C1(COCC=C)CCCN1C(=O)Cn1cc(CNC(=O)CC2CCCCO2)nn1 C#CC1CCC(C(=O)NCC2C=CCN2C(c2ccncc2)=O)CC1 N1(C(CCCOCC=C)=O)CC2COCCC2(NC(=O)CC2CCC2(C)C)C1 CCCC(C)(C)C(=O)NCC1CN(C(c2ccn(C3CC3)n2)=O)C2CC12 C(=O)(C(C)N(OC)C(=O)C1COCCC1NC(c1ncn(C)n1)=O)OC Cc1cc(CNC(c2occc2CNC(=O)Cc2coc(C)n2)=O)sn1 c1(CN(C)C)cn(CCF)nn1.C12CN(C1)C(=O)CC1(CC1)CC(=O)NCC2F c1(OC)c(C(=O)N(C(CNC(=O)C=Cc2sccc2C)C2CC2)C)csc1C C#Cc1cc(NC(=O)C(c2ccccc2)NC(c2cscc2Cl)=O)cc(F)c1 N1(C(CN(CCC)C(c2ncoc2CC)=O)=O)CCC(OCCN(C)C)C1 N1(C(CCOC)=O)CCC12CN(C(C13CCC(CF)(C1)OC3)=O)C2 Cc1ccc2ccccc2c1C(c1nnnn1C)NCCC1=CCCCC1 N1(C(C(SC)SC)=O)CCC2(CCCN2C(C2(C(=O)N(C)C)CC2)=O)CC1 c1(C(N2C(CN(C(=O)C(C3CCOCC3)O)C)CCC2)=O)ccc(O)nn1 C(=O)(CCC(C)(F)F)N(CCNC(C(C)(COCc1ccccc1)OC)=O)C1CC1 Cc1cc(C(=O)NCCCCCCNC(=O)C(O)Cc2cnc[nH]2)c(C)o1 N1(C(C(C(C)NC(=O)C2=CCCC2)(C)C)=O)CC(C2=NOCC2)C1 CC(C)CCCCCC(=O)NC1(C2CCN(C(c3cncc(C#N)c3)=O)C2)CC1 N1(C(C2CCC(CC)CC2)=O)CCC(CO)(NC(=O)CCc2ccnn2C)CC1 c1(C(=O)NCCC(C)N2CCC2)n[nH]c2c1CN(C(=O)CCc1cn(C)nn1)C2 c1(C(=O)NC2CCC(C)N(C(c3cc(F)ccc3F)=O)C2)ccc2c[nH]nc2c1 c1(N2C(CNC(=O)CCC[N+](=O)[O-])CCC(C)(C)C2)nc2c(F)cccc2o1 c1(C(N2C(CNC(C(C)C#N)=O)CCCC2)=O)cc(N)c(F)cn1 C(CCCC(C)(F)F)NC(C1(CC=C)CCCN1C(c1occc1COC)=O)=O C1(C(N(CC(=O)Nc2ccccc2Cl)C)=O)CCCN(C(c2ccc(O)cc2)=O)C1 C1(C(=O)NCC2(C)CCCC2NC(C2CCCCNC2=O)=O)CCOC2(CCC2)C1 c1(C(=O)NC(C)CN(C)C(c2cc(Br)n(C)c2)=O)cnn2c1CN(C)CC2 C1(C(C(CC)C(=O)NCCOCCOC)=O)(COCCNC)CC12CCC2 Cc1cc(C(N2CC(NC(=O)COC3CCCC3)C(F)C2)=O)c(Br)cc1F O=C1C2CC(C(N3CCC(Cn4cc(-c5nccs5)nn4)C3)=O)CN2C(=O)N1 Cc1ccc(NC(C23CC(C(=O)Nc4ccccc4)(C2)C3)=O)nc1C N1(C(CNC(C)=O)=O)CCC(C2CC2)C1CNC(c1cn(C)nc1-c1cccs1)=O c1(-c2ccc(C(N(CC)CC)=O)cn2)ccc(C)nc1F c1(N(CC(C)NC(C2(C=C)CCOCC2)=O)C)nc(Cl)nc2[nH]cnc12 c1(C(=O)NC2CC(C)N(C(=O)CC3(C)CC3(Cl)Cl)CC2)cnc2c(c1)nnn2C CCC(CC)C(C(=O)N1CC(NC(c2cc(Cl)ns2)=O)C(C(F)F)C1)OC N1(C(c2c[nH]c(=S)cn2)=O)CCN(C(=O)CNC(N)=O)CC1.C(C(=O)OC)NCC#C Cc1ccc([N+](=O)[O-])c(C(=O)NCC2CCN(c3nccc(C4CC4)n3)CC2)c1 C1(CC=C)(NC(=O)COCP(C)(C)=O)CCN(C(c2cnoc2C2CCC2)=O)C1 C1(NC(CCCOCCOC)=O)CCCC(C(=O)NC2CC(CSC)C2)CC1 N(C)(C1CCOc2ccc(F)cc21)C(CC(C)CCC1=CN=CN(C)N1C)=O Cc1cc(O)cc(O)c1C(N1CCNC(C(=O)NCC23CCN(CC2)C3)C1)=O Cc1cc(C#N)nc(N2CC(NC(=O)C(C(C)C)c3ccc(F)cc3)C(C)C2)n1 Cc1cc(CNC(=O)C(C)C(C)NC(=O)C(C)(C)F)cc(C)c1 c1(C(=O)NC2CN(C(C(C)CC#N)=O)C2)c[nH]c2ccc([N+](=O)[O-])cc12 N1(C(=O)CCCC2CCCC2)CCCN(C(c2ccc(C(F)F)o2)=O)CC1 C(=O)(C1=CCCC1)NCC(C)(C1CCC1)NC(c1conc1C(F)F)=O Cc1cn2cc(C(=O)NC(C)(C)CNC(C3(CCF)CCOCC3)=O)nc2s1 N1(C(CCCCCC)=O)CC2(C1)CN(C(c1nc3c(s1)COCC3)=O)CC2CO N1(C(C(c2ccc(C)cc2)C)=O)CCCCC(NC(=O)Cn2ncc(Cl)c2C)C1 O=S1(=O)CC=CC1CN1CCCCC1C1CCOCC1 c1(C2C(C(N(CC(O)CNC(=O)Cc3cccc(Cl)c3)C)=O)C2)ccc(F)cc1F C1(C(=O)NCC2CCN(C(=O)CSCc3ccccn3)C2)CCCS1(=O)=O C1(OCC#C)CCCN(C(C2(n3cc(-c4cncnc4)nn3)CCOCC2)=O)C1 N1(C(C=C(C)C(C)C)=O)CC(CC(N2CC(C(C)(C)C)C2)=O)CC1(C)C C(=O)(C(C(C)(C)C)SC)NC(CC)(CNC(=O)C(N1CCOC1=O)C)CC c1(C(C(=O)N2CC(CCCCN(C(C(F)=CCC)=O)CC)C2)(F)F)ccc(F)cc1 CN1CCCC(CC(=O)NCC2CC2NC(c2cccnc2OC(F)F)=O)C1 Cc1ccc2scc(CC(N3CCN(C(=O)CC4=CCCC4)CCC3C)=O)c2c1 N#CC1CCC(C(N2CCN(C(=O)C3=CCC3)CC2C(F)F)=O)CC1 C1(NC(CCCOC)=O)CC(C)CN(C(=O)C(=O)NCC2CC2)C1 C(=O)(C(C)(O)C(F)(F)F)N(C)CCC1CCN(C(c2scnc2Cl)=O)CC1 c1(OCC)cncc(C(=O)N(C)CC2CC(O)CN2C(=O)C(C)COCC)c1 C1(C(=O)NC2CCCN(C(C(N3CCNC3=O)C)=O)C2)Cc2cc(Cl)ccc2O1 n1(CC(N2C(C(=O)N(C3CCCC3CCO)C3CC3)CC2)=O)cnnc1O C1(c2nnnn2C2CCCC2)(Nc2c(OC)nn(C)c2)CCCN(C)CC1 N1(C(CN(C2CCC2)C)=O)CC(F)CC1CNC(=O)COCC1CCCCO1 CC(C)CC(C(=O)NC(CNC(c1cc(N)c(O)c(F)c1)=O)C1CC1)C(N)=O c1(C(N(C(C)CNC(C2CCOC2)=O)C)=O)cnc(C(F)(F)F)c(Cl)c1 c1(C(=O)NCC2N(C(C3C(C)C3)=O)CC2)ccnc(OCCO)c1 C(CCCCC(=O)NC(CNC(=O)C(O)Cc1ccccn1)CC(C)C)SC C(=O)(C=C1SCC(=O)N1C)NCc1c(NC(C2(OC)CC2)=O)cccc1.N1(C)CC1 N1(C(c2c(SCC)cc(Cl)cc2)=O)CC2CCC(C1)N2C(=O)C(C)CC(C)C CC(C)(C)C(C(=O)NCCn1cc(CO)nn1)NC(=O)C(O)c1cnc[nH]1 C(=O)(CCCN(C)N=O)N1CC(NC(C2(CC#C)CCCCO2)=O)C(OC)C1 C1(C(=O)NCCc2c(C)ccs2)CCCN(C(c2cnsc2C)=O)C1 C12(NC(Cc3c(C)cc(F)cc3)=O)CCC(CN(c3ncnc(C)c3Br)C1)C2 c1(C(C(=O)N(CCN(C(C2CCC(=O)O2)=O)CC)CC)O)cc(F)ccc1C C(C1=CCN(C(=O)Cc2cn[nH]c2)CC1)NC(C1CCN(C2CC2)S1(=O)=O)=O c1(NC(C2CCN(c3ncccn3)C2)=O)cccc(C(F)(F)C(F)(F)Cl)c1 CC1COc2ccc(C(N3CCC(C)N(C(=O)CCc4cscn4)CC3)=O)cc21 c1(NCC(COC)O)ccc(S(=O)(=O)NC2CC3(CCC(CO)OC3)C2)c(Br)c1 N1(C(C(CCNC(C2CC(C)(F)C2)=O)O)=O)CCC2(CC1)N=N2 N1(C(C2C(CC)CN(C(=O)CC(C)N(C)C)C2)=O)CCCC(C)C1C N1(C(C2(Br)CC3(CCCC3)C2)=O)CCC2CCCC12CNC(=O)C1CC1 C1(N(C(=O)Cc2cncnc2O)C)CC2CC1N(C(=O)CNS(=O)(=O)N(C)C)C2 C1(C(N2CCC(F)(C(=O)NC3CCCSC3)C2)=O)=CC(NC(=O)N(C)C)=CCC1 CCC(F)C(=O)NCC1(NC(C2CC(O)(C(F)(F)F)C2)=O)CC1 c1(C(N2CCC(CC(=O)NC3CC(C)OCC3)C2(C)C)=O)cnn2ccccc12 c1(C(=O)NC2CCCCN(C(c3n(C)nc(O)c3)=O)C2)cccc2nc(S)oc12 C1(CCCC)CCC(N=c2[nH]c(=NCc3cc(Br)ccc3F)[nH]c3ncn(C)c23)C1 c1(CC(Cn2cc(CCSCC)nn2)CO)ccc(F)cc1 C1(NC(C(CC)N(C)C)=O)CN(C(c2ccc[nH]2)=O)C(C)(C)C1 Cc1cccn2nc(C(N3CC(NC(=O)CC4CCOC4)C(C)(C)C3)=O)cc12 c1(C(N(CCN(C(=O)C(O)c2ccsc2)CC)CC)=O)ncn(C)n1 C1(CNC(CCC=C)=O)CCC2(CO1)CN(C(=O)C(O)Cc1ccc(F)cc1)C2 C1(CNC(CC2N(C(C)=O)CCC2)=O)C2CCCC2N1C(=O)C(C)CC(F)F N1(C(CCNC(C)=O)=O)CC(NC(c2cnc3n2CCS3)=O)CC12CCCOC2 c1(OCC)ncc(C(=O)N(C)CC2(CNC(=O)CN3CCOCC3)CC2)cn1 c1(CNC(C2CC(NC(c3c(C)cno3)=O)C2)=O)ccnc(C)n1 C(=O)(C1=CCOCC1)NCCCN(C(=O)CN1CCCNC1=O)C(C)C C12(NC(C3CCCCC3O)=O)CCCN(C(=O)CO)CC1C2 C1(NC(c2cc3ccsc3s2)=O)CCN(c2nnc(CO)s2)CCC1CO N1(C(c2cc(C)no2)=O)CC2C(C1)N2C(c1cccnc1C(F)F)=O C1(CC)(NC(c2c(C)nn(C)c2-n2cc(C)cn2)=O)CCCN(C(=O)C2CC2)C1 O=C(CCC1CC(NC(=O)CC2CCOC2=O)C1)NOCC1CCCO1 C1(OCCCN(C)CCNC(C2CCCO2)=O)CCNCC1CC(F)(F)F c1(N2CC(=O)N(CC(C)C)C2=O)nc(N(C)C(=O)OC(C)(C)C)c2c(n1)CCC2 C1(C(=O)NN2CCC(N(C)C(c3ncc(C(F)F)s3)=O)C2)CC2CCC1CC2 c1(CNC(CNC(=O)OC)=O)cc(C(=O)Nc2ccncc2Cl)n(C)n1 c1(CC(=O)NC2C(NC(C(CCC(C)C)O)=O)CCC2)ccc2ccccc2c1 C(=O)(C1SCCc2sccc21)N(CCC(C(C)C)NC(c1cccc[n+]1[O-])=O)C C1(C(=O)NC(COCCNC(=O)COCCOCCO)(C)C)CCC(=O)NC1 C1(C(N(C2CC(NC(c3c(C(=O)OC)coc3)=O)C2)C)=O)CCC2CC2CC1 CC1CCc2[nH]c(=NCc3ccc(C#N)cc3)nc(N3CCC(C)(C)CC3)c2C1 C(=O)(C(O)CCCC)N1CC2C(C(N3CC(CCC)C(CC)C3)=O)(C2)C1 CC(C)(C)CC(O)CC(=O)NCC1C(C(N2CC3(CC=CC3)C2)=O)C1(C)C c1(C(N(C)CC2=CC(Cl)=CC=NC=C2)=O)cccc2ccc3ccccc3c12 C=CC1(CC(N2CC(NC(C3CCC3CN(C)C)=O)CC2CO)=O)CCCCC1 N1(C(=O)CCC2CCC2)CC2CN(C(=O)CC3CCCC3)CCC2(CO)C1 c1(N2CC(CN(C(C(C)CN(C)C)=O)C)OCC2)[nH]cnc2nc(Cl)cc1-2 CN1CCN(C(=O)Cc2ccon2)CC1CNC(c1cccc(C2CCC2)c1)=O CC1CC=C(C(=O)N(CCNC(c2noc3c2COCC3)=O)CC2CC2)CC1 Cc1ccc(C=CC(N2CCCC2C(C)NC(=O)C(C)C)=O)nc1 N1(C(c2nc(OC)oc2)=O)CCC2(CC1)CN(C(c1ncc(C)nc1OC)=O)C2 c1(CC)nc(C)c(C(N2CCC(OCCNC(c3nc(Cl)oc3C)=O)CC2)=O)s1 C1(CC(N2C(C(C)O)COCC2)=O)CCCN(C(=O)CC2=CCCC2)CC1 C12(C)CCN(CC1)C(=O)N2.c1(CCNC(=O)OC(C)(C)C)nc(I)cnc1N C(=O)(C(CNC(=O)CC1CCC(F)(F)C1)CF)N1C(CSC)CCC1 C1(CC(=O)NCCOCC(=O)NCC(CCC)C)CCC(=O)N1C C1(C)(C(=O)NCCOC(C)=O)CCN(C(C2CCC(C)(C)O2)=O)C1 Cc1c(CN(C)CCN(C(=O)C2=NOC3(CCC3)C2)CCO)[nH]c2ccc(F)cc12 CC1(C)CN(C(=O)CCC2CCOCC2)CCC1NC(c1cccnc1Cl)=O c1(C(=O)OCCCC2C(C(=O)OCC)C2)nc(=O)n(C)[nH]1 C1(NC(c2c(C)nn(C(C)(C)C)c2)=O)CCN(C(C2CC(F)(CO)C2)=O)C1(C)C C1(C(=O)NCCCCNC(C(CC)OC)=O)CC(=O)NC(=O)N1 C1(C(=O)NCC(CCC)OC)CC2CCC(C1)N2C(=O)CCc1cccn1C CC(c1ccco1)=CC(=O)NC1CCCCC1NC(C1CC1C(C)(C)C)=O CC1CN(C(c2ccn(C)n2)=O)CC(C)N(C(c2cc(Br)no2)=O)C1 C(=O)(C(=O)C(C)(C)C)NC(CNC(C(c1cn(C(C)(C)C)nc1)=O)=O)C1CC1 N1(C(C(C)OC)=O)CCN(C(c2csc([N+](=O)[O-])c2)=O)CC1CC(F)(F)F c1(SC)ccc(OC(C)(C)C(=O)N(C)CCNC(=O)CC2CCCCCO2)cc1 N1(C(COC(CC)CC)=O)CCC(CC(=O)NCC2(O)CCCC2(C)C)C1(C)C c1(CCC(=O)NC2CCC2NC(c2ncccc2O)=O)ccc(Cl)cc1Cl Nc1c(Cl)cnc(C(=O)NC2(CCNC(C3CC=CCC3)=O)CC2)c1Cl c1(CNN2C3C(C(N4C(C#N)C5CC5C4)=O)C(C3)C2)ccc2nc(Cl)ccc2c1 C1(CNC(c2ccc(F)c(F)c2F)=O)CC2COCC2N1C(C1(F)CCCC1)=O C(=O)(C1=CCCC1)N(C)CC1CCCN1C(c1cnn(C(F)(F)F)c1)=O c1(C(=O)NC23CC(C(=O)Nc4cc(C)no4)(C2)C3)cc2cccc(F)c2s1 c1(CC)c(N2CCOC(CNC(C3CC4CCCC(C3)C4)=O)C2)nc(C)nc1Cl Cc1cccc(COC(C)C(=O)NCC(O)CN(C)C(c2[nH]c(O)nc2C)=O)c1 C1(C(=O)NC2(CNC(C(C)NC(C)=O)=O)CCC2)CC(c2cccc(F)c2)=NO1 C#Cc1ccc(Cl)c(C(=O)NCC2(C)CCCN(C(C3(CO)CCCC3)=O)C2)c1 C1(CNC(c2cccc(COC)n2)=O)CCC12CN(C(=O)Cc1cnccn1)C2 Nc1nc(Cl)ccc1C(=O)NCC1CCCCN1C(C1CC2(CCC2)CO1)=O C(=O)(CC(CN(C)C)C(F)F)NC(CC)(CNC(=O)CNC(=O)C1CC1)CC c1(C(N(CC(CC)NC(C2CCCC23CCC3)=O)C)=O)ccc(P(C)(C)=O)nc1 C1(NC(CC2CCC(NC(CCSCCC)=O)CC2)=O)CCCC12CCC2 N1(C(=O)CCNc2ncccn2)CCC2CN(C(c3csc(C(F)(F)F)n3)=O)C2C1 c1(C(=O)NC2CCCC(N(C(=O)CC3CCOCC3)C)C2)cc2cccnc2s1 c1(CC(=O)NCC2(O)CN(C(C3CC4CC3C4)=O)C2)cc(F)cc([N+](=O)[O-])c1 N1(C(COc2cc(C)on2)=O)CC2(COC(CNC(C34CCC(C3)OC4C)=O)C2)C1 CC#CCCCC(=O)N1CCN(C(=O)CSc2ccccc2C)C(CO)C1 c1(CNC(N(CC(C)CN)C)=O)csc(-c2ccccc2)n1 C#Cc1cnn(CC(N2C(C(=O)NC(C)COCC3CC3)CC2C)=O)c1 C1(NC(CNC(C)=O)=O)CC2CC1N(C(C1(Sc3cccc(C)c3)CCC1)=O)C2 c1(C(N(Cc2c(CC)cccc2)Cc2ccccc2)=O)ccc(I)c(Cl)c1 CC(C)C(N=[N+]=[N-])C(=O)NCC1CCN(C(C2(CO)CCCO2)=O)C1 N1(C(c2cn(CCNC(c3c(CC)nco3)=O)nn2)=O)CCOC(C)(CC)C1 C1(CC(=O)NC(CCNC(c2c(COC)ncs2)=O)C)CCC(C)CC1 C1(O)(C(C)NC(=O)Cn2ncccc2=O)CCN(C(c2cccnc2)=O)CC1 N1(C(c2cc(C)ncc2C)=O)CCOC2(CCN(C(c3cc(C)ns3)=O)C2)C1 N1(C(C2NC(=O)SCC2)=O)Cc2nccn2CC(NC(C2CC2(Cl)Cl)=O)C1 CC(C)(C)CCC(=O)NCC1(C(C)(C)O)CN(C(=O)CSCC2CCCO2)C1 c1(C(N(C)CC2CCN(C(c3c(CCC)occ3)=O)C2)=O)cc(OC)nc(Cl)c1 C1(N2CCC2)(C(N2CC(F)(CNC(=O)CSC(F)(F)F)C2)=O)CCCO1.C(=O)OC C1(C(N(C2CCCN(C(C3(C(=O)C4CC4)CCC3)=O)C2)C)=O)CC2CCCC2C1 c1(C(=O)NC(CSCC)C(=O)NCCC2CCCC2OC)ccc(O)nc1 c1(C(=O)NC2C(CNC(c3c(SC)cc(F)cc3)=O)C2)c(C)c(C)cc(C)c1C c1(OC)cc(CNC(=O)CC(O)CNC(=O)Cc2cn(C)nc2C)n(C)n1 C1(NC(C2(CC)CCC2)=O)CC2(CCCN(C(c3cc(C)c(F)cc3F)=O)C2)C1 C(=O)(CCC(C)SC)N(CCN(C(=O)C(C1(O)CCCC1)F)CC)CC C1(CNC(c2cn(C3CC3)nn2)=O)CCCN(c2ncccn2)C1 c1(C(=O)NCCN(C(c2cnc[nH]2)=O)C2CC2)cc2nccc(Cl)c2s1 c1(C(CC)(C)C)ccc(C(=O)NCC2CN(C(c3c(SC)noc3C)=O)C2)cc1 C1(C(N(C2CCN(C(c3cc(F)ccc3F)=O)C2)CCC)=O)CCCCNC1=O C(=O)(NNS(=O)(=O)c1ccc(Br)c([N+](=O)[O-])c1)c1c(OC)cc(Br)cc1 O=C(C1=CCCCO1)NCC1CN(C(=O)CC2COC(=O)N2)CC1C(F)(F)F CC1(C)C(NC(=O)Cc2ccns2)CCN1C(c1cc(N)c(F)cn1)=O CC1CCN(C(c2ccc(C3CC3)o2)C(=O)NCCOCC2CC2)CC1C c1(CN(CCNC(C2C(C(C)C)C2)=O)C(C2CC2C(F)F)=O)cccc(Br)c1 C(CCCC(=O)N(C)CC1CCN(C(C2(CO)CCCC2)=O)C1)OC C12(NC(C(C(C)C)SCC)=O)CCN(C(=O)CC3CN4CCC3CC4)CC1C2 C(CCC(O)C(=O)NCC1CCCN1CC)NC(C(CC=C)OC)=O N1(C(c2c(CCC)n[nH]c2)=O)CCC(C(=O)N(C(CO)C2CC2)C)C(C)(C)C1 C1(NC(CSCC=C)=O)CC(C(=O)NN2CC=C(C=C)C2)C12CCC2 c1(CN2CC(CC#N)CC(C(=O)OC)C2)scc2c1OCCO2 c1(C(=O)NC(CC2CN(C(C(C)CC3CCC3)=O)C2)C)cc(N)cnc1Cl N1(C(=O)NC2CCC(C(C)(C)C)CC2)CCOc2cc(Cl)c(Cl)cc21 C(C)(CCCC(=O)N(C1C=CCC1)C)NC(CNC(=O)OCC)=O CCC(F)(F)CC(=O)NCCOCCCNC(C1(C)CC(C)=NO1)=O C(CC(=O)N1CCCc2ccnn21)N(C(c1ccc2cncn2c1)=O)CC1CC1 C1(C(N(CCC(=O)OCC)C)=O)CN(C(=O)Cc2cccc(O)c2)CCC1O C#CC1(C(=O)Nc2ccc(F)cc2)CN(C(c2cc(CO)oc2C)=O)C1 C#Cc1cncc(C(N2CCCCC2C(C)NC(c2ccc(Br)o2)=O)=O)c1 C1(CNC(C(CCC)CC)=O)CN(C(=O)Cc2c(Cl)cnn2C)CCC1(F)F C(=O)(C(C)(C)Oc1ccccc1)N(CC(CNC(CSCC#C)=O)O)C c1(SC)cc(C(N2CC(CNC(c3c(C)ccn3C)=O)CC2C)=O)nn1C C1(NC(C2C(COC)C2)=O)CCCC1NC(c1cn(CCC(C)(C)C)nn1)=O c1(C(N(C)CCNC(C2CN(C3CCOC3)C2)=O)=O)ccc2c(c1)CCCS2(=O)=O C#CCC(C(=O)NC1CC(=O)C1)N(C(=O)CNC=O)C(C)CC C(=O)(C(C)CCCC(C)C)N1C(CC=C)(C(=O)NC2CC3CCCC3C2)CCC1 c1(OC)cnc(Br)cc1C(=O)N(CC(=O)NC(c1ccc(Cl)cc1)C)C c1(C(N2CC3OC(C)C3C2)C(=O)NCc2ccco2)cncc(S(C)(=O)=O)c1 CC1(NC(=O)C(O)C(F)(F)F)CCN(C(=O)C(C2CCCCCC2)F)CC1 c1(C(=O)NCC(C)NC(=O)C(O)C(F)(F)c2ccccc2)nn(C)c(Cl)c1Cl c1(OC)cccnc1C(=O)NCC#CCNC(=O)CN1CCCNC1=O N1(C(C(CC)(CNC(=O)CCC2CCCO2)CC)=O)CCC2(CNC(=O)O2)C1 CC1(C)NC(=O)CC1C(N1CCCC(NC(c2cccc(C3CC3)n2)=O)C1)=O C=CC1CN(C(=O)CC2CC(=O)NC2=O)CC1NC(=O)C(CC)(CC)OC N1(C(C(CC=C)C)=O)CCC(N=[N+]=[N-])(C(=O)NCCC(C)(C)N(C)C)C1 CS(=O)(=O)c1ccccc1CCNC(=O)NC1(CC2(C#N)CCCC2)CC1 c1(C(=O)NC2(CNC(C(CC)(C)O)=O)CCC2)cc2c(Cl)c(OC)ccc2[nH]1 N1(CC)CCCCC1CNC(=O)C(CCC1CC1)NC(c1cc(Cl)ns1)=O C1(C(=O)NCC(CC(=O)NC(CCCC)CC)O)CN2CCN1CC2 Cc1cccc(C(C)C(=O)NCCC2CSCCN2C(=O)Cn2cncn2)c1 CCCCCCCCC(C)C(=O)NC1CCCCN(C(c2c[nH]c(C#N)c2)=O)C1 Cc1cc(C(=O)NC2CC3CC2N(C(c2cn(C)ccc2=O)=O)C3)c(C)nc1C C1(F)(C(N(CCCSC)C)=O)CCN(C(=O)CN(C2CCC2)C)C1 Cc1ncc2n1CCN(C(C1COC3(C1)CN(C(c1cnccn1)=O)C3)=O)C2 C1(CNC(CC(C)NC(N)=O)=O)CN(C(=O)C(C)(F)F)C2(CCOCC2)C1 c1(C(=O)NCC2C(NC(c3ccc(OC)nc3)=O)COC2)ccc(N)cc1Cl C(=O)(C1CCc2nccn21)NC1CCCC(NC(CN(C(=O)OC)C)=O)C1 C1(C2N(C(C)(C)C)CCCC2)CCN(C(C(C)(C)C)=O)CC1C(=O)NOC(C)(C)C CCC(CC)C(C(=O)N1CCOCC1C(N1CCOC(C2CC2)CC1)=O)OC c1(N(C)CC2CC3CC3C2)nc2c(c(=NCC3CCC(C(F)(F)F)O3)[nH]1)SCC2 c1(C(N2CCC(N(C(=O)COC3CCCCC3)C)C2)=O)cc2c([nH]1)CCCC2=O C1(OC)CCC2CN(C(=O)CN(C3CCCC3)C(=O)Cc3cn(C)cn3)CC12 C1(C(=O)NCCC2CC(NC(c3n(C(CC)CC)ncc3)=O)C2)CCC(C)CC1 c1(CC)ncoc1CNC(=O)CC1CCN(C(=O)CCc2cnoc2)C1 CCC(C)(C(=O)OC)NC(c1cc(N2CCCC2)ncn1)=O.C12CC1CNC2=O c1(OC)ccc(F)c(CN2CCC(=O)N(CC(=O)OC(C)C)C2=O)c1Br C1(CC)CCN(C(=O)CC2(OC)CCC2)C1C(N1CC(CO)C(O)C1)=O C(=O)(C1=CCN(C(c2cccc(C3CC3)c2)=O)C1)C(COCCOCC)=O C1(CC(=O)NCC2(C(N)=O)CN(C(=O)CSCC3CCCO3)C2)NC(=O)NC1=O Cc1nc(C(=O)NCC2CC3CC3N2C(=O)C(C2CCOCC2)F)ccc1C#N N1(C(C(CC)(F)F)=O)CCOCC(F)(CNC(c2ccc(Cl)nc2NC)=O)C1 c1(CC(=O)NC2CCC(NC(Cc3[nH]c(=N)sc3)=O)C2)ccc(F)cn1 C1(CN(C)CCn2cnccc2=O)CCN(C(=O)CSC(F)(F)F)CC1 C1(CNC(C2C(NC(COCCC)=O)CCC2)=O)COCC(=O)N1C N1(C(CC=CC=C)=O)CCC2(CC1)CN(C(c1ccc(F)c(N)c1F)C1CC1)C2 N1(C(C(=O)NC2CCC2)=O)CC2(CCCN(C(c3cn(C4CC4)nn3)=O)C2)C1 C12(NC(c3scc(C)c3)=O)CCCC(CN(C(C3CCC=CCC3)=O)C1)C2 C1(CN2CCC(O)(c3ccc(Cl)cc3)C2)CC[Si]2(CCCC2)CC1 N1(C(C2(C)CCCN(C(=O)CC3CCCNC3=O)C2)=O)CC(O)C2(CCCC2)C1 c1(C(=O)OCC)cccnc1NCC#CCNC(=O)CC1(NC2CC2)CCCC1 N1(C(C)=O)CC2CN(C(=O)CC(C)(F)F)CC2(C(F)(F)F)C1 N1(C(CCOC)=O)CCC(C2(NC(c3cccc(C)c3Cl)=O)CC2)CC1 N1(C(c2cccc(C)c2)=O)CC(C)N(C(=O)CC2CCCC(C)(C)O2)CC1C C1(Cc2[nH]c(=N)sc2)CC2(CCOC2)C1.C1C(=O)NCCCN1CCO C1(C(=O)NCC(C)N(C)C(c2cccc(C3CCOC3)c2)=O)CCCC2(CC2)C1 C1(N(C(=O)CCOC2CCCOC2)CCC)CCN(C(=O)C(C)(C)CF)CC1 c1(OC)ccccc1C(=O)NCC1CCC(N(C(=O)C=CC2CC2)C)CC1 Cc1cc(O)cc(=O)n1CCC(N1CC(NC(=O)C(F)CC2CCC2)C(F)C1)=O N1(C(C2CC(C)(C)C2)=O)CC(CNC(=O)CC2SC(=N)NC2=O)OC(C)(C)C1 c1(C(N2CCC(O)(CNC(c3ncc(OC)cn3)=O)C2)=O)c([N+](=O)[O-])cnn1C c1(OC(C(N2CC(N(C(c3cnc(CC(C)C)[nH]3)=O)C)C2)=O)C)cccc(F)c1 CC(C)CCCC(=O)NC(CC(=O)NCC1(O)CCC1)C1CC1 C1(NC(CC2CC(C)(C)OC2)=O)CC2CN(C(c3ncccn3)=O)CC12 CC1=C(C)CN(C(=O)C(O)C2CN(C(C3CNC(=O)C3)=O)C2)C1 CN1CCc2cc(CN(c3cccc(F)c3F)C(=O)NCC(O)C3CNC3)ccc21 CCC(C(F)(F)F)NC(=O)CNC(=O)CCN1CCCC1=O c1(OC)cccc(CO)c1.C1(CC(N2CC(C(=O)O)C2)=O)CCS(=O)(=O)C1 CCCCC1C(=O)NC(C)(CC)C(=O)N1.C(CCN=[N+]=[N-])NC(=O)COC(=O)CO Cc1c(CCNC(C2CCCCN2C(c2coc(C(C)C)n2)=O)=O)cnn1C C1(NC(Cc2c(OC)cccc2)=O)CN(C(c2cc(C3CC3)no2)=O)CC12CC2 C1(C(N2CC(Nc3ncc(OC(C)C)cn3)C2)=O)CC2CCCN(C1)C2 C1(CCNC(c2c(CC)cno2)=O)CCN(C(=O)C(C)(C)NC(=O)OC)CC1 C1(O)(CNC(c2ccccc2OC2CCC2)=O)CCN(C(c2ccnnc2)=O)C1 c1(C(N2CCCC(NC(c3cccc(F)c3O)=O)CC2)=O)cnc2ccnn2c1 c1(CN2CC3(N(C(c4n(C)ccc(=O)c4)=O)CC3)C2)ccc(N)c([N+](=O)[O-])c1 CCCC(C(=O)N1CCC(O)(CN(C(=O)C(C)SCc2ccccc2)C)C1)OC O=c1[nH]c(CCC(N2CCC3CN(C(C45CC4C5)=O)CC23)=O)nc2ccccc12 N1(C(CS(CC)=O)=O)CCCC2(CCN(C(=O)C(CCSC)NC(C)=O)C2)C1 C(c1cccc(F)c1)=CC(N1CC(C(C)NC(c2cnco2)=O)OCC1)=O N1(C(CC=C(C)C)=O)CCC(C2CCN(C(c3nccc4occc34)=O)C2)C1 C1(CC)CN(c2ccnc(N3CC(C(N4CCCC4)=O)C(O)C3)n2)CCS1 N1(C(C)C)CCC(CNC(=O)CNC(c2n[nH]c(=N)[nH]2)=O)C1 c1(C(=O)NCC2N(C(C=C(CC)C)=O)CC2)ccc(-c2sccc2C)s1 C(CCC(C)NC(=O)C(CC)N1CCCC1=O)NC(C=C(C)CNC(=O)N(C)C)=O N1(C(c2c(CC)con2)=O)Cc2ccccc2C(CNC(=O)C(O)CC(N)=O)C1 CCC(C)C(CC(=O)N1CCC(SC)C1)NC(c1ccco1)=O N1(C(CC=C)=O)CCCCC(NC(c2[nH]c(C)c(C(N)=O)c2CC)=O)C1 c1(CC)c(C(=O)NCc2ccoc2C(=O)N(C(C)C(F)(F)F)C)ccn1C Cn1c(CC(=O)NCCC2(NC(=O)CC3CCNC(=O)C3)CC2)nnc1S N1(C(c2cc(CC)oc2C)=O)CCC(C2CCCN(C(C3(C)CC(F)C3)=O)C2)C1 c1(CC)nc(C)ncc1C(=O)N(C(CNC(c1nccnc1N)=O)CC)C CCCC(CCCNC(=O)Cn1cncn1)NC(=O)C(C)NC(C1CCC1)=O CC(CC(F)(F)F)N(C(=O)C(c1ccco1)NC(C1CCCC1)=O)C C1(CC(=O)NC(C)CNC(=O)CC2(C)CCC2)CCN(C)C1 C1(CCC(=O)NCC(C)C2CC2)CCN(C(=O)Cn2ccnn2)CC1 c1(C(N2CC3C(CC(=O)NC(CCCC)COC)C3C2)=O)cc(O)cc(F)c1 C1(C(=O)NCC2(F)CC(NC(C(CC)F)=O)C2)CN2CCN1C(C)C2 C1(NC(CSC(C)C)=O)CCCCC1CNC(C1CCCC1)=O n1(CCOCC)nnnc1C(c1ccoc1)NCc1nocc1C(C)(C)C C1(C(N2CCC(NC(C3(C=C)CCCC3)=O)C2)=O)CC(=O)CC(=O)N1 C1(C(=O)NC2CC(NC(C(c3nccc(C)c3)(F)F)=O)C2)CCN(C)S1(=O)=O N1(C(c2onc(COC)n2)=O)CCN(C)CC1CNC(c1ccc(Cl)nc1O)=O C1(CON(C)CCc2cn(CCO)nn2)CCN(C(C2(C(F)(F)F)CC2)=O)C1 C1(C(=O)OC)Cc2ccc(O)cc2CN1C(c1ccc(CC(C)C)cc1)=O C=CC(C)(O)CC(=O)N(C1CCN(C(c2ncccc2OC)=O)C1)CCC C1(CC)(NC(C2CCC3(CCC3)O2)=O)CCCN(C(c2c[nH]cc(C)c2=O)=O)C1 Cc1c(C(=O)NCCC(O)CNC(=O)C=CCF)cnn1C(C)C(C)(C)O CC(CO)C(=O)NCC(C)(C1CCC1)NC(c1ccoc1C1CC1)=O C(=O)(CCC(=O)NN(C)C)N1CC(C(=O)NC(C)C(=O)NO)CC(C)C1 c1(NC(COC(C)(C)CNC(c2cccc(=S)n2O)=O)=O)cccc2cc[nH]c12 C1(C(=O)NC(C(C)NC(=O)Cn2cc(CN(C)C)nn2)(C)C)CC(F)C(=O)N1 N1(Cc2cccc(NC(c3cc(OC)c(C)[nH]3)=O)c2)CC(C(=O)O)C2(CCC2)C1 c1(C(N2CCC(C)(CNC(C(CC=C)C)=O)C2)=O)c(C)ccc2ccccc12 C1(C(=O)NCCOCCCNC(COCC(=C)C)=O)CC(F)(F)C1 c1(CC(=O)NC(CC=C)CNC(=O)CCS(C)=O)ccc2c(c1)CC(C)O2 c1(Oc2c3c(ccc2)C(OC(C)C)CC3)cc([N+](=O)[O-])ccc1N c1(NC(C2CCN(C(Cn3c(C)ccn3)=O)C2)=O)ccc(N2CCCC2)nc1 c1(SCC(=O)NCC2N(C(CC(=O)OC)=O)CC2)ccc(Br)cc1C Cn1c(C(=O)NC2CCC2CNC(c2cnc3n2CCCC3)=O)cnc1[N+](=O)[O-] CC1CN2CCN1C(C(=O)NCC1CCCN(C(c3ccc(F)c(Cl)c3N)=O)C1)C2 c1(C(N(C2CCN(C(=O)CC=C)C2)CC#C)=O)c(F)cccc1Cl C1(NC(c2cc(SCC)ncc2)=O)CC(O)CN(C(c2sccc2C(C)=O)=O)C1 Cc1nn(CC(=O)NC2CC(C(C)NC(=O)CO)C2)c(C)c1C=NO C(c1cccc(F)c1)=CC(N1CC(CNC(=O)C(O)CC2CCCC2)C(O)C1)=O C1(CNC(CCCN(C(C)C)C)=O)CCC(NC(C2CCC23CCC3)=O)CC1 C1(C(=O)NC(C2CN(C(C3(C4CCCO4)CC3)=O)C2)C)CC2C(C1)C2(C)C c1(C(C)=O)ccncc1-c1cn(CCCN(C(C)C)C2CC2)nn1 Cc1ccccc1-c1cc(C(=O)NC(C2(CNC(C3C(C)C3C)=O)CC2)C)no1 C1(C)(C(=O)NC(CC)CNC(=O)C(C)OC2CCOC2)CCC(=O)N(C)C1 C1(NC(COCCC)=O)CCCC(NC(=O)CC2CCOCC2OCC)C1 S(=O)(=O)(c1ccc2cccnc2c1Br)Nc1ccc2[nH]c(=N)sc2c1 N1(C(CCCOC)c2nnnn2C2COC2)CC(C(=O)OC)CC1=O C1(CSCC)CCCC1C(=O)NC1CCC(CC)C1.n12cc(nn1)C1(CC1)C2 C1(CNC(CC(CC)(C)C)=O)CCN(C(C2CCCCS2)=O)C12CCC2 N1(C(C=CC2N(C(Cc3n(C)cnc3)=O)CCC2)=O)CCCC12CCCCC2 C1(OC2CN(C(CC(C)OC)=O)C2)CCN(C(=O)CC2CCCS2(=O)=O)CC1 c1(C(N(CC(C)N(C)C(C2C3CCCCC23)=O)C)=O)ccc(C#N)c(O)c1 Cc1cc(F)c(CN2CCC(CC(=O)Nc3cccc(C(C)C)c3C)C2)cc1F C1(NC(c2n(C)c(O)nc2)=O)C2CCN(C(C3CCCN3C(N)=O)=O)C2C1(C)C CCCC(C(O)C(=O)Nc1cc(C)cnc1F)NC(=O)C(C)C(F)(F)F C#CCC(CC(F)F)C(=O)N1CC2CC(C(=O)N(CC(=O)OC)C)CC2C1 O=C(CC(F)(F)C(F)(F)F)NC1COCCC1CNC(C1CCCOC1)=O C1(CNC(CC(CN(C)C2CC2)O)=O)CC2C(C1)C2(F)F.c12nnc(s1)C2 N1(C(c2c(C)ncs2)=O)CCCCCC1CNC(c1cc(C(N)=O)[nH]n1)=O N1(C(C2CCCN(C(CC)=O)C2)=O)CC(C2CN(C(=O)Cc3cncnc3)C2)C1 c1(NC(C(CCC)NC(c2cc(C#N)[nH]c2C)=O)=O)ccc2ccoc2c1 CC1CCCC1(C)C(N1CCCC1)=O.C1(CC2CC2)CC(=O)N2CCC(CC2)N1 c1(C(=O)NC(CNC(c2cncn2C2CC2)=O)CO)ccc2c(c1)OCCO2 c1(C(=O)NC(CNC(C=C(C)Cl)=O)C2CC2)cc(C(F)(F)F)n[nH]1 C1(C(=O)NC2CCC(F)CC2)(NC(C(c2ccnn2C)C)=O)CCC(C)(C)C1 CC1(CNC(=O)C(C#N)NC(c2ccco2)=O)C=CCCC1 CCC(O)C(C)C(=O)NCC1(C(=O)N(C(C)CCC(C)C)C)CCC1 C1(O)(CC(=O)NCC2COCC2NC(=O)C(F)=C2CCC2)CCOCC1 Cc1cnc(C(=O)NC2CCCCC2CNC(C2CC(C)(O)C2)=O)cn1 c1(C(=O)NC(CNC(C(C)CC2CCCC2)=O)C)ccc(Cl)c(N2CCCC2)n1 N1(C(CSCCOC)=O)CCCC(C)(CNC(c2ncc(C(N)=O)cc2Cl)=O)C1 CC(C)C(F)C(=O)NCC1CCC(NC(=O)C(C)(C)C2CCCCO2)CC1 c1(NC(C)CCN2CCc3ccccc3C2)ccc(S(=O)(=O)NC2CC2)cc1Br c1(C(N2CCCC(NC(=O)Cc3ccsc3)C2)=O)cccc2c1NCC2 c1(CC(C)NC(=O)C(c2cccs2)NC(=O)C(N)=O)cccnc1 N1(C(c2c(C)nc(C)n2O)=O)CC2CC3CC2C1C3NC(=O)C1=NOCC1 Cc1cc(OC(c2cccc(C(N)=O)c2)=O)ccc1F N1(C(C(C)NC(C)=O)=O)CC2CCCC(C1)C2C(=O)Nc1cc(O)ncc1Br c1(C(=O)NCC2CCC(NC(C(F)=CCC)=O)C2)sc(-c2cnn(C)c2)nc1C c1(C(=O)OC)ccc(OC)c(C(=O)O)n1.c1(C)cn(CC2CCCN2C(=O)CC#N)nn1 CC(C)CCCC(C)C(=O)NC(CO)C(N1CCCC(O)(CN(C)C)C1)=O c1(C(N2CC3(CC(CC(=O)NCc4cc[nH]n4)C3)C2)=O)ccc2nncn2c1 CC(C(=O)N1CCC(N(C)C)C1)S(=O)(=O)c1ccccc1.C12CCN(CC1)C2 CC(C(=O)OCCN(C(=O)C(C)n1cccc1)C)OC(C)(C)C N(C1CC2(CN(C(=O)C(=Cc3ccccn3)C)C2)n2ccnc21)C(C1C(=C)C1)=O C1(NC(C2(CCC)CC2)=O)CN(C(c2ccc(=O)n(C(C)(C)C)c2)=O)CCC1O C1(CC(=O)N2CCCC2)CC(=O)N1.c1(CC(=O)NC(C)C)ccn(C)c1 C#CCC(C(=O)OC)NC(=O)CCC1CCN(S(=O)(=O)Cc2ccccc2)CC1 c1(OC)ccc(NC(C2CCCC(=O)O2)=O)c(C#N)c1 C1C(C)CN=C2C=C(N=C(C(C)(C)C)N2)C(=O)N1.C(C)(C)(C)OC(C)=O.C(F)(F)F c1(CC)cnc(Cl)[nH]c1=NC(C)CCNC(c1c[nH]c(=O)cn1)=O c1(C(N2C3(CNC(c4c(C)scc4)=O)CC(C2)C3)=O)cccn(C2CCC2)c1=O C1(NC(c2cn[nH]c2)=O)CCN(C(C2CCC=CCCC2)=O)CC(O)C1 C1(C(=O)NC(CCSC)CO)(NC(c2ccc(N)cn2)=O)CCC(C)(C)C1 CC(CNC(=O)C(c1cncn1C)O)CC(=O)N(C)Cc1cnc[nH]1 C(=O)(C(C)(C)n1cnnn1)NC(C)C(C1CCCCC1)NC(c1ncn(C)n1)=O C(C)(CCC(=O)N1CCC(C(C)(C)NC(=O)CCCCOCC)C1)OCC C1(CC(=O)NCC2COCC2NC(=O)CCC2(F)CCCC2)CCCNC1=O C1(CCC(=O)Nc2cnc(C(F)(F)F)cn2)COCCC1=O C1(C(=O)NC(CCCOC)(C)C)CNC(=O)CN1C(=O)C=CC1CCC1 c1(C(N2CC(CCOC)N(C(=O)C=CC(C)C)CC2)=O)cc(C)cc(C)c1C C(=O)(C(C)(O)C(F)(F)F)NC1C(COC)CN(C(=O)CCC=C(C)C)C1 CN1CC(C(N2C3CCC2C(CNC(c2n[nH]cc2Cl)=O)C3)=O)CCC1=O c1(CC(=O)OC)ccc(F)cc1C.c1(C(C#C)NC)ccc(Cl)cc1 C1(CNC(c2ccc(C(C)C)cc2O)=O)COC(C)(C)CN1C(=O)CC C(CC(=O)NOC(c1ccccc1)C1CC1)N(C(C)C)C(C1CCN1C)=O c1(NCc2ccc(CC)s2)ccc(S(=O)(=O)N2CC=CC(O)C2)cc1C#N c12nc(C)c(s1)[nH]2.N1(C(=O)NCc2cc(C)[nH]c2)CCOCC1c1ccc(Cl)s1 CCC1=C(C(=O)N2CC(CNC(=O)C(C)CC3CC3)C(O)C2)CCCO1 CCC(CC)C(C(=O)NC(C1CCCN1C(C1(C)CCC(F)(F)CC1)=O)C)OC C12(C(=O)NCCN=S(C)(C)=O)COC(C1)C(NC(=O)C=CC1CCOC1)C2 O=C(C1=NOC2(CCC2)C1)NC12CCC(C(N3CCCC3CC3CC3)=O)(CC1)C2 C#CCCC(C(=O)NCC)NC(=O)CC1(NCC(C)=CCC)CC1 CS(=O)C=CC(=O)N1CCCC1(C)CNC(=O)CC1CC2(CC2)CO1 Cc1cc(C#N)cc(Cl)c1NC(C1CC2CC1(CO)C2)=O C(C(=O)NCCN1CCCOC1=O)(C(C)(C)C)NC(CN(C(C)=O)C)=O C1(O)(CNC(c2c(C)ccnc2C)=O)CCCN(C(=O)Cc2c[nH]nc2C)CC1 C(c1ccccc1C#N)=CC(=O)NCC(C)(CC(C)C)NC(C(C)OC)=O N1(C(Cc2c(C)scc2)=O)C2CCC(C2)C1CNC(=O)C(C)(C)CF c1(OC)cc(C(=O)N(C)CCN(C(=O)C#CC2CCCO2)C)cc2c1OCCO2 C1(C(N2CC(CC(N3CCOC4CC34)=O)(OC)C2)=O)(CC)CCNC1=O n1(CC=C)nnnc1C(c1ccc(CCCOC)o1)NC(C)CCF C1(CNC(C(Cn2ccc(C)n2)C)=O)CN(C(c2ccnnc2S)=O)CC12CC2 C12(C(=O)NC3CC(C)N(C(c4c[nH]c(=N)o4)=O)C3)CCCC(C1)OC2 N1(c2nc(C)c(F)cn2)CCC2(CCCC2C(N2CCc3ccccc32)=O)C1 C1(NC(COCC(=O)NC)=O)CN(C(=O)CN(C)C2CC2)C2CCCCC12 C1(CNC(c2cn(C(CC)=O)nc2)c2nnnn2CCOCC)CC2CCC1O2 c1(CC(=O)NCC(CN(C(CNC(CCC)=O)=O)CC)(C)C)cccnc1F c1(CC(=O)NCC2C(CNC(=O)NC3CC3)C2(F)F)c[nH]nc1O.C1(=O)CN1 c1(C(N(C2CCN(C(CCc3nc(C)[nH]n3)=O)C2)CC2CC2)=O)ccccc1C C(=O)(C#CC1(CC)COC1)NC(C(C)NC(CC(CC)C)=O)(C)C c1(OC)cncc(C=CC(=O)NCC2(CNC(c3cccnc3O)=O)CCC2)c1 c1(C(=O)NC2C(NC(c3ccc(C)c(N)c3)=O)C2)csc2c1CCCC2 c1(OC)cc(CN2CC3(CCN3C(=O)CN3CCCCCC3)C2)cc(F)c1 N1(C(CCC#CC)=O)CC(NC(c2nnn3ccccc23)=O)CC12CCOC2 N1(C(C2C(C)N(C(c3ccc(OC4CC4)o3)=O)CC2)=O)CC2C(C1)C2(F)F C(CC(C)C(=O)NCc1ccc(C(=O)NC2(CC(N)=O)CC2)s1)=CCC c1(C(=O)NCC2(CNC(c3ncccn3)=O)CC2)ccc2c(c1)C(=O)NC2 C1(C(N(CCOCCNC(c2c(OC)nccc2)=O)C)=O)CCCCC1C1CC1 C(=O)(CCC(=O)NC(C)CC(C)NC(=O)CCCOC(C)=O)NC(C)(C)C c1(C(=O)NCC(C)(CC(C)C)NC(c2c(C)ncs2)=O)cc(C#N)c(O)nc1N C1(C(C)NC(=O)CC2(C)CCCO2)CCN(C(=O)CC2C=CCCC2)CC1 N1(C(CCCC=C)=O)CCC(C)C(CC(=O)NC2(c3nn[nH]n3)CC2)C1 Cc1ccc(NC2CCOC(C3CCCCC3)C2)c(OCc2cc[nH]c2)c1 C1(NC(C(CC)O)=O)CC2(C1)CC2NC(=O)Cc1cn(C)nc1C(F)(F)F c1(C(N2CC(F)(CNC(C=C3CCN(C)CC3)=O)C2)=O)[nH]nc2c1COC2(C)C C(C)(C(C)NC(=O)CN(C(C)C)C(C1SCC=C1C)=O)(C1CC1)OC CC1COC(CNC(=O)C(Cc2cn[nH]c2)NC(=O)C(F)=CC2CC2)C1 c1(C(=O)NCCn2cc(CNC(C34C=CC(CC3)C4)=O)nn2)c[nH]c2cnccc12 N1(C(c2ccsc2Cl)=O)CCCC2C1CCN2C(c1ccc(O)nc1Cl)=O C(CCC(C)CC(=O)N1CC2(C1)CN(C(=O)CC1(C)CCS(=O)(=O)N1)C2)=C(C)C C(C(=O)NCC1(C(C)(C)C)CCN(C(=O)C=Cc2cncn2C)C1)(C(C)C)SC C1(NC(C(=O)NCC2CC2)=O)CC2CN(C(=O)CC3(O)CC3)CC2C1 S(=O)(=O)(c1ccc(NCc2cccc([N+](=O)[O-])c2)nc1)NCC(CC)(CC)CO C1(CCNC(COCC(=C)C)=O)CC(OC)CN1C(C1CCC(F)CC1)=O c1(C(=O)NC(CC)CNC(c2c[nH]c(=N)s2)=O)nn(CC)nc1Br c1(CC(N2CC(C3CN(C(C4CCCCCC4)=O)C3)C2)=O)ccc2c(c1)CCC2 c1(CNC(C(C)C(F)(F)F)=O)ccc2c(c1)CCC2NC(c1c[nH]nc1C1CC1)=O N1(C(CCC(C)C)=O)CCC(C2CCCN(C(c3ccnc4cc[nH]c34)=O)C2)C1 c1(CNC(NC(C)CN2CCCC2)=NCCc2cccs2)ccc(S(N)(=O)=O)o1 c1(C(=O)NC2C(NC(C(C(C)C)NS(N)(=O)=O)=O)C2)cc2cn[nH]c2cn1 C(C(C)(C)n1cccn1)NC(C=CC(C)NC(C1CCN1C(C)(C)C)=O)=O N1(C(CSc2n(C(C)C)cnn2)=O)CC(C2CN(C(C3CC3(F)F)=O)C2)C1 C(C)(CCC=C(C)C)(C1CC1)NC(C(CC)C)c1nnnn1-c1cccc(OC)c1 CC(C)C(CNC(C1(C2CC2)CN(C(c2cc(Cl)cs2)=O)C1)=O)C(C)C Cc1ccc(C(N2CCC(C)(CC(=O)NCC(C)(C)CCO)C2)=O)cc1O N1(C(c2c(CC)nn(C)c2)=O)CCCC2OCCN(C(=O)C(C)C3CC3)CC12 N1(C(C2(CC)CNC(=O)C2)=O)CCN(C(=O)Cn2nccc2C)C2COCC12 N1(C(CSCC=C)=O)CC2CCC2(CC(=O)N(C2CCC2)Cc2ccccc2)C1 CCCCCCC(CC)C(=O)N1CCC2(CCCN(C(=O)C=CC3CCC3)C2)C1 c1(N2CC3CC(NC(C4(COC)C=CCC4)=O)C3C2)ncc([N+](=O)[O-])c(C)n1 C1(C(=O)NC2CCC2NC(=O)CC2OCCCO2)(OC)CCC(F)(F)CC1 C=CCC(C)(CC)C(=O)N1CC(C(=O)NCCCCF)C2(CC2)C1 C1(NC(C(CN(C(Cn2nnc(C)n2)=O)C)C)=O)CCCN(C)CC1 c1(C(N2CC(O)(CNC(c3cc[n+]([O-])cc3)=O)C2)=O)cc(O)ncc1F Cc1cccc2c(=O)n(CC(=O)OCc3cccc([N+](=O)[O-])c3O)cnc12 S(=O)(=O)(c1cccnc1NC(C)(C)CO)NCc1ccc(C(C(C)C)O)cc1 C1(NC(Cc2c(CC)noc2CC)=O)CC2CN(C(c3c[nH]c(Br)c3)=O)CC2C1 C1(O)(CNC(=O)C=CC=C(Cl)Cl)CCCN(C(=O)C(CO)NC(=O)C(F)(F)F)C1 C(CCCCN=[N+]=[N-])NC(C1C(NC(CC(CC)O)=O)CC1)=O S(=O)(=O)(c1ccc(NCC2(S(C)=O)CC2)nc1)NCCn1c(CC)nnc1 c1(C(=O)NCC23CC(CNC(C=CC(=O)N(C)C)=O)(OC2)C3)ccc(F)c(F)c1 N1(C(C2N(C(c3ncc(C)cc3F)=O)CCC2)=O)CC2(C)CC1CCO2 c1(C(=O)NCC2CCN(C(CC3(C=C)CC3)=O)C2)c[nH]cc(C)c1=O CC(C)(C)C(=O)C(=O)NC1CCCN(C(C2CCCCS2)=O)CC1 N(C1CCN(C)c2ccccc21)C(C1C(C)N(C)CC1)=O Cc1ccc(F)c(C(N2CCCCC2c2ncc(C)s2)C(=O)NCCC#N)c1 c1(NC(C(=O)NC2CC(N)C23CCC3)=O)cc(Br)c(F)cc1F C=CCCC(O)CN(C(=O)C(C)(C)C1CCCN1C(=O)CCC=CC)C C1(CNC(=O)C(O)Cc2cnc[nH]2)CCCCN1C(=O)CCC1CC2(CCC2)C1 C1(OC)(CO)CCCSC1.C12COCC1n1cc(nn1)CN(O)C2=O c1(CC(=O)NC2CC2CNC(=O)CN2CCCC2)nc2ccccc2s1 CC(C)C(CNC(=O)Cc1cnns1)NC(=O)Cc1cnsc1 c1(N(C)CCNc2cccc(C)n2)nc(=N)[nH]c(=NCC23CCCC2OCC3)[nH]1 Cc1ncnc(O)c1Sc1cnn(CC2CCCCC2)c1 c1(C(CNC(C2CC2C(N)=O)=O)NC(CCCSC(C)C)=O)ccc(F)cc1 C(=O)(C(C)(C)CF)OCCNC(C1(c2ccccc2Br)CC1)C C1(C(CNC(=O)NC2CCN(C(=O)OC(C)(C)C)C2)=O)CCc2ccccc2O1 c1(NC(C)=O)ccc(C(=O)NNC(=O)NC2(OCOC)CC(CO)C2)cc1F C1(OCCC(=O)N(C2CCN(C(C(C)OCCOC)=O)C2)C)CCCCCC1 C(=O)(C1=NOC(C)(C)C1)NC1C2CCC(F)(F)C12.CN1CCC2(C1)C(=O)N2 C1(Nc2nc(C)cc(CC)n2)CC2COCC(C1)N2C(=O)C(COC)OC C1(CNC(C2CC(CC)OCC2)=O)CCCN(C(=O)CC(=O)OC(C)(C)C)CC1 c1(NC(C(N2CCCCC2CCF)c2cn(C)nn2)=O)cc(O)c2ccccc2c1 N1(C(CC(C=C)C)=O)CCC(CO)(CNC(C2(CN3CCOCC3)CC2)=O)CC1 N1(Cc2n(C)nc(C(F)(F)F)c2Cl)CCc2[nH]c3c(F)cccc3c2C1 C1(C(=O)OC)CCC(C(=O)NCC2(CNC(c3nnc(C)s3)=O)CC2)CC1 C(=O)(C1=Cc2ccccc2C1C)NC1CCC(NC(c2cc(C(C)=O)oc2)=O)C1 N1(C(CC2ON=C(CC)C2)=O)CC(CO)C2(CCN(C(c3cncs3)=O)CC2)C1 c1(NC)ccccc1C(N1CCC(C(C)(C)C(=O)NC(C2CCCC2)CO)C1)=O C1(CCNC(Cc2nc(C)[nH]n2)=O)CCN(C(=O)CCOC2CC2)CC1(F)F C1(NC(=O)Nc2[nH]nc3n(Cc4ccccc4)nc(C)c32)CC1C1(C)CCOCC1 C1(CNC(CS(CC)=O)=O)CN(C(c2ccc(F)c(N)c2)=O)CCC1C CC1=C(C(=O)N2CCC(NC(=O)C(F)(F)C(F)(F)F)C2)C(C)n2ncnc2N1C C1(NC(=O)CCF)CCCCC1NC(c1ccc(F)cc1)c1nn[nH]c1Cl C1(C)(C(=O)OC)CC(O)CN1C1(CNC(C2CC2C(=O)NC2CC2)=O)CC1 C1(C(N2CCC(C)(NC(COC)=O)CC2)=O)CCCC2(CCOCC2)O1 N1(C(COCCCC#C)=O)CC(C2CC2C(N2CCCCC2CSCC)=O)C1 C1(NC(=O)CC2(C(F)(F)F)CC2)COC2C(NC(C3(O)CCSC3)=O)COC12 c1(C(C(=O)NCCC(C)N(C(=O)C#CC2(C)CC2)C)(C)C)cc(F)ccc1F c1(CC)cc(F)ccc1C(=O)NCC1CN(C(=O)Cc2cn(C)nn2)CC1C C1(SCCC2CC(NC(C(COC)(C)O)=O)C2)CC(C)CC(C)C1 N1(C(c2cc(CC)no2)=O)CC2CC(NC(c3ccn(C(C)C)c3C)=O)CC1C2 N1(C(C(C)CO)=O)CC2CC(C1)C2NC(c1cnn(CCO)c1)=O N1(C(C(CC#C)C2CC2)=O)CCCN(C(=O)CC2OCCC2(C)C)CC1 C12(CNC(c3cnc(CC)s3)=O)CCC(CC1)N(C(=O)CCOC(C)C)C2 CC1C(NC(=O)C(c2cccc(Cl)c2)O)CCN1C(=O)CCc1ccoc1 c1(CC)nn(C)c(Cl)c1C(N1CCC(CN(C(=O)C(=O)NC2CC2)C)C1)=O c1(NC(C2(OC)CCN(C(=O)CSC(F)F)CC2)=O)ccc2c(c1)OC(CN)C2 c1(C(N2CC(NC(CCSCC)=O)C2)=O)cn(C)nc1C1CCOC1 Cc1cc(C(=O)NC2CC(OCC(N3CC4CC3CN4C)=O)C2)c(O)nn1 CC1CCc2ncc(C(=O)N(CC(C)NC(=O)C#CC(C)(C)C)C)n2C1 CC1COCCN1C(C1CCCC(CNC(=O)CCc2nc(=N)[nH][nH]2)C1)=O c1(CNC(=O)CSC(CC)C2CCNC2=O)cccc(C(F)(F)F)c1 CCS(=O)(=O)c1cccc(C(=O)NC(C)CNC(c2cc(F)cc(Cl)c2O)=O)c1 N1(C(C(CC)SC)=O)CCCCCCC1C(=O)Nc1cc(C)ccc1CO Cc1cc(CNC(=O)C(F)CC2CCOC2)oc1C(=O)N(CCC(C)C)C CC1CC(C(=O)NC2CC(NC(=O)CC3CC4CCC3CC4)C2)CC(C)C1 C1(F)(C(=O)NCC2(C)N(C(C(F)=CC)=O)CCC2)CCC(F)(F)CC1 c1(C(=O)NCCN(C(C(C)=CC)=O)CC(C)O)ccc(COCC)cc1 N1(C(c2cc(OC)n[nH]2)=O)CCC(C(=O)NCc2ncsn2)C1(C)C Cc1cc(NC(C2CN(C(C3(C#N)CC3)=O)CC2(F)F)=O)c(O)cc1F N1(C(c2cccc(Br)c2F)C(=O)NCCCOC)CCC(S(=O)(=O)C(C)C)C1 C(CCCC(C)(C)CNC(C1CC2CCC1NC2=O)=O)(OC)OC C123CCC(CO1)(C2)NC(=O)NC3.C1(=Cc2c(C)n[nH]c2)CCC(F)(F)CC1 C(=O)(CCCC1CC1C)N(C1CCN(C(C2(C)CC=CC2)=O)C1)CCC N1(C(c2n(CC)ccc2)=O)CCCCC1C(C)NC(=O)Cc1ccns1 c1(C(N2CCC(C(C)NC(c3cnc(=N)[nH]c3)=O)CC2)=O)ccc2[nH]ccc2n1 c1(C(=O)NCC(CC)(CC)NC(=O)CSCC2CC2)cc(Cl)ccc1C(F)F N1(C(CCC(=C)Cl)=O)CCC(C2CC2)(CNC(c2cnc(-c3cccs3)o2)=O)C1 c1(CCC)ccc(C(=O)NCCC(C)NC(=O)C(C)(C)C2CCOC2)cc1 C1(NCc2onc(COC)n2)CCN(C(=O)COCCF)C1(C)C.C1C(=O)N1 c1(CN(C2CCCN(CC#C)C2)C(C2CCCN(CC)C2)=O)ccc(Cl)cc1F C1(CNC(c2c(CC)occ2)=O)CCCN(C(C2CCS2(=O)=O)=O)C1 Cn1ncc2cc(NC(C3(C)CCCN(Cc4cccc(O)c4Cl)C3)=O)ccc12 Cc1noc(C)c1C(C)C(=O)N(CCNC(=O)CC(C)C1CC1)C(C)C C1(NC(CNC(C)=O)=O)CCN(c2cc(F)ncn2)CC12CCC2 C1(C(=O)NC(CC)CNC(C23COCC2C3)=O)CC2(CSC2)C1 c1(C(=O)NCC2C(NC(CCCCOCC)=O)CC2)cccc(N)c1C(F)F Cc1ccc(C(N2C3CCC2CN(C(C2(O)CC(F)(F)C2)=O)C3)=O)cc1C#N N1(C(CCC(=O)OCC)=O)CCN(C(=O)CS(C)(=O)=O)CC1CC(F)(F)F N(C1c2ccccc2CC1NC(=O)C(F)(F)CO)C(Cc1cnc(C)s1)=O C1(CNC(C(c2ccccc2Br)(C)C)=O)COCCN1C(=O)COCCF Cc1nn(C)c2ncc(C(N3CCC(C)(NC(=O)C4=CCCCO4)C3)=O)cc12 c1(C(=O)NCC23CC(CNC(CCCCC#C)=O)(C2)C3)cc(C)c(S(N)(=O)=O)cn1 c1(NS(CCN(C(=O)NC)CC)(=O)=O)ccnc2cc(C(F)(F)F)nn12 CC1CCC(CNC(=O)COc2ccccn2)N(C(C2CC3(CC3)C2)=O)C1 Cc1cc(N(C(C)Cn2cnnc2)C)nc(=NC(C)CC2CC2)[nH]1 C1(CCC)(C(=O)NC(C)C(=O)N(C(C)C(=O)N(C)C)C)CCC1 Cc1ccc(C(=O)NC(c2ccnn2C)C(=O)NC2(CCF)CCC2)s1 C1(OC(C2CN(C(N(C)CCOC(C)(C)C)=O)C2)=O)CCOCC1 c1(CN2CC3C(C(N4C5CCC4CC(O)C5)=O)C3C2)ccc(Cl)cc1[N+](=O)[O-] C1(N(C(C(C)OCCCC)=O)C)CCN(C(C2CCC(CC)CC2)=O)CC1.CC(C)C C1(OC)CCCCC1C(=O)NC(C)CC1(O)CCN(C(C2CSC2)=O)C1 c1(C(=O)NCC(C)CN(C)C(c2n[nH]cc2Cl)=O)cncc2ncccc12 N1(C(C(C)S)=O)CC2(CC(NC(=O)CC3CCOCC3)CO2)C1 Cc1cc(CC(=O)NC2(CNC(C3CC4C(C3)C4(F)F)=O)CCOC2)ccc1O CC(C)C(C)(CNC(=O)CC1CC=CCC1)NC(=O)CCc1ccc[nH]1 C1(CNC(C(n2cc(C)nc2)(C)C)=O)CCN(C2CCCc3ccc(F)cc32)C1 C1(NC(CN(C(C)C)C)=O)CCCC(CNC(C23CSCC2C3)=O)C1 C1(CNC(C2CC(CNC(=O)CCOCC(F)F)C(O)C2)=O)CC2(CCC2)CO1 N1(C(C(CC(F)F)N(C(C(C)=C2CCCC2)=O)C)=O)CCOC(C)(C)C1C C(=O)(CC(C)C(C)C(C)C)N1CCC(CNC(c2ccc(C)cc2O)=O)C1 N1(C(CNC(=O)OCC=C)=O)CC2CC1CN(C(=O)CCc1cc(Cl)cs1)C2.OCC C1(NC(c2cc(Cl)on2)=O)CS(=O)(=O)C12CCN(C(C1(CO)CC1)=O)CC2 C1(C(N2CCCC(CC(C)C)C2)=O)CC2CC1CN(C(=O)CSC(C)C)C2 C1(CNC(=O)CCC2=CCCCC2)CC2(CCN(C(=O)C(F)OC(F)(F)F)CC2)C1 C(=O)(C(C)CCCCCC)NC(CNC(c1cccc(OCCC)c1)=O)CC c1(OCC)cc(C(N2CCC(NC(c3coc(C(C)C)n3)=O)CC2)=O)ccn1 CCCC(CCCNC(=O)CC1(N2CCCC2)COC1)NC(=O)CCS(C)=O Cn1ccc(C(=O)NC2CCCC2n2cc(C3(C)CCOC3)nn2)n1 C1(NC(C2C(OCC)C2)=O)CC(N(C(=O)CC2(O)CCC2)C)C1 c1(C(=O)NCC(CNC(c2cnc(Cl)s2)=O)O)ccnn1CC1CCC1 C(=O)(C#CC1(C)CCCO1)N1C(C(=O)NCCNC(C)=O)(CC)C=CC1 Cc1c(Br)noc1C(=O)NCC1(CN(C)C(C23CCC(C2)C3)=O)CC1 C1(NC(C2(C)CCNC2)=O)CC2CCC1C(NC(=O)CN1CC3CC3C1)C2 CC(C)CC(CNC(C1CCCO1)=O)NC(C1(C)CC(C#N)C1)=O n1(CCC)nc(C)cc1C(=O)NC(C)C(C)NC(=O)CC1(OC)CCOCC1 CCCC(CC)C(=O)NC(C)(CC)CC(=O)NC(COCC)CC CC1(C(N2CC(CC(F)(F)F)C2)=O)CC(O)CN1C(c1ccc(Cl)cn1)=O C1(NC(c2c(C(C)=O)c[nH]c2C)=O)CCCN(C(=O)CN2CCCC2CO)CC1 c1(C(=O)NC(C)CS(C)(=O)=O)cc(NC(C2(c3ccccc3F)CC2)=O)nc(Cl)c1 C12(CNC(C3(C)CCCO3)=O)CCC(CNC(C3COC(=O)N3)=O)(CC1)CO2 N1(C(C2(C#C)CC2)=O)CC2CCC1C(CNC(c1ncsc1C(C)C)=O)C2 N1(C(CCCc2onc(CC)n2)=O)CCCC(CN(C)CCc2ccon2)C1 N1(C(c2ccc(SC)cc2)=O)CCC(CC(=O)Nc2cc(Cl)ccc2I)C(O)C1 c1(C(=O)OC)cc(F)cc(S(=O)(=O)NCc2ccc(Cl)c(C)c2)c1F S(=O)(=O)(c1ccc(=NCCc2ccc(OCC)nc2)[nH]c1)NC(CCC)C1CC1 C1(CC#C)(C(=O)NCC=CCNC(=O)C=CC(C)CC)CCOC1 N1(C(C2(c3cc(C)no3)CC2)=O)CC=CC(NC(c2cc(C(N)=O)ccn2)=O)C1 N1(C(C2CCC(CC)O2)=O)CCC=C(C(=O)NC(C)C(F)(F)F)C1 c1(NCC)ccc(F)c(Cl)c1F.C1(C(=O)NC2CN(CC)C2CCC)CCCC1(F)F Cn1nnc(C(N2CC(O)(CCNC(c3ccccc3Br)=O)C2)=O)c1N N1(C(c2c(C)c(N)n(C)n2)=O)CC2CN(C(c3sccc3Cl)=O)CC2C1 C1(F)(C(N2CC(CN(C(=O)CC34CCC(CC3)C4)C)OCC2)=O)C(C)(C)C1(C)C c1(C(N(C(CNC(c2c(C)cc(SC)o2)=O)C2CC2)C)=O)cnn2c1CCC2 N1(C(C(c2cccc(Cl)c2)C)=O)CCN(C(=O)Cn2cnc(C(N)=O)n2)CCC1C C1(O)(CN(C(c2cnc(CC)[nH]2)=O)CC)CCCN(C(=O)C(C#N)C(C)C)C1 N1(C(c2cnn(C(C)(C)C)c2)C(=O)NCCCSC)CCSCC1c1nccs1 CCC(CC(=O)NCc1nc(C(=O)NC2CC2C)c(C)o1)OC CC1CCC(NC(=O)Cc2cc(Cl)ccc2Br)CN1C(=O)CSC(C)(C)C c1(C(=O)NCCN(C(c2occc2Cl)=O)CC)cccc2cccnc12 O=C(C#CC1CCC1)NCCCNC(c1cnn(C(C)C)c1F)=O CCC(CCOC)C(=O)NCC1CCCN1C(c1conc1SC(C)C)=O C12(CNC(C(C)(O)C3CCOC3)=O)CC(CN1C(=O)C(C)(C)c1ccccn1)C2 C(=O)(N=c1c(Br)c[nH]cc1Br)C1N(C(c2ccc(C)c(Cl)c2F)=O)CC(F)C1 c1(CC)noc(C)c1C(=O)NCC1CN(C(c2cnn(C(C)C)c2)=O)CC1C CC1(CC(=O)NCC2(O)CCOC2)CCN(C(c2cn(C3CC3)cn2)=O)C1 C1(CNC(C2N(CC)CCC2)=O)N(C(=O)C(CC2CCC2)OC)CCCC1(C)C c1(C(N2CC(C)N(C(=O)C=Cc3ccoc3)CCC2)=O)cc2c(n1C)CCOC2 CCCCC(CNC(=O)C1=CCN(C(c2cnnc(C)c2)=O)CC1)CCC Cc1nccn1CCC(=O)NC(CO)C(=O)NC(C)Cc1ccco1 c1(C(N2CCC(NCCOCCOC)CC2C)=O)cc(Cl)c(Cl)cc1O c1(C(=O)NC(CC)CN(C)C(C2CC(=C3CC3)C2)=O)c(C(F)(F)F)n[nH]c1C c1(C(=O)NC(CNC(C2C(c3c(C)ncs3)C2)=O)CO)cccc(N(C)C)n1 c1(N2C(CC#N)CN(C(C3CCSCC3)=O)CC2)ncnc2cccnc12 C1(NC(C(C=C)O)=O)CCC2(CC1)CN(C(c1csc(Cl)c1OC)=O)CCO2 c12n[nH]c(n1)S2.CCCCOC1CNC1 c1(CCC(=O)NC(CC(C)NC(c2cn(C3CC3)nn2)=O)C)ccc(Cl)c(F)c1 CC1OCCCC1C(=O)NC1(C)CCN(C(=O)CCC2CCC(=O)NC2)C1 N1(C(C)=O)CC2CC2(CN(C(C)C(=O)O)C(c2coc(Cl)n2)=O)C1 CCCCC(O)C(C)C(=O)NC1CN(C(c2cc(COC)cn2C)=O)CC1O c1(C(=O)NCc2ccccc2)nc(=NCc2ncco2)cc[nH]1 c1(NC(c2ccc(CS(C)(=O)=O)o2)=O)cccc(F)c1C(F)F Cc1cc(C)n(CC(=O)NCc2cc(C(=O)NCCC3CCCN3C)co2)n1 CCC(C)CCC(=O)N1CC(NC(=O)CN(C(=O)C(O)c2ccsc2)C)C1 C(=O)(C(O)CC(C)(C)C)Nc1c(C(=O)Nc2ncc3cn[nH]c3n2)ccc(OC)n1 c1(C(C)=O)cc(C(=O)N(C(Cc2cc[nH]n2)C(=O)N2CCC2C(C)(C)O)CC)no1 C1(C(N2CC(CC)OCC2)=O)CC(C)CCN1C(=O)C(O)C1CC1 CC1CC(C)(C(=O)NCC(C)CNC(C2CCCC(C)(C)O2)=O)CCO1 C(C(=O)N1CCOC(CN(C)C(c2cn(C)cc2C)=O)C1)(C(C)C)SC c1(C(=O)NCC(CC)(CC)NC(c2c[nH]nc2F)=O)ccc(N)c2ncccc12 n1(CCNC(c2nccc3[nH]ccc23)=O)ccc(=NC(=O)C=Cc2ncc[nH]2)nc1O N1(C(C(C)C(F)F)=O)CC2CCCN(C(=O)CC(F)(F)F)C2C1 C12(CNC(c3cccc(C(F)(F)F)n3)=O)CCC(CC1)N2C(c1ccon1)=O C1(CC(N2CC3CCC(C2)N3C(C2CC(CC3CC3)C2)=O)=O)CCCCC12CC2 C12CCC(CC1)N(C)C(c1cnc[nH]1)C(=O)N2.CCCCCCSC c1(C(=O)NCCNC(CCC2(C)CC2)=O)nc2ccccc2cc1C1CC1 N1(C(C2CCN(C(C)=O)CC2)=O)CCC(NC(=O)C(C)CC(C)C)C(C)(C)C1 C1(C)(CCC(=O)NCC(C)OC(F)F)CCCN1C(=O)Cc1ccsn1 N1(C(C(C=C=C)C)=O)CCC2(C(=O)NC(c3cnn(C)c3)CC)CCCC12 Cc1ccc(-c2noc(-c3cnn(CC(O)CO)c3)n2)c(C#N)c1 CC1CC=C(c2cc(CNC(c3ccc(O)c(C#N)c3)=O)n[nH]2)CC1 N1(C(CCCOCC=C)=O)CCCC(C2CN(C(C3(Br)CC3)=O)C2)C1 c1(C(=O)NCC2N(C(c3ccc(C(C)(F)F)nc3)=O)CC2)ccc2ocnc2c1 C1(NC(c2nn(C)c(Cl)c2)=O)CCC12CCN(C(=O)CC(C)(C)C1CC1)CC2 Cc1ccc2nc(C(N3CCCC(n4cccc4)C3)C(=O)NC3(C)CC3)cn2c1 C(N=c1[nH]c2c(c(=NC3CCCC(C)(C)C3)[nH]1)SCC2)c1c(C)c(Br)ccc1 c1(NC(C2CC3(CCCCC3)C2)=O)cnc2c(O)cccc2c1 C1(COC)C(C(=O)NCCS(N)(=O)=O)CCN1C(=O)COC1CC=CC1 c1(C(=O)Nc2ccc(NC(C(C)OC)=O)cc2C)c(C)nc2ccc(Br)cn12 CC(C)(CC(=O)NCC1CN(C(c2cc(N)cnc2Cl)=O)C1)C(F)(F)F C1(C2CC2)(C(=O)NC2(C=C)CCC2)CN(C(=O)CCc2ccsc2)C1 C1(C2(C)CC2)CCc2sc(C(=O)NC3CCCN(C(c4ccc[nH]4)=O)C3)cc2C1 CCC(CC1CCCCC1)C(=O)NCCn1cc(-c2cc(C#N)cs2)nn1 S(=O)(=O)(c1cc(F)cc(Br)c1)N1CCCC(CNS(c2c(C)nn(C)c2)(=O)=O)C1 C(=O)(C(C)C(C)O)N(C1CCN(C(c2ccnn2C2CCC2)=O)CC1)CC#C Cc1cc(C(N2CCCC(C(C)Nc3cc(O)ncn3)C2)=O)nc(C)n1 C1(CC(=O)OC)COC2(CCC2)CN1C(=O)C(N1CC=C(C#N)CC1)=O c1(C(=O)NC2CC(CNC(=O)C(F)C(F)(F)F)C2)csc([N+](=O)[O-])c1 Cc1ccc(C#N)cc1NC(=O)CNC(C1CCCC(F)C1)=O CCCCC(O)C(=O)N1CCC(CNC(=O)Cc2ccc(Cl)s2)(COC)C1 C1(N(C(c2n(CC)ccn2)=O)C)CCC(NC(=O)C(O)Cc2ccccc2)CC1 c1(C(=O)NCC(C(=O)N2CC(COC)OCC2)N=[N+]=[N-])cnc2ncnn2c1 c1(C(=O)NCCC2N(C(C3COC(=O)O3)=O)CCSC2)ccc2sccc2c1 c1(NC(C=C(CNC(CC(=O)NCC)=O)C)=O)c(OC)cccc1C C(=O)(C(C)CC(=O)N1CC=C(C(=O)N2CCOC(C(C)C)C2)C1)OC N1(C(CC)=O)CCC(C(CO)NC(c2ccnc(C(C)(C)C)n2)=O)CC1 N1(C(c2cc(CC)[nH]n2)=O)CCC2CCN(C(=O)CCC3(C)CC3)CC2C1 C=C=CC(C)C(=O)N1CCC1CCCn1ccc(C(=O)NCc2cc(C)[nH]n2)n1 Nc1ccc(C(N2CCN(C(=O)Cc3cccc(F)c3)CC2C(F)F)=O)cc1O c1(C(C)C)ccc(C(O)CN(C(=O)Nc2nc(Cl)sc2Cl)Cc2ccccc2)cc1 S(=O)(=O)(c1ccccc1Cl)NC(=O)C1=CCCN(Cc2cc[nH]c2)C1 C1(CC(=O)NC2CCC(CCNC(c3cnc(S)nc3)=O)C2)CN2CCN1CC2 C12CCN(CC1)N(CC=CC=C(Cl)Cl)C2C1CCOC1.C1(F)C(=O)N1.CC c1(COC)cccc(-c2ccnc(C(=O)Nc3nc(O)cs3)c2)c1 Cc1noc(C)c1S(=O)(=O)N1CCCCC1C(=O)N(CCCCO)CC1CC(N)C1 n1(CC(=O)N(C2CN(C(=O)CCCN(C)C)CC2O)C)ncc(O)nc1=O c1(NC(C2CCCN(CCN3CC(C)(C)C3)C2)=O)nccc(Oc2ccccc2)n1 C1(C(=O)NC2CCC(CC(=O)N(CC=C)CC=C)C2)NC(=O)OC1(C)C CN1CC=CCC1CC(=O)NC1(C)CC(NC(C2(F)CC=CC2)=O)C1 Cc1nc(C(C)C)oc1C(=O)NCC(C)(C1CC1)NC(=O)CC1C=CS(=O)(=O)C1 N1(CC(=O)NC2(CC(=O)NCC3COC(CF)C3)CC2)CCC(C(N)=O)CC1 C1(NC(C(C)NC(C2CCN(CC3CC3)CC2)=O)=O)CCC([N+](=O)[O-])CC1 C1(NC(CSC)=O)(CNC(=O)Cc2cccc(Cl)c2F)CCCCC1C C1(CNC(C(COCC)OCC)=O)CN(C(c2cc(OC)n(C)n2)=O)CCO1 c1(OC)cc(CCC(=O)NCCNC(C23CCC(F)(CC2)C3)=O)cnc1Br C1(CNC(C(CSC)OC)=O)CCN(C(=O)Cn2nnnc2C)CC1O C1(O)(C(=O)NC(C(=O)OC)C)CCN(CC(C)CO)CC1 c1(CSCC(N2CC(CC(C)NC(=O)C(O)C3CCC3)C2)=O)ccccn1 C1(CC)(NC(=O)CC2CC=CCC2)CCN(C(=O)Cc2c(C)n[nH]c2C)CC1 C(CC(=O)NNc1cccc(Br)c1F)c1c(C)cccc1 N1(C(Cn2c(CCC)ncc2)=O)CCCC(NC(=O)C(C)(C)n2cnnn2)CC1 CC1C(NC(=O)CC2COC(C)(C)O2)CCCN1C(=O)CCc1cccc(Cl)c1 c1(C(N2CC(C)C(NC(C3CCCCC34CC4)=O)C2)=O)cccc2c1OCCC2 c1(NC(=O)Nc2ccc(NC(=O)NC)cc2)ncc2c(n1)NCCC2 C1(CNC(Cc2ncc(CC)[nH]2)=O)CC2CCC1N2C(=O)Cc1cc[nH]c1 O=C(C(CCC1CCCCC1)N1CCN(CCF)CC1)NCC1CCOC(C(F)F)C1 CCCC(O)CC(=O)N1CCN(C(c2ccc(OC)cc2Cl)=O)C(CO)C1 C1(CC(=O)NCCOCCC(=O)NC(C=C)CO)CC(O)C1(C)C Cc1cccc(S(=O)(=O)N2CCOCC2c2ccc(F)c(F)c2F)c1F c1(C(=O)NC(CNC(CCOCCOCC)=O)(CC)CC)cnc2scnc2c1 C12CC3(CC(C3)NC1=O)C2.c1(C(=O)NC)scnc1C(C(CC=CCC)=O)CC N1(c2nnc(COC)s2)CCC(NC(C2CCCS2)=O)C(F)C1 C1(C(N(CCCCCC)C)=O)CC2CCC1N2C(=O)CCC1CC1 c1(OC)cc(C)ccc1CO.N12CCC(C1)NC(=NC)NCC2=O CC1CC(C(=O)NC(C)(CNC(=O)Cn2ccc(C(F)F)n2)C2CC2)=NO1 C1(CNCCC2N(C(=O)OC(C)(C)C)CCOC2)CCC2(CCC2)CO1 C1(CNC(c2nccc(CC)c2)=O)CN(C(=O)CCC2(O)CCC2)CCC1C NS(=O)(=O)C1(C(=O)NCC2CCC(NC(c3c[nH]nc3C3CC3)=O)C2)CC1 C1(C(=O)NC2(CNC(CCC(C)(C)F)=O)CCOC2)CCS(=O)(=O)C12CCC2 CCCC(C)(CC)NC(C1(N(C(=O)CCC2CC2(C)C)C)CC1)=O C1(CCOC)(NC(CC2CC(=C)C2)=O)CCN(C(=O)Cc2ccsc2)C1 c1(C(=O)NCCN(C2CCN(C)C2=O)CC)cc(C)c(Br)s1 CC(F)(F)CCCNC(C1CCCN1C(c1cnc(O)o1)=O)=O Cc1nc(CNC(=O)CC2COCCN2C(C2COCCN2C)=O)c(C)o1 C1(CNC(C=CC(=O)OCCCC)=O)CC2(CCC2)CN1C(C1CC1Br)=O C1(NC(c2cccnc2)=O)CCCN(C(C2CC2c2cccnc2)=O)CCC1 C1(NC(=O)Cc2ccon2)CCC2(CCCN2C(=O)Cc2cnc[nH]2)CC1 c1(SCCC2N(C(C(=O)Nc3n(C)c(Cl)nc3)=O)CCC2)cccc2nsnc12 N1(C(c2ccc(OC)nc2)=O)CC(OC)CC(NC(c2cnc(SC)[nH]2)=O)C1 C1(C(N2C(C(=O)OC)CCC2)=O)CCN(C(C2CC=CCN2C)=O)CC1(C)C N1(C(C2(CNC(c3c(CC)ccs3)=O)CC=CC2)=O)CCCN(C)CC1C C(C(COC)C(=O)NC1(F)CCN(C(=O)COc2cc(C)on2)C1)OC COn1cnc(C)c1C(N1CC(NC(C2CCN2C2CCCC2)=O)C(SC)C1)=O C(=O)(C(O)C(F)(F)F)NC(C)CC(=O)NCCC1CCCC1 C(=O)(CCC(=O)OC)N(C(C)CNC(=O)C(F)C1CCCC1)C c1(C(=O)NCCC2(O)CN(C(c3cc(CC)[nH]n3)=O)C2)nsc2ccc(C)cc12 c1(C(=O)NCC2(NC(c3c(OCC)nccc3)=O)CC2)cc(C)c(C)nn1 C1(N(C(=O)Cc2ccco2)C)CCCN(C(=O)CCc2ccccc2)C1 C(CC(C)C)(C(=O)NCCC1CCCO1)N(C(C(C)=C(CC)C)=O)C CC(C)C(F)(F)CC(=O)NCC1CCCCN1C(=O)C(C)SCc1ccccc1 n1(CC)ncc([N+](=O)[O-])c1C(N1CC(O)(CNC(C2C(F)(F)C23CCC3)=O)C1)=O c1(N2C3CN(C(C(=C)C(F)(F)F)=O)C(C3)C2)ccc2c(c1)N(C)CCC2 N1(C(CC2N(C(C)C)CCC2)=O)CCN(C(=O)C=CSc2ccccc2)CC1C N1(C(c2n[nH]cc2C(F)(F)F)=O)CCOC(c2cn(CC3CCOC3)nn2)C1 CCC(C)(C)C(O)C(=O)N1CCC2(C1)CN(C(c1c[nH]cc1C1CC1)=O)C2 c1(CCC(=O)NCC(F)CNC(c2cccc(O)n2)=O)ccc(O)c(F)c1 c1(OC)ccc(CN2CCCC(C(N3CC4CC4C3C#N)=O)C2)c(Br)c1 c1(C(=O)N(c2ncc(C(C)C3CC3)s2)CCO)cccc(-c2nnco2)c1 c1(C(=O)NC2CN(C(C3CCC(=O)NC3)=O)C2)cc2cn[nH]c2cn1 O=C1Cc2cc(C(=O)NC3CCCC3NC(c3ccn(C4CC4)n3)=O)cnc2N1 N1(C(C=Cc2occ(C)n2)=O)CCCC1C1CCCN1C(C1CCC2(CC2)C1)=O n1(CC2(C(C)NC(C3C(CC)C3)=O)CC2)cc(-c2ccccc2)nn1 c1(C(=O)NC2C(CNC(=O)CCC3OCCO3)CC2)cccc(Cl)c1F C(=O)(C1=C2CCCN=C2NN1)NCC(CC=C)NC(=O)Cc1ccc(Cl)nc1 Cc1c(F)ccc(CNC(=O)C(CCC2CC2)NC(=O)CSC2CC2)c1F CCCC(CC(=O)N1CCN(CC(C)O)CC1)NC(c1coc(CCC)n1)=O N1(C(C2(C(=O)OCC)CC2)=O)CCC2CN(C(=O)C3=COCCO3)CC2CC1 c1(CCN2CCCC(N(C(c3ccc(O)cc3F)=O)CC)C2)ccc(C)c(Cl)c1 C1(CNC(c2cnc(CC)o2)=O)CCC2(CO1)CC(NC(=O)C(F)CC(C)C)C2 C(=O)(CCCCc1ccccc1)NC(C)(CNC(=O)COc1ccsc1Cl)CO Cc1cc(C#N)cnc1C(N1CC(C)(NC(C2CC2(C)Br)=O)C1)=O C1(C(N2CC(CCC)C(OC)C2)=O)CC2(CCO1)CC2.C12CCN1C2=O N1(C(C(CCC)C)=O)CCC2CCN(C(=O)Cc3cc4ccccc4s3)CC2C1 N1(C(=O)OC)CCCC(C(=O)NCCNC(C2CC(=O)N(C3CCCC3)C2)=O)C1 CCCCCC(F)C(=O)NC1CC(N(C)C(c2ccc(CO)cc2)=O)C1 C1(C(C)C)CN(C(=O)Cc2cccnc2)CCN1C(=O)Cn1nc(O)ccc1=O Cc1scc(C(=O)NC(CNC(C2CCN(C(N)=O)CC2)=O)C(C)C)c1N Cc1ncccc1C(=O)NC1CN(C(C2CCC(F)(F)C2)=O)CC1O c1(C(=O)NCC(CCOC)NC(C2CCC3CC23)=O)nc(-c2cccs2)oc1C N1(C(c2cc(C)c(I)cc2)=O)CC2CC(O)C1C2N(C(=O)OC(C)(C)C)C1CC1 Cc1c(C(N2CC(N(C)C(c3ccc(CCF)cc3)=O)C2)=O)cnn1C(C)C O=C1Nc2ccccc2CC1NC(C1(O)CCC(C(F)(F)F)CC1)=O N1(C(C2(OCC)CCC2)=O)CCC(CC(C)NC(=O)COC2CCCCO2)CC1 C1(NC(CCC(C)SC)=O)CCCN(C(=O)CC2(C)CC(F)(F)C2)CC1 CCC(CC(F)(F)F)C(=O)NC(CNC(c1ccnc2ncnn12)=O)C(C)(C)C C1(C(N2CC(C)CC(NC(COCCOC)=O)C2)=O)C2(CCC2)C12CCC2 c1(OC)ccc(F)c(C(=O)N(C2CCN(C(c3nccc(C)n3)=O)CC2C)C)c1 N1(C(c2c(C)nc(Cc3ccccn3)s2)=O)CC2CCCC1C2CCO C(=O)(C(C)CCC(C)(C)C)N1CCC2(C(CSC(C)(C)C)C2)CC1.C1(=O)C2CC2N1 N1(Cc2scc(C)c2)CCN(c2ccc(OCCCO)cc2)CC1 c1(C(=O)NC2(COC)CCN(C(=O)C(O)C(C)C)CC2)cc(Br)c(F)c(F)c1F c1(C(=O)NC(CC(C)OC)C)ccc2nc(O)n(-c3c(C)cccc3C)c2c1 Cc1cc(F)cnc1C(=O)NCC1(NC(=O)COCCN(C)C)CCC1 c1(CNC(=O)NCC(c2ccc(Cl)cc2)C)ccc(N)c(F)c1 N1(C(C(CC(C)C)OC)=O)CC2C3CCC(C2C1)N(C(=O)C1=CCSC1)C3 C1(N(C(=O)COC2CC=CC2)CC)CCCN(C(=O)C=Cc2ccc(Cl)s2)C1 C(=O)(C(CCC(C)C)NC(=O)CNC(=O)C(F)(F)F)NC(CCC#C)C(=O)OC C1(CCO)CC2(CCN(c3ccnc(N(C)CC4CCC5(CC4)CC5)n3)C2)CO1 N1(C(c2n(CCCC)ncc2)=O)CCCCC1CCNC(c1nn(C)cc1N)=O C1(CC(=O)NCCC(C)N(CCC)C)CN(C(C2CSC2)=O)CC12CC2 Cc1[nH]nc2c1CCCC2C(=O)NCC(C)Oc1ccccc1F C(=O)(CCP(C)(C)=O)NCC1(COC)CCCN1C(=O)CCc1ccc(C)s1 CC(C)C(O)C(=O)NCC1CN(C(c2coc(Cc3ccccc3)n2)=O)CC1C N1(C(C=CC(=O)OCC)=O)CCCN(C(=O)CN(C)C2CC2)C(C(C)C)C1 C1(NC(C2CCCO2)=O)CN(C(=O)CC2CC2)C2(CCOCC2)C1 C1(C(C(=O)NCCOC)N(C2CCCCC2)CC2CC2)C2CCOCC12 CC1CC(C)N(C(CCC2CCCOC2)C(=O)Nc2ccccc2Cl)C1 C1(NC(c2n(CC)cc(Cl)c2)=O)CN(C(C2CC2OC)=O)C2(CCCCCC2)C1 C1(C)(CNC(CC2(N(C)C(C3(O)CCCCC3)=O)CC2)=O)CC=CCC1 CCC(C)CCCC(=O)NCCC(C)(C)CNC(=O)CCCC1CCCC(=O)N1 c1(C(=O)NC2C(NC(C3CC(C)(C)OCC3)=O)CC2)ncc(F)c2ccccc12 c1(OC)cc(CN2CCC(NC(C3CCNC(=O)C3)=O)C(O)C2)c(Cl)cn1 C1(C(=O)Nc2c(C(=O)OC)scc2)CN(Cc2scnc2Cl)CC(F)(F)C1 n1(CCN(C)C)cc(C(=O)NCC(O)CNC(C2CN(C)C(=O)N2)=O)ccc1=O N1(C(C23CC(C(=O)NC(CC#N)=O)(C2)C3)=O)CCCCC1C#N c1(CC)cc(C(=O)N(C(C)C(=O)N(C)CCF)C2CC2)n(C)n1 Cn1cncc1C1CCCC1C(=O)NCC(O)CC1CCCC1 CC12CCC(C(=O)NCCNC(=O)C(C)(C)CN3CCOCC3)(CC1)OC2 c1(CCCNC(c2cnn[nH]2)=O)cn(Cc2ccc(C(=O)O)o2)nn1 CC1(C)CCCC(C(N2CCOCC2CC(N2CCC2C2CCCC2)=O)=O)C1 C1(NC(CCOC)=O)CN(C(c2c(C)nn(C)c2C)=O)CC1C#N Cc1cc(S(=O)(=O)NCC(C)CCO)ccc1C1(C)NC(=O)NC1=O C1(C(=O)NC2CC(NC(C(C(CC)O)(F)F)=O)C2)Cc2ccccc2N(C)C1=O CCCCCC(O)CC(=O)NCC1C2CN(C(=O)Cn3c(C)csc3=O)CC12 Cc1cncc(C=CC(=O)NCC2CC2CNC(C2CCN(CC(F)(F)F)C2)=O)c1 c1(C(=O)NC(C(=O)NC(C#C)C(C)OC)c2cccs2)nc(=N)cc[nH]1 c1(CC)nc(Cl)c(F)c(=NC(C)CNC(c2ccc(CSC)o2)=O)[nH]1 CCCC(C(O)C(=O)Nc1conc1C(C)C)NC(=O)CCc1csnn1 CN1CC(C(=O)NC23CC(CNC(c4cc(C(F)F)cs4)=O)(C2)C3)NC1=O CC(C)C(O)CC(=O)N1CC(F)(F)CC1CNC(c1ccnn1C1CCCC1)=O C(=O)(CCCC(=O)OC)N(CCC(=O)NCC1CC1)CC#C Cc1nc(C)oc1C(=O)NC(C(N1CCCC1(C)CC1CC1)=O)(C)C.S(C)(=O)(=O)N CC1(C#CC(=O)N2CCC(CCNC(=O)Cn3nnc(C4CC4)n3)C2)CCCO1 C1(C(=O)NCC(CNC(C(C=CC)O)=O)(C)OC)CC(=O)CC(=O)C1 CC(C)C(F)(CNC(c1cnn(C(F)F)c1)=O)C(=O)N1CCC(O)C(F)(F)C1 Cn1nc(C(N2CC(CNC(C3CC3F)=O)C3(CC3)C2)=O)c(Br)c1Cl CCC(C)(C)C(O)C(=O)NCC(C(=O)NCCCn1ccnn1)C(C)C CCCC(C(=O)NCCN(N1CCCC(C)C1)C)NC(=O)OC(C)(C)C.C(C)=O c1(C(N2C(CCN(C(CN(C)CCO)=O)C)CCCC2)=O)cnn2cccnc12 c1(C(C2CCCC2)NC(CCNC(CC2C(OCC)CC2)=O)C)cnc(C)o1 C1(C(=O)NCC=CC(=O)NCCOC)CC1(C)C(C)C c1(C(N(CCCNC(CCC=CCC=C)=O)C)=O)cccc(F)c1C C=CCC(C)(CC)C(=O)N(CCC(=O)N(C1CC2CCC1O2)C)OC C12(NC(C(C)P(C)(C)=O)=O)CCC(CN(C(=O)Cc3cc(F)ccc3F)C1)C2 c1(C(=O)NCC(C)(CO)NC(=O)C(O)CN2CCCC2)ccc(O)nc1 N1(C(C(C(C)C)F)=O)CCC2(NC(C3CNC(=O)N3)=O)CCCC12 Cc1cncnc1N1CCCC(CNC(c2nn[nH]c2C(F)(F)F)=O)C1 Cc1c(NC(=O)NC2CCC(NC(C3CC34CCC4)=O)CC2)cccc1F c1(OC)cc(N2CCC(N(C(=O)COCCC3CCCC3)C)C2)nc(Cl)n1 c1(OC)cc(Cl)c(Cl)cc1CC(=O)NC1CN(C(c2ccc(C)cc2)=O)CC12CC2 C1(Nc2cccc(C3CC(=O)N(F)C3)c2)CNCC12CCOCC2 C1(N(C)C)CCC(NC(c2cscc2C(N)=O)=O)C1.c12cc(no1)CC(=O)C2 S(=O)(=O)(c1c[nH]c(C(=O)NC(C)CNC(=O)C(C)Cc2ccnn2C)c1)NC C1(OC)CCCC(C(=O)NCCC2CC(NC(c3ncc(C)cn3)=O)C2)C1 C1(NC(CCC2(C)CN(C(CCCCSC)=O)C2)=O)CCCCC1(C)O c12ccc(cc1Cl)S(=O)(=O)N(C)Cc1nnc(n1C)CN2.N1(SC)CCOCC1 c1(COC)nn[nH]c1C(=O)NC1CCC1C(=O)N(CCC(C)(C)C)C C(C(CC(C)C)NC(C1CCCN1CC(F)(F)F)=O)NC(CCOCCC)=O C1(C(=O)NC(C(=O)N(CC2=CCSC2)C)C2CC2)CC2(CCC2O)C1 N1(C(C2CCC2C(F)(F)F)=O)CCC(C(F)(F)F)C(NC(=O)CC2CCOC2)C1 Cn1nc(O)cc1C(N1CCC2CC12C(N1CCCC1CC(N)=O)=O)=O C#CCCC(=O)NCC1C=CC(NC(=O)C(C2CCCCC2)C)C1 C1(NC(c2ccc(C(C)C)o2)=O)(CO)CCN(C(C2CCOC2C2CC2)=O)C1 C1(C(N2CCC(O)(C(N)=O)C2)=O)(CC)CCN(C(C2CC2(F)F)=O)C1 C(=O)(CCCCC1CC1)N(CCNC(C1(c2ccccc2F)C(C)C1)=O)C1CC1 c1(NC(CC2(CSC)CC2)=O)ccc(NC(=O)C=CC(C)(C)C)c(C)c1 C(=O)(C1=CCCC1C)N(CCCNC(C(CC)C#N)=O)C(C)C c1(C(=O)NC(C2(O)CN(C(=O)C=Cc3cnc[nH]3)C2)C)ccc2ccncc2n1 Cc1cnc(C(=O)NC2CCC23CN(C(=O)CC2OCCC2C)C3)cc1Br C=CCCC(C(=O)N1CC(c2cc[nH]n2)C1)NC(C1(C)CC=CCC1)=O C1(NC(C=CCCC)=O)CCCN(C(c2ccccc2-c2ccncc2)=O)C1 Cc1nnn(CC(=O)NCC(c2ccccc2)CNC(=O)C=C2CCC2)n1 C1(NC(Cc2nc(C)sc2)=O)CN(C(c2cc(C#N)[nH]c2C)=O)CC1(C)C N1(C(C(CCC)OC)=O)CC=C(CNC(c2ccc(=O)n(CCOC)c2)=O)CC1 C1(C(N2CCC(CNC(C3(C)CCC3)=O)C23CC3)=O)CC(O)c2ccccc2O1 C1(C(=O)NC2CC(n3cc(COCC(C)O)nn3)C2)CC2CCC1C21CC1 CC1NC(=O)CCC1NC(c1cccnc1CNC(=O)C(F)C(C)(F)F)=O c1(NC(C2C(C(=O)Nc3ccc(CO)c(Br)c3O)C2)=O)c(Br)ccc(F)c1F C1(NC(c2c(OC)nccc2C)=O)CCCN(C(=O)CCOCC2CC2)CCC1 N1(C(C(CC)(C)C)=O)CC2CC(C1)N2.c1(SCC(=O)OC)ccncc1 C(=O)(C(CC(C)(C)C)N(CC(C)C)C(c1cccc(F)c1)C)NCC C(=O)(N=c1ccc(Cl)n[nH]1)C12C(CN(C(C3CCCC(OC)C3)=O)C1)C2 c1(C(N2CCC(NC(C3CCCC(N(C)C)C3)=O)C2)=O)cc2n(n1)CCNC2=O c1(CC)nncn1NC(=O)CCC1CCN(C(c2cnn3ccccc23)=O)C1 c1(C(=O)NCCNC(CCCN(C(C)=O)C)=O)ccccc1C c1(C(=O)NC2CC3CCC(C2)N3C(=O)CC2CSC2)ccc2c(c1)NCCC2 c1(CNC(c2cc(C(=O)OC)on2)=O)cnc(CN2CC(O)CC2C(C)C)nc1 CC1CN(C(=O)C(C)(C)N(C)C)CCCN1C(=O)CC1(O)CCCOC1 C1(CNC(C(CC)NC(N)=O)=O)CCC2(CN(C(c3cncnc3)=O)C2)O1 c1(COC)ccc(C(=O)N(CC(C)N(C)C(c2cc(-c3ccco3)c[nH]2)=O)C)s1 c1(NC(C2CC(NC(C(c3ccc(C)cc3)C)=O)C2)=O)c(F)cc(C#N)cc1F C1(C(N2CCCC2CC2CC2)=O)CCN(C(=O)C=Cc2cccs2)O1 c1(C(N2CCC(NC(C(C)C3CCCC3)=O)C2)=O)nccc2ccsc12 c1(C(=O)Nc2cnc(CC)nc2)ccc2c(n1)CN(C(C1(C#N)CC1)=O)CC2 N1(C(COCCCCCC)=O)CCN(C)CC1CNC(=O)CC1CCCOC1 C(C(CC(F)(F)F)NC(C)=O)NC(C1(C)CCCN(CC2(CC)OCCO2)C1)=O C1(C)(C(=O)NCCOCCN(C)C(C2CCCS2)=O)CCCCO1 C1(C(N2CC(O)(C(C)NC(CN(C(COC)=O)C)=O)C2)=O)CC2(C1)CC2(F)F C1(C(N2CCC(CCNC(C3OCCCO3)=O)CC2)=O)CC2CC(O)CC(C1)C2 C1(NC(=O)CCCC2CCC2)CN(c2ncnn3cccc23)Cc2nccn2C1 C1(C(=O)N(CCCCNC(=O)CC(C)OC(C)=O)C)(CC)CCOCC1 C(=O)(CCCCC(F)F)N1CCCC(C2N(C(CC(=O)N(C)C)=O)CCCC2)C1 N1(C(c2c(CC)c(C)sc2)=O)CCC(C)(NC(CC2CC(COC)OC2)=O)CC1 C1(C(N(CC(C)(C)NC(C(C)=CC2CC2)=O)C)=O)CCC(C)(C)OC1 Cc1ccc(C(N2CCC(F)(C(=O)NC3CC(C)C3)C2)=O)cc1C CC1CN(C(c2ccc(OCCO)cc2)=O)CC1CCNC(C12CC(F)C1C2)=O Cc1cnncc1C(N1CC2C(CNC(=O)C(c3ccc(F)cc3)CO)C2C1)=O CC1(CNC(=O)C(F)n2cccn2)CCCN(C(=O)CSC(F)(F)F)C1 N1(C(c2c(CNC(C(F)=C(C)C)=O)ocn2)=O)CC2CC(O)CC2C1 N1(C(c2c(C)cc(C)s2)=O)CCC(N=[N+]=[N-])(C(=O)NC(CC2CCCC2)CO)C1 C(=O)(C1=CCCN(C(C23CCC(C2)C3)=O)C1)N1CC(OC(C)C)C1 c1(C(=O)NC(CN(C(C(C)OCCC#C)=O)C)CC)cn(CCC(C)(C)C)nn1 c1(NC(C2CCN(C(c3c(OC)cccc3O)=O)C2)=O)cc(S(C)(=O)=O)ccc1C c1(OC)ccc(I)cc1C(N1CCCC1C(=O)NCc1cncc(Br)c1)=O C(=O)(CCC(C)(C)F)N1C(C(N(C)CP(C)(C)=O)=O)CCC1 CCC(CNC(c1ccn(C)n1)=O)(CC)C(=O)NCCCN(C)C(C)=O C1(CC)CN(C(=O)CSC2CC2)CCN1C(c1sc(CC(C)C)nc1C)=O N1(C(c2ccc(C)s2)=O)CCOC2(CCCCC2NC(c2c[nH]nc2C)=O)C1 C1(CC(=O)NC2CC2CNC(=O)NC(=O)C(Cl)(Cl)Cl)CCC(=O)N1 C1(C(=O)OCC)(C(=O)NC2CC(C)OC2=O)CCOCC1 C(C(CC(=O)N1CCCC(C(C)(C)C)C1)OC)NC(CN(C)CC)=O CC1(C)CC(NC(=O)Cc2cscn2)CN(C(c2cc(-c3ccco3)on2)=O)C1 CCS(=O)(=O)CCNC(C1CC(O)CN1C(C1(CC2CC2)CCC1)=O)=O C(C(CC(C)C)C(=O)NC(CNC(C1CCN(c2ccccc2)C1)=O)CO)OC CC(C(=O)NCCOC1CCN(C(=O)CCN2CCCCCC2)C1)C(F)F c1(CC)sccc1C(=O)NCC1(COC)CN(C(=O)CC(O)c2ccccc2)C1 Cc1ccc(F)c(CC(N2CC(F)(F)CC2CCNC(C2(O)CC2)=O)=O)c1 c1(C(N2CCC(OCC(=O)NCC(=C)F)C2)=O)ccc(C2CC2)cc1 c1(NC2CCN(CCC)C2)cc(N(C)Cc2ccc(C3CC3)s2)nc(C)n1 N1(C(C(C2CCOCC2)C)=O)CCOC(CC(=O)NCCc2ncon2)C1 N1(C(=O)CC2C=CCC2)CC2(C(=O)NCC3CCC4CC34)CC1CO2 C=Cc1cncc(C(=O)NCc2ccnc(C(=O)NC3CCN(C)CC3)c2)c1 N1(C(c2c(Cl)cn(CCC)n2)=O)CCCCCC1CNC(=O)CCF c1(CC)oc(C(=O)NC2COCC2C(=O)NCCCC2CCCCO2)cc1C C1(CNC(NC2C(C)(C)OCC2)=NCCCCl)CCC(c2ccccc2)=NO1 N1(C(CC(CC)CC)=O)C2COCC1CC(NC(c1c(C)cncc1C)=O)C2 C1(C(=O)NCc2n(C(C)C)ncn2)CCC(C2CC2)N1C(c1sccc1C)=O c1(C(C(=O)NCCC(=C)CNC(c2cc(=O)cc(Cl)[nH]2)=O)(F)F)cc(F)cc(F)c1 N1(C(C2C(CC)CCCC2)C(=O)NC2COC2)CCC2(CC1)CCN(C)C2=O C1(C(N2C(OCC(N(C)OCC3CC3)=O)CC2C)=O)CCCC12CCC2 C=CCCCN=C(NC1CC1)N1CN(C)C(=O)C1C C(=O)(CC1CCc2ccccc21)NC(C)(C)CCNC(C1CCCO1)=O c1(C(=O)NC(C(C(C)C)Nc2ccccc2)C)cccc(C2CC2)c1Cl C1(C)(CC)CC(NC(=O)NCCC(N)C2(C)CC2)C1 N1(C(C(CNC(c2ccc3[nH]ccc3c2)=O)OC)=O)CCC(C)C2(CCC2)C1 CCN=c1[nH]c(C(=O)NCC(C)(O)CNC(=O)C(C)(C)C2CCOCC2)cs1 c1(C(=O)NC(C2CCCN2C(c2cc(O)cc(F)c2)=O)C)cccn2nccc12 C(=O)(CC1OCc2ccccc21)N1CC=CC(NC(C(C)(C)N(C)C)=O)C1 N1(C(c2ccc(OC)cn2)C(=O)NC2CCCCC2)CC2CCCC(C2)C1 c1(C(N2CC(CCC)C(NC(=O)CC3CCC(C)O3)C2)=O)cc(F)ccc1F c1(C(N2CCC(C(C(N3CCC(COC)(CO)C3)=O)F)C2)=O)cc(F)ccc1F CCCCC(C(=O)N1CCC2CC12C(=O)N(CCC(=O)NC)CC)C(C)C c1(SCC)cnc(O)c(C(=O)NC2CCC(C)N(C(c3ccccc3F)=O)C2)c1 CON(CCC(=O)N1CCCCC(C)(C)C1)C(=O)C(C)CC(F)F Cc1ccc(SCC(=O)NC(CNC(c2ccc(C)c(F)c2)=O)C2CC2)c(C)c1 C1(NC(C(C)OC2CCCC2)=O)CCCCC1NC(c1cnc(O)o1)=O CCC(C)CC(C(=O)NCC1C=CCC1)NC(=O)Cc1cc(C)cs1 c1(SC)ccc(-c2nc(C3CC(O)C3)n(Cc3ccsc3)n2)cc1 c1(CNC(c2n(CC)ccc2)c2nnnn2CCSC)cn(CC)c(C)cc1=O N1(C(c2scc(COC)c2)=O)CCC2CCCN(C(=O)C=C(Cl)Cl)C2C1 c1(CN2C(C)(C(N3CCC(CN(C)C)C3)=O)CCC2)cccc([N+](=O)[O-])c1Br c1(CNC(=O)NCC2(C(C)(C)OC)CC2)cc(CSC2CCC2)no1 C(=O)(CC(=O)Nc1nccs1)NCCNC(C1CC(OC(C)(C)C)C1)=O c1(CC(=O)NC2C(C)N(C(=O)CC3(CO)CC3)CCC2)c[nH]c2cc(F)ccc12 c1(C(=O)NCCOCCNC(c2cc(C)c(C)s2)=O)cccc(Cl)c1O c1(CN(c2n(CC=C)c(C(C)(C)[N+](=O)[O-])nn2)C)cccc(C#N)c1 C=C1CC2(C1)CC(C(=O)NCC(CC=C)NC(=O)COCCC)C2 C1(C(N(C)CC2C(C)OCC2)=O)CCCCN(C(=O)CC2CC3(CC3)C2)C1 N1(C(c2c(C)nsc2C)=O)CCC(NC(=O)CC2(C#N)CCC2)C(C)(C)C1 C1(NC(C2CCCS2(=O)=O)=O)CCN(C(C2(CO)CC2)=O)C1Cc1ccccc1 c1(C(N(CC(C(=O)NCCn2c(C)ncc2)C)C)=O)ccn(C)c(=O)c1 C(=O)(C#CC1CCCC1)NC1CCCN(C(c2cc(C)nnc2)=O)CC1 c1(C(=O)NCCCNC(c2n(CC)nnc2C)=O)ccc(Cl)c(Cl)c1O C1(C2CCCN(C(=O)CC3CC3)C2)(NC(=O)COC2CCOCC2)CC1 C1(C)(C(N2CCC(OCCNC(c3c(C)n(C)cc3)=O)C2)=O)CCCCCC1 Cc1ccc(C=CC(N2CC(N(C)C(c3ccnn3CC3CCC3)=O)C2)=O)s1 N1(C(=O)CC2CCCC(F)(F)C2)CC2(CCCCN2C(=O)Cn2nccn2)C1 c1(CNC(c2ccc[nH]2)=O)cc(O)nc(CNC(C2CC3(C2)CC3F)=O)n1 Cc1cccc(OCC(N2CC(C(N)=O)(CNC(C3(C)CCCC3C)=O)C2)=O)c1 CC1(C)C(NC(C23CC(C#N)(C2)C3)=O)CCN1C(c1ccc(Cl)o1)=O N1(c2snc(CC)n2)CC2CCC1C(NC(=O)Cc1ccc3ncsc3c1)C2 C1(C(N2C(C)(C(=O)NCCC(COCC)O)C=CC2)=O)CCC(O)CN1C C1(NC(C=CC)=O)CCCN(C(=O)Cn2cc(C(F)(F)F)nn2)C1C N1(C(c2cccc(C)c2)=O)CCC2CCC(C1)N2C(c1cccc(F)c1O)=O CC(CC(N)=O)C(=O)NCC(n1cc(-c2cc(CC(F)(F)F)ccc2F)nn1)C c1(CC)ccc(C(C)NC(=O)NCCS(=O)(=O)CCO)cc1F CC1CC(=O)NC1C(=O)NCC(C)(F)CNC(=O)CN1CCOCC1 C1(C)(N(N2CCNC(=O)C2)C)CC12CCN(c1cnc(=N)[nH]c1)CC2.C=O N1(C(CC)C(=O)NC2CCC2CNC(=O)C=NOC)CCC(C(F)(F)F)CC1 c1(NC(C=CCCCCC)=O)ccc(C=CC(=O)NC2(C(O)CO)CCC2)cc1 C=CC(C)(C)C(=O)NCCCCNC(c1cn(C2CC2)nc1-c1ccco1)=O Cn1ccc(=O)c(C(=O)NC(C2CCCC2)CNC(c2ncc(Cl)nc2Cl)=O)c1 c1(NCC2CCCCO2)ccc(S(=O)(=O)NC2COCCN2CCSC)cc1Cl CC1CCN(C(C23CCC(F)(CC2)C3)=O)CCN1C(C12CC(C)(C1)OC2C)=O CC1(C)COCC(NC(=O)C(CO)NC(=O)CCP(C)(C)=O)C1 n1(CC)ccc(=NC(=O)CC(C)C2CCCN(C(=O)C(F)(F)C(C)O)C2)[nH]1 C1(C(=O)NCC2CCN(C(C3CN(C)C(=O)N3)=O)C23CC3)CC2(CCCCC2)C1 C12CC13CCN(CC3)C2=O.C1(c2cccc(Br)c2)(CNC(C)=O)CCCCC1 N1(C(C(C)NC(C2CC(F)(CO)C2)=O)=O)CC(CCC2CS(=O)(=O)C2)OC(C)(C)C1 Cc1ccc(F)c(OCC(=O)NC(CNC(=O)CSC2CC2)C2CC2)c1 C1(C(N2C(C3CCN(C(CSCC(N)=O)=O)C3)CCC2)=O)SC2C=CC1C2 C(=O)(CCCCCNCC(c1ccccc1)N(C1CC1)CC)OCC=C c1(C(=O)NC2(CNC3CC3c3cccc(Cl)c3)COC2)ccc(F)c(I)c1 c1(-n2cc(C(=O)NC(CC)(C)CNC(c3n[nH]cc3C)=O)nn2)cccc(Cl)c1 C=C(C)c1ccccc1NC(C1CCCCCC1)(c1nnnn1C1CCCC1)C C1(C(N2CC(CNC(CN3CC(=O)NC3=O)=O)OCC2)=O)CC2(CCC2)CO1 C#CCC(C(=O)NC(C)CN1CCCCC1)NC(c1ccnnc1)=O C1(O)(CCNC(CC(C)c2ccncc2)=O)CCN(C(c2coc(Br)n2)=O)C1 C(=O)(C(=O)N=S(C)(C)=O)N(C1CCN(C(=O)CCn2cc(Cl)cn2)C1)CC C1(C(=O)NCC(C)CN(C)C(c2cc(N(C)C)ccc2F)=O)C2CCC(F)(F)C12 N1(C(C(Cc2ccccc2)OC)=O)CC2CC(N(C)C(C3CC(F)(F)C3)=O)C1C2 C1(NC(C2C(C)(C)C2)=O)CCN(C(=O)Cn2cc(Cl)cn2)C12CC2 C(=O)(C(F)CC(C)(C)C)N(C(C)CNC(C1CCC(F)(F)C1)=O)C CC1(C)C(CNC(C2CC2C(F)(F)F)=O)CCN1C(=O)Cc1cccc(O)c1 c1(CNC(CCN(C(COCCCCC)=O)C)=O)c[nH]nc1C(C)C C1(C(N)=O)CCC(C(=O)OCC(=O)NCCn2cc(CC3CCCC3)nn2)C1 C1(C#N)(C(=O)NCCC(C)NC(=O)C(O)Cc2cnc[nH]2)CC12CCC2 CCCC(CC)CCC(=O)NCCCCNC(c1cnn(CC2CCC2)c1)=O C(=O)(C(CC1CCCO1)C(F)(F)F)NCC(C)N(C(=O)OC(C)(C)C)CC C(=O)(CC(C)C(C)(C)C)NCC1C(CNC(c2c(C)n(C)nc2C(F)(F)F)=O)C1 C(CC(C)(C)CC(=O)N(C1CCN(C(C2OCCOC2C)=O)CC1)CCO)OC C1(NC(CC2CCCN(C(C(C(C)C)=O)=O)C2)=O)CCn2nccc2C1 c1(C)cn2c(n1)CCCC2.N(C(=NCC1CC1)NC1CCC(O)CC1)C(CC)CC CC(C)CC(CNC(=O)CCN1CCOCC1)NC(C1CN(C)C1)=O c1(C(N2CCC(c3ncco3)C2)C(=O)NC(CC)C)ccc(C2CC2)o1 c1(OCCCc2n(C)cnn2)nc(=NCC2C3CCC(F)(F)C23)[nH]c2c1CSC2 c1(NCC(=O)NC(C)(C)CNC(=O)CC2CC(F)C2)cccc(C#N)c1 c1(OC)ccc(C(=O)NC2CN(C(c3ccc(C)o3)=O)CC2C)c2sccc12 c1(C(=O)NC(CNC(CCCCCOCC)=O)C)c[nH]c2c(Cl)cccc12 C(c1cc2ccccc2o1)=CC(=O)NCC1CN(C(CSCC(N)=O)=O)C2C1C2 CC1CN(C(C2CCC2(C)C)=O)CCCN1C(c1ccnc(C(F)(F)F)c1)=O C1(CC2CCCCO2)CN(C(C2(NC(=O)C=CC=C(Cl)Cl)CC2)=O)CCC12CCC2 Cc1cnc[nH]c1=NCCCC(=O)NC(=O)CC1CC1(C)C N1(C(CCN2CC(=O)NCC2)=O)CCC2CN(C(c3ccoc3)=O)CCC12 CC1COC2(C1)CN(C(C1CCN(C(c3sccc3C)=O)C1(C)C)=O)C2 C(C(C(=O)N1CCC1C(C)NC(=O)CCCOC(C)(C)C)NC(C)=O)OC.CCF C#CCC(C)(C(=O)NC(C)CN(CCCC)C)NC(c1ccc(=O)n(C)n1)=O C1(C(N(C)CC2CCCCN2C(C2CC2c2cccnc2)=O)=O)COCC(C)(C)O1 N1(C(CSCC)=O)CC2C3CCC(C2C1)N(C(C1(C)C=CCCC1)=O)C3 CON1CC(C(=O)N(CCCCC(=O)NC2CC(C(F)(F)F)C2)C)CC1=O C1(NC(c2nn(CC)nc2C)=O)CN(C(c2ccc(=O)n(C)c2)=O)C(C)(C)C1 N1(CC#C)CC2CCC1C1CN(C(c3nccnc3OC)=O)CC21 C#Cc1cnc(C(=O)NCc2ncccc2C(N2CC(S(C)(=N)=O)C2)=O)c(C)c1 C1(COC)(CNC(=O)Cc2nc[nH]n2)CCN(C(c2cc(Br)no2)=O)C1 C1(C(=O)NC(COC)COC)C(C(C)C)CCCN1C(=O)C=Cc1nccs1 c1(OCC)cccc(C(=O)NC2(CCNC(C3CC3OC)=O)CCCC2)c1N N1(C(C=C(C)C(F)F)=O)C2CCC1C(C)C(NC(=O)CC(C)(O)C1CC1)C2 C(C(C)(C)C#CC(=O)NCc1cn(CCOC)nn1)NC(c1c(CC)csc1)=O C(=O)(C1=NN(C2CC2)C(=O)CC1)NCC1CCN(C(c2ccc(C)c(F)c2)=O)C1 CC1C(C(=O)NCCc2ccnn2C)CCN1C(=O)CSC1CCCCO1 N1(C(C(=O)NCCC2CCC(C)(C)O2)=O)CCC12CCC(F)(F)CC2 C1(C(=O)NCCCN2CCN(C3CCNC3=O)CC2)CCC2(CCC2)CC1 C(=O)(C(C)C(O)CC)NCC1N(C(C=Cc2c(COC)cccc2)=O)CC=C1 C(C(C(=O)N(CCO)OC)C(C)C)NC(C1=C(C)CC1)=O N1(C(c2nc(C)[nH]n2)=O)CCC2(C1)CN(C(=O)C(c1c(C)noc1C)C)CCO2 C=CCCCCCCC(=O)NC(C(N1CCCC(C(F)F)C1)=O)c1ccoc1 C(c1csc(C)n1)=CC(=O)OC(C1CC2C=CC1C2)=O.C123CC(C1)(C2)NC(=O)CN3C C1(C(N2C(CNC(C=Cc3c(C)ccs3)=O)CC(O)C2)=O)CCC(=O)N(C2CC2)C1 Cc1cnn2ccc(C(N3CCC4C(NC(=O)CC(C)(C)C)CC34)=O)nc12 C1(O)(C2N(C(CCOC)=O)CCC2)CCN(C(=O)C=C(C)C)C1 CC(C)C(CCC(=O)N1CCC2CC12)NC(=O)NC1(C2CCCO2)CC1 c1(C2C(C(=O)NCCOCCNC(c3n(C)nnc3)=O)C2)ccc(F)cc1F C(=O)(CC(C)CCCCC)N1CCC(O)(CN(C(C2(C)CC(=C)C2)=O)C)CC1 N1(C(C(OC)OC)=O)CCN(C(C2CS(=O)(=O)C2)=O)C2(CCC2)C1 n1(CC)nc(CNC(=O)N(C)Cc2ncon2)c(Br)n1 c1(C(=O)NCCCN(C(C2CCCCC2)=O)CC)cc(F)cc(Br)c1C c1(CCCNC(COCCCC)=O)ncc(Br)cc1NC(C1CC1CF)=O c1(OC)ccc(C(N2CCC3CC23C(=O)N(CC(O)CN(C)C)C)=O)cc1 N1(C(C(COC)C)=O)CCC(O)C1C(=O)NCCCCC(N)=O c1(CC=C)cccc(C(=O)N(CC(C)C)C2CC2)c1.C1(C(C)C)C(=O)N1 N1(C(C(C)OCC)=O)CC(NC(c2nccc(C(F)F)n2)=O)C(O)C1 C(CCOCC(N)=O)(C(=O)N1CC(OC)C1)NC(C1C(CCC)C1)=O C1(CNC(c2scc(COC)c2)=O)CN(C(=O)CC2CSC2)CC1C(F)F Cc1cc(CCC(=O)NCCOCCNC(C2(c3ccc(Cl)cc3)CC2)=O)nn1C C(=O)(C(CO)C(C)(C)C)NC(CNC(Cc1c(C)nc[nH]1)=O)(C)CC(C)C n1(CC#C)cccc1C(=O)NCc1ccc(C(N2CCC(COC)C2)=O)s1 C1(CC(=O)NCC=CCNC(=O)COCC2CCCC2)CCCCC1(F)F CCC(C(=O)NC(C)(C)CN(C(=O)C(C)n1cnnn1)C)n1ccnc1 c1(C(=O)NC(C(C)NC(CN2CC(CC)C2)=O)C)ccc(C2CC2)c(C)c1 CC(C)C(C(C)NC(c1cnc(C2CC2)[nH]1)=O)NC(c1coc(Br)n1)=O Cc1ccc(C(=O)NC23CC(C2)N(C(c2cn(C)nc2C(C)(C)C)=O)C3)c(C)c1 N(C(=NCCNc1ccccn1)NCCc1ccn(C)n1)CC1(C=C)CCC1 N1(C(C(C2CC2)OCC)=O)CCOCC(C)(CNC(c2c(CO)noc2C)=O)C1 Cc1ccnc2ccc(C(=O)NCC(C)CN(C(=O)Cn3cc[n+](C)c3)C)cc12 c1(C(N2C(CN(C(C(C=CCCC)O)=O)C)CCC2)=O)ccc(=O)n(CCO)c1 C1(CC)CCN(C(C2CN3CCC2CC3)=O)C(C(N2CCC2C(C)O)=O)C1 Cc1ccc(C(=O)NCC2CN(CCc3ncccc3Cl)CC2(C)C)c(Br)c1 N1(C(c2cn(CC)nn2)=O)CCC(C)(CNC(C2(c3cc(C)on3)CC2)=O)C1 C=C(Cl)CC(C(=O)NCC1CCCC(C)(C)C1)NC(c1cccc(C#N)c1)=O O=C1CC(=O)CC(C(=O)N(CC(=O)NOCCF)CCN2CC3C=CC2C3)C1 C=CC(CCC)CC(=O)NCCC1(C)CCN(C(c2cn(C)nc2C(F)F)=O)C1 S(=O)(=O)(c1ccc(C#N)cc1Cl)N(CCC(C)CCO)C(C)(C)C c1(C(=O)NCC(CNC(CCNCCOC)=O)O)cc(OC)cc(Br)n1 C1(O)(CN(C(=O)CC2CC=CCC2)C)CCN(C(=O)C(F)OC(F)(F)F)CC1 CCC(C)(CC)C(c1nnnn1CCC1CC1)NCc1ccn(C2CCC2)c1 Cn1cc(NC(=O)Nc2ncccc2C(F)F)c(C(N)=O)n1 C1(CC(=O)N(C)CC2(NC(C(C)n3ccnc3)=O)CC2)CCCCCC1 N1(C(C(CC)OC)=O)CC(C)Oc2cc(F)ccc21 CC1CN(C(c2cc(-c3ccccn3)no2)=O)C12CCC2 c1(N2C(C)C(NC(c3ccc(-c4cccs4)o3)=O)CCC2)ccnc2ncnn12 C1(CCNC(c2cc(C)nn2C)=O)CCCN(C(c2ccc(F)cc2C)=O)CC1 C1(CNC(C(COC)C)=O)CCCCN(C(c2cn(C(C)(C)C)nc2C)=O)CC1 c1(OC)cnccc1C(=O)N(C1CCCN(C(=O)CC2CC3CC3C2)C1)C CCC(CC(=O)NCCC1CCN(C(=O)CC(C)C(C)C)CC1)C(C)C N1(C(COCC#C)=O)CC2(CCC(CNC(=O)COCc3cc(C)on3)O2)C1 C1(CC(=O)NC(CCCNC(CCCOCCC)=O)C)CCC(C)(C)C1 C(F)(F)(C(F)(F)F)c1scc(C(=O)NCC(C)NC(C(CC)NC(C)=O)=O)c1 C(=O)(C(COC)CC)NCCN(CCC)C(C1(C)CC1C)=O.c1ccc(Cl)nc1 N1(C(COC(CC)(C)C)=O)CCC(C)(C(=O)NC2(CCO)CC=CC2)CC1 C1(CNC(=O)C(=O)NC2CCOCC2)CC(F)(F)CN1C(C1CCC(F)(F)C1)=O N1(CC)CC(C(=O)N(C2CCCC2)CCNC(=O)CC(C)F)CC1=O C(CCC(=O)N1CC=CC1CNC(=O)CC1CCCC1C(=O)O)=CC(C)C c1(C(N2CC3OCC(NC(c4occ(C)c4)=O)C3C2)=O)ccc(F)c2c1CCC2 C1(S(N)(=O)=O)(C(=O)NC(CCCC)CNC(=O)CCF)CCCC1 N1(C(Cc2c(C)nc[nH]2)=O)CC2(CCCC2NC(=O)CC2CCC2C)C1 C(=O)(C(c1cccs1)=Cc1ccccc1)NC(CC=C)CNC(=O)CC1CC=CC1 C(=O)(C1=CC2(CCOC2)C1)NC(C1CCN(C(CC(CC)C)=O)C1)C CC1(C)CC(NC(c2cscc2SC2CC2)=O)CN1C(=O)CCF N1(C(CCCC#C)=O)CCC2(CC(NC(c3n[nH]c4ccc(F)cc34)=O)CO2)C1 C1(NC(c2cnn(C)c2)=O)CN(C(C2C(C(C)C)CCC2)=O)CC2(CC2)C1 c1(C(=O)NCC2(F)CC(NC(C3(OC)CCOC3)=O)C2)cc(Cl)n(C)n1 n1(CC(N2CCCC(N(C(CN(C)C(=O)C3CC3)=O)C)C2)=O)ccc2ccccc12 N1(C(=O)OC(C)(C)C)CCOCC(CNC2CCCN(CCO)C2)C1 Cc1nc2cc(C(=O)NCC(C3CC3)NC(C3CCCO3)=O)cc(O)c2o1 c1(C(=O)NC(CN(C(C2(n3ccnn3)CC2)=O)CC)C)cc(OC(C)C)ccc1C C(C(=O)NOC(C)CC(C)C)(C(C)C)NC(CCSCCC)=O c1(-c2nc(C)nn2-c2nnc(S)nc2O)ccc(N=[N+]=[N-])cc1 CC(=O)C(C)CCC(=O)N1CCC2(CC(CO)C2)C1 C(C(C)(C)C#CC(=O)N1CC(O)(C(N)=O)C1)NC(C(C1CC1)SC)=O c1(CC(C)C)ccc(CC(=O)NC(CNC(=O)C(O)C2CCC2)C2CC2)cc1 C1(NC(c2cc(C)oc2C)c2nnnn2C(C)C)CC2CCC(C1)S2(=O)=O c1(CCC2ON=C(C)C2)csc(=NC2CCSCC2)[nH]1 C1(C)(C(c2nnnn2-n2cccn2)NCC(C)(C)COC(N)=O)CC=CCC1 C1(NC(C(C)(C)Cc2ccccc2)=O)CC2CN(C(=O)C=Cc3cc[nH]n3)CC12 c1(C(=O)OC)nc(C(=O)NC(c2nocc2C(=O)NC2CCOC2C)C)cs1 N1(C(c2c(OC)c(C)sc2)=O)CCC(NC(=O)C(C)SC(F)(F)F)C1(C)C c1(OC)ccc(C(N2CCC(C)C(NC(c3cn(C)cn3)=O)C2)=O)c(N)c1 c1(CC)ccccc1CC(N1CCC(NC(=O)C(c2c[nH]ccc2=O)=O)CC1)=O c1(N2CCC(C#C)CC2)ccncc1S(=O)(=O)NCC1CCNC(=O)C1 CCCC(C)CC(=O)N1CCC(F)(CNC(=O)CCc2nc(C)no2)C1 Cc1cc(Cl)cc(C(=O)NCC2(CNC(c3sccc3CN(C)C)=O)CC2)c1N c1(CNC2CC(C)CN(C(c3n[nH]c4c3COC4)=O)C2)c(F)cc(O)cc1F N1(C(C2C(C(C)C)CCO2)=O)CCC(C)(C(=O)NCCN2CCCC(O)C2)CC1 Cc1nc2ncc(C(N3C4CCCC3CN(C(=O)C(O)C(C)C)C4)=O)c(=O)n2[nH]1 N1(C(c2c(C(C)(C)C)noc2)=O)CCC(C(F)F)(CNC(c2cnccn2)=O)C1 N1(C(c2c(OC)cccn2)=O)CC(CNC(C23COCC2C3(F)F)=O)CC(C)(C)C1 c1(C(=O)OCC)oc(NC(=O)NCC2CN(C(C)C)CC2C)nc1CC C(=O)(C1CCCc2ccccc21)NC1CC(NC(c2ccnc3ncnn23)=O)C1 c1(CC(=O)NCC2CN(C(C3(CC)CCOC3)=O)C2)c[nH]c2ccc(Br)cc12 N1(C(c2ccc(CC)s2)=O)CCC(C)(C)C(C(=O)NC2CCC(C)(C)CC2C)C1 C(=O)(C(CO)C(F)(F)F)N1CCC(NC(c2cc(C)nc(C)c2)=O)C(CO)C1 C(c1cc[nH]c1)=CC(=O)N(C(C(=O)OCCC)C)C(=O)CC1CCCCC1 CC12CCC(C(=O)NC3CCCC3NC(c3cnc(C4CC4)o3)=O)(CO1)C2 C1(C(N(CC#CC)C)=O)CCN(C(=O)C(N2CCOCC2)C)C12CCC2 c1(C(N(CCN(C(C)C)C(c2ccc[nH]2)=O)C)=O)cc(C(F)(F)F)c[nH]1 c1(NC(N2C(Cc3ccc(C)c(C4CC4)c3)CC2)=O)cc2c(nc1O)CCN(C)C2 C(=O)(C(CC(F)F)N(C(=O)C(N1CCOC1=O)C)C)NCC(C#C)C(C)C c1(C(=O)NCCC2CN(C(c3ccon3)=O)CC(C)O2)ncc2[nH]ncc2n1 Cc1cc2c(C(N3CC=CC(NC(c4snc(Cl)c4Cl)=O)C3)=O)cccc2[nH]1 c1(-c2nc(COCC)nn2Cc2ccncc2)ccc2[nH]ccc2c1F CCC(CCC(=O)NC1CSC1)NC(=O)Cc1cnn(C)c1C c1(NC(c2n(CCCC)nnn2)CCOC)ccc(OC)nc1C.C1CCC1 N1(C(C2(COC)CCCO2)=O)CCCCC(NC(c2ccc(NC)cc2Cl)=O)C1 c1(C(=O)NC2C3CC(NC(=O)CCc4nncs4)CC32)ccc(Cl)c(F)c1F C12(NC(c3cccc4nonc34)=O)CCC(CC1)N(C(=O)CC1CCCCO1)C2 C1(C(=O)NCCC(C)C)Cc2cccc(OC(C)(C)C)c2O1 C(CCN=C(NCC1CC(OC)(OC)C1)N1CC(O)C2(CC2)C1)OC C1(C)(CNC(c2n(CC)ccc2)=O)CCCN1C(=O)Cc1cnoc1 n1(CC(=O)NCCOC(C)=O)cc(CC(=O)NCC2(CC(N)=O)CC2)nn1 Cn1cncc1C(O)C(=O)NCC1(F)CC(CNC(C2CC2c2ccccn2)=O)C1 c1(CCC(=O)NC(CNC(c2ncccc2O)=O)C2CC2)cc(Br)ccc1F C1(NC(C2N(C(C)=O)CCC2)=O)CC2CC1N(C(c1cnccc1C)=O)C2 C12(C(N3CCCC(NC(CC(C)(F)F)=O)CC3)=O)CCCCC1NC(=O)C2 c1(N(CC(C)C(C)(C)C)C)nc(N2CCOC(C#N)C2)nc2c1CC(C)CC2 c1(C(=O)NC2C3CCN(C(CCNC(=O)C=CCl)=O)C32)cnn2ccsc12 N1(C(C(C=C)CC)=O)CC(NC(c2ccc(C)c(O)n2)=O)C2(CCC2)C1 CC(C1=CCN(C)CC1)NC(C1CCCCCCN1C(=O)CN1CC2CC2C1)=O C(C)(C(C)(C)C(=O)N(CCOCCO)CC)NC(CC=C=C)=O C1(CC=C)(NC(=O)COC2CC(F)(F)C2)CCN(C(c2cccc(C3CC3)c2)=O)C1 c1(NC(C2C(CNC(C(C)=C(CC)C)=O)C2)=O)cnc(CC2CC2)nc1 CC1(C)CCCC(O)(C(=O)NCC2CC2NC(=O)CCSN2CCCC2)C1 N1(CCC)C(=O)NC(c2nn(C)cc2I)C2=C1C(C)(CCC)NC2=O C(=O)(CCC(C)(C)C(=O)NCC1CCCN1C(C1CCC([N+](=O)[O-])CC1)=O)OC C(=O)(CS(=O)C(F)(F)F)N1CCN(C(CSCC#C)=O)CC1C(F)F C#CCCC(O)C(=O)N1CC2CC(N(C(=O)CCCCSC)C)C1C2 N1(C(C(C=C)(C)O)=O)CC(C2CCN(C(c3nscc3Br)=O)CC2)C1 C1(CC)CN(C(=O)CNC(=O)C(F)(F)C(F)F)CCC1NC(c1ccc(C)s1)=O C(C)(CCC(=O)OC)OC1CC(NC(C=CC=CC)=O)(CO)C1 C1(C(=O)NCC(CCCC)NC(c2cnn(C(F)(F)F)c2)=O)CC2CCCC2C1 C1(CNC(C(C)OCC(C)C)=O)CCCCN(C(c2cnc(C(F)(F)F)s2)=O)C1 c1(N(C)C2CC2)nc(=N)[nH]c(=NC2CCCN(C(C3CCCN3C3CC3)=O)C2)[nH]1 C#CCCC(C(=O)OC)NC(C1C=CC(NC(c2csnc2OC)=O)C1)=O c1(C(=O)NCCN2CCCC2)ccc(CNC(c2ccn(CC(F)F)n2)=O)o1 c1(C(N(CCCN(C)C(c2cc(F)cc(F)c2)=O)C)=O)cc(F)ccc1Cl c1(C(N2CCC(NC(C(C)C)=O)C2C)=O)cc(Cl)c(F)cc1N N1(C(C=C(CCC)C)=O)CC2CCCC1C2CNC(c1ncnn1C(C)C)=O c1(C(N(C(c2ccccc2)C(C)NC(C(C)O)=O)C)=O)ccc(C2CC2)c(Cl)c1 c1(C(N2C(NC3(CCOC)CC3)CCC2)=O)ccc(C#N)c(Cl)c1 N1(C(C2C(CCOC)C2)=O)CC(O)CC1C(=O)NCc1ncc(C)o1 C12(COC)CC(NC(c3cnc(C4CC4)cc3C)=O)(CN1C(=O)CCCC(C)=O)C2 CS(=O)(=O)C1(C(=O)NC2CCCC2NC(=O)CNS(=O)(=O)C2CC2)CC1 c1(C(=O)NC(CC2CCCC2)CO)cccc2c1COC2 Cn1nc2c(c1C(N1CC3OCC(NC(C4(Cl)CC4(C)C)=O)C3C1)=O)CCCC2 CCCC(C(=O)N(C)CC1CCCN1CC)NC(=O)CC1CC(C)=NO1 c1(C(N2CC3C(C(N4CC5C=CC4C5)=O)C3C2)=O)ccc(F)c(Br)c1F C(C(C)(C(=O)NCCc1cnnn1C)NC(c1ccn(C)c1)=O)SC C(=O)(C1OCCc2ccccc21)N1CC(N(C)C(C2CC23CC3)=O)C1 C1(C(NOC(C)(C)C)=O)CCN(C(=O)CC2CCOC2)C12CCC2 c1(C(=O)NCC2C(NC(=O)C(=O)Nc3ccccc3)C2)cc2n(n1)CCCC2 C1(C(=O)NCC2(C)C=CCC2)(CCNC(=O)CC2CCS(=O)(=O)C2)CCOCC1 C(=O)(C(C)(C)CN(C)C(=O)NC1CC(C(=O)OC)C1)OCC c1(CNCCN(C(C(C(C)C)OCC)=O)CCCN(C)C)coc2c(C)cccc12 c1(N2CCN(C(Cc3nc(SCC)sc3)=O)CC2)cnc2nc(C)cnc2n1 c1(C(=O)NC2CN(C(c3scc(C)c3C)=O)C(C)CC2)cc2cnccc2o1 c1(C(=O)NC2CC2CNC(c2cc(-n3ccnc3)ccn2)=O)cnc(O)c(F)c1 c1(C(=O)NCC2CCN(C(C3(CCF)CCC3)=O)C2)cnnc2ccccc12 c1(C(=O)NC2(CNC(C(C3CCCOC3)OC)=O)CCOC2)cc2occc2n1C N1(C(CCN(C)C(=O)OC(C)(C)C)=O)CCCCC1CNC(C1COCCOC1)=O N1(Cc2n(C)ncc2)CC2CCN(C(c3ccc(OC4CC4(F)F)cc3)=O)C2C1 C1(NC(c2ncnc(C)c2C)=O)CC2CCC1CC2NC(C1CC2(CCC2)C1)=O Cc1cccc2nc(NC3C4CN(C(C5CC56CCC6)=O)CC34)sc12 C(=O)(N=c1cc[nH]cc1F)C1C2(CCN(C(=O)Cc3ccc(OC(C)=O)cc3)C2)C1 C#CCC(C(=O)NC)NC(=O)C(CCOC)NCc1conc1C C(=O)(C(CN(C)C)C(C)C)N(CCNC(C(C)=NOCC#N)=O)C.c1(S)cccc(C)c1 C1(CNC(C(C)CF)=O)CN(C(=O)C=Cc2ccc(Br)cc2)CC1(C)C c1(CC(=O)NCC(C)NC(C2CCC(CC)CC2)=O)ccc2cc(O)ccc2c1 CCCC(C(=O)NCC(=O)OC)NC(=O)CC1CCCO1 N1(C(CCC2C(C)(C)C2)=O)CC(CNC(=O)CSc2cccnc2)CC12CCC2 O=c1oc2cccc(CNC(C3CCNC3)C3CCC3)c2[nH]1 C1(C(=O)NCC(=O)NCC2(C(=O)NC)CC2)CC2(C1)CC2C(=O)O.C(C)(C)(C)N CC1(NC(C2CNC(=O)N2)=O)CCC(NC(C2(F)CCOC2)=O)CC1 C(C)(C(C)(C)C(=O)N1CCC(F)CC1)NC(C(CC)NC(N)=O)=O N1(C(c2ccn(C)c2)=O)CCCC2(C1)CN(C(=O)CC1CCC3CC13)CCO2 CC1=C(C(=O)N2CCC(F)(C(=O)N(CC#N)Cc3ccccc3)C2)CCCO1 C(=O)(C1CCCc2ncc(C)n21)N(C1CCCN1C(=O)CN(C)C(C)=O)CCC CC1CCC(NC(=O)C(n2nnnc2C(C)(C)C)C)CN1C(=O)CC(C)(C)C c1(C(N2CCN(C(c3c(C)ocn3)=O)CC2C)=O)ncnc2cc[nH]c12 CC(CS(C)(=O)=O)C(=O)N1CCC(NC(=O)CCC2OCCO2)C(C)(C)C1 c1(C(=O)NCCC(C)NC(C(C)N2CCC2)=O)cc([N+](=O)[O-])cnc1O c1(C(=O)NC(CNC(CSCC#C)=O)C(C)(C)C)cnc2ccccn12 O=C(CCCCCCCCCO)NCCC1(NC(c2cn3c(n2)SCC3)=O)CC1 N1(C(CCN(C)CC)=O)CCOC(C)(CNC(c2cccc(F)c2Br)=O)C1 CC1=C(C)CC(C)(NC(=O)C(c2cnn(C)c2)NC(C2CC2C(C)C)=O)CC1 C1(NC(c2c(CC)nco2)=O)CCCN(Cc2ccc(Cl)cc2C)CC1 CC1(C)CC(NC(=O)NCC2(CF)CC2)CO1 N1(CCn2cc(CCC(=O)NC)nn2)CCN(C(=O)C2=NOCC2)CC1=O N1(C(C(C)=CC)=O)CCCn2nc(C(=O)NCCCc3ccccc3F)cc2C1 C1(CCCC)CCC(C(=O)Nc2cccc(NC(C3CC3C3CC3)=O)c2)CC1 C(=O)(CCC(C)(C)C#N)NCC1C(NC(C(CN(C)C)(F)F)=O)C1 C(=O)(C#CC1(C)COC1)N1CCC(NC(C(C(C)C)SCC)=O)C12CC2 C1(N(C)C)(C(N)=O)CN(C(=O)CN2CCSCC2)C1.C1CC(=O)NCC1 Cc1n[nH]c(C)c1CCC(=O)N(CCCCCNC(c1ccncc1)=O)C Cc1cc(CNC(C2COCC2NC(c2nccnc2O)=O)=O)cc(F)c1 C(=O)(CCC(=O)NN(C)C)N1CCN(C(C2CC(C(=O)OC)CC(CCl)C2)=O)CC1 C1(N(CC#C)C(c2cc(CC)c[nH]2)=O)CCN(C(=O)CN(C)CCC)CC1 N1(C(C=CCOC)=O)CC(CC(N2C(C(=O)OC)CC2C)=O)C2(CC2)C1 C(=O)(C(C)N=[N+]=[N-])N1CCC(C(C)C(=O)NC2(C3CCCCC3)CC2)C1 n1(CCC(C)C)cc(C(=O)N(C2CCOC2)C2CC2)nn1 Cc1cc(NC(C2CC(F)CN(Cc3ncccc3F)C2)=O)c(I)cc1F N1(C(C2C(CCC)CCC2)=O)CCN(C(=O)Cc2ccc(Cl)c(F)c2)C(CO)C1 c1(C(=O)NCCC2(OC)CN(C(c3cn(C)c(=O)cn3)=O)C2)cc2scnc2[nH]1 Cc1cc(C(N2CCC(C(C)C(=O)NCCc3cccnc3O)C2)=O)c(N)s1 c1(C(=O)NC2C=CCN(C(C(CC(C)C)O)=O)C2)ccc([N+](=O)[O-])cn1 C1(NC(C=C(CC)CC)=O)CC2CN(C(c3cncnc3C(C)C)=O)CC12 C12(C(N3CC(O)(C(C)NC(c4cc(C(F)(F)F)[nH]n4)=O)C3)=O)CCC(C1)C(C)O2 C(C)(CN=c1nc(N(C)C(c2cccs2)C)c2c(F)cccc2[nH]1)N(CC)CC C(CN=C(NCC1CCN1CC)NCC(c1cccc(Cl)c1)CO)SC N1(C(C(F)=CC)=O)CC2(CC(NC(=O)C(C)C(C)(C)C)C2)C1 c1(NCCn2nc(OC)c([N+](=O)[O-])c2)cc([N+](=O)[O-])n2cccc2c1 c1(OC)ccc(C(=O)N(C)CCNC(=O)COCC(F)F)s1.C12CCC(C1)S2 N1(C(CNC(=O)NC)=O)CCC(C(C)NC(=O)Cc2c[nH]nc2C)C1 C1(C(=O)NCC(C2CCCCC2)NC(c2csnn2)=O)(COC)CCOC1 C1(C(N2CC(C=C)C2)=O)CCCCCN1C(c1ccn(C)c(=O)c1)=O C1(CNC(COCCCCC)=O)CC(O)CN1C(c1cscc1C)=O C1(O)(CNC(C(CC)N(C)C)=O)CCCN(C(=O)CCCN)C1.C(C)(C)SC C(CN=c1cccc(S(=O)(=O)N2CCCC2C(C)C)[nH]1)(N(C)CC)C1CC1 c1(OCC(=O)N(C2CN(C(=O)Cc3scnc3C)C2)CC)cccc(OC)c1 C1(O)(CCNC(C2(CCCC)CCC2)=O)CN(C(=O)CCOCCOC)C1 C(CC1CC1)(C(=O)NCC1(c2cc[nH]n2)CC1)N(C(C1CCCC1O)=O)CCO N1(C(CCC(C)(C)C)=O)CCN(C(=O)Cc2ccccn2)CC(O)C1 N1(C(c2cc(OCC)cc(=O)o2)=O)CC(CNC(=O)C(C)NC=O)C2(CCC2)C1 c1(C(=O)NC2CCC(C)N(c3ccnc(SC(C)(C)C)n3)C2)ccc([N+](=O)[O-])cn1 Cc1cc(C)c(CNC(C2CCCC(CC3CC4(CCO3)CC4)C2)=O)c(O)n1 Nc1ncnc2c1ncn2CCC1CC2CCC12 C1(CC)(CC)CCN(C(=O)C(CCC)NC(=O)C(CO)OC)C1 C(C1CCOC1)=CC(=O)N(CCCNC(C=C(C)C)=O)C c1(NC(N2CCCC2c2nncn2C)=O)ccc(C2CCOC2)cc1F C12(NC(C(C)SCC3CC3(C)CC)=O)CCCC1N(C(C)=O)CCC2 c1(OC)ccccc1NC(=O)CC(N(C1CCSC1)C)C1CC1 CC(CC(=O)NC12COC(CNC(C3(O)CCCC3)=O)(C1)C2)C(F)(F)F C(c1ccc(F)cc1F)=CC(=O)NC1CCCC1NC(C1CN2CCC1CC2)=O c1(C(=O)NCC(CNC(C(C)N(C)C)=O)C(F)(F)F)ccc2c(c1)OCCN2 C(=O)(CC1=CCOCC1)N1CC(CC(C)NC(=O)C=CC2(C)COC2)C1 N1(C(CCC2N(C(C3CCN(C)C3=O)=O)CCCC2)=O)CC2C=CC1CC2 N1(C(c2c(CC)cno2)=O)CCC2(CCN(C(=O)C(C)(C)C3CCOCC3)C2)C1 N1(C(c2c(CC)noc2C)=O)CCN(C(C2CC(F)C(=O)N2)=O)C(C(C)C)C1 N1(CC(=O)NCC#C)CCCC(NC(=O)C(C)OCC(C)C)C1 c1(C(=O)NC(C(C)NC(Cc2c(C)ccnc2)=O)C)ccc(S(N)(=O)=O)c(F)c1 C1(NC(CCC=C)=O)CCN(c2ncccn2)CC1O.c12ccnc(c1)NC2=O c1(COC)cncc(NC(=O)CCN(C(c2ccnnc2C)=O)CC2CC2)c1 C1(CCC(=O)NCCC(CC)C)CN(C(=O)CC2CCC(=O)C2)CC1C C1(C(=O)NC(c2csc(CN3C(=O)CCC3=O)n2)C)CCCN(C2CC2)C1 C1(NC(=O)Cc2cncnc2O)CN(C(c2c[nH]ccc2=O)=O)CCC1O C1(C(=O)NC(c2ccccc2O)C)CN(C(=O)C(O)C2CC2)CCN1C c1(C(=O)OC)c[nH]ccc1=NC(CNC(c1cnns1)=O)C(C)C(C)C c1(C(=O)NCC(CC)NC(c2ccc(C(C)(C)C)[nH]2)=O)ccc(Br)s1 CC1CN(C(c2cnc(O)s2)=O)C(C)CN1C(c1cccc2c1CCO2)=O c1(C(=O)NCC2N(C(C3N(CC)CC3)=O)CCCCC2)cc(C)c(F)cc1N c1(C(N(C)CCN(C)C(C2(Cl)CC2(C)C)=O)=O)c(Cl)cnn1C Cc1cccc(CC(=O)NCC2C=CCN2C(=O)COC2CCCOC2)c1F C(=O)(C(C)C(=O)N1CCC(C(=O)N(C2CCCCCC2)C)(C(C)C)C1)OC N1(C(COC(CC)CC)=O)CCN(C(c2cn(C)c(=O)n2C)=O)C(COC)C1 C1(COC)(CNC(c2ccccc2OC)c2snnc2C)CCOCC1 C1(C(N2C(C(=O)OC)C=CC2)=O)CC1C1CN(C(C2(C(=O)N(C)C)CC2)=O)C1 N1(C(C(C)C)=O)CCC(OCCNC(C2CCC2c2nc[nH]n2)=O)CC1 Cn1cccc1-c1cc(N2CC(O)(C(Cl)(Cl)Cl)C2)n[nH]1 c1(CC(=O)N(c2ccccn2)CCNC(CC2C(C)(C)C2)=O)cc2ccccc2s1 Cc1ccc(SCC(=O)NCC2(F)CCN(C(c3[nH]ncc3C#N)=O)C2)cc1C c1(C(N(C2CCN(C(=O)C(=O)N=S(C)(C)=O)C2)CC)=O)cncc2c[nH]nc12 c1(OC)ccc(C(N2CC(O)(C(C)NC(c3csc(F)c3)=O)C2)=O)c(F)c1F c1(NC(=O)Cc2noc(-c3ccccc3)n2)ncc(Br)cc1I C(C1CCN(C(C2CC23CC3)=O)CC1)=CC(N1C(CN(C)C)CCC1)=O Cn1ncc2c1CC(CCNC(=O)CC1CCCO1)CC2 c1(OC)cc(C)c(C)cc1NC(C1CCN(Cc2cc(C)cnc2F)CC1O)=O C1(CC(N2CC(CC(C)(C)C)C2)=O)CC(F)(F)CN1C(c1ccc(=N)[nH]c1)=O C(N=c1[nH]c2cc(Br)cnc2s1)C1(N2CCOCC2)CCCC1.O=C(C=CCF)NC c1(CNC(=O)NC(C)C(F)(F)F)cnc(Br)c(F)c1 Cc1cc2[nH]c(C(=O)NC3CN(C(c4ccoc4)=O)CC3C3CC3)cc2s1 CC1OC2CCC1(C(=O)NC1CC(CC(=O)NC3CC4(CCC4)C3O)C1)C2 C1(NC(c2cc(OC)c(O)cc2)=O)CCN(C(c2cccnc2S)=O)CC1(C)C C1(NC(=O)NCC(CC)NC(c2cc(C3CC3)nn2C)=O)CCN(C(C)=O)CC1 Cc1cc(C(=O)N(CCNC(C2CC(=O)N(C3CC3)C2)=O)C2CC2)ncc1Cl CC1CN(C(=O)CCC2CCC(=O)N2C)CC1CNC(=O)COc1ccccc1Cl c1(C(=O)NC2C3CN(C(c4cccc(CC)c4F)=O)CC32)cccc2nonc12 CC1(NC(C2CC(NC(=O)CC3CC4(CC4)C3)C2)=O)CCC(O)CC1 c1(C(=O)NC)cc(N)c(OC)cc1F.c12ccc(cn1)NC(CO)CNC2=O C1(NC(c2cnn(C)n2)=O)CCCCCN(C(c2cccc(OCCF)c2)=O)C1 c1(C(=O)NCC2(NC(CCC3CCC(=O)N3)=O)CCOCC2)csc([N+](=O)[O-])c1 C1(NC(CCOCC#C)=O)CCN(C(=O)CNC(C2CCCC2)=O)CC1O C1(CN(C(=O)COC2CCOC2)C)CCCN(C(C2(CCO)CC2)=O)C1 C=CCC(C(=O)NC1CC(OC2CC2)C1)NC(C1(C)CC(C)(C)C1)=O C(CO)(C(C)NC(c1sccc1C1CC1)=O)NC(C1CN(C(=O)NC)C1)=O C(CC(C)C(C)C)NC(=O)CCc1nncs1.C(C=C)OCCSC C1(C(N2CC(OC)C(NC(C3CC3C#N)=O)C2)=O)CC2(C1)CC(O)C2 N12CCC(NC(CC(=O)O)C(=O)O)C(C1)C2=O.Cc1cccc(-c2ccsc2)c1 C#CCCCC(=O)NC1(CNC(=O)CCc2ccncn2)CCC1 N1(C(c2c(C)snn2)=O)CC2CCC(C1)N(C(c1cc(Cl)ccc1F)=O)C2 c1(OC)ccc(C(=O)NC2CCN(C(c3cnc(O)c(C)c3)=O)C(C)C2)nc1N N1(C(C(n2ncc(C)c2)C)=O)CCC(C=CC(N2CCCC(C)C2CO)=O)CC1 Cc1nc[nH]c1CNC(C1CN(C(=O)C(C2CCOCC2)O)C1)=O Cc1cc(Cl)ccc1C1CC1NC(=O)C(N)c1ccsc1 c1(CNC(C(C)Oc2cccc(C(C)=O)c2)=O)cc2ccccc2o1 Cc1ncc(CCCC2(CC(=O)N(C(=O)CC3CC3(C)C)C3CC3)CCCC2)o1 Cc1cccc(OCCC(=O)NCCC(C2CCC2)NC(=O)C(C)(C)C)c1 N1(C(c2cc(CC(C)C)[nH]n2)=O)CC2CC(NC(=O)CCc3ccc[nH]3)C(C2)C1 c1(OC)ccc(CC(=O)N(CC(C)NC(=O)C(C2CCCCC2)O)C)nc1 CC1c2cc(F)ccc2CCN1C(=O)NCc1cc(C2CC2)on1 c1(C(=O)NC(CN(C(=O)C=CCN(C)C)CC)C)cnc(C(C)C)o1 Cc1ccc(CCC(=O)NCC(C2CCC2)NC(=O)C=CCF)c(C)c1 O=S(=O)(c1ccc(=NCC2=NOCC2)[nH]c1)N1CC(C2CC2)C1C1CC1 C(=O)(CC(C)C(F)(F)F)N1C2CN(C(Cc3c(C)nn(C)c3)=O)C(C2)C1 N1(C(=O)CC23COC(CF)(C2)C3)CCCC(O)(CNC(=O)C(F)(F)CO)C1 Cc1cccc(CC(=O)OCC2(CNC(=O)COc3csc(Cl)c3)CCC2)c1 c1(CC(=O)NCC2C=CC(NC(C3(C(F)F)CCCO3)=O)C2)cccc(F)c1F C1(C(N(CCC)OC)=O)CC2CN(C(C3CC4(CC4)CO3)=O)CC2C1 c1(N(C)CC)nc2ccsc2c(=NC(C)c2c(C)n[nH]c2C)[nH]1 C(=O)(NNc1ncccc1C)C1(C(=O)OCC)CNC1 C1(CCNC(COCCCC)=O)C(C)CCCN1C(=O)Cn1nccc1C N1(C(CCC(=C)C)=O)CCC2CCCN(C(c3ccco3)=O)C2C1 c1(C=O)cc(Br)c2[nH]ncc2c1.CC1(C)CC2(CC2CNC(=O)OC(C)(C)C)C1 c1(SC)cccnc1C(=O)NC(CNC(C1CSCCS1)=O)C1CCC1 C1(C(=O)NC2CCC2O)CCCN(C(=O)CCCc2ccccc2Cl)C1 c1(C(=O)NCC(C2CC2)NC(C(C)C2CC2)=O)ccc2c(c1)CN(C)C(=O)N2 C1(C(=O)NCC2(CC)CCCCO2)CCN(C(=O)CN(C)C(C)C)CC1O O=C(C1=COCC1)NCCN(CCOCCO)C(c1cc(C2CCC2)no1)=O C1(NCCOc2cc(C)cc(C)c2)CC(=O)CC12CCC2 C1(C(=O)Nc2cncc(C#N)c2)CC2(CCN(S(=O)(=O)CCBr)CC2)C1 C#Cc1cc(NC(c2nnnn2C(C)C)C2CC23CCC3)cc(Br)c1 C1(CNC(C2CCN(C(C)=O)C2)=O)CCCCN(C(C2(F)CCCC2)=O)C1 C1(C(=O)NC(C)CNC(=O)C(C)(C)CN(C)C)CCc2ncncc2C1 C(=O)(CC(C)C(C)(C)C)NC(C(=O)N(C(CCCC)C)C)CCC c1(C(=O)NCC(C2CC2)NC(C(C)OCCO)=O)cccn1C1CCCC1 CCC(CC(=O)NC(CCNC(=O)CCc1cc(Cl)no1)C(C)C)SC c1(C(=O)NCC(CNC(c2n[nH]c(=N)[nH]2)=O)O)cnc2c(c1)CS(=O)(=O)CC2 NCCS(=O)(=NC(=O)CNC1(c2ccccc2Cl)CCCC1)c1ccccc1 C(=O)(CC(O)CC(C)(C)C)N1CCN(C(c2cncc(SC)c2)=O)C(C2CC2)C1 N1(C(C(COC)OC)=O)CCC2(CC1)OC1(CO)CC2(NC(C2CCSC2)=O)C1 C(N=c1[nH]c(=NCCC(F)(F)F)c2ncccc2[nH]1)c1ncc(C)o1 N1(C(c2nc(C)sc2)=O)CC(O)CC1C(N1CCCC(N(C)C)C1)=O C(=O)(CCC(C)(C)NC(C1CN2CCC1CC2)=O)NC(CCOCC)C c1(C=O)ccc(F)nc1F.N12CC(C(C)(C)C1)N2C.C1(C(F)(F)F)(C=O)CCC1 c1(NC(CC2(OC)CN(C3CC3)C2)=O)ccc(I)nn1 C1(NC(CCSCCOC)=O)CC(CC(=O)N(C2CC(C)(C)C2)C)C1(C)C N1(C(C2(COC)CC2)=O)CCOC2(C1)CN(C(c1ccc(=O)n(O)c1)=O)C2 C#CC1(C)CCN(C(C2CC(OC)CN2C(=O)CSC(F)F)=O)CC1 N1(CS(CC)(=O)=O)CCC(CN=C(NCc2cc(C)on2)NC(C)COC)CC1 N1(C(c2c(C=C)cccc2)=O)CC(C2CCCN(Cc3cccc(F)c3I)C2)C1 N1(C(Cc2cccc(C)c2)=O)C2CCC1CC(CNC(=O)C(C)C(F)(F)F)C2 N1(C(CCS(CC)=O)=O)CCC(CC)(Cc2cccnc2Cl)C1 c1(C(=O)NC(C(=O)NC(CC)CN2CCCC2)CC)cn(C)c(=O)n1C c1(C(N(C2CN(C(C3OCCN(C)C3)=O)C2)C)=O)ccc2[nH]ccc2n1 Cc1cc(C(N2CCC(O)(C(C)CNC(=O)COCC(C)(C)C)C2)=O)cn1C N1(C(CSc2ccc(C)c(C)c2)=O)C2CCC1CN(C(=O)CC1(C)CC1F)C2 C1(CCC)CN(C(C2CCC(F)(F)C2)=O)CCN1C(=O)CN(C)C(C)C N1(C(C(CC(C)C)NC(C=C(C)C(C)(C)C)=O)=O)CCC(F)(F)C(O)C1 Cc1ccc(OCC(=O)NCC2CCC(NC(C34CCC3C4)=O)CC2)cc1 CC(C)C(C)(C(N)=O)NC(=O)C1=NOC(CNC(c2cccn2C2CC2)=O)C1 Cc1ncc(SCC(F)F)c(NC(=O)NCc2cccc(C)n2)n1 c1(COC)ccc(CN2CCC(O)(C(=O)NCc3cncnc3)C2)cc1 Cc1cn2ccnc(C(=O)N(C(C)CNC(c3cccn3C)=O)C)c2n1 C12(CNC(=O)OC(C)(C)C)CCC(CC1)N2C(c1cc2c(s1)CSC2)=O c12cc3ccc1cc3[nH]2.N1(C(c2cnc(C)c(Cl)c2)=O)CCN2CCOCC2C1 C1(C(=O)NCCC(=O)N(C(c2cccnc2)C)C)CCC=CCCC1 c1(C(=O)NCCOCCN(C(=O)C#CC2CC2)C)cc(Cl)nc(Cl)c1 c1(CNC2C(C(=O)NCc3cnccn3)CCC2)c(O)cc(Br)cc1F C1(NC(C(C)(C)C2CCOC2)=O)CCOC(C(=O)NCC2CC(=O)N(C)C2)C1 c1(CNC(C=C2CCN(C(C3(C#N)CCCO3)=O)CC2)=O)cc2cccnc2o1 C1(CNC(C2CC2Cl)=O)CN(C(C2C3CCC2(c2ccco2)C3)=O)CCO1 c1(SCCNC(C)(C)C)ccc(N2CCC(N)CC2)cc1 C1(C(=O)NCC2(F)CCN(C(CCNC(=O)NC)=O)CC2)CCC2(CCC2)CO1 S(=O)(=O)(c1cc2sc(=NC3COC(CCOC)C3)[nH]c2cc1Cl)NCCCC c1(C(=O)OC)ccccc1CN1CCCC1.C1(C)(C2CC2)CNC(=O)C(=O)N1 Cc1ccnnc1C(N1CCCC(C(=O)NC(c2noc(C(C)(C)C)n2)C)C1)=O c1(C(=O)NC2CC(C)(CNC(CC(C(C)C)C)=O)C2)cc(F)c2ncccc2c1 c1(C(N2C(C)CC(NC(c3c[nH]c(=O)cn3)=O)C2)=O)cc2ccc(O)cc2n1C N1(C(C(C(C)C)NS(N)(=O)=O)=O)CC2(C1)CN(C)C(=O)CO2 C1(C(N2CCC(N(C)C)C2)=O)CN(C(c2ccncc2)=O)CC(C)(C)C1 N1(C(COC)=O)CC2CC(NC(C3CC(=O)N(C)C3c3ccccc3)=O)CC2C1 O=C(C1=CCCC1)NCC(N1CCC(N2CCOC2=O)CC1)=O C#CCCCC(=O)N(CC(C)NC(=O)Cc1cncc(Br)c1)CC c1(C(=O)NC(COC)C)csc2c1CCN(C(c1ccncc1F)=O)C2 c1(C(N2CCC(C3N(C(C(C)OCCCC)=O)CCC3)C2)=O)cccnc1O C=CC(C)CC(=O)N1C(C(=O)N(C2CCN(C)C2)C)CCC1C1CC1 C1(NC(C(CC)N(C(CC=CCC)=O)CCOC)=O)CCCC(C)C1C C1(N=[N+]=[N-])(C(=O)NCC2CCCN(C)C2)CCN(C(=O)C(O)Cn2cncn2)C1 C1(NC(CCCCSC)=O)CC12CCC(NC(=O)CCc1nnc(C)n1C)CC2 C(CCC(C)C(=O)N1CCC(OCCNC(=O)C(C(C)(C)C)N(C)C)C1)OC C(=O)(CC(C)F)N(C(C)C(=O)N(C1CC1C1CC1)C)CC C1(CC)CC(C(=O)NCC(C2CCCC2)NC(=O)CCC2CCCCC2)CCO1 N1(C(C)=O)CCCC(C(CC(=O)N(C2CCC(NS(=O)(=O)C3CC3)CC2)C)=O)C1 CC(C)C(C(=O)OCc1noc(-c2ccccc2)n1)Sc1ccccc1 c1(SCC#C)cccc(C(=O)NCC2CC(O)(CNC(=O)CC3CC3)C2)c1 N1(C(c2c(OC)nsc2)=O)CC(O)CC1CNC(=O)CC1CC12CC2 c1(CN2C(CCC(=O)NCc3ccsc3)CCC2)ccc2ccoc2c1 C1(NC(C2(SC)CC2)=O)COCCC1NC(c1ccnc(-c2ccccn2)n1)=O c1(C(=O)NCCCC(C)NC(C(C)n2cncn2)=O)c(C(F)(F)F)cccc1O C(=O)(C(C)(C)CCCF)N(C)CCNC(=O)CCc1cccnc1F C(=O)(C(O)CC(C)(C)C)NCC1CC(C(N(c2cnn(C)c2C)CC)=O)C1 c1(C(=O)NC2(CNC(C3C(C)(CC)C3)=O)CCOCC2)cc2n(n1)CCCCO2 c1(OC)ccc(C(=O)NCC(C)(C)NC(c2ccc(C)nc2)=O)c(C)n1 C1(C(N2CCC(OCC(=O)N(C)CC3CC(O)C3)C2)=O)CC(N=[N+]=[N-])C1 C=CC(C)(O)C(=O)NCC=CCNC(c1cnc(-c2ccoc2)s1)=O C1(CNC(C(c2ccc(Cl)cc2)(C)O)=O)CN(C(c2ccoc2)=O)CCC1(F)F C(=O)(C(C)(C)CCS(C)(=O)=O)NC(C)C(CO)NC(c1cc(N)c(F)cn1)=O C1(C(=O)NCC2CCN(c3c(C)cc(C#N)cn3)C2)C2Cc3c(Cl)cccc3C12 C(=O)(C1=NNC(=O)C1)NCCC(C)CCNC(C1(c2cccs2)CCCCC1)=O C1(C(c2nnnn2C)NCCCC(CO)O)CC2(C1)CC1CCC2C1.C1(CC)CC1 C1(C(=O)NCC2(C)CCN(C(C3C(C)(C)C3(F)F)=O)C2)CC2C(C1)C2(F)F C1(N(C(=O)CO)C)CCCC(CNC(=O)CC(C2CC2)C2CC2)C1 N#Cc1cc(C(N2CC(O)CC2C(=O)Nc2c(F)cc(Br)cc2Cl)=O)ccc1O C1(C(=O)NCCOC)CC(C(=O)Nc2sccc2C(=O)OC)CCO1 N1(C(C(CC=C)CNC(C2(CC)CCCC2)=O)=O)CCC2(CCCCC2)C1 CN1C(=O)c2ccc(C(N3CCCc4ccc(F)cc43)=O)cc2S1(=O)=O N1(C(C(C)OCC)=O)CCCC(C)C1CNC(c1ccc(N)cc1F)=O c1(C(C(=O)NC2CN(C(C(CSC)(C)C)=O)CC2O)C)cccc2ccccc12 N1(C(C(C(=O)OC)C)=O)CCCN(C(c2ccc3ncnn3c2)=O)CCC1 C1(C(=O)NC2(CNC(C(CCC)N(C)C)=O)CCC2)CCCCC1C1CC1 c1(OC)nc(C)ccc1C(=O)NC(CNC(=O)C#CC(C)(C)O)C(C)(C)C CN=c1[nH]c(=NCCc2cnc3n2CCCC3)[nH]c(=NC2CCOC2)[nH]1 c1(C(N2C(CNC(C3(O)CCC3)=O)CC(C)(C)C2)=O)nsc2c(Cl)cccc12 C1(CNC(c2cnc(SC)s2)=O)CC(C)(C)CN1C(=O)Cc1cnc(C)s1 C1(C(CNC=O)NC(C(C)OCCC=C)=O)CCCCN1C(=O)OC CN1CCc2nc(C(=O)NC3CCCC(N(C(=O)Cn4ncnn4)C)C3)sc2C1 N1(C(CSc2cn(C)nc2)=O)CCC(C)(NC(=O)C(F)C(C)(C)O)CC1 c1(OC)c(SCC2CCC(C)CCC2)cccc1Cl Cc1cc(F)c(Cl)cc1C(=O)NC1CCCC(NC(C2(n3cccn3)CC2)=O)C1 C(=O)(CCCCCF)NC(CCCC)CNC(=O)C(c1ccccc1)C1CCCC1 c1(C(N2CC(OC)(CNC(C3CC34CCC4)=O)C2)=O)ccc(=O)n(C(C)C)c1 N1(C(c2c(CC)ncs2)=O)CCC2(CC(NC(C3(O)CCCCCC3)=O)CO2)C1 c1(NC(c2cnsc2)=O)cc2c(=O)cc[nH]c2s1.c12cn(nn1)C1CN(C1)C2=O c1(C(=O)NC(CCC)Cc2ccccc2)cccc(Cl)c1SC CC1CN(C(=O)CSC2CCC(F)(F)CC2)CCCN1C(=O)Cc1cn(C)cn1 C12(C(=O)NCCN(C(C3CN4CCC3CC4)=O)CC)CC3CC(C1)CC(O)(C3)C2 CCC(C)CCC(=O)N(C1CN(C(=O)C2=CSCS2)CC12CC2)C C1(NC(CC(=O)N(C)C)=O)CN(C(=O)CCC(F)(F)F)CCC12CCOCC2 c1(C(C)CC(=O)NCC2(C(F)(F)F)CCC(=O)N2)ccc2c(c1)OCO2 c1(C(=O)NCC2N(C(C3C(CC)CCC3)=O)CC(C)(C)C2)cc2ccncc2o1 C(=O)(C(CCC)N(C)C)NC1(CNC(CCC=CC=C)=O)CCOC1 C#CCCCCCC(=O)N1CC2C(CNC(c3cc(S(C)(=O)=O)co3)=O)C2C1 c1(C(=O)NC(CNC(c2csc(F)c2)=O)C2CC2)cnn2c1CCC2 Cc1c(C(N2CCCCC2CNC(C2CC3CCC2O3)=O)=O)cnn1CCC#N N1(C(C(=O)NC(c2cccc(OC)c2)CF)C)CCOc2ccccc21 C1(N(C(C)C)C)CCN(C(C)CNC(=O)CN(C2CCCC2)C(C)C)CC1 c1(C(=O)OCC)sccc1S(=O)(=O)N1CCCCC1C(CO)CO Cc1cc(NC(C2CC2F)=O)ccc1NC(c1nn(C)c(Cl)c1Cl)=O N1(C(=O)NC(C)(C)C)CCC2(CCCC2NCCCc2ccc(OC)nn2)C1 C(C)(C)(CC(=O)NCCC(C)CCNC(=O)CCc1csc(C)n1)SC c1(C(C)NCc2cn(-c3c(F)cc(F)cc3Cl)nn2)cc(Cl)cc([N+](=O)[O-])c1 c1(C(C(=O)NCC2C(CNC(C(C)O)=O)C2)(C)C)ccc(Cl)cc1F C1(C(N(C)CCC2CCCCN2C(=O)CCc2cnn[nH]2)=O)OCC2CCCC12 O=S(=O)(N1CCC(OCCCO)CC1)N1CCc2cc(Br)ccc2C1 c1(C(N2CC(N(C(c3ccc(CN(C)C)[nH]3)=O)C)C2)=O)cc([N+](=O)[O-])sn1 c1(C(N(C2CN(C(=O)CC3CC(C)(C)C3)CC2(C)C)C)=O)ccn2c1CSCC2 CN1CCC(N)(C(=O)NCC2CCCC2C(F)(F)F)C1 N1(C(c2cnnc(Cl)c2)=O)CCC2(CCCC2CNc2nccc(CO)n2)CC1 c1(OC)ccc([N+](=O)[O-])c(N2CCCC2c2ccc(F)cn2)n1.C1(CC)CC1 Cc1ccc(C(=O)NCC2CCCN2C(C2CCCN2C)=O)nc1C C1(N)(C(=O)NCC(Cn2cc(C(C3CC3)OC)nn2)(F)F)CCCS(=O)(=O)C1 C(C(=O)NCC1CCCN1C(=O)C(C1CCOCC1)O)(C(C)C)OCC(C)C CC(CCC1CCCC1)C(=O)N1CCCC(Cc2cn(C3CC4CC4C3)nn2)C1 Cc1cc(C(=O)NCC(C(C)(C)C)NC(=O)CCc2nncs2)c(C)o1 C1(NC(c2cc(CC)ncc2)=O)CN(C(=O)C(C)(O)CC)CC1N=[N+]=[N-] C(CCC(=O)NC(=O)NCC(O)Cc1cccnc1)N(C(=O)OCC)C C1(C(=O)NCC(CNC(C2(C(=O)OC)CC2)=O)O)CCCCC12CCC2 C(CCCCC(=O)NCC(C)C(F)F)NC(C(CC)(C)C)=O Cc1cc(-c2csc(C3CCCN3c3ncc(C)c(C)n3)n2)ccc1Br c1(OCC)cccc2c1CCC2NCCCCCC1CC1 C1(NC(COC(CC)C)=O)C2CN(C(c3ccc(-n4cccn4)nc3)=O)CC12 C(=O)(C1=CCCOC1)NC(C(C)(C)NC(c1cnc(C(C)=O)s1)=O)C Cc1cc(N2CCCC2CS(N)(=O)=O)nnc1C Nc1ccc(C(=O)NC2CCCC2NC(=O)CC2CC(=O)C2)cc1C(F)(F)F c1(C(=O)NCCC2(OC)CN(C(C3C4C5CCC(C5)C34)=O)C2)cnn2c1OCC2 c1(C(=O)NCC(C)N(C(c2c(COC)nn(C)c2)=O)CC)nc(OC)ccc1Cl c1(C(N2C(CCNC(C3C(CC)C3)=O)CSCC2)=O)ccc2n[nH]cc2c1 N1(C(C(CCC)NC(=O)CC2(O)CCCCC2)=O)C2C=CCC1CCC2 C1(C(N2C(CNC(C3N(S(C)(=O)=O)CCC3)=O)CCC2)=O)COC2(CCC2)CO1 Cc1ccc(NC(C2C3CC3CN2C(=O)CC2(O)CCCC2)=O)cc1Cl N1(C(Cc2ccn(C(C)C)n2)=O)CCC(C2CC2)C1C(=O)NOC1CCC1 C(C(C(C)C)NC(c1cc(F)c[nH]1)=O)NC(C(C)OCCOC)=O c1(NC(C(C)NC(C(CC)CC)=O)=O)nc(C)ccc1O C(=O)(CC(F)(F)F)N(CCCNC(COCC)=O)CC C1(NC(C2CCC2)=O)CC(=O)N(C)C1.c1(CC(=O)NC2(C)CC2)ccccc1 C1(C2CCOCC2)(C(N2CC(NC(Cc3cnc(C)o3)=O)C2)=O)CC1(F)F c1(C(N2CCN(C3CCC3)CC2)C(=O)NCC(=C)C)ccc(C(F)F)cc1F c1(N(C)C)ccc(CNc2cc(C(=O)NCC(O)C(F)(F)F)n(C)c2)cn1 N1(C(C2ON=C(C)C2)=O)CCCC(OCCN)C1 CC1C(NC(=O)C=C2CCC(C)CC2)C(C)CCN1C(=O)Cc1cscn1 C1(NC(=O)C=CC=C(Cl)Cl)CC2CC(C1)N(C(c1cc(C3CCCC3)no1)=O)C2 C=C(C)CC(C(=O)NCC1COCCN1C)NC(=O)COc1cc(C)on1 c1(CC(=O)NC2CN(C(CC3(C#N)CC3)=O)CC(F)C2)cn2ccccc2n1 C1(NC(Cc2c(C)nsc2)=O)CCCC(C(=O)N(CCCCN(C)C)C)CC1 C(C)(CCC(=O)NC(c1cnn(C)c1)C(=O)NCCC1CC(O)C1)OC C1(NC(C2(C)COC2)=O)CN(C(c2nncn2C2CC2)=O)CC1C(F)(F)F C1(C(N2CCC(CN(C(CN(S(CC)(=O)=O)C)=O)C)C2)=O)CC2CCC1O2 N1(C(=O)CCc2ccc(F)cc2)CC2CC(C1)CN(C(=O)C(F)(F)C(F)(F)F)C2 C(=O)(C1=C(C)OCCC1)NC(CCOC)CNC(c1n[nH]c(C)c1C)=O c1(OC)csc(C(=O)NCC2CN(C(C3CC(C)=NO3)=O)CCO2)c1OC c1(C(=O)NC2CCN(C(c3c(OCC)ccs3)=O)C2(C)C)n[nH]c2c1CC1CC21 c1(OC(C)C)ncccc1C(N1CCCCC1C(=O)N(CCO)C1CC1)=O N1CCC2(N)CCCC12.C(=O)(C1=CCCCCC1)C(c1scc(C)c1)=O C1(NC(=O)NC)CCC(OC2CCOC2C)CC1 C(C)(C)(CC(C)(C)C)NC(C(C1CN(C(C)=O)C1)F)=O.N12CCC(C=CC1=O)CC2 C1(NC(C(=O)NCc2n(CC)ccc2)=O)C2CCOC2C1(C)C C(N=c1[nH]c(N2CCCC(C3(C)CC3)C2)nc2c1CCC2)C1CCN(C)CC1 c1(C(N2CC(O)CC(NC(c3cnc(OC)s3)=O)C2)=O)ncnc2c1CCC2 C(=O)(C1=NNC(=O)C1)N(C1(c2cccnc2)CC1)C.C12(CO)CN(C1)C2=O C(=O)(C(F)CCCC)N1CC(COCC(=O)NC2CCOC2)C(C(F)(F)F)C1 c1(C(=O)NCCCN(C(=O)CCn2cncn2)C(C)C)cc2n(n1)C(C)CCC2 N1(C(C2C(=C)CC2)=O)CC(NC(C2(C#N)CC=CC2)=O)CCC1C C(=O)(C(C(C)c1ccccc1)N1CCC1)NCCCOC.C1(C)C(=O)N1C N1(C(C(COC)C)=O)CCC(C)(C)C(CNC(c2csc(C)n2)=O)C1 C1(C)(C(N(CC)Cc2nccn2C)=O)CCCN(C(=O)C(=O)NCC(F)(F)F)C1 CC(CCCCNC(=O)CCNC=O)NC(c1cn(Cc2cccnc2)nn1)=O CC1CN(C(=O)C(CNC(C2CC(C3CC3)=NO2)=O)CC2CCCC2)CCN1C CC1C(O)CCCN1C(=O)CCC(C)(C)NC(=O)C=Cc1cccnc1 c1(C2C(C(N(C3CN(C(C4CN(C(C)C)C4)=O)C3)C)=O)C2)ccc(C#N)cc1 CCCC(CC)CCC(=O)NCC(CC(=O)N(C1CCSC1)C)OC Cc1noc(C)c1C(C)C(=O)NC(CNC(c1cncc(N)c1)=O)CO c1(C(N2CC(O)(C(C)NC(=O)C=CC3CCCO3)C2)=O)cc2cnn(C)c2s1 c1(-n2ncc(CNCc3cc(SC)nn3C3CCCC3)c2)ccc([N+](=O)[O-])cc1 c1(C(=O)NC(C)CNC(=O)C(C)SC(F)(F)F)ccc(C(F)(F)F)s1 CCCC(CC)C(=O)N1CCCCCC1CNC(c1ncc(C(F)F)s1)=O CCCCCCCN(C)C(C1CC(C)N1C(=O)C(C)C(=O)OCC)=O C=CCCC(C(=O)NC(c1cnc[nH]1)C)NC(=O)CCCCC N1(C(C(CC)COC)=O)CCCC(O)(CCNC(=O)Cn2ccccc2=O)C1 c1(O)cc(N)ccc1F.C1(C(N(C(C)C)C)=O)CCC(C(=O)O)C1 C1(C(=O)OCC)CCN(C(=NCC(C)(C)C2CCCCC2)NCC2CC2)CC1 c1(C(C)NC(=O)N(C)CC2CC(C)(C)C2)nc2c([nH]1)CCCC2 C1(CNC(Cn2c(C)cc(C)n2)=O)CN(C(=O)C(C)C(C)(C)C)C2(CCC2)C1 n12ccc3nc(ncc13)N1CC(C(C)C1)C2.c1(SCC)cc(Cl)cnc1Cl C1(N(C(C2(CC=C)CCCN2C(c2cc(C#N)cs2)=O)=O)C)CC(C)CC(C)C1 N1(C(C(CCC)C#N)=O)CCC2CCN(C(c3oc(C)nc3C)=O)CC12 c1(OC)cc(Br)c(C(N2CCOC(c3noc(C(C)C)n3)C2)=O)cc1OC c1(-c2n(CCC(C)C)ncc2)cccc(NC(=O)NC(C)CCCCO)c1 c1(C(C(=O)NCCN(C(c2cc(OC)no2)=O)CC)C)cccc(S(C)(=O)=O)c1 N1(C(CSSC)=O)CC(NC(=O)CCCc2nncn2C)C(C)(C)C1 c1(C(=O)NC(CC2CC2)C(=O)N(C2CCOC2=O)C2CC2)ncncc1Cl C(C1CCCCC1)=C(C(=O)NC(CN(C(c1c(OC)nsc1)=O)C)C)F C1(C)(C(N(C2CCCC2)CCNC(CCCOCC=C)=O)=O)CC2C=CC1C2 CC(C)C(CNC(=O)CC1OCCO1)NC(=O)CC(C)C1CCCO1 N1(C(c2cc(C#C)c(C)cc2)=O)CCC(NC(=O)C(CC)OC)CC(C)(C)C1 c1(CC)cc(C)c(C(=O)NC2CC=CCC2C(=O)NOCC2CCCC2)o1 N1(C(=O)NC2CCN(C(=O)NC)C2)CCN(c2cc(F)ncn2)CC1 N1(C(C(C)CC(F)F)=O)CCC(C2CCOCC2)(CNC(C2(F)CCC2)=O)C1 C(N=c1[nH]c2c(c(=NCc3nnc4n3CCCCC4)[nH]1)SCC2)c1cnc[nH]1 C1(C(=O)NCC2(CNC(C(C)(C(C)C)OCC)=O)CC2)CC(C)CC(C)(C)C1 C1(O)(CNC(C(c2c(C)nn(C)c2)C)=O)CCN(C(c2ccn(C)c2C)=O)CC1 CC1(C)OC2(C(N3CC=CC3CNC(C3(c4ncco4)CC3)=O)=O)CCC1CC2 C1(OC)CC2C1CCN2C(=O)C(CCSC)NC(=O)C=C=C(C)C N1(C(C(C(C)C)C)=O)CC2(CO)CC1(C(=O)NCc1ncc(CO)[nH]1)C2 N1(C(C(CC(=C)C)C)=O)CCC2(NC(=O)CC(C)C(F)F)CCCC12 Cc1nnc(OC(F)F)c(NC(=O)Nc2cc(Br)ccc2N(C)C)c1C C(CC(F)F)(C(=O)NCc1cc(NC(N)=O)n[nH]1)N(C(=O)CC1(C)CCOCC1)C Cc1cnc(F)cc1-c1nc(CC2CCC2)nn1C1CCN(CC(F)(F)F)CC1 N1(Cc2cc(C)ncn2)CCCN(C(=O)Cc2nocc2C)CC1 N1(C(CC(=O)OCC)=O)CC(N(C)C(C2CC=CCN2C)=O)C2(CC2)C1 C1(CC)CN(C(C2(C#N)CCCO2)=O)CC1NC(=O)COCc1cccnc1 CC1CC(NC(=O)C=CCl)CN1N(c1cccnc1)C(=O)CNc1ccnc(O)c1 N1(C(C(C2CCCO2)NC(c2cc(C)sn2)=O)=O)CCC(CCF)CC1 N1(C(C(c2cccc(Br)c2)C)=O)CCC2(CC1)OCCC2NC(C1CC1C)=O CC(C(=O)NCC(CC(F)(F)F)NC(=O)Cc1cc(C2CC2)no1)C(C)(C)C c1(-c2cn(CC(CCNC(C3CN(C)CC(C)O3)=O)(F)F)nn2)cc2cccnn2c1 C1(NC(C2CCCCC2)=O)CC2CCCC(C1)N2C(=O)CCC(F)F C=CCCCCC(=O)NCCCNC(C1OCC2CCCC12)=O c1(C(=O)NCC(CC)NC(=O)C(F)(F)C2CC2)ccccc1-c1nc[nH]n1 C(C)(C(C(=O)NCCCCN(C(=O)CCCN(C)C)C)N(C)C)OC n1(C(C)C)ncc2c(N3CCC(F)C3)[nH]c(=NCC3CCc4nccn43)nc12 N1(C(C(CC(C)C)(F)F)=O)CCC(NC(c2n[nH]cc2C(C)C)=O)CC(C)(C)C1 C(=O)(C1=C(C)OCC1)NCC1(NC(c2cc(COC)[nH]n2)=O)CCCCC1 N1(C(Cc2ccc(C#C)cc2)=O)CCC(C)C(NC(=O)C=CCOC)C1C c1(C(N(CC(C)NC(=O)CC2CCC23CCC3)CC)=O)ccc(S(C)(=O)=O)s1 C(=O)(CC1=NN(C)C(=O)C1)NC(CC(=O)NC(CC)C(C)CN(C)C)C1CC1 Cc1cc(C)cc(N=c2scc(-c3cnnn3C)n2Cc2c(Br)nnn2C)c1 N12CCN(CC1)c1cc(n[nH]1)C2.c1(N(C)C2CC2)ncsc1C(c1cccnc1)C1CC1 C1(NC(C(C)(Cl)Cl)=O)CC2CCC1N(C(=O)C=Cc1cnccn1)C2 C1(=O)CC(C)CC(=O)C2CC3C(COC)N1C2C3C(=O)OC.OC C1(C)(C(=O)OCc2cc(C)ncn2)CCCS1(=O)=O N1(Cc2ccc(COC)s2)C(=O)CCN(CCN2CCNCC2)C1=O c1(CNC(C2CCN(C(c3c(COC)cc[nH]3)=O)C2)=O)cc(F)ccc1F c1(C(=O)NCC(CNC(=O)Cc2ccc(F)c(C3CC3)c2)F)csc2ccncc12 N1(C(Cn2ncc(C)cc2=O)=O)CC2CCC(C1)N2C(=O)Cn1cnnc1O C1(CNC(C(C)SC(C)C)=O)CN(C(c2ccncc2N)=O)CCC12CCOC2 C1(CNC(CC2CCC(=O)C2)=O)CCCN(C(=O)CSc2ccncc2)C1 CCC(C(=O)NCC1CCC(CNC(=O)C(Cl)=CCl)CC1)C(F)(F)F c1(COC(c2c(NCC3NCC(C)(C)OC3)cccc2)=O)ncnc2sccc12 CC1CCN(C(c2ccccc2NCC(F)(F)F)=O)CCN1C(C1CC=CC1)=O c1(C(N2CCCCC(N(C)C)C2)C(=O)NCC=C)cc(Cl)cc2cccnc12 c1(C(N(CCCCNC(=O)CC(=O)NC2CC2)C)=O)c(F)cc(F)cc1F N1(C(CNC(=O)NC)=O)CC(O)C(O)C1CNC(=O)CC1CC2CCC1O2 C12(NC(CS(=O)(=O)NC)=O)CCCC1N(c1ccnc(S(C)(=O)=O)n1)CCC2 c1(-n2cc(C(CC(=O)O)Sc3ccc(Cl)cc3)nn2)ccc(Cl)c(Br)n1 c1(C(N2CCC(N(C(C3CC(C#N)C3)=O)CC)C2)=O)cc(F)c(F)c(F)c1F C1(CNC(C(=O)N(C)C)=O)CC(C)(C)CCC1NC(=O)CC1CCCC1(F)F c1(C2N(C(C(=O)NCC3CC34CCOC4)=O)CCC2)nnc2n1CCOC2 O=C(C1=CC2C=CC1C2)NC(CC1CCCC1)C(=O)NCC(c1ccsc1)O O=S(=O)(c1ccc(NCc2csc(C(F)F)n2)cc1Br)NCCc1ccoc1 C(=O)(C(C)(CO)ONC(=O)CN(CCCO)C(=O)C=Cc1cn(C)cn1)OC c1(C(N2CC(CNC(=O)COC(F)F)CC(C)(C)C2)=O)ccc2n[nH]cc2c1Cl C(CCC(COC)C(N)=O)n1cc(CCC(C=C)C)nn1 C1(NC(c2ccc(C3(C(=O)OC)CC3)[nH]2)=O)CC2CN(C(=O)Cc3cnc[nH]3)CC12 CCC(CC(=O)NCCC(O)C(=O)N(C1CCOC1)CC)C(F)F c1(C(=O)NC(CNC(c2cnc(CC)s2)=O)CC(C)C)ccc(S(=O)(=O)NC)o1 n1(CC)nc(C(N2CCC2CC(=O)NCc2cc(Cl)ccn2)=O)cc1O C1(CN(C(CC2(OCC)CCC2)=O)C)CCCN1C(=O)C(O)CSC C1(C(N2CC=CC(NC(c3c(C)cc(CC)o3)=O)C2)=O)CCc2n[nH]cc2C1 N1(C(C(CCC)NC(N)=O)=O)CC2CN(C(=O)CP(C)(C)=O)CC2(C)C1 N(C(=NCCC1CCCO1)NC(C)CNC1(COC)CC1)C(CC)C C1(C)(C(N2CC(C)C(NC(c3cc(Cl)no3)=O)C2)=O)CCN(C)C1=O N1(C(CCOCC(C)(C)C)=O)CCC(CO)CC1(C)C C=CCN=C(NCc1cc(Cl)ccc1OC)NCC(F)(F)C1CCC1 C(C)(C)(C(=O)NCc1cn(CC2CCCN2C(=O)CC(=O)NC(C)C)nn1)SC N1(C(c2c(C(C)C)c(F)ccc2)=O)CCN(C(=O)C=CC(C)(C)C)CC12CC2 C1(C(F)(F)F)(C(=O)NCC(C)NC(C2(C#N)CCOC2)=O)OC2CCC1CC2 c1(C(=O)NC2CCC(C)(NC(=O)Cn3ncnn3)CC2)cnn2cccc(Cl)c12 C(=O)(CC1=Cc2ccccc2C1)NC1C(NC(Cc2cc(COC)on2)=O)CC1 C(=O)(CCC(=O)N1CCN(C2CCN(C(=O)C(C)O)CC2)CC1)NCCC CC1CC(c2ccccc2)(C(=O)NC2CC(CCNC(=O)CC3CCCO3)C2)C1 c1(C(=O)NCC(CO)NC(CCCCC(N)=O)=O)cnc2ncnn2c1O C1(C(=O)NCC2CCN(C(CC(=O)OC(C)(C)C)=O)C2)CS(=O)(=O)CC12CCC2 c1(C(N(CC(CC)NC(C2CCC2CF)=O)CC)=O)csc(-c2ccc(C)o2)n1 c1(CCN2CC(=O)N(c3cc(F)c(I)c(F)c3)CC2)nc(Cl)cc2ccccc12 C1(NC(C2CS(=O)(=O)C2)=O)CCN(C(=O)CC(F)(F)Cl)C1C1CC1 C12(C(=O)NCC3C(NC(c4ccc(CC(C)C)s4)=O)C3)CC3CC(C1)CC(C)(C3)C2 N1(C(C(Cc2c(C)nn(C)c2C)C)=O)CCC(C2CCN(C(=O)CC3CC3)C2)CC1 C(=O)(C1=COCCC1)NC(C(N1C(CC)CCOCC1)=O)(C)C1CCC1 CCCC(C#N)C(=O)NC1(C(N2CC(=O)NC(C)C2)=O)CCCC1 C#Cc1ccc(F)c(C(N2CC3CCC2C(NC(C2CC2F)=O)C3)=O)c1 N1(C(C(c2ccc(Cl)c(F)c2)NC)=O)CCC(O)CC12CCCC2 C(=O)(C(C)C(C)(F)F)NC1CCC(CNC(CCCOCC=C)=O)C1 C1(N=[N+]=[N-])(C(N(CCCc2ccco2)C)=O)CCN(C(C2CC(=O)NC(=O)C2)=O)C1 c1(C(=O)NCCc2ccsc2Br)nocc1-n1cc(C2CC23CC3)nn1 N1(C(CCN(C(C(CC(=C)C)OC)=O)C)=O)CC=CCC(C)(C)C1 c1(C(N2CC(CN)OCC2)=O)cc(F)cc(C(F)(F)F)c1N CC1CCC(NC(=O)C(C)(C)OCC(F)(F)F)CN1C(c1ccc(=O)n(C)n1)=O C1(NC(C(C2CN(C(=O)CC3CC(O)C3(C)C)C2)OC)=O)CC2CCCC2C1 c1(NC(CCC=C)C)ccc(S(=O)(=O)N2CCCC(N(C)C)C2)cc1C#N N1(C(C2CC(CC)N(C(=O)CSCCC#N)CC2)=O)CCN2CCCC2C1 N1(C(C2N(CCC)CCC2)=O)CC2C(C(=O)NC3(CC)CCCC3)C2C1 N1(C(CCC(C)C)=O)CCCC12CCCN(C(=O)Cc1ccccc1S(C)=O)C2 Cn1ccc(C(=O)NC2CC(O)(C(=O)NC3CC3)C2)n1.C12(CCC1)C(=O)NC2 c1(C(N(C(C(=O)NCCC2CCC2)C2CCOC2)C)=O)cc2ncccc2[nH]1 C1(C)(NC(C2CC(SC)C2)=O)CCCN(C(=O)CCc2ncccn2)C1 c1(CC(=O)NCC(CN(C(c2c(C)noc2N)=O)C)C)cccc(Cl)c1Cl c1(COC)nc2n(n1)CC(N1CCC3(CCCNC3)C1)CC2 C(=O)(C1CCCc2cncn21)NC(CN(C(CCCC#CC)=O)C)C Cc1cn2c(n1)CC(C(N1CCC(CNC(c3cnc4[nH]ncc4c3)=O)C1)=O)C2 C1(N(C)C)(NC(=O)NCC2(C(C)(F)F)CC2)Cc2ccccc2C1 N(C(=NCCSCC1COC1)NC(C1CCCC1)C)CC.c1ccccc1 Cc1cc(=Nc2nc3c(s2)CSC3)[nH]n1-c1ccc2cccc(Br)c2n1 c1(C(N2C(CC)CN(C(c3ccn(CC#N)n3)=O)CC2)=O)ccc2c(n1)CCC2 N1(CC(N2C(CNC(C(CC)N(CC)CC)=O)CC2)=O)CCCNS1(=O)=O c1(C(=O)NC2C3(CC(NC(CCCSC)=O)C3)C2)cccc(C#CCO)c1 c1(C(=O)NCC2=CCN(C(c3[nH]c(=NC)sc3)=O)CC2)c(C)nc(CO)nc1C N1(C(C(C)OC2CCCC2)=O)CCC(N(C)C(c2ccc(C(F)F)o2)=O)C1 Cc1ccc2c(c1)C(=O)N(CC(=O)N(CCC(O)C1CCC1)C1CCCC1)C2=O C(=O)(CC(CC(N)=O)CC(C)C)NCC1N(C(CCOCCC)=O)CCOC1 C(=O)(C1=CCCCCC1)N1CCN(C(C(CC=C)C)=O)C(c2ccncc2)C1 c1(OC)c[nH]nc1C(=O)NC1CCC(CNC(C2(C(C)C)CCC2)=O)C1 C12(CNC(Cc3c(C)nccc3)=O)CC(CO1)N(C(C1CS(=O)C1)=O)C2 C1(C)(CNC(C2(COC)CCC2)=O)CCN(C(C2CCCC2C#N)=O)CC1 c1(C(N(C)Cc2ccccc2)=O)cn2c(n1)CN(C(c1cnn(C)c1Br)=O)CC2 C(=O)(C(C(C)(C)O)NC(c1coc2c1COC2)=O)N(CC(COC)O)C c1(NCCC2CCN(C(=O)CCC3CCOC3)CC2)c(F)cccc1[N+](=O)[O-] CCCCCCC(=O)NC(C1CCCN(C(C2SCC=C2C)=O)C1)C c1(CN2CC(C(N3CCC3CO)=O)SCC2)cccc(OC(F)(F)F)c1Br CN1CCCC(F)(C(N2CCC(CNC(C3CC(=O)CCO3)=O)CC2)=O)C1 Cc1cc(CS(=O)(=O)NC(C(N2CCN(C(C)C)C(C)C2)C)=O)ccc1F C(=O)(C#CC1CCCCO1)NC1C(CNC(c2cnc(CCC)s2)=O)CC1 C1(N(CC(=O)OC(C)(C)C)C(=O)CC)CCN(Cc2ccccc2)CC12CC2 c1(NC2(c3n(CCOCC)nnn3)CCOC2C)cc(S(N)(=O)=O)ccn1 c1(C(=O)NCC2CCC(C)CN2C(=O)Cc2ccns2)cc2ccc(F)cc2o1 N1(C(CC(CC)NC(c2c[nH]c(C#N)c2)=O)=O)CCC(C)(C)C1CO N1(C(C2CNC(=O)O2)C(=O)NCC(CC)CC)CCC(OC(C)C)CC1 C1(NC(C(C=C)(C)CC)=O)CCC2CN(C(C3CC3F)=O)CCC2C1 n1(C(C)(C)C)cnnc1C1CC1C(=O)NCC(C)NC(c1cnc(O)o1)=O CC1(C)C(CNC(C2(c3ccc(F)c(F)c3)CC2)=O)CCN1C(=O)C1=CCSC1 C1(CNC(C2(NC(C3CC(OC)(OC)C3)=O)CC(CO)C2)=O)CCC(O)CC1 c1(SCC)ccc(CC(=O)NC2C(CCSCC3(C(=O)N)CCCC3)C2)cc1 C1(C(N2CCCOCC2)=O)COCCN(CC2CCNC2=O)C1 c1(C(=O)OC(c2c(F)cccc2Cl)C)ccc2nc(O)n(C)c2n1 C(=O)(C(C)(C)C(O)CC)NC(CC=C)CNC(=O)Cc1nc(C2CC2)nn1C C1(C(=O)NCC2CCC(NC(c3ccn(CC)n3)=O)C2)C2CC3C(C2=O)C13 CC(CC(=O)N(C(C)C(=O)NCc1nnc(O)o1)C1CC1)N(C)C C1(CC)CN(C(=NCCc2cn3c(n2)SCC3)NCCc2ccccc2)CCS1 CC(CC(=O)NC1(C(=O)O)CC(F)C1)C(F)(F)F Cc1nnc2cnc(C(N3CCN(C(=O)CC4(O)CC4)CC3C(C)C)=O)cn12 CC(C)(CC(=O)NC1CCC(NC(c2cnc(Br)s2)=O)C1)C(F)(F)F Cc1c(C(=O)NC(CNC(=O)CC2CCC(=O)N2C)C2CC2)cccc1N C(=O)(C1=C(Cl)CCCC1)NC1C2C(C(=O)NCC3COCC(C)O3)C3C(C2)C13 Cc1nn(C)c(C)c1OCC(=O)NC(C)C(CO)NC(=O)CC1CCNC(=O)C1 c1(OC)cccnc1C(=O)NCCCCNC(=O)CC(C)NC(C1CCCCC1)=O C(CCCCCNC(=O)CC1CCC(O)C1)N(C)C(c1cnc(C(C)(F)F)s1)=O N1(CC(=O)NC2CCC(NC(CC3(OCC)CC3)=O)CC2)C(=O)C(C)C(C)C1=O C1(CNC(CCc2ccc(C)o2)=O)C2CCC(C2)N1C(c1cc(C2CC2)n[nH]1)=O C1(C(N(CC(O)COC(c2ccccc2)C)C(C)C)=O)CNCC1C1CCCC1 C(CC(C)(C)C(=O)NC1CCC(NC(c2scnc2C2CCCC2)=O)C1)SC c1(C(N2C3CC(NC(CCCOCC=C)=O)C2CC3)=O)cc2oc(Cl)cc2[nH]1 C1(C(N2C(CCCNC(c3cnccc3Cl)=O)CCCC2)=O)CC(C2CC2)=NO1 c1(C(=O)NC(C(=O)N(CC(C)(C)O)C)Cn2cncn2)c[nH]c(=S)cn1 N1(C(C2(C(=O)OC)CC2C)=O)CCC(C2CC2)(CNC(=O)CC(C)(C)OC)C1 CC1CCC(CC(=O)N(C2CN(C(c3cn(C4CCOC4)cn3)=O)C2)C)O1 N1(C(=O)C(F)(F)CO)CC2CCC(NC(CCC(=O)OCC)=O)CC2C1 C(CC(=O)NCC1(n2cccn2)CC1)(C(C)(C)C)NC(CC1(CC(C)C)CC1)=O c1(OC)cc(C(c2cccc(F)c2)NC(C(C)(C)CO)c2nnnn2C)cc(C)c1 C(=O)(CC(C)C(F)F)NC1(C(=O)NCC=CC(=O)Nc2c(OC)ccnc2)CCC1 O=S(=O)(c1ccc(NCC2CC=CC2)c(Br)c1)N1CC(CO)CC(C(F)(F)F)C1 N1(C(c2nc(C)sc2)=O)CC2CCN(C(C3CN(C4CCOCC4)C3)=O)CCC2C1 c1(C(=O)NCC2(CC(N3C(CC)C=CCC3)=O)CC2)cnn2ccccc12 c1(NC(C)C)cnccc1C(N1CC2CC2(C(=O)NCCCCC2CC2C)C1)=O c1(C(=O)NCCOC2CCN(C(c3cn(C)nn3)=O)C2)cccc(Br)c1O N1(C(C=CC(C)C)=O)CCCC(C)(CNC(C2(c3cccnc3)CCC2)=O)C1 C=CC(CC)CC(=O)NCCC(C)NC(=O)C(C)OCC(C)C c1(C(C2CC(NC3CCN(C)CC3)C2)CC)cnn(C)c1Cl C1(CNC(CC(CC)O)=O)CCCC2(CN(C(c3cn(C)nn3)=O)C2)O1 CCS(=O)(=O)C1(CNC(=NCc2ccc(F)cc2)NC(C2CCCO2)C)CC1 c1(C(=O)NC(CC)CN(C(C2CC2C)=O)CC)ccc(C(C)=O)c(F)c1F N1(C(=O)C(=O)NCCOCC(CC)N(C)C)CCC(CF)C1 C(C(CNC(=O)Cc1ccccc1SC)C(F)(F)F)NC(C=CC=CCC)=O C1(C(=O)NCC(C2CC2)NC(=O)COC(F)(F)F)(OC)CCCCC1 c1(CC)cnc(O)c(C(=O)NC2(CC)CCCN(C(C3CC(=C4CC4)C3)=O)C2)c1 N1(C(C(C)OC2CCCCC2)=O)CCCC(C)(CNC(C23CC(C2)C3)=O)C1 N1(C(c2cn(CCNC(C3(CC)CCC(C)C3)=O)nc2)=O)CCC(C)(F)CC1 C1(C(=O)N(C)CC2CCN(C)CC2)(CC)CCCN(C(C2CC3CCC3C2)=O)C1 C1(C(N2CCC(C)C(NC(c3csc(O)n3)=O)C2)=O)CCC2CCCCC2C1 C(=O)(CC(C)C(F)F)NC(CCOC)C(=O)N1CC(C)(O)C1 n1(CC(=O)NC(C(C)C)CNC(C2(F)CCOCC2)=O)cc(C#N)c(O)nc1=O C(CNC(=O)C(C)(C)C1CCCO1)(CC(F)(F)F)NC(CCc1n(C)cnc1)=O c1(C(=O)NCCN(C)C(=O)C2CC2)c(F)cc([N+](=O)[O-])cc1Cl.C1(N)CCCC1CF N1(C(c2cn(C(C)C)nn2)=O)CC2(CCC2)CC1CNC(c1c[nH]nc1F)=O c1(-c2nc(C)nn2C2CCOC2)ccnc2[nH]c(-c3cnccn3)nc12 C(=O)(C1=NOC(C)(C)C1)NC(C(C)NC(c1cc(C(F)F)no1)=O)(C)C C(=O)(CC(CC)C(C)C)NCC1N(C(c2cccc(CCC)c2)=O)CC1 N1(C(=O)CC(O)Cc2ccccc2)CC2(C34CC(CC5CCC5)(C3)C4)CCC1CC2 c1(C(=O)NC(C(CO)NC(c2ccc(C)c(C)c2)=O)C)cnc(P(C)(C)=O)cn1 c1(C(C)(C)OC)nc(CCC(F)(F)F)nn1-c1ccc(C(C)(C)C)cc1 c1(SCC(=O)NCC2N(C(C(CC)n3cncn3)=O)CC=C2)cnn(C)c1C N1(C(COCc2nnc(C)s2)=O)CC(NC(c2cnn[nH]2)=O)CC(O)C1 CCC(N=c1cc(C)nc(N2CCC(C)(C)CC2)[nH]1)c1nccs1 C1(O)(C(C(=O)NCCc2cc(C)on2)NC(=O)CC2CC=CC2)CCCCC1 Cc1cc(Cl)ccc1OCCC(=O)N1CCC1CNC(c1n[nH]c(=N)s1)=O c1(CCCC)cc(NC(C)CNC(c2ccnn2C2CC2)=O)n2ncnc2n1 Cc1c(C(N2CC3C(C(N4Cc5ncsc5C4)=O)C3C2)=O)sc2ccccc12 C12(CNC(C3CN(S(C)(=O)=O)C3)=O)CCCC1N(C(=O)CN1CCSCC1)CC2 N1(c2nc(C)cc(CC)n2)CC2CC1CN(C(C1CNc3ccnn3C1)=O)C2 CCC(O)C(F)(F)C(=O)NC1CCN(C(=O)C=CCOCC(F)(F)F)C1C n1(CCC(N2CCC(COC)(NC(c3csc(C)c3C)=O)C2)=O)nc(C)c(C)c1C c1(C(C)NC(c2ccsc2Cl)=O)ccc(CNC(=O)C(C)c2ncco2)cc1 C(=O)(C1=CCCSC1)N(CC(CNC(C1C(c2cccc(C)c2)C1)=O)O)C C=CC(C)(C)CCCN=c1nc2c(ncn2C(C)C)c(NC2CC(C)C2(C)C)[nH]1 C(N=c1ccn2nccc2[nH]1)C1CC(NC(C2C(=O)NCCC2)=O)C1 S(=O)(=O)(C1CCC(C#N)C1)NCC(C(=O)OCC)(C(=O)OC)C(F)(F)F C1(C(N2CC(NC(CSCCC)=O)C(n3cccn3)C2)=O)CCc2ccnn2C1 N1(C(c2n(CC)nnc2)=O)CCC2CCN(C(=O)Cc3ccc4nn[nH]c4c3)CC12 Cc1ccc(O)c(C(N2CCC=CC2C(=O)N(C)Cc2ncccn2)=O)c1 C(C(C)(C)CN(C(=O)C(n1cc(Br)cn1)C)CC)NC(C(F)OC)=O c1(C(=O)NCCN(C(c2occc2Cl)=O)CC)cnc(C(F)F)c(F)c1 C(=O)(C(C)N=[N+]=[N-])NC(C(=O)NC(C=C)C1CC1)CC1CCC1 c1(CNC(C(=O)NC(c2cc(OC(F)(F)F)cc(Br)c2)C)=O)nc(Cl)ccc1F N1(C(C=C(C)C(F)F)=O)CCC(C(=O)NC(c2nccn2C)C)(C(C)C)C1 N1(C(COc2c(OC(C)C)cccc2)=O)CC(NC(C2(C)COC2)=O)CCC1C N1(C(C2(COC)CCCO2)=O)CCN(CC(=O)NCC2CCCN2N=O)CC1 n1(COC)nccc1C(=O)NC(C)CCCNC(c1ncoc1-c1ccon1)=O c1(C(C)CNC(=O)C(=O)NC(c2ncc(C(C)(C)C)o2)C)cccc(F)c1F c1(C(=O)NC(C(C)C)(C)C)ccc(CNC(c2cn(CCO)nn2)=O)cn1 c1(-c2scc(C(=O)NCC#CCNC(C(C)CN(C)C)=O)n2)ccccc1Br C1(CNC(c2cscn2)=O)CCC2CN(C(c3cccn3C3CC3)=O)CC12 C1(Cc2ccc(NC(CN3CC(C)N(CC)CC3)=O)cn2)CCCC(C)(C)CC1 C12(C(=O)NC(C3CCCC3)C#C)CC(CO1)N(C(=O)CCCC(=O)OC)C2 C1(CN(C(=O)CC2CCC(F)(F)C2)C)CN(C(C2CCCN2C)=O)CCO1 N1(C(CC)=O)CCCCC1C(N1C(CNC(c2cnc(CC)[nH]2)=O)CCC1)=O N1(c2cc(NC(c3cnc(Br)s3)=O)ncn2)CC2(CCCC(C(=O)O)O2)C1 C(CCC(C)C)(C(=O)NCCC(C)(O)C1CC1)NC(CCC)=O C1(COC)(CNC(=O)Cc2cnoc2)CCCN1C(C1CCCCN1C)=O C=CC(C)(C)CC(=O)N1CCCC1CN(C(=O)CCOCC(C)(C)C)C N1(C(C(CNC(C(C=C)OC)=O)C(C)C)=O)CC2(CCC(=O)O2)C1 c1(C(=O)NCC(CC)NC(c2csc(C)c2N)=O)cnc2n1CCS2 C12(NC(c3c(OCC)scc3)=O)CC(COC)(C1)OC21CCN(C(=O)CSC)CC1 C1(C(N2C(CO)CC(OC)C2)=O)CC(=O)NC(=O)C1.c12ccnc(c1)OC2=O Cc1[nH]c(C)c(C(=O)NCCC2CC(C(N3CC=CC(O)C3)=O)C2)c1C Cc1ccc(CC(=O)NC(C)(CNC(c2ccnn2CCF)=O)CO)cc1C c1(C(=O)NC2C(NC(c3ccnc(C)c3N)=O)C2)ccn2c(Br)cnc2c1 C(=O)(CC(O)C(C)C)NCC=CCNC(c1c(C)n(-c2cccc(Cl)c2)nc1)=O c1(C(=O)NC(CNC(C(COC)C)=O)CC2CCCCC2)ccnnc1NC1CC1 c1(N(CC=C)C(c2cnccn2)=O)ccc2cnn(C(C)=NO)c2c1 N1(C(CSCC)=O)CCOC2CCN(C(C3CCC(=O)NC3)=O)CC12 C12(C(=O)NCCCN(C)C)CC(CN(C(=O)COCC3CCCO3)C1)C2 C1(C2CCN(C(c3c(F)c(F)cc(F)c3F)=O)C2)(NC(C2C(C)(CC)C2)=O)CC1 CN1CC(CNC(C2CC2CNC(=O)C(F)(F)CO)=O)CC1=O C(=O)(C#CC1CCC(=O)CC1)N1CC(=C(CNC(CSc2nc(C)[nH]n2)=O)F)C1 C(=O)(CCCS(N)(=O)=O)NC1C(C)CN(C(=O)CCOC2CCOCC2)CC1 N1(c2c(C)c(N(CCCN(C)C3CC3)C)ncn2)CCc2ccccc2C(C)(C)C1 C1(C(=O)NC2CCC(N(C(c3sccc3OC)=O)CC)CC2)CC(=O)NC(=O)C1 c1(C(N2CC(CCCCSC)C2)=O)ncc(F)c(OC)n1.c12nocc1C(=O)NC2 c1(NCc2nc(C)no2)[nH]c2ccccc2c1C(C(CC)(C)OC)OC C1(NC(CCC(N)=O)=O)CC2CC(NC(=O)Cn3nnc(C(C)(C)C)n3)C2C1 N1(C(C2(C#C)CCCC2)=O)CC2(CNC(=O)C(CC)n3nccc3C)CC1CO2 c1(SCCOCCCNC(C(=O)N(C2C(C(C)O)C2)C)=O)ccccc1 C(=O)(CC1=CCCCC1)N(C1CC(C#N)C1)CC(=O)NCCc1ncccn1 N1(CC(N2CC3(CC(CC(=O)OC)C3)C2)=O)C(C)CCC(C(=O)O)C1C N1(C(C(C(C)C)F)=O)CCC(NC(=O)C(C)OCc2ccccc2C)C12CC2 c1(C(N2C(C)(C(=O)N(C3CCC(C(=O)O)C3)C3CC3)CC2)=O)ccc(F)cc1Cl Cc1ncncc1C(=O)NC1CN(Cc2ncccc2Cl)CC1O CCC(C(=O)NCC1CC(NC(c2ccoc2CC)=O)C1)n1ccc(C2CC2)n1 C(C)(C(C(=O)NCC1CC1(Cl)Cl)NC(=O)C(O)CCSC)OC C1(CNC(C2CC3CCC2O3)=O)CCC2(CN(C(c3c(F)ccnc3Cl)=O)C2)O1 c1(CC)nc(C)oc1C(N1CCC(CF)(NC(c2ccnnc2C)=O)C1)=O C12(NC(c3csnn3)=O)COCCC1CN(C(=O)CCOC1CC1)C2 C1(CNC(CCOC(C)C)=O)CCCCCN1C(=O)C=CCN1CCCC1 c1(C(N(CCC)CCNC(C23CCN(CC2)C3)=O)=O)ccc(F)c(O)c1 CC1ON=C(C(=O)N(C2COC3(C2)CN(CC(=O)NCC#N)C3)CC2CC2)C1C C1(C(N(CCOCC(F)Cl)CC)=O)CCOCCN1C(=O)COC C(C(=O)N1CCCO1)NC(c1cc(CNC(=O)CC2CCCC23CC3)[nH]n1)=O N1(C(CC)=O)CCCC12CCCN(C(=O)Cc1ccc(-n3cnnn3)cc1)C2 N1(C(c2ccc(N)c(C)c2C)=O)CCCC2(NC(c3ccon3)=O)CCCC12 N1(C(C2(NC(=O)COC(F)(F)F)CCC(C)(C)C2)=O)CC2(CCCCC2)C1 N1(C(C2CC(CC)C2)=O)CCC(CNC(=O)Cc2cccc(C)c2F)(OC)CC1 c1(-c2ccn(C)n2)ccc2[nH]nc(NC(c3cccc(I)c3F)=O)c2c1 C1(CC(N2CC(N(C(c3c(C)cccc3)=O)CCO)C2)=O)CCCC(F)(F)C1 C1(NC(c2c(C)cno2)=O)CC2(C1)CC(CNC(c1ccc(C(N)=O)o1)=O)C2 C(C)(C)(C(=O)NCCC1CC(NC(=O)Cc2cc[nH]n2)C1)OCCC c1(NC(N2CC3C(Nc4cccc(CC)n4)(C3)C2)=O)ccc([N+](=O)[O-])cc1Cl N1(CCc2cn(CC3CC(NC(c4c(OC)scc4)=O)C3)nn2)CCN(C)CC1 C1(NC(=O)Cn2cncn2)CCN(C(=O)CC2CC3C=CC2CC3)C12CCC2 c1(-c2ccc(C3(NC(N4CC5CC4CC5O)=O)CC3)cc2)ccc2c[nH]nc2c1 C1(NC(=O)NC(C(=O)OCC)C)CC(C)CN(C(=O)Cn2cnnn2)C1 CC(C)CCC(=O)C(=O)NC1(C(=O)N(CC(F)Cl)C)CC1 c1(C(=O)NCCCCCNC(C2CCC(C(=O)OC)C2)=O)cccc2nc[nH]c12 N1(CCC(=O)N(C2CCCC2)CC(ONC(=O)C2CC2)=O)CCOC1=O C12(NC(CC3CN(C)C3)=O)CCC(CN(C(C3(C#N)CC4(CC4)C3)=O)C1)C2 C1(NC(c2n(C)cc(Br)c2)=O)CCC2CN(C(=O)Cc3cc[nH]c3)CCC2C1 c1(NC(CC)C(F)F)nc(Cl)cc2c(N)cccc12 C(=O)(CCCCCNC(N)=O)NCC1(NC(c2cnc(OC)s2)=O)CC1 C1(C(=O)NCC(CNC(C(C)=C(C)C)=O)(C)C)CCN(c2ccccc2C)C1=O S(=O)(=O)(c1ccc(Cl)c([N+](=O)[O-])c1)NCCS(=O)(=O)NC C#CC1(C(=O)NCC2(COC)CCC2)CCN(C(=O)C(C)CC=C)C1 c1(CN(C(=O)CC2C=CCCC2)C)ccc2c(c1)CCCS2 C=CCC(C(=O)NCC(C(N1CCC(C#N)(CCC)CC1)=O)OC)C(C)C c1(C(c2n(CCOCC)nnn2)NCCS(C)(=N)=O)cccc(Cl)c1Cl c1(C(C)=O)ccc(C(=O)NC(CNC(=O)CCCN(C)C)CO)o1 C12CC(C13CCC3)N2.N=c1ncn(CC(=O)NCC(N2CCC(C(N)=O)C2)=O)[nH]1 C1(N=[N+]=[N-])(C(=O)NCCCOCCOC)CCN(C(=O)C(C2CC2)SC)C1 C1(CC=C)(NC(=O)CSC(F)F)CCCN(C(=O)CC(C)(C)C)C1 CCCC(CNC(=O)C(F)=C(C)C)C(=O)N(C)CC12CCC(CC1)C2 N1(C(C(C)n2cccn2)=O)CCCC2C1CCN2C(=O)Cn1nnc(=O)[nH]1 c1(C(N(CCCN(CC)CC)CC)=O)c(O)nnc(CNC)c1NC C1(C(N(C)Cc2cnn(C)c2)=O)CN(C(=O)CCc2nc[nH]n2)CC1(F)F C(C(=O)NCC1CCC(NC(c2ncccn2)=O)C1)(C(C)C)OCC N1(CCCC(=O)N(C2(C(=O)OC(C3CCCCC3)=O)CC2)C)CCC(=O)CC1 c1(OC)cc(O)ncc1C(=O)NCC1C=CCN1C(=O)C(C)OC c1(C(=O)NCC(C)CN(C(=O)CCSc2nnnn2C)C)cccc(N(C)C)c1 C12CCCCC1NC(=O)C2.N1(C2(NC(=O)CN3CC4CC4C3)CC2)CCOCC1 n1(C(C)C)ncc(Cl)c1C(=O)NCCCC1CCCN1C(=O)CN1CC(C)(C)C1 C1(C(=O)OC)(C(=O)NCCCOC2CCCCC2)CC(O)C1(C)C Cc1cnccc1CNC(=O)CN(C(C1CC2CCC2C1)=O)C1CC1 N1(C(c2c(CC)nccc2)=O)CCC(O)(CNC(c2cc(C)cc(F)c2)=O)CC1 Cc1cnc2c(C(=O)NC3CC4CN(C(=O)CN5CCCCC5)CC34)cnn2c1 Cc1ccc(N(C(=O)CCCC2CCC2)C(c2cccs2)=O)cc1.C(CCSC)N C1(CC(=O)NC2CC(OCC(=O)N(CCCn3cccn3)C)C2)CCCC1O C1(C(=O)NCC(C(C)C)NC(c2ccn(CC)c2C)=O)CC2(C1)CC21CC1 N1(C(CC=C)=O)CCCC2(CCCN2C(C2(C3CCCO3)CCCO2)=O)C1 C1(C)(C(C)NC(c2nc(C3CC3)cs2)=O)CCN(C(=O)C(F)=CCCF)C1 c1(C(=O)NCCCC2N(C(C(CCC)OC)=O)CCC2)ccc(S(N)(=O)=O)cn1 C1(C(=O)NC(C(C)NC(C2OCC2(C)C)=O)(C)C)CCCN(CC(F)F)C1 C1(C(=O)NCC(C)CN(C(=O)Cc2cccc(Cl)c2)C)(CC)CCNC1=O N1(c2c(F)ncc(-c3c(C)ccc(CO)c3)c2)CCc2c(O)noc2C1 C1(N(C(C(C)(C)N2CCCC2)=O)CCO)CCCCN(C(C2(O)CCC2)=O)C1 c1(CC)cc(C(N2CC(NC(c3ccc(CC#N)cc3)=O)CC2C)=O)sc1C c1(C(=O)OCC)cc(CO)ccc1Cl.C12CC1C(=O)OCCO2 C1(CC(N2C(CC)C=CC2)=O)CCCCN1C(c1cccc(CNC(C)=O)c1)=O C(C(=O)N(C)CCN(C)C(c1nccc(C)n1)=O)(C(C)C)OC C1(CNC(C2CC(OCC)C2)=O)CC2CCC1N(C(=O)CC1(C)CCC1)C2 C(CCCC(F)(F)F)N1CCOCC(C(=O)NCC(C2CCCCC2)O)C1 CC(=O)CCN=C(NC(=O)Nc1ccccc1)NC1CC1C1CCOCC1 c1(C(=O)NCCCCNCC(COC)O)cccc(OCc2ccccc2)c1 CC1Cc2cc(C(=O)NCC3CCC(C(=O)O)CC3)ccc2N1 C1(CC=C)(NC(=O)C(CCO)N(C)C)CC2CCC(C1)N2C(=O)CSC(F)F c1(C(=O)N)c[nH]nc1NC(C1C(C(=O)NC2(c3cc[nH]n3)CC2)C1)=O.CC(F)F c1(C(=O)NC2CCC(NC(C3C(=C)CC3)=O)C2)cc(S(=O)(=O)NCC)ccc1C c1(C(=O)NCC2N(C(C(N3CCSCC3)C)=O)CC2)ccnn2ccnc12 Cc1nn(C)c(C(=O)NC2CC3CC(NC(=O)CSc4ccccn4)C3C2)c1Cl Cc1ccc(CCC(N2CCN(C(=O)CSc3cnoc3C)CC2C)=O)cc1C C1(NC(C(CCF)NC(c2n(CC)nc(C)c2)=O)=O)CCn2cnnc2C1 C1(NC(C2C(=C)C2)=O)CCCC(NC(=O)Cn2ncc(Cl)c2C)C1 c1(C(=O)Nc2n(C)ccn2)cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O C(C(C)(C)CC(=O)NCC1(n2nccn2)CC1)NC(C1CC(N(C)C)C1(C)C)=O N1(C(CC(C)F)=O)CCOCC1CN(C)C(C1CC(F)C(=O)N1)=O N1(C(COC(CC)(C)C)=O)CCN2C(=O)C(NC(=O)CNC(=O)OC)CC2C1.C(C)=O N12CCCC3(CCN(C3)N(C)c3cc1ncn3)C2.c1(CN)c(C)cnn1C.CC CC12CC(C(N3CC4=C(C3)CN(C(C3(C#N)CCCC3)=O)C4)=O)(C1)C1(COC1)O2 C1(NC(c2cc(COC)[nH]n2)=O)CCN(C(=O)CC2(OC)CC2)CC1(C)C C(=O)(C1=CC(O)C(NC(c2cccc(O)c2)=O)C1)NCCC(C(C)C)C C1(CNC(C(c2cccc(Br)c2)N)=O)CCC2(CCOCC2)O1 c1(C(=O)OC)ncc(NC(=O)C(C)Sc2cccs2)cc1F C1(C(=O)NC(C(CO)NC(C2(CC)CCOCC2)=O)C)CC2CCC(C1)N2C c1(C(N2CC(OCCNC(c3cccc(C)c3F)=O)C2)=O)ccc2nsnc2c1 N1(C(c2c[nH]c(=NC)o2)=O)CC2(CCCC2)C1C(=O)NCc1ccnc(O)c1 c1(OCC(N2CCN(C(CCSCCC)=O)CC2CO)=O)cccc([N+](=O)[O-])c1 C1(CNC(C2(CC=C)CC2)=O)CN(C(C)=O)CC2(CCC2)O1.C12CCC1C2 CC1(CC2CCC2)CCCN1Cc1sc(Br)c(Br)c1F CC1(N2CCOCC2)CCN(C(c2ccc(N3CCOCC3)cn2)=O)CCO1 c1(CSc2snc(C)n2)ccc(C(=O)O)cc1.C1CCC(=O)NCCn2cc1nn2 CC1(CNC(c2csc(=N)[nH]2)=O)CCCN1C(c1cc(C(F)(F)F)n[nH]1)=O c1(CNC(C(N2CCC(SC(c3ccccc3F)C)C2)=O)=O)csc2cncn12 C(=O)(C1=CCS(=O)(=O)C1)N1CCC(C)C1.N1(C(C2C3CCC23)=O)CCOC(C)C1 N1(C(c2c(C)coc2)=O)CCC2CN(C(=O)C3=CCC(C)CC3)CC2C1 c1(C(N)=O)cnc(N2CCC(CF)(NC(=O)COc3ccon3)C2)c2ccsc12 C1(F)(C(=O)NC(CSCCCC)=O)CC(CNCC2(N3CCC(C)C3)CC2)C1 CC(C)(CCCF)NC(=O)NCC1(N2CCOCC2)CC1 C12(CNC(C3C(C)C3C)=O)CCCCC1N(C(=O)COCCN(C)C)CC2 c1(C(=O)NC2(C3CN(C(C=CS(C)=O)=O)C3)CC2)ccc2cnccc2c1 Cn1nc(O)cc1NC(C12CC1CN(C(c1cnn(C3CCOCC3)c1)=O)C2)=O N1(C(C(CC#C)O)=O)CCCC(O)(CCNC(c2ccc(C(C)C)cc2)=O)C1 C1(C(=O)NC(C2CCN(C(Cc3c(C)cccc3)=O)C2)(C)C)CN2CCC1CC2 Cc1ccc(C(N2CCN(C(=O)CC3CC(F)C3)C(CCO)C2)=O)c(F)c1Cl C1(C(=O)NC(CNC(C23COCC2C3(F)F)=O)C2CC2)CCC(=C(F)F)CC1 C1(C(=O)NC(C(C)N(C(=O)C=Cc2cccc(C)c2)CCC)=O)CCCC(C)C1C c1(C(=O)OC)cc(O)c(NC(=O)NC2C=CCCCC2)cc1F N1(C(C(CCC)OC)=O)CCC(CO)(CNC(c2[nH]c(O)nc2C)=O)CC1 C1(CC)CCN(C(=O)Cc2cn[nH]c2)C1CNC(=O)CCOCC1CCC1 C1(NC(C2CCC2)=O)CCC2CN(c3[nH]cnc4nc(Cl)cc3-4)CCC2C1 Cc1cn(CC(F)(F)F)[nH]c1=NC(=O)C(C)c1ccc(Cl)c2ccccc12 Cc1ccc(N(C(CCC2CCC2)C(=O)NCCCNC2CC2)C)c(Br)c1 C1(=CC(=O)NC2(CNC(C(C)OC3CCCC3)=O)CC2)CCCCC1 C1(C(C)(C)C)CC(c2nnnn2CC(F)F)(NCCCC2CCCCC2)C1 C=CCCCCC(C)(c1nnnn1Cc1ccco1)NCC1CCOC1 c1(N2CC3OCC(C(=O)NC(CC)CO)C3C2)ncnc2scc(C)c12 C1(NCC)CCCCN(N2CCCN(C(=O)OC(C)(C)C)CC2)C1 CCN=c1[nH]c(C(=O)NC2CCC2NC(c2ccc(C)cc2F)=O)cs1 CC1c2cc(Cl)c(Cl)cc2CCN1C(=O)C(=O)NCCc1cccc2cnccc12 N1(C(CCOCCC)=O)CC(C)C(NC(C2C(C)C2C)=O)C(C)C1 C1(CC)CC2CCC1N2C(C12CC1CCN2C(=O)CCc1ccccc1)=O Cc1cccc(Cl)c1CC(=O)N(C(C)C(C)S(C)(=O)=O)C c1(SC)ccc(-c2nc(-c3coc(C)n3)n(CCS(N)(=O)=O)n2)nc1 C1(CC(=O)NC(CC)CC)CCCN(C(c2cccn2CCOC)=O)CC1 c1(C(COC)NC(=O)NC2CCN(CC(F)(F)F)C2)ccncc1 C(CC(=O)NC1CCNC(=O)C1)(C(F)(F)F)NC(COCCCOC)=O C(=O)(C(C(CC)CC)OC)N1CCC2(C(C(N3C(C#C)COCC3)=O)C2)C1 C1(OC)(CNC(c2nc(C(C)C)oc2C)=O)CCN(C(C2CC2[N+](=O)[O-])=O)C1 C(=O)(C(F)C(C)C)NC1CCN(C(C(=O)NCCOC)=O)C1 c1(C(CC)NCCC2CC2C(=O)OC(C)(C)C)cn(-c2ccccc2)nn1 C1(O)(CNC(C2(OC)CCOCC2)=O)CCCN(C(C2(CO)CC2)=O)C1 c1(OC)ncccc1C(=O)NCC1C=CCN1C(C1CCCC1SC(F)F)=O c1(C(=O)NCC(CNC(c2c(CN(C)C)noc2)=O)O)cc(O)cc([N+](=O)[O-])c1 C1(C(=O)NCC(CCC)OC)N(C(=O)CSCCOC)CCC1(C)C CC(C)CS(=O)(=O)CCC(=O)Nc1ccc(N2CCCCCC2)nc1 c1(C(N2CCC(N(C(CCCCN(C(C)=O)C)=O)C)C2)=O)cccc(=O)n1C CCC(C)(O)CNC(C1(C2CCCO2)CCC1)=O C#Cc1cc(NC2CN(C(=O)C(CC(C)C)OCOC)C(C)(C)C2)ccc1C C1(C)(OC)CCN(C(=O)CSCCN(C(=O)CN2CC(C)(C)C2)CCO)CC1 c1(OC)cccc(C2CC(O)CN2C(=O)CCn2cc(CC3CCCO3)nn2)c1 Cc1cc(=NCC(C)N2CCCCC2)[nH]c(=NC(C)CN(C)C)[nH]1 C1(CNC(C(CC(=C)C)OC)=O)CC2CCC1N(C(=O)CNC(N)=O)C2 c1(C(=O)NC(CCOC)CNC(c2cc(C(F)F)ccn2)=O)ccn2c1CCC2 c1(C(N2C(C(N3CCC(CCOC)C3)=O)CC3CC32)=O)cc(C)c(O)nn1 C1(NC(C(C)OC(c2ccccc2)=O)=O)CCN(c2ccccc2)C1=O C1(=CC(N2CC(CCO)(NC(c3c(C)con3)=O)C2)=O)CCC(C)CC1 C(CC1CCC1)(C(=O)NC1CC(CNC(C2CCCC2O)=O)C1)OC CCC(C(=O)OCC)C(=O)NC1CCCC(CNC(c2cnccn2)=O)C1 c1(C(C)(C)C(N2CC(NC(c3cnc(S)nc3)=O)C(O)C2)=O)cc(Cl)cc(Cl)c1 Cc1cc2c(cc1C(=O)NC1CC(F)(CNC(=O)Cc3ccoc3C)C1)OCO2 Cc1cc(C(N2CC3CC3(CNC(c3sc(C#N)cc3Cl)=O)C2)=O)cc(C)c1F c1(C(=O)NC2CN(C(C3=NOC(C)C3)=O)CC(F)C2)ccc2c(c1)NC(=O)C2=O Cc1ccc(C(O)CNC(c2cnn(C)n2)=O)cc1C c1(OC)cc(C(=O)NCCCCCNC(C2(OC)CCOC2)=O)n(C)n1 C1(CCC(=O)NCC=C)CCN(C(=O)Cc2scnc2C)C1 N1(CC2CCC(C)(C)O2)CCC(O)C(C(=O)NC2(c3ccc(F)cc3)CC2)C1 C1(C(=O)NCCOC2CN(C(C(C)N(C)C)=O)C2)OCCOC1C c1(C(N(C)CC2N(C(c3c(C)cns3)=O)CCC2)=O)c(C)n(C)c2ccccc12 N1(C(c2ccc(NC)cc2)=O)CC2CC1CCC2NC(C1CCCC(=O)N1)=O CC1CN(C(c2csc(CO)n2)=O)CC1(C)C(=O)NCC1CCC(F)C1 c1(C(=O)NC(CCNC(c2c(C#C)c[nH]n2)=O)C)ccccc1S(=O)CC CC1(C(=O)NCC2CN(C(c3c(F)cccc3F)=O)CCO2)CC2(CCC2)C1 C(=O)(C(C(C)C)NC(=O)C(C)C#N)NCCc1c(C)nns1 C1(C(C2CN(Cc3ccc(Cl)s3)C2)=O)CCN(S(=O)(=O)C(F)F)CC1 Cc1cnc2c(C(N3CC(N(C(=O)C(C)O)C)C(C)(C)C3)=O)cnn2c1 c1(OCC)cnc(C(N2CCC(C(=O)N(CC(F)F)C)(SC)C2)=O)cn1 c1(C(C)NC(c2cc(I)cn2C)c2n(CCC)nnn2)cc(F)cc(F)c1 N1(C(=O)NC(c2cc(C)sc2C)C)C2CCC1CC(CC(F)(F)F)C2 c1(C(N2CCCC(CCNC(C3(C)CC3(F)F)=O)C2)=O)cccc(P(C)(C)=O)c1 c1(C(=O)NC2C(NC(c3oc(CC)c(C)c3)=O)CCC2)cnc2n1CCCCC2 N1(C(c2c(C)cc(C)[nH]2)=O)CCN(C(=O)COc2ccc(O)cc2)C2CC12 CC1(C#N)CCN(C(C2CCN2Cc2cccc(O)n2)=O)CC1 N1(C(c2cc(C)on2)=O)CCC(n2cccn2)(C(=O)NCC2(O)CCCC2)CC1 c1(OC)ccc2c(c1)CN(C(=O)N=c1[nH][nH]cc1C1CC1)C2 C1(COC)CN(C(=O)CC2CSC2)CCN1C(C1CCCN(C(C)C)C1)=O C1(NC(c2cc(C(=O)OC)nn2C)=O)CN(C(=O)C=C(C)C(F)F)CC12CCC2 c1(C(=O)NC2C(NC(C(CC)N3CCCC3=O)=O)COC2)cnc2ccnn2c1 Cc1cccc2cc(C(N3CCC(=CCNC(=O)Cc4ccco4)CC3)=O)nn12 C(=O)(CCCC(=O)C(C)(C)C)N1CC(COC)(NC(C2CCCC(F)C2)=O)C1 Cn1cc(S(N)(=O)=O)cc1C(=O)NCC1C2CCC(C2)N1C(c1cc(O)cs1)=O Cc1ccc(C=CC(N2CC(CC(C)NC(C3(C)CCC(=O)C3)=O)C2)=O)s1 c1(C(N2CC3(CN(C(C(CCC)CC)=O)C3)C2)=O)ccc2c(c1)C(=O)CCN2 Cc1csc2ncnc(NC3CC3C(=O)Nc3cc(Cl)ncc3F)c12 C1(N(C)C)CCC(NC(=O)C(=O)Nc2ncc[nH]2)CC1.N12CCOC(C1)C2=O C12(C(=O)NC3CC(N(C(Cc4cnc(C)s4)=O)C)C3)CCC(CC1)OC2 N1(C(C2C(C)CC(=O)NC2)=O)CCC2(CC1)CC(NC(=O)CC1CC1)C2 C1(C(C)NC(=O)CN2CCCCC2=O)CN(C(=O)C=CC(F)F)CCCO1 C1(N2C(=O)C(O)C2)CCCN(C(C2CC3(CC3)C2)=O)C1.c1(SCC)cccnc1 N1(C(CC2(C(=O)OC)CC2)=O)CCC(C2CCCN(C(C3CCN(C)C3=O)=O)C2)C1 C1(C)(NC(CCC(C)(C)NC(=O)CNC(N)=O)=O)CCCCC1(C)C C(=O)(C(O)CCC(C)C)NCC1(F)CCN(C(c2c(O)ccc(C)n2)=O)C1 O=S(=O)(c1ccc(N2CC(CO)OC(C(F)(F)F)C2)nc1)NCCC1CCCC1 C1(C(=O)NC(C)(C)CNC(C2CCC(F)C2)=O)CC2CC1CC2(F)F C=CC(CC)CC(=O)NC(c1ccc(F)cc1F)CNC(=O)C(N)=O N1(C(Cc2ccc(OC)cc2)=O)CCC2CN(C(=O)CC3(CCOC)CC3)C2C1 C(=O)(C(CO)NC(N)=O)NCCC(=O)N(C1(c2cc[nH]n2)CC1)C C(C)(C)(CCC(=O)N1CCC=CC1COC)NC(c1c(CC)cno1)=O c1(OC)cc(C(=O)NC2CN(C(C3CC3C(C)C)=O)CC23CC3)cc(N)c1O c1(OC)ccc(CCC(N2CC(F)CC2C(=O)NC2CC(F)C2)=O)cc1 CN1CC(C)(C(=O)NC2CC(CCNC(c3occ4c3CCC4)=O)C2)CCC1=O c1(C(=O)NCC2(CNC(c3cc(OCC)no3)=O)CC2)cn(C)c(=O)cn1 C(=O)(C(F)(F)C(C)O)NCC1(CO)CCN(C(C2(COCC)CC2)=O)C1 n12cnc3c(nc(N(C)CP(C)(C)=O)nc13)N(C)CC2.C(O)(C(C)C)C1CCC1.CO C1(CN(C(c2nc(C(C)OC)sc2)=O)C)CCCCN1C(=O)Cc1cnc[nH]1 C1(C2(O)CN(C(=O)C(F)C3CCOC3)C2)(CNC(=O)CCF)CC1 c1(OC)cc(C(=O)NC2CC3CC(NC(C4C=CCC4)=O)C2C3)cc([N+](=O)[O-])c1 C1(CN(C(=O)CN2CCOCC2)C)CCCN1C(=O)CC1CSCCS1 N1(C(C)C)CCOC(C(=O)NC(C)(CNC(C2CC2(C)Br)=O)C2CC2)C1 c1(C(N2CCOC(C3CC3)C2)C(=O)NCCC#N)ccc(CC2CCC2)cc1Br C=Cc1cc(C(=O)OCC2CCC(NC(=O)OC(C)(C)C)C2)cc(F)c1 C1(CC(=O)NC(c2ccnn2C)C(=O)NC(c2nn(C)cc2O)C)CC2C=CC1C2 c1(OC)ccc(C)cc1-n1cc(C2CN(C(=O)CC3(C)OCCO3)C2)nn1 c1(CC(=O)NCCOCCNC(=O)CCC2CCCOC2)cccc2nsnc12 C1(CNC(CC(C(C)C)O)=O)CC12CCN(C(=O)CN1CCCCCC1)CC2 C1(C(=O)OC(c2ccccn2)=O)CC(P(C)(C)=O)C1.c12ccc(cc1)c(=O)n2C CCC(CNC(=O)CN1CCN(C)C1)(CC)NC(=O)CCSCC(C)C n1(CC)nnc(C)c1C(=O)N(C)CC1CCCN1C(c1scnc1Cl)=O c1([N+](C(=O)NCC2CN(C(C)=O)CC2C)(C(c2ccccn2)=O)[O-])ccc(C)c(F)c1 N1(C(C(C(COC)C)C)=O)CCCCCN(c2nc(C(C)C)cc(C)n2)CCC1 C(CC(C)C(=O)NCC1CN(C(c2cc(-c3ccccn3)no2)=O)CC1O)OC c1(CN(C(=O)C(C)(C)C2CCCN2C(C2CCCS2)=O)C)ccc(O)cc1 c1(C(=O)NC(C)CN(C)C(C2CN(C3CCCCC3)C2)=O)cn2cccnc2n1 O=[N+]([O-])c1cncnc1NCC1CC1(F)Br Cc1noc(C)c1Nc1ccc(C(=O)OCc2ccc(N(C)C)s2)nc1 C(=O)(C(C)(C)C(O)C(C)C)N(CC(CNC(c1ccc(CC)nc1)=O)O)C C(=O)(C(C)CCCC(C)=O)NC1CCC(CN(C(c2c(CC)nn[nH]2)=O)C)CC1 N=c1[nH]c(C(F)(F)C(=O)NC2CCC(CCNC(=O)Cc3ccsn3)C2)cs1 c1(CCC)ccc(S(=O)(=O)N2CCC(C(=O)NC3CC3C(=O)O)C2)cc1 N1(C(c2cc(C)no2)=O)CCCN(C(c2cc3ccccn3c2)=O)C(C)C1 c1(C(=O)NC2(C)CC(NC(=O)CCc3nc[nH]n3)C2)ccc(O)nc1 c1(CC(C(=O)NCCCCOC)NC(=O)C(O)C2CCCC2)ccc(C)cc1 C(=O)(CCCC(=O)N(C(C)Cc1ccccc1C(F)(F)F)C)NCCNC(C)=O N1(C(CCC2(CCC#C)N=N2)=O)CC(C2CC2NC(=O)NC2COCC(C=C)C2)C1 c1(C(=O)NCCC2CCN(C(CC(CCCC)O)=O)CC2)cc2ccncc2[nH]1 C1(NC(C2(CC)CN(C(C3CCC(=O)N3)=O)C2)=O)CCC(=O)N(C)C1=O C1(C(=O)NCCCC(C)NC(c2cnnn2-c2ccccc2)=O)CC(=O)N(C)C1 C1(C(=O)NC(CC)CN(C(=O)Cc2cncs2)CC)C(C)(C)C1(C)C C1(C(=O)NCC(=O)OCC)CC=CC(NC(c2c(C#N)cnn2C)=O)C1 c1(NC(N2CCC(CNC(C3CCC(C(C)(C)C)CC3)=O)C2)=O)ncn2c1CCC2 C1(C)(C(N(CCCNC(C2C(C(C)C)OCC2)=O)C)=O)CCN(C)C1=O O=C(CCc1cn[nH]c1)NCC1(C(=O)NC2CC(CCN)C2)CC1.C(=O)O Cc1ccc(-c2cn(Cc3cn(-c4ccc(F)c(C)n4)nn3)nn2)c(N)c1 CCC(C)(C)CC(=O)N(C(C)(C)CC(=O)N1CCCC(CCF)C1)C C=C1CC(C(=O)NCC2CCC(C(=O)NCC=CBr)C2)(COC)C1 c1(Nc2c(C(=O)Nc3n(C)nc4c3CCC4)scc2)ncnc2ccc(F)cc12 c1(CC(=O)NCC2CCN(C(C3(CCC)CC3)=O)CC2C)cn2cccnc2n1 C1(CCOC)(C(=O)NC(C)CF)CCN(C(=O)CCC2CC2(F)F)CC1 N1(C(COC(CC)C)=O)CCCCC1CN(C(=O)CC1CC(C)C1)C CCCC(C)CN=c1[nH]c(=NCc2nncs2)[nH]c2c1CCCCCC2 C(=O)(CCCCCC(C)O)NCCC1CCN(C(CSC)=O)C1 N1(c2nc(O)cc(C)n2)CCC2(CC1)CC2C(N1CCCC1CNC(N)=O)=O C1(CCCC)CN(C(=O)CC=Cc2ccccc2)CCN1C(c1ccc[nH]1)=O c1(C(=O)NC(C(=O)NC2CCCC(CC)C2)c2cccs2)cnc(C)nc1C Cc1[nH]c(=N)nc(O)c1CC(N1CCCC(C)C1CNC(C1(CO)CC1)=O)=O N1(C(CN2CCC(C(CC(=O)OC)(C)C)CC2)=O)CCCC(O)C1C C1(CNC(CC=C=C)=O)CN(C(c2nc(OC)ccc2C)=O)CCCO1 CS(=O)CCC(=O)NCC(C)(C)OCCNC(C1(O)CCC1)=O C1(C#N)(CC)CCCN(C(C2CCCN2C(C2CCC3CC3C2)=O)=O)C1 c1(C(=O)NCC2CCCN(C(CCOCCC)=O)CC2)cc2cnc(Cl)cc2s1 c1(CC)nc2c(C(=O)NCC3CCCCN(C)C3)ccnc2[nH]1 N1(CC(=O)NCC(C)O)CCN(C(=O)COc2ccc(Cl)cc2)CC1=O C1(C(=O)NCC2(C)CCN(C(C(CSC)C)=O)C2)COC2COCC12 C1(NC(C(CCC)(C)C)=O)CCN(C(c2ccc(C)c(F)c2)=O)CCC1CO C1(CNC(C(C=C)(F)F)=O)CN(C(=O)CC2CCCCC2(C)C)CC12CCC2 C=C(C)CC(C(=O)NC1CCN(C)C1(C)C)NC(=O)C#CC(C)C c1(C2(C)CC2)cncc(C(=O)NCC(C)(C(C)C)NC(=O)CCC2CC2(F)F)c1 N1(C(C(C)=C2CCC2)=O)CCN(C(C2CCCO2)=O)CC1c1ccc(F)c(F)c1 CC1CC(NC(C2(C)CC2(F)Cl)=O)CN1C(=O)COCC1CCOC1 c1(C(C)(C)SCC2CCCC2c2nc[nH]n2)nc(CNC(=O)OC(C)(C)C)no1 N1(C(c2cn(C3CC3)cn2)=O)CCC(F)(C(=O)NCCc2nccs2)C1 N1(C(C(C)(C)c2cc[nH]n2)=O)CCOC2(C1)CN(C(=O)C1=C(Cl)CCOC1)C2 C1(C(=O)NCCC(=O)N(CC(c2ccccc2)NC(N)=O)C)CCCNS1(=O)=O CC1CCC(C)(C(=O)NC2CN(C(=O)COC3CC3(F)F)CC2C)C1(C)C C1(NC(CC2CC(NC(N)=O)C2)=O)CC2CCCCC12.C1(NC=O)CCC1 C1(CCOC)(NC(c2ccc(CO)nc2)=O)CCN(C(=O)C=C(C)Cl)C1 CCCCCCCC(F)C(=O)NCC12CC1CN(C(=O)Cc1cn[nH]c1)C2 C=CC(C(=O)NCCCC)CCN(C(C=CCNC)=O)CC.OC c1(C(=O)NCC2C(NC(c3cc(CCC)nn3C)=O)C2)ccc(C2CC2)nc1O c1(C(=O)OCC(=O)NC2CC(C(C)(C)C)CC2O)cc([N+](=O)[O-])cc([N+](=O)[O-])c1 c1(C(=O)NC(C)C(C)C(=O)Nc2ccccc2F)cc2cccn2cn1 C(=O)(C(C)C(F)F)N1C(CN(C(=O)Cc2cccc(O)c2)CC)CCC1 c1(C(N(C(c2ccccc2)C)C2CC2)=O)ccc(CCN)cc1 c1(C(=O)NCC2CCC(NC(c3ccc(O)nc3)=O)C2)nnc(O)nc1O C12CCC(CC1)CN(C)C2=O.CC(C)CC(=O)NC1CCN(c2ccncc2)C1 Cc1cc2sc(CNC(N3CCN(CC(N4CCCC4)C)CC3)=O)cc2s1 C1(S(N)(=O)=O)(C(=O)NCCCN2CCN(C(C(C)(C)N(C)C)=O)CC2)CCCC1 CC1(C)C(C)(C(=O)NCCC2(O)CCN(C(c3cn[nH]c3)=O)C2)C1(C)C N1(C(C2CCC(=O)NC2)=O)C2CCC1C(CNC(c1coc3c1COC3)=O)C2 C1(CC(=O)NC2CC(CNC(COC(C)(C)C(F)(F)F)=O)C2)CC(F)(F)C1(F)F N#Cc1cncc(CN2CC(F)CC(NC(c3cn4c(n3)CCC4)=O)C2)c1 C1(O)(CN(C(=O)CC2(CC#N)CC2)C)CN(C(=O)CCCC2CCC2)C1 c1(C(N2CCC(NC(C(F)(F)C3(COC)CCC3)=O)C2)=O)oc(Br)nc1C N#Cc1cncc(CN2CC(NC(c3cc(Cl)ncc3C(F)(F)F)=O)C(O)C2)c1 CC(C)(C)CCCC(=O)N1CC(CNC(=O)CCCc2ncco2)OC(C)(C)C1 N1(C(CCOC(C)=O)=O)CC2CC3CC2C1C3NC(=O)Cc1c(Cl)cccc1Cl Cn1nc(CNC(c2c(F)cncc2F)=O)c2c1CCN(C(c1cccs1)=O)C2 C(=O)(C1Cc2ccccc21)N1CC2N(C(c3cc(OC)c(O)cc3)=O)C(CC2)C1 Cc1c(C(N2CCOCC2C(=O)NC(C)CCC2CCCC2)=O)cccc1C#N c1(NC(c2cccc(C)c2I)=O)cc(S(C)(=O)=O)ccc1OCCN c1(CNC(COCCOC)=O)ccc(CN(C)C(C23CCC(CC2)C3)=O)cc1 C1(CNC(c2cc(OC)nn2C)=O)C(C)CCCN1C(=O)CN1CCNC(=O)C1 C(=O)(C1=CC(C)(C)C1)NCC=C(C(=O)NCC(CSC)(C)O)C c1(OC)ccccc1-n1nnc(C(=O)NC2COCC2NC(=O)CC2CC2)c1C C=CCC(C(=O)N1CCCC(OC2CC2)C1)NC(c1nscc1C)=O C(=O)(C1=NNC(=O)CC1)NCCCC(CCC)NC(c1nnc(O)cc1C)=O c1(C(=O)NC2COCCN(C(C3OCC(C)C3)=O)C2)cccc2c1C(=O)NC2 C(=O)(CCC(=O)NN(C)C)NCC(C(=O)NC(C1(O)CCC1)C)(F)C(C)C C(c1ccc(C2CC2)cc1)=CC(=O)NC1CC(NC(c2ccccc2C2CC2)=O)C1 C(CCS(C)=O)(C(=O)NC1(F)CCCN(C(C2CN(C(N)=O)C2)=O)C1)N(C)C c1(C(=O)NCC2N(C(C(C)S(C)(=O)=O)=O)CC=C2)c2ccccc2nn1C Cc1cc(CC(=O)NCC2C(C)CCN2C(c2ccsn2)=O)ccc1O N(C1CCOc2c(C)cccc21)c1c(C)c(N2CCC(CC#N)C2)ncn1 C1(C(=O)NCCc2nc[nH]n2)CC2CC2N1Cc1ccccc1I c1(CN(C(=O)C(F)NC2CC(Oc3ccccc3)C2)CC)cccnc1 c1(C(=O)NCC(CC)NC(C2CCN(C)C(=O)C2)=O)cccc2[nH]c(C)cc12 c1(OC)cccc2[nH]c(C(=O)NCC(C)(C)NC(=O)C(OC)OC)cc12 c1(CNC(c2cc(C(C)=O)cs2)=O)cc(NC(C2(CC#C)CCC2)=O)ccn1 C(C1CCCN1C(C1CCCCCC1)=O)=CC(N1CC(CC(C)(C)C)C1)=O C12(CC(=O)N(CCC(N)=O)CCCN)CCC1CCN2C(N)=O CN1CCC(C(=O)NCCC2(NC(c3ncsc3C(F)F)=O)CC2)C1 c1(C(N2CC3C(NC(C(n4ncc(C)c4)C)=O)C(C3)C2)=O)cc(C)c(C#N)cn1 C(=O)(C1=C(F)CN(C(=O)CC2C=CCCC2)CC1)N1C(C)(C(=O)OCC)CCC1 N1(Cc2c(C)noc2)CCC(NC(=O)C(=O)Nc2nn(C)c(Cl)c2Cl)C(O)C1 c1(OCCOC)cccc(C(=O)NCC2CC2CNC(c2ccc(Cl)n2C)=O)c1 C1(OC)CC(C(=O)NC2CCCC2CNC(=O)CCc2ncc[nH]2)CC1OC Cc1cnnc(O)c1C(=O)NCCCC(C)NC(C1CCC=CCC1)=O [N-]=[N+]=NC1CC2(C(=O)NC3CCNCC3)CC12 S(=O)(=O)(c1cc(F)cc(F)c1)N1CCC(CC(=O)Nc2ccnc(Br)c2)C1 c1(C(F)F)ncc(Br)c(NCC2CC3CC2CC3O)n1 N1(C(C(C(=O)OC)OC)=O)CCOC(C(N2CCSC(C)C2)=O)CC1 N1(C(c2cc(OC)n[nH]2)=O)CCC2(CC1)C(NC(=O)CCCC(F)F)CS2(=O)=O C(=O)(C1=CCCCCC1)N1CCC(C(C(=O)NC(C#C)CC(C)(C)C)C)CC1 c1(C(N2C3C(CNC(C(C(C)C)O)=O)C(C3)C2)=O)ccn2ccnc2n1 c1(OC)cncc(CNC(C2(CO)CN(C(c3cnn(C4CC4)c3)=O)C2)=O)c1 c1(CC(=O)NC(CNC(c2n(CC)ncn2)=O)CO)ccncc1Cl N1(C(=O)OC(C)(C)C)CCCCC12CCN(C(=O)CCc1ccc3[nH]ccc3c1)C2 C1(=CCNC(COCCCC)=O)CCN(C(C2(COC)CC(F)(F)C2)=O)CC1 Cc1ccc(C(=O)NC2CCC2CNC(c2n[nH]cc2C2CC2)=O)c(N)c1 Cn1nc(C(F)(F)F)cc1NC(=O)NC(c1ccccc1F)C(F)(F)F N1(C(CC2(C)CCN(C(=O)Cc3cscn3)C2)=O)CC2CCCCC2C1 c1(CC(CN(C(C(C)OC)=O)C(c2nccn2C)C)O)ccccc1 C1(CC(=O)N)CCCCC1(F)F.N1(C(C=NOC)=O)CCC(C2C(CC)C(C)(C)N2)C1 c1(CC(c2ccccc2Br)NC(=O)NC2CCCC2O)ccccc1Br CC1CCC(CNC(=O)CCCC2CCOCC2)CN1C(=O)CC1CSCCS1 c1(C(C(=O)NC2COC2)N(CCCC)C)occc(=O)c1OC CCC(C(=O)OC)C(=O)N(CCCNC(=O)CCC1(C)CC1)C(C)C CN1CC(C)(C)CC1C(=O)NC1C(C(=O)NCC2CCC=CCC2)C1(C)C N1(C(C(CCC)CNC(=O)C(C)(CC)CO)=O)CC2(CCC(O)CC2)C1 C(CO)(CCCCNC(c1c(C)cccc1Br)=O)NC(CCCC)=O C1(CC=C)(NC(C2CCC2(C)C)=O)CN(C(C2(Cl)CC2(C)C)=O)C1 c1(OC)cc(C(=O)NCC(C2CC2)NC(=O)CCC2CCCC2)ncn1 C(=O)(CCOCC1CCC1)NC(C(=O)N(CC#C)CC1CC1)C1(C)CC1 C1(N(C(C=CC)=O)CC)CCCN(C(c2c(C3CCCCC3)noc2C)=O)CC1 N1(CC(=O)N(CCN(C(Cc2c(C)non2)=O)C(C)C)C)CCCNC1=O C1(C(N2CCCC(NC(c3cnc(OCC)nc3)=O)C2)=O)CCc2nccn2C1 C1(C(C)C)CN(C(=O)CN=S(C)(C)=O)CCC1NC(C1(C2CC2)CCC1)=O CN1CC(C(=O)NC2CC(C)(NC(=O)COCc3nc[nH]n3)C2)CC1=O C(=O)(C(=O)N=S(C)(C)=O)N(C1CCN(C(=O)CN2C(=O)C(=O)N(C)C2=O)C1)CC N1(C(CC2CC(=O)C2)=O)CC2CC(C(N3CC4CC4(CO)C3)=O)C(C2)C1 c1(-n2cc(CNCCN)nn2)cccc2c1CN(S(C)(=O)=O)C2 C1(C2CCN(C(C3CCOC3C(C)C)=O)C2)(NC(c2c(CC)nn[nH]2)=O)CC1 c1(C(=O)Nc2cc(OC)cc(Br)n2)cc(-c2cnn3c2CCC3)c(C)cc1F c1(CN(C)C(C2C=CCCC2)=O)cccc(CNC(c2c[nH]ccc2=O)=O)c1 CCCC(C)(C)CC(=O)N1CCCC(C)C1CNC(=O)CCc1ccccc1O C(CC(C)(C)C)(C(=O)N(CC)CC)O.N(S(=O)(=O)NCc1ccccc1)(CC)C N1(C(C2(N)CC3(CCCC3)C2)=O)CCc2c(Cl)cc(Cl)cc2C1 C=C1CCC(C(=O)NC2CCCCC2CNC(c2cncnc2)=O)CC1 Nc1c(C(N2CCC2CN(C(=O)C(CC2CC2)CC2CC2)CC)=O)ccc(Cl)c1Cl C(=O)(C1=CCCCC1C)NCC1CCCC(NC(C(C)(C)N(C)C)=O)C1 C1(NC(c2n(C)ccn2)=O)CC2CCC(C1)N2C(=O)CC1CCC(=O)NC1=O C1(N2CC3C(NC(C(C)SCCCC)=O)C3C2)CCc2ccccc2NC1=O C=CCC(CC=C)C(=O)N1CC(C)(CNS(=O)(=O)CC2CCC2)C1 N1(C(C2(C)CCCCO2)=O)CCCC(C2CN(C(=O)CN3CCNC(=O)C3)C2)C1 C1(CNC(CCCC(=C)C)=O)CCC(C)(C)CN1C(c1ccnn1CCOC)=O C(=O)(CCCCCF)N1CCCC(NC(c2ccc(N3CCCC3)nc2)=O)C1 C1(NC(C(C=C)O)=O)CC2CC(NC(=O)CSc3cnn(C)c3)CC12 C(=O)(C1=C(Cl)CC1)N(CCC(C)NC(C1C(c2ccccc2)C1(F)F)=O)C c1(C(=O)NCCCN(C(C)C)C(C2C=CCCC2)=O)cc2nc(=O)ccn2[nH]1 N1(C(c2n[nH]c(C)c2Br)=O)CCCCC(NC(C2CC=CCC2)=O)C1 CCCC(C(=O)NCc1nc(C(=O)NC(C)C=CCOC)co1)OCC C=CCC(C(=O)NCC(C)(C)CC=C)NC(c1sc(C)nc1C)=O C1(COC)CN(C(=O)CC2CCCC2)CCN1C(=O)C(O)Cc1cnc[nH]1 C(=O)(CCCCC(F)F)N(C1CCN(C(=O)CC2COCC(C)(C)O2)C1)CCC c1(C(N2C(C(NOCC(CC)C)=O)CCC2C(C)C)=O)cc(C)c(N)cc1F C=CC(C)(O)C(=O)NC1CCC(N(C(=O)CCC2CC2C)C)CC1 c1(C(=O)NCC(c2ccc(F)cc2F)NC(C(CC)OC)=O)ccc(C#N)cn1 C(=O)(C(F)(F)C(F)(F)F)N(CC(C)(C)CNC(C1CCCC(=O)N1C)=O)C c1(C(=O)NC2(CNC(C(CC)C(C)O)=O)CCCCCC2)cc(C#N)ccc1N N1(C(=O)CC2CCC3CC23)CCC(n2cc(CCC3CCCO3)nn2)(CCO)C1 C1(C(=O)OC)(CC2CCN(C(CNC(=O)Cc3cccc(C)c3)=O)C2)CCC(O)CC1 Cc1ccsc1CCC(N1CCC(N(C)C(c2ccn(CCF)n2)=O)C1)=O c1(CC(C)N(C)C)nc(-c2ccc(C(F)(F)F)nc2)nn1C(C)C(F)(F)F C12(C(=O)NCc3c(C)nncc3)C(NC(c3cc(N)cc(F)c3)=O)C3CC1C2C3 c1(OCC)cc(C(F)(F)F)ccc1C(=O)N(CC(C)NC(C1CCC(=O)C1)=O)C N1(C(CC2CN(C(CC(CC)C3CC3)=O)CC2C)=O)CC2CCCC2C1 C1(C(N(C(CC)CNC(c2cc(CO)[nH]n2)=O)C)=O)CC(O)C1(C)C C1(O)(C(C)(C)NC(C(C)N(C)C)=O)CCN(C(c2ccc(C(N)=O)cn2)=O)CC1 Cc1ccc2c(c1)CC(C(=O)NC1CC3(CCCN(c4nnnn4C)C3)C1)O2 c1(-c2cc(C(N(C3CCN(C(C4(F)C(C)C4)=O)C3)C)=O)sn2)ccc(Cl)cc1 c1(C(=O)NCC(C)NC(c2cscc2F)=O)csc2c1CCC(C)(C)C2 c1(C(N2CCC(N(C(CCC(C)SC)=O)CCO)CC2)=O)n[nH]c2c1COC2 CC(C)(C)CCCC(=O)NCC#CCNC(=O)C(Cc1ccc(F)cc1)C1CC1 CC(C)(C)C#CC(=O)N1CC2CC1CN2C1CCCCN(CC(F)(F)F)C1=O C1(NC(CSC)=O)CC(C)(C(=O)NCCN(CC(F)F)CC)C1 C(C(C(C)(C)C)NC(=O)C(C(C)C)c1ccc(F)cc1)NC(CNC(C)=O)=O c1(CNC(C2(CNC(C(C)CC#N)=O)CCCO2)=O)cccc(F)c1O C1(NC(CC2ON=C(C)C2)=O)CC2(C1)CC(CNC(c1nc(O)c(C)s1)=O)C2 Cc1cccc(C(N2CCCCC2CNCc2ccc(Br)c(Br)c2)=O)c1C#N C12(C(=O)NCCC3CC(C(F)(F)F)CO3)CCC(C(F)F)(CC1)C2 c1(C(N2CC(CCNC(C3(CF)CCC3)=O)C2)=O)cc(O)ncn1 Cc1ncc(C(N2CCN(CCNC(=O)CC3CCC3)CC2)=O)n1C C1(SC)CCC(C)(CC(=O)NCC(CO)NC(=O)CC(C)N(C)C)CC1 C1(C(=O)O)COCCN1N1CCC2(CC1)OCCc1ccsc12 C1(NC(CCP(OC(C)(C)C)(C)=O)=O)CCCC2(CCC2)C1O c1(-c2cn(CCC(N3CCC(CN(C)C)C3)=O)nn2)cccc(CC(=O)O)c1 c1(OC)cccc(C(O)C(=O)NCC(C)CNC(c2c[nH]ccc2=N)=O)c1 C(=O)(CC(C)(C)C1CC1)N(C)CC1CC1(F)F.C12CC(C1)NC(=O)C2 C=C(C)CC(C(=O)N1CC(OC)C1)OCCC(=O)NCC(CC)C(C)C C1(C(CNC(CCCNC(C)=O)=O)C)CCN(C(C2(C)CC2C)=O)CC1 C(=O)(C1=CC2CCCC12)N1CCC(NC(=O)COCC2CCCC2)C(F)C1 CCS(=O)(=O)CC(=O)NC1CC2(C1)CC(C(N1CCOCCC1C(=O)OC)=O)C2 N1(C(C2C3CC4C(C3)C24)=O)C2CCC1CN(C(c1cccc(F)c1CC)=O)CC2 C(=O)(CCC(=O)NC1CC(F)(CNC(C2OC3CCC2C3)=O)C1)OC c1(C(=O)NC(CC#C)C(=O)NCCCn2cnnn2)cc2n(n1)CCO2 C(=O)(C(C(=O)N1CC(CNC(C2SCCCS2)=O)C1)OC)OC C(=O)(CCCC(C)(C)NC(=O)CCC(C)OC)NCC(CC)CC CC1CN(C(=O)CSc2nncn2C(C)(C)C)CC(C)C1NC(=O)CC1CSC1 Cc1cc(=O)n(C)cc1C(=O)N(C)CCN(C)C(C1(C)CC2(CCC2)C1)=O CC(C)CC(C)CC(=O)N1CCOC(C)(CNC(c2ccc3cccnn23)=O)C1 CC1(C(N2CC(NC(c3ccc(CO)cn3)=O)C(CO)C2)=O)CC2CCC1C2 Cc1c(F)cc(C(=O)NC2CCCN(C(C3CC(O)C3)=O)CC2F)cc1F c1(C(=O)NC(CC=C)CNC(=O)COCCCCCC)scc(Br)c1C c1(C(=O)NC(CNC(CCC#CC)=O)(C)C2CCC2)cc(C(N)=O)cc(C)c1 C(=O)(C1CCc2ccccc21)N1C(CNC(C=C(C)C(C)C)=O)CC2(CC2)C1 C1(C(N(C)CC2(NC(C=CSC)=O)CC2)=O)CCc2nncn2C1 CC1(C)OCCC1C(N1CC(NC(c2cc(Cl)cnn2)=O)C(O)C1)=O N1(C(C2CCC(NC(CC)=O)CC2)=O)CC2CC3CC2C1C3 c1(C(=O)N2C3CCN2C3)cc(C)on1.C(=O)(CCC=C(C)C)OC.S(C)(=O)(=O)N N1(C(=O)OCC)CCn2ncc(C(=O)Nc3ccoc3C(F)(F)F)c21 c1(N(C)CCC2CCCN(C(=O)OC(C)(C)C)C2)ccccc1S(C)(=O)=O c1(OC)ncccc1S(=O)(=O)N1CC2(CC(NC(c3cc(Br)c[nH]3)=O)C2)C1 c1(C(N(C(C)CNC(=O)CN2CCC2C)CC)=O)ccccc1-n1ccnn1 N1(C(C(C)OCC)=O)CCC2(CC1)C(NC(c1cc(C(F)F)no1)=O)CS2(=O)=O N1(C(=O)Nc2cccc(COC)c2)CC2(CC(Cc3nc(C(C)(C)C)n[nH]3)C2)C1 CC(CCCCN=c1cc(C(F)(F)F)nc[nH]1)NC(C1CCCSS1)=O c1(C(=O)NC2CC3CN(C(COC(CC)C)=O)CC32)nccc2occc12 CN1CCCC1(C)C(N1CCN(CC(N2CCC(c3ccc(F)cc3)C2)=O)CC1)=O c1(C(N2CC3CN(C(=O)CN4CCCCC4)CC32)=O)ccc([N+](=O)[O-])c(F)c1F c1(C(=O)NC(C2CN(C(c3coc(Br)n3)=O)CCO2)C)cc(O)nc(Cl)c1 N1(C(c2cc(NC)ns2)=O)CC2CC2(CNC(=O)CCc2cc(C)sc2C)C1 Cc1cc(Cl)cc(C(=O)NC2CN(C(C3CCCNS3(=O)=O)=O)CC2C)c1N c1(C(=O)NCCC(C)CCNC(C2(C)CCOCC2)=O)nncc2c1CCCC2 C(C)(CCC(C)(C)C)NC(C(CCC1CCC1)NC(c1c(C)nccc1)=O)=O C1(C(=O)NC(CC)CNC(c2onc(C)c2C)=O)CC(c2ccccc2F)=NO1 C1(CC)CCCN(C(C)=O)C1C(N1CCN(C2CCC3(COC)C2C3)C(C)C1)=O CC1c2ccccc2CC1OC(C1CCN(C2COC2)C1)=O c1(C(=O)NC(C(=O)N(c2cnccn2)C)=O)cccc(F)c1CN1CCOCC1 CC(C)(C)CCCC(=O)N1CCCC1CNC(C1CC12CCCC2)=O N1(C(=O)OC(C)(C)C)CC(n2cc(CC(C)N)nn2)CC1C(=O)O N1(C(c2cccs2)=O)CCN(C(C2(C3CCC3)CC2)=O)C2COCC12 C1(C)(CCNC(c2c(C)nns2)=O)CCN(C(C23CCCC2(C(N)=O)C3)=O)CC1 Oc1cc(Cl)c(-c2noc(-c3cc(Cl)ccc3OC(F)(F)F)n2)cc1Cl N1(C(c2ccc(O)cc2Cl)=O)CC(C2CCCN(C(=O)C(F)Br)C2)C1 N#Cc1ccc(CC(N)C(=O)NCc2ccc(Cl)c(Br)c2)c(Cl)c1 C1(CNC(C2(C)CC2(F)Cl)=O)CC2COCC2N1C(c1cc(Cl)ccc1Cl)=O c1(C(=O)OC)coc(C(N2CC(CCCCNC(=O)CNC=O)C2)=O)c1 c1(-c2nnc(CC(c3ccc(F)cc3)CC)o2)cccc(O)c1 C(=O)(CCCCCN)NCC1CCC(CNC(C=CC=CCC)=O)C1 C1(C(=O)NCCCO)(CNC(CC(C)F)=O)CC12CCC2 C=C=CC(C)C(=O)NCC1CCC1C(=O)NC(c1ccccc1)CF C(=O)(CCC(O)C(C)(C)C)NCC(C)N(C(=O)C=C1CCSCC1)C C(C(O)CO)(C1CCC1)C1(NC(=O)CC2CC2)CC1 CC(=O)CCN=C(NCCC1(C(=O)N(C)C(C)C)CCC1)N1CCC2(CCC2)C1 Cc1ncc(CNC(C23CC(NC(=O)Cn4cccn4)(C2)C3)=O)s1 C1(CCC(=O)NC2(CCC)CC2)CCCCN(C(=O)C(F)C(C)C)C1 c1(CN2C(CNC(C)=O)CCC2)ccc([N+](=O)[O-])cc1Cl.C1(c2cnc[nH]2)C(=O)N1 c1(C(=O)NC2(COC)CCN(C(C3COC(=O)O3)=O)C2)nnn2c1C(=O)NCC2 c1(CC(C)N(C)C(C2CCN(Cc3cnccn3)CC2)=O)cccc(F)c1 C12(C(=O)NC3C(C)(C)COC3=O)CCC(CN(C(=O)C=CC(F)(F)F)C1)C2 C12(CCC1)C(=O)NCC(=O)NCCN(CC)CC2.C(CO)OC N(C(=NCC#Cc1cnn(C)c1)N1CCCC(OC(C)(C)C)C1)C(CC)C c1(SC)ccc(OC)cc1.C(C(CCO)N(C)C)NC(CCN(C)C)=O N1(C(c2c(COC)cco2)=O)CC(OC)C(N)C1.C1(=O)C(C)N1.C(N)(=O)N c1(OC)ccc(C(N2CCCC(F)(CNC(c3ccccc3I)=O)C2)=O)cc1C C(=O)(C(F)CCC(C)C)NCC1CC(C(N(c2cccc(C#C)c2)C)=O)C1 CN1CC2C(C(N3CC=CC3C(=O)NCc3ncc(CO)[nH]3)=O)C2C1 C(=O)(C1(C)CCn2c(C)nnc21)NCC1C(NC(C=C(C)C(F)F)=O)CCCC1 N1(C(c2c(C)n[nH]c2C)C2CC2)C(=O)NC(CC(N2CCOCC2)=O)C1=O c1(C(N(CC(C)OC)CC)=O)cnn(CCCC2CN(C(=O)C3CC3)C2)c1 N1(C(c2cc(-c3ccccc3)[nH]n2)=O)CCC2CN(C(C3CCCC3)=O)C2C1 c1(CS(=O)(=O)NC2CCCC2)cccc(C)c1.CC(C(=O)NCC1CCCO1)=C1CC1 N1(C(CC2C(C)(C)C2)=O)CC(NC(=O)CCCOCCc2ccccc2)C(O)C1 N1(CC(C)C)CCC(C(N2CC=CC2CNC(=O)Cc2ccon2)=O)CC1 C12(NC(CCC#C)=O)CCOCC1CN(C(c1ccsc1SC)=O)C2 c1(C(N2CC(NC(=O)CCc3cc(Cl)no3)C2)=O)cc2c(F)ccc(F)c2[nH]1 C1(C(=O)NC)CN(C(CC2(C)CC2)C(=O)NC(C)COC)CC12CC2 CCCCCCCCC(CC)NC(c1cnn2c1NCCC2)=O C1(NC(COC(C)C)=O)CCC(CNC(c2cc(C3CCC3)[nH]n2)=O)C1 C1(N(C)C(c2cc(O)nn2C)=O)CC2CC1N(C(C1(C)C=CCCC1)=O)C2 CCC(C)(C)C(C)CC(=O)N(CCCOCCNC(C1CCOC1C(C)C)=O)C C1(F)(CNC(c2cc(COC)no2)=O)CCC(NC(C2CCC(C)(C)O2)=O)C1 Cc1cc(C)c(CC(=O)N(C2CCN(C(c3ccc(C(C)C)nc3)=O)CC2)C)s1 N(C1c2ccccc2C2CC12)C(=O)Cn1cc(CC(CO)C2CC2)nn1 O=C(C1=CS(=O)(=O)CCC1)NCC1CN(C(C2(F)CCOC2)=O)C2COCC2O1 c1(NC(=O)CC2CC(NCc3ccc(F)c(I)c3)C2)cc2ccccc2cc1O c1(OC)cccc(C(c2nnnn2C)NCc2cnc(C3CCC3)s2)c1O c1(NCC2C(C)CCCN2C(=O)CC2CCOC2)ncc([N+](=O)[O-])c(=N)[nH]1 c1(CNC(c2n(CCC)nnn2)(C2CCCO2)C)nc(C)c(C)o1 c1(CC)cc(C(N2CC3(C(=O)NC4CCN(C(C)=O)C4)CC2CO3)=O)cc(Cl)n1 N(C1CN(C(C2(F)CCC2)=O)CCc2ccccc21)C(=O)CCc1ncccn1 N1(C(CCCC(C)O)=O)CC2CCCC(NC(=O)C(c3ccccn3)C)C2C1 N1(C(C2C(C)(C)CCO2)=O)CC=C(CCNC(c2cnco2)=O)CC1 c1(CC)onc(C)c1C(=O)NCCOC1CN(C(=O)C(C)O)C1 N1(C(c2noc(CC)c2C)=O)CCC(O)(CNC(C2NC(=O)C3CC23)=O)CC1 C(=O)(CCCCCCCSC)NC1C(C)CN(C(C2CCc3cnnn3C2)=O)C1 O=C(C#CC1CCOC1)NCC1CN(C(=O)Cc2cccc(C3CC3)c2)C1 c1(C(=O)NC2C(NC(c3n(C)ccn3)=O)CC(F)(F)C2)ccc2c(c1)ncn2C c1(C(C)C)nc(=NCC2CCN(C(=O)C(O)Cc3ccccc3)C2)s[nH]1 C1(C(N2CCC2C(=O)N(c2ccccc2)Cc2cscc2Br)=O)SC2C=CC1CC2 n1(CCC)nccc1C(N1CC(O)(C(C)NC(=O)CSc2ccccc2)C1)=O C1(C(=O)Nc2cnc(CC)[nH]2)(NC(C2CCCCC2=C)=O)CCN(C)C1 Cc1cccc(CCC(=O)NC2CC2CNC(c2cscc2C)=O)c1 c1(C(N2CC(CNC(CC(C)CC(C)(C)C)=O)C2)=O)nn(C)c2ccc(F)cc12 N1(C(c2cc(CC)[nH]n2)=O)CCCCC1C1CCCN1C(=O)CCC(=O)NC c1(CNCC2C(C(N3CCCC(C#C)C3)=O)CCO2)cccc2ccoc12 c1(CN(C)C(c2cccc(N)n2)=O)nc(C(F)(F)F)n2c1CCCC2 c1(OC)ncnc(Cl)c1NC(C1CCN(c2ncnc(Cl)c2F)CC1O)=O c1(CCCC(=O)NC2CC2CNC(=O)C(F)=CCCF)cccc(OC(F)(F)F)c1 c1(C(=O)NCC(=C2CN(C(CCOC)=O)C2)F)ccncc1C(F)(F)F CC1CN(C(C2CCC3(CCC3)CO2)=O)CCCN1C(=O)CCC(N)=O C(=O)(CC(CC)CCC)NC(CCNC(c1cn(CCC=C)nn1)=O)(C)C N1(C(C2COCCN(C(C3C4CCC(F)(F)C34)=O)C2)=O)CCC2(CC1)CC(O)C2 c1(OC)ccccc1C(O)CNC(=O)C(N1CCOC(CS)C1)=O C1(C(=O)NCC(C(=O)NCc2c(CC)con2)OC)CCCCCCC1 c1(COCC)cc(C(N2CCCC(C(C)C(=O)OC)C2)=O)sc1Br Cc1ocnc1CC(=O)NCC(C)(O)CNC(c1cc(C2(O)COC2)on1)=O c1(C(=O)NCC2(C)OCCN(C(C(C)OCC)=O)C2)[nH]nc2c(=O)n(C)cnc12 CC1CN(C(c2c[nH]c(=N)o2)=O)CCC1N(C)C(c1ccccc1Cl)=O c1(C(N2CC(O)CC(NC(C(C(C)(C)O)F)=O)C2)=O)cccc(S(N)(=O)=O)c1 C=CC(CCC)CC(=O)N(C)CC1Cc2ccccc2O1 C1(CNC(CCOC)=O)CN2CCCCC2CN1C(c1n[nH]c2c1CC1CC21)=O Cc1cc(CC(=O)N(CCC2CCCCCC2)CCO)ccc1Cl c1(CC(N2C(CN(C(C(C)OCC#C)=O)C)COCC2)=O)ccc2ocnc2c1 Cc1[nH]cc(C(=O)NC2CC3CC(NC(c4cc(Cl)cn4C)=O)CC23)c(=O)c1Cl CC12CCC1CN(C(C1(NC(=O)CC3CC4(CC4)C3)CCCC1)=O)C2 c1(OC(C)C)cccnc1C(=O)NCC1CC(O)CN1C(C1CC1CF)=O C(CC(O)C(=O)NC1CC(CO)N(C(C2CCC(C(N)=O)CC2)=O)C1)N(C)C C1(CC(=O)NCCSC(C)C)CCCCN1C(C1(C)CCOC1C)=O C1(NC(C2C(C)CN2C(c2scnc2Cl)=O)=O)CC2(CCCCC2)C1 N1(C(CCC2C(C)=NOC2=O)=O)CC2CCC1C(NC(c1cscn1)=O)C2 N1(C(C(C(=O)OCC)OC)=O)CCN(C)CC1C(=O)NCC(C)(CO)OC c1(OC)ncc(C(C(=O)NCC2CCOCC2)N2CCC2C(C)C)cc1Cl N1(C(=O)Cc2cc(Cl)cc(Cl)c2)CC2OCOC2C1 C(CC(C(=O)NCc1ccc(C#N)s1)NC(=O)C(F)C1CCC1)OCC c1(N(C2CCCNC2)C(=O)CN2C(=O)CCC2=O)nc2ccccc2o1 Cc1nc2cc(C(N3CCOCC(CNC(C4CCC4(F)F)=O)C3)=O)cnc2[nH]1 C1(C(C)NC(=O)CC2(C)CC(C(=O)O)C2)CCC(NC(=O)Cn2nnc(=O)[nH]2)CC1 C1(CNC(c2cccc(N)c2F)=O)CCn2cncc2C1 CCC(CNC(c1cnc(NC)cn1)=O)(CC)NC(=O)C(C)C1C(CC(C)C)C1 c1(C(=O)NC2(CCNC(c3ccc(CO)nc3)=O)CCC2)ccc(O)c(Cl)c1 N1(C(C=CC=CC)=O)CC(NC(=O)CCC2CCC(O)CC2)CC(F)C1 CCC(CCCC(=O)N(C)C)NC(=O)CSC.N1CCN(C(=O)C(O)CSC)CC1 C(=O)(CC(C)C(F)(F)F)N(CCOC)CCNC(=O)COCCc1ncnn1C c1(CCCC(=O)N(CC(C)(C)NC(=O)CCF)C)ccc(F)cc1 N1(CCCCc2c(C)ccs2)CCN(C(=O)Cc2cnccn2)CC1C1CC1 c1(C(=O)NCC(C(C)(C)F)(C)F)ccc(S(=O)(=O)N2CCCC2)cc1 C1(CC=C)(NC(c2ncc(C)o2)=O)CCN(C(=O)CN(c2ccncc2)C)C1 C1(CN(C(c2cc(CC)on2)=O)C)CCCC(NC(c2cc3n(n2)CCC3)=O)C1 C=CCC(C(=O)N1CCC(C)(Cn2cc(C(O)CC)nn2)CC1)C(C)C C1(NC(C=CC=CC)=O)C(C)CN(C(c2cc(CC(=O)OCC)on2)=O)CC1C C(=O)(N=c1[nH][nH]c2cc(Cl)ccc12)C12CN(C(C(CC)C)=O)C(C1)CO2 C1(CC(N2CCC(C)(NC(C3(CC)CCOCC3)=O)C2)=O)CCCC(C)(C)O1 C1(C(=O)NC(CN(C(=O)CCSc2ccccc2)CC)C)Cc2nccn2C1 C(=O)(C1=C(Cl)CCOC1)N1CC(C(C)NC(c2ccc(-c3ccccn3)o2)=O)C1 C1(C)(CC)CCN(C(C2(CCOC)C=CCN2C(C2CC2COC)=O)=O)C1 CCCC(CCCNC(c1scc(C)c1Cl)=O)NC(C1CCC(C(F)F)CC1)=O c1(C(=O)NC2CC(C)(COC)N(C(C3CC(=O)N3)=O)C2)cc(C)c(F)cc1F CCC(CC(=O)NCC1CN(C(C23CC(F)(C2)C3)=O)CCO1)SC C1(CC)C(=O)NCCN1C(C1CCN(C(=O)C=CC=C(C)C)CC1O)=O N1(C(C=C(C)C2CCCCC2)=O)CC2CN(C(C3(C)CCCOC3)=O)CCC12 N1(C(C=CC=C=CC)=O)CCOC2CN(C(=O)CC3CCn4cncc4C3)CC12 C1(CNC(c2cc(C)no2)=O)CCC2CN(C(c3cc4c(ncn4C)s3)=O)CC12 C1(O)(CN(C(COCCC(C)C)=O)C)CCCN(C(C2CC(C3CC3)C2)=O)C1 n1(CC(=O)NC2COCCC2NC(c2ccc(CO)cn2)=O)cnc([N+](=O)[O-])c1 N#CC1(CC(N2CCOC(CNC(C3CCC4CC34)=O)C2)=O)CCCCC1 N1(C(C=CC(C)C)=O)CCN(C(=O)C=C2CCC2)C2CCC12 C1(NC(C2CN(C(C)=O)C2)=O)CCC12CN(C(C1COCCN1C=O)=O)C2 C1(C(N2CCC(CCC(N3CCC(N(C)CC)C3)=O)C2)=O)CCC(=O)N1C Cc1nc(CCCC(=O)N2CC(O)(CNC(=O)CCNC(C3CC3Br)=O)C2)cs1 CN(C1CS(=O)(=O)c2ccccc21)CC(=O)Nc1ccc2c(c1)OCCO2 C1(CC)OCCC1C(=O)NC(CNC(=O)C=Cc1cocn1)C1CCC1 N(C)(C1CCCc2cccnc21)CCc1ccc(OC)nc1 C1(NC(C)CS(N)(=O)=O)(CO)C2CCCNC2C1(C)C CC1CN(C(C2CCCC2O)=O)CCCN1C(=O)CCCCC(N)=O c1(C(=O)NCC(C2N(C(C3CC(C(C)=O)C3)=O)CCC2)(C)C)c(C)noc1C(C)C N1(C(CC2(COC)CC2)=O)CC2CC(CNC(C3CSCCS3)=O)CC1C2 c1(C(N2CCC(N(C(CC=CC=C)=O)C)C(C)C2)=O)cc2c(ccn2C)[nH]1 c1(C(=O)NCCCN(C)C(C2CCC(C)(O)CC2)=O)ccc2c(c1)CCO2 c1(C(N(CC(CC)NC(C2CC3C(C2)C3(F)F)=O)C)=O)c[nH]c2nc(F)ccc12 N1(C(C2CCCO2)=O)CCNCC1.CC1CCN1CCC(=O)N1CCCC1 C(C)(CNC(=O)CCc1ccc(N)cn1)(C(C)C)NC(C(C)=C1CCCC1)=O N1(C(c2cc(COC)no2)=O)CCC(NC(C2CC(C)CO2)=O)C(C)(C)C1 C(=O)(C(C)(C)C(=O)OC)N(CC=CC(=O)NCC1N(CC)CC1)C C(=O)(C1=CCCC1C)NCCSCC(=O)N(CCCO)C c1(C(N(CCNC(=O)C=C(CC)c2ccccc2)CC)=O)cccc([N+](=O)[O-])c1Cl C1(NC(c2csc(Cl)c2)=O)CC2CN(C(C3CCOC3)=O)CC12 c1(NC2CC(NC(C3CC3C3CCCC3)=O)C2)ncccc1[N+](=O)[O-] c1(C(N(C)CCOCCCNC(=O)CN(C)C2CC2)=O)cnc[nH]1 N1(C(COC(=O)CO)=O)CCC(C2CC2)C1CNC(C1COCS1)=O c1(C(N)=O)cnc(C(=O)Nc2cccc(NC(=O)C(C)n3cnnn3)c2)c(Cl)c1 C#Cc1cncc(C(=O)NCC(C(=O)NC2CC2CC(C)C)OC)c1 c1(C(=O)NC2CC2CNC(c2cn(C3CCOCC3)nn2)=O)cnc(O)c(Cl)c1 C1(C)(C(=O)NC2C(C)CCN(Cc3cnn(C)c3)C2)CC2(C1)CC(F)(F)C2 c1(C(=O)NC(c2cc(Cc3ccc(F)cc3)no2)C)ccc([N+](=O)[O-])cc1 C(C)(C)(C(=O)NC1CC(CCNC(C2CCCN2CC)=O)C1)OCC c1(OC)nccc(C(=O)NCC(C)C(=O)NCC(O)C(C)O)n1 N1(C(c2ccc(CNC(C(C3CCC3)OC)=O)o2)=O)Cc2cccc(C)c2C1 c1(SCCC)ccc(CNC(C2C(CNC(=O)CC3CCCN3C)C2)=O)cc1 c1(Cn2cc(CCC)nn2)cc(C)ccc1C(=O)NCc1cccc(Br)c1 c1(CCn2cncc2)ccc(-c2ccc(-c3ccc(C=O)o3)cc2F)cc1C.CO C(=O)(C(C(C)NC(c1ccnc(C)c1C)=O)C(C)C)NC1(C)CC(C(=O)OC)C1 N1(C(C(N)=O)=O)CCOC2CN(C(=O)CCCc3cccnc3)CC12 c1(OC)ccc(F)c(CN2CC3CCN(c4ncc5c(n4)CCC5)C3C2)c1F Cc1cc(C)c(C(N2CC3CC3(NC(=O)CCn3cnnn3)C2)=O)c(=O)o1 C1(C(=O)NC(CCC)CCC)CCCCCCN1C(=O)C=C(C)C(C)C CC1(C)C(C(N2CCCC(C3CCCCN3C(C3COC(=O)C3)=O)C2)=O)C1(F)F N1(C(Cc2c(C)n[nH]c2C)=O)CC(C)(C)OCC1CNC(c1cnsc1)=O c1(CC)ccc(C(=O)NCCC(C)NC(c2cnn(C3CCCC3)c2)=O)[nH]1 c1(C(=O)NCCCCCNC(c2cc(C(C)=O)no2)=O)nc(C)ccc1O N1(C(C2(C)CCN(C)C2=O)=O)CCC2CN(C(=O)CC3COCCO3)C2C1 c1(C(=O)NCC2(OC)CN(C(CCCCC)=O)C2)ccc2nc3n(c2c1)CCC3 S(=O)(=O)(c1ccc(N(C)CC2CCOC2)nc1)N(C1CC(C)OC(C)C1)C c1(CC(=O)NC2(COC)CCNCC2)ccc2c(Cl)ccnc2c1 C1(NC(C(C)SCC)=O)CCC(C(=O)NCc2sccc2-c2ccccc2)CC1 C1(COC)CCCN1C(c1ccc(C(=O)Nc2ccccn2)o1)C(=O)NCCC#N c1(C(N2CCC(CNC(C3CCC(F)(F)C3)=O)C2)=O)cc(Br)ccc1Cl N1(N2C(N(C(c3ccn(C)n3)=O)CC)CC2)CCOC(CC(N)=O)C1.C(=O)CSCC N1(C(C2(C)CC2)=O)CC(C2CC2)(C(=O)NCC2CC2(Cl)Cl)C1 c1(NC2(C(C)(C)O)CN(C(COc3cc(C)on3)=O)C2)ccc(C#N)nn1 C1(C)(CNC(c2ncc(C)cn2)c2cccs2)CCCC(F)(F)C1 C(=O)(C#CC1CCCOC1)N1C(CNC(CCc2ccc(SC)cc2)=O)CCC1 N1(CC)CCN(CC(=O)N(C(C)CCNC(c2cncs2)=O)C)CC1 CCCCCCCCC(C)C(=O)N1CCN(C(c2cc[nH]c3nccc2-3)=O)CC1 c1(OC)c(C(C(F)(F)F)NC(=O)OCC2CCCC2C)cnn1C c1(C(N(C2CCC(NC(=O)C3=CSCS3)C2)C)=O)cc(Cl)ccc1Cl C1(C(=O)N(CC(c2ccccc2)N(C)C)C)CC12CCN(CCCC(F)(F)F)CC2 CC(C)CC(C(=O)N1CCCC(C(=O)Nc2cnccc2C2CC2)CC1)C(C)C C1(C(=O)NC(CCNC(C(CC)CC(C)C)=O)(C)C)Cc2ccccc2C1(C)C c1(CC(=O)NCC(C)CN(C(=O)C2=CCSC2)C)c(Cl)cccc1Br C(=O)(C1c2ccccc2OCC1(C)C)N1CCC(N(C(c2coc(C)n2)=O)CC)C1 C1(CNC(CN(C2CC2)CC)=O)CCCCC1NC(c1oncc1CC)=O Cc1sc(O)nc1C(=O)NCCN(C(=O)C(c1ccccc1Cl)C)C C(=O)(C(CC)(CC)CO)NC1C(CC)CN(C(c2cc(F)cnc2Cl)=O)CC1 CC(C)(CC(F)C(=O)NC1CCCC(C(N)=O)C1)NC(=O)CC=Cc1ccccc1 Cc1ncsc1C=CC(=O)NCC1(C(=O)NCC2CC(C)CO2)CC1 N1(C(C2(C)N(Cc3c(C)cc(Cl)nc3)CC2)=O)CC23CCCCC2(C1)C(=O)NC3=O CCC(CC(=O)N(CCC(=O)OC)C)N(C)C(C1CCCN1CC)=O N1(C(c2c(OC)nc(C)cc2)=O)CC2OCCN(C(=O)CC(C)SC)C2C1 CC1(C)CN(C(C23CCC(O)C2CC3)=O)CCC1NC(c1cnc(C2CC2)o1)=O c1(C(=O)NCC(=O)NC2(CN(C(C3CC(C)C3)=O)C)CC2)ccc(N)cc1 C1(CN(C)C(c2ccnn2C2CCCC2)=O)CCN(C(=O)Cc2cnn(C)c2)C1 C12(C(=O)NCC3(OC)CN(C(c4cc(Br)co4)=O)C3)CCC(CC1)C2 C1(CNC(C2CN(C)C2)=O)CN(C(c2ccc(-c3cccnc3)o2)=O)CC1O CC(CC(C)(F)F)C(=O)N1CC2(CCCC2NC(c2ccc(N)c(F)n2)=O)C1 N1(C(CC(=O)NCC#C)=O)CC(NC(=O)CC2CCSCC2)CC12CCC2 c1(N2CC=CC(Nc3nc(C)[nH]n3)C2)ncnc2c1ncn2C N1(C(CC2CC(=O)OC2)=O)CC2(C1)CN(C(=O)CC1CCCCC13CC3)C2 CC1(C)OCCC1CC(=O)NCC1C2CN(C(=O)CC3CCCC3O)CC12 c1(C(N(C2CCCN(C(=O)C3=CCCS3)C2)CC2CC2)=O)ccnc2[nH]ncc12 C=CCCC(C(=O)NCCC1CCCC1(C)C)NC(C12CC(CO)(C1)C2)=O c1(C(=O)NC(C2C(C(=O)NCCC(C)(C)OC)C2)C)cc(C)n(C)c1 CC(C)C(CCN(C)C(C1CCCOC1)=O)NC(=O)CCCc1cnn[nH]1 CC1CC(C(=O)NCC2CCCOC2)CN(C(C2(CC3CC3)CC2)=O)C1 N1(C(C2N(C(=O)CCCCC#N)CCN(C)C2)=O)CCCCC(C)(F)C1 Cc1cn2c(n1)CC(C(=O)NC1CCC(CNC(C3OCCC3C(C)C)=O)C1)C2 Cn1ccc2c(C(=O)NC3CC3C(=O)Nc3nccc(Cl)c3Cl)cccc12 Nc1cc(C(=O)NCC(C2CCCC2)NC(C2C3COCC23)=O)cc(Cl)n1 C1(NC(C(C=C)O)=O)CC2CCC1CN2C(=O)C(C)(F)c1ccon1 c1(C(N2CC(NC(c3ccn(C)c3)=O)C(C#N)C2)=O)ccc(C#N)c(F)c1 C1(C#N)(OC)CC(C(=O)NC(CNC(=O)CN2C(=O)CNC2=O)C(C)(C)C)C1 c1(C2(C(=O)NC3C(C(=O)Nc4cccc(F)n4)CCCC3)CC2)ccc(F)c(Br)c1 C(=O)(CCC=CBr)NC(C)C(C)(C)NC(c1cnn(C)c1N)=O C1(NC(C(P(C)(C)=O)O)=O)CCN(C(c2ccc(C(F)(F)F)o2)=O)CC12CCC2 N1(C(=O)Nc2ccc(F)cc2)CCN(CCNC=O)C(c2ncc[nH]2)C1 N1(C(c2c(C)nc[nH]2)=O)CC2(CC(CNC(c3ccc(O)c(N)n3)=O)C2)C1 c1(C(=O)NC(CF)CF)ccc(SCCc2ccco2)cc1 N1(C(c2n(CCC)ncc2)=O)CC(NC(=O)Cn2nnnc2C)CC(O)C1 C(CC(COC)(c1nnnn1C1CCOCC1)NCC1CNC(=O)O1)OC C1(NC(C(COC)C)=O)CCCCC1CN(C(=O)CCC1CCCC1)C O=C(C1=C(F)CN(C(C2CC3CCC3C2)=O)CC1)NCC12CCCC(CO1)C2 N1(C2CC3(CN(C(C(CN)c4ccccc4)=O)C3)C2)CC2CC(F)CC2C1 Cc1cc2c(cc1C)OC(C(N1CCn3c(-c4ncnn4CCF)nnc3C1)=O)C2 CC1=C(C(=O)N(C)CC2COCCN2C(=O)C=Cc2cccc(Cl)c2)CCC1 C1(NC(=O)Cc2nc[nH]n2)CCN(C(=O)COCc2ccc(F)cc2)CC1 C(=O)(CCN=c1[nH]ccs1)NC1CCC(CCNC(CCCC(C)=O)=O)C1 CC(C)CC(O)CC(=O)NCC1CN(C(c2cc(C#N)c[nH]2)=O)CCN1C CC1(C)CC(NC(C2CC23CCN(C(c2c[nH][nH]c2=N)=O)C3)=O)C(C)(C)O1 N1(C(CC(C)C2CC2)=O)CC2CCC1C(CNC(c1cn3cnnc3cn1)=O)C2 CC(=Cn1ccnn1)C(=O)NC1CC2CC1N(C(=O)CC1CCCN1C(C)C)C2 N1(C2C(C)C2)CCN(C(=NCC2CCCCC2)NCC2CCC(F)(F)CO2)CC1 C(=O)(CCS(C)(=O)=O)NCCCN(C(c1noc(-c2ccccc2Cl)n1)=O)CC C1(NC(=O)Cn2ncccc2=O)CC2CC1CN(C(=O)C=CC1CCCCC1)C2 N1(C(C(CC)(C)C#N)=O)CCC2(CC1)CC(NC(C1(C)CCC(C)CC1)=O)C2 c1(COC)cc(C(=O)NCC2C(C)CCN2C(c2cc[nH]c2C)=O)c(C)o1 C=CC1CN(C(=O)CN2CCCS2(=O)=O)CC1NC(=O)C(=O)N(C)C c1(C(=O)NC(C)CN(C(=O)CCC2CCOC2)C)c(Br)c2ccccc2n1C C(=O)(C(C)(C)CCC(=O)N(CC(O)CN(C)C(c1ccc(CO)nc1)=O)C)OC N1(C(CCCCCOC)=O)CCC(C)(C)C(CNC(=O)CC(C)C(F)(F)F)C1 Cc1cc(C(N2CCC(NC(=O)CC(O)C(C)C)C(O)C2)=O)c(F)c(F)c1 C(=O)(C1=CNC2=NCCCN12)N(CCCNC(c1ccn(CCC)n1)=O)C(C)C CC(C)C(O)CC(=O)NC1CC1CNC(=O)CCC1CCC(C)O1 c1(OC)ccc(OCc2cn(CCNC(c3cn(C(C)C)nn3)=O)nn2)cc1 C1(CC)OCCCC1C(=O)NC1CN(C(c2cnns2)=O)C1 N1(C(C2CCN(C)CC2)=O)CC=C(CC(=O)Nc2cncc([N+](=O)[O-])c2)CC1 c1(C(=O)NCC(=O)NCCCCNC(CC2(C)CC2)=O)cn(C(C)(C)C)nn1 CCC(C)(C(=O)N1C2CCC1CC(CNC(c1c(Br)nnn1C)=O)C2)C(N)=O CC1(C)NC(=O)CC1C(=O)NCC(C)(O)CNC(=O)CCc1ccon1 C(=O)(CCC(=O)N1CC(F)CC1C(=O)NCCOC(CC)CC)NCC O=C(CCC(F)(F)C(F)F)NC1CCCC12CN(C(c1n[nH]cc1Cl)=O)C2 n1(CC(=O)NC2CN(C(C3CCCC3F)=O)C2)cnnc1O C1(CC(C(=O)NCC(F)F)N(C2CCCC2)CC)CCCC(C)(C)O1 CC(CSCc1ccccc1)C(=O)N1CCCC1CNC(C1CC(Cl)(Cl)C1)=O N1(C(CN2CC(C)(NC(CC)=O)C2)=O)CCC(C)(C(F)(F)F)C1 N1(C(C=CCN(C)C)=O)CCCC(CN(C)C(C2CCCC(=O)N2)=O)C1 C1(C(=O)NC2C(NC(C3CC4(CCOC4)C3)=O)CCC2)CCCC(F)(F)CC1 C12CC13CCN(C3)C2=O.c1(COC)cccc(-c2ccc(CC#N)cc2)c1 C#Cc1cccc(C(=O)NC(C)CN(C)C(C2CCN(C)C2)=O)c1F c1(CN(CC(F)(F)F)C(c2c(C(C)C)csc2)=O)ccnc(C(=O)O)c1 C(C)(C)(CC(=O)NCCCCCn1cc(C(C(C)C)NS(N)(=O)=O)nn1)SC C1(C(=O)NC(C2(O)CN(C(=O)CCC3CC3)C2)C)OCCOC1(C)C c1(C(=O)NCC2CN(C(c3nncc(OC)c3)=O)C2)ccc2nnc(S)n2c1 C(=O)(C(C(C)(C)C)NC(c1csc(F)c1)=O)NC1C(C=C)OCC1 N1(C(c2n[nH]c(O)n2)=O)CCC2CCN(C(C3CCC(=C(F)F)CC3)=O)CC2C1 C(=O)(CCCCCCN=[N+]=[N-])NCCCCCCN(C)C(c1ccc(CO)o1)=O C1(C)(NS(C2(C(=O)OCC)CC2)(=O)=O)CCN(c2ccc(F)cc2)CC1 N1(C(C2(CCC)CC(=O)C2)=O)CC2(C(=O)NC(c3ccnn3C)C)CCC1CC2 C(=O)(C1=CCC(F)(F)CC1)N1CCN(C(CN(C(C2C(C)(CC)C2)=O)C)=O)CC1 C1(C(=O)OCC)(NC(=O)CCc2ccccc2F)CC=CCC1.C1(NC=O)CC1 c1(C(N2CC3CCC2CN3C(C2CC3CC2C2CC32)=O)=O)cc2n(n1)CCCC2=O CC1COC(C)(C)CN1C(C1CN(C(c2c[nH]c(=NC)s2)=O)CC1(C)C)=O S(=O)(=O)(c1ccc(N2CCCC(CC3CC3)C2)nc1)NCCc1cn(CC)nc1 C12(C(=O)NC(C)CN(C)C(c3cnc(N)c(Cl)c3)=O)CCCCC1NC(=O)C2 C1(C(=O)NCCC2CCN(C(C3CCN(CCF)CC3)=O)C2)CCCC1C1CC1 c1(NC(C2CCCN(c3snc(C)n3)CC2)=O)cc(=O)n(C)c(O)n1 C(=O)(C1=C(C)OCCS1)N(CCNC(=O)COc1cc(C)ccc1F)CC C1(C2(O)CCC2)(C(N2CCC(C(C)NC(C3C(=C)CC3)=O)CC2)=O)CC1 C1(NC(C2CC(SC)C2)=O)CCN(C(C2CCC(N(C)C)CC2)=O)C12CC2 n1(CC(=O)NCC(CC(C)C)NC(=O)C(C)(F)F)cc(F)ccc1=O C1(C(=O)Nc2cc(OCC)no2)(NC(=O)C(C)C(F)F)CCCCC1 N1(C(C(=O)Nc2cccc(C)n2)=O)CCc2cc(F)c(F)cc21 c1(CC)c(C(=O)NC(C2CCCCN2C(=O)CSC2CC2)C)ccn1C C1(OC)CCCC(C(=O)NCC2CCCN2C(=O)C(F)F)C1 N1(C(CC(C)OC)=O)C2CCC1(CNC(C1CCCCS1)=O)CC2 C1(CC)CCCN(C(C2CC(N(C)C(C3(C#N)CC3)=O)C2)=O)CC1 C1(CN(C)C(C2(CCF)CCC2)=O)CN(C(C2CCC(O)C2)=O)CCO1 CC1(C)CN(C(=O)C(O)C2CCC2)CC1NC(=O)CCc1cncnc1O C#CC1(C(=O)NCC2(C)CN(C(C3CCCCN3C)=O)CC2C)CCCCC1 C1(C(=O)NC2C(COC)C2)CC2CCC1CN(C(c1c(OC)ccnc1F)=O)C2 N1(C(c2c(CC)cc(Br)cc2)=O)CCC2CCN(C(=O)C3=CCOC3)CC12 CC1C(NC(c2cc(Cl)sc2Cl)=O)CCN1C(C1CC1c1ccccc1)=O N1(C(C2N(CC)CCC2)=O)CC(NC(=O)C=CC(C)C)CC(F)C1 C(=O)(C1c2c[nH]nc2CN1C(=O)CCCC1CC1)NC1CN(C)C(=O)C1 c1(N2CCC(NC(c3ccc(CC4CC4)cc3)=O)CC2)ccc([N+](=O)[O-])cc1Br CON1CCC(CC(N2CC3(CCN3C(=O)C=C(C3CC3)C3CC3)C2)=O)CC1 S(=O)(=O)(c1cccnc1NCC1COC(C)(C)CO1)NC(c1n(C)cnc1)(C)C C1(CCCC)CCCC(NC(C2(c3cccc(C(=O)O)c3)CC2)=O)CC1 C(=O)(C(C)(C)CC(=O)N1CCOCC1CN(C)C(c1nc(Cl)cs1)=O)OC N1(C(CSC)=O)CC2(C1)CN(c1ccc(OC(F)F)c(OC(C)C)c1)CCC2(F)F c1(C(=O)NC(C)C(CO)NC(c2cnn(C)c2Cl)=O)csc2ccc(F)cc12 c1(OC)cc(C(=O)NC(CNC(C23CC(C2)C(C(F)(F)F)O3)=O)CO)sc1Cl c1(CCCC)ccc(C(=O)NC(CNC(=O)C(C)OCCN(C)C)CO)cc1 c1(C(=O)NC(C)CCCNC(c2ccc(C(C)(C)C)s2)=O)ncnc(O)c1F C(CNC(=O)CC1CCCN(C)C1)(CC)(CC)NC(C=CC=CCC)=O Cc1cc(CC(=O)NC2(C)CCCN(C(C34CC(C)(C3)C4)=O)C2)ccc1F C1(NS(NCC(=O)C=O)(=O)=O)CCS(=O)(=O)C2(CCOCC2)C1.CC(C)(C)O O=C(C1CCCc2sccc21)NCC(O)CNC(C1CC2CCC1O2)=O CC1(CNC(C2CCCOC2)=O)CCCN1c1ncnc(=N)[nH]1 C1(C(=O)Nc2cc(C)no2)CCC2(CN(Cc3cc(I)c[nH]3)C2)O1 c1(NC(C(c2cn(C)nn2)NC(c2cccnc2O)=O)=O)ccnn(C)c1=O C1(NC(c2cc(C)cc(C)n2)=O)CN(C(=O)CSc2nc[nH]n2)C2(CCCC2)C1 c1(C(N2CCC(C)(NC(C=CC=CC)=O)CC2)=O)ccc(S(=O)(=O)NCC)cc1 C1(N(CCCC2CCCC2)C(C2CCNCC2)=O)CCN(c2ccccc2)CC1 C1(NC(C(CC)OC)=O)CN(C(c2ccn(C(C)C)c2CC)=O)CCC1(C)C Cc1ccccc1C=CC(=O)NC(CCN(C)C)C(=O)NCC(=O)CC1CCC1 c1(Cn2cc(C3N(C(CCSCC)=O)CC(O)C3)nn2)ccc(COC)c(F)c1 c1(C(C)C)cnc(O)c(C(=O)NCC2CC2NC(c2cc(C(F)(F)F)c[nH]2)=O)c1 C(=O)(C(C)C1=CCCC1)N(CCN(C(c1coc(COC)c1)=O)CC)CCSC C1(NC(Cc2c(C)scc2)=O)CN(C(c2ccnn2CCOCCO)=O)CC12CC2 C1(C(=O)Nc2ccc(-c3c(C)nccc3)s2)CCc2ccccc2N1CCCO c1(C(N(C2CN(C(CNC(=O)OC)=O)CC2O)C)=O)nc(C)c(N)cc1C C(=O)(CC1=CCOCC1)N1CC(CC(=O)NCc2ccccc2Cl)C2(C1)CC2 C1(CNC(C2CCCSC2)=O)CCN(C(c2cc(C3CCCC3)on2)=O)C1 Cc1cnc2n1CCC(NC(=O)NCc1ccc(C#N)c(Br)c1)C2 C#CC1(C(=O)NCC=C)CCN(C(=O)CC23CCCC2C3)C1 CC(C)(C(=O)NCC1CCN(C(C2COCOC2)=O)CC1)C(N)=O c1(C(N2CC(N(C)C(C3CC34CCC4)=O)C2)=O)ccnc(OC2CCC2)c1F Cc1nc(CC(=O)NC(C)(C)C(C)NC(c2ccc(CO)s2)=O)c(C)s1 N1(CCOC)CCCC(C(=O)NCC(C)CN(C)C(SS(C)(=O)=O)=O)C1 c1(C(=O)NCCC(=C)CNC(c2ccnnc2S)=O)cc2cccc(C)n2n1 C=CCC(CC=C)C(=O)NC1CCCC12CN(C(c1sc(C#N)cc1Cl)=O)C2 Cc1nc(C2CC2)ncc1C(=O)NC(C1CN(C(C2CCC2)=O)C1)C C1(CC(=O)NC(C(=O)NC)C2CC2)CC(F)CN1C(c1ccc(C#N)[nH]1)=O C1(NC(CSc2cc(C)on2)=O)CC12CC(NC(=O)C(=O)Nc1ccccc1)C2 C1(C(=O)NCC2(CN(C(=O)C(C)OCC(F)(F)F)CC)CC2)ON=C(C)C1C N1(C(=O)OC(C)(C)C)CC2CCCCC2C1NC(c1cn(C)nn1)C1CC1 c1(OC)cccc(CC(O)C(=O)NCCCCCCN(C)C(c2cnns2)=O)c1 Cc1cccnc1C=CC(=O)NCC1CCN(C(=O)COc2ccsn2)C(C)C1 c1(CSc2n(C3CCS(=O)(=O)C3)nnn2)ccn2ncnc2c1 C1(OC)CN(C(=O)C=Cc2ncc[nH]2)C(C)(CNC(=O)CSCC(F)F)C1 CC1CCN(C(=O)COCC(F)F)CC1.C(CC(C)C)NC(=O)CSC(F)F Cc1cccc2c1OC(C(N1CCCC(C)(CNC(C3CCCCC3)=O)C1)=O)C2 N1(C(=O)C(F)C2CCC2)CCC2(CC1)CC(N=c1cc(Cl)c(O)n[nH]1)C2 N1(C(C(CCC)N(C)C)=O)CC(C)(C)CC1CNC(C12CCCC(CO1)C2)=O c1(COC)nocc1C(=O)NC(C)CCNC(=O)C=CCOC N1(C(C)C)C(=O)COCC1C(N1CCOCC1CCNC(c1nnn(C)n1)=O)=O CC(C)C(=O)C(=O)N1CCC1C(=O)N(C)Cc1cccc(O)c1 CN1CCCC(N(C(C2(C)CNC(=O)N2)=O)CNC2CCCN2C2CC2)C1 N1(C(c2cc(OC)ns2)=O)CCC(C(C)NC(C2(OC)CCCOC2)=O)CC1 c1(C(N(CC(CNC(CCc2cc(C)nn2C)=O)C)C)=O)cnc2occc2c1 C12(C(N(C3CCN(C(C)=O)C3)C)=O)CC(CN1C(=O)CCc1cnco1)C2 C1(C(=O)NCC#CCNC(COCC(=O)NC)=O)CC(C)(C)CC(C)(C)C1 c1(CNC(CNC(c2ccccn2)C)=O)cn(Cc2cccnc2)nn1 C1(C(=O)NC(CCCCNC(c2nc(C)sc2)=O)C)CCc2nncn2CC1 C#CCC(C)(C(=O)NC(CO)CC(C)(C)C)NC(=O)CC1C=NN(C)C1=O C(=O)(C(C)CC(N)=O)N1C(C(=O)NCc2nnc(C)o2)CC=CC1 N1(C(C2=NNC(=O)C2)=O)CC2CCCC(NC(C3CCC4(CCC4)C3)=O)(C2)C1 N1(Cc2c(C(=O)O)ccs2)CC(C(N2CCC3(CC3)C2)=O)C(O)C1 C(CC(CNC(C1CCC1(F)F)=O)NC(=O)CSc1ccncc1)OC c1(C(C)NC(C2CSCCN2Cc2cccn2C)=O)ncc2ccccn12 C(=O)(C(CCc1cnn(C)c1)NCCOC(C)(C)C)NCCCC(C)=O CC1(C)CC(CNC(=O)CN2CCCC2=O)N(C(=O)Cc2cccc(F)c2)C1 N1(C(CCC(C)(C)O)=O)CCC=C(C(=O)N(C(C)(C(F)(F)F)c2ccccc2)CCl)C1 c1(-c2cccc(C3(C(=O)NCCCCC#C)CC3)c2)cccn2ccnc12 c1(OC)cc(OC)cc(O)c1Cl.c1(C(=O)OC)cc(-c2ccccn2)ns1 C1(CC)C(NC(=O)Cc2cnoc2)CCN1C(c1cncc(C(C)C)c1)=O c1(OC)ccc2[nH]cc(C(=O)NCC(C)NC(=O)C3=CC(C)CC3)c2n1 c1(CC(=O)NC(C(N2CCC(CSC)C2)=O)CC2CCCC2)ncccc1C c1(CN(CC(=O)Nc2ccccc2)C)cccc(Cl)c1 N1(C(c2cncc(N)c2)=O)CC2(CCC2)CC1C(=O)NC1CCN(CCO)CC1 n1(CCC)ncc(C(=O)NCC2(F)CCN(C(c3cc(C)cs3)=O)C2)c1C N1(C(C(C)OC)=O)CCN(C(C23CCC(F)(CC2)CC3)=O)C2COCC12 c1(C(=O)NCC=CCNC(c2cnc(C(=O)OCC)s2)=O)nccc2n[nH]cc12 CCCS(=O)(=O)CC(=O)NC(C)(C)CCCNC(=O)Cc1ccoc1 c1(C(=O)NCC=CCC(N2CC=CC(OC)C2)=O)[nH]ccc(=O)c1C c1(CC(=O)NCC(CC=C)NC(=O)C=Cc2ccccn2)cccnc1C CN1CCC2(CCCN(C(c3cc(C(=O)O)ncn3)=O)C2)C1=O C1(NC(CC2CC(C(C)(C)C)C2)=O)CCCCN(C(=O)Cn2cc(C3CC3)nn2)C1 N1(C(C(C)=CC=C)=O)CC(C2CC2C(=O)NC2CC3(C2)CC3(F)F)C1 C(=O)(C1=CC2(CCOC2)C1)NC(CNC(c1c(C)c(Br)cnc1)=O)(C)C C1(CC(=O)Nc2cncc(C)n2)CC(N=c2[nH]cnc3cc(I)sc23)C1 C1(C(=O)NCC(c2ccccc2)NC(c2c(C(C)C)con2)=O)CCCN(C)C1 C12(CN)CC(C(=O)NCc3cnc(C)o3)C1C2 c1(C(=O)NC2(F)CCN(C(C(CC)N(CC)CC)=O)C2)cc(F)cc2cc[nH]c12 C1(OC)CN(C(=O)CCC(=O)NC2C=CCN(C(C)=O)C2)CC1CO Cc1ccc2c(c1)nc(CNCc1cc3n(c(=O)c1)CCS3)n2C Cc1cnc(C(=O)NCCC2CCN(C(c3ncc[nH]3)=O)C2)c(O)c1 C(=O)(C1=COCCO1)N1CCCC(CNC(CC2(C)CCOCC2)=O)C1 C1(C(=O)NCCCCCNC(Cc2c(C)n[nH]c2C)=O)OC2CCC1CC2 N1(C(CCCN=[N+]=[N-])=O)CC2CN(C(=O)C=CCF)CCC12 Cc1ccc(CC(N2CCC(O)(CNC(=O)COCCOCCO)C2)=O)cc1O C1(O)(NC(COC2CC(NC(c3c(CC)cns3)=O)C2)=O)CCC(C)C1 C(CC(=O)NC1CC2CCC1N(C(c1cccc(F)c1O)=O)C2)(C(F)(F)F)OC C(=O)(CCCCC(N)=O)NCCN(CC(C(=O)OC)C)C(=O)COC1CCC1 C1(C(=O)NC2CCOC2c2ccnn2C2CCCC2)CCC2(CCC2)CN1 CC(CCCC(F)(F)F)NC(=O)NCCc1cccc(C#N)c1 c1(C(N(CCC)CCNC(c2ccc[nH]2)=O)=O)cccc(C#CC2CC2)c1 C(=O)(C#CC(C)(C)C)NC(C1CCCCN1C(=O)COC1(C)CCOCC1)C C1(C(=O)NCC(C)(C)NC(=O)CNC(CN(C)C)=O)CC2CCCCC12 CCCCCCCCC(C)C(=O)N1CCC(N)(Cc2cccnc2OC)CC1 C1(NC(C(C(=O)OC(C)C)c2ccccc2)=O)CC(C)(C)OC1=O c1(C(=O)NC(CN(C(C2(C)CC(=C)C2)=O)CC)CO)cnn(C(C)C(C)C)c1C CCC(CC)(C(=O)N1C2CCC1C(NCC1CCCCCC1)C2)c1ccccc1 C=C(F)CN=c1nc(N2CCSC(c3ccccc3)C2)cc[nH]1 C1(CNC(c2ncc(OC)nc2)=O)CCN(C(=O)CO)C12CC2.C1(CN)CCCC1 N1(C(CCc2n(CC)ccn2)=O)CC(CNC(c2[nH]c(=N)sc2CC)=O)C(C)C1 C1(CNC(C2CCC2)=O)CCCN(C(C2CC2c2nc[nH]n2)=O)CC1 C(=O)(CCCCCN(C(=O)CNC(=O)C1CC1)C)NC1(CC#C)CCCCC1 C1(C(N(C2CN(C(C3COCCC3(F)F)=O)C2)C)=O)NC(=O)C2CCC12 c1(C(N2C3CN(C(C=CC(=O)N(C)C)=O)C(CC3)C2)=O)cc2cnc(F)cc2s1 CCCCC(C)C(=O)N1CC(CNC(=O)C=C2CCSCC2)C(O)C1 Cc1ccc(C(N2CCCCC(N(C)C(c3ccc(O)c(F)c3)=O)C2)=O)cc1F C(=O)(CCCC(F)(F)CO)NC(CNC(c1c(C)ccnc1)=O)C(C)C C1(C(=O)NC2CCCC(CNC(c3ccc(Cl)cc3)=O)C2)CC2C=CC1CC2 C1(NC(COCCC=C)=O)CN(C(C2CCCC2(F)F)=O)CCC1F c1(NCC(CC=C)NC(c2ccc(C)nn2)=O)ncc(Br)cc1C#N c1(CC)ccc(NC(=O)C2=CCN(C(c3cnn(C(C)C)c3)=O)C2)cc1O c1(N2CCCC(NC(CC3(C)CCOCC3)=O)C2)ncc(C#N)cc1Cl C1(C(=O)OCc2n(C)c(=O)ccc2)COc2c(ccc(Cl)c2F)C1 CC(Cc1cnc[nH]1)C(=O)N(C)CCn1cc(C(N2CCCC2)C2CC2)nn1 C1(NC(Cc2ccn(CC)n2)=O)CC2(C(=O)Nc3cc(Cl)n(C)n3)COC1C2 C1(CC)CCCC1C(=O)NC(C(N1CCOC1C1(C)CC1)=O)c1ccoc1 C1(c2n(CC)nnn2)(NCCN2CCN(S(C)(=O)=O)CC2)CC2CS(=O)(=O)CC12 CC(CNC(C1CC=CC(O)C1)=O)C(F)C(=O)N1CC2(CC2)CC1CO c1(OCC)nc(C)ccc1C(=O)NCC(O)CNC(C1CC(CC2CC2)C1)=O CCC(C)(CCNC(C12CC3CC1C2C3)=O)NC(=O)CCCOC(C)C C1(C(=O)NC2CC(NC(c3cc(C)nc(N(C)C)n3)=O)C2)C2CCCCCCC12 N1(C(c2ccc(C)o2)=O)CCCC(C)C1CNC(c1nn(C)cc1C)=O c1(C(N2CCCC(Nc3ncnc4ccsc34)C2)=O)ccc2n[nH]cc2c1 C1(N(C(c2cc(Cl)no2)=O)CC)CCN(C(C2CCCN(C(=O)OC)C2)=O)CC1 Cc1nc(O)sc1C(N1CC(OC2CC(=O)N(C)C2)C1)=O.C1CC(=O)NCCO1 C1(NC(=O)NCCc2cnc(C)[nH]2)CCC2CC2CC1 N1(C(c2n(COC)ncc2)=O)CC2CCC(C1)C2NC(C1CC2(CCC2O)C1)=O C(=O)(C1CC(=O)Nc2cc(F)ccc21)N(C(C(C)C1CC1)C(=O)O)C1CC1 C1(C(C(c2n(C)ncc2)NC(=O)C(=Cc2c[nH]cn2)F)=O)CC2(CNC(=O)O2)C1 C1(NC(CC(C(C)OC)NC(c2nc(CC)oc2C)=O)=O)CCOCC12CCC2 C(=O)(CCC(C)(C)C)N1CC(CNC(C(CN(C)C)(F)F)=O)C(n2ccnn2)C1 C1(NC(C)=O)CCc2onc(C(N3CCC(O)C(O)c4ccccc43)=O)c2C1 c1(C(=O)NCC(=O)N(CCC(=O)OC)C)ccc(=O)n(-c2ccccc2)n1 C(=O)(C1=CCCCCC1)N(C)CC1CCN(C(c2c(O)ccc(SC)c2)=O)CC1 N1(C(CCC2(NC(=O)NCc3ccno3)CCCC2)=O)Cc2ncsc2C1 c1(NC(C(=O)NCc2cnc(OCC)nc2)=O)cc(C)oc1NC(=O)NC C1(C(=O)NC(CCN(C(COC(C)C)=O)C)C)CCCC12CCC2 c1(C(=O)NCC2(C(=O)NC(CCOC)COC)CCCC2)nc(Cl)oc1C C(=O)(C(C)S(=O)(=O)C(C)C)OCCNC(C1C(CC)C1)=O c1(C(=O)NC2CCC(C)N(C(c3c(O)ncnc3O)=O)C2)c[nH]c2nccc-2c1 C1(C)(CC)CCC(C(N2CC(CNC(=O)CNC(=O)C(F)(F)F)C3CC23)=O)O1 c1(C(C(=O)N2CC(NC(c3c(C(C)C)onc3)=O)C2)(C)C)ccc(C#N)cc1 C1(C(C)C)(C(=O)N(CCC(=O)N(C)CCn2cncn2)C)CCOCC1 N1(C(C(CC)O)=O)CCN(C(c2cc(C3CCCN(C)C3)no2)=O)C(CCO)C1 Cc1ocnc1CNC(=O)CN(C(c1cn(C2CC2)cn1)=O)CC1CC1 C12(C(N3CCC(N(C(c4c(C)scn4)=O)C)C3)=O)CC3CC(CC(C3)C1)C2 c1(C(N2CC(NC(c3c(C)nn[nH]3)=O)CC23CCC3)=O)cc2cccc(C)c2o1 C12C(C1(C)C)C(=O)NC2.C1(COC)(CNC(=O)CC2CCOCC2)C=CCC1 N#Cc1cc(F)ccc1-c1cccnc1C(=O)Nc1cc(Br)cc(I)c1 C(=O)(C1=CC2(CCOC2)C1)Nc1c(C)ncnc1C.C123CC(C)(CN1C2=O)C3 C(CC(C)N=c1[nH]c2c(c(=NCCCc3cnn(C)c3)[nH]1)CCC2)OC Cc1ccc(C(=O)NCC2CC3CN(C(c4nc(C)sc4C)=O)CC23)cc1Cl C(=O)(C(C)(C)CC1CCC1)NC(C1CCN(C(CC)=O)C1)C c1(C(C)C)c(C(=O)NCCCCN(C)C(C2CCCS2)=O)cnn1C N12CCCC(C)CCCCC=CC=CN(C)C=CC(Cl)=CC=C1NC(=O)C2=O n1(C(C(=O)N(C2CCC(=O)N2)C(C(=O)NC)C)C)c(C)nc2ccccc12 C1(CNC(c2c(CNC(C3C(C(C)C)OCC3)=O)noc2)=O)CC(O)C(O)C1 C1(CNC(=O)NCc2ccc(NC)cc2)CCCC(C)(C)C1 c1(C(=O)OC)cc(C(N2CCCC(NC(C3CC(C)=NO3)=O)CC2)=O)cc(F)c1 C(N=c1[nH]cnc(Cl)c1C#N)C1C(NC(c2c(Cl)cn(CCC)n2)=O)CCC1 C1(NC(CCCNC(N)=O)=O)CC(CO)N(C(=O)CCF)C1 C(=O)(C(C)(C)CC(F)F)NCCNC(C(C)NSC(F)(F)F)=O c1(CC(=O)NC2CN(C(C(C)NC(=O)C(C)(C)C)=O)CC2C)ccnc(F)c1F C1(C(=O)NCC(C(C)C)NC(=O)Cc2cccc(C3CC3)c2)CCC(C)(C)OC1 CC(O)C(C)C(=O)NCCC(O)CNC(c1c[nH]cc1C1CCC1)=O Cn1cc2c(C(N3CCC(=CCNC(=O)CN4CCCC4)CC3)=O)cccc2n1 CC1(C)CCCC(C(=O)NCC(C)(C2CC2)NC(=O)C=Cc2ccccc2Cl)C1 C=CCCC(CCC)(c1nnnn1CC1CC1)NC1CC12CC(O)C2 Cc1ncc([N+](=O)[O-])cc1C(=O)NCC(C(C)C)NC(=O)C1=NOC2COCC12 CCC(C)(COC)C(=O)N1CCCC(N2CCN(C(=O)CN=S(C)(C)=O)CC2)C1 c1(NC(C2CC(F)(F)C2)C)nc2cc[nH]c2c(=NC2CC3COCC(C3)C2)[nH]1 N1(C(=O)CCCCC2CCCCC2)CC(F)(F)CC1CNC(C12CCC1CC2)=O N1(C(C(CCC)C)=O)CCC(COC)(NC(c2cc(C(C)(C)C)[nH]c2C)=O)CC1 c1(C(=O)NCC2(CC)CCOC2)ccc(CNC(=O)Cc2cncnc2)cc1 N1(C(CN(C2CC2)CC)=O)CCC(NC(C2CCCN(C(=O)C3CC3)C2)=O)CC1C c1(C(=O)NC(C)CC2CCN(C(=O)C3=NOCC3)CC2)cccc2ncn(C)c12 C=C(C)CC(C(=O)NOCC(N1CC(CO)C(O)C1)=O)OC(C)=O C1(C(N2CC(CC=C)(NC(=O)CC3C(C)C3(F)F)C2)=O)CC2(CC(=O)C2)C1 C1(C(=O)NC2CC3(CCN2C(=O)Cn2cccn2)CC3)CCn2nnnc2C1 Cn1cc(Br)c(CC(N2CC=CC(NC(=O)C(=Cc3ccccc3)F)C2)=O)n1 C(=O)(C(CC#N)c1ccccn1)NC1(C(C)C)CC1 C1(NCC(COCC(C)C)O)CC(NC(c2ccc(OC3CC3)cc2)=O)C12CCC2 O=C(CCCn1cccn1)NCC(C1CCC1)NC(=O)CC1CCC1 C=Cn1nccc1C(N(C)CCOC)=O.N12CC(C1)C2.C12CC1NC2=O C1(C(C)C)CCOC1C(=O)NC(c1cccnc1)C(=O)NCc1cnc(O)o1 c1(C(=O)OCC)ccc2c(c1)C(CNC(c1[nH]cc3c1CCC3)=O)CCC2 c1(C(C)C(=O)NCC(CO)NC(=O)CS(=O)(=O)NC2CC2)nc(F)ccc1Cl N(C1CCCc2ccc(Cl)cc21)C(c1c(C)scc1)c1nnnn1C C(C(F)(F)C(=O)N1CC(NC(=O)CC2CCC(=O)N2)C(c2ccccc2)C1)OC C1(c2cn(CCCC(=O)N(C)C3CC3)nn2)C2CCCCC12.c1ncc(Br)cn1 C1(NC(c2cnn[nH]2)=O)CCC2CN(CC(=O)Nc3ncc(F)cn3)CC2C1 C(CC(C(=O)NC1CN(C2CC2)C1)OCC=CCl)NC(=O)C=C1CCOCC1 c1(C(=O)NCCNC(c2coc(O)n2)=O)ccc([N+](=O)[O-])cc1Br CC(C)CCCCC(=O)N1CC2(CCCC2NC(=O)CCc2nncn2C)C1 N1(C(CC(C)F)=O)CCN(C(c2c[nH]nc2-c2cccnc2)=O)CC1C1CCC1 CCC(C)C(C)(O)CNC(C1C(CC)CCN1C(c1sc(C)cc1C)=O)=O c1(C(=O)NC2(CN(C(C(CCC)CC)=O)C)CC2)c(C)nn2ccccc12 N#Cc1ccc(C(=O)NC2CC(C(N3CCC(F)(CO)C3)=O)C2)s1 c1(C(N2CCN(C(CNC(C(C#C)(C)C)=O)=O)CC2)=O)cc(C)cnc1F N1(C(Cc2cc(C)no2)=O)CCC(C(=O)NCCCC2CCC2)C12CC2 C1(CNC(Cc2nnc(C)o2)=O)CCN(C(C2CCCN2S(C)(=O)=O)=O)C1(C)C Cc1[nH]cc(C(=O)NCC2(O)CN(C(C3CCC(C#N)C3)=O)C2)c(=O)c1Br N1(C(c2cnc(C)s2)=O)CCC2(CC1)CC2CNC(c1cnc2c(c1)COC2)=O Cc1nc2cc(C(N3CC(NC(C4CC5CCC(C4)O5)=O)C(O)C3)=O)ccc2s1 Cc1ccc2nc(CNC3CCN(C4CCCC4O)CC3)cn2c1 C1(CCC)CN(C(c2ccc(Cl)cc2N)=O)CCN1C(=O)C(O)CCSC CC1=C(C(=O)N(CC(C)(C)NC(=O)C(C)n2cccn2)C)CCC1 c1(C(N(CCCC2CCCC2)C)=O)c[nH]nc1C1CC1NC(=O)CC1CCCOC1 C1(NC(c2cn(CC=C)nc2)=O)CCC(NC(C2(O)CCOCC2)=O)CC1 N1(C(c2cc(-c3ccc(C)s3)[nH]n2)=O)CCC(NC(C2(C(C)C)CC2)=O)C(O)C1 CC(=O)C(C)CC(C)C(=O)N1C(C(=O)NCC#CCOC)CC2CCCC12 C1(C=O)CN(N2C(C)C(N(C)C)CCC2)CC(C)(C)O1.c1(C=O)cc(C(N)=O)cs1 c1(C(N2CCCN(CC(C)NC(=O)C(C)(F)F)CC2)=O)cnc2[nH]cncc1-2 C(=O)(CS(=O)(=O)CCOC)NCC1(NC(C2C(C=C)C2)=O)CCCCC1 C(=O)(CCC(=O)N1CCC(C(=O)NCCc2cccc(C)n2)(C(C)C)C1)OC CCCCC(=O)NCc1nc(CNC(C2CCC(=O)O2)=O)cs1 c1(CNC(C(=O)OCC)CC2CCCO2)ccc(Cl)c(-c2ccccc2)c1 c1(C(=O)NC2(C(N(CCCCOC)C)=O)CCCC2C)cc(C)cc(O)n1 N1(C(C(C(C)C)SCC)=O)CCC2CN(C(c3c(C)nnn3C)=O)CC2CC1 Cc1ccc(C(=O)NCC2CCC(CNC(=O)C(C)C3CCC3)CC2)c(N)c1 C1(C(=O)NC2CN(C(Cn3nnc(=N)[nH]3)=O)C2)CC(=O)N(c2ccccc2)C1 C(=O)(C(C(C)(C)C)N(C)CC)N(C(C)CNC(C)=O)C(c1ncc(C)cc1Br)=O N1(C(c2c(C)n(C)nc2)=O)CCC(C)N(C(=O)C(N2C(=O)CCC2=O)C)CC1 C1(C(N(CCSc2ccccc2)CC)=O)C=CCN(C(=O)C(C)(C)C)C1 c1(OCC)ccc(CCC(=O)NCC(C2CCC2)NC(=O)Cc2cnns2)cn1 N#Cc1cc(NC(=O)NCC(CO)CC(F)(F)F)cc(-c2ccc(F)cc2)c1 Cc1ccc(CC(=O)NC2CC(CO)N(C(c3cnc(C4CCC4)s3)=O)C2)cc1 C1(CC(=O)N=CC(=O)O)CC(N(c2cccc(CCC(=O)OC)n2)C2CC2)C1(C)C Cc1cc(NC(c2cn(CCNC(C3COCC(C)O3)=O)nn2)=O)cc(Cl)c1 N1(C(C2(OC)CCC2)=O)CC(CNC(c2scnc2Cl)=O)C(O)C1 c1(C(N2CCCCC(C(=O)NCc3ccns3)C2)=O)cccc2cc[nH]c12 c1(CC(=O)NCC2N(C(C=CCN(CC)CC)=O)CCC2C)ccc(C#N)nc1 n1(CCC(=O)NC2C(CNC(=O)CCn3cnnn3)CC2)cc(Cl)cn1 C1(C)(CNC(C2C(C)(C)C(F)(F)C2)=O)CN(C(=O)CC(Cl)Cl)C(C)(C)C1 N1(C(COCCOCC)=O)CCC(O)(CNC(=O)C(C)CSC)C1.C(C)=O CCC(CC(=O)NCC1CCCN(C(c2cnc(=N)[nH]c2)=O)C1)OC c1(N2C(CC)CN(C(=O)CCc3cn[nH]c3)CC2)nc(C#N)nc2ccccc12 C1(C(=O)OC)CCCC(C)(C)C1.c12ncc([nH]1)CC(=O)ONC(=O)NC2CC C(C(CNC(=O)Cn1nc(C)c(C)c1C)C(F)(F)F)NC(C1C=C(C)CS1)=O CCC(F)(F)CC(=O)NC(C1CCCN1C(c1ccc(C#N)cn1)=O)(C)C n1(CCOC)cccc1C(=O)NCC1(NC(c2ccc(CN=[N+]=[N-])o2)=O)CCC1 CN1CCN(C)c2cc(NC(=O)CNc3cc4ccncc4cc3F)ccc2C1 c1(C(=O)NCCC2CCCN(C(CS(CC)=O)=O)C2)cc2c(cc1OC)OCO2 C12(C(N3CC(CC=C)(NC(c4coc(CO)c4)=O)C3)=O)CCCC1C2(F)F c1(C(N2CC3(C2)CN(C(c2ccnn2C(F)F)=O)C3)=O)cc2c(Cl)cccc2[nH]1 c1(OC)ccc2c(CC(=O)NCCCCNC(=O)C(C(C)C)C(C)C)c[nH]c2c1 c1(C(=O)NCC(=C)CCNC(=O)CC(C)c2ccco2)cc(C)nc2ncnn12 N1(C(CC(CC)C2CCC2)=O)CCC(O)(CC(=O)Nc2cncnc2C#N)CC1 Cn1c(C(N2CC(F)(F)CC2CCNC(C2CCO2)=O)=O)cc2sccc12 c1(C(N2CCCC(NC(CCn3c(C)ncc3)=O)C2)=O)nnn2c1CCC2 C1(N(C(CC)=O)C)CN(C(=O)Cc2ccc(CO)c(C)c2)CC12CC2 N1(C(C(C)OCCCC)=O)CCC(CNC(=O)Cc2c(C)cccc2F)C12CC2 C12(CNC(C=NOC)=O)CCCCC1N(C(C1CCC(C(N)=O)O1)=O)CC2 c1(OC)cc(C#N)ccc1CNC(=O)NCCC12CCCC1C2 N1(C(C)=O)CCN(C2CCN(C(C3(C)CC3F)=O)CC2)CC1 CCCC(C(=O)N1CCN(CCCNC(C2CCNC2=O)=O)CC1)NC(N)=O Cc1ccc(C(=O)NC2CCCC2NC(C2CCCN(C)C2)=O)nn1 c1(OC(C)C(N2CCCC2C2(NC(c3cnc[nH]3)=O)CC2)=O)ccccc1 N#Cc1cc(C(N2CCC(C3CCCCN3C(C3(CN(C)C)CC3)=O)CC2)=O)c[nH]1 N(C(=NCCCCF)NC1CCCC1)C1N(C(CC)=O)CCC1 C1(OC)CC(NC(=O)COC2CCCC2)CN(C(C2CCC2(F)F)=O)C1 N1(C(C2C(=C)C2)=O)CCC(C(F)F)(CNC(=O)CC2CCN(CCC)CC2)C1 N1(C(CCCCCC)=O)CCCC2C(NC(=O)C#CC3CCOCC3)C(C)(C)C12 c1(C(N(CCNC(c2nc(C)nn2C)=O)CC)=O)cncc2ccsc12 C1(CNC(=O)CCc2nnc(C(F)F)o2)CCC2(CCC2)CN1C(=O)C(F)F c1(C(N2CCCC(N(c3nc(CC)nc(=N)[nH]3)CC3CC3)C2)=O)cccc2c1OCC2 C(CCC(O)C(=O)NCCN1CCC(C)(C)C1)NC(C(C)NC(=O)OCC)=O CC(O)(CC(=O)NCC1(F)COCCN(C(C2CC2F)=O)C1)P(C)(C)=O c1(CC)cncc(C(=O)NC2CCC(CNC(c3nc(C(C)(F)F)cs3)=O)C2)c1 C(C(C(C)C(C)C)NC(=O)CCSCC(=O)NC)NC(c1c(C)nc(CC)s1)=O c1(C(=O)NCC2CC2NC(C23CC4CC2C3C4)=O)cc(OCCF)ccc1Cl C(C(C)(C)CNC(=O)C(C)CN(C)C(C1CCN1C(C)(C)C)=O)SC C(=O)(CC(C)C)NC(CC)CNC(=O)CCOC1CC1 CONS(=O)(=O)c1ccc(C(=O)NC(C)CNC(=O)C(C)C(C)(F)F)cc1 C1(NC(=O)COCCCF)C2CC3CN(C(c4ccc(Cl)c(Cl)c4)=O)C1C3C2 C(c1ccc2c(c1)CCO2)=CC(N1CCN(CC2CCC(F)(F)CC2)CC1)=O C(=O)(CC(C1CC1)NC(C1CC(F)(F)C1)=O)NC(CCN(CC)CC)C C1(C(=O)NCC(C)NC(C2CNC(=O)N2C)=O)CC(=O)N(C)C1 C(=O)(n1cnc2ccccc2c1=O)OC(C(C(CC)CC)C)=O c1(NCC(CC=C)C)ccc(S(=O)(=O)NC(CSCC)CC(C)(C)C)c(Cl)c1 c1(C(=O)NCC(N(C(=O)CCCn2cncn2)CC)C2CC2)cc(SC)n(C)n1 C(C)(C)(CC(=O)NC1(C)CC(NC(=O)Cc2ccn(CC(C)C)n2)C1)OC CCC(CC(=O)N(C)CCN(C(=O)Cc1cnnn1C)C)C1CC1 C1(CCNC(CCCNC(C(CC)OCC)=O)=O)CCC2(CCC2)O1 C1(OC)CCOCC1NC(=O)C(C)N(C(=O)C=Cc1nccs1)C1CC1 C1(NC(CC2(C)CCOC2)=O)CCN(C(=O)CNC(C2CCCC2)=O)C1(C)C N1(C(C2C(CN(CC)CC)OCC2)=O)Cc2cccc(O)c2C1.C1CC(=O)N1 c1(C(N2C(C(=O)NC(C)CCO)CC(C)(C)C2)=O)cnn2ccccc12 c1(NC2C3CN(C(c4ccc(C(F)(F)F)o4)=O)CC32)ncnc2c1COC2 Cn1nc(Br)c2ccc(C(=O)NC3CN(Cc4cccc(Cl)c4[N+](=O)[O-])C3)cc12 c1(C2N(C(c3cnn(C)c3-c3nn[nH]n3)=O)CCC2)ccc(Br)cc1Cl n1(C2(NC(CC(=O)OC)=O)CC2)ccnc1 N1(C(C)=O)CCc2cc(S(=O)(=O)N(C(C)Cc3ccccc3C)C(C)C)ccc21 C1(NC(C2CCN(C(=O)NC)C2)=O)CN(C(c2nnc(C)s2)=O)CCC1C(F)(F)F c1(C(=O)NC2(COC)CN(C(N)=O)C2)cc2c(s1)CCSC2.C1(=O)CCCCN1 Cc1ccc2cc(C(=O)NC(C)(CNC(C3CC34CCC4)=O)C3CCC3)cn2c1 N1(C(c2c(OC)cncn2)=O)CC(C(=O)N(CC(C)CO)C)C(F)(F)C1 CN1CC(F)CC1C(N1CC=CC1CNC(=O)CC(C)(C)C)=O C12(C(=O)NCC3CCN(C(CCC=C)=O)C3)CCC(C(F)F)(CC1)CC2 n1(C(CC)C)nc(C(N2CC(NC(c3c[nH]ccc3=N)=O)C2)=O)cc1C C(=O)(C(C)(O)C(F)(F)F)N1CCC(=C)CC1C(=O)NCC1CCOC1C(C)C Cc1cccc(CCNC(=O)C(C2CCN(C(c3cc(C(N)=O)co3)=O)C2)C)c1 c1(C(N2CC(N(C(c3c(OC)ncnc3C)=O)C)C2)=O)csc2ccc(F)cc12 CCS(=O)(=O)CC(=O)N1CCCC(NC(c2ccccc2COC)=O)C1 C1(CNC(C=CSC)=O)CC2CCC1N(C(=O)CCOc1cccnc1)C2 c1(C(C)NC(=O)Cc2cnnn2C)cc(Cl)ccc1OC(F)F C1(CC)CCCC2(CCN(Cc3ccc4c(C)noc4c3)C2)O1 c1(C(=O)NCCN(C(C)C)C(C2COCCO2)=O)ccc(F)cn1 N1(C(C(c2cnn(C)c2)OC)=O)CC=CC(NC(=O)CC2(C)CC2(Cl)Cl)C1 C(CCNC(C1(n2cccc2)CC1)=O)(C(C)C)NC(Cc1nc(C)[nH]n1)=O CC1CCC(C(=O)NCC(C2CC2)NC(=O)C(C)(C)Nc2ccccn2)C1 C1(NC(=O)CCc2cn[nH]c2)CN(C(C2CC2c2ccccc2)=O)CCC1O c1(C(N2CC3CC(n4cc(-c5nc(Cl)cs5)nn4)C3C2)=O)cc2ncccc2s1 N1(C(CC(CC)O)=O)CC2CCN(C(c3cccc(C(F)(F)F)c3O)=O)C2C1 c1(C(C2CCCC2)NC2CC(CCC)C2)cccc(OC)c1 Cc1cc(O)nc(C)c1C(=O)N(CCCN(C(=O)C(C)(O)C1CCOC1)C)C c1(CCC(N2CCOC(CNCc3cncs3)C2)=O)cc(Br)ccc1Cl C=CC(F)(F)C(=O)N1CCN(CC(C)NC(c2ccc(C(C)C)cc2)=O)CC1 C1(CC(=O)NC2C(C)CN(C(c3cnc(Cl)nc3)=O)C2)Cc2cc(F)ccc2O1 N1(C(CNC(C2C(C)C2)=O)=O)CC(NC(C2CCCC23CC3)=O)Cc2ccccc21 C(=O)(C1=C(Cl)CCCC1)NC(CC)CNC(=O)C(C(C)C)c1cncs1 N1(C(c2ccc(C)s2)=O)CC2CCCC2(C(N2CC3(CCC3(C)C)C2)=O)C1 c1(CC)onc(C)c1CN(C)CC1N(C(c2oc(C3CC3)nc2C)=O)CCC1 N1(CCN(C)C)CC(F)(F)CC1(C)CNC(=O)CC1CCCOC1 c1(C(N2CCCC(n3nc(C)nc3C)C2)C(=O)NC)cc2cccc(OC)c2o1 c1(CC)onc(C(=O)NCCNC(C2CCN(C(C3CCSC3)=O)CC2)=O)c1C CCCC(CCC)CC(=O)N1CC(C2CCCCN2C(c2ccc([N+](=O)[O-])o2)=O)C1 CCC(CC(=O)NOC(=O)CCOCCN(C)C)CC(=O)OCC1CC1 N1(C(C=CC(C)C)=O)CC2CC(NC(c3cn4cnnc4cn3)=O)CC(C2)C1 CN(CC1(C)Oc2ccccc21)N1CCCC1OCc1ccccc1 CC(CC(=O)N1CCCCC1CCC(=O)N(C1CCOC1)C)C(F)(F)F C(=O)(C1CCCc2nn[nH]c21)N1CCN(C(C(C)(C)Br)=O)CC(O)C1 C#CCCCCCC(=O)N(CCCNC(=O)Cc1csc(C)n1)CC c1(C(N(C)CCN2CCN(C(c3ccc(O)cc3)=O)CC2)=O)cc2ncsc2[nH]1 CC1CN(C(c2ccc(C#N)[nH]2)=O)CC1CCNC(C1(N2CCOC2=O)CC1)=O c1(OC)ccc(C(=O)Nc2cc(C(F)(F)C(F)(F)F)ccn2)c2cnccc12 C1(C(=O)NCCCCC=C)CCCC(NC(C2(n3cccn3)CC2)=O)C1 C1(CNC(CCC=CCC=C)=O)CN(C(=O)C(C)C2=CCCC2)CCC1(C)C C1(C)(COC)CC(NC(=O)CSC2CC2)CN1C(=O)CN(C)C.C(=O)CC(C)(C)C C1(C(N2CC3N(C(C(COC)(F)F)=O)C3C2)=O)CCC2CC1CO2 O=C(C1=CC2=C(Cl)N=CNC2=NC1)NCCN1CCCN(C(C2CC2F)=O)CC1 CC1CC(CNC(=O)C(c2ccc(Cl)s2)C)CCN1C(=O)CCC1CC1(F)F C1(C(=O)NCC2(C)CCOC2)CCCCCCN1C(c1cc(CO)[nH]n1)=O c1(-c2c(C(=O)NCCN(C)C(C34CCC(CC3)O4)=O)nco2)ccc(F)cc1F c1(C(=O)NC(c2ccccc2F)C)cc2c(C3=CCC(C)CC3)cccc2s1 c1(C(=O)NC(c2ccccc2)CNC(C=CC(=O)OCC)=O)nnsc1N C1(NC(=O)CO)CCC2CCN(C(c3nncs3)=O)C1C2 c1(N(C)CC)ccc(COC(C)C)cc1.C1(=O)C(C#N)N1 C1(CN=C(NC2CCN(CC=C(C)C)CC2)NC(C)C)CC2C(O)CC2O1 C(=O)(C1=C(C2CC2C)N(CCSCC)C(=S)NC1c1cccc(=S)n1O)OC Cc1cncc(CCC(=O)NC2CCCC2(C)CNC(=O)Cn2cc(Cl)cn2)c1 C1(C)(CC=C)CN(C(c2cc(CNC(=O)CC=CC)no2)=O)C1 C1(C(=O)NC2(CNC(CC(C)N(C)C)=O)CCC2)CCCC(C)(C)O1 N1(C(c2cn(CC)nc2)=O)CCN(C(=O)C(C)OCc2cccc(C)c2)C(C)C1 C1(CNC(C2C(=C)CC2)=O)COCCN1C(c1ccc(-c2cn[nH]c2)cn1)=O c1(C(N2CC(CC)C2)=O)cc(Br)ccc1CN(c1ccnc(C)n1)C c1(OC)ccc(C(=O)N(C(C)CNC(c2cccnc2C)=O)C)c2ccccc12 Cc1nc(CCC(=O)OCc2cnc(C3CCC3)o2)cs1 C1(CC(=O)NCC(CNC(COCc2n(C)ccn2)=O)(C)C)CCCC(C)(C)C1 Cc1cc(O)ccc1CC(=O)NCC(C1CCCCC1)NC(C1CC1CF)=O N1(C(c2cnn(CC)c2C)=O)CCC(C2(NC(c3occ(C)c3C)=O)CC2)CC1 C1(SCC(=O)NCc2cc(C(=O)NC3CCC(C(F)(F)F)C3)co2)CC=CCC1 c1(CC(N2C(C(N3CC(C)OCC3)=O)CC(F)C2)=O)cc(Br)ccc1Br O=C(C1=C(Cl)CCCC1)NC1CCCC(NC(C23CCC(CC2)CO3)=O)CC1 Cn1c(C(=O)NCC2(F)CCN(C(=O)CCF)CC2)cc2ccsc12 n1(C(CC)CC)nc(C(=O)NC(C)CCNC(=O)CC23CC(C2)C3)ccc1=O C(C(CC1CC1)C(=O)NC1(C)CCOC1)NC(c1cnc(C)s1)=O Cc1c(NC(=O)CC(CC2CC2)NC(=O)C(C)CC(F)F)cccc1C#N C1(NC(C(CC)NC(C)=O)=O)CC2(C1)CC(NC(C1OCC1(C)C)=O)C2 C=C1c2ccccc2C(=O)N1CC(=O)OCC(=O)OC1C2CCOCC12 C1(F)(C(=O)NCCOC2CCN(C(C(c3ccc(C)o3)C)=O)C2)CCS(=O)(=O)C1 C(=O)(C1CCCc2ncnn21)NCCCN(CCCNC(C(C)C1CCC1)=O)C c1(C(N(C2CCN(C(C(C)NC(CC)=O)=O)C2)C)=O)ccc(C(C)C)cn1 c1(C(N(CCOCCN(C(C2N(CC)CCCC2)=O)C)C)=O)c(O)cccc1Cl C12(CNC(C3(CC)CC3)=O)CCCC(CN1C(=O)CCc1cnc(O)[nH]1)C2 c1(CC)c[nH]ccc1=NCCOc1cccc(F)c1 c1(C(N2CC3C(CN(C(c4[nH]cc(CC)c4)=O)C)C3C2)=O)cc(F)c(F)cc1Cl N1(C(C2(CC(C)C)CC2)=O)CC2CC1CN(C(=O)C(c1cccc(O)c1)C)C2 c1(CC)c(C(=O)NC2(C3CN(C(=O)CCc4cn[nH]c4)C3)CC2)cccc1F Cc1cc(I)ccc1COC(C)(C)C.c12ccc(cc1)c1cnc(nc1)c(=O)o2 Cc1nc(C(=O)NC2CN(C(=O)Cc3ccc(F)cn3)CC2O)c2ccnc-2[nH]1 CCC(O)CCCN1CCCC1Cn1cc(-c2cccc(Br)n2)nn1 c1(OC(c2sc(Br)cc2Cl)=O)csc2ncccc12 N1(C(CC(=C)C)=O)CCC(c2ccccc2)C(NC(C2CCCC(F)(F)C2)=O)C1 c1(N2CCC(C)(C(N)=O)C2)nc2ccsc2c(=NCC2CC3(CCC3)CO2)[nH]1 C#Cc1ccc(C(N2CC(NC(c3nn(C)c(C)c3Br)=O)CC2C)=O)cc1 N1(C(C(C)(C)C(F)F)=O)CCC(CNC(=O)C(O)C(F)(F)F)C(F)(F)CC1 Cc1ccc(CNn2cccn2)c2c1CCC2.N1(C=O)CCOCC1 c1(C(=O)NCC2C(C)CCN2C(=O)CN(CC(C)(C)C)C)ncn2ccccc12 Cc1nnsc1SC1CCCN1C(=O)C(=O)OC(=O)C(F)(F)F N1(N(C)CC=CC(=O)N)CCN2CC(O)CC2C1.C1(C#N)(C=O)CC1(C)C c1(C(N2CCC(N(CCO)Cc3sccc3Cl)CC2)=O)cc2cnccc2[nH]1 N(C(=NCC1CCC1)N1CC(O)C(C)(C)C1)CC(C)(C)OC(F)F C(=O)(CC(F)(F)C(F)(F)F)N(C1CCCCC1)CCNC(C(C)C#N)=O c1(C(N2C(CNC(c3c(C)nc(Br)cc3)=O)CCC2)=O)ccc2cnnn2c1 N1(C(C2N(C)CC(C)(C)C2)=O)C2CCCC1CC(NC(c1sccc1CO)=O)C2 Cc1c(CNC(=O)NCC23CCCC2CNC3)cccc1C(F)(F)F C=Cc1cc(C(=O)NCC(C)NC(=O)C(CCSC)NC(C)=O)cc(F)c1 Cc1cc(NC(c2nnnn2C2CCCC2)C2(CC#N)CC2)cc(C)c1Br N1(C(c2c(CC)[nH]c(=N)s2)=O)CCCC(CNC(c2ccnn2CCF)=O)CC1 N1(C(Cn2ncc(S(N)(=O)=O)c2)=O)CCC2CN(C(=O)C=CCF)CCC2C1 C1(NC(c2c(COC)occ2)=O)CC2CC1CC21CC1.C12(CCSC1)C(=O)N2 CC1Oc2cc(F)ccc2C1n1cc(CC2CCC3(CC2)NC(=O)C3=O)nn1 C1(C(CNC(CSc2nc(C)[nH]n2)=O)O)CCN(C(C2(C#N)CC2)=O)CC1 N1(C(COCCOC)=O)CCC(C)(CNC(c2ccc(C(C)(C)C)[nH]2)=O)C1 c1(CC(=O)NC2CC3CC2N(C(c2c[nH]nc2O)=O)C3)c[nH]c2ccccc12 N1(C(C(C)CC(N)=O)=O)CC(C(=O)NCCCOCCO)CC12CCC2 c1(C(=O)NCCOCCNC(Cc2c(OC)ccnc2)=O)cc2sccc2s1 c1(CNC(N(C)CC2CCC(F)C2)=O)cccc2cc[nH]c12 N1(C(c2cc(COC)oc2C)=O)CCN(C(=O)CCCC(C)(C)C)CC(CO)C1 N1(C(C2CCC(C)O2)=O)CCC2(CCCC2Nc2cc(S(C)(=O)=O)ncn2)CC1 C1(C(=O)NC2C(NC(c3c(C)nc(CCC)s3)=O)CC2)CC(=O)NC1(C)C S(=O)(=O)(c1c[nH]ccc1=NCCC=C(Cl)Cl)N(C)CC1CC1(F)F C12(NC(CC(C=C)CCC)=O)CCCC(CN(C(=O)C(C)(C)O)C1)C2 C(=O)(C(O)C(C)(C)C)NCC(C(C)(C)C)NC(c1c(C)nc(CCCC#N)o1)=O n1(CC)c(-c2cn(CC(N3CC(O)(c4cc[nH]n4)C3)=O)nn2)c(C)sc1=O N1(C(CCC=C=C)=O)CC2(CC2)CC1CNC(c1ccnn1CCCC)=O N1(C(C(C)n2cncn2)=O)CCOCC(NC(C2CC3C(C2)C3(C)C)=O)C1 C1(OC)(CNC(=O)N(C)Cc2[nH]c(C)nc2C)CCC(C)(C)CC1 Cn1ncc2c1CC(CC(=O)NCCN1CCOCC1)CC2 N1(C(C(C)O)=O)CCC2(CC1)CC(NC(c1scnc1C(C)(C)C)=O)C2 Cc1cc(C(=O)NCCC(C)NC(=O)C(=O)NC2CC2)c(C)n1-c1ccccc1 C#CC1(C(=O)NCC2(CO)CC3(CC3)C2)CCN(C(=O)CCc2ccoc2)C1 C1(Cn2cc(C3N(C(Cc4ccn(C)c4)=O)CC3)nn2)CCCOC1(C)C Cc1cccc(OCCC(=O)NC23CC2CN(C(=O)C(C)SC(F)(F)F)C3)c1 c1(C(=O)NC23C(CCN(C(C(=O)NC4CC4)=O)C2)CC3)cc2cc(Cl)ncc2[nH]1 n1(CCOC2CN(C(CN(C)C3CC3)=O)CC2C2CC2)ncc2ccccc12 C=C(Cl)CCC(=O)NCCSCC(=O)NCc1cncc(CC)c1 Cc1cc(C(=O)NC(Cc2nncn2C)C(N)=O)cc(F)c1 C(=O)(C(C)(C)CCN(C)C)N(C1CCCN(C(=O)C(N2CCCCC2)C)C1)C CC1CN(C(C2(C3CCCN3C(c3nnc(O)nc3O)=O)CC2)=O)CC(=O)N1C Cc1c(F)ccc(CN2CCN(c3cc(C(F)(F)F)ncn3)C(C(C)C)C2)c1F Cc1cccc2c(C(N3CCOCC3c3nncn3C)=O)n[nH]c12 CSC=CC(=O)NC1(CNC(=O)C(C2CCOCC2)C)CCCC1 c1(OC)ncc(C(=O)NC(CNC(=O)Cn2cc(C(=O)N(C)C)nn2)C2CCC2)s1 CCCC(C)(C)CC(=O)NC(CC(C)C)C(=O)NCC1CC2(CC2)C(=O)O1 CC(C)CC(C(=O)N1CCN(C(C2CCC(N=[N+]=[N-])C2)=O)CC1C)N(C)C C(=O)(C(C)CCC)N1CC(C)(C(N(CC(=C)C)C)=O)C1 CC(C(=O)NC1(C)CCN(C(c2c(F)cncc2Cl)=O)C1)C(F)(F)F c1(C(=O)NCCN(C(C(C#C)(C)C)=O)CCOC)ncnc(OC)c1F c1(C(N2CCC(NC(CCC(C)(F)F)=O)C2)=O)occ2c1CCOC2 c1(C(N(CC(C)NC(C2(F)C3CCCC23)=O)CC)=O)cccc(Br)c1F c1(NC(CC2OCCN(C(CCCC#CC)=O)C2)=O)cc(O)c(C)cc1C C(C(=O)N1CC(NC(=O)CCc2nncs2)C1)(N(C)C)C1CC1 C(CCC(=O)NCCc1ocnc1CNC(=O)CCC1CCCCO1)NC(C)=O Cc1nc(COCC(=O)NC(C)CNC(=O)CCc2cc[nH]n2)cs1 c1(C(=O)OC(c2ccco2)(C)NC(=O)C(C)C2CCC2)cc(C#N)c(N)cc1O n1(C(C(=O)OCC)C)cc(C2CCCN2C(c2cn(CC)nn2)=O)nn1 c1(CC(=O)NCC2C3N(C(CC(C)C)=O)C(CC3)C2)ccc(F)cc1[N+](=O)[O-] CCC(C(=O)NCC12CC1CN(C(c1coc(C)n1)=O)C2)C(C)(C)CC N1(C(C#C)C)CCC2CC(C(N3CC(=O)NCC3C(=O)O)=O)C2C1 c1(C(=O)NC2CCN(C(c3c(F)ccc(C)c3)=O)CC2)cc(N)c(C#N)c(F)c1 C=CC1(CC(=O)NC2CC(C(C)NC(=O)C(C)C(O)CC)C2)CCOCC1 O=C(C1Cc2ccccc21)N1CC2CCCC(C1)N2C(=O)C1=NOCC1 c12ccc(Cl)c(Cl)c1C(=O)OC1CN(C1)C(=O)N2.C(CCl)O.N(F)F N1(C(C(C)CC2CC2)=O)CC2CCN(C(=O)CCN=c3[nH]ccs3)CC2C1 c1(SCC(N2CCC(CNC(C(C)Cc3ccncc3)=O)C2)=O)ccc(O)cc1 C1(NC(CS(=O)(=O)NCC)=O)(CC)CCCN(C(=O)CCC2CCCO2)C1 c1(C(N2CC(O)(CNC(=O)CC3CCCCO3)C2)=O)cncc2c(F)cccc12 c1(CN(C(C(C)OC)C(=O)N2CCC(OC3CCC3)C2)C)ccc2c(c1)OCO2 C1(N=[N+]=[N-])(C(=O)NCc2n(CC)nnn2)CCN(C(=O)CCN(C)CCO)C1 C1(NC(CC)=O)CC2(CCN(C(c3ccn(C4CCCC4)n3)=O)CC2)C1 C1(NC(=O)C(Cn2cncn2)NC(C2CC2Cl)=O)CC(=O)NC(=O)C1 c1(C(N(C2CN(C(COC(C)=O)=O)CC2O)C)=O)cn(C(C)C)c(=O)nc1O N1(C(Cc2ncc(C)s2)=O)CC=CC(NC(=O)C(C)(C)C2CCCCC2)C1 C(=O)(C1=C(Cl)CCOC1)N1CC(CCNC(=O)CCC2CC3CCC2C3)(OC)C1 C1(NC(c2cocn2)=O)CN(C(c2ccoc2C2CC2)=O)CCC1c1ccccc1 C(CCCNC(=O)CC1CSC1)(c1ccccc1)NC(CNC(N)=O)=O c1(N2CCCC(CCC(C)C)C2)nc(NC2(C(=O)N(C)C)CC2)c2ccsc2n1 c1(-n2ncc(C(N(CCNC(C(C)SCC)=O)C(C)C)=O)c2)ccc(C)cc1 N1(C(CC(CC#C)NC(C2C=C(C)CS2)=O)=O)CCC(C2CCCC2)C1 c1(C(N2CCC(C)(c3ccc(C)cc3)C2)C(=O)NCC)cccc(I)c1 N1(C(c2c(CCC)nco2)=O)CCC2(CC1)CN(C(=O)CC1COCC(C)O1)C2 N1(C(CCCC)=O)CCC2CN(C(=O)C3=CCCS3)CC2C1.N12CCCC1C2=O c1(C(=O)NCC(C2(O)CN(C(C3CCOCC3)=O)C2)(C)C)ccn(C2CC2)n1 c1(OC)cc(C(=O)NC23CC2CN(C(c2c[nH]nc2C(C)(C)C)=O)C3)ccc1C c1(C(=O)NCC(C)NC(=O)CCC2CC2CC2CC2)cc2c(cc1O)OCO2 c1(N2CC=C(C)CC2)nc2c(c(=NCc3ccc(C)c(N)c3)[nH]1)SCC2 C1(C(=O)NC2CCC(NC(CCc3[nH]c(=N)sc3)=O)CC2)Cc2nncn2C1 CC1(C)CCC(=CC(N2CCN(C(=O)C(C3(O)CCCC3)F)CC2CO)=O)CC1 CCCCC(C)C(=O)N1CC(NC(=O)Cc2ccc(OC(C)C)cc2)CC(C)C1 N1(C(c2c(C)scn2)=O)Cc2ccccc2C1CNC(=O)Cc1ccon1 N1(C(C(CC=C)N(C)C)=O)CCC(O)(CCN(C(C)C)CC)CC1 c1(C(=O)NCCC2CCCN(C(c3cncc(C)c3)=O)C2)coc(S(N)(=O)=O)c1 S(=O)(=O)(c1cc(Cl)ccc1OC(F)(F)F)NC(C(=O)OC)CC1CCC1 C#Cc1cccc(C(N2CCCC(N(C(=O)CCC3CCCN3C)CC)C2)=O)c1 N1(C(c2cc(C)c(C)nc2O)=O)CCCC2CN(C(c3ccoc3)=O)CCCC12 C1(OC)CC(CCNC(=O)C(C)Cc2cnn(C)c2)N(C(=O)CCCC2CC2)C1 C1(CCC)CN(C(=O)Cc2csc(NC=O)n2)CCN1C(c1nonc1C)=O c1(N2CCC(SC)CC2)ncccc1S(=O)(=O)N1CCCC1CC1CC1.NC C12(C(C)C)COC(C(=O)NC(CC3CC3)CNC(=O)COCC3CCCO3)(C1)C2 N1(C(C(CC)C)=O)Cc2ccccc2CC1C(=O)NC(c1ccc(F)cc1)C Cc1c[nH]cc(C(=O)NCCN(C(C2CS(=O)C2)=O)C(C)C)c1=O C1(C(N2CCC(CNC(C3(C=C)CC3)=O)C2)=O)CCCC(=O)N1C CC(C)C(C(=O)N(CC(N)=O)C)C(C)NC(c1cnn(C)c1N)=O CC1CCC(O)CN1C(c1cc(CNC(c2cnnn2C)=O)no1)=O c1(NC(C2CCOC2)C)nc(N2CCC=C(Cl)C2)cc(=NC)[nH]1 N1(C(=O)OCC)CCCC1(C)C(N1CCC(CCNC(=O)C=CC(C)C)CC1)=O N1(C(c2cccc([N+](=O)[O-])c2)=O)CC2CC(N=c3[nH]c(Cl)ncc3[N+](=O)[O-])C2C1 N1(C(C(=O)NC)CCCCOC)CCc2cc(-c3ccccc3)oc2C1 CCCCCC(F)C(=O)NC1(CF)CCN(C(c2cc(C(F)F)n(C)n2)=O)C1 Cn1cc(C(=O)NCC(C2CCCCC2)NC(=O)Cc2csc(C(F)F)n2)cn1 Cc1cccc(C(=O)NC(C)CNC(C2CCOC2c2cccnc2)=O)c1N O(N(C)C(=O)CNC(=O)C(CCF)NC(=O)C(C1(C)CC1)C1CC1)CC CC1CCC(CCC(=O)Nc2ccc(-c3ccccn3)cc2Cl)C1(C)C c1(C(N2C(CCNC(=O)C(F)C3CCC3)CSCC2)=O)ccc2[nH]ccc2c1 c1(C(N2CC(NC(C(CC)O)=O)C3(C2)CCC3)=O)coc2c1C(=O)NCC2 c1(SC)ccc(OCC(N2CC(NC(C3CN(C4CC4)CCO3)=O)C2)=O)cc1 c1(C(=O)NC2C(CNC(c3c(C)nc4sccn43)=O)C2)coc2c(Cl)cccc12 Cc1cccc(CNC(C2(O)CCN(C(=O)Cc3cc(Cl)ccc3O)C2)=O)c1F c1(C(=O)NC2CC(NC(C3CC34CCCC4)=O)C(O)C2)ccc2c(c1)CC2 C1(CNC(CC(C)C2CCCC2)=O)CCCCN1C(c1coc(CO)c1)=O C1(C)(C(=O)NCCCC(CO)NC(Cc2ccc(C)s2)=O)CCC(=O)NC1 C(=O)(CC(CN(C)C)C(F)(F)F)NC(C)CNC(c1cc(F)c(Cl)cc1F)=O c1(CC)ccsc1C(N1CC(CC(C)(C)CNC(C2(Cl)CC2(C)C)=O)C1)=O Cc1nccnc1C(=O)NCC1(CCCNC(C2CCS2(=O)=O)=O)CCCC1 c1(C(=O)NC2(C)C(NC(C(n3c(C)ncc3)C)=O)CCC2)ccn2nccc2c1 C1(C(c2n(CCC3(C)CC3)nnn2)NCc2cccc(Cl)c2)CCCCC1(F)F C=CCC(CC=C)C(=O)N1CCCC(C)C1CNC(c1ncnn1CC)=O N1(C(c2cc(OCC)no2)=O)CC(OC)CC(NC(=O)C(O)CSC)C1 c1(OC(C)C(N2CC3(CCCC(NC(N)=O)O3)C2)=O)cnc2ccccc2n1 CN1CC(C(N2CCC2CC(=O)N(C)Cc2nnnn2C)=O)CCC1=O c1(CSC)ccc(NC(c2cnn(-c3ccc(Br)cc3Cl)c2)=O)cc1C(=O)O C1(CNC(C(C)OCCCC)=O)COCCN1C(c1cc(C(C)C)sn1)=O c1(C(=O)NC(CC)CNC(C2C3CCCOC23)=O)cc(C2CC2)n(C)c1C c1(CC(=O)NC23C(CN(C(C4CC(C)(O)C4)=O)C2)C3)ccc2sccc2c1 C1(CC)CCCCC1C(=O)NCCCN(C(c1c(Cl)cnn1C)=O)C1CC1 CC(c1ccccc1)=CC(=O)NCC1N(C(C2(N(C)C)CC(O)C2)=O)CCOC1 c1(C(=O)NCc2scc(CNC(CC=CC)=O)n2)cc2cnccc2o1 C1(CC(=O)NCC(C)CNC(=O)C=C2CCC2)CCCC(=O)N1 c1(NC(C2CCC(NCc3cc(OCC)ncc3)C2)=O)ncc(Br)cc1F C1(NC(=O)C(Cl)CCl)COCCN(C(=O)Cc2cccc(Br)c2F)C1 CC(CCC(=O)NC1(CCN2CCCC2)CC1)NC(=O)C=CCN(C)C C12(CC(=O)N(C)CC3CCN(C(C4C(C#C)C4)=O)C3)CCCN1CCC2 N1(C(C2(C(=O)OCC)CC2)=O)C(C(N2CCSCC2)=O)CC1C Cc1cnn(CC(=O)NC2CC(NC(C3CCCN3C(N)=O)=O)CC2O)c(=O)c1 c1(NCC)scnc1C(=O)NC(c1ncc(C(N)=O)s1)C.C(C(=O)OC)S C1(CC(=O)NCC2CC(C(N3C(C(=O)NC)CC3)=O)C2)CCC(O)C1 c1(CCCC(=O)NC2(CF)CCN(C(C=CC(N)=O)=O)C2)c[nH]c2ccccc12 c1(C(N2CCC(N(C(C3COCCS3)=O)CC)CC2)=O)cc2c(F)cccc2s1 C1(C(=O)NCC(C#C)CC2CC2)CNC(=O)CN1C(=O)CN1C(=O)CCC1=O CS(=O)(=O)c1ncccc1C(=O)NC1CCC(CCNC(c2cc[nH]n2)=O)C1 c1(CC(N2CCC(C(N(CCC)Cc3ocnc3C)=O)C2)=O)cncc(C)c1 c1(CC(=O)NC(CN(C(C=CC(C)C)=O)C)C)ccc2c(c1)CCO2 c1(CCOC(C(C2CC2)OC)=O)nc2ccccc2s1 c1(-c2n(C3CCC(C)(C)C3)nc(C3CC34CC4)n2)ccc2ncccc2c1 N1(C(CCOC)=O)CC(C(=O)NCC2(N(C)C)CCCC2)OC(C)C1 C1(C(=O)NCC(COC)NC(C2CCC2(F)F)=O)CCCC(CF)C1 C1(N(C(CCc2onc(CCC)n2)=O)C)CCN(C(C2CC(O)C2)=O)CC1C C(CCC(=O)NC(c1ccccc1)C(C)NC(=O)CC=C(C)C)NC(C)=O N1(C(C=Cc2cncc(C)c2)=O)C2CCC1C(C)C(NC(c1cc[nH]n1)=O)C2 C(CN=c1[nH]c(=NC2CCCn3cnnc32)c2c(ncn2C)[nH]1)(C1CC1)SC C(N=c1[nH]c(=NC)[nH]c(=NCCc2ccc(C)o2)[nH]1)c1cc(CC)on1 c1(C(N(C2CN(C(c3cccc(C4CC4)c3)=O)C2)C)=O)ccc2ncnc(O)c2c1 c1(OCC(=O)NC2(C)CC(NC(=O)CC3=CCCC3)C2)c(O)cnc2ccccc12 CCCN=C(NCC(c1cccs1)OC)NCc1c(C)cccc1F C(=O)(CCCCC1CC1)NCCC1(OC)CN(C(=O)CCc2ccccc2O)C1 c1(SC)ccc(F)c(-c2csc(CN(CC(=O)C(C)C)C(=O)CC3(O)CCC3)n2)c1 c1(C(N2C(C)(NC(=O)C3=CCCCC3)CC(O)C2)=O)cnc2c(c1)CCC2 c1(CCC=C)cccc(S(=O)(=O)NCC2(CCCO)CCOCC2)c1 c1(C(=O)NC2CN(C(C(CC)OCC)=O)CC2C)nn(C)cc1S(N)(=O)=O Cc1cc(OC(C)C(N2CCN(C(C3CCCC3C)=O)C(CO)C2)=O)ccc1Cl C1(C(N2CC(CNC(C3COC4COCC34)=O)OCC2)=O)Cc2ccncc2C1 Cc1[nH]c2ccc(Br)cc2c1CN=c1[nH]c(N)cc2c1CCCC2 C12(CNC(C=C(CC)C)=O)CC1CN(C(c1cscc1C(N)=O)=O)C2 C(C(CSC)CC)c1n(C(CC)Cn2cncn2)nnn1 C1(C#N)(C(=O)NC(CC(=O)NC(C=C)C)C)CC12CCC2 N1(C(c2cccc(C)c2Cl)=O)CC2CN(C(c3coc(O)n3)=O)CCC2(CO)C1 N1(CC(C(N)=O)NC(C(C)OC(F)F)=O)C(=O)c2ccccc2C1=O CC1CCN(C(c2ncoc2C2CC2)=O)CCN1C(=O)Cc1cccnc1 N1(S(C)(=O)=O)CCN(C(c2cnn(CO)c2N)=O)CC1.C1(C)CC(CO)CO1 Oc1ncc(Br)c(F)c1CSCC(Oc1cccc(Br)c1)Oc1ccsc1 C1(=O)CC(C)(O)C(=O)C(CC)C(=O)NC(C)C(=O)NCC(CC)N1C C1(C(=O)NC(CNC(C(N2CCNC2=O)C)=O)CO)CC(=O)N(C2CCCC2)C1 C1(CC(C)NC(=O)C(C)N2CCC2)CC2CCC(C1)N2C(c1cocn1)=O C(=O)(CCC(N)=O)N(C)CCNC(=O)NC1CC1.c1c[nH]c(-c2ccccc2)c1 N1(C(c2c(C)cc(C)s2)=O)CCCCCC(NC(C2CCc3[nH]ncc3C2)=O)C1 C(CS(=O)(=O)CC(=O)NC1CC(NC(=O)CCc2ccc(SC)cc2)C1)OC C1(CNC(=O)CN2CSCCSC2)CC12CCN(C(C1(CO)CCCO1)=O)CC2 c1(N(CCN(C)C(c2ccn(CC(F)F)n2)=O)C)nc2ccc(F)cc2s1 c1(-c2ccc(CN(C(C)C)C)s2)ccc(O)c(F)c1 C(=O)(C(C)(C)CCNC(c1ccn(CC)c1C)=O)N1CCC(=C)CC1 CC(C)C(C(=O)N(C)C)NC(C1OCCC1CNC(c1ccn(C(C)C)c1)=O)=O C1(C(=O)NC(C)(CNC(=O)CC2C(C)(C)C2(C)C)CO)CC12CCCCCC2 C1(C(=O)NCc2cnc[nH]2)CCN(C(c2cccc(Cl)c2)=O)CC1O C(=O)(CCCC(C)NC(c1nsnc1O)=O)NCC(C#C)C(C)C N12CCC(C)(CC1)NCC2=O.C(=O)(C(F)=CCCF)CCC.OCC Cc1[nH]nc2c1CCC(C(=O)NCC1CC1NC(=O)Cc1c[nH]c3cnccc13)C2 n1(CC)ccnc1C(=O)NC1CCOC1C(=O)NCC(c1ccn(C)n1)O Cc1oc2ccccc2c1CN1CCN(C(c2cccc(CF)c2)=O)C(C)C1 Cc1cc(C(=O)NC2CCN(C(c3cccs3)=O)CC2O)cc2[nH]ccc12 N1(C(CCNC(C)=O)=O)CCCCCC(NC(=O)CSCC(F)(F)F)C1 C(=O)(C1CCCc2nc[nH]c21)NC1C(C)CCN(c2snc(C(=O)OC)n2)C1C CCC1=NOC(C(=O)NC2COCCC2C(=O)N(CC(F)F)C(C)C)C1 C(CC(C)(C)C(=O)NC1CC12CCCC2)NC(CCC(C)NC(N)=O)=O CC1CCN(C(=O)CC2=CCCC2)C1C(=O)N1CC(O)CO1 c1(OC)cc(C(N2CC=CC2CNC(c2cnn(CCO)c2)=O)=O)ccc1Cl C1(C(=O)Nc2nnn(C(C)(C)C)n2)CC2CCC(C1)N2CC1(N(C)C)CCSC1 c1(C(=O)NC(C)CNC(=O)C(F)(F)CC2CC2)nccc2ncccc12 c1(-c2n(C3(C)CCN(Cc4nnn(C)n4)C3)ccn2)cnn2c1CCC2 C1(NC(C2CC(F)(F)C2)=O)CC(CO)N(C(=O)CC2(O)CCC2)C1 N1(C(c2cc(C)nc(O)c2)=O)CC2C3CCC(C2C1)N(c1ccnc(C#N)n1)C3 c1(C(=O)NCCOCCCNC(c2cnsc2)=O)c[nH]c2ccccc2c1=O c1(C(N2C(CNC(c3c(C)c(N)cnc3)=O)CC2)=O)csc2c1CCC(C)(C)C2 CC1(C)CN(C(c2cc(Cl)sc2Cl)=O)CCC1NC(=O)CCCCCn1cnnn1 C(=O)(C(F)C1CC1)NCCN(C)C(=O)NC(=O)CCSC(F)(F)F.C(C)(C)(C)O c1(C(=O)NC2CSC2)ccc(N)cn1.CN(CCOCCOC)C(=O)C1CC1 C(C)(C)(CC(F)C(=O)N1CCSC2(CCC2)C1)NC(c1ccc(CC)o1)=O C1(CNC(c2cc(C)sc2)=O)CCN(C(c2oc(C(C)C)nc2C)=O)C12CC2 N1(C(COCCC)=O)CC(NC(=O)CC2CCC(F)(F)C2)CC(O)C1 CC1(C)CN(C(C2(C(F)(F)F)CC2)=O)CC1N=c1nc(CC2CC2)[nH]s1 C(=O)(CCCCCN=[N+]=[N-])NC(CC#C)C(N1CC(F)(F)C(F)(F)C1)=O C(=O)(C(C)C(O)CC(C)C)NCC1(NC(CCCCNC(C)=O)=O)CCC1 Cc1cc(C(=O)NCC(C(=O)N(CC(C)N(C)C)C)N(C)C)cc(F)c1 c1(OCC(=O)NC2CN(C(C3CCC4CC34)=O)CC2(F)F)cc(Cl)ccc1Cl N1(C(C=C2CCN(C)CC2)=O)CC2CCC1CN2C(c1ccn2nccc2n1)=O Cc1ccc(CN2CCC3(CC3C(=O)Nc3cncc(O)c3)C2)cc1C#N c1(N2C(C)CC(CNC(c3cccc(=O)o3)=O)C2)ncc2c(c1C#N)CCC2 C1(CNC(CN(CCOC)C)=O)CC(C(F)(F)F)CN1C(C1CC1C)=O C1(C(=O)NCC(C)(C)SC2CCN(CC)C2)(COCCNC=O)CCN(C)C1 c1(C(=O)NCC(C2CCCC2)NC(C2(c3cccs3)CC2)=O)coc(Br)n1 c1(C(=O)NC2(CO)CCCN(C(C(CC(N)=O)O)=O)C2)cnc2cccnn12 CC1CCc2sc(C(=O)NCC3CC3NC(c3cc(F)c(Cl)cc3Cl)=O)cc2C1 c1(CNC(C2CC2C(F)F)=O)ncsc1C(N1CC(O)C1)=O C(=O)(CC(C)(C)C#N)NCC(CCC)NC(C1(C)CC(C)=NO1)=O C1(CCN)CCC(=O)N(C(c2ccc(CC(F)F)cn2)=O)C1=O C1(C(N(CC(O)C2CC2)C)=O)CC2CCC(C1)N2C(C1CCCC(=O)CC1)=O N1(C(CC2CC(C)C2)=O)CC2(CCOCC2)CC1CNC(=O)CCSC(F)(F)F c1(C(=O)NC(C)CCNC(=O)CN2CCCC2=O)ccc2c(c1)C=CS2(=O)=O C1(NC(C=CCCC)=O)COCC1NC(C1SCC=C1C)=O C12(NC(c3scc(OC)c3)=O)CCCC1(F)CN(C(c1nn(C)c(Cl)c1Cl)=O)C2 C#CC1(C(N2CCC(CO)C(C)C2)=O)CCN(C(c2cnc(C)c(C)c2)=O)CC1 C(=O)(CCCC(=O)NC1CC1CNC(c1ccnc(CO)c1)=O)OCC c1(C(=O)NC2CCC(C)(NC(c3ncccc3Cl)=O)CC2)cccc2c1CCO2 CC(C)CCC(O)C(=O)N1CC(C2CN(C(c3n[nH]cc3C3CCC3)=O)C2)C1 C1(C(N(C2CCCN(C(C3C(C)(C)C3(C)C)=O)C2)C)=O)CC2(CCOC2)C1 N#Cc1c[nH]c(C(N2CCCOC(CCNC(c3ccc(F)c(F)c3)=O)C2)=O)c1 C1(C(c2ccccc2)SC)CCCN1N1CCn2c(C(N)=O)nnc2C1 C=CC1(CC(=O)NC2CCCC2O)CN(C(=O)C(C)C2(O)CCC2)C1 CN1C2CCC1CC(C(=O)NC1CN(C(c3ccnc(Cl)c3N)=O)CC13CCC3)C2 N1(C(c2cccc(F)c2)=O)CCN(C(c2cc(F)c(Cl)cc2F)=O)C2CCCC12 C1(CC)CC(C(=O)NC2CCN(C(c3cncc(C)n3)=O)C2C(C)(C)C)CCO1 C(=O)(CCCC(C)C)NCC(C1N(C(C(CC)n2cncn2)=O)CCC1)(C)C C1(C(=O)NC2C(OC)CN(C(=O)C=Cc3ccccc3)C2)CC2(CCCC2)C1 c1(C(=O)NC(CCN(C(=O)CC(C)(F)F)C)C(C)(C)C)nnn2c1CSCC2 CC1CN(C(C2OC3CCC2C3)=O)CCC1C(=O)NCc1cccc(O)c1 c1(OC)ccc(NC(=O)C(C)(C)C2CCN(C(c3n[nH]c4c3COC4)=O)C2)cc1O CC(C)CC(C)C(=O)NC(C(=O)NCc1c(O)cccc1Cl)C(C)(C)C C(N=c1[nH]ccc(C#N)c1[N+](=O)[O-])C1C(C)CN(C(=O)CC(=O)NC2CC2)C1 Cc1sccc1CNC(=O)NCc1nnsc1C1CC1 N1(C(C(Cc2cn(-c3c(SC)cccc3)nn2)C)=O)CC(C)(C)OCC1COC C1(NC(C(C2CC(F)(F)C2)OCC)=O)CC12CCN(C(C1CCC(=O)O1)=O)CC2 C1(CNC(CCC(C)OC)=O)CC2(CCN(c3ccncc3C#N)C2)CO1 c1(CC(=O)N(C2CCN(C(C3CC34CC4)=O)C2)CCC)ncc(C)s1 N1(C(CCCCCC#C)=O)CCC2CCC(C1)N2C(C1CCC2(CCC2)O1)=O C1(CN(C)C(c2ccns2)=O)CCCC(OC(C2CCC(C(=O)N(C)C)CC2)=O)C1 CCCC(C(=O)N1CCC(C(C)NC(=O)C(Cl)=CCl)CC1)NC(N)=O N12CCC3C(C1)CN3C(=O)C1(CC1)CNC2=O.C1(N)CCCC(OCC)C1.OC C1(NC(=O)C(Cl)=CCl)CC2CN(C(C3(F)CCCC3)=O)CCN2C1=O C1(Cc2ccc(C(=O)N3CC(n4cc(C5CCC5)nn4)CO3)o2)CCCCC12CC2 C(=O)(CC1=NNC(=O)C1)N1CC(CCNC(C(C)OCC)=O)OCCC1 c1(OC)ccc2c(c1)CCCC2C(=O)NC1CC1NC(c1ccc(C)nc1O)=O N1(C(C=C)=O)CCC(C2CC2)C1CCNC(=O)C(O)CCSC C(CN=c1[nH]c(N(C)CC2CC2C)nc2cc[nH]c12)SC(C)C CC(O)(C(=O)NCC1CC(O)CN1C(c1cc(Cl)cnc1O)=O)C(F)(F)F c1(C(C)NC(=O)N(C(C)CO)C)cccnc1.CC(C(=O)NC1CC1)OCC1CC1 CC1CN(C(=O)Cc2c(Br)cnn2C)CCN1C(=O)CCC1CCCOC1 O=C1NCCCC1n1cc(C2CC2)nn1.c1(C)ccsc1Br C(C)(CC(=O)NCC(=O)N(CCO)CC1CCC1)NC(C=CC)=O c1(OCC)ccc(C(=O)NC(C)CNC(c2occc2C)=O)cc1OC C1(C(=O)NCCCCCCN(C(C2C(=C)C2)=O)CC=C(C)C)CNC(=O)C(C)(C)C1 N1(C(Cc2ccc(C(=O)OC)s2)=O)CC(CCNC(=O)CCSC)OC(C)C1 c1(CN2C(C(N3CC(C(=O)NCC)(COC)C3)=O)CC2)ccc(O)nn1 O=C(CC(F)(F)C(F)F)N1CCN(C(c2ccc(F)cn2)=O)C(CC(F)F)C1 Cc1cccc(C(F)(F)C(=O)N(CC(C)N(C(C2CCCN2C(C)C)=O)CC)C)c1 C1(NC(Cc2c(C)ccs2)=O)CCSC12CN(C(=O)C(C)S(N)(=O)=O)C2 C1(C(=O)NC(C)CN(C(=O)COCC(F)(F)F)C)CCN(C2CC2)S1(=O)=O N1(C(c2c(C)onc2-c2cccs2)=O)CC(NC(C2CC(C)(C)O2)=O)C(C)(C)C1 C1(C(=O)NC(C)CCNC(=O)CCOc2cccc(Cl)c2)Cc2ccccc2S1 C(=O)(CC1OCc2ccccc21)NC(C(C)(C)C)CNC(c1ccnc(O)c1)=O C(CC(C)C)(C(=O)NC1CCCN(C(=O)CC2CCCC2)CC1)NC(=O)OC C12(COC)CN(C(=O)C=Cc3cocn3)C(CNC(=O)C(=O)Cc3cccs3)(C1)C2 Cc1cc(F)ccc1CC(=O)NCC(C)N(C)C(C12CC(C)(C1)C2)=O C1(CNC(c2c(C)ncnc2)=O)CCN(C(=O)CC2CN3CCC2CC3)C1(C)C O=CN1CCCN(C(C2CSCN2C(C2CCCC2O)=O)=O)CC1 c1(C(=O)NC2C(CNC(C3CN(S(CC)(=O)=O)C3)=O)C2)cccc2c1C(=O)NC2 c1(C(=O)NC2(CC(=O)NC(C(=O)OC)(C)CO)CCC2)ccc2n[nH]cc2c1 c1(C(N(CC(C)O)CCNC(C2(C#C)CCC2)=O)=O)cc2c(C)ccc(C)c2[nH]1 N1(C(S(C2=NC(=O)NCC2)(=O)=O)=O)CCc2ccc(Br)c(F)c2C1 C1(NC(=O)C=Cc2ccccc2)CN(C(c2cc(C3CC3)ccn2)=O)CC12CC2 Cc1ccc(C(=O)C(=O)NCC2CC(NC(=O)COc3cccc(Cl)c3)C2)cc1 N1(C(C(CC)CC)=O)CC2(CCCC2N=c2[nH]c(C(F)F)nc(=N)[nH]2)C1 N1(C(CC2C(C)CN(C(c3cncnc3)=O)C2)=O)CC(C)(C)CCC1CO N1(C(C(C)(O)Cn2ccccc2=O)=O)CC2CC(C1)N(C(=O)CCN1CCC1)C2 c1(NC(Cc2n(C)nc(C)c2C#N)=O)cc(C(=O)O)cc2ccccc12 CCCCC(C(=O)N1CCCN(C(c2oc(CCC)nc2C)=O)CC1)C(C)C C1(CNC(C=CCN(C(=O)C(c2cccnc2)O)C)=O)CC(C#N)C1 c1(N)nc2ccccc2o1.c1(CN2CC(CO)N(C)CC2)ccc2ncoc2c1 O=C(C#CC1CCCCC1)N1CC(NC(C23CCC2CC3)=O)C(F)C1 C1(C2CCC2)(C(=O)NC(CNC(=O)Cc2cnccn2)C2CCC2)CC1 C1(c2nnnn2C2CC(F)(F)C2)(NCc2scc(C)c2)CCOC1C C#Cc1cc(F)c(C(N2CC3(CCN(C(=O)C(C)NC(N)=O)C3)C2)=O)cc1F c1(NC(C(C2CN(C(C3(COC)COC3)=O)C2)O)=O)ncc(Br)[nH]1 C1(NC(=O)Cc2ccco2)CCCN(C(c2ccc3cccnn23)=O)CC1F C(CN=C(NCCc1cc(O)cc(O)c1)NC(c1ccc(C(C)C)cc1)C)SC N1(C(c2cc(CC)sn2)=O)CC(C(=O)N(C)CCC2CCCCC2)OC(C)C1 N1(C(c2c(CC)non2)=O)CCC2(C1)CN(C(=O)CCCCCOC)CC(C)O2 C1(C(C)C)CC(CC(N2CCCC2(C)CNC(C23CCC(CC2)C3)=O)=O)CCO1 C1(F)(NC(COCCC=C)=O)CCCN(C(=O)C(CC2CCOCC2)OC)C1 C=CCCCCN=c1[nH]c(=N)[nH]c(=NCC2(OCCOC)CCC2)[nH]1 CC1CC(CNC(c2ncc(Cl)cc2F)=O)CCN1C(C12CSC(C1)C2)=O N1(C(c2c(OC)cc(C)cn2)=O)CCCC2(NC(=O)CSCCN(C)C)CC2C1 C1(NC(c2c(C#C)c[nH]n2)=O)CN(C(=O)C(=O)NCCOCCOC)C2(CCC2)C1 N1(C(c2ncn(CC)n2)=O)CCOc2cccnc2C1 c1(CC(=O)NC(C)C2CC2)cncnc1O.C(C(=O)NO)C1(C(C)(F)F)CC1 N#CC1(C(=O)NCc2cccc(C(=O)NC3CC4CCC(C3)C4)n2)CC2CC2C1 N1(C(C2C(OC)C2)=O)CCCC1C1CCN(C(=O)CSCC(F)(F)F)C1 C1(C)(SC2(C(=O)NCCNC(CCC(=O)c3cn(C)nc3)=O)CC2)CCNC(=O)C1 C(=O)(C(C1=CCCSC1)N(C)Cc1cnn(C)c1C#N)Nc1nnc(C(C)C)s1 CC(=O)C(C)CC(C)C(=O)NC1(C)CN(C(C2CCCC(=O)N2C)=O)C1 C(=O)(C#CC1CC(F)(F)C1)NCC1(C)N(C(c2ncc(OCC)nc2)=O)CCC1 C1(C(N2CCCC(C(=O)NC)C2)=O)COC2(COC2)C1 Cc1ccc([N+](=O)[O-])cc1C(N1CC(NC(c2cc(CO)on2)=O)C(C)C1)=O c1(C(=O)NCC2C(NC(Cc3ncc(C)s3)=O)C2)cc(C)c(O)c(C)c1 c1(C(N2CC(NC(C(C(C)C)(C)C)=O)C(F)C2)=O)ccc(C#N)nc1O C(=O)(C(C)(C)CC(=O)NCCCSCC(C)C)NCCn1cc(C(=O)OC)nn1 C=CC1(CC(=O)NCC2SCCS2)CN(C(c2cnc(N)cn2)=O)C1 C(=O)(CCCCC(C)C)NCC1(C)N(c2nnc(C(=O)OC)s2)CCC1 C#Cc1cccc(NC(=O)C(CC(C)C)ONC(=O)C2(COCC)CCC2)c1 c1(NC(C2N(Cc3cc(C)c(Br)cc3)CCC2O)=O)cc(C)c(F)c(C)c1 N1(C(c2c(C)occ2)=O)CC2(C1)C(NC(=O)C(O)CC(C)C)CCS2(=O)=O c1(OC)cc(Br)c(CNCC2CCCCC23CCC3)c(F)c1F N1(C(CCCC(OC)OC)=O)CC2CCCC(C1)N2C(c1cc[n+]([O-])cc1)=O C1(NC(=O)CN2CCSCC2)CN(C(=O)C=C2CCCCC2)C2CCCC12 CN1CCCC(F)(C(=O)NC(C2CCN(C(C3CS(=O)(=O)C3)=O)CC2)CO)C1 C1(C(=O)NOCC2CCCO2)C=CCN(C(C23CC2CNC3=O)=O)C1 N1(C(C2(OC)CCN(C(C(C)SCCCC)=O)C2)=O)CC2(CCC2)CC1C C1(NC(=O)NCC(=O)NCC=C)CCN(C(=O)CCSC(F)(F)F)CC1O Cc1ccc(C(N2CCC(C(C)NC(C3SCCS3)=O)C2)=O)c(C2CC2)n1 Cc1nc(N(C)CCN2CCOC2=O)cc(NCC2(C(F)(F)F)CCN(C)C2)n1 C1(NC(CCC2(C)CCCN2C(c2ccc[n+]([O-])c2)=O)=O)CCn2ccnc2C1 C1(C#N)(C(=O)NCC(C)(C2CC2)NC(c2ccc(-c3ccco3)[nH]2)=O)CC12CCC2 C(=O)(CC(C)(O)COC)NCC1C(CNC(c2cn(CCC=C)nn2)=O)C1 c1(C(C)=O)cc(N2CC(NC(C3CCCC(O)C3)=O)CC2C)ncn1 C(=O)(C1Cc2ccc(Cl)cc21)N1C2CN(C(C3Cc4nncn4C3)=O)CC1CC2 N1(C(CCCOC(C)C)=O)CC=CC(NC(c2ncnn2C)=O)C1 C1(CC(=O)NCC2(CSCC)CC3CC3C2)CC2(C1)CN(C(=O)C1CC1)C2 Cn1ncc(CNC(c2cc[nH]c(=N)n2)=O)c1C(=O)NCC1C(CO)C1(F)F C(N=c1[nH]c2cc(Br)cnc2s1)C1CN(C(CCOCCOC)=O)C(C)C1 N1(C(C(CCC)OC)=O)CC2CCC(C1)N2C(=O)C=CCN(C)C c1(CC(=O)NCC(C)(C)NC(c2n(CCC(=O)OC)ncc2)=O)ccc(F)nc1 C1(C(=O)NC2CN(C(c3c(C)[nH]nc3CO)=O)CC2(C)C)CCn2nccc2C1 CC(C(=O)N1CCC(CN(C)C(c2cncnc2C2CC2)=O)CC1)C(C)O C1(OC)CN(C(=O)CCc2cnc(C)s2)CCC1NC(c1cnc(O)s1)=O N1(C(=O)C=C2CCCC2)CC(CO)C2(C1)CN(C(=O)COCC(F)F)C2 C1(N(C(CC=C(C)C)=O)C)C2CN(C(c3cn(C(C)C)cn3)=O)CC12 N1(C(CCOCCOC)=O)CC(C)C(C)(CNC(=O)C(C)C(C)(C)C)C1 CC1CCCn2cc(C(N3CCCCC3CNC(=O)Cn3cnnc3O)=O)nc21 c1(C(=O)NC(CC)CNC(=O)Cn2cccnc2=O)sc(S(N)(=O)=O)cc1C N1(C(CCSC)=O)CCC2(CCCCC2NC(c2cc(F)c3c(c2)CCC3)=O)C1 N1(C2CCN(C(c3oc(CC)c(CC)c3)=O)CC2)CC2CCC(C1)NC2 c1(C(=O)NCC(C)N(C)C(C2CC2c2nncn2C)=O)ccc2nc(O)oc2c1 C(=O)(CS(=O)(=O)CC1CCCO1)N(CC(CNC(CCSCC(C)C)=O)C)C C1(C(=O)NC2CC(C(F)C(N3CCC(CSC)CC3)=O)C2)CCCN1C=O Cc1cc(Cl)ccc1OCCC(N1CC2CCC2(NC(=O)C=CC2CCC2)C1)=O c1(CCCN(CC(CCC(=O)OC)O)C2CC2)c[nH]c2ccccc12 C1(C)(CNC(C2ON=C(C)C2C)=O)CC(F)(F)CN1C(=O)CCn1cncn1 c1(OCC)cnc(C(N2CC=CC2CNC(=O)C(C)CC2CCCCC2)=O)cn1 C(C1CCCCC1)=C(C(=O)NC(CC)CNC(=O)COC1(C)CCC1)C c1(C(=O)NCC(CCOC)NC(=O)C(F)=CCCF)c[nH]c2cc(OC)ccc12 C(c1ccc(F)cc1)=CC(=O)NC(C1(O)CN(C(C2CCCN2C)=O)C1)C CCC(CC(=O)NC(C(N1CC(O)(CN(C)C)C1)=O)C1CC1)C1CC1 c1(C(=O)NCCC2(NC(CC(C)(C)OC)=O)CCC2)sc2ccccc2c1C C1(CC=C)(NC(=O)CNC(C2CC2OC)=O)CCCN(C(c2cc(C)ns2)=O)C1 N1(C(c2nc(C(C)C)oc2)=O)CCC(C(=O)NCC(O)CC(C)(C)C)C1(C)C n1(CC)nc(C)cc1CN=C(NC1CCN(C(=O)NC2CC2)CC1)NC1CC1C Cc1ccnnc1C(N1CCCC1C(C)(C)C(=O)NC1CCOCC1C)=O C(=O)(C1=CCN(C)C1)NC1(CF)CCN(C(c2c(C)nc(C3CC3)s2)=O)C1 C1(C(=O)NCC(C)NC(C2CC2C2CCCO2)=O)(COC)SCCCS1 N1(C(C(=O)NCC2CC2)=O)CC(C2CN(C(C3CC4CCCCC4O3)=O)C2)C1 C(=O)(C(O)CN1CCCC1)NCC1CC(C(N(C)CCn2cncn2)=O)C1 c1(C(N2CC(NC(c3c(OC)ccc(O)c3)=O)C(O)C2)=O)cc(Cl)cc(Br)c1O C12CC3(C1)CC(C3)NC(=O)c1c(C)nc(s1)N2.C(=O)(CCN1CCC1)NC1CC1 c1(C(=O)NCc2n(C)nc(CN3CCCC3)c2)cc(C#N)c2ccccc2n1 c1(N(C(C(=O)NCCOC)C2CC2(Br)Br)CCC#C)ccc(Cl)cc1OC c1(C(=O)Nc2c(Br)cc(Cl)nc2Cl)cc(-c2cccnc2F)c2[nH]ccc2c1 c1(CCC)nc(C(=O)NC(C)CNC(=O)COC2(C)CCCC2)cs1 c1(OC(CC)C)ccc(C(=O)NCC23CC(NC(=O)C(C)O)(C2)C3)cc1 c1(CC(=O)NC2CCC(NC(c3c(C)nns3)=O)C2)ccc2[nH]ccc2c1 C(=O)(CCC(C)CN(C)C)N1C(CCNC(c2ccc(OC)cc2)=O)COCC1 C(c1ccc(C)c(Cl)c1)=CC(=O)NC(C(=O)NC(CCOC)CNC(C)=O)C c1(S)ccccc1Cl.C1(C(C(=O)CSCC(F)F)=O)(CO)CCCC1 C1(CC(=O)NCC(c2ccccn2)NC(c2cccnc2)=O)CCCC(C2CC2)O1 C(=O)(C1=CCC(NC(C2CCOCOC2)=O)C1)NC1CN(CC)CC1C c1(OCC)ccc2cc(C(=O)NCCC3CN(C(=O)CCN(C)CC)C3)[nH]c2n1 C1(CC(=O)NC(CC(=O)NC)(C)C(=O)O)CCN(C(=O)OC(C)(C)C)CC1(F)F C(=O)(C#CC1(C)CCCO1)NCC(CC(C)C)(C)NC(c1cc(C(C)C)no1)=O C1(CC(=O)N(C2CCCC2O)C)CCCC1CNC(c1ccc[nH]1)=O C1(C2CCN(C(C3CC4CC4C3)=O)CC2)(NC(c2occ(S(C)(=O)=O)c2)=O)CC1 N1(C(CCCSC)=O)CCC2(C)CN(C(=O)CCC3NC(=O)NC3=O)CC12 N1(CN(C)C(C2(NC(=O)CN(c3ccsc3)C)CC2)=O)C(=O)NC(=O)C1=O N1(CCNC(C2(C)CCCO2)=O)CCN(C(C2OCCO2)=O)CC12CCC2 Cc1cc(CNC(=O)Cn2cccnc2=O)oc1C(=O)NC1(CF)CCC1 C(CO)(CC(O)C(C)(C)C)NC(=O)NC(c1cccc(OC)c1)c1ccccn1 CN(C)S(=O)(=O)N1CCc2ncnc(N3CCCC(c4ccc(F)cc4)C3)c21 C1(C(=O)NC23CC(NC(=O)CCc4cnco4)(C2)C3)CC2OC(=O)OC2C1 CCC(CC(F)F)C(=O)NC1(CCO)CCOCC1 c1(C(N)=O)cc(C(=O)CC2CCN(C3CCCSC3)CC2)ccc1OC(F)(F)F C(=O)(C(CC(C)(C)C)OC)N1CC(C#C)(C(=O)NC2(CO)CC(O)C2)C1 O=C1CC(=O)NC(C(N2C3CCC2C(CNC(c2cscn2)=O)C3)=O)C1 N1(C(c2cc(CC)ncc2)=O)CC(NC(c2sc(C)c(C)c2C)=O)C2CC2C1 C1(C(N2C(C3(C(=O)NCC(CO)OCC)CC3)CCC2)=O)CCCC(C)CC1 C1(NC(=O)CCc2cncc(Br)c2)CCCN(C(=O)C2=CCSC2)CC1 C1(C(N2CCC(NCC=CCOC)C2)=O)CC(O)CN1C(C)=O C1(NC(c2n(C=C)ncc2)=O)(CC)CCCN(C(c2n[nH]c(C)c2O)=O)C1 c1(OC)ccc(F)cc1C(=O)NC(C1CCCC1)CNC(C1CCC1F)=O N1(Cc2cnn(C3(C)CCN(C(C(C)(C)OC(C)C)=O)C3)c2)CCS(=O)(=O)CC1 c1(C(=O)NC2CCCC2CNC(C2(c3ccsc3)CC2)=O)cc2ncccc2[nH]1 c1(C(=O)NC2CCCN(C(C(CC)(C)CO)=O)CC2)cc(N)c(C)cc1Cl C1(C(=O)NC(CCOC)CNC(=O)CC2CS(=O)(=O)C2)CCC(C)CC1 c1(C(=O)NCC2(O)CN(C(c3c(C)nsc3)=O)C2)cc2ccc(Br)cc2o1 C1(NC(C(C(C)O)(F)F)=O)CC2(CCC(Nc3ncc(Cl)cn3)CC2)C1 c1(NCCCC)ccc(S(=O)(=O)N2CCCC(OC)C2C)cc1NC(C)=O CCC1=NOC(C(=O)NCCn2cc(CNC(C3CN(C(C)=O)C3)=O)cn2)C1 c1(C(=O)NCCCCCN(C(C2CC(C)OC2=O)=O)C)cnc2ccccc2c1 C1(NC(c2c(SC)scc2)=O)CCN(C(c2cc(F)n[nH]2)=O)C(C2CC2)C1 Cc1conc1C(=O)NC(C)(CNC(c1ccn(CCN(C)C)n1)=O)C1CC1 Brc1cnc[nH]c1=NCc1ccc(-c2ccccc2)s1 c1(N2CCC(OC(c3nc(-n4cnc(=N)[nH]4)sc3)=O)C2=O)cc(F)cc(F)c1 N1(C(c2c[nH]c(=N)o2)=O)CCCC(C2CCCN(C(c3cnco3)=O)C2)C1 c1(C(=O)NC2CC(C(N3CCC(C#N)C3)=O)C2)cc(O)c(O)c(Cl)c1 c1(C(N2CC3CN(C(=O)COCCF)CC3C2)=O)ccc2occc2c1 N1(C(C(CC)=CC)=O)CCC(NC(c2ccoc2Cl)=O)C1C(C)(C)C CC1CN(C(=O)C=Cc2cccnc2)C(C)CN1C(=O)CCC1(C)CC1 c1(C(=O)NCCn2nnc(=N)[nH]2)nc2c(s1)CCCC2.C12C3CN(CC13)C2=O Cc1c(C(=O)NC2CCCCC2NC(C2C3CCC23)=O)cnn1CCC(C)C N1(C(CCCC)=O)CCN(C(=O)C(O)C(F)F)C(CO)C1 N1(C(CCC=C)=O)CCN(c2nc3cc(Br)cnc3s2)CC(C)(F)C1 CC1(C)CCC(C)(NC(C2CCCCN(C(c3cccc(F)c3N)=O)C2)=O)CC1 Cc1cccc(CCC(=O)N(CC(C)(C)CNC(C2CCC2C)=O)C)c1Br c1(C(=O)NCC(CC)NC(c2coc(C)c2)=O)cc(C(=O)OC)cc(C)c1 N1(C(c2c(CC)n(C3CCC3)nc2)=O)CC2CN(C(=O)C(OC)OCC)CC2C1 CCCCCCC(C)C(=O)NCCCC1CN(C(c2[nH]nnc2CC)=O)CCO1 c1(C(=O)NCC2C(CC(=O)NCCCSC)C2)c(C)cccc1Cl CC(C)CC(C)CC(=O)N1CC(C(N2CCC(C)C2)=O)C(C2CC2)C1 N1(C2CCN(C)CC2)CCC(N=c2nc3c(ncn3C)c(NC3CC3)[nH]2)CC1 CC1CCc2ncc(C(=O)NCCCN(C(=O)CC3CCCN3C)CCO)n2C1 N1(C(C(c2ccccc2)SC)=O)CCCCC1CNC(c1nocc1C1CC1)=O CCC(CC(=O)N(C(C)C(=O)NC(C)Cn1cccn1)C)OC C1(CNC(Cc2c(C)ccc(F)c2)=O)CC2(CCC2)CN1C(=O)C(F)=CCCF C1(N(C)C)CCN(C(=O)COC2CCN(C(=O)CCCF)C2)CC1 c1(CC(=O)NC(C)C(C)NC(=O)C2=CCCCC2)ccc2[nH]ccc2c1 N#CC1(C(=O)NC2CN(C(C3CCC4(CC3)CC4)=O)C2)CC12CCCC2 c1(C(=O)NCC(CC)NC(C2CC23CCC3)=O)c(C)cc(OC)cc1F Cc1cn2cc(C(=O)NCCC3(CNC(=O)C(C)C(F)(F)F)CC3)nc2s1 CN1CCC(OCC(=O)NCC2(O)CCN(C(=O)Cc3ccc(F)cc3)C2)CC1 C(=O)(C1=NN2CCCN=C2N1)NCC(C)NC(=O)CC1(O)CCN(C)CC1 C1(NC(c2scc(C)c2)=O)CCN(C(c2ncc(C)o2)C)C(C)C1 N(C(=NCCC(C)N1CCOCC1)NC1CCC1)CC1(CC)CCCCCC1 c1(CN(C(=O)NC2CCCO2)Cc2c(CC)[nH]nc2Cl)cc(Cl)ccc1Cl C1(NC(C2(Br)CCCCC2)=O)CCC2CC1CN2C(C12CC3CC1C2C3)=O N1(C(Cc2cn(CC)nc2)=O)CCC(NC(=O)Cc2cccc(C)c2F)C12CC2 c1(CNC(c2nc(C(=O)N(C3(CC)CCC3)C3CC3)co2)=O)ccc(Cl)cn1 C(=O)(CS(=O)(=O)CC(=O)NCC(O)CNC(C1(O)CC2CCC1C2)=O)OC C1(C(=O)NCC2N(C(c3c(N)nccn3)=O)CC(F)(F)C2)CCn2nnnc2C1 C12(NC(C(C)(C)SC)=O)CC1CN(C(c1nc(C)sc1C)=O)C2 c1(NC(Cn2nc(C)c(Cl)c2C)=O)cnn2cc(C#N)cnc12 C(=O)(C#CC1(C)CCCO1)NCCC1CCN(C(C(C(C)C)C)=O)CC1 C1(O)(CN2CCC(N(C(=O)C(C)CSC)CCC)C2)CN2CCC1CC2 C12(NC(c3c(COC)cc[nH]3)=O)CCCC1N(C(=O)CCOC)CCC2 Cc1cccc(C(=O)NCCN(C(C23CC(C2)C(C(N)=O)CO3)=O)C(C)C)c1F C1(C(=O)NC2CCCN(C(C3N(C)CCC3)=O)C2)C2C3CC4C1C1C2CC3C41.CC c1(C(=O)NC2CC(C)(NC(=O)C(F)(F)C(F)F)C2)cnc2c(c1)CCCC2 C(c1ccc(NC)cc1)=CC(=O)N(CCOCCN(C(C(CC=CC)C)=O)C)C c1(NC(=O)OC(C)(C)C)cc(O)nc(NCc2ccnn2-c2ccccc2)n1 n1(CC(=O)OC2CCC2c2cncc(Br)c2)cc(F)ccc1=O c1(NC(C(C2CCN(C(c3ccc[n+]([O-])c3)=O)CC2)C)=O)ccc(Cl)nc1 c1(NC(=O)NC(c2c(OCC(F)(F)F)cc(Cl)cc2)CO)ncc2n1CCCC2 C12(NC(C(CC)OC)=O)CC(C)(C1)OC21CN(C(c2cncc(Br)c2C)=O)C1 c1(NC2(c3nnnn3CC)C(CCCC)CCC2)c(CC)ccc2[nH]ccc12 C1(CCCCC)CCC(C(=O)NCCC(C(C)C)NC(c2cc(C)[nH]n2)=O)CC1 C1(CCC)CCCCC1C(=O)NC(CCC)C1CC1.C12CCN1C(=O)NC2 CC1CCCC(C(=O)N(CCCCNC(c2cc(Cl)ns2)=O)C)CC1 Cc1cc([N+](=O)[O-])cc(C(N2CCC3(NC(=O)CCC4CCC4)CCCC23)=O)n1 c1(CCC(=O)N(CC(CC)NC(=O)C(O)C(C)C)CC)nc2ccccc2s1 CCCCCC(CC)C(=O)N(CC(=O)NCCc1nccn1C)CC(C)C C(=O)(CC1=CCN(C(C2CCC2)=O)CC1)NCc1c(CC)nccn1 CCCC(C)(C)CC(=O)NC1CCOC(C(=O)NC2(C)CC(O)(CO)C2)C1 C1(NC(C2ON=C(C)C2)=O)C2CN(C(=O)Cc3cncnc3)CC12 CC(=O)CCCC(=O)NCC1C(C)CCN1C(=O)Cn1ncc(O)nc1=O c1(C(=O)NCCOCCCN(C(c2cnc(CC)s2)=O)C)cn(C)c(O)n1 C(=O)(C(C)CCCC)NCC(N1CCN(C(CC(C=C)C)=O)CC1)C(F)F c1(OC)cccc(Cl)c1C1(C(=O)NCC(C(C)C)NC(C2CCN(C)C2)=O)CC1 C1(O)(CC(C(=O)NCC2C(C)OCC2)NC(=O)COCC2CC2)CCCCC1 CC#CCC(C(=O)NCCN1CC=CCC1)NC(c1cc(OC)cnn1)=O C(=O)(C(F)C(C)COCC)N1CC(CC=C)(C(=O)OCC)C1.c12sccc1C2 N=c1[nH]c(=NCC2CCCC2C(F)(F)F)[nH]c(=NCc2cccnc2Br)[nH]1 N1(C(c2cn(CCOC)nc2)=O)CC2CN(C(=O)Cc3nc(C)no3)C2C1 N1(CCN2CCCC(F)(F)CC2)CCC2(CC1)CC2(C)NS(C)(=O)=O CC1CC(NC(=O)CC2COCC2O)CCN1C(c1ccn(C(F)F)n1)=O C1(C(=O)NC2CC(C)(C)N(C(=O)Cc3ccccn3)C2)CCc2n[nH]cc2C1 c1(C(=O)NCC2(CNC(C=Cc3c(C)cco3)=O)CC2)n[nH]c2ccc(F)cc12 Cc1cc(C(N2CCN(C(=O)Cc3cc[nH]c3)C(CCO)C2)=O)c(C)nc1C C1(CC(N2CC(F)(C(=O)OC)C2)=O)CC2(CCOCC2)CN1 c1(NC(N(C(C)Cc2ccccc2)CC)=O)cncc(Cl)c1 C12(C(=O)NCC3C(NC(CCCN(C)C)=O)CCC3)CCC(CC1(F)F)C2 C1(CC)CN(C(=O)C(Cc2ccco2)NC(C2C3CCC(F)C23)=O)CCCO1 C1(N(C(=O)C(F)=C2CCCC2)CC)CCCN(C(=O)Cn2nnc(=N)[nH]2)C1 c1(C2CC(C(=O)NC(c3n(C)ccn3)C(F)(F)F)C2)cccc(C#N)c1 Cc1sc2cncn2c1C(=O)NCC(n1cc(CCCC(C)O)nn1)C C1(NC(c2scc(C(=O)OC)n2)=O)CS(=O)(=O)CC1NC(c1cc(C)oc1C)=O N1(C(Cc2c(C)nc[nH]2)=O)CCC2(CCC2)C(NC(=O)CC2CCCC(=O)N2)C1 C1(CNC(c2c(OC)scc2)=O)CCN(C(=O)CN2CCOC2=O)CC1C n1(CC(N2CC(C)N(C(c3ncccn3)=O)CC2)=O)ncc2ccc(F)cc12 C1(NC(CCCC=C)=O)CCN(C(C2OCCOC2C(F)(F)F)=O)CC(C)(C)C1 CC(C)CC(C(=O)NCCn1ccnn1)ONC(C1(C)CC2CCC1O2)=O C=CC(CCC)CC(=O)NCC1CCCCN1C(c1cn(CC)nc1C1CC1)=O C1(CC)CCCN(C(C2C=CCN2C(=O)C=C(C)C(F)F)=O)C1 c1(Nc2cccc(F)n2)cnc(Br)c(Cl)n1.N12CCCC1C(=O)NC2=O c1(C(N(C2CCCN(C(C3N(C)CCC3)=O)C2)C)=O)cnc2cc(Br)ccn12 c1(OC)ccc(C(=O)NC2COCCC2NC(c2cn(C3CC3)cc2C)=O)nn1 C1(NC(C2CCN(C(C)=O)CC2)=O)C(C)CCN(C(=O)CSC2CC2)C1C C12(NC(COCCOCC)=O)CCCC1N(C(=O)Cn1nc(C)cc1C)CCC2 Cc1nnc2n1CCCC2C(=O)NCC(C)N(C)C(C12CC3CC1C2C3O)=O N1(C(C(C)(C)OC(C)=O)=O)CC2(C1)SCCC2NC(c1cnn2c1CCC2)=O N1(CC(=O)NC(CC2CCN(CCCNC(CCC)=O)C2)=O)CCCCCC1 c1(OC)cc(OC)c(C(N2CCCC2c2cn(C3(C(=O)O)CC3)nn2)=O)cc1OC O=S(=O)(c1ccc(NCC2CN(c3nncs3)C2)c(F)c1)NC1CCCC1O c1(NCc2ccc(OCC)cc2)cc2ccc(-c3cc(F)cc(C#N)c3)cn2c1 CC(C(=O)N1CC(CC(C)(C)CNC2(C)CSC2)C1)C(=O)OC(C)(C)C C1(CC(N2CCCC(N(C(CC(C=C)C)=O)C)C2)=O)CC(C)(C)OC(C)(C)C1 C#Cc1ccc(CC(=O)NC(C)(C)C(C)NC(=O)Cc2c[nH]ccc2=O)c(F)c1 C1(CNC(c2cncc(C)n2)=O)CN(C(=O)C(C)C(C)O)CCC1C C(=O)(C(Cc1cnc[nH]1)NC(=O)Cn1cccc1)NCCC1(C)CC1 N1(C(CC)C(=O)NCC(=O)N(CC(C)C)C(C)C)CCc2ccccc2C1 C(=O)(C#CC1CCOCC1)NCCC1CCC(C)N(C(=O)CCCF)C1 C1(C(=O)NC2CN(C(C3(Br)CC3)=O)CC2C(F)F)CC2C=CCC(C1)C2 c1(SC)ccc(Cl)c(C(=O)NC(C)C(C)NC(=O)C(C)(C)n2cnnn2)c1 c1(N(C)C)ccc([N+](=O)[O-])c(C(=O)NC(c2cncnc2)CC2CCC2)c1 c1(C(=O)NC(C)C(C)NC(C2(C#N)CCOCC2)=O)cccc(OC(F)(F)F)c1F c1(NC(=O)CSCC(F)(F)F)cc(N2C3CCC2CC3)nc2ccccc12 C12(C(N(c3cncc(C#N)c3)C)=O)CCC(NC(c3sccc3Cl)=O)(CC1)C2 c1(OC)cc(C(N2CCC(CN(C)C(c3cncnc3)=O)CC2)=O)c(N)c(C)c1 n1(CC)nnc2c1CCC(C(N1CC(NC(=O)CC3(C(F)F)CC3)C1)=O)C2 C(=O)(CC(C)(C)CCOC)N1CCC(C(=O)NC(C2CCOCC2)C#C)OCC1 Cc1nnc2n1CC(C(N1CCCC1Cc1cn(CC(C)N(C)C)nn1)=O)CC2 CC(C)C1CC(=O)NCCC2CC(C2)C(=O)SCC(=O)N1.C(C)(C)(C)OC1CC1 N1(C(C2CCN(C(C)=O)C2)=O)CC2CN(C(=O)C=CC3CC3)CC2C(F)(F)C1 C1(C(N2C(CNC(C3C(C)(C)CCO3)=O)CC(O)C2)=O)CCC2CC1CO2 c1(C(N2CCC2(C)CNC(=O)OC(C)(C)C)C(=O)NCC=C)ccc(F)cn1 C1(C)(C(N2C(CN(C(=O)CCN3CCCCCC3)C)CCC2)=O)COC(=O)C1 Clc1cc(Cc2nc(C3CC3)nn2C2CCCCC2)cc(Cl)c1 N1(c2ncnc(OC)c2C)CCC(C2CC2)(CNC(c2cnc3n2CCC3)=O)C1 C1(C(=O)NCC(COCC)C)C=CCN(C(C2CC(=O)C2)=O)C1 N1(C(C=CCC)=O)CCC(C2CCCN(C(c3c[nH]cc3Br)=O)CC2)CC1 C1(C(N2CC(O)(CC=C)C2)=O)CN(C)CCN1C(=O)CCCOCC N1(C(c2cocn2)=O)CCC(C(N2CC(c3cccnc3)C2)=O)(CF)C1 N1(C(C(CCC)N(C)C)=O)CCN(C(=O)C(C)O)CCC1C c1(CNC(=O)CO)ccc(C)cc1.C1(C(=O)NC2CCC2CF)CCCN1CC c1(CNC)ccc(C(C)C)cc1S(=O)(=O)Oc1cc(C)c(F)c(C)c1 C#CC12CCC(C(N3CCC(C)(NC(c4cc(Br)no4)=O)CC3)=O)(CC1)CC2 C(Cc1ccoc1)(C(=O)NCCCCCNC(C)=O)NC(C)=O.c1(C=O)cccs1 C=CCC(F)(F)C(=O)N(CC(=O)Nc1cn(C)nc1C(C)C)CC1CC1 C=C=CC(C)C(=O)N1CCOC(CN(C)C(c2cnn(CCC(C)C)c2C)=O)C1 c1(OC)cnc(C(=O)NC(Cc2cn[nH]c2)C(=O)N2CCC(C(F)F)C2)cn1 C1(C)(C(=O)NCC(C)CNC(=O)CC2COCCO2)CC2CCC(C1)S2(=O)=O c1(C(C)C)cc(C(=O)NC2CC(C(C)NC(=O)CCC(C)N(C)C)C2)nn1C CCCCC(CC)N(C(=O)Cc1csc(C(C)C)n1)C1CC1.C1CCO1 C(C(N=[N+]=[N-])C(=O)NC1C(n2cc(NC(=O)C(C)CCO)nn2)CCC1)OCC c1(C(=O)NCC2C(C)CCN(C(C3(C(N)=O)CC3)=O)C2)cccc2ccn(C)c12 C1(CC(=O)NC2CCCN(C(Cn3ccc(C)n3)=O)CC2)CCCC2(CCC2)O1 c1(C(=O)NC(CNC(c2cnsc2)=O)CO)csnc1Br C(CCCC(=O)N1CCCCC1C(=O)N(CC(O)COC)C(C)C)OC c1(C(=O)NCC2N(C(C3=NOC(C(C)(C)C)C3)=O)CC2)cc2cc(O)ccc2[nH]1 N1(CCC(C(=O)OC)(C)O)CCNCc2cccc(Cl)c21 Cc1c(Cl)ccnc1C(N1CCC(CF)(NC(c2ccnc(S)c2)=O)C1)=O C1(CCCC=C)NC(=O)N(C(c2ccc(Br)cc2C)C)C1=O C1(NC(c2csc(C(F)(F)F)c2)=O)CS(=O)(=O)CC1NC(c1cnsc1)=O Cc1cccc(C(=O)NC2(CC(=O)NCC3(CCO)CC3)CC2)c1N CCC(CC)CCC(=O)NCC1(C(N)=O)CN(C(=O)CCCS(C)(=O)=O)C1 c1(C(N(C2CC3CNC2C3)CC2(C)OCCO2)=O)ccc(N)c(O)c1 c1(CC(=O)NC2CCCN(C(CC3(C#N)CC3)=O)CC2)cc2ccccc2s1 c1(OCC)ccc(C(=O)NC(CNC(C2CC2Br)=O)C(C)C)c(F)c1F C1(C(=O)NC(CCNC(CCCCSC)=O)C(C)C)(OC)CC2CCC1C2 c1(-c2ccc(C)o2)nc(CCC(=O)N(C)Cc2ccccc2)n(CCC(C)C)n1 c1(C(C(=O)NCCC(C)N(C)C(c2cc(CO)[nH]n2)=O)O)ccccc1 n1(C(C)C)ncc2c(N3CCC(F)(CNC(C4CC45CC5)=O)CC3)ncnc12 Cc1ccc2[nH]nc(C(=O)NC3CCN(C(=O)C(F)=C4CCCC4)CC3C)c2c1 c1(C(=O)NC2CCN(C(CN(C)CC)=O)CC2C)ccc2cc(F)c(F)cc2n1 N1(Cc2c(C(=O)OC)cccc2)CC2C=CC2C1C(=O)OC c1(NC(=O)Cc2ccccc2NC(C2(O)CCCC2)=O)nc2ccccn2n1 c1(C(N2CCCC(c3cc(C(N)=O)on3)C2)=O)cccc2c1OCCC2 C(=O)(C(CO)C(F)(F)F)N1CCC(CC#C)(C(N2CC(n3ccnn3)C2)=O)C1 N1(C(c2ccc(CC)[nH]2)=O)CCCC(C)(CNC(=O)Cc2c[nH]nc2O)C1 c1(C(N2CCC(NC(c3cc4c[nH]nc4s3)=O)C2)=O)ccc([N+](=O)[O-])cc1O Cc1ccc(F)cc1S(=O)(=O)N1CC(CO)C1.c12ncc(cc1[N+](=O)[O-])c(=O)[nH]2 Cc1cnc(C2(NC(=O)CC3CCCN3C(=O)CCOC3CCCC3)CC2)[nH]1 c1(CN2CC(CNC(=O)Cn3cc(Cl)cn3)OCCC2)cccc2c1CCOC2 NS(=O)(=O)c1ccc(CC(N)CC(=O)Nc2nnc(-c3ccc(Cl)c(Cl)c3)s2)cc1 C(=O)(CC(C)P(C)(C)=O)NCC(C1CCN(C(c2ccc(C)c(N)c2)=O)CC1)C C1(C(N2CCCCC2CN(C)C)=O)(CC)CCCN1C(c1cnsc1)=O c1(C(C)C)cnc(Cl)[nH]c1=NCC1(C(=O)N(C2CCCC23CC3)C2CC2)CCCC1 C(=O)(C1CCc2ccccc21)N(CCC(=O)NCCCCCCO)C1CC1 N1(C(COCC)=O)CC2(CNC(c3ccc(NS(C)(=O)=O)cc3)=O)CCC1CC2 c1(C(=O)NC(CCNC(C2C(CC)N(C)CC2)=O)C)occ2c1CCCC2 N1(CC(C)C)CCCC(N(C(C2CN(C(C3CC=CCC3C(C)=O)=O)C2)=O)CC)C1 c1(C(N2CC3C(NC(C(c4ccn(C)c4)C)=O)(C3)C2)=O)cccc2c1CCC2 Cc1nnc2cnc(C(=O)NCC3C4CN(C(C5CC6CC5C6)=O)CC34)cn12 c1(C(=O)NC2C(NC(=O)Cc3ccc(Br)nc3)CCC2)ccc(Cl)c(F)c1 C1(C(N(CCN(C)C(c2cc[nH]c(=N)n2)=O)C)=O)CC2(CCO1)CC2 C(C1CCCCCC1)=CC(=O)NC1CC1CNC(C1COC2(CCC2)C1)=O Cn1cc(C(=O)NC2CC3(C2)CC3NC(c2ncccc2F)=O)nc1C(F)F N1(C(C(C)(C)N(CCCO)C(C2CCC2)=O)=O)CCC(C2(O)CC2)CC1 NS(=O)(=O)c1ccc(C(=O)NC2CC(CNC(C3CCC4C3C4(F)F)=O)C2)nc1 N1(CC(N2C(C(C)NC(=O)CSC3CC3)CCCC2)=O)CCC(=O)NC1=O C(C(O)CC(=O)NC(C1CSC1)C)NC(C(C)SC(C)C)=O c1(C(=O)NCC2N(C(c3c(C)sc(Br)c3)=O)CC2)cc2c(s1)CN(C)CC2 N1(C(CC(CC)(F)F)=O)CC2(CNC(C3CCCOC3)=O)CC1CCO2 C(c1ccc(Cl)c(OC)c1)=CC(N1CCC(N(C(C=C(CC)CC)=O)C)C1)=O Cc1cc(C(N2CCN(CC3(C4CCC4)CCC3)CC2)=O)c(C)n1C c1(C(=O)NC(CC)CNC(c2csc(O)n2)=O)cc(C2CCCC2)n(C)n1 O=C1CCC(C(=O)NC(CC2CC2)CC(=O)NCc2cncnc2)CN1 C(=O)(CC(F)(F)F)NCCCN(CC(=O)OC)C(C1CCCN1C(=O)C(C)C)=O C1(CCO)(NC(C2CC(N(C)CC)C2)=O)CN(C(c2cnc(C(C)C)o2)=O)C1 S(=O)(=O)(c1ccc(Br)cc1Cl)N(C)CC1CN(C(c2cc(O)cc(O)c2)=O)C1 c1(OC)cscc1C(=O)NCCC1CC1C(=O)NC(c1cnn(C)c1)CO C1(NC(c2cc(CC)c(C)s2)=O)CN(C(=O)CN2CCOC2=O)CC(C)(C)C1 n1(CCOC)cc(C#CC(C)(C)NC(c2cccc([N+](=O)[O-])c2I)=O)nn1 c1(C(N2C3C(C(N4CCC(NC(C)=O)C4)=O)C(C3)C2)=O)cccc2ccccc12 c1(SCC)ccccc1-n1cc(CC2CCCN(C(C3CCOC3)=O)C2)nn1 C(c1cnccn1)=CC(=O)NCCC1CCN(C(C(C)(C)c2ccc(Cl)s2)=O)C1 C1(NC(CCn2ncc(C)c2)=O)CCC(C(N2CC3CC2CS3)=O)CC1 c1(CC)conc1C(=O)NC1CC(C(=O)N(C)CCOC(F)F)C1 C(=O)(C(C1CC(NC(=O)CSCCC(C)C)C1)N(C)C)NCCOC c1(NC(N2CCC3CN(CC(=O)OCC)CC32)=O)cc(C)c2sccc2c1 C1(NC(C=C(C)C)=O)(CO)CCCN(C(=O)CCN(S(C)(=O)=O)C)C1 c1(CC(=O)N(CC(CC)NC(C2C3CC(=O)CC23)=O)C)cc(C)cc(F)c1 C1(C(=O)NCC(CNC(c2cc(C)nnc2)=O)(C)C)CCC(F)(F)CO1 c1(CC)[nH]nc(C(=O)NCC(CCNC(=O)C(C)N(C)C)OC)c1[N+](=O)[O-] C1(NC(c2nc(C)nc(O)c2)=O)CCC2(CC1)CN(C(c1ccncc1N)=O)C2 C12(C(=O)NC3CN(C(=O)CN4CCCC4=O)CC3O)CCC(C(F)F)(CC1)C2 c1(C(N2CCC(CN(C(c3cccc(C)c3F)=O)C)C2)=O)cc(F)c(C)cc1Cl c1(CN(C)C(C2CC3CC2C3)=O)nc2ccccc2n1-c1ccccc1 N1(C(Cc2cccc(OCC)c2)=O)CCC(NC(=O)CSCC(C)C)C(C)C1 c1(C(N2C(C(N3CC4CCC3C4)=O)CC(OC)C2)=O)cnc2ncccn12 C1(NC(C2CN(CC(C)C)C(=O)C2)=O)CC2CCC(C1)N2C(C1CCCCO1)=O C1(COC(c2occ(C(=O)OC)c2)=O)CC(OC)CN1C(c1ccnc(O)c1)=O N1(CCNC(C2(C)CC2(F)Cl)=O)CCCN(C(C2(n3cncn3)CC2)=O)CC1 C1(C(C(=O)NCCCCCC)(C)C)CCCN(C(=O)C=Cc2cnccn2)C1 C=C(C)CC(C(=O)NC)NC(C1(COC)CC1)=O N1(C(=O)CC2CC2)CCC(C2CCCC2)(c2cn(CC3CNC(=O)CO3)nn2)C1 N1(C(C(C)OCC2CC2)=O)CC2(C1)CN(C(=O)C(F)CCC(C)(C)C)CCO2 N1(C(c2cc(C)nc(C)c2)=O)CCC(C(=O)NC2CCC2(C)C)=C(F)C1 c1(SCC)cc(Cl)c(NC(=O)OC(C)(C)C)nc1C.C12CCC(C)(C)CN1CC2 N1(C(CNS(CC)(=O)=O)=O)C2CCC1(CNC(c1ccc(C(F)F)cc1)=O)CC2 C[Si](C)(C)c1ccc(C(N2CC3(CCN(C(=O)CC4CC4)C3)C2)=O)o1 c1(CC)onc(C(=O)NCC(C2CCOC2)NC(C2(C)CC2)=O)c1C N1(C(=O)C(F)CC2CCCC2)CCC2(CC1)CN(C(C1(O)CC3CCC1C3)=O)C2 C1(NC(=O)CN2CCCC2=O)CC2CC1CN2C(=O)CN1C(=O)CCC1=O CC(=O)CCCC(=O)NCC(CO)NC(=O)CC1CSCCS1 c1(NCCc2nc(C)[nH]n2)ccc(S(=O)(=O)N(C(C)CC#N)CC(C)C)cc1Cl c1(C(=O)NCC(CNC(c2cn3ccsc3n2)=O)OC)cnc2ccncc2c1 c1(CN(C(c2ccc(C)o2)=O)CCNC(=O)NCC(C)C)cccc(Cl)c1 c1(C(=O)OC)nccnc1C(=O)C(c1c(C(C)N)noc1)=O.C(CC(N)=O)N C(=O)(CCCCC(C)CC)N1CC(C(=O)NCCCCC=C)C(C)(C)CC1 Cc1c(C(N2CC(NC(c3csc4ccccc34)=O)C2)=O)oc2ccc(F)cc12 c1(C(c2n(CCOC)nnn2)NCCC2CC(F)(F)C2)nc(Br)c2ccccn12 O=C(C1CCCn2cnnc21)NCC1CCN(c2ncnc3ccc(O)nc23)C1 N1(C(C(C=C)O)=O)CCC2CCC(C1)N2C(C1CCC(=C2CCC2)CC1)=O c1(C(CNC(=O)C2=CCCCC2)NC(C23CCC(CC2O)C3)=O)cc(F)cc(Cl)c1 CC1(C#CC(=O)N2CC(C3(NC(=O)CCc4ccc[nH]4)CC3)C2)CCCO1 c1(C(C(=O)NC(CN(C(C2C(C(=O)OCC)C2)=O)C)(C)C)C)ccccc1OC c1(NC)cccc(C(=O)N(C2CCN(C(=O)CCc3cnc(C)s3)C2)C)n1 c12ccc(cn1)c(=O)[nH]2.N1(CC)CCN(CC(=O)Nc2ccnc(SC)n2)CC1 C(c1cccc(C#N)c1)=CC(N1CCC(C)C1c1noc(-c2ccccc2)n1)=O C(=O)(C#CC(C)(C)O)N(CCNC(C(C)Sc1ccc(C)cc1)=O)C(C)C C(c1ccnn1C)=CC(=O)NCCN(CCC)C(C1COCCC1C)=O C(CCN=C(NCCN1CCN(C)CC1)NC(C)CC(F)F)N1CCC(SC)C1 CC1(C)CN(C(C2(c3cccs3)CCC2)=O)CC1N=c1cnc2ccccc2[nH]1 C1(CC)(NC(=O)C(CC)Oc2ccccc2)CN(C(c2ccsc2)=O)C1.C1(=O)CN1 c1(C(=O)NC2C(C)CN(C(=O)Cn3nccn3)CC2)cc(=O)c2ccncc2o1 N1(C(C=CC)=O)CC2CCC1C1CN(C(C3(OCC=CC=C)CCC3)=O)CC21.C(C)=C C1(NC(C(CCC2CCC2)NC(C2CC(OC)C2)=O)=O)CCC12CCCC2 C1(N(C(C2CCC(F)(F)CC2)=O)CC2(CO)CCC2)CCC12CCNCC2 C1(C(=O)NC(=O)COCC(C)(C)C)CCCCN1C(C1CC1F)=O.C1C(O)CN1C C1(N)CN(C(=O)C=C(CCC)C(=O)NCc2ccnc(C#N)c2)CC1C1CC1.CCC=C c1(C(N(C2CC23CN(CC2CCNCC2)C3)CCC)=O)cc(C(F)F)ccc1C C1(CC=C)(CN2CCCC2c2nc(C)no2)CNCCO1 C1(NC(c2cccc(Cl)n2)=O)CCCC12CN(C(c1cnns1)=O)C2 c1(-c2cn(CCC(C(c3c(O)nnc(C)c3C)=O)=O)nn2)ncn2ccccc12 CCCC(C(=O)NC1CCCC(NC(c2cnccc2N(C)C)=O)C1)C(C)C C1(CNC(C2CCOC2)=O)CCCN1C(c1cc(C2CC2)no1)=O C12(CN(C(C3C(C(C)NC(C4(C=C)CC4)=O)C3)=O)C)CCC(CC1)C2 C(=O)(C(C#N)C(C)(C)C)N1CC(NC(C=Cc2ccc(OC)cn2)=O)C(OC)C1 N1(C(CNC(C)=O)=O)CCC(CNC(=O)Cc2nc(C3CCOC3)n[nH]2)(OC)C1 c1(NCc2ccc(C(N(CCn3cccn3)OC)=O)o2)nccc(Br)c1Cl Cc1nc(C(N2CCC(C)(NC(C3(CC4(O)CCCCC4)CC3)=O)C2)=O)c(C)o1 N1(C(C(c2ccccc2)NC(C)=O)=O)CCN(C(c2nncn2C)=O)CC(C)(F)C1 C1(C(=O)NCC(C2(O)CN(C(C3C(C)(C)C3(F)F)=O)C2)(C)C)CCCC1(F)F n1(C(C)C)ccnc1CNC(C1CCCC1CNC(C1CCCCO1)=O)=O C1(C(=O)NCC(CNC(C(CCC)NC(N)=O)=O)O)CCCC12NC(=O)NC2=O N1(C(CC(=O)NC(CCC(C)C)C)=O)CCC2NCCC2C1 N1(C(C(CO)NC(c2[nH]cc(C(N)=O)c2)=O)=O)CCCC(O)C1 C1(NC(CSCC#C)=O)CC2CCC(C1F)N2C(c1cn(C2CC2)nn1)=O C1(C(=O)NC(C)CNC(=O)Cc2ccc(CC(=O)N(C)C)cc2)CC(S(C)(=O)=O)C1 C1(C(=O)NCCN(C(C(CCC)(C)C)=O)C)CCc2cc(C)ccc2O1 c1(CC(C(=O)NCCC(=C)CNC(=O)CC2(CSC)CC2)O)ccccc1Cl CCCCC(CC)C(=O)NCCCCN(C)C(c1ccnn1C(C)C)=O C(=O)(C(F)C1=CCCCC1)NC1(CC=C)CN(C(=O)CC2(O)CCOC2)C1 CC(CC(=O)N(C)CCNC(=O)CC(c1ccccc1)N(C)C)c1cccs1 c1(C(=O)NC2CC(CNC(c3ccc(OC)nc3C)=O)C2)cc(C)c(C)cc1C N1(C(=O)C=Cc2cnc[nH]2)CCC(O)(CNC(c2cc(F)ccc2C(F)F)=O)CC1 C1(C2CCN(C(=O)C3=C(Cl)CCCC3)C2)(NC(c2cc3c(s2)CCCC3)=O)CC1 c1(C(N(C2CCN(Cc3cnn(C)c3SC)C2)CC)=O)cc(C)nc2ncnn12 C(=O)(C(C)(C)CC(=O)NC(CCC1CC1)C(=O)N1CCC(SC)CC1)OCC c1(C(=O)NCC2CCN(C(c3c(CC)c[nH]c3)=O)CC2C)nn(C)c2c1CCC2 C#CC(C1CC1)NC(C1CC1C(C)NC(C1CCC1)=O)=O c1(C(=O)OC)nc[nH]c(=NCCN(C(=O)Cc2cc(Cl)n(C)n2)C)c1OC C=CC(CCC)CC(=O)N1CC(OCC(N2CCCC(CO)CC2)=O)C1 N1(C(C2CC(C)(CN(C)C)C2)=O)CCC(NC(=O)Cn2cccn2)C(F)C1 c1(CC)cccc(C(N2CC(NC(=O)CC3CCCCCC3)CC2CO)=O)c1F c1(C(C(=O)NC2CC2)N(CCC)Cc2ccc(C(F)F)cn2)sc(CC)cc1Br N1(C(Cc2nc(=N)[nH][nH]2)=O)CCC2CN(C(c3cc4occc4s3)=O)CC2CC1 Cc1nnc(CCNC(=O)CN2CCCC2)n1C.C12(CCC1)CC(=O)N2 c1(OC)ccnc(CNC(C2CN(C(=O)Cc3csc(C)n3)CCO2)=O)n1 c1(C(=O)NC(C)C(=O)NCCC2CCCO2)c[nH]c2ccccc12 c1(-c2nc(C(c3nccs3)=O)[nH]n2)ccccc1NC(C=CC=CC)=O N1(C(c2scc(OC)c2)=O)CCC2(CC1)CC2NC(C12CCCC1C2(F)F)=O C1(C(=O)NC(C(CC)C)c2ccco2)CCCC(NC(C2CCOC2CC)=O)C1 C1(NC(C=C(CCC)C)=O)(CO)CCN(C(c2nn(C)c(Cl)c2Br)=O)CC1 C(=O)(C(C)C(O)C(C)C)NC(CN(C(c1cc(OC)nn1C)=O)C)C C1(CC(N2CC(O)(CN(C)C(c3nnn(C)c3N)=O)C2)=O)CCC2CC2C1 C(=O)(C(=O)N=c1cc(C)o[nH]1)N(C(CNC(C(CC)(C)OC)=O)C)C C12(C(=O)Nc3c(C)csc3)CC(CO1)N(C(N1CCN(c3ccccn3)CC1)=O)C2 C1(CCNC(C23CC(C)(C2)C3)=O)CCC(=O)NC1=O N1(C(C2Cn3c(C)nnc3C2)=O)C2CCC1CN(C(C1(C)C=CCCC1)=O)CC2 N1(C(C(CCSC)O)=O)CCCCC(NC(=O)COC2CCOC2)C1 C=CC1OCCC1C(=O)NCc1ccccc1CN(C(=O)Cc1cc(C)on1)C N1(C(CC(CC=C)NC(c2ccn(C)c2C)=O)=O)CCc2cccc(C)c21 c1(N2C3CN(C(C(CCC)OC)=O)CC2CC3)ncc2c(n1)CCOC2 c1(NCC(N2C(C)CC(NC(=O)CO)CC2)=O)ccc(C(C)(C)C)cc1[N+](=O)[O-] C1(CN(C(c2cc(CC)on2)=O)C)CCCN(C(c2cc(C)sc2N)=O)C1 C(=O)CC(=O)N1CCC(C(=O)NC(C)(C)CCN(C)C)O1.C#CCOCC N1(C(CCC)=O)CCC(O)(C(=O)NCC2COCC2N(C)CC)CC1 N1(C(C(CNC(CC(C)C(C)(C)C)=O)CC2CC2)=O)CCc2cc(F)ccc21 C(=O)(NN1CC2CCCC2C1)N1C(CN2CC(C)(C)C2)Cc2ccccc21 N1(C(C(C)C)=O)CC(NC(C2(N(C)C(C)C)CC2)=O)CCC1C C(C)(C(C)(C)C(=O)NC(c1nc[nH]n1)CO)NC(c1c(C)cccn1)=O C1(CN(C(=O)CN2CCC(C)(NC(c3ccc(F)s3)=O)C2)C)CCCCC1O Cc1cc(=NC2CC3CN(C(=O)CCc4ccc(Cl)s4)CC23)[nH]c(C(C)(C)C)n1 c1(C(=O)N(CC2C(NC(CSc3cn(C)nc3)=O)C2)C2CC2)ncccc1N c1(C(N2CCC(OC)C2)C(=O)N(c2ccccc2)C)cc(F)ccc1Br CC(C)C(O)(C(=O)NC(CNC(=O)CC(C)(C)S(C)(=O)=O)C1CCC1)C(F)(F)F C12(NC(C=C(C)C(C)(C)C)=O)CCCCC1N(C(c1cc(Cl)c(Cl)n1C)=O)CC2 C1(CNC(=O)NCC(CC)NC(C)=O)CC2(CCC2)CN1 Cc1cc(C(=O)N(c2nnc(N)s2)C(c2ccc(C(N)=O)[nH]2)=O)cnc1C Nc1cnc(Br)c(C(=O)NCC2(CO)CCOCC2c2ccccc2)c1 c1(C(N2CC(NC(C3C(C=C)OCC3)=O)C(O)C2)=O)ncnc(O)c1F C1(C(N(C)CC2CCN(C(=O)Cc3ccoc3)C2)=O)CCCN1S(=N)(=O)N(C)C C(=O)(C(CC(C)C)n1ccnc1-c1cccc(C(=O)OC)c1)N1C2(CC)CC(C1)C2 c1(NC(C(C2(O)CCCCC2)CC)=O)ccc(NCC(F)(F)C(F)F)cc1F CC(C)CC(=O)NCCC(=O)NCC1CCC1NC(=O)Cc1nnc(O)s1 c1(C(C)C)cc(C(=O)O)c(N(C(C)CNC(c2cccs2)=O)C)s1 C(CC(O)CC(=O)N1CCC(NC(C2CCN2C(=O)OC(C)(C)C)=O)C1)SCC C(=O)(C(CNC(c1ncc(F)cc1C)=O)C(C)(C)C)Nc1cccc(OCC)c1 C1(CC(=O)NCC2CCCC2)CCCC(NC(=O)CC2(c3cc[nH]n3)CC2)C1 C1(C(=O)NCCCC2(CNC(CCC(C)C)=O)CCCC2)CCc2c[nH]nc2C1 C(C1CCN(C(=O)C2=CCCOC2)CC1)=CC(=O)NCC1CCCCC1 N1(C(C(C)Oc2ccccc2)=O)CC(F)(F)CC1C(=O)NC(=O)C1CC1.C12CC(C1)O2 C12(CNC(CSC)=O)CCCC1CN(C(=O)C(C)(O)C=Cc1ccccc1)C2 N(C1C(=O)Nc2ccc(Br)cc21)C(C1CC2C=CC1C2)=O c1(N2CCC(CCOC)(NC(=O)C(F)(F)C3(O)CCC3)C2)ncnc2sccc12 N=c1[nH]cc(C(N2CC(N)(c3nn[nH]n3)C2)=O)c2cc[nH]c12 C(CCCCCNC(=O)Cn1cc(C2CCOC2)nn1)NC(C1(CC)COC1)=O CC(F)(CNC(=O)C(C1(O)CCCC1)F)CNC(C1CC(C)(F)C1)=O C1(CCC)CN(C(c2cc(Br)n(C)n2)=O)CC1NC(=O)CN(C)C(C)=O Cc1nccc(N2CCN(C3CCN(C(=O)Cc4cc(C)nn4C)CC3)CC2)n1 CC1(C)CCc2[nH]nc(C(N3CC(CNC(=O)C(C)(C)C(N)=O)C3)=O)c2C1 C1(CC)CCCCC1OCC(=O)NCc1ocnc1NC(C1CC2CCC1O2)=O c1(CN2CCC(CC(=O)NCC3CCC(F)C3)C2)c[nH]c2ccc([N+](=O)[O-])cc12 CC1COCC(CNC(=O)CC2CC(NC(c3sccc3F)=O)C2)O1 c1(C(=O)NCC(O)CC(=O)NC2CC(C3CC3)C2)ccc(O)c(F)c1 C(=O)(CCC(C)NC(c1cnn(C(F)F)c1)=O)NCC(CCOC)O C1(NC(CC(CC)C(F)F)=O)CCc2ncc(C)n2C1 c1(C(N2CC(CC)C(NC(=O)C3=CCCC3)CC2)=O)c(C)cc(Cl)cc1N N1(C(c2ccc(C)s2)=O)C2CCCC1CN(C(c1n[nH]c(C)c1F)=O)CC2 c1(C(=O)NCC(CCCC)NC(=O)Cc2coc(C)n2)cncc(F)c1C C(=O)(C(C)(C)C(F)(F)F)N1CCC(C(C)NC(c2[nH]c(C)c(C(C)=O)c2C)=O)C1 c1(C(=O)NC(CNC(C(CC(C)C)O)=O)(C)C2CCC2)ccc2occc2c1 CC1CCN(C(c2cccs2)=O)CCC1N1CCC(O)C(C)(C)C1 c1(C(=O)NC(C)C=CC(=O)N2CCC2c2cc(O)no2)ccc(O)cn1 c1(C(=O)NCC(CNC(c2cc(C)c(N)cc2)=O)(C)C)n[nH]c2ccc(Cl)cc12 CCC(C)C(C)C(=O)NCC1CCCN1C(c1sc(-c2cnn(C)c2)nc1C)=O CC(C)(CCl)C(=O)N1CCC(O)(CNC(C2(F)CCOCC2)=O)C1 c1(CNC(c2nn(C)c(O)c2)=O)nc(CC2CCCC2(F)F)cc(O)n1.C1C(=O)N1 Cc1nc2ccc(C(N3CCN(C(=O)CNc4ccccc4)C4CC34)=O)cc2o1 CC(CC(=O)N1CCN(CCCNC(C2COCC2(C)C)=O)CC1)C(C)(C)C N1(Cc2ccc(Cl)cn2)CC(=O)N(Cc2ccc(C#N)cn2)C1=O c1(NC(C(N(C(C2C(=C)C2)=O)C)C2CC2)=O)cc(C)c(F)c(C)c1 Cc1ccc(O)c(CC(=O)NCSCC(C)(O)CNC(=O)CC2(C(F)(F)F)CC2)c1 CC1CCCN1CC(=O)NC1C(C(=O)N(C)Cc2cocn2)C1(C)C C1(C(N2C(C)CC2)=O)CC2C=CC1N(C(C1(C#N)CC=CC1)=O)C2 N(C(=NCCCOc1ccc(Cl)cc1)NCc1cnco1)C(C=C)C CCS(=O)(=O)CC(=O)N1CC2(CC(NC(=O)CCC(F)(F)F)C2)C1 c1(CNC2C(C(C)NC(N3CC4CCCCC4C3)=O)C2)cnn(C)c1S(C)(=O)=O Cc1ccc(C(N2CC(NC(c3cnc(C4CC4)s3)=O)C3CC23)=O)nn1 n1(CCNC(C2(CCNC(=O)Cc3nc(=N)[nH][nH]3)CCC2)=O)c(C(F)F)nnc1S Cc1cccc(CC(=O)NCCC2CCC(NC(c3cc[nH]n3)=O)C2)c1C c1(C(N(CC(C)CNC(=O)C(O)C2CCC2)C)=O)cc(O)cc(Cl)c1 c1(OC)cnccc1C(=O)NC1(C(=O)NCC2(OC)CC2)CCSC1 n1(CC)nc(C(=O)N(C)CC=CC(=O)NC2CCOC2)cc1O N1(C(c2ccc(COC)o2)=O)CCC2(C(=O)NCCc3cnnn3C)CCCC12 c1(C(=O)NCCN(C(=O)Cc2ccn(C)n2)C)ccc(Br)cc1OCF CCC1=C(C(=O)Nc2ccccc2)C(c2n[nH]cc2Br)NC(=O)N1CC=O c1(OC)ccnc(NC(C2CC2OCc2ccccc2)=O)c1I c1(C(=O)NC2C(CNC(c3scc(C(C)=O)c3)=O)CCC2)nccc2ccncc12 C1(CNC(c2cc(C(C)C)on2)=O)CC(C(=O)NCCn2cc(CO)nn2)=NO1 c1(C(N(C2CN(C(=O)C(F)(F)CC3CC3)CC2F)C)=O)ccc2nc(S)oc2c1 c1(C(N2CC(NC(CC3C(OC)CCC3)=O)C2)=O)cnccc1S(C)(=O)=O [N-]=[N+]=NC1CCC(C(N2CCCC(CN3CCOCC3)C2)=O)CC1 N1(C(CC(C(C)OC)NC(C2(C)CNC(=O)C2)=O)=O)CC2CCC(C1)N2C Cc1cncc(C(=O)NC(C(=O)NCC2COCCO2)c2cccs2)n1 C12(NC(c3cnn(CC)c3Cl)=O)COC(C1)C(NC(=O)CCCCSC)C2 N1(C(C(CC)C(C)C)=O)CC2(CCC2)CC1C(=O)N1CC(O)CCO1 c1(OC)ccccc1NC(=O)C(c1ncccc1C)N(C)CC1(C(N)=O)CC1 c1(C(=O)NC2C(CNC(c3ncn(C)n3)=O)C2)cc2ccccc2oc1=O CCCCCC(C)(C)NC(c1cc(N(C)C)ccc1F)c1nnnn1CCC1CC1 N1(C(C=NOC)=O)CC2CCC2(CNC(=O)C(C(C)C)NC(=O)OC(C)(C)C)C1 C(=O)(C(CC(=C)C)NC(=O)CCn1cnnn1)NCCC#C N1(C(c2ccc(CSC)o2)=O)CCC(C2CC2)C1CNC(=O)CCC=C(C)C Cc1ccnc(C(N2CC(C)(C(=O)NCc3cccc(C4CC4)c3)C2)=O)c1.OC C(=O)(C1=NN2CCCN=C2N1)N1CC(C2(NC(C3C4CCCCCC34)=O)CC2)C1 C1(CC)C(NC(C2CCC(O)CC2)=O)CCN1C(C1COCCO1)=O Cc1cc(C(=O)NC(CCO)c2cncs2)c2nccn2c1 c1(CC(=O)NCC(C(C)C)NC(C23OCC(CC)(C2)C3)=O)ccc(OC)c(F)c1 c1(C(c2ccc(-c3ccoc3)s2)NC)ccccc1Br CC(CC(C)(C)C)C(=O)NCC1CC(O)(CNC(c2cccn3nccc23)=O)C1 C(=O)(C(C(C)C)N(C(c1ccccc1C(C)C)C(=O)NC1CCC1)C)OC C#CC(CC(C)C)NC(=O)CC(O)CNC(=O)C(C)(Cl)Cl N1(CC=O)CCCCCC1.C1(CCC)CCCC1C(=O)NOCCCOCCO C=CCC(C)(C)C(=O)N1CCC(OCC(N2CCC(C(C)(C)O)C2)=O)C1 c1(N(C(=O)CS(=O)(=O)Cc2cccs2)CC2N(C(C)=O)CC2)cc2n(n1)CC(F)C2 C1(NC(CC(C)OC)=O)CCN(C(c2c(Cl)c(C)nn2C)=O)CC12CCC2 c1(C(=O)NCC2CC(CNC(=O)CCc3ccncc3)OC2)cnn2c1NCCC2 C1(CN(C)C(c2cc(-c3ccncc3)[nH]n2)=O)CCCN(C(=O)CC#N)C1 N1(C(C2CCN(CC)C2)=O)CCCCC1C(N1CCC(C(N)=O)C1)=O C1(C(C)C)CCC(C(=O)N(C)CCc2ncccn2)N1C(=O)C(C)C1CCCC1 c1(C(N2CC(N(C(c3nc(C)n(C)c3)=O)C)C(O)C2)=O)nnc(O)nc1O N1(C(CSCC)=O)CCN(C(=O)Cc2nccn2C)C(C)C1 C=CCC(C)C(=O)N1CCC1CNC(c1nnc(C)s1)=O CC(N=c1[nH]c(N2CCC(C)C(F)(F)C2)nc2cccnc12)c1ccc(C#N)cc1 N1(C(C(CC)(F)C(=O)OC)=O)CCCC2(CCN(C(=O)CNS(=O)(=O)CC)C2)C1 N1(C(C2C(C#N)C2)=O)CCN(C(c2ccnc(CO)c2)=O)C(CCCCC2CC2)C1 C1(C(N2CCCC(NC(C3CCC(SCC)CC3)=O)C2)=O)CCCC(=O)N1C c1(N2CC3C(C)C3C2)nc2ccc(Cl)cc2c(=NC2CCCCC2N(C)C)[nH]1 c12cccc(c1F)N(S(C)(=O)=O)C2=O.c1(C(C)(C)C)ncccc1OC(F)F CCCC(CC)C(=O)NCC1CCN(C(C2CCC(N(C)C)CC2)=O)C1 c1(C(N2CCC(CCOC)(NC(c3oc(C)nc3C)=O)C2)=O)ccc(O)cc1F C1(NC(c2c(CC)[nH]cc2)=O)CC=C(C(=O)NCC(O)COC(C)C)C1 C1(CNC(c2ccc(CC)s2)=O)CCCC2(CN(C(=O)CC3CC4(CC4)C3)C2)O1 c1(C(N2CCN(C(C=CCCC)=O)C3C2C3)=O)ccc2c(c1)CCC2 c1(C(N2CC(CC(C)NC(C=C(C)C(C)(C)C)=O)C2)=O)cc2n(c1)CCSC2 Cn1nc(CC(=O)NCCNC(c2coc(Cc3ccccc3)n2)=O)cc1Cl.C C(=O)(C(C)C(O)C(C)CC)N.C(=O)(CCCCCn1cc(C)nn1)OCC C(CC(C)C)(C(=O)NCC1CC1)ONC(COCCOC)=O N1(C(c2ccc(CN(CC=C)C)cc2)=O)CCC(F)C(NC(=O)C2=NOCC2)C1 C(=O)(CC(C)(C)CC(F)F)N(C(C)C)CCN(C)C(C1CCN2CCOCC12)=O S(=O)(=O)(C1(C)CC1C)N(CC)Cc1ccccc1.C12(CCC(=O)N1)CNC2 CCCC(C(=O)N(CC(C)NC(=O)OC(C)(C)C)C)NC(=O)Cc1conc1C c1(C(N2C(CC)CN(C(c3oncc3C)=O)CC2)=O)n[nH]c2ccccc12 c1(C(=O)NCC2CN(C(c3ccc(C)n3C)=O)C(C)(C)C2)ncnc2sccc12 Cc1cc(C(=O)NCc2ccc(C(C)NC(C3(O)CCC3)=O)cc2)nc(O)c1 CC1(C)CC(NC(=O)C2=CCCC2)CN(C(c2ccc(OCCO)cc2)=O)C1 c1(C(N2C(C)CC(CNCC(=O)OC(C)(C)C)C2)=O)[nH]nc2c1CCC2(C)C N1(C(C(C2(O)CCC2)NC(CN(CCC)C)=O)=O)CCCN(C=O)CC1 c1(CC)ccc(C(=O)N(CC(C)NC(=O)C(C#N)C2CC2)C)s1 c1(NC(CC(C)OC)=O)ccc(NC(c2cnn(C)c2C(C)(F)F)=O)c(C)c1 CC1CN(C(C2(C(=O)NC3CC3)CC2)=O)CC(C)C1CNC(C1CC(O)C1)=O CCC(O)C(C)(C)C(=O)N1CCC2(C1)CN(C(c1nccc(Cl)c1F)=O)C2 c1(CC(=O)N(CC(CNC(c2ccc(C)o2)=O)C)C)c(C)noc1C C=CCC(CC)C(=O)N1CCOCC(CNC(=O)CCSc2cccc(C)c2)C1 C=CCCCCN(C)CCOCCNC(C1CC1c1cncs1)=O C1(C(C)NC(CN(CCCCCC)C)=O)CCCN(C(=O)CC2(O)CCC2)C1 c1(NC(C2N(C(C(C(C)C)O)=O)CCCC2)=O)cc(Br)ccc1C#N C1(C(N(CC(=O)NCC)CC2CC2)=O)CCC(COC(C)(C)C)C1 c1(C(=O)NCC(C)N(C)C(C2CCOC3(CCC3)C2)=O)cccn2c(O)nnc12 Cc1cc(C(=O)NCC23CCC2CCN3C(c2nnc(S)n2C)=O)c(C)n1C c1(C(=O)NC2CC(N(C(C(c3ccccc3)SC)=O)C)C2)cc(F)c(F)c(F)c1 C1(C(N2C(C(=O)NC(CC(C)C)(C)C)CC2)=O)CC2CC(=O)C1O2 C12(C(N3CCC(CC=C)(NC(=O)Cc4cscn4)C3)=O)CCCC1OCC2 C1(NC(COc2ccc(C)cc2C)=O)COC2(CCCN(C(=O)OC(C)(C)C)C2)C1 c1(NCC2N(C)CCN(C(C3CCCO3)=O)C2)ncnc2c1CCCC2 C1(NC(CCOC(C)C)=O)CCN(C(C2CC3CCC2C3)=O)C(C)C1 C(C(C)(C)CNC(=O)C(C)Cn1ccc(C)n1)N(C(C1C(C(=O)OC)CC1)=O)C C(=O)(CCCc1nc(C2CC2)no1)NC1C(CNC(CNS(N)(=O)=O)=O)CC1 c1(C(N2C3C(NC(C(c4cnn(C)c4)C)=O)C(C3)C2)=O)ccc2c(c1)CC(=O)N2 N1(C(CS(=O)(=O)NCC)=O)CCCC2(CNC(c3ccc(C#N)s3)=O)CC12 Cn1ncc2cc(C(=O)NC3CCC(CNC(C4CC(Cl)(Cl)C4)=O)C3)sc12 C1(C(CNC(S(c2ccn(C)n2)(=O)=O)=O)(C)O)CC2(CCCCC2)S1(=O)=O C12(NC(c3cc4ccccn4n3)=O)CCCCCC1N(C(=O)Cn1ccnn1)CC2 C1(CCC)(NC(c2nn(C)c(Cl)c2Cl)=O)CCN(C(c2sccc2F)=O)CC1 C=CCC(C(=O)NC1(C(=O)NC(c2cccc(O)c2)C)CCN(C)C1)C(C)C C(CC(C)C(=O)N(CC)CC1CCCN1C(=O)CCn1cnnn1)=CCC C1(CN(C)C(c2cc(-c3ccccc3)c[nH]2)=O)CCCN1C(=O)CC1C=CCC1 c1(NC(=O)NC2C(c3onc(COC)n3)OCC2)cccc2cc(Br)cnc12 c1(OC)cccc2[nH]cc(COCC(=O)NCCC(O)CNC(=O)C(C)=CC)c12 C(=O)(CN=S(C)(C)=O)N1CC(N(C(CN(CCC)C)=O)C)C(F)C1 C(=O)(CC(C)CC(C)C)NCC(C(C)(C)C)NC(c1c(C)nco1)=O C1(NC(CC(CC)C2CC2)=O)CN(C(=O)C(F)C2CCCC2)CC12CCCC2 c1(CN2C(NC(=O)OC(C)(C)C)CCCC2)cccc(OC(F)F)c1C Cc1cn(C)cc1C(=O)NCC(C1CCOC1)NC(c1c(C)coc1C(C)C)=O C1(CNC(C2C(COCCOC)C2)=O)CCN(C(=O)Cc2scnc2C)C1 S(=O)(=O)(c1ccc(C(C)NC(c2cccc(N(C)C)n2)=O)cc1)NC(C)C C1(C#N)(CC(=O)NCC(CC)NC(=O)CCc2ccc(C)nc2)CCOCC1 C(=O)(C(O)CC(C)(C)C)NC1CCC(NC(c2cccc(C)c2)=O)CC1 N1C(=NCC2CCC2)N2CCC(C2)OCC1.OCC(C(F)(F)F)c1ccccc1 c1(C2(O)CN(C(=O)NC(c3ccc(Cl)cn3)C)C2)ccccc1Br C=CCC(C(=O)NCCNC(=O)Cc1ccc(C(N)=O)cc1)c1ccccc1 CCCCCCCN(C(=O)C(N)C(C)C)C(C)CC C1(NC(CCOCC)=O)CN(C(c2cnc(C)nc2C)=O)CCC1c1ccccc1 Cc1nc(C(=O)NCC(CNC(=O)C(C)(C)Nc2ccccc2)CO)n[nH]1 N1(CC)CCC(NC(c2cnn(CCNC(=O)CN3CCC(O)CC3)c2)=O)CC1 N1(C(C(=CC2CCCC2)C)=O)CCC2CN(C(c3n[nH]cc3Cl)=O)CCC2C1 N1(C(CCOCCC)=O)CCN(C(=O)CN(S(=O)(=O)CC)C)C(C(C)(C)C)C1 c1(NC)ncccc1C(=O)NC(C1CCN(C(=O)CC(F)(F)Cl)C1)C N1(C(C(C)CC2CC2)=O)CC2(C=C(C(=O)N(CCC(N)=O)C)CO2)C1 c1(C(=O)NCC2CC(C)(C)CN2C(C2CCC2F)=O)ccnc2cc(Cl)ccc12 CCC(C#N)C(=O)N1CC(CO)(NC(C2CCCCC2c2nc[nH]n2)=O)C1 N1(C(c2ccc(SC)cc2)=O)CCC2(CCN(C(C3CCOC3(C)C)=O)C2)C1 C(C(C)(C)CC(=O)N1CCC(NC(=O)C(O)Cc2cccc(Cl)c2)CC1)N(C)C C1(=O)C(C(C)C)OC(=O)C2CC(C)(C2)N1.C(C(=O)N(C)C)N(CC)CC c1(C(=O)OC)ccc(NC(C2(CNC(c3nccn3C)=O)CC2)=O)c(C)c1F C1(C(=O)NCC2CCN(CC)C2)CN(C(=O)CC2CCSCC2)CC1(F)F C=CC(C)(C)C(=O)N1CC(NC(=O)CC2C(=O)NN=C2C)C(O)C1 C1(C(=O)OC)C(NCc2n[nH]c(CO)n2)C2CCCC12 CCC1=C(C(=O)NC2(CF)CCN(C(c3csc(C)c3)=O)C2)CCCO1 c1(N2CCC(N(C(=O)NC3C(CC)CCCC3)C)CC2)nc(C)cc(=N)[nH]1 N1(C(c2cc(C)c(C)nc2)=O)CC2CCC(N(C)C(c3ncc[nH]c3=O)=O)C2C1 C(=O)(CC(C)(C)C(F)F)C(C1N(C(N(CCOCCNC(=O)NC)C)=O)CSC1)=O CON(CCC(=O)NC1CC(SC)C1)C(=O)CCC(CC)OC C1(F)(CNC(c2nc(OCC)sn2)=O)CCN(C(=O)Cc2[nH]cnc2C)CC1 c1(C(C(=O)NCC(C)(C)NC(c2cnsc2)=O)OC)ccccc1Br n1(CC(N2CC(COC)(NC(=O)CC3CC(C)=NO3)C2)=O)nnc2ccccc12 N12CC(CC13CCC3)CC(=O)Nc1c(csc1C)C2=O.CCCSC1CC1 N1(C(C(C)O)=O)CCC(N(C(=O)C(O)c2ccco2)Cc2ccccn2)CC1 N1(C(C2(SC)CCC2)=O)CC2CCC2(CCNC(c2c(O)cccc2F)=O)C1 C=CCC(CC)C(=O)N1C(CC(=O)NCCC2CCSC2)C2CCCC12 CC(C)CC(CNC(c1cc(C(C)C)[nH]n1)=O)NC(C1CN(C(N)=O)C1)=O c1(OC)ccsc1C(N1CCC(N(C)C(c2csc(CN(C)C)n2)=O)C1)=O C12(CNC(COCC#C)=O)CN(C(=O)Cn3cc(C)cn3)CC1CCO2 c1(C(N(C(C)C(=O)NC(c2ccncc2F)C)CC)=O)c[nH]c2nccc-2c1 CC1(C)CN(C(=O)CC2CCCCCO2)CCC1NC(=O)CNS(=O)(=O)C1CC1 N1(C(c2cc(OCCO)cnc2F)CC)CCS(=O)(=O)CC1C N1(CC(N2CC(OC)C(NC(c3ccc(Cl)cc3C)=O)C2)=O)Cc2ccccc2C1 C(C(O)CC(=O)NOCC(F)(F)F)NC(c1cc(C)c(C)nn1)=O C1(NC(C2(CCCC)CC2)=O)C=CCN(C(c2cc(C)nn2C(C)(C)C)=O)C1 c1(CCC(N2CCC(CNC(c3ccc(=O)oc3)=O)C2)=O)ccccc1[N+](=O)[O-] N1(C(C2CC(C)=C(C)CC2)=O)CCC(CCNC(=O)C2=CCCC2)C(F)(F)C1 N1(CCC(=O)Nc2ccc(C(=O)NCC(CC=C)NC(C)=O)s2)CCC(O)CC1 c1(C(=O)NCC2CCN(C(c3cc(C)nn3C)=O)CC2C)cc(S(N)(=O)=O)cs1 c1(CCCSC)cnn(C(=O)NCCCC2(NC(CSCCCC)=O)CC2)c1 N1(C(C=COCC)=O)CC=CC(C(N2CC(CC(F)(F)F)C2)=O)C1 C(N=c1nc(C(C)C)cc(C)[nH]1)C1(C)CCCN(C(C2CC3(CC(=C)C3)C2)=O)C1 C1(NC(C=C(CC)C)=O)CC(CNC(=O)CNc2ccccc2C(C)C)C1(C)C C1(CN(C(=O)Cc2cnc(O)[nH]2)CC)CCCN1C(=O)CC1COCC1O C1(NC(C(C=CC)O)=O)CCN(C(C2CCCCN2S(=O)(=O)C(C)C)=O)CC1 C=CCC(CNC(C1C(CNC(=O)C(C)C2CC2)C1(C)C)=O)CC(C)C c1(NC2(C)CCCC2)ncccc1S(=O)(=O)Cc1ccc(F)c(F)c1.C1(CN)CC1 N1(C(c2cc(C)ncc2)=O)CCCC(NC(=O)CCC2CCC(=O)N2)C1C N1(C(C2C(C(=O)OC)C2)=O)CCC2(CC1)CCN(C(=O)CCNCCC(C)(C)C)C2 N1(C(C2C(C(C)=O)C2(C)C)=O)CCC2(CCN(C(C3CC4CCC3O4)=O)CC2)C1 CC1CN(C(=O)C(F)(F)C(C)O)CCC1CNC(C1CCC2(CC2)C1)=O C1(CC(=O)N(CCCCCNC(=O)C(CO)NC(=O)C(F)(F)F)C)SC(=N)NC1=O Cc1cc(C(=O)NC(C)CCNC(=O)CSCc2ccncc2)c2nccn2c1 C1(NC(c2cccc(-c3ccc[nH]3)c2)=O)CN(C(C2(CCF)CCC2)=O)CC1F O=C1CC(=O)CC(C(N2CCOCC2Cc2cn(-c3ccccc3)nn2)=O)C1 CS(=O)C=CC(=O)NCCOCCNC(c1nc(-c2ccccc2)sc1N)=O N1(C(CCCOC(C)=O)=O)CCCOC(CNC(c2cc(C(N)=O)cn2C)=O)C1 C1(NC(CC(CC)C)=O)CC2CCC(C1)N2Cc1cc2ccccc2s1 C1(NC(c2ccc(OC)s2)=O)CC(CC(=O)NC2(C)CCSCC2)C1(C)C c1(OC)ncc(F)c(=NC(=O)c2ccn3ncc(Br)c3n2)[nH]1 Cc1cc(C#N)cnc1C(N1CCCCC1CCNC(C1(NC(C)C)CC1)=O)=O Cc1sc(Br)nc1C(=O)NC1(CCNC(C2C=CCC2)=O)CCCC1 c1(CNCCc2ncc(C(C)(C)C)s2)cccc2cccc(Br)c12 c1(NCC23CC(NC(c4c(C)nn(C)c4Cl)=O)(C2)C3)ncnc2c1cnn2C(C)C c1(N2CC(F)C(F)C2)nc(=NCc2cocn2)[nH]c2c1CSC2 C(CC)(C(=O)NCCC1CCN(C(c2csc(C(F)(F)F)n2)=O)C1)OCC N1(c2onc(C)c2C)CCN(C(=O)C2CC2)CC1C c1(C(N2CC3CN(Cc4cncs4)C3C2)=O)cc2ncccn2n1 c1(C(=O)NC(C2(O)CN(C(=O)C(O)CN3CCOCC3)C2)C)ccc(C(F)F)o1 N1(C(CCCC)=O)C(CNC(=O)C(c2ccc(F)c(F)c2)=O)CC2CCCC12 CCC(C(=O)NCc1ncoc1C1CC1)N(C(=O)CC(C)n1ccnc1)C C1(C(=O)NCCc2c(C)ncs2)CCC(O)CN1C(=O)CCCOC(C)C CC1(C)CCC(C(N2CC(CNC(C3CC4(CCCC4)C3)=O)C(F)(F)C2)=O)CC1 c1(CSCC)ccc(C(=O)NC2CCC2NC(=O)C(=O)Nc2ncc[nH]2)cc1 C1(F)(CNC(c2cccc(F)c2O)=O)CCN(C(=O)C(F)(F)c2cscn2)CC1 N1(C(C23CC(C)C2C3)=O)CCC(c2n[nH]c(CNC(=O)CSC(C)C)n2)CC1 N1(C(CCc2c[nH]c(=N)[nH]2)=O)CC2ON=C(CNC(=O)CN3CCCC3)C2C1 C1(CC(N2CC(C)(NC(C(c3c(C)cccn3)(F)F)=O)C2)=O)CCC(C)(C)CC1 c1(CC)cc(CCNC(N2CCC(c3cc(CC)on3)C2)=O)n(C)n1 C(CC(=O)N(C(C)CNC(C1CN2CCN1C(C)C2)=O)C)(C(F)(F)F)OC Cc1nc2ccccc2n1CC(=O)NCCC(C)CCNC(c1n[nH]cc1Cl)=O C(=O)(C1=NN(C)C(=O)CC1)NC1CCCCN(C(C(C(C)C)F)=O)C1 N12CC3CC(C3)(C1)C(=O)N(CC=C)CCC2=O.C1(C)C(=O)N1.C(=O)(CO)NC c1(C(N(CCC(=O)NCC(c2cnn(C)c2)O)CC#C)=O)c(CO)n[nH]c1C C(=O)(C(C)(C)C(=O)OC)N(CCN1CCN(C(c2cc(CCC)on2)=O)CC1)C C1(C)(CNCCCS(=O)(=O)N(C)C)CCCNS1(=O)=O Cc1sc(-n2cnnn2)c(C(=O)NC(CNC(C2CC2F)=O)C2CC2)c1C C(=O)(C1=NOC(C)C1)NC1CCCN(C(CCSC(c2ccc(C)cc2)=O)=O)C1 N1(C(C=CC)=O)CCCC2C(NC(=O)CC3=NNC(=O)C3)C(C)(C)C12 N1(C(c2cccc(C)c2Cl)=O)CCC2C(CCN2C(c2ccc(O)cc2Br)=O)C1 N1(C(C(F)=CCC)=O)CCCC2(CNC(=O)C(c3ccccc3)=O)CCCC12 CC1=C(C(=O)N2CC(NC(=O)CCc3ccn(C)c3)CC2(C)C)CCC(C)(C)C1 C1(C(N(CCCCCNC(COCc2cc(C)no2)=O)C)=O)CCCCC1F Nc1c(F)ccc(F)c1C(=O)NC1CC2(C1)CC(NC(C1CCCN1C(N)=O)=O)C2 N1(C(c2nccc(CC)c2)=O)CC(C(=O)NCC(C)(C)C(C)(C)C)OC(C)C1 Cc1c(C(=O)NC(CNC(=O)C(C)C2CCCC2)C(C)C)noc1C1CC1 CCS(=O)(=O)CC(C)(C)CNC(=O)Nc1cc(N(C)C)cc(C)c1 N1(C(c2nc[nH]n2)C2CC2)CC(O)(C2CCC2)C1.CC1=CC(=O)NC1 c1(OC)cc(OC(C2(Nc3ccc(F)cc3)CCNCC2)=O)ccc1C(F)(F)F Cn1cc(C(=O)NCCCCNC(C2(CCF)CCC2)=O)c(Br)n1 C=C(C)C(O)CC(=O)N1CCCC(N(C(=O)CCSCC(C)C)C)C1 C1(NC(CN(CCC)C)=O)CN(C(c2cccc3nccn23)=O)C2CCCC12 CC1(C)C(C(=O)NCCCC2CCN(C(C3CC(n4cnnc4)C3)=O)CC2)C1C#N N1(C(C(CC)C)=O)C2CCC1C(F)C(NC(c1cc(N3CCCC3)ncn1)=O)C2 C1(CC(=O)NCCCC(=O)N(CC(CC)O)C)CC(=O)NC1=O c1(C2C(Cn3cc(CC4N(C(CC5(C)CC5)=O)CCC4)nn3)C2)cnccc1Cl C(=O)(CCS(C)(=O)=O)NC(C(C)NC(c1cnn(C(C)C)c1Cl)=O)(C)C c1(C(=O)NC2CC3CN(C(CS(CC)=O)=O)C2C3)ccc([N+](=O)[O-])n1C c1(C(N2C(C(C(NOCc3cccc(C)n3)=O)C)CCC2)=O)ncc(F)cc1N c1(N2CCC(CC=C)C2)[nH]c(=NC(C)c2ccc(Cl)cc2)nc2sccc12 c1(C(=O)NC(CN(C(C2CCCC(OC)C2)=O)C)C)n[nH]c2ccccc12 C1(CC(=O)NC(c2ccc[nH]2)C)C=CC(NC(=O)Cc2ccccc2)C1 c1(OCC(C)C)ccc(C(N2CC(CNC(=O)C(c3ccccc3)C)C2)=O)cc1 N1(C(C(CC2CN(C(=O)CC(C(O)CO)C3CC3)C2)F)=O)CCOCC1 C(CC(C)(C)C(=O)NC(CCC(C)CCO)(C)C)NC(=O)OC n1(CC(=O)NCC(C)(C2CCC2)NC(C(COC)C)=O)ccc2cc(F)ccc12 C1(CC(=O)NC(CC#C)C(N)=O)CN(C(c2cccc(CC)c2)=O)C(C)(C)C1 C1(C2CC2)(CNC(C2CC(OCC)C2)=O)CCN(C(C2(OC)CCCOC2)=O)C1 C(N(C1CC1)N(C)C1CCn2ccnc21)c1ccc2ccc(C)cc2c1 N1(Cc2c(C)noc2C)CCOCC(NCc2cc(N3CCCC3)nc(Cl)c2)C1 CCCC(CNC(c1ccnn1CC)=O)NC(=O)CCCc1ccsc1 c1(NC(N2CC(c3ccccc3)CN(C)C2)=O)cn2c(Br)cnc2s1 c1(C(N2CC(C)C(C(N3CCc4nn[nH]c4C3)=O)CC2)=O)cccn2nccc12 N1(C(C=CC)=O)C(C(=O)Nc2ccnc(Br)c2)CC2CC12 c1(N2CCC(N(C(C(CCC)C(C)C)=O)C)C2)ncc([N+](=O)[O-])cc1Br Cc1ccc(C2CCC(c3nnc(C4CCC4)n3C3CC(OC(F)F)C3)C2)n1C CC(CC1CCC1)C(=O)NCCCCNC(C1CS(=O)C1)=O c1(C(N2CCC(OC)(CNC(C3CC(O)CN3C)=O)C2)=O)cnc2[nH]cnc2c1 c1(NC(C(C2CN(C(C3CC4(CCO3)CC4)=O)C2)OC)=O)ccc2c(c1)COC2 c1(C(N2CCN(C(CN(CC(C)(C)C)C)=O)CC2CO)=O)ccc(C#N)cc1O c1(NC(CNC(C2C(C(=O)OC)CCCC2)=O)(C)C)cc(=O)n2ccccc2n1 C#CCCCC(C)C(=O)NCC1CCN(C(c2ncc(C(F)F)s2)=O)C1 C(=O)(C(C)CCCOC)NC(CNC(c1c(CC)n(CC)nn1)=O)(C)CC CC(C)(C)C(CNC(=O)Cc1ccco1)NC(c1ncccc1C(F)(F)F)=O c1(C(=O)NCCCNC(C2C(C)OCCC2)=O)cnn2c(Br)cccc12 c1(CCC(=O)N(C2CCN(C(C(F)OC)=O)CC2)CC2CC2)cccc(F)c1F n1(CC(=O)NC2CCCC2CNC(C2(CF)CC2)=O)ccc([N+](=O)[O-])n1 N1(C(c2c(CC)ccs2)=O)CC(CNC(C2(C)CCC23CCC3)=O)CC(C)(C)C1 N1(C(c2nc(C)n(C)c2C)=O)CCCC2CN(C(c3cnnn3C3CC3)=O)CC12 c1(C(N(CC(CC)NC(C2CC3CCC(C2)S3)=O)C)=O)ncncc1C#N N1(C(C(C2CCN(C(CN(CC(C)(C)C)C)=O)C2)(C)C)=O)CC2C(CO)C2C1 Cc1ccc2cc(COC(C34OCCCC3C4(F)F)=O)oc2c1 N1(C(c2scc(C)c2)=O)CC=CC(NC(=O)CCc2ccc(CO)cc2)C1 CCCC(C)(O)CC(=O)NC(C)(CNC(=O)Cc1ccc(C)cc1F)CC1CC1 N1(C(c2c(C)nc(C(F)F)o2)=O)CCC2C(CCC(=O)N2C2CC2)C1 N1(C(Cc2ccn(CC)n2)=O)CC(NC(=O)C(O)CN2CCCC2)C(C(F)F)C1 C1(CCC(=O)N(CCCN(C(C(F)=C(C)C)=O)C)C)CCCCN1C N1(C(C(C2CCC2)OC)=O)CC(NC(=O)CCNC(C)=O)CC(C)(C)C1 N1(C(C2(CC#C)CCCCO2)=O)CC2CCC1CC2NC(=O)C(F)OC(F)(F)F N1(C(C(C)C(F)F)=O)CC(C(=O)N(CC(C)(F)F)C)CC(C)(C)C1 c1(C(N2CCN(C(C(C)n3cccc3)=O)CC2C)=O)ccc2nn(C)cc2c1 CCCCCCCCC(=O)NC1CC(CNC(=O)CC2OCCOC2(C)C)C1 c1(NC(C(c2ccoc2)NC(C(CC)CCOC)=O)=O)cccc(N=[N+]=[N-])c1 N1(C(c2ccc(C(C)C)s2)=O)CCCCC1CNC(=O)CSc1nncs1 CCC(C(=O)NCC(C1CCCCC1)O)N(C(=O)Cc1cnn(C)c1)CC.C(N)=O C1(CNC(c2cc(OC)ns2)=O)CC(NC(c2cnc(O)s2)=O)C1(C)C C(=O)(C(O)CC(C)(C)C)NCC(C1CCC1)NC(c1cc(NC)no1)=O N1(C(C2CC(C(C)C)C2)=O)CC(NC(=O)C(=O)NC(C)C)CC1(C)C c1(OC)ccc(C(C)NC(=O)C(C)(C)C2CCCN2C(=O)CS(C)(=O)=O)cc1 N1(C(CCCC#C)=O)CCN(C(c2cccc(F)c2SC)=O)CC1CS(C)(=O)=O C12(NC(C(CCSC)NS(CC)(=O)=O)=O)CCCC1N(C(=O)C=C1CCC1)CC2 N1(C(C(C2CC2)OC)=O)CC2CCC1C(NC(=O)Cc1ccc(C)s1)C2 N1(C(c2c(C)cco2)=O)CC(C(=O)NCC(C)(C)CCO)C(C)(C)C1 C1(C(c2scc(C)n2)C(=O)NC2CCOCC2)C2CCC1CNC2 C1(C(=O)NC2C(NC(C=CSC)=O)CCCC2)CCCCC(C)(C)C1 N12CCC(n3cccn3)(CC1)C2=O.C1(NCc2occ(C)c2)CCN(C)CC1C C1(NC(C(CC)C)=O)CN(C(=O)CN2CCC(O)CC2)CC12CCSCC2 N1(C(C)C)CCC(NC(c2ccc(C(N)=O)cn2)=O)C(C)C1 N1(C(CC=C)=O)CCN(C(=O)C(c2ccccc2)OC2CCCC2)CC(CO)C1 C(C1CN(C(C2CCOC2=O)=O)Cc2ccccc21)NC(=O)CCc1cnco1 c1(OC)ccc(CC(C)OC(=O)CC2(O)CCN(C(C(C)(C)C)=O)C2)cc1.C1(C)CC1 c1(C(=O)NC2CCC(NC(C3CCC(=O)NC3)=O)C2)ccc2ncnc(O)c2c1 C(=O)(CC(C)(C)CNC(C1CC1OC(C)(C)C)=O)NC(C#C)C(C)OC c1(C(=O)NCC2(O)CCN(C(C3CC=C(C)CC3)=O)CC2)cc(C)c(=O)n(C)c1 C(=O)(CC(C)(C)CC(=O)N1CCCC1C(C)NC(=O)C(C(C)O)N(C)C)OC c1(C(N2CC(C)N(C(=O)CCCn3ccnn3)CC2)=O)cc2c(cn1)OCCC2 C1(NC(c2c(C(C)C)c[nH]c2)=O)CCCN(C(c2ccc(C(C)(F)F)nc2)=O)C1 n1(CC(N2CC(O)CC(NC(c3nocc3Cl)=O)C2)=O)ncc2cccnc12 C1(C(=O)NC2CN(C)CC2(F)F)CC2C=CC1N(C(=O)CCc1nccs1)C2 CCCC(C(O)C(=O)NOC1CC1)NC(=O)C(C)(O)CSC c1(OC)cc(C)cc(C(N2CC3(C2)CN(C(c2c(OC)noc2C)=O)C3)=O)c1N N1(C(C(CC)(C)CC)=O)CCN(C(c2cccc3oncc23)=O)C2(CCC2)C1 CC(C)CC(C(=O)NCC1CCC1NC(=O)CCC1CC1)N1CCCCCC1 c1(C(N2C(C3CN(C(C4C(C(=O)OC)C4)=O)C3)CCCC2)=O)ccnc(F)c1O N1(C(C(CC)F)=O)CCc2ccccc2C1CNC(=O)Cc1coc(C(F)F)n1 S(=O)(=O)(c1csc(CCNC(c2ccc(C3(C)CC3)cc2)=O)c1)NC c1(C(=O)NC2CCCC(NC(=O)C3=COCC3)C2)cnc2nccn2c1 c1(C(C)C)cc(Br)cc(C(F)(F)F)c1O.C12(CCOCC1)CC(=O)NC2 c1(C(N2CCC(C3N(C(=O)C#CC4CC4)CCC3)CC2)=O)cc(O)cc([N+](=O)[O-])c1 N1(C(C(C=CC)O)=O)CC(CO)C2(CCN(C(c3ccncc3F)=O)CC2)C1 C(CC(F)F)(C(=O)NCC1CCOC1)N(C(c1c(C)nncc1)=O)C C1(C(N2CCN(CCCNC(=O)CC3CS(=O)(=O)C3)CC2)=O)Cc2nncn2C1 C1(N(C(C(=O)NCCCSC)CC2CC(F)(F)C2)CC2CC2)CCCC(O)CC1 c1(C(C(=O)N(C)CCN(C)C(C2(Cl)CC2(F)F)=O)O)ccc(C#N)cc1 C(=O)(C#CC1(C)CC1)NC(C1CCCCN1C(c1nnc(O)cc1C)=O)C Cc1c(C(N2CCC(N(C3CC34CCC4)C)CC2)=O)cccc1F C(C(C)(C(C)C)NC(C1C(Cl)(Cl)C12CC2)=O)NC(Cc1ccc(C)s1)=O CN1CCC(C(=O)NCC(C)(C2CC2)NC(=O)CCc2ccncn2)C1=O C(=O)(CC(C)P(C)(C)=O)N1CCC(NC(c2cc(NC)nc(Cl)c2)=O)C(F)C1 C1(NC(c2c(C)cco2)=O)CCN(C(=O)Cc2cccc(C#N)c2)CCC1CO C1(C(=O)NCc2cccc(Br)c2)CCN(Cc2cccc(I)c2)CC1 C(=O)(CS(=O)(=O)CCOC)N1CCC(N(C(c2cccc(CC)c2)=O)C)CC1 CCC(C)(O)CC(=O)N(C)CCOCCCNC(c1cccc(CN=[N+]=[N-])c1)=O c1(OC)ccc(CNC(C2CC(C)CN(C(=O)CSC)C2)=O)c(F)c1 C1(C(N2CC3C(C(=O)NC4(CCOC)CCCC4)(C3)C2)=O)Cc2ccccc2C1 C1(CNC(c2c(C)ccc(Cl)c2)=O)CN(C(C2CC3CC3C2)=O)C2CCCC2O1 C1(C)(C(=O)NCCOCC(=O)NC)CCCN1C(C1(C)CC(C#N)C1)=O C(=O)(CCCCC(C)C)NC(CNC(c1cnc(OC)nc1C)=O)(C)C1CCC1 N1(C(c2cnc(NC(C)=O)o2)=O)CCC(NC(=O)CC2OCCC2(C)C)C1(C)C Cc1cc(CC(=O)NCC2(NC(C34CC(C3)C4)=O)CCC2)on1 C1(C(N(C2CCN(C(C3(C#C)CCC3)=O)CC2)CCC)=O)OCCOC12CCC2 CC1(NC(=O)CC2(NC(=O)Cn3ccnc3)CCC2)CN2CCC1CC2 c1(C(N2CCCC(CNC(CNC(CCCCC)=O)=O)C2)=O)cnc(N)c(N)c1 CC(C)(C(=O)N1CC(C2CCOCC2)(F)C1)n1cc(N)cn1 N1(C(CC=CC=C)=O)CCCC1(C)CNC(=O)Cc1coc(-c2ccccc2)n1 n1(CCC)cc(C(=O)NCC(F)CNC(=O)C(C)(C)c2ccns2)nn1 CCC(C)(CCNC(C1CCC1C)=O)NC(=O)CCC1CCC(=O)N1 c1(C(C)C(N2CCC(NC(=O)CC3CN(C(C)C)C3)C2)=O)cc2ccccc2o1 N1(C(C(C2CC2)OCC)=O)CCC(O)CC1C(=O)NC1CCCCC1C#N C1(N(C(C(=O)NCCC)=O)CC)CCC(N(C(=O)CCN(S(C)(=O)=O)C)C)CC1 c1(NCC(C(=O)NCC(CNC(C)=O)(C)C)c2ccccc2)c(C)n[nH]c1C n1(CCC)cc(C(=O)NC(C2CCCN2C(=O)CNC(N)=O)C)c2ccccc12 N1(C(C(CCC)OC)=O)CCC(C(=O)Nc2cccc(OCC)c2)CC1(C)C n1(CC(=O)NC2C=CC(CC(=O)NCc3ccco3)C2)cccnc1=O C1(C(N2CCN(CCc3ccccc3)CC2)C(=O)NCC(=C)C)C2CCOCC12 c1(C(N2CC(C)C(NC(C3CC4(C3)CC3(CC3)C4)=O)C2)=O)cccc2c1CCN2 C1(NC(=O)CN(C(c2ccc(O)cn2)=O)C2CC2)CCN2CCCC12 c1(CC2(C(N(CCC)C(c3ccccc3)C)=O)CNC2)ccc(Cl)cc1 c1(CCC)ccc(C(=O)NCCCN(C2CCCC2)C(=O)CO)[nH]1 C(=O)(C(CC(C)C)C(N)=O)N1CC(NC(c2cc3sccc3[nH]2)=O)CC(OC)C1 C(C)(C(C(=O)N1CC2C(C(=O)N(C)C)C2C1)NC(=O)CC(C)(F)F)OC N1(C(=O)C=CC2CCCN2)CCCC(N)(CO)C1 c1(C(=O)NC(CNC(c2c(NCC)scn2)=O)(C)CO)ccc(NC(C)=O)cn1 N1(C(C2N(C(CN(CC(C)(C)C)C)=O)CC2C)=O)CCC(C)(CO)C1 N1(C(=O)NCc2cn(C3CC(=O)NC3)nc2)CCOC(C2CCCC2)C1 C(=O)(C(C(C)C)n1cnc(C)c1)NCC1(NC(c2c(COC)ccs2)=O)CCC1 C1(CCC(=O)OC)(C(=O)NCCNC(=O)C(C)N(C)CCn2ccnc2)CCC1 C1(COC)(NC(=O)CC(C)N(C)C)CN(C(C2(OC)CCCC2)=O)C1 C1(C(=O)NC2(CO)CCN(C(=O)CCn3cnnn3)C2)CCOC2(CCC2)C1 c1(C(=O)NC(C2(O)CN(C(CC3C(CC)C3)=O)C2)C)ccc(C)c(F)c1 CCCCC(CNC(=O)CN1CCOC1=O)NC(C1(CC2CC2)CC1)=O C(C1c2ccccc2CCN1C(C1CCOCC12CCC2)=O)NC(=O)C1=CCC1 CCCCC(CC)CC(=O)NC(C)C(C)(C)NC(c1cc(CC2CC2)ncn1)=O c1(C(N(C2CCCN(C(=O)CNS(C)(=O)=O)CC2)CC)=O)cccc2c1COC2 c1(C(=O)NCC(C)(C2CCC2)NC(C(C)n2cnnn2)=O)cc(F)ccc1N N1(C(COCCOC)=O)CC2CCC(C1CO)N2C(c1cccc(F)c1)=O N1(C(C(c2ccccc2)NC(CC=C=C)=O)=O)CC(O)C(O)C1CO C1(C)(C(N2CCC(CN(C(=O)CCNS(C)(=O)=O)C)CC2)=O)CC(O)CN1C C(=O)(C(O)Cc1ccccn1)NCC(CC)NC(c1ncsc1Br)=O CC1CCC(NC(=O)C(C)(C)c2cccs2)CN1C(C1CC(O)CN1C)=O c1(C(=O)NC(C)CCNC(C2CCCC23CC3)=O)cc2c(s1)CC(C)(C)C2 CCC1=NOC(C(N2CCC(C(CO)NC(=O)Cn3ncccc3=O)CC2)=O)C1 C1(C(N(CC(C)CC)C(C2(C3CC3(C)C)CC2)=O)=O)CC(C(C)C)=NO1 C(=O)(C(C(C)C)OC(C)C)Nc1ccn(CCCOC)n1.C12(CCOC1)C(=O)NC2 N1(C(CC(=O)OC)=O)CCN(C(c2cccnc2C)=O)CC1CC(F)F N1(C(CCSCCC)=O)CC(F)CC1C(=O)N(C1CC(O)C1)C N1(C(C=Cc2c(C)coc2C)=O)C2CCCC1CN(C(c1ccco1)=O)CC2 N(C(=NCCn1cccn1)NCCC1(O)CCOCC1)C(CCC)C1CC1 N1(C2CN(C(C(Cc3ccsc3)NC=O)=O)C2)CC(NC(C2(F)CC2)=O)CC1=O C1(C(NOC(C(C)n2ccnn2)=O)=O)CCCCN1C(=O)CCN(C)C c1(CC(=O)NCCC(C)N(C)C(c2coc(CC(C)(C)C)n2)=O)ccccc1Cl C12(C(N3CC(C)(C)C(NC(=O)C(F)C(C)(C)O)C3)=O)CC(CO)(C1)OC21COC1 c1(CN2CCC(C#N)(Nc3cnc(Cl)cn3)C2)ccc2[nH]ccc2c1 Cc1sc(O)nc1C(=O)NCC(CC1CC1)C(=O)NC1CCN(C)C1=O C(=O)(C(C)Cc1ccco1)NC(CNC(C(C)NC(c1ccoc1)=O)=O)(C)C CCC(C(C)(C)C#N)NC(=O)NC(c1nnc2n1CCC2)C CCCC(C)(CCC)C(=O)N1CCC(O)C(NC(=O)CCc2ccsc2)C1 C(=O)(C(CC(C)C)N(C)C(C1CC1C(F)F)=O)N(CC=C)CC Cc1ccc(O)c(C(N2CCC(n3cc(CC(C(=O)O)C4CC4)nn3)CC2)=O)c1 c1(C(=O)NCCC(C)NC(c2cccc(S(C)=O)c2)=O)cc2c(F)cccc2[nH]1 C1(CC)CC(CC(=O)NCCOCCOCCOC)C1.C12(CCC1)C(=O)N2 c1(C(N(C)CCNC(c2c[nH]c(C#N)c2)=O)=O)ncc(Br)cc1C(F)F N1(C(C=Cc2scc(C)n2)=O)CCN(C(=O)C(CO)C(C)(C)C)C2(CCC2)C1 c1(N(C(C)C(=O)NO)CC=Cc2ccoc2)cn(CCN=[N+]=[N-])nn1 c1(CC)cccc(C(=O)NC2(CC(=O)NCC(O)C(F)(F)F)CC2)n1 c1(OCC(=O)NC2CN(C(CC3C(=O)NCCC3)=O)C2)ccc(F)cc1O C1(N(C(c2cc(OC)ns2)=O)C)CCN(C(=O)CCN2CCC(F)C2)CC1 N1(C(C(CC(N)=O)O)=O)CCS(=O)(=O)C(CCNC(=O)CN2CC3CC3C2)C1 N1(C(c2cnc(OC)s2)=O)CC2(CC2)CC1CNC(=O)CC1CCN(C)C1 C(C1c2ccccc2CCN1C(C1CC1C#N)=O)NC(C=Cc1ncc(C)[nH]1)=O [N-]=[N+]=NCCCC(=O)N1CCN(C(=O)CNC(=O)CSc2ncccn2)CC1 C1(C(=O)NCC2C(NC(C3CCC(N(C)C)CC3)=O)C2)CCCC1P(C)(C)=O N1(C(C(CC)C(C)C)=O)CCC2CCC(C1)N2C(c1cc(C(=O)OC)n(C)c1)=O C1(NC(c2c(CC)ncs2)=O)CN(C(c2[nH]c(C)cc2C(=O)OC)=O)CC1C C12(NC(CC(CCC)C)=O)CCCC1N(C(=O)C(C1CCOCC1)C)CC2 N1(C(c2cc(C(C)C)[nH]n2)=O)CC2CCC1CC2NC(=O)CCn1cnnn1 CS(=O)C=CC(=O)NCCCCCCNC(c1cccc(Cl)c1)=O C(=O)(CCCCCNC(C1CC1OC(C)(C)C)=O)N(CC(C)(C)O)C c1(CN(c2cnccc2C(N2CC(NC(N)=O)C2)=O)C)cc(O)ccc1Cl c1(C(N(CCN(C(=O)CCOC2CCC2)C)C)=O)cc2c(nn1)CCC2 N1(C(C2CCCN(CC(C)C)C2)=O)CC2(C1)SCCC2NC(=O)CNC(N)=O N1(C(C(C=C=C)C)=O)CC2CC(NC(=O)CC3(O)CCCCC3)C(C2)C1 c1(C(N2CCCC(CCNC(CCCCOC)=O)CC2)=O)cc2cccnn2c1 N1(C(CC(CC)SC)=O)CC(NC(=O)C(C)(C)C)CC1(C)C C1(C(N(C)CC2C(NC(C(C=C=C)C)=O)CCC2)=O)CN2CCN1CC2 c1(NC2(c3nnnn3C3CC3)C(C)SCC2)cc(F)c(CCO)cc1Cl S(=O)(=O)(CC(C)(C)Cc1ccccc1)N(CC(=O)OCC=C)C N1(C(Cc2cccc(OCC)n2)=O)CCC(C)(C)C1CNC(=O)C#CC(=O)NC c1(CCNC(C2CCC(NCc3csc(Br)n3)C2)=O)ccccn1 C1(CC)CN(C(=O)C(C(C)C)C2CCC2)CCN1C(c1ccc(C(C)C)o1)=O CC(C)CCCCC(=O)N1CC(C(C)NC(=O)Cc2cncc(O)c2)C1 c1(C(=O)OC)ccc(OC)cc1NC(C1CC1C(=O)Nc1cccc(Cl)n1)=O N1(CC(=O)NCC2(F)CC(NC(=O)CC3CCS(=O)(=O)C3)C2)CCCCCC1 c1(NC(=O)CCn2cccc2)ccc(O)c(Br)c1.C12CCC(C1)CNC2=O C1(COC)(NC(=O)CN(C2CCCC2)C)CN(C(=O)CC(C2CCC(=O)N2)C)C1 C1(NC(c2cc(CC)sn2)=O)CC=C(C(=O)NC2(C)CCCC2(F)F)C1 c1(C(N2CCC(N(C(c3sc(C4CC4)nc3C)=O)CC)C2)=O)cc(C)cc(F)c1 C=CCC(CC)NC(=O)Cn1cc(CNC(=O)COc2ccsn2)nn1 N1(C(C2N(C(c3c(C)nco3)=O)CCSC2)=O)CCn2nc(C(F)(F)F)nc2C1 C(CCCC(C)(C)NC(=O)C(C)C1CC1)NC(CCc1nc(C)c(C)[nH]1)=O C(c1cnc(O)nc1O)=CC(=O)NC1CN(C(CN(C)CC)=O)C(C)C1 c1(C(C(=O)NCC(C)N(C(C2CN(C(C)C)C2)=O)C)O)cccc2c1OCC2 C1(C(=O)NC2CN(C(CC3(N(C)C)CCCC3)=O)CC(F)C2)CCC2(CC1)CC2 CN1CCN(C2CCN(C(=O)NC3CC3(C)C(F)F)C2)CC1.c12ccccc1O2 c1(CCNC(N(CC(F)F)CC#C)=O)c(F)cccc1Cl C(=O)(CS(=O)C(F)(F)F)NCCC1CCCN(C(c2nc(C(C)=O)sc2)=O)C1 c1(C(=O)Oc2c(C(=O)OC)nc(C)[nH]2)ccc2c(-c3ccccc3OC)n[nH]c2c1 CC(C)(C)C(C(=O)NC1CN(C(C2(c3ccnc(Cl)c3)CC2)=O)C1)n1ccnn1 Cc1nc(CCCC(=O)NC(c2cn(Cc3cc(C)on3)nn2)(C)C)cs1 Cn1nccc1C(O)C(=O)N1CCC1CNC(=O)CCCNC(c1ccsc1)=O C12(OC)CCC(C(=O)NC3CCC(C(=O)NC4CCOCC4C)C(O)C3)(CC1)C2 C(=O)(CCC(C)CC)NCC(c1ccccc1)CNC(C(C#C)(C)C)=O CC1(C)CC(NC(=O)CC2(NC(=O)CC3(C)CCOCC3)CC2)CCO1 CC1CCCC(O)C1.C1(=O)CC(C2CCC2)CN1.C(=O)C(=O)C(C)C C=CC1(CC(=O)NCCNC(c2cc[nH]c2-c2ccccc2)=O)CCC1 C1(NC(C(CC)n2cccn2)=O)CCN(C(=O)CC(=O)NCC)CC1 N#CC1(C(=O)NCC(C2CC2)NC(C2COCCO2)=O)CC2CCC1CC2 CC1CC(NC(c2cnccn2)=O)CN(C(c2cnc(Br)nc2)=O)C1 C(=O)(C(CN=[N+]=[N-])NC(=O)CCc1cn(C)nn1)NCCn1cnc(C)c1C c1(CNC(C2C(C)C2C)=O)cn(CCNC(=O)CCCNC(=O)C(C)(C)C)nn1 Cc1noc(C)c1CNC(C)(CCCl)c1nnnn1C(c1ccccc1)C Cc1ccc2oc(C(=O)NC3CN(C(=O)C(C)OC4COC4)CCC3C)cc2c1 c1(C(N2CC(C(C)NC(C3CC(C)(c4ccccc4)C3)=O)C2)=O)ncc[nH]c1=O C1(OC)CC(C(=O)NC(C)CNC(c2sccc2CSC)=O)CC1OC C1(CC(=O)NC(c2ccnc(F)c2)C2CC2)Cc2ccccc2C1=O CC(C)(C)C#CC(=O)NCC1CCCCN1C(=O)CCCCCN1CCCCC1 N1(C(C(C)Cc2ccco2)=O)CC2CC2C1C(=O)NCCCSC(F)F CCC(F)(F)CC(=O)NCC(CC1CC1)C(N1CCSCCC1C)=O C1(CCNC(C=CCC)=O)CN(C(C2(COC)CCCC2)=O)CC(C)O1 C1(C(=O)NC2CC3CC(O)C2C3)CC2CCC1N2CCCc1ccccc1Br c1(C(=O)NCC2N(C(CC3C(OC)CC3)=O)CCCCC2)ccc2sccc2c1 CC1CC2(CCN(C(=O)CC3(CNC(C4CCN(C)C4)=O)CC3)C2)CO1 C(CC(C)(C)NC(=O)Cn1cc(Cl)cn1)NC(COCC(C)C)=O c1(NC(Cc2cccc(CN=c3[nH]cc(C)s3)c2)=O)cc(Cl)ccc1OC(F)F c1(C(=O)NC2(C3N(C(C(CC)CO)=O)CCC3)CC2)cccc2n[nH]cc12 C1(C(=O)NCC(C)(CO)NC(c2cccc(C(F)(F)F)n2)=O)OCCC1(C)C C=CC(CC(=O)N1CC(C(F)(F)F)CC1CNC(=O)C=[SH]CC)c1ccccc1 CC1=C(C(=O)NC(C2CCCCC2)CNC(C2CC3CCC2O3)=O)CCO1 C1(C(=O)NC(C2CN(C(c3ccc(CO)nc3)=O)C2)C)CCC2(CCC2)C1 C1(NC(C(CCC)N(C)C)=O)CCN(C(c2ncoc2C(C)C)=O)CC1O c1(C(=O)NC(C2CCN(C(C3CS(=O)(=O)C3)=O)C2)C)ccc(CN(C)C)o1 C1(C(=O)NCC(c2ccccc2)OC)CC(NC(=O)OC(C)(C)C)C(O)C1 C12(NC(c3cc(SC)c(C)o3)=O)CCC(C1)N(C(C1(CC(C)C)CCCC1)=O)C2 N1(C(c2c(C)cc(CC)o2)=O)CC2CC1CCN2C(=O)Cc1cc(C)[nH]n1 C(CC(C)(C)NC(C1CCCN1C(=O)CC1(C)CC1)=O)N(C)C N1(CC(C(C)(C)O)O)CCCCC12CCC2 n1(CCC#C)cc(C(=O)N(CC(C)N(C)C(C2CCC2(OC)OC)=O)C)nn1 C(C(=O)NCc1cccc(NC(=O)C(C)(C)c2cccs2)c1)(C(C)C)NC(C)=O N1(C(C(C)CC2CC2)=O)CC(C2CCCN(C(C3CC(C4CCCCC4)C3)=O)C2)C1 c1(C(=O)NC2C(CNC(C3C(=C)C3)=O)C2)ccccc1C(C1CCC1)=O C(=O)(CCC(C)(F)F)NC(CCC(=O)NCC(=O)NCCCC)C c1(CC(C(=O)N(CCCCC=C)C)N)cncc(Br)c1 c1(NC2C(C)NC(=O)CC2)ccc(C#N)c(F)c1C#N c1(C(N2CCC(n3cc(CCS(N)(=O)=O)nn3)C2)=O)cc(F)c(Cl)cc1F CC1CN(C)CCN1C(=O)CC1CCC(NC(C2CC3(CCC3)C2)=O)CC1 c1(C(=O)NCCC2(O)CN(C(Cc3c(C)cnn3C)=O)C2)nnc(O)nc1O C1(NC(=O)Cn2cc(C3CC3)nn2)CCCN(C(=O)CCn2cccc2)C1 C#CC1(O)CC(C(N2CCC(C(=O)NCc3cnccc3C)(CF)C2)=O)C1 c1(C(N2C3CN(C(c4c(N)cc(F)cc4)=O)C(CC3)C2)=O)cccc2cnccc12 c1(CC)ccc(CN(C(=O)C(=O)NC(CCF)C(=O)OC)C)cc1 C1(NC(=O)C=C2CN3CCC2CC3)CC2(CCCN(C(=O)CSc3nncs3)C2)C1 CC1CNc2ccc(C(=O)NCC(C)(C3CC3)NC(c3ccoc3Br)=O)cc21 C1(C(=O)NC(C)CCNC(c2ccn(C)c2)=O)CCC2(CCOCC2)CO1 c1(C(N2CC(CNC(c3cc(C(C)=O)on3)=O)C2)=O)cc2scc(Cl)c2[nH]1 c1(OC)ccc(NC(=O)NCCCCN2CSCCSC2)c(OC)c1Cl c1(CC)ccc(C(=O)NC2(C)CC(NC(=O)CCC3CC3(C)C)C2)cc1N c1(CC(=O)NC2(CO)CCN(C(=O)CC3CCCC3)CC2)c(F)ccc2occc12 C=CCCC(F)(F)C(=O)NC1CC2CC(C1)N(C(C)CC1CCOC1)C2 c1(CC(N2CC(CC(C)NC(c3ccc(Cl)o3)=O)C2)=O)c[nH]c2ncccc12 C1(C(N(CCCC)CCOC)=O)CC(C)(NC(C2CC(F)(CF)C2)=O)C1 Cc1cc(C(=O)NCC2CCCC2C(=O)NCCCCCCF)c(O)nn1 c1(CNC23C(CN(C(c4c(OC)cncc4)=O)C2)C3)cc(C)nc(C)c1 c1(OC)cccc(NCC2(CNC(c3ccc4sccc4c3)=O)CC2)c1[N+](=O)[O-] c1(NC(c2c(C)nc(NC(c3ccc(Cl)cn3)=O)s2)=O)cccnc1[N+](=O)[O-] c1(NC(C2(C)CCCO2)=O)c(-c2cncc(Br)c2)noc1C1CC1 C(=O)(CCC(C)C(C)(c1cccnn1)NCCCN(C)C)OC C1(OCCNC(C23CC(OC)C2C3)=O)(NC(C2CCC(C)CC2)=O)CC(F)(F)C1 c1(C(C)(C)C)cc(C(N2CC(CCNC(C3(c4cc[nH]n4)CCC3)=O)C2)=O)no1 c1(C(N(CC(CNC(Cc2cccc(OCC)c2)=O)O)C)=O)cccc(F)c1C Cc1nn(-c2ccccc2F)cc1C(N1CCC(O)(C(=O)N(C)C)C1)=O C(C)(C)(C(=O)NCC1(NC(=O)CCN2CCCCC2)CC1)NC(=O)OC c1(C(=O)NC(N2CC(COC)C(F)(CO)C2)=O)cnc2cc(C)nn2c1 CN1CC=C(CC(=O)NC2CN(C(c3csc(CO)n3)=O)C3CC23)CC1 C(=O)(C(C)CC(F)F)NC1C(NC(CCc2cc(C)sc2C)=O)CC1 Cc1cc2[nH]c(=NC(COCc3ccccc3)C(C)C(C)C)ccc2cc1C Cc1ccc2cc(C(=O)NC3C4CC3N(C(C3CC5(CC5)CO3)=O)C4)cn2c1 C1(CC(N2CCC(N(C(=O)CN3CCS(=O)CC3)C)C2)=O)CCCCC1(F)F N1(C(c2scc(OC)c2)=O)CCC2(C1)CN(C(=O)CC(C)P(C)(C)=O)C2 c1(OC)cccc(S(=O)CC(=O)N2CC3CCCN(C(c4cccs4)=O)C3C2)c1 C(=O)(C1=Cc2ccccc2OC1)N(CCCNC(c1c(CC)c[nH]n1)=O)C(C)C c1(C(N2CC(CC)N(C(=O)CC3CCCC3O)CC2)=O)ccc2ncn(C)c2n1 CC(C)C(O)CC(=O)N1CC(NC(=O)CC2(C)OCCO2)C1 Cn1ccc2cccc(CNc3cnc(F)cc3C(=O)NCCF)c12 C(=O)(C(CC(C)C)N(C)C(c1cnn(C(C)C)c1)=O)NC(CC#CC)C N1(C(c2ccc(C)s2)=O)CC(NC(C2CCn3nccc3C2)=O)C2CCCCC12 Cc1cnc(CNC2CC(C(=O)NCC3CCCO3)C2)cn1 N1(C(c2ccc(C)c(C(F)(F)F)c2)=O)C2CCC1CC(NC(C1(CF)CC1)=O)C2 CCCC(C)CCCC(=O)N1CCCC1C(C)NC(=O)Cc1nc(=N)[nH][nH]1 C1(OC)CCCCC1NC(C1C2CC1N(C(c1c(C)noc1C)=O)C2)=O Cc1ccc(C(=O)N(CC(O)CN(C(=O)CC(C2CC2)C2CC2)C)C)cc1Cl CCC(O)CC(=O)N1CCCC(CCNC(c2cc(C(N)=O)co2)=O)C1 C=CC(C)CCN=c1[nH]c(=NC2CCOC2CC)c2cccc(F)c2[nH]1 N1(C(Cc2nc(C)[nH]n2)=O)C2CCC1C2NC(=O)CN1CCC(CO)CC1 C(=O)(C(C(C)O)N(C)C)NC1CC(C(C)NC(c2c(C(C)C)noc2)=O)C1 c1(NC(C2(OCC)CC2)C)nc(=NC(C)c2ccsc2)[nH]c2ccsc12 C1(NC(CC(COC)COC)=O)CC2CCCC(C1)N2C(=O)CN1CC2CC2C1 C1(NC(Cc2c(C)ncs2)=O)COCCC1NC(C1(c2cscn2)CC1)=O N#Cc1ccncc1C(N1CCC(O)(CNC(=O)CC2(CO)CCCC2)C1)=O N1(CC)CCC(C(=O)NCCN(C(=O)COc2ccccc2)C(C)C)C1 C(C(C)(O)CNC(c1coc(-c2ccsc2)c1)=O)NC(COC(C)C)=O c1(NC(c2c(C)ncs2)=O)ccc(C#N)c(C(F)(F)F)c1.C12CN(CC1C)C2=O Cc1nc(C[N+](C(CN(C)C)C(C)C)([O-])[O-])co1.N1(C)CCCC1CC=O C1(CCN2CC(C)(C(=O)NCC3(F)CCCC3)C2)COc2ccccc2O1 N1(C(c2n[nH]c(C)c2Cl)=O)CCC(NC(=O)C(F)C2CCC2)C(O)C1 N1(C(c2cn(C)nc2)=O)CC2C(NC(=O)CCC(c3ccccc3)C3CC3)C1C2 CC(C)CC(C)(O)C(=O)Cc1cc(-n2cc(C(=O)NC34CC(F)(C3)C4)nn2)no1 N1(C(C(C(=O)OC)C)=O)CCN(C(C2CC(F)(F)C2)=O)CC1CC(F)F N1(C(CCc2cc(C)on2)=O)CC2CC(C1)N2C(C1(C)CCCCC1C)=O C(N=c1[nH]c(=NC)[nH]c(=NCC2CCOC2)[nH]1)c1cc(CCC)no1 c1(C(=O)NCC2CN(C(COC)=O)CC2(C)C)ccc2nn[nH]c2c1O N1(CC2CCCC(OC(C)(C)C)C2)CCOc2cc(Cl)ccc2C1 C12(CC(=O)NCC3(O)CN(C(Cc4n[nH]c(=NC)s4)=O)C3)CCCCC1C2(F)F C(=O)(CCCCCSC)N1C(CNC(C2(CC=C)CCCC2)=O)(COC)CCC1 N1(C(c2cc(CNC(COCC)=O)on2)=O)CCC2CCC(O)C1C2 CC1Cc2ccccc2N1C(C1CC2CC2N1C(c1ccc2nccn2c1)=O)=O c1(C(=O)NC(C2CCN(C(=O)C(C)N(C)C)C2)C)ncc(F)cc1F c1(C(=O)NCC2CCCCN2C(c2cc(F)cc(F)c2)=O)cccc2c[nH]nc12 c1(C(=O)NC2CN(C(C3C(C(C)O)C3)=O)C2)cccc(C(N)=O)c1 N=c1ccc(C(N2CCC(C3CCN(C(=O)CNC=O)CC3)C2)=O)c[nH]1 N1(C(C2CCCCN(C(CSC(C)C)=O)C2)=O)CCC2(CNC(=O)O2)C1 C(c1ccc(F)c(F)c1)=CC(=O)NCCCN(C)C(C1CCCC(C)(C)C1)=O C#CCCC(=O)N(C1CC1)CC1CCCN1C(=O)CN1CCOCC1 S(=O)(=O)(c1ccc(NC(C2(CF)CC2)C2CC2)cc1Cl)NCC1(N2C(=O)OCC2)CC1 CCC(C)C(CC(=O)NC(c1cc[nH]n1)C)NC(=O)C=Cc1cc[nH]n1 N1(C(C(CC)C(C)C)=O)CC2CCCC2C1C(=O)NC(CC1CC1)C1CC1 c1(CN2CCN(C(c3c(OC)cccn3)=O)C3C2C3)c[nH]c2ccc(Cl)cc12 N1(C(CC=C=C)=O)CCN(C(c2cn(CC)cn2)=O)CC1CC(F)F Cc1cc(C(=O)NC2CC(CO)N(C(=O)CC(F)(F)C(F)F)C2)c2c(c1)CCO2 N1(C(c2c(C(C)C)cco2)=O)C2CCC1C(NC(=O)Cc1n[nH]cc1Br)C2 C1(F)(C(N(CC(C)NC(COc2cccc(C(C)C)c2)=O)C)=O)CCS(=O)(=O)C1 CC1(C)CC(=O)NC1COC1CCC(OC(=O)C=Cc2ccc(Cl)cc2)C(O)C1 N1(C(CN(CCC)C)=O)CCCC2CCN(C(c3cn(CC(N)=O)nn3)=O)CC12 C(=O)(C(C)(C)CN(C)C(c1ocnc1CCC)=O)NCC(C#C)C(C)C N1(C(CC=CC)=O)CC2(CCCC(CNC(=O)C=Cc3sccc3C)O2)C1 Cc1cc(C(=O)NC2CC(C)N(C(C3CC4(CC4)C3)=O)C2)c(O)cc1F C(CN=c1cc(C2CC2)nc(C2CC2)[nH]1)=CNC(=O)CSc1nnc(C(F)(F)F)s1 C1(NC(=O)CC2CC(NC(=O)NCC#CC(F)(F)F)C2)CCC2(CC1)CC2 c1(C(N2CCCC(F)CC2)C(=O)NCCC)cc2cc(Cl)ncc2o1 C1(N(C)C)CCC(C(N2CC(CNC(=O)CCc3cnn(C)n3)C2)=O)C1 c1(C(N2CC(C)CC(C)C2)C(=O)NC2(C)CC2)cc(Cl)c2c(c1)OCCCO2 S(=O)(=O)(c1cccc(N(C)CCOCCOC)c1)N1C(CCCC)CCC1.C(C=C)OC Cn1cncc(C(N2CC(O)(CNC(C3CCCCC3O)=O)C2)=O)c1=O Cc1c(C(=O)NC2C=CCN(C(c3c(Cl)nsc3Cl)=O)C2)ccc2[nH]ccc12 CC1(C(=O)NCc2nc(C3CC3)no2)CCCN(C(c2ccc(=O)oc2)=O)C1 C1(COC)(NC(=O)Cc2ccnn2C)CN(C(C2(C)CCCO2)=O)C1 C1(C(=O)NC(C)CC2CCC2)CC2(CC(NC(C3CC(O)C3)=O)C2)C1 c1(C(N2CCC(OCCNC(C3CC3Cl)=O)C2)=O)cnc2ccccc2c1 C1(=O)C(C)(C)N1.C(CC(C)NC(N)=O)N(CC)CC.C(C)(=O)NCC CCC(C)C(O)C(=O)NCC1CC2(C1)CN(C(=O)Cc1cncn1C)C2 CC(c1ccccc1F)=CC(=O)NCCNC(=O)C(F)(F)C1CCCC1 CCC(F)(F)C(=O)NCC(C)(F)CNC(=O)CC(C)C1CCCC1 c1(C(=O)NCc2ccc(C(=O)NC(c3ncnn3C)CC)nc2)ccc(F)c(C)c1 C1(NC(C=CCC)=O)CCC(CNC(=O)C(CC)NC(C)=O)C1 N1(C(CCN2C(=O)CCC2)=O)CC2COCC(C1)C2NC(C1CC12CC2)=O CCCC(C)(C)CC(=O)N1CCC(C2CCCN2c2nccc(CC#N)n2)CC1 c1(C(C)N(CCCOC2CCC2)C(c2ccsc2)C)nnnn1C1CCC1 N1(C(c2cc(C)c(Cl)cc2)=O)C2CCC1C(CO)N(C(=O)C(C)CC1CC1)C2 N#Cc1ccc(O)c(NC(C2(CNC(c3ncoc3C3CC3)=O)CC2)=O)c1 N1(C(c2ccc(NC(C3C(OCC)C3)=O)cc2Br)=O)CCN(CC)C(=O)C1 c1(C(=O)NC(C)CN(C(=O)Cn2cc(CO)nn2)C)cn2cc(Cl)cnc2n1 C1(C(=O)NC2CCC(OC)C2)C=CCCN1C(=O)Cn1nnc(C)n1 c1(OC)ccc(Br)cc1C=CC(=O)NCCOCCNC(=O)Cc1cnoc1 C1(NC(c2n(C(CC)C)ncc2)=O)CC12CCN(C(c1n[nH]c(C)c1Cl)=O)CC2 N1(C(C(c2ccc(C)s2)C)=O)CC2C3CCC(C2C1)N(C(=O)CN(C)C)C3 c1(C(=O)NC(CN(C(c2c(C)n(C)nn2)=O)C)C)cc(O)nc2c1CCCC2 [N-]=[N+]=NC1CCCC1OC1CN(C(C=O)CCNC(=O)C=CCO)C1 N1(C(C(C)CC(N)=O)=O)CC(C)(C)OCC1CNC(=O)CC1CCSCC1 C1(CNC(C=C(C)CNC(=O)CN2CCCCC2)=O)CCCC12CC2 C1(CCN)CN(C(=O)Nc2csc(C3CCCN3)c2)CCO1 C1(CC=C)(OC)CCOCC1.C1(NCc2nnnn2CCOCC)CC2C=CC1C2 c1(SCC(N2CC(N(C)C(C3(F)CCOC3)=O)C2)=O)ccc(F)cc1 C1(NC(C2CCN(C(C)=O)CC2)=O)CN(C(c2cc3ccsc3s2)=O)C(C)(C)C1 c1(C(=O)NCCN(C(c2cccc(CC)c2)=O)C)cccc([N+](=O)[O-])c1OC C1(CNC(c2ccc(CC(C)C)s2)=O)C2CN(C(C3CCC3(C)C)=O)CC12 c1(C(N2CCC(N3CCN(C(C4C(OC)C4)=O)CC3)C2)=O)cnc2[nH]nnc2c1 N1(C(CC(CCOC)(C)C)=O)CCCC12CCN(C(=O)C(F)C1CCCC1)C2 c1(OC(C(=O)NCCC(C)NC(c2c[nH]c(C(F)(F)F)c2)=O)C)cccnc1 c1(C(Cc2onc(-c3cccc(C(=O)OC)c3)n2)C)cccc2c1OCC2 N1(C(C)=O)CCc2cc(C(C3(n4cc(-c5ncsc5C)nn4)CC3)=O)ccc21 CCCC(C(=O)NC1(CCOC)CCN(C(=O)CCOCC(C)C)C1)OC C1(C(C)(C)C)CC(C(=O)N(C2CCCN(C(C3CSCCS3)=O)C2)CCO)=NO1 C1(C(=O)NC(c2ccccn2)Cc2c(C)cccc2)CCCN(C(=O)C(C)C)CC1 c1(C(N2CCS(=O)(=O)C(CO)C2)C(=O)NCCSC)c(Br)ccc2ccccc12 CC1(C)CC(C)(CNC(C2C(C)(C)C2(F)F)=O)CN1C(C1CC2CCC1CC2)=O n1(CCC)ncc(C(=O)N(C(C)CNC(=O)C(c2ccc(OC)cc2)C)C)c1C C(=O)(C1=NNC(=O)CC1)NCCC1N(C(c2cn(C(C)(C)C)nc2)=O)CCSC1 N1(C(CCCN(C)C)=O)CC(C)(C)OCC1CNC(=O)CCSCC(N)=O CC(CO)C(=O)N1CC(c2ocnc2C(=O)OCC#N)C1.C12CC(F)(C1)CNC2=O C1(CNC(c2ncccc2CO)=O)CC12CCN(C(c1cncc(Cl)c1)=O)CC2 C1(NC(C2(OC)CC(CF)C2)=O)CC2(C1)CN(C(=O)C(F)C1CCC1)C2 c1(-c2onc(CN3CCC(C(N=S(CC)(C)=O)=O)CC3)n2)cn2c(n1)CCCC2C C=Cc1ccc(C(=O)NC(CC(=O)N2CCOCC(C)C2)C(C)OC)cc1 C(=O)(CCCCC(C)(C)C)N1C(CC)CN(C(C2CCC(O)C2)=O)CC1 N1(C(c2cccc(OC)n2)=O)C2CCC1CC(O)(CNC(C1CCSCC1)=O)C2 C12(NC(C(C=C)O)=O)CC(CNC(C3CCC4(CCC4)OC3)=O)(C1)OC2(C)C C(C1CCCCC1)=CC(=O)NCC1CCC(NC(c2ccncc2F)=O)CC1 C(=O)(N1OC2C=CC1CC2)c1cc(CNC(c2ccc3nonc3c2)=O)sc1 N1(C(C(CC)C)=O)C2CCC1C(F)C(NC(c1snc(Cl)c1Cl)=O)C2 c1(OC)c(C(N2CCCC2C(C)C(=O)O)=O)cccc1F N1(C(c2nc(C)[nH]n2)=O)CCN(C(c2ncn(C(C)C)n2)=O)CC1CO c1c(C)cc(C)cc1C.c1(CNC(C(CC)C)N)ccccc1CO C1(C(=O)NCc2ccncc2)C2CCCC1CN(Cc1c(F)cc(Cl)cc1F)C2 N1(CCC)CC(C(N2CCOC(C3CN(C(=O)CNC(=O)CC)C3)C2)=O)CC1=O N1(C(CC(CC)C)=O)CCCOC(CNC(=O)CCc2ccccc2OC)C1 c1(CC)nc(O)c(C(=O)NCC(C)NC(C23CCCC2C3(F)F)=O)cc1C c1(CC)cncc(CC(N2CC(CNC(C3(CC)CCC3)=O)(OC)C2)=O)c1 N1(C(c2ccn(CC)n2)=O)CC(CNC(=O)CSC(C)C)OC(C(F)(F)F)C1 N1(CC2CCN(C(C3CC(OC(C)C)C3)=O)C2)CCCCC1C.C(C)(C)(C)OC.O c1(CC(=O)NCCN(C(=O)C(O)CC2CCOCC2)CC)cncc(C#N)c1 c1(C(=O)NCC(N(C(=O)C=CSc2nc[nH]n2)C)C2CC2)cc(Cl)cn1C Cc1ccc2sc(N3CC4CCCC(NC(c5cnccc5Cl)=O)C4C3)nc2c1 c1(C(=O)NCC2N(C(CNC(=O)OC)=O)CC(OC)C2)n[nH]c2ccc(F)cc12 C1(NC(Cc2n(C)ncc2)=O)CCCCC1NC(C1C2CCC1(c1cscn1)C2)=O S(=O)(=O)(c1cccs1)N(C(C(=O)NC12CC(NC(COC)=O)C(OC1)C2)C)C C1(C)(CNC(CSCC=C)=O)CCC(NC(=O)C(c2cccc(Cl)c2)O)CC1 C1(N(C)C)CN(C(=O)CNc2ccc(N3CCCC3)cn2)CCC1(F)F N1(C(=O)Nc2ccc(OCC)c(C)c2)CCC2(CC1)C(F)(F)C21CCC1 c1(OC)ccc(C(=O)NCC2CCN(C(=O)C(=O)NCC(F)(F)F)C2)nc1 N1(C(C(CCOC)C)=O)CCC2(CC1)CC2C(=O)NCC(C(C)C)OC CC(C(C)(C)NC(c1csc(O)n1)=O)NC(=O)C=Cc1ccco1 C12(CNC(CCc3scc(C)n3)=O)CC(NC(c3snnc3C)=O)(C1)C(C)O2 C(C(C(C)(C)C)NC(=O)CCCF)NC(CCN(C(CCC)C)C(C)C)=O CN1N=CC(CC(=O)NC2CC(OCC(N3CCC(F)CC3)=O)C2)C1=O.C1CN1 N1(c2nnc(C)s2)CCc2c(c(CNC(=O)C(F)F)nn2C)C1 CCC(CC(F)F)C(=O)NCC(C)CNC(C1(c2cccnc2Cl)CC1)=O CN1CCC2CC1CCN2C(c1cccc(F)c1CO)=O C=C=CC(C)C(=O)NCCOC1CCN(C(c2nocc2CC)=O)CC1 CCC(O)C(C)C(=O)NC(C)(CC)CCNC(=O)Cc1ccc(OC)nc1 CN1CCN(C(C2CC(F)C(=O)N2)=O)C(C(=O)NCc2csc(CCO)n2)C1 CC1OC2(COC(=O)CCCCCCCNC(=O)OC(C)(C)C)CCC1CC2 c1(C(=O)OCC)cc(C(N2CC(O)CC2c2cccc(F)c2)=O)cc([N+](=O)[O-])c1 C(=O)(C=CS(C)(=O)=O)N1C(CNC(=O)C(c2cnn(C)c2)O)CC(OC)C1 C(=O)(CC1OCc2ccccc21)NCC1CCN(C(C(C)(C)O)=O)C1 C#Cc1nccnc1NC(C1C=CCN1C(=O)C(c1ccc(O)cc1)C)=O C(=O)(C(CC(C)(C)C)NC(c1csc(=N)[nH]1)=O)NC(c1ncccc1F)C O=C1CN(CC(=O)NCC(O)CC(=O)NCC2CCC(F)(F)C2)C(=O)N1 c1(C(C)C(=O)N(C(C(=O)O)C2CC2)C)cccc(Br)c1 Cc1ccc(CC(=O)NC2CCC(CNC(c3csnc3C(C)C)=O)C2)cc1Cl C1(C(=O)NC2CC(C)(NC(c3cn(C4CC4)nn3)=O)C2)C2CCC1(C(F)(F)F)C2 C(=O)(C#CC1CCCO1)NC1CCC(NC(Cc2ccc(OCC)cc2C)=O)C1 N1(C(=O)CC2(C(F)(F)F)CC2)CCCC(C2CCCN2C(=O)CCC(F)F)C1 C(=O)(C(O)C(F)(F)F)N1CCCC(OC2CN(C(=O)C(F)C3CCCC3)C2)C1 c1(-n2ccc(C(=O)NC(C)(C)CNC(C3C4COCC34)=O)n2)ccc(F)c(Cl)c1 Clc1nc2cc[nH]c2c(=NCCc2nc(C(c3ncccn3)N)cs2)[nH]1.C1CC1 C1(C)(CC(N2CCC(OCC(=O)NC(C3CCC3)C)C2)=O)CCCCC1 Cc1nc(C)c(C(=O)NC2C3CN(C(=O)CCC(N)=O)CC23)c(C)n1 N1(C(=O)Nc2cc(CCN)on2)CCN(c2cccc(Cl)c2)CC1.CC(=O)SC c1(C(=O)NCC(=CC(=O)N(C(C(N)=O)C2CC2)CC)C)cccnc1 N1(C(c2c(OC)cc(C)s2)=O)CCN(C(C2(C3CCCCO3)CCC2)=O)CC1C c1(C(=O)NCCCN(C(=O)C(C2CCC(=O)N2)C)C(C)C)ncsc1C1CC1 c1(CCCOC)cnc2[nH]cnc(N3CC4CC(C3)N(Cc3ccccc3)C4)c1-2 C1(NC(=O)CCCc2cnco2)CCCN(C(=O)CCO)C1.C1(=O)CCCNC(=O)N1 C1(NC(c2cc(Cl)no2)=O)COCCC1C(=O)N(C1CC1)CC1CCNC1 C1(C)(C(=O)NCCN(C)C)CCN(CCCNC(CN(C(C)=O)C)=O)CC1 N1(C(C(CC)C)=O)CCC(C(=O)N(C)CCNC(c2nc(Cl)cs2)=O)CC1 CC1CCN(C(=O)Cc2cn[nH]c2)CC1NC(c1cc(SC(F)(F)F)ccn1)=O C(=O)(C(C)(C)C(=O)NC1CCCC(NC(=O)CSCc2ccc(Cl)cc2)C1)OC C(C(=O)NCC1CN(C(c2cc(N)ccc2F)=O)C2CC12)(C(C)(C)C)N(C)C CN1CCC(C(N2CCC(C(N)=O)CC2)=O)(NC(C2CC2(C)C(F)F)=O)C1 Cc1ncc2n1CC(NC(C1CC3CCC(C1)N3Cc1cnco1)=O)CC2 c1(N2CCC3(C)C(C2)C3(Cl)Cl)ccncc1S(=O)(=O)NCc1cccc(Cl)n1 C1(O)(CCNC(C2(CC#C)CCCC2)=O)CCN(C(=O)CCNS(C)(=O)=O)CC1 C1(C(N2C(C(C)NC(c3c(CC)csc3)=O)CCC2)=O)COC(C)(C)CO1 C1(CNC(C(C)(C)COCC(F)F)=O)CCCN(C(=O)CC2CCC(=O)N2)CC1 C1(CNC(C)=O)CCCN1C(=O)C(c1ccnn1C)NC(=O)C(O)C1CCC1 n1(N2CC(NS(c3c(C)cc(C)cc3C)(=O)=O)C2)ncc2cccc([N+](=O)[O-])c12 Cc1cncc(C(N2CCC(C(F)F)(CNC(=O)CCN3CCC3)C2)=O)n1 N1(C(C2CCN(CCC)CC2)=O)CCC2CC1CN2C(C1CC(=O)NC(=O)N1)=O C1(OCC#C)CCCN(C(=O)C(N2CCOC(c3noc(C)n3)C2)=O)C1 CC1(C)C2CCC(C(=O)NC3CC4CC(NC(C5(N(C)C)CCC5)=O)CC34)C1C2 C1(NC(CC2(C=C)CCOCC2)=O)C2CCN(C(c3cnsc3C)=O)CCC12 C(=O)(C1=CCCCC1)NC1C(OC)CN(C(C23CC(C2)C3)=O)C1 N1(C(C(CCC)C#N)=O)CCC2(C(=O)NCC3(CF)CC3)CCCC12 N1(CC(C)C)N=C(C(=O)N(CCCNC(C2C(Cl)(Cl)C23CC3)=O)C)CCC1=O C1(O)(CN(C(=O)CC2CCC2(C)C)C)CCCN(C(=O)CC2(C)CC(F)(F)C2)C1 N1(C(CC(CC)C2CC2)=O)C(CNC(=O)CCCC(C)C)CC2CCCCC12 c1(OC)nc(C)c(C(=O)NC2CCC(C(=O)Nc3ncccc3O)C2)s1 C1(NC(C2CCC3CC3C2)=O)CCCCC1N=c1cc(Cl)nc(C2CCCO2)[nH]1 O=C(C1=NOC2(CCC2)C1)NC(CCCNC(=O)C=Cc1ccccc1)C1CC1 N1(C(C(C)C2(O)CCC2)=O)CCCC1(C)CNC(C1(C)CCCS1)=O N1(C(C(CC(C)C)N(C)C)=O)CCOCC(C)(CNC(c2ccnnc2O)=O)C1 n1(CCOC)ncc(C(=O)NC2CC(F)(CNC(c3c[nH]nc3F)=O)C2)c1C [N-]=[N+]=NCC(C(=O)NCCCc1cccnc1)NC(C1CC=CCO1)=O N1(C(C)=O)CCC(c2n[nH]cc2CNC(c2csc(-c3ccccc3)c2)=O)C1 CCC(CC(=O)NC1CN(C(=O)CNC(=O)Nc2ccoc2)CCC1F)C(C)C N1(CCN)CCN(CCO)CC1.c1(C(=O)NCc2c(C)cns2)cn(C)c(C)n1 c1(OC)cc(N(C)C)ccc1C(N1CC(CNC(=O)C2=COCCC2)C1)=O CN1C(=O)COc2ccc(C(=O)NCC3CC3NC(=O)C=Cc3ncc[nH]3)cc21 N1(C(C)C)C(=O)COCC1C(=O)N(C(C)CCNC(=O)C(c1cccn1C)=O)C C1(NC(C2(CC)CC2)=O)CC2CC(NC(=O)CN3CCC3C)CC2C1 c1(C(C)(C)C)ccc(C(N2CCC(C(=O)NCc3sccc3Br)CC2)=O)cc1 C1(C(=O)NC2C(C)(C)C(O)C2)C2CC3C(C2NC(C2C=CCS2)=O)C13 c1(C(=O)NC(CCCC)CNC(=O)Cc2cccnc2C)ccc(O)c(C)c1C C(CCCCCC(=O)NCc1nccs1)n1cc(CN(C(C)C)C)nn1 C1(NC(c2cccc(OC)n2)=O)CCN(C(=O)CC2CCN(C)C2)C(C)C1 c1(C(=O)NC(C(C)C)CNC(=O)Cc2cnsc2)cc2cccnc2[nH]1 C1(OC)CCC12CC(C(N1CCCC1CNC(=O)C(C)OC(C)C)=O)C2 C1(CC)CN(C(=O)C(CC(C)C)N(C)C(C2(n3ccnn3)CC2)=O)CC(=O)N1 c1(N2CC(C)C(NC(=O)CC(C)(C)C3CC3)CC2)ncnc2ccccc12 c1(C(N(CCCNC(C(C)Cn2ccnc2)=O)C)=O)nc(Cl)c(Cl)s1 N1(C(CNC(=O)CC2CC=CCC2)=O)CCCC(OCc2cc(C3CC3)[nH]n2)C1 C1(C(F)(F)F)(OC)CC(NC(=O)NC(C)CN(C)C)C1 C1(C=O)CC(=O)N(C(C)C)C1.c1(C(=O)NC(C(C)F)C)csc(CO)c1 c1(CC(=O)N(CC(O)CN(C)C(C2CCCC23CC3)=O)C)csc2nccn12 C1(CNC(C(C)NC(C)=O)=O)COCCN(C(=O)NC2CN(CC(F)(F)F)C2)C1 c1(OC)cc(C(=O)NCCC(C)N(C)C(C2CC(O)CN2C(C)=O)=O)ncn1 c1(C(=O)NCCC2(CNC(=O)Cn3cnnc3O)CC2)cc2cnccc2o1 n1(CCC(=O)NC(CNC(Cc2scc(C)c2)=O)C(C)C)cccnc1=O N1(C(C=C(CC)CC)=O)CCC2(NC(c3coc(C(=O)OC)c3)=O)CC2C1 C(CSC1CCC1)(C(=O)N)C(c1ccccc1)=O.C12CCCC1C2.C(CCOC)S C=CC(C)(C)CC(=O)N1C2CCC1C(CNC(C1(CO)CCCO1)=O)C2 CCC(C)(C)C(=O)C(=O)N(CCC(=O)NC1CCOC(C)C1)C(C)C c1(C(N2CCC(CNC(CCCCC#C)=O)(OC)C2)=O)ccc(F)cc1[N+](=O)[O-] c1(SC)cccc(F)c1C(=O)NC1CCC1NC(c1cnc(C)[nH]1)=O c1(OCC)cc(C(=O)OC(=O)C(O)(CSC)CSC)ccc1F c1(C(=O)NC2(C)CC(NC(C3ON=C(C)C3)=O)C2)cc2c(C)c(F)ccc2[nH]1 N1(c2nnc(C)o2)CCC2(CN(C(=O)Cc3ccc4n[nH]cc4c3)CCO2)C1 c1(COCC)cc(C(=O)NC2CN(C(=O)CC(=O)OC)CC2O)ccc1OC C=CC1(C(=O)Nc2cnccn2)CCN(C(=O)C(O)CC(C)C)C1 Cc1nc(C(=O)NCCC(C)NC(=O)C=Cc2cnc(C(C)(C)C)s2)nn1C Cc1ccn(C(C)CC(=O)NCC2(CCNC(C3(C)CCCO3)=O)CC2)n1 c1(C(=O)NC2CC(C)CN(C(c3ccn(C)n3)=O)C2)cc(O)c(O)c(Cl)c1 Cc1ccc(C#N)cc1C(N1CCC(NC(=O)CC(C)F)C12CC2)=O C1(CC(N2C(CN(C)C(c3ccc(-c4ccco4)[nH]3)=O)CCC2)=O)CCC(O)C1 N1(C(C23CCC(C)(OC2)C3)=O)CC2CCC(C1)N2C(c1c[nH]nc1C(C)(C)C)=O Cc1cc(C(=O)N(C)CC2CN(C(C3(C)CC(C#N)C3)=O)CCO2)ncc1F c1(SCC(=O)NC(CN(C(CC2(C=C)CC2)=O)C)C)nc2ccccc2o1 c1(C(C)Br)ccc(C(=O)Nc2n[nH]cc2NC(C2(O)CC2)=O)c(O)c1 CCC(C)(O)C(=O)N.c1(CN2CCN2C(=O)CCc2ccoc2)ccc(Cl)nc1 C(=O)(C1CC(=O)N(C)c2ccccc21)CC(c1coc2ccccc12)C(=O)OC C1(F)(CNC(C(C)n2ccnc2)=O)CCN(C(C2CCCO2)=O)CC1 Cn1cc(C(N2CC(CNC(c3ocnc3C3CC3)=O)C2)=O)c(=O)n(C)c1=O N1(C(C(CCC)N(C)C(C2CCCCN2CC)=O)=O)CCCC(C)(CN)CC1 c1(C(N2CCCC(CCNC(COC)=O)C2)=O)cc2c(s1)CCC(C)C2 C12(NC(c3cc(=NC)[nH]cc3)=O)CCC(CC1)N(C(=O)CCSCC(N)=O)C2 CCCC(C(=O)NCCc1ccc(C)cc1)NC(C1(C)CC(C)=NO1)=O C(=O)(CCN=C(NC(CC)C)N1CCN2C(=O)CCC2C1)Nc1ccc(F)cc1 N1(CC(CC)SC)C(=O)CN(CCC(N2CCN(c3cnccn3)CC2)=O)C1=O c1(C(=O)NCC2(F)CC(NC(c3ccc(CN(C)C)o3)=O)C2)cc(C#N)no1 c1(SCCC(=O)NCCNC(C(C)C2CCOC2)=O)nnnn1C1CC1 C(=O)(CC(CCCCC)SC)NC(CNC(CC=C=C)=O)(CC)CC c1(CCNC(C2(C)N(C(CCc3scc(C)c3)=O)CC2)=O)cccnc1F C1(C(=O)NCc2cc(CC3CC3)on2)CC2CC(C1)N(Cc1cnnc(O)c1)C2 c1(C(=O)NCC(C)NC(=O)C(C)(C)NS(C)(=O)=O)c(O)ncc2c1CCC2 N1(C(c2ccc(C)cn2)=O)CCC(NC(C2CCCCC2N(C)C)=O)CC(O)C1 c1(C(N(CCNC(C#CC(=O)OC)=O)C(C)C)=O)ccc(C)c2[nH]c(C)cc12 CC(C)C(C(=O)NCCNC(=O)C(N)=O)N.C1(C(=O)NC)CCN1C(=O)OC(C)(C)C c1(C(=O)NCC(C)N(C(c2ccco2)=O)CC)cc2c(cc1Cl)OCO2 CCN=c1[nH]cc(C(=O)NC(C2CCCC2)CNC(=O)CC(C)COCC)s1 c1(C(=O)NCC(C2CC2)Nc2cc(C(F)(F)F)ncn2)ccc(C2CC2)cn1 CC1=C(NC(=O)C(N2CC(C(=O)NC)OC(C)(C)C2)=O)c2ccccc2S1(=O)=O C(=O)(CCS(=O)(=O)Cc1ccccc1)NCC(CC)(CN1CCCC1)CC Cc1cccc(C(C)NC(C2CCC(C(C)C)N2C(c2nnsc2N)=O)=O)n1 C1(c2cn(Cc3cccnc3F)nn2)CCCN(C(C2(CC(C)C)COC2)=O)C1 CC(C(=O)NCCCNC(c1cc(C#N)ccc1F)=O)C(C)S(C)(=O)=O C1(CNC(C2C(OCC)CC2)=O)CN(C(C2CCC(C)(C)CC2)=O)CC1(C)C C1(C(C)CNC(c2ccn(CCF)n2)=O)CCN(C(c2cnn(C)n2)=O)CC1 c1(C(=O)NC2(CO)CCCN(C(C3CCCSC3)=O)C2)ccnc2ccnn12 N1(C(CS(=O)(=O)NCC)=O)CC2CCCC1C2CNC(=O)Cn1cc(Cl)cn1 c1(C(N2CCC2CNC(C23CC4CC2(CO)CC4C3)=O)=O)ccc2cnsc2c1 O(S(=O)(=O)c1ccc(F)cc1)C(c1c(C)nc(-c2ccc(Br)cc2)s1)=O CCS(C)(=O)=NC(=O)c1cc(Br)ccc1OC(F)(F)F N1(C(C(CC)CC)=O)CCCC(NC(=O)CC2CC(OC)C2)C(F)C1 C(=O)(CC1COc2ccccc21)N1CC=C(CNC(C2CC(C(=O)OC)C2)=O)CC1 C1(NC(C(c2ccccc2)OC)=O)CC(C)(NC(=O)C(C)OC(C)=O)C1 N1(C(C)C)CC(C)OC2(CCN(C(c3conc3Br)C(=O)NC3(C)CC3)C2)C1 CC1(CC(=O)NC2CCCN(C(c3cc(C4CC4)cs3)=O)C2)CCOCC1 S(=O)(=O)(c1cc(Cl)ccc1F)N1C(CNCc2ccc(C(=O)O)cc2)CC(F)C1 C1(NC(C2(C(=O)OCC)CC2)=O)C2CCC(C2)C1C(N1CCCC(C#N)C1)=O N1(C(C=C(C)CCCC)=O)CCCCC1CC(=O)NCCc1cn(C)cn1 C1(CNC(C2N(C)CCC2)=O)CCCC(CNC(c2ccncc2F)=O)C1 c1(C(N2CCC(c3ccc(Br)cc3)C2)C(=O)NC(C)(C)C)ccncc1Cl c1(CC)nn(C)c(C(=O)NC2CN(C(=O)CC3C(C)C3(F)F)CC2OC)c1Cl Cc1cccc(C(N2CC(NC(c3nnccc3C)=O)C(C)C2)=O)c1Br CC(F)(F)C(C)(C)C(=O)N1CCCC(F)(CNC(=O)CCc2cccs2)C1 c1(C(N2CCOCC(NC(C34CC(C)C3C4)=O)C2)=O)ccc(P(C)(C)=O)nc1 CC1(C)CN(C(c2cc3sccc3[nH]2)=O)CC1NC(c1ccc(NC=O)cc1)=O N1(C(c2c(Cl)cn(C)n2)=O)CCC2CN(C(C3CCCC3)=O)CC2C1 C(=O)(C(CC(C)C)NC(=O)CCCn1cc(-c2cncc(C)n2)nn1)OC c1(C(=O)NC2C(C)CN(C(=O)C(C)(C)CC#N)CC2)ccc2ccsc2c1 C12(NC(c3c(C)nc(C(C)C)s3)=O)CCN(C(=O)C=CCO)CCC1C2 C1(NC(C(CC)F)=O)CCCN(C(=O)CSc2nncn2C2CC2)C1C c1(CC(N2CC3C(NC(=O)CSC(F)(F)F)(CCC3)C2)=O)ccc2ccoc2c1 C(=O)(CCC(CC)NC(C1(OC)CCOC1)=O)NC(CC#CC)CC N1(C(c2c(C)ncc(N)c2)=O)CC2CC(NC(c3n[nH]cc3Cl)=O)CC2C1 C12(NC(c3c(C#N)nc[nH]3)=O)CCC(n3cc(CC4CCS(=O)(=O)N4)nn3)(CC1)C2 C1(CNC(C(C)(C)SC)=O)CCC2(CN(C(=O)C(F)OC(F)(F)F)C2)O1 CC1CC(NC(c2cnn(-c3ccccc3F)c2)=O)c2ncnn21 c1(C(N2CC(NC(CC(C=C)C)=O)C(C)C2)=O)cccc(O)c1Cl Cc1cc(C(F)F)nn1CC(N1CC(C)(NC(C2CC(C)(C)O2)=O)C1)=O C(=O)(CCC(C)(C)[N+](=O)[O-])NCC(C)CN(C)C(C1(C)CCN(C)C1=O)=O C1(C(=O)NC(CCNC(C=CSC)=O)C)CCN(C(=O)Nc2cccnc2)CC1 Cc1nc2cccnn2c1C(=O)NC1CC2CN(C(C34CCC(C3)OC4)=O)CC12 c1(CN2CCC(O)(C3(C)N=N3)C2)cc(S(=O)(=O)Nc2ccccc2)c[nH]1 N1(C(C(CC)CO)=O)CCC(CNC(=O)C(c2ccc(OC)cc2)O)C1(C)C C1(CNC(C=CCC)=O)CN(C(c2cc(-c3cccs3)on2)=O)C2CC12 C12(C(=O)NCC(CC=C)NC(=O)C3=CC(C)CC3)CCC(C(F)F)(CC1)C2 N1(C(c2cc(CC)n(C)n2)=O)CCCC12CCN(C(=O)Cc1sccc1Cl)C2 C1(C(N2CCC(CN(C(C3(CC#C)CCCCC3)=O)C)C2)=O)CCCCNC1=O Cc1cc(O)nc(CNC(=O)C(CC(C)C)NC(=O)C=C2CCC(C)CC2)n1 C12CN(CC1C)C(C)CCc1nc(cs1)C(=O)N2.c1(CSCC)cn(CSC)nn1 Cc1c(C(=O)N(C)CC2CCCN2C(C2CCC3(C2)N=N3)=O)cccc1[N+](=O)[O-] CCN=c1ccc(C(N2CCOCC(NC(C34CCC(O)(CC3)C4)=O)C2)=O)c[nH]1 CC(C(=O)Nc1ccc2c(Cl)nccc2n1)S(=O)(=O)C1CCOCC1 c1(C(N(C2CCC(NC(=O)C(C3(O)CCCC3)F)C2)C)=O)ccc2c(c1)CCC2 C12(NC(CP(C)(C)=O)=O)CCCCC1CN(C(=O)Cn1nnc(=O)[nH]1)C2 c1(OC)cccc(C(N2CC3C(CNC(=O)Cn4c(C)csc4=O)C3C2)=O)c1O c1(C(=O)NCC(=O)NC(CCSC)CO)ncc[nH]c1=O c1(C(=O)NC2C(NC(CC3(C=C)CC3)=O)CCC2)c(C)[nH]c2ncccc12 N1(C(CCSCCCC)=O)CCN(C(c2cc(C)n(C3CC3)c2C)=O)C2CCC12 CCCCCCC(C)C(=O)NCc1csc(C(=O)NCCCN2CCC2)c1 C1(C(N2CC3C(C(=O)NC4CCN(CCC)C4)(C3)C2)=O)CC12CCOCC2 c1cc(=NCCC2CCOC2)[nH]c(NC2CCSC2)n1 c1(C(N(CC(CN(C(=O)CC2CCCO2)C)O)C)=O)nnc(O)c2ccccc12 CC(C(C)C(=O)NCC1(O)CN(C(=O)CC2CCC(=O)N2)C1)S(C)(=O)=O C1(CNC(CC=C(C)C)=O)COCCN1C(C1CC2CC2C1)=O n1(CC)ccc2cc(NC(C3CC4(CC4)CN3Cc3cncnc3)=O)ccc12 CC1(NC(=O)CCCc2ncco2)CCN(C(=O)CC(=O)NCC(F)(F)F)C1 C1(C(=O)NC(C(C)C)(C)CNC(=O)COC(F)(F)F)CCC(C)(F)CC1 c1(CCC)ccc(C(=O)N(CCNC(=O)C=C=C(C)C)CC)cc1 c1(C(N2C3CN(Cc4nc(C)sc4C)CC32)=O)cccc([N+](=O)[O-])c1C CC(C)CC(C)C(=O)NCC(CO)NC(=O)CCc1cscc1Br CC(N=c1ccc(Br)c(S(=O)(=O)NC2CCCCC2F)[nH]1)C(C)F c1(N2CC(C(=O)OC)C(SC)C2)ncnc2cc(-c3nn[nH]n3)ccc12 c1(C(N2CCCCC(N(C(=O)CC3COCCO3)C)C2)=O)ccncc1N=[N+]=[N-] c1(SCc2ccc(CN(C)C(c3nnnn3C)=O)cc2)cccc2c1CCC2 Cc1csc(C)c1NC(=O)CC1COCCN1C(c1ccn(C)c1)=O CC(C)C(CNC(c1cc(O)n(C)n1)=O)C(=O)NCC1(C(N)=O)CCCC1 c1(C(C)C(N2CC(C3CN(C(c4cc[nH]n4)=O)C3)C2)=O)ccc2c(c1)C(C)(C)CO2 N1(C(C(CCCC=C)NC(=O)CCOC)=O)CCN2C(=O)NCC2C1 c1(C(=O)OC)cc2cc(n1)C(=O)N2.C(C)(C(C)SC)NC(=O)Cc1ccon1 c1(NC(C(C)(C)C)(CC)c2nnnn2C2COC2)cc(Br)c2c(c1)OCCCO2 Cc1ccc(C(=O)NC(C2CN(C(=O)Cn3ncn(C)c3=O)C2)C)c(O)c1C CCC(C#CC(=O)NCC(S(C)(=O)=O)C1CC1)NC(=O)OC(C)(C)C Cc1cc(Br)cc(S(=O)(=O)N2CCC3(CCN(Cc4c(C)nn(C)c4Cl)C3)C2)c1 N1(C(C(C)S(C)(=O)=O)=O)CCCC12CCN(C(C1CCCS1)=O)C2 Cc1cnc(C(N2CCN(C(=O)COC3CCC3)CC2CC2CC2)=O)cc1C C(c1ccc(C)c(C)c1)=CC(=O)NCC(CNC(c1cnc(C)s1)=O)C CC(C)CC(O)C(=O)N1CCCCC1C(C)(C)CNC(=O)CCCC1CC1 C1(NC(Cc2c(C)noc2Cl)=O)COC2CN(C(=O)C(C)CC3CCC3)CC12 N1(C(CN(C)C)=O)CCC(F)C(NC(c2cccc(CN3CCOCC3)c2)=O)C1 c1(C(N(C(CNC(c2c(C)ncn2C)=O)C)C)=O)c(F)ccc2[nH]ccc12 C1(CC(C(=O)NCCCSC)N(C(CC)C2CC2)C)CCCC(C)(C)C1 c1(OC)cc(CN2CCC3(CC3C(=O)Nc3c(O)cccc3Cl)C2)cc(Cl)c1 C=CCCCCCCC(=O)N(CCC(C)NC(=O)C(N1CCCC1CC)=O)C C1(NC(C2(COC)CC2)=O)CCN(C(c2cnc(C(C)=O)s2)=O)CCC1CO N1(CCC)CCN(C(c2cn(CCC)nn2)C(=O)NCc2ccc(F)cc2)CC1 CC(CCC(=O)NNC(=O)N(CC(F)C(=O)O)CC(F)(F)F)c1ccccc1 N1(C(CCN(CC)CC)=O)CC2CC1(C(=O)NC(CN1CCCC1)CO)C2 N1(C(C(CC)OCC)=O)CCN(C(=O)CCCC(N)=O)CC12CCC2 n1(CCC2CN(NC(C3CCCCO3)=O)C2)cc(CCC2CCCO2)nn1 c1(C(=O)NC2CN(C(CCCC)=O)CC2c2cnn(C)c2)ccc(OCC)cc1Cl c1(C(N2C(C(N(CC)Cc3ccc(Br)cc3)=O)CSCC2)=O)cc(C#N)ccn1 c1(C(=O)NCC(CN(C(C2N(C(C)=O)CCC2)=O)C)O)nnccc1Br CC(C)CC(C)CC(=O)NCCC(C)NC(c1nc2n(c1Br)CCC2)=O c1(C(=O)NC2CCCN(Cc3cccc(-c4cc[nH]n4)c3)C2)cc2sccc2[nH]1 c1(CC)nccn1C(C)CC(=O)NC(C)(C)C(C)NC(C1CC(OC(C)C)C1)=O C(N=c1cc(C(=O)OC)nc(CC)[nH]1)C1CC(NC(c2n(CC)ncc2Cl)=O)C1 C12CCN(CC1(F)F)C2=O.c1(C(=O)Nc2ccno2)nc(C(F)(F)F)no1 c1(C(N2CCC(C(C)CNC(=O)CCNS(C)(=O)=O)CC2)=O)cc([N+](=O)[O-])n[nH]1 Cc1cc(NC(C2(C(C)NC(=O)CCc3cnn[nH]3)CC2)=O)cnc1C c1(N2C(C)C(NC(=O)C(F)(F)C(O)C3CC3)C(C)CC2)ncc([N+](=O)[O-])cc1Br N1(C(c2ccc(C)c(O)n2)=O)CC(NC(c2nccnc2N)=O)C2CCCC2C1 CCCCC(O)CC(=O)NCCOCC(=O)NCC1(CO)CC(C)(C)C1 N1(C(C(C2CCN(C(c3cc(C)nc(C)c3)=O)C2)C)=O)CC(F)(F)CCC1C C(=O)(CCCC(=O)NCC(CC)(CC)NC(c1n[nH]cc1C)=O)OCC N1(C(C(C)Cn2ccnc2)=O)CC2CCCC2C1C(=O)NCC1(CN(C)C)CC1 CCC(C)(C)C(O)C(=O)NCC1(C(=O)NCCCC(C)(C)CO)CC2(CC2)C1 C(=O)(CCCC(F)(F)CO)NCC1CC(C)(CNC(=O)CN2CC3CCC2C3)C1 c1(N(CCNCC(O)Cc2cnn(C)c2)CC)ccc(COC)cc1[N+](=O)[O-] c1(OC)coc(C(N2CC(F)(CNC(C3CC(C(F)F)C3)=O)C2)=O)cc1=O c1(C(=O)NC2(C)CCCN(C(C3(F)C(C)C3)=O)C2)c(Cl)ccc(Cl)c1Cl c1(N2CCn3c(C(C)C)cnc3C2)nc(=NC2CCOC2)[nH]c2c1SCC2 CC1=NOC(C(=O)NCC2COCC2NC(=O)C(c2cscc2Br)=O)C1 C(=O)(C(C)(C)CC(F)(F)F)NCC(CN(C(C(c1c(C)ccnc1)(C)C)=O)C)C CC1OC2(C(=O)NCCn3cc(CCC(c4ccc(F)cc4)O)nn3)CC1(N)C2 Cc1cc2c(C(=O)NC3CC(NC(=O)C=Cc4scnc4C)C3)nccn2n1 c12cccc(c1Cl)OC2.c1(CC=C(C)C)ccc(NC(=O)OC(C)(C)C)cc1 c1(NCC(c2cc(OC)ns2)N2CCCC2)nccc(=NCC2CCCCC2(F)F)[nH]1 C#CC1CCCC(CNC(=O)C(C)(C)CNC(=O)C=Cc2ccc[nH]2)C1 n1(CCC(=O)NC2CN(C(C3(C)CCOC3)=O)C2)cc[nH]c(=O)c1=O c1(N2CCCC(NC(CC(C(C)C)O)=O)C2C)nc2cc(Br)cnc2s1 CC1(C)CC(NC(=O)NC2CC(=O)CC2C(=O)O)CCN1 c1(CC(C(=O)NCC2N(CC)CC2)NC(c2cnc(Cl)s2)=O)cnn(C)c1O N1(C(c2c(C)oc(C)c2C)=O)CCN(C(c2cc(C#N)oc2C)=O)CC12CCC2 c1(C(=O)NCC(C)N(C)C(c2ccc(C#N)cc2F)=O)cc2ccccc2s1 O=S(=O)(c1ccc(NC2CC=CCC2)cc1Cl)NCC(F)Cl CN1CC=C(CC(=O)NCC(C(C)(C)C)NC(c2ccc(CO)nc2)=O)CC1 C(=O)(C(C)(C)C(=O)N1CCC(C(=O)NC2CCCCC2C(C)C)CC1)OCC C(c1cccc([N+](=O)[O-])c1)=CC(=O)NCC(CNC(c1c(C)nn(C)c1C)=O)F C1(NC(CCCCSC)=O)C2CCCC1CC(NC(c1nnsc1C)=O)C2 C1(NCCCC(=O)N2CCCCC2)C2CN(c3ncccn3)CC12 N1(C(C2(CSC)CC2(F)F)=O)CC(NC(=O)CCC(N)=O)CC(C)C1 C1(CCNC(c2cnncc2O)=O)CCCN(C(C23CCCC(CO2)C3)=O)CC1 C1(NC(C2Cc3nnsc3S2)=O)CCCN(C(C2CCC(F)CC2)=O)CC1 CC(Cc1cnn(C)c1)C(=O)NC1C=CC(CNC(c2coc(CC3CC3)n2)=O)C1 O=C(C#CC1CCC1)NC1CC(F)(CNC(c2n[nH]c(C3CC3)c2Cl)=O)C1 c1(NC2C3CCN(c4ncnc(COC)c4F)C3(CO)C2)ccc2nncn2c1 N1(C(CC2(C)CCC2)=O)CCN(C2CCCC2NC(=O)COCCCF)CC1 N1(C(CC2(OC)CCC2)=O)CCCN(C(c2cc(F)c(O)c(F)c2)=O)C(C)C1 c1(CC(=O)NC2(CNC(C3(C=C)CC3)=O)CCOC2)cncc(Br)c1 N1(C(C2CCCN(Cc3ccncc3)CC2)=O)CCC(N2CCC2)(C(=O)O)CC1 c1(C(N2CC(F)CC(NC(C3(C)CC(=C)C3)=O)C2)=O)cccc2nonc12 c1(C(=O)NCC2C(NC(=O)Cc3cncs3)C2)ccc(Cl)c(Cl)c1 c1(NCCNC(C2CCCN(C(C3C(=C)C3)=O)C2)=O)ncnc2c1CCC2 c1(C(N(C)CC2COCCN2C(=O)CC(C)F)=O)cc(F)c(N)cc1F CC(O)(C(=O)N1CCCC1Cc1cn(Cc2ccc(Br)s2)nn1)C1CCCO1 C=CC1(CC(N2CC(N(C)CC)C2)=O)CN(C(C2CC(CC)=NO2)=O)C1 c1(C(=O)NCCN(C(CCN(CCC)CCC)=O)CCC)cc(C)c(Cl)cn1 Cc1cc(CN(C(=O)C=CC(C)NC(C2(C)CC3CC3C2)=O)C)nn1C C1(CNC(c2[nH]cc(CC)n2)=O)CCC(F)(CNC(=O)CCC2CCOC2)C1 C12(CN(CC(C3CCC3)OC)Cc3cccc(Br)c3)COC(C(F)(F)F)(C1)C2 C1(NC(CC(C)n2cccc2)=O)CN(C(C2(C#N)CCCC2)=O)CCC1CO Cc1ccc(F)c(C(N2CC(CNC(=O)C=Cc3cccnc3)C(F)(F)C2)=O)n1 c1(OC)cc(C)ccc1C(N1CC(NC(=O)CCCCn2ccnn2)C2CC12)=O C1(NC(c2nc(C(C)OC)oc2)=O)CC2CCC(C1)N2C(c1cnccc1C)=O N1(CCNC(=O)Cc2n[nH]cc2Br)CCN(C(=O)C(N2CCCC2)C2CC2)CC1 c1(CC(=O)NCCC2CN(C(c3occ4c3CCC4)=O)C2)cn2c(n1)CCCC2 c1(C(N2CC(NC(c3c(SC)ccs3)=O)C(C)C2)=O)ccc(F)c(C)c1F N1(C(C2C(OC(C)(C)C)C2)=O)CCC(C(O)CNC(C2CCOC2)=O)CC1 c1(CNC(c2cc(O)cs2)=O)cc(C(N2CC(CF)C2)=O)no1 C1(C(N2CCC(CC#C)C2)=O)CN(C(C2COCC(C)O2)=O)CC1CC c1(C(N)=O)cc(C(=O)NC2CCN(C(=O)C3=COCCC3)C23CC3)ccc1O c1(C(N2CC(CCNC(=O)CSc3ccccc3Cl)C2)=O)csc([N+](=O)[O-])c1 C1(N(C(CCC2(C)CC2)=O)CCO)CCN(C(=O)CC2C=CCCC2)CC1 c1(C(C(=O)NC2CCCC(CNC(COC)=O)C2)=O)ccc(F)c(F)c1F N1(C(c2cccc(C(F)F)c2)=O)CC(C2CN(C(c3cc4[nH]ccc4s3)=O)C2)C1 c1(N2CC3C(NC(CC(CC)O)=O)C3C2)ncnc2cccc(C)c12 Cc1ccncc1C(=O)NCc1nnn(C)c1C(=O)NCc1ncccc1Cl Cc1cc(=O)c(C(N2CCCC(CCC(N3CC(O)C(C)(C)C3)=O)C2)=O)c[nH]1 C1(NC(C=CCOCCOC)=O)CCOC(C(=O)NC2(CCCF)CC2)C1 c1(C(N2CCCC(NC(=O)CN3CC4C=CC3C4)C2)=O)ccc2c(c1)NCC2 C(=O)(C(O)C(F)(F)F)NCc1cccc(C(=O)NC(C#C)(C)C)c1 c1(CC(=O)NCC(CN(C)C(c2cc(O)ccc2N)=O)O)ccc(F)c(F)c1 CN1CCOC(C(=O)NC2CC3(C2)CC3NC(C2CN(S(N)(=O)=O)C2)=O)C1=O C1(C)(C(=O)NC)CCN(C(=O)C=CCNC(=O)COCCSC)C1 Cc1ccc(F)cc1C(N1CCC1(C)CC(=O)NCC1(C2CC2)CCCO1)=O C1(CNC(CSCCCC)=O)CCN(c2ccc(C(F)(F)F)cn2)CC1C N1(C(c2ccc(OC)cn2)=O)CCCC12CCN(C(=O)C(F)CC(C)C)C2 C1(C(N(CC#CC)CC#C)=O)(CC)CCCN1C(=O)Cc1ccsc1C C12(C(=O)NCCCCN(C)C(C3CC3F)=O)CC(F)(C1)C2 Cc1cc(C(=O)N(CCC(=O)NC2CCCC(C)CC2)CC2CC2)nnc1O N1(CC(C)C(=O)NCC2(NC(c3cnccn3)=O)CC2)CCOCC(CO)C1 C12CCCCC1C(=O)N(C(C)(CO)C1CCC1)C2=O.C1(CC)COC(C)C1 C=CCC(C)(CC)C(=O)NCCC(CNC(=O)CCc1ccccn1)OC CCN=C(NCCF)NC1CC(OC)C(c2ccc(OC(C)(C)C)nc2)C1 C=CCC(C)(C)C(=O)NCC1(COC)CCCN1C(C1CCCS1(=O)=O)=O CC(C)(F)CCC(=O)NC(CNC(c1cccc(-c2cccnc2)n1)=O)CO c1(CNC(=O)NC(c2ccc(OC)cc2)C(C)C)nnc2c(C#N)cccn12 c1(OC)cc(I)ccc1Nc1nc(C(C)(C)C2CC2)cs1 N1(C(c2c(N(C3CCC3)C(C3CC=CC3)=O)n[nH]c2)=O)CC(O)(C2CC2)C1 CCN=C(NCC1CCC1C)N1CCN(c2ncnc(N(C)C)c2C)CC1 c1(C(C)OC)nc(C)c(C(=O)NC(CNC(c2cc(O)ncn2)=O)C(C)C)s1 c1(C(N(CCN(C)CCNC(C2CCOC2C(C)(C)C)=O)C)C2CC2)ccccc1 C(=O)(CCCCCOC)N1CC(CCC)C(C(=O)NCC(C)CC(F)(F)F)C1 N1(C(CN(C(C2C=CCCC2)=O)CC)=O)CCC(C)(C)C1C CCC(CC(=O)NCCOCCNC(=O)C(F)CC1CCC1)OC c1(NC(C)C(=O)NC2CC(N(C(=O)CNC(C3CCSC3)=O)C)C2)cccnc1 C1(N(C(c2c(C)noc2N)=O)C(C)C)CCSC2(C1)CC(C(N1CCCC1)=O)C2 N1(C(=O)COC(F)F)CC2CN(C(c3cnn(C4CCCC4)c3)=O)CC2C1 c1(N2CC(NC(c3cc(C)no3)=O)C(C#N)C2)cc2ncnn2cn1 C(=O)(CCC(=O)N(C)C)NC1C(CNC(c2c(COC)ccs2)=O)CC1 C1(C(=O)NCC(CCOC)(C)O)N(C(=O)Cn2nnc(C)n2)CCCC1(C)C C(C(C(=O)NOCC(F)F)NC(C1Cc2nccn2C1)=O)SCC c1(C(N2CC3(C2)CC(=O)N3)=O)ccc(F)c(F)c1.C(C)(C(=O)OC)SCCC C1(C(=O)NC(C#C)CC(C)C)CCCN(C(=O)C(=O)NC2CC2)C1C C1(N(CC)CC)CCN(C(C2CC(C)CO2)=O)CC1.CCC(CC)N(CCC(=O)N)C c1(CC(=O)NC2C=CCN2C(=O)C#CC2CCCO2)cccc2sccc12 C12(C(=O)NCc3n(CC)nc(C)c3)CCC(CC1NC(C1CCC(O)C1)=O)C2 N1(CC#C)CCCN(C(=O)C(=O)NCC)CC1.c1cc(N)ccc1CC c1(OC)ccc(C(=O)NOCc2cn(C3CC4(CCCC4)C3)nn2)c(Cl)c1OC c1(C(=O)NCC2(CC)N(C(CCOCC)=O)CCC2)cc(OC)cc2c1CCC2 c1(C(N2CCN(Cc3ccc(C)c(C)c3)C(C)C2)=O)ccc2ncoc2c1 CCCC(C(=O)OC)NC(C1CN(C(=O)C(C)(C)CC)CC1CO)=O C1(O)(CNC(C2CC(C)N2C(=O)CC2(O)CCC2)=O)CC2CCC1C2 c1(C(=O)NCC(CCNC(CSC(C)(C)C)=O)(C)C)nccc(N)c1Cl Cc1nn(CC(F)(F)F)c(C)c1C(=O)Nc1ccc[n+]([O-])c1 N1(C(CCc2c(C)ncs2)=O)CC=CC(C(=O)NCC2CCC3(CC3)C2)C1 C1(C(=O)NCC(C(=O)NCC)(C)C)CCCN(C(C2CCCC(=O)N2C)=O)CC1 c1(N)ncnc2cccc(Br)c12.C12CCCN1N(CC)C2.C1(C=O)(OC)CCC1 c1(C(N(C(CNC(c2[nH]c3cc(C)oc3c2)=O)C)C)=O)ccc2oc(O)nc2n1 c1(C(N2CC(N(C(CC(CCC)C)=O)C)C(O)C2)=O)cc(OC)ccc1[N+](=O)[O-] C(=O)(C(O)CNS(C)(=O)=O)NC1C(=O)C1CCNCCN(C(CC)C)C c1(OC(CN(CC(C)(C)C)C(C)=O)=O)ccn2nnnc2c1.C12CCN(C1)C2=O c1(C(N(CC(C)CNC(=O)CCC2(C)CC2(F)F)C)=O)cc2c(s1)CCC(C)C2 n1(CC(=O)NC2C(NC(C(N)=O)=O)CC2)cc(Br)c(C2CC2)n1 CC(C)C(C(=O)NCC(C)(C)NC(=O)Cn1ncccc1=O)c1ccn(C)n1 C(=O)(C(O)CC[S+](C)C)N1CC(CNC(c2cc(CC)ncc2)=O)OCC1 Cc1cc(C(=O)N(C2CCN(C(C3CC3C)=O)CC2)C)c(C)nc1C Nc1ncc(C(=O)NC2C=CCN(C(c3ccc(F)c(Cl)c3)=O)C2)cc1CO N1(C(C(C(C)C)OCC)=O)CCC2(CCN(C(C3CCCSC3C)=O)C2)C1 C1(C(=O)NC(CCC)CO)(CF)CCN(C(=O)C(Cl)Cl)C1 c1(CNC(c2c(NC(C(C(C)C)NC(C)(C)C)=O)c[nH]n2)=O)cc(Br)ncc1Br N1(C(CCc2cccc(OC)n2)=O)CCN(C(n2nc(C)ccc2=O)=O)C2CC12 C12(NC(CC3C=CC(NC(c4n(COC)ncc4)=O)C3)=O)CC1COC2(C)C n1(CCCCC(=O)N(CCN(C(C(C)SCC)=O)C)C)cnc2c(N)ncnc12 C1(NC(C(CN(CC)CC)F)=O)C(C)(C)C(NC(=O)CN(C)C(C)=O)C1(C)C N1(C(C(C)NC(=O)NC)=O)CCC(O)(C(C)NC(c2cnn(C)c2OC)=O)C1 c1(C(=O)NC(CC)CNC(=O)CSc2ccc(F)cc2F)c(C)cc(C)oc1=O Cc1ncc(CCCOc2cc(F)n[nH]2)cn1.N12CCC(CC1)C2=O c1(C(=O)NCC2N(C(C(CCC)OC)=O)CCC2)c(C)c(C)nc2ccccc12 Cc1ncc(NC(c2nc(CNC(C3CCCC(C#N)C3)=O)oc2C)=O)cc1Cl N1(C(C2(C)CCCN2Cc2ccc3c(c2)CCO3)=O)CCCC2(CCNC2=O)C1 N1(C(C(CO)OC)=O)CCC(O)(CNC(=O)C(c2ccccc2)c2ccn(C)n2)C1 N1(C(c2[nH]c(=NC)sc2)=O)CC2CCCC1(CNC(c1c(SC)cnn1C)=O)C2 N1(C(c2c(C)n[nH]c2)=O)CCN(C(c2cnc3ccoc3c2)=O)C(C)C1C Cc1ccc(C(=O)NC(C)CNC(=O)Cc2ccccc2O)c(C)n1 c1(CC)nc(O)c(C(N2CC(NC(c3cnnn3C)=O)CC2C)=O)cc1C c1(C(N2CC(N(C)C(C3CCCC(C(N)=O)C3)=O)C2)=O)n[nH]c2ccccc12 N1(C(CC(C)(C)N(C(C(C(C)C)SC)=O)C)=O)CCSC2CCCC12 CN1CC(C(=O)N(C2CC(NC(=O)C3CC3)C2)C)C(c2ccccc2)C1 C=CC(O)C(=O)N(C)CCOCCNC(c1coc(C(F)(F)F)n1)=O CC1CCC=C1C(=O)N1CCC1(C)CC(=O)N(CCN1CC=CC1)CCO C12(CNC(c3cnn(C4CCC4)n3)=O)CCC1CCN2C(C1CC(O)C1)=O N1(C(CCCCN(C(C)C)C)=O)CCCCC(CNC(=O)C=CC2CCCC2)C1 c1(CNC2C(C)N(C)CC2)cc(Cl)c2c(c1)OCCO2 c1(C(C)C(=O)NC2COCC2NC(C2CC(=C3CC3)C2)=O)ccccc1F Cc1c(Cl)cnn1CC(=O)NCC(C)(O)CNC(=O)Cc1cccc(F)c1 C=CCN=c1[nH]c(C(N2CCCC2CNC(=O)CCC(C)C)=O)cs1 N1(C(CSCC#C)=O)CCN(C(=O)C(C)n2ccnc2)C(C2CCCC2)C1 N1(C(CC(C(C)C)NC(CC)=O)=O)CCN(C(=O)OC(C)(C)C)C2CCC12 C12(C(N3C(C)CCC(NC(=O)C=CC4CCC4)C3)=O)CC3CC(C(=O)N1)C2C3 C(c1ccccc1[N+](=O)[O-])=C(C)C(=O)NCC1CC1NC(=O)Cc1cn(C)nc1C Cc1cc(O)nc(N2CCN(C(c3ccc(C)c(C)c3)=O)CC2)n1 C1(C(=O)N(C)Cc2ncccn2)(COC)CN(C(=O)CC2CCC(C)C2)C1 C(=O)(C1=CC2CC(C1)CC2O)NC(CC)(C)CNC(c1cc(C(N)=O)[nH]n1)=O N1(C(Cc2c(C)nc(S)s2)=O)C2CCC1CN(C(C1CCC(F)(F)CC1)=O)C2 C1(C(N2CCC(C)(F)CC2)=O)CN(C(=O)C(O)CC(N)=O)CC12CCC2 N1(C(C2N(C(c3c(CC)nns3)=O)CC(F)(F)C2)=O)CC2C=CCC(C2)C1 C(=O)(C1=CCS(=O)(=O)C1)NCC1C=CC(CNC(CC(C)c2ccccc2)=O)C1 C1(CNCc2n(CC(F)F)ccn2)CCCN(CC2(c3ccc(Cl)cc3)CC2)C1 c1(C(=O)NC2(C)CC(NC(C(C(CC)O)(F)F)=O)C2)cc2ccc(Cl)cc2[nH]1 c1(NC2CCCN(C(c3cc(C)c(Br)c(C)c3)=O)C2)ncc2c(Cl)cccc2n1 c1(C(=O)NC2CN(C(COCCCOC)=O)CC2C)cccc(C)c1F c1(C(N2CCC(N(CCC)C(C3CC3C)=O)CC2)=O)cc2c(F)ccc(F)c2[nH]1 N1(C(C(CCNC(Cc2nc(C)oc2)=O)O)=O)CC(C)OCC1C c1(CN(C(c2cc(Br)nn2C)=O)CC)ncc(Cl)n1C C#CCC(C)(C)C(=O)NC1CCN(C(=O)CCCc2ccc(SC)cc2)CC1F N1(C(c2c(C)cccc2C)=O)CCC2CN(C(C3C4CC5C(C4)C35)=O)C2C1 C(=O)(C(C)(C)CSC)N(CC(CC)(C)NC(c1cnn(C(F)F)c1)=O)C N1(C(C(C)=CC2CC2)=O)CCCCC(CNC(C2CCN(CC(C)C)CC2)=O)C1 Cc1ccccc1C1(C(=O)NC2CCC(NC(=O)CC3CCOC3=O)CC2)CC1 N1(C(C2N(C)CCCCC2)=O)CC(NC(c2cnn(C)c2)=O)C2(CCC2)C1 C#Cc1ccc(C(=O)NC2CC(C)N(C(=O)C=Cc3ccn(C)c3)C2)cc1C N1(C(CC2C=CC(NC(c3cnc(C)nc3)=O)C2)=O)CCC(F)C(O)C1 c1(C(=O)NC(C)CC2CN(C(C3CC3C)=O)C2)ncc(Br)cn1 C1(CN2CC(C)(CCC(N3CCCOCC3)=O)C2)CC2CC1CC2O C1(CC=C)(NC(C2C3CNC(=O)C23)=O)CCN(C(C2C=C(C)CS2)=O)CC1 C12(C(N3CC(CNC(c4ccn(CC(F)F)n4)=O)C3)=O)CC3CC(CC(C3)C1)C2 CC(=O)C(C)CC(C)C(=O)NC1(C(=O)N(CC(O)C(F)(F)F)C)CC(C)C1 C1(C(=O)NC(C(C)OC)C(=O)N2CC(C(N)=O)C2)CCC2(CCC2)O1 C1(NC(c2cccc(C)c2I)=O)CCN(C(=O)C(O)C(C)C)CC1(C)C C#CC1(C(N2CC=C(CO)C2)=O)CN(C(C2CCC(=O)N2)=O)C1 N1(C(C=CCC)=O)CCC(C(N2CC(C(N)=O)(N(C)C)C2)=O)C12CC2 C12(CNC(=O)NCCOCC3CCC=CO3)CC(C1)C(C(F)(F)F)O2 C1(CC(N2CCN(C)C(CNC(=O)C3=NOCC3)C2)=O)CCn2cncc2C1 C1(C)(C(=O)NC(C2(CNC(=O)CCc3ncc(F)cn3)CC2)C)CCCOC1 N1(CC(N)=O)CCN(C(=O)CN(C(C2CC(=O)CC(=O)C2)=O)C2CC2)CC1=O C1(NC(C(C)c2cccs2)=O)CC(F)CN(C(c2nc(F)ccc2Cl)=O)C1 C1(Cl)(C(N2CC3C(CN(C(C(CCOC)OC)=O)C)C3C2)=O)CC2CCC1O2 C(=O)(C=CS(F)(F)(F)(F)F)N(C1CCN(C(c2cccs2)=O)CC1)CCC Cn1c(C(N2CC3CC3(NC(c3coc(CS(C)(=O)=O)n3)=O)C2)=O)nnc1S C1(C(=O)NC2(C(=O)OCC)CCCCC2)CC12CCN(Cc1cnc(Br)s1)CC2 c1(C(=O)NC(C(C)(C)C)CNC(c2ccoc2C(F)(F)F)=O)cc(O)cc(=O)o1 C=CC(C)(C)C(=O)N1CC(NC(c2ccnn2C(C)CC)=O)C(C)C1 c1(C(N2C(C)CC(CNC(CSC)=O)C2)=O)cc(S(=O)(=O)N2CCCC2)c[nH]1 Cc1nc2c(C(N3CCC(NC(c4cnccc4C)=O)C34CC4)=O)cccc2o1 N1(C(CCC(C)OC)=O)CCCC(C2(NC(c3ccc(C)nn3)=O)CC2)C1 c1(-c2ncccc2CNC(c2ccc([N+](=O)[O-])cc2)=O)ccc(F)c([N+](=O)[O-])c1 N1(C(CC2CN(C)C2)=O)CCC2CN(C(c3cncc4c3CCC4)=O)CC2C1 C(c1cccc(F)c1)=C(C(=O)NC1CCC(NC(c2n(CCC)ncc2)=O)C1)F N1(C(C(CC)SC)=O)CC2CCC(C(N3CC(OCCNC(C)=O)C3)=O)(C2)C1 C1(NC(c2n(C(C)C)ncc2)=O)CCCN(C(=O)Cc2ccns2)C1 c1(CN2CC(CNC(CC(CC)O)=O)C2)c[nH]c2cc(C)ccc12 n1(C(CC)C)nnnc1C(c1cc(C(F)F)on1)NCC(=O)OCC1CC1 C12(C(=O)NC3CC4C(NC(C(C)CS(C)(=O)=O)=O)C4C3)CCCC1CC(=O)CC2 C(CCCN=c1[nH]cc([N+](=O)[O-])cc1CO)NC(c1c(CC)c[nH]c1)=O N(C(=NCC=CCl)NCC(N1CCN(C)CC1)(C)C)C(Cc1c(OC)cccc1)SC N1(C(c2c(OC)cc(C)s2)=O)CCN(C(C2CC23CCSCC3)=O)CC2(CC2)C1 c1(CCC(N2CCC(C)(N(C)C(C3COCC3C(N)=O)=O)C2)=O)ccc(O)nn1 c1(SCC(N2CC(C=C)C(NC(C3(O)CCC3)=O)C2)=O)ccc([N+](=O)[O-])cc1 c1(C(C(=O)NC(CC)C2CC2)NC2CCCO2)nc(C)ccc1Br.N12CCC(C1)C2 c1(C(=O)NC2C3(CC(NC(c4scc(C)c4)=O)C3)C2)cc(F)cc(Br)c1 C1(C(N(C)Cc2cscn2)=O)C(NC(c2ccnnc2)=O)C1(C)C N1(c2[nH]c(N3CCN(CC4CCC4)CC3)nc(=N)n2)CCN2C(=O)NCCC2C1 c1(NC(CCCC2(NCc3occ(C)c3)CCC2)=O)cn(C)nc1C C1(C(=O)NC(C(C2CCC2)OCC)=O)CCc2nc(C(F)(F)F)cn2C1 N1(C(c2c(C)noc2N)=O)CCC(C)C(NC(=O)CC2CC2C(F)(F)F)C1 c1(CNS(CC2(CC(=O)O)CCC2)(=O)=O)csc2cc(Cl)ccc12 N1(CC(=O)NCC2CN(C(=O)Cc3ccccc3)C2)CCC(F)CC1 CCC(CC(=O)NC(C)CCNC(=O)COCc1cc(C)no1)C1CCC1 C=CC1(O)CCN(C(C2C3CC4C(C3NC(c3ccon3)=O)C24)=O)C1 c1(C(C)C)nnc(C(=O)NCCOCCCN(C)C(C2CC(O)C2)=O)s1 C1(NC(c2cccnc2)=O)CCN(C(c2c(Br)ccnc2F)=O)CC1F c1(C(=O)NCCCCC(C)NC(CC2CC(CC)C2)=O)cc2nc(C)ccc2o1 N1(CC)CCC(N(c2cnn(-c3cccc(Cl)c3)c2C)c2ccccn2)C(O)C1 c1(COC(C(=O)N(C(CN(C(COCCC=C)=O)C)C)C)C)ccccc1Cl N1(C(C=CCCC)=O)CCCC(C2CN(C(=O)CCCCCN(C)C)C2)C1 c1(C(N2CCC(F)(CNC(=O)C=CCF)C2)=O)cc(F)c(C2CC2)cc1F CCCCC(C(=O)N1CCC(C(C)(C)NC(=O)C(=Cc2c[nH]cn2)F)C1)N(C)C CC1COCCN1C(C)CNC(c1ccsc1C(=O)OC)=O Cn1cnc2nc(=NC3CC(C)(C)C3)[nH]c(NCCC3CC4CCC3C4)c12 c1(C(N(CC(C)NC(c2c(NC(=O)NCC)scn2)=O)C)=O)cc(O)cc(O)c1 c1(C(=O)NCC2C3N(C(CSSC)=O)CC(CC3)C2)ccc(F)c2ccsc12 C(CC1=CCCCCC1)NC(C1=CCN(C(C(C)OC(C)(C)C)=O)C1)=O CC1(CNC(C2CC2F)=O)CN(C(c2c[nH]nc2-c2cccs2)=O)CCO1 c1(C(=O)NCC(CCOC)NC(c2ccc(Cl)o2)=O)cc(C2CCC2)n(C)c1C N1(C(C2(N(C(c3cc(Cl)no3)=O)C3CC3)CCC2)=O)CCC(NC(C)=O)C1 c1(C(=O)NCCCCC2CN(C(C3(CCCC)CCCC3)=O)C2)cnncc1C Cc1cc(C(N2CCC(CNC(C3OCCC3c3cnn(C)c3)=O)C2)=O)c(C)s1 n1(CC)ncc(C(=O)NC2CCN(C(C3CC3(C)C(F)F)=O)C2(C)C)c1[N+](=O)[O-] N1(C(C(C)NC(CC)=O)=O)CCC(C)(NC(C2CC2(C)C)=O)C1 N(C1CCSc2ccc(Cl)cc21)C(N1CCCC(Oc2cccc(Br)c2)CC1)=O c1(CC)ccc(C)cc1OC.C1(N2N(CCCN(C)C)C2=O)CCN2CCCC1C2 Cc1cc(C(=O)NC(C)C(=O)NC(C)C(=O)NCC2CC2)ns1 N1(C(C(CNC(C(C)OCCC=C)=O)OC)=O)CCC2(CC2)C1 CS(=O)(=O)c1cc(C(=O)NC2CCC(NCc3cc(Br)c[nH]3)C2)ccc1F C1(COC)(NC(c2ccc(C(N)=O)o2)=O)CCN(c2nc(Cl)c(C#N)s2)CC1 Cc1c(C(=O)NCC2C(C)CCN2C(c2ccc(F)cc2F)=O)nn(C)c1Br N1(C(C=Cc2c(C)ncs2)=O)CCCC(C2CC2NC(C2(O)CCOCC2)=O)C1 C1(C)(C(N(C)CC2N(C(C=CC(CC)C)=O)CC(F)C2)=O)COC(=O)OC1 C=CCC(C)(C)CCNC(c1ncoc1C1CC1)c1nnnn1CC1CCOC1 c1(C(N2CC(NC(CCC=C(C)C)=O)C(C)C2)=O)cccc(Br)c1F c1(NC(C(C(CC)C)OC)=O)c(C)nc2ncnn2c1C N1(CC(=O)OCCCC)CCC2(CC1)CCN(C)C2=O c1(CN2CC3C(C(=O)NCCCCCO)C3C2)cc(O)c(Br)c(O)c1 C1(C(=O)NCC(C)C)CC2(C1)CN(C(c1cnc(C(C)(C)C)o1)=O)C2 CC1C(CC(=O)NCC(C2CCCC2)SC)C1(F)F.C1(OCC=O)CCCCC1 N1(CCC(=O)NCC2C(N(C)C(C3C=CC=CC=C3)=O)C2)Cc2ccccc2C1 N1(C(C2(C)CC3C=CC2C3)=O)CCCC(C2CN(C(c3cnsc3)=O)C2)C1 c1(SCC(F)(F)F)nnnn1CC(=O)NCCCC(C)NC(C1OCCCO1)=O C1(CCOC)CN(C(C2(F)CCC2)=O)CCN1C(=O)CCc1ccc(C)nc1 Cn1cc2c(n1)CCC(C(N1CC(C#N)(CNC(=O)OC(C)(C)C)C1)=O)C2 C1(CCCC)CN(C(c2ccnn2C)=O)CCN1C(C1CCS(=O)(=O)N1)=O C(=O)(C(C)C1CCC1)N(C1(CNC(C2(C)CC2C)=O)CC1)C N1(C(CNC(C)=O)=O)CCN(C(=O)CC(C)(C)c2ccccc2)CC2CCCCC12 CC1=CCC(C(=O)N(CCCCCCNC(c2ncc(C(F)(F)F)s2)=O)C)CC1 c1(-n2cc(CCC(=O)NCCNC3CCCCC3)nn2)ncccc1Br C1(CNC(CCC(=C)Cl)=O)CCCC2CN(C(C3(C)CCCC3C)=O)CC12 CCC(CC)C(C)C(=O)N(c1cc(Br)c(C2CC2)s1)CCc1nn[nH]n1.CO N1(C(c2nnc(C)s2)=O)CC2(CNC(=O)Cc3cccc(Cl)n3)CCC1CC2 C(=O)(C1=CC2(CCOC2)C1)NCCC(CC)(CC)NC(C(CCCC#C)C)=O C(=O)(CCC(C)(C)N(C)C)N(CCCNC(Cc1c(C)ocn1)=O)C Cc1c(C(N2CC(CC(C)NC(C3CCOC(C)C3)=O)C2)=O)ccn1CC1CC1 N1(C(CCC)=O)CC(NC(c2cn3c(C)cccc3n2)=O)CC12CCCCC2 C(=O)(CCCC(=O)NC1CC(C)(NC(=O)CC2CCC2C)C1)OCC Cc1cnc(C(N2CCC(C)(CC(N3CC(O)(c4cnn[nH]4)C3)=O)C2)=O)c(F)c1 C1(N(C(CN(C(C)=O)C)C)C(C2CCCC2)=O)CNC(=O)CN1C(c1cnn[nH]1)=O c1(C(=O)NC2CCCN(C(c3cnns3)=O)C2)ccnc2ccncc12 C(=O)(CCCCCC(C)(C)C)N1CC(OCCC(=O)NC2C(OC)C2)C1 N1(C(c2cn(C)nn2)=O)CC(O)CC1CC(N1CCCCC1C1CC1)=O C(c1cnccn1)=CC(=O)NC1(CNC(=O)CC2(C(F)F)CC2)CCOC1 C1(C(N(CC(C)O)CCNC(=O)C(C2CC2)C2CC2)=O)CCC(C)(C)CO1 c1(C(N2CC(CCNC(CNC(=O)OC)=O)C(C)C2)=O)cc(OC)ccc1Br C1(C(=O)NC(C(=O)Nc2cccc(C)c2)CC2CCC2)CCCCCCC1 c1(CN2CC=CC(NC(CN(C(COC)=O)C)=O)C2)c(Br)nc2n1CCOC2 C1(=O)CCCC(=O)N1.c1(N(C2CCN(C(C3CC3)=O)C2)CC)cc(=O)c(O)c[nH]1 c1(CC(N2C(CNC(C(C)SCCCC)=O)CC(F)C2)=O)cc(F)ccc1C c1(OC(=O)CCNC(N2CCCC2c2ncccn2)=O)ccccc1 C12(n3cncn3)CC(CN1c1nnc(C3CC3)n1CC1CC1)C2 c1(C(CO)NC(CN(c2nc3ccccc3s2)C)=O)cc2ccccc2s1 C(=O)(C(C)(C)CCOC)N1CC2C(C(=O)NC3(CC=C)CCCC3)C2C1 CC1CCC(CC(=O)NCCC(C)N(C(=O)CCC(=O)N(C)C)C)OC1 N1(C(c2occ(C(N)=O)c2)=O)CCCN(C(=O)CCCC(F)(F)F)C(CO)C1 c1(C(N2CCC(CNC(C(C(CC)CC)OC)=O)C2)=O)cnn2c(N)ccnc12 C(=O)(CCCC(F)(F)F)N1CCC(NC(c2c(C)cc(SC)o2)=O)CC1 N1(C(CCNC(=O)NC)=O)CC(C)CCC1CNC(c1cc(CS(C)(=O)=O)on1)=O N1(C(C=CS(C)=O)=O)CCN(C(=O)C#CC2CC2)CC1CC(C)(C)C Cc1ccc2c(C(N3CCC(NC(=O)Cn4ccc(C)n4)C34CC4)=O)coc2c1 C1(NC(C(CCC)(C)C)=O)CN(C(=O)CC2CC(OC)C2(C)C)CC1N=[N+]=[N-] C1(NC(c2c(C)[nH]nc2Cl)=O)CS(=O)(=O)C12CCN(c1ncc(C(F)F)cn1)CC2 N1(C(C2C(=C)C2)=O)CCC(CCCNC(c2cnc(C)cn2)=O)CC1 CCCCC(CNC(c1c(Cl)cnn1C)=O)NC(C1(CO)CCOCC1)=O c1(C(=O)N(C)C)n[nH]c2c1CN(C(C1(CNC(CCSCC(C)C)=O)CC1)=O)CC2 c1(C(CCOC(C)(C)C)NC(=O)Nc2c(CC)[nH]cc2)ccc(OC)cc1 N1(Cc2cc(C(N(C)CC)=O)no2)CCCC(CC(=O)NCC(C)C)C1 C(c1ccncc1)=CCNC(C1(NC(C(N2CCNC2=O)C)=O)CCC1)=O C(C(F)(F)C(F)(F)Br)C1C(N2C(=O)CN(CCC(C)C(C)(C)C)C2=O)C1 C=CC(CC)CC(=O)N1CCCC1CN(C(=O)CC(C)(C)c1ccccc1)C c1(C(=O)NCC(=O)NC(C(=O)OCC2(CCC=C)CC2)C)ccc(C)cc1 Cc1ccc2sc(C(=O)NC3CC3NC(c3cc(F)c(F)cc3F)=O)cc2c1 N1(C(c2c(C(C)C)cnn2C)=O)CCC2CN(C(=O)COC3CC=CC3)CCC12 N1(C(c2n(C)nnc2)=O)CC2CCC(C1)C2NC(c1cc(F)c(F)cc1Cl)=O c1(C(=O)NC2C(OC)CN(C(=O)CCCC(C)=O)CC2)nnn2c1COCC2 c1(CNC(C2(C)C(C3(C(=O)NCC)CC3)CC2)=O)ccc(Cl)c(NC(=O)NC)n1.NC N1(C(CCc2cccc(C)c2)=O)CC2(CCCC2NC(=O)C#CC2CCCO2)C1 N1(C(c2cc(C(C)(C)C)n[nH]2)=O)CC2CC1C2CNC(C1(C)CCCS1)=O n1(CC(N2CC3C(NC(=O)CCOCC(F)F)(C3)C2)=O)ccc(O)nc1=O C(CC(F)F)(C(=O)N1CC2C(C1)C2(C)C)N(C(CSCCCC)=O)C N1(C(C(=O)OCC)=O)CC(OC)CC1C(=O)NCCC(F)=C(F)F C(C)(C(=O)NCCOCC(=O)NCC(C)(C)F)SCC N1(C(C(CCCC#C)C)=O)CCC2(C=C(C(=O)N3CC(=O)NC(C(C)C)C3)C2)C1 C(CCC(C)(C)NC(c1ccc(C2CC2)o1)=O)OC.C12CCN1C(=O)C2 c12cc(oc(=O)c1)C(=O)O2.C12(C)CCC(CC1)CNC2=O.N1(CC)CC2CC2C1 n1(C(C)C)ncc(C(N2CCC(CO)(NC(C3CC3(C)C(F)F)=O)C2)=O)c1Cl C(C(=O)Nc1ccc(C(=O)NC(c2c(C)n[nH]c2C)C)nc1)(C(C)C)OCC C(=O)(N=c1nc(C2CCOCC2)[nH]n1C)N1CCC(CN(CCC)C)C1 c1(CC(C2CCCCC2)C)nc(-c2cncc(F)c2)nn1CCN(C)C CC1CSCCCN1C(=O)C(CCOCCOC)NC(=O)C=Cc1cccnc1 c1(CC(=O)NCC(CCC)(C)NC(c2cnc(C)s2)=O)cccc(F)c1F c1(OC)ccc(C(=O)NCC(C)N(C(C2CCCN(C)C2)=O)CC)cc1C(F)F CC(CN(C)C)CCC(=O)NC1(F)CCC(NC(C2(SC)CC2)=O)C1 O=C(CC(F)(F)C(F)(F)F)NCC(C1CC1)NC(=O)C1=C(Cl)CCOC1 C1(C)(C(N2CC(CNC(C(COC)OC)=O)C(C)C2)=O)CC2(CCC2)C1 C1(NC(c2cc(C)nn2C)=O)CS(=O)(=O)CC1NC(C1(C#N)CCC1)=O C1(C(=O)NCC=CCNC(C2(CCCC)CCCC2)=O)CCc2nn[nH]c2C1 c1(C(=O)NC2(C)CCCN(C(C(C=CCCC)O)=O)C2)[nH]c(C)c([N+](=O)[O-])c1C c1(C(=O)NCc2ccc(Cl)cc2Cl)ccc2c(-c3ccncc3F)cccc2n1 c1(C(=O)NCC2(NC(C3CCCC3)=O)CCC2)ccc2c(O)nncc2c1 C1(C(N2CCC(NC(c3ccnc(C(F)F)c3)=O)(CO)C2)=O)CC(C2CC2)=NO1 C1(Cl)(C(=O)NCC(CN(C(CCn2c(C)cc(C)n2)=O)C)C)CC12CCOCC2 C1(=O)CS(=O)(=O)CCOCCN1C.C=CC1(CC(=O)N(C)CCOCC)CC1 CCS(=O)(=O)CC(=O)N1CCCC1(C(N1CCOC(C#N)C1)=O)C(C)C O=C(C1=C(F)CNCC1)NC1CC(c2cccc(F)c2)C12CCC2 c1(C(=O)NC(CC)CNC(=O)C(C)N(C)C)cc2n(n1)CCNS2(=O)=O C12(C(=O)NCCC(C)NC(=O)CC3CC4(CCC4)CO3)CCC(C#N)(CC1)CC2 C(=O)(C(C)CC(N)=O)N1CCCC(CN(C(C(C)=C2CC2)=O)C)C1 c1(C(N2C(CN(C(CNC(C(CC)C)=O)=O)C3CC3)CCC2)=O)snc(O)c1Cl c1(C(=O)NCC(C)N(C(C(CC)N(C2CC2)CC)=O)C)cc(OC)c(O)c(OC)c1 c1(OC(N(CCNC(CCCNC(C)=O)=O)C2CC2)=O)c(Cl)ccc(F)c1N Cn1cc(CC(=O)NCC(c2ccccc2)NC(C2(CO)CCCO2)=O)cn1 CCCCC(O)CN(C(=O)CC1C2CN(C(=O)C3=NOCC3)CC12)CC C1(C)(CNC(CN2CCC(C)C2)=O)CN(C(=O)CCN2C(=O)CCC2=O)CCO1 C(=O)(C1=NOC(C)C1C)NC(C1CCN(C(C2CCN(C(C)=O)CC2)=O)C1)(C)C N1(C(COCC)=O)CCCC1C1CCCN1C(c1c(Cl)cnn1C)=O c1(C(=O)NCC(CNC(C(C)N(CC)CC)=O)C)cc2c(Cl)cncc2s1 CC1(C(=O)NCC(c2ccc(F)cc2)NC(=O)CC(F)(F)F)CC2(CCC2)C1 C(C(C(=O)N1CC(COC(C)=O)C1)C(C)C)NC(c1cccc(C)c1)=O c1(-n2cc(-c3sc(OC)c(CO)c3)nn2)ccc(Cl)c(C)c1C(=O)OC N1(CC)CC(N=c2[nH]c(=N)[nH]c(=NCc3nc(Br)n(C)n3)[nH]2)C1 C1(CNC(CCS(C)=O)=O)CCCC2(CN(C(C34CCC(C3)C4(C)C)=O)C2)O1 C12(CC1)C(=O)N(CCNC(C1CC1CO)=O)CCO2.CN(C)CCO CC1(C)CCOC(CC(=O)NC(CNC(=O)C=Cc2cncs2)CO)C1 N1(C(C(C=C)C)=O)CCC2(C1)CN(C(c1cc(OC)cnn1)=O)C2 C#Cc1ccc(C(N2CC(C3(NC(=O)Cc4ccc(F)cc4)CC3)C2)=O)c(C)c1 C#Cc1c[nH]nc1C(=O)N(C1CC(C#N)C1)CC(=O)N(CC(C)(CC)OC)C N1(C(C(C)C)=O)CC(NC(=O)CCc2cnoc2)C(F)C1 c1(CN2C(C(=O)NC3(c4cccc(Cl)c4)CC3)CC(F)C2)ccccc1[N+](=O)[O-] C1(SCc2cn(CC3(CS(C)=O)CCCC3)nn2)CCCCNC1=O N1(C(C=C(C)C2CC2)=O)CCC2(CCCC2CNC(C2CCCC(=O)O2)=O)CC1 C1(C)(NC(CC(=O)OC)=O)CCCCC1C(=O)NCC1CCn2cncc2C1 c1(C(=O)NC(CNC(C(C)n2cccn2)=O)C2CC2)nccnc1N C1(C(N(CC(CN(C)C(C23CC(C(C)(C)C)(C2)C3)=O)O)C)=O)CC2(CCCO2)C1 C1(NC(C(CC)CC)=O)CC2(CCN(C(c3ccc(O)cc3C)=O)C2)C1 C1(NC(C2(CCC)CCC2)=O)CCN(CC(=O)NC2CCCC2SCC)CC1 CCCCCCC(F)C(=O)N(C1CN(C(c2cnc(C)[nH]c2=N)=O)CC12CC2)C CC1CCCN(C(C2CCCCN2c2ccnc(Br)n2)=O)CC1 c1(C(N2CC(C=C)C(NC(C3(CC)CCOCC3)=O)C2)=O)cc2ncccn2n1 C(=O)(C(C)(O)C(F)(F)F)NC1C(NC(c2nn(C)c(O)c2)=O)CCCC1 c1(C(N2CC(c3cccc(C)c3)CC2C)=O)cnn2cc(C(=O)N(C)C)cnc12 CC1(C)CC(CC(=O)NCc2ccc(O)cn2)N(C(=O)CC2CCC(C#N)C2)C1 c1(C(N2CC(C)(NC(C3CC(S(C)(=O)=O)C3)=O)C2)=O)cccc2cnsc12 c1(C(=O)NC(CNC(=O)C=CCO)C2CC2)c[nH]cc1-c1ccc(Cl)s1 N1(C(CC2C(CC)C2)=O)CC(C2CCCN(C(c3cnsc3)=O)C2)C1 C1(NC(C2CCCC2)=O)CN(C(=O)Cn2ncc(Br)n2)CCC1F C1(CNC(C(C)(C)n2cncn2)=O)C2CN(C(=O)CC3CC4CC4C3)CC12 C(=O)(C(C(F)(F)F)C(F)(F)F)NC1(C2CN(C(Cc3cnc(C)[nH]3)=O)C2)CC1 N1(Cc2ccc(COCC)o2)CC(=O)NCC1Cc1ccc(F)cc1 N1(C(CCNC(N)=O)=O)CC(NC(c2ccc3n[nH]cc3c2)=O)CC2(CCC2)C1 c1(C(=O)NCCC(CNC(=O)C=C2CCCCC2)O)cc2n(n1)CCC2 c1(C(N2CC(C(F)(F)F)CCC2C)C(=O)NC)ccc2sc(C(=O)OC)cc2c1 N1(C(C(C)C2CCC2)=O)C2CCC1CN(C(C1CCc3ncncc3C1)=O)CC2 CC1CN(C(=O)Nc2cnc(Oc3cccc(Cl)c3F)s2)CC(CCO)O1 C1(CCCCC)CCC(C(=O)NCC23CC(NC(C4CC4(F)F)=O)(C2)C3)CC1 N1(C(c2c(CNC(C3CC4CC4C3)=O)scc2)=O)CCCCC1C(F)F c1(C(N2CCC3C(CCN3C(=O)C(F)F)C2)=O)cc2ccccc2nc1O c1(CC(=O)N(C2CC3CN(C(C=C(CC)C)=O)C2C3)C)nc(C)n2c1CCCC2 C1(C(=O)NC2CCCN(C(COCc3onc(C)n3)=O)C2)CC2(COC(=O)N2)C1 N1(CC(C(c2ccccc2)OCCOC)=O)CCC(C(C)C#N)CC1 C1(C(N2CCC(C(C)N)C2)=O)CCN(C)CC1.c1(C(C)(C)C)ncnn1C C(C)(c1ccccc1)=CC(=O)NCC12OCC(CNC(C(C)OCC=C)=O)(C1)C2 C1(CCNC(COCCCOC)=O)CCC(C)N(C(=O)CCc2scnc2C)C1 N1(C(CCCCC)=O)CCC2CCCC12CNC(=O)C=Cc1cccc(C#N)c1 c1(SC)ccc(CNC(C2N(C=O)CC(C)C2)=O)cc1.c1(N)ccc(C(F)(F)F)nc1 N1(C(C(C)NC(=O)NC)=O)CCC(NC(c2cc(C(C)C)on2)=O)C(CO)C1 N1(C(CC(COC)NC(c2cc(=N)[nH][nH]2)=O)=O)CCn2nncc2C1 N1(C(c2c(CC)cno2)=O)CCCC2(CCCN2C(c2cnn(C(C)C)c2)=O)C1 C1(C(=O)NCC(CC(=O)N2C(C)CCC2C)OC)CC2C(C1)C2(C)C N1(C(CCC)=O)CCN(C(c2c(C)noc2C(F)(F)Cl)=O)CC1CO CCC(C)(CC(=O)NC(CN(C(=O)C(C)OCC(C)C)C)CC)C(=O)OC C(CC(=O)N1Cc2ccccc2CO1)NC(C1CCN(C(=O)NC)CC1)=O Cc1cc(Cl)ccc1CCCCOC(=O)C#CC1CCCC1.C1(=O)CCN1C(C)C Cc1[nH]c(=NCCOCCN(C(=O)CC2CCOC2)C)ccc1[N+](=O)[O-] C1(N(C)CC2CCCO2)CCN(C(C2CC(=O)N(C3CCCC3)C2)=O)CC1O C=CCCCCCCC(=O)NCC1CCC(NC(C2CCC(C)CC2)=O)C1 C(CCCC(=O)N1CC(c2nnnn2Cc2ccccc2)(OC)C1)(C1CC1)NC c1(OCCn2cc(NC(N3CCCC(C(C)(C)O)C3)=O)nn2)cccc(Cl)c1Cl N1(S(c2ccc(P(C)(C)=O)cc2)(=O)=O)CCOc2c(F)cc(F)cc2C1 c1(C(N2CCC(F)(CNC(c3cccc(OC)n3)=O)C2)=O)ccc(OC)cc1F C1(NC(C2N(C)CCC2)=O)CCC2CN(C(c3cccn3C)=O)CC2C1 Cn1c(C(N2CC=C(CNC(C3CN4CCC3CC4)=O)CC2)=O)cc2sccc12 c1(CC)nnc(O)c(C(=O)NCCCCC(C)NC(=O)C(C)=CC2CC2)c1CC c1(OC)cc(O)ncc1C(=O)NCC(C)CNC(c1ccc(SC2CC2)cc1)=O N1(C(C(CC=C)(C)C)=O)CCC2(CC1)CC2C(=O)NC1CCN(S(C)(=O)=O)CC1 C1(CC)CN(C(=O)Cc2ccsc2C)CCN1C(c1ncn(C(C)(C)C)n1)=O c1(OC)ccc(F)c2c1CN(C(c1ccn3c(C)cnc3c1)=O)CC2 C(=O)(C(Cc1ccco1)C(F)(F)F)NC1C(NC(C(OC)OC)=O)CCC1 C12(C(=O)NC(c3nc(C)sc3)C)CCCC1CN(C(=O)CC1CC=CC1)C2 CCC(CC(=O)NCC(CNC(C12CCC(OC)C1C2)=O)OC)CC(C)C c1(OC)cc(C(=O)NC2CCN(c3nnc(C#N)s3)C2)cc([N+](=O)[O-])c1C c1(CN(C(=O)CN(C(C)COC(C)C)C)CC2CCC2)cc2ccc(Cl)cc2o1 CC(C)(C)CCC(F)C(=O)NCC1OCCC1C(=O)Nc1cnc(O)c(F)c1 C(C(=O)NCC(O)CCNC(=O)C(F)(F)C1CCOCC1)(C(C)C)SCC c1(C(N2C(CN(C)C(C3CC=CCO3)=O)COCC2)=O)cc2cc(Cl)ncc2[nH]1 c1(C(=O)NCCCN(C(CCOC)=O)CC2CCCC2)cc(C)n(C)c1C C12(C3(O)CN(C3)C1)CC2.c1(C(=O)NC(C23CC(C)C2C3)=O)cc(CN(C)C)c[nH]1 CCCCC(CC(=O)NCCCOC(F)(F)F)NC(c1cccc(C)c1O)=O CN1CCCC(C(=O)N(C)CC2(O)CN(C(=O)CC3CC4CCC3C4)C2)C1 N1(CC(C)C)N=C(C(=O)NCCCN(C(=O)CN(C)C)C(C)C)CCC1=O c1(C(N)=O)ccc(C(F)(F)F)nc1N.N12CCC(CC1)C(=O)NCCNCCC2 N1(C(c2c(CC)[nH]nc2Cl)=O)CC(CNC(C2(C)CNC(=O)C2)=O)OC(C)(C)C1 c1(C(N2CC(CNC(C3C(C(N)=O)C3)=O)C3(C2)CC3)=O)cc2ccccn2c1 CCCC(C)(C)CC(=O)N(CCNC(=O)C(C)ONC(=O)OC(C)(C)C)C1CC1 C1(C(N2CCC(CCNC(C(CCC)O)=O)C2)=O)CC2(CCC2=O)C1 c1(C(=O)NCCC(C)N(C(c2ccc(COC)o2)=O)C)c[nH]cc(C)c1=O C1(C(N(C(C)CNC(C2CNC(=O)N2)=O)C)=O)C2CCC1(c1cccnc1)C2 C1(C(=O)NCC2CCCN(C(=O)CC3CCCCC3O)C2)Cc2ccccc2O1 C1(NC(C(CC)O)=O)C2CC3C1C3C2C(N1CC(C)(C)C1C(=O)OCC)=O C1(NC(c2c(C)cccc2F)=O)CC2CCC(C1)N2C(C1CCCS1(=O)=O)=O c1(OC)ncc(C(N2CCC(CNC(=O)CCc3cnc[nH]3)C2)=O)cn1 c1(C(=O)OCC)ccccc1C1CN(C(C2CCC(Nc3cccn3C)C2)=O)C1 c1(C(C(=O)N(C(CCNC(CCSCCCC)=O)C)C)C)cccnc1 C1(OC)CCC(C(N2CCC(C)(CO)C2)=O)N(C(c2cccc(CO)n2)=O)C1 C1(n2c(C(C)(CCC3CC3)NCCCOC3CCC3)nnn2)CCC(F)(F)CC1 c1(CNC(C2CCN(CCCc3ccccc3Cl)C2)=O)cc(Br)cc2[nH]ncc12 C#Cc1cccc(C(N2CCCC(NC(=O)CCOC(C)C)CC2)=O)c1F CC1CC(C(=O)N(C(C)C(=O)NCC(O)C(F)(F)F)C)CN1C C12(C(=O)NC3CCC(CNC(c4ccc(N)c(O)c4)=O)C3)CCCN(CCC1)C2 C(=O)(CC(COC)NC(=O)C=NOC)N(C(C#C)C)C C(=O)(CCCC(=O)NCCN(CC(C)O)C(c1nn(C)cc1C(F)(F)F)=O)OC N1(C(=O)CCCCc2ccc[nH]2)CC2CCC(C1)N(C(c1ccc(O)cn1)=O)C2 c1(OC)nc(C)cc(=NC(=O)c2ncc(-c3ncc(Cl)cc3F)cn2)[nH]1 N(C(=NCCc1cccs1)NCC(c1cnn(C)c1)(C)C)Cc1n(CC)ncn1 Cc1ccc(C(=O)N(CC(O)CN(C(=O)C(C)c2cccs2)CC)C)c(C2CC2)c1 CC1(C(N2C3CCC2COC3)=O)CCCN(c2ncc(Br)c(C(F)(F)F)n2)C1 N1(C(CCc2cc(OC)no2)=O)CC(CNC(C2CC23CCCC3)=O)CC1(C)C N1(C(c2c(CC)occ2C)=O)CC2CC(NC(=O)C=Cc3ncco3)C(C2)C1 CC(C(C)NC(C1(CN(C)C)CC1)=O)NC(C1(C#N)CC1)=O c1(C(N2CCC(OCCN(C)C)C2)C(=O)N(CC=C)C(C)C)ccnc(Cl)c1 N1(C(=O)C(C)(F)C(=O)OC)CC=C(C(C)(C)C)CC1.CCCC(C(O)C=O)N C12(C(=O)NCCCCC3CN(C(c4c(OC)c[nH]n4)=O)C3)CCCCC1C2 CN1CCCCN(C(C2C3CC3CN2C(=O)CCC2(C)CC2)=O)CC1 C1(C(N(C2CN(C(=O)C(C)(C)CC#N)CC2O)C)=O)C2CCCCCCC12 c1(OC)ccc2cc(C(=O)OCC3CCN(C(C)=O)C(C)C3)[nH]c2n1 C=CCCCCCC(=O)NCC1CCCCN1C(c1ccc(F)cc1C#N)=O C1(CNC(=O)CC2CS(=O)(=O)C2)CCN(C(=O)C(c2ccc(Cl)cc2)(F)F)CC1 c1(NC(C(=O)NCCC2COCCO2)=O)nc2cc(Br)cnc2[nH]1 C12(C(N3C(COC)CN(C(=O)C=CCF)CC3)=O)CCC(C)(CC1)OC2 C1(NC(C(C)OCCC=C)=O)CCCC(NC(C2(C)CCN(C)CC2)=O)CC1 C(CC(=O)NCC1C=CCN1C(c1occc1C)=O)(C(N)=O)NC(C)=O c1(C(N(C(CNC(C2CC(CC)(CC)C2)=O)C)C)=O)nc(C2CC2)oc1C c1(C(C(N2CC(CNC(C3C(C)(CC)C3)=O)C2)=O)O)cnn(C)c1 C(C(CC(C)C)C(=O)N(CC(C)O)CCNC(=O)CCOC)OC N1(C(c2csc(Cl)c2)=O)CCC2(CCN(C(c3ncc(Cl)cn3)=O)C2)C1 c1(C(C)C(=O)NCC2CCN2C(=O)COC(F)F)ccc(Br)cc1 N1(C(c2c(C)c(O)ccc2)=O)CCN(C(=O)CC2COC(=O)C2)CC(C)(F)C1 Cc1ccc2ncc(C(N3CCC(C)C(CNC(=O)C(C)(C)CC#N)C3)=O)n2c1 N1(C(=O)CCOCC2CCCO2)CCC2C1CCCN2C(C1CCCCCC1)=O CCCCC(C)C(=O)N1CCC(CF)(NC(=O)Cc2ccc(CO)c(C)c2)C1 O=C(CCS(=O)(=O)c1ccc(F)cc1)NCC1CCCN(C(c2ccsn2)=O)C1 C1(O)CCN(CC2CC2)C1.C1(C=O)CN(C(=O)CNC(c2ncccn2)=O)CS1 c1(C(=O)NCCCC(C)NC(C2N(CC)CC2)=O)oc2ccccc2c1OC c1(CC)cccc(C(=O)NC2CCCC2CC(=O)NCC(O)CN2CCCC2)n1 C1(NC(c2c(C)cn(C)c2)=O)CC2(C1)CC(C(=O)NCCN1CCOCC1C)C2 Cc1ncc(Cl)cc1CC(=O)NCC1(F)CCN(C(C2CCCCC2(F)F)=O)C1 N1(C(CCCCC=O)=O)CCC(O)(CN2CCCCC2)CC1.C1(S)CC1 c1(C(N2C(CNC(C3CCC3(F)F)=O)CCCC2)=O)cccc2nc(CO)[nH]c12 C(N=c1nc(N2CC3CC3C2)c2c([nH]1)CCCCC2)C1CC=CC1 c1(C(N(CCNC(C2CC2c2ccc(OCCF)cc2)=O)CC)=O)ncc[nH]c1=O C=CC(C)C(C)C(=O)N1CCC(C(C)NC(=O)CCS(N)(=O)=O)CC1 C(C)(CC(=O)NCC(O)CCNC(=O)C(N1CCSCC1)C)=C(C)C C1(CC(=O)N(CCCSCC)C)(N)CN(C(=O)C(C)C)C1.OC N1(C(C(COCC)(F)F)=O)CC2(CO)CC1(C(=O)NCC=CC(C)(C)C)C2 C1(CCNC(C(CC)=CC)=O)CCCN(C(=O)C(C)(CC)CC)CC1 N1(C(C(CCC)OC)=O)Cc2[nH]nc(C(=O)NC(C)CCF)c2C1 C1(NC(C(CC2CCC2)NC(=O)Cn2cnnc2O)=O)CCC2(CCC2)C1 C(=O)(CC(O)CC(C)(C)C)N1CCC2(C(CNC(CNC(CCC)=O)=O)C2)CC1 N1(C(CN(C(C(C)C)=O)C)=O)CC2(CCN(C(=O)C=Cc3nccs3)CC2)C1 N1(C(C(CC(C)=O)C)=O)CC(NC(c2cc(Cl)cnc2F)=O)C(C#N)C1 C1(C(N(C2CCN(C(C3CC(C)C3)=O)C2)CC#C)=O)Cc2cc(Cl)ccc2O1 N1(C(c2c(C)[nH]c(C#N)c2)=O)CC2(CCCC2NC(=O)CC(Cl)Cl)C1 N1(C(COCC(=O)NC)=O)CC2(CNC(c3ccccc3S)=O)CCCC2(F)C1 CC1CN(C(=O)COc2ccc(Br)cc2)CC1NC(=O)CC1CCCO1 Cc1cc(CCC(=O)N(CCNC(C2(C#N)CC3CC3C2)=O)C(C)C)ccc1Cl Cn1cnc2cnc(N3CC=CC(NC(C4CCCC4c4nc[nH]n4)=O)C3)nc12 C1(NC(=O)CCOc2ccccc2F)CCC12CCCNC2 C(c1cncc(F)c1)=CC(=O)NC(C)(C)CCNC(=O)CNc1cncc(Cl)c1 C(N=c1nc(N2CCC(COCC)C2)cc(C)[nH]1)c1ccc(C(F)F)c(F)c1 N1(C(C2(C(=O)OCC)CCCC2)=O)CCC2(C1)CN(C(=O)C=CS(C)=O)CCO2 C1(NC(c2ncn(CC)c2)=O)CC(SC(C)(C)C)CC1O CCC(CC(F)F)C(=O)NCC1CCC1NC(C12CC(C1)C(C(F)(F)F)O2)=O C(=O)(C1=C(C)S(=O)(=O)CC1)NCC(CNC(CCNC(COC)=O)=O)OC N1(C(C(c2cccs2)SC)=O)CC(C2CN(C(=O)CC3COC(C)(C)C3)C2)C1 Cc1ccc(O)c(NC(c2csc(-c3cnn(CC#N)c3)n2)=O)n1 N1(C(C2CCN(CC)C2C)=O)CC(C(=O)OC)C2(CCCCCC2)C1 N1(C(C)=O)CCCN(CC(=O)NCCNC(C2CCC(OC(F)F)C2)=O)CC1 C(=O)(C(C)CNC(c1coc(C(=O)NCCO)n1)=O)OC.C(=O)C(C)(C)C C1(NC(CN(C)C)=O)C2CCN(C(=O)C(C)N(C)C(=O)OC(C)(C)C)C12 c1(CCN(C(=O)CSCCOC)C(C)(C)C)ccccc1.c1(C(C)N)ccc(C(F)(F)F)s1 C1(CC)C(NC(=O)CCCN2CCCC2)CCCN1C(C1CC1c1ccco1)=O C(=O)(C(F)C(C)(C)O)N(CCCN(C(Cc1ccc(CC)cc1)=O)C)C(C)C C=CCCC(=O)NC1CC(C)(NC(=O)CC(c2ccccc2)N2CCCC2)C1 N1(c2ncc(C(=O)OCC)cn2)CCC(C)C(NC(c2cc(C)on2)=O)C1CC Cc1cc(C(=O)NC2CCCC2CNC(=O)CC2CCCN2C)c(Cl)cc1N c1(C(=O)NCCOC2CCN(C(C(CC)(F)F)=O)C2)ccnn(C)c1=O C1(NC(c2ccc(CNC(C(C(C)C)O)=O)cn2)=O)CCCC(C)(C)C1 CC1(C)CCc2cc(C#N)c(NC3CN(C(=O)CCC4CCC4)C3)nc21 CCC(CC(=O)N1CC(OC)CC1C(N1CCC(CC(N)=O)C1)=O)OC n1(CC)ncc(Br)c1C(=O)NC(C)C(C(C)C)NC(=O)C#CC1CC1 S(=O)(=O)(c1cccc2c(C(=O)NC(C)(C)C)cccc12)N1C(C)(CC)CC1 c1(CCC)nc(C)cc(=NC2CC3CN(C(=O)CCc4ccccc4C)CC23)[nH]1 N1(C(C2C(C=C)CC2)=O)CCC(N(C(=O)COCC)CCO)CC1.C1C(=O)O1 c1(OC)cc(C(N2CCSC(C)(C)C2)C(=O)NCC2CCC2)ccc1OC(C)C C(=O)(C(O)CC(F)(F)F)NCC1CCC(CN(C(Cn2ncc(C)c2)=O)C)CC1 Cc1nc2c(C(N3CC4CC(NC(C5CC5F)=O)CCCC4C3)=O)ccnc2[nH]1 CCCCCCC(C)C(=O)NC1CC(NC(=O)CC2CCN(OC)CC2)C(O)C1 Nc1c(C(=O)NC2CCC2NC(c2cn(CCO)nn2)=O)cc(F)cc1F c1(C(=O)NCC2(CCCNC(C(C(C)C)O)=O)CCCC2)cnn2c1OCCC2 C1(OC)CC(C(=O)NCCc2ccncc2)N(C(C2CCCN2C(C)C)=O)C1 c1(C(=O)NC2C(C)CCN(C(CCCCCC)=O)C2)cc2c(C)cccc2[nH]1 CC1(C)COc2cc(C(c3nnnn3C3CC3)NCc3sc(Cl)nc3Cl)ccc21 C1(O)(C(=O)NC(C(N2CCC(CC#C)C2)=O)COC)CCCCC1 C(=O)(C(O)C(F)(F)F)NC(C(C)(C)NC(C=CC(c1ccc(C)cc1)=O)=O)C c1(CC(=O)NC(C(C)NC(C2(S(C)(=O)=O)CCC2)=O)CO)c[nH]c2cnccc12 C1(C(=O)NC2CCC3(CCC3)C2)CCCN(C(c2ccc(CO)s2)=O)CC1 Cc1cc(Br)cnc1C(N1CC2(CC(CC(=O)NCCCn3ccnc3)C2)C1)=O c1(C(N2CCCN(C(c3cncc(CC)c3)=O)C2C)=O)ccc(Cl)c2occc12 C1(CNC(COCC)=O)CC2(CO1)CN(c1ncncc1C#N)C2 N1(C(C2(Cl)CC2)=O)CC(NC(C2(c3ccc(O)cc3)CC2)=O)C2(CCC2)C1 C1(NC(C(c2ccco2)NC(C=C(COC)C)=O)=O)CCCC12CC2 C(=O)(CCc1cscn1)N(C1CN(C(=O)C=CCF)C1)CC1CC1 N1(C(CC(CC#C)c2ccccc2)=O)CC(NC(C2(O)CCC2)=O)CC(C)(C)C1 c1(CNC(N(CCCOCC(F)(F)F)CCC)=O)cc(F)ccc1Cl c1(C(C)C)cc(C(=O)NC(C)CC(C)NC(=O)C(F)CC2CCCC2)on1 c1(OC)ccccc1CNC(=S)NC(c1ccc(SC)cc1)C1CC1 C1(C(F)(F)C(=O)NCC(C)(C(C)C)NC(=O)CCOC(C)=O)(OC)CCOCC1 C1(C(=O)NC(c2cccc(F)c2)(CCOC)C)CCCN(c2cc(NC)ncn2)C1 Cc1cc(Cl)c(C)c(C(=O)N(CCCNC(C2CCCCO2)=O)C)c1N N1(C(CN(CC#C)C(c2ccn(CCF)n2)=O)=O)CC(C)CCC1C C1(C)(CNC(c2sc(C)c(O)n2)=O)CC(F)(F)CN1C(c1ccc(C(F)F)o1)=O CCCCC(CC)C(=O)N(CCC(=O)N(C)CC1(O)CCCC1)C Cn1c(C(c2nnnn2C2CCOC2)NCCCCF)cc(=O)n(C)c1=O c1(C(N(CCC)CCNC(=O)C2=CC3C=CC(C2)C3)=O)cc2sc(=O)n(C)c2s1 c1(OC)cc(CC(C)NC2CC(=O)N(c3cccc(F)c3)C2)ccc1O c1(NC(C2CCCN2C(c2ccc(Cl)cc2Cl)=O)=O)cncc([N+](=O)[O-])c1 C1(C(C(=O)OC)C)CCCN(C(C2(NC(c3cc(C)sc3C)=O)CC3(CC3)C2)=O)C1 C1(C)(C(N(CC(=O)NC2CC(C)N(C)C2)CC)=O)CCCCC1O c1(OC)cccc(C(N2CC=CC2CNC(c2sncc2C)=O)=O)c1N CC1CC2(CCN(C(c3ccc(C(N)=O)cn3)=O)CC2)CN1C(=O)CCC1CC1 C(C)(CN=C(NCC(F)F)N1CCC(O)C1)(N1C(COC)CCCC1)C1CCC1 c1(C(=O)NCCN(C)C(c2ncn(C)n2)=O)ccc(=O)n2c1CCC2 C(=O)(CCCCC(C)C)NCC1N(C(CC(=C=C)C)=O)CC(C)C1 C1(C(=O)NCC(CN(C(C(C)(c2ccccc2)OC)=O)C)C)CC2(C1)CC2(F)F C1(CN(C(=O)CC2CC(OCCF)C2)C)CCCCN1C(C1CS(=O)C1)=O n1(CC)c(CNC(=O)C(C)N(C(=O)CSc2cn[nH]c2)C)nnc1O c1(NC(COC(C)C)=O)ccc(S(=O)(=O)NC(=O)OCCCN(C)C)cc1 C(=O)(CC(C)(CC)C(=O)OC)NCCNC(C(CC)(CC)c1ccccc1)=O CCC(CC)CC(=O)NCC1CCN1C(=O)C(C1(O)CCCC1)F CN1CC2C(CCN2C(C2CCC2C2CCC2)=O)CC1=O C1(c2n(CC(=C)C)nnn2)(NCC2CCCNC2=O)Cc2ccc(F)cc2C1 C#Cc1ccc(Cl)c(C(=O)N(C2CCN(C(=O)CC3(C)CC3F)CC2)CC)c1 CCCCC(C(=O)Nc1cc(F)ccc1OC)n1ccnc1-c1ccc(SC)o1 N1(C(c2ccc(C)s2)=O)CC(C(=O)NCCS(C)(=N)=O)C(F)C1 c1(CN2CCCC(NC(Cn3ncc(C#N)c3)=O)CC2)[nH]nc2c(F)cccc12 c1(C(C)=O)cc(N(C)C)ccc1F.c12cc(F)ccc1NC1CC(C1)C(=O)NC2 CCCCCCCC(=O)NCC1C(CC)CCN1C(=O)CCN1CCC(F)C1 C(=O)(C(C)CC(C)C)N1CC(C(N2CC(CC)(OC)C2)=O)OCC1 N1(C(C2CN(C(C)=O)C2)=O)CC(N(C(=O)CC2CC(C)=NO2)CCO)C2(CC2)C1 n1(CCOCC)nnnc1C(c1ccccc1)NCCNCC(C1CCC1)F c1(C(=O)NCC(COC)NC(=O)CN2CCC(N(C)C)CC2)c(C)ncn(C)c1=O CC(C)C(C#N)C(=O)N(CCCNC(C1CCN(C)C1)=O)Cc1cccnc1 c1(OC)ncc(C(N2CCC(C)(NC(=O)Cc3nnc(C)o3)CC2)=O)cc1Br c1(CC)c(C(=O)NCCC2(NC(=O)Cc3cncnc3O)CCC2)cccc1C N1(C(=O)Nc2nc(F)ccc2Br)CCC2(CC1)C(O)CC2O c1(CC(N2CC3C(CNC(=O)COCC(F)F)(C3)C2)=O)ccnc(F)c1F CC1CN(C(C2(C3CC3)CCCO2)=O)CC1NC(=O)CCCn1ccnn1 CC(=NO)c1cc(C(N2CC(O)(CCNC(=O)COCCN(C)C)C2)=O)cnc1O Cc1cc(C(N2CC(N(C(=O)C(F)C3CCC3)C)C2)=O)nn1CC(F)F CC1(C)CC(NC(C23CC=CCN2CCC3)=O)CCN(C(C2CCS2(=O)=O)=O)C1 S(=O)(=O)(c1cc(Cl)ccc1F)NC1CN(C(=O)Cc2ccc(Cl)cn2)CC12CC2 N1(C(C(C=C)OC)=O)CCN(CCN(C(=O)Cc2ccoc2)C)CC1 CC(C)C(C(=O)NCC1CCN(C(=O)CCNc2ccccn2)C1(C)C)C(C)C C1(C)(CO)CC(NC(C(C2CCN(C(=O)CCCN3CCCC3)C2)C)=O)C1 c1(C(=O)NCCC2CC3N(C(C(C)=CC)=O)C(CC3)C2)cc(S(C)(=O)=O)oc1C C1(OC)(CNC(c2ccnn2C2CC2)=O)CN(C(C2CCC3CC23)=O)C1 c1(-c2c(OCCC)ccc(NCc3ccc(C)nc3)c2)cccc2[nH]ncc12 C(=O)(C(C)(C)CN(C)C(c1cccc(O)c1)=O)NCC(C(=O)NC)O Cc1ccc(C)c(C(=O)N(C)CC2CCCN2C(C2CC3CCCC3C2)=O)n1 c1(C(=O)NCC(CNC(c2cc(CC)oc2C)=O)C)cnc(O)c(C(F)(F)F)c1 C1(NC(C=CCNC(c2cc(Cl)ns2)=O)=O)CCC(O)C(O)C1 C1(CC(=O)NCc2ccc(C(=O)NC3C(CCC)C3)s2)CCCOCC1 C1(COC)(NC(C2COCC2C(N)=O)=O)CCN(C(=O)C(C)CS(C)=O)CC1 N1(C(C(C)OCCC=C)=O)CCC(NC(C2C(c3nc(=N)[nH][nH]3)C2(C)C)=O)CC1 c1(CC(N2CC(COC)N(C(=O)C3=C(C)OCC3)CC2)=O)cccc2sccc12 CC1(CNC(=O)CCCn2ccnn2)CCC(NC(=O)C(F)F)CC1 C1(CC)CN(C(c2cnn(CC)c2)=O)CCN1C(C1(c2ncccc2F)CC1)=O C1(NC(=O)CCSc2ccccn2)CCCN(C(c2ccc(C3CC3)s2)=O)CC1 c1(C(N(C2CCN(C(c3cc(OC)nn3C)=O)C2)CC)=O)cc2sccc2cn1 c1(C(N2CCC(N(C(=O)C(C3CC3)OCC)CCC)C2)=O)oc2ccccc2c1C c1(SCC(=O)NCC#CCNC(C2C(C(N)=O)OCC2)=O)ccc(Cl)cc1 c1(NC(C)=O)nc(C)c(S(=O)(=O)N2CCC3C2CCN3C(=O)CCc2ccoc2)s1 C(CS(=O)(=O)CC(=O)N(CCCN(C(c1coc(N(C)C)n1)=O)C1CC1)C)OC c1(N2CCOCC(NC(C3CC34CCOCC4)=O)C2)ccc(F)cc1[N+](=O)[O-] C=C(Br)CCC(=O)NCCN(C12CCC(CC1)C2)C(c1ccncc1)=O C(N=c1[nH]c2c(c(=NCC34CC(CCO3)C4)[nH]1)CSC2)C1C(C)CCC1 c1(C(=O)NCC(CC)NC(=O)CCCC(C)=O)cccc2nc[nH]c12 c1(C(=O)NCC(C)N(C)C(C2CC2C(C)O)=O)nnc(C(F)(F)F)s1 c1(C(=O)NC2CC(CC(=O)NCC(CO)C3CC3)C2)cc(C2CC2)no1 C1(C(=O)OC)C(N2CCCC(CNc3ccccc3)C2)CCCN1C N1(C(c2c(C(C)C)c[nH]n2)=O)CC2CC(NC(=O)C#CC3CCCO3)CC(C2)C1 CCC(C(=O)NCC1CN(C(=O)CC2COC(C(F)(F)F)C2)C1)C1CCOCC1 CC1Cc2cccc(C(N3CC=CC(NC(=O)Cc4cnc[nH]4)C3)=O)c2O1 C1(NC(C=CC=CCC)=O)CCN(C(c2ccc(C)cc2Br)=O)CC1F C12(CNC(C3C(OCC)C3)=O)CC(CO)(CN1C(C1(C)CCOCC1)=O)C2 Cc1cc(C(N2C(C)C3CC2C3NC(=O)CNC=O)=O)c(C)c(C)c1 C1(CC(=O)NC(C2(O)CN(C(c3c(OC)csc3)=O)C2)C)CCC2(CCC2)O1 c1(CNCC2(C(=O)Nc3c(SC)cccn3)CC2)c[nH]c2ncc(Br)nc12 c1(CC)ccc(F)cc1C(=O)N(C)CC1CCCN(C(=O)COC2(C)CCC2)C1 c1(NC(=O)NC(CSC)(C)CC)cc(OC(F)F)ccc1F n1(CC(C)O)cc(C(N2CCC(NC(c3ccon3)=O)C2C2CC2)=O)ccc1=O c1(CNC(N(CCc2ccc(C)cc2)C)=O)ccc(C(F)(F)F)c(C)n1 C(=O)(C1=CCCCCC1)N1CCCC(C(=O)NC2CCS(=O)(=O)C2)(CC)C1 N1(C(C2(OC)CC2)=O)CC(NC(=O)CC=C(C)C)C2CCCC2C1 Cc1ccc2c(c1)CCC2C(=O)NOCCC1CCO1 C1(C(=O)NC2CC(C)CN(C(=O)C(C)(C)c3cccs3)C2)CC2(C1)CC1(CC1)C2 CCCCC(=O)C(=O)NC1COCCC1NC(c1cn(C)nc1CC)=O N1(C(C=CC(CC)=CC)=O)CCCC(NC(=O)Cc2ncoc2C)C1C C1(CNC(c2nc(C(C)OC)oc2)=O)CN(C(c2ccncc2Cl)=O)C(C)(C)C1 c1(C(=O)NC(C(=O)NCCC=C=CC)(C)C2CCC2)cnc(CC)nc1 N1(C(CCCC)=O)CC2(CNC(C3(Cl)CC3)=O)CCC1CC2 C#Cc1cc(C(=O)NCC(CNC(=O)C(C(C)O)N(C)C)C(F)(F)F)cc(N)c1 Cc1cc(C)n(CC(=O)NCCC2CC(C(=O)NC3(CC(F)(F)F)CC3)C2)n1 C1(NC(C(C)CNC(C2(CN(C)C)CC2)=O)=O)CC2CCC(C1)N2C C1(NC(CNC(C)=O)=O)CCCN(C(c2cn(C(C)(C)C)nc2Br)=O)C1 N1(CC(=O)NC(C2CN(C(C3CCC(C(F)(F)F)O3)=O)C2)(C)C)CCCCCC1 c1(C(=O)NCCCC(CCC)NC(c2cnn[nH]2)=O)cc(OC)ccc1[N+](=O)[O-] Cn1[nH]c(=Nc2ccccc2C(F)(F)F)cc1-c1ccc(COC2CCC2)cc1 c1(CN2CCN(CC(=O)Nc3cc(O)ccc3C(F)F)CC2)c(F)cc(Br)cc1Br CN=c1[nH]c(=NCCC2(CO)CC2)[nH]c(=NCC2CC2C2CCCCC2)[nH]1 c1(C(=O)NC(CCCNC(C2CC=C(C)CC2)=O)C)cc2ccccc2s1 c1(OC)cnc(C(N2CCOCC2CNC(c2conc2C(C)(C)C)=O)=O)nc1 Cc1cc(-c2cnc(CNC(c3ncc(C)cc3Cl)=O)nc2)cc(F)c1 C1(CCC)CN(C(c2cnccc2F)=O)CCN1C(c1nccn1CC)=O C1(SC)CC(C(=O)NCCC(C)NC(=O)Cc2ccsn2)C1 C12(CNC(C(C(C)C)OC)=O)CCC(CN(C(C3CC4CCC4C3)=O)C1)C2 c1(C(=O)NC2C(NC(C34CC(C(N)=O)(OC3)C4)=O)CCC2)nc[nH]c2nccc1-2 C1(C(=O)NCC(=O)NCC(N2CCCC2CC)=O)(CN2CC=CC2)CC12CCC2 N1(C(C(CC)SC)=O)CCC2(CNC(=O)C(C)Sc3ncccn3)CCCCC12 C(=O)(C(C)(C)C(C)(F)F)NCC1C(C)CCN1C(=O)Cc1cnccc1Cl CC1(C(N2CC(CNC(C3(C)CCCO3)=O)C2)=O)CC1(F)F N1(C(CCC(C)SC)=O)CCC2(CC1)C(NC(=O)CC1CCC1)CS2(=O)=O c1(C(=O)NC(CC)CN(C(=O)Cc2ccsn2)C)cc(C2CCCO2)n(C)n1 c1(OC)cc(NC(C2(NC(=O)C(c3ccccc3)C)CC2)=O)cc(Cl)n1 C12(CNC(C(C)C3CCC3)=O)CC(CO1)N(C(=O)CCCCCF)C2 CCC(COC)C(=O)N(C(C)(C(=O)N(C1CCN(C(C)C)C1)C)C1CC1)C c1(SCC2(CSC)CC2)ccc2oc3ccccc3c2c1 Cc1ccsc1CC(=O)NC(CC1CC1)C(=O)NC(C)(C)CN1CCCC1 c1(C(c2nnnn2CCCF)NC(c2c(I)cnn2C)CCC)ccncc1C c1(C(=O)NC2C(C)(C)CN(C(=O)C(N)=O)CC2)ccc2ncccc2c1F C(N=c1[nH]c(Cl)nc2c1CSC2)C1CCCC(C(C)(C)CN2CCCC2)C1 N#CCCCCC(=O)N1CCCC(CCNC(=O)CSCc2cccs2)C1 N1(C(C2=CN(CC)CC2)=O)CC2OC(=O)N(C)C2C1.C12CCCCC1CNC2=O N12CC(C)(C)C1C2=O.C1(C)(CC=CCC)CCN1C(=O)OC(C)(C)C c1(OCC(=O)NC2COCC2NC(c2cc(O)cs2)=O)cc(F)cc(Cl)c1 C(c1ccc(F)nc1)=CC(=O)NCC1(F)CN(C(c2ccn(CCCC)n2)=O)C1 C(=O)(CC(C(F)(F)F)NC(c1cccc2c1CCC2)=O)N(C(C(C)SC)C)C C1(Nc2c(C)c(Br)ncc2)C2CC(O)C1N(C(=O)OC(C)(C)C)C2 CC1(C)CN(C(=O)CC2CN(C(c3cccc(=O)o3)=O)CC23CC3)CCCO1 C(=O)(C=CS(=O)(=O)CC)NC1C(CC)CN(C(=O)CCc2cc(OC)no2)CC1 N1(CC=C)C(=O)NC(c2oc(O)nc2O)C(C(=O)OCC)=C1c1ccc(F)cc1 Cc1[nH]c(=N)ccc1C=CC(=O)NCC1(O)CCN(C(=O)CCCCC(F)F)C1 c1(C(=O)NCC(CNC(C2N(C(CC)=O)CCCC2)=O)O)ccc(Cl)c(N)c1 C(=O)(CCCCC(C)=O)N1C(C(=O)NC(C=C)C)(COC)C=CC1 CC1CC(C(N2CC(N(C)C(c3cnn(C4CC4)c3)=O)C(O)C2)=O)CC(C)O1 C(=O)(C(C)(C)CS(C)(=O)=O)NCC1N(C(CCCC(=O)NCC)=O)CC(O)C1 c12cc(no1)CN2.C1(CC(=O)CCN(C(=O)CN)CCF)CCOC1.CO CC(C)C(C)CC(=O)NCCN(C(=O)COC1(C)CCCC1)CCCCO N1(C(C(CCF)NC(C2CC(SC)C2)=O)=O)CCC(C2CC2)C1 c1(NCCCN(C)C(=O)OC(C)(C)C)nc2cc[nH]c2c(=NCC=CCO)[nH]1 C1(c2nnnn2C2CCC(F)(F)CC2)(Cn2cc(CO)nn2)CC2C=CCC12 Cc1ccc2c(c1)CC(C(=O)NCC(O)CNC(c1cc(Br)nn1C)=O)S2 C(CC1=CCOCC1)NC(C1(NC(=O)Cc2ccno2)C(C)C1)=O C1(C(N(CC)Cc2cncn2C)=O)CC=CCN1C(=O)C1=COCC1 CC(C)C1=NOC(C(=O)NCC(=C2CN(C(=O)Cc3ccc(CO)cc3)C2)F)C1 C(=O)(C1=C(C)CCOC1)N1CCC(N(C(=O)CC2CCCCC2(C)C)CC#C)C1 c1(C(N(C2CCN(C(C=CC=CCC)=O)C2)CCC)=O)ccc(C)n1C CN1CCC(N(C(=O)C(N2CCCC(CN3CCOCC3)C2)=O)CC2CC2)CC1 N1(C(C(CC)F)=O)CC(C)C(C)(CNC(=O)CN2CC(=O)NC2=O)C1 C(=O)(CC(C(F)(F)F)n1ccnc1)NC(CNC(CNC(CCCCC)=O)=O)CC C(C(=O)NCc1ccnc(C)n1)(C(C)C)NC(CCC=CCC=C)=O C12(NC(CC3C(C)C3(F)F)=O)CC1CN(C(=O)CCC1CCN(C)CC1)C2 Cc1cc(C(N2CCC(C(=O)NCC3SCCS3)(C(C)C)C2)=O)nc(C)n1 C=CCCCC(C(=O)NCCCC1CCOC1=O)NC(C1OCCC1CC)=O N1(C(CCCC(=C)C)=O)CCCC2(CC(NC(=O)CSc3ccncc3)CO2)C1 C(=O)(C1CCc2nccn21)NC1(C(=O)NC(C2CCCC2)CC)CCCCC1 N1(C(C2NC(=O)OC2)=O)CCC(CO)(NC(c2cc3sccc3s2)=O)CC1 c1(OC)ccc(C(N2CC(CN(C)Cc3cn(C)nc3C)C2)=O)c(Br)n1 C(=O)(C1OCCc2c(Nc3ccnc4[nH]nnc34)cccc21)OC C1(CC(=O)N(C)CC2(NC(CN(C)CCO)=O)CC2)CCCCC12OCCO2 CCCC(CC)CCC(=O)NCCCCCC(=O)NC(c1ccc(O)nc1)C CCCC(CC(C)C)C(=O)N1CC2CN(C(C3CCc4ccccc4C3)=O)CC2C1 c1(CNC2(CC)CCOC2)ccccc1S(=O)(=O)N(C)C c1(C(=O)OC2(C#C)COC2)cnc2c(c1)c(C(F)(F)F)nn2C C(C(C)(C)C(=O)C(C)C)N(C1CCN(CCOC)CC1)C CCN=c1[nH]cc(C(=O)NCC(C)CN(C(=O)C(C)(C2CC2)OC)C)s1 CCCC(CC)CCC(=O)NC(C)C(C)(C)C(=O)NCc1cnc(C)cn1 C(=O)(CC(C)CC(=O)N(C)CCNC(=O)CCCOc1ccccc1)OC c1(C(=O)NC(C(=O)OCC)C2CC2)cncc(CNC(C2CCCOCC2)=O)c1 C1(NC(c2c(C)cccc2F)=O)CC2CCC(C1F)N2C(=O)CC1(O)CCOC1 N1(C(c2ccc(Cl)o2)C(=O)NC(CC)C)CCCC(c2cc(C)[nH]n2)C1 Cc1cc(=NC(C)CCNC(=O)C(=O)OC(C)(C)C)[nH]c(C)n1 N1(C(Cc2c(C)nn[nH]2)=O)CCC2(CC1)CCN(C(C1CCCC(F)C1)=O)C2 c1(C(=O)NC(C)CNC(=O)CCn2cnc(=N)[nH]2)c(S(C)(=O)=O)cnn1C C1(NC(CCC=CC)=O)CC2(NC(c3ncc(Br)cc3C)=O)COC1C2 c1(CC(N2CC(CNC(CCC(C)O)=O)N(C)CC2)=O)ccc2c(c1)CCCO2 C(C(=O)NC1CC1)(C(C)CC)N(C(CCC)CCO)C c1(C(N2CC(CC(N3CCCC(OC4CC4)C3)=O)OCC2)=O)cccc(C#N)c1 CC(C(=O)NCC1CC(O)CN1C(=O)CC1CC2C=CC1CC2)C(C)(F)F CC(CC(C)NCC(C(=O)CCCc1ccccc1)=O)N1CCCC1CCCO.N c1(C(=O)NCCN(C(c2n(CC)ncn2)=O)CC)cc2c(s1)COCC2 C1(COC)CC(C(=O)NCC(C)(CO)NC(C)=O)N(C(=O)OC(C)(C)C)C1 CN1CCN(C(c2cc(O)cc(Cl)c2)=O)CC1CNC(=O)C(C)(C)C1CCCO1 C1(C)(C(=O)NCC(C(=O)NC)O)CCN(C(=O)C(C)=C(C)C)CC1 c1(CNC(C2CC(OC)CN2C(=O)C(C)(C)CCF)=O)cc(C)cc(C)n1 c1(CC(=O)NC(CNC(CN2C(C)CCC2)=O)C2CCC2)nnc(S)nc1O Cc1[nH]nc2c(C(=O)N(C)CC3C4CN(C(C5COC(=O)N5)=O)CC34)cccc12 N1(C(CCc2ccc(OC)nc2)=O)CCN(C(c2sc(C)nc2C)=O)CC1CO C(=O)(CS(=O)(=O)C1CC1)NCC1CN(C(C(CC=C)(C)C)=O)CC1C c1(C(=O)NC(c2ncc[nH]2)CC)n[nH]c2c1CN(C(=O)CNC(=O)C(C)(C)C)C2 CC1CN(C(c2cc(I)cnc2Cl)=O)Cc2ccc(Br)cc2O1 c1(C(=O)NCCN(C(c2c(C)nc(C)o2)=O)C(C)C)c(C2CCC2)cccc1F C1(CC)(OC(C(=O)NC)(C)C)CN(C(C2CCC(C(N)=O)O2)=O)C1.OC C(=O)(CCCC#CC)N1CC(OCC)(COC)C1.C1(=O)C(CCF)N1 C1(NC(c2ncc(OC)nc2)=O)CCN(C(=O)CCc2cn[nH]c2)CC1F N1(C(C(CC)NC)=O)CCC2CN(C(c3cc(Cl)on3)=O)CC2CC1 c1(C(N2CCC(C)(CNC(C(C)CCO)=O)C2)=O)cnc2occc2c1 c1(CNC(C2OCCN(Cc3c(OC)cc(O)cc3)C2)=O)cc(C#N)ccc1Cl C#CC1(O)CCN(C(=O)C(C)=CCNC(C2(CC3CC3)CCOC2)=O)CC1 N1(C(c2ccc(C)s2)=O)CCCC2C(NC(=O)CCCCC(C)(C)C)C(C)(C)C12 CCCC(CNC(=O)C(CCSC)NC(=O)Cn1c(C)ccc1C)CCO N1(C(C(C)c2cccs2)=O)CC(c2nc(C3CC34CC4(F)F)no2)CCC1C N1(C(C(C)OCCOC)=O)CCN(C(=O)C2=NN(C3CC3)C(=O)CC2)CC2(CC2)C1 c1(CC(=O)NCC2C(NC(C(C)NC(C)=O)=O)CC2)cn2ccsc2n1 c1(OC)cc[n+]([O-])c(C(=O)NC2CCN(C(C3(CSC)CCCC3)=O)C2)c1 C#CCCCCCCC(=O)NC1CC(C)CN(C(=O)C(c2c(C)noc2C)C)C1 c1(C(=O)NC2CCC(NC(C(CC#C)O)=O)C2)ccnc2ccc(O)cc12 CC1CCN(C(c2cnc(N)c(N)c2)=O)C(C)C1NC(=O)C(O)C(C)(C)C N1(C(c2c(C)n[nH]c2)=O)CCCCC(NC(C2C=CC=CC=C2)=O)C1 C(=O)(CS(=O)(=O)CCO)N1CC(NC(C2CC(C(C)C)C2)=O)C(C)CC1 c1(C(N(CC(C)NC(C(C)CC(F)F)=O)C)=O)cn2c(n1)CCCC2 C1(CC=C)(C(=O)N(CC(CC)NC(=O)CN2CSCC2=O)C)CCCCC1 C1(C(=O)NC(C2CCN(C(C3(C#N)CC3C(C)C)=O)CC2)C)CCC(C)(C)CC1 c1(C(=O)NCCC2CCCN(C(C(C(C)C)OCC)=O)C2)cc2ncccc2[nH]1 C1(NC(C(C(C)O)(F)F)=O)CCN(C(=O)Cn2ccc(=O)n(C)c2=O)CC(O)C1 C1(F)(CNC(CN(S(CC)(=O)=O)C)=O)CC(NC(c2sccc2SC)=O)C1 N1(C(c2cc(COC)on2)=O)CC(NC(C2(C3(C)OCCO3)CC2)=O)CC(O)C1 C(=O)(C(c1ccccc1)=CC(C)(C)C)NCC1CC(NC(CCCC(=C)C)=O)C1 Cc1cc(Cl)ncc1S(=O)(=O)N1CCC(NC(c2ccc(F)c(F)c2)=O)C1 C1(C)(C(N2CCC(OC)C2)=O)CC(O)CN1C(=O)C=C1CCOCC1 C1(N(C(=O)C=CC=C(Cl)Cl)C)CCC(NC(=O)CCSC(F)(F)F)C1 C1(C(N(CC(c2ccccc2)O)C)=O)(NC(=O)CCSC)CCCC1 c1(C(=O)NCc2c(C(=O)NCC(C#C)CC)scc2)cnn2c1OCC2 c1(OC)cc2c(cc1Cl)CN(C(c1ccc(C)nc1C)=O)C2 C(=O)(CCCC(=O)NCC1CC(O)CN1C(=O)C(C)(C)NC(=O)OC)NCC C(=O)(C(O)CC(C)C)N1CC(F)(C(N2CCN(C(CC)C)CC2)=O)C1 CCCCC(CC(=O)N1CC(C(C)OC)C1)NC(=O)CC(O)CC(C)C N1(C(C(c2cnn(C)c2)C)=O)CC2CC(C(=O)NCc3cc(=O)cc[nH]3)C2C1 C12(COC)CCCCC1NC(C(=O)NCc1cccc(COC)c1)CC2 N1(C(C2(CCOC)CC2)=O)CCC2CN(CCNC(c3cccs3)=O)CC2CC1 CON(C(=O)C(C1CCCCC1)NC(=O)OC(C)(C)C)C(C)C c1(NC(C2C3CN(Cc4c(C)n(C)nc4)C2C3)=O)cc(Cl)ccc1I N1(C(CCCC(CC)NC(=O)C(C)(C)CF)=O)CC2(CCNC(=O)O2)C1 Cn1cccc(C(=O)Nc2ccccc2Oc2ccc(Cl)cc2)c1=O CCC(CCCC(=O)NC(CO)C(=O)N(C)C)NC(c1cc(C#N)cn1C)=O Cc1cc(F)c(CC(N2CC3(NC(=O)C=Cc4cocn4)CCC2C3)=O)cc1F C(CC(C)C(=O)NC(C)CCNC(c1cccc(CO)c1)=O)=COC C(CCCC)(CCC)NC(c1n(CCCCCC)nnn1)c1cnn[nH]1 C=CC(C)(C)C(=O)NC1CCC(CCNC(C2CCCCN2C(=O)C2CC2)=O)C1 N1(C(CSCC)=O)CCOC2CCN(C(c3cc(Br)ccn3)=O)CC12 C1(C(=O)O)CCS(=O)(=O)CC1.C1(COCCOCC)(C)CC1 C=CCCCCCC(=O)N(C)CC1CCCN1C(=O)Cn1cc(C=CC=C)cn1 O=C(CC1=CCOCC1)NCC1(CCNC(C2CN3CCC2CC3)=O)CC1 C(=O)(C(O)CC(F)(F)F)N1CCC(NC(C(C)(C)CCCl)=O)C(F)C1 Cc1ccc(Cl)c(F)c1C(=O)NCC1CN(C(=O)CC2OCCO2)C2(CCC2)C1 Cn1nc2c(c1-c1ccc(C3COC(=O)N3)s1)CN(CCN1CCCCCC1)CC2 c1(C(=O)NC(CC=C)CNC(C2CC2F)=O)cc2c(Cl)cncc2s1 N1(C(CC(C)(C)NC(CCC(C)OCC)=O)=O)CC2CCCC2C1 N1(C(c2occc2C2CC2)=O)CC2CCN(C(=O)NC3CC=CC3)CCC2C1 C=C1CCN(C(C2CC(O)C(F)C2)=O)C(C(=O)NCCC23CC(CCO2)C3)C1 c1(C(=O)NC(C(C(C)C)NC(=O)CN2CCS(=O)CC2)C)cc(F)c(F)c(F)c1 c1(CNC(C(C2CC2)SC)=O)cncc(C(=O)NC2CC23CCC3)c1 C#CCCCC(=O)NC1CCCC1NC(C1(CC(C)C)CCC1)=O C(=O)(CCCCCS(N)(=O)=O)NCC(CCNC(C(C)CO)=O)O N(C(=NCC(C)c1c(C)noc1C)NCc1cccnc1)C(COC)C N1(CCc2cn(CCCC(=O)NCc3c(C)nc(C)[nH]3)nn2)CCS(=O)(=O)CC1 Cc1ncc(C#N)c(N2CC3CC(NC(c4ccn(CC5CC5)c4C)=O)C3C2)n1 c1(N2CCN(C(=O)NC3CCc4cnnn4C3)CC2)cccc2ccccc12 c1(OC)ccc([N+](=O)[O-])cc1.c1(NC(C2CCCCO2)=O)ccc(C(C2CC2)O)cc1 C1(C(N(C(CNC(C(CC)OC)=O)C)C)=O)(CC)CCNC1=O c1(NCC)cncc(C(=O)NCCC2CCCCN2C(=O)CN2CC=CC2)c1 C1(NC(c2c(C)nsc2)=O)CCCCN(C(c2cccc(N)c2C(F)F)=O)C1 C1(NC(CCC(CC)C)=O)CC12CCC(NC(=O)Cn1cnnc1O)CC2 CCCC(C)(CC)C(=O)N1CCC(CCCNC(c2cn(C(C)C)nn2)=O)CC1 c1(CNC(C(c2ccc(C)s2)N(C)Cc2cccc(Cl)c2)=O)cc(Br)cnc1Cl C12(NC(c3scc(C)c3Cl)=O)CCCC(NC(=O)Cc3ccsc3)(C1)C2 CCCCCCCC(=O)N1CCC(C)C1CNC(=O)Cc1ccc(OC)cn1 C1(O)(CN(C(C(CC)c2ccccc2)=O)C)CCN(C(=O)C(CCO)N(C)C)CC1 c1(C(=O)NCc2cccc(CNC(C3C=CCCC3)=O)c2)cc2occc2[nH]1 C1(C(=O)N(C(C2CCCSC2)=O)Cc2cnnn2C2CC2)CCC(=C2CCC2)CC1 C1(CNC(=O)C=C2CCC2)CN(C(=O)Cc2cnc3ncccn23)CC12CCC2 c1(-n2c(C3CC34CC4)nc(C(CC)O)n2)cn2ccccc2n1 N1(C(c2c(C)scc2)=O)CC(C(=O)NC2CCNC(=O)CC2)C(F)(F)C1 C(=O)(C1CCNC(=O)CCO1)OC1CCN(C(CC)=O)CC1.C(C)(C)OC c1(OC)cc(C(=O)NC(C(=O)NCC2(CCO)CN(C)C2)C2CCCC2)sn1 c1(CC(N2C(C(=O)NCCN3C(=O)CNCC3)CSCC2)=O)cc(F)cc(F)c1F C=CCCCC(C(=O)N1CCC(c2cc(C#N)n(C)n2)C1C)NC(C)=O c1(SCC(N2C(CN(C(C(C(C)OC)O)=O)C)CC(F)C2)=O)nc(C)cc(C)n1 C=CC(C)(C)CCN=C(NCC(C)SC1CC1)NCC(C)C c1(NCCNc2n(CC)ncc2)nc(OC)cc(N2CC(C(N)=O)C3(CC3)C2)n1 c1(CNC(C2C(OCC)C2)=O)nc2c(s1)CN(C(c1csc(C)c1OC)=O)CC2 C1(C(=O)NC2(CNC(C(COC)C)=O)CC2)CCc2ccccc2CC1 Cc1nc(-c2ccc(Cl)cc2)sc1CNC(c1cc(Br)n(C)c1)C C1(C(=O)NCC(CCOC)NC(C2(C)CCC2)=O)CCc2cnn(C)c2C1 C12(C(=O)NC3CCC(N(C(c4c(C)nc(C)o4)=O)C)CC3)CCC(CC1)C(C)O2 C(=O)(C(CCS(N)=O)N(C)C(=O)OC(C)(C)C)N(C)C(n1cc(CC)nn1)C N1(C(C(CC(=C)Cl)NC(=O)CC2COCC(C)O2)=O)CCCCC2(CCC2)C1 C1(CC(C)NC(=O)C(N2CCC(CS(C)(=O)=O)C2)=O)COC(C)(C)O1 C1(C(=O)NCC(C)(C)OCCNC(c2cc(C)c(C)[nH]2)=O)C2CCCCCCC12 c1(CC)nnsc1C(=O)NCC1CCCN1C(C1CCN(S(C)(=O)=O)C1)=O c1(C(=O)NC(C2CN(CC3CCCCO3)CCS2)=O)ccnc2c1OCO2 Cc1c(C(=O)NCC(C2CCCC2)NC(=O)CC(=O)NCC)c(C)n2ccncc12 N1(C(c2cncc([N+](=O)[O-])c2)=O)CCC2CCCNC2C1 N1(C(CN(C(C)C)C)=O)CCCC2(C1)CN(C(=O)C(c1ccc(Cl)c(Cl)c1)C)C2 C#Cc1ccc(NC(C2CCN(C(=O)CC3C(C)(C)C3(C)C)CC2)=O)cc1 c1(C(N2CC(NC(C=C(CC)C)=O)CC23CCC3)=O)[nH]cc2c1CCS2(=O)=O Cc1cc(C(N2CCC(CCCn3cc(C(C)(C)OC(=N)O)nn3)C2)=O)ccn1 c1(CC(C)C)n[nH]c(=NC2CC(CNC(c3cccc(=O)n3C)=O)C2)s1 C(C(C)(C)CC(=O)NC1CC2CC1N(C(=O)CCNC(=O)NC1CC1)C2)N(C)C CC#CCCC(=O)NCCC1CCCCN1C(=O)CC1OCCCO1 C1(CNC(CC(=O)OC)=O)CN(C(c2ccoc2Cl)=O)C2COCC2O1 c1(OC)ccc(Cl)c(C(=O)Nc2cccnc2Sc2nc(C)cs2)n1 c1(CCC(=O)NC2CCC(NC(C3(CO)CCOC3)=O)C2)cccc(C(F)F)c1 C(C(=O)N1CCCC(CNC(CCCC)=O)C1)(C(F)(F)F)C(=O)N=c1cco[nH]1 Cc1cnc2cc(C(N3CC4CCCC4(CNC(=O)C(C)(F)F)C3)=O)nn2c1 c1(C(=O)NC2C(NC(c3cc(C)ncc3)=O)CCC2)cncc2c1CCNC2=O Cn1c(C(=O)NCCc2ccc(CNC(C3(C)CCOC3)=O)cc2)cnc1Cl CCC(C)(C)C(O)C(=O)NC(C1CN(C(=O)Cn2ccnc2C)CCO1)C C1(Cc2cn(C(C)C(N3CCC(CN4CCCC4=O)C3)=O)nn2)CC(C)(F)C1 C(=O)(C(F)CCC(C)(C)C)NCC1CN(C(C(CCC)(C)C)=O)CC(C)(C)C1 Cc1cccc(C(=O)NCC(C)(F)CNC(C2CC23CCC3)=O)n1 C1(CCC(=O)NC2CC(C(C)NC(CCOCCOC)=O)C2)CCCCO1 c1(OC(C(=O)NCC2CCC(NC(COCCC=C)=O)C2)C)ccc(F)cc1Cl C1(C(=O)NCC(CO)NC(c2ccc(C(C)C)c(Cl)c2)=O)CC2COCC(C1)C2 C1(C(N2CCCC(CCC=C)C2)=O)(C(=O)O)CCCNCC1 N1(C(C2(C)CC(C)C2)=O)CC(N(C(=O)Cc2ccc(F)cn2)C)C2(CC2)C1 c1(C(=O)NC2CCC(CCNC(c3ccc(CC)o3)=O)C2)cccc2occc12 C(C(CC(C)C)C(=O)NCc1nncn1C)NC(c1c(C)c(O)ccc1)=O N1(C(C2CN(CC)C(=O)C2)=O)CC2(CCC(NC(=O)CC3CC4CC4C3)CC2)C1 Cc1nn(C)c(N)c1C(=O)NC1CC(NC(=O)CSCc2ccncc2)C1 c1(C(=O)NCC2(OC)CN(C)C2)n[nH]c2c1CN(C(c1ccc(F)cc1O)=O)C2 Cn1cc(C(=O)NCC2CCN(C(C3(n4cncn4)CC3)=O)C2)c2ccccc12 C1(CC)CCN(C(C2CCCC2F)=O)C1CNC(c1ncccc1N)=O C1(NC(C2C(CC)N(C(=O)CCc3cc(C)no3)CC2)=O)CCOC2(CCC2)C1 N1(C(c2ccc(C)c(O)c2)=O)CCN(C(c2coc(C(F)F)c2)=O)CC(C)C1 c1(C(=O)NC2(CNC(c3cn(CC)nc3)=O)CC2)ccc(Br)c(OC)c1 C1(C(=O)NCC2(C)CCN(C(c3ccc(COC)cc3)=O)C2)CC(C)OC(C)C1 C(=O)(CC(C)(C(F)F)N(C)C)Nc1ccc(NC(C(C)n2ccnc2)=O)nc1.CC N1(C(CC=CC=C)=O)CC2(CCC2CNC(C2CN(C)CC2C(F)(F)F)=O)C1 N1(CC)CCCC(C)(CNC(=O)CCc2csnn2)C1 C(CNC(C1CCS(=O)(=O)N1)=O)(CC(F)(F)F)NC(c1c(N)cncc1)=O CCC(C)C(O)C(C)C(=O)N1CCC(C(=O)N2CC(C3CCCCC3)C2)=C(F)C1 C1(C(=O)NC(C)(C)CNC(C2(C(C)(F)F)CC2)=O)CCc2nnc(O)n2C1 Nc1ccccc1CC(N1CCC(CN2CCCCC2)C1)=O N1(C(COCCCCCC)=O)CC(CNC(C2C=CCCC2)=O)C(F)(F)C1 C1(CCNC(=O)Nc2c(C(C)C)cncc2)COc2ccccc2O1 N1(C(Cc2noc(C)c2C#N)=O)CCN(C(C2CCCC2O)=O)CCC1C C1(C(=O)NCC2CCN(C(C3N(C)CC(O)C3)=O)CC2)CCCCN1N=O C1(C)(CN(C)C)CCCN1C(=O)CC1CN(C(=O)OC(C)(C)C)C1(C)C C(C)(N=c1[nH]c(=N)c2[nH]cc(Br)c2[nH]1)C1C(C)CCCC1 c1(C(N(C2CCN(C(c3ccon3)=O)C2)CC)=O)csc2cc(Cl)cnc12 N1(C(C(C=CC)O)=O)C2COCC1CC(NC(C1(COC)CC=CC1)=O)C2 CCC(C)C(O)CC(=O)NC1CCC(C(=O)NCCOC(CC)CC)C1 C1(C(=O)NC2(C(=O)NC3C=CC(C(=O)NC)C3)CCCC2)COCCN1C C1(CC)(CC)CC(NC(=O)C(=O)NC2CC2)CN1C(c1ccccc1)=O C(=O)(CC(C)C(=O)N1CCOC(CCCNC(=O)C=Cc2cnc[nH]2)C1)OC C=CCCC(C)(C)C(=O)NCC(C1CC1)N(C(=O)C(C)N1CCC1)C N1(C(CN2C(C)CCC2)=O)CCC(N(C(=O)C(O)C2CC2)CCO)CC1 C1(C)(CC(=O)N(CC(C)NC(C2(CF)CC2)=O)C)CC1(F)Cl n1(CC(CC)C)ccc(=O)n(C(=O)c2ccc(F)cc2[N+](=O)[O-])c1=O N=C(CNOCC(F)(F)F)c1ccc(F)cc1F.C1C(=O)N1 C(=O)(CCCCCN(C(=O)CN1CCSCC1)C)N1CC(C#C)(F)C1 C12(C(=O)NC(CCC)C(=O)NC)CC(CO)(CN1C(=O)COCCCN(C)C)C2 C1(C(N(C(C)CN(C(=O)C(C)(C)N(C)C)C)C)=O)CC2(C1)CC1(CC1)C2 c1(C(N(C(CNC(CC=C)=O)C2CC2)C)=O)ccc(C)nc1C1CC1 N1(C(c2cccc3ncc(C)n32)=O)CCC2(CC1)COC(CNC(=O)C(F)F)C2 N1(C(C2(C)CC2c2cccc3ccccc23)=O)C2CCCC1CC(F)(F)C2 n1(C2(NC(C3N(c4nccc(OCC)n4)CCSC3)=O)CC2)cc(C)ccc1=O C1(CCC)(NC(=O)C(CC)OC)CCCN(C(c2nccc(OC)c2O)=O)C1 C1(C(=O)NCC(C)(C2CC2)NC(=O)CCCC2CC2)CCC(C(N)=O)O1 Cc1ccnc2sc(C(N3CC(C4CN(C(c5sccc5Cl)=O)C4)C3)=O)c(C)c12 Cc1cc(C(=O)N(CCCCCNC(C2(C#N)CC23CCC3)=O)C)cc(C)n1 CC1C(C)N(C)CCN1C(=O)CONC(=O)c1cnco1 c1(C(=O)NC(CNC(Cn2c(C=C)ncc2)=O)C2CC2)cc(C)c2n[nH]cc2c1 N1(C(c2c(CC)cc[nH]2)=O)CCN(C(C2CC(CF)C2)=O)C(CCOC)C1 N1(C(C2CN(C)C2)=O)CCC(CNC(c2cccc(C#N)c2F)=O)C(F)(F)CC1 c1(OC)ccc2c(C(=O)NC(CN3CCCC3)C(=O)O)ccnc2c1 N1(C(C(C(C)C)N)=O)CCOCC(C(=O)N(C)CCc2ncon2)C1 c1(C(=O)NC2C(NC(C3(C)CSC3)=O)CCC2)c(Cl)cccc1Cl C1(N(C(=O)COCc2nc[nH]n2)C)CN(C(=O)C(C)(C)CC2CC2)CC12CC2 c1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)c2ccsc2)cc2n(n1)CCCC2 C1(CC#C)(NC2CCC(c3cc[nH]n3)O2)CCN(C(=O)OC(C)(C)C)C1 C(=O)(CCCCC#N)N1CC(C=C)(CC(=O)NCC2CCCSC2)C1 c1(CNC(C)(CCC2CC2)c2nnnn2C2CCC2)cccc(C(F)F)c1F C1(NC(CC(C)NC(=O)NC)=O)CC2CC(CNC(=O)OC(C)(C)C)C2C1 Cc1cc(C)c(C(=O)NC(CNC(c2nn(C)c(C)c2Cl)=O)CO)cc1Br C#CCCN=C(NCC(C(C)C)c1ccccc1)NCC(C)(C)F N1(C(C(C(=C)Cl)(C)C)=O)CC(C)CN(C(=O)C=C2CC3CCC(C2)N3C)C(C)C1 c1(C(=O)NC(CC=C)CNC(=O)CCC2CCCO2)cccnc1OCCOC C(C(=O)NCC1CC2CC2N1C(=O)CN(C)C(C)C)(C(C)(C)C)SC N1(C(c2nccnc2OC)C(=O)NCCCC)CCCCC1CC C(C)(C)(C(C)CC(=O)N1CC(=O)NC2(CC2)C1)NC(C(C)OCC=C)=O C12(CC)CCN(CC1)C(=O)c1ccc(cn1)C1(CC1)C(=O)N2.C1(CC)CC1(C)C c1(C(=O)NCC(CN(C(CN(CCOC)C)=O)C)(C)C)cc(OC)ncc1Cl c1(C(N(CCNC(c2c(C)cc(N)cn2)=O)C)=O)cccc2nc(N(C)C)oc12 N1(CC=C)CCCC(CCC)C1.C1(=O)C(C)OCCOCCN1.C1CS1 N1(C(CCc2scc(C)c2)=O)CCC(c2cn(C3CC4CCC3C4)nn2)C(O)C1 c1(C(N(CCOCCCN(C(c2cc(C)no2)=O)C)C)=O)cccc2c[nH]nc12 Cc1cnc(NC(C(C2CCN(C(C3CCCOC3)=O)C2)C)=O)c(C)c1 c1(C(=O)NCCN(C(C(C)C)=O)C(C)C)cc2sc(Br)cc2s1 C1(NC(=O)NC2CC(CC(=O)OC)C2(C)C)CCn2c(O)nnc2C1 n1(CCC)ccnc1CNC(c1[nH]ccc1CNC(C1CCCC1C(N)=O)=O)=O C1(OC)CN(C(C2C3CN(C(=O)COC4CC=CC4)CC23)=O)CC1F N1(C(C(C(C)(C)C)=O)=O)CCCC2(C1)CN(C(c1cnc3ccsc3c1)=O)C2 c1(NCC(N2C(CCNC(C(COC)O)=O)CSCC2)=O)cc(F)cc(F)c1 C1(C(=O)OC)CCCC(NC(=O)C(Cn2cccn2)NC(C2CN(C)C(=O)N2)=O)C1 CC1CCc2nc(C(=O)NCC34CCC(NC(c5cnc[nH]5)=O)(CO3)C4)cn2C1 N1(C(CN(C(C=C(CCC)C)=O)C2CCC2)=O)CC(C)CC1CC C1(N(C(CCN(C(CCC)C)C)=O)C)CCCC(NC(c2ccc(CC)o2)=O)C1 C=C(C)CC(C)C(=O)N1CCC1CNC(=O)CCN(CCCCC)C c1(NC(c2cncc(NCc3c(C)cccc3Cl)c2)=O)cccc2c(I)n[nH]c12 N1(C(C(=O)NC)=O)CCC(C)C1c1ccccc1.c1(N2C(=O)CCC2)ccccc1C c1(CNC(C(CC=C)(C)C)=O)cnn2c1CN(C(c1coc(C(C)=O)c1)=O)CC2 CC(O)CCCCCC(=O)NCC1C2CN(CC3CCOC3=O)CC12 C1(CN(C)Cc2ccc(OCCC)cc2)Cc2cccc(C)c2O1 C1(O)(C(=O)OCC)CC(CNC(c2n[nH]cc2-c2ccncc2)=O)C1 CC1CC=C(C(=O)NCC(c2ccccc2)CNC(C2(C3CCC3)CC2)=O)CC1 c1(C(N(C2CCCCC2)CCNC(c2ccncc2O)=O)=O)ccc(O)nc1 CCCC(C)(CCC)C(=O)NCCC1CC(OC)CN1C(c1csc(CO)n1)=O C(CCN=c1[nH]cnc2c1COC2)OCCNC(c1ccc2c(O)nncc2c1)=O C1(NC(C(C)Sc2nncn2C)=O)COC2(C1)CN(C(c1cn(CC)nn1)=O)C2 Cc1nn(C)c(C)c1NC(=O)NC(=O)NCCCOC1(CCO)CS(=O)(=O)C1 C#CC1CN(C(C2CN(C)CCN2C(=O)CN2CCSCC2)=O)CC1O c1(C(=O)NCCCOCCCNC(CC(C)C)=O)cc(-n2cccc2)ccc1Cl c1(N2CC3CC(OC)C3C2)nc(=NCc2ccc(Cl)s2)[nH]c2c1CCCC2 c1(CNC(C2CCCN2C(=O)CC2=CCCC2)=O)ccc(O)cc1Cl c1(C(=O)NC(C)CNC(c2cnc[nH]2)=O)ccc(O)nn1 S(=O)(=O)(c1cnn(C)c1)NC(C(=O)NC1CCN(C(c2c(C)ccn2C)=O)C1)C Cc1cnc2c(C(N3CC(C)C(NC(c4cnsc4)=O)C(C)C3)=O)cccc2n1 N(C1COc2cc(Br)ccc21)C(c1cccc(S(C)=O)c1)C Cc1cc(CC(=O)NCC2(NC(c3cnn(C(C)C)c3)=O)CC2)on1 c1(NCc2ccc(C#N)cc2[N+](=O)[O-])cn2ccc(C3=CCC(O)CC3)cc2n1 C1(CC(N2C(CCCC)CCC2)=O)CN(C(=O)C(F)=C(C)COC)CCO1 C1(NC(C(C)Cc2cnn(C)c2)=O)C=CCN(C(N)=O)C1.C12(CCCC1)C(=O)N2 C1(NC(c2c(CCC)nco2)=O)CN(C(c2cc(Cl)ccc2C)=O)CC1(C)C Cc1ccc(OC(C)(C)CNc2cnn(C(F)(F)F)c2)c(C)c1 C(=O)(C1=CS(=O)CCC1)N1CC(N(C(c2c(Cl)cn(C)n2)=O)CCO)C1 C(=O)(C(O)C(C)C)NC(CNC(CCC)=O)C1CCC1.c12cccc(c1)S2 N1(C(C2CCN(C(=O)C(C3CCOCC3)O)C2)=O)CC2C3CCC(C3)C2C1 CC(C)(C(=O)NC(CC1CC1)CO)C1CCCN1C(=O)C=Cc1ccco1 CCCCC(C(=O)NCC(=O)NCc1cccnn1)C(C)C C1(C(=O)NCC#CCNC(CCc2cccc(OC)c2)=O)CC2(CCCO2)C1 N1(C(CC2N(C(C(C)CO)=O)CCOC2)=O)CC(CO)CC1(C)C c1(NC(C)CNC(=O)CCCC2CCCCC2)ncc([N+](=O)[O-])cc1F N1(C(C(C(=O)OC)OC)=O)C2CCC1CC(C(=O)NCC=CC(C)(C)C)C2 CC(O)C(C)CNC(C1(CNC(c2cc(CO)[nH]n2)=O)CCCC1)=O N1(C(CCCNC(c2ncn(CC)c2)=O)=O)CC2(CCCO2)C1 c12nc(oc1C)CNC1(CC(C)C1)CNC2=O.c1(C(=O)OC)nnsc1C C=C(C)c1cccc(NC(=O)CC(C2CC2)NC(=O)COCC2CCCO2)c1 CCC(C)CCC(=O)NC12COC(C1)C(NC(c1ccc(C(N)=O)c(Cl)c1)=O)C2 CN1CC(C)(NC(=O)C(O)C2CN(C(=O)C(C)(C)C3CCOC3)C2)CCC1=O CC1CC(CC(=O)NCCCC2CCCCC2)CN1C(c1coc(CO)c1)=O CCCC(CCC)=CC(=O)NC(C)(C)CC=CC(N1CCC(C)(O)C1)=O c1(C(=O)NCC2CC(O)(CNC(C(CC)C(C)C)=O)C2)cnc2nccnc2c1 c1(C(N(CCOC)CCNC(c2cn(C)nc2C)=O)=O)cn2cccc(Cl)c2n1 c1(C(C(N2CC(NC(Cc3cc(CC)no3)=O)C2)=O)=O)ccc(C2CCC2)cc1 c1(N(CC(=O)NC(C)(C)Cc2ccc(C(F)(F)F)cc2)C(C)=O)ccccc1Cl C1(C(=O)NCc2conc2C)(CNC(CCCOCCOC)=O)CC12CCC2 CC1C(NC(c2ccc(C3CC3)o2)=O)CCCN1C(c1cccnc1N(C)C)=O c1(COC)cc(C(N2CC(O)(CN(C(=O)CC3(C)CCC3)C)C2)=O)c(C)o1 C(=O)(CCCCC(F)F)NCc1cn(CC(C)NC2CC2c2cnn(C)c2)nn1 c1(CN2C(CNC(c3c(C)noc3C)=O)CCC2)ccc2ccn(C)c2c1 c1(C(=O)OC)nc(CNC(=O)OC(C)(C)C)oc1C.C12CC(O)CN1C(=O)N2 C1(CC(N2CC(c3nncn3C)C2)C)CN(C(C23CSCC2C3)=O)CCC1(C)C C1(OC)CN(C(c2c(Br)ncn2C)C(=O)NCc2ccc(F)cc2)C2(CCC2)C1 O(NC(=O)CN=c1nc(N2CCOC(CN(C)C)C2)c2c([nH]1)CSC2)CC N1(CC(=O)NCC(CNC(c2ccc(C(F)(F)F)nc2)=O)CO)CCOCC1=O CCC(C)(CC(=O)N1CCSCC1CCNC(=O)C(C)(C)CF)C(=O)OC C1(CNC(c2cc(Br)cs2)=O)CC(F)(F)CN1C(c1ccc[nH]1)=O C12(NC(C(Br)=C(C)C)=O)CC(C(F)(F)F)C1CN(C(c1ccco1)C1CC1)C2 C12(C(=O)OC)CCCC(C(N3CCN(C(C4CCCN4C)=O)CC3C)=O)(CC1)C2 CC1CCC(OCC(=O)NC(C)CCNC(c2cccnc2N)=O)CC1 C(=O)(C(CO)C(C)(C)C)NC1(CCOC)CCN(C(c2ccc(CCC)s2)=O)C1 CC1(C)OCC(C=CC(=O)NC2CC23CC(NC(c2cnc4sccn24)=O)C3)O1 C1(C(=O)NC(Cc2cccc(I)c2)CO)CC12CCN(C(=O)C(O)CCl)CC2 C(=O)(C(CN(C)C)C(C)C)NCC(C(=O)OC)NC(=O)CC12CCCC1C2 c1(C(=O)Nc2nc(C(=O)Nc3cc(C)ns3)n(C)c2)cc(I)cnc1Cl O=C(NNS(=O)(=O)N1CCOCC1)NCc1ccc(CCBr)cc1 C(=O)(C1=CCCC(C)(C)C1)N1C(CNC(C(C(C)C)C2CCC2)=O)CCCCC1 c1(CC(=O)NC2C(NC(Cc3c(C)ocn3)=O)COC2)cnccc1Cl c1(C(=O)NCC2(NC(c3nc(Br)c[nH]3)=O)CC2)nn2c(c1Br)CCC2 CC(C(=O)N(C1CCCN(C(c2cncs2)=O)C1)CCO)C1=CCCC1 C(C(C)(CO)CO)NC(C(c1cnn(C)c1)NC(c1c(C)ncs1)=O)=O c1(C(=O)NCCC(C)N(C(C(C)OC2CCCCC2)=O)C)c(N)cc(Cl)nc1Cl c1(C(=O)NCc2ccc(C(N3CCCC(SC)C3)=O)nc2)c(F)cncc1F N1(C(CN2CC(C)C2)=O)CCC2(CC1)CCN(C(C1CCN(C)S1(=O)=O)=O)C2 C(=O)(C1CCCc2cncn21)NC1(CO)CCN(C(C2(CC)CC2)=O)C1 C(c1cnc(O)nc1O)=CC(=O)NC1CCN(C(c2c(C)noc2C)=O)C(C)C1 Cc1c(Br)ccnc1C(=O)OC1CCCCC1C c1(-c2onc(C3CCC(O)CC3)n2)cc(Cl)cc(Cl)c1 C1(OC)CN(C(=O)C=C2CCCC2)C(C)(CNC(=O)C=Cc2ccc(Cl)s2)C1 C=CC(CCC)CC(=O)NCC1(NC(c2cc(F)cc(Cl)c2)=O)CCCCC1C C(C(C)(CC(C)C)NC(c1cc(C(=O)OC)ncc1F)=O)NC(C(F)=CC)=O CC(C)(C)C(CNC(c1c(N)cnn1C1CCCCO1)=O)NC(C1CC(O)C1)=O c1(NC(N2C3C(C)(CCC3)CCC2)=O)cc(S(N)(=O)=O)c(Cl)cc1Cl CC1C(NC(=O)C(c2ccc(F)cc2)=O)C(C)CCN1C(=O)CCC1CCCO1 C12=CC(=O)C(=CN1)N2.C1(NC2(c3n(CCC)nnn3)CCC2)CCCCC1CO C1(CC(=O)N(C2CCN(C(=O)CC3=CCCC3)C2)CCC)CCC(=O)NC1=O Cn1ccnc1CNC(=O)CC1(NCc2cnn(C3CC3)c2)CCC1 C1(=CC(=O)NCCCN(C(=O)CCN(C)C(C)=O)C(CC)C)CCOCC1 C1(C(=O)NCC(C2CCC2)NC(Cc2ccc(C)nc2)=O)CC2CCC1CC2 c1(C(N2CC(O)CC(NC(C(C=C)(C)C)=O)C2)=O)cc2c(o1)CCC(C)(C)C2=O C(=O)(CC(F)(F)C(F)(F)F)NC(CCCC)CNC(c1ncoc1C(C)C)=O N1(C(c2nc(CCC)sc2)=O)CCCCC1CCCNC(c1cnc(Cl)s1)=O c1cnc2cccc(Nc3cc(NC4CCn5ccnc54)ncn3)c2c1 C1(CNC(CCC#C)=O)CCCN(C(=O)C(C)OCc2ccc(C)cc2)C1 c1(CC(C)C(=O)N(CCCCCNC(c2cc[nH]n2)=O)C)ccc(F)cc1F CC(C)(C)C(C(=O)NCCCn1cc(C2CCCCO2)nn1)C1CCCCC1 C=C(Cl)CCC(=O)NCC1CCCCC1NC(c1ccn(-c2ccccc2)n1)=O N1(C(C=C(COC)C)=O)CCCC(NC(=O)CCOc2ccc(C)cc2)C1 N1(C(C(C)(C)NC(=O)C2=CCOC2)=O)CC(NC(C2CCCC2)=O)C2CCCC2C1 CC1(C)CN(C(C2(n3cccn3)CC2)=O)CCC1C(=O)N(CCC1CC1)C1CC1.C(C)=C c1(N(C(C(C)n2ccnc2)=O)CCO)ccc(C(C)C)cc1.C12CCN1C2=O N1(C(=O)C(CO)c2ccccc2)C2CCC1CN(C(C13CCC(F)(CC1)C3)=O)C2 c1(C(N(C2CCN(C(C3(F)CCS(=O)(=O)C3)=O)CC2)C)=O)cnn2cnnc2c1 C1(OC)CN(C(=O)C=Cc2ccoc2)CCC1NC(=O)Cc1ccnnc1O N1(C(c2cc(C(C)=O)[nH]n2)=O)CCCC1(C)C(=O)N(C1CC1C)C c1(NC(COC2CC(NC(C(C(CC)O)C)=O)C2)=O)ccc(F)c(F)c1C C1(CC(=O)NCc2ccco2)CCCN(CC(O)COC(F)(F)F)C1 C(=O)(C1CCCc2nncn21)NC1(C2CCN(C(CC(C)C3CCC3)=O)C2)CC1 c1(COC)cccc(-c2nc(C(F)F)nn2CCOc2ccccc2)c1 N1(C(COC(CC)(C)C)=O)CCC2(CC1)C(OC)CC2NC(=O)CC1=CCCC1 N1(Cc2nnc(C)s2)CCN(CC(N2CC(Cc3cc[nH]c3)C2)=O)CC1 C=CC1(C(N2C(CNC(C3CCc4cnnn4C3)=O)CC3CC23)=O)CCCCC1 C1(NC(C(c2c(C)nn(C)c2C)O)=O)CC2(CCCCN2C(c2cn[nH]c2)=O)C1 c1(CNC(=O)SCC(=O)NCCCC)cccc(Cl)c1CC.c1(S)cccnc1 N1(C(c2nc(CC)sc2)=O)CC2(CNC(C3CC(F)(F)CS3)=O)CCC1CC2 N1(C(C2(OCC)CCOC2)=O)CC2(CCCN(C(C3CC3F)=O)C2)C1 C=C(C)C(C)(O)C(=O)N(C1CN(C(=O)C(=O)NCCOCCO)CCO1)C CCCCC(O)CC(=O)N1CC(C(=O)NCCn2ncnn2)C(C)C1 CC12COCC1CN(C(=O)C1=CCC(NC(C3OC4CCC3C4)=O)C1)C2 C(=O)(C(C)(C)CC#N)N1C2CN(C(c3c(OC)cccc3)=O)CC21 c1(C(N2CCC(C(N3CC4C=CC4C3)=O)CC2)=O)n[nH]c2ccccc12 CCC1=NOC(CONC(=O)CC2CCCC2)C1.C(=O)CCC C(=O)(C1=NOC2(CCC2)C1)NC(CNC(C(c1ccccc1F)C)=O)CO c1(C(N(CCN(C(CC(n2ccc(C)n2)C)=O)C)C)=O)ccc(C(N)=O)cn1 Cc1cc(C(=O)N(CCNC(=O)CCC2(C#N)CCC2)C(C)C)ccc1F c1(CNC(C(=O)NC2C(C(C)C)OCC2)=O)sc(Br)nc1C c1(C(N2CCCC(NC(=O)CC3CCC3)CC2)=O)ccn2c1CCCC2 C(=O)(CC=C(Cl)Cl)N(C(C)C(=O)NCCSCCOC)CC#C C1(CC(=O)Nc2ccc(C(N3CCOCC3)CF)cc2)CSC2CCCC12 C1(C(N2CCC(OC)(CNC(=O)CC3CC(F)(F)C3)C2)=O)CC12CCCCC2 c1(C(N2CC(O)(C(C)NC(C(CC)n3cncn3)=O)C2)=O)cnc(N)cn1 CCC(CN(C)C)CC(=O)NCCN(C(=O)CCCC1CCCCC1)C Cc1cc(C)n(CC(=O)N(C2CC(NC(=O)C(C)NC=O)C2)C)n1 C1(NC(C(c2cccc(F)c2)C)=O)CCN(C(=O)Cc2ccn(C)n2)CC1(C)C c1(CC)cc(C(=O)NC(C)(CNC(=O)C(CC(C)C)N(C)C)CC(C)C)ccc1F c1(NC(C2N(Cc3c(OCC)cccc3F)CC(F)C2)=O)cn2ccccc2n1 CCCC(C(O)C(=O)N(C1(C)CC1)CC)NC(=O)COCCOCC C1(CSCC(=O)NCC(C)N(C(C2C(=C)CC2)=O)C)CCCCO1 N1(C(c2c(C)nn[nH]2)=O)CC2CC(C1)N(S(=O)(=O)c1cn[nH]c1)C2 n1(CCCC)ccc(C(=O)N(CCC(C)NC(=O)C(C)c2ccco2)C)n1 N1(C(C2=NOC(C)C2)=O)CCC2CCCC12C(=O)NCc1cccc(F)c1F n1(CC)cc(C(N2CC(c3cc(CNC(c4cc(Cl)ns4)=O)no3)C2)=O)c(C)n1 C1(F)(C(=O)NCCCNC(c2c(CCC)n(CCO)nc2)=O)CCCCCC1 C(=O)(NNC(=O)C(C)NC(=O)C1CC1)C1C(c2nc(C)sc2)OCC1 c1(NC(=O)OCC)ccc(NC(C2(N)CCCOC2)=O)cc1C c1(C(=O)NCC(C)NC(=O)Cc2ccccc2CC#N)cccc(O)c1F c1(NC(C23C(CN(C(c4ccc(CC)nc4)=O)C2)C3)=O)c(Cl)ccnc1Cl CCCC(O)C(CO)NC(=O)C(O)CCCNC(c1ccc(N)cn1)=O CCCCC(CC)C(=O)NCC1CN(C(=O)CCCC(=O)N(C)C)CCCO1 C#CC1(C(=O)NCC(O)CN(C(=O)C(C2(C3CCCC3)CC2)OC)C)CCCC1 c1(NC(c2n(CCOC)nnn2)(C)CCCl)cc(N=S(C)(C)=O)ccn1 c1(C(N2C(C(=O)NCCNC(CCC)=O)COCC2)=O)cccc2nccn12 C1(C(=O)NCC2CN(C(c3nc(C)sc3C)=O)C3C2C3)CCCC12CCOCC2 C#Cc1ncc(F)cc1NC(=O)C(N1CCCC1c1ccc(F)cc1)=O C1(NC(C2(N(C(c3c(C)n(C)cc3)=O)C3CC3)CCC2)=O)CC2CC1C(O)C2O c1(OC(C)(C)C)cccc(S(=O)(=O)N2CC(C(=O)O)C3CC23)c1 C1(NC(c2coc3c2COC3)=O)CCCC12CCN(C(C1CC3CC3C1)=O)CC2 N1(C(C=Cc2nc(C)sc2)=O)CCC(C2(NC(C34CC(C)C3C4)=O)CC2)CC1 C12(NC(C=CC(=O)N(C)C)=O)CC(NC(=O)C(F)C3CCC3)(C1)C2 c1(C(=O)NC(CC)CNC(c2ncc[nH]2)=O)cnc(NC2CC2)s1 C(=O)(C(F)CCC(C)(C)C)N1CCCC(CCC(=O)NCc2cn(CC)nc2)C1 N1(CC(=O)NCC2CC(NC(C(n3c(C)cc(C)n3)C)=O)C2)CCCCCC1=O C(N=c1[nH]c2cc(Cl)cc(Cl)c2o1)C1C(C)CCN(C(=O)CCCCCF)C1 CCCCC(CNC(c1cnc(Cl)s1)c1nnnn1CCC1CC1)CCC Cc1ccc(-c2cn(C3CC(NC(c4cccc(F)c4F)=O)C3)nn2)c(F)c1C C1(C(=O)OC)(NC(=O)C(F)(F)F)CC(N2CCCC(F)(F)C2)C(O)C1 C1(NC(C(C)OCCN(C)C)=O)CC2(C1)CC(NC(c1cc3n(n1)CCC3)=O)C2 c1(CC)nnc2n1CCCC2C(=O)N(CCNC(=O)C1=CCC1)CC c1(OC)ccccc1C(C)C(N1CCCC1C(=O)Nc1cnnn1C)=O c1(NC2CC(C=C)OCC2)cc(Br)ccc1S(=O)(=O)N1CC(C2CC2)OC(C)C1 c1(OC2(C(=O)NC3(CO)CN(C(COC)=O)C3)CC2)noc2c1COCC2 C(=O)(NNc1ncc(Br)cn1)Nc1c(OC(C)C)cc(F)cc1 C(CCCCC(=O)N(C)CC1CCCC2CC12)NC(CCc1onc(C)n1)=O C12(NC(c3c(C(C)C)ocn3)=O)CCCC1N(C(c1ccn(C)n1)=O)CC2 CC1C(C)N(C(c2cnc(N)c(Br)c2)=O)CCN1C(=O)CSc1n[nH]c(O)n1 CN1CCc2cc(C(=O)NCCC3CN(C(C4CCCNS4(=O)=O)=O)C3)sc2C1 C1(NC(CC2C(NC(CCCNC(C)=O)=O)CC2O)=O)CCC(=O)NC1(C)C N1(C(Cc2nc(=N)[nH][nH]2)=O)CC2(CCCC2NC(C2CCCC2O)=O)C1 C1(CNC(c2cccc(OC)n2)=O)CC2(CCC2)CN1C(C)C(N)=O C1(C(=O)NC2(CNC(c3coc(CO)c3)=O)CCC2)COCCN1CC(F)(F)F c1(OCC(=O)NCc2ccc(C(NOCCCCC)=O)o2)ccc(Cl)cc1 C=C(C)CCCC(=O)N1CC(CCNC(=O)Cc2coc(C)n2)C(C)C1 N1(C(c2c(C)c[nH]n2)=O)C2CC1CN(C(C1CCOC1C)=O)C2 c1(C(N2CCC(O)(CNC(c3c(C)n[nH]c3C)=O)CC2)=O)cnc2scc(C)n12 n1(CC(=O)NC(C(=O)N(CCC)CCN(C(C2CCC2)=O)CC)C)cnnc1O Cc1ccc(OCCC(=O)NCCNC(c2ccc(C#N)[nH]2)=O)c(C)c1 Cc1cc(Cl)ccc1OCC(=O)NCC1(C)CCN(C(C2CCOC(=O)N2)=O)C1 C12(OC)CC(C(N3CCCC3CNC(c3cccn3C)=O)=O)C(C1)C2 C1(C(C(=O)N(CC(CC)(C)OC)C)C)CCCN(C(=O)CN(C)C(N)=O)C1 c1(CCC)cc(C(=O)NCC23CC2CN(C(C2(C)CCOCC2)=O)C3)c(C)o1 CC1CCC=C1C(=O)NCCN(C)C(c1cnn(C2CC2(F)F)c1)=O c1(C(=O)NCC2OCCCN(C(C(=O)NCC)=O)C2)ccc2c(c1)CC(C)O2 N1(C(C(C2CC2)SC)=O)C(C(=O)N(CCCF)C)CCC1C1CCCC1 Cc1cc(C(c2nnnn2CCCC2CC2)NC(c2cnn(C)c2C)C)ncn1 c1(C(N(C(CNC(C2(CC=C)CCOC2)=O)C)C)=O)[nH]nc2ncc(Br)cc12 Cc1cc(C(N2CCC(CC(=O)NCC34CCCN3CCC4)CC2)=O)cc(O)c1 Cc1cc(C(C)NCC(c2ccccn2)C)sc1-c1cnn(C)c1 C1(C(N(C2CCN(C(c3ccc(C)nc3)=O)C2)CC)=O)CCC(=O)N1C C1(C)(C(N2CC(CCNC(c3nc(COC)[nH]n3)=O)(OC)C2)=O)CCN(C)C1=O N1(C(C2C(CC)C2)=O)CCCC(C2CCN(C(=O)C#CC3(C)CCCO3)CC2)C1 CC1CCn2cc(C(=O)NCCC3CCC4(CCC4)O3)nc2C1 c1(C(N2CCC(O)(C(C)NC(C(C(CC)O)C)=O)C2)=O)cc(F)c(F)cc1Cl c1(C(=O)NC(C(C)(C)NC(c2c(C)n[nH]c2C)=O)C)cc(Cl)c(F)c(Cl)c1 C(=O)(C(CC(C)C)NC(C1CC1CF)=O)N1CC(NC(=O)OC)C1.C=O C1(C(N(C(C=C)C)C)=O)(CNC(=O)C(C)c2ccsc2)CC12CCC2 C12(C(CC)=O)CC(C(=O)N(C)Cc3cscn3)(C1)C2 c1(C(C)=O)cc(C(=O)N(CC(C)(C)CNC(c2cscc2C)=O)C)oc1C N1(C(C(c2ncc(CC)o2)(C)C)=O)CC2CC3CC2C1C3NC(c1cscc1C)=O CC1(C)CN(C(C2CCC3CCC2N3C(=O)C2=CCSC2)=O)C12CCC2 N12CC3CC3C1C(=O)NC(CC)C2=O.C(CCCN(CC)CC)OCC C1(NC(=O)COc2ccon2)COC2(CCCN(C(c3csc(S)n3)=O)C2)C1 S(=O)(=O)(c1ccc(=NCCN2CC(C)CC(C)C2)[nH]c1)NCc1c(C)cccn1 C(=O)(C(C)CCCc1ccc(N)cc1)N1C(CNC(CCNC(=O)OC)=O)CC1 N1(C(CSCCC)=O)CC(NC(C2Cc3ccncc3C2)=O)CC12CCCCC2 N1(C(C(=O)NCC2CC2)=O)CC2CCC2(CCNC(c2ccnnc2O)=O)C1 CN1C(=O)CN(CC(=O)NC2CN(C(C3(O)CC3)=O)CCC2CO)C1=O C(=O)(CCCCCF)NCc1c(C2CCN(C(C3C(=C)CC3)=O)C2)n[nH]c1 C=CCCCCC(=O)NCc1nc(CNC(C2CC2(C)C)=O)cs1 n1(CC(N2CC(CNC(=O)CCc3csnn3)C(O)C2)=O)cnc([N+](=O)[O-])c1 c1(CCC)nc(C(=O)NCC=CCC(=O)N(C(C)CC)CCOC)co1 C1(C(N2CCCC(NC(c3cccc4sccc34)=O)C2)=O)CCCCC1C1CC1 N1(C(C2N(C(C=C(CCC)C)=O)CC(O)C2)=O)CC2CN(C)CC2C1 C(=O)(C1=CC2(CN(C(=O)CC3(C)CCCCC3)C2)OC1)NC1CC(C)OC1=O C1(CNC(COCCC)=O)COCC1NC(c1cc(Cc2ccccc2)c[nH]1)=O C(=O)(C1Cc2ccc(C)cc21)NCCC(C)NC(c1ccc(SC)cn1)=O C1(C(=O)NC(CCC)CO)CCCN(C(c2cc(Cl)n(C)n2)=O)C1 C12(C(N(CC(C)NC(=O)Cc3ccc(C4CC4)cc3)C)=O)CCC(CC1)CO2 N1(C(c2cc(CCOC)on2)=O)CC(F)CC1CN(C(=O)C=CC(C)(C)C)C Cc1c[nH]cc(C(=O)NC(c2ccccc2)c2cn(C)nn2)c1=O c1(C(=O)NCCCS(C)(=O)=O)c(-c2ccc3ncoc3c2)ccc2c1OCO2 C(=O)(C(C(C)O)N(C)C)N(CCCNC(=O)CN(C1CCC1)C(C)=O)CC c1(CNc2c(C(N3CCC(C#N)C3)=O)cc(Cl)nc2)ccc(Br)c(F)c1F c1(C(=O)NC2C(C(=O)NCCNC(N(C)C)=O)COC2)cnc2n1CCC2 c1(C(=O)Nc2c(C(=O)OC)ccc(OC(F)F)c2)ccc(C)c(F)c1O N1(C(CC2CCCN(C(C3C(C)=CCS3)=O)CC2)=O)CC2CCCCC2C1C CC(C)(C)CCC(=O)NC1CCC(NC(C2(C(C)(C)C)CCCC2)=O)C1 c1(C(=O)NC(CCC)C(=O)NCC(C)(C)C(C)C)ccc(O)c(F)c1 N1(C(=O)NC2CCCC2F)CCCN(C(=O)C(c2ccccc2)C2CC2)CC1 Cc1cc2sc(C(N3CCOC(CNC(C4C=CCC4)=O)C3)=O)cc2s1 CCC(C)(C)C(C)CC(=O)N1CCC(C)(CNC(=O)C=C(C)c2cccs2)C1 c1(Oc2cccc(NC(C=COC(C)=O)=O)c2)ccccc1[N+](=O)[O-] C1(C(=O)NCCCCNC(c2c(C(C)C)nns2)=O)CCCC2CCCN12 c1(C(=O)NC(CC)C(=O)NCCC(C)O)oc(C)cc1C C1(C(=O)NC2CCN(C(CC(C)(F)F)=O)CC2O)Cc2ccccc2C1 N1(C(C2C(CCOC)C2)=O)CCCN(C(=O)C(C)n2cncn2)CC1 c1(C(N2CCCC(n3cc(COC)nn3)C2C)=O)c2c(nn1C)CCC2 Cc1c(NC(C2CCC=CC2NC(=O)Cn2cncn2)=O)cccc1C(=O)O CC(C(=O)NCCCN(C(=O)CC1CC(=O)NC(=O)C1)CCO)S(C)(=O)=O C1(C(N2CCC(N(CC#C)C(C3CC(C)CO3)=O)CC2)=O)Cc2ccccc2C1 C1(CNC(C2N(CC)CCC2)=O)CC2(CCN(C(C3(C4CC4)CC(=O)C3)=O)C2)C1 c1(NC2CCC(OCC)CC2)nccc(=NC2COCC2C2CC2)[nH]1 N1(C(c2c(CCCC)ocn2)=O)CC(NC(=O)Cn2cccnc2=O)C(O)C1 Cc1[nH][nH]c2ncnc(=NC3CCC(NC(C4CC5(CCCC5)CO4)=O)CC3)c1-2 C12(CNC(C(C)Cn3cccn3)=O)CC(CO)(CN1C(C1CC(=O)C1)=O)C2 Cc1c(Br)ccc(N2CC(CNC(C3(O)CCSC3)=O)OC(C)(C)C2)c1[N+](=O)[O-] C(=O)(C1=CCCCCC1)NC(C1CCOC1)CNC(c1ccc(C)n1C)=O N1(C(C(Cc2c(C)noc2C)C)=O)CCCCC(NC(=O)Cc2cncn2C)C1 c1(C(=O)OC)ccc(C(=O)N(C)CCN(C(=O)CC2CC3COCC23)C)cc1Cl N1(C(C)CNC(=O)N(C(C)Cc2ccc(C#N)cc2)C)CCc2ccccc21 C1(C)(CNC(C(C)(C)OCC)=O)COCCN(C(C2(CSC)CC2)=O)C1 c1(CC(N2CCCC(CNC(C(C(C)C)(C)C)=O)C2)=O)ccc2c(c1)CCCC2 c1(C(N2CCCN(C(C(C=C)O)=O)C(C)C2)=O)oc2c(F)cccc2c1C C1(C)(CNC(C=NOC)=O)CC(F)(F)CN1C(c1cc(C(=O)OC)c[nH]1)=O C1(C(=O)OCC)(C(=O)NCCN(C)C(c2cc(CC)c(C)[nH]2)=O)CC1S(C)(=O)=O C=CC1CN(C(=O)CCCC(C)NC(C2(OC)CCOC2)=O)CCO1 Cc1cc(F)c(C(=O)NCC2(CNC(c3[nH]nc4ncccc34)=O)CC2)cc1Br c1(N(C(=O)C(=O)NCC(C)Cn2ccnc2)CCOC)cccc(F)c1 c1(N(C)C(C2CCCC(=O)C2)=O)cc(N2CCCCC2)cc(F)c1 C(C)(C)(CC(=O)OC1(CCO)CN(C(=O)CN(c2ccncc2)C)C1)OC c1(OC)c(C)csc1C(=O)N(C)CCOCCSc1ccnc(C)n1 C(=O)(C#CC1CCC1)NCC1CCC(F)(CNC(C(c2ccccc2Cl)C)=O)C1 Nc1cc(F)c(C(N2CC(NC(c3cnc(C(F)(F)F)o3)=O)C(F)C2)=O)cc1F N1(C(c2csc(C)c2)C(=O)Nc2ccc(OC)cc2C)CCN2CCCCC1C2 CC(C)(C(=O)NC1CCc2ncnn2C1)C1=CCN(C(C2CSCC(=O)N2)=O)C1 N1(C(c2n[nH]c(C)c2F)=O)CCCC2C1CCN2C(c1cc(Cl)cc(Cl)c1)=O c1(OC)cc(C)ccc1C(N1CCC(C)(NC(C2COC(=O)O2)=O)C1)=O c1(C(=O)NC2C=CCN(C(c3ccc(NC)c(F)c3)=O)C2)cnn2c1CCCC2 C1(C)(CNC(CCN(CCCCC)C)=O)CCCC1NC(=O)CCCOC O=C(N=c1[nH]oc2ccncc2c1=O)C1C=CC1=Cc1cccc([N+](=O)[O-])c1 c1(C(=O)NC(CN(C(c2cnc(CCC)s2)=O)C)C)nccc(Br)c1O C1(C(C)NC(c2csc(C3CC3)c2)=O)CCCCN1C(c1nn(C)cc1N)=O N1(C(C2CCN(C(c3c(C)c(F)ccc3)=O)CC2C)=O)CCc2cc(C#N)ccc21 N1(C(C)=O)CCCC1C(=O)NC1(CNC(c2cncs2)=O)CCC1 S(=O)(=O)(c1cnc(Cl)nc1)N1Cn2c(-c3c(SC)nc(NC(=O)OC)cc3)cnc2C1.OC C1(C)(OC(C=COc2ccc(OC)cc2)=O)CCC(=O)CC1 C(=O)(C1CCOc2ccccc21)NC1(CC=C)CCN(C(c2nonc2N)=O)C1 c1(C(=O)NCC2CCN2C(C2(C3CC3)CCCO2)=O)ccc(-c2cscn2)nc1 c1(C(=O)NCC(C)(CO)NC(=O)CC2CCOC2)cn2c(n1)CCCC2 c1(C(=O)NCCC(C)NC(C(C(C)C)OCC)=O)c(C)ccc(F)c1Br CC(C)C(F)C(=O)NCC(C1CCCC1)NC(c1cn(C)nn1)=O C1(C2(O)CN(C(c3cnsc3)=O)C2)(CNC(C2(C(C)(C)C)CCCCC2)=O)CC1 c1(CCCNC(N2CC(O)(C3CC3)C2)=O)cncc2ccccc12 N1(C(c2cn(CC=C)nc2)=O)CCC=CC1C(=O)NCc1nnc(O)n1C C(=O)(C(F)(F)c1nc(C)cs1)NCCN(C(=O)CC1(CO)CC1)CC C12(NC(C(COC)C)=O)CCC(CN(C(c3csc4nnsc34)=O)C1)C2 N1(C(C2C(CC)C2)=O)CCCC1C1CCCCN1C(=O)Cc1ccnc(C)c1 N1(C(C(C(C)NC(CCC(C)C)=O)C)=O)CCc2nncn2CC1 N1(C(C2C(C)C2C)=O)CC(F)(F)CC1(C)CNC(C1CCC(F)CC1)=O c1(C(=O)NC(C(=O)N(C(C=C)C2CC2)C)c2ccco2)nnc(S)n1C c1(OC)ccc2c(c1)CCC(NC(=O)N(C)CC1(C(C)C)CCC1)C2 c1(COCCSC)ccc(C(=O)NCCCNC(c2ncccn2)=O)o1.OC Cn1ncc(C(=O)NC2CCCC2NC(c2cc3occc3s2)=O)c1C#N Cc1c(C(c2nnnn2CCCF)NCC2(n3cccn3)CCC2)cncc1Br c1(OC)cc(C(=O)NCCC(C)(C)NC(c2cc(C(F)F)on2)=O)ncn1 C1(C(C)C)CN(C(=O)C(F)C2CCCC2)CC1C(=O)NCCC(C)CO Cc1cccc2cc(C(=O)NC3CCC(NC(C4CCCCNC4=O)=O)C3)oc12 CC(C(C)(C)C(=O)N1CC2(CC=CC2)C1)NC(=O)CC1CC=CCN1C C1(CC)CNC(=O)CN1C(=O)CC1C(NC(c2cc(OC)no2)=O)CC1O c1(C(=O)OCC)ccc(C(=O)N(C)CC2OCCC2(C)C)nc1C N1(C(CCN(C(C)=O)C)=O)CC2CC(NC(C3CC(C)CC(C)(C)C3)=O)C(C2)C1 N1(C(C2N(C(C(CC3CC3)OC)=O)C3C(C2)C3)=O)CC(=O)NC(C(C)C)C1 c1(NC(CCN(C(c2c[nH]c(=NC)o2)=O)CC)=O)cc(O)ncc1F c1(C(=O)NCC(N(C(C=CC(CC)=CC)=O)C)C2CC2)ccc(F)c(O)c1F N(C(=NCC1C2CCC12c1ccccc1)NC(CC)CC)C1CCN(CCC)C1 c1(CC)cc(C(=O)NC2CCC(NC(=O)CCCc3nc(C)cs3)C2)cc(N)c1 C1(COC)(NC(=O)COC)CCN(C(=O)Cc2cccc(N)c2F)CC1 N1(C(C(C2CCCC2)OCC)=O)CCCCC1CNC(c1cccs1)=O CC(C(=O)NCCCN(C(=O)CCNS(=O)(=O)C(F)(F)F)C1CC1)C(F)F C1(NC(c2c(OC(C)C)cccn2)=O)CN(C(=O)CCOCC2CCC2)CC1(C)C CC(C)C1CCC(=O)NC(COC(C)C(C)C)Nc2c(cccc2Cl)C(=O)N1 c1(CNC(c2cn(C)nn2)CC)ccc(F)nc1 c1(OC)nccc2c(C(=O)NCC(C)NC(=O)Cc3ccc(C)c(C)c3)c[nH]c12 c1(C(=O)NCC(C(C)C)NC(=O)C(c2ccccc2)O)cc(Cl)ncc1N C(CC(C(=O)NCC1(C(C)C)CCCC1)NC(=O)Cc1c(C)n[nH]c1C)OC N1(C(c2nc(CCC)sc2)=O)CCC2C(CCCN2C(=O)C(C(C)C)C(C)C)C1 c1(C(N2CCC(N(C(c3cc(C)nnc3C)=O)CC)C2)=O)ccc(C)c(C)c1N N1(C(C(C)OCCCC)=O)CCCC(F)(C(=O)NCc2ncnn2C2CC2)C1 C(=O)(C(C)P(C)(C)=O)Nc1c(C)cc(CNC(C(C(C)C)NC(C)=O)=O)o1 C1(NC(C2C(CC(C)(C)C)C2)=O)CCC2(CCN(C(=O)CCF)CC2)C1 c1(C(=O)NCCCN(C(C(C(C)C)N(CC)CC)=O)C2CC2)cc2ccccn2n1 C(C)(C)(CCC(=O)N1CCC=CC1C(=O)Nc1ccc(F)cc1C)OC n1(CC)c(C)cc(C(=O)NCCCCN(C(=O)C(N2CCC(C)C2)=O)C)c1C C1(C2CCN(C(c3ccn(-c4cccnc4)n3)=O)CC2)(NC(C2(Cl)CC2)=O)CC1 n1(CC)nc(C(=O)NC2CC2CNC(c2cnc(O)c(F)c2)=O)ccc1=O c1(C(=O)NC2CCC(NC(CCSCCC)=O)CC2)cc(F)c(C)cc1F C1(NC(CCN(C)CCO)=O)CC2CC1N(C(c1nc(=O)n(C)[nH]1)=O)C2 c1(CCNC(c2c(CNC(CC(C)OC)=O)occ2)=O)ccncc1C C=CCCC(C(=O)N(C)CC1(O)CCCC1)NC(c1cc(C)cc(C)n1)=O C(=O)(CCCC(=O)NCC1C(C)CCN1C(=O)COC1CCCC1)OCC c1(C(=O)Nc2c(C)cc(OC)c(Br)c2)cc(Cl)nn2ccnc12 CC1(C)CN(C(=O)Cn2cccn2)C(CNC(=O)CCN2CCOCC2)CO1 c1(C(N2CC(C)C(CNC(C3C=CCC3)=O)CC2)=O)cc2cc(F)ccc2[nH]1 Cc1nccc(C(=O)NC(CNC(=O)Cc2cccnc2C(F)(F)F)C(C)C)n1 c12ncnc3c1ncn3CCC1CN2C1.Cn1cc(C(C)NC(CC(F)(F)F)=O)cn1 c1(OCC)cccc(C(=O)N(CCCCN(C(=O)CCOC(C)=O)C)C)c1N C(CC(C)(F)F)NC(C(C1CCN(C(=O)CN(C)C2CC2)C1)C)=O C1(C(C)C)CN(C(C2CCC3CCC(=O)N23)=O)CCCN1C(=O)CN1CC=CC1 C1(C(N2CC(CCCCNC(C(c3ccccc3)SC)=O)C2)=O)CCOCC1(C)C C1(NC(c2c(OC)nsc2)=O)CCC2CN(C(c3cccc4c3CCN4)=O)CC2C1 N1(C(C(C)=CC)=O)CCCC2CN(C(=O)CC(C(F)(F)F)OC)CC12 C1(CC(=O)N(CC(C)O)CCNC(=O)C2=CCOC2)(OC)CCOCC1 c1(C(N2CCC(NC(COCCC=C)=O)CC2C)=O)cc(C)c(Cl)cc1C CC1(C)CC(NC(=O)COc2ccc(N)cc2)CN1C(C1CCCS1(=O)=O)=O N1(C(c2cc(CC)n(C)n2)=O)CCC2CC2(C(N2CC(N(C)CC)C2)=O)CC1 S(=O)(=O)(CC(=O)NCCC(C(C)C)NC(=O)CN(CC(=O)N(C)C)C)NC c1(NC(C2CC(C)CN2Cc2ccccc2OC(=N)O)=O)cc(Cl)c(F)c(Cl)c1 C1(NC(CNC(CC)=O)=O)CC2CN(C(C3(CC)CCNC3=O)=O)CC2C1 c1(NC(C2C3(CCN(C(C=COCC)=O)C3)C2)=O)cc(C)cc(Br)c1F c1(OCCNC2CCCN(C(CC(C=C)CCC)=O)C2)ccc2ccccc2c1 C1(CC(=O)OC)(NC(C2CC2C(C)C)=O)CCN(C(=O)Cc2ccc(C)nc2)C1 N1(C(CN(CC(C)C)C(C2CC23CCCCC3)=O)=O)CC(C)CCC1C c1(CC)onc(C)c1C(=O)NCCCC(C)NC(=O)CC1CCCC1OCC C12(NC(C3CCN(C(CCC)=O)C3)=O)CC1CN(C(=O)CCCc1nccs1)C2 C1(C(=O)NC2C(NC(CNC(=O)OC(C)(C)C)=O)C2)(CO)CC(F)(F)C1 N1(C(C(Cn2cncn2)NC(Cn2c(C)ccn2)=O)=O)CCCOCC1 Cc1cnc(C(=O)NC2C3CC2N(C(=O)Cc2cnc(C)[nH]2)C3)c(Br)c1 N1(C(CCCCC#C)=O)CC2(CCCC2)C1C(=O)NCC1(CC)CCCCO1 Cc1ccc(C(=O)NC(C2CCN(C(C3OCCC3(C)C)=O)C2)(C)C)cc1CO c1(N)ccccc1.CCC(CNC(CC(C=O)C)=O)N(C(=O)C(F)=CCCF)C c1(CNC(CN(C(=O)NC(CCC)CO)C)=O)nc(COC)no1 C12(C(N3CC(CNC(c4ccc(CC)s4)=O)(CC)C3)=O)CC3CC1C2C3O N1(C(c2c(C#C)cnn2C)=O)Cc2ccnn2CC(NC(C23CCCC2C3)=O)C1 N1(C(c2c(COC)nn(C)c2)=O)CC2CCC1CC2NC(c1cc(OC)ns1)=O C1(NC(=O)NC(CC)COC(F)(F)F)(COC)CC12CCOCC2 CCC1=NOC(C(=O)NC2CC(NC(=O)CC(C)c3ccccc3)C2)C1 c1(C(N(c2cccc(C)c2)C(=O)CN2CCC3CC23)=O)cncc2ccccc12 c1(C(CO)N)ccccn1.C1CC(=O)NCCCN1C(=O)CC1CCC1C.CO c1(C(N2C(CN(C)C(c3ccc[nH]3)=O)CCC2)=O)c(F)cc(Cl)cc1F CC(C(=O)NCC1CC(C)CN(C(=O)CCN2CCCCC2)C1)C(F)(F)C(F)F C1(CNC(C(CC)N(CC)CC)=O)C2CCN(C(=O)C(C)C3=CCCC3)CC12 N1(C(CC2(C=C)CCC2)=O)CC2COCCC2(NC(=O)CN2C(=O)CCC2=O)C1 C1(C(N(CC(=O)NC2CC2)C)=O)C(C)CN1C(=O)CC(=O)N(C)C c1(CC)cc(F)ccc1C(=O)NC1CCCN(c2cc(OC)ncn2)C1C c1(C(=O)NCC2(CNC(C3CC(C(C)C)OCC3)=O)CCC2)cc2ncccc2o1 c1(CC(=O)NC2CC(NC(c3[nH]n(C)c(=O)n3)=O)CC2O)ccccc1S(C)=O C1(NC(Cn2c(C)ccn2)=O)CC(NC(c2ccc(CN(C)C)s2)=O)C1(C)C CC1CN(C(=O)CN2C(=O)CCC2=O)CCCN1C(=O)Cc1n[nH]c(=N)s1 Cc1cc(C(N2CCC(C)(CNC(C34CC3CNC4=O)=O)C2)=O)nc(O)n1 n1(CC(=O)NC2(C)CN(C(=O)Cc3nnc(O)s3)C2)cc(S(N)(=O)=O)cn1 Cc1cc(Cl)ccc1C(=O)NCC(O)CCNC(=O)CCn1cncn1 N1(C(CCOCC(C)C)=O)CC=CC1CNC(C12CC(C1)C2)=O Cc1ccc(C(N2CCC2C(N2CCCC(CC3CC3)C2)=O)=O)c(O)c1 CC(C(F)C(=O)N1CC(NC(c2ccc(CC(N)=O)cc2)=O)CC1C)C(F)(F)F N1(C(Cc2c(C)nc(C3CC3)s2)=O)CC(C)C(NC(c2csc(C#N)c2)=O)C(C)C1 N1(C(CC(C)=C(C)C)=O)C(C(=O)NCC(C)CC(C)O)C2CC(O)C1C2 n1(CCC(=O)NCC(CO)NC(C2CCN(OC)CC2)=O)ncc2c1CCCC2 c1(NC(=O)C=Cc2cccc(F)c2)cc2cccnc2c2ccccc12 C1(C)(NC(=O)OC(C)(C)C)CCCCCCC1.N12CCCC1CN(CC(C)O)C2=O C(=O)(C(C(C)C)c1cnn(C)c1)NCC1(C(C)NC(c2c(CC)nco2)=O)CC1 C(=O)(C(C)(C)S(C)(=O)=O)NC1CN(C(CCN(C(CCC)C)C)=O)CC(F)C1 C(CC(N)=O)(C(=O)N1CCC(OCCF)C1)NC(c1c(CC)nc(C)o1)=O N1(C(C2(CNC(C(C(C)C)OCC)=O)CCCO2)=O)CCN2CC(O)CC2C1 C#Cc1ccc(C(=O)NC(C)(C)CN2CCN(C(=O)CC3OCCC3C)CC2)cn1 C(=O)(C1COc2ccccc21)N1CCN(C)CC1CNC(=O)CCOC1COC1 c1(CNC(c2cn(C)nc2CC)c2n(CC=C)nnn2)ccc(C#N)cc1 CCCC(C(=O)NC1CCCC1(C)CNC(c1cc(C(C)C)n(C)n1)=O)C(C)C C12(F)CCCN(C1)C2=O.c1(CNC(=O)CNC(=O)C2CC2)cccc(F)c1Cl N1(C(CC(C)N(C)C(C2CCSCC2)=O)=O)CCC2(CC1)N=N2 CC(C)C(C(=O)NCC1CC1CNC(=O)C1=CCC1)C1CCC1 C(c1ccccc1C)=CC(=O)NC(C(C(=O)NCCCOC)C)C C#Cc1cnc(C(=O)NC2CC2CNC(=O)C(C)(C(C)C)NC(C)=O)c(C)c1 C=C=CCCC(=O)NCCC(=O)NCC1CCCN1C(=O)C(C)SC C(N=c1[nH]c(N(CCC(C)C)C)nc(=N)[nH]1)C1CCCC(C)CC1 c1(CNC(C23N(C(CC4(C)CCC4)=O)CC(C2)C3)=O)[nH]ccc(=O)c1O c1(C(N2CC(OC)C(NC(=O)CC(C)SC)C2)=O)cccc(=O)n1C CC1(c2cn(-c3cccnc3F)nn2)CCN(C(=O)CCOC2CCOC2)C1 c1(C(=O)NCCCCCCN(C(C(CC)C(=O)OC)=O)C)cc2cccnc2s1 C=CCCCCC(=O)N1CCCC(C)(CNC(c2ccc(C(C)(C)C)s2)=O)C1 CC(C)CCCCC(=O)NC(C1CCN(C(=O)Cc2cc(Br)ccn2)C1)C C(C)(C)(CCC(=O)NC(Cc1cc[nH]n1)C(N1CCC(C)(C#N)C1)=O)OC C12C3CCN(C13)C(=O)C=CCCC(=O)N2.c1(NC2CCOCC2)c[nH]nc1OC N1(C(C2(COC)CC2)=O)CCC(C2CCCN2C(c2nnn(C(C)(C)C)n2)=O)CC1 c1(CNC(C(COC)C)=O)cc(F)ccc1NC(C1CCCC(CF)C1)=O N1(C(C(C)=C(C)C)=O)CC2(C1)C(NC(c1ccnn(C)c1=O)=O)CCS2(=O)=O C(=O)(C1=C(Cl)CC1)NC(CNC(c1cc(C(CC)C)no1)=O)C N1(C(C2CC(C)(NC(CC3CCCC(C)(C)C3)=O)C2)=O)CCOCC(F)(F)C1 n1(CC)nc(C(=O)NCC2(CNC(c3ccc(O)nn3)=O)CC(F)(F)C2)c(C)n1 C1(N(C(C2C(=C)C2)=O)CCO)CCN(C(=O)CCC(=O)N(CC)CC)CC1 c1(C(=O)OC(C)=O)n[nH]cc1C(=O)NC(CCNC(CC=CCC)=O)C CON(CCC(=O)NC1(C)CC1)C(=O)Cc1ccnc(O)c1.C1CC1.OC N1(C(=O)OC)CC2C=CC1C(C(=O)NC1CC(CNC(c3cnc(SC)s3)=O)C1)C2 c1(C(=O)NC(C2CCCCC2)CNC(C2(CC#C)CCC2)=O)c(CO)n[nH]c1C c1(C(N2CC(=C(CCCC(=O)NC)F)C2)=O)ccccc1CC(=O)OC c1(C(N2C(CN(C(c3c(C)ocn3)=O)C)CCCC2)=O)cc(F)ccc1O c1(SC)ccc(CCC(=O)NC(C)(CNC(c2sccc2F)=O)C(C)C)cc1 c1(C(=O)N(C2(C(C)C)CCNC2)C2CC2)cccc2ccccc12 Cc1nc2c(s1)CN(C(C1CN(C(=O)C(C)(F)c3ccon3)CC1(C)C)=O)C2 c1(CNC(C2C(CO)CCN2)=O)csc(CN)c1 N1(C(c2c(CC)[nH]cc2)=O)CC2CC2(CNC(=O)CC2CC=CCC2)C1 N1(C(C(C)OCCC=C)=O)CCCC1C1CCN(C(c2oncc2C)=O)C1 Cc1cncc(C(N2CCCC(CNC(c3cn(CCCF)nc3C)=O)C2)=O)n1 C(=O)(CC(C)(C)C(C)=O)NC12CC(C(=O)Nc3cnc(COCC)nc3)(C1)C2 c1(C(=O)NCCC2CN(C(c3c[nH]cc3C3CC3)=O)CCO2)cnn2c1CCC2 CC1(C)C(NC(=O)CCC2CC2)CCN1C(=O)CC1CCCCCO1 CCCC(CC)C(=O)NCC(C)(C(C)C)NC(=O)CCCOc1ccccc1 n1(CC)cc(C(F)(F)C(=O)N(C)CCN(C(=O)C(C)NC(c2cccs2)=O)C)cn1 c1(C(=O)NCC(CNC(C(CC)SC)=O)OC)onc2c1CCCC2 c1(C(=O)OC)cc(NCC(C(C)(C)C)OC)cc(C(=O)N(C)C)c1 N1(C(CSC(C)C)=O)CC23CCCC2(C1)CN(C(=O)C(C)Sc1ccccc1)C3 c1(NC(CCOCCNC(CCC(C)=O)=O)=O)ccc(F)cc1F Cc1nn(CC(N2C(C(=O)NC(C3CCCCC3)C)CC2C)=O)c(=O)o1 C(=O)(C1=NOC(C)(C)C1)N(CCCC(N1CC(CC)(CC)C1)=O)C CCCCCC(C)(C)CNC(=O)C(CCC)NC(=O)C(C1CC1)OCC C1(CNC(C2(CCOC)CCC2)=O)CC(C)CCN1C(=O)CC1CC1(C)C c1(C(=O)NC(CN(C(C(C)c2cncs2)=O)C)C)cc(C2CCCCC2)n(C)n1 C12(CC(=O)NCC3=CCCOC3)CCC1CN(C(=O)Cn1cncn1)C2 c1(-n2c(C)nnc2)ccc(NC(=O)NCc2ccc(C(F)(F)F)[nH]2)cc1 Cc1noc(C(=O)NCCC2(NC(=O)CC(C)C)CC2)n1 CC(C)C#CC(=O)NCCN(CC(=O)NC1CC(CO)(CO)C1)C1CC1 C(=O)(C1=C(C)OCCC1)N1CCC(C)(C(N2CCC(O)(CCC)CC2)=O)C1 c1(C(=O)NC2CN(C(C(C)(C)C3CC3)=O)CC2C(F)(F)F)cc2sc(Cl)cc2s1 CC(CNC(c1cccc(CO)n1)=O)C(F)C(=O)N1CC(C)(CO)C1 N1(C(c2ncc(C)cc2F)=O)C2CC=C(C(=O)N(CC(O)CO)C(C)C)C1CC2 c1(NC(C2CC(=C)CN2Cc2ncccc2C)=O)c(C(=O)OC)cc(Br)cc1Br CC(C)P(=O)(CC(=O)NCC1CCC1NC(=O)C(C)(C)N1CCCC1)C(C)C C1(N(C(C2CCCC2F)=O)CC)CCCN(C(C2CCC3(CC3)C2)=O)CC1 C1(NC(C2(N(C)C)CCCC2)=O)CCC(C)(CNC(=O)C(=O)Nc2ccncc2)C1 c1(C(N2CC3CCC2CN3Cc2ccc(O)cc2Br)=O)c(O)ccc(F)c1F N1(C(COc2c(C)occc2=O)=O)CCCCC12CC(Nc1ncccn1)C2 c1(NC(=O)NCC2(C)CC2c2cc(Cl)cs2)nc2ccc(Br)cn2n1 CC1(C(=O)NCCC2CCN(C(=O)CNS(=O)(=O)C3CC3)C2)CC2CC2C1 N1(C(C(C)(C2CC2)OC)=O)CCC(CNC(c2ccc([N+](=O)[O-])s2)=O)C(F)(F)CC1 N1(C(c2ccc(NC=O)cc2)=O)CCC2CN(C(=O)Cc3csc(Cl)c3)CC2C1 c1(C(N2C3(CNC(C(C)OC)=O)CCC(CC3)C2)=O)cn2c(n1)CCCC2C c1(CC(=O)NCCC2CCCN2C(C2CCC(F)CC2)=O)cccc2ccoc12 N1(C(C=C(C)C)=O)CCN(C(=O)CCCC(F)F)C(CCC)C1 c1(C(=O)NC(C(=O)NCC2CNC(=O)CO2)C2(C)CC2)ccc2[nH]ccc2c1 C(=O)(C1=CC2C=CC(C1)C2)N1CC=CC(C(=O)Nc2c(OC)cccc2)C1 N1(C(Cn2cc(C(C)O)nn2)=O)CC(C2CCN(C(c3ccc(Cl)s3)=O)CC2)C1 C1(NC(CC2CCC(=O)NC2)=O)CCC2CC1CN2C(c1ccc2c(c1)NCC2)=O c1(CNC(CCC(C)N(C)C)=O)cccc(C#N)c1.C1(=O)CCN1 Cc1n[nH]c(C)c1S(=O)(=O)N1CCC2CN(C(c3ccnc(O)c3)=O)CC2C1 Cn1nc(I)cc1CC(N1CCC(C#N)C1)=O C12(NC(C(CC)OC)=O)CCCC(NC(=O)C(C)NS(=O)(=O)CC)(C1)C2 Cc1ccc2c(C(=O)NCC3CCC(C)CN3C(=O)CCCCCO)cnn2c1C c1(C(=O)NC(CN(C(C(C=C)(C)C)=O)C)C)cc2c(Cl)cc(Cl)cc2[nH]1 C(=O)(C(C(F)(F)F)C(F)(F)F)N(CCCNC(C1CCC(C(C)C)CC1)=O)CC N1(C(C(CC=C)C)=O)CC2(C)CC1C2NC(=O)CCCSC(C)(C)C CCS(=O)(=O)CC(C(=O)NCCOCC1CC1)N1CC(CCOC)CC1CO C(=O)(CCCCC(N)=O)N1CC(CN(C)C(C2CC3C=CC2C3)=O)OCC1 C1(C(=O)NC2CC(C#C)C2)CCN(C(=O)Cn2cc(Cl)cn2)CC1O Cc1ocnc1CNC(=O)C(C)(C1CCC1)NC(c1ccn(C)c1)=O N1(C(CC2(N(C)C)CC2)=O)CCCCC1CC(N1CC(N2CCCC2)C1)=O S(=O)(=O)(c1cc(Br)c(Br)s1)N1C2(CN(C(c3ccc(C(C)(C)C)cc3O)=O)C2)CC1 CC1CN(C(c2coc(Cl)c2)=O)CC2(CCN(c3cncc(C#N)n3)C2)O1 C1(CCNC(C(C)n2cccc2)=O)CSCCN1C(=O)COC1CCC1 C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)NC1C(NC(CC(C=C)(C)O)=O)CC(F)(F)C1 Cc1oc(C)c(C(N2CC3CC3(CNC(=O)C(c3cccnc3)C)C2)=O)c1C C(CC(C)(C)C(=O)NCC(C)(C)OCCNC(=O)CC(C)c1ccncc1)OC Cc1cccc(OCC(=O)NCC2CC(C)N(C(c3ccns3)=O)C2)c1 N1(C(c2nc(CCN(CCOCC)C)c(C)s2)=O)CCCCC1C(=O)OC C(=O)(CC(CNC(C1CCCSC1)=O)C1CCC1)NCCOC c1(C(N2CCC(NC(C3C(=C)CC3)=O)C2(C)C)=O)cc(F)cc(Br)c1F Cc1ccccc1C(=O)NCC(=O)NCC(O)CNC(=O)CC1NC(=O)NC1=O C=CC1(C)COCCN1S(=O)(=O)CC1CC1C(C)(F)F CCC(O)C(F)(F)C(=O)NCC1CCC(F)(CNC(C2CC(=O)N(O)C2)=O)CC1 C1(NC(C2C(=C)CC2)=O)CCC2CC1CN2C(c1cc(OC)ncc1Cl)=O CC1CN(C(C2C3CN(C(=O)CN(C)C)CC23)=O)CCC1O c1(NCCc2c(C)nc(C)nc2O)ncccc1S(=O)(=O)N1CCCCCC1C c1(CCCC)ccc(C(N2CC(NC(=O)C(C)CC(F)F)C(SC)C2)=O)cc1N CC1CCCCCN1C(=O)CN(C(=O)CCc1ccn(C)c1)C S(=O)(=O)(c1ccc(F)c([N+](=O)[O-])c1)N1CCC(CC(N2C(C)(C(C)C)CC2)=O)C1 c1(N2CCCC(NCCN(CC=C)CC)C2)cc(N)nc(C)n1.C(CO)O C1(C(=O)NCC23CC2CN(C(=O)CC24CC(C2)C4)C3)Cc2ccccc2O1 c1(CC(=O)NC2CN(C(C=C(CC)CC)=O)CC23CCC3)coc2cc(Cl)ccc12 c1(C(=O)NC(CCC=C)C(=O)N2CCCC2CN=[N+]=[N-])ccc(C#N)c(C)n1 C=CCC(C)(CC)C(=O)N(CCCCCC(=O)NCc1ncoc1C)C C1(N)CCC2(CCC2)C1.CC1CC(C(=O)N(C)CCOCCC(=O)NC2CC2)CCS1 C1(C(N2CCN(C(C=C(CC)CC)=O)C(C3CCC3)C2)=O)CCCC(C)(C)CC1 c1(CC)ocnc1C(=O)NCC1(CNC(c2ncoc2-c2ccccc2)=O)CC1 c1(CNC(CCc2nc(C)c(C)o2)=O)n[nH]c2c1CN(C(=O)C(F)C1CC1)CC2 CCC(F)(F)C(C)(C)C(=O)NC1CC2CC(C1)N(C(=O)C(C)(COC)OC)C2 N1(C(c2cc(C)c(C)nc2)=O)CCC2(CC2)CC1C(=O)NCC#CC1CC1 c1(SCC(=O)NC(CCC2CC2)C(=O)Nc2ccc(O)nc2)ccncc1Cl C(CCO)(C(F)F)NC(C1(CNC(C2CCN(C)C2)=O)CC=CC1)=O c1(C(N2CCC(C(C)NC(c3cnnn3C)=O)CC2)=O)cc(F)cnc1Cl N=c1cc(C(=O)NCC2CCN(C(C3CCCN3N=O)=O)C2)[nH]c(=N)[nH]1 c1(OC)cccc(OC)c1CC(N1CCC(c2cn(CC=C(C)C)nn2)C1)=O c1(C(N2CC(N(C)C(C3CCC4(CCC4)CC3)=O)C2)=O)ccnc(P(C)(C)=O)c1 C#CC(CC(C)(C)C)N1CCOCC1.c12cccc(n1)C(C)(C)NC2=O c1(C(N2CCC(C3N(C(CCC(=C)C)=O)CCCC3)C2)=O)ccc(C)nc1OC C(=O)(CN=[N+]=[N-])N(CC(N1CC(CC(C)C)C1)=O)CCC c1(CCC)nc(CCSc2ccncc2)nn1-c1ccc(-c2ccc(F)cc2)cc1 Cc1ccc(C(=O)N(C)CCc2cnc(NC(=O)C3=CSCCO3)s2)c(C)c1 C(CCCCCNC(C1CCSC1)=O)N(C(=O)CC1CCC(C(F)(F)F)O1)C c1(CC)ccc(S(=O)(=O)NC2CCC(C(=O)Oc3ccc(C(C)=O)cc3)CC2)cc1 Cc1oc(S(C)(=O)=O)cc1C(N1CCCC1CCNC(C1(C)CC1(F)Cl)=O)=O c1(CC2N(C(=O)Nc3nnn(C(C)(C)C)n3)CCC2)cnc(O)nc1O C(=O)(C(O)CCC(F)(F)F)N1CC2C(CNC(C3CC4(CC(=C)C4)C3)=O)(C2)C1 N1(C(CC(C(C)C)c2ccccc2)=O)CCC(NC(=O)C2=C(Cl)CC2)C12CC2 Cc1cc(C(=O)NCC2(NC(=O)C=CCc3ccccc3)CCC2)c(Br)s1 C1(N(C(c2nccc(C)c2)=O)C)CN(C(=O)CCCn2ccnc2C)CC12CC2 c1(CC(=O)NCC(CNC(C2CCC(CC)C2)=O)C)cccc2c1OCCO2 c1(C(N2CC(NC(c3c(C)cc(CC)o3)=O)(CO)C2)=O)nnn2c1C(=O)NCC2 c1(-c2ncco2)cccc(F)c1.N12CC3C(C3C1)CN1C(CCC1)C(=O)NC2=O CS(=O)(=O)c1ccccc1S(C)(=O)=NC(=O)c1ccccc1CSCc1ccccc1 C=CCCCC(C(=O)NC12CCC(CC1)C2)NC(c1ccc(CC)nc1)=O C(=O)(CCC(=O)c1ccc(Cl)cn1)NC1CN(C(C(CN(CC)CC)F)=O)C1.C(=O)OC c1(C(=O)NC(CC)CNC(C2(C3CCC(C)O3)CC2)=O)cc2cccnc2o1 C1(CNC(CSCC=C)=O)CN(C(=O)CCc2ccc(C)nc2)CC12CC2 N(C(=NCCCC(F)F)NCc1ccn(C(C)C)n1)CC1N(CC)CCC1 C1(NC(c2cc(COC)no2)=O)CN(C(c2coc3c2COC3)=O)CC2(CC2)C1 C(c1cn(C)nn1)=CC(=O)NC1C(NC(C(C)=CC2CC2)=O)CCC1 CC(C)(CCNC(C1CCCN1C1CC1)=O)C(=O)NCc1ccc(F)cn1 CC(C)N=c1[nH]c(=NCc2nc(Cl)cs2)c2cc(F)cc(F)c2[nH]1 c1(C(=O)NCC2CC(NC(COCCC=C)=O)C2(C)C)ccc(C)c(NC(C)=O)c1 c1(C(=O)NC2(C3CCN(C(C(C)O)=O)C3)CC2)cc2cc(Br)ccc2c(=O)o1 C1(C)CCN(C)CC1c1ccnn1C.C1(N(CC)CC2COC2)CC(CN)C(O)C1 N1(C(C23N(C(C4CCCCC(=O)N4)=O)CCC2C3)=O)CCC(C2CCC2)CC1 c1(C(N2CCCC(CCNC(C(C)O)=O)C2)=O)cc(N)cc2ccccc12 c1(-c2ccc(C3(CO)CC3)cc2)cc(C)c(C)cc1Cc1c(OC)cc(Br)cc1 S(=O)(=O)(c1ccc(NC(c2ccc(C)s2)C)nc1)NC(COC)(C)CC C1(CCNC(=O)C2CC2)(NC(=O)CO)CCCN(C(C2CC3CCC2CC3)=O)C1 C(=O)(C1CCCc2nnn(C)c21)N1CCC(NC(c2c(C)cc(O)cc2)=O)CC1 c1(C(=O)OCC)cc(N(C(C)CNC(c2cnc(CC)s2)=O)C)ncn1 C1(NC(c2c(C)cc(F)cn2)=O)C2CC3CN(C(=O)C(C)CN(C)C)C1C3C2 c1(N(C)Cc2ccc(C)cc2Br)[nH]c(=NC(C)c2nc(=N)[nH][nH]2)nc2scnc12 c1(OCC)ccc(C(=O)N(C(CNc2ncncc2C#N)C2CC2)C)cc1 c1(C(N2CCC(C)C2CNC(c2ccc(C(N)=O)cc2)=O)=O)cc(O)cc(Cl)c1 N1(C(CCCN(C(C)=O)C)=O)CCC2CN(C(=O)C(n3ccc(C)n3)C)CC2C1 C1(CNC(C2CN(S(CC)(=O)=O)C2)=O)CN(C(=O)C(C)c2cccs2)CC12CCC2 C1(C(=O)Nc2c(CC)nn(C)c2)N(C(c2ccn(C)n2)=O)CC12CCCC2 C1(CC=C)(C(=O)NCC(C(C)C)NC(c2cn(CC)nn2)=O)CC=CC1 c1(C(=O)NC2C(C)(C)CN(C(=O)CP(C)(C)=O)C2)ccc2c(c1)NC(=O)C2=O C1(CNC(C2CCC(F)(F)C2)=O)CCN(Cc2cc(Cl)ccn2)CC1(F)F C1(NC(c2c(C#C)cn(C)n2)=O)CN(C(C2CC2COC)=O)C2(CCOCC2)C1 c1(CNC2C(NC(C(C(=O)OCC)(C)C)=O)C2)ccc2nnnn2c1 N1(C(c2cc(CC)no2)=O)CCC(C2CC2)C1C(=O)NCC1CCCCCCC1 C1(C(=O)NC(c2ccccc2)C(=O)OCC)CCCCN1C(c1sc(Cl)nc1C)=O CCC(C(C)CN(C)C)NC(=O)C(C1CCCC1)NC(c1ccc(C(C)=O)o1)=O N1(c2c(OC)ccnc2)CCN(N(Cc2ccco2)C2CC2)CC1 c1(C(=O)NCC2CN(C(=O)C(F)(F)C3(O)CCC3)C2)cccc2c1C(=O)NC2=O c1(OC)ccc(C(=O)NCC2CC(CNC(C3CCN(C)C3=O)=O)CO2)c(F)n1 N1(C(C2CC2(F)F)=O)CCCC(C2CN(C(C3(O)CCOCC3)=O)C2)C1 Cc1ccc(CCC(=O)NCCC2CC(NC(=O)CN3CC=CC3)C2)cn1 C(=O)(C(C(C)O)N(C)C)NC(C1C(C(N2CC(CC)(CO)C2)=O)C1)C N1(CCC(=O)NCCN(C(C23CC(C(=O)OC)(C2)C3)=O)CC)CCc2ccccc2C1 Cc1sc2ncc(C(=O)NCC(C)NC(=O)C=CCF)n2c1C CCC(C)CC(C)C(=O)N1CC(N2CCCSc3ccccc32)C1 CCCC(C)C(=O)NCC(c1cccc(C(F)(F)F)c1)NC(C1CC(C#N)C1)=O CC1(C)CC=C(C(=O)NCC2CC3(C2)CN(C(=O)CC(F)(F)C(F)F)C3)CC1 C1(NC(=O)C2=CCC2)COCCC1NC(c1c[nH]nc1C1CCCC1)=O N1(C(c2nc(C)n(C)c2)=O)CCC(NC(c2cnc(C3CCC3)o2)=O)C(CO)C1 C1(C(=O)NC2(C(N3CC(NC(=O)NC)C3)=O)CC2(C)C)CCCCCN1C C1(C(C)C)CN(C(=O)OC(C)(C)C)CCN1C(c1ccc(C2(C)CCO2)cc1)=O c1(N2CCC(NC(c3cn(CC)nc3)=O)(COC)CC2)ccc([N+](=O)[O-])cn1 Cc1cnc(O)cc1NC(C1CC1NC(c1cccnc1O)=O)=O N1(C(CN(C(COC)=O)C)=O)CCN(C(C2CCCN(C(C)C)C2)=O)CC1CF CC1CC(NC(=O)COCCNC(c2cncn2C)=O)CS1 CC1CSCCN(C(C2(CF)CCN(C(c3cnc(Cl)n3C)=O)C2)=O)C1 N1(C(C2(F)C(C)OCC2)=O)C2CCC1CN(C(c1nnn3c1CCCC3)=O)C2 C=CC(C)CC(=O)NC(CCC)C(=O)N1CCCC(C)C1 C=CC1OCCCC1C(N1CC(CCNC(=O)CSc2cccc(F)c2)C1)=O Cc1cc(F)cc2c1CCC2NC(=O)C(N1CC2(CCCCO2)C1)=O c1(CSC=CC(=O)NC2C(NC(c3ccco3)=O)C2)n[nH]cc1Br N1(C(Cn2c(C)ccn2)=O)C2CCCC1CN(C(=O)C(C)(C)NC(N)=O)C2 c1(C(N2CC(NC(C(C=C)(F)F)=O)C(O)CC2)=O)cc2cn[nH]c2cn1 Cc1cc(-c2ccc(C(N3CCC(O)(c4cnn[nH]4)C3)=O)cc2)oc1C CCCCC(C(=O)NC1CCC1)N1CC[Si](C)(C)CC1 Cc1ncc(C(=O)NCC#CCNC(c2cncn2C2CC2)=O)cc1CC(C)C N1(C(C(=O)NCC2CCC(C(F)(F)F)O2)=O)CCOC(C2CCCO2)C1 c1(C(N2CC(Oc3cc(Br)cnc3I)C2)=O)ccc(NC2CCC2)cc1O Cc1ncc(C(N2CCN(C(c3cccc(F)c3)c3nnnn3C)CC2)=O)cn1 c1(C(=O)NC2CCN(C(C(C)n3cncn3)=O)C2C2CC2)ccc2occc2c1 C(=O)(CCC(C)S(C)(=O)=O)N(CCNC(C(F)OC)=O)C1CC1 N1(C(CN(C)C(=O)C2CC2)=O)CCC(NC(=O)Cc2cnccc2Cl)C(CO)C1 c1(NC(C(C=C=C)C)=O)cccc2cccc(Cl)c12 C1(CC(=O)N(C)CCOCCCNC(=O)C(F)C2CCOC2)CCCN1C c1(C(N2C3CC(OCCCC#C)CC2CC3)=O)cc(S(N)(=O)=O)ccc1F C1(NC(CSCCC)=O)CC(C(=O)NC(C)C(=O)NCC)C1 C12(NC(c3cccc(F)n3)=O)CCCC1N(C(c1coc(Cl)n1)=O)CC2 C(=O)(CC(C)P(C)(C)=O)NCC1(F)CC(NC(Cn2nc(C)c(Cl)c2)=O)C1 N1(C(c2c(C)scn2)=O)CC(NC(c2ccc(CSC(F)F)o2)=O)C2CC12 c1(C(N(CCOCCC(N2C(CC(=O)NC)CC2)=O)C)=O)cncc(Cl)c1 c1(CNC(CCN(C(c2c(CC)c[nH]c2)=O)C(C)C)=O)cc(Cl)ccn1 C=CC(C)(CCOC)C(=O)NCC(C(C)C)NC(c1nnc(C(F)(F)F)s1)=O c1(C(=O)NC2(C(=O)OCC)CC(C(F)F)C2)cc(S(=O)(=O)N(C)C)cn1C c1(NC(CNc2nnc(SCC)s2)=O)ccc(O)cc1O C(CCC(=O)NC1CCCC1NC(c1nscc1Br)=O)N(C)C c1(C(N(CCCNC(CC=C=C)=O)C(C)C)=O)cn(C)nc1CC(C)C C(=O)(C1=C(S(=O)(=O)N=S(=O)(N(C)C)N(C)C)CCCC1)N1C(C)CC(C(=O)O)C1 C1(C(=O)NCCN(C)C(c2c[nH]c(C#N)c2)=O)CC2(CCC(F)(F)CC2)C1 c1(N2CC=CC(N(C(C3CCC4(CC3)CC4)=O)CC)C2)nc(C#N)ncc1Cl N1(NC(=O)OC(C)(C)C)CC2CCC1C1CN(N3CCCC3CCO)CC21 C1(C(C)NC(C(c2ccccc2)SC)=O)CCCN(C(=O)CC2CC(C)=NO2)C1 c1(C(=O)NC(CC(N)=O)c2cn(CCCOCC(F)F)nn2)cc(Br)c(Br)cn1 C1(=O)CCC(=O)OC2(CN(C(C(C=CC)O)=O)C2)CCN1.C(C)(C)(C)OC N1(C(c2cc(F)c(F)c(F)c2)C(=O)NCCCSCC)CCOc2ncccc2C1 c1(C(=O)NCC2(C)C(C)CN(C(c3ccccc3)=O)C2)c[nH]c2cc(F)ccc12 c1(C(c2ccccc2)CCC#N)ccccc1CCC(=O)CNCC(F)(F)F.CO C1(C(=O)NCC(N(C(c2nc(C)oc2)=O)C)C2CC2)CCCn2cnnc2C1 CS(=O)CCC(=O)NC1CCC(NC(C2CC23CCCC3)=O)CC1 c1(C(=O)NC(C)C(N)=O)cc2n(n1)CCN(C(c1cnc3c(Cl)cccn13)=O)C2 c1(CN2CC3(CC(NC(=O)Cc4cccc(Cl)c4)C3)C2)ccc2c(c1)CCCC2 C(=O)(CCCCCNC(=O)C(C(C)C)NC=O)NCCN(CC)CC C1(NC(c2c(CCC)n(CC)nn2)=O)CC2CN(C(c3[nH]cnc3C)=O)CC12 N1(C(C(C=C)(C)C)=O)CCC=C(C(=O)N2CC(F)(F)CC2CO)C1 c1(OC)cc(C(=O)NCC2CC2NC(=O)C(c2cccs2)C2CC2)cc(Cl)c1 C1(CNC(c2ccc(CC)o2)=O)(NC(=O)NC)CC12CCC2.c12nc-1n[nH]2 c1(OC)cc(C)c(C(=O)NC2(C3CCN(C(=O)C4=CCCC4)C3)CC2)cc1Br CCC(CC(=O)NC1(C)CC(C(=O)OC)C1)NC(=O)C(CNC)CC c1(C(C)C)ccc(F)cc1C(=O)NCCC1CC(NC(c2sccc2Cl)=O)C1 c1(C(N(C2CCN(C(=O)CSCC(F)(F)F)C2)CC#C)=O)cc(CC)cc(F)c1 c1ccc(C)cc1CN1CCOCC1c1ccccc1.N1(CC)CCOC(C#N)C1 C(CCCC(C)(C)C(=O)NNC(=O)C1(CO)CCCO1)NC(C(C)=CC)=O C(CC1=CCN(C(c2ccc3scnc3c2)=O)CC1)NC(c1nc(C)n(C)n1)=O n1(CCC)c(C(=O)NC2CN(C(N3c4scnc4C3)=O)C2)nnc1C.C1CC1 Cc1cc2c(C(=O)NC3(CCO)CN(C(c4snc(O)c4Cl)=O)C3)nccn2n1 c1(C(C(=O)NCCSC)N(CC(=O)OCC)C)ccc(OC)c(SC)c1 CCC(CC)C(F)C(=O)N1CC2(CC(C(N3CCOC(C)C3CO)=O)CO2)C1 c1(OC)ncnc(Cl)c1NC(C12CC(NC(c3cccc(F)c3Cl)=O)(C1)C2)=O CC(N=c1[nH]c(N2CCC3(CSC3)C2)nc2ccsc12)C1CSC1 c1(C(=O)NC2CN(C(C(=O)NCC)=O)C(C)C2)cnc2[nH]ncc2c1 Cc1cnc(C(=O)NC2CCCC2NC(C2CCCCC2)=O)cc1Cl CC1(NC(=O)CNC2CC3CC3C2)CCCCCC1.C1(C=O)CCC1 C(c1ncc(C)[nH]1)=CC(=O)NCCCN(CCC)C(c1cnc(SC)[nH]1)=O C(=O)(CC(C(F)(F)F)OC)N1C(C(=O)NCC2(C(=O)OC)CC2)CC(F)C1 Cc1ccc(N)cc1C(N1CCCC1CNC(C1CC2(C1)CC2(F)F)=O)=O c1(OC)ccc(Cl)c(C(N2CC3CCC3(C(=O)NCCC(C)(C)O)C2)=O)c1F N1(C(CN2C(C)CC2)=O)CCCC1CN(C)C(c1cnn(CC(F)F)c1)=O c1(CCC(=O)N2CCC2c2nc(-c3ccccc3)no2)c(F)cccc1Cl c1(C(N2CC(C)N(C(=O)C(F)C3CCC3)CCC2)=O)cnc2c(c1)OCC(=O)N2 CC(C)(C)C(CNC(C1CCSCC1)=O)NC(c1cccnc1-n1cccn1)=O c1(C2C(CCCC(C)CF)=NN=NNC(CCOCC)CN2)c(F)cccc1Br Cc1ccnc(CCC(=O)NC2CC2NC(C2(C(F)(F)F)CC=CC2)=O)c1 c1(C(N2CC(CNC(CCC(=C)Cl)=O)C(O)C2)=O)ccc(OC(C)C)c(F)c1 N1(C(COCCC#C)=O)CCC(=C)CC1C(N1CC(C)CC1CC)=O C1(NC(=O)Cc2cnc[nH]2)CC2(CCC(NC(=O)CC3(C(F)F)CC3)CC2)C1 c1(C(N2C(CNC(C(=O)NC(C)C)=O)CC2)=O)nc(O)[nH]c(=O)n1 c12nncn1C2.C1(C(=O)NCC#C)CCC1 c1(C(N2CCCC(F)(CNC(C3C(C)CC(=O)N3)=O)C2)=O)cc(O)cc(N)c1Cl N1(C(CNC(=O)OCC)=O)CCCC1CNC(=O)CCC1CCCN1C n1(CC#C)cccc1C(N1CCC(C(C)N(C(c2cc[nH]c2C2CC2)=O)CC)C1)=O C12(NC(c3ncn4ccccc34)=O)CN(C(=O)C3=CCOC3)CC1CS(=O)(=O)C2 c1(C(N2C(C(=O)Nc3c(C)nn(C)c3)CC(C)C2)=O)cnn2ccncc12 C1(C(N2C(C#C)CCC2)=O)COCCN(C(C2CC(C)C2)=O)C1 N1(C(C=CCC)=O)CCC(OC2CC(CCCCC(=O)NC(C)(C)C)C2)CC1 c1(C(=O)NC(C(c2c(OC)cccc2)OC)C)ccn2nnnc2c1 C1(NC(C2C(C)(C)COCC2)=O)CCC2CCN(C(=O)Cc3ccccc3)C12 C(C(C)N=c1[nH]c(-c2ccccn2)nc2[nH]cnc12)N(C(=O)C#CC(=O)N(C)C)C.C N1(C(C2C(C(C)C)OCC2)=O)CC2CCC2(CNC(=O)Cn2ccnn2)C1 C(c1ccccn1)=CC(N1CC=CC(NC(C2(n3cnccc3=O)CC2)=O)C1)=O c1(CC)nc(C)ncc1C(=O)NCCC1(CNC(c2ccc(C#N)cn2)=O)CC1 c1(COC)ccc(CC(=O)NC2CC(NC(=O)Cc3ccsc3Cl)CC2O)cc1 c1(N2CCCC(C=C)C2)nc(N2CCC(CN(C)CC)CC2)nc2ccsc12 N1(C(C2(S(C)(=O)=O)CCC2)=O)CCC(C2CC(NC(=O)C(=O)NCC(F)F)C2)C1 N1(C(C(C)(C)NC(=O)OC)=O)CC=CC(NC(=O)CCNC(=O)CO)C1 C=CC(O)(C(=O)N(CC(O)CNC(=O)CCCN=[N+]=[N-])C)C(F)(F)F c1(C(=O)NC2CCCCN(C(C3=NOC(C)C3C)=O)C2)ccc(P(C)(C)=O)cn1 N1(C(C(C)SCCCC)=O)CC2(CCCCN(C(C3CC(CF)C3)=O)C2)C1 C1(C(=O)NCCCOCCNC(C(c2cnccn2)C)=O)CCc2n[nH]cc2C1 N1(C(COCCC=C)=O)CCC(NC(C2CC3(C2)CC(F)C3)=O)C(F)C1 c1(CN2CCN(C(c3ccc(O)cc3C(F)(F)F)=O)CC2)cc(F)c(O)c(Br)c1 C(=O)(C(C)(C)C(C)(F)F)NCC1C(C)CN(C(c2ccc(CO)c(Cl)c2)=O)CC1 C1(NC(C2(NC(c3ccncn3)=O)C(C)CCC2)=O)CNC(=O)C12CC2 c1(CCOCC(=O)NCC2CN(C(C(C)OCC)=O)C2)cccc(F)c1 C1(C(=O)NCCC(C)NC(C2(N=[N+]=[N-])CC2)=O)CCCC1c1ccccc1 C1(C(=O)NCC(C)NC(=O)CSC(F)F)CCCN(C(c2ccsc2)=O)C1 CC(C)(CS(N)(=O)=O)C(=O)C(=O)COC.C1(C(=O)NCCN)CCOC1 C1(NC(C2CC(OC)C2)=O)CC2CC(C1)CN(C(=O)C(C)=C1CCCC1)C2 c1(C(C(=O)NCC=CCNC(c2cc(CCC)on2)=O)O)cccc(C)c1 c1(C(=O)NCCCN(C(c2c(CC)oc(C)c2)=O)C(C)C)n[nH]c2c1COCC2 C(CC1=CCOCC1)NC(C1(CNC(c2c(C#N)scc2)=O)CCC1)=O Cc1cccc(C(=O)NCC2(C)CN(C(c3csc(C(C)C)n3)=O)CCO2)c1Cl c1(NCC(=O)Nc2cnns2)cc(O)nc2ccccc12 c1(OC)cccc(C(=O)NCCC2CC(NC(C3(C)CCC(=O)N3)=O)C2)c1 c1(NCC2N(C(CC(CC)(F)F)=O)CCCCC2)ccncc1[N+](=O)[O-] O=C(N=c1nn[nH]n1-c1ccccc1)N1CC(CCN2CCOCC2)C1 CCCCCCC(F)C(=O)N(C)CC1(O)CN(C(C2CC3C=CC2CC3)=O)C1 c1cc2c(cc1CCCn1cc(-c3cc4ccccc4s3)nn1)OCCO2 N12CCCC3CN(CCC13)C(=O)CCC2=O.c1(CC2CC2)cn[nH]c1 c1(OC)ccc(Cl)c(C(=O)NCCOCCCN(C)CC(=O)Cn2cc[n+](C)c2)n1 Cc1cc(C(N2CCN(C(=O)CNC(=O)CCCCO)C(C)C2)=O)c(O)c(C)c1 C1(CNC(c2cnc(Cl)[nH]2)=O)(CO)CCN(C(=O)C=Cc2ccco2)CC1 CC(CC(C)(F)F)N=c1ccc(Br)c(S(=O)(=O)N2CCCCCCC2CO)[nH]1 c12ccnc(c1)NC2=O.n1(CCC)cccc1C(=O)NC1CN(C(=O)C2CC2)C1 c1(CC)cncc(CNC(C2CCN(C(=O)CCOCCOC)CC2)=O)c1 CC1CCC(C(F)(F)F)CN1CCn1cncn1.C12COCC1N2 C1(CC=C)(C(=O)NC23CC(CNC(c4cnsc4)=O)(C2)C3)CCCC1 c1(CNCc2cn(CC)nn2)c(C)cc(CC2(CC(=O)OC)CC2)cc1C.NC1CC1 C1(CC)CCN(C(=NCCC2CCC2)NCC2(C)CCCO2)C1 Cc1cc(C(N2CCC(NC(C3(O)CCC3)=O)C2C2CC2)=O)sc1-c1ccccc1 c1(NC(C2CC(Nc3ncc(SC)cn3)C2)=O)cc(C)c(F)cc1Br c1(C(N(C2CCCN(C(C(CC)CC)=O)C2)C)=O)cc2c(nc1N)CCCC2 Cc1cc(C2(C(=O)NCC3(NC(c4cc(O)nc(O)n4)=O)CC3)CC2)ccc1F c1(NC(C(N)Cc2ccc(C(F)F)cc2)=O)ccc(Br)c2c1CCCC2 c1(N2CCS(=O)(=O)CC2)[nH]c(=NC2CC(CCO)C2)nc2scnc12 c1(NC(C)=O)ccccc1CC(=O)N(CC(O)CNC(=O)COC1CC=CC1)C c1(C(N2C(CN(C(=O)C=Cc3nccs3)C)CCC2)=O)c(N)cccc1Cl N1(C(CC(C)N(C)C)=O)CCC2(CCN(C(c3ccc(P(C)(C)=O)o3)=O)CC2)C1 C1(NC(CCSCC)=O)C(C)CN(C(c2ccncc2-n2cccn2)=O)CC1C c1(CCC)nnc(S)n1CC(=O)NC(C)CN(C(=O)CC(C)CC)CC c1(CNC(N(C)Cc2ccc[nH]2)=O)cnc2ccccn12 CC(CC(=O)NCCOCCNC(=O)CC1CCCO1)c1cccnc1 c1(C(N2CC(CNC(C3CC(=O)CC34CCC4)=O)C2)=O)ccc2c(n1)CCCN2 n1(CC(=O)NC(COC)CNC(c2sc(C)cc2C)=O)cnc([N+](=O)[O-])n1 N1(C(C2C(C)(C)CO2)=O)CCC(c2ccccc2)(NC(=O)C=C(Cl)Cl)C1 C(=O)(C(CCCCSC)NC(c1cn(CC2CC2)cn1)=O)N1CCC(COCC)C1 C1(NC(C(C=C)(F)F)=O)CCN(C(c2cccnc2C(F)F)=O)C(C)C1 C1(NC(=O)NCCCN(c2ncccn2)C)CCCC(c2ccccc2)CC1 c1(CC)nnc(C(c2nnnn2CCCOC)NCC(C)CCO)n1C c1(CC(=O)NC(C(C)C)CNC(c2ccnn2C2CC2)=O)nc(F)c(F)cc1F C(CN=c1cc(C)nc(-c2cccnc2)[nH]1)OC(C(c1cnn(C)c1)OC)=O c1(CC(=O)Nc2cccc(CNC(C3C(C)(C)C3)=O)c2)ncn2c1COCC2 C(=O)(C(C)(Cc1ccccn1)NC(=O)NCCNS(=O)(=O)CC)NC c1(OC)cccc(C(=O)NCC2CN(C(=O)C(C)(C)OC)CC23CC3)c1N CCCCCC(O)CC(=O)N1CCC2CC12C(=O)NCC1(CO)CCCC1 Cc1ccc(-n2cc(C3CN(C(c4cc(C)sc4Br)=O)C3)nn2)c(C)c1 C1(NC(COC(CC)(C)C)=O)CC(N=c2nc(C#N)[nH]cc2Cl)C12CCC2 C1(CN(C(C(C)OC)=O)C)C2CN(C(c3ccc(-n4ccnc4)cn3)=O)CC12 C=CCC(COC)NC(=O)CSCCOC1CC1(F)F.C1(=O)CC(=O)N1 Cc1nnc2n1CC(C(=O)N(C)CCN(C(=O)C(C1CCCCC1)F)C)CC2 c1(CCC)cc(C(N2CC(OCCNC(=O)C3=C(Cl)CC3)C2)=O)ccc1Cl C(=O)(C(C)(C)C(N)=O)NCC1(C(=O)NCC(C2CCC2)OCC)CCC1 CCCC(CC(C)C)C(=O)NCC1CC(F)(F)CN1C(=O)C=Cc1ccnn1C c1(C(=O)NC(C2(O)CN(C(=O)CC3CCC(C)(C)C3)C2)C)[nH]nc2ncccc12 Nc1ccc(C(=O)NC2CCN(C(=O)CC3CCS(=O)(=O)C3)C2)c(O)c1 C1(C(=O)NC2CCC(O)C2)(CC)CCCN(C(c2ccnnc2)=O)C1 c1(C(N2CCC(c3ccc(C(=O)OC)cc3)C(O)C2)=O)cc([N+](=O)[O-])cn1C CC(C(=O)N1CCC(CC(=O)NCC=CCl)CC1)C(C)(C)C N1(C(c2c(OCC)ccs2)=O)CC(CNC(C23CCC(CC2)C3)=O)CC1C CC(C)C(C(=O)N1CC(N(C)C(C2CN(C)C(=O)N2)=O)C1)Sc1ccccc1 CC(C)C1=NOC(C)(C(=O)NC2CC3CC2N(C(c2ccncc2F)=O)C3)C1 N1(C(CC(C(F)F)NC(=O)Cn2cc(C3CC3)cn2)=O)CCOC2C(O)CC12 Cc1ccc(CNC(C2(NC(C3C(C)(C)C3(C)C)=O)CCSC2)=O)cn1 C1(C(=O)NC(CNC(=O)C(C)(C)Br)CO)(OC)CCC(C)(C)CC1 c1(C(C)C(=O)NC(C2CCCN2C(=O)CC2CC=CCC2)(C)C)ncccc1F CC1CC(CCNC(=O)CCn2cnnn2)CN1C(c1ccn(C)n1)=O C1(S(C)(=O)=O)(C(=O)NCC(C)N(C(c2cncc(O)c2)=O)CC)CCC1 C1(C(=O)N)CC1C1CN(C(C2(C)CCOCC2)=O)C1.C1(OC)(CNC)CCC1 C(c1ccc(OCC)nn1)=CCNC(CSCCOCC)=O c1(C(=O)NCCN(C(=O)C=Cc2ccoc2)CCC)cc(CC(C)C)nc(O)c1 C1(Cl)(C(=O)NCC(CNC(=O)Cc2nc(C(C)(C)C)cs2)OC)CC1(C)C c1(C(=O)NCCCOCCNC(C2CCNC2=O)=O)cccc2cnccc12 N1(C(c2scc(C)c2)=O)CCCCC1C1CCCN1C(=O)CNS(=O)(=O)C1CC1 Cc1oc(C#N)cc1C(N1CC(CNC(C2CCCN2N=O)=O)C(O)C1)=O c1(C(C)=O)cc(C(=O)NCC(C)NC(=O)C(N2CCC(O)CC2)C)c(C)o1 N1(C(COC)=O)CCN(C)C(CNC(=O)CC2CCC2(C)C)C1 N1(C(C2N(C(C)=O)CSC2)=O)CCCC(N(C(=O)CCN2CCC2)C)C1 C(CC(C(C)(C)C)NC(=O)CC12CCC(CC1)CC2)N(C)C(c1cn(C)nn1)=O C1(NC(c2occc2Br)=O)COC2(CCN(C(c3cnc4cc[nH]c4c3)=O)C2)C1 CN1CC(C(=O)NCC2CC(CNC(c3cn[nH]c3)=O)CO2)OCCC1=O c1(CN(C(=O)CCn2cc(-c3ccccc3N)nn2)C)cc([N+](=O)[O-])sn1 c1(CC)n[nH]cc1C(=O)NCC(O)C(=O)NCCn1nncc1C c1(SC)c(C(=O)NCCCCN(C(=O)COc2ccccc2F)C)cccc1F Cc1c(C(=O)NCC2CN(C(c3coc(C(C)(C)C)n3)=O)CC2C)cccc1N C(=O)(C(CCC(F)(F)F)C(C)C)N1CCC(CN(C(C(C=C)(C)C)=O)C)C1 c1(OC)ccc(C(N2CCC(C(F)CNC(=O)C(C)(C)C(C)O)CC2)=O)cc1O c1(N(CC(C)OC)C)nc(N2CCC3(CCOCC3)C2)nc2c1CC(C)CC2 CS(=O)c1ccc(CC(=O)NCc2nc(CNC(C3(C)CCOC3)=O)cs2)cc1 C1(C(N(C2CN(C(C3CC(C#N)C3)=O)C2)C)=O)OCCC1NC(=O)OC(C)(C)C C(=O)(NNC(=O)CCCc1ccccc1)NCC(=C)Cl Cc1cncc(NC(=O)CC2(C)CN(C(C34CC(CC(C)C)(C3)C4)=O)C2)n1 c1(CC)nccnc1C(=O)N(CCNC(=O)C(C(C)C)SC(C)(C)C)CCSC c1(C(N2CCC(N(C(c3cc(OC)nnc3)=O)CC)CC2)=O)nccc(Cl)c1C N1(C(C(CO)N(C)C)=O)CCC2(C(=O)NC3CNC(=O)C34CC4)CCCC12 C1(NC(CNC=O)=O)CCCC(NC(=O)C(c2ccc(Cl)cc2)(F)F)CC1 C12CN(CCO1)CCNC2=O.c1(C(=O)OC)cn(Cc2nccs2)nn1 CC(C(=O)NCC1CN(C(c2cncc(F)c2Cl)=O)CCO1)P(C)(C)=O C(C)(C)(CCC(=O)NC(C)CCCCNC(C1COCCO1)=O)OC CCC(CC(F)(F)F)C(=O)OCC(=O)NCC(C1(O)CCCC1)(F)F C(=O)(CCCCC(C(F)(F)F)NCC1(C)SCCCS1)OC C(=O)(C#CC1CCOCC1)N(C)CC1(NC(=O)CC2CCC(F)(F)C2)CC1 c1(C(=O)NCCCN(C(Cn2ncc(C)c2)=O)C(C)C)cnn2cccnc12 n1(CC(=O)NCC2(NC(CC)=O)CC3CCC2C3)nc(C)c2cccnc12 Cc1c(O)ccc(C(N2CCN(CCNC(C3CC3(F)F)=O)CC2)=O)c1C C1(C(=O)NCC2(O)CN(Cc3nc(C)on3)C2)CCCC(C)C1 c1(CC)oc(C(=O)NC(C(=O)N2CCC(C)(N(C)CC)C2)C(C)C)cc1C N1(C(C2(C)N=N2)=O)CCN2CCN(C(c3cccnn3)=O)CC2C1 Cc1cc(F)ccc1-n1nnnc1S(=O)(=O)NC1CCN(C2COC3(CCC3)C2)C1=O N1(C(C2(C(CC)=O)CC2)=O)CCCC(C)(C(=O)NCc2conc2C)C1 CC1CN(C)CC(NC(c2cn(C3CCN(c4nnc(O)s4)CC3)nn2)=O)O1 C1(NC=O)(CO)CC2CCCC12.c1(CC(=O)NCc2ncn[nH]2)ccc(O)nn1 C1(NC(C2CCN(C(C3(CC#C)CCCO3)=O)C2)=O)CC(C)OC1=O c1(OC)cc(C(N2CCC2(C)C(=O)Nc2c(O)cccc2Br)=O)ccc1C(C)=O C1(NC(C2CC23CC3)=O)CN(C(=O)CCc2ccc(Cl)c(F)c2)CCC1F c1(CNC(c2cncc(Cl)c2Cl)=O)nc2c(s1)CN(C(C1CC(F)C1)=O)CC2 C(CCCCC(=O)NC(Cc1ccoc1)C(=O)NC1CC12CC(O)C2)OCC N1(C(c2cccc(C(F)F)c2)=O)CCC2C1CCCN2C(C1CC2CCC1O2)=O Cc1sc(C)c(C(=O)N(CCCCNC(C2CC3(C2)CC3F)=O)C)c1Br c1(CCC)nc(=NC2CC(F)(CNC(=O)CCc3ncc(C)[nH]3)C2)s[nH]1 Cc1noc(C)c1C(N1CC(C(C)NC(=O)C(C)n2cccn2)C1)=O C1(F)(CNC(CC2N(C)C(=O)CC2)=O)CCCN(C(c2cnnn2C)=O)C1 C1(NC(C(CC)NC)=O)CCCCCC1NC(=O)C=CC1CCCCC1 CCC(CNC(=O)C(C)NC(c1ccoc1)=O)(CC)NC(c1ccn(C)c1)=O c1(C(=O)NOC2(CN3CCOCC3)CC(N)C2)ccc(F)cc1C.CO c1(OC)ccc(F)c(C(=O)NC2CCN(C(C3CC(C)=NO3)=O)C2C(C)C)c1F C(=O)(C(C)C(O)C(C)CC)NC(C(C)NC(C(CCC)F)=O)C C(CCCCCNC(=O)CSc1ccc(Cl)cn1)NC(C1(C)CC1F)=O c1(C(=O)NCC2CC(NC(C3C(CC)CC3)=O)C2(C)C)cccc2nc[nH]c12 O=C(C1CCCc2c(O)cccc21)NCC1CC(O)CN1C(=O)COC(F)(F)F C1(CN(C(Cn2c(C)ccn2)=O)C)CC(F)CN1C(=O)CNc1cccc(Cl)c1 Cc1nc(NCCCCN2CCCC2)cc(N2CCC(CO)CC2)n1 N1(CC)CCOCC1C(=O)NCC1CN(C(=O)CC=C(Cl)Cl)CC1C CN1CC(CCC2(C(=O)NC(=O)C3=CCSC3)CCCC2)C2(CC2)C1=O c1(OC)ccc(CC(=O)NC2CC2CNC(=O)COCC(C)(C)C)nc1 C1(CC(=O)N(CC(C)CNC(=O)CCC2CC2(Cl)Cl)C)CC2CCC(C1)C2 C(C#CCN=c1nc2c(ncn2C)c(NCC2CC(C)(C)CCC2O)[nH]1)OC N1(C(C(C2CCCC2)OC)=O)CCN(C(c2cccc(=O)n2C)=O)CC(C)(F)C1 C1(C(=O)NC(C2CCCN2C(c2cncc(Cl)c2)=O)C)CN2CCC1C2 N1(C(CNS(N)(=O)=O)=O)CC2(C1)SCCC2NC(=O)C(c1ccc(Cl)nc1)(F)F N1(CCN(C(C(CSC)C)=O)C)CCC(NC(=O)C(C2(O)CCCC2)F)CC1 C(=O)(CCC(F)(F)F)N1CC(CC(C)NC(CN(CC#C)C(C)=O)=O)C1 C#CC1CN(C(c2ccnc(C)c2)=O)CCN1C(=O)CC1(N(C)C)CC1 C(=O)(N=c1cc[nH]cc1O)C1CCCCC1CNC(=O)C=Cc1cc(F)cc(F)c1 c1(SC)cccc(CC(=O)NCc2ccnc(N3CCOCC3)c2)c1 c1(OCC(=O)N(CC(C)CNC(=O)C(=O)NCC(F)F)C)ccc(F)c(Cl)c1 C1(C(=O)NCc2cc(C)oc2)CCCC(NC(C2CCN2C)=O)CC1 N1(C(c2cnn(C(C)C)n2)=O)C2CCC(C2)C1C(=O)NCC1CCN(C)CC1 C1(CC(=O)N(C(C)CO)C)CCN(C(C)CN2CCCC2)C1 c1(C(=O)NC(CC)(C)CNC(=O)CCc2ccco2)cc(=NS(C)(=O)=O)cc[nH]1 C1(C(=O)N(C(C)CNC(C2CC23CCC3)=O)CC)CCN(CCc2ccccn2)CC1 c1(OCC)cc(C(N2CC(NC(C3CCS3(=O)=O)=O)C(O)C2)=O)cc(F)c1 c1(C(=O)NCCOC2CCN(C(CC(CC)(F)F)=O)C2)cnc2c(c1)CCC2 n1(CC)c(C)nc2cncc(C(=O)NCC(C)(C)C3CC3)c12 C(C)(CCC(=O)NCC1CC1CNC(=O)C=Cc1nccs1)SC C1(C(=O)NCCCN(CCCNC(C(C)C(C)O)=O)C)CN2CCN1CC2C c1(C(N(C2CC(C)C2)CC(C)C)=O)ccc2ccoc2c1.C12CCN(CC1)C2=O c1(C(=O)NC2CCN(C(C(=O)NCC)=O)C2C(C)(C)C)cc2c([nH]1)CCC(C)C2 Cc1ccccc1CN(C)C(C1(C)C=CCN1)=O C(=O)(C1CCCc2nccn21)NC1CCC(CNC(CCCCCN(C)C)=O)C1 N1(C(C=C(C)C(F)F)=O)CC=CC1C(=O)N(CC(C)O)CC(C)O C(c1ccncc1)=CC(=O)NCCCCNC(C1CC(C2CC2)C1)=O C1(C(=O)NC(C)(C)CC(N)=O)CN(C(C2C(C)(C)C2(C)C)=O)CC1(C)C CC(Cc1cnn(C)c1)C(=O)NCC1CC(NC(=O)CSCc2ccccc2)C1 N1(C(CC(C)F)=O)CCCCCC1C(=O)NCCC1CC(C)(C)CO1 C1(C(N2CCCC(C)(CNC(CC=C=C)=O)C2)=O)CC2(CO1)CC(F)(F)C2 C1(CNC(C(CC)OC)=O)CCN(C(c2cnc(C3CC3)s2)=O)C12CC2 c1(OC)cc(C)cc(C(=O)NCC23CCC2CN(C(=O)CCC(C)(C)F)C3)c1N C12(NC(COc3cc(C)on3)=O)CCCC1N(C(c1cnc(F)c(C)c1)=O)CC2 C(=O)(C1=NOC(C)(C)C1)N(CC)CC1CCN(C(c2cnc(C3CC3)s2)=O)CC1 N1(C(=O)Cc2cccnc2)CCC(C(=O)NCC2CC(O)C(O)C2)(CF)C1 c1(C(N2CC(C=C)(CC(=O)NC(C)C(O)C(C)C)C2)=O)cn2c(n1)CCC2 C(C)(CCC(=O)NCC1(CNC(=O)CC2CCCC(=O)N2)CC12CCC2)OCC Cn1c(=O)c2cc(C(N3CCC4(C(=O)Nc5cn[nH]c5)CC4C3)=O)sc2n(C)c1=O c1(CC(=O)NCC2N(C(Cc3nccc(C)n3)=O)CC2)ccc2sccc2c1 c1(CC(=O)NC2CC(NC(=O)C(O)c3cnc[nH]3)C(O)C2)ccc(Cl)c(Cl)c1 C1(NC(C(C)N(CCC)C(c2sccc2CO)=O)=O)(CO)CC2CCCC12 c1(C(N2CCN(c3cc(C)ccn3)CC2)C(=O)NC)cnccc1CO C1(NC(c2c(CC)ocn2)=O)CCC12CCN(C(C1CCCC(=O)CC1)=O)CC2 O=C(C1=CCCC1)NC1C=CCC(C(N2CCC2C2CCOCC2)=O)C1 c1(C(N2CC3C(CNC(c4n(CC)ncn4)=O)(CC3)C2)=O)cc(Cl)cc(Cl)c1O CC(C)CCCCC(=O)NCC1(CC(=O)NC2CCCC23CC3)CC1 N12CC3C(C3C1)C2=O.CC(C)(CC1CC1)Cc1cn(CCC(F)(F)Cl)nn1 O=C(CCC(=O)N1CCCC(NC(=O)Cc2ccsn2)C1)c1cccc(F)c1 CC1(C)C(C)(C(=O)NCC2(NC(=O)CCc3csc(=N)[nH]3)CCOCC2)C1(C)C N1(C(C(C)C2CCC2)=O)CCCC2(CCN(C(c3cc(=O)n(C)cn3)=O)C2)C1 N1(C(CC(=O)OC)=O)CCC(NC(=O)C(C)(N(CCCSC)C2CC2)C2CC2)CC1 C(=O)(C(C)C(C)(C)C)N(C1CCN(C(C2(C(C)(C)C)CCCC2)=O)C1)CCC Nc1cccc(Cl)c1C(=O)NCCCNC(=O)CC12CCCC1C2 C1(C(=O)NC(CCC)C2CC2)COCC1NC(c1csnc1OCC)=O N1(C(C(C)C)=O)CC(NC(=O)CSCC)CC1(C)C.C(c1ccccc1)=CC=O c1(CC(=O)N(CCCn2cc(C(C)(C)OC(=N)O)nn2)C2CC2)c(F)cc(F)cc1F c1(-c2cncc(C(Nn3c(C)nnc3)=O)c2)n[nH]c2ccc(Cl)cc12 C1(CCC)CCN(C(C2(N(C(=O)CC=CCOC)C(C)C)CC2)=O)C1 C1(C(=O)NCCC2CC(NC(C(C(C)C)O)=O)C2)CC2CCC(C1)N2C(N)=O c1(NC(CCOCCCNC(CCc2n(C)cnn2)=O)=O)cccc2c1OCO2 C(=O)(C(F)(F)CO)NC1C(CC(=O)NCC(C)OCC#C)CCC1 c1(CC(=O)NCc2cc[nH]c2)cccnc1Cl.c12cccc(c1)C(=O)NC2C N1(CC(=C)CC)CCC(O)(C(N2CCOCC2C)=O)CC1 CCCC(O)C(=O)NC1(CCOC)CCN(C(=O)CN2CCC(O)CC2)C1 C(=O)(C1c2ccccc2CN1Cc1ncc(-c2cc(C)[nH]n2)cc1F)OCC c1(CC(=O)NCC2CN(C(CCCOCC)=O)CC(C)O2)ccc2nn[nH]c2c1 C1(NC(C2C(C)CCC2)=O)CC2(C1)CC(CNC(=O)CN1CC(C)(C)C1)C2 c1(C(N(C2CCC(CNC(=O)NCCCl)C2)C)=O)cn2ccnc2c(=O)[nH]1 CCC(CNC(C1CCC(C)CC1)=O)(CC)C(=O)N(CCC1=CCCCC1)C C(CCS(C)(=O)=O)NC(C=CCN(C)C(C1CCCN1C1CC1)=O)=O C1(NCC2CC(O)C2)CCOC12CCN(C(c1cnc(O)o1)=O)CC2.C1(N)CC1 Cc1c(C(=O)OCc2ccnn2C2CC2)ccc2n[nH]cc12 N1(C(C(=O)Nc2c(OC)ccc(OC)c2)c2cc[nH]n2)CCOCCC1(C)C C1(C(N(C)CC2CCN(C(c3csc(Cl)n3)=O)C2)=O)CN2CCC1CC2 C1(CC(N2C(CNC(C3(CC#C)CCCC3)=O)CCC2)=O)CCCCC1O c1(C(=O)NC2CN(C(C(CC(C)C)F)=O)CC23CC3)cc2cccnc2cn1 Cc1c(Br)ccc(C(=O)NC2C3CN(CC(O)C(F)(F)F)CC23)c1F C1(NC(=O)C=Cc2cncs2)CN(C(C2C3CC4C(C3=O)C24)=O)CCC1CO Cc1cscc1C(=O)NC1CCC(CNC(c2n[nH]cc2-c2ccncc2)=O)C1 CC1CCC(C(=O)NCC2C(CNC(=O)CSCC(F)F)C2(F)F)CC1 O=C(CC(F)(F)C(F)(F)F)NCC1CC1CNC(C1(CCF)CC1)=O N1(C(c2ccc(OC)cn2)=O)CC2CCC2(NC(=O)COc2ccc(Cl)cc2)C1 Cc1nc(CCC(=O)NCC2CCCCN2C(C2CC2(C)C)=O)oc1C C(=O)(C1=CC2C=CC(C1)C2)NCC(C)NC(c1cc(C)c(CO)cn1)=O CP1(=O)CCN(CC(=O)NCC(=O)NC2CCC(F)(F)CC2)CC1 N1(C(c2c(CC=C)cccc2)=O)CC(O)CCC1C(=O)N(C)CC1(C#N)CCC1 c1(OC)ccc(CN2CC3(CC3C(=O)NC3CCC(F)(F)C3)C2)c(Cl)c1 C=C(C(=O)NCC1COC2CNCC12)C1CCC1 c1(C(=O)NC2(CCCNC(CCC(=O)NC)=O)CC2)cc(S(N)(=O)=O)c(C)o1 Cc1cc(C(=O)NC2CC(NC(=O)Cc3cc[nH]n3)CC2O)cc(C)n1 N1(C(C(CCN(C)C)NC(C2CC3CCC3C2)=O)=O)CC2(CC(=O)NCC2)C1 N1(C(CC(C)O)=O)CCOC2(CCN(C(c3c(C4CC4)cnn3C)=O)C2)C1 c1(C(=O)NC2CC(N(C(C(C(C)C)OC)=O)C)C2)cc2c(s1)CCCC2 C#Cc1cccc(OCC(N2CCCC2CCNC(=O)CCc2cnoc2)=O)c1 N1(CC2C(CCC)C2)C(=O)CCN(Cc2cccc(S(=O)(=O)N(C)C)c2)C1=O C1(N(C(=O)C=CCO)CC)CCN(C(=O)CCOC2CCCOC2)C1 CCCC(O)CC(=O)NC1CC12CC(NC(=O)CN(C)Cc1ccc(C)cc1)C2 c1(C(C)C(=O)NCCOCCN(C(=O)C(N2CCSCC2)C)C)ccc(F)cc1 C(CC(C)(C)C)(C(=O)NC(C)(C)CN(C(=O)CC1CCCOCC1)C)OC C1(C(=O)NCC(CCCC)NC(=O)Cc2cccc(O)c2)CC2(C1)CC2(F)F c1(C(=O)NCC2(NC(=O)COC(F)F)CCOCC2)c[nH]c2c(Cl)cccc12 Cc1cnc(CC(=O)N(C2CCC(NC(=O)C(C)(C)O)C2)C)s1 C1(N(C(CN(C)C(=O)Nc2cnn[nH]2)=O)C)CCN(C(=O)OC(C)(C)C)C1 N1(C(C2C(CC)CCO2)=O)CCC(C2CN(C(=O)C(C)n3cccn3)C2)CC1 Cc1ccc(F)c(C(=O)NC2(CCNC(=O)CC3CCC(C)C3)CCOCC2)c1 Nc1c(C(=O)NCCC2CC(NC(c3ccoc3)=O)C2)nnc2ccccc12 c1(C(C)(C)C)ccc(C(=O)CCC(N2CCC(O)C(F)(F)C2)=O)cc1[N+](=O)[O-] C1(CC(=O)N(c2cccc3cc[nH]c23)CC(=O)O)Cc2cc(C(F)(F)F)ccc2O1 C1(S(N)(=O)=O)(C(=O)NC(CN(C(c2ocnc2C2CC2)=O)CC)C)CC1 CC(C)CC(F)(F)C(=O)NC1CCN(C(c2ccc3c(c2)OCO3)=O)CC1C C1(CCC(=O)NCCOCCOCC)CCCCN1C(=O)CCCF C1(C(N2CC3N(C(C4CCN(C)CC4)=O)C(C3)C2)=O)CC2CCCCCC12 c1(COC(N(CC(=O)OC(C2COC(=O)C2)C)CCC)=O)ccccc1Cl N1(C(c2c(C)nn(CC(F)F)c2C)=O)CC2(CC(NC(=O)CCC(C)C)CO2)C1 C(=O)(CC(O)C(C)C)N(C1CCCN(C(=O)COCCF)CC1)CC N1(C(C(F)=CC)=O)Cc2nccn2CC(NC(=O)CCC(C)N(C)C)C1 O(P1(=O)CN(c2cccc(Br)c2)C(C)=N1)CC C1(C(N2CCC(N(C(=O)Cn3ncccc3=O)C)C2)=O)CCc2nc[nH]c2C1 CC(C)C(COCC(N)=O)C(=O)N1CCCC(C(=O)NCC(N)=O)C1 c1(CC(=O)Nc2ccc(CC(=O)OCC)cc2)cc(C)c(Br)c(C)c1 C1(NC(C(C)=CC)=O)CCC(CNC(C2CC(N3CCCCC3)C2)=O)CC1 C1(Br)(C(=O)NCC(=O)NCC(C)C)CCC1 Cn1cc(C=O)c(Br)n1.N1CCC(n2cc(CN3CC4CC4C3)nn2)C1 c1(N(C(N2CCC(CCO)CC2)=O)C2CC2)cccc(Br)n1 c1(NC(C(C)Nc2ccc(-c3nc(C)on3)cc2)=O)ccc(S(C)(=O)=O)cc1 c1(CC(=O)NCCCN(C(C2(C)CS(=O)(=O)C2)=O)CC)ccc(Cl)nc1C C1(CC#C)(C(=O)NCC(=O)OCC=C)CCN(C(=O)Cn2cc(C)cn2)C1 C12C(O)C(O)CN1C(=O)N2.CS(=O)C1CN(C(C)(C)C)C1 c1(C(N2CC(OCCNC(c3cc(O)cs3)=O)C2)=O)nccc2c(F)cccc12 C(CC(=O)NCC(CC)(CC)SC)(CC(C)C)NC(C=CC)=O c1(C(C(=O)NC2C3CN(C(C4N(C(C)=O)CSC4)=O)CC32)C)ccc(F)c(F)c1 C1(CC=C)(C(=O)OCC)CCN(C(=O)C(=Cc2ccccc2F)C)CC1 N1(C(CCSCC)=O)CC(O)CC1CC(=O)NC(C)CSC c12cc(Cl)ccc1C(=O)C(=O)NC2.Cn1nncc1C1C2CNCC12 Cc1ccc(C(=O)NCCOCCc2ccc(Br)cc2)cc1C N1(CC(COCCOCC)O)CCN(C(=O)Cc2cnnn2C)CC1 c1(CC)ccc(C(=O)NC(C)(C)CNC(=O)CC2CN3CCC2CC3)cc1CC C1(CNC(C2(c3cccs3)CC2)=O)C(C)CCCN1C(c1ccc(OC)cn1)=O c1(C(=O)NCCCN(C(CCC#CC)=O)CCO)ccc(C)c2c1CCCN2 CCC(CC)CCNC(=O)C(C1CCN(C(=O)CC2CC(=O)C2)CC1)C Cc1cccc2c(C(N3CC(CNC(=O)COC(C)(C)C)CC3(C)C)=O)n[nH]c12 N1(C(C2(C#C)CC2)=O)CCOCC(NC(c2nsnc2O)=O)C1 C1(NC(c2nnc(-c3ccco3)o2)C)CCC(NC(=O)OC(C)(C)C)CC1 Cc1c(C(=O)NC2CCCC(CNC(C3CC(C)(C)C3)=O)C2)cnn1CC(F)F c1(C(=O)NCc2cccnc2Cl)ccc(OC)c(-c2c(OC)cccn2)c1 C(=O)(C(CO)C(F)(F)F)NCc1cccc(C(=O)NCC(C(C)O)O)n1 N1(C(c2c(C)csc2)=O)CCOC2(CCC(Nc3cccc(F)c3C#N)CC2)C1 N1(C(C2(C(C)C)CCC2)=O)CCOC(CC(=O)NC(C23CCC(CO2)C3)C)C1 CC1(C)CN(C(C2CC3CCC3C2)=O)CCC1NC(c1ccc(CO)c(Cl)c1)=O C(C)(CNC(=O)CNc1ccnnc1S)(C(C)C)NC(C(C)OCCC(C)C)=O c1(OC)cc(F)c(C(=O)NCC2CN(C(c3c(C)nsc3N)=O)C2)c(F)c1 c1(NC(C(CCNC(=O)C(=C2CCCCC2)F)OC)=O)ccc(C2CC2)cc1 c1(C(CCC)NC(C(=O)NC(CC#C)C)=O)ccc(O)cc1 Cc1nc(Cl)nc(N2CCC3(NC(c4c[nH]c(C(N)=O)c4)=O)CCCC23)c1F C1(NC(=O)C=CC2CC2)CN(C(=O)CCc2nc[nH]n2)C2CCCC12 C1(C(=O)NCC2CCCC2NC(c2ocnc2C2CC2)=O)(COCC)CC=CC1 N1(C(CCOCCC)=O)CCC(NC(c2ncc[nH]2)=O)C1C c1(C(N2CC3(CN(C(c4cccc(C)c4F)=O)C3)C2)=O)ccc(F)cc1C#N N1(C(c2ccc(CC)o2)=O)CC2CC(C(N3CCC3CC)=O)(C2)C1 C#Cc1ccc(C(=O)NC2CC3(NC(=O)CC4CCCC(C)(C)O4)COC2C3)nc1 N1(C(C(C)CO)=O)CCCCC(CNC(c2cncn2C)=O)CC1 Cc1nc2c(C)cc(C(N3CC4CN(C(=O)C(C)C#N)CCC34)=O)cn2n1 C1(NC(C(C(C)OC)NC(=O)C=C2CCC2)=O)CCCC(C)(C)C1 CCC(CN(C)C)C(=O)N(C)CC=CC(=O)NCC(CSC)OC CN(C)S(=O)(=O)NCC(N1CCCC1C1(O)CN(C(=O)CCc2nc[nH]n2)C1)=O CC1CCN(C(c2c[nH]c(=N)o2)=O)CC1NC(=O)Cn1cc([N+](=O)[O-])cn1 c1(CNC(N(C(CC#C)C)C)=O)cnc(NC(C)(C)C)nc1 N1(C(C(CCC)N(C)C)=O)CC(C2CN(C(c3cccc(C4CCC4)c3)=O)C2)C1 C=CCCCCCC(=O)N1CC(N2CCN(C(C3(C4CCCO4)CC3)=O)CC2)C1 C#Cc1cnc(C(=O)NC2CC(O)C2CC(=O)NCC(CCC)CCCC)c(C)c1 c1(C(=O)NC2C(C(=O)NCCC(=O)NC)C2)ccc(SC)o1 C1(NC(CC=C)=O)CCC(CNC(C2(c3ccccc3)COC2)=O)C1 C(C)(CCC(=O)NCCc1cccnc1)NC(C1C(C(=O)OC)COC1)=O Cc1nnc(SN2CCCSCC2)n1C(c1ccccc1)C c1(C(=O)NCC2(O)CC(NC(C3C4CNC(=O)C34)=O)C2)cccc2c1OCCC2 C1(NC(=O)C(O)CN2CCOCC2)CC2(C1)CC2NC(c1csc(Cl)n1)=O N1(C(C(C(C)C)NS(C)(=O)=O)=O)CC2(C1)CN(C(=O)CS(=O)(=O)C1CC1)C2 O=C(C1CCOc2ccc(Cl)cc21)NC1CCN(C(C2(C(F)(F)F)CCC2)=O)C1 c1(NC)ccc([N+](=O)[O-])cc1C(N1CCC(NC(=O)COC)C1)=O S(=O)(=O)(c1cccc(=NCC(C)C(C)O)[nH]1)N(CC)Cc1cccs1 C12(CC)CN(C(=O)CCOC3CCOC3)C(CNC(c3nc(=O)n(C)[nH]3)=O)(C1)C2 C1(CNC(COC)Cc2ccc(F)cc2)COCC(=O)N1C C(=O)(CCCC(C)O)N1CC(C2OCCN(C(Cc3c(C)nn(C)c3)=O)C2)C1 Cc1cc(C(=O)NC(C)C(C)(C)NC(=O)C=Cc2c[nH]nc2C)ncc1C(N)=O N#CCCCCC(=O)NC12CCC(CC1NC(C1CS(=O)(=O)C1)=O)C2 C1(NC(CC2(C=C)CC2)=O)CC(C)(NC(c2ccsc2C(F)F)=O)C1 C1(C(N(CCCN(C(=O)COC2CCCOC2)C)C)=O)Cc2cscc2C1 c1(C(=O)NCCN(C(C(C=C)O)=O)C)cc(C)ncn1 c1(C(N2CCC(N)(SC)C2)=O)ccc([N+](=O)[O-])nc1 N1(c2nccc(C)n2)CC(NC(=O)CSc2cccc(Cl)c2)C(C)(C)C1 c1(C(=O)NC2(C(N3CCCC(CC(=O)NC)C3)=O)CCC2)nc(C)ccc1F n1(CC(=O)NCC=CCNC(c2cc(C)c(Cl)s2)=O)ncn2cccc2c1=O C1(C(C)C)CCCN(C(=O)NCCC2CC2)CC1 c1(SC)cc(C(N2CCN(C(c3ccc(C)nc3O)=O)CC2CO)=O)cc(Cl)c1 CC(=O)C(C)(C)CC(=O)NC(C1CCN(C(=O)CC(C)C(F)F)CC1)C Cc1cc2c(N(C3CCNCCC3(F)F)C(c3cncnc3)=O)ncnc2[nH]1 N1(C(C(C)N(C(C)=O)C)=O)CC(O)(C2(CNC(=O)CCCN(C)C)CC2)C1 c1(C(C(N2CC(NC(Cc3c(C)ncs3)=O)C2)=O)N(C)C)ccc(F)cc1 C1(C(c2nnnn2C)C)CCC2(CCCCC2)O1.n12nnc(n1)CNC2 O=C(C#CC1CCC1)NC1CCC1CNC(C1(C2CCCO2)CCCC1)=O c1(OC)cc(C#N)ccc1C(=O)NCC1CN(C(=O)CCCCOC)CCCO1 C(=O)(C1=C(C)CCC1)NCC(CO)NC(C(c1cccc(OC)c1)C)=O Cc1ccnc(C(=O)NC(C)(CNC(=O)CC2(n3ccnc3)CC2)CO)c1N N1(C(CC(=O)NCC#C)=O)CCC2(CC1)CC2NC(c1n[nH]cc1C)=O c1(C(N2CC(NC(C3SCCS3)=O)C(F)CC2)=O)ccc2nc(O)[nH]c2n1 C(=O)(CCC1=CCCCC1)NC(C(=O)NC(c1cncs1)C)CO CC1=C(C)CC(C)(C(=O)N(CCCCNC(C2CCCCN(C)C2=O)=O)C)CC1 Cc1nc(C)n(O)c1C(=O)NC(CO)C(C)NC(c1c(C)ccn1C)=O N1(C(C(=O)NC(c2cc(Br)ccc2F)C#C)C)C(=O)c2ccccc2C1=O C(=O)(C1CCCc2nccn21)N1CC(C)C(NC(C2CCc3nccn3C2)=O)C1 C1(C(=O)NCC2CCN(C(c3c(C)cnn3C)=O)C2)CCCC(F)(F)CC1 Cc1cnn(C)c1C(=O)NC(C1CCCN1C(C1CCCC1c1nc[nH]n1)=O)C N1(C(COC(C)=O)=O)CCC(NC(=O)C2CC2)C12CC2.C1CCC(=O)N1 C1(CNC(C2(CCOC)CCCC2)=O)CN(C(C2(C)CCCS2)=O)CCCO1 c1(CC)ccccc1C(C(=O)Oc1ccccc1C)NC(C1CCCC1)C CC(C)CCC(F)C(=O)NCc1ncoc1CCNC(=O)C1=C(Cl)CCCC1 c1(OC)ccc2c(c1C(N1CCCC(NC(=O)CC3C=CCCC3)C1)=O)CCC2 c1(C(N(C(c2cn(C3COC3)nn2)C)C)=O)cc(S(=O)(=O)N(C)C)ccc1I N1(C(c2c(CC)scc2)=O)CC2CCN(C(=O)Cc3ccc([N+](=O)[O-])cc3)CC2C1 N1(C(c2cc(OC)ncn2)=O)CC2(CCCC2)C1C(=O)NOCCCC1CC1 Cc1[nH]c(C(=O)NC2C=CCN(C(=O)CC3CCCC(C)C3)C2)c(C)c1C C1(CNC(CSCC=C)=O)CC2(CCN(C(c3ccc(OC)nc3)=O)CC2)CO1 N1(C(c2cccc(OC)c2)=O)CCN(C(c2ccc(F)cn2)=O)CC(C)(F)C1 c1(OC)ccc2nc(N3CCN(c4ccnc(O)c4)CC3)c(Br)n2n1 N1(C(C2CN(C(C)=O)C2)=O)CC2(NC(c3[nH]nnc3C3CC3)=O)CC1C2 CC(C)(CNC(c1ccn2cncc2c1)=O)C(=O)N1CC(C)(O)CO1 c1(NCc2c(C)ccc(F)c2)nc(=NC(C)c2ncccn2)[nH]c2ncn(C)c12 C(=O)(C(F)CCC(C)C)NCC(C(=O)NCc1ccc(OC)cc1)O Cc1cn(C)nc1C(=O)NC1CCCC1(C)CN(C)C(c1ccc(F)cc1)=O CCC1=NOC(NC(=O)C=CC(C)(C)NC(=O)CC(C)C2CCCO2)C1 C1(O)(C(N2CC(NC(=O)C(F)(F)c3cncs3)C(O)C2)=O)CCCCCC1 c1(OCCOC)cccnc1C(N1CCC1CC(=O)NCC1(C)CC1(Cl)Cl)=O c1(CCCOC)nc(-c2cnn(-c3ccccn3)c2)n(-c2ccc(F)nc2)n1 c1(NCC(CCC)OC)nc(N2CCC(C3CC3)C2)nc2c1ncn2CC C1(C)(CC)C=C(C(=O)NC(CC(N)=O)C(=O)NCC2CCOC(C)(C)C2)C1 c1(C(=O)NC2CN(C(CC3CC(N(C)C)C3)=O)CC23CC3)ccn2cnnc2c1 O=C(C1=CCCN(C(=O)C=Cc2ccsc2)C1)NC1CCOC(C2CC2)C1 CCC(CC(F)(F)F)C(=O)NC1(c2ccc(F)c([N+](=O)[O-])c2)CC1 n1(CC)ncc(C(=O)NC(C)C(C)NC(c2cc(C(F)(F)F)on2)=O)c1C N1(C(c2cc(C(C)=O)oc2C)=O)CCCC2CCN(C(=O)CC3=CCCC3)CC12 C(C)(C(CC(=O)N1CCC12CC(CNC(C1CC1C1CCCO1)=O)C2)OC)OC c1(C(=O)NC2C(NC(Cc3ccc(C)cc3Cl)=O)CC2)cc(F)cc([N+](=O)[O-])c1 c1(C(N2CCC(NC(C(C(=O)OC)C)=O)CC2C)=O)cc(C)cc2ccncc12 CCC(O)C(F)(F)C(=O)N1CC(O)(C(C)NC(c2cn(CC)nn2)=O)C1 C(CC(=O)Nc1cnc(SC)nc1)(C(F)F)NC(C(C)OCC)=O N1(C(=O)Nc2nccc3c2CN(C(C)C)C3)CCC2(CC1)OCCc1ccsc12 C#CCC(C(=O)NCC1CCCN(C(=O)Cc2cscn2)C1)C1CC1 c1(C(N(C)CC2CCCN2C(C2(C)CC3(CC3)C2)=O)=O)ccc2c(ccn2C)c1 C(=O)(C(C(CC)CC)OC)NCC(CCC)NC(C1CS(=O)C1)=O C#Cc1cnc(C(N2CCCC(C(C)C(=O)NCC(C)CCO)C2)=O)c(C)c1 Cc1c(NC(=O)C(CCOCCO)NC(=O)C(C)C(F)F)cnn1C(C)C C(=O)(C(Cn1ccnn1)NC(C1CCCC1F)=O)N1CC(C(C)C)C1 C(=O)(C(C)(C)C(C)(C)c1ccccc1)N(CC(C)NC(c1ccncn1)=O)C C(=O)(C(CNC(C1CNC(=O)O1)=O)CC1CCCC1)Nc1cn(CCC)nc1 C1(O)(CN(C)C(=O)COc2cccnc2)CN(C(c2cc(CO)on2)=O)C1 C1(C(C)NC(C2(CC=C)CCC2)=O)CCCN(C(=O)C=CCN(C)C)C1 C(=O)(C1=C(Cl)CCOC1)N1CCN(CC(N2CCN(C)C(C3CC3)C2)=O)CC1 CC1(C(=O)NCCCCC2(NC(c3coc(C4CC4)n3)=O)CC2)CC2(CC2)C1 N1(CC(N2CCC(N(C(CC3(NC(C)=O)CC3)=O)C)C2)=O)CCC(F)CC1 CCC(C)(O)C(=O)N1CCC(CNC(=O)C(c2ccc(Cl)nc2)(C)C)C1 Cc1cc(C(=O)N(C)CC2CCCN2C(c2ccc(Br)c(F)c2)=O)c(C)cn1 c1(C2(C(=O)NC34CC(NC(C(C)=C(CC)C)=O)(C3)C4)CCCC2)ccc(C)cc1 C1(C(N(C)Cc2cn[nH]c2)=O)CC12CCN(C(C1CC1C#N)=O)CC2 C1(C(=O)NCCOC(N(C)C)=O)C2C(CN1C(c1nnc(C(F)(F)F)o1)=O)C2(C)C c1(C(=O)NCCC2(O)CN(C(C3C(CC)CCC3)=O)C2)cc(Br)oc1C C1(NC(C2C(CC)CCN2C(=O)CN2CCCC2)=O)CCCC1C1CC1 c1(CC(=O)NCC2(C)CCN(C(=O)CO)C2)c(F)ccc(Br)c1F c1(OCC)cc(N2CCC(C)(CNC(C3OCCC3C)=O)CC2)nc(C)n1 Oc1nc(NC2CC2)nc2c1ncn2Cc1cc(Cl)ccc1-c1ccncc1F N1(C(CCC(N)=O)=O)CC2CCC1C1CN(C(C3(O)CCOC3)=O)CC21 c1(C(N2C(CO)CC(NC(CC=CC=C)=O)C2)=O)nc2cnccc2s1 C1(NC(C2CCCN(C(c3n(CC)ccc3)=O)C2)=O)CC2CN(C(C)=O)CC12 c1(CC(N2CC(N(C(C(C)C(F)(F)F)=O)C)C(O)C2)=O)c[nH]c2ccncc12 c1(OC)ncccc1S(=O)(=O)NC(=O)CC1COCC(C)(C)O1 c1(C(N(CCC(C(C)C)NC(C(C(CC)C)OC)=O)C)=O)cccc2cncn12 c1(C(=O)NC2C3(CC(NC(C4C(C=C)OCC4)=O)C3)C2)cccc2c1ccn2C C1(NC(C2C(C)(C(C)C)C2)=O)CCCN(C(c2cnn(C)c2C2CC2)=O)CC1 C(=O)(C(C)C(C)COC)NCCOCCNC(C1(C(=O)CC)CC(=C)C1)=O.C1(C)CC1 C(C)(CNC(=O)COCC1CCC1)(C(C)C)NC(C(n1ncc(C)c1)C)=O C1(C(=O)Nc2ccc(=O)n(C)c2)(NC)CCCN(C(c2ccnc(OC)c2)=O)C1 n1(CC)cc(CC(=O)NCC2CC2NC(=O)C(c2ccc(OC)cc2)(C)O)c(C)n1 CC(C)C(C(=O)NCCC1CC(NC(c2cc(O)cs2)=O)C1)C1CCCCC1 C1(C)(C(N2CC(NC(CSCCC)=O)C(OC)C2)=O)CC(C(C)C)=NO1 CCC(CC)(C(C)C)NC(c1cc(CNC(C2CC(O)C(F)C2)=O)on1)=O N1(C(C(CC(=C)Cl)NC(=O)CN(CC)CC)=O)CCc2cccc(O)c21 N1(C(c2c(C=C)cnn2C)=O)CCCC2(CC(NC(C3CCC(=O)NC3)=O)C2)C1 c1(C(=O)NCC(CN(C(=O)CC2COCCO2)C)O)ccc2c(c1)C(=O)CCO2 C1(C(N(C(C)CCNC(=O)C(F)C(C)(C)O)C)=O)CCC2(CCC2)CC1 N1(C(CC2(CC)CCCC2)=O)CCN(C(=O)C=CC(=O)NC2CC2)C(C2CC2)C1 C(C)(CS(C)(=O)=O)NC(C(C1CN(C(CCOC)=O)C1)OCCC)=O c1(C(N2CCC3C(CCN3c3cc(O)ncn3)C2)=O)c[nH]c2ccccc2c1=O C1(C(=O)NC(CNC(c2cccc(SCCC)c2)=O)C)CCc2cnc(C)n2C1 C(c1ccc([N+](=O)[O-])s1)=CC(=O)NCCCCCNC(C1CC1c1nc[nH]n1)=O N1(C(C2CC(C)(CC)C2)=O)CCC(CCOC)(NC(=O)CCc2nccs2)CC1 c1(C(N2CCC(CN(C)C(C3CC3(Cl)Cl)=O)C2)=O)nnc(O)cc1O n1(CC)ccc(C(=O)NC(C(C)NC(C23CSCC2C3)=O)C(C)C)cc1=O n1(CC(N2CC3C(NC(C4(CC=C)CC4)=O)C(C3)C2)=O)nc(C)c2cccnc12 c1(CC(C)NC(C2CCN(C(=O)CC3CCCN3C)CC2)=O)ccc(F)c(F)c1 N1(C(c2ccnc(C)n2)=O)CC(C(=O)NC(C)C(C)n2cccn2)OC(C)C1 c1(N(C(c2ccccc2F)(C)C)C)ncccc1NC(=O)OC(C)(C)C C=C(Cl)CCC(=O)NC1(C2CCCN2C(=O)CN2CCCC2)CC1 N1(C(CCNC(N)=O)=O)CC(n2cc(-c3ncccc3Br)nn2)C(O)C1 N1(C(C2CN(CCOC)C(=O)C2)=O)CCC2(NC(c3ccc(C)o3)=O)CC2C1 C1(CC(=O)N(C2CCN(C(=O)NC3CC4CC4C3)CC2)CCC#N)SC(=N)NC1=O N1(C(c2c(C)onc2O)=O)CCC(C)(CNC(C2(C)CCCC2C)=O)CC1 C1(C(=O)NCCC(=O)NCCOC)CC(C)(C)CCN1C(=O)Cc1ccsn1 N1(C(C(c2ccc(Cl)s2)C)=O)CCC(N(C)C(C2CC(n3cncn3)C2)=O)CC1 C=CCC(CNC(=O)C=Cc1cncn1C)C(=O)Nc1cscc1CC c1(C(N2CCC(CNC(=O)CCCC(F)(F)F)C2)=O)cnc2ncc(Br)cc2c1 CC(C)C(C)CC(=O)NCC1CCN(C(c2csc3cncn23)=O)C1 C1(C(=O)Nc2ccc(Cl)c(O)c2)CCN(C(=O)CCCN2CCCCCC2)O1 CC(CC(F)F)C(=O)N1CCC(O)CC1C(=O)NCc1cccc(O)c1 C1(CNC(CN(S(CC)(=O)=O)C)=O)CC(C)(C)CN1C(C1CCC(C)(C)OC1)=O c1(C(N2C(CNC(CCCC)=O)CCC(C)C2)=O)cc2c(s1)CCCC2 C=CCC(C(=O)NCC(CC(C)C)C(=O)N(CCCCSC(C)(C)C)C)C(C)C C12(NC(CC3CC(NCc4n(C(C)(C)C)nnn4)C3)=O)CCCCC1OCC2 CC(CC(=O)N(C)CC1CCN(C(C2CC3CC2C2CC32)=O)C1)P(C)(C)=O c1(C(N2C(CCNC(C3(OC)CC(C)C3)=O)CCCC2)=O)ccnc2[nH]ncc12 Cc1cc(Cl)c(C(=O)N(CC(C)CNC(c2cncs2)=O)C)s1 C(=O)(C(C(=O)NC1CC(NC(=O)CC(F)(F)Cl)C1)C1CCCC1)OC(C)(C)C C1(C(C)NC(c2cnsc2)=O)CN(C(C2CCCO2)=O)CCO1 S(=O)(=O)(c1ccc(N)cc1)NC(C12CCC(CC1)N2CS(=O)(=O)c1ccc(Br)s1)C c1(C(=O)NC(CC#CC)C(=O)N(C)CC2COC(=O)N2)cccn2ccnc12 c1(OC)ccc(C(=O)NC2COCCN(C(c3cc(Cl)ccn3)=O)C2)c(F)c1 c1(Cc2n(C(=O)OC)nc(Br)n2)ccc(Br)c(N2CCCC2)c1 CCCC(C(O)C(=O)NCc1ccc(C)c(F)c1)NC(c1c[nH]c(C)c1)=O N(C(=NCc1ccnn1C)NC1CCN(C(=O)CC)C1)Cc1ccn(CCC)n1 N1(C(C(C)OCCOC)=O)CC(NC(=O)CN2CSCCSC2)C(C)C1 N1(C(CCN(C)CC)=O)CCC(O)(C(C)NC(C2(C(C)(F)F)CCOCC2)=O)C1 CC1CN(C(=O)CCC=CCNC(=O)C(F)(F)c2ccncc2)CC(C(N)=O)O1 C1(C(N2CC(C)(C)C(CNC(=O)C3CC3)C2)=O)CC2(C1)C(F)(F)C21CCC1 CC(CC(=O)N1CC2CCC1C(NC(C1(CC3CC3)CC1)=O)C2)C(C)(C)C CCCC(C)(CCC)C(=O)NCC1CCC(NC(=O)C(C)OCC(C)C)CC1 n1(CC(=O)N(C2CCN(C(=O)COCC(=C)C)C2)CC#C)ncc(Br)n1 C(=O)(CCCC(=O)NCC1CCCN1C)OCC.n12cc(nn1)C(=O)NCC2 C(=O)(C(C)CCC(C)(C)C)NCC1C(OCC)CN(C(=O)CC(C)C(C)C)C1 Cc1ccc(C(N2CC(CNC(=O)C(O)c3ccco3)C2)=O)c([N+](=O)[O-])c1 CCC(O)C(=O)N1CCCC1CC(=O)Nc1ccncn1 c1(CN(C(=O)Cc2ccc(N(C)C)cc2)C)cccc([N+](=O)[O-])c1S(C)(=O)=O C12(C(=O)Nc3cccc(NC(C4CCC(CC)C4)=O)c3)CCC(=O)N1CCS2 Cc1nn(C)cc1C(O)C(=O)N1CC(N(C(=O)COC2(C)CCC2)C2CC2)C1 N1(C(C(CC)C)=O)CCn2nc(CNC(C3CC(CC4CC4)C3)=O)cc2C1 C1(C(N2CC3CN(C(CCCOC(C)=O)=O)CC32)=O)Cc2ccccc2O1 C1(NC(C(C)OCOC)=O)CN(C(=O)CC2(O)CCCC2)C(C)(C)C1 c1(N(CC(=O)NCCOC)C)nc(=NC(C)c2cnc[nH]2)[nH]c2c1CCCC2 C1(C(=O)NCCCN(C(CSCC#C)=O)C)Cc2ccccc2O1 N1(C(CN(C(CC2C(=O)OCC2)=O)C2CCC2)=O)Cc2cccc(F)c2C1 N1(C(CSCC(=O)OC)=O)CCC(CO)(NC(=O)C(C)COc2ccccc2)CC1 c1(C(C)=O)cccnc1OC(F)(F)F.C1CCCN1C1CCCC1 c1(CC)cccc(C(=O)N(CCCNC(C2CSCCS2)=O)CCO)c1O CN1CCN(C(c2cccnc2C2CC2)=O)CC1C(=O)NC1CC(C)(O)C1 CCCS(=O)(=O)C(C)C(=O)N1CC2(CCN(C(C3CCCCS3)=O)CC2)C1 c1(OC(F)(F)F)ccc(C(=O)NCC(n2cc(CN)nn2)C)nn1.CC(C)O C=CCC(CC)C(=O)N1CCC(CNC(=O)CCn2c(C)csc2=O)CC1 c1(CN2C(c3scc(C(=O)OC)n3)CCC2)c[nH]c2ccc(C#N)cc12 Cc1ccc(C(CCc2ccc(C)o2)NC(=O)Nc2nc(C(F)(F)F)cs2)cc1 CC(C)(C)C(C)(C)C(=O)N1CC(NC(c2cnc(C(N)=O)s2)=O)C1 C1(NC(CCCCC=C)=O)CN(C(c2scnc2Cl)=O)CC2(CCOCC2)C1 c1(-c2n(CCOC)nc(-c3cccs3)n2)ccc2c(c1)C(C)CO2 c1(OCC)ccccc1C(C(=O)NO)NC(C1(C(=O)OC)CC1C(F)(F)F)=O C(=O)(CC(C)(C)C(=O)OC(C)(C)C)NC1CC(NC(c2cc(OC)nc(Cl)c2)=O)C1 C1(C)(CNC(CC2CC(C(=O)OCC)C2)=O)CCCN1C(=O)Cc1cn[nH]c1 Cc1cccc(C(=O)NC(COC(C)C)C(=O)NCCC2CC2C)c1C#N N1(C(CCCC=C)=O)CC(NC(c2cccc(Cl)c2OC)=O)CCC1C C(=O)(C(C)(COC)OC)NC1CC(C(C)NC(C(C2CCCC2)OCC)=O)C1 N1(C(CCC=C)=O)CCC2(CC1)CC(NC(C1(CC(C)C)CC1)=O)CO2 N1(C(=O)NC(C#C)CC)CCOc2cc(Cl)ccc21 c1(C(=O)NCCC(C)NC(CCNC(C)=O)=O)cccc2c1oc(=O)n2C Cc1ccnc(C(=O)N(C(C)(C(=O)NC2C=CCCCC2)C2CC2)C)c1F C1(CC)(NC(C2(C)CC(F)(F)C2)=O)CCN(C(=O)C(C)Oc2ccccc2)CC1 CC1(C)CN(C(c2cc(CO)on2)=O)CC1NC(=O)CN1CC2CC2C1 C(=O)(CCC(O)C(C)(C)C)NCC1OCCN(C(c2cc(Cl)cc(C)c2N)=O)C1 c1(CC(=O)NC2C(NC(CC3C(C)CCC3)=O)CCC2)sc(O)nc1O c1(C(=O)NCC2(F)CCCN(C(C(F)=CC)=O)C2)ccn2ccnc2n1 C1(O)(C(=O)NCC2=CCN(C(C=C(C)C(F)F)=O)CC2)CCc2ccccc2C1 N1(C(c2nc(C)n(C)n2)=O)CCN(C(=O)C(F)C(C)C)C(C)C1 C(C(C)(C)CC(=O)NCCCC(C)NC(=O)C(C)C1CCCC1)OC C1(CC=C)(NC(=O)CC2(CC)CCOCC2)CCCN(C(=O)C(C(=O)OC)OC)C1 N1(C(c2cncc(SCC)n2)=O)CCC2CN(C(c3cnc(C)nc3)=O)CCC12 C(=O)(C1=CCCCCC1)NC1CC(NC(c2cc(C)nn2C2CCC2)=O)C1 C1(C(=O)NCC2CN(C(C(CC)O)=O)CC2C)CC(C2CC2)=NO1 N1(C(c2ccc(C(C)(C)C)o2)=O)CC(CNC(=O)CC2COCCO2)C(O)C1 C1(OC)CC(C(=O)NC2C=CCN(C(c3ccc(Cl)s3)=O)C2)C12CCC2 N1(C(C(C)(F)F)=O)CC2CC(C(=O)NC3(CCO)CCC3)CC2C1 C1(C(CNC(C2N(C(C)=O)CC2)=O)F)CCN(C(c2oc(CO)cc2C)=O)CC1 c1(C(N(CCCNC(C(F)OCC)=O)C2CC2)=O)coc(SC)c1 c1(C(N(CC(C)N(C(C(=Cc2ccncc2)C)=O)C)C)=O)c(F)ccc(F)c1O Nc1cccc2ccc(C(=O)NC34CC3CN(C(C3CC3C(F)F)=O)C4)nc12 C1=CCCOC(CNCCN2CCC(CC3CCCCC3)CC2)C1 c1(C(=O)NCC2N(C(C(C)C)=O)CC(C(F)(F)F)C2)cc2c([nH]1)CCCC2 C1(Cc2ncc(CC)s2)CCN(C(=O)C(c2cccc(Cl)c2)N)CC1 C12(NC(COCC)=O)CC3CCC(C1C2)N3C(C1CCCC1c1nncn1C)=O Cn1c(C(N2CCC(CCNC(C3CCCC4(CC4)C3)=O)C2)=O)cc2sccc12 c12ccc(cc1)OC2.Cn1cc(CC(=O)NC2CC2NC(c2cnn[nH]2)=O)cn1 C1(C(=O)NC2CN(Cc3ccccc3)CC(C)O2)C2C3CCC(C3)C12 C1(O)(C(C(=O)NCCN(CCO)CC)F)CN(C(=O)C(C)N2CC(C)C2)C1 c1(-c2cn(CCCC3N(C(CC4(C)CCCC4)=O)CCC3)nn2)ccnc(O)c1 C#Cc1cnn(C)c1C(=O)NC1CC2(C1)CC2NC(=O)Cn1nnc(C2CC2)n1 c1(CNC(C2N(C(c3nccc(CC)c3)=O)CC(C)C2)=O)cc(Cl)c(Br)cn1 Cc1cnc(O)cc1NC(CC(C)(C)C#N)c1nnnn1C1CCC1 CCCCCC(O)CNC(=O)C(C)(C)CNC(=O)C(C)CCOC C1(NC(CC2(NC(c3c(C)cc(C)s3)=O)CC2)=O)CN(C)CC12CC2 C#Cc1cc(NC(c2conc2CNC(c2[nH]ccc2CC)=O)=O)cc(F)c1 C1(C(=O)NCc2cc(OCC)no2)CCC(C)CN1C(c1cc(CC)ccn1)=O N1(CC2CC(C(=O)NC(CC)(C)C)C2)CC2(CCN(CC(C)(C)O)C2)C1 C#Cc1cc(C(=O)NCCC2CCCN2C(=O)C2=C(C)OCC2)ccc1C S(=O)(=O)(c1cn[nH]c1)NC1C=CC(C(=O)N(c2cccnc2Cl)CCO)C1 C1(NC(C2CCC(O)CC2)=O)CC(NC(C23CCCC2(C(=O)O)C3)=O)CC1O C=Cn1nncc1C(=O)NC(C(=O)NC(COC)C1CCC1)C(C)C c1(C(N2C(CNC(C(C)C3=CCCC3)=O)C=CC2)=O)ccc2oc(O)nc2c1 c1(C(=O)NC(C)CC2CN(C(C3(O)CCSC3)=O)C2)ncccc1Br N1(C(CCC2CCC(C)O2)=O)CCC(C2(NC(=O)CC3(C)CC3)CC2)C1 N1(C(C(C)Cc2ccncc2)=O)CC(NC(C2(CO)CCC2)=O)C(C2CC2)C1 CC(C)CC(C)(O)c1cn(-c2cncc(C(=O)N(C3CCN(C)C3)C)c2)nn1 C1(C(=O)NCC23CCN(CC2)CC3)CCCCN(C(=O)CSCC(F)(F)F)C1 C(=O)(CCCC(C)(C)NC(=O)CSC(F)(F)F)NC(c1n(CC)ncn1)C C1(N(C(=O)C=Cc2ccco2)CC)CCN(C(=O)C(O)CCSC)CC1 N1(c2ncnc(C)c2Br)CCC(C2CCN(C(C3(CCF)CC3)=O)CC2)CC1 C(C(C(F)(F)F)N1CCN(C(=O)C(F)=C(C)C)CC1)NC(C1C(OC)CCC1)=O C1(SCC)C(NC(c2nncn2C)=O)CCN1C(=O)C(C)Oc1ccccc1Cl C1(C(=O)NC2(CN(C(=O)CNC(=O)C(C)(C)C)CC)CC2)CSCN1C N1(C(c2c(C)nsc2C)=O)CC(C(=O)O)CC2=CCC12 CCP1(=O)CC(C)CN(C(=O)CC(O)C(C)(C)C)C1 N1(C(c2cnc(OC)nc2)=O)CCCC2(NC(c3nc(C)c(C)s3)=O)CC2C1 C1(C(N2C(=O)CN2CC)=O)CC(O)CN1C(=O)CC(F)F.c1(CC)ccccc1 Cc1csc2[nH]c(C(=O)NC3CCC(NC(C4(C(F)F)CCCC4)=O)CC3)cc12 C1(NC(c2cc3c(s2)CCC3)=O)CC2CN(C(C3CCCC3(F)F)=O)CC2C1 c1(OC)ccc(Cl)c(CC(N2CCN(C(=O)CC#N)CC2c2nccn2C)=O)c1 C1(CC)CN(C(=O)C(c2ccccn2)C)CCN1C(c1ccc(F)cc1Br)=O N1(C(C(CCSC)OC)=O)CCN(C)C(CNC(c2c(F)cccc2Cl)=O)C1 N1(C(C(C(C)(C)C)N(C)C)=O)CCC(CCNC(c2cncc(Cl)c2)=O)CC1 C(=O)(CC(F)(F)C(F)(F)F)NCC1CCCC(CNC(C(CSC)C)=O)C1 c1(CN(C)C(=O)NCC(C2CCC(=O)N2)(C)C)cc2cc(Cl)ccc2[nH]1 C(=O)(C1=NOC2(CCC2)C1)N1C(C)C(C(=O)NCCCc2ccsc2)CC1 C1(C(=O)NN(C)C(C2(CC3CC(=C)C3)CCCC2C)=O)CC2CCC1CC2 c1(C(N2CCC(NC(c3c(CC)onc3C)=O)C2)=O)cccn2cnnc12 N1(C(CCc2ncc(C)[nH]2)=O)CCC(CO)(NC(c2cnn(C)c2Br)=O)C1 C1(CC=C)(N)CCNC1.C(=O)(CCCC1CCCCC1)C(C1(CCN(C)C)CC1)=O N1(C(=O)C2CC2)CCC(O)(NCc2cc(OC)ncc2)CC1 C1(OC)CC(C(=O)OC)CN(C(c2ccc(C(C)(C)C#N)cc2)=O)C1 c1(CC(=O)N(CCC)CCNC(C2C3COCC23)=O)cccc(OC)c1F C1(NC(CC2CCN(C)C2=O)=O)CCN(C(C2(F)CCCC2)=O)CC1(C)C C1(C(=O)Nc2cn(C)nc2C)(CC)CCN(C(=O)CC(=O)NC2CC2)C1 C1(CC=C)(NC(C2CCC(=O)N2C)=O)CCCN(C(c2nc(O)sc2C)=O)C1 C1(=O)CCCC(=O)C(=O)c2coc(n2)CNC(=O)CC2(C)CCN12.COOC c1(C(C)C)cc(NC(C2C3CC2N(C(c2cc(Br)cs2)=O)C3)=O)n(C)n1 C1(CNC(C23CCCCC2C3)=O)CN(C(c2cc(=O)cc[nH]2)=O)CCCO1 N1(C(Cn2ncc(C#C)c2)=O)CCCC(CC=C)(NC(=O)CCNC(=O)CC)C1 N1(C(CCC(C)SC)=O)CC(CNC(c2cc(Br)n(C)c2)=O)C2(CC2)C1 Cc1nn(C)c(C)c1C(=O)NC1CCCN(Cc2noc(C(C)(C)C)n2)C1 Cc1sc(S(=O)(=O)Nc2c(F)cc(F)c(F)c2F)cc1[N+](=O)[O-] C1(C(=O)NC)C2CN(CC(c3cccc(OC4CC4)c3)=O)CC12.OC C1(NCc2c(Cl)ccs2)CC2(CO)COC1C2 C1(N(C)C(C2CCCS2)=O)CCCN(Cc2cn(-c3ccn(C)n3)nn2)C1 c1(C(C(=O)N(CCC(=O)NCC2CC2CNC)C)S(C)(=O)=O)ccccc1.CC C1(C(=O)Nc2onc(C)n2)CCCN(C(CC2CCCO2)C(=O)NC(C)C)C1 CCC1=C(C(=O)N2CC(C(=O)NC(C)(C(=O)OC)C3CC3)CC23CCC3)CCCO1 Cc1nc(CC(N2CC(NC(c3nn[nH]c3Cl)=O)C(C)C2)=O)c(Cl)s1 N1(CCCC(=O)NCCCOC)CC=CC(O)C1 CCCCC(C)CCC(=O)N1C2CC1CN(C(c1ccc(Br)c(Cl)c1)=O)C2 C=CCC(CC(F)F)C(=O)N1CC(N(C)C(C2CN(C)C(=O)N2)=O)C2(CC2)C1 Cc1cc(=NC(CNC(c2cccc(C3CCOC3)c2)=O)C(C)C)[nH]c(Cl)n1 C123CCCC1CN(C2)C(=O)c1ccnc(c1)N3.C1(C=O)CC2CC(=O)C1C2.CO N1(C(CCOC(C)=O)=O)CCC(O)(CNC(c2cc(C3CCCO3)n(C)n2)=O)C1 c1(C(=O)NCC2CCCN(C(C(CC)CO)=O)C2)ccc(C(C)C)nc1C CCCCCC(CC)C(=O)NC1CCN(C(c2ccc(N)cc2OC)=O)C(C)C1 C=CCCCCCCC(=O)N1CCCC1CNC(C1COC(C)(C)O1)=O N1(C(=O)NCCOCC(C2CC2)OC)CC2C(CO)C2C1 C1(c2n(CCCC)nnn2)(Nc2ccc(C(=O)OC)nc2)CCOC(OC)C1 C(=O)(C(O)C(O)C(=O)NC(c1ccccc1CCC(F)(F)F)=O)OC(C)(C)C N1(C(=O)NCC2CCC(c3ccc(OC)cc3)C2)CC(C)C(CO)CC1C C=CCCCCCCN=c1nc2cccc(Br)c2c(NC2CNC(=O)C2)[nH]1 C1(OCC(=O)OC2CCN(c3ccccc3C(F)(F)F)C2=O)CCCC(F)(F)C1 c1(C(=O)OCC)cc(C)c(NC(N(C(C2(N)CCOC2)C)CC)=O)o1 C=CCC(F)(F)C(=O)NCC1CCCN(C(c2ccc(CC#N)cc2)=O)C1 C1(CC=C)(C(=O)NCCC2(C)CCOC2)CCCN1C(C1COCCO1)=O C(=O)(C1Cc2c(Cl)cccc21)NC(C(CO)NC(CNC(CC)=O)=O)C Cn1nccc1C(C)(C)C(=O)NC1CC1NC(C1(c2ccccc2)CC1(Cl)Cl)=O C1(F)(CNC(CCOCC#C)=O)CCCN(C(=O)Cc2ccc(Cl)nc2)C1 c1(C(=O)NC(C)C(C)NC(C2CCC(C(F)(F)F)CC2)=O)cc(O)cc(F)c1F C1(NC(=O)CN2CCOCC2)CCC12CN(C(C13C4C5C6C4C1C6C35)=O)C2 c1(CC(=O)NC(CNC(c2c(C)c(C(C)C)[nH]n2)=O)(C)C)cccc2nonc12 Nc1ccc(S(N)(=O)=O)cc1C(=O)OCc1ccc(=N)[nH]c1 c1(C(N2CC(C)N(C(=O)CCCn3ccnc3)CC2)=O)ccc2ncccc2n1 C1(C)(CNC(COCCOCC#C)=O)CCN(C(=O)CN2CC3CC3C2)C1 C1(C(N(CCCN(C)C(c2cc(N)nc(Cl)c2)=O)C)=O)CC2CCC(C1)C2F Cc1c(C(=O)NC2CCCC2(C)CN(C)C(C2C(C)C2C)=O)cnn1C Nc1c(Cl)c(C(N2CC(C(=O)O)OCC23COC3)=O)cc(F)c1Br C1(C(=O)OC)C(C(F)(F)F)CCN1CCS(=O)Cc1cnn(C)c1 c1(CC(C(=O)NCC2(NC(C34CC(C)C3C4)=O)CC2)O)cccc(Cl)c1Cl CC1(C)CCC(C(=O)NCC(O)CC2CCC2)(NC(C2CC3CCC3C2)=O)C1 c1(C(N2C(C)C(N3CCOCC3)CC2)=O)cc2c(s1)CCCCC2 C1(NC(c2c(C(N)=O)coc2)=O)COC2(CNC(c3cn4c(n3)CCC4)=O)CC1C2 N1(C(C2=CCN(C)C2)=O)CC2CCC(C1)C(NC(c1cc(Cl)nnc1O)=O)C2 N1(C(CN(C(COC)=O)C)=O)CCCCCC(NC(c2cn[nH]c2)=O)C1 c1(OCC#C)ccc(NC(=O)CNC(=O)C(=O)N(CCC(C)O)C)cc1 C1(c2nnnn2C(C)(C)C)(NC2(C)CC(CO)C2)CCN(C(C)(C)C)CC1 C(=O)(CC(C)(C)CNC(=O)C(C)(C)N=[N+]=[N-])NC(CC)C(C)(C)O c1(C(=O)NC2(CNC(C(CC)SC)=O)CCCC2)csc(Cl)c1Cl C1(NC(CCCOC(C)C)=O)C2CCC1N(C(C1CCN(C3CCCC3)C1)=O)C2 C(=O)(CC1=CCN(C)CC1)NCCCCC(C)NC(c1cc(C2CCC2)[nH]n1)=O Cc1ccccc1NC(C1CCOC1CNC(=O)C(C)C#N)=O O=C(CC(C(F)F)c1ccc(F)cc1Cl)NC1CN(C(=O)CSC2CC2)C1 Cc1cc(C(N2CC(C)(NC(=O)C(n3ccc(Br)n3)C)C2)=O)sn1 C1(CCC)CC1N=c1nc2c(ncn2C)c(NCC(C)(CC)c2ccccn2)[nH]1 C(=O)(C1SCCc2ccccc21)N1CC(C)C(CNC(C2(O)CCC2)=O)C1 Cc1cc(CCC(N2CCCCC2CCNC(=O)CC2CCNC2=O)=O)nn1C Cc1[nH]nc2ccc(C(=O)NC(C3CCCN3C(C34CC(C3)C4)=O)C)cc12 c1(C(N2C(CCNC(C(C)OCC)=O)CCC2)=O)ccc(Cl)c(F)c1 O=C(C1=CCCSC1)NC1COCCN(C(C2(c3ccc(O)cc3)CC2)=O)C1 C1(C=O)CCC(C)(C)OC1.C12CN(C1)C(=O)C(C)NC2=O.CCC(=O)OC N1(C(C2(O)CCN(C(C3N(C)CCC3)=O)C2)=O)CCn2ccnc2C1 Cc1cccc(-n2ncc(CNC(=O)C(=O)NC3(C)CCNC3=O)c2C)c1 Cc1c(C(=O)NC(c2cn(CCF)nn2)C)cc(C(F)(F)F)cc1[N+](=O)[O-] N1(C(c2ccc(OC)c(C(F)(F)F)c2)=O)CCN(C(C2CCCO2)=O)CC(O)C1 C(CCC1CC1)(C(=O)NCC(O)C1CCC1)NC(c1cc(C)ns1)=O N1(C(CCc2onc(C)n2)=O)CCN(C(C2(C)CC2(F)F)=O)CC1CO Cc1ncc(C(N2CCC(CN(C)C(C3CC3c3cnnn3C)=O)C2)=O)[nH]1 c1(C(N(CCCCNC(c2cc(C3(C)CC3)on2)=O)C)=O)ccc([N+](=O)[O-])nc1 N1(C(C2CCC2)=O)C2CCC1C(C(=O)NCC=CCCC)C2 C=CC(CC)C(=O)NCC1(C(N2CC(CC)(CC)C2)=O)CCOC1 C1(C)(CNC(C(C)(CO)OC)=O)CCC(NC(c2c(C)coc2C)=O)CC1 Cc1cc(C(=O)NCC2CN(C(c3ccc(Cl)cc3N)=O)CC2C)nc(C)n1 C1(C(=O)NCC2CC(CNC(CCCN(C(C)=O)C)=O)C2)C(C#N)C1(C)C C12(C(N(C3CC(NC(C(CC)C)=O)C3)C)=O)CCC(CC1)C2 C1(C)(CNC(CC(COC)C)=O)CCN(C(c2cc(=O)c(OC)co2)=O)CC1 C1(OC)CCN(C(=O)NCCCC(OC)OC)C(C)C1 c1(C(N2CC(NC(c3cccc(C(c4cnsc4)=O)c3)=O)C2)=O)cc(O)ncn1 CON(C)CCN=c1nc(N2CCc3c(sc(N)c3C(=O)OC)C2)c2sccc2[nH]1 C=CC1(C(=O)NC(C)CC2CN(C(=O)C(F)(F)c3cnccn3)C2)CCCCC1 C(=O)(C(F)(F)C(O)C(C)C)NCC1CN(C(C(C)OCc2ccc(C)cc2)=O)C1 C(C(C)(C)C(=O)NCC1CCCC(NC(C2(C(=O)OC)CC2)=O)C1)N(C)C n1(CC)nccc1C=CC(N1CCC1CNC(=O)C(F)=C1CCCC1)=O C123CC(C1)(C2)C(=O)NC(C1CCCOC1)C(=O)N3.C(C)(C(C)(C)C)=C(CC)CC C12(NC(CCC#C)=O)CCC(C(=O)NC3C4CCCCC34)(CC1)C2 C(CS(=O)(=O)CCOC)NC(C(C1CCCC1)NC(C=CC(CC)C)=O)=O Cn1ccc2ccc(C(N3CCCC(F)(CNC(=O)CC4CC4)C3)=O)cc12 c1(C(N2C(C)CN(C(C3CNC(=O)C3)=O)CC2)=O)cc(F)cc2c1CCC2 C(=O)(C1=CCCC1)N(C1CCC(NC(c2cc(C(F)(F)F)nn2C(F)F)=O)C1)C c1(OC)ccnc(C(=O)NC23CCN(C(C45CCC(CC4)CO5)=O)CC2C3)c1C Cc1ccc(Cl)c(-c2nc(Cc3cnn(C)c3)nn2C2CCCCCC2)c1 C=C1CCN(C(=O)CCN=[N+]=[N-])C(C(=O)NCCOCCCO)C1 c1(N(CC(C(C)(C)C)N2CCOCC2)C)ccncc1S(=O)(=O)NC1CCCC1 C1(CC(C)C)(C(=O)NCC2CCCC(CNC(=O)C3=C(Cl)CC3)C2)CCNC1=O C(C)(CNC(c1cc(C(C)C)on1)=O)(CC(C)C)NC(c1cn(CC)nc1C)=O C1(NC(CN(CC(=O)Nc2nnnn2C2CC2)C)=O)CC(C#N)C1 C1(O)(CNC(C(CC)CC)=O)CCCN(C(C2C3C4CCC(C4)C23)=O)CC1 C1(CC(=O)NCCC2(NC(C(c3ccc(C)o3)C)=O)CC2)OCCCC1(C)C C1(CNC(c2c(C(C)C)cco2)=O)CC(C)N(C(=O)COc2ccc(O)cc2)C1 CCC(C)CCCC(=O)N1CC(NC(c2csnc2C)=O)C(O)C1 Cc1cc(C(N2CCC(C(=O)N(C)CC3CCN(C)CC3)C2C)=O)ccn1 N1(C(Cc2n(C)cnc2)=O)CCC2OCCN(C(c3ccn4cccc4c3)=O)C2C1 C(C(CC(C)C)NC(c1cnc(C(C)C)s1)=O)n1cc(C(CC)O)nn1 N1(C(C(CCC(C)C)O)=O)CCOC2CCN(C(c3c[nH]c(=N)s3)=O)CC12 CCCCCCCCCC(O)CC(=O)Nc1nc(C)c(CC(=O)O)s1 c1(C(N2CCCC(C(=O)NC(CCC)CCO)C2)=O)cccc(Br)c1Br N1(C(CC(CC)SC)=O)CC(C2CCN(C(C3CC4CCCCC34)=O)CC2)C1 c1(C(C)C)nc(=NCCC(C)NC(C2OCC2(C)C)=O)s[nH]1 Cc1cc(C(=O)NC2CCC2CNC(=O)CN2CCC(=O)CC2)n2nccc2n1 CCC(Cc1ccccc1C)C(=O)NCC1CC(O)CN1C(=O)CCNC(N)=O c1(C(N(CCN(C(CN(CCC)C)=O)C)C)=O)cnn(-c2ccc(Cl)cc2)c1C C1(CCC)(NC(C=C(CCC)C)=O)CCN(C(=O)C(C)(COC)OC)CC1 C1(NC(C2CCCN(CC)C2)=O)CC2CCC1N(C(=O)C1=CCCOC1)C2 C1(O)(C(N2CC(C(C)NC(c3cnn(CC(F)F)c3)=O)C2)=O)CCCCCC1 c1(C(=O)OCC)c(C)[nH]c(C(N2CC3CC3(C(=O)N(C(C)C(C)C)C3CC3)C2)=O)c1C C(=O)(C1=CCCC(C)(C)C1)N1CCCC(NC(c2c(C)oc(C)c2Br)=O)C1 C(=O)(C1=CCOC1)N.n1(CCC(=O)NC(C2CCCO2)C)cc(C)nn1 C(=O)(CCCCc1cnc[nH]1)N(CCCNC(c1cc(Br)cs1)=O)C C(=O)(C1=CC2CCC1C2)N1CC(CNC(=O)COCc2ccccn2)OCCC1 C1(NC(c2ccc(Cl)o2)=O)CN(C(=O)C(F)(F)c2ccccc2)CC1O N1(C(C=CC=CC)=O)CC(CNC(=O)CC(C)C2CC2)C2(CCC2)C1 N1(CC(C)NC(=O)C(=O)NCCC23CC(CO2)C3)CCCC1=O CC(O)(C(=O)NC1CC2(C1)CC(C(=O)Nc1ncn(C3CC3)n1)C2)C(F)(F)F N1(C(CCNC(=O)NC)=O)CCC(NC(=O)CCc2nccn2C)C1(C)C C12(NCC(=O)NCC3CCC(NC(C(F)OC)=O)CC3)CCC(CC1)CC2 c1(C(C)=O)cc(C(=O)NCC(C)C(=O)NC(C2CCCCC2)C)no1 CCC(C)C(O)CC(=O)NC1(CC(=O)NC(c2cnn(CC)c2)C)CCC1 c1(OCCC(N2CC3C(CNC(c4nsnc4O)=O)C3C2)=O)c(F)cccc1F c1(C(N2C(C(=O)Nc3c(OC)ccnc3)CC2)=O)cccc(Cl)c1C N1(C(C2C=CCCC2)=O)CC(NC(C2(c3ccc(Cl)nc3)CC2)=O)C2(CC2)C1 N=c1ccc(C(N2CCCCC(CNC(=O)CC3C=CCC3)C2)=O)c(Cl)[nH]1 S1(=O)(=O)C2=CNC=CC2=NCCN1.C(CC(C)(C)NCC1CCOCC1)N(C)CC N1(C(C2CN(S(CC)(=O)=O)C2)=O)CCOC(C)(CNC(C2CC2CF)=O)C1 C1(C(=O)NCC2CN(C(CCC(C)(C)OC)=O)CC2C)CN2CCN1CC2C CC(C)CCC(=O)NCC1CC(C)N(C(c2cccc(C(N)=O)n2)=O)C1 N1(CCCC(=O)NC2CC3C(NC(=O)C(=O)NC4CC4)C3C2)C(=O)CNC1=O c1(OCC(N2C(C(=O)NC3(C)CC=CC3)CCC2)=O)nc(O)nc(O)n1 C1(CNC(C(CC)(C)O)=O)CN(C)CCN1C(=O)Cc1cccc(CSC)c1 CCC(C)(C#N)C(=O)N1CC2CC2(NC(c2cscc2C(F)(F)F)=O)C1 c1(C(=O)NC(CN(C(=O)Cc2ccsc2C)CC)C)c(C)nc(C)n1O Cc1cc(C(=O)NCCCNC(=O)C=CC(C)(C)C)ccc1N1CCOCC1 N1(C(C(C(C)(C)C)N(C)C)=O)CC(C2CCN(C(=O)Cc3cncn3C)CC2)C1 CC(CC(=O)NC(C)(C)C)C(=O)OCC(C)(C)Cn1cc(CCCCCO)nn1 c1(OC)cc(CN2CCC(CNC(=O)CC(O)Cn3cncn3)C2)cc(F)c1 N1(C(C(SC)SC)=O)CC2COCC2(CNC(C2(c3nn[nH]n3)CC2)=O)C1 N1(C(C(COCC)NC(=O)CCCC2CCCO2)=O)CCC(F)(F)C(C)C1 C1(NC(CCCCNC(N)=O)=O)CC2CC(NC(c3coc(C(F)F)n3)=O)CC12 C1(C(C)(C)C)CC(=O)CC12CCC2.C1(N)CC=C(C(=O)N2CC(O)(CCO)C2)C1 N1(C(Cc2c(C)ocn2)=O)CCC(C)(NC(=O)C=CC2CC2)C1 c1(CC)cnc(CN2C(CNC(C3CCCN(S(C)(=O)=O)C3)=O)CC(O)C2)nc1 c1(C(=O)NCC2(CNC(C(C3CC3)OC)=O)CC23CCC3)cc(F)c(C)cc1F n1(CC(N2CC(NC(C(COC)(C)C)=O)C3C2C3)=O)cc(Br)c(O)nc1=O C(CCCC(C)NC(C1CC(C)=NO1)=O)NC(CC=CC=C)=O O=C(C#CC1CCC1)N1CC(n2nccn2)C1 N1(C(C(CC)NCc2ccccc2)=O)C2CCC1CC(NCc1c(C)ncn1C)C2 C1(CNC(=O)CC2CCCSC2)C(O)C(O)CN1C(=O)CC1CCOC1=O C1(C2CC2)(C(N2C(C)CSCC2)=O)CN(C(C2C3CCC(F)C23)=O)C1 Cc1cc(C(=O)N(CC(=O)NCC(c2cccs2)O)C2CC2)cc(C)c1 Cc1cc(C(N2CCC(OCCNC(C3CCCCN3C)=O)CC2)=O)c(C)s1 Cc1cc(C(=O)NC2CN(C(=O)CC(F)(F)F)CC2CO)c(C)n1C1CCCC1 C(=O)(C(C)(C)C(C)NC(=O)C=CC(=Cc1ccsc1)C)OCC c1(C(=O)OC)nc2c(COC)cccc2s1.S1(=O)(=O)CC(=O)NCCN1CC C1(C(=O)OC)(C(=O)Sc2ccccc2OC2C3CCC(F)(F)C23)CCC(O)CC1 C1(C)(C(N2CCN(C(C#C)C)CC2)=O)CN(C(=O)Cc2ccn(C)c2)CC1C Cn1cccc1COC(C1(CC(=O)O)CCC1)=O c1(CN(C(=O)CC(C2CC2)NC(c2cncs2)=O)C)cn(C)cn1 C1(N(C(C(C)SC(C)C)=O)C)CN(C(=O)C=CC(c2ccc(F)cc2)=O)CC1O Cc1ccc(F)c(C(N2CC(NC(C3CC3C(N)=O)=O)C(C(F)F)C2)=O)c1 C1(CC)CN(C(c2ccoc2)=O)CC1C(=O)N(C1CCC1)C1CCC1 C1(C)(N(c2ccccc2)C(CN(CCC)C)=O)CCCN(C(C2CC2F)=O)C1 C12(C(=O)NC(C(=O)NCCC3(CSC4CC4)CCC3)C3CCCO3)CCC(C1)C2 N1(C(C(C)(C)n2cc(Cl)cn2)=O)CC2CCC1CN2C(=O)COC(F)F.C1C(=O)O1 c1(SC)cccc(F)c1C(=O)NCCC1(CNC(C2CCCC3(CC3)C2)=O)CC1 CC1(C)CCC(NC(C)(CCN2CCCCC2)c2nnnn2CC2CCCO2)C1 C1(C(=O)NC(CNC(COCCCCOC)=O)(C)C2CC2)CCCC1(F)F N1(C(=O)CCCN2CCCC2)CCSCC1Cn1cc(CCn2cccc2)nn1 N1(C(c2cc(OC)ns2)=O)CCCC(N(C(=O)CCCF)C)CC1 c1(-n2ccc(CS(CC3C(C)(C)OCC3)=O)n2)ccc(S(C)(=O)=O)cc1 C(CO)(CCS(C)(=O)=O)N(c1ccc(NC(C(CC)C)=O)c(C)c1)CC N1(C(COC(C)C)=O)Cc2nccn2CC(NC(c2nncn2C2CC2)=O)C1 c1(C(=O)NC2(CNC(c3c(C)csc3)=O)CC2)cc2ccc(Cl)cc2[nH]1 C1(NC(C2CCS(=O)(=O)C2)=O)CCCC(NC(C2(CC(F)F)CCC2)=O)C1 N1(C(c2c(C)cns2)=O)CCC(NC(c2cc(C(C)(F)F)n[nH]2)=O)CC1C C(=O)(C#CC1CCOC1)N1C(CNC(c2cc(OC)nn2C)=O)CC1 C1(NC(=O)CCCCNC(=O)C2=COCCO2)CC2CC1CC2(F)F c1(OC)cccc(CN2CCC(NC(C3CCNC(=O)C3)=O)C2)c1 c1(C(N(CC(C)(C)NC(CC2CCN(C)CC2)=O)C)=O)cc2cc(Cl)sc2[nH]1 c1(OC)cc(CNC(=O)C(C)(O)CC(C)C)c(-n2cc(C(C)O)nn2)cc1Cl N1(C(c2[nH]c(=NCC)sc2)=O)CCCC(C2CCN(C(C3(C)CC3Br)=O)C2)C1 Nc1c(C(N2CC3(CCNC(=O)COC(F)F)CCC2C3)=O)cc(F)cc1Cl c1(C(=O)NCC2OCCN(C(C3=C(C)CCC3)=O)C2)cc(C)cc(F)c1N N1(C(=O)CN2CCSCC2)CCC2(CCCN2C(=O)CC2(CO)CCC2)CC1 CCCCC(C)CCC(=O)N1CC(N(C(=O)CC(O)CCCCC)C)C(O)C1 C(=O)(Nn1cnn(C)c1=S)C12N(C(CN3C(C)CCC3)=O)CCC1CCC2 N1(C(c2c(C)n[nH]c2)=O)CC(C(=O)NCC(F)Br)C2(CC2)C1 N1(C(C2N(C(c3c(C)ccnc3)=O)CSC2)=O)CC2(CCC2(C)C)C1 N1(C(CCCNS(C)(=O)=O)=O)CCOCC(C)(NC(=O)C(F)(F)CO)C1 c1(CCC=C)ccc(C(N2CCC23CCCC3)C(=O)NCCCF)cc1 c1(C(C)C(=O)NCC2(CNC(C3CC3C)=O)CC2)ccccn1 N1(C(CCc2cccc(C)n2)=O)CCN(C(=O)CN2CCC(C)C2)CC(CO)C1 N1(C(CC2CCN(C)C2)=O)CCCCC1CCNC(c1nnn(C)n1)=O c1(C(N2CCC(CCCNC(CC(=O)NCC#C)=O)CC2)=O)cc(C)ccc1Cl C1(CNC(C(CC#C)NC(=O)Cc2cn(CC)nn2)=O)CCCCC1(C)C C1(C2CCN(C(C3(CO)CC3)=O)CC2)(NC(C2N(C(C)C)C(=O)COC2)=O)CC1 C=CCC(C)(C)CC(=O)NC1CN(C(C2CC3(C2)CC32CC2)=O)CC1(C)C c1(C(=O)NC2C(CNC(C3C(CC(C)C)C3)=O)C2)ccc(C(F)F)cn1 Cc1ccc(F)c(CC(N2CC(NC(=O)CC3CC(C)C3)CC(F)C2)=O)c1 CC(C(=O)NCCCC(C)(F)F)NC(=O)CCOC1CC1 c1(C(N2C(C(C)NC(C(CCC)OCC)=O)CCC2)=O)cnn2cc(C)cnc12 C1(NC(Cc2c(C)nc(SC(F)F)s2)=O)CN(C(=O)CCSC2CC2)CCC1C Cc1ccc(CCNC(=O)C(Cc2cn[nH]c2)NC(C2CC(F)CN2C)=O)cc1 CC1CC(CO)CCN1C(=O)NC(c1cccnc1Cl)c1ncnn1CCCl CN1CCN(C)C(C(=O)N(C2CC(NC(C3CN4CCC3C4)=O)C2)C)C1 c1(CN2C(CC(NOC(C3CCCC3)=O)=O)CC2)ccncc1F N(C(=NC1CCC1)N1CCC(OC2CCCC2)CC1)C1CCS(=O)(=O)N1 Cc1nc(C(=O)NCC23CC2CN(C(=O)CC(F)(F)F)C3)ccc1[N+](=O)[O-] C(=O)(C#CC1(C)CCCO1)NC1CC2(CC(C(=O)NCc3c(C)cccc3C)C2)C1 C#CC1CN(C(=O)C(C)CN(C(=O)C(C)CC(N)=O)C)CCO1 C(=O)(C#CC(C)(C)C)NC1C(NC(CCOc2ccc(OC)cc2)=O)CC1 N1(C(C2CC(C)N(C(=O)OC(C)(C)C)CC2)=O)CCCC12CCOC2 N1(C(C2N(C(c3ccc(CC)nc3)=O)CCCC2)=O)CCC2(CCCOC2)C1 N1(C(C(CC2CCOCC2)NC(Cn2ccc(C)n2)=O)=O)CCCCCC1C C1(N=c2nc(C3CC3)[nH]s2)(CCNC(c2cc(-c3ccoc3)on2)=O)CCC1 N1(C(c2cc(C)n(C(C)(C)C)n2)=O)CCC(NC(C2(C)CNC(=O)C2)=O)C(F)C1 CC(CCCNC(=O)CSCc1cccs1)NC(=O)CC1COC2CC12 c1(CC(N2CC3(CCN(C(CCC=CC)=O)C3)C2)=O)cn(C)c2ccccc12 C1(c2nn[nH]n2)CCC(C)=CC1C.C12(CCC1)C(=O)N(C(C)C1CC1)N2.C12CCN1C2 C1(CC(=O)OC)(NC(=O)NC2CCCN(c3cnn(C)c3)C2)CCOCC1 Cn1ncc(C(=O)NCC2(NC(=O)C=CC(c3ccccc3)=O)CCOC2)c1N c1(NC(=O)C2=NOCC2)cc(N(C)C)ccc1C(=O)NC1CCC(C(=O)OC)C1 N1(CC(=O)OC)CCC(CNC(=O)CC2CC2c2cccc(Cl)c2)CC1 c1(CC)cc(CN(C)C)on1.C123CC(C1C2)n1cc(nn1)CN(C)C3=O c1(C(N2CCC(c3ccon3)C2)C(=O)NC(C)C)ccc(O)nc1 C#CC1(C(=O)NCC2CCCCCC2)CN(C(=O)Cn2cc(CC)cn2)C1 N1(C(c2c(-c3ccn(C)n3)[nH]cn2)=O)CCC(CNC(=O)COC(F)F)C1(C)C C(=O)(C(O)C(F)(F)F)N(CCNC(C1C(C)COCC1)=O)CCOCCO C1(C(=O)NC(C(C)O)C(=O)NC2C=CCCC2CO)CC(=O)CC12CCC2 C1(NC(C(C)N(C(CCN(C)CC)=O)C2CC2)=O)C(C)(C)C1(F)F c1(CN2CC(C(=O)Nc3nc(O)nc(O)n3)OCC2)ccc2ccoc2c1 C(CCC(=O)NCC(CCc1ccccc1)NC(=O)C=CCO)C1C(C)C1 C(CC1CC1)(CC(=O)NCc1cccc(C(=O)O)n1)NC(COC)=O c1(C(N2C3CC(CNC(C4(OC)CC4)=O)C2CC3)=O)cc2cc(F)ccc2o1 CCC(C)(O)C(=O)N1CCC(c2ccccc2)(NC(=O)C=Cc2cccn2C)C1 N1(C(C2(F)CN(C(C(CC)OC)=O)C2)=O)CC(OC)C(SC)C1 C(=O)(C(F)CC(C)(C)NC(=O)C1=C(C)CCOC1)N(CCF)CC n1(CC)c(C(N2CCCC(O)(CCNC(=O)C(Cl)=CCl)C2)=O)nc2ccccc12 CCC(CC(=O)N(C1CC(C(C)C)C1)C)NC(=O)CCCC#N C1(C)(C(=O)NCC(COC)(O)CO)CCN(C(=O)CC(C)C2CCCCC2)CC1 CCC(C)C(C(=O)NCCNC(C1(c2ccccc2)CC(F)C1)=O)NC(C)=O CCC(CC)CCCC(=O)NOCC(=O)N(C(C)C(C)(C)O)C C(N=c1ccnc(C(C)C)[nH]1)C1CCCN(C(C(CC)(C)C)=O)C1 Cc1cc(CNc2ncc(-c3ccoc3)cc2I)cnc1F c1(C(N(C2CCCC2)CCNC(C2(COC)CC2(F)F)=O)=O)cc2nc(C)sc2[nH]1 C1(C(=O)NCC(CCC)C)CCN(C(=O)CC2CC(NCC)C2)O1 N1(C(CCC#C)=O)CC2(CC(C(=O)NCc3ccnc(OC(F)F)c3)CO2)C1 C(=O)(CCS(=O)(=O)NC)NCC1N(C(C(C)=C(CC)C)=O)CC(O)C1 C1(C(=O)NC2C=CC(CNC(C3(C)CC(=C)C3)=O)C2)CCn2c(C)cnc2C1 N1(C(c2[nH]cc(CC(C)C)c2)=O)CC2CCCC(NC(C3CCCO3)=O)C2C1 Nc1ncc(C(=O)NCC2CCC2NC(=O)C=Cc2ccsc2)cc1Br N1(C(C23N(C(c4c(C)cncn4)=O)CC(C2)C3)=O)CCCCC(CO)C1 n1(CC)c(SNCc2cccc(Cl)c2)nc2ccccc12 C1(C2CCCOC2)(NC(C2C3CCN(C(c4cc(C)c(O)nn4)=O)CC32)=O)CC1 c1(OC)ccc(F)c(C(=O)NCCCOCCCNC(=O)Cc2ncccc2C)c1 N1(C(CCCC(C)O)=O)CC2CCN(C(=O)CC3CCC(=O)N3)C2C1C C(CCCCC(=O)NC(C)CCCCNC(=O)Cc1cn(C)nc1C)OC N1(C(C2C(CC(C)(C)C)C2)=O)CC2(CC2)CC1C(N1CC(O)(C(F)F)C1)=O N1(C(c2ccc(N(C)C)cn2)=O)CCN(C(=O)Cc2cnoc2)CC1CCO N1(C(CC(C)C2CC2)=O)CC(C)CN(C(C2(C(=O)NC3CC3)CC2)=O)CC1C C(C(=O)NCC1(C(N)=O)CN(C(c2csc(Cl)n2)=O)C1)(C(C)C)OCC(C)C C1(C(C)=O)CCN(S(=O)(=O)NC(=O)CN2CC(C)CC(C)C2)CC1 n1(-c2c(OC)cccc2)cc(C(=O)N(C2CC2C2CCCCC2)C)ccc1=O C1(C(N2C(C)(CNC(c3c(C(N)=O)scn3)=O)CCC2)=O)CN2CCCC2CO1 C1(OCC)CN(C(=NCCNC(C2(CC3CC3)CC2)=O)NCC)CC1O C#CCC(=O)N(C(CCn1ccnn1)C1CCC1)CC1(c2nn[nH]n2)CCC1 CN1CCN(C(C2CCCN2C(=O)Nc2ccccn2)=O)C(C(C)(C)C)C1 C(=O)(C1=CCCCC1C)N1C(CNC(c2ccc(OC)cc2)=O)CC(F)C1 c1(C(=O)NCC(CO)NC(c2ncoc2C2CC2)=O)ccc(F)cc1.C1CSCCS1 c1(C(=O)NC2C(C(=O)NCCCC(C)(C)OC)CCC2)cc2ccccc2[nH]1 S1(=O)(=O)c2ccc(cc2)N1.C=CC1CCCCN1CCN1CCN(C)CC1 c1(C(N2CCC(F)(CNC(C3CN(C)C(=O)C3)=O)C2)=O)cnc(OCF)c(Cl)c1 c1(C(=O)NC2C3(CC(NC(C(c4ccc(C)o4)C)=O)C3)C2)cc(C)c(=O)n(C)c1 c1(CC)nc(O)c(C(=O)NCC(CO)NC(c2cnccc2C)=O)cc1C CC(C(C)(C)CO)NC(=O)C(C)(C)C1CCN(C(c2ccncc2F)=O)C1 C1(C)(CNC(c2c(CC)noc2C)c2n(CC=C)nnn2)CCCCC1 N1(C(C2(C)CNC(=O)C2)=O)CCOCC(NC(C2CCSCC2)=O)C1 CC1(NC(=O)C=Cc2cncs2)CCN(C(c2ccsc2-n2cnnn2)=O)C1 Cc1cnn(C(C)C(=O)NCC(C(=O)N2CC(C)(C)C2)N(C)C)c1 N1(C(CC=CC=C)=O)CCOCC1CCNC(c1ccc(-c2ccncc2)o1)=O C1(NC(Cc2c(C)cnn2C)=O)CC2(C1)CN(C(C1CCN(C3CC3)C1=O)=O)C2 CC(C)C(O)CCNC(=O)C(C1(C)CC1)NC(c1nccn1C(C)C)=O C1(C(N(CC)Cc2ccncc2)=O)N(C(C2CCNC2=O)=O)CCC1(C)C C(C(CC(C)C)C(=O)NC1COCC1CO)NC(c1c(C)scc1)=O Cn1[nH]cnc1=NC(=O)C1CCC(NC(c2ccc3c[nH]nc3c2)=O)CC1 CC(C(=O)NC1CC(F)CN(C(c2cnc(O)c(C(F)(F)F)c2)=O)C1)S(N)(=O)=O c1(C(CC)C(=O)N2CCC(c3csc(=N)[nH]3)C2)cccc(Br)c1 c1(C(=O)NC(C)CCCNC(=O)CC2CCCN2C)cc2c(cc1Cl)OCCO2 N1(C(c2c(C(C)C)nn(C)c2)=O)CCC(NC(=O)C=CS(C)=O)CC(C)(C)C1 C1(C(=O)NC2C(C)N(C(C3CCC(F)C3)=O)CCC2)CC(C2CCOCC2)=NO1 C#Cc1ccc(C(=O)NC23CCC2CN(C(=O)C=Cc2cn(C)cn2)C3)cc1F C(C)(C(=O)NCC=CC(C)(C)C)(C1CCC1)NC(C(C1CCC(=O)N1)C)=O Cc1nc2c(C(=O)NCC34CC(NC(c5ccon5)=O)(C3)C(C)O4)ccnc2[nH]1 C(=O)(CC(C)C(F)(F)F)NCCCC1(NC(c2noc(CC)c2C)=O)CC1 C1(CC)(NC(=O)C(C)N(C)C)CCN(C(c2nc(C)oc2C)=O)C1 CCC(CC)CC(=O)N1CC(CCNC(C2CCCC2C(N)=O)=O)(OC)C1 c1(CC(N2CCOCC2)C)nc(-c2ccc(C3CC3)cc2)nn1N(C)CCO c12ccc(cc1)CC(=O)N1CCSC(C1)C(=O)N2.c1(OC)cnn(C(C)(C)C)c1 N1(C(c2cc(Br)cc(C)c2N)=O)CCN(C(=O)CCCC(C)C)C2COCC12 C1(C(N2CCC(C#C)(O)C2)=O)CN(C(=O)CCCCSC)CC(F)(F)C1 C(N=c1[nH]c2cc(Cl)ccc2s1)C1(C(C)(C)C)CCN(C(C2CCCC2O)=O)C1 C1(NC(C)=O)CC2CCC(C1)N2C(C1(C#N)CCCO1)=O C1(C(=O)NCC(Cl)Cl)CC(CNC(C2(C(F)(F)F)CC2)=O)C1 C1(NC(c2ccc(C#C)cc2)=O)CC2CN(C(=O)CCCC(C)O)CC2C1 CC1CCCC(C)N1C(=O)C(N1CCCC(C)(CNC(=O)CC2CC2)C1)=O Cc1nn(CC(N2CCC3(NC(c4ccnn4CCF)=O)CC3C2)=O)c(C)c1Cl C1(C(=O)NCCCCN(C(CN(CCC#C)C)=O)C)CCCCN1C(C)=O C1(NC(COc2c(OC)cccc2)=O)CCN(CC2CCOC2)CC1C C#Cc1cncc(NC(=O)CN(C(=O)C(C(=O)OCC)OC)C)c1 C(C(C)S(C)(=O)=O)(c1nnnn1CC(F)F)NCC(c1nc(C(F)(F)F)cs1)C C1(C(=O)NC2C(C)(C)CN(C(=O)Cn3cnc(=N)[nH]3)C2)CC2(C1)CS(=O)(=O)C2 C(C)(C)(CC(=O)N=c1ccn(C2CCC2)[nH]1)NC(COCCOC)=O c1(OC)ccc(F)c2c1NC2=O.c1(C(N2C3CNCC23)=O)ccnc(OC)c1 N1(C(C2(c3ccn(C)n3)CC2)=O)CCC2(C1)CN(C(N1CC(C)(C)C(O)C1)=O)C2 C1(CNC(=O)CCC2CCCC2)CN(C(c2cnc(C3CCC3)s2)=O)CCCO1 CC1(NC(c2cccn2C2CC2)=O)CCN(C(=O)CC=C(Cl)Cl)C1 c1(C(=O)NCC(C)(C2CC2)NC(C2C(OCC)CC2)=O)c(Br)noc1C CCCCCCCC(=O)NC1CCC(C(=O)NC2CCCOC2)C1 C12(C(=O)NCC3(C)CCN(C(Cc4nc(C)oc4)=O)C3)CCCC1CCC2 Cc1c[nH]cc(C(=O)NC2CCC(C)(CNC(c3cn(C)cn3)=O)CC2)c1=O O=C(NNC(=O)C12CC(C1)C2)NC1(CF)CCCC1 c1(C(=O)NC2CC(C)CN(Cc3ncccc3Br)C2)ccc2ccccc2c1 N1(C(CC2(C=C)CCC2)=O)CCCC(C2CN(C(C3CC4C=CC3C4)=O)C2)C1 CSC1=C(C(=O)N2CCOC(CNC(=O)C(c3ccc(F)cc3)=O)C2)CCCC1 C=CCC(CC)C(=O)N1CCC(C(=O)NC(c2ccoc2)C)(CC)CC1 N1(C(C(CC)OC)=O)CC2CCC1C2NC(c1cccc(C(N)=O)c1C)=O C(C)(C(=O)NCC(C)(C)CN(C(=O)CSCc1cscn1)C)(C1CC1)OC C1(CNC(=O)CC2CNC(=O)O2)CCN(C(C2CCS(=O)(=O)CC2)=O)C12CC2 C1(CNC(C(C)N(C(CN(CC)CC)=O)C)=O)COC2(CCC2)C1 c1(C(=O)NCC(CC)NC(C2(CNCC)CC2)=O)cccc(Cl)c1-n1cccc1 C12(NC(c3cnc(C)s3)=O)CC1CN(C(C13CCCC1(C(N)=O)C3)=O)C2 C1(CC)CN(C(=O)Cc2csc(-c3ccc(Br)cc3)n2)C(CC)CO1.CCNC N=c1[nH]c(CCC(=O)N2CCC2CNC(c2sccc2F)=O)cs1 N1(C(CN(C(C2C=CCCC2)=O)C2CC2)=O)CC2COCC2(CO)C1 N1(CC(=O)NCCN(C2CCCCCC2)C(C2CNC(=O)O2)=O)C(=O)CCC1=O CC(CCCCNC(=O)C(F)C1CCCC1)NC(=O)CCS(C)=O N1(C(CC2CC(SC)C2)=O)CCC(F)(NC2CC2(C)CO)CC1 N1(C(c2ccc(-c3nc[nH]n3)nc2)=O)CC2CC(C1)N2C(=O)CC1CC1 C1(C(=O)NC2(NC(C(C)OCCC#C)=O)CC2C)CCN(C(C)C)C1 c1(C(=O)NC(C(=O)NCCSCCOC)C2CCOC2)ccc(F)cc1C c1(C(N2CCC(C(=O)NCC#C)C2)C(=O)NC(C)(C)C)cccc(C(C)C)n1 C(=O)(CCC(C)(C)C#N)NC(CC)(C)CNC(C1CC(OC(C)=O)C1)=O c1(C(=O)NCCNC(C2CN(C(CCS(C)=O)=O)C2)=O)cn(C)c2ccc(F)cc12 c1(COC)ccc(C(=O)NC(CNC(=O)C2=CCCC2C)C2CCC2)cc1F CN1CCC(C(=O)NCc2cn(C3(C(=O)O)CCCOC3)nn2)C1c1ccccc1 c1(C(N2CCCC2c2ccon2)=O)ccc(Cc2cn(C3CCOC3)nn2)cc1 N1(C(C(COC)NC(C)=O)=O)CCC2(CC1)CC(NC(=O)CSCC(C)C)CO2 CC1CCN(C(c2ncsc2C(F)(F)F)=O)CC1CNC(=O)COc1ccsn1 CC1CN(C(c2cnccc2Cl)=O)CCC1CNC(c1ccc(C#N)cc1)=O C(=O)(CS(=O)(=O)C(C)C)CCC(Cn1cc(-c2cccc(OC)c2F)nn1)F N12CC(CC1(C)C)C(=O)N(C)CC2=O.C1(NC(=O)C2CC2)CCCC1C#N C1(=CC(=O)NC(C)CNC(=O)CCC2CC(CC3CC3)C2)CCCCC1(C)C N1(C(c2cnc(C)s2)=O)CC2CCCCC2(CNC(c2occc2Cl)=O)C1 Cc1ccc(I)cc1NC(C1(C)CCN(c2ncc(Br)c(C(F)(F)F)n2)C1)=O N1(C(c2ccc(NC)c(F)c2)=O)CCN(C(=O)C(=O)C2CC2)C(C)C1C N1(C(c2cc(SC)c(F)cc2)=O)C2CCCC1CC(NC(=O)CC(C)O)C2 c1(CC)c[nH]c2ncnc(N3CCC(CNC(c4ccc(C)nc4CC)=O)C3)c12 N1(C(C(CC=C)C)=O)CC2(C(N3CCC3(C)C(=O)OC)=O)CCC1CC2 c1(C(=O)NCC2N(C(c3[nH]cc(C(N)=O)c3)=O)CC=C2)cccc2ncccc12 C1(NC(C(F)=CC)=O)(CF)CCN(C(C2C3CCC2(c2cnco2)C3)=O)C1 N1(CC(=O)N(C)CC2CCSCC2)C(=O)CCCC1=O N1(C(C(CC)N(C)C)=O)CC2CC1CCC2NC(c1ncc(C)o1)=O c1(OC)cc(F)ccc1CNC(=O)C(=O)NC(C1CCOC1)CO C1(N(C(C2CCC(F)(F)CC2)=O)CC2(C#C)CCCC2)C2CC(O)C1N(CC)C2 Cc1ccc2ncc(C(N3CCCC4(NC(=O)C(C)C(C)(F)F)CC4C3)=O)n2c1 c1(C(=O)NCCCN(C(C2(COC)CC=CC2)=O)C)cc(C)c(C)c(F)c1 CC(CNC(C)(C)C1C(C(C2CCC2)N(C)C)C1)CC1CCC1 C12(C(N3CC(NC(c4ccncc4-n4cccn4)=O)C3)=O)CCCCC(F)(C1)C2 C12(C)CCN(CC1)C2=O.c1(OCC2CC(NC(C3(C#C)CC3)=O)C2)ccccc1 c1(CN(C)Cc2cccc(C)c2)cc2ccc(F)cc2nc1O n1(CC(=O)NC(CNC(C=Cc2n(CC)ncc2)=O)CCCC)nc(Cl)ccc1=O C(=O)(C(F)C(F)(F)F)NC1C(NC(c2oc(CC)c(C)c2)=O)CCC1 c1(N(C(C=CC(=O)NCC2(CSC)CC2)=O)C)ccccc1.C1(C2CC2)C(=O)N1 CC1CN2CCN1C(C(N1CC(F)CC1CNC(c1ccc(Cl)c(F)c1)=O)=O)C2 N1(C(C#CC(=O)N(C)C)=O)CCC2C(CCCN2C(=O)C=Cc2cccnc2)C1 C1(CC(=O)N(C2CN(C(c3ccc(-c4ccncc4)o3)=O)C2)C)OC(C)(C)OC1=O c1(OCC(c2ccc(OC(F)(F)F)cc2)=O)cncc2ccc(F)cc12 C(C(C(=O)N1CCC(CF)C1)NC(c1cnnn1C)=O)OCC c1(CC=C(C)C)ccc(C(N2CCCC2CC(=O)Nc2csc(C)n2)=O)nc1 CC1C(=O)N(CCO)CN1C(c1ccc(OC(C)(C)C)cc1F)=O c1(C(=O)Nc2ccnc(C3CC3)c2)cnc(C2CC2)[nH]c1=N CCC(C)C(=O)N(CCNC(c1ocnc1-c1ccccc1)=O)CC1CC1 Cc1ccc(C(=O)Nc2ccc(NC(=O)CC3CCCC(C)C3)cn2)nc1 N1(C(C2(CO)CC2Br)=O)CCC(c2cc(-c3ccccc3)[nH]n2)CC1 c1(C(N2C(CCCNC(C(=O)NC(C)C)=O)CCC2)=O)cc(F)ccc1Br CC(CC(F)F)C(=O)NC(CO)C(C)NC(c1cncc(-n2cccn2)n1)=O CCCCCC(C)CC(=O)N1CCC(NC(c2cncs2)=O)C1C(C)C C1(C(=O)NCC2CC(NC(C3CNC(=O)N3)=O)C2)C2CCCCC12 N1(C(C2(C(=O)NCCSCC)CCC(N)C2)=O)CC2C3C=CC(O3)C2C1 C1(C2=CCOCC2)(CN2CCC(SC3CCN(C)C3)CC2)CC1 C1(C(N(CC(C)C)CC)=O)CCC2(CC2)N1C(=O)C(CC(C)C)N(C)C c1(N2CCc3cn(nn3)-c3cc(cc(Cl)c3)C2=O)ccc(C(F)F)cc1F.CC C1(C(=O)NC(CC(N2CCN(C(=O)Cc3cc[nH]c3)CC2)=O)=O)CCCC12CCC2 N1(C(c2c(CC)nns2)=O)CCCCC(NC(=O)C(=O)CCc2ccccc2)CC1 c1(OC)ccc(Cl)c(C(=O)NC2CCCC2CNC(C2CCCOC2)=O)n1 C1(NC(c2n(-c3c(C)cccc3)nnn2)c2nnn(C)n2)CC(C)(C)C12CC2 CCC(O)CCN=c1cc(C)c(S(=O)(=O)NC2CCCCC2CC)c[nH]1 N12CC34CCCCC3(CN(C4)N(C)c3nc1c1c(F)cccc1n3)C2.C1CC1.CC C1(C(=O)NCC(C)N(C(C2CC(OCC)C2)=O)C)Cc2ccccc2C1(C)C S(=O)(=O)(c1ccc(NC2CCCC2S(C)(=O)=O)c(Cl)c1)NCC(CC)(CC)OC N1(C(C(C(C)C)SCC)=O)CCC(O)(C(=O)NC(C)CC2CCCCC2)CC1 C1(CC(=O)NCC(CCOC)NC(=O)C=Cc2ccc(C)s2)CCC(=O)NC1 c1(CC(=O)NC(CC=C)CNC(=O)C(C)(C)C)ccc(C(=O)N(C)C)nc1 C=CC1CN(C(=O)Cc2nccn2C)CC1NC(c1nn[nH]c1C(F)(F)F)=O c1(C(=O)NC2(CCNC(C(C)Oc3ccc(C)cc3)=O)CC2)cc([N+](=O)[O-])sn1 C(CCCOC)(C(=O)N(C1CCCC1(C)O)C)NC(COCC=C)=O N1(C(c2c[nH]c(=N)s2)=O)CCC(NC(C2CCN(CC(F)F)CC2)=O)CC(O)C1 c1(C(C(=O)N(C2CCN(C(C3CC34CC(O)C4)=O)C2)CC)O)cc(F)cc(F)c1 CC(C)CC(CNC(=O)C(c1cnn(C)c1)O)C(=O)N1CCC(F)(CF)C1 C1(C(=O)NC(CCCC)COC)CCCCCCN1C(C1CCC(CO)CC1)=O c1(C(=O)NCC2N(C(C3C(C)(C)CO3)=O)CCC2)csc2c1CCCC2 c1(OC)ccc(OC)c(C(=O)NC(CNC(c2occc2Br)=O)CO)c1 C1(CNC(C2C(C)(C(C)C)C2)=O)C(C)CCN1C(=O)COc1cncc(Cl)n1 C1(CNC(C2(OCC)CC2)=O)CC2CC1CN2C(c1nc(Cl)cs1)=O c1(C(=O)NC2(CCOC)CCN(C(=O)C(C)CO)C2)cccc2c1OC(C)(C)C2 C(c1cn(C)nn1)=CC(=O)NC(C)CCCNC(=O)Cc1cncnc1 C1(CC(=O)OCc2cnc(-c3ccccc3Cl)s2)CCC(F)(F)CO1 Cc1cc(O)nc(C)c1C(N1CCC(NC(=O)CSc2cccnc2)C(F)C1)=O C1(C(F)(F)F)c2cn(nn2)C2CC3(CC23)C(=O)N1.C1(OCC(=O)O)CCCCC1 CC1(C)CN(C(C2CCCCO2)=O)CC1NC(c1cnn(CC2CCCC2)c1)=O C1(NC(c2cncc(C)c2)=O)CC(C(=O)NCc2cc(C)[nH]n2)C12CCC2 n1(CC=C(C(=O)N(CC(C)NC(=O)C=CC(=O)N(C)C)CC)C)cncn1 c1(C(N2C(COCCOCCC(=O)OC)CCC2=O)=O)cnc2c(c1)CCC2.C1(CC)CC1 C1(CC(=O)N(CCCN)C(C)C)NC(=O)NC1=O.n1(CC(C)C)ccnc1C(C)C C(CC(C(=O)NC1CC12CCC2)NC(=O)C=CCOCCOC)=CC c1(OC)cc(C)c(Cl)cc1C(N1CC2(CCN(C(=O)CC3CCCC3)C2)C1)=O N1(C(C(F)=CC)=O)CCC2(CC1)CC(NC(=O)CCc1c(C)nn(C)c1C)CO2 c1(C(C(C(C)N)=O)=O)ccc2c(n1)NCC2.C1(O)(CN)CN(C=O)C1.n1(C)cnnc1 C1(C(=O)NCC(C)F)CC12CCN(C(C1CCOCC1)=O)CC2 C#CCC(C(=O)NC(CC1CCOCC1)C(=O)N1CCCCC1)C1CC1 c1(C(=O)NC2CCC(NC(c3ccsc3)=O)C2)ccc(Cl)cc1C(F)(F)F C(c1ccc(F)c(C)c1)=CC(=O)NCC1N(C(c2ncc(C)cn2)=O)CCCC1 c1(N2CC(NC(c3cccnc3C3CC3)=O)(CO)C2)ncc(F)cn1 c1(NC2C(NC(CCCCC(=O)NC)=O)CCCC2)nc2cc(F)c(F)cc2s1 C1(C)(C(N2CC(CCC=C)(C(=O)NC3(CC4CC4)CC3)C2)=O)CCC(C)C1 S(=O)(=O)(CC(=O)NCC1C2CN(Cc3cccc(F)c3)CC12)NC C(=O)(C(CC(C)(C)C)NC(C1CCC(=O)NC1)=O)N1CCC(C(C#C)C)CC1 CC1(C)CC(NC(=O)COc2cccc(F)c2)CN1C(c1cc(C2CC2)on1)=O Cc1nc(CO)sc1C(=O)NC12CC(NC(C3CCCN3C)=O)(C1)C2 N1(C(Cc2n(C)nnc2)=O)C2CCCC1CN(C(c1cc(C3CC3)no1)=O)CC2 N1(C(C(C)OCC)=O)C2CCC(C2)C1C(=O)NCC1(CC2CC2)CC1 c1(C(=O)NCC2(C)C(C)CN(C(=O)CC3CC3(C)C)C2)cc2c(s1)CCSC2 CC1(C)C(NC(c2cc(Br)n[nH]2)=O)CCN1C(=O)Cn1nc(O)ccc1=O Cc1cc(C(N2CCC(=C(F)F)CC2)=O)c(C)c(Cl)c1 C12(C(=O)NCC3N(C(c4nc(OC)oc4)=O)CCC3)CCC(C1)C(C)(C)O2 C12(OC)CCC(C(=O)NC34CC3CN(C(c3cnn(C5CCC5)c3)=O)C4)(CC1)C2 C(C1=CCN(C(c2ccc(O)cc2F)=O)CC1)NC(=O)CCc1cccc(Cl)c1 Cc1c(C(=O)NCC2C(C)CCN2C(=O)CNS(N)(=O)=O)cnc2ccccc12 N1(Cc2cc(=N)[nH]cc2)CCN(C(c2nncs2)=O)C(=O)C1.C1CCS1 C1(OC)CN(C(=O)C(C(C)(C)C)n2cc(CNC(=O)C(C)O)nn2)CC12CC2 C(=O)(CC(C)P(C)(C)=O)NC1(COC)CCN(C(=O)CCCC2CC2)CC1 C1(c2cn(CC(CC)O)nn2)CN(C(c2cn(C(C)C)cn2)=O)CCN1C N1(C(C2(CSC)CC2)=O)CCC2(CCCN(C(c3cccnc3C(F)F)=O)C2)C1 N12CC(CC(C)C1)NC(=O)C2c1ccnc(SCC)c1.C(=O)(CCOC)OCC c1(OC)c(F)cc(C(=O)NCCN(C)C(c2n[nH]c3c2COC3)=O)c(N)c1F N1(C(C(C)OCCC=C)=O)CCOC(CN(C(=O)C(C)(C)c2cc[nH]n2)C)C1 C(C(=O)NCCOCCCNC(=O)C(C)c1ccco1)(C1CCC1)OC C1(CNC(C2(CC)CC2)=O)CCOC1NC(CC1(NCC)CCC1)=O c1(NC(CC)COC(F)F)ncc(OC(F)F)cn1.c12nnnn1C2(C1CCCO1)C C1(C(N2CC(CNC(C3N(C(CCC)=O)CCCC3)=O)C2)=O)CCC2CC1C2(C)C c1(C(=O)NCC(CN(C(c2c(C)cno2)=O)C)O)coc2c(F)cc(F)cc12 c1(C(N(CCCNC(C2CC2C2CC2)=O)CC)=O)[nH]c2cccc(C)c2c1C c1(OC)ccc(CN2CCCC(NC(=O)C(O)C(C)(C)C)C2C)cc1Br c1(C(=O)NCCC2CCC(NC(CN(C)C3CC3)=O)C2)ccc(C#N)s1 c1(C(N2CC(C(=O)OC)C(C)C2)C(=O)NC2CC2)cc(C)ccc1C(C)C Cc1cc(Cl)ccc1C(=O)NC(CNC(=O)CSC(F)(F)F)Cc1ccccc1 c1(CC)nc(C)oc1C(N1CCOC(CC(=O)N(C(C)CC(=O)OC)C)C1)=O C1(NC(=O)C(C)Oc2ccccn2)CCC(C)(C(NC(C=C(C)C(F)F)=O)CN)C1 C(=O)(C#CCNC(c1nscc1C)=O)NC(C#C)CC1CC1 C12(C(=O)NCC(CCCC)NC(c3cc(C)cs3)=O)CCC(O)C1CC2 C1(NC(N(CC(COC)(F)F)C)=O)CCCC(C(=O)OC)C1 c1(CC(C)(C)C)noc2nc(C3CC3)cc(C(=O)OCC3CC(=O)NC3=O)c12 c1(CC=C)ccc(OC)c(NC(N2CCOC(CC(C)C)CC2)=O)c1 N1(C(c2ccc(CC)cn2)=O)CC(CNC(=O)C=Cc2cn[nH]c2)C(C)(C)C1 CC(CF)CC(=O)NCCN1CCC(NC(C2(Cc3ccc(Cl)nc3)CC2)=O)C1 C(=O)(CCN(C)C(C1(N(CCCO)C)CC1)=O)N(CC(C)O)C1CC1 C1(C2(O)CCOCC2)(C(=O)NCC2N(C(C3CC(C#N)(OC)C3)=O)CC2)CC1 N1(C(C2(CCC=C)CC2)=O)CCC(NC(=O)C(CC)OC2CCCC2)C(C)(C)C1 C(=O)(C(C)(C)CC1CCC1)N(C1CCC(NC(c2c(C)csn2)=O)C1)C Cc1c(Cl)ccc(C(=O)NCC(C)CNC(=O)C(C(C)C)N(C)C)c1F C1(CC)C(C(N2CCCC2CC2CCCC2)=O)CCN1C(=O)CC1CCCCC1 C1(NC(CCc2ccnc(C)n2)=O)CC2CCC1N(C(=O)COCCN(C)C)C2 Cc1ncc(C(=O)NC2CC3CC2N(C(=O)CCc2nncs2)C3)c(C(C)C)n1 c1(NC(CC(CC)O)=O)cnn2c1CN(C(=O)COCC(F)(F)F)CC2 C(=O)(C1=NNC(C(F)(F)F)C1)NC(CNC(C(c1ccncc1)C)=O)CC(C)C CC1CCOC(C(N2CCOCC2C(=O)NC2(CO)CC(O)C2)=O)C1 c1(CN(C(C(=O)NCCC)CC)C)cc([N+](=O)[O-])oc1C c1(C(C(C)OCC)NC(=O)NC2CC(n3cccn3)C2)ccccc1 C(=O)(C1=CCC2CCC1N2C(C1(C)CCCC1O)=O)NC1CC(CC(=O)OC)C1 c1(C(=O)NC2CC(N(C(CC=CC=C)=O)C)C2)sc(Cl)c(Cl)c1N CC1CCC(F)(C(=O)NC(CC(=O)N2CCC2)C2CC2)CC1 C(=O)(C(CC(N)=O)NC(=O)CC1CC=CC1)NCc1cc(C(C)C)on1 Cc1cc(C(N2CCCN(C(=O)CC3CSC3)CC2C)=O)c2ccc(F)cc2n1 C#CCC(CC(=O)NC(CO)CC=CC)NC(C1(CC)CCCCO1)=O C#Cc1cncc(C(=O)NC(CC2CC2)CC(=O)N(CCCO)CC2CC2)c1 Cc1cc(C(=O)N(C2CN(C(c3cc[nH]c3)=O)C2)C)c(O)nc1C C(=O)(CCC(=O)NN(C)C)N1CCC2C(C(NOCCOC)=O)C2C1 C1(C(N2C(c3nnc(C)o3)CCCC2)=O)CCCN(c2ccccc2)C1=O c1(OC)ccc(C=CC(=O)NC2C=CCN(C(C3(O)CCCC3)=O)C2)cc1F C1(NC(c2oc(C)c(CO)c2)=O)C2CC3C1C3C2C(=O)NCc1cccc(F)c1 N12CCC3(CC1)C(C3(F)F)C2=O.c1(OC)cc(Br)ccc1CCC(=O)NC(C)CO C(=O)(CCN1C(=O)CCc2ccccc21)NCCC1CCN(C(C=NOC)=O)C1 C1(NCC2CCC2)CCC1C(=O)NC1(CN(C(=O)CC2CC2)C)CC1 Cc1[nH]nc(Br)c1C(c1nnnn1C1CCOC1)NC(c1cccc(C(F)F)c1)C C(CN=C(NCc1ccc(F)c(F)c1)NC1CCOC1)C1(O)CCCCC1 C(=O)(C(C)(C)CCF)NCC(CC)NC(c1ccnc(C(C)(C)O)c1)=O CCC(C)C(C(=O)NCC1CN(C(=O)CSCCOC)CC1C)NC(C)=O CC1CN(C(c2cnc(S)nc2)=O)CCC1NC(c1ccn(C(F)(F)F)n1)=O C(=O)(C(O)CCS(C)=O)N(C1CCN(C(=O)COc2ccc(F)cc2O)CC1)C C1(N(C(C(C)C2CCC2)=O)C)CCN(C(C2CCCN2C(N)=O)=O)CC1 CC(CCC(=O)NCc1cnsc1)NC(=O)C(C)CN1CCCC1 C1(C(=O)OCC)CC(Cn2cc(CN3CC4CC4C3)nn2)CO1 N1(C(c2c(SC)csc2)=O)CCC(O)(C(C)NC(c2cc(Cl)ccc2C)=O)CC1 C1(F)(C(=O)NCC(N2CC(C)(C)C2)C)CCCN(C(N)=O)C1 N#Cc1cc(C(N2CCC(N3CCN(C(c4cccnc4O)=O)CC3)C2)=O)no1 C1(N(C(C2CC2n2cccn2)=O)CC)CCN(C(=O)Cc2cncs2)CC1 n1(CC)ncc(C(=O)N(C2CCN(C(c3cc(C4CC4)ns3)=O)C2)CCO)c1C N1(C(c2c(C)nc(C)o2)=O)CCCC(N(C(=O)CC2CCOC2=O)CCO)CC1 N1(C(CN2CCC(C)CC2)=O)CCOCC(C(=O)NC2CC(C)(C)C2)C1 c1cn2c(C(c3nnnn3CCN3CCOCC3)NC3CCCSC3)cnc2s1 C1(NC(Cc2ccc(CCC)cc2)=O)CN(C(c2cc[nH]c2C)=O)CCC1C c1(C(N2C(C)(C(=O)Nc3ccc(Cl)cc3CO)CCC2)=O)cc2ccccc2cn1 c1(CNC(c2n(CCOC)nnn2)CC2CC2(Cl)Cl)nnc2nc(C)ccn12 C(=O)(C#CC1(C)COC1)NC(C)Cn1cc(CNC(=O)CN2CCCNC2=O)nn1 Cc1oc(C(F)(F)F)c(C(=O)Nc2ccnn2-c2cccc(C#N)c2)c1C c1(C(=O)NC(CNC(C(CC)Br)=O)C(C)(C)C)cnc2scnc2c1 C1(CNC(c2c(C)ccc(F)c2)=O)CC2COCC2N1C(c1cccc(Cl)c1)=O N1(C(=O)NC(c2cccc(C)c2)C(C)(C)C)CCSC2(CCCC2)C1 C(CCC(O)C(=O)NC1CCCC1(C)N(C)C)NC(CC(CC)SC)=O CC(C(CO)NC(c1nc(C2CCCC2)no1)=O)NC(=O)CNC(C1CCC1)=O Cn1ccc(C(=O)NCC(C)(O)CNC(C2CCCN2C2CCCC2)=O)n1 C1(NC(CCn2c(CCC)ncc2)=O)CCN(C(=O)C(CC)C(C)C)C12CC2 c1(N2CCCC(c3oc(CC)c(C)n3)C2)cccc2c1OCCC2O c1(C(=O)NCC(CCOC)NC(=O)C(O)C(F)F)nc(Cl)ccc1OC N1(c2nc(N3CCC(F)(N(C)C)C3)nc3c2CCC3)CCOc2ccncc2C1 C1(OC)CC2(CCC(NC(C3CC3c3ccoc3)=O)CC2)C1 N1(C(c2c(C)nn(C)c2)=O)CCN(C(c2ccc(C(N)=O)cc2)=O)C2CCC12 C1(OC)(CNC(=O)C(O)C2CN(C(C3CN(C)CCO3)=O)C2)CCCCC1 c1(C(c2nnnn2C2CCOC2)NC2(CC)COC2)ccn(CC(F)(F)F)c1 C12(CNC(c3c(C)c(Br)no3)=O)CN(C(c3cnc[nH]3)=O)CC1CCO2 CCC(O)C(F)(F)C(=O)N(c1ccccc1C#N)C(C1CCOC1C)=O O=C(CC1=CCOCC1)NC(c1ccc(F)cc1F)CNC(=O)CS(=O)(=O)CCO C1(C(=O)N)(C)CCCCC1.CC(Cc1ccco1)C(=O)NCCC(C)c1cn[nH]c1 c1(C(=O)NCCC2CCN(C(C3(C#N)CCC3)=O)C2)ccc2c(O)nncc2c1 N1(C(Cc2nc(C)[nH]n2)=O)CC=C(CNC(=O)CC2CCC(=O)C2C)CC1 CCCC(C#N)C(=O)N1CC(NC(c2ccc(N(C(CC)CC)C)cc2)=O)C1 Cc1nccc(C(=O)NCCCNC(=O)CC2CCC2(C)C)n1 CCC1(C)CNC(=O)CCN(C2CC2)C1=O.c1(CC(=O)NC)cc(C)nn1C Cc1ccccc1C(C)NC(=O)C(C1(O)CN(C(=O)Cn2cc(Cl)cn2)C1)F N1(CCO)CCCN(C(=O)CC2CNCC(F)C2)CC1.c1(C(=O)N)cscn1 C1(NC(C(C)N(C(c2cc(C)ncc2C)=O)C2CC2)=O)CCn2nccc2C1 C1(NC(=O)COc2ccc(Br)cc2)CCSC12CN(C(C1CC1[N+](=O)[O-])=O)C2 c1(SC)nc(O)c(C(N2CC3(CC(NC(=O)CNC=O)CO3)C2)=O)cc1C#N Cc1cc(OCC(N2CCCC2CCNC(c2cnn(C)c2N)=O)=O)cc(C)c1 C1(NC(COC)=O)CCCC12CN(C(c1sc(-c3ccccc3)nc1C)=O)C2 N1(C(=O)C(F)(F)F)CCCC(CO)CC1.c1nncn1C1CC1 c1(C(N2CC3CN(C(=O)CCCCBr)CC32)=O)cccc2c1C(=O)CC2 C(N=c1[nH]c(=NCCC2CCSC2)[nH]c2cccc(F)c12)C1C(C)(C)CC(=O)N1 CC1CCC(C)N1CC(=O)NC12CC(C1)N(C(=O)C(=O)NCC(F)F)C2 N1(c2snc(CC)n2)CCCCC(CNC(c2n[nH]cc2CC)=O)C1 N12CC(F)CC1CNC(C1CC1)C2=O.CC(C(=O)NC1(C)N=N1)ONC=O Cc1ccc(C(N2CCOC(CCNC(C3CCCC3C)=O)C2)=O)c(N)c1 N1(Cc2cc(C)on2)CCN(C(C2(CC(C)C)CCC2)=O)C(C)C1 N1(CC)CCCC(C(=O)NCCCC(C)NC(c2cc(C(C)(C)C)nn2C)=O)C1 C1(c2ccccc2)(C(N(C2CCN(Cc3cccnc3)C2)C)=O)CC(F)(F)C1 C1(NC(CN2CC(=O)NCC2)=O)CCC2CC1CN2C(c1nc(Cl)sc1Cl)=O c1(C(=O)NCC2CC(NC(c3nc(C(C)(C)C)oc3)=O)C2)cnc(S)nc1 C1(NC(C(C2CCC2)OC)=O)COC2(C1)CN(C(=O)Cc1ccsc1C)C2 Nc1c(C(=O)NC(CNC(c2ccc(Br)o2)=O)CO)cc(Cl)cc1Cl C1(NC(=O)Cc2sc(O)nc2O)CCCN(C(=O)Cc2cocn2)CC1 CCC(CCC(=O)OC(C)(C)C)S(=O)(=O)N(CC(N)CC)C1CC1 c1(C(N2CCCC(CC(=O)Nc3cc(CCC)no3)C2)=O)cc(F)ccc1O c1(NC(CC#CC)CO)cc(Br)ccc1S(=O)(=O)NCC1CC(O)C1 C(=O)(C1=CC(C)(CC)C1)N1CCC(C(C(=O)N(CCC(=C)C)CC)C)CC1 O=C(CC(C1CC1)C1CC1)N(C1CCCC1)CC(=O)NCc1csc(O)n1 N1(C(c2n(CC)cc(Cl)c2)=O)CCCC(NC(=O)CCCn2ccnc2)C1C C(c1ccccn1)=CC(=O)NCCCCCNC(C1CCC1c1nc(S)n[nH]1)=O N1(C(=O)NCc2cccc(C)c2I)CCC2(CC1)CC(O)CO2 C(=O)(C1Cc2ccccc21)N1C(CNC(c2cnc(CCCC)s2)=O)CC(O)C1 Cc1ccc(C(C)NC(c2conc2CNC(C2OC3CCC2C3)=O)=O)cc1 C1C(CCC)C(=O)N1.C#CCN(CCOC)C(C)=O Cc1cc(C(N2CCCC(N(C(=O)Cc3[nH]cnc3C)C)C2)=O)c(C)[nH]1 c1(SC)c(NC(=O)C(=O)NC2CCC(C)(C)C2)cccc1F N1(C(C(C2CC2)OCC)=O)CCCC1C(C)NC(c1cc(-c2cccs2)on1)=O CN1CCc2nc(C(=O)NCC3(C)CCCN(C(C4CC=CC4)=O)C3)sc2C1 C1(C(=O)NC(c2ccncc2)C)(CC)CCN(C(=O)CSC)CC1 Cn1cnc2c(NC3CCC3)[nH]c(=NCCSc3cnccn3)nc12 CC1OC2(CNC(c3n[nH]cc3Cl)=O)CC1(NC(c1cc(Cl)ccc1F)=O)C2 CCCC(C(=O)NCC1CN(C(=O)C(C)SC(F)(F)F)CC1C)S(N)(=O)=O C1(C)(NC(CC(=O)NCC#C)=O)CCN(C(C2CCCS2)=O)C1 C(=O)(C1=CC2CC=CCC12)NCC1(O)CN(C(c2cc(C)c(N)cn2)=O)C1 C1(NC(C2C(C)(c3cccs3)C2)=O)CN(C(c2ccc(F)s2)=O)CCC1O N#CC1(C(=O)NCC2(F)CC(NC(=O)CNC(=O)C3CC3)C2)CCCCCC1 N1(C(C(C(C)(F)F)(C)C)=O)CCC2(CCN(C(C34CCCC3(C(N)=O)C4)=O)C2)C1 c1(OC)ccc(C(=O)NCC(CC(C)C)NC(c2cccc(CO)n2)=O)c(F)n1 C1(C(N)=O)CC2(CCC(C(=O)N=c3cc[nH][nH]3)CC2)C1 c1(-c2nc(CCC(=O)NCC(C)(CO)C(C3CSC3)=O)on2)ccc(Cl)cc1 c1(C2(NC(C(n3cc(CCNC(C)=O)nn3)C)=O)CC2)ccnc(Cl)c1F C(=O)(C(CCSc1nc(N(C)C)no1)NC(N)=O)NCCN(C)CCO N1(C(c2cccc3oncc23)=O)CCC2CN(C(c3ccco3)=O)CCC2C1 c1(C(N2CCCC(CCNC(=O)C3CC3)C2)=O)cncc(CC(F)(F)F)c1 Cc1cn2ccc(NC(C3CCC4(CN(c5snc(Cl)c5C#N)C4)O3)=O)cc2n1 CC(Cc1ccccc1)C(C(=O)NC1CCC1)N1CCCCC1C(C)(C)O.C(CO)N Cc1cc(CNC(=O)CCN(C(=O)CC=C(Cl)Cl)CCO)nnc1C CCC(C)(CO)C(=O)N1CC2CC2(C(=O)NC2CC(CCO)C2)C1 N1(C(C2N(C(c3c(C)nccn3)=O)CC(O)C2)=O)CCC2(CC1)CC2C#N CC1CCCN(C(=O)CSCC2(C(=O)N)CC2(F)F)C1CO.C1(S)CCOC1=O C1(NC(CCc2cc(C)nc(C)c2)=O)CN(C(c2ccc(F)s2)=O)CC12CCC2 C1(CC)C(=O)NCCN1C(=O)CC(C(C)C)NC(C1(C)COC(=O)N1)=O C1(NC(COC2CC(NC(C(C)(C)F)=O)C2)=O)CC12CCOC2 C1(N(C)C)CCC(CC2CC2)CC1.c12cn(nn1)CC(=O)N2CCS(C)(=N)=O C1(NC(CCCCCC)=O)CN(C(c2ccc(C#N)nc2O)=O)CC1C1CC1 c1(C(=O)NC2CCC23CN(C(=O)Cn2cncn2)C3)cc2nc(=O)ccn2[nH]1 c1(C(N2C(CNC(c3cocc3C)=O)CC(OC)C2)=O)cncc2cccnc12 n1(CCOC)nc(-c2ccc(C(F)(F)F)nc2)nc1CC(C)CC(F)F c1(C(=O)NCC2(C)N(C(C(C)CO)=O)CCC2)cc2n(n1)CCO2 N1(C(C=COCC)=O)CCCC(NC(c2cnc(N3CCOCC3)s2)=O)C(F)C1 c1(C(N2CCN(C(C(CC)F)=O)CC(CO)C2)=O)ccc(S(C)(=O)=O)cc1 c1(CNC(CC(=O)OCCOC)=O)cnc2ccccn12 C1(NC(C=C(CCC)C)=O)CCN(C(C2CC(=O)N(OC)C2)=O)CC1C C(=O)(C(C(C)C1CC1)N1CCCC(O)C1)NCCCSC.C(C)(C)(C)O C1(O)(CNC(C(CC(CC)CC)F)=O)CC2CCC(C1)N2C(C1CCC(=O)C1)=O c1(C(=O)NCC2C(CNC(CC3(COC)CC3)=O)C2)cc(C)c(Br)c(Cl)c1 c1(OCC)nccc(OC)c1C(=O)NCCCNCC#N.c1(N)cccc(OC)c1 CN1CCCC(CC(=O)NC2CCCCC2NC(c2n[nH]cc2C2CCC2)=O)C1 O=C(C1=NOCC1)NC1CC(NC(C2CCCN2CCC(F)(F)F)=O)C1 CCC(C)CC(C)C(=O)N1CCC(N(C(=O)CC(C)C2CCCO2)C)CC1 N#Cc1ccc(C(=O)NC2CCCC(CNC(C3CC34CC4)=O)C2)s1 C(=O)(C(C)CC(N)=O)NC(C1(C(=O)NC(C)CC2SC(=N)NC2=O)CCC1)=O n1(CCC)nccc1C(=O)N(CC(C)CNC(c1nocc1Br)=O)C c1(C(N(C2C(C)CCN(C(CC(C)F)=O)C2)C)=O)ccn2nnnc2c1 C1(N(C(=O)C=Cc2nn[nH]n2)CC)CC2CCC1CC2 C1(CCNC(CC2C(CC)C2)=O)CSCCN1C(=O)Cn1cnc(C#N)n1 N1(C(c2c(C)cc(N)cc2)=O)CCC2(C1)CN(C(C1CCn3nncc3C1)=O)C2 N1(C(C2(c3ccn(C)n3)CC2)=O)CC2CCC1CN2C.c1(NCCO)ccccc1 C#Cc1cnn(C)c1C(N1CC(=O)CC1C(N1CC(=O)NC(C)C1)=O)=O C1(N(C(=O)CC(F)(F)c2ccccn2)C)CC2C(O)C(O)CC12 c1(N(CCN2CCC(CC)C2)CCNC(C)=O)cc(C(F)(F)F)cnc1C c1(C(N2CCC(NC(c3ccc(OC)s3)=O)CC2C2CC2)=O)ccc2nonc2c1 c1(C(N2C(c3ccc(C(F)(F)F)cc3)CCC23CC3)=O)ccc2c(c1)CCCN2 c1(C(N(CC(C)NC(C2(CC#C)CC2)=O)CC)=O)cccc2sccc12 c1(C(=O)NC(CC)CN(C(=O)C(c2ccnn2C)C)C)ncc(C)cc1F c1(N2C3CN(Cc4c(C)c(F)c(F)cc4)CC32)ncnc2[nH]cc(C#N)c12 C1(C(C(=O)NCCN(C(c2nc(CCC)oc2)=O)C)O)CCC(F)(F)C1 C(=O)(C1CCCc2nn[nH]c21)NC(CNC(c1c(CC)scn1)=O)(C)CC(C)C N1(C(c2c(C)noc2C)=O)CCN(C(=O)Cn2nnc(=O)[nH]2)C(CCO)C1 CC1CC(CNC(=O)CCc2cncn2C)CN1C(=O)CCCCC1CC1 C(=O)(CCC(C)(C)[N+](=O)[O-])NCC(N(C(C(C=CC)O)=O)C)C1CC1 C=CCCCC(C)(C)C(=O)N1CCC(CC(=O)NC(COCC)C(C)C)CC1 c1(CNC(CCOC)(C)c2nnnn2C)cccc(C)c1F C1(CC(=O)NCC(CN(C)C(c2ccc(Cl)[nH]2)=O)O)CCCN1C N1(N(C(c2c(-n3cc(-c4cc(C)nn4C)nn3)ccs2)=O)C)C(C)COCC1C c1(OC)c(NC2CC(NC(c3ccc(CO)c(F)c3)=O)C2(C)C)ncnc1Cl N1(C(CC=C=C)=O)CCC(C)C1CNC(=O)CC1CCC(OCC)CC1 CC1(CNC(c2ccc(N)cc2)=O)CCCN1C(C1CC2C=CC1C2)=O C(=O)(C(C)(C)CCNC(c1ccc(F)c(Cl)c1)c1nnnn1C1(C)CC1)OCC C1(NC(c2ccc(C)c(N)c2)=O)CC2(CCC(NC(C3CC3(Cl)Cl)=O)CC2)C1 C(=O)(C(C)(C)CCCF)N(CCN1CCN(C(C(CCC)O)=O)CC1)CCOC C(=O)(CCC(=O)NCC(C(C)(C)C)NC(=O)CCCc1nc(CC)no1)NCC O=C(C#Cc1cc(Cl)ccc1N1CCCC1)NC12CCCCC1C2(F)F CC1Cc2ccc(OC3CC3)cc2N1C(=O)NCCC(O)C1CCCC1 CCC(C(=O)NCCN(C(=O)Cc1ccsc1)C(C)C)SC c1(C(N2CCC(C)C(CNC(=O)C(F)(F)C3CC3)C2)=O)cc2ccc(F)cc2s1 CC(C)(C)C#CC(=O)N1CC(C)(C(=O)NC2(CO)CC(F)C2)C1 C(CCC(=O)NC1CC(F)(CNC(C2CCC(C)O2)=O)C1)=CC CCCCC(C)C(=O)NC1CC(F)(CNC(=O)CN2CC(=O)N(C)C2=O)C1 c1(N(C2CCN(C(Cc3cnc(C)[nH]3)=O)C2)C)c(C)noc1C c1(C(=O)NCC2CCC(C(=O)Nc3c(OC)nccc3)C2)cccc2occc12 N1(C(=O)Nc2ccc(CC(=O)OC)cc2SC)CCC2(CCSC2)C1 c1(CC(=O)NCC2CC(OC)CN2C(=O)CCCC#N)c[nH]c2ncccc12 C1(C(=O)OC)CCCCN1C(C12CC(NC(=O)Cc3ccc(O)nn3)(C1)C2)=O C1(CC(N2CC(C)C(NC(=O)CNc3cccnc3)C2)=O)CCCCC(=O)N1 c1(CNC(=O)NCC2(c3ccncc3)CC2)nc2ccccc2[nH]1 C(C(C)(C)CC(=O)NCCCOCCN(C)C(c1conc1C(C)OC)=O)OC c1(C(=O)NCCc2cccc(C)c2)ccc2cc(Br)cnc2c1 N1(CC(=C)C)C(=O)NC(c2cccc(C(=O)OC)c2)C(C(=O)OCC)=C1COC C1(C)(NC(c2cccc(CC)n2)=O)CCCN(C(=O)CC(C)COC)C1 C(=O)(CCCCC(=O)N1CCC(C2(NC(c3cccc(CF)c3)=O)CC2)C1)OC C1(C(N(CCNC(=O)CC2(N(C)C)CCCC2)C2CC2)=O)CC12CCCC2 c1(C(=O)NC2CN(C(C3CCCC(=O)N3)=O)CC2F)c(F)ccc(Cl)c1F c1(CNC(=O)NCC(=O)NCC(C(C)NC(CCC)=O)=O)cc2cccnc2s1.NCC CCC(C#N)C(=O)NC1CC(CNC(c2ccc(CNS(C)(=O)=O)o2)=O)C1 c1(NCCN(C(=O)NC(c2cccnc2)C)CC)ccc(Cl)c(N)c1 C1(C(=O)NC23CC(CNC(c4ccn(CCC)n4)=O)(C2)C3)CN(C)CC1C CCCC(CC)CCC(=O)NCC(C)C(=O)NCCN1CCCC(O)C1 S(=O)(=O)(c1cccc(=NC(C)c2cccc(Cl)n2)[nH]1)N(CCOC)C C(CC(=O)NCC(C)(C)C1CCCO1)(C(F)F)NC(C(=Cc1ccccc1)C)=O C1(CC(=O)NCCOCCCNC(C2C(C)(C(F)F)C2)=O)CC2(CC2)CO1 CN1CCCCC1CC(N1CCC(N(CCO)Cc2ncc(C(F)F)o2)C1)=O c1(C(N(C(CC(=O)N(CCCC)CC)C)C)=O)nnc(S)n1C C(=O)(CC(C(F)F)NC(C)=O)NCCN(c1ccccc1)CCC CCCCC(C(=O)N1CCCN(C(=O)C(C2CCCCC2)F)CCC1)C(C)C C1(C(=O)NCC(C)(CO)NC(C(c2cn(C)nc2)O)=O)CCCCCC1 c1(C(N2CCCC2c2ncc(C)s2)C(=O)NCC)ccc2c(c1)CCC2 C1(C(=O)NC2(CSC)CCC2)CN(C(=O)C(C2(O)CCCC2)F)CC1F CC1(C)Cc2cc(C(N3CCN(C(=O)C=C4CC4)C(CO)C3)=O)ccc2O1 C1(C(N2CCC(C(C(=O)N(CC(N)=O)CC)F)C2)=O)CC2(CCC2)C1 C1(C(=O)NC2C=CCN(C(C(OC)OC)=O)C2)COc2ccc(O)cc2O1 C1(Cn2cc(C3CN(C(C(CO)N(C)C)=O)C3)nn2)CC(F)(F)C1(F)F CC1(C)NC(=O)CC1C(=O)NCC(C1CCCN1C(C1CCC(=O)C1)=O)(C)C Cc1cc(Cl)cc2cc(C(=O)NCC(C(F)(F)F)c3ccccc3)oc12 c1(C(=O)NCC2(F)CN(C(C3C(C)C3(F)F)=O)C2)cc(N(C)C)nc(Cl)c1 C=C(C)c1cccc(NC(C2CC(O)CN2C(c2cc(C)sc2N)=O)=O)c1 C1(NC(=O)Nc2ccc(C(=O)NC(C)C)c(F)c2)CCc2ccccc2C1 CON1CCC(C(=O)NCC2CC2C(=O)NCCC2CC(C)(C)C2)CC1 C1(C(=O)NCC2C(NC(Cc3c(C)ocn3)=O)C2)CCC2CC2CC1 C(CO)(CCCCNC(C1CCC(=O)N1)=O)NC(Cc1c(C)ccs1)=O c1(CN2CC(C(=O)Nc3c(C(=O)OC)cc(C)cc3)C2)ccc(OC)c(C)c1C c1(C(=O)NC2(CC(=O)NC3CCN(CC)C3)CC2)cccn2cncc12 C1(CCOC)CN(C(c2cc(OC)ncc2C)=O)CCN1C(C1CC1C1CC1)=O CCC(CCOC)C(=O)N1CC=CC1CNC(c1cccc(OCC(F)F)c1)=O C1(CC)(NC(C2CCCCN2C(=O)Cn2cccn2)=O)CCCCC1 CCCC(O)CC(=O)N1CCC(C(C)(C)C)(NC(c2cnc(C(C)C)nc2)=O)C1 Cc1cc(C(=O)NC2CC(N(C)C(c3ccn(CCN(C)C)n3)=O)C2)ncc1F c1(C(N(CCCCCCNC(C2C(Cl)(Cl)C23CC3)=O)CC)=O)cc2c(o1)CCCC2 CC(C)C(O)C(F)(F)C(=O)N(C)CC1CC(C)C1.C(=O)(C(C)C1CC1)N C1(C)(NC(C(CNC(C=C(C)C(F)F)=O)CC2CCCC2)=O)CN2CCC1CC2 N1(C(CCc2ccc(C(C)C)cc2)=O)CCC2(NC(=O)CC3(C)CC3)CC2C1 N1(C(CCCCN(C)C)=O)CCC2(CC1)CC2C(=O)NC(CO)CCF C=CC(CC)CC(=O)NC(c1ccc(F)cc1)CNC(c1nnn(C)c1C)=O N#CC1CC(C(N2CCC2CNC(=O)CCCC2CCOCC2)=O)C1 C#CCC(O)C(=O)NCC1CCN1C(c1ccc(Br)s1)=O c1(CC(C(C)=O)OC(c2nc(Cl)sc2Br)=O)ccc(Br)cc1F c1(C(=O)NCC2CCN(C(C3CN(C)C3)=O)C2)c[nH]cc(Br)c1=N C(CC(O)C(F)F)NC(C(C1CC(NC(=O)CCC2CCOC2)C1)F)=O n1(CC(=O)NCCC(C)N(CCC)C(C2CCOC2)=O)cnc(C(F)(F)F)c1 C1(C)(OC)CCCN(C(=O)COC23CCC2CN(C(=O)Cc2cn[nH]c2)C3)CC1 N1(C(c2nc(OC)nc(O)c2)=O)CC2CCCC(C1)N2C(=O)CC(F)(F)C(F)F CC(O)CC(=O)NCC(C)(F)CNC(c1sccc1Cl)=O C1(C(=O)NCC2COCCN2C)(CC)CCN(C(=O)Cc2ccc(C)cc2)CC1 C(C)(C(=O)N1CC(C(N)=O)C1)S.C(=O)(COCCF)N(C(C)C)C CCCC(C)(CC)C(=O)NC1CC(CCNC(c2ncc(N)cc2Cl)=O)C1 N1(C(CC(C)SC)=O)CC2CCC1C(NC(=O)C=C(C)c1cccnc1)C2 c1(SNC(CNC(=O)Cc2cnoc2)=O)cccc2ccccc12 C(C1COC(C)(C)O1)=CC(=O)NC1CC(CNC(C=CCOCCOC)=O)C1(C)C C1(NC(C(C)OC2CCCC2)=O)CCC2(CCN(C(c3cncc(Cl)c3)=O)C2)C1 C(=O)(C1=NOC2(CCC2)C1)NCC1C(C(N2C(C)CCC(CO)C2)=O)C1 N1(C(CC(COC)C)=O)CCC(C)(C)C(CNC(=O)C(F)(F)C2CC2)C1 CCCCC(C(=O)NC1CN(C(=O)Cc2ccc(CO)cc2)CC12CC2)C(C)C C12(C(N(CCCN(C(C)=O)C)C)=O)CCC(NC(C3CC3C(F)F)=O)(CC1)C2 N1(C(C2C(C)(C)C(F)(F)C2)=O)CC2CCOC2(CNC(C2CCCN2C2CC2)=O)C1 C12(NC(C(CC=CC)C)=O)CCOC(CNC(c3csc(C(C)=O)n3)=O)(C1)C2 CC1(C)CS(=O)(=O)CCN1CCNC(=O)CC1CCCN(C(=O)C(O)CC[S+](C)C)C1 CC1C(NC(C2(Br)CC2)=O)CCN1C(=O)Cc1ccccc1 Cc1cnc2scc(C(=O)NC3CCC(CN(C(=O)C(F)(F)C(C)O)C)CC3)n12 N1(C(c2c(C)ncs2)=O)CCCCCC1C(=O)NOCCCN(C)C N1(C(CC2(C)CC(NC(CC3ON=C(C)C3)=O)C2)=O)CC(O)C(O)C1 c1(C(N2CC(F)CC(NC(CN(C(COC)=O)C)=O)C2)=O)ccc(C#N)c(C)n1 Cc1cc(Br)cnc1Sc1cccc(C(=O)OC(C)(C)C)c1 C1(CNC(C(C)(CC2CC2)OC)=O)CC2(CC2)CN1C(=O)CCN1CCCCC1 N1(C(c2c(CC)nccn2)=O)CCC(C2CC2)(CNC(=O)CCCC2CC2)C1 C(=O)(C(CCC(C)C)NC(c1cnn(C(C)C)c1)=O)N(CC=C)CCC C1(C2CC2)(CNC(c2n(C)c([N+](=O)[O-])cn2)=O)CCN(C(=O)C(F)OC(F)(F)F)C1 c1(C(N(CC2N(C(C3N(CC)CC3)=O)CCC2)CC)=O)cc(C2CC2)ccc1F Cc1nc(C)c(CCC(=O)NCC2CCN2C(c2cccc(C)c2Cl)=O)c(O)n1 CCC(CC)C(C)C(=O)NCC(CC)NC(=O)CN1CCC(O)CC1 O=C(CCCCC(F)F)NCC1CCCN1C(C1(c2ccccc2)CC1(F)F)=O c1(C(=O)NC(CCSC)C(=O)NCCC2NC(=O)NC2=O)cc(C#N)ccc1N CC(C)(C)S(=O)(=O)CC(=O)N1CC2CCN(C(C3C=CCCC3)=O)C2C1 C(=O)(CC(F)(F)C(F)(F)F)N(C)CC1N(C(CCn2ccc(C)n2)=O)CCOC1 C12(COC)CN(C(C34CCCCC3C4)=O)C(CNC(c3cc(C)cs3)=O)(C1)C2 C1(C(N(C(CN(C(CCC=C(C)C)=O)C)C)C)=O)CCCOC1C C(=O)(C(F)CC(C)(C)C)N(C(CNC(c1ccncc1F)=O)C1CC1)C c1(C(=O)NCC(C)NC(c2n(C(CC)C)ncc2)=O)ccc2c(c1)CCO2 c1(C(N2CC(F)(CNC(C(C)(CO)OC)=O)C2)=O)ccc2nc(C3CC3)[nH]c2c1 C(=O)(C1=CC2(CCN(C(=O)Cc3ccn(C)n3)C2)C1)N(CC(=O)OCC)CC=C C1(CNC(c2c(C)nsc2)=O)CN(C(c2ncoc2CO)=O)CC1N(C)C C(=O)(C1CCOc2ccccc21)N(C)CCOCCN(C(=O)C(C)(C)O)C N1(C(c2cncc(OC)c2)=O)CCC(NC(c2cc(C3CC3)on2)=O)C1(C)C C(C(C(C)(C)C)NC(c1cnn(CC(F)(F)F)n1)=O)NC(c1nc(CC)oc1)=O CCCCC(CC(=O)N1CCC1C(C)O)NC(c1cccc(C)c1O)=O C12(CNC(CC3CC(=O)C3)=O)CN(C(c3cccc(O)n3)=O)CC1CS(=O)(=O)C2 c1(C(=O)NCC(CC(C)C)NC(CC2(OC)CCC2)=O)cc2cccc(C)c2s1 C1(NC(=O)CCc2cccc(F)c2)CCN(C(c2n[nH]cc2Cl)=O)C12CC2 C1(CNC(C(c2c(C)cccc2)(C)C)=O)CCC(C)(C)CN1C(=O)C(C)C1CC1 c1(C(=O)NC2(CO)CN(C(COCC=C)=O)C2)ccc2c(c1)nc(CO)n2C N1(C(C(C)CN2CCOCC2)=O)CC2(CC(NC(c3cnccc3Br)=O)CO2)C1 C1(C(=O)NC(CN(C(c2ncc(C)cc2C)=O)CC)C)CCN(S(N)(=O)=O)CC1 C(CC(C(=O)NC1CC2(C1)CC2C(=O)N(C1CCCCCC1)C)OC)OC C1(NC(c2nc(C(C)C)oc2)=O)CN(c2nccc(C#N)n2)CCC1C C(=O)(CC(COC)COC)NCC1(COC)CN(C(C2COCCN2C=O)=O)C1 CC1CC(=O)NCC1C(N1CC(C)(CCC(=O)NC2CCCCNC2=O)C1)=O c1(C=O)cc(C)c(C)nc1O.Cc1cc(O)cc(C)c1.C1C(=O)NCC2C1C2 C1(C(=O)OC(C)(C)C)CCOC(c2cnn(C)c2)C1.C1(Br)=C(C)CNC1 n1(CC)nnc2c1CCN(C(c1n[nH]c3cc(Cl)ncc13)=O)C2 C1(CC(=O)NCC(COCC)C)COCCN1C(=O)COC1CCCC1 C1(C(=O)NC(C=C)C(F)(F)F)CCN(C(c2cc[nH]c2C2CC2)=O)CC1O C1(CC)CCC(C)CN1C(C1(NC(c2cncn(C)c2=O)=O)CC1C)=O C1(C(N(CCO)Cc2cc(C)no2)=O)COCCN(C(=O)CNC(N)=O)C1 c1(C(=O)NC2C(SC)CN(C(=O)Cc3cc[nH]c3)C2)cc(C)c(Cl)cn1 c1(C(=O)NC2CC(=O)N(C3CN(C(C4(CF)CC4)=O)C3)C2)cc2ccc(F)cc2s1 c1(CC)sc(C)cc1NC(C1CCC(C2CC2)N1C(c1ccc(OC)nn1)=O)=O Cn1ncc(CC(C(N2CCC(C#N)C2)=O)C2CC(c3ccccc3)C2)c1O Cc1nc(N(C)C)sc1CCNC(C1CC1NC(=O)C(C)(C)c1cscn1)=O C(C(C(=O)N1CCCC1CCNC(=O)CCCF)NC(C)=O)OC c1(CN(C)CC2CCN(C(c3ccc(Cl)cc3O)=O)C2)cc(Cl)ccc1[N+](=O)[O-] C1(CCC(=O)NC(C(C)C)C2CCC2)CCCCN1C(=O)CN1CC2CCC1C2 N1(C(c2ccc(C=C)cc2)=O)CCC2C(CCN2C(=O)CC(C)F)C1 C1(NC(Cc2cc(C)ncc2)=O)CCCN(C(=O)CCc2ccco2)C1C(C)C C=CCC(F)(F)C(=O)N1CCC(n2cc(CC(C)O)nn2)CC1 C(=O)(CC1=CCN(C(=O)CC(C)n2ccnc2)CC1)N1CCCC(C#C)(C)C1 c1(CNC(C(=O)NN2CCOCC2)=O)ccc(SCC)c(F)c1.Cc1c(C(=O)C)cnn1C CCCC(C)CC(=O)NC1CC(F)(F)CC1NC(c1ccc(Cl)cc1OC)=O C1(NC(CCCOCC=C)=O)CCC2(CC1)CC(NC(=O)CN1CCCCC1)C2 CN1CCN(c2cc(-c3cnc(C(=O)Nc4cnccn4)cn3)ccn2)CC1 C(C)(C(=O)NCC(C)(C1CC1)NC(=O)OC(C)(C)C)SC C1(C(N(CCNC(=O)C=CBr)C2CC2)=O)CCC2C(CC1)C2(F)F N1(CC(=O)NC(C(C)(C)NC(C(C)OC2CCCC2)=O)C)CC(=O)NC1=O C1(CNC(CCN(C(CC)CC)C)=O)C2CN(C(C3(CF)CC3)=O)CC12 Cc1c(C(=O)NC(C)CCNC(C2(C(C)C)COC2)=O)cnn1C(C)(C)C CCCC(C(=O)NCC(C1CCCCC1)NC(c1ccccc1)=O)NC(C)=O Cc1nc(NC(=O)N=c2ccn(-c3cccc(F)c3F)[nH]2)nc2ccc(F)cc12 C12(NC(=O)Cc3cscn3)CCCN(C(=O)Cc3c(F)cncc3Cl)CC1C2 C(=O)(CC(C)P(C)(C)=O)NC1CCC(NC(COc2ccc(C)cc2)=O)C1 N1(C(C2(OC)CCC2)=O)CC(CNC(=O)CCCc2ccncc2)CC(C)(C)C1 N1(C(C2(C)C(C)CCC2)=O)CC(F)CC1C(=O)NCc1c(F)cncc1F c1(C(N2CCC(NC(C(CC)N3CCCC3=O)=O)C2)=O)cc(C)nn1C C(=O)(C(C(=O)OC)SC)NC(C1CC=CCC1)C(=O)NCC(=C)F c1(C(=O)NCC2(NC(c3cocn3)=O)C(C)CCCC2)cc2ccc(Cl)cn2c1 c1(C(=O)NCC(C(C)(C)C)NC(=O)CN2CCCC2)cc(S(N)(=O)=O)cs1 c1(C(=O)NC(C)C(=O)NCc2ccncn2)cc(S(C)(=O)=O)co1 C1(CNC(C(c2n(C)cnc2)O)=O)C2CN(C(=O)CN3CCSCC3)CC12 N1(C(C=CCCC)=O)CCCCC(NC(=O)C(c2ccc(C)cc2)C2CC2)CC1 C1(C(=O)NC(c2ccccc2)CNC(C2(NC(C)=O)CC2)=O)CCC(=O)N1C C1(NC(CC=C(C)C)=O)COC2(C1)CN(C(C13CC(F)C1C3)=O)C2 c1(-c2cn(CC(CN(C)C)O)nn2)ccncc1Br C#Cc1ccc(C(=O)OC)cc1.C12CCC(CC1)CC(=O)NOC2.C1(CC)C(=O)N1 N1(C(C(C(=O)OCC)F)=O)CC2CCC(C1)C(NC(=O)Cc1nn(C)cc1Cl)C2 C1(NC(=O)COCc2cccc(Cl)c2)CC2CCC1N2C(c1ccon1)=O C1(NC(c2ccn(C(F)F)n2)=O)CC2(CCN(C(=O)CC=C(Cl)Cl)C2)C1 c1(C(=O)NCC2C(CNC(C=C(CC)C)=O)C2)oc2ccc(Cl)cc2c1C CC1CCCC=C1C(=O)N1CCC2C(C(=O)N(CCCO)CCO)C2C1 C1(NC(c2c(C)nc(C(C)C)o2)=O)(CO)CCCN(C(C2(C)CCCN2C)=O)C1 CC1CCN(CC(N2CCSCC2C(=O)NCCCC2CCOC2)=O)CC1 c1(C(N2CC(C)(C(=O)Nc3cncnc3)C2)=O)n[nH]c2ccccc12 c1(CC(n2cccn2)C)nc(Cc2cccs2)nn1-c1ccccc1OC(F)F c1(C(N2C(CNC(C=CCN(CC)CC)=O)CCC2)=O)cccc2nc(Cl)cn12 C1(C(N2CC(OCC3(C(=O)Nc4ccc(F)s4)CCC3)C2)=O)CN(CC)CCN1C c1(CN2C(CCC(N3C(C(=O)OC)CSCC3)=O)COCC2)ccc(F)c(F)c1 C(=O)(C(C)(C)CS(C)(=O)=O)NC(C(C)NC(c1cccc[n+]1[O-])=O)CO C(=O)(C1=CC(C)(C)C1)N(C1CC(NC(=O)CCc2ccccc2C#N)C1)C Cc1ccc(Br)c(Cl)c1C(=O)NCC(C)(C(C)C)NC(c1cnns1)=O C(=O)(CCCCCCS(N)(=O)=O)NCC(CO)NC(C1(NC(N)=O)CCCCC1)=O C1(C(=O)NC(C2(O)CCN(C(c3c(CC)cncc3)=O)C2)C)CCC2CC1CO2 c1(CC)noc(C)c1NC(C1CCC(C)N1C(=O)CN1CCC(F)CC1)=O Cc1ccc(C(N2CCCC(C)(NC(C3CC(C)CO3)=O)C2)=O)c(C)c1 N1(C(C(CC#C)C)=O)CC2(CCN(C(c3ccc4cnccc4n3)=O)CC2)C1 c1(N2CCC(CNC(c3c(C(C)C)sc(Cl)n3)=O)CC2)cc(C(N)=O)nc(Cl)n1 N1(C(Cn2ncc(C)c2)=O)CC2(CC(NC(C3(C(N)=O)CC3)=O)CO2)C1 CCCCC(O)C(=O)NC1CCN(C(c2ccnc(C3CC3)n2)=O)CC1O S(=O)(=O)(c1cccc(C#N)c1)N.C1(C2CN(C(=O)CC3CC3)C2)(NC(C(F)=CC)=O)CC1 N1(C(C(CCOC)OC)=O)CCC(C(=O)NCC(N2CCOCC2)=O)CC1C C(CC(=O)N1CCC(NC(=O)CCC(=O)Nc2nnc(C)s2)C1)(C(C)C)OC N1(C(=O)NC(c2ccccc2OCC)CC)CC(Cc2ccsc2)C(C)CC1C c1(C(N2CC(CNC(C3C(C)C3C)=O)OCCC2)=O)c[nH]c2cc(F)c(F)cc12 N1(C(c2n(C)cc(Cl)c2)=O)CCN(C(c2ccc(C#N)n2C)=O)C2CC12 n1(C(C)C)cnc2c(N(CCCO)C)[nH]c(=NCCC3C4CCCC34)nc12 n1(C(=O)NCC2(C(C)NC(C3CC3C(F)F)=O)CC2)cc(OC(F)F)nn1 Cc1c(C(=O)NC(C(=O)N(CC(N)=O)C)c2ccoc2)nnn1C Cc1cc(C(N2CCCN(C(c3cscc3C)=O)CC2C)=O)cc(C)c1F N1(C(c2nc(OCC)oc2)=O)CC(C(=O)NCC2CCCCN2C)C(C)(C)C1 c1(N(C)C)ccc(Cl)nc1NC(=O)NCCC1CCCC2CC12 C1(NC(=O)C=CC2CCCC2)CC2CN(Cc3cccc4[nH]ccc34)CC2C1 CCC(CC(=O)NCC(C)NC(=O)Cc1csc(-c2ncccn2)n1)C(C)(C)C C(=O)(C(C)(C)S(C)(=O)=O)N(C1CCCN(C(=O)CC(Cl)Cl)CC1)C c1(C(c2nnnn2Cc2ccoc2)NCC2CC(C)C2)cc(Br)cc(Cl)c1F CN1CCCC(c2cccc(NC(=O)C(F)(F)F)c2)C1.N12CCN(CC1)CCC2=O c1(C(=O)NCc2ccc(O)cc2F)cccc2c1CN(C(=O)CC1CCO1)CC2 C1(C(C)(C)NC(CCSCC)=O)CCN(C(C2CSCC(=O)N2)=O)CC1 CC1CC(NC(=O)Cc2cnoc2)CCN1C(c1ccnnc1O)=O Cc1cc(C(=O)NCCN(C(=O)CCn2nc(C)c(C)c2C)C)c2n[nH]cc2c1 c1(C(=O)NCC(C)NC(=O)C(O)Cc2ccccn2)ccn2ncccc12 C1(C(=O)NC(CNC(=O)CC2CCCC(C)C2)C(C)C)(CC)CCNC1=O c1(OCC)ccccc1C=CC(=O)NC(C1CCCCC1)CO C1(NC(CCSC)=O)CC2(NC(c3cn(C)c(C(=O)OC(C)(C)C)n3)=O)COC1C2 N1(C(CCCOCC)=O)CC(CNC(=O)CSc2cn[nH]c2)C2CC12 c1(C(=O)NCC2(C)N(C(CC=CC=C)=O)CC(OC)C2)cc2nccn2c(O)n1 C1(C(N2CCN(C(C3CC=CCO3)=O)C(CCO)C2)=O)CCc2ncsc2C1 C1(NC(C(N)=O)=O)CC2CCC(C1)N2C(C1COC(=O)N1)=O CCCCCC(O)C(=O)NC(CCC)C(O)C(=O)N1CC(S(N)(=O)=O)C1 N1(C(C(C2CCCN(C)C2)(C)C)=O)CC2(CC(NC(=O)C=CC3CCCO3)C2)C1 CCC(CC)C(C(=O)NC1(C(=O)NC)CCC1)N(CC)Cc1cc(C)ncn1 C12(C(N(C)Cc3ccc(CNC(C4CNC4)=O)cc3)=O)CCC(C1)C(C)(C)O2 CC1CN(C(=O)CCN2CCCC2)CCCN1C(=O)C(C)n1ccnn1 C1(C(=O)NCCCCc2cc(C)no2)COC2(C1)CN(C(C1CCNC1=O)=O)C2 C=CCCC(C)N(C(=O)CC(C)c1ccco1)C1CCCCC1 c1(OC)cc(Br)c(C)nc1NC(C1CC1C(=O)Nc1cc(C#N)cnc1C)=O CC1=NNC(=O)C1CC(N1CC=CC(NC(C2(C)CC2(F)F)=O)C1)=O N1(C(C2(OC)CC(C)(C)C2)=O)CCC=C(C(=O)N(C(C)CS(C)=O)C)C1 CC1CN(S(=O)(=O)c2cccnc2NC(CC2OCCO2)CO)CC2(CCC2)O1 C(C(=O)N1CCOC(C(=O)NOCC=CCl)CC1)(C(C)(C)C)N(C)C C=CCCCC(C(=O)N(C1CCN(C)C1)C)NC(c1cc(F)ccc1C)=O N(C(=NCCCF)NC(Cc1ccccc1)CO)CC(C)C(F)F N1(C(C2CCC(n3cc(CN(C)CC)nn3)C2)=O)CCc2scc(C)c2C1 c1(OC)nc(=NC2CN(C(c3cccnc3)=O)CCC2C(F)(F)F)nc(OC)[nH]1 C1(C(=O)NC(C(=O)Nc2cncc(C)c2)c2ccoc2)CC2CC(=O)C1O2 CC1=CCC(C(=O)NC2C3CN(C(C4CC(c5ccccc5)C4)=O)CC23)CC1 C(=O)(CCP(C)(C)=O)c1nsc(Sc2cn(CC)nc2)c1Br CC1(C)CC(c2nnnn2CC2CC2)(NCc2nnc(C(F)(F)F)s2)C(C)(C)O1 CC1(NC(=O)CCS(C)(=O)=O)CCCN(C(=O)CCn2cc[nH]c(=O)c2=O)C1 C1(C(N2CCCC(CCn3cc(C(C)(C)N(C)C)nn3)C2)=O)CCOCC1(C)C O=C1CCC(C(=O)NC2CC(CCNC(c3cnn(CC4CCOC4)c3)=O)C2)O1 C1(C(=O)NCCCC(CCC)NC(c2ccoc2CC)=O)CC2(CCCC2)CO1 c1(OC)ncnc(OC)c1NS(=O)(=O)CC1CNCCO1.C(C)(C)O Cc1cc(C)c(C)c(C(=O)NC2CC(C)(NC(c3cc(CO)on3)=O)C2)c1C Cc1nc(O)ccc1C(=O)NCC1CC(C(N2CCC(C)(CCO)CC2)=O)CO1 c1(N2CC=CC(OC)C2)nc(=NCc2nnc3n2CCCC3)[nH]c2c1CSC2 N1(C(C(CC)n2cncn2)=O)CCCC(NC(C2(C(F)F)CCOCC2)=O)C1 C=CCC(CC=C)C(=O)NC1CCOCC1NC(=O)C=CC(C)C c1(C(CNc2cncn2C)NC(CNC(C2C(COC)C2)=O)=O)ccccc1Cl CC1(F)CCCN(C(=O)CC2COCCO2)C1 N1(C(C2C(C)=CCS2)=O)C2CCCC1CN(C(c1ccc(F)cn1)=O)C2 C(CCCCC(=O)N1CCCC1C1CCN(C(=O)Cn2cc(CO)nn2)C1)OC c1(C(N(C2CCN(C(C3CC(C)CO3)=O)C2)CC#C)=O)ccc2[nH]cc(C#N)c2c1 c1(CC)nc(C)c(CC(N2CCCC2CNC(=O)COCCSC)=O)c(C)n1 N#Cc1ccc(C(=O)NC2C3CC4C2C4C3C(=O)NCC=CCl)cc1 N1(C(C2(C(C)(C)O)CC2)=O)CCOC(CCCNC(=O)CN2CC=CC2)C1 N1(C(CCC=CC(C)C)=O)CCC2CCCC12CNC(=O)CCn1cncn1 C1(NC(C(CCC)OC)=O)CC2(C1)CC(CNC(=O)C=Cc1ccnn1CC)C2 C1(NC(Cc2cc(C)sc2)=O)C(C)(C)C(NC(=O)CCC(C)CN(C)C)C1(C)C C(C(N=[N+]=[N-])C(=O)NCC(Cn1cc(-c2ccccc2Cl)nn1)OC)OCC N1(C(C(CN(CC)CC)F)=O)CC2(C1)SCCC2NC(c1cnc2sccn12)=O C#Cc1cc(C(=O)NC(C2CCCN2C(=O)Cn2ccnc2C)(C)C)ccc1Cl c1(OC)ccc2c(=NCc3cccc(N)c3)[nH]c(=NC3CC(F)(F)C3)[nH]c2c1 C1(C2CCN(C(c3coc4c3CCCC4)=O)CC2)(NC(C=COCC)=O)CC1 C1(C(N(CC(CC)C)C)=O)CCN(C(=O)Cc2cc[nH]n2)C(C)(C)C1 C(C)(CSC)(C(=O)NC1CCS(=O)(=O)C1)NC(CC1C(CC(C)(C)C)C1)=O C12(C(=O)NC3(Cc4ccc(Br)nc4)CC3)CCCC(C1)NC2 C(=O)(C(C)(C)CC(C)=O)N1CCN(C2CCN(C(CCC=C)=O)C2)CC1 C1(C(=O)NCC(N(C(c2c(CC)n(C)cc2)=O)C)C2CC2)OCC2COCCC12 c1(OC)ccnc(O)c1C(=O)NC1CC(C)(NC(C2CC=CC2)=O)C1 c1(NC(=O)CN2CCC3(CSC3)C2)cn2cc(Cl)ccc2n1 c1(OC)ccc2cc(CN(c3ccc4ncsc4c3)c3ncccc3Cl)oc2c1 C(=O)(CCCCCCN=[N+]=[N-])N1C2C(CNC(C3C(C)OCC3)=O)CC(CC2)C1 Cc1ccc(SCC(=O)NC(C)C(C2CCCCC2)NC(=O)CCF)cc1 N1(C(C(COC)OC)=O)CCN(CCCC(=O)OC(C)(C)C)CC1 C1(C)(CC)CC(C(=O)NCCN(C(=O)CCC(N)=O)CCOCCO)CCO1 N1(C(C2(C(=O)OCC)CC2)=O)CCN(C(=O)CCc2nc(O)n[nH]2)CC2(CC2)C1 C1(CN(C(C2(OC)CCSC2)=O)C)CCCN(C(c2ncccc2C)=O)C1 C1(CNC(c2snc(Cl)c2Cl)=O)CC2CCC(C1)N2C(c1cccc(O)n1)=O CCCCC(O)CC(=O)N1CCCC1CN(C)C(c1ccc(Br)nc1N)=O C(C(O)CCNC(c1ccnnc1)=O)NC(C(C)OCC(C)C)=O N1(C(c2cc3ncccc3s2)=O)CCC2(CC1)CC(O)CCO2 c1(C(=O)NC(C2CN(C(C3CCCC(OC)C3)=O)C2)C)cc2cccc(C)c2o1 N1(C(Cc2noc(C)c2C#N)=O)CCC2(CCCN(C(=O)C(F)OC(F)(F)F)C2)C1 C1(OC)CC(C(=O)NCCc2cscn2)N(C(c2ccc(C)cn2)=O)C1 C(CNC(=O)CCC(=O)c1cccs1)(C(C)(C)C)NC(C1CC(C)(CC)C1)=O N1(C(C2C=CCN(C(C(CC)CC)=O)C2)=O)CC2C(C1)C2(F)F CCCCC(CC)CCC(=O)N(C1CCCN(C(C2CCCN(C)C2=O)=O)C1)C C(=O)(CC1=CCCCC1)NC1C(NC(c2nccc(C(C)(C)C)c2)=O)CCC1 c1(C(=O)NC2(CCOC)CCN(C(=O)C=C(C)CCC)C2)c[nH]cc(Cl)c1=O C(=O)(CCC(C)(F)F)NCC(C1CCCCC1)NC(Cc1nc(C)sc1C)=O c1(CNC(=NCCC=C)NCC2(CO)CCCOC2)coc2c(C)cccc12 Cn1cc(-c2ccoc2C(=O)NCC(O)CNC(=O)Cc2ccsc2)cn1 CC(C)CCCCC(=O)N1CC=CC1(C)C(=O)NCCN1CCCCC1=O CCCC(F)C(=O)N(C1CCCCCC1)CCNC(C1CCCC1F)=O c1(OCC)nccc(C)c1C(=O)NCC(O)CNc1ccc(C(C)(C)C)cn1.CO c1(NC(=O)CCC=CBr)ccc2cc[nH]c2c1.C12CC(F)(C1)CNC2=O C=CCC(C)(C)C(=O)N1CCC(CN(C)C(c2occc(=O)c2OC)=O)C1 c1(OC)cc(OC)cc(NC(C2CN(Cc3nc(Br)cn3C)C2)=O)c1 c1(OC)ccccc1C(C)(C)C(=O)NC1CN(C(=O)CC2CCCC2C)CC1C CCC(C(=O)N1CC(O)(CCO)C1)N(C)C(c1coc(N(C)C)n1)=O C=CCC(CC(=O)N1CC2(CC(O)C2)C1)NC(c1ccc(C)nc1O)=O CC(C)CC(C)C(=O)N1CCC(C(=O)NCCCNC2CC2)O1 C#Cc1ccc(C(=O)NC2CCN(C(C3CC(S(N)(=O)=O)C3)=O)CC2O)nc1 Cc1cc(C(=O)NCCCN(C(=O)CC2CCCC(C)(C)O2)C)cc2c1CCC2 C1(Cc2ccc(OCC(=O)NC3(CC(C)(C)C)CC3)cc2)CCSC(C)(C)C1 C1(C(=O)NC2C(NC(CCc3ccn(C)n3)=O)C2)CC(c2cccc(F)c2)=NO1 c1(CNC(C2(OC)CN(c3ccnc(C)n3)C2)=O)c(Cl)sc2nnsc12 c1(NC)cc(C(=O)NC2CCC(C)N(C(c3cc(Cl)n(C)n3)=O)C2)cc(Cl)n1 N1(CC(C)C)CCC(C(N2CC(NC(C3CCCCC3O)=O)CC2CO)=O)CC1 N1(C(CC2C(OC)CC2)=O)CCC(N(C(c2ccc(C(C)C)s2)=O)C2CC2)CC1 CC1c2nccn2CCN1C(=O)C(CC(F)F)N(C(=O)C(c1cncnc1)C)C C12(NC(C3CN(C)C(=O)C3)=O)CCC(NC(C3CCCC(C)(C)O3)=O)(CC1)C2 c1(C(N2CC3CC3(C(=O)NCc3cccnc3Cl)C2)=O)cc2cc[nH]c2cc1Cl CCC(CC)(CC)C(=O)N1CCC(C)N(C(c2noc3c2CCCC3)=O)CC1 C1(N(C(=O)C(c2cc(Br)ccc2F)F)C)CC2CC1CC21OCCO1 N#CC1(C(N2CC3CC(C(=O)NOCC(F)(F)F)(C3)C2)=O)CC(F)(F)C1 Cc1ccc(C(C)C)c(C(=O)NCC(C)(C2CCC2)NC(=O)CC2CCC(C)O2)c1 Cc1ccc(C(F)(F)F)cc1OC(c1occc1NC(C(=O)NC1CC1)=O)=O Cc1cccc2sc(C(N3CC(NC(C4SCCCS4)=O)CC(C)C3)=O)c(Cl)c12 N1(C(c2ccc(OC)nn2)=O)CCC2(CCCN2C(c2ccoc2C(C)C)=O)C1 C1(CN(C)CC2CCC2)CCCCN1C(C1CCN(C)C1c1ccccc1)=O c1(OCCCC(=O)NCCC(C)N(C(C(C)(C)OC)=O)C)ccc(C)c(C)c1 C1(CNC(CCOCC)=O)C2CC1N(C(C1CC(OC)C1)=O)C2 c1(C(=O)NC(C(N2CCC(C(CC)CC)C2)=O)CC2CC2)c[nH]c(=N)c(C)c1 c1(N(CCNC(c2c(C)nc(C)[nH]2)=O)C2CC2)ncc(Cl)cc1[N+](=O)[O-] C1(C(=O)NC(CCNC(Cc2c(CC)con2)=O)C)CCC(C)(C)O1 C1(N(C)C)CN(C(=O)C(C)(Cl)Cl)CC1NC(=O)C(N1CCCC1)c1cccs1 C(C1c2ccccc2CCN1C(c1ccc(C(C)C)nc1)=O)NC(C=CSC)=O N1(C(C=Cc2cncc(C)c2)=O)CCC(C)N(C(C2CCCCS2)=O)CC1 N1(C(c2nn(CC)c(C)c2)=O)CCC(F)C(NCc2ccc(CC(C)C)cc2)C1 S(=O)(=O)(C1Cc2ccccc2C1)NC1CCC(N=[N+]=[N-])CC1 Cc1cc(C(=O)NC2CCC(CCC(=O)N3CC(CC(C)C)C3)C2)cnc1O N1(C(CC(C)c2ccco2)=O)CCC(C)(CNC(C2CC(n3ccnn3)C2)=O)C1 C(=O)(C#CC(C)(C)C)NCC(C)(CNC(=O)Cn1cnc(C(F)(F)F)n1)OC C1(C(=O)OCC(C2(C)CCCCC2)=O)CC12CCS(=O)(=O)CC2 C1(NC(CNC(c2ccc(C)s2)=O)=O)CC(NC(=O)C2CC2)C2CC12 C(=O)(CCC(F)(F)C(F)F)N(CC(CNC(c1occ(C)c1)=O)O)C CC1(CNC(=O)C(C2CCC2)NC(=O)C2=CCSC2)CC2(CCC2)C1 c1(C(=O)NCC2CN(C(c3c(CC)c(C)sc3)=O)C2)ccc2oc(O)nc2n1 C12(C(=O)NCC3N(C(CCC=CC)=O)CC(F)C3)CC(CO)(C1)OC21CCC1 C#CCCN=c1scc(-c2cccc(C=C)c2)n1CC1CCN(CC)C1 Cc1cc(I)c(C(N2CCCOC(C(=O)O)C2)=O)cc1C c1(OC)ccnc(Br)c1NC(c1cc(C(=O)Nc2cncc(C(F)(F)F)c2)no1)=O Cc1c(C(=O)NCC(C)N(C)C(c2ocnc2C2CC2)=O)c(C)n(C)c1Br C(=O)(CC(C)(C)C(=O)CO)NCCC1CCN(C(CC2(NC(C)=O)CC2)=O)C1 C1(C#N)(C(=O)NCC(CCOC)NC(=O)CCN2CCCCC2C)CCCCC1 c1(OC)c(C)[nH]ccc1=NCC1(C)CC2(C1)CC2(F)F C1(NC(C2CN(C)C2)=O)COC2(CCN(C(=O)Cc3cc(Br)ccc3Cl)CC2)C1 C#CC1CCCCN1C(CCc1ccccc1)C(=O)NC1(C)CC1 N1(C(c2c(C)ccc(OC)n2)C(=O)NC2CCC2)CC2CC(C)(C)C2C1 CC(C)(C(=O)NC1CN(C(c2ccncc2-n2cccn2)=O)CCC1CO)C(F)F N1(C(c2c(C)nc(O)[nH]2)=O)CCN(C(=O)C=CSc2nc[nH]n2)C(C)C1C Cc1ccc(CCC(=O)NC23CC(NC(=O)CC4CCC(=O)N4)(C2)C3)nc1 C1(C(=O)NC(c2ncccn2)CC)(CC)CCN(C(c2ccc(CO)o2)=O)C1 C1(C(=O)NCC2(SC)CC2)CCC(O)CN1C(c1ccnc(OC)n1)=O c1(C(C)(C)C)cccc2nc(NCC(=O)NC(N3CCCC3)=O)nn12 C1(CC(=O)NC(CCOC)(C)C)CC(NC(c2cnn(C)c2Cl)=O)C1(C)C C(CC(C)(C)C(=O)NCC1CN(C(=O)C(F)=C2CCC2)C(C)(C)C1)SC C1(CNC(c2c(COC)scc2)=O)CCN(C(=O)CN2CCC(C)C2)C12CCC2 Cc1ncc(C(=O)NCC2C=CCN2C(=O)CCCc2cccnc2)c(O)n1 c1(C(N2CCN(C(c3cc(Br)no3)=O)C3C2C3)=O)cc2c(o1)CCCC2 c1(C(N2C3(CCN(C(C(C)C)=O)C3)CCC2)=O)ccc2c(c1)CCCCC2=O N1(C(C(C)(C)Cl)=O)CCCCC(CNC(C2CN3CCC2CC3)=O)C1 C(=O)(CCCCCNC(c1nccnc1C)=O)NCc1n(CC)nnn1 C1(C(=O)NCC2CC(C)N(C(=O)CC(C)(C)C3CC3)C2)COCCN1C=O c1(N(c2ccccc2)CC=C)nccc(Br)c1C.N12CCC(C1)C2C(=O)NCC N1(C(CC2(OCC)CCC2)=O)CCN(C(C2C3C4CCC(C4)C23)=O)CC12CC2.OCC C(=O)(C(CC(F)F)NC(c1cc(C)sn1)=O)N1CCC(N(C)CC)C1 C12CCCCN1C(=O)CC2.N1(CC(=O)NCCOCCCCC)CCC(C)C1 CC(=O)CCCCC(=O)N1CCC(NC(=O)CC2CCC(=O)N2)C(CO)C1 N1(C(COCCOC)=O)CCC(O)(C(C)NC(=O)CCc2ccnc(Cl)c2)C1 C1(C(C)(C)C)CN(C(=O)C(C)(F)F)CC1NC(c1ncc(F)cn1)=O C1(CNC(c2c(SC)scc2)=O)CN(C(=O)CSC(F)(F)F)CC12CCC2 C(=O)(C1=C2CCCN=C2NN1)NCC1CN(C(C2(C)CN(C)C(=O)CC2)=O)C1 CCCC(CCCNC(c1ccc(C(F)(F)F)cc1)=O)NC(C1CCOC1)=O C1(C(N2C(CCNC(C=C(COC)C)=O)COCC2)=O)CCCC1C1CC1 c1(CNC(C(C)NC(C)=O)=O)ccc(CNC(=O)CC2CC23CC3)s1 C1(C(N(CC(=O)NCc2nn(C)cc2C)CCOC)=O)CCC2CC1CO2 C12(CCNC(C=CCCC)=O)CCC1CN(C(=O)C(F)(F)Sc1cnn(C)c1)C2 C(=O)(C#CC1(C)CCCO1)NCCCOCC(N1C(CC#C)CCC1)=O C1(C2CCOCC2)(NC(CCCCN(C(=O)CCn2ccnc2)C)=O)CC1 C(=O)(C(C)(CC)CC)N(C(CC)CC(=O)NCC1CCOCC1)C c1(CC(=O)NCC(CC)(CC)NC(c2nc(C)nn2C)=O)cccc(Cl)c1Cl c1(OCCN(c2nc(C)c(C)s2)C(CC)CO)ccc(F)cc1 Cn1c(C(=O)NC2CC3CCC(C2)N3c2nc(C(C)(C)C)ns2)ccc1[N+](=O)[O-] N1(C(C(C2CC2)OC)=O)CCCC1C1CCN(C(=O)Cc2n[nH]c(C)n2)C1 c1(SCc2c(CCCC)cccc2)cc2cccc(OC)c2o1 C1(C(=O)NCCC2N(C)CCC2)CCN(C(=O)CN(C2CCCC2)C)C1(C)C C12(C(N3CCCC(SCC(N4CC(OCC(C)C)C4)=O)C3)=O)CCC(C1)OC2C CCCCC(CC)CCC(=O)NC1(C)CC(NC(=O)CC2(O)CCC2)C1 CCCCCC(CC)C(=O)NC(C)(CNC(=O)Cc1c(F)cccc1C#N)CC N1(CCCNC(CNC(CCC)=O)=O)CCN(CC2CC(OC(C)C)C2)CC1 CC(C)(CCC(=O)N1CC(CNC(=O)C2=CCOC2)C2(CC2)C1)N1CCOCC1 N1(C(c2c(C)occ2)=O)CCCC(C)C1CNC(c1cn2ccsc2n1)=O CC1(C)C(C(N2CCCC(CCCCNC(c3ccnnc3O)=O)C2)=O)C1(F)F CCC1=C(C(=O)NCC(c2ccc(F)cc2)C(=O)OC)SCCO1 Cc1cnc(NCC(O)CNC(C2CCC3CC3CC2)=O)nc1S(C)(=O)=O c1(C(=O)NC(C(C)NC(c2ccc(C(C)=O)o2)=O)C)cc2ccccn2n1 C1(C(N2CC(NC(C(COC)C)=O)C(C)C2)=O)CCOC(C)(C)C1 C1(C(=O)NCCN(C(=O)CCC(=O)N)C2CC(F)(F)C2)COC2(CCC2)CO1.CC N1(C(CC2(C)CC(F)(F)C2)=O)CCN(C(=O)C(C2CCCCC2)F)C(CCO)C1 CC(CNC(c1c(F)ccc(F)c1F)=O)CN=c1[nH]nc(CO)s1 c1(OC)c(C(=O)NC(C)CCN(C(=O)CC2CCC(=O)N2)C)c(C)nn1C N1(C(C=CCOC)=O)CC(NC(=O)C(O)Cc2cnn(C)c2)C(F)C1 c1(OC)ccc(Cl)c(C(=O)NCC(C(C)C)NC(=O)C(C)(C)C#N)c1F C1(CC(=O)O)(CNC(C(=O)NCCOCC2CC2)C2CCOC2)CCCC1 c1(CSC)noc(CCC(=O)N(C(CNC(C2CC(C)(O)C2)=O)C2CCC2)C)n1 c1(C(=O)NC23CCN(C(c4n(C)cnc4)=O)CC2C3)ccc(S(C)(=O)=O)s1 C1(N(C(=O)CC(O)C2CC2)C)CCC(NC(c2ncsc2C(F)(F)F)=O)CC1 C12(NC(CCC=C=C)=O)CCOCC1CN(C(c1ccncc1Br)=O)C2 C(C(C(=O)N1CCN(C)C2(CC2)C1)C(C)(C)C)NC(C(C)NC(=O)C1CC1)=O CC(C(=O)NC1CCC(CNC(c2occc2C2CC2)=O)C1)C(C)S(C)(=O)=O C(=O)(C(C)(O)CC)NCCC(=C)CNC(c1coc(CC)c1)=O CC1(C)CCCC2(CCN2Cc2ncn3ccccc23)C1 Cc1ncc2n1CC(C(=O)NCC(C)NC(=O)CC1CCNC1=O)CC2 c1(C(N2CCN(C(CCCC)=O)C(C3CCCC3)C2)=O)cccc2cncn12 c1(C(=O)NCCC2CSCCN2C(C2CCCOCC2)=O)ccc(=O)n(O)c1 C(=O)(CCCC(=O)NC1(CCO)CN(C(C2CCN(C)C2=O)=O)C1)NC CCC(CC)CC(F)C(=O)NCC(C1CCN(C(=O)CCc2nccs2)CC1)F C1(C(=O)NCc2cc(C)cc(F)c2)CC2(CCN(C(=O)C(C)(C)C(F)(F)F)C2)C1 N1(C(CC)C)CCN(C(=O)CN(C(=O)Cc2ccnn2C)C(C)=O)CC1 C(=O)(CC(=O)N(CC(O)CN(C(=O)CC1CC1)C)C)NCC.C(C(C)(C)C)S c1(C(=O)OC)cnc2[nH]c(O)nc2c1.N12NN=NC1=NCC1CN(CCO1)CC2 C1(F)(CC(=O)OCC)CCN(C(=O)Nc2occ(C)c2C)C1 Cc1cc(O)c(C(=O)NCCCNC(C2CN(C)C(=O)N2)=O)cc1Br Fc1cccc(-c2cn(CCc3noc(Cc4cnn[nH]4)n3)nn2)c1F c1(CN2CCC(O)(C(=O)NCCNC(C)=O)CC2)ccc2n[nH]cc2c1 c1(C(=O)NC(CNC(C2CCC(CC)CC2)=O)CCOC)ncsc1S(N)(=O)=O c1(OC)c(F)ccc(Br)c1-n1cc(-c2ccc(C3CNC(=O)C3)cc2)nn1 C1(N(C(c2n(CCC)nc(C)c2)=O)CCO)CCCN(C(=O)C=CCO)C1 C1(NC(CC2CC(NC(C(C)OC)=O)C2)=O)CC(=O)N(C(C)C)C1 N1(C(c2n[nH]c(C)c2Br)=O)CCCC2CN(C(c3ccnnc3)=O)CCC12 C1(CNC(c2cc(C)ncc2)=O)COC(C)(C)CN1C(c1cccnc1CO)=O c1(C(=O)Nc2c(CC(OCC)OCC)cccn2)coc2c1CSC2 C(=O)(CCCC(C)=O)NCC1CC(NC(C(CC)Oc2ccccc2F)=O)C1 c1(C(=O)NC2(CC=C)CCN(C(c3cccn3C)=O)C2)cccc(C)c1N C(=O)(C1CCCc2ccnn21)NC(C(C)NC(C1(CCC)CC1)=O)CO C(=O)(C(C)(C)CSC)N(CC(C)NC(c1cn(CCOCC)nn1)=O)CC C(=O)(C(C)(C)C(=O)N1CCN(C(c2ccc(C(F)(F)F)o2)=O)C(C)C1)NC c1(C(=O)OC)csc(C(c2nnnn2-c2ccccc2)NC(C)(C)C)c1 N1(Cc2c(C)cncc2)CC2(CCC2)CCC1C(C)C c1(C(=O)NCC(CC(C)C)NC(c2ccnc(C#N)c2)=O)cccc(F)c1F c1(CC(=O)NCCCC)csc(=NCc2ccc(Cl)nc2)[nH]1 C1(C(N(C)Cc2coc(C(F)(F)F)c2)=O)CN(C(=O)C(F)OC(F)(F)F)CCO1 CCC(C(=O)NCCC1(O)CCN(C(c2ccc(C)c(O)n2)=O)C1)C(C)C S(=O)(=O)(c1ccc(NC(=O)Nc2cccnc2)cc1)NC1C(C)CCCC1 N1(C(CC(CC=C)NC(C2CC(=C3CC3)C2)=O)=O)CC2(C1)NC(=O)NC2=O N1(C(c2nnc(C(CO)(F)F)o2)=O)Cc2ccccc2C1 c1(CC(N2CCC(NC(=O)CN(C3CC3)C(=O)C3CC3)C2)=O)ccnc(F)c1F c1(C(=O)NCC2N(C(c3c(CC)oc(C)c3)=O)CC2)nccc2cc[nH]c12 c1(CC(=O)NCC(N(C(C(c2cnn(C)c2)C)=O)C)C2CC2)ncn2c1CCC2 C(=O)(C(CC(F)F)CCO)NCC1(OCC)CN(C(C2CCC3(CC2)CC3)=O)C1 O=S1(=O)CCC(c2nc(-c3ccc(Cl)cn3)nn2Cc2ccccc2OC(F)F)N1 C1(C(=O)NCC(CNC(C(CC(C)C)N(C)C)=O)C)CC2C=CC1C21CC1 c1(OC)ccc(Br)c(C(=O)NCC(C)CN(C)C(c2ccc(F)cn2)=O)c1 c1(C(=O)NC2CC(CNC(C(C3CCC(=O)N3)C)=O)C2)cc2ccc(O)nc2s1 c1(CC)ccc(CC(=O)NC2CCCC2NC(=O)CC2(C)CCCO2)cc1 c1(OC(CC)C)ccc2[nH]ccc2c1C(C)NC(c1nn[nH]n1)C c1(NC(CC2(C)CN(C(c3cccc(Cl)c3Br)=O)C2)=O)ccccc1C(N)=S N1(C(CC2C(C)(C)C(O)C2)=O)CCCC(C(=O)NCC2CC(N3CCCC3)C2)CC1 N1(C(C2CC2C(F)(F)F)=O)CCC2C1CCN2C(C12CC(CCC(F)(F)F)(C1)C2)=O C(C(O)C(=O)NC(CC1CCCC1)C(=O)NCC1C2CCCC12)=CC N1(C(=O)CCN2CCC2)CCCC(C2CCN(c3ncnc4cccnc34)C2)C1 Cc1c(NCCN2CC=CCC2)nc[nH]c1=NCC1CC2(CCCCC2)CO1 C1(N(C(C(=O)NC)C(CC(C)C)OC)C)(OC)CCCC(C)(C)C1 Nc1sc2c(c1C(=O)NCCC1CCN(C(C3(Cl)CC3(F)F)=O)C1)CCC2 c1(C(C(=O)NC(CO)C(=O)OC)NCc2c(COC)noc2)c(C)cccc1Br CC1CN(C(c2sccc2CO)=O)CC(CCNC(C2CC(=O)C2)=O)O1 CCC(C)CC(=O)C(=O)NC1CCCC1CC(=O)NC1(CCCF)CC1 c1(C(N2CC(C)N(C(C3CC4CCC3CC4)=O)CC2)=O)cn2ccccc2n1 C1(C(=O)NCCNC(=O)NC)CCN(C(C2CCCOCC2)=O)C1C C(CC1=CCN(C(=O)CC2CCC3(CCC3)CO2)CC1)NC(c1cc(O)cs1)=O c1(C(=O)NC(C)(C)CCNC(=O)CC2(O)CCOC2)c(O)nnc2c1CCC2 c1(SC)cccc(C(=O)NC2CCN(C(=O)CCc3cnn(C)n3)CC2C)c1Cl N1(C(c2c(OCCC)oc(C)n2)=O)CCCCCC(NC2CC(C)CCO2)C1 c1(C(C)=O)ccc(OC)c(NC(c2n[nH]cc2NC(=O)C2CC2)=O)c1 N1(C(c2[nH]c3cc(C)oc3c2)=O)CCCC2C1CCCN2C(=O)CC1CCC1 C(=O)(C1=CCCCC1C)NCC1(NC(c2cc(C)cc(O)n2)=O)CCCC1 c1(CC(=O)NCCC2CCCN(C(C(C)c3cccs3)=O)C2)c(F)cccc1Cl C1(N(C(C(C=C=C)C)=O)Cc2ccccc2)CN(Cc2cc(Cl)n(C)n2)CC1(C)C c1(C(=O)OC)ccc2sc(NC3C4CCC3N(C(=O)CC3(CO)CC3)C4)nc2c1 N1(C(C=CCC(C)(C)NC(C2(C)CCCCO2)=O)=O)CC(O)(C2CCC2)C1 c1(N2CC(CC(C)NC(=O)C3=CC4CCCC34)C2)ncnc2c1c(Br)nn2C Cc1nc(C)c(C(N2CC(CNC(c3cc[nH]c3C3CCCC3)=O)CC2C)=O)o1 c1(C(C)=O)c(Cl)nc[nH]c1=NCC1(NC(c2nccnc2C)=O)CCOCC1 Cc1ccc(C)c(SCC(N2CCSCC2CCNC(=O)Cn2cccn2)=O)c1 C1(NCc2ccc(C(=O)O)o2)C2CC1CN(C(c1ccc(F)c(O)c1)=O)C2 c1(CNC(C(C)OCCCC)=O)cccc(C(=O)NCCC(C)c2cn[nH]c2)n1 C1(CNC(C(C)OC2CCCC2)=O)CCCC1NC(C1CCN1C1CCCC1)=O N1(CC(N)CNC(=O)NC(C2(C)CCC=CO2)C)C(=O)c2ccccc2C1=O Cn1cc(Br)c(C(=O)NCC(C)(CO)NC(=O)CCCC2CCC2)cc1=O C1(CC)CCN(C(=O)C(=O)C2CCCC2)C(C(=O)Nc2ccc(F)c(CO)c2)C1 c1(C(=O)NCCCNC(=O)CCc2ccco2)cn(C2CCC2)nn1 N1(C(CCC2(C)CC2)=O)CCC(C2CC2)C1C(=O)NCC1(O)CC=CC1 c1(N(C(C2CC2(C)C2CCC2)=O)CC)cn(CC(C)(C)C)nn1 C1(C(C)NC(c2cn(CCC)nc2)=O)CCCCN1C(C1CN(C2COC2)C1)=O C12(CNC(c3cnc[nH]3)=O)CCC(CC1)N2C(c1csc(-c2ccoc2)n1)=O C(c1cnc[nH]1)=CC(=O)NCC(N(C)C(c1ocnc1C1CCC1)=O)C1CC1 N1(C(C2CC(C)(C)OC2(C)C)=O)CC2CCN(C(=O)CN=S(C)(C)=O)CC2C1 c1(-c2onc(NC(C(CCCCC)O)=O)n2)noc2cc(OC)ccc12 c1(NC2C3CN(Cc4nn(C)c(CC)c4Cl)CC32)c[n+]([O-])ccc1[N+](=O)[O-] N1(C(CCSCC)=O)CCC2CN(C(=O)Cn3ccnc3C(C)C)CC2C1 Cc1nc2nccc(C(N3CCC(CC4CC4)C3)=O)n2n1.C12(CC1)C(=O)NC2=O C1(NC(CNC(CCN(C)CCO)=O)C(=O)Nc2ccc(F)cc2)CCC(F)CC1 c1(CC(N2CCC(CN(C)C(C3CCCOC3)=O)C2)=O)cnc2ncccn12 C(C(COC)C(=O)NCc1nnn(C)c1C(=O)N(Cc1cncn1C)CC)OC C(=O)(CS(=O)(=O)CC(F)(F)F)N1CCN(C(C2CCCC(=O)N2)=O)C(CO)C1 Cc1cnc(C#N)nc1N1C2CCC1C(CN(C(=O)C=CCN1CCCC1)CC)C2 CCC(CC)C(=O)N1CC(O)(C(C)NC(=O)C(C)NC(=O)Nc2ccccc2)C1 Cc1c(N)ccc(C(=O)NCCCOCCNC(C2CC23CC(C)(C)C3)=O)c1F C=Cc1cncc(C(=O)NCC2N(C(=O)CN(C)C(C)C)CCC2(C)C)c1 c1(C(N2CC(NC(c3cc(COC)no3)=O)C(OC)C2)=O)cnc(C)c(C)c1 C(=O)(CCCC(C(=O)Nc1ccc2c(c1)CCC2)N1CC(C)CC(C)(C)C1)OC C(CC(F)F)(C(=O)N1CCC(NC(N)=O)C1)N(C)C(C1CC=CC1)=O S(=O)(=O)(c1ccc2[nH]c(=NCC3CCCSC3)sc2c1)N1CCC(OCC)C1 C1(C(=O)NCc2ccc(C(=O)NC3C(OCC)CCC3)cn2)CC(=O)OC1(C)C C(=O)(C1=C(Cl)CCOC1)N1C(C(N(CC)Cc2ccoc2)=O)CN(C)CC1 c1(N(C)C)cc(C(=O)NC(c2ccccc2F)Cc2ccccc2Cl)cc(Cl)n1 c1(NC(N2CCC(OC(C)=O)CC2)=O)c(C)oc2cc(O)ccc12 N1(c2nc(C)nc(Cl)c2)CC(NC(=O)C(C)S(N)(=O)=O)CC2(CCC2)C1 c1(OC)ccc(CN(C(C)C)CC2COC(=O)O2)c(C)c1 C(=O)(C#CC(=O)N(C)C)N(C)CC1CCN(C(C2(CCOC)CC2)=O)C1 CCC(C)(COC)C(=O)NCC(C)NC(=O)COCc1cccc(C)c1 c1(CN(C)C(C2CNCCN2C)=O)ncc2ccccn12.CSC N1(C(C(=O)NCC2(C)CC(F)(F)C2(F)F)=O)CC2CCC1C(CO)C2 Cc1ccc(C(CCO)NCC(=O)Nc2ccc(CNC(N)=O)cc2)cc1 c1(C(=O)NC(C(=O)NCC(=C)C(F)(F)F)(C)CSC)ccc(F)c(F)c1 C1(NC(CCOCCN(C)C)=O)C=CC(CNC(c2coc(Cl)c2)=O)C1 N1(C(CC2CCCC(=O)C2)=O)CCC2(C=C(C(=O)NCCCCO)C2)C1 Cc1nc(N2CCC(F)(F)C(C(=O)Nc3ccc(CO)cc3)C2)c2sccc2n1 C1(N(C(CN(S(C)(=O)=O)C)=O)C)CCCC(N(C(=O)COCC(C)(C)C)C)C1 N1(C(C(C)(C)OCCC)=O)CC2C(CNC(=O)C(C)C(C)C)C2C1 N1(c2nc(N3CCC(C)(OC)CC3)c3c(n2)CSC3)CC2(CCC2)OCC1C C1(C(=O)NCC(CC)(C)C)N(C(=O)CSc2ccccn2)CCCC1(C)C c1(OC)nc(=NC2CCCCC2C(=O)NC(c2ccc(F)cc2)C)nc(OC)[nH]1 N1(C(CC(CCC)(C)O)=O)CC2CCCN(C(=O)C=Cc3cnc(C)s3)C2C1 C1(NC(C=C(CC)C)=O)C2CC(O)C1N(C(C13CC=CCN1CCC3)=O)C2 C1(CNC(CC(COC)C)=O)CCN(C(c2ccon2)=O)C12CCC2 CC(C)(C)CC(C)(C)C(=O)NCC1COCCN1C(c1cnc2c[nH]nc2c1)=O C1(C(N(CCC(=O)Nc2ccnn2C2CC2)CC)=O)C2CCC(C2)C1(C)C S(=O)(=O)(c1c(F)cccc1F)NC(=O)COc1cccnc1 C1(NC(C2(COC)CC=CCC2)=O)CC(F)CN(C(=O)C=C2CCOCC2)C1 C1(C(=O)NC(COC)CNC(c2ccc(C)cn2)=O)CCC2(CCCO2)CC1 C1(NC(C2C(=C)CC2)=O)(CO)CCN(C(c2cc(SC)n(C)n2)=O)C1 C(=O)(CCC(C)(F)F)NCC1N(C(c2ccc(SC)o2)=O)CC(F)C1 C(=O)(C1=CCOCC1)NC1CN(c2cccc(NC(COCCSC)=O)c2)C1=O c1(CC)cc(OC)ccc1C(N1CCCCC1CCNC(C1CC1C)=O)=O CC1CN(C(=O)CCC2CCCO2)CCN1C(=O)COCCC1CCCCCC1 S(=O)(=O)(c1ccc(Cl)cc1)N1C(C(N(CC(C)C)CC)=O)CCCC1 CC1C(NC(c2cncc(F)n2)=O)CCCN1C(c1cc(Cl)nc(=N)[nH]1)=O c1(C(=O)NC(C2CCCN2C(=O)CC2CCC(=O)NC2)C)cncc(F)n1 C1(CC)CN(C(C2C(C)OC(C)C2C)=O)CCC1N=c1[nH]c2ccc(Cl)cc2s1 N1(Cc2ncn(C)n2)CCC(F)(C(=O)NC(c2cccnc2)C2CC2)CC1 c1(CN(C(CN(C(c2cc(OC)cs2)=O)CC)=O)C)nnc(C)n1C c1(C(=O)NC(CNC(C(C)(C)c2cscc2Cl)=O)CO)ccn2cccc2c1 N1(C(c2ncn(C(C)(C)C)n2)=O)CC2CCCC(C1)N2CCOCCC1CC1 c1(C(=O)NC2CCC(NC(C3(COC)CC=CC3)=O)CC2)cc(C)c(=O)n(C)c1 C1(O)(CC(=O)NC(C2CCN(C(C3CC34CCCC4)=O)CC2)CCC)CCCOC1 CC1CN(C(=O)CCN2CCNC(=O)C2)CCC1CNC(=O)CCSC(F)(F)F C12(NC(C(=O)NCC)=O)CCCN(c3ncnc(Cl)c3OC)CC1C2 C(=O)(CCC(=O)Nc1cc(C)ccn1)N(CC(=O)NC1CCCCC1)CC C(=O)(CCCN(C)N=O)N1CCC(O)(C(=O)NC(C2COC(C(=O)O)C2)C)CC1 C(=O)(CS(=O)(=O)C12CC(C1)C2)NCCC1N(C(COCC(=C)C)=O)CCOC1 C(C(O)C(=O)NC(CC(=O)OC(C)(C)C)C1CC1)=CC C12(C(N3CC(c4nncs4)C3)=O)CCCN(CC1)C2.C=C1CC2(C1)C(=O)NC2.NC C(=O)(C1=CCC(F)(F)CC1)N(C1CCCN(C(c2cc(N)ccc2F)=O)C1)CC C1(C(=O)NC(C)CN(C)C(c2cc(Cl)cc(F)c2N)=O)COc2ccccc2C1 C(CNC(=O)C(=O)NCCC1OC(C)CC1C)(C(C)(C)C)OC C(=O)(CCCCCN(C)C(C1CCS1(=O)=O)=O)NC(c1cnns1)C C1(C(=O)NC2COCC2NC(c2ccsc2OC)=O)(OC)CCCCC1 C1(CNC(C=C(CC)CC)=O)CN(C(c2coc(C(=O)OC)c2)=O)CC12CCC2 C1(OC)CN(C(=O)CC2CN(C(c3nc(C)oc3C)=O)CC2C)CC1NC(C)=O O=C(NN1CCCC1CCO)C1CCCN(c2nnnn2CC2CCC3CC23)C1 c1(OC)ccc(Cl)c(CC(=O)NC(CNC(=O)C(F)CC2CC2)C2CCC2)c1 c1(C(=O)NCC2C(NC(c3n(C)ncc3)=O)C2)c(F)ccc2ccoc12 C(C(C)(C)C(=O)N(C)CC1(C)CCCC1NC(c1ccoc1)=O)OCC c1(C(N2C(C(=O)OC(COC(C)=O)CO)CC(O)C2)=O)cc(C)nc2oncc12 c1(CC)cc(C(=O)NCC2CC2NC(C2CCCNS2(=O)=O)=O)ccc1F C=CCC(CC(=O)NCCCOCC(C)C)NC(=O)CC1C=NN(C)C1=O N1(C(c2cc(C)oc2C)=O)CCC(F)(F)C(CNC(=O)CC2CCC(O)C2)C1 CC1(C)CCC(CC(=O)NCC2CN(C(=O)C(N3CCCC3)C3CC3)C2)C1 C1(OC)(CNC(=O)CC2CC3(CCC3)C2)CCN(C(=O)CCSC2CCCC2)C1 c1(C(=O)NCCCC2N(C(CCOC)=O)CCC2)ccc(-c2ncccn2)cc1 N1(C(C2C3(CCN(C(=O)CCc4ccncn4)C3)C2)=O)CC2CCC1C(O)C2O N1(C(C2C(NC(C3C(C(=O)OC)C=C3)=O)CC2)=O)CCCC(C)C1CO C(=O)(C1=CC2(CCOC2)C1)NC1CC(CNC(CCC(C)(C)NC(C)=O)=O)C1 C(=O)(C1=NNC(=O)C1)N1CCCC(C(=O)NCc2nnn(C)n2)C1 C(=O)(C1=CCCCC1)N(CC(C)CNC(=O)CC1(C)CC1(F)Cl)C C(N=c1[nH]c(=NCc2cc[nH]n2)c2cc(Cl)ccc2[nH]1)C1(C)CCOC1 C(CC(N=c1cc(Cl)c(O)n[nH]1)C(C)C)NC(C1(CCCC)CCCC1)=O C1(NC(C=C(C)Cl)=O)Cc2ccccc2C1NC(c1c(C)cc(Cl)cc1N)=O c1(C(N2CC(O)(CCNC(C3CCCCC3F)=O)C2)=O)ccc(F)cc1F N1(C(C(C2CC2)NC(c2n(C)cc(Cl)c2)=O)=O)CCC2(CNC(=O)O2)C1 c1(OCC)ccc(F)c(C2CCC(C(N3CCC(C4CCCO4)C3(C)C)=O)C2)c1 c1(C(=O)NC2CC3CN(C(C4(C#C)CCCC4)=O)C2C3)nccc2ncncc12 N1(C(C(CC#C)O)=O)CCC(C=C)(C(=O)NCc2ccnc(OC)c2)C1 N1(C(CC(=O)NC)=O)CCC(O)(CNC(C2C(C(C)C)C2[N+](=O)[O-])=O)C1 C1(C)(CNC(CN(C(=O)Cc2ccon2)CCC)=O)CCOC1C N1(C(C(C)(C)NS(C)(=O)=O)=O)CCC(C2OCCC2NC(C2(F)CCCC2)=O)CC1 C1(C(=O)NCCCCO)CCCCCCN1C(=O)CCN1CCOCC1 c1(C(=O)NC2CCC(N(C(=O)CCCN=[N+]=[N-])C)C2)cc(N)c(F)cc1F N1(C(C(CC=C)C)=O)CCCC(NC(=O)C(C)(C)C)C1C(F)(F)F Cc1nc2cccc(C(=O)NCC3CCC(NC(=O)Cc4cccnc4)C3)c2[nH]1 C1(CC(=O)OC)CC(C)(C)CN1Cc1c(CNC(CS(=O)(=O)NCC)=O)noc1 C(C)(C)(CCC(=O)NCC(CC(=O)N1CCCCC1CC(C)C)C1CCC1)OC C=CC1(CC(=O)NCC2CCCN(C(C3CCCCCCC3)=O)C2)CCOCC1 N1(C(C(C)n2cnnn2)=O)CCCC(N(C(=O)Cn2ccc(C(F)(F)F)n2)C)C1 C1(C(N2C(CN(C(c3ccc(CC)nc3)=O)C)COCC2)=O)CCCCC(=O)C1 Ic1cnc(C(c2nnnn2Cc2ccccc2)NCCc2sccc2Cl)s1 c1(C(C(N2CCCC2CCCNC(C2CC2[N+](=O)[O-])=O)=O)OC)ccc(Cl)cc1 C1(NC(=O)O)CC2CC1N(C(=O)C(C)(O)C1CN(CC)C1)C2.c12cc([nH]n1)C(=O)N2.OC C1(NC(c2c(OC)n(C)nc2)=O)CC(O)CN(C(=O)Cn2nnc(=O)[nH]2)C1 CC1OCCC1CN(C(=O)CCN(CCCNC(=O)Cn1cccc1)C(C)C)C c1(OC)nc(Cl)cc(=NC2CCN(CC)CCC2(F)F)[nH]1.c1(CC(=O)O)cnn(C)c1 CCC(C)CCN=c1[nH]c2c(c(=NCc3ccc(Cl)c(Cl)c3)[nH]1)COC2 C(=O)(C(C)(C)C(C)(F)F)NC(C)C(CCc1ccccc1)NC(c1cc[nH]n1)=O n1(CC(N2CCC(C(C)NC(CC(C)F)=O)CC2)=O)ncc2ccccc2c1=O N#Cc1ncc(C=CC(=O)NCCc2noc(-c3ccccc3)n2)cn1 C12(C(N3C(C)(C(=O)NCC4(CO)CC4)CCC3)=O)C(=O)C3CC1C2C3 c1(C(=O)NCc2cccc(O)n2)cnc2ccc(-c3cnn(CCO)c3)cn12 C=C(C(=O)NCCC(C)N(C(=O)CCc1ccc[nH]1)C)C(F)(F)F c1(NC2(C(=O)Nc3cccc(C(CC)(C)C)n3)CC2)ccc2c(c1)OCCO2 C1CCCCCC(=O)N1.C1(F)(CSC)CCN(C(=O)CCCc2ncco2)C1 C1(NC(c2c(C(C)C)cccc2)=O)COCCN(C(=O)C=CC=C(Cl)Cl)C1 C=CCCC(C(=O)N1CCC1(C)C(C)C)NC(=O)C(C)C(=O)OC(C)(C)C CC1(C)CCCC(C)(NC(C2CCCN2C(C2CCC(C3CC3)C2)=O)=O)C1 C1(n2cc(CC(C)O)nn2)CCC(C)(C)N(C(=O)C(C)(C)CCF)C1 N1(C(C(=O)NC(C)C)=O)CCN(C(C2CCSCC2)=O)CC1C N1(C(CCc2ccc(C)nc2C)=O)CCC(O)(C2(NC(C3CC3F)=O)CC2)CC1 C1(C(=O)OCC)(Cc2ccccc2N(C)C)CCCN(CC2CCCO2)C1 Cc1ccc(CN2CCOCC2c2nnc(-c3cccnc3)o2)c(C)c1C C1(C(N(CC(=O)NCC(C)CCCO)C2CCC2)=O)C2CCCCCC12 C(=O)(CC(C)(C)N(C(=O)Cc1ncccc1F)C)NC(C)CCCC N1(C(CC(=C=C)C)=O)CCCC(C)(CNC(C2OCCCO2)=O)C1 c1(C(N2CC(O)(CNC(c3ccc(Cl)cn3)=O)C2)=O)nnc(O)cc1O c1(CNC(CN(C)Cc2c(COC)cc(OC)cc2)=O)ccc2nc[nH]c2c1 CC12COCC1CN(C(=O)C(CC1CC1)NC(=O)CCC(=O)C1CC1)C2 C1(NC(CC2CC(C)C2)=O)CCCC1CNC(c1ccccn1)=O c1(OC)ccc(C2(C(=O)NC3CCCC(C4CCCCC4)C3)CCC2)cc1O N1(C(c2c(OC)nsc2)=O)CCC(NC(=O)CC2CC(N(C)C)C2)C(C)(C)C1 c1(OC)cccc(C)c1C(=O)NCC1CCCN1C(=O)C(O)CC(C)C c1(CCNCCN(CC(C)C)C)ccc(S(=O)(=O)N(CCC(N)=O)C)cc1C#N Cc1ccnn1C(C)C(=O)NCCCCCN(C)C(c1coc(Cl)c1)=O C(N=c1nc(N(CC(CCO)OC)C)c2c([nH]1)CSC2)c1cnn(CC)c1C C1(C(=O)NCCCSC)CC(C)CN(C(C2CC(CF)C2)=O)C1 C(=O)(C(C)C(O)CC(C)C)N(C(CN(C(CCC#C)=O)C)C)C C(=O)(CS(=O)(=O)C(C)(C)C)N1CC(C(C)NC(CC(C=C)C)=O)C1 c1(C(C)NC(C2N(C(c3ccc(OC)s3)=O)CCC2)=O)ccc(Br)c(F)c1 c1(C(=O)NC2C(n3cc(COCCCC)nn3)COC2)nc(C)[nH]c1[N+](=O)[O-] CCC(C(=O)NCCCC(c1ccccc1)NC(C1CCCOC1)=O)n1cccn1 C#Cc1ccccc1CCN(CCOc1ccccc1)C(C1(F)CNC1)=O C1(CN(C(c2cccc(COC)n2)=O)C)CCCN(C(=O)C2=CCCSC2)CC1 c1(CCNC(C=C(C)C(C)C)=O)cc(C(=O)N(C)C(c2ccco2)C)no1 C(=O)(CCC(=O)NCC(C1CCCN(C(=O)CC(F)F)C1)(C)O)NCCC c1(C(C(=O)NCC2CC2)N(C2CCN(C3CCCC3)CC2)CC)cccnc1C c1(OC)ccc(CN=C(NCc2ccsn2)NC(C)C2CC2)cc1F c1(SC)ccnc(C(=O)NCCC(C)NC(c2cocc2C)=O)n1 CCC(CC)(CC)C(=O)N(CCC(=O)Nc1c(C)cccc1C)CCO CC(CC(=O)N(CC(O)CN(C)C)C)N(C)C.C12(CCCC1)C(=O)N2 c1(SC(C(=O)NC(CC)CNC(=O)C(=O)NCC)C)cccc(C)c1 C1(CC(N2CCC(NC(C3C(CC)CCC3)=O)C2C)=O)CC2(CCC2)CO1 C(=O)(C(C)(F)C(C)(C)F)N1CCC(CC(C)NC(c2cnc(C(C)O)s2)=O)CC1 c1(CNC(=O)NCC2(C)C(C)(C)C2)nc(C(F)(F)F)n2ccncc12 c1(C(=O)NCC(C2CC2)NC(C2(C(=O)OC)CC2C)=O)cc(SC)ccc1N c1(C(N(C2CN(C(C3N(C(C)=O)CC(O)C3)=O)C2)C)=O)ccc2c(c1)N(C)CC2 c1(CC(=O)NC(CCC)CNC(=O)CC(=O)N(C)C)cccc(NC(C)=O)c1 c1(CC)nc(C)sc1C(N1CC=CC(C(=O)N(CCCOC)C)C1)=O C1(C(N2CCN(C(=O)C(Cl)Cl)CC2)=O)CCN(Cc2ccnnc2O)CC12CC2 C(c1cccn1C)=CC(=O)NCC(C)(C)NC(C(c1cnn(C)c1)C)=O C1(NC(=O)Nc2ccc(SC)cc2)CC2CCC1CN2C(=O)COC(C)(C)CC N12CCOC(C1)C(=O)O2.C1(CC(C2CCOC2)NC(C=CC)=O)CCCCC1 C1(CN)CCCC(NC(C2(c3cccnc3)CCCC2)=O)C1 N(C(=NCc1cccc(OC(F)F)c1)NCC(C)(C)C)C1C(C(F)F)C1 N1(C(c2csc(C)c2C)=O)CCN(C(C2CCC(C)O2)=O)CC1CC(C)(C)C C(=O)(CC(C)CN(C)C)NC(C)CCCN(C(c1ccccc1)=O)C1CC1 C1(CCC(=O)NCc2c(CC)nco2)CCCCN(C(c2coc3c2COC3)=O)C1 C1(CC)CC(C(N2CCCC2(CNC(=O)C=Cc2cscn2)COC)=O)CCO1 C1(Nc2cccc(C(=O)OCC)c2)CCN(C(=O)COc2cnccn2)CC1O c1(C(CNC(c2cc(Cl)cnn2)=O)=O)cccc([N+](=O)[O-])c1 Cc1cc(NC(N)=O)ccc1NC(=O)C(C)C(C)(C)O.C1(C)(C)C(=O)N1 c1(CC)cccc(C(N2CC(NC(=O)CNC(=O)C(F)(F)F)CC2C)=O)c1C c1(C(=O)NCC2C(CNC(Cc3cc(C)on3)=O)C2)ncc([N+](=O)[O-])n1C C1(C(=O)NCC(=O)NCC(C)C)CCCCN1C(=O)CC1CCCC1C N1(C(C2(CCC)CC2)=O)CCC2CCN(C(c3ccc(Br)o3)=O)C2C1 c1(C(=O)NCCC2(NC(C=C(C)Cl)=O)CC2)ccsc1CN(C)C c1(C(=O)Nc2ncc(C(C)=O)nc2)cc2ccc(-c3ccc(I)cc3)cn2n1 N12CCOC(C1)CCNC(=O)Cc1nc(cs1)CC2=O.C(C)(C)SC C1(OC)CC2CCCC2N1S(=O)(=O)NC1CCN(C(=O)NC2CCCC2)CC1 N1(C(c2c(N)ncc(C)c2)=O)CC2(CCC(NC(c3sc(C)nc3C)=O)CC2)C1 C1(C(=O)NCCCC2OCCC2(F)F)CC12CCSCC2 C1(NC(c2n(C(C)C)ccc2)=O)CN(C(C2CCCC(=O)CC2)=O)CC1C1CC1 Cc1ncccc1CCCn1cc(C(N2CCC(c3nc(=N)[nH][nH]3)C2)(C)C)nn1 N1(CCCCNC(c2c(C)cns2)=O)CCCN(C(C2C(C#N)C2(C)C)=O)CC1 C1(CNC(Cc2ccc(C)nc2)=O)CN(C)CCC1O.C1=CC(=O)NC1(C)C C(=O)(CCN=c1[nH]c2ccccc2s1)NC(CNC(C1CC(OC)C1)=O)(C)CO c1(OC)ccc(C(=O)NCC(O)CN(C(=O)CCc2cccnc2C)C)cc1Cl C(=O)(C(C1CC1)N(CC)CC1CC1)NC(COCC)C c1(C(N2CC(NC(C3CCCN3CC(F)F)=O)C(F)C2)=O)cc2c(o1)CCCC2 c1(C(N2CC3CC(NC(CC(C=C)CC)=O)C3C2)=O)c(F)ccc(F)c1Cl c1(NC(CCN(C(CC)=O)C)C)cc(C(C)=O)c([N+](=O)[O-])cn1 C(=O)(CC1=CCOCC1)NCC1C(NC(CCc2cccc(OCC#N)c2)=O)C1 N1(C(CCN(C)C(c2cnn(C)c2)=O)=O)CCN(C(=O)CC(=O)OC)C(CO)C1 C12(NC(c3ccc(COC)[nH]3)=O)CC1CN(C(=O)CCC1CC(F)(F)C1)C2 CCC(CNC(Cc1ccc(Cl)cc1)CO)(CCC(=O)O)C(=O)O Cc1ccc(C(=O)NCC2CC(CNC(C3CCC(C)(C)C3)=O)C2)n1C CCC(F)(C(=O)NC1CC2CCC(C1)O2)C(=O)O CC(C)CC(C)CC(=O)N(C(C)C(N1CCC(OC(C)=O)C1)=O)CCO c1(C(=O)NC2C(OC)CN(C(=O)C3=COCCO3)C2)cc(C)c2c(c1)CCC2 C1(C(=O)NCCCNC(CCOc2ccc(C#N)cc2)=O)CC2CCCCN2C1 C1(CNC(c2c(CC)con2)=O)COCCN(C(c2cn(C(C)C)nc2C)=O)C1 CCCCC(O)CC(=O)N(CCNC(c1n[nH]c2cccnc12)=O)CC1CC1 c1(SC(C(N2CC3C(C(=O)NCCNC(C)=O)C3C2)=O)C)ccc(F)c(F)c1 N1(C(C(C(COC)C)C)=O)CC2CCC(CNC(c3ccsc3C(=O)OC)=O)C2C1 CCCCCCCCCN1CCSC1.c1(C(C(=O)OC)NCC)ccc(C(F)(F)F)cc1 C(=O)(CCCCC(C)=O)NC1COCC1N=[N+]=[N-].C12(CC=C)CN(C1)C2=O C1(CNC(c2c(CCC=C)ocn2)=O)CC2CCC(C1)N2C(=O)CC(C=C)CC c1(CC=C)cc(C(N2CC(OC)C(NC(=O)C(CCN(C)C)OC)C2)=O)c(C)o1 C1(=CCNC(CCSc2n(C)nnn2)=O)CCN(C(c2ccoc2)=O)CC1 CC1(C)CCCC(c2[nH]nc(C3CC(C=O)C(O)C3)n2)O1 c1(C(=O)NCCC(C)N(C(c2nc(C)oc2)=O)C)cnc2scc(C)n2c1=O C#Cc1ccc(C(N2CCC(C(=O)NC(C)(C#N)C3CCC3)C2)=O)nc1 c1(N(C(C)Cc2ccccc2)C)ccc(S(=O)(=O)NCCCSC(F)F)cn1 c1(NC(=O)NC)cccc(C(=O)NC(CNC(C2CCCN2CC)=O)C(C)C)c1 C1(NC(=O)Cc2cscn2)CCCC2CN(C(C3(C4CCOCC4)CC3)=O)CC12 C#Cc1cc(C(=O)NC2CCN(C(c3cc(N)ccc3Cl)=O)C2CC)ccc1Cl C1(C(=O)NC2CCCN(C(C3(F)CCCCC3)=O)CC2)CC2C=CCC(C1)C2 N1(C(C2(C)CCOC2)=O)CC2CCC1C(CNC(=O)C1=CCOC1)C2 C1(NC(CNC(c2c(C)cco2)=O)=O)CC2(C1)CC2N=c1[nH]cc(C#N)cc1C c1(C(=O)NCCC2CC(NC(c3snc(C)c3N)=O)C2)n[nH]c2c1CCC2 CC1CN(C(=O)CCCC2CCC2)C1C(N1CC(N2CCOC2=O)C1)=O C=Cn1nncc1C(=O)NC1CCCC1NC(c1nccnc1C)=O Cn1cnc2nc(N3CC4CC=CCC4C3)nc(NCC3(C4CC4)CC3)c12 c1(C(=O)NCC(C2CC2)NC(c2c(C)nn(C)c2F)=O)cc2c(C)n[nH]c2cn1 c1(C(=O)NC(CNC(CS(=O)(=O)N(C)C)=O)(C)C)cn2c(n1)COCC2 C12(CNC(CC(C)C(F)F)=O)CCC(CN(C(=O)C(O)C(C)(C)C)C1)C2 c1(CC)ncc(C(=O)N(CCC(C)(C)NC(c2c[nH]cc2C)=O)C)s1 Cc1ccc(C)c(CN2C3CCC2CN(C(=O)C=CC2CC2)C3)c1O C(=O)(C1=NN(C)C(=O)CC1)N1CCC(n2cc(C3CCOCC3)nn2)(C(=O)OC)C1 C(CCC(=O)NC1CCC(NC(C2(C3CC3)CC2)=O)C1)OCC C1(N(C(=O)C(CO)NC(N)=O)CC)CCN(C(=O)C(F)Cc2ccccc2)CC1 N1(C(C(C)n2cnnn2)=O)CC2CC2(CNC(c2cnn(C)c2Cl)=O)C1 c1(CCC)onc(C)c1C(N1CCC(CN(C(c2nonc2CC)=O)CC)C1)=O N1(C(C(CCNC(c2ccc(SC)o2)=O)O)=O)CCSCCC1C C1(N(C(C(C=C)O)=O)C)CN(C(c2cc(C3CC3)ccc2Cl)=O)CC12CC2 C1(CNC(CC2CN(C)C2)=O)CN(C(C2C=CCCC2)=O)CC1O C(=O)(C1=CCC(F)(F)CC1)NC1CC(C)(C)N(C(c2cc(C3CC3)cs2)=O)C1 C12(NC(c3c(CNC(c4cncc(C)n4)=O)nnn3C)=O)CC1COC2(C)C Cc1ccc(Cl)c(C(N2CC(C3CN(C(C4(C)CCC45CCC5)=O)C3)C2)=O)c1O C1(F)(CNC(C(COC)(C)O)=O)CC2CCC(C1)N2C(=O)Cc1cccc(F)c1 C1(CNC(c2c(C)cc(C)s2)=O)CC2(CCN(C(=O)CN3CC4CC4C3)CC2)C1 C(C(C)C)(C(O)C(=O)N(C)CC1CCCN(C(=O)CCSC2CCCC2)C1)OC C1(c2nn[nH]n2)(NC(=O)Nc2cccc(Cc3ncc(C)s3)c2)CC2CCC1C2 C1(CC)CN(C(c2c[nH]nc2C(C)C)=O)CCC1NC(=O)C=Cc1cnccn1 C(=O)(C1=C(Cl)CCCC1)N1CC(CNC(=O)CC2C=CCC2)OCCC1 Cc1cc2ncc(C(=O)NC3CCCC(NC(=O)C=CC4(C)COC4)C3)cn2n1 C1(OCC)C(C(=O)NCCC(C)N(C(=O)Cn2ccnn2)C)C1C N1(Cc2cn(CC)nn2)CCC(NC(C2CN(C(C)=O)CC2OCC)=O)C(C)C1 n1(CC(=O)N(CCN(C(C2(C)CC(C)=NO2)=O)CC)CC)c(=O)oc2ccccc12 CCC(CC(=O)N(C)CCSC)N(C)C(c1nonc1N)=O C1(C(=O)NCCN(CC)CC)(CO)Cc2ccccc2C1.C1(C(=O)N)CCC1C C1(NC(C2(CCOC)CCN(C(CCC=C)=O)C2)=O)CCc2nn[nH]c2C1 c1(C(N2CC(NC(C(C)NS(C)(=O)=O)=O)C(O)C2)=O)cn2cccc(F)c2n1 Cn1c(C(=O)NCCN(C(c2ccc(O)nn2)=O)CC2CC2)nnc1S C(C(=O)NCCOCCOCCNNCC(=O)NC1CC1)(C1CCC1)OC N1(C(=O)NCc2cnc(-c3ccsc3)s2)CC2CC2(CO)C1 C1(C)(NC(c2n(C)ncc2)=O)CCCN(C(c2cc(C(F)(F)F)ccc2Cl)=O)C1 C1(C(=O)NCC2(CN(C)C(C3(c4ccccc4)CCCO3)=O)CC2)COC(=O)N1C Cn1cnc2c1CCCC2C(=O)NC1CN(C(c2cc3scnc3[nH]2)=O)CC1O C1(COC)(NC(=O)C(=O)NCC2CCC(=O)C2)CCCOC1 c1(CC(=O)NCCC2(NC(C3C(C#N)C3)=O)CCC2)ccc2nonc2c1 c1(-c2c(C)cc(C(=O)O)o2)cnn(NC(=O)C2CS(=O)(=O)c3ccccc32)c1 N12CCCC(C1=O)C2.n1(C(C)C)cc(CNC(=O)CCCOCCS)nn1 CCCC(CCC)=CC(N1CCC(C)(NC(c2cc(-c3ccco3)cs2)=O)C1)=O CC1CC2CCN1C(=O)O2.c1(OC(C)(C)C)cscc1Br Cn1cc(Cl)c(C(=O)NC(CC(=O)NC(C(O)CO)C2CC2)C2CC2)n1 C(CCCCC(=O)N1CCC(C)C(NC(C2(C)CC=CCC2)=O)C1)NC(C)=O c1(C(N2C3CC2CN(S(=O)(=O)Cc2cccnc2)C3)=O)cc([N+](=O)[O-])ccc1Cl C1(=O)C(C(C)C)N1C(C)C(C1CCCCC1)=O.C(C)(C)(CC)N.C(CC#N)SC CC(CC(F)(F)F)C(=O)N1CC=C(CCNC(c2n[nH]cc2Br)=O)CC1 CCC(C(=O)NCCCCCC1CC1)N(C(=O)CCC1OCCO1)C c1(C2CCCN2CCC(C)(C)NC(=O)CNC(=O)C(N)=O)nc2ncccn2n1 c1(NC(C2CCCC(NC(C3CCCC3)=O)C2)=O)cc(F)cnc1Br C1(CC(=O)NC(CCC)C2CCC2)COCCN1C(C1CCCCC1)=O c1(C(=O)NC(CCNC(C2CCC(CC)O2)=O)C)cn(C2CC2)nc1C C(C1CCCCC1)=C(C(=O)NCC1N(C(C(=CC2CCCC2)C)=O)CC(O)C1)F c1(CNC(C2C(C)COCC2)=O)ccc(CNC(c2cnc(C(F)F)s2)=O)cc1F C(C(=O)OC(CNC(Cc1scc(C)c1)=O)C)(C(C)(C)C)N(CCN)C.C(CO)O C(=O)(CC(O)(C(F)(F)F)c1nc(C)cs1)Nc1onc(-c2scc(C)n2)n1 C1(C(=O)NCCCCCNC(CSCC=C)=O)CC2CCCCCC12 N1(C(C(CCC)F)=O)CC2(CCCC2)C1C(=O)NC(C)C(=O)NC(C)(C)C S(=O)(=O)(CC(=O)NCC(C)(C1CCC1)NC(c1cc(=O)n(C)o1)=O)N(C)C C1(C)(C(=O)NCCCCCNC(c2nc(C(F)(F)F)cs2)=O)CCC1(C)C(=O)OC C1(NC(C2(CCC)CC2)=O)CC(C)N(C(=O)CCc2ccnc(C)n2)C1 C1(NC(CC2CC(=O)NCC2)=O)CC2(C1)CN(C(=O)CCc1cnccn1)C2 C1(CNC(c2cc(CC)sn2)=O)CN(C(=O)CNS(N)(=O)=O)CC12CCC2 c1(C(N2CCN(C(c3n(C)c(Cl)c(Cl)c3)=O)CC2)=O)cc(=O)nc2cccnn12 c1(C(=O)NOC2CCC2C(N2CCCC2)=O)ccc2occc2n1 c1(C(C(=O)NC2CC(NC(C3(Cl)CC3)=O)C2)SC)cc(F)cc(F)c1 c1(C(N(C2CN(C(C3(COC)COC3)=O)C2)C)=O)coc2cc(F)ccc12 C1(C(=O)NCCSCc2ccc(C(=O)O)o2)C2CCC1(c1ccccn1)C2 C=CC(CC(=O)NCC(C)CN(C(=O)Cc1nonc1C)C)c1ccccc1 C1(NCc2cn(-c3c(C(=O)NCC4(C=C)CCC4)con3)nn2)CC2CCC2C1 n12cc(nn1)CCNC(=O)CC2.CC(C#N)COCCO Cc1cc(C(C)NC(C2CC(C)(F)C2)=O)ccc1Br C1(C(=O)NCc2cn(-c3cnnn3C)nn2)(CC)CNC(=O)C1 C(=O)(CCC(F)(F)Cn1cc(CCCSC)nn1)NC(CCCC)COC C1(NC(C2(C(=O)OC)CC2C)=O)CCN(c2nnc(C(C)C)o2)C1 N1(C(C(C)N(C(C)=O)C)=O)CC(NC(c2cn(C(C)C)cc2C)=O)CC(C)C1 c1(C(CC)(C)O)cn(C2CC(NC(=O)CCCn3cc(C)cn3)C2)nn1 Cc1ccnc(CNC(C2C3CC3CN2C(=O)CC2CCCCC2)=O)n1 C(=O)(C(C)(C)COC1CCCCC1)NC1C(NC(C(C)NC(N)=O)=O)C1 CCC(C(=O)NCCCC1CCCN1C(=O)Cc1ccn(CC)n1)n1cncn1 c1(OC)cc(C)cc(C(N2CCN(C(c3cncs3)=O)C3CC23)=O)c1C N1(C(C(CNC(C(C2CCC2)OC)=O)OC)=O)CCCC(O)(CO)C1 Cc1cc(C(N2CCOC(CN(C)C(C3(C)CC3(Cl)Cl)=O)C2)=O)c(N)c(Cl)n1 C12(NC(c3cn(CC)nc3)=O)CCCC1CN(C(c1cc(F)c(Cl)cc1F)=O)C2 CC1=C(C(=O)N2CCOCC2CNC(c2c(C)ccnc2O)=O)CCC1 c1(OC)cc(Cl)c(Cl)cc1C(N1CCC(NC(C23CCCC2C3)=O)C(F)C1)=O Cc1ccccc1C(F)(F)C(=O)NCC1CCCN(C(=O)C(C)(F)F)C1 c1(C(N2CCC3CN(C(C=CC(=O)N(C)C)=O)C3C2)=O)c[nH]c2cc(Cl)ccc12 CC1CC(C)CCN(C(=O)C(CCS(C)(=O)=O)NC(c2ccc(Cl)cc2)=O)C1 CC1CCC(C(=O)NC2CCN(C(C3(C4CCC4)CC3)=O)C2C)CC1 C1(C(=O)NCC(C)NC(C(CC)Oc2ccccc2F)=O)CCn2cncc2C1 C(=O)(CCc1nncs1)N(CCNC(C1(CCCC)CC1)=O)C1CC1 CC(C)CC(CNC(c1cc(C(C)(C)C)on1)=O)NC(=O)CC12CCCC1C2 CCS(=O)(=O)c1ccc(C(=O)NCCC2CC(NC(=O)C(C)SC)C2)cc1 c1(C(N(CCOC)CCNC(C2CC(O)C2)=O)=O)ccccc1S(=O)CC C(=O)(CCS(C)(=O)=O)N(CC(C)NC(C1CCC(CCCCC)CC1)=O)C(C)C c1(OC)ccc(C(=O)N(C)C)cc1NC(=O)CN1CCS(=O)C(C)C1 c1(C(N2CC(C(C)NC(C3N(C(C)C)CCC3)=O)OCC2)=O)cc(O)cc(F)c1 c1(C(N(C2CCN(C(C3CC(SC)C3)=O)C2)CC)=O)ccc(S(C)(=O)=O)s1 C1(NC(CC(C)(C)CNC(c2cc(F)c[nH]2)=O)=O)CCn2cnnc2C1 CC1CC(NC(C2CCC(F)C2)=O)CN1C(=O)CCc1nccs1 c1(C(N(CC(C)N(C(=O)CCCCCn2cnnn2)C)C)=O)cnc(O)c(F)c1 C(=O)(C(C)C(C)(F)F)NCC1OCCN(C(C2(C(F)F)CC(=C)C2)=O)C1 N1(C(C2N(CC)CC2)=O)CC(C(=O)NCC(C)(C)C2CC2)C2(CC2)C1 Cc1cc(C(=O)NCC=CCNC(=O)CC2CCC(C)C2)ccn1 C1(CC)CCCN(C(C2CC=C(C)CC2)=O)C1C(N1CC2CC2C2CC12)=O C12(NC(C(CC)C#N)=O)CCC(NC(C3CCC(C)=C(C)C3)=O)(CC1)C2 C12CN(CC1NC(=O)C=CBr)C2=O.C1(CC)C2CC(=O)CC12 c1(CC(C(=O)NC(c2ccccc2)c2cccs2)O)ccc(Cl)cc1Cl c1(NC(c2ccc(Nc3ccnc(SC)n3)cc2)=O)cc(Cl)c(F)cc1F c1(NC(COC2CCN(C(C3(C)CCOC3)=O)C2)=O)cc(O)ncn1 C(c1ccc(Oc2ccc(C3NC(C4C(C(CCCC)NCC)(I)CC4)C3)cc2)c(O)c1)=C c1(C(=O)NC(C)C(C)NC(c2nccc(Cl)c2O)=O)ccc(F)cc1[N+](=O)[O-] N1(C(C(=O)C2CCCC2)=O)CCCN(C(c2cc(Cl)ccc2F)=O)CCC1 c1(CCC=O)ccc(Cl)cc1.N1(CC(F)F)CCN(CC(O)C2CCC2)CC1 Cc1c(C(=O)NCCCC(C)(C)NC(=O)CCCC#N)cc(C(C)C)n1C C1(CNC(c2n(CC#C)ccc2)=O)CN(C(=O)CCSC(F)(F)F)CCC1C CC1(C(=O)NC2COCC2NC(=O)CN2CCC(C(N)=O)CC2)CCC(=O)NC1 c1(C(C)NC(c2nc(CC(=O)OC)no2)CC)cccc(OC(F)F)c1 C12(CC)CCC(CC1)N2C(c1cn(C2CC(N)C2)nn1)=O c1(C(=O)OC(C)C)cc2cc(-c3cnoc3)ccc2oc1=O.CCC1C(=O)N1 C#Cc1cccc(CCN=C(NCc2ncccc2F)NCC2CCCO2)c1 C1(C(=O)NCC2(C(=O)N(C3CCC(C)(C)C3)C)CC(=C)C2)CCCCC1(C)C c1(C(=O)NC2(CO)CCN(C(C3ON=C(C)C3)=O)C2)cc([N+](=O)[O-])n(C)n1 c1(C(=O)NC(CN(C(C(C=C)c2ccccc2)=O)CC)C)cccc(NC)n1 N1(C(C23CCC(OC)C2C3)=O)CCC=C(CNC(C2CC2F)=O)C1 C1(NS(c2cc(C)c(Cl)cc2)(=O)=O)CCN1C1c2ccccc2-c2ccccc21.CNC c1(C2CCN(C(=O)CC3CCCOC3)C2)cccc(Br)c1 c1(C(=O)NCC2(NC(Cc3ccc(C)s3)=O)CCOC2)ccn(C)c(=O)c1 C1(NC(C2CCC(CC)O2)=O)CCC2CN(C(c3c[nH]nc3C(F)F)=O)CC2C1 C(=O)(C1=CC2C=CC1C2)N1C(CC(=O)NCC(F)(F)CO)CC(O)C1 O=C(CCC(=O)N1CCN(CCCc2ccc(F)cc2)CC1)NC1CCOC1 C(N=c1[nH]c(=NC(C)CC(C)O)[nH]c2cc(OC)ccc12)C1CC(=C)C1 c1(C(=O)NC2CN(C(CSCC(C)C)=O)C2)coc(C(F)F)c1 c1(NC(C(N2CCC(c3c(C(=O)OC)cccn3)CC2)=O)=O)cc(F)c(C)c(Br)c1 N12CCCN(CC1)C1(CCCC1)C2=O.O=C1NCC(Cn2cc(CO)nn2)O1 n1(C(C(=O)NCCCN(C(C2CCC(OC)CC2)=O)C)C)c(C)cc(O)cc1=O CC(C)C(CCN(C(=O)C=Cc1ncc[nH]1)C)NC(=O)CNS(N)(=O)=O C#Cc1ccc(NC(=O)C(Cn2cncn2)NC(=O)C(C)(C#N)CC)c(C)c1 C(=O)(C(C)(C)C(F)F)NCc1c(C(=O)NCc2nc(C)on2)occ1 c1(C(=O)OC)cnn(C(=O)NC2(C3CCC3)CCC2)c1.C12C3CN(CC13)C(=O)NC2 Cc1ccc(-c2cnc(C3(C4OCCO4)CCC3)[nH]2)c(Cl)c1 CC1(C#CC(=O)N2CCOC(CCC(=O)NCCCCF)C2)CCCO1 c1(CCC(=O)NCc2ccc(C)c([N+](=O)[O-])c2)c(C)nc2c(c(O)nn2C)c1C C1(CC(N2CCC(C=C)C2)=O)CN(C(=O)C=C(C2CC2)C2CC2)CC1(C)C C(=O)(CCCc1ccsc1)NCCC1CN(C(C(C)NC(c2cccs2)=O)=O)C1 C(CCC(C)(C)NC(=O)CCCN(C(=O)CC(Cl)Cl)C1CC1)OC CC1(NC(c2ccccc2)=O)CCN(C(=NCCF)NCC2CC2(Cl)Cl)C1 N1(C(C(C)O)=O)CC2CC(C1)C2NC(c1cnc(C(=O)O)nc1)=O N1(Cc2ccc(N)cc2C(F)(F)F)CCOCc2ccccc21 c1(C(N(C2CC(NC(C3C=CCCC3)=O)C2)C)=O)ccccc1C1CCOC1 C1(C(=O)NCC(C2CCOCC2)NC(C(C)C)=O)(N(C)C)CCOCC1 N1(C(CN(C)S(N)(=O)=O)=O)CCc2[nH]nc(CNC(=O)C(F)=CCCF)c2C1 c1(C(CCC(=O)N2C(CCNC(C(=O)NCC)=O)CCC2)=O)cc(F)ccc1F CC1CN(C(c2ccc(Cl)cc2Cl)=O)CCC1CNC(=O)CNc1cncnc1 c1(-c2nc(C(CC)CC)nn2CCOC)cc(O)nc(CN(C)OCC(F)F)n1 N1(C(C2(SCC)CC2)=O)CCN(C(=O)C=Cc2cncc(C)c2)CC2(CC2)C1 C1(C2CN(C(=O)Cc3nnc(S)n3C)C2)(NC(c2cn(CCC)nc2C)=O)CC1 CCC(CNC(c1cccc(C(F)(F)F)c1)=O)(CC)Nc1ccnc(C)n1 N1(C(C2C(COC)C2)=O)CCCC1CN(C(=O)C=CSC)C C=C=CC(C)C(=O)N1CCC(CN(C)C(c2cnn[nH]2)=O)CC1 Cc1cc(=NC2CCCN(C(=O)C(O)C(C)(C)C)C2)[nH]c(S(C)(=O)=O)n1 CP(C)(=O)CCC(=O)N1CCC2CC2(NC(c2ccc3nn[nH]c3n2)=O)CC1 C1(CC(=O)N(C2CCCC(NC(C3CCOCC3)=O)C2)C)CCC2(CC1)CC2 c1(OC)ccc2[nH]cc(NC(=O)CSCC3CC4(CO3)CC(=O)C4)c2c1 c1(Nc2c(C)cc(Br)cc2Cl)cc(Br)cc2ccccc12 N1(C(CCCCCC)=O)CCCC(C2CC2NC(c2ccc3[nH]ccc3n2)=O)C1 C1(C)(C(=O)NC2C(NC(C3(CC#C)CCOCC3)=O)CC2)CC=C(C)CC1 C12(CNC(CC(C)(C)n3cc(CC4CCC(=O)NC4)nn3)=O)CC1CCC2(F)F CCC(COC)C(=O)NC1(C)CC(C(=O)NCc2cc(OC)no2)C1 c1(OC)cc(C(=O)NC2CCCC2CNC(=O)CCC(C)CN(C)C)cc(C)n1 C1(C)(C(=O)N(c2scc(C(C)C)n2)C(C)C)CCCN(c2ccc(C#N)cn2)C1 N1(C(CCc2cnc(C)o2)=O)CCC(NC(c2ccnn2C)=O)C12CC2 c1(C(C(=O)NCC2CC(NC(C=Cc3occ(C)n3)=O)C2)C)ccc(F)c(F)c1 CC1CCCn2cc(C(N3CC4CC(NC(c5cn(C)nn5)=O)CC4C3)=O)nc21 C(C(C)(C)CC(=O)NC1CC2(C1)CC2C(=O)N(CC(F)F)C1CC1)N(C)C C=C(C)CC(C)C(=O)N1CCC(C)(NC(c2ccc(C(F)(F)F)c(OC)c2)=O)C1 C(CCCC(=O)N(C)CC1CCN(C(=O)Cc2ccn(C(F)F)n2)C1)SC Cc1cc(C(N2CCN(C(C3(C(C)(C)O)CCC3)=O)CC2C2CC2)=O)cc(N)c1 CC1(C)CC(CNC(C2CCC(=O)O2)=O)CN(C(C2CC3(C2)CS(=O)(=O)C3)=O)C1 C1(CN(C)C(C2CCOC2)=O)CN(C(c2coc(Cl)n2)=O)CCO1 C1(NC(c2cc(C(C)C)no2)=O)CCC12CCN(C(c1cn(C)[nH]c1=N)=O)CC2 c1(C(N(CCOC)CC2CCCN2)=O)cc2cccc(F)c2o1 c1(C(=O)NCC2CN(C(c3cn(CCC)nc3C)=O)C2)cccc2nc(S)oc12 c1(C(N2CC(OC)C(NC(=O)Cn3nc(C)cc3C)C2)=O)cnn2ccccc12 C1(NC(COCCCCC)=O)CC(C)N(C(c2ccc(CC3CCCC3)[nH]2)=O)C1 Cc1cc2sc(C(=O)NC3CCCC(NC(=O)C4=COCC4)C3)cc2s1 C1(C(=O)NC2CCN(C(C)C)CC2)CCCCC(F)(F)C1.N12CC(C1)CC2=O C(N=c1ccc(S(C)(=O)=O)c[nH]1)C1(OC)CCC1.c12c(ccc(F)c1OC)OC2 C(N=c1[nH]c(=NC2CCCN(C)C2)[nH]c2c1CSC2)c1cc(C)nc(O)c1 N1(C(C2(NC(c3c[nH]ccc3=O)=O)CCN(C)C2)=O)CC2CCC(CN(C)C)C2C1 CCC(CC(=O)NCC1COCCN1C(=O)CSc1nncn1C)OC c12ccc(cc1)C(=O)NCC1(CC1)NC(=O)COC2.n1(CC)cnnc1C1CC1 O=C(N=c1cc[nH]cc1Cl)C1CC2CC2N1Cc1ncc(Cl)cc1Cl C1(CF)CCCCN1Cc1cccc(Cl)c1.c12cc(cs1)c1noc2n1 c1(OC)cccc(C2(C(N3CC(NC(=O)CC(C)n4ccnc4)C3)=O)CC2)n1 CC(C)C(C(=O)NCc1ccccc1O)NC(=O)COc1cccnc1 CCCCCC(C)CC(=O)NCCOC(C)(C)CNC(=O)C(C#N)CCC c1(C(C)C(=O)OCCOCCn2nnc(C(C)(C)C)n2)ccc(Cl)cc1F C1(C)(C(=O)NC(c2cn(-c3cccc(OCC)c3)nn2)CC(N)=O)CC(C)=NO1 c1(C(=O)NC2CC2)cnc(CC2(CNC(C3CC4CC4C3)=O)CC2)s1 c1(C(C(=O)NC2CCN(C(COCCOCC)=O)C2)O)ccc(OC)cc1 c1(CC(=O)NC2C(OC)CN(C(=O)C=CC=C(Cl)Cl)C2)cn2cc(F)ccc2n1 c1(CC(=O)NC(CN(C(CCCC(C)=O)=O)C)C)ccc2oc(O)nc2c1 C1(C(CNC(C(C=CCCC)O)=O)O)CCN(C(C2(C)CC=CCC2)=O)CC1 c1(C(=O)NC2C(CNC(C3(C)CC(C)=C(C)CC3)=O)C2)cc(N)cc([N+](=O)[O-])c1 N(C(=NCCc1ccc(F)cc1)NC1CC(F)(F)C1)C(c1ccc(C)cc1)C Cc1nccc(C(N2CCOCC(NC(=O)CCC(F)(F)F)C2)=O)c1C C(C)(C(CC(=O)NC(C)CCOC)NC(=O)COc1ccccc1C)OC Cc1cnc(NC2CCC(=O)NC2C)c(S(=O)(=O)N2CCN3CCOCC3C2)c1 C1(C(N2CCC(C)(CNC(CCC(=C)Cl)=O)C2)=O)CCC(C#N)CC1 c1(OCC(=O)N(C2CCCN(C(=O)CCc3nc(=N)[nH][nH]3)C2)C)cc(F)cc(Cl)c1 C[Si](C)(C)C#Cc1ccc(F)c(Nc2cc(Br)ncn2)c1 C1(C(=O)NCC(C)(C)NC(CN(C)C)=O)CC2C=CC1C2 C1(C)(CC(=O)NC2C(CCC)C2)CCN(C(C2(CO)CCC2)=O)C1 C(N=C(NCC(=O)NC(C)(C)C)N1CCCCC1)C1N(C)CC(F)C1 c1(NC(CCCn2cc(CCP(C)(C)=O)nn2)=O)cncc(C(N)=O)c1 S(=O)(=O)(c1ccc2c(c1)C(=O)NC2=O)N1C(C(=O)OC(C)(C)C)CC(O)C1 N1(C(c2nc(CC)oc2)=O)CCC2(CC1)C(NC(=O)CC1CCOC1)CS2(=O)=O C(=O)(C(F)CC1CCOC1)N(C)C(c1cnn[nH]1)C1CC1 c1cnn2c1CN(S(=O)(=O)C(F)(F)F)CC2.[SH](=O)(=O)C(F)(F)F C(N=c1nc(C(C)C)c(Cl)c[nH]1)C1CCC(CNC(C(CC)(O)C2CCC2)=O)C1 C(=O)(C#CC1CCCC1)N(C(C)CNC(=O)C(c1cnn(C)n1)=O)C C1(C(N2CCC(CC3CC3c3ccc(F)cc3)CC2)=O)CCCC12CNC2 c1(OC)ccccc1SC(C)CC(N)=O.c12cccc(c1)CC(=O)N2 c12cc(-c3nncn3C)c(cc1Cl)-c1cn-2nn1.N1(OC)CC2(N)CCC1CC2 c1(CC)ccc(OC)c(Cl)c1.C12(c3nn[nH]n3)CCN(C1)CCNC2=O N1(C(C2(CNC(c3cc(Cl)no3)=O)CCCO2)=O)CC(O)(C2CC2)C1 c1(C(=O)NCC(CCNC(CC(CC)OC)=O)OC)cc(OC)cnc1F c1(C(=O)NCC2CN(C(c3cnc(C)o3)=O)C(C)(C)C2)ccc(Cl)c([N+](=O)[O-])c1 c1(CC(C)SCC2(C(F)(F)F)CCOCC2)cccc(COC)c1 c1(C(=O)NC2CC3CN(C(c4c(C)nsc4)=O)C2C3)cccc2cncn12 C(C)(N=c1[nH]nco1)C1N(C(c2c(C)nc(CC)s2)=O)CCCC1 c1(C(S(Cc2c(Cl)cn(C)n2)=O)C=Cc2ccccc2)cccc2[nH]ncc12 c1(C(N2C(CN(C(c3c[nH]c(=NC)o3)=O)C)COCC2)=O)sc(C)c(C)c1C N1(CC)C(=O)CCC1C(=O)NCC(C)N(C)C(c1cc(C2CC2)ns1)=O Cc1cccc(C(N2CCC(C(C)C(=O)NCC=C3CCSCC3)CC2)=O)c1 N1(C(C2C(C)=C2)=O)CC(NC(c2c[nH]nc2C2CCCO2)=O)Cc2ccccc21 C(=O)(C1=CCS(=O)(=O)C1)NCC=O.N1(N2CC(C)(C#N)C2)CCCC(F)C1 C1(NC(N)=O)COCC1.C1(NC(CN(CC(C)(C)C)C)=O)CN(C(=O)CNC)C1 N1(C(CN(CC)CC)=O)CCC(F)(CNC(c2c(C3CC3)noc2C)=O)C1 Cc1cc(C(=O)NCC2(F)CC(NC(C3(CC4CCC4)CCC3)=O)C2)on1 C12CN(CC(C)N1C(C1CC1Cc1cccc(F)c1)=O)C(=O)O2.C(C)(C)(C)OC C(=O)(C(CC(C)(C)C)OC)N(CC(C)(C)CNC(c1ccc(CO)s1)=O)CC C(C(=O)N1CCOC(CCC(=O)NCC(CC)CC)C1)(C(C)C)N(CC)CC c1(C(=O)NCC(CC(N2CC(C(=O)OC)C(C)C2)=O)C)ccc(C)c(F)c1 C1(C(=O)NCC(C)CNC(C2CC2c2cnc[nH]2)=O)CCC(C)(C)CO1 Cc1noc(C(C)C)c1CN1CCCCC1c1cn(CC2CC2)nn1 Cc1cc(=O)ccn1CC(N1CCC(CCNC(c2ccc(SC)s2)=O)C1)=O Cc1nc2ncccn2c1C(N1CC(CNC(c2cc3ccc(F)cc3s2)=O)C1)=O c1(C(N(CC(CNC(C(=O)NCCOC)=O)C)C)=O)ccn2ccnc2c1 c1(C(=O)NC2CC(F)(CNC(C3C(C)CC(=O)NC3)=O)C2)nccc2n[nH]cc12 CN1C2CCC1CC(C(=O)NCCOCCCNC(C1CC(N(C)C)C1)=O)C2 C1(OC)CC(NC(c2cc[nH]n2)=O)C12CCN(C(c1cc[nH]c1C)=O)CC2 Cc1cc(C(=O)NCC(C)NC(C2C=CC=CC=C2)=O)cc2nc[nH]c12 C(=O)(CC(CC(C)C)NC(=O)C(C)(C)C)NC(C(=O)OC)CO Cc1cncc(CC(=O)NCCN(C)C(c2ncc(F)cn2)=O)c1 C1(CC=C)(C(=O)NCC(=O)NCCOC)CCCC1.C1CC(CC)(CCl)C1 CCCCCS(=O)(=O)CC(=O)NC1CN(C(c2cnc(C)o2)=O)CC1F c1(SC(C(=O)NCCCC(C)Nc2cn(CC3CC3)cn2)C)ccccc1Cl C1(O)(CNC(C2C(=C)CC2)=O)CCCN(C(=O)Cc2nncn2C(C)C)CC1 C(CCC(C)CC(=O)N1CCCC(CNC(c2ncc(C)cc2F)=O)C1)=C(C)C N1(C(C2(NC(=O)OC(C)(C)C)C(C)C2)=O)CC2CCCCC2C1 C(=O)(C1=NN(C)C(=O)CC1)N1CCN(C(c2cc(C)n(C)c2)=O)C(CF)C1 C1(CCC(=O)NC2C(CCC)C2)CCN(C(C2CCCN(CCC)C2)=O)CC1 CC(CCCCCO)NC(=O)CC1CCN1C(C12CCCC1C2)=O C(=O)(C(O)CC(C)(C)C)NC1C2N(C(c3c(C)n(C4CCC4)nc3)=O)C(CC2)C1 c1(OCC)ccccc1NC(=O)C(C)(CSC)NC(c1csc(C)c1C)=O c1(OCC=C)c(OC)cc(CN2CCCC(CCO)C2)cc1OC n1(CC(=O)NCC2(O)CCC23CCC3)ccc2ncc(Br)cc12 CCCC(C)CC(=O)N1CCC(C(C)(C)NC(c2cc(C)cnc2F)=O)CC1 c1(C(=O)NCC2C(NC(c3cccc(OCC=C)c3)=O)C2)ccc(=O)n(C)c1 C(=O)(C(=O)C(C)(C)C)N1CCCC(C(C)NC(c2c[nH]nc2-c2ccco2)=O)C1 N1(C(CCOCCC)=O)CCC(C)(CCNC(=O)Cc2ccccc2C(N)=O)C1 c1(-c2c(C(=O)NC(CNC(C(CC#C)C)=O)C(C)C)c[nH]n2)ccc(F)c(F)c1 C12(C(=O)NCC3C(NC(=O)CCNC(c4ccccc4)=O)C3)CC3CC1C2C3 C1(CC(=O)NC2(c3ccccn3)CC2)CCCN(C(C2CCCC(=O)N2)=O)C1 C1(CC=C)(NC(c2nn(C)c(Cl)c2Cl)=O)CCCN(C(=O)C=CC)C1 C#CC1(C(=O)NC2CCCC2CC=C)CCN(C(=O)CC2CCCOC2)CC1 C1(C(=O)NCc2ccc(F)cn2)(NC(C(C)O)=O)CCN(C)C1 C1(C(=O)NCC(CCC)OCC)CCN(C(=O)C2=C(C)OCCS2)C(C)(C)C1 N1(C(CNC(CCC)=O)=O)CC(OC(N2CCCC(C)C2)=O)CC1CCCOC C1(C(=O)NCCSC)CCC(n2cc(C3(CCO)CC3)nn2)C1 C(=O)(C1=CC2(CCOC2)C1)N1C2CC(CNC(C3(CC)CCCC3)=O)CC1CC2 O=C1NCC2(CC(NC(=O)CC3(N(C)C(C4C=CCC4)=O)CC3)C2)O1 c1(CC)nc[nH]c1C(=O)NC(C)(CNC(=O)CC1CNC(=O)O1)C1CC1 c1(OC)ncc(C(=O)NC(C)CCN(C(=O)CCc2nccs2)C)c(C)n1 c1(C(=O)OC)cc(C(=O)NC2(CNC(=O)C(F)Cl)CCOCC2)ccn1 C(CCC)(C(=O)NCC1(CC(=O)NC2CCN(C(=O)CC)C2)CCCC1)=CCC c1(CO)nc(C(=O)N(C(C)C(C)NC(C(C)OCCOC)=O)C)co1 CC1C(C(=O)NCCN(C)C2CC2)CCCN1C(=O)CCC1CCCO1 C1(C(=O)NCCC(C)(C)NC(c2c(COC)nn(C)c2)=O)OCCOC12CCC2 N1(C(CC2CCC(OC)CC2)=O)CCN(C(c2cc(C)[nH]n2)=O)C(CO)C1 c1(C(=O)NC2CN(C(C(C)C3CC3)=O)CC2O)cc2c(s1)CCS(=O)(=O)C2 CCCC(C)(C)CC(=O)NC1CC2(C1)CC(NC(=O)C(c1cnn(C(C)C)c1)=O)C2 CCC(CC(C)C)C(=O)NC1CN(C(=O)C=CI)CCC1C(F)(F)F O=C(CCCCCNC(=O)CCC1CCCCO1)Nc1ccc(F)c(CO)c1 N1(C(=O)NC(c2ccco2)=O)CCN(C(=O)C(C)NC2(C(=O)OC)CCCC2)CC1 c1(OC)cccc2cc(C(=O)N(CCCNC(=O)CC3CCCCC3)CCO)oc12 C1(NC(CC(CC2CC2)NC(C2(C(=O)NC)CC2)=O)=O)CC2CC1C(O)C2O C1(C(N2CCC(c3c(C)c[nH]n3)CC2)=O)CC12CCc1cc(Br)ccc12 CCCCC(F)C(=O)N(C1CC1)CC1CCCN1C(=O)C(O)CN(C)CC N1(C(C2CC(OC)C2)=O)CCC(CO)C(NC(=O)CCC(N)=O)C1 C1(C)(CNC(CC(C)(C2CCC2)N(C)C)=O)CCCN(C(C2(CCO)CC2)=O)C1 C1(NC(C2CC3(CC(=C)C3)C2)=O)CC12CCC(NC(=O)C1=CC(C)(C)C1)CC2 C1(COC)(CNC(C2CCCCN2C)=O)CCCN1C(=O)CCN1CCC1 N1(C(CNC(=O)NCC)=O)CC2CCN(C(C3CC3CCOC)=O)C2C1C C1(NC(CCc2c(C)ncs2)=O)CCC2(CC1)CN(C(=O)C(F)=C1CCC1)C2 Cc1nn(CC(=O)N(CCC(=O)NCCCCC2CC2)CCO)c(=O)o1 C(=O)(C1c2c[nH]nc2CN1C(c1ccc(C#N)cn1)=O)NC1(CCC)CC1 C#Cc1cncc(C(=O)NCCC2(C(N3CCCC3C=C)=O)CCCC2)c1 C(c1ccc(OC)cc1)=CC(N1CCC(CN(C(c2cc(OC)ns2)=O)C)C1)=O C12(C(=O)NC3CCN(C(=O)C=CC4CCCC4)C34CC4)CC=CCN1CCC2 c1(C(=O)NC2CCC(CNC(=O)C3=CCCCCC3)C2)cn2cc(Cl)cnc2n1 C(=O)(C(F)C(F)(F)F)N1C(CC(=O)N(C2CCC2)CCC)CC1 C1(NC(=O)CCSC(F)(F)F)CCCCN(C(C2CCC3CCC2O3)=O)C1 C1(CCNC(c2n(CCCF)nnn2)c2cc(C3CC3)on2)CCCCC12CC2 c1(CCC(=O)NC(CCNC(C2C(C(C)(C)C)C(=O)C2)=O)(C)C)nnc(O)nc1O Cc1cc(C(O)C(C)NC2(C)CCOC2Sc2ccccc2)ccc1F C(=O)(C(C)C(O)CC(C)C)NC(CC)(C)CCNC(=O)C(O)C1CC1 N1(CC)CC(C(=O)NC(C)(C)CNC(c2cnc(C)s2)=O)NC1=O N1(C(c2cn(CC)nc2C)=O)CCC(C2CC2)(CNC(=O)C(C)C2CC2)C1 N1(C(c2c(CC)n(C)cc2)=O)CCCC(NC(C2(C)CC=CCC2)=O)C1C CCC(C(=O)NC1(C)CCCN(C(=O)CCc2cc(C)n(C)n2)C1)C(C)C N1(C(C(C=C)O)=O)CCC(NC(c2cncc(C)n2)=O)C1CC C1(CC(=O)NCCCCN(CCCNC(COCC=C)=O)C)CCCC(F)(F)C1 c1(SCC(=O)NCC(C)(O)CNC(C2CCSCC2)=O)nc2ccccc2[nH]1 N1(C(c2c(C)cc(C)[nH]2)=O)CC2C3CCC(C2C1)N(C(=O)CN1CC2CC2C1)C3 C(C(C)CC(=O)NOCC1(C)CCC1)NC(C1C(CC)CCCC1)=O N1(C(CCC=CCC=C)=O)CCC(COC)(NC(=O)CC(C)c2ccccc2)C1 CC(C(C)(C)NC(C1CCC1)=O)NC(=O)COCC1CCCOC1 N1(C(c2ccc(CN(C)C)nc2)=O)CCc2cc(O)c(C(=O)ON)cc2C1 N1(C(CC2C(C)=NOC2=O)=O)CCOCC(C)(CNC(=O)Cn2cncc2C)C1 N1(C(Cc2c(C)nn(C)c2Cl)=O)CCN(C(=O)CCc2ccco2)CC(C)(F)C1 C12(Cn3cc(C4(C)ON=C(C)C4)nn3)CCCC1CC(=O)N2 N1(C(C(OC)OC)=O)C2CCC1CC(CC(C)NC(c1ncsc1C)=O)C2 C1(C(=O)N(C(C)CC2CC2)C)(CC)CCCN1C(c1ccoc1)=O c1(COC(C23CCC(NC(C4CCCO4)=O)(CC2)CC3)=O)ccc(F)c(F)c1Cl C1(NC(c2sc(Cl)cc2Br)=O)CN(C(c2cnco2)=O)CC2(CCC2)C1 CC(C)C(C)(O)C(=O)NC(C)C(=O)N=CCC1(CCO)CCC1 c1(C(N2CCCC(Cc3nccs3)C2)=O)cnc(C(F)(F)F)nc1O N1(CC(=O)N(C(C)C)CCN(C)C(c2ccc(C(C)(C)C)o2)=O)CCC(F)CC1 C1(F)(C(N2C(CNC(C3(COC)CC3)=O)CC(COC)C2)=O)CCCN(C)C1 C1(C(=O)NCC(C2CC2)SC)CCC(C(C)C)N1C(=O)C(C)SC(C)C CC1CN2CCN1CC2C(=O)N(C)CC1CCCN(C(C2C3CC4C(C3)C24)=O)C1 Cc1c(C(c2nnnn2C)Nc2cc(CO)ccc2Cl)cc(C#N)n1C Cc1cc(Br)cc(COC(c2cccc(C(N)=O)c2)=O)c1F C1(NC(C(C)C(C)(C)C)=O)CN(C(=O)Cc2cc[nH]n2)C2(CCCCC2)C1 N1(C(c2sc(C)c(O)n2)=O)CCCN(C(C2CC(C)CC(=O)N2)=O)CCC1 C1(N(C(C(C(C)C)NC(c2ccn(C)c2)=O)=O)C)CC2CCC1CC2 C1(C(N2CC(C#C)(C(N3CCCC(CCF)C3)=O)C2)=O)CC12CCOCC2 C(=O)(C1CCOc2ccccc21)NC(C)CCNC(=O)CCC#N C12CC3(CCOCC3)CN1C2=O.CCC(Br)C(=O)OC(C)(C)C c1(N(CC(C)CO)C)[nH]c(=NCC2(CO)CC2)nc2c1CCCC2 C(=O)(C1=CCCOC1)N1C(C2(C=O)CC2)CCCC1.CC(C)CCF Cc1nnsc1C(=O)NCC1CC(CNC(C2CCCN2C(C)C)=O)C1 C1(CNC(CSCC=C)=O)CCCC1C(=O)NCC#CCCO c1(C(=O)NCCNC(c2ccc([N+](=O)[O-])c(O)c2)=O)ccc2c(c1O)CCCC2 C(=O)(C1=C2CCCN=C2NN1)N1CCCC(NC(c2cc(C)oc2)=O)CC1 c1(C(N2C(NC(=O)Nc3ccc(OCC)nc3)CCC2)=O)c(C)nc(O)nc1O Cc1cc(Cl)ccc1Cc1nc(-c2cscn2)nn1C1CCOC(C)C1 N1(C(c2cc(C(F)(F)F)cc(C)c2)C(=O)NCCCSC)CCSC2CCCC12 CC(C)CCCCCC(=O)NCC1CC2CCC1N2C(=O)CN1CCC(C)(O)C1 c1(OC)c(C(N2CCCC2C(N2CCC(O)(CO)C2)=O)=O)cnn1C N1(C(C(CC)SC)=O)CC(CNC(c2cn(CC)cn2)=O)OC(C)(C)C1 c1(OCC=C)ccc(CNC(=NCC)NCCCOC2CCCCC2C)cc1 C12(CNC(c3c[nH]nc3F)=O)CC1CN(C(c1cccc(C3CCC3)c1)=O)C2 N1(C(CCC)=O)CCOc2ncc(-c3ccc(C)c(CC4CCC4)c3)c(C)c21 N1(C(CSCC#C)=O)CCN(C(=O)CC(C(F)(F)F)c2nccn2C)C2(CCC2)C1 C=C=C(C)CC(=O)NC1CN(C(=O)CN(C(C)=O)C2CC2)C1 C1(C2CCN(C)CC2)(C(=O)NCCC2(C(N3CCC(OCC)C3)=O)CC2)CC1 CC1(C)OC2(C(N3CCCC3CCCNC(=O)CC3=CCCC3)=O)CC1C2 CN=c1nc(N2CCN(C)CC2)[nH]c(=NCCOCC(F)(F)F)[nH]1 n1(CC(C)O)cnc2c(N3CCN(C(=O)C(n4cc(Cl)cn4)C)CC3)ncnc12 c1(C(N2CC(CC(C)NC(CN(CC)CC)=O)C2)=O)cnc(C(F)(F)F)cn1 Cc1c(C(=O)NC(C)CNC(c2ccc(-c3ccccn3)o2)=O)nnn1C(C)C N1(C(CSCC#C)=O)C2CC=C(C(=O)NC3CC(O)C34CCC4)C1CC2 c1(CCN(C)C)ccc(NC(=O)CC2(NCc3ccc(CBr)cc3)CCC2)cc1 CN1CC(Cn2cc(C3C4CN(C(=O)OC(C)(C)C)CC34)nn2)OCCC1=O CC1CC(=O)NC1C(=O)NC1CC(NC(c2ccnn2CCC(F)(F)F)=O)C1 C(CCN(C(=O)C(C)C1CCCC1)C)(C(C)(C)C)NC(C(C)=NOCC#N)=O C#CCC(CC#C)C(=O)NCCC1CCN(C(=O)C2=NOC(C)C2C)CC1(F)F CCCC(CCC)C(=O)NC1CC(NC(=O)CC(C)C(=O)OC)CC1O C1(C(=O)NCCOCCC)CCN(C(=O)CCCC2CC2C)CC1O C1(NC(C2C(CC)CCC2)=O)CCC(C)N(C(=O)Cc2nccs2)C1 CCCCCCCCCC(=O)N1CC(NC(c2ncn(C)n2)=O)CC12CCCC2 C(=O)(C1=COCCO1)N1C(CNC(c2csc(-c3cccs3)n2)=O)CC(OC)C1 C12(C(=O)NC(C#C)C(C)OC)CCC(CC1NC(=O)CCc1ccncc1)C2 C#CC1(O)CCN(C(=O)C(=O)NC(c2ccc(Cl)cc2)c2ccccc2)C1 Cc1ccc2nonc2c1C(=O)N(C(C)CC1CN(C(c2ccsc2Cl)=O)C1)CC c1(CN2CC3C(C(=O)NCC4CCN(CC)C4)C3C2)c(F)ccc(Br)c1F C1(C(=O)NCCNC(c2coc(Cl)c2)=O)(Cc2ccccc2)CCOCC1 c1(OC)ccc(C(=O)NC(C2(CNC(c3cc(C)[nH]c(=N)n3)=O)CC2)C)c(C)n1 C1(NC(Cc2cc(C)on2)=O)CCC(NC(c2ccccc2Br)=O)CC1 C1(C(C(=O)NCCOC)N(C2CCNC2=O)C)CCN(CCF)CC1 c1(N(CC)CC)ccc(C(=O)N(CC(c2ccccc2Cl)C)CC)cc1 c1(C(=O)NCC2(NC(C(COC)C)=O)CC2)c(C)nn(-c2cccc(Cl)c2)c1C c1(OC)ccc2c(c1)NC(=O)C2CC(=O)NCCNC(c1cc(CCO)on1)=O N1(C(COCC(=O)NC)=O)CC2CCN(C(c3ccccc3C(C)C)=O)C2C1 C1(F)(CNC(C(C2CCCC2)OCC)=O)CCN(C(=O)C(O)C2CC2)CC1 CN1CCC(N=c2[nH]c(=NCc3ccnc(OC(F)F)c3)[nH]c3c2CSC3)C1 C1(C(N(CCNC(=O)C=Cc2cocn2)CCOCCO)=O)CC2(C1)CC21CCC1 N1(C(=O)OCc2ccccc2)CCC2(CC1)CN(Cc1n(C(C)C)ncc1F)C2 C1(SC)CCN(c2ccnc(NC(=O)NC3(c4ncco4)CC3)n2)CC1 CC(C)CCCC(=O)NCC12CC1CN(C(=O)CC1NC(=O)NC1=O)C2 C1(C(=O)NC2CN(C(=O)C=CC=C)C2)CC1C1CCCC1.c1(NC(=O)CO)ccoc1 c1(C(=O)OC)cnccc1C(=O)NC1(CCO)CN(C(=O)CSCC(C)C)C1 C1(N(CCNC(c2cccc(COC)c2)=O)CC)CCS(=O)(=O)CC1 Cn1ccc(CNC2(c3cccc(C(=O)O)c3)CCCCC2)cc1=O C(=O)(CC(F)(F)CC(=O)N1CCC(C)N(C(=O)CSCC(F)(F)F)CC1)OC CCC(C)C(C(=O)N1CC2CC1(C(=O)N(C)Cc1nnnn1C)C2)N(C)C N1(C(CCC(C=C)C)=O)C2CCCC1CC(NC(c1ncoc1Br)=O)C2 c1(NC(=O)COC(C(F)F)c2cccs2)c[nH]cc1Br c1(OCC=C)ccccc1C(N1CCCC(CN(C(=O)C(=O)NC(C)C)C)C1)=O n1(CCC(=O)N(CC(C)NC(C2CC(C)(C)O2)=O)CC)nc(C)nc1C n1(CC)nc(C(N2CCCC(CC(=O)N(C(C(N)=O)C3CC3)C)C2)=O)c(C)n1 C=Cc1ccc(C(=O)NCC(C2CC2)NC(=O)CCNC(=O)C=CCl)cc1 CC(C)(C)CCCCCC(=O)NCCC1CN(C(=O)Cc2cnccn2)CCO1 c1(C(=O)NCC2CCC(C(=O)NC(c3ccncc3F)C)O2)cc(O)ncn1 C(=O)(C1=C2CCCN=C2NN1)NCC1(C)CCN(C(C2CCCSC2)=O)C1 N1(C(C2(C#N)CCN(C(c3ccccc3)=O)C2)=O)CCc2sc(Br)c(Br)c2C1 Cc1cc(Cl)cc(C(N2CC3CCCC2C3CNC(C2CCCSC2)=O)=O)c1N C1(CC=C)(C(N2CCOC(CC(N)=O)C2)=O)CCN(C(c2ns[nH]c2=O)=O)C1 c1(C(N2CC(NC(C=C(CC)CC)=O)C(C)C2)=O)cc(Br)c(O)cc1F CN1CCC(C2CCN(C(=O)NCc3snc(Cl)c3Cl)C2)CC1 C1(F)(C(N(C)CC2(NC(c3n(C(C)C)ccc3)=O)CC2)=O)CCOCC1 C1(n2cc(CNC(COC)=O)nn2)CCCN(C(C2(N(C)C)CC2)=O)C1 C1(NC(CSCCOC)=O)CCCC(C(=O)N(CCCC(C)(F)F)C)CC1 c1(CC)n[nH]c(=NC2CC(CNC(c3cc(C)nc4ccnn34)=O)C2)o1 CCC(CC)(CCNC(c1cc(C2(C)COC2)no1)=O)NC(C1CC1F)=O CON(CCC(=O)N(C(C)C(C)C)C1CC1)C(=O)CN1C(=O)CNC1=O N=c1nc(C(F)(F)F)[nH]c(=NC2CC(CNC(=O)C3CCc4c[nH]nc43)C2)[nH]1 c1(CC(N2CCC(O)(C(C)NC(CC=C)=O)C2)=O)nc([N+](=O)[O-])n[nH]1 c1(C(=O)NC(CN(C(COCCCC)=O)CC)C)cnc(C(C)(C)C)o1 C1(CCC(=O)NCC=C(C(=O)N(CCCOC)CCO)C)CCC(=O)C1 C1(C)(NC(C2C(C)C2)=O)CCCN(C(C2C(C)(C)C2(C)C)=O)C1 n1(CC(C)C)cc(NC(c2n[nH]cc2CNC(=O)CC2(N(C)C)CC2)=O)cn1 C1(CC=CC)CCCN(C(=O)C(CCNC(c2occc2COC)=O)OC)C1 N1(C(C2CCC3(CC2)CC3)=O)CCC2C1CCCN2.c1(SC)ncc(Br)c(N)n1 CCCCCCC(C)C(=O)NC1(C)CC(NC(c2cc3cnccc3[nH]2)=O)C1 c1(CS(C)(=O)=O)nc(=NCC2CC3CC3C2)s[nH]1 Cc1nc(=NC(=O)c2cccc(CC3CCC4(CCC4)CO3)c2)n(C)[nH]1 C(=O)(CCCC(=O)N(C)C)NC(C)C(CO)NC(C1CCN(C2CCSC2)CC1)=O c1(C(=O)NCC2(F)CC(NC(c3cc(OCC)n[nH]3)=O)C2)sc2nccn2c1C c1(C(=O)NCCC(CNC(=O)CC2CCC2CF)O)cc(C(F)(F)F)ccc1F c1(C(N2C(CCNC(CCC(C)SC)=O)CCCC2)=O)ncnc(O)c1Br N1(C(C(C(C)(C)O)F)=O)CCc2c(CNC(C3CC(=O)N3)=O)cccc2C1 N1(C(C(C=C)OC)=O)CCOCC1C(=O)NCC1CCCC1CC c1(C(N2CCC(C)(NC(c3[nH]cc(C)c3)=O)C2)=O)cc2ccc(Br)cc2s1 C(=O)(N=c1ncn(C(=O)OC)[nH]1)c1nc(CC=C)c2n1cccc2 N1(C(c2c(C)[nH]c(=N)s2)=O)CCC2(C1)CN(C(=O)Cc1ccc(Cl)cn1)C2 C(=O)(CC(O)CNC(=O)C1=C(Cl)CC1)NC(c1cnccn1)C C(=O)(C(C)(C)CC(C)(C)C)NC1CN(C(C=CC=CC)=O)C2(C1)CCC2 C1(C)(C(N(C(CNC(C2CCC(O)C2)=O)C2CC2)C)=O)CCC(=O)C1 Cc1cccc(C=CC(=O)NC2CC3CC2N(C(C24CCC(CC2)CC4)=O)C3)c1 C1(C(=O)NC2CCC(CNC(C3(CSC)CC3)=O)C2)CCCCCS1(=O)=O CCC(CC(=O)NC1CC2CCC1N2C(c1ccoc1Br)=O)C(C)(C)C c1(OC)ccc(CN(C(=O)CN2CCS(=O)CC2)C)c(C)c1 c1(C(CC(=O)NC2(CO)CN(C(CCCOCCC)=O)C2)O)cccc(F)c1 N1(C(C2CCC(=O)O2)=O)CCCN(C(c2cscn2)=O)CC1 C#Cc1ccc(C(=O)N(C2CCC(NC(c3ccc(N)c(Cl)c3)=O)C2)C)c(F)c1 c1(C(N2CCC(CC=C)(NC(=O)C(C)C(C)(C)O)C2)=O)nc(C)c(C)[nH]c1=O c1(CCC)c(C(=O)NC23CC(NC(C4CC4C(C)C)=O)(C2)C3)cnn1C c1(OC)ccc(CCN2CCCC(C(=O)NC(c3ccc(Cl)cc3)C)C2)c(Cl)c1 C1(C(=O)NC(C2(O)CCN(c3nnc(C4CC4)o3)C2)C)Cc2cccc(F)c2O1 C(=O)(C(C)(C)CCC#N)N(CC(C)(C)NC(C(CC1CCC1)OC)=O)C c1(C(=O)NCC(C)NC(=O)C(C)C2(O)CCC2)cc(Br)c(O)nc1C C1(OC)CCCC(n2cc(CCN3CCCC3)nn2)(C(=O)NC(C)C2CC2)C1 Cn1nc(O)cc1C(=O)N(C1CCCCC1)CCNC(c1occc1C1CC1)=O C1(CNC(C(C(C)C)NC=O)=O)CCC2(CN(C(=O)C=CCN3CCCC3)C2)O1 C1(C(=O)NC2CC(CCNC(c3c(C)nc(Cl)cc3)=O)C2)CCCC2CCCN12 C(=O)(C(=O)C(F)(F)F)NCCC1(CNC(C(CCOC)C)=O)CC1 Cc1ccc(CC(N2CCCCC2CCNC(c2cccc(F)c2)=O)=O)c(Cl)c1 CCC(CC)CCCC(=O)NC1CC(CC(=O)Nc2cc(C#N)c(Cl)cc2F)C1 c1(C(=O)NC(CN(C(C(CC)CC)=O)C)C)cc2c(C)n[nH]c2cn1 N12C3CCC1CC(C3)C2=O.Cc1ccc(C(=O)Nc2cc(CC3CC3)on2)nc1 c1(CN(C(C2(C#C)CC2)=O)C)ccc(CNC(c2n[nH]c(C)c2Cl)=O)cc1 CCC(C)(C)CC(=O)N1CCOCCC1C(=O)NC(C)CS(N)(=O)=O C(CC(C)(C)C(=O)N1CCCN(C(c2nccc(OC)c2N)=O)CC1)SC Cc1cc2ncnc(NC3CS(=O)(=O)CC3NC(C3CC(N(C)C)C3)=O)c2[nH]1 c1(OCC)ccc2c(c1)CCN(C(c1ccc(CO)o1)C(=O)NCCCSC)C2 C(CCC1CC1)(C(=O)NC(CCC)COC)NC(c1cc(COC)on1)=O c1(OC)nc(N2CCCC(NC3CC(OC)C3)C2)c2ccc(NC(C)=O)cc2n1 N1(C(Cc2nc(=N)[nH][nH]2)=O)CCN(C(c2cccc(Cl)c2F)=O)C2COCC12 c12cnc(Cl)cc1C(=O)N2.c1(C2(NSCCCC)CCC2)cc(OC(C)=O)ncn1 N1(C(c2c(C)cncc2C)=O)CC(O)(C2CCN(C(=O)C(C)CS(C)=O)CC2)C1 CCC(C)(CO)C(=O)NCC1(CNC(c2ccnn2CC2CCC2)=O)CC1 c1(C(N2CC3C(NC(C4(SC)CC4)=O)C3C2)=O)cnn2c1OCC(F)C2 C1(C(N2CCC(NC(=O)Cc3cocn3)C2C2CC2)=O)CC2CCC(C1)C2O c1(C(=O)NCC(CN(C(c2[nH]c(=NC)sc2)=O)C)C)ncc(C)cc1OC N1(C(=O)Nc2n(C=O)cnc2)CCOC2(CCN(C(=O)Cc3cccc(O)c3)C2)C1 c1(OC)ccc(C(=O)NCCC(C(C)C)NC(=O)CC(C)F)cc1C1CC1 c1(C(N2CC(NC(c3cscc3Br)=O)C2)=O)cccc([N+](=O)[O-])c1O Cc1ccncc1C(N1CC(NCc2cccc(-c3ccncc3)c2)C(C)C1)=O N1(C(COCCCC#C)=O)CCC(N(CCC)C(C2CCN(C)C2)=O)C1 N1(CC(N2CCCC(C(C)NC(c3cnn(CCF)c3)=O)C2)=O)CCP(C)(=O)CC1 c12ccc(cc1)C(=O)CN2CCC.c1(CC(=O)OC)cccc(F)c1 CCC(C)CC(=O)NCC1CCC(F)(CNC(C2(SC)CCC2)=O)C1 C1(C(N(C)CC2N(C(COCCOC)=O)CCC2)=O)CC(C(C)(C)C)=NO1 c1(CN(C(=O)CCc2cn(C)nn2)C)ccc(S(=O)(=O)CCO)cc1 c1(C(=O)NCC2C(C)CCN2C(=O)C2=NOCC2)cc2n(n1)CCO2 N1(CCCCOCC#C)CCCC2CNCC12 N1(C(c2occ(C)c2)=O)CC(O)CC1C(N1CCC(O)(CC(C)C)C1)=O Cc1nc(-c2cc(CC(N3CCC(N(C)C(C4C5CCCC45)=O)C3)=O)cs2)cs1 CC(C)(O)C(C)(C)C(=O)N1CCC(O)C(NC(C2CCCC(CF)C2)=O)C1 CN1CCN(C(=O)C2=NOCC2)CC1CNC(c1ccc(-n2ccnc2)nc1)=O Cc1cccc(C)c1N1C(=O)C1C.C(=O)(C1=NNC(=O)C1)NCCNC(=O)C(C)(C)C N1(C(c2c(C(=O)OC)c(C)on2)=O)CCC(NC(=O)CNS(C)(=O)=O)C(C)C1 c1(CCC(=O)NC2CC(C)N(C(=O)CCCF)C2)ccc(F)c(Br)c1 N1(C(c2c(C(C)=O)nccc2)=O)CC(NC(=O)C=Cc2cocn2)CC(F)C1 c1(OC(c2ccc(C)cc2F)=O)ccc2cccc(F)c2n1 CC(C)(CC(=O)NCC1CC12CCN(C(c1cn[nH]c1)=O)CC2)C(F)(F)F CCC(CC(C)C)C(=O)NC(CN(C)C(c1ccccc1OC)=O)(CO)CO c1(CN(C(C2(C(F)(F)F)CC(F)(F)C2)=O)CC)c(OC(F)(F)F)cccc1F Cc1cccnc1C=CCNC(N1CCC12CC(O)C2)=O c12ccc(F)c(c1)-c1cn(nn1)C(C(=O)NCC(CC)C)CO2.C(C)(=O)NC C1(NC(C2CC(SC)C2)=O)CC(C)CN(C(c2cc(O)ncc2Br)=O)C1 C1(CC(=O)NCC(CCOC)NC(=O)CCn2cccn2)CCCC(=O)N1 C1(C(N2CCC(C)(NC(C)=O)C2)=O)CC2(CC(NC(=O)OC(C)(C)C)C2)C1 N1(C(c2cc(CC)no2)C(=O)NCC2CC2)CCC(C2CCCC2)C1 N1(C(C(=O)NCc2cc(C(=O)OCC)no2)=O)CCC(=O)N2CCCCCC12 c1(C(N2CC(NC(C(C#C)(C)C)=O)C(C)C2)=O)c[nH]c2cc([N+](=O)[O-])ccc12 c1(C(N(CC(=O)NCCCN(C)C)CC#C)=O)cncc(OCC#C)c1 C1(NC(=O)COCCF)CCC(F)(CNC(=O)CCSCc2ccccc2)C1 C1(COC)(CNC(=O)CCSc2nnnn2C)CCCN1C(c1cccs1)=O c1(C(=O)NC2(C)CN(C(CCc3cc(C)sc3C)=O)C2)cc(Br)cc(C)c1N c1(C(N(CCN(C)Cc2cccn3cnnc23)C)=O)cc2sc(C(=O)O)nc2s1 C1(C(=O)OCC)OC(C)(C)OC1CNC(c1nccc(Br)c1C)=O C1(OC)C2CCC1N(C(=O)NC1CC3(C1)CC(C(=O)OC(C)(C)C)C3)C2 c1(C(N2CC(CC)(NC(=O)Cc3occc3C)C2)=O)cc(O)ncc1F C1(O)(NC(CCNC(=O)NC)=O)CCN(c2ncc(Cl)c(C)n2)CC1 c1(OCC(=O)NCC(CN(C)C(=O)NC2COC2)O)cnn(C)c1 C1(C(N2C(c3cn(C)nc3SC(C)(C)C)CCC2)=O)COC2(C3CC3)CC1C2 C1(CC(=O)NC2COCC2O)CN(Cc2ccnc(C(F)(F)F)c2)CCO1 c1(C(=O)NC(CC)CN(C(=O)C=NOC)C)ccc(C2CC2)nc1 C1(C)(CC)C=C(C(=O)NCC(O)CNC(C2CCN2C)=O)C1 c1(C(C(N)=O)NC(C(=O)NC(c2ccccc2OC)CC)=O)cccc(Br)c1 CC1C(=O)N(CC(=O)Nc2cccc(C(=O)NC(C)(C)C)c2)C(=O)C1C c1(-c2ccc(CN(C)Cc3cccc(Br)c3)o2)cc(F)ccc1F C1(NC(C(C2CCN(C(=O)CC3CCC3C)C2)C)=O)CC(C)(C)OC1=O C12(C(=O)NCCCCN(C(c3n(CC)cnn3)=O)C)CCCN1CCC2 CC1CCN(C(=O)CNC(=O)CCC(N)=O)CC1CC1(O)CC2CCC1O2 C=C(C)CC(C(=O)OC)NC(C1(NC(=O)C(=O)CC(C)C)CCCC1C)=O c1(C(=O)NC2C3(CC(NC(CCS(C)(=O)=O)=O)C3)C2)cnc2cc(O)ccc2c1 S(=O)(=O)(CCC(=O)NC1CCCC1CNC(=O)Cc1csnn1)NC N1(C(c2cc(C)nc(C)n2)C(=O)N(C(CC)C)S(C)(=O)=O)CCN(CC)CC1(C)C c1(C(=O)NC(C(C)NC(Cc2c(C)scc2)=O)CO)nn(C)cc1Cl Cc1cc(C(N2CCCC(CNC(C3CC34CC4)=O)C2)=O)n2nc(C)c(C)c2n1 C(C(C)C)(C(O)C(=O)NCC1CC2(CC2)CN1C(C1CC(F)(F)C1(F)F)=O)OC C(C(C)(O)CCC)SC.N1(C(CCOCCOC)=O)CC2(C1)C(=O)N2 C(C(C)C(C)C(=O)N1CCCOC(CNC(c2ncccc2N(C)C)=O)C1)OC c1(C(NOc2cccc(F)c2)=O)cc(Br)c2occc2c1.CCCN1CC1 N1(C(C(CC)(C)O)=O)Cc2ccnn2CC(NC(c2cccc(CO)n2)=O)C1 C(=O)(CC1C(=O)Nc2c(F)cccc21)N(CCCNC(C(CC)C)=O)CCO C12(C(N3CC4(CN(C(c5cc(OC)ns5)=O)C4)C3)=O)CCCC(=O)N1CCC2 c1(NC(N(CCN2CCCC2)CC)=O)cccc2[nH]c(Cc3ccccn3)nc12 N1(C(C2C=C(C)CS2)=O)CCC2(C(=O)NCC(C)CCCO)CCCC12 c1(NC2CN(C3CCN(CC)C3)C(=O)C2)nccc2[nH]nc(C(C)C)c12 N12CCC(C)C(C1)CC2=O.CCS(=O)(=O)NCCC(=O)OC c1(C(N(CC(C)O)CCNC(c2cnc(CCCC)s2)=O)=O)cc2occc2[nH]1 CCCCCCC(C)CC(=O)N1CC(O)(CNC(c2ccncc2N)=O)C1 C#CCC(C)(C(=O)NOCCC(C)O)NC(c1c[nH]c(=N)c(C)c1)=O N1(C(C(C)(O)C2CCC2)=O)CC=C(C(=O)N2CCCC(F)CC2)C1 N1(C(C2CCC(NC(=O)CC3CCC3)C2)=O)CCOC(F)C1 c1(C(N2C(CCC#C)CCC2)=O)cc2ccccn2c1 C1(C(=O)NCC(CN(C(=O)CCC2CCCCO2)C)(C)C)CC(=O)N(O)C1 c1(C(=O)NCCN(C(C(C=C)O)=O)C2CCCC2)cc(C(F)F)ncn1 c1(OC)cc(C(=O)NC2CC2NC(=O)CC2COC(C)(C)C2)c2c(c1)CCC2 N12CC3CC1(CO3)C2=O.CC(C)(C)OC(=O)NCC1COC1 CC1COC(C(=O)NCCc2nncn2C)c2ccccc21 N1(C(C2C3COCC23)=O)CCN(C(C2(O)CC3CCC2C3)=O)CC(O)C1 C1(O)(CCNC(=O)NCCCCSC)CCOC1 C(=O)(C1CCCn2cnnc21)C(C1Cc2ccncc2C1)=O.C12(N)CN(C1)C2 c1(CC)[nH]nc(C(N2CC(=C(F)CNC(=O)CC3CC=CCC3)C2)=O)c1Br c1(C(N(C(CN(C(C(CCCCC)O)=O)C)C)C)=O)ccc([N+](=O)[O-])c(C)n1 C1(NC(C2(C)ON=C(C)C2)=O)CC2CC1N(C(c1nc[nH]c1C(F)(F)F)=O)C2 N1(c2ncnc(C)c2C#N)CCC=C(C(=O)Nc2cnc(Cl)c(Cl)c2)C1 Cc1ncc(CCNC=O)s1.C1(c2nnnn2C2CCC2)(C)CC1(C)C C12(NC(C3(C)CC3)=O)CCC(CC(=O)NC(CNC(C3CC34CC4)=O)C)(CC1)C2 N1C(NCC23CCC(CC2)OC3)=NCCCOCCN2CC1CC2=O.CCOCC c1(CNC(C2(c3c(Cl)cccc3Cl)CC2)=O)cc(Cl)ccc1[N+](=O)[O-] N1(C(c2csc(C)c2N)=O)CC2CC(NC(=O)C(c3ccncc3)C)CC2C1 C1(CNC(Cc2ccn(C)n2)=O)CN(C(=O)Cc2cccnc2)CC1O C1(CC=C)(NC(c2cnoc2-c2cccs2)=O)CN(C(C2CC(SC)C2)=O)C1 c1(SC)cncc(C(N2CCN(c3ccc(C(N)=O)cc3)CC2)=O)c1 C1(C(=O)NCc2ccc(CCO)cc2)(COC)CCC(=O)CC1 C1(NC(C(CCOC)NC(=O)CC2CCCC(=O)N2)=O)CC2(COCCO2)C1 N1(CC(=O)OCC)CCN(N2Cc3ccccc3C2CO)CC1 c1(C(=O)N)n[nH]c2c1CCC2.C1(NC(C2CCN2C(C2(C)C(C)C2)=O)=O)CC(F)(F)C1 c1(C(=O)NCCCOCC(C)(C)NC(C2(C)CCC(=O)N2)=O)csc2c1CCCC2 C(C(C)C(C)C(=O)NC(C1CN(C(=O)CCOCC2CCCO2)C1)C)OC C(CC(O)C(=O)N(CC(N1CCCC(CCO)C1)=O)CC(C)C)SC c1(C(C(=O)NCCCC)N(CCC)C)cnn(CCC)n1 N1(C(CC2(N(C)C)CC2)=O)CCOC(C(=O)NCCCn2cccc2)C1 C(=O)(CCC(=O)NN(C)C)NC1CCN(C(Cc2cc(C)nc(O)c2)=O)CC1 C(=O)(CC(C)(C)C(F)F)NCCOCCN(C(c1c(CC)con1)=O)C N1(C(C(CCC)(C)CC)=O)CCn2c(CNC(c3ncn(CC)n3)=O)nnc2C1 c1(-n2cc(C(N3CCCC3CCCO)C(=O)NCCOC)nn2)ccc(C)c(F)c1 C1(C(=O)NCC(CNC(C(CC)C)=O)O)C2C3CC4C1C1C2CC3C41 c1(CNC(=O)CC2CCCN2C(=O)CCC2CCOC2)cc(Cl)cc(Cl)c1O c1(CC)ccc(C(=O)N(C)CC2CCCN(C(c3cn(C)[nH]c3=N)=O)C2)cc1 C1(C(=O)NCCCNC(C2CCC(C(C)(C)C)C2)=O)CC2C(C1)C2(F)F N1(C(C(CCC)OCC)=O)CC2(CCC2NC(=O)C=Cc2cncc(C)c2)C1 c1(C(C(=O)NCc2nnn(C)n2)N(C2CCCC2C#N)C)ncccc1F c1(C(C(=O)NC(CCCC)CNC(c2cnn(C)c2N)=O)O)ccc(F)c(Cl)c1 N1(Cc2cccc(OC)c2)CCCC(NC(=O)CCc2c(F)cccc2F)CC1 c1(C(=O)NCC2N(C(C(F)OC)=O)CCC2)cc(C2CC2)nc2ccccc12 c1(OCC(N2C3(CNC(c4c(OC)csc4)=O)CC(C2)C3)=O)cccc(C)c1F CC1(C)CN(C(C2(N3CCCC3)CC2)=O)CC1NC(C1CC=CCO1)=O C(=O)(C1=C(F)CN(C(=O)C(C)O)CC1)NCCc1cnc(C)s1 C1(C(=O)NC2(CNC(C=C(C)C(F)F)=O)CC2)CCCOC1C CC#CCC(C(=O)N(CC(C1CC1)OC)C)NC(c1cc(C)n(C)c1)=O C=C(Cl)CCC(=O)NC1CCCN(C(c2cnc(C)s2)=O)C1 Cn1nnc(CNC(=O)CC2CCCN2C(=O)Cc2cncs2)n1 C1(N(C)C(c2ccccc2)=O)CCCN(C(=O)CC2CCCC2(F)F)CC1 N1(c2nnc(CSc3ccc(C(=O)OCC)cc3)n2C)CCN(CCO)C(=O)C1 C1(NC(=O)CN2CCSCC2)CC2CN(C(c3ccnnc3)=O)CCN2C1=O C1(C)(C(=O)NC(COCC)C(=O)NCC(C)(F)C(C)C)COCCO1 N1(C(CN(CC(C)C)C(C2CCSC(C)C2)=O)=O)CCn2ccnc2C1 c1(C(CNC(C2C(C(C)C)C2)=O)NC(=O)CCc2cccs2)cccc(Cl)c1 N1(C(c2c(CC(C)C)cccc2)=O)CC2(CCN(C(C3CCC(C)O3)=O)C2)C1 N1(C(CC2SCC(C)C2)=O)CCCC(CCC(=O)NC(C(N)=O)C2CC2)C1 C(=O)(C1CCCc2nncn21)N(C(c1cn(-c2ccc(Br)cc2)nn1)C)C CCCC(C(=O)N1CCC(c2ccccc2)(NC(c2cn(C)nn2)=O)C1)OCC c1(OC)c(N2CCCC(C)(NC(c3cncc(C)n3)=O)C2)ncnc1Cl C(C(C(C)(C)C)NC(C1C2CC1N(C(C1CCCC13CC3)=O)C2)=O)N(C)C N1(C(C(C)(O)C2CCC2)=O)CCC(NC(c2ccc3nccn3c2)=O)CC(O)C1 c1(C(N2C(C)CC(NC(Cn3c(C)cc(C)n3)=O)C2)=O)ccn(C(C)C)c(=O)c1 C1(NC(CCc2ccc(C)s2)=O)C2CCCC1CC(NC(c1csc(Cl)n1)=O)C2 CC1CN(C(=O)Cc2cccs2)CC1NC(C1C2CC1(c1cccnc1)CO2)=O c1(CCC)nc(=NC(C)CNC(c2ccc(C3CC3(F)F)cc2)=O)s[nH]1 N1(C(CCOC)=O)CC(CNC(c2cc(OC)cc(COC)c2)=O)CC1(C)C n1(CCC)cc(C(=O)NCCC2CCN(C(=O)CC(C)C)C2)cn1 Cc1nc(SNC(=O)Cn2cc(C(C)N(C(=O)C(C3CCCCC3)C)C)nn2)cs1 C(C(CNC(C1CCOC1)=O)CO)NC(c1ccc(SC(F)(F)F)o1)=O c1(C(=O)NCCOCCNC(C2(CC(C)C)CCC2)=O)cnc(N(C)C)nc1 c1(NC2C(NC(C3N(CC)CC3)=O)C2)cccc(C(=O)NC2CC2)c1 C1(C(=O)NCC2(O)CC(C(=O)NC3CCN(C(C)C)CC3)C2)(CC)CCCCO1 c1(CC)ccc(C(=O)NC(C)C(C)NC(=O)C(C)Nc2nc(C)cs2)cn1 N1(C(C2N(CC)C(=O)CC2)=O)CC2(CCCN(C(C3(O)COC3)=O)C2)C1 C1(N2C(=O)COC2)CCCN(C2=NCCCN2NCC2CCOC2)CC1 CS(=O)CCC(O)C(=O)NC1CCN(C(c2cnn(C(C)(C)C)c2)=O)CC1 C1(NC(c2scnc2C(F)(F)F)=O)CN(C(c2ncc(F)cc2F)=O)CC12CC2 N1(C(C2CCN(C(C(C)C)=O)C2)=O)CC(NCCN2CCCCC2C)C(F)(F)C1 c1(C(=O)NC2(C)CN(C(c3cc(O)ccc3Cl)=O)C2)cnc2occc2c1 C1(NC(=O)CCC(=O)c2ccc(Br)s2)CCCCC12CCC2 C1(NC(CC(C)SC)=O)CCC(N(C(=O)Cc2sc(SC(F)F)nc2C)C)CC1 C1(OCCOCCNC(C2CS(=O)(=O)CC23CC3)=O)Cc2cc(F)cc(F)c2O1 c1(-c2ccc(C)o2)cn2cnc(C(=O)Nc3nccs3)c2s1 c1(NC(C2CCCN(C(c3cncc(C#N)c3)=O)CC2)=O)ccccc1C(N)=S C1(C(N(CCC)CC2CCCCO2)=O)CCN(C(C2(CC)CCCC2)=O)C1C n1(CC)nc(C(=O)NC(CNC(=O)C(C)(C)COC)C2CCC2)cc1C C1(O)(CNC(c2c(C)ocn2)=O)CCN(C(c2csc3cncn23)=O)CC1 N1(C(CC2CC(NC(C34CCCC3C4)=O)C2)=O)CCc2cncnc2C1 C1(C(=O)NCC2C(OCC)CN(C(C(F)=CCC)=O)C2)CCc2nncn2C1 N1(C(c2c(COC)cc[nH]2)=O)CC2(C)CC1(C(=O)NCc1csnc1OC)C2 N1(C(c2c(CCC)cccc2)=O)CC2(CC2)CC1CNC(C1CCCOC1)=O c1(C(N2C3CN(C(C(CC=C)(F)F)=O)CC2CC3)=O)ccc2c(ccn2C)c1 C1(CNC(C2CCCCN2C(c2cccc(C3CC3)c2)=O)=O)CC12CCOCC2 c1(C(N(C2CC(NC(=O)CC#N)C2)C)=O)cc2scc(Br)c2s1 C1(C)(C(=O)NCC2CCC(NC(CC=CCC)=O)C2)COCCO1 C1(CNC(C2OCCC2C(=O)NC2CC(OC(C)C)C2)=O)(CO)CCOCC1 c1(C(N2CC(CNC(C(C)CC(F)F)=O)OCCC2)=O)ccc2ccnn2c1 c1(C(=O)NCC2(NC(C(CC)(C)C(N)=O)=O)CCCC2)cscc1S(C)(=O)=O c1(C(C)C)nc(Cl)cc(=NCC=C2CC(CN3CCSCC3)C2)[nH]1.C1(=O)C(C)N1 CCCCCCCCCCNC(=O)CN(c1cc(NCC(F)(F)CC)nc(C)n1)C C(=O)(C(C)C(=O)N1CCCC(CC(N2CCC2CSC2CC2)=O)C1)OC CC(=Cn1ccnn1)C(=O)NCC(O)COc1ccc(C=O)cc1 CC(CCNC(C1CCCC1NC(c1ccc2occc2c1)=O)=O)CC(C)(C)C n1(CC)cc(Cl)cc1C(=O)NC1C=CCN(c2ccnc(C3CC3)n2)C1 CC1(C)CN(C(C2(F)CC2)=O)CCC1NC(c1cc(Cl)c(N)cc1F)=O CC1CCN(C(c2ccc(F)cn2)=O)C1CNC(=O)C(C)(F)c1ccon1 CC1(C)CN(C(C2(F)CCOCC2)=O)C1Cc1ccccc1F c1(C(N(CCCCN(C(C(c2cnn(C)c2)C)=O)C)C)=O)c[nH]c(=S)cn1 N1(C(CCCc2onc(C)n2)=O)CC(C)(C)CC1CNC(=O)C(CO)N(C)C c1(-c2ccc(CNCCN(CC)Cc3nc(C)c(C)o3)o2)ccccc1Cl c1(OC)ccc(Br)c(C(=O)NC23CCN(C(=O)Cc4coc(C)n4)CC2C3)c1 N1(C(CSCCCC)=O)CCCCC(NC(=O)CCc2ccnc(C)n2)C1 Cc1cccc2cc(C(=O)NC(CNC(=O)CC3(C)CC3(Cl)Cl)CO)sc12 CC1CC(C(=O)NC(CN(C)C(c2cccnc2S)=O)(CO)CO)C1(C)C N1(C(C(CC)(CO)OC)=O)CCCCC12CN(C(=O)C=CCF)C2 c1(C(N2CCC(COCCOC)C2)=O)cnc(C2CC2)nc1O.C1(C)C(=O)S1 C1(C(=O)NCc2ccc(C)s2)CC(NC(=O)Cn2[nH]cnc2=N)C12CCC2 Cc1c(NC(=O)C(C2CCC(C)=C(C)C2)N(C(C)C)CC2CCCO2)cccc1Cl C1(NC(C2(C(N3C(CC(=O)NC)CC3)=O)CCCCO2)=O)CCN(C)C(C)C1 c1(CC)cc(C(=O)N(C2CCN(C(=O)CN(C3CCCCC3)C)C2)CC)n(C)n1 CC1(C)C(CC(N2CC(C(O)C(N3CC4CCCC34)=O)C2)=O)CC1O N1(C(C(C)(C)C2CCC2)=O)CCC(CNC(c2ccc([N+](=O)[O-])o2)=O)C(O)C1 C1(C(N2CC(NC(c3ncc(OC)cn3)=O)C(OC)C2)=O)CCC(C)(C)CO1 CS(=O)(=O)C1CC(NC(C2CN(Cc3cc(O)cc(Cl)c3)CCO2)=O)C1 N1(C(c2cc(F)c(O)c(F)c2)=O)CCC2CCN(C(C3C4COCC34)=O)C2C1 C1(NC(C(C(=O)OC)F)=O)CCCCN(C(c2cnc(C3CC3)[nH]2)=O)C1 c1(C(=O)NCC2N(C(CC=CC=C)=O)CCC2C)cc2c(F)cccc2s1 C(N=c1cc(C(C)(C)C)nc[nH]1)C1N(C(c2ccc(SC)cc2)=O)CCCC1C C1(C2CC2)(CNC(C2CCCC2O)=O)CCN(C(=O)CC2CSC2)C1 Cc1cc(Cl)c(NC(c2ccc(C(F)C(F)(F)F)cn2)=O)cc1Cl N1(C(C23CC=CC(C2)OC3)=O)C2CCC1C(CNC(C1CCC(F)C1)=O)C2 c1(C(=O)NC(C2(CNC(c3cc(N)cc(O)c3)=O)CC2)C)n[nH]c2c1COCC2 C(=O)(C1=CCCCC1C)N(CCNC(C1NC(=O)NC1=O)=O)CC C1(C(=O)NCC2(F)CN(C(CC3CC(=O)NC3)=O)C2)CCC2(CCOCC2)O1 C1(C(=O)NCC(C#C)C(C)C)CCN(C(=O)C=Cc2nccs2)C(C)(C)C1 N1(C(CC(=O)NC)=O)CC(C)CN(C(c2cccn(O)c2=O)=O)CC1C c1(NC2CCC3CN(C(COC)=O)CC3C2)cc2nc(O)oc2cc1[N+](=O)[O-] C1(CCn2cc(CN(C(c3ccc(Br)cn3)=O)CC)nn2)CCCC(C)C1 C1(CN(C(=O)CC2CCOC2)C)(NC(=O)OC(C)(C)C)CC1(C)C c1(C(=O)NC2(CC=C)CCCN(C(COCCC)=O)C2)ccc2cnc(C)n2c1 CC(C)C(O)C(F)(F)C(=O)NC1CCN(C(c2cc(C(F)(F)F)c[nH]2)=O)CC1 N1(c2nnc(C)c(C)n2)CCC(C2CCCN(C(=O)C(C(C)C)NC(C)C)C2)C1 c1(C(=O)NCC2CN(C(c3cnsn3)=O)C3CC23)noc2cc(F)ccc12 C(C(C(=O)N)NC(=O)CCOC1CCC1)OCC.N(C=O)CCC=CCO c1(OC(C)(C)C)ccccc1F.N1(C=O)CCCC1Cn1cc(CNS(N)(=O)=O)nn1 C1(C)(C(N(C2CCN(C(c3cccc(C(N)=O)n3)=O)C2)CC#C)=O)COC(=O)C1 CCC(C(=O)NC1CC(N(C(N)=O)CC)C1)SC.c1(C(C(=O)N)O)cccnc1 C1(OC)CC(CNC(=O)CC2CCNC(=O)C2)N(C(=O)COC(F)(F)F)C1 N1(C(CCCCOC)=O)CC2CCOC2(CNC(=O)C(C(C)C)NC(C)=O)C1 N1(C(CC2CC(OC)C2)=O)CC(C)(C)CC1CC(N1CCC(CC(C)O)CC1)=O C1(F)(C(=O)Nc2cc(C(=O)OC)n(C)c2)CCN(C(=O)Cc2cccc(Cl)c2)CC1 C1(C(=O)OC)COCCN(C(C2(C)CCN(C(=O)Cn3c(O)nnc3O)C2)=O)C1 C1(NC(COCC(C)C)=O)CCCCC1NC(=O)CCF NC(=O)CC(O)C(=O)N1CCC(NC(c2ccsc2C(F)F)=O)C1 c1(C(=O)NCC2(NC(C3CCC(C)(C)C3)=O)CCOC2)cc([N+](=O)[O-])ccn1 C=CC(F)(F)C(=O)NC1CC(NC(c2cc(-c3ccccn3)no2)=O)C1 Cc1cc(C(N2CC(O)CC2C(=O)NC2CC3C=CC2C3)=O)ccc1I CCCCC(CC(=O)N1C2CCCC1CC2)NC(C1CCCN1C1CC1)=O c1(C(=O)Sc2ccccn2)ccnc(C(c2cn(C(C)(C)C)nn2)OC)n1 CCC(C)C(C(=O)NCC1CN(C(c2ccc(COC(F)(F)F)cc2)=O)C1)OC C(=O)(CCCN(C)N=O)N(C)CC1CN(C(c2n(CC)ccn2)=O)C1 CC1CCC(CNC(=O)CCC2CC2)N(C(=O)CN(C)C2CC2)C1 C1(c2n(C(CC)(C)C)nnn2)(NCCCC2CCC2)CCC(C2CC2)C1 C1(CNC(CSCC=C)=O)(NCCCC2(CCC(=O)NC)CCCC2)CCCC1 c1(C(N(CCCNC(C2COC(C)C2)=O)C(C)C)=O)ccn2nccc2n1 C1(CCC)(NC(C2CCC(=O)O2)=O)CCCN(C(c2csc(O)n2)=O)C1 C#Cc1ccc2c(c1)CN(C(=O)NCCc1ccccc1)CC2 C1(C(=O)NCCC2(O)CCN(C(c3c(CC)[nH]nc3Cl)=O)C2)COCC(C)(C)O1 C1(NC(C2CCN(CCOC)C2)C)CCN(C)C1(C)C.C(C)(C)(C)OC(=O)O Cc1oc(C(N2CCC(C(C)C(=O)NCc3ccsc3)C2)=O)cc1CO C1(N(C(C(C)NC(C2(NC=O)CC2)=O)=O)C)CCN(C(=O)CCOC(C)(C)C)C1 N#CC1CCC(CC(N2CC=CC(NC(=O)CCc3ccncc3)C2)=O)C1 N1(C(=O)COCCOCCOCCO)CC2CCC1CN2C1CCc2ccc(F)cc21 CC(C(=O)NC1CCN(C(c2ccnc(C3CC3)c2)=O)C1C)C(C)S(C)(=O)=O CC(C)(CC(N)=O)NC(=O)CC1CC(F)CN1C(=O)COC1CC(N(C)C)C1 C(=O)(CC(C(=O)OC(C)(C)C)C(C)C)N1CCCC(CNC(C=CCCC)=O)C1 C=CCCCCCCCC1C(=O)C(CC)N1CC(=O)NCCOCC N1(C(CCC)=O)CCCC1(C)CNC(=O)C(N)COCc1ccccc1 N1(C2CCN(C(C(CSC)C)=O)C2)CCN(C(c2nocc2C)=O)CC1 C1(Nc2c(C)ccc(S(=O)(=O)N(C)C)c2)CCC2(CC1)C(=O)Nc1ccccc12 c1(CC(=O)NCCc2cn(Cc3cscc3Br)nn2)ccc(F)c(Cl)c1 c1(C(N2C3CN(C(C=CCCCCC)=O)C(C3)C2)=O)cc2cc(Cl)ccc2n1C c1(SC)cccc(C(=O)NC2(C(=O)NCC(CC3CC3)CO)CC(F)(F)C2)c1 c1(Cc2c(C(N(CCOCCO)CC)=O)scn2)cc(C2CCCN2C)[nH]c1 CCCCC(C)(F)C(=O)NCC1=CCCN(C(=O)Cn2cccc(N)c2=O)C1 C(=O)(CCCS(C)(=O)=O)NCC(=C)CCNC(c1c(C)nsc1C)=O N1(C(CCC(C)SC)=O)CCC(F)(CNC(=O)CC(n2nc(C)cc2C)C)CC1 C1(C)(NC(CCN(C(c2cc(C)oc2)=O)C(C)C)=O)CCSCC1 CC1(C)CCC=C1C(=O)N1CC(N(C)C)C(CNC(c2cncnc2)=O)C1 c1(C(N(c2cc(C)nc(C)n2)Cc2onc3c2CCCC3)=O)c(C)cc(O)nc1C c1(CC(C)C)n[nH]c2ccc(NC(N3CCCC3c3ccccc3F)=O)cc12 C1(CCC(=O)NCC(CC)OC)CCN(C(C2(CC)CCCC2)=O)CC1 N1(C(C2(CC)CCCCCC2)=O)CCC2(C1)CN(C(=O)CC(C)F)C2 N1(C(c2c(C)nc(Br)o2)=O)CC(CNC(=O)CC2CCCCO2)CC(C)(C)C1 c1(CNc2c(CNC(C3CCN(C(C)=O)C3)=O)cccc2)cnc(O)nc1O CC(c1ccccc1F)=CC(N1CCC(NC(=O)CC23CCCC2C3)C1)=O CCS(=O)(=O)CC(=O)NC(C)(C)CCCNC(C1COCCN1C=O)=O C(C)(C(C)(C)C(=O)NCCCn1cnnc1)NC(C(C)CCN(C)C)=O c1(C(c2n(CCSC)nnn2)NCc2nc(C3CC3)no2)cc(Cl)c(Br)cc1F N1(C(C(C(C)C)F)=O)CC2CCC(C1)C(NC(c1ncn3cc(Cl)ccc13)=O)C2 c1(N(C2CCN(C(=O)CC3C=CCC3)C2)C)ccc([N+](=O)[O-])cn1 c1(N(C(C2C(NC(c3cccc(F)c3)=O)C2)=O)CCO)cccc(Cl)n1 CC(C)(C)CC(O)C(=O)NC(C1CCCC1)CNC(c1cc[nH]c2nccc1-2)=O N1(C(=O)NC(c2nncs2)C)CCOc2ccc(Br)cc21 C1(C)(NC(C2CC(C)C2)=O)CCCN(C(c2cncc(O)c2)=O)C1 c1(C(=O)OCC)cnc(NC2CC3(C2)CC(C)C3)n2ncnc12 CC1CC(C(=O)NCc2cnn(C)c2O)N(C(C2CCCSC2C)=O)C1 C1(C(N(C)Cc2cn(C)nn2)=O)CN(C(=O)CCC2CNC(=O)N2)CC1(F)F C(C(=O)N1OC2CCC1CC2)C1(C)CCN(C(=O)C(=O)NC2CC2)C1 C12(CNC(=O)CCN3CCCC3)CC(CO1)N(C(C1(CO)CCC1)=O)C2 c1(C(N(C)CC2CCN(C(C(CC)F)=O)C2)=O)cnc2ccnn2c1C c1(OC(CC)C)nccc(C(=O)N(C)CCNC(C2(COC)CC2)=O)c1F C(=O)(C1CCCc2n[nH]cc21)N(CC(CNC(C1(COC)CCOCC1)=O)O)C c1(OCC(=O)NCC#CCNC(CC2CCC(C)CC2)=O)ccccc1C#N N1(C(Cn2ncc(C)c2)=O)CCCCC(CCC(N2CC3CC(C)C3C2)=O)C1 CN1CCN(C)C(CNC(C2CCN(C(=O)c3ncccc3O)O2)=O)C1 n1(CC(=O)NC23CC(CNC(C4CNC(=O)C4)=O)(C2)C3)cnc([N+](=O)[O-])n1 Cc1ncc(C(=O)NCC(C)(C)OCCOCCNC(=O)CN2CCC2C)c(=N)[nH]1 Cc1cccc(Br)c1C(C(=O)NCc1cccc(=O)o1)NC(C1CCC2(CC2)C1)=O C1(NC(c2cn(CC=C)nn2)=O)CC2CCC(C1)N2C(c1cccc(N)n1)=O N1(C2CN(C(=O)CCc3cccs3)C2)CCN(C(C2CCN2C2CCCC2)=O)CC1 N1(C(C(CCCC)F)=O)CCN(C(C2CC2(F)Cl)=O)C(C)C1C CN1CC=C(CNC(=O)CC2CCC(NC(=O)CNS(N)(=O)=O)C2)CC1 c1(C(N2CCN(C(C(C(CC)C)C)=O)CC2C)=O)cncc(P(C)(C)=O)c1 C1(C(=O)NCC2CCN(C(C(CCC)N(C)C)=O)C2)Cc2c(C)cccc2O1 c1(C(N(CCCNC(c2cnc(N)cn2)=O)C)=O)ccc(N=[N+]=[N-])cn1 N1(C(c2c(CC)con2)=O)CCC2(NC(=O)Cc3ccnc(Cl)c3F)CC2C1 n1(CC(=O)N(CCCNC(C2C(=C)CC2)=O)C2CC2)cc(Br)c(C)n1 CC1(CNC=O)COCCN(C(=O)CCF)C1.C(O)(C(F)(F)F)C1(C2CSC2)CCC1 C1(NC(=O)CSCC2CCOC2)CCC12CN(C(=O)CCc1cnccn1)C2 C1(C(=O)NCC(C(=O)NCC2CN(C3CC3)C2)OC)CCCSC1C N1(C(c2ccc(C)o2)C(=O)NCC2CCOCC2)CCC2CCCCC12 CC1CN(C(=O)CCc2cn(C)nn2)CCC1NC(C1CCC=CO1)=O c1(SC)ncc(NC(=O)CC2CC2(F)Cl)s1 N1(C(C(CC=C)CC)=O)CC(C)OC2(CCN(C(c3ccoc3CC)=O)CC2)C1 CC1(C)CCC=C1C(=O)N1CCCC(N2CCN(C(=O)C=C3CCSCC3)C2)C1 N1(C(c2conc2C)C(=O)NC(C(=O)NC)CC(C)C)CCOC2(CCN(C)CC2)C1 c1(N(C)C(c2ccccc2OCC(F)(F)F)=O)ccc2c(n1)NC(=O)CO2 C1(C(=O)NCC2CN(C(c3c(C)nn(CCO)c3C)=O)C2)CC(=O)CC12CCC2 c1(C(=O)NCC(CN(C(=O)Cc2nnn(C(C)(C)C)n2)C)O)nccnc1N(C)C c1(Nc2ccc(Cl)cc2)cnc2[nH]c(=NCC34CCCCC3C4)sc2c1 Cn1c(Cl)cnc1C(F)(F)C(=O)NCC1CCCN(S(=O)(=O)C(F)(F)F)C1 C1(F)(C(=O)NCCCCCSC)CCCN(C(=O)CC[SH](CC(N)=O)CC)CC1 C1(C)(NC(C2CCN(C(C)=O)CC2)=O)CCCN(C(n2cnc(Br)n2)=O)C1 C#Cc1cn(C)nc1C(N1CCC(NC(=O)CC2COCCN2C)C1(C)C)=O Cc1ccc(C(=O)NCC2CN(C(=O)CC3CC3(Cl)Cl)C2)nc1O c1(CNC2CCN(C(C)Cc3cc(Cl)cc(Cl)c3)C2)cccc2nonc12 S(=O)(=O)(c1cc(C)ccc1C)NCC(=O)NCCC1CN(C(CC(C)SC)=O)C1 N1(C(C(CC)NC(N)=O)=O)CCCCCCC1C(N1CC(F)CC1C)=O c1(NC(C(=O)NC(c2cc(Br)no2)C)=O)cccc(SC(F)F)c1 C(=O)(CC1=CCCCC1)NCCC1N(C(c2cnc(OCC)s2)=O)CCCC1 C1(CC(N2C(CCNC(CCCC#N)=O)CCC2)=O)CCC(=O)NC1=O Cc1cnn(C)c1C(=O)NCC1(C)CC(NC(=O)C(C)CF)C1 C1(C(N2C(CNC(c3cccc(OC)n3)=O)CCC2)=O)CCC(C2CC2)C1 c1(-c2cn(C3C4CN(C5=CCC(C)CC5)C(C4)C3)nn2)cc(F)c(Br)cc1F c1(CN2CC3CN(C(=O)Nc4cccc(OC)c4)CC32)cc(F)cc(C)c1O C1(CCC)CCC(C(=O)N(CCCNC(=O)CCC(F)F)CC)CC1 N1(C(CC(n2ccc(C)n2)C)=O)CC(NC(=O)C=Cc2cc[nH]c2)CC1CO N1(C(C(C)NCCC(=O)OC)=O)CCc2cncnc2C1 c1(C(C)NC(C2N(C(C3(C(=O)OCC)CC3)=O)CC2)=O)cc(C)on1 C(=O)(C(C)(C)c1nncn1C)NC1(CCNC(=O)OC(C)(C)C)COC1 S(=O)(=O)(c1ccsc1C(=O)NCC(O)CCC1CC1)NC(C)(C)C c1(C(N(C(CNC(C(CC)COC)=O)C2CC2)C)=O)cn(CCO)c(=O)nc1O c1(C(N2C(C)(C)C(NC(C3OCCO3)=O)CC2)=O)cc2ncccc2o1 C1(NC(c2cn(CC)nn2)=O)COCCN(C(c2cc(C(F)(F)F)c(Cl)cn2)=O)C1 N1(C(CC(C)(C)O)=O)CC2(CCC2)CC1CNC(c1cc(C2CC2)[nH]n1)=O CCC(C)C(CC(=O)NC1CCC(C(C)C)CC1)NC(=O)C(C1CCOCC1)O CCC(C)(O)C(=O)NCC(C)(C1CCC1)NC(c1cc(C#N)cs1)=O CN1C(=O)CC(C(=O)NC2CCN(C(c3c[nH]c(=N)o3)=O)C23CC3)C1=O N1(C(c2c(CC)cno2)=O)CCN(C(=O)C=CCCC(C)C)CC1CC1CC1 C1(CC(NOCC(=C)Cl)=O)CN(C(=O)C(C2CCCCC2)O)CCO1 C(=O)(C(C)(F)C(=O)NCC(C)NC(=O)COc1c(C)cccc1Cl)OCC C1(N(C(Cc2n(C(C)C)cnn2)=O)C)C2CN(C(=O)CC3CCCO3)CC12 C(c1ccc2c(c1)COCC2)=CC(=O)NCC(F)CNC(C1CCCOCC1)=O N1(C(C2CC(C)CN(C(c3cnn4c3CCC4)=O)C2)=O)C2CCC1CC(=O)NC2 C1(F)(CNC(C2CC(C)N2C(=O)Cc2ccon2)=O)CCN(C)C1 N1(C(C(CC)O)=O)CCC(C)(C)C(C(=O)NCCc2cccnc2O)C1 N1(C(CSCC=C)=O)C2CCC1CC(CC)CN(C(c1cc(C(=O)OC)on1)=O)C2 c1(C(=O)NC(CNC(C2(COC)CC=CC2)=O)CO)cc(C)c(N)cc1F CON(C(=O)C1CCC(C(N2CCCC2)=O)O1)C(C)CC(=O)O C1(CNC(c2cn(CC(C)C)nc2)=O)CCCCC1NC(=O)C=CC1CCC1 c1(C(N2C(C(C)(C)NC(CCCOCC)=O)CCC2)=O)ccc2ccn(C)c2c1 C1(NC(C(C)(C)NC(C)=O)=O)CC2CCCC(C1)N2C(C1CCCC(=O)N1)=O N1(C(CSC(C)C)=O)CC(NC(c2ccc[n+]([O-])c2)=O)C(c2ccccc2F)C1 c1(C(N2C(CCNC(C3(OC)CCSC3)=O)CCC2)=O)c[nH]c(=O)cn1 c1(C(N(C2CN(C(=O)C=C3CCCC3)CC2O)C)=O)cc(-c2cn[nH]c2)ccn1 C1(NC(COCC#C)=O)C=CCC(C(=O)NCCN(CC(C)C)CCC)C1 C1(OC)CC(NC(c2cc(CC3CC3)on2)=O)CN(C(=O)Cc2cnc(C)[nH]2)C1 CCC(C)CCCC(=O)Nc1cccc(NC(=O)C(C(C)C)C2CCC2)c1 N(C(=NCCCOC(F)(F)F)NCC1(C)COC1)Cc1c(CC)onc1C c1(C(=O)NC(CCNC(C(F)=CC)=O)C)ccc(F)cc1CC Cc1ccc(C)c(C(N2CCN(C(c3ccsc3C(F)F)=O)C(C)C2)=O)c1N c1(NC(C2(O)CCN(C(C3CC4CCC3O4)=O)C2)=O)ncc(Br)cc1I C1(CC)CN(C(C2CC(C3CC3)=NO2)=O)CCC1NC(c1cccnc1C)=O C1(CC=C)(NC(c2ccoc2Cl)=O)CCCN(C(=O)CCc2ccccn2)C1 C1(NC(C2(C#C)CCCC2)=O)CC2CCC1CN(C(c1cc(C(N)=O)no1)=O)C2 N1(C(COCCOCC#C)=O)CC(NC(=O)CCSC(F)(F)F)CC1(C)CC c1(C(=O)NC(CCC)CNC(=O)CC2C(=O)N(C)N=C2C)cccc2cc[nH]c12 c1(C(=O)NCC2C(NC(c3c(C)ccnc3O)=O)CCC2)cc(Cl)c([N+](=O)[O-])[nH]1 CCC(CC)CN=c1[nH]c(=NCc2cccc3[nH]ncc23)c2ncccc2[nH]1 C1(C(=O)OCC)CCN(N2CCC(c3sccc3C)CC2)CC1 C1(C(=O)NCCOc2c(C)cccc2)CC2CCC(C1)N2C(c1ccsn1)=O Cc1nn2c(C)c1C2.c1(C(CNC(=O)NCC2CCCO2)C)cnn(C)c1 C1(C(N2C(C(N(C3CC4CC4C3)C)=O)CC2)=O)(CO)CC(C)(C)C1 C(c1ccc(Cl)cc1F)=CC(=O)NC1C(CC)N(C(C2CC3(CC3)CO2)=O)CC1 C1(C(=O)Nc2cccc(C)c2)CC(C)CN(c2ncc(C)c(C)n2)C1.C1CC(=O)N1 C(CS(=O)(=O)NC(C(C(F)=CC)=O)CCNC(=O)CC#N)N C1(C(=O)NCC=CCNC(C2CC(CCO)C2)=O)CC(=C(F)F)C1 c1(C(=O)NC2CCCC(NC(C3(C)CC(C#N)C3)=O)C2)ccc(Br)nc1O N1(C(C2N(C)CC2)=O)CCN(C(C2CC3OCCCC23)=O)CC1CC(C)(C)C C1(NC(c2c(C)nns2)=O)CC(O)CN(C(=O)CC(C(F)F)n2ccnc2)C1 N1(C(CCOC(C)=O)=O)CC2ON=C(CNC(=O)CSC(F)(F)F)C2C1 CC(C)CCC(F)C(=O)NC1CCCC1CNC(C1CC(=O)C1)=O Cc1nccc(Br)c1NC(C1CC12CN(C(C1(F)CCCC1)=O)C2)=O N1(C(C(CCC)NC(c2ccc3n[nH]cc3c2)=O)=O)CCc2cnccc2C1 C#CC1CCN1C(=O)C(C)N(C(=O)C(CC)SC)CCC CC(C)S(=O)(=O)c1ccc(F)c(C(N2CC3CC3(CNC(C3CCO3)=O)C2)=O)c1 C=CC(CCC)CC(=O)N1CCC(C(C)C(=O)N(C2CCOCC2O)C)CC1 CC(C)C(C)C(CNC(=O)C(C)(C)c1ccc(Cl)s1)NC(=O)CCC(F)(F)F c1(C(=O)NCC(C2CCOC2)NC(CSC(C)C)=O)cc(Cl)c(F)cc1O N1(C(C2N(N=O)CCCC2)=O)CC(NC(=O)C=Cc2ccco2)CC2(CCC2)C1 c1(CCC(=O)NC(CNC(C2C(C=C)C2)=O)(C)CC(C)C)ccc2c(c1)OCO2 c1(C(=O)OC)ccc2c(c1)CCC2NCc1csc(C(F)(F)F)c1 C#CC1(F)CCN(C(=O)C(CC=C)NC(C2CC23CCCC3)=O)CC1 Cc1ncccc1C(C)NC(C1C2CN(C(=O)C(O)CC3CCCC3)CC12)=O C(=O)(CCCC(C)c1ccccc1)N(C(C1CN(C(CN2C(C)CC2)=O)C1)C)C(C)C CN1CC(C)(NC(C2C=CCN(C(=O)CC3(O)CCCOC3)C2)=O)CCC1=O c12ccc3cc(oc3c1)-c1cccc(c1F)CNC2=O.c1(OC(C)=O)ncccn1 N1(C(CSCC=C)=O)CCCC(n2cc(CNC(=O)C=CC3CCOC3)nn2)C1 N1(C(c2cc(CC)nn2C)=O)CCC(C)C(CNC(c2cc(F)cnc2Cl)=O)C1 C(CCCOC)(C(=O)N1CCC(CO)C1)NC(c1cc(CC)on1)=O C1(C(N2CC(CC(C)NC(=O)CC3CC3C)C2)=O)C=CCCC1 c1(C(N2C(CNC(c3ccc(CO)o3)=O)COCC2)=O)[nH]nc2ncccc12 N1(C(=O)NCC2C(C)(C)C(O)C2)CCC12CC(O)C2 CC1=C(C(=O)N2CCN(C(=O)CP(C)(C)=O)CC(C)C2)C(=O)OC1(C)C N1(C(C=CSC)=O)CCN(C(=O)Cc2ccnc(C(N)=O)c2)CC2CCCCC12 C(=O)(C1CCc2nccn21)N(C(CN(C(C1CCC(C#C)CC1)=O)C)C)C c1(CC)ccc(C(N2CC3CC2C3C(N2CCOCC2CC)=O)=O)cn1 C(=O)(C(C(C)(C)C)c1ccccc1)NC1(CF)CCN(C(C2C(C(C)O)C2)=O)C1 c1(C(=O)NCC(CNC(c2nccc(C#C)c2)=O)F)cc2ccccc2nc1O Cc1c(Br)ccc(CNC(=O)Cc2ccc(Cl)cc2C(F)F)c1F C1(C(=O)NC2CCC(n3cc(CCC4CC4)nn3)C2)C2CCCCC12 C1(NC(C2(C)CCCC2)=O)CC2CN(C(=O)Cc3cc(Cl)cc(Cl)c3)CC2C1 CCC(CC)C=CC(=O)NCC(CNC(=O)CC1OCCCO1)CO N#Cc1ccccc1CC(=O)NC1CN(C(=O)Cc2ccc(F)nc2)CC1F c1(OC)c(C(C)NC(c2nc(C(F)(F)F)no2)C)cccc1Cl Cc1cc(C)cc(S(=O)(=O)N2CC(N(C)C(c3n[nH]cc3I)=O)C2)c1 C1(CC)C(NC(=O)Cc2ccn(C)n2)CCCN1C(C1C2CCC(=O)C12)=O c1(C(=O)NCC23N(c4cc(C)nc(CO)n4)CC(C2)C3)cnc2[nH]cnc2c1 CC(C)(C)CC(C(=O)NC1(CO)CCCC1)Nc1cn(-c2ncccc2Cl)nn1 N1(CC(=O)NCC(CO)NC(C(=Cc2ccncc2)C)=O)C(=O)C(=O)N(C)C1=O N1(C(C)=O)CCN(C(=O)Cc2cc(Cl)cs2)C2C1C2(F)F c1(OC)cccc(CC(N2CCCC2C(N2CCCC(Br)C2)=O)=O)c1 CCCC(C(O)C(=O)NCC1CC1c1ccoc1)NC(c1c[nH]cc1C1CC1)=O c1(C(C(=O)NC(CC(C)NC(=O)CN=S(C)(C)=O)C)C)c(Cl)cccc1Cl C(=O)(CS(=O)(=O)C1CC1)NC(C)CCN(C)C(c1ccnn1CC1CCC1)=O C1(C(N(CCCNC(=O)C(C)(C)c2cnc[nH]2)C(C)C)=O)CCCCN(C)C1=O N#CC1Cc2cccc(C(=O)NCC(O)CNC(c3csc(C(F)(F)F)n3)=O)c21 C1(CNC(COCCCCC)=O)CCN(C(C2(N(C)C)CC2)=O)CC1O c1(OC)ccc(C(N2CC(O)CC2CC(=O)C(n2ccnc2C)C)=O)c(C)c1 C1(C(=O)OCCN(C)C(C2CC2)=O)CCCCCCN1C(=O)CN(CC(C)(C)C)C c1(OC)ccnc(-c2nc(-c3c[nH]nc3F)n(Cc3cccs3)n2)c1 n1(CC(=O)NC2C(NC(CCc3c(C)ncs3)=O)CC2)ccc(O)nc1=O C(=O)(C1=CCCCC1C)NC(c1ccccc1OC)CNC(CCOC)=O CCC1=NOC(CC(=O)N(CCCNC(c2cncc(C)n2)=O)CCO)C1 c1(C(N2CCN(C(C#CC)=O)CC2)C(=O)N(C)C)nccc(OC)c1OC N1(C(c2ccc(CCC)[nH]2)=O)CCCCC(CNC(c2ccsn2)=O)CC1 Cc1cc(=NCC2CCC(F)(F)CC2)[nH]cc1S(=O)(=O)NC1CN(C)CCC1C C1(C(=O)NC(CNC(C(N2CCC(C)CC2)=O)=O)C)CCCC(=O)N1C C1(CNC(C2CN(C(C)C)C2)=O)CC2(CO1)CN(C(c1cc(Cl)ccc1N)=O)C2 C1(NC(C(=Cc2ccco2)C)=O)CCCC2CN(C(=O)Cc3ccco3)CC12 C1(NC(c2ccn(CCCC)n2)=O)CCC(NC(=O)Cc2ccsc2C)CC1 C1(CNC(c2cc(CC)sn2)=O)CCN(C(c2cccn(C)c2=O)=O)CC1O Cc1ccc(CC(=O)NCCC2CCN(C(C3CN(C(C)C)C3)=O)C2)cc1 n1(CC)ncc(C(=O)NCCC(C)N(C)C(c2cnn(C)n2)=O)c1C(F)(F)F CC1(C)CC(C(=O)N2CCN(C(=O)CC3CCCNC(=O)C3)CC(O)C2)=NO1 N1(C(c2cc(SC)oc2C)=O)CCN(C(c2cnoc2C)=O)C(C)CC1C c1(NCC(CC)N(C)C)cc(Br)ccc1S(=O)(=O)NCC(CO)C1CC1 c1(C(N2CCOCC(CNC(COCC=C)=O)C2)=O)cnc2cc(O)ccc2c1 c1(-n2c(C3CN(C)CC3O)nc(-c3cccnc3)n2)ccc(F)cc1F Cc1cc2ccccc2n1CC(=O)NCC1CC(C)(C)CN1C(=O)CP(C)(C)=O C1(C(C2CN(C(=O)CC(C)N(C)C)CCO2)C)CCS(=O)(=O)CC1 Cn1cc2c(n1)CCN(C(=O)CC1CCN(Cc3cc(Br)c(F)cc3Cl)CC1)C2 c1(OC)cc(OC)nc(N(CCCCN(C)C(c2cccc(Cl)c2C)=O)C)n1 C1(C#CC(=O)NC(C(COC)(F)C(C)C)=O)(C(CC(O)C2CCC2)=O)COC1 C=CCC(C(=O)N1CC(O)(C(F)C(=O)NCCc2ccnn2C)C1)NC(C)=O N1(CC)CCOC(CC(N)=O)C1.C12CC(O)C1CC(=O)N2.C=CCC=O c1(C(N2C(CN(C)C(C3COC4(CCC4)C3)=O)CCC2)=O)cc(N)c(F)cc1F C1(CC(=O)NCCC(=O)NC(C)C)CCCCC1NC(=O)CCC1CCCC1 c1(CCNC(=O)C(CC(C)C)OC(F)(F)F)cccc2c(C)c(C(=O)OC)oc12 c1(C(=O)NCC2CC(F)(CNC(CCCCC)=O)C2)cc2c(cc1Cl)OCCO2 C(C1OCc2ccccc21)N(C)C(CC(c1ccc(F)cc1Cl)(F)F)=O CC1=C(C)CC(C)(NC(C2CCC(O)CN2C(=O)Cc2cccc(C)c2)=O)CC1 N1(C(c2cc(C(C)=O)sc2)=O)CCC(O)(C2CCN(C(C3CC34CC4)=O)CC2)C1 C1(NC(=O)CCN(C2CCCC2)C2CC2)(CF)CCN(C(c2cc[nH]c2)=O)C1 N1(C(CN(CCC)C)=O)CCN(C(c2cn(-c3cccc(C)c3)nn2)=O)CC1C C1(NC(CCc2ccn(C)n2)=O)CCCCN(C(C2CC3CC2C2CC32)=O)C1 c1(NC(=O)NC(C)C(F)F)cccc(CC(=O)NCCNC2CCCC2)c1 CCCC(CNC(=O)COC1CCN(C(c2cc(CC)no2)=O)C1)CCO C1(C(=O)NC2C(NC(=O)Cc3ccnc(F)c3F)CCC2)CCc2ncsc2C1 C1(NC(c2c(C)csc2)=O)CCOCC1NC(=O)Cc1cc(-c2ccco2)on1 C(=O)(C1=CCCOCC1)NCc1ccc(C(N2CC(C)C(C)C2C)=O)o1 C12(CNC(C(CC)F)=O)CCCCC1N(C(=O)CC1(OC)CCCC1)CC2 C1(NC(C2C(C)(C)C2)=O)COC2(C1)CN(C(=O)Cn1nc3c(n1)CCCC3)C2 N1(C(c2nccc(OC)c2)=O)CCN(C(=O)C(C)(C)c2ccns2)CC1C C1(C(N2CC3C(NC(=O)C4CC4)C(COC3)C2)=O)COc2ccc(O)cc2O1 N1(C(C(=O)NC2(C)CC2)c2ccsn2)CCCC(CON)C1.N(C)C C1(C(C)NC(=O)CCOCc2ccccc2)CCCN(C(c2cc(Cl)on2)=O)C1 CCC(CC(=O)N1CCC(C(=O)N(C)Cc2nc(C)no2)CC1(C)C)C(C)(C)C CCC(C)(F)C(=O)NCC1CC(NC(c2ccoc2C(C)C)=O)CC1O Cc1cc(Cl)c(Cl)cc1C(=O)NC1CC1CNC(=O)C(C)Cc1ccc(F)cc1 C1(C(=O)NC2C3CN(C(C(C=C)(F)F)=O)C2C3)Cc2ccc(OC)nc2C1 C(=O)(C1=C(CC)OCCC1)OCC(C)CNC(=O)C(CC1CCCC1)NCC C1(CNC(C=C(C)C(C)(C)C)=O)CN(C(C2(F)CCCOC2)=O)CC1O C1(CC(=O)NC2C(CNC(CC(=C)C)=O)C2)=CC=CC=CC=C1 CC1(C)CC(NC(c2ccncc2C(F)F)=O)CN1C(c1cnn2ccsc12)=O C1(OC)CC2CCC1N(C(C1(COC)CN(C(c3cc(C#N)oc3C)=O)C1)=O)C2 CC1CCOC2(CCN(Cc3ccc(-c4cc(Br)nc(Br)c4)s3)CC2)C1 N1(C(CNC(=O)C(F)F)=O)CC=CCC2(CCCC2)C1 S(=O)(=O)(c1ccc(NCCC2CC(C)(C)C2)cc1Br)NC1CCN(C)C1 C(C(CC(F)F)C(=O)NCCOc1ccon1)NC(=O)OC(C)(C)C C1(O)(N(C)CCC2CCN(C3CCC3)C2)CCNCC1 N1(C(CCC#C)=O)CC(C)(C)OCC1CNC(C1(OC)CCCSC1)=O N1(C(c2cc(OCC)no2)=O)CCC(C)C1CNC(=O)CC1CCCSC1 Cc1[nH]c(C(=O)NCC2CN(C(C3OCC4CCCCC34)=O)C2)c(C)c1[N+](=O)[O-] CCCC(CC)C(=O)N1CCC(CNC(=O)C(COC(C)C)NC(C)=O)(CC)C1 c1(COC(=O)CCc2nncs2)c[nH]c(=O)cn1.c12ccc(o1)C(=O)NC2 C1(NC(C2CCOC2)=O)CCCCN(C(c2cn3ccsc3n2)=O)C1 c1(C(N(CC(=O)OCC)CC2CNC(=O)C2)=O)ccncc1Cl C1(CCOC)CCCC1NC(=O)COC1CN(C(C2CN(C(C)C)C2)=O)C1 C1(CC(=O)N(C2CCC2)CC#C)CN(CCC(=O)CC2CCOC2)CC1C C1(OCC=C)CCCN(C(=O)NC(c2ccccc2F)C2CC2)C1 C(=O)(C1CCCc2nn[nH]c21)NCC1CC(NC(=O)C=CC2CCCC2)C1 C1(C(=O)NC(C(C)(C)OC)C)C(C)OCCN1C(c1cncc(Cl)c1)=O C(=O)(CC(C)(C)CC(=O)OC)NC1CN(C(C=CC)=O)C2(C1)CCC2 C1(CNC(=O)CCc2nc[nH]n2)CC2CCC1N2C(C1(C2CCCCO2)CC1)=O C1(C(=O)NCC2CCNC(=O)C2)CC2CC1CN(C(C1CC1c1ccsc1)=O)C2 C=C(C)CC(C)C(=O)NCC(C)(C)OCCNC(C12CC(F)(C1)C2)=O c1(C(=O)NC(CCNC(c2cncc(OCC)c2)=O)C)cnc(O)c(Br)c1 c1(-c2n(C(COCC)C)nc(C(C)O)n2)ccc(S(=O)(=O)CCO)cc1 C(=O)(C1CNC(=O)c2ccccc21)NC(CCOC)CNC(=O)CCSC N1(CCNC(=O)OC(C)(C)C)CCC(C(=O)NCC2CCC2F)CC1 c1(C(=O)NC(CCNC(c2c(C)onc2O)=O)C)ccc2cc(C#N)ccc2c1 c1(CN2CC(OC)CC(C(=O)OC)C2)ccc2c(c1)C(=O)N(C)C2 C1(CC)CN(C(c2ccon2)=O)CCC1NC(c1n[nH]cc1C(F)(F)F)=O C12(COC)CN(C1)C2=O.c1(C(=O)NCC2CN(C3CC3)C2)cc(C)c[nH]1 O=C(CCCC(=O)C1CC1)NCC1CN(C(C2OCCC2C2CC2)=O)CC1O c1(C(=O)NCC2C(CNC(C3OCCN(CC)C3)=O)C2)nnn2c1CCCC2 N1(C(CCC=CC)=O)CC(CCNC(=O)COCC(C)C)OC(C)C1 CC1CC(NC(=O)CCc2cnn[nH]2)CN(C(C2(C(N)=O)CC2)=O)C1 C(=O)(CC(C)C(F)F)NCC(C(C)C)NC(CC1CCC(OCCC)CC1)=O C(CC(=O)NNC(=O)NCSCCOCC)(C(C)(C)C)NCC1(n2ccnn2)CC1 C1(C(N(CCCn2cccn2)C)=O)CCCN(C(C23CC(C#N)(C2)C3)=O)CC1 Cc1c(O)ccc(C(=O)NCCNS(C)(=O)=O)c1C.N12CCCC(O)(C1)NCC2 C(=O)(C(C)(C)CCC)NCC(CCCC)NC(c1ccc(C)nn1)=O CCC(CCCO)NC(=O)CC1CCCN(C(=O)C=Cc2ccc(C)o2)C1 C1(CC(N2C(CN(C(c3c(C)cco3)=O)C3CC3)CCC2)=O)CCCCCO1 C1(CNC(C2C(CCOC)C2)=O)CC2CCC1N2C(=O)CSc1ccccc1C N1(C(C(CCC)NC(N)=O)=O)C2CCC1CC(F)(NC(=O)CC(C)(F)F)C2 c1(NC(CC2OCCN(Cc3cc(C)nc(C)c3)C2)=O)cnc2[nH]ncc2c1 CCC(C)C(CNC(=O)CCC1CCCN(C(c2nn(C)cc2Cl)=O)C1)CO N1(C(C2(OC)CCC2)=O)CCC(C2CC2)(NC(=O)Cc2nocc2C)C1 c1(C(=O)NC2CCCC(N(C(=O)C=CBr)C)C2)cnn2ccc(O)nc12 C(c1cncn1C)=CC(=O)NC(C1(C(N2C(CC=C)CCC2)=O)CC1)C C1(NC(CNC(=O)NC)=O)CCCC(C(F)(F)F)C1 c1(C(C(=O)NC(C2CN(C(c3cnc(C)s3)=O)C2)C)C)ccccc1F c1(C(=O)NCC2CC(COC)CN2C(c2coc(OC)n2)=O)ccc(C#N)cc1 N1(C(C(=O)N)=O)CCCC2(CCCC2)CC1.CC1(c2nn[nH]n2)CCCCNC1 N1(C(=O)Cc2cccnc2Br)CC2CCC1CN2C(=O)CC1CC=CCC1 c1(C(=O)OC2CC(C(C)(C)C)C2)cccc2ncccc12 C(CNC(=O)COc1cccc(Cl)c1C)(C(C)C(C)C)NC(C(CC)=CC)=O c1(C(=O)NC2CC(NC(C(COC)C)=O)C2)cc(C)cc2c(C)ccnc12 c1(C(=O)NCC2C(NC(=O)Cc3csc(C4CC4)n3)C2)ncncc1F Cc1cc(C(N2CC(C)C(NC(C3CCOCC3)=O)C(C)C2)=O)c(N)c(F)c1 CC1(C)NC(=O)CC1C(N1CC=CC1C(=O)NC(C1CCC(=O)N1)c1cncs1)=O c1(C(=O)NC(CC)(C)CNC(c2cnn(C3CC3(F)F)c2)=O)cccc(F)c1 C1(NC(Cn2ncc(C)c2)=O)C2CC(NC(c3nc(O)sc3C)=O)CC12 Cc1cc(F)ccc1CC(=O)NC1CC(NC(=O)C(C)C2CCCC2)C1 CCCCCC(C)(CC)C(=O)NCCCC(CCC)NC(=O)C(F)(F)CN(C)C n1(C(CC)C)nccc1C(=O)NCCC(C)NC(=O)C(c1cnn(C)c1)C C1(NC(c2cc(C)n(C3CC3)c2C)=O)CC2CC1CN(C(=O)Cc1cnnn1C)C2 CCC(C)(C)C(=O)C(=O)N1CCCCC1CNC(C1(C)CCC(O)CC1)=O S(=O)(=O)(c1cnn(C)c1)CNCC(=O)NCC1C(NC(c2c(C)cncc2C)=O)C1 c1(C(N2CC3CCCN(C(C4C5COCC45)=O)C3C2)=O)ccc(Cl)c2occc12 n1(CC(=O)NC2CC(NC(c3cncc(C(N)=O)c3)=O)C2)cc(Br)ccc1=O C1(NC(CC2(C)OCCO2)=O)CCCC(CNC(C2(c3ccsc3)CC2)=O)C1 C#Cc1ccc(C(=O)N(C(C)CC(N2CCC(C(N)=O)C2C)=O)C)c(C)c1 C1(NC(=O)OC(C)(C)C)CCC2C(C1)C2(F)F.CC1(C)COC(=O)NCC1 C1(C(=O)OCC)CCC2OCCN(C(c3cc(Br)sc3I)=O)C2C1 C1(n2cc(-c3ccccn3)nn2)CN(C(=O)C(C)OC(C)=O)CC1O C1(NC(c2cc(CC)c(C)s2)=O)CCN(C(=O)CSc2ccc(C)cc2)C(C)C1 N1(C(c2c(C)n[nH]c2)=O)CCC(CNC(c2ccnnc2S)=O)CC1 N1(C(c2cc(C(N)=O)[nH]c2)=O)CC2CN(C(=O)C=Cc3cccc(F)c3)C2C1 C1(C(N2CC(C3N(C(C4(OC)CCC4)=O)CCC3)(O)C2)=O)CS(=O)(=O)CC(=O)N1 c1(C(N(CCNC(CCC(CC)C)=O)C)=O)c[nH]c2c(Br)cccc12 c1(C(C(=O)NCC(C)(C)NC(CC2CCN(C)C2)=O)CO)ccc(Cl)cc1 C1(N=c2[nH]ccnc2F)(C(N2CCCC2COC(F)(F)F)=O)CCCC1 C(C(N=[N+]=[N-])C(=O)N1CC=CC1C(=O)N(CC(C)(C)COC)C)OCC c1(C(=O)NCC(CNC(C2CC3C(C2)C3(C)C)=O)OC)c(C)cc(C)oc1=O CC#CCCC(=O)NC(C1CCCCC1)C(=O)NCC1(CC)CCC(=O)N1 C1(C(N2CCC(N(C)CC3CN(C(C4CC4)=O)C3)CC2)=O)C2C3CCC(C3)C12 C(=O)(C#CC(C)(C)C)Nc1cc(CNC(C(N2CC(N=[N+]=[N-])C2)C)=O)ncc1 C12(CNC(=O)Cc3cccc(Cl)c3)CCCC(CN1C(C1CC1CF)=O)C2 C1(CC=C)(C(=O)N(C)CCOCCNC(=O)CC2CC(C)C2)CCC1 c1(OCC)ccc(C(N2CC(NC(c3cc(C)co3)=O)CC(C)C2)=O)cc1Cl N1(C(CCCC#C)=O)CCCC(F)(CNC(C2(C)CC2(C)C)=O)CC1 N1(C(CN(CCOC)C)=O)CC2CC(C(N3CC4CCN(C)C4C3)=O)CC2C1 c1(CC(=O)NC2(CNC(C3C(=C)C3)=O)CCC2)ccc(C(C)=O)c(F)c1 C#CC(C)(C)C(=O)NC1CC2(C1)CC2NC(C1CSCC(=O)N1)=O c1(C(=O)NCC2(C(C)(C)C)CCN(C(C3C(CC)C3)=O)C2)nnc(C)cc1O CCCCC(CC(=O)Nc1cc(C)ccc1O)NC(=O)C(O)Cc1cccc(F)c1 C1(C(=O)NCC(COC)C)CC(C)CCN1C(=O)CN(C)C(=O)C1CC1 N1(C(c2ccc(C(=O)OC)s2)=O)CC2CCN(C(=O)C=C(C)Cl)CC2C1 N1(C(CC2C(C)=NNC2=O)=O)CCCC(F)(CNC(C2CCS(=O)(=O)N2)=O)CC1 c1(C(=O)NCC2CCCC(NC(C3(F)CC=CC3)=O)C2)cc(Cl)cc(Cl)c1 N1(C(CSC)=O)CCN(C(C2CCN(C3CC3)CC2)=O)CC(C)(F)C1 c1(C(=O)OC)csc(Cn2cc(CNCCO)nn2)c1.C12CC(CO1)C2 Cc1nc2ncc(C(=O)NC(CNC(C3CC(O)CN3C)=O)C(C)C)c(=O)n2[nH]1 S(=O)(=O)(c1ccncc1)N1C2CN(C(c3cc(COC)nn3C)=O)C(C2)C1 N#Cc1nc[nH]c1C(N1CCC(CNC(=O)C=CSCc2ccco2)C1)=O Cc1cc(NC(C2(CO)CCN(C(=O)CC(C)(C)C)C2)=O)cc(O)c1 C1(CNC(C2(CCCNC(C=CCCC)=O)CCC2)=O)CCCNC1=O c1(OCc2cc(C(N3CC4CCC3C4)=O)no2)ccccc1Cl c1(C(=O)NCC(CC)NC(C2CCCCC2(C)C)=O)ccc(CO)cc1F C1(NC(Cc2cnc(C)s2)=O)CCCCC1CNC(=O)COc1ccccc1F c1(C(=O)NCC(C)(C)NC(c2cc(C#N)c[nH]2)=O)c(N)cncc1Br N1(C(C(c2ccc(Cl)cc2)CC)=O)CCn2c(CS(N)(=O)=O)nnc2C1 C1(CC(N2CC(OCCOC)C2)=O)CN(C(=O)CCC=CC(C)C)CC12CC2 C1(N(C(COc2cccc(CC)c2)=O)C)CCCN(C(=O)CC(F)F)CC1 CC1=C(C(=O)NCC2CCC(C)N(C(C3CC3F)=O)C2)Cn2ncnc2N1C C1(CC)C(C(=O)NCCN2CC3CC3C2)CCCN1C(C1CCN1C)=O c1(NC(C(=O)NCCc2c(C)cc(Br)c(F)c2)=O)cc2n(n1)CC1(CC1)C2 C(c1cc(OC)c2c(c1)OCCO2)=CC(N1C(CNC(C(CC)(C)O)=O)CC1)=O N1(C(COCc2cc(C)[nH]n2)=O)CCCC(CCC(=O)NC(C)C(F)(F)F)C1 O=C(C1=C(Cl)CCOC1)NC1CCCC1CNC(c1ccoc1Br)=O S(=O)(=O)(c1cccc(Br)n1)NS(CCOCC)(=O)=O.C12CN(C1)C(=O)OC2 C12CCC(CC1)C(=O)N2.N1(C(CC)=O)CCC(NC(c2ccc(O)nn2)=O)CC1 C1(OC)C2CCC1CN(C(C1(CCNC(=O)CC3CC(C)=NO3)CC1)=O)C2 Cc1cnc(N)c(C(=O)NCC2(F)CCC(CNC(C3CN(C)C(=O)N3)=O)C2)c1 C1(NC(C=C(C)C(C)C)=O)CC2CN(C(C3(C)CC3)=O)CCN2C1=O c1(C(=O)NC(CC)CNC(=O)C(CCO)N(C)C)cc2ccc(F)cc2nc1C c1(C(=O)NC(CCCC)CNC(=O)CCCCC(F)F)cc2c(cc1C)OCO2 N1(C(C2C(COC)C2)=O)CCCC(NC(=O)Cc2ccc(CSC)cc2)C1C c1(CC(=O)OCC2CCCO2)cn(CC2CCCCO2)nn1 C1(COC)CCCCN1C(=O)C(=O)NC1CC(=O)N(C(c2ccc(N)cn2)C)C1 c1(N2CCOCC(OC)C2)nc2c(c(=NC3C4COCC34)[nH]1)CCC2 O(NC(=O)CC(C)(O)COC)CC(=O)NC(CC=C)(C)C c12cc(F)ccc1C(=O)N1CC(C)(C1)c1cn-2nn1.C1(C(=O)O)(COC)CC1 c1(N2CC(C(C)NC(C3CCC=CCC3)=O)OCC2)cc2nncn2cn1 CN=c1nc(C(=O)NCCC2CC(NC(c3cc(=O)cc(Cl)[nH]3)=O)C2)cc(C)[nH]1 N1(S(CCCC)(=O)=O)CCC(C(F)(F)F)C(F)(F)C1 C1(C)(C(=O)NC2CCC(F)(CNC(C(C)=C3CC3)=O)C2)CCC(C)C1(C)C CCCCC(C(=O)N1CCC(C)C(NC(C2C(OCC)C2C)=O)C1)C(C)C CC(C)(C)CC(F)C(=O)NC(CCNC(=O)CN1CCCCC1=O)C(C)(C)C c1(C(N(C(CNC(CCCOCC)=O)C2CC2)C)=O)cc2ccc(Cl)cn2c1 Cc1[nH]nc(C(=O)NCCn2cnc(C(=O)NC(C)C(C)F)c2)c1C C#CCCCOCC(=O)NC(CNC(C1(C2CCCO2)CCC1)=O)CO N1(C(C2C=C(C)CS2)=O)CCC(NC(=O)CC2CCC=CCC2)C(O)C1 CCC(C)CCCCC(=O)N1CCC(n2cc(CCCC(C)=O)nn2)C1 C1(CNC(C(C)OCC#C)=O)CC(C(C)(C)C)CCN1C(c1nc(=N)cc[nH]1)=O N1(C(CC=C)=O)CCc2sccc2C1CNC(c1cc(S(C)(=O)=O)co1)=O C1(CC(=O)NCCc2ccc[nH]2)CCCCN1C(c1nc[nH]n1)=O CC(C)CC(O)C(=O)NC(C)(CNC(=O)COC(c1cccnc1)N)C1CCC1.C(C#N)O CCC(C)CCCC(=O)N(C1(CC(=O)NCc2cnc(OC)c(C)c2)CC1)C c1(-c2cccc(N(CC#C)C(C(C)C#N)=O)c2)cc(C(F)(F)F)ccc1C(F)(F)F c1(OC(C)C(=O)NCCCNC(c2coc(C(F)F)c2)=O)cccc(F)c1 Cc1cnc(C(=O)NCCCC(CO)NC(=O)CC2CSCCO2)c(F)c1 c1(COC(C)C)cccc(NC(c2ccc(CO)cn2)=O)n1.C(CO)SCC1CC1 c1(C(=O)NC23CN(C(CSCC=C)=O)C(CC2)C3)cn2c(n1)CCCC2 Cc1c[nH]c2ncc(C(N3CC=CC3CNC(c3ccc(Cl)o3)=O)=O)cc12 C1(C#N)(C(N2CC(CNC(C(c3ccccc3)C)=O)OCC2)=O)CCCOC1 C1(NC(C(C)(C)SC)=O)CC2CC(NC(C3(C)COCCO3)=O)CC2C1 CC(C(=O)NCC(C1CCCCN1C(=O)COCC1CCC1)(C)C)C(F)(F)F N1(c2cccc(C(=O)OC(C)(C)C)n2)CCN(C2CCNC2=O)CC1C C12(C(=O)O)CCC(CC1)N(C(C1CC3(CCC3)C1)=O)C2 N1(C(C(c2ccoc2)NC(c2c(CC)cc[nH]2)=O)=O)CCNC(=O)C1 c1(OC)ccc(C(N2CC3CN(C(c4cn(C(C)(C)C)nn4)=O)C3C2)=O)c(Cl)c1 O=C(CCCC(F)(F)CO)NCCC1CN(C(C2CC3CCCCN3C2)=O)C1 C1(CCC)(NC(=O)CCc2ccccc2C)CCCN(C(c2nnc(C)s2)=O)C1 N1(C(c2n(C)ncc2Cl)=O)CC2COCCC2(NC(C2CCC23CCC3)=O)C1 C(=O)(CS(=O)(=O)Cc1cccs1)N1C(CNC(C(CC)COC)=O)CCCC1 c1(-c2c(C(N3CC(C=C)C(O)C3)=O)cccn2)nccn2nccc12 c1(C(c2nc(C3CC34CC4)nn2CC(F)(F)F)(C)C)cccc(C#N)c1 C#CC1(C(=O)NCC(O)CC)CN(C(C2CCC(=O)C2)=O)C1 C1(NC(C(C)c2ccco2)=O)CC=C(C(=O)NCc2cccc(C#N)c2)C1 N1(C(Cc2n(C)cnn2)=O)CCC(CNC(=O)CC2(C)OCCO2)CC1 C(C)(N=c1[nH]c2cc(Br)ccc2o1)C1N(C(C2C(OC)CCC2)=O)CCCC1 C#Cc1cc(C(c2nnnn2C2(C)CC2)NC2(C)CCOC2=O)cc(COC)c1 N1(C(CC2C(C)CCC2)=O)CCC(C)(CN(CCC#N)C=O)C1.C1(C)CC1 C1(CCOC)CCCN(C(C(=O)NC2CC2)C2CC2(C)Br)C1 C=CC1CCCC(NC(=O)CCCCN(C(=O)C(c2ccn(C)c2)C)C)C1 c1(C(=O)NC(C)CCNC(C2CC3CCC2O3)=O)ccc2c(c1)CC(=O)N2 Cn1oc(C(N2CCN(CC3CN(C(=O)C#CC4CC4)C3)CC2)=O)cc1=O c1(C(=O)NCCN(C(C2CCN(OC)CC2)=O)CC)cc2cnccc2o1 C1(F)(CNC(C2N=C(C)SC2)=O)CCN(C(=O)CC(C)n2ccnc2)CC1 S(=O)(=O)(CCC(=O)N1CCN(C(c2ccc(-c3cnccn3)s2)=O)CC1C)NC O=C(CCCc1ccsc1)NCCN(C(=O)C(O)C1CCCC1)CCOCCO c1(C(N2CC3C(NC(c4cn(C5CC5)nn4)=O)(C3)C2)=O)ccc([N+](=O)[O-])[nH]1 S(=O)(=O)(c1ccc(NC(C2CC(=O)NC(=O)N2)=O)cc1)N(CCCC)C N1(C(C(C)N(C)C)=O)CC(NC(=O)C(C)Sc2ncccn2)C(C)C1 C1(NC(C(CC)n2cccn2)=O)CC2C1CCN2C(c1csc(C2CC2)n1)=O C(C(C)CC(=O)NC1(C)CCC(C)C1)NC(C1(CC=C)CCC1)=O c1(C(N(CCCC(=O)NCCC(C)N(C)C)C)=O)cc(C#N)cs1 c1(C(N(CC(C)O)CCNC(CCNC(C)=O)=O)=O)[nH]c2c(Cl)cccc2c1C CC1(C)OCCC1CC(N1CCCC1CC(N1CC2CC1CO2)=O)=O NS(=O)(=O)N1CC(C(=O)NC2(CO)CCCN(C(=O)CN3CCCNC3=O)C2)C1 c1(C(N(C(C(C)NC(c2ccco2)=O)=O)C2CC2)C)cccnc1 C(=O)(CC1OCCc2sccc21)NCCC1(NC(C2OCC(C)(C)C2)=O)CCC1 C1(NC(C2CCN(C(c3cn(CCC)nc3)=O)C2C)=O)CC2CCC(C1)C2O C1(N(C(=O)CNS(C)(=O)=O)C)CN(C(c2coc(CS(C)(=O)=O)n2)=O)CC12CC2 C1(C)(CC(=O)N(CCN(C(C(c2ccc(OC)cc2)O)=O)C)C)CCS(=O)(=O)N1 N1(C(CCOCCOC)=O)CC(C)C(C)(C(N2CC(N(C)C)C2)=O)C1 N1(C(C(CCC)F)=O)CCC2CN(C(c3cnc(C)o3)=O)CC12 C1(C(C)NC(c2nc(COC)oc2)=O)CCCN(C(=O)C(C)NC(N)=O)C1 C=CC(C)CC(=O)N(C1CCN(C(=O)C=C2CCC(C(C)(C)C)CC2)C1)C C(=O)(CCCCN(C)C(C12CC(C#N)(C1)C2)=O)NC(C)Cc1nccn1C CCCC(CCCO)C(=O)NCc1cccc(SC(F)(F)F)c1 C(=O)(C(C(C)C)NC(=O)C(C(C)C)NC(=O)CN)NCCCOCCCC C=CCC(CNC(c1ccc(C)n1C)=O)C(=O)Nc1cncc(NC)c1 c1(C(=O)NCCC(=O)N2CCC2C(=O)Nc2ccco2)cc(F)c(Br)c(F)c1 N1(C(c2c(CC)nn(C)c2)=O)CC2CCC(C1)C2CNC(c1cncc(C)c1)=O C(=O)(CCCCCCSC)NC1C(CNC(C2N(C(=O)NC)CCC2)=O)CCC1 c1(C(N2CC(COC)N(C(c3ncccc3C)=O)CC2)=O)cc(O)cc(N)c1C c1(C(N2C(C(CNC(C=C(C)C)=O)(C)C)CCC2)=O)cc2cc(C)c(Cl)cc2[nH]1 Cc1cc(CCC(=O)NC2(CCNC(=O)C(C)CO)CCCC2)n(C)n1 c1(C(N2C(CNC(CC(CC)SC)=O)C=CC2)=O)ccc(N)c(OC(F)(F)F)c1 Cc1csc(C(N2CCCC2C(C)NC(C2(CCN3CCCC3)CC2)=O)=O)c1 c1(N(C)C)ncccc1OCC(N)=O.C12CC(O)C1CC(=O)NOC2 C12(C(N3C(C)(CNC(=O)CCC4NC(=O)NC4=O)CCC3)=O)CCCC(CO1)C2 C12Cc3ccccc3N(C1)C(=O)N2C(C)(C)C.Cc1cncc(NC2=NCCS2)c1 N1(C(c2scc(OC)c2)=O)CCN(C)CC1C(=O)NCc1cnn(C)c1O c1(C(=O)NC2CN(C(CC3CC(=C)C3)=O)C2)cc(Br)cc(F)c1F c1(C(C(C)C)=O)ccc(NC(C2(c3ccccc3)CCOC2)=O)cc1 c1(C(=O)NCC(C)NC(=O)CC2(C)CC2(F)Cl)ccc2[nH]ccc2n1 c1(C(N(CC(CC)NC(=O)CCCNC(=O)C2CC2)C)=O)ccc(C)c(C)c1F Cc1ccc(C=CC(=O)NC2C=CC(CNC(=O)CC3CC4(CCC4)C3)C2)cn1 N1(C(c2cccc(C(=O)OC)n2)=O)CC2CCC(CNC(=O)CC3CSC3)C2C1 c1(C(=O)NCCC2(CNC(=O)CC3CSCCS3)CC2)ccc2cccnc2n1 C1(C2(O)CN(C(C3CC(F)(F)C3(F)F)=O)C2)(CNC(C(CC)C)=O)CC1 C1(C(C)NC(c2c(C(C)C)c[nH]n2)=O)CN(C(c2cncn2C)=O)CCO1 Cc1nn(CC(N2CCC(C3CCCCN3C(=O)CC3OCCO3)C2)=O)c(=O)o1 C1(NC(C(CCC)C)=O)CCN(C(c2coc(CC)n2)=O)CC1c1ccccc1 C1(C(=O)NCC#C)CCCN(CC(CC)=CCCC)CC1 c1(-c2cn(C3CN(C(=O)Cc4cnoc4)CC3O)nn2)ccc2ccccc2c1 C1(CNC(=O)Nc2cnc(C(F)(F)F)cn2)CC12CCSCC2 C1(C(N(C2CCN(C(=O)OC(C)(C)C)C2)C)=O)CCCOC1.C12CN(C1)C2=O C1(CC(=O)NC(CCOC)COC)CN(C(=O)C(C(C)C)NC=O)CCO1 C(=O)(CCCCCCNC(=O)COCc1nc[nH]n1)N(c1cscn1)C CC(C)(O)C#CC(=O)NCC1CC2CCC1N2C(C1CSCCS1)=O C(=O)(C1=CCCCO1)NCC(C1CCCCC1)NC(c1cc(C(C)(C)C)no1)=O N1(C(C(C)OCOC)=O)CC(O)(C(C)NC(c2ccc(C3CCCCC3)o2)=O)C1 c1(OC)ccsc1C(=O)NC(C)(CNC(=O)C(C)C1(O)CCC1)C1CCC1 c1(CCNC23C(C)(C)OCC2C3)ccc(Cl)c([N+](=O)[O-])c1 c1(C(N(CC(C)NC(=O)C(C)(C)CO)CC)=O)ncnc2c1ccn2C1CC1 CCCCC(O)C(=O)N(CCNC(C1CC(O)C1)=O)CC C(=O)(C(CCOCCC)NC(C12CC(CO)(C1)C2)=O)N1CC(O)(CC=C)C1 c1(C(=O)NCC(C)NC(c2cc(Br)cnc2O)=O)cc2[nH]ccc2s1 C1(C(N2CCC(C)C2)=O)C2CC1N(C(=O)CCOCC1CCC1)C2 c1(C(=O)OC)ccc2c(c1)nc(N1CCC(C(=O)OC)CC1(C)C)n2C Cc1ccc(SCC(N2CC(F)CC2CNC(C2C3CCCC23)=O)=O)cc1C C1(C)(CNC(C2(OCC)CCC2)=O)CCC(NC(=O)Cn2cnnc2O)C1 N1(C(COC(C)(C)C)=O)CC2(CC2)CC1CNC(=O)C(O)Cc1ccccc1 CC1(C)C=C(C(=O)NC23CC(CNC(c4ccccc4C(F)F)=O)(OCC2)C3)C1 c1(C(=O)NCCOCCCNC(C2(C)CC3CCC2C3)=O)ccc2cnoc2c1 c1(C(C(F)(F)F)NC(=O)NC2CCC3(CC2)CNC3)ccc2ccccc2c1 c1(C(=O)NCC2C(NC(c3n(C)nnc3)=O)C2)cnc2sccc2c1 N1(C(COCC(=O)NC)=O)CCN(C(=O)CCCSc2ccccc2)C2CC12 N1(C(CC(C=C)CCC)=O)CCCCC2(CCN(CC(=O)NCCC)C2)C1 C1(CN(C(=O)CCN2CCCS2(=O)=O)C)CCCCN1C(=O)CC1CSCCS1 CC(C)(C)C(CNC(=O)CC1(O)CCC1)C(=O)N1CC2C=CC2C1 c1(C(=O)NC(C)CN(C(=O)CSC2CCOC2=O)CC)cnnc2ccccc12 c1(C(=O)NCC2(NC(c3ccc(C)nn3)=O)CCCC2)ccccc1P(C)(C)=O c1(CCCNC(=O)NCC2(CC)CCC(=O)N2)nc2c(C)cccc2o1 c1(C(=O)NCC(CC=C)NC(C2CC(O)CN2C(C)=O)=O)c[nH]c2cnccc12 c1(C(N2C(CNC(C3CC(F)C3)=O)CC(F)C2)=O)cccc2occc12 C(C(C)(C)CO)N(CCC)C(C1CCC(n2cc(-c3ccn(C)n3)nn2)C1)=O N1(C(C(CC)N(C)C)=O)CCC(C2OCCCC2NC(C2COC(=O)O2)=O)CC1 Cc1cc(N)c(C(=O)NCC(C)NC(c2nnc(O)nc2O)=O)cc1C C1(C(=O)NCC2(CC=C)CN(C(c3c(SC)cnn3C)=O)C2)CC2CCC1CC2 O=C(C1=CC2(CCOC2)C1)NC1CC1CNC(C12CCC(O)(CC1)CC2)=O c1(NC(C2(F)CC(N)C2)=O)ccc(N(C)C)c(C(N)=O)c1 CCC(CNC(c1cc(O)ncc1F)=O)(CC)C(=O)N(C1CCOC1)CCO c1(C(=O)NCC(CCC)NC(c2ccoc2)=O)ccc(CC)nc1C Cc1ccc(I)cc1C(N1CC(NC(=O)Cc2cccnc2C)C(C)C1)=O N1(C(c2c(C)cncc2)=O)CCCC(F)(CNC(c2cn(C)nc2C(C)C)=O)C1 N=c1[nH]nc(Cl)cc1C(N1CC(F)CC1CNC(c1cc(C(N)=O)[nH]n1)=O)=O c1(C(=O)NC(C2CCCN2C(=O)CC2CCC(=O)O2)C)csc(-c2nc[nH]n2)n1 c1(C(=O)NC)cccnc1NC(C1CCCN(Cc2cc(C)n(C)n2)C1)=O C1(NC(c2cc(=N)[nH]cc2)=O)CCCC2CN(C(c3ccc(Cl)[nH]3)=O)CC12 c1(CC)ccc(Cl)cc1CN(C)C(C1CCCN(C)C1c1ccnn1C)=O C(=O)(C1=CC2CCCC12)Nc1cccc(CNC(c2cn(C)c(Br)c2)=O)c1 N1(C(c2cn(CC)nn2)=O)CCC(C2CCN(C(=O)C(C)(C)c3ccns3)C2)C1 N1(C(C2(CC=C)CCCCC2)=O)CC2CCC2(CNC(=O)CCS(N)(=O)=O)C1 CC1(C)CC(C(=O)NCC(C)(O)CO)CN(C(=O)CSC(F)F)C1 C1(NC(COCCCC(C)C)=O)C2CC3C1C3C2C(=O)N(C1COC(C)C1)C1CC1 C1(O)(C(C)NC(CC2(C(=C)F)CCC2)=O)CCN(C(c2cnn(CC)c2)=O)CC1 C1(NC(C(C)(C)CCl)=O)COC2(CCN(C(=O)CNS(C)(=O)=O)C2)C1 C(=O)(C(CCC=C)NC(=O)C(F)OC(F)(F)F)NCC1(C(F)(F)F)CC(=C)C1 C1(NC(C(C)OCC=C)=O)CCN(C(=O)CCCn2ccc(C)cc2=O)CC1C C1(NC(c2ccc(OC)o2)=O)CCC2CN(C(=O)CN3CC(C)(C)C3)CC2C1 O=C1CC2(CCN1)CN(C(=O)COC(F)F)C2 C(=O)(C(CCC)C(C)C)NC1(CC=C)CN(C(=O)Cc2ccccn2)C1 c1(CN(C)CC2CCCN(C(CCc3cccc(C)n3)=O)C2)cc(Br)ncc1F c1(OC)cc(Br)ccc1C(N1CC(Cn2cc(C3CCOC3)nn2)C(CO)C1)=O CCS(=O)(=O)CC(C)N=c1[nH]c2c(c(=NCc3nnnn3C3CC3)[nH]1)CCCC2 c1(NC(C(c2cccnc2)NC(=O)OC)=O)cc(C)cn(C)c1=O N1(C(COCCC)=O)C2CCC1CN(C(=O)C(C1CCC(F)(F)CC1)OC)C2 N1(C(Cc2c(C)ncs2)=O)CC2CCN(C(=O)CCCc3cccnc3)C2C1 C(=O)(CC(CC)OC)N1CC(CNC(C2(CCC)CCCC2)=O)C1 C1(C(=O)NCC23C(CN(C(CNC(N)=O)=O)C2)C3)CCCN(S(N)(=O)=O)C1 c1(C(N2C3CC(NC(c4cc(Cl)ccc4F)=O)C2CC3)=O)cn2c(n1)COCC2 N1(C2CCCN(C(C=C(C)C(C)(C)C)=O)C2)CCN(Cc2cnsc2)CC1=O CC1SCCC1N=c1cc[nH]cc1S(=O)(=O)N(C)Cc1cccs1 N1(C(c2cc(CC)n(C)n2)=O)CC(C)N(C(=O)CC2C=NN(C)C2=O)CC1C C1(F)(C(N(CCC)CCNC(c2c[nH]nc2C(C)(C)C)=O)=O)CCOCC1 c1(C(C(=O)N(C2CCN(C(c3c(CC)[nH]cc3)=O)C2)CC)C)c(Cl)cccc1Cl c1(CC(=O)NC(CN2CCCC2)CO)cccc2c1OCCCO2 c1(C(=O)NCC2N(C(C(CCC)O)=O)CC(OC)C2)cn(CC)c2ccccc12 CC1CN(C(c2ccc[n+]([O-])c2)=O)CCCN1C(=O)Cc1ccc2c(c1)COC2 N1(C(CC(=O)OC)=O)CCC2CCN(C(C3Cc4n[nH]cc4C(=O)N3)=O)CC12 CC(=O)CCCC(C)C(=O)N1CCCC(C(C)C(N2CCS(=O)(=O)CC2)=O)C1 n1(CC(C)N(C(=O)C(C)Cc2ccccc2F)CCN)cnc2sccc2c1=O c1(C(N2CC(NC(c3ccn(C)c(=O)c3O)=O)C2)=O)nn(C)c2c1CSCC2 C1(NC(CC(C=C)CC)=O)CCC2(CC1)CC2NC(c1cc(F)cc(F)c1O)=O c1(C(N2CCN(C(C(c3cncn3C)C)=O)CC2CO)=O)cnc2c(c1)COC2 C1(CNC(=O)COCC2CCOC2)CC(F)(F)CN1C(C1CC12CCCC2)=O c1(C(=O)NCC2C(NC(COCC(=C)C)=O)CC2)ccccc1SC N1(C(c2cnco2)=O)CC2OCC(C(N3CCN(n4ccnc4O)CC3)=O)C2C1 n1(C(C)C)nccc1C(=O)NCC1CCN(C(=O)Cc2cnn(C(F)F)c2)C1 C1(CNC(c2c(CC)cccn2)=O)CC2(CCN(C(=O)C(C)(C3CC3)OC)C2)CO1 N(C(=NCC1CC1)N1CCN(c2nncs2)CC1)C=O.CC(C)CC(C)CCO C1(=O)C2=NOC(C2)CN1.c1(CSc2c(C(OC)OC)cccc2)ccnc(C)n1 Cc1ccc(C(=O)NC2CC(C)(NC(C3C(Cl)(Cl)C34CC4)=O)C2)c(Cl)c1Cl c1(N(C(C)C)C)ccccc1C(=O)NC1CN(C(=O)CC2(C)CC2(Cl)Cl)C1 Cc1nocc1CC(N1CC(NC(C2CC2c2cnn(C)c2)=O)C1)=O N1(CC)CCC(OCCOC(=O)CCc2cn(C)nn2)C1=O C1(COC)CCN(C(c2ccc(CN(CC)CC3CCCCO3)s2)=O)CC1 N1(C(C(CC)C(=O)OC)=O)CC2CC1(C(F)(F)F)C2.c12cn(nn1)C2 CC(=NO)c1cc(C(=O)NC(C)CNC(c2cccc(N)n2)=O)cnc1O c1(OCC)ccc(CC(=O)NCc2ccc(C)cc2)cc1NC(C1(OC)CC1)=O c1(C(=O)NCC2(C(=O)NCC3CC(OC)C3)CC2)cnc(N(C)C)s1 N1(C(C(CCC)c2ccccc2)=O)CCC2CC(NC(=O)C=CS(C)(=O)=O)CCC2C1 C1(C(=O)CC)CCCCC1C.C1(C(C(=O)N(CCCOC)C)O)CCOCC1 c1(-c2ccc(CNC(C(C)C3(C(N)=O)CC3)=O)o2)cc2ccccc2s1 Cc1cc(C(=O)NC2(C(=O)N(C)Cc3nc(C)cs3)CCCC2)cc(C)n1 n1(CC(=O)NCC(C)NC(=O)C(CO)C(C)(C)C)ncc2cccnc12 C(=O)(C(CC(C)C)OC)NC1(CF)CN(C(C(C)NC(COC)=O)=O)C1 c1(C(=O)OC(c2c(F)cccc2F)C2CCCCCC2)cncc2sccc12 N1(C(c2cc(C#C)cc(C)c2)=O)CC(C)Oc2cc(C)c(Br)cc21 c1(C(CC)(C)C)cn(C2CC3(C(=O)N(C4CC4)CC4CCC(=O)O4)CC23)nn1 C(=O)(C(C)(O)CCS(C)=O)N1CC(O)(CCNC(c2ccc(C)c(C)n2)=O)C1 C1(NC(=O)C(C)(C)C)CCC(NC(=O)CCC(=O)NC(C(=O)NCC)CC)CC1 n1(CC(=O)NC2C(CNC(C(COC)OC)=O)CC2)nc(C)c2cccnc12 c1(CC(=O)OCC2(C)CNC2)ccccc1NC(c1ccc(OCC#N)cc1)C c1(C(=O)NCC(C)NC(CC(c2cccs2)N(C)C)=O)cc(F)c2cn[nH]c2c1 C(C(O)CC(=O)NCCC(Cl)Cl)NC(c1c(C(C)C)cco1)=O C1(NC(c2cn(C)c(Br)c2)=O)CC2CC1N(C(C1CCC13CCC3)=O)C2 N1(C(c2c(CC)c[nH]n2)=O)CCC(C2CCN(C(=O)Cn3ncnn3)C2)C1 c1(C(=O)NCC(C)=CC(=O)NCc2ncnn2C2CC2)oc(C)cc1C Cc1cc(C(=O)NCC2CC2NC(c2ccnn2C(C)C)=O)cnc1OC(F)F N1(C(=O)NC2(C)CCCO2)CCOC(CC(=O)NCCCNC(=O)C(F)(F)F)C1 CC1(CNC(=O)CC2CC2)CCN(C(C2CC2OC(C)(C)C)=O)CC1 C1(C(C)O)C(C2CC2)CCN1C(=O)COC(=O)NCc1cccc(C2CC2)c1 C#Cc1ccc(C2CC2C(=O)NC(CCNC(C2CC3(CCC3)C2)=O)C(C)C)cc1 N1(C(c2onc(CC)n2)=O)CCC(C)C1CNC(c1cnns1)=O CCCS(=O)(=O)C(C)C(=O)N(CCCNC(c1cnnn1-c1ccccc1)=O)C N1(C(CC2CC(=C)C2)=O)CCN(C(c2oc(C)nc2C)=O)CC1 Cc1ccc(NS(=O)(=O)CC(C)c2ccccc2)c(Cl)n1 c1(C(N2CCC(N)(CC)C2)=O)cccc2c1OC(C)(C)C2 c1(CCNC(CN(CCC)C(=O)N)=O)ccc(OCc2ccnn2C)c(N)c1 N1(C(C2C(C(N)=O)C2)=O)CCN(C(c2csc3nnsc23)=O)CC(O)C1 C1(CC)C(C(=O)NC(CCO)C(C)C)CCN1C(=O)C(F)=CC1CC1 C=CC1(C(=O)NC(CNC(c2c(F)cccc2Cl)=O)CC(C)C)CCOCC1 C(=O)(CCCCC(F)(F)F)N1CCC(N(C(=O)C(C(C)O)NC(C)=O)CC)CC1 C(CCN=C(NCC(c1cccc(F)c1F)(F)F)NCC1CCCS1)OCC N1(C(CCc2ccn(C)n2)=O)CC=C(CCNC(C2C3CCCCCC23)=O)CC1 c1(C(N2CCC(CNC(CNC(CN(C)C)=O)=O)C2)=O)cnn2ccc(O)nc12 N1(C(c2ccc(OC)cn2)=O)CCC(CNC(=O)Cc2c(C)noc2C)C1(C)C c1(C(=O)NC(C)CNC(C2CCc3nncn3C2)=O)cc2c(nc1O)CCC2 C1(C(C)NC(=O)CCc2cscn2)CCC(F)(F)CC1 c1(C(N2C(C)(CC(=O)NCC(C(C)C)(C)O)CC2)=O)cncn(C)c1=O N1(C(S(Cc2ccc(NC)cc2)(=O)=O)=O)C(C)C(=O)OCC1(C)C.C1CO1 N1(C(c2nc(-c3cccc(C)n3)sc2)=O)CCC(N(C(=O)C(C)C)C)C(C)C1 C1(NC(C(CC2CN(C(C3(OC)COC3)=O)C2)F)=O)CCCC(C2CC2)C1 c1(CCC(N2CC(C(C)(C)O)(CNC(C(F)=C(C)C)=O)C2)=O)cccc(O)n1 c1(CC)nc(C(=O)NC2CC(CNC(=O)C(C)(C)c3ccncc3)C2)c(N)s1 C(C(C)(CC(C)C)NC(C1CC(F)C1)=O)NC(c1ccc(COC)o1)=O Cc1nc2cc(C(=O)NCc3csc(CNC(=O)CC4CC4)n3)cc(O)c2[nH]1 N1(C(C(CC)(C)C)=O)CCC(O)C(C(=O)Nc2sccc2C#N)C1 N1(OC(C)(C)C2(CC(C)(C)C)CC2)CCN(C(=O)CCN(CCCO)C(C)C)CC1 CCCCC(O)CC(=O)NC1CC(NC(=O)CC2CCS(=O)(=O)CC2)C1 n1(CCC(=O)N(CC(C)N(C(C(CC(C)C)O)=O)C)C)cnc2c(N)ncnc12 c1(C(N2C(CN(C(=O)Cc3cn[nH]c3)C)CCCC2)=O)cc([N+](=O)[O-])c[nH]1 c1(C(=O)NCC2(C)CCN(C(c3cc(=O)cc[nH]3)=O)C2)cc2cccc(Cl)c2[nH]1 C#CCCCCCC(=O)N1CCCC(C(=O)NC2CCN(CC#C)CC2)C1 N1(C(C(C=C)(C)C)=O)CC2CCCC(NC(=O)CCc3ccccc3Cl)C2C1 C12(SCCC(=O)NCc3n(C)ncc3)CC3CC(CC(C3)C1)C2 N1(C(C(C2CCCCC2)C)=O)CC2CCC(C1)C(NC(C1CC1C)=O)C2 C1(C(N2CC(OC)C(C(=O)NC(CN(C)C)CCO)C2)=O)CC2CC(=O)C1O2 N1(C(C2CCC(C(=O)OC)CC2)=O)CCC(NC(c2cc(Br)c[nH]2)=O)C(F)C1 C(=O)(C(C(C)(C)C)NC(=O)CCOCC1CCC1)N(CC(CC)C1CCC1)CC C(C(C)(C)CNC(c1nc(C(C)(C)C)cs1)=O)N(C(c1cncn1CC)=O)CC Cc1ncsc1CCNC(=O)CC(C)c1ccco1.C12CC(C1)C(=O)N2C N1(C(C(c2ccc(C)o2)C)=O)CCOC(C)C1C(N1CC2(CC(O)C2)C1)=O Cc1c(C(N2CCCC(C(=O)O)C2)=O)[nH]c2cc(F)cc(F)c12.C(C)(C)(C)NC(C)C C(=O)(C1=CS(=O)CCC1)NC1(COC)CCN(C(=O)C(C)(C)N=[N+]=[N-])CC1 C1(NC(C2CCCC2)=O)CC2CC1N(C(c1cc(C3CCCC3)ccc1Cl)=O)C2 CC(CN(C)C)CCC(=O)N1CC(C(=O)NC(c2ccccn2)C)C2(CC2)C1 C(C(C(F)(F)F)N1CCN(C(=O)C=C2CCC2)CC1)NC(C1(CSC)CC1)=O N1(CCC)CC(C(=O)N(CC(C)(C)CNC(C2CC(C(N)=O)C2)=O)C)CC1=O c12ccnc(n1)N(Cc1nc[nH]n1)C2.N1(CC)CC(CC(N)=O)C(O)C1 c1(C(=O)NCC2CN(C(C(CC)SC)=O)CC23CCC3)ccnc(S(N)(=O)=O)c1 c1(NC(C)=O)ccc(C)c(C(N2CCC(O)C(C(=O)NCc3nn[nH]n3)C2)=O)c1 c1(CN(C(=O)C(O)C(F)F)C(=O)NC(C)(C)C)cccc(C(N2CCCC2)=O)c1C C1(C(=O)NC2CC(O)C2)CCN(C(=O)C2CC2C2CCC2)O1 c1(SCC(=O)NC(C2CCN(C(C3(O)CC3)=O)C2)C)nc2ccccc2o1 CC(C)CC(CNC(C1CN2CCC1C2)=O)C(=O)NC1CC(C)CC(C)C1 N1(C(CCC(C)(C)OC)=O)CCC(C)(C)C(NC(C2CCCCCC2)=O)C1 C(=O)(CCCS(C)(=O)=O)N(C1CCN(C(=O)CCn2cnc([N+](=O)[O-])c2)C1)CC c1(C(N(CC(CNC(C=C(C)c2cccs2)=O)O)C)=O)ccnc2nc(C)nn12 N1(C(C(=O)NCC)CCC2CC2)CCN(S(=O)(=O)NC(C)C)CC1 C1(CC(=O)NCc2c(SC)con2)CCCC(NC(=O)CCc2ccccc2)C1 c1(C(=O)NCc2c(-n3cnc(C#N)n3)cccc2)cc(Br)cc([N+](=O)[O-])c1 C(CCCCC(=O)N1CCCC(CNC(c2cccc(N)c2O)=O)C1)SC C1(C(N(C)CC2CN(C(C)=O)C2)=O)CCc2ccnn2C1.N12CC(C1)SCC2=O Cc1ccccc1C1CCCCN1C(c1sccc1N(C)C)=O C(=O)(CC1CCc2ccccc21)NC(CNC(CS(CC=C)(=O)=O)=O)CCCC c1(C(C)C)nc(NCc2cc(Br)no2)cc(=NC(CN(C)C)C(C)C)[nH]1 N12CCCC(CC1)OC2=O.C12(O)C(=O)C3CC1C2C3.C(F)(F)(Cl)OC(C)(C)C n1(CCn2cc(C3(C)CN(C(C4CCC=CCCC4)=O)C3)nn2)cccc(O)c1=O c1(NC(N2CCC(Cc3ccc(O)cc3)C2)=O)cc(F)c2c(c1)OCCO2 C1(C(=O)NC(C2N(C(c3ncc(OCC)nc3)=O)CCC2)C)COCCC1(F)F N1(Cc2c(F)ccc(C)c2)CC(C(N2CC3CCC2C3)=O)CC(F)(F)C1 c1(C(N2CCCC(C)(NC(CC3(C)CC3)=O)C2)=O)cc(F)c(Cl)cc1F C1(NC(CCNC(=O)OCC)=O)CN(C(=O)C#CC2(CC)CC2)CC1C1CC1 C12(NC(CC(C)N3CCCC3=O)=O)CCC1CN(C(c1c(O)cccc1F)=O)C2 c1(C(=O)NC2(CCNC(C3(CC=C)CCOCC3)=O)CC2)cc2cnccc2[nH]1 c1(C(N2CC3C(C(=O)NCCC(OC)OCC)(C3)C2)=O)c(F)ccc2[nH]ccc12 Cn1nc(C(N2CSCC2C(N2CCCC(F)(CO)C2)=O)=O)ccc1=O Cc1occc1C(=O)NCC1CCN1C(c1coc(C2CCCC2)n1)=O c1(C(=O)NC(c2ncc(C)cc2C)C(=O)OC)ccc(S(C)(=O)=O)s1 C1(N(CC(N2CCCC2C(N2CCC(CCF)CC2)=O)=O)C)CC(S(C)(=O)=O)C1 C=CC1(CC(=O)NC2CCN(C(C3CCSC(C)C3)=O)C(C)C2)CCOCC1 c1(C(=O)NCC(C)NC(c2c(N)ccc(C)c2F)=O)ccc(Cl)c2occc12 c1(C(N2CC(=C)C2)=O)csc(=N)[nH]1.C1C(=O)N(C)CC(=O)NCCO1.C1CO1 c1(C(=O)NC2C3CN(C(COC)=O)C3CC2)c(C(F)F)ccc2ccccc12 C1(C)(C(=O)NCC2(F)CC(NC(C(C)(C3CC3)NC(C)=O)=O)C2)CCC12CCC2 C#Cc1cnc(C(N2CCC(NC(=O)CCC=CC=CC)C(C(N)=O)C2)=O)c(C)c1 O=C(C1=CNC2=NCCC2=C1)Nc1ccc(C(F)(F)F)cc1.C12CCN(C1)C2=O Cc1cc(C(N2CC(CNC(c3nccnc3N)=O)C2)=O)c(N)c([N+](=O)[O-])c1 CC1(C)CCC(CC(=O)NCC2CCC(C(=O)NCC3CCC3(C)C)CC2)C1 CCC(CC(=O)N1CC=C(C(=O)N2CCCC(CO)CC2)CC1)C(C)C c1(OC)c(Cl)ccc(C(N2CCC(O)C(NC(=O)CC3CC=CC3)C2)=O)c1F C(CCCCCNC(=O)CC1CCCCC12CC2)N(C(C(C)=C(CC)C)=O)C c1(N(C(c2nnnn2C2(C)CC2)C2(CCl)CCC2)C2CC2)nc2cnccc2o1 N1(C(C(C)C2CC2)=O)CCC(C)(CNC(=O)C=CCN2CCOCC2)C1 C1(C(C)C)(C(=O)NCCCSc2ccccc2F)CC(F)(F)C1 CC1=C(C(=O)NC2CC(O)(CNC(=O)C(O)CC(N)=O)C2)Cn2ncnc2N1C c1(OCC)cc(OC)cc(C(O)CNC(c2cccc(F)c2)C(C)(C)C)c1 N1(C(=O)NC2C(C=C)CC2)CC(CO)CC(C)(C)C1 c1(C(=O)NCC(CNC(c2cnn(CC3CCC3)c2)=O)OC)n[nH]c2c1CSCC2 c1(C(C)C(=O)NCC2(O)CCNC2)cnccn1 C1(C(=O)NCc2ccc(COC)o2)CCN(C(C2CCC3(CC3)C2)=O)C1C c1(NCc2c(C)cc(Br)cc2C)cccn2ncnc12 C(=O)(C(C(F)(F)F)C(F)(F)F)N1CCC(CCNC(=O)C=C2CC2)C1 c1(C(=O)NC2C(=O)NCCN(C(=O)NCNC(=O)C(Cl)(Cl)Cl)C2)ccc2ncoc2c1 C(=O)(C1=C(Cl)CCC1)NCC1C(NC(Cn2nnc(=N)[nH]2)=O)CCCC1 CC1CC(CNC(=O)Cn2ccc(Br)n2)CN(C(=O)COC(=O)CO)C1 N1(C(CN2C(C)CCC2)=O)CCC2C(C(=O)NCCN3CCCCCC3)C2C1 C=CC(CC)C(=O)NCC(CC1CCCC1)C(=O)NC1(C(N)=O)CCOCC1 C(=O)(C#CC1CCOC1)NCc1ccc(CNC(CC2(C)CCOCC2)=O)cc1 CCCCC(CNC(=O)CNS(=O)(=O)CC)NC(=O)CSc1ccc(C)s1 CC1CC(CNC(=O)CC2(CO)CCOCC2)CCN1C(c1ccncc1Cl)=O Cc1cc(C(N2C3CCC2C(CNC(C24COCC(C2)C4)=O)C3)=O)c(N)c(C)c1 c1(C(=O)NCCCN(C(=O)C=CC(C)(C)C)C(C)C)n[nH]c2c(=O)n(C)cnc12 N1(Cc2ccc(C=C)cc2)CCC2(CC1)CC2(C)C(=O)NCc1nn[nH]n1 C1(C)(NC(CC=C=C)=O)CCN(C(=O)COc2ccc(CC#N)cc2)C1 N1(C(=O)Nc2c(C)cccc2)CCN(C(c2cc(O)cc(Cl)c2)=O)CC1C Cc1cccc(CN2C(C(N3CCCC(NC(=O)C4CC4)CC3)=O)CCC2)c1C C=Cc1cncc(C(=O)NCCCCC(C)NC(C2CCN2S(C)(=O)=O)=O)c1 Cc1ccc(C(=O)NC2CCCCN(C(C3C=CCS3)=O)CC2)c2ccccc12 S(=O)(=O)(c1cccc(C(N2CCC(C)(NC(C3CC(C)(C)C3)=O)C2)=O)c1)N(C)C CC(CC(C)(F)F)C(=O)NC(C)CN(C1(C(N)=O)CC1)Cc1ccccc1 c1(NC(=O)CCN2CCCC2)cccc(NC(C2CCCC(C(N)=O)C2)=O)c1 C(CCNC(C1(C)C=CCN1C(=O)C(C)N1CCCC1)=O)(C(C)C)OC C1(N(C(=O)C(F)OC(F)(F)F)CCNC(c2ncsc2Br)=O)CCCCCC1 C(c1cc2ccccc2o1)=CC(=O)NCC1N(C(c2nc(CC)[nH]n2)=O)CC=C1 N1(C(CC(c2cccs2)SC)=O)CCN(C(N2CCCC(N(C)C)C2)=O)CC1C C1(NC(c2[nH]cc(CC)c2)=O)CC12CCC(NC(=O)C1=C(C)CCC1)CC2 CN1C(=O)CCC1CCNC(=O)NCC1CCN(S(C)(=O)=O)C1 c1(C(C)C)ccc(C=CC(=O)N(CCCNC(c2cc(C#N)no2)=O)C)cc1 Nc1ccc(C(N2CCCCC2CNC(=O)C(=Cc2c[nH]cn2)F)=O)cc1O N1(C(c2cc(C(=O)OCC)on2)=O)C2CCC1C1CC1(NC(C1CCCS1)=O)C2 N1(C(CCC=C)=O)CCCC(C2CCCN(C(c3ccc4scnc4c3)=O)C2)C1 Cc1cc(N(C(=O)CONC(=O)C(C)CC2CC2C)C(C)C)cc(O)c1 C1(C(=O)NCc2ccc(CNC(C(C)(C)C3CCC3)=O)cc2)CC2(CCC2)CO1 N1(C(=O)NC2CCN(c3ccccc3)C2)CCOC2(C1)C1CC=C(C2)N=N1 CCC1c2cccn2CCN1Cc1nnc(-c2ccnc3ccnn23)o1 c1(OC)ccc(C=CC(=O)NC2CC(CNC(C3(C#N)CC3)=O)C2)cc1OC C(=O)(C1=CCCSC1)NCC1C(C(=O)NCCN2CC(C)OCC2)CCC1 C1(C)(C(=O)NC2CCC(C(=O)NCC=CC)CC2)CCC(=O)CC1 c1(N2CCCN(C)C(=O)C2)nc(=NC2CCC3(CC3)C2)[nH]c2cc[nH]c12 C1(N(C(C=CC=CC)=O)CCNC(=O)C(C)CC)CCN(C(=O)NC(C)C)C1 C1(C(N(C(c2ccccc2)CNC(C23CCC2CC3)=O)C)=O)Cc2nccn2C1 C#Cc1cnn(CC(=O)NCC2CCC2NC(c2ccc(CC)[nH]2)=O)c1 c1(C(=O)NC2CCCN(C(C3(OC)CC3)=O)C2)c(O)ncc2c1CCC2 CC(C)(CNC(=O)C(CC1CC1)N(N(C)C)C(C1CCCOC1)=O)CC1CCCC1 N1(C(=O)NCC(=O)N(CC(F)(F)F)CC)CC(NC(=O)C=CCn2cnnn2)C1 CC(C)CCCCCC(=O)NCC1CCCC(CNC(c2nsnc2O)=O)C1 n1(CCC(=O)NCC(CO)(CO)NC(C=C(C)C(F)F)=O)ccc2cccnc12 c1(C(N2CC(CC(C)NC(c3cc(CC)sn3)=O)C2)=O)cnn2c(C)ccnc12 c1(OC)cc(CC(=O)NC(C)C(C)(C)NC(c2csc(C(=O)OC)n2)=O)ccn1 c1(C(=O)NCCCN(C(c2c(Cl)cc(C)s2)=O)CCO)c(F)c(F)cc(F)c1F C1(C(N(C2CCN(C(CCC=CC(C)C)=O)C2)C)=O)COCC1(C)C N1(C(C(CC(C)C)OC)=O)CCC2(CC1)CC2C(N1C2CCC1CC2)=O.C1C(=O)N1 C1(C(=O)NCCNC(c2c(C)oc(CO)c2)=O)CCC(C2CC2)C1 C=CC1(CC(=O)N(C)CC2(N3CCCC3)CC2)CN(C(=O)Cc2cccc(F)c2)C1 c1(-c2n(C(c3cnn(C)c3)C)nc(-c3ccccn3)n2)cccc2cnsc12 C1(C(N(CC(CN(CCCOC)C)O)C)=O)CC(=O)N(CC(C)C)C1.C(C)(=O)O C1(NC(c2n(C(C)C)ccc2)=O)C2CC3C1C3C2C(N1CCCC1CCO)=O c1(NC(C2CN(C(c3cccc(CO)c3)=O)CCC2O)=O)ccc2nonc2c1 Cc1cc(C(CC)NC(C2CCCC2CNC(=O)COCC(C)(C)C)=O)no1 CCC(C)(C)C(O)C(=O)NCC1CC2CC2N1C(c1cc(OC(C)=O)ccc1O)=O C(CCCOC(C)C(=O)NCC(CC)N(C)C(C)=O)OC N1(C(Cn2c(C)nnn2)=O)CCN(C(=O)Cc2cc(Br)ccc2F)C(C(C)C)C1 N1(C(CNC(=O)OC)=O)CCC(C)(C(=O)NC2CCC(NC(C)=O)CC2)C1 N1(C(c2nc(C)c(C)[nH]2)=O)CC(NC(c2ccc(C)n2C)=O)C(C)(C)C1 c1(C(N(CCCCNC(c2c(C)cc(CC)o2)=O)C)=O)cccc(CC)c1N c1(C(C)C)cc(C(=O)NCC(C(C)C)NC(=O)CNC(=O)C(F)(F)F)n(C)n1 C1(NC(CC2CCC(=O)N2)=O)CC2CCC1C(NC(=O)CCN1CCCC1=O)C2 c1(CC)nc(C#N)cc(=NCCCNC(c2cnn(C3CCC3)c2)=O)[nH]1 c1(OC)cc(NC(=O)C(F)CC2CN(C(c3[nH]c(C)c(C)c3C)=O)C2)ccc1OC CC(C)(CN1CCCC(O)C1)C(F)C(=O)N1CCCCO1 C12(NC(C(F)OC)=O)CC(CNC(C3CC3c3ccccc3Cl)=O)(C1)OC2C C1(NC(=O)C=CI)CC12CC(NC(C1CCN(CC(F)(F)F)C1)=O)C2 C(=O)(CCCCC(C)C)NCC(C)N(C(COCC#C)=O)CC CC(C(F)(F)F)C1(O)CC(C(=O)NC(=O)NCC(=O)NCCN(C2CC2)CCCl)C1 C=CCCC(C)(C)C(=O)N1CCCC1C(=O)NCc1cc(O)cc(F)c1 C1(NC(=O)C=CC2CCCN2C(=O)CCc2cccs2)CCC(C2CC2)C1 c1(C(c2n(CCCSC)nnn2)NCC(C)C(C)(F)F)cnc2ccccc2c1 Cc1ccc(Cl)c(F)c1C(N1CCC(n2cc(CCO)nn2)CC1)=O C(=O)(C(CCC)CCCO)NC(CCNC(CS(CCC)(=O)=O)=O)C(C)C C1(NC(=O)CCOCCOCCO)CC(F)CN1C(=O)Cc1c[nH]nc1O C=CCC(C(=O)NCCC(O)CNC(=O)CSc1nncn1C(C)(C)C)C(C)C c1(C(=O)NCC(CNC(c2nc(C)[nH]n2)=O)CO)cc2cc(Cl)cnc2o1 N1(CC(O)Cc2ccccc2)CCC2(CCOCC2)C1 Cc1cn(C)nc1C(=O)NC1CC(=O)N(C2CN(C(=O)C(C)(C)N(C)C)C2)C1 C(=O)(N=c1ccn(C2CC2)[nH]1)C1CCC(Cc2ccc(CC=C)cc2)CC1 c1(C(=O)O)cnc(Cl)[nH]c1=NC(CNC(=O)C(CO)c1ccccc1)C1CCC1 c1(C(N2C(C)CC(NC(=O)CS(=O)(=O)N(C)C)CC2)=O)cnn2ncccc12 c1(C(N2CCC(C(CNC(c3c(C)nns3)=O)(C)C)CC2)=O)c(O)cccc1F CCCC(F)C(=O)NC1CC(CNC(C2SCCCS2)=O)C1(C)C c1(NC(C=Cc2ccc(OC)cc2)=O)ccc([N+](=O)[O-])c(O)c1 C(=O)(C1=C(C)CCCC1(C)C)NC1CC(OC)CN(C(=O)CC(F)(F)C(F)(F)F)C1 N=c1ccc(C(=O)NC2CC3(C2)CC3NC(c2cc(Cl)cs2)=O)c[nH]1 C12(C(=O)OC)CC1CCN2C(=O)Nc1cc(C)oc1C C1(C(=O)NCC(CC)(C)OC)CCCCCCN1C(c1cc(C)co1)=O Cc1c[nH]nc1C(=O)NCc1c[nH]nc1C(=O)NCC1CCC(C)C1 CC(C)(C)CC(O)CNC(=O)CC1(C)CCN1C(C1CN(C(N)=O)C1)=O C12(NC(=O)Cc3ccsn3)CCCC1CN(C(c1c(CC)c[nH]n1)=O)C2 Cc1ncncc1C(=O)N(CC(C)(C)CNC(C1(C2CCCCO2)CC1)=O)C c1(C(=O)OC)ccc(CNC(C2CC(C)CN(CC3CCOC3)C2)=O)cc1F C12CCCN1C2=O.C1(C(N2CC(CN3CCOCC3)C2)=O)(CN(C)C)CCCC1 c1(N2CCN(C(C(=O)NCC34N(C)CC(C3)C4)=O)CC2)nc2ccccc2s1 Cc1cc(NNC(=O)C(N)C2CCCC2O)nc(=N)[nH]1 N1(C(C(C)OCCCC)=O)CC2C3CCC(C2C1)N(c1ccc(C#N)nc1)C3 c1(OC)cc(C(=O)NC2CCC(CNC(=O)Cc3cn(C)nc3C)C2)c(Cl)cn1 C12(OC)CCC(C(=O)N(CCC(N3CCCC34CC4)=O)C3CC3)(CC1)C2 N1(C(C2C(C(=O)NCC#C)C2)=O)CC(c2ccccc2)(NC(=O)C=C(C)C(F)F)C1 c1(NC(C2CC(=C)CN2Cc2ncc(-c3ccccc3)cn2)=O)cc(F)nc(F)c1 N1(CCNC(c2c(CC)nn(C)c2)=O)CC2CCCC1C2c1nnc(O)n1C C1(C(N2C(CN(C(=O)CCC(N)=O)C)CCCC2)=O)CCc2nc[nH]c2C1 c1(C(N(C)CC2(CNC(C(CC)F)=O)CC2)=O)cc2c(OC)ccc(Br)c2[nH]1 Cc1csc2ncc(C(=O)N(C)CC3CN(C(C4(O)CCC4)=O)CCO3)n12 N1(C(Cc2nc(C)c(C)s2)=O)C2CCCC1CN(C(=O)C(C)(C)C(N)=O)CC2 N1(C(c2c(C)scn2)=O)CCC(C(F)(F)F)C(NC(C2(C)CCOC2)=O)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1C(C)CN(C(C2C3CCCC23)=O)CC1 N1(C(C=NOC)=O)CCN(C(c2cnn3c2C(=O)NCC3)=O)C2CS(=O)(=O)CC12 c1(C(N2CC(NC(c3c(SC)snn3)=O)C(C)(C)C2)=O)csc2c1CCC(C)C2 C1(C(=O)NC(CCNC(CN(C(C)C)C)=O)(C)C)Cc2c[nH]cc2S1(=O)=O Cc1ccc(Cl)c(C(=O)NC(CNC(c2cnc3cccnn23)=O)C2CC2)c1N Cc1onc(Cl)c1C(=O)NCC1CCC(NC(=O)COCC(F)F)C1 N1(C(C(c2cccc(C#N)c2)C)=O)CCCN(C(=O)CN2CC(C)(C)C2)CC1CO C1(CNC(CC(C)C2CCCC2)=O)CCC2(CN(C(=O)COC3COC3)C2)O1 C12(CNC(=O)C(=O)Nc3nncs3)CCCC1N(C(=O)CSc1cccs1)CC2 C(CCCCC(F)F)NCc1onc(-c2cc(N)ncn2)n1 C1(NC(C(N2CCC(C(C(=O)OC)C#N)CC2)=O)=O)CCc2c[nH]nc2C1.C1CC1 N1(C(c2cc(-n3cc(C(C)N(C)C)nn3)ncc2)=O)CCC2C(O)CCCC2C1 c1(OC)cc(Cl)c(Cl)cc1NC(=O)CC1CN(Cc2nc(Cl)ccc2Cl)C1 N1(C(CC2(COC)CC2)=O)CCCC2CN(C(=O)CC(C)(C(F)F)N(C)C)CC12 c1(C(=O)NC2(CC=C)CCN(C(=O)CNS(=O)(=O)CC)C2)cccc(C#C)c1F N1(C(c2ccn(C)c2)C(=O)NCC(C)C)CCn2c(-c3cnn(C)c3)nnc2C1 N1(C(C2CN(C3CCC3)C2)=O)CCCN(NC(CCc2onc(CC)n2)=O)CC1C N1(C(C(C(C)(C)C)OC)=O)CCC2(CC2)CC1C(=O)Nc1cc(C)cc(F)c1 N1(C(CCCC#CC)=O)CCC2CCCC12C(=O)NC1C=CC(C(=O)NC)C1 Cc1cc2nc(-c3cn(CC4CCC(C(F)(F)F)OC4)nn3)cn2cc1C C1(C(C)C)CN(C(C2C=CCCC2)=O)CCN1C(=O)C1=C(Cl)CCC1 C1(C2CCOCC2)(C(=O)NCCC2N(C(CSCCC)=O)CCSC2)CC1(F)F C1(C(=O)NC(c2ncc(C)cn2)C)C2CCN(C(C3CC3C3(C)COC3)=O)CC12 N1(C(CC(C(F)F)NC(c2cccc(CC=C)c2)=O)=O)CCC(O)CC(C)C1 C1(NC(C(=O)Nc2cccc(CS(N)(=O)=O)c2)=O)C2Cc3ccc(Cl)cc3C12 c1(NC(C2CC2C(CCN2CC(C)(C)OCC2)=O)=O)c(Cl)cc([N+](=O)[O-])cc1Br c1(CC(=O)NC(C(=O)NCCc2c(C)n[nH]c2)C2CCCO2)cccc(O)c1 N1(C(c2ccc(CO)cn2)=O)CC2CCC(NC(C3(C4CCC4)CC3)=O)CC2C1 c1(C(N2CCC(N3CCN(C(C(CC)(F)F)=O)CC3)C2)=O)cncn(C)c1=O c1(CC(N2CCN(CC(=O)Nc3occc3Br)CC2)=O)cccc(F)c1F c1(C(=O)NC2CC(CCOC)C2)cc2ccccc2cc1F.CCC1(C)C(=O)N1 CC1CCN(C(=O)NC(c2nnc(S)n2C)C)CC1F N1(C(C(C)(C)C2CCC2)=O)CCOC2(C1)CN(C(C1CC(n3ccnc3)C1)=O)C2 N1(C(CCSCC)=O)CCC(NC(c2nnc(C)cc2O)=O)CC(C)(C)C1 C1(CC(=O)NC(C)(C)CNC(C23CC(CCO2)C3)=O)(COC)CCOCC1 c1(C(=O)NC2C(CC)CN(C(c3c[nH]nc3C)=O)C2)ccc(=O)n(C)c1 CCCCCC(=O)NCCC1CN(C(=O)CC(c2ccon2)C2CCCC2)CCO1 C(C(=O)NN1CCCC1)=CCC.N12CC(C1)CC2=O.C(C)(C)O C=CCC(C(=O)N1CCC1CNC(c1cnc(C)o1)=O)C(C)C C1(C(N2C(CNC(C(C)C3CCOC3)=O)CC2)=O)CCCS(=O)(=O)C1 C(C(CN=c1nc(N2CCCCCC(C)CC2)c2c([nH]1)COC2)C(C)C)OC c1(CC(=O)NC2CN(C(C=CCOC(C)(C)C)=O)CC(F)C2)ccc2n[nH]cc2c1 C#CCC(C(=O)NC(c1cncc(F)c1)C)NC(=O)C=C(C)C(=O)NC CC1CCC(C(N2CCN(C3CCC3)CC2)=O)CN1C(C1CC1C(C)(C)C)=O C(=O)(C(C)(C)C(C)(C)O)N(CCC(C)CC(F)F)CC(=O)O c1(C(=O)NC(C(C)(C)C)CNC(C2CCCCC(=O)C2)=O)cccc2cnsc12 N1(C(Cc2cc(C)[nH]n2)=O)CCC(CCNC(c2nc(Cl)sc2C)=O)C(F)(F)C1 C1(C(N(C)CC(=O)NCC2CC(O)C(F)C2)=O)CCCC(C#N)C1.C1C(=O)O1 c1(C(=O)NCC23C(CN(C(C4CC(OC)C(OC)C4)=O)C2)C3)cc2c(s1)CCC2 Cn1ccnc1COCC(=O)NCCC1CN(C(=O)CN2CCSCC2)C1 C#CC1CC2CCC1N(c1cc(NCC3(OC)CC3)nc(C)n1)C2 N1(C(CC2OCC(C)(C)C2)=O)CC2CCCC(C1)N2C(c1coc(C2CC2)n1)=O c1(C(C)C)cc(C(N2CCC2CNC(c2cccn2Cc2cccs2)=O)=O)cs1 N1(C(C2N(S(CCC)(=O)=O)CCCC2)=O)CC(N(C(=O)CC)C)C2(CC2)C1 c1(C2CN(CC(c3nc(-c4ccncc4)no3)C)CC2O)nc2ccccc2[nH]1 c1(C(N(CCNC(C2CN(S(CC)(=O)=O)C2)=O)C(C)C)=O)c(Cl)ccc(F)c1F C1(CCOC)NC(=O)N(C2CCN(Cc3ccc(C)cc3C)CC2)C1=O c1(OC)ccc(C(=O)N(CCNC(=O)CSCC(F)(F)F)C2CC2)c(Cl)c1 C=C1Cn2c(C(N3CC4=C(C3)CN(C(=O)C=Cc3cnc[nH]3)C4)=O)nnc2S1 C(=O)(CCCCCOC)N1CC(CC(=O)NCCOC(CC)(C)C)C(C)C1 C1(C(=O)NCCCCN(C(CC2C(CC)C2)=O)C)CCn2cnnc2C1 Cc1nc(Cn2cc(-c3ccnn3Cc3cccnc3)nn2)c(C)s1 C1(CC(=O)N(C(C)C(=O)N2CC(n3ccnn3)C2)C)CC2(CC2)C1 CC1(C)CCC(C(=O)NCC2CCCCN2C(C2CCC(C(N)=O)CC2)=O)O1 N1(C2(C(N(CCN(C)C(C3(N(C)C)CC3)=O)C)=O)CC2)CCOCC1 C=CCC(CNC(c1cncc(OC)n1)=O)C(=O)NCc1nc(C)sc1C Nc1cc(C(N2CCC(NC(c3ccc(Cl)c(O)c3)=O)C(F)C2)=O)nc(O)c1 C(=O)(CCCC(=O)NC1CC(C)(NC(=O)CC(C)COC)C1)NCC Cc1cncc2cc(C(N3CC(NC(c4ncn5ccccc45)=O)C3)=O)sc12 C1(NC(=O)C=Cc2ncc[nH]2)CC2CC1CN2C(c1ccoc1C(F)(F)F)=O N1(C(=O)C2=CCCN(C(c3occ4c3CCC4)=O)C2)CC2C3C=CC(O3)C2C1 C(C)(CCC(=O)N(C(C)CNC(c1cnc(-c2ncccn2)s1)=O)C)SC c1(C(=O)NCC2CCN(C(CCN(C)CC)=O)C2)ccc2c(c1)C(C)CO2 N1(C(C(C)SC(C)C)=O)CCC(C)C1CNC(C12CSCC1C2)=O c1(C(=O)NCCNC(N(C)C)=O)ccnn1C1CC1.C1(C(C(=O)N)O)CCCC1 N1(C(C2CN(c3ccccc3)C2)=O)CCc2ccccc2C1.c12cccc(n1)O2 C(CNC(c1c[nH]ccc1=O)=O)(CC(=O)NCC(c1cn(C)cn1)O)OC C(N=c1ccnc(C(C)C)[nH]1)C1(C)CCN(C(CCCNC(C)=O)=O)C1 CC(C)CC(C(=O)N(CC(O)CN(C)C(C1CCCN1N=O)=O)C)N(C)C N1(C(c2ccc3c(n2)CCCC3)=O)CC2(CCN(C(C3CC4CC4C3)=O)CC2)C1 N1(C(c2c(C)nc(C)n2O)=O)C2CCC1CN(C(c1ccc3c(n1)NCC3)=O)C2 c1(CCNC(c2cn(C)nc2Cl)c2n(CCCOCC)nnn2)cnc(C)nc1 C12COCCC1CC(=O)N2.N1(CC)CCCC1CNC(C1(CC2CC2)CC1)=O C1(NC(CC(C)SC)=O)CCN(C(c2cnsn2)=O)C1c1ccccc1 C1(NCc2cn(C(C)C)nc2)CCN(C(=O)CC2CC(O)C2(C)C)CC1F N1(Cc2c(=O)cc[nH]c2)CCOCC12CCOCC2 N1(C(C2CC3(C(OC)CC3)C2)=O)CCCOC(CCNC(=O)CCCCSC)C1 c12c(ccc(C(C)C)c1C(F)(F)F)S2.CCCCC(C)(c1nnnn1C(C)C)NCC Cc1ccc(C)c(CC(=O)NCC2CCN(C(C3(C)C=CCC3)=O)C2)c1 C1(NC(c2cc(OC)no2)=O)CCN(C(=O)CC2CC=CC2)CCC1CO C12(N(C3(CNC(=O)C4CC4)CC3)C(C3(c4ccno4)CC3)=O)CCC(CC1)O2 C(=O)(CCCC(=O)NC(CC)CNC(=O)CC1CC(F)(F)C1(F)F)N(CC)CC C(=O)(CCCNC(N)=O)NC(CN(C(=O)CCN1CCC1)C)CO CCC(=O)CCC(=O)NCC(O)CN(C)C(C1(C)CCCS1)=O C(=O)(C(CCCOC)NC(=O)CC1CCC(=O)CC1)N(C(CC)CC)CCO C1(NC(c2cn(CC)nc2C2CC2)=O)CC2C1CCN2C(c1snnc1C)=O N1(C(CC2C=CC(C(=O)NC3C(=C)C3C(=O)OC)C2)=O)CC=C(C)CC1 c1(C(=O)NC2(CCC(N3CC(C#C)(O)C3)=O)CCC2)ccc2[nH]nc(Cl)c2c1 C1(CNC(CC(=O)NCC#C)=O)CC(O)CN1C(c1cnc(SC)s1)=O CC(C)(C)CC(O)C(=O)NCC1C=CC(NC(=O)C=CC2CCCC2)C1 CC1CCN(C(C2CCCC2F)=O)CCN1C(C1CC2CC2C1)=O C1(NC(=O)C(c2ccccc2)O)CC2CCC(C1)N2C(c1cccc(F)c1)=O C=C(Br)CC(C)(C)C(=O)NC1C=CCN(C(=O)CC2CC(C)(C)CO2)C1 c1(C(=O)NC2CC(C(C)NC(C(C(C)O)(F)F)=O)C2)cccc2cc[nH]c12 C12(NC(C3CCC=CCC3)=O)CN(C(=O)CCn3ccnn3)CCCC1C2 C(CC(=O)N1CCNC(=O)CC1)(C(F)(F)F)NC(CC1(C)CCOC1)=O N1(C(c2n(CC)ncc2)=O)C2CCC1CN(C(c1ccc(F)c(CSC)c1)=O)C2 C1(NC(CCCOCC)=O)CC(F)CN(C(c2cscc2C)=O)C1 C1(N(C)C(c2cn(C3CC3)nc2C(F)(F)F)=O)CC2CC1N(C(C1CCC1)=O)C2 N1(C(c2ccn(CCOC)n2)=O)CC(NC(=O)CC(C)C(=O)OC)CC2(CCC2)C1 Cc1nc(C(=O)NCC2CCCC2NC(c2csc(C3CCCO3)n2)=O)n[nH]1 N1(C(C=CC=CC)=O)CCCC1C1CCCN1C(=O)CCCCCCSC c1(C(N(CCC(C)NC(=O)CCCc2ccsc2)C)=O)cc2ccc(O)cc2[nH]1 N1(C(COCCCCC)=O)CCC(OCCCNC(=O)CC2CCC(C)C2)CC1 c1(OC)c(C(=O)NC2C=CCN(C(C3CC(C(F)(F)F)C3)=O)C2)nc(O)nc1O N1(C(C(CCC)O)=O)CCOCC(CNC(=O)C(=O)C=Cc2ccc(F)cc2)C1 C#CCCCCCCC(=O)NC1CCCC1C(=O)NCc1ocnc1CC C(C)(CCC(=O)N1CCCC1C1(NC(=O)CO)CC1)OC N1(C(c2cc(Br)c[nH]2)=O)CCC2(CCC2)C(CNC(C2(CO)CCC2)=O)C1 CC1CC2(CCN1C)c1nnnn1CCN2.c1(CCS)cccc(F)c1F C=CC1CCN(C(=O)C#CCNC(=O)CC2CC(C)=NO2)CC1 N1(C(CCCC)=O)CC(CNC(C2CC=C(C)CC2)=O)OC2(CCC2)C1 N1(C(c2ccc(Br)c(C(F)(F)F)c2)C(=O)NC(C)(C)C)CCCC2(CCCO2)C1 C1(NC(Cn2ncc(CC)c2)=O)CN(C(c2c(C)noc2N)=O)CC1CC1CC1 Cc1ccc(C(C)CC(=O)NC2(c3ccc(Br)cc3)CN(C(=O)CCBr)C2)cc1 c1(C(=O)OC)nc(=NCC(CCOC)NC2(O)CCC2)cc(C(C)(C)C)[nH]1 C(CCC(CCC)NC(=O)C=Cc1ccoc1)NC(C1C(C=C)C1)=O c1(C(=O)NC2(CCCC(=O)NC3(c4cccs4)C(C)(C)C3)CCC2)ccc(C#N)[nH]1 Cc1ccc(O)cc1NC(=O)COc1cnc(F)cc1C(=O)NC(C)C C1(NC(C2CN(C(N)=O)C2)=O)CN(C(C2CC23CCCC3)=O)CC1F C(=O)(CCS(=O)(=O)N(C)C)N(CCC)CCNC(c1cccc(CCF)c1)=O CCC(C)(C)C(O)C(=O)NC(c1nocc1C(=O)NCC(C)(F)C(C)(C)F)C c1(C(=O)NC(C(CO)NC(C(C)OCC=C)=O)C)ccccc1N(C)C(C)C C1(CNC(C2C(C3C(C)C3)C2)=O)CCN(C(c2cnccn2)=O)CC1(F)F N12CCCC(C)(C1)C2=O.C1(CC)CCC(C(N2CC(CSCC(C)(C)C)C2)=O)O1 N=c1nc2c(c[nH]1)CC(C(=O)NCC1CCN(C(c3csc(Cl)c3)=O)C1)CC2 N1(C(c2ccc(C#C)cn2)=O)CC(C2CN(C(c3c[nH]c(=N)s3)=O)C2)C1 C1(NC(C2(C=C)CC2)=O)CC2(C1)CC(CNC(=O)CC1CCC=CCCC1)C2 c1(C(N2C(CNC(C(CO)OC)=O)CC(O)C2)=O)cc2cccnn2c1 C(C)(CCC(=O)N(C)CCc1ncon1)NC(CC(C)F)=O N1(C(CC2(C(=C)F)CCC2)=O)CCN(C(C2CC(C3CC3)=NO2)=O)CCC1C N1(C(c2nc(C(=O)OC)sc2)C)CCCCCC1CCNC(=O)CCC1(C)CC1 C1(C)(CNC(c2cc(OC)n(C)n2)=O)CCCN(C(c2ccncc2F)=O)C1 c1(OC)c(C(N2CCOCC2CNC(C2CC23CCCC3)=O)=O)nc(O)nc1O CCC(C)CC(=O)C(=O)N1CCN(C(C2CCOC(CC)C2)=O)CC(CO)C1 C(N=c1nc(C(F)(F)F)[nH]s1)C1CCC(NC(c2nccc(SCC)c2)=O)CC1 Cc1cc(C(=O)NC2CC23CCN(C(=O)Nc2cn[nH]c2)CC3)c(C)cc1F CC1CCc2[nH]c3c(C(=O)NC4CNCCS(=O)(=O)C4)cccc3c2C1 c1(C(=O)NCC2CCC(F)(CNC(CCSCC)=O)C2)ccc2nn[nH]c2c1 c1(N(C)C)cncc(C(=O)NC2CCC2CNC(c2c[nH]ccc2=O)=O)c1 C1(N(C(C2CC(CC)C2)=O)C)CCN(C(C2CC(=O)N(C)C2)=O)CC1 CCCCC(O)CC(=O)NC(c1cccc(OC)c1)CNC(c1csc(=N)[nH]1)=O c1(CC)nn(C)c(Cl)c1C(=O)NC1CCCC1CNC(c1cc[nH]c(=N)c1N)=O C(=O)(CCCCCC(C)C)NCC(C)(C(C)C)NC(CC(CC)C)=O N1(C(c2cnc(C(C)O)s2)=O)CCCOC(CNC(C2(CC(F)(F)F)CC2)=O)C1 CC(CC(=O)NOCCF)NC(c1cncc(C#N)c1)=O Cc1cccc(CC(=O)NCCC(C)N(C(=O)Cn2cnc(C(N)=O)n2)C)c1C c1(CNC2C(C(=O)NCc3cccc(-c4ccoc4)c3)C2)cc(O)cc(F)c1 N1(C(CC(C=C)(C)C)=O)Cc2ccccc2C(Nc2ncnc3c2COC3)C1 c1(CN2CCC(CNC(c3ccc(Cl)c(O)c3)=O)C2)cnc(O)nc1O C(CCCCC(=O)NC1CC2(C(N3CCC(C(F)F)C3)=O)COC1C2)OCC C1(C(=O)NCC=CCC(=O)NC(c2onc(C)n2)CO)CC(C)(C)CO1 c1(C(N2CC(O)(CNC(C3(C(C)(C)O)CC3)=O)C2)=O)snc(Cl)c1Cl C12(NC(C=CC(=O)OCC)=O)CCN(C(=O)C(=O)NC3CC3)CC1C2 c1(C(=O)OC)c(C)[nH]c2ccccc2c1=Nc1ncc(C(=O)O)s1 N1(C(C(C)OCCOC)=O)CCC(C(N2CC3(C2)CN(C)C3)=O)CC1C c1(C(N(CC(CNC(C(C(=C)C)(C)C)=O)C)C)=O)c[nH]c2cccnc2c1=O C(=O)(CC(C)(C)n1cc(C(C2CCCNC2)C)nn1)N(CC(=O)OC)C(C)C C1(C(C)C)CN(C(c2ccn(C(C)(C)C)c2)=O)CCCN1C(=O)CCN(C)C Cc1cccc2c1S(=O)(=O)CC2NC(=O)CC(C)(F)F Cc1cn2c(C(=O)NC3CCC(NC(=O)CC4CCC(=O)O4)C3)c(C)nc2s1 C1(OCC(=O)NCCCN(CC)CC)CCN(C(C2CC(C)=NO2)=O)CC1 C1(C(=O)NC2CC(C)(C)N(C(=O)CCc3cnc(O)[nH]3)C2)CCc2c[nH]nc2C1 N1(C(C(c2cccc(F)c2)C)=O)CCN(c2cnc(F)cn2)C(C(C)C)C1 C12(NC(=O)C=Cc3cnc[nH]3)CCCN(C(=O)CCc3ccccc3Cl)CC1C2 C1(C(C)NC(=O)C(C2(O)CCCC2)F)CCCN(C(c2ncccc2O)=O)C1 C(CC(C(=O)NCCc1ccccc1F)NC(=O)CC1COCCO1)SC Cc1cc(N)c(C)nc1C(=O)NCC(=C1CN(C(c2c(F)ccnc2Cl)=O)C1)F C1(CCOC)CN(C(C2(CSC)CC2)=O)CCN1C(=O)CN1CCOCC1 c1(C(=O)NC2CCC2CNC(=O)C(c2ccc(Cl)cc2)(F)F)n[nH]c2c1CCC2 n1(CC)ccc(C(=O)NCC23CN(C(=O)CC4CC5(CC5)C4)C(C2)CO3)cc1=O C1(NC(C(C)C2CCCO2)=O)CN(C(=O)CCNC(C2CCC2)=O)C2CCCC12 CCC(C)CC(C(=O)NCCC(C)CO)NC(C1OCCC1C)=O C(=O)(C(O)C(C)C)N(C(C)CNC(=O)CNC(c1ccccc1OC)=O)CC N1(C(c2cccc3c2OCC3)=O)CC2(CCN(Cc3c(F)cccc3I)CC2)C1 c1(C(N2CC(NC(C(CC#C)C)=O)CC2(C)C)=O)ccc2ncc(Br)n2c1 N1(C(CC2(C)CC2(F)Cl)=O)C2CCC1CC(NC(=O)CCn1cnnn1)C2 c1(CC(N2CCN(C(=O)CCc3cncs3)C3CC23)=O)cnc(O)nc1O Cc1cncc(C(C(=O)NC(C)C)N(Cc2ccccc2)Cc2ccon2)n1 CCCCC(CN=c1ncc(CO)c[nH]1)NC(c1ccn(C(C)C)n1)=O C1(NC(C2C(C)(C)OC(=O)C2)=O)CN(C(=O)CCc2cncnc2)CC(F)(F)C1 C(=O)(C(O)C1=CCCCC1)N(C)CC1CCCCN1C(C1CC(C)(C)CCO1)=O c1(C(=O)NCCN(CC(=O)N(c2ccccc2)C)C(C)=O)cnn(C)c1Cl N1(C(C)C)CCCC(C(=O)NCC(C)CN(C(=O)CCC2CCCO2)C)C1 c1(C(=O)NC2CN(C(c3cc(CC)cc(N)c3)=O)C(C)C2)cc(C)c(C)nc1O N1(CC2(NC(c3n(CCC)ccc3)=O)CC2)CCN(C(=O)C(O)C2CCC2)CC1 C1(NC(=O)C(C2CCOCC2)O)CC2(C1)CN(C(c1scnc1C1CC1)=O)C2 N1(C(C2(CC#C)CC=CCC2)=O)CC2CC(NC(c3cccc(O)n3)=O)CC1C2 N(C(=NCCCN1CCOCC1)NCC1CCCO1)C(c1cc(C)cc(C)n1)C C(=O)(C(C)C(=O)NCCCCNC(C1(F)CCC1)=O)OC N1(C(C(C)(C)Sc2ccc(Cl)cc2)=O)CC2(CCN2C(=O)CSC(F)F)C1 c1(NC(=O)NC2CN(CC#C)C2)ccc(F)cc1C#N CC1=C(C(=O)N2C3CCC2C(F)C(NC(C2CC2(C)C)=O)C3)CCS1(=O)=O n1(CC)nc(C(=O)NC2CCC(CNC(C3CCN(O)CC3)=O)C2)c(C)n1 C1(C(=O)NC(c2ccccn2)(C2CCCCC2)C)CCc2nnn(C)c2N1 N1(C(c2c(C)nco2)=O)CC2(CC2)CC1CNC(c1cc(C)ns1)=O C12(C(=O)NC3CCN(C(C4OCCN(C)C4)=O)C3)CC3CC1(CO)CC3C2 C1(CNC(c2scc(C)c2Cl)=O)(NC(=O)Cc2c(Cl)cnn2C)CCCCC1C c1(C(N2CCCC(CNC(C3(CCF)CC3)=O)C2)=O)ccn2cnnc2c1 C=CC1(C(=O)N(CC(CC)NC(c2cc(C)sc2F)=O)C)CCOCC1 CC1CCN(C(=O)CCF)CC1CC(=O)NCCOc1cccnc1 CC(C)(C)S(=O)(=O)CC(=O)N1CCN(C(=O)C2=CCCCO2)C(CCO)C1 c1(C(=O)NCC(C)NC(=O)CCCn2ccnn2)cn(CCN2CCOCC2)nn1 N#Cc1cc(F)c(NC(C2CC(F)CN(Cc3ccc(CO)cc3)C2)=O)c(F)c1 C(=O)(C1=CCCCO1)NC(C(C)C)CNC(=O)C=C1CCN(C)CC1 N1(C(C2N(C(C)C)CCOC2)=O)Cc2ccc([N+](=O)[O-])cc2C1 c1(C(=O)NC2C(NC(Cn3c(CCC)ncc3)=O)COCC2)ccc(F)c(C)c1 C1(CNC(C2C(C=C)C2)=O)CC(F)(CNC(=O)CCCN2CCCC2)C1 CC1(NC(c2coc3c2CSC3)=O)CCCN(C(=O)CCn2cncn2)C1 N1(C(=O)COCC2CC2)CCCN(CCCCNC(C2(F)CC2)=O)CC1 N1(C(C(C)OCCN(C)C)=O)CC2(COC(CNC(=O)C3=NNC(=O)C3)C2)C1 CC1CCN(C(=O)C(=O)N=S(C)(C)=O)CCN1C(C1CCCC(=O)N1C)=O C=C1CCC(C(=O)NC2CCC2NC(=O)C(C)Oc2ccccc2C)CC1 N1(CC(=O)NCC(C)(C)NC(=O)CC2CCOCC2)CCN(C2CC2)C1=O O=C(C1=NOC(c2ccccc2)C1)NCC1CCN(C(=O)CC2CSC2)CC1O c1(NCC2N(C(=O)C=C3CCCC3)CCC2)cc(C(F)(F)F)nc2ncnn12 C1(CC)CCN(C(=O)CSC(C)(C)C)C1C(=O)NC1CC(O)C(O)C1 C1(OC)CCC(C)(C(=O)NC2CCCN2C(=O)CCCC(=O)OCC)CC1 C1(CNC(C(CCC)O)=O)CC(C)CCN1C(c1cnc(C2CCC2)cc1C)=O c1(C(=O)NCCOC2CN(C(C3(C#N)CC3)=O)C2)ccc2c(c1)C(=O)NCC2 C(=O)(CS(=O)C(F)(F)F)NCCNC(C(c1c(OC)ccc(F)c1)(F)F)=O C1(F)(C(=O)OCC)CCC(CNC(=O)C(C)(C)C2CCCC2)CC1 CCC(C)(C)CCCC(=O)N1CC2CC(NC(C3C(F)(F)C34CCC4)=O)C1C2 C(CNC(c1c[nH]c(C)c1)=O)(C(C)(C)C)NC(C(COC)O)=O C(=O)(C1=CNC2=NCCC2=C1)N1CC(C2CN(C(C3(C)C(C)(C)C3(C)C)=O)C2)C1 CCCC(C#N)C(=O)NC(Cc1c(C)cccc1Br)C(=O)NCC(C)(C)C(C)(C)O CCC(CC1CCCC1)C(=O)N1CCCCC1CNCCNC(C1(F)CCC1)=O C1(C(C)C)CN(C(=O)CCCCCF)CCN1C(C1C(C)C1C)=O O=C(C#CC1CCCO1)NC12CCCN(C(c3cccc(Cl)c3O)=O)CC1C2 c1(C(C(=O)NCC(C2CC2)NC(=O)CC2CCOC2)O)ccc(Cl)cc1Cl N(C(=NCc1ccccc1-c1ccccc1)NCC1CCCCC1)C1CC(CC)C1 C1(CNC(Cc2ccn(C(C)C)n2)=O)CN(C(c2ccnc(S)c2)=O)CC1C CC(C(C)C(=O)N(C1CCN(C(=O)OC2CCC2)CC1)C)NC(=O)OC(C)(C)C CC1=NOC(=O)C1CC(=O)NCCOCCN(C)C(C1(Cl)CC1(F)F)=O C(=O)(C1=C(SC)CCCC1)N1CC2C(CNC(C=C(CCC)C)=O)(CC2)C1 N1(C(c2ccc(C(C)C)s2)=O)CCCC(N(C(=O)C(C)OCC2CC2)C)CC1 C1(NC(C(C)n2ccnc2)=O)CN(C(C2(C#N)CC=CC2)=O)CC1(C)C c1(NC(c2cc(Br)cs2)C)[nH]c(=NCc2cncc(C#N)c2)nc2c1ncn2C C1(C(N2CCC(CCNC(c3c(C)onc3)=O)CC2)=O)Cc2nn[nH]c2C(C)C1 C(=O)(C1=CCCC1(C)C)NC1CCCN(C(c2cccc(OC)c2)=O)CC1 C1(NC(CCCOC(C)=O)=O)CN(C(c2cc3occc3s2)=O)CC2CCCC12 C1(CNC(CC=CC)=O)(CO)CCN(C(=O)CCC(=O)N(CC)CC)C1 c12cc(on1)C(=O)N2.C(CCCO)C1CN(C(C)C)C1 C(=O)(CCCC(=O)OC)NC(CNC(C1(COC)COC1)=O)C1CCC1 CC(CN(C)C(C1(NC(=O)CCc2nncn2C)CC1)=O)C(F)(F)F CCC(C)C(O)CC(=O)NCC(C)(C)CC(=O)N1CC(=O)NC(CC)C1 c1(C2C(C(=O)NCCCCNC(C=C(COC)C)=O)C2)cccc(OC(F)F)c1 n1(CC(=O)NC2(CNC(C=CCC)=O)CCC2)nnc(-c2ccoc2)n1 C(C(F)(F)C(=O)N1CCCC1CNC(C1CC=CCN1C)=O)OC CCC(CCC(=O)N1CCOCCC1C)NC(C1CC2CCC1O2)=O C1(C(=O)NC(C(=O)NCCCN(CC)CC)CCF)CC12CCOCC2 CC(O)CCN=c1cc[nH]cc1S(=O)(=O)N1CCCC(C2(C)CC2)C1.CC CCC(C(=O)N(CC(C)(C)NC(=O)Cc1ccc(C)c(C)c1)C)C(C)(F)F CCN=c1[nH]c(C(=O)NCC2(F)CC(NC(=O)C(C)(C)C(F)F)C2)cs1 CC(CC(=O)N(CC(O)CNC(c1cnoc1-c1ccccc1)=O)C)C1CC1 c1(NC(C2N(C(c3c(C)oc(-c4cccs4)n3)=O)CC2)=O)cccc(F)c1F c1(CC(N2C(C(=O)Nc3nccc(C)n3)CC2)=O)ccc(Br)cc1Br C1(C(C(=O)NC2(CCOC)CCC2)C)CCN(C(c2nscc2C)=O)CC1 CC#CCCCC(=O)NC1(CF)CCN(C(=O)CCC2CC(OC)C2)C1 C(N=c1[nH]nc(C(F)(F)F)s1)C1OCC(CNC2(CC(=O)OC3CC3)CC2)C1 C12(CNC(C3(CC4CCCC4)CCC3)=O)CC(CN1C(=O)Cc1cncnc1)C2 c1(NC(c2ccc(-c3c(C)nc(C(C)C)o3)cc2)=O)ccc(OC(F)(F)F)c(Cl)c1 C1(CC(=O)NCCOCCNC(C=Cc2n(CC)ncc2)=O)CC2(CCC2)CO1 C12(CNC(C=CC(C)C)=O)CCCC1N(c1cc(=O)n(C)c(O)n1)CC2 c1(C(N2C(c3cn(CC(=O)NC)nn3)C(C)CC2)=O)ncnc2c(C)csc12 C1(C(N2CC3CCN(C(CS(N)(=O)=O)=O)C3C2)=O)CCOCC12CCCCC2 N1(C(C(CCSC)NC(=O)C(C)CC#N)=O)CC2CC(O)CC2C1 N1(C(=O)CN2CC3CC3C2)CCC2CN(C(c3ccn(CCO)c(=O)c3)=O)C2C1 c1(CC(C(=O)NCC(C)NC(C2(F)CC2C)=O)C)ccc2ccccc2c1 C1(CNC(c2c(CC)ocn2)=O)CN(C(c2nnccc2C)=O)CCC1(F)F C1(C(=O)NCC2CC2)COCCN1C(C1CCC(NC(Cc2cc(C)[nH]n2)=O)C1)=O N1(C(c2ccc(CC)[nH]2)=O)CCCC(Cc2cn(Cc3ncon3)nn2)C1 C(=O)(CCCC(C)(C)C#N)N(CCC(C(C)C)NC(=O)CC1=CCOCC1)C N1(C(COC(C)=O)=O)CCC(C)C(N(C)C(C2C=CC=CC=C2)=O)C1 C1(CC)(NC(C2CN(C(=O)OC)C2)=O)CCN(C(=O)Cc2cn[nH]c2)C1 C1(C(=O)NCCC2N(C(c3c(C)nc(CO)s3)=O)CCCC2)CCN(C)C(=O)C1 C12(C(N3CC(NC(C4(C)CC(C)(C)C4)=O)C3)=O)CCOC1CC(=O)NC2 C1(O)(CCNC(c2ccc(C#C)o2)=O)CCCN(C(c2c(C)ncnc2C)=O)C1 C(CCC(F)(F)F)N(C(C1(NC(=O)CCc2ccn(C)n2)C(C)C1)=O)C CS(=O)(=O)c1ccc(F)cc1C(c1nnnn1C(C)(C)C)NC1CC(=C2CC2)C1 C1(C(N(CCC)CC2CC2)=O)C(NC(c2ccc(CO)o2)=O)CC1O N1(C(C2N(C(Cn3ncc(C#C)c3)=O)CC(OC)C2)=O)CC2(COC(C)(C)C2)C1 c1(OCC#C)ccc(CN2CC(C(=O)NCC3CCCN(C)C3)C2)cc1 N1(C(C=CC)=O)CCCC(N2CCN(C(=O)C(=C3CCCCC3)F)CC2)C1 c1(OC)nc(C(N2CCCC2CN(C(=O)C(C)SC(F)(F)F)C)=O)ncc1F CC1(C)CCC(CNC(c2coc3c2CSC3)=O)N(CC(=O)NC2CC2)C1 N1(C(C(c2cccc(OC)c2)C(C)C)=O)C2CCCC1CN(C)C(=O)C2 C1(NC(CN(CCOC)C)=O)CC(F)(F)CC1NC(=O)CC(=O)NC1CC1 c1(CC(=O)NC2C(C)CN(C(c3nncn3C)=O)CC2)cccc2c1OCO2 C1(C)(CNC(C(CC)n2cccn2)=O)CCCN(C(C23CCC(CC2)CO3)=O)C1 Cc1ccc(C(=O)NC2CCCC2CNC(=O)CS(C)(=O)=O)c(O)n1 c1(C(N2CC(C)C(CNC(=O)CCF)CC2)=O)cccc2c1CC(=O)N2C C1(C)(NC(C(C)OCc2ccccc2F)=O)CCN(C(c2coc(Cl)c2)=O)C1 c1(CC(=O)NC2C(F)CCN(C(C3(C)CC3)=O)C2)ccc(F)c(Cl)c1F CC(C(=O)NCC(C)(F)CNC(=O)CC1OCCCC1(C)C)S(N)(=O)=O C1(CC(=O)NCC(C)NC(C2(c3ccccc3F)CCCC2)=O)CCC(C)(C)O1 C(c1ccc(O)cc1)=CC(=O)NCC1(O)CN(C(C2(CF)CC2(F)F)=O)C1 Cc1[nH]c(=N)sc1C(N1CCC1CNC(=O)CCC1CCC(=O)N1)=O c1(C(N2C(C)(C)CC(NC(c3csc(Cl)n3)=O)C2)=O)cc(Cl)cc(F)c1N C(CCC(C)C)(C(=O)NCCCOCC1CCC1)NC(CN(CC=C)C)=O.C1CC1 CC1(C(N2C3CC2CN(C(=O)Cc2cccc(C#N)c2)C3)=O)CCC2CC2C1 C1(C(=O)NC2CC(CCNC(Cc3c(OC)nccc3)=O)C2)OCC2CCCC12 CN1CCN(C(=O)NCCc2ccc(Cl)cn2)c2cc(Cl)ccc21 C(C)(CCCCNC(c1cc(OC)n(C)n1)=O)NC(CC=CC)=O CC(CCC(=O)N1CCCC(N(C)C(C2CS(=O)(=O)C2)=O)CC1)S(C)(=O)=O c1(C(CNC(C(C2CCC2)OCC)=O)NC(=O)CC)ccc(CC2CCC2)cc1 C(c1ccc(OC)c(OC(F)F)c1)=CC(=O)NCC(C)(C)NC(C(COC)O)=O c1(CC)cncc(CNC(=O)CSCCNC(C2(O)CCOC2)=O)c1 N1(C(C2(SC)CN(C(=O)CC3CCCC(=O)N3)C2)=O)CC2CC(O)CC2C1 N1(C(C(=O)NCC)=O)CC2CCCC(CNC(c3csc([N+](=O)[O-])c3)=O)C2C1 N1(C(c2ccc(CO)c(Cl)c2)=O)CCC2CCC(C1)N2C(=O)CC1CSC1 S(=O)(=O)(c1cccc(Br)c1)N1C2CN(C(c3c(CC)nccc3)=O)C(C2)C1 c1(C(=O)NC(C2N(C(c3cnc(C)[nH]3)=O)CCCC2)C)ccc2cncn2c1C c1(C(=O)NC23C(CN(C(C=COCC)=O)C2)CCC3)ccc(Cl)c2ncccc12 N1(C(c2ccc(C)n2C)=O)CCCCCC1C(=O)NC1CCCC(O)CC1 Cn1cc(Cl)c(C(c2nnnn2C2CCC2)Nc2cccc(CCCCO)c2)n1 C(=O)(CCS(=O)(=O)c1ccc(F)cc1)NCC(C)NC(C(CC)(C)O)=O c1(OC)cccc(C(=O)O)c1O.c12ccc(cc1)C(=O)N1CC(C1)N(C)C2 c1(OCC(N2CC(CC(C)NC(C(CC)SC)=O)C2)=O)cccc(Cl)c1C c1(CNC(C2C=C(C)CS2)=O)cncc(C(=O)NCC(C)(C)CN2CCCC2)c1 CC1=CCC(C(=O)NCCC2CCC(NC(=O)CC3CCN(C)CC3)C2)CC1 n1(CC)nc(C2CC2)cc1C(C(=O)NCc1ccco1)N1CCCC1 C(=O)(C(=O)C(C)CC)NCCn1ccc(C(=O)NCCN(CC(C)C)CC)c1 c1(C(N2CCC(N(C)C(C3CC4CCC3O4)=O)CC2)=O)ccnc2[nH]ncc12 C12(OC)CCC(C(=O)NCC3(CNC(=O)C(F)C(F)(F)F)CC3)(CC1)C2 N1(C(=O)OC(C)(C)C)CCCC(CC(=O)NC2CCC23CCC3)C1C c1(CC)cccc(C(=O)N(CC(O)CNC(C2(CC)CCC2)=O)C)c1O c1(NC)cccc(C(=O)NCC(C2CCN(C(c3ccns3)=O)CC2)F)n1 CCCCCC(C)(CC)C(=O)NC1CCN(C(c2cccc(C)c2O)=O)C1 CC1(CNC(=O)CP(C)(C)=O)CN(C(=O)C(=Cc2cccnc2)F)CCO1 N1(C(C2(CC=C)CC2)=O)C(C(=O)NC2(CO)CCCC2)CC1C c1(C2C(NC(=O)Nc3cnn(C4N(C(C(C)(C)C)=O)CCC4)c3)C2)ccccc1Cl C1(O)(NC(CC(=O)OC)=O)CCN(C(=O)C(=O)Nc2cccc(OC)c2O)CC1 O=C1N=C(C(=O)NCCCC2(NC(C3CCCC(F)C3)=O)CC2)c2ncccc21 C(=O)(C1Cc2c(Cl)cccc21)NCCNC(c1c(NS(C)(=O)=O)cncc1)=O C1(CC(=O)NCC(F)F)CCCNC1=O.C12OCCC1C(=O)N(C)C2 CC1=NN(C)C(=O)C1CC(=O)NC1CCN(c2nccc(C(F)(F)F)n2)C1(C)C S(=O)(=O)(c1cc(Cl)c(Br)cc1F)Nc1cccc(C(N2CC(C)OCC2)=O)c1 C#CC1(NC(=O)CC23CCC2CN(C(=O)C(O)C(C)C)C3)CCCOC1 Cc1cn2c(C(=O)NC3CC4CCC3N4C(C3CCCC3C)=O)cnc2s1 c1(NC(C2CC(F)CN2C(c2ccncc2Br)=O)=O)ccc(O)c(F)c1F C#CC1C(C(=O)NC(CCCC(c2ocnc2C2CC2)=O)C)C1(C)C c1(CCC(=O)NCCC2CCCN2C(=O)CCC2CC2)ccc(Cl)nc1 c1(C(N(CCCCCNC(C2(C(F)(F)F)CC2)=O)C)=O)ccc(N)c(N)n1 C1(NC(C2(C(=O)OC)C(=C)CC2)=O)C2CC1N(C(c1ccc(C3CC3)cc1)=O)C2 c1(C(N(CCOCCN(C(C2C(CC)C2)=O)C)C)=O)ccc2cc(F)ccc2n1 N1(C(c2cc(CC)sc2)=O)CCN(C(c2cnn(C)c2)=O)C(C)C1C C1(NC(c2[nH]c3c(C)cc(C)cc3c2)=O)CC(N=c2nc(C(C)C)[nH]s2)C12CCC2 C1(C(=O)NCC2C(C(N(CC(CC)OC)C)=O)C2)COCCO1 Cn1sc(C(=O)NC2CC=CCC2C(F)(F)F)cc1=O c1(C(=O)Nc2cc(C(=O)NCCc3c(C)ncs3)n(C)c2)cccn2nccc12 C1(N(C(=O)C(c2cccc(Cl)c2)C2CC2)CC)CCCN(C(=O)C=CCO)C1 c1(OC)ccc(=NC(=O)CC2CCN(C(c3ncc(C)cc3F)=O)CC2)[nH]n1 c1(CC)cc(C(=O)NCC(C)N(C(=O)C(C)(C)C2(O)CCOC2)C)nn1C C1(CC)(NC(C2(C)CC2(F)Cl)=O)CCN(C(CCC(=O)NC(C2CCC2)=O)=O)CC1 C(=O)(CCCCCC(C)(C)C)N(CCC(C)NC(c1n[nH]c(C)c1Cl)=O)C Cc1cc(NC(C23CSCC2C3)=O)ccc1NC(=O)CC(C)C1CCCCC1 N1(C(CCCOC(C)C)=O)CCN(C(=O)C(C)C(C)(F)F)CC1c1nccn1C C1(C)(CC(=O)NC(C2CC=CCC2)C(=O)N(CCN(C)C)C2CC2)CCCCC1 C1(N(C)C(C2CNC(=O)CC2C(F)(F)F)=O)CCCN(C(c2ccoc2)=O)CC1 C1(CNC(C(C2CC2)OC)=O)CC12CCN(C(=O)C(c1cccc(F)c1)F)CC2 N1(C(=O)CCF)CCCC(C2CCN(C(c3ccc(F)cc3)=O)CC2)C1 c1(C(=O)NCC(CC)NC(C2CC(SC)C2)=O)ccc2cc(O)ccc2c1 C(C(C)C(F)C(=O)NCC1CCC(C)(O)CC1)OC(C)C.C1CC(=O)N1 C(=O)(C(C)P(C)(C)=O)N(CC(CC)NC(c1nccnc1C)=O)C n1(CC(=O)NC2CCC(CNC(C3C(C)=C3)=O)C2)cccnc1=O CCC(C)(O)C(=O)Nc1cccc(NC2CCN(c3cc(OC)ncn3)C2)c1.C(N)=O Cc1cccc2cc(S(=O)(=O)OC(CC3CC3)Cc3ccccc3)sc12 c1(C(=O)NCC2(OC)CN(C(c3c(OCC)scc3)=O)C2)ccc(C)c(C)c1O N1(C(C(CNC(C)=O)(C)C)=O)CCCC(C2(NC(=O)C(C)(F)F)CC2)C1 C=CC1CN(C(c2sccc2Cl)=O)CC1NC(=O)C=Cc1cccnc1C C1(NC(c2ccc(C#N)o2)=O)CC(CNC(c2ncc[nH]c2=O)=O)C12CCC2 c1(CN=C(NCc2n(CC)cnn2)NC2CC2C)cccc(F)c1C#N n1(CC#C)cnnc1C(=O)NCCC1(NC(=O)CCc2ccccn2)CCC1 CC1(CNC(c2ccc(CNC(=O)CC3C=CCC3)nc2)=O)CC=CCC1 c1(C(=O)NCC2(OC)CN(C(c3n(CC)ccc3)=O)C2)cc2c(C)nn(C)c2s1 CCC(C)C(C(=O)NCC1(CC)CCOC1)N(C(=O)CCCCCOC)C C1(CC(=O)NC2(CC)CCCC2)CCN(C(C2C(C)C2C)=O)CC1 C1(C(F)C=O)(C(=O)O)CCCCC1.C1(O)(C(F)CN2CC(CC)C2)CCOCC1 c1(CNC(C2(C)CCN2C(=O)Cc2cncnc2)=O)ccc(O)nc1 Cc1ccc(C2(C(=O)NC3CC(N(C)C(C4CCCO4)=O)C3)CCCC2)cc1 c1(C(C(=O)NCC(C)(C2CC2)NC(CC2CC(=C)C2)=O)(F)F)cc(Cl)ccc1F c1(C(N2CCC(CNC(C3(C)C(CC)CCC3)=O)C2)=O)c[nH]cc(Br)c1=N C12(CNC(C(CN(C)C)NC(c3c(C)cco3)=O)=O)CCC(CO1)C2 C1(C(=O)NC2CCN(C(Cn3cnc(C#N)n3)=O)CC2)CC2C=CC1C21CC1 C1(NC(Cn2c(C)nc(C)n2)=O)CN(C(=O)CC2CCCN(C)C2)CCC1F N1(C(Cc2cc(C)nn2C)=O)CCOCC(NC(=O)COc2ccccc2F)C1 c1(N(C)C)ccc(C(=O)NCC2CC2CNC(=O)Cc2nccn2C)nn1 N1(C(c2c(C)n(C)cc2)=O)C(C(=O)NC2CCCC3(CC2)CC3)CC2CCCC12 CC1=C(C(=O)NCC2CCC(C(=O)NCC#CC3CC3)C2)CCC1 c1(C(N2C(CNC(CC(CCC)C)=O)CCC2)=O)cc(C(C)C)ccc1F O(C1CCCc2ccccc21)CC(N1C(CNC(CSCCC)=O)CCC1)=O CCC(C)CCC(O)CC(=O)N1CC(NC(c2cccnn2)=O)CC2(CCC2)C1 Cn1c(C(N2CCCCC(CNC(c3cnns3)=O)C2)=O)cc(Cl)c1Cl C1(C(N2CCC(OC)(CO)C2)=O)CCCC(NC(C2CNC(=O)N2)=O)CC1 c1(C(C)C(=O)NC2C3CN(C(=O)C=CC(=O)N(C)C)CC23)ccccc1N(C)C CS(=O)(=O)c1cnc(N2CC(NC(C3CCCC3)=O)CC3(CCC3)C2)c(Cl)c1 C(=O)(C1Cc2ccc(Cl)cc21)N1CCC(C)(CNC(C2CCC(=O)O2)=O)C1 c1(C(=O)NCCN(C(C23CCCC2(C(N)=O)C3)=O)CC)cc2ccncc2[nH]1 C1(C(=O)NC(C)CNC(=O)CN2CCCC(O)C2)CCC2(CCC2)C1 C1(NC(=O)CCc2cccs2)CCCC2(CN(C(=O)C(=O)Nc3ccccc3)C2)O1 Cc1cc(C(N2CC(F)CC2CC(N2CCC(OC3CCC3)C2)=O)=O)cnn1 CC1CCCCC1CNC(=O)C=CCN(C)C(c1ccoc1Cl)=O c1(NCc2nccc(SC)n2)c2c(cc3c1CCC3)CCC2 c1(C(N2CCC(N(C)C(c3cnn[nH]3)=O)C2)=O)c(N)cc(Cl)nc1Cl N1(C(C2C(C(=O)NCc3c[nH]c4cccnc34)C2)=O)CCCC2CCCCC12 N1(C(C(CC)=CCCC)=O)CC(CC(N2CC(c3cc(O)no3)C2)=O)CCC1C N1(C(C(C2CCC(=O)N2)C)=O)CC2(CCCCN2C(c2nn(C)c3c2CCC3)=O)C1 C(C)(c1ccco1)=CC(=O)N(CCOCCCNC(C(C1CC1)OCC)=O)C C1(CNC(C(C#C)(C)C)=O)(CO)CCCN(C(=O)Cc2cc(C)ccc2O)C1 C1(CN(C(C2(CCOC)CC2)=O)C)CN(C(c2cn(C(C)C)nn2)=O)CCO1 C1(C(N2C(C)CN(C(c3cc(=O)cc(Cl)[nH]3)=O)CC2)=O)CCc2nncn2CC1 c1(C(N2CC(O)(CN(C)C(c3cnnn3C)=O)C2)=O)ccc2cc(Cl)ccc2c1 C(CC(C)C(=O)c1ccc(C(=O)NCC=C)[nH]1)=CCC.C1COCCO1.OCC C1(NC(C(CC=C)(C)C)=O)C2CCC1CN(C(c1cc(F)ccc1O)=O)C2 C1(NC(CC(CNC(c2ocnc2C)=O)OC)=O)C2CCC(F)(F)C12 N1(C(CC)=O)CCC2CCN(C(c3ccccc3CC)=O)C(C)C2C1 C(=O)(C#CC1CCCC1)N1CC(CNC(Cc2cc(C)c(Cl)cc2)=O)C(F)(F)C1 N1(C(CNC(CC)=O)=O)CC(CNC(=O)C=C(C)C(C)(C)C)OC2CCCC12 N12CC3CN(C(=O)O)CC3C1C=C(C(F)(F)F)OC(C)(C)CC2CC(O)C(O)C CC1(C)CC(C(N2CCC(C(F)F)CC2)C(=O)NC(C)(C)C)CC(C)(C)O1 C(=O)(C#CC(C)(C)C)NC1C(CNC(c2n(C)ccn2)=O)C1 c1(C(N2CCCC(Cn3cc(CO)nn3)C2)=O)ccc(F)c2[nH]ccc12 C(=O)(CCCCCNC(C1(C#N)CC(C)C1)=O)NC1C(CC=C)COC1 c1(NC)ccc(C(=O)N(C(C)CN(C)C(C2CCN(S(C)(=O)=O)C2)=O)C)nc1 c1(CC(=O)NCC(C(C)C)NC(CC2(C=C)CC2)=O)ccc(F)cc1Cl CC1(CNC(C2(c3cccc(Cl)c3)CC2)=O)CCN(C(=O)CN2CCNC2=O)C1 Cn1cc(CCNC(C2(CCNC3CC=CC3)CC2)=O)n(C)c1=O C1(NC(C)=O)CCC(C(=O)NC2CCCC(C(=O)NC(C)(CO)CCF)C2)CC1 Cc1c(CC(=O)NCCC2CC(NC(C3CC4CCC4C3)=O)C2)cnn1C C=Cc1cc(C(=O)NC2CCN(C(C34CCC(CC3)C(C)O4)=O)C2)cc(F)c1 N1(C(c2nc(C(C)C)sc2)=O)CCC2CCN(C(=O)C#CC3CCCCC3)C2C1 O=C(CC1CCCCC1)CCC1CCCC1.N12CCC(C1)C2 c1(C(N2CCC(OCC(N3CCC(CCC)CC3)=O)C2)=O)ncc(F)cc1N CN1CC=CCC1CC(N1CCCCC1CCNC(c1cc(C(N)=O)c[nH]1)=O)=O N1(C(C(C)C2CCCO2)=O)CC(NC(=O)CCS(C)(=O)=O)C(C)(C)C1 c1(C(=O)NC2CC(CCNC(C(COC)O)=O)C2)cnc2c(c1)CNC(=O)N2 CCC(C(C)C)NC(=O)C(C1CCCO1)NC(=O)CNC(N)=O C1(CC)CCN(C(=O)OC)CN1C(=O)C(F)CC1CN(C(=O)CCCNC(C)=O)C1 Cc1cc(C(=O)NCCOCCN(C(=O)CCC2CC3CCC2C3)C)ccc1Cl C(CCC(C(=O)NCC(C)CC(F)(F)F)NC(=O)CC(O)C1CCCC1)OC C(=O)(CCC(=O)NC1(CNC(=O)CCc2nc(C3CC3)no2)CCOC1)N(C)C CCCCC(C)CCC(=O)NC(CC(=O)NCCOCCCO)C(N)=O N1(C(CCCCN(C)C)=O)CC(NC(c2n[nH]c3c2COC3)=O)C2(CC2)C1 C(=O)(CCCC(F)F)NCc1ccc(CNC(c2ccc(C#C)o2)=O)cc1 c1(CC(=O)NC2(CF)CCN(C(CCN(C(CC)CC)C)=O)C2)noc(C)c1C#N C1(CSC)CCCN(CC2CCN(c3nncs3)CC2)C1 N1(C(c2ncn(CC)c2)=O)CCC(C(=O)NC(c2ccsc2)C)(OC)C1 N1(C(C2(CNC(c3ccc(C)cc3C)=O)CC(=C)C2)=O)CCOCC(CO)C1 n1(CCC(=O)NCC(c2cc(Cl)ccc2F)(F)F)nc2ccccn2c1=O C(=O)(CCC(F)(F)F)NCCCN(C(c1cc(C)cc(C)n1)=O)CC N#CC1CCCN(C(C2C=CCN(C(c3ccoc3C3CC3)=O)C2)=O)C1 C(=O)(C(F)(F)C(F)(F)F)NC1CCC(NC(c2ccc(OC)cc2OC)=O)CC1 Cc1cc(CC(=O)NCC2CCN(C(=O)CC3CCCC3)C(C)C2)ccc1Cl C1(C(=O)NC(CN(CCCC)CC(C)C)C)CCN(CCOC)CC1O CC1CCCN1CC(=O)NCC(C)=CC(N1CCCC1CCO)=O C(CCCC(c1nnnn1CC(F)F)NCCc1c(C)noc1C)(OC)OC C1(NC(CCC(=C)Cl)=O)CCCN(C(=O)C(C)CCCc2ccccc2)CC1 CON(CCC(=O)N1CC=CC(O)C1)C(=O)Cc1cnccn1 C12(CCNC(CCN(CC)CC)=O)CCC(C1)N(C(c1cc(C)nc(C)n1)=O)C2 CCC(CC)(CC)C(=O)NCC(CC(=O)NCc1ccnc(OC)n1)OC C1(NC(=O)C=Cc2ccc(Br)o2)C2CCC1N(C(c1ccn(C(F)F)n1)=O)C2 c1(C(=O)NC(CCCC)CNC(c2cnc(C(C)C)[nH]2)=O)n[nH]c2cccnc12 c12cc(c(C)c(Br)c1)OC2=O.c1(NC(=O)NCC)cc(Cl)ccc1C(=O)OC C1(NC(c2ccccc2C(F)F)=O)CC2CCC1N(C(=O)CCOC1CCC1)C2 N1(C(C(C(C)=O)(F)F)=O)CCCCC2(CCCCN(C(=O)CCSC(=N)N)C2)C1 C(C(N)=O)(C(C)C)SCC(C(=O)c1ccccc1)NC(CNC(C)=O)=O c1(C(=O)NC(CNC(c2ncc(C)cn2)=O)C(C)C)ccc(O)cc1C c1(C(N2CCC(C(=O)NCCC=C=C)CC2)=O)cncc(C=C)c1 CC(C)C(CNC(c1cc(F)ccc1F)=O)C(=O)NCC1(CCO)CN(C)C1 C1(CC(N2CCC(N(C(c3cc(OC)ns3)=O)CC)CC2)=O)CCCC2(CCC2)O1 Cc1c(C(=O)NC2(CO)CCCN(C(=O)CC(C)O)C2)sc2ccccc12 C1(C(=O)NC(CSCC)C(=O)NCC2=C(C)CC2)CCOCC1(C)C CC1(C)CCOC1CC(=O)NCC(=C1CN(C(C2CCC(C(N)=O)O2)=O)C1)F c1(C(=O)NC2C(CNC(C(COC)O)=O)CC2)cccnc1N c1(NC(C(C2CCN(C(c3ccc(C#N)o3)=O)C2)C)=O)ccc(F)cc1CO N1(C(C2C(C)C2(F)F)=O)CC(C2(NC(=O)CCSC3CCCC3)CC2)C1 C12(NC(=O)CCCc3cccnc3)CCCC1N(C(=O)Cc1cscn1)CC2 c1(C(=O)NCC2(F)CC(NC(c3c(OC)csc3)=O)C2)nccn2nc(C)cc12 c1(OC)ccc(N2CCC(Oc3ccccc3S)CC2)nn1.C1CCC1 C(CCCC(=O)N1CCCC1CC(=O)NCCCc1ccnn1C)(OC)OC O=C(CCCC(F)F)NC1CN(C(=O)CNC(c2ccc(O)cc2)=O)C2CC12 CC#CCC(C(=O)NCCN(C)CCF)NC(C1(OC)CCSC1)=O C1(OC(=O)NCC2N(C(=O)NCC)CCCC2)CCc2n[nH]cc2C1 C1(CC(N2CC(C)(NC(c3ccc(COC)o3)=O)C2)=O)CCC2(CC1)OCCO2 C#Cc1ccc(C(=O)N(C(C)(C)CC(=O)NCC(C)(C)C(C)C)C)o1 n1(CC)nc(C(=O)NC2C3CCC2N(C(c2ccnc(O)c2)=O)C3)ccc1=O c1(C(=O)NC(C2(O)CCN(C(C3CCC(OC)CC3)=O)C2)C)c[nH]cc(Cl)c1=O C(=O)(CCC=CBr)N1C(CN(C(c2cc3n(c2)CCC3)=O)CC)CCC1 C1(N(C(CCN(c2ccccc2)C)=O)C)CN(C(C2CC=CCC2C)=O)CC1O C1(NC(c2ncc(OC)cn2)=O)COC2(CCN(C(=O)C3=C(Cl)CCC3)C2)C1 CCCCC(CC)C(=O)N1CCN(C(=O)CC2(OC)CC2)C(CO)C1 c1(CC(=O)NC2(C)CC(N)C2)ccccc1N N1(C(CNC(C)=O)=O)CC(C)(NC(C2=NC=NCCN2)=O)C1 N1(C(CCC#C)=O)CC2CC(NC(c3cnc(-c4ccccc4)[nH]3)=O)C1C2 C1(CNC(C=NOC)=O)C2CN(C(=O)C(=O)NCCOC3CC3)CC12 CC1CCCCC1(CNC(=O)CNS(C)(=O)=O)NC(C1CCCC1F)=O C(CN=c1cc[nH]cc1S(=O)(=O)NCc1ccc(CSC)o1)OCC(F)(F)F C(CN=C(NC(C1CN(C)CCO1)C)NCC(=O)NC(C)(C)C)OCC=C C1(NC(C=Cc2ncn(C)c2)=O)CN(C(C2CC(F)C(=O)N2)=O)CC1(C)C c1(C(N2CC(O)(CN(C(CSCCOC)=O)C)C2)=O)cnn2ccccc12 Cc1cccc(C)c1CC(N1CCCC(CNC(c2ccns2)=O)C1)=O C1(NC(CC2CC(=C)C2)=O)CC2CC1CN2C(=O)C(c1ccc(F)cc1F)=O C(=O)(CCCCC(N)=O)NCCC1(C)CCN(C(c2nc(Cl)cs2)=O)C1 C(=O)(C(CC(F)F)NC(C1CC(C2CC2)C1)=O)NCC(C)(C1CC1)OC.C1CC1 c1(OCCC)ccc(F)cc1NC(c1cc(C2CC2)ccn1)c1nnnn1C c1(NCC2(OC)CCCCC2)nc(N2CCCC2)nc2ncn(C)c12 Cc1ccc2c(c1)C(C(=O)N1CCCN(C(C3CC4(CCC4)C3)=O)CCC1)C2 C12(NC(C(=Cc3ccco3)C)=O)CCC1CN(C(c1cccc(F)c1C)=O)C2 N1(C(C(=O)N(C(C)(C)CC(C)C)C)=O)CCC(F)(F)C(C(F)(F)F)C1 c1(NCCC2CCCN(C(C3(CO)COC3)=O)C2)ccc2nnnn2n1 c1(C(=O)NCC(C)(C)OC)cc(C(=O)N(CCN2CCCC2)CCSC)c(Cl)cn1 S(=O)(=O)(c1cc(C(F)(F)F)cc(F)c1)NC(c1ccc(Cl)cc1)C(=O)OCC C1(C)(C(N(CC)Cc2ccc(Cl)cc2Cl)=O)COC(=O)N1C C1(CNC(c2ccc(C)o2)=O)CC2CCC(C1)N2C(=O)CNc1ccccn1 CC1=C(C(=O)NCC(CNC(=O)C(O)Cc2ccccn2)OCF)CCCO1 c1(C(C)COC)ccc(Oc2ccccc2)nc1OCC1CC1.C1(CCN)CCC1 c1(CNC(CC2C(=O)NC(=N)S2)=O)cc(O)nc(CNC(=O)CC2CC=CC2)n1 C(=O)(CC1CCOc2ccccc21)NCCN(C(COCc1onc(C)n1)=O)C N1(C(c2cc(C)sc2)=O)CCN(C(c2cc(F)c[nH]2)=O)CC1CC(F)F c1(COCC)ccccc1.C1C(CO)O1.C1CO1.C1CO1.C(CO)NC(C)C C(=O)(CC(C(C)(C)C)NC(c1ccc(CO)o1)=O)NC(C)CSC(F)F C=CC1(C(=O)N(C)CCOCCNC(C2(C(C)(C)O)CCCCC2)=O)CCCCC1 C(=O)(CCCC(=O)N1CCCC(C)(CNC(c2nc(Cl)cs2)=O)C1)OCC c1(C(N2CC(NC(C=CCC)=O)C3(C2)CC3)=O)cc(C)c2ccccc2n1 C(=O)(C(CNC(C1CCCNC1=O)=O)CC1CC1)NC1C=CC(CC(=O)OC)C1 CC(C)CCC(=O)C(=O)N1CC(NC(=O)CCn2ncn(C)c2=O)C2(CCC2)C1 C1(C(N(C(CN(C(C)=O)C)C)C)=O)CCN(C(C2C=C(C)CS2)=O)CCO1 c1(NC)cnncc1C(=O)NCCC1CC(NC(c2cc(C3(C)CC3)n[nH]2)=O)C1 C1(NC(CC=C=C)=O)CCCC(C(=O)NOCc2ccccc2COC)CC1 CC1(C(N2CCCCC(CNC(=O)CC3CCOCC3)C2)=O)CCCNS1(=O)=O N1(C(C2CN(C(=O)NCC=C3CCCCC3(C)C)C2)=O)CCN(CC)C(C)(C)C1 N1(C(CCC(C)OC)=O)CCCC(O)(Cn2cc(CC(C)(C)C)nn2)CC1 c1(C(=O)NCC2CC(NC(C(CC)OC)=O)C2)ccn2c(C(F)(F)F)nnc2c1 c1(C(C(=O)NCC(F)F)N(CCC)CC2CCSCC2)cc(OC)c(F)c(F)c1 c1(CCC(=O)N(CCCN(C(C(C)SCC)=O)C)C)c(C)nc2ncnn2c1C CC1C(NC(C2CCCC3CC23)=O)C(C)CCN1C(C1CC(C)(F)C1)=O C1(C(N2CCC(O)(C(C)NC(COCCCC#C)=O)C2)=O)CCCC(=O)N1C N1(C(Cc2n(C)ncc2Cl)=O)CC2CC1CCC2NC(=O)COC1CC=CC1 C#CC1CCC(NC(=O)C=CCC(C)(C)NC(c2cnncc2C)=O)C1 O=C(C(C1=NOC2(CCC2)C1)N1CC2CC=CCC2C1)NCC1CC1 C(CCCCC(=O)NC1CCCCC1F)N(C(CN(C(C)C)C)=O)C C1(C)(CC)CC(NC(=O)Cn2cc(-c3cncc(F)c3)nn2)CN1C(=O)C1CC1 CCCCCC(O)C(=O)NC1CCC1CNC(c1ccc2ncnn2c1)=O N1(c2cc(NCc3cccnn3)nc(COC)n2)CCCC2(CCC(=O)NC2)C1 C12(NC(C=C(C)C)=O)CCCC(NC(C3CCC(C(C)(C)C)O3)=O)(C1)C2 CCCCCCCC(=O)N1CC(C)(C)CC1CNC(C1CCCC(C)(C)C1)=O N1(C(CCCCN(C)C)=O)CCC(C(N2CCCC(F)(F)CC2)=O)CC1(C)C Cc1cc(C(=O)NC(CC(=O)NCC(c2cnc[nH]2)C)CC(C)C)ccc1C#N c1(C(=O)OC)cc2cccc(OC)c2[nH]1.C123C(C1)(C2(F)F)NC3=O C(=O)(C(O)CCCNC(=O)C(C)(F)n1cccc1)NCC1CCCN(C)C1 c1(NC(C(=O)NC(CCNC(C23CC(OC)C2C3)=O)C)=O)cc(C)cc(C)c1 Cc1ccc(C(N2CCN(CC(F)F)CC(O)C2)C(=O)NC=O)c(F)c1F N1(CC(=O)NCCCC(C)(C)NC(CC2(OC)CC2)=O)CCCCCC1=O N1(C(C(C(C)C)n2ccc(C)c2)=O)CCN(C)C(CNC(=O)Cn2ccnn2)C1 CCC(CC)CCC(=O)NCC(C)(CNC(=O)C(CC)C1CCOCC1)OC c1(OC)nccc(C(=O)N(CC(C)NC(C2CCN(C)C2)=O)CC)c1Br CC1=C(C)CC(C)(NC(C2(NC(=O)CC3C=CCC3)CCC2)=O)CC1 N1(C(CC(C)SC)=O)CC(C)OC2(CCN(C(=O)C(C)(C)N3CCCC3)C2)C1 CC1(C)CCC(NC(=O)C(N)=O)C(CNC(=O)CCC(=O)c2cccs2)C1 n1(CC(=O)NC2C3CCN(C(C(CC=CC)C)=O)C32)c(=O)oc2ccccc12 c1(-c2n(C3CC(C)N(C)C3)ccn2)cccc(C#N)n1.c1(S)cccc(=S)n1O C1(N(C(=O)Cn2nc(C)c(Cl)c2C)C)CCCN(C(=O)C=CC=C(Cl)Cl)C1C n1(CC(C)C)cc(NC(=O)CCSCCCNC(=O)OC(C)(C)C)c(C)n1 N1(C(COC(C)=O)=O)CCCC1CCNC(=O)C(C)CO c1(C(N(C2CCN(C(C3CC4(CC4)C3)=O)C2)C)=O)cnn(Cc2ccco2)c1 Cc1cc(C(=O)NCC2(O)CN(C(=O)CC3CCCOCC3)C2)c(F)cc1F C1(NC(c2ccnc(CC)n2)=O)CCCN(C(=O)Cn2c(C)ccc2C)C1CC N1(C(C2COC2)=O)CCCC1C1(C(=O)NC(C2CCCC2)CO)CC1 CC1(C)CCCOC1CCNC1(C)CCCN(c2cc(C=O)ncn2)C1.C(N)=O N(C(=NCCN1C(=O)COc2ccccc21)NCc1ccccc1F)C(C)CF c1(CNC(N2C(C)CN(C(=O)OC(C)(C)C)CC2)=O)ccc2ccccc2c1 Cc1ccc(-n2cc(C3CCCN3C(C3CCCCS3(=O)=O)=O)nn2)c(F)c1 N1(C(CN)=O)CCC(CN)(CF)C1.c1(C(=O)N)cccc(NC(=O)NS(C)(=O)=O)c1 C=C(C)CC(C(=O)OC)N(C(c1cc(F)ncc1F)C(=O)NCCCOC)C C(=O)(C(F)CC(C)(C)NC(=O)C=Cc1ccncc1)NCc1c(CC)cccc1 C1(NC(C2(C)CC2Br)=O)CC2CCC(C1)N2C(C1CC12CC2)=O c1(C(N2C(CCNC(C(CCCOC)C)=O)CSCC2)=O)ccc2ccnn2c1 N1(C(CCCC(C)NC(=O)CCC2CCCCC2)=O)CC(=O)N2CCCC2C1 CP1(=O)CCN(CC(N2CC3CCN(C(=O)CCCCC(N)=O)C3C2)=O)CC1 C1(F)(CNC(c2c(OC)c(F)ccc2)=O)COCCN(C(C2C3COCC23)=O)C1 N1(C(CC(C=C)CC)=O)CC(NC(=O)COC2CC=CC2)CC12CCOCC2 CCCCC(C(=O)N(C1CCN(C(c2nc(Cl)sc2Cl)=O)C1)C)NC(N)=O c1(C(N2CCCC(N(C(=O)CCC(=O)NC)CC)CC2)=O)cc2c(nn1)CCC2 C1(CNC(Cc2cc(C)ns2)=O)CC(O)CN1C(C1CC1c1cccs1)=O C(CC(C(=O)N1CCC(O)(CCO)C1)NC(C1CC(C)C1)=O)=CC C1(CN(C(=O)Cn2ncccc2=O)C)CN(C(C2CN3CCC2C3)=O)CCO1 c1(C(=O)NCCCC(C)NC(=O)CCC2CC2C)c[nH]c2c(C#N)cccc12 CCC(C)(C)C(C(=O)NC1(C)CC1)N1CCC(C(O)C(F)(F)F)C1 c1(C(=O)OC)cc(NC(C2CCCC(C(F)F)CC2)=O)ccc1OC c1(C(=O)NCC2(CN(C(=O)CC3CCCN3C)C)CC2)cccc(N)c1O N1(C(C2CCN(C(C)C)CC2)=O)C2CCC1CN(C(=O)CNS(=O)(=O)N(C)C)C2 CC(C(C)(C)NC(C1CSCCS1)=O)NC(=O)CSCCN(C)C CC1CCC=C1C(=O)N(C1CCC1)CCNC(C1CCCOC1C)=O C(c1ccc(C)c(Cl)c1)=CC(=O)NCCC(CNC(c1cc(SC)oc1C)=O)O C1(N(C(=O)CSc2cnn(C)c2)C)CCOCC1NC(C1CCN(C(N)=O)C1)=O C(C(=O)NCCC1CC(NC(=O)COC(F)F)C1)(C(C)C)SC c1(C(=O)NCCC(=C)CNC(=O)C(C)OC2CCCC2)ncnc(O)c1Cl C(=O)(CC(C)C(=O)NCC1(CNC(c2cc(C(C)C)n(C)n2)=O)CC1)OC C1(Cl)(C(N(CCCCN(C(=O)C(F)C2CCCC2)C)C)=O)CC1(F)F Cc1nsc(C(=O)NC2(CF)CN(C(C3CCOCC3)=O)C2)c1N CCC(CC(F)(F)F)NC(c1[nH]nnc1C)c1nnnn1C1CCCC1 C1(CC=C)(C(=O)Nc2ccccc2C2CC(N(C)C)C2)CNCCO1 C1(C(N(C2CN(C(c3cscn3)=O)CC2O)C)=O)CC2(CCC2)CCO1 c1(C(C)C)ccc(C(=O)NCCC(O)CNC(C2CC(C(N)=O)C2)=O)cn1 Cc1cncc(C(=O)NCCC(C)CCNC(C2(C3CCCO3)CCCC2)=O)c1C N1(C(CC(C(F)F)NC(C(CC)O)=O)=O)CCC2(CC1)CN(C)C2 C1(NC(CCC(C)SC)=O)CCC2CCN(C(=O)C(C)SC(F)(F)F)C1C2 Cc1nnsc1C(=O)NCC1CCC(NC(c2cc(-c3cn(C)nn3)on2)=O)C1 Cc1cc(N2CCOC(CF)C2)nc(=NCCCOCC2CC2)[nH]1 c1(C(=O)NCCC2N(C(c3n(CC)cc(Cl)c3)=O)CCC2)noc2c1CCCC2 CCC(C)C1C(=O)N1CCCNC(C)=O.c1(C(=O)OC)c[nH]c(=NC)o1 N1(C(CC(=C)C)=O)CC2(CC(NC(=O)C(C)(C)C3CCOC3)CO2)C1 Cc1coc2ccc(C(=O)NCC(C3CCN(C(C4CCSC4)=O)C3)(C)C)cc12 c1(CCC)cnnc(C(=O)NC2(CNC(C3C4CC4C4CC34)=O)CC2)c1 C(=O)(C1=CCCCCC1)NCC(CNC(C1(CC)CCCO1)=O)(C)O Cc1cccc(C(N2CC3(NC(C4CCC(=O)N4C(C)C)=O)CCC2C3)=O)c1Cl C(CCO)(C(F)F)NC(C1CC(F)CN1C(c1cnc[nH]c1=N)=O)=O C(=O)(C(C(=O)N1CCC(F)(C(=O)NCC2CN3CCC2C3)C1)OCC)OC c1(NC(C=Cc2c(C)nccc2)=O)c(F)cc([N+](=O)[O-])cc1F c1(C(N2CCN(C(C3CC3(F)F)=O)C(C3CCCC3)C2)=O)ccc2nsnc2c1 C12(CNC(CN(CCOC)C)=O)CC(CO1)N(C(=O)CN(S(C)(=O)=O)C)C2 N1(C(C(CCC)C)=O)CCCC(C)C1CNC(=O)CCNC(=O)OC C(C(CN=c1[nH]c2c(c(=NCC3CCCN(C)C3)[nH]1)CCC2)OC)OC c1(CCCOC)cn(CCC2CN(C(=O)CN3CCOCC3)C2)nn1 C1(CNC(CCc2ccc(C(=O)OC)[nH]2)=O)CCC(C)N(C(=O)C=CBr)C1 n1(CC)c(C)nn(CC(=O)NCC(CO)NC(=O)C(O)CCSC)c1=O Cc1cnc(C(=O)NCC(C2CCCN2C(=O)C(C#N)C2CC2)(C)C)cc1C N1(C(c2cnn3ccsc23)=O)CCC2CN(C(=O)C3CC3)CCC2C1 c1(CNC(=NCCCOC(C)C)NC2CC(F)(F)C2)nn(C)cc1S(N)(=O)=O Cc1nsc(N(C(C)CNC(C2CCC(=O)NC2)=O)C)c1C#N C(=O)(CCCCC(=O)NCC12CC1CN(C(C1(c3cncs3)CC1)=O)C2)OC C(C(C)C(C)C(=O)NCC1(CNC(=O)CCc2cccc(C)c2)CC1)OC C1(NC(COCC(C)(C)C)=O)CN(C(c2cccc(C(F)F)c2Cl)=O)CC12CC2 C#CCCCC(=O)NC(C)(C)CN(C)C(c1cc(C)n(-c2ccccc2Cl)n1)=O CON1CCC(C(=O)N(CC(=O)NC2CC2C(F)(F)F)C)CC1 C1(CCCC)CN(C(=O)CCCSC)CCN1C(=O)CNC(=O)CCC c1(C(=O)NC2C(NC(=O)Cn3cccnc3=O)CCCC2)cnc2c[nH]nc2c1 C(C(O)C(C)(C)C)c1cn(CC(=O)N(CC(C2CCCC2)C)C)nn1 N1(C(C(N2C(C)CCC2C)C)=O)C2CCCC1CC(NC(c1ccccc1Cl)=O)C2 N1(C(c2c(C)c[nH]c2)=O)CCC2CC12C(N1CCC(CCO)CC1)=O N1(C(c2c(C#N)ccs2)=O)CC(NC(=O)C=Cc2nccs2)C(N=[N+]=[N-])C1 N1(C(C(C)c2ccsc2)=O)CSCC1C(=O)NC(c1ccncc1)C c1(C(=O)NC2(CNC(C3CCCN(CC(C)C)C3)=O)CCC2)cc(=N)[nH]c(Cl)n1 C12(NC(=O)C3=CCOCC3)CCCC1N(C(=O)CCc1nc[nH]n1)CCC2 C#Cc1cc(F)cnc1NC(C1CC12CCN(Cc1ccc(CO)o1)C2)=O c1(C(=O)NC2(CNC(C(C(C)(C)C)OC)=O)CCCCC2)cncc2nc[nH]c12 C1(N(C(COCCC=C)=O)C)CCC2CN(C(=O)CC3CCCCN3C)CC12 C1(CNC(CCNC(C2C(C)C2)=O)=O)CN(C(C23CSCC2C3)=O)CC1(F)F c1(C(N2CCC(NC(c3ncnc(O)c3Cl)=O)(CO)C2)=O)cnc2ncccn12 CC(C)C(C)(O)C(=O)N1CC2CCC2(NC(C23CC(F)(C2)C3)=O)C1 C(=O)(CC(C)N=c1[nH]c2c(c(=NC(C)CCSCC)[nH]1)SCC2)N(CC)CC Cc1ccc(C(=O)N(CCC(=O)NCCC(O)C2CCC2)CCO)s1 CCCCCCCCCCCC(=O)N1CCCN(C(=O)CC2CCCC2)C(CO)C1 C1(NC(C(C)OC(C)(C)C)=O)CN(C(=O)CCCCC2CC2)CC1(C)C Cc1cc(C)c(CNC(=O)C(c2ccnn2C)NC(C2CC(=C3CCC3)C2)=O)s1 N1(C(C=C(CNC(C)=O)C)=O)CC(C)CN(C(=O)C(C)(C)NC(C)(C)C)CC1C C(=O)(C(C)(C)COCC(F)F)NCC(CCOC)Nc1cscc1C c1(C(=O)NCC=CCC(=O)N(C(CC)CC)CC)cnc(C)c(C)c1 CN1CCCCC1C(=O)N(C1CCCN(C(=O)CN2CCNC2=O)C1)C c1(OC)cncc(NC(=O)CN2CCC2CNC(=O)C(O)CN(C)C)n1 N1(C(C2CCC(NC(C(C)N(CC(F)(F)F)C)=O)CC2)=O)CC2CC(F)CC2C1 N1(C(c2c(C(C)C)noc2)C(=O)NC2(C)CC2)CCCC(COC(F)F)C1 C1(C(=O)NC(C)COC(F)(F)F)CC2(CCC2)CN1C(=O)C1=CCN(C)C1 N1(Cc2c(C)non2)CC2CC1CN2C(c1ccc(C(F)(F)F)o1)=O C1(NC(c2c(C)nsc2)=O)CCC(N(C(=O)Cc2ccsc2Cl)C)CC1 Cc1nn2c(C(=O)NCC3(O)CCN(C(=O)C=Cc4cscn4)C3)c(C)nc2s1 CC1CCN(C(c2ccccc2OCC(F)(F)F)=O)C1CNC(=O)C(C)(C)CF C#CCC(C)C(=O)N1CC(CCNC(=O)CC2(C(F)F)CC2)C(C)C1 C1(c2cn(CC3CN(C(c4conc4C(C)C)=O)C3)nn2)(OCC)CCCCC1 C(=O)(CCCCCCN=[N+]=[N-])NC(C)CN(C)C(c1cc2ncccc2s1)=O C1(C(=O)OC)CCc2sc(NC(c3cncc(C(C)(F)F)c3)=O)nc2C1 C1(NC(C2CC(Cl)(Cl)C2)=O)CC2CCCC(C1)N2C(=O)Cn1nccn1 N1(C(C2CCC(=O)C2)=O)CCC2CC(CNc3cc4nncn4cn3)CCC2C1 CC1(C)CCN(C(=O)C2=CC3C=CC2C3)CC1C(N1CC2(CCOC2)C1)=O CCC(F)(C(=O)OC)C(=O)N1CCC(CCNC(=O)CCCSC)C(F)(F)C1 C1(NCc2nnc(-c3ccc(C)cc3)o2)CCSC(C)(C)C1 N1(C(C2(C(=O)NC)CC2)=O)CCC2(NC(C3(O)CCC(CCC)CC3)=O)CCCC12 c1(CN2CC(C)(C(=O)NC3CC(O)C3)C2)cc2ccccc2cc1O C1(O)(C(C)NC(=O)Cc2c[nH]nc2O)CCN(C(C2CCNC(=O)C2)=O)C1 CC1OC2(CO)CC1(C(=O)NCC1CN(C(C3CC3(Cl)Cl)=O)C1)C2 N1(C(CC2CN(C(C)=O)C2)=O)CCCC(NC(c2cc(C)cc(C)c2)=O)C1C CC1CCC(NC(c2cncc(N)c2)=O)CN1C(c1ccccc1O)=O n1(CC(N2CCCC(CNC(c3c(C)ncnc3)=O)C2)=O)nc(C)c(Br)c1C C1(CN(C(N(C)Cc2cn(CC)nc2C)=O)C(C)C)CCC(C2CC2)C1 c1(C(=O)NC2C(NC(C(CC=CCC)C)=O)COCC2)cc(C)c(Cl)cc1OC C1(c2nc(C)nn2CCN(C)C)CCC2(CC1)CC(O)C2 c1(C(=O)NC2CCC(C)N(C(c3ccccc3Cl)=O)C2)cc(C#N)c(O)nc1N C(C(=O)N=c1cc(CC)n(C)[nH]1)NC(C1CC(NC(C2(CO)CC2)=O)(OC)C1)=O c1(C(=O)NC2C(CNC(c3n[nH]c4ccccc34)=O)C2)cccc2sncc12 N1(C(C(CC(C)C)C)=O)CCC(C)(C)C(CNC(C2CCN2S(C)(=O)=O)=O)C1 C1(C(N2CCC(NC(CCSCCC)=O)CC2C)=O)CCCC12CCOCC2 CCCC(C)CCCC(=O)NC(C1CCN(C(=O)C2=NOC(C)(C)C2)CC1)C c1(C(=O)NCC(C2CCCCC2)NC(CC(C=C)C)=O)c[nH]c(=N)nc1CC C1(CN(C(C2C(CNC(c3cn(CC)nn3)=O)CCC2)=O)C)OCCC1(C)C c1(C(=O)NCCCCn2cc(CC(C)(C)OC)nn2)cccnc1S n1(CC(C)C)cc(C(=O)N(C2CC(NC(c3ccco3)=O)C2)C)c(C2CC2)n1 Cc1nc(C(=O)NCC2CCCCN2C(c2ccc(C(F)F)cc2)=O)ccc1Br N1(C(C)=O)CCC(C)(NC(C2CCN(C(c3cc(C)c(Br)s3)=O)CC2)=O)C1 c1(C(=O)NCCNC(C2CCC(C)(CC)O2)=O)ccc2c(c1)NC(=O)CN2C C1(C(=O)NC2(CF)CCN(C(c3nccc(N)c3)=O)C2)CCc2ccnn2C1 C1(C(C(N2CC(CNC(=O)Cc3cncs3)C2)=O)O)CCCCCC1 N1(C(CC(=C)Br)=O)CCOC(CNC(C2C3CC4C(C3)C24)=O)C1 N1(C(C2C(O)CCN2Cc2cnccn2)=O)CCN2CCOCC2C1 C(CC(C(C)(C)C)NC(=O)C1=CCCS1)N(C(C1C(C)OCCC1)=O)C Cn1nc(C(N2CC=CCC2C(=O)NCCc2ccnn2C)=O)cc1Cl C1(C(=O)NC(CNC(COCc2cc(C)on2)=O)(C)CO)CCCC(C)C1 C1(C(N2C(C(=O)NCC3(CO)CC(=C)C3)CC2)=O)CCC2(CCC2)O1 CC1(NC(C2COCCO2)=O)CCN(C(c2ccc(Cl)s2)=O)C1 N1(C(C(CCC)C)=O)CCC(COC)(NC(c2nn(C)c(C)c2Br)=O)CC1 c1(C(=O)NC2CC(NC(c3c(OC)nc(C)cc3)=O)C2)cc(C)ccc1[N+](=O)[O-] CCC(F)(F)CC(=O)NCC1(F)CN(C(=O)C=CI)C1 N1(C(c2cnn(CC)c2Cl)=O)CCN(C(c2ncnn2C)=O)CC1C C1(NC(=O)NCCN2CCC(CCC)C2)OCCC(N)C1O C(=O)(C(CC)CC(F)(F)F)N(CCC)CCNC(=O)COCC1CCCOC1 c1(C(N2CCC(NC(c3c(OC)nccc3)=O)CC2)=O)c(F)ccc2ccoc12 C1(C(=O)NC(C)COC(F)F)CCCN1C(c1ccc(CO)s1)=O c1(C(=O)NCC(C2CC2)NC(C2CCC=CCC2)=O)ccnc(O)c1F C1(NC(CS(=O)(=O)NCC)=O)CC2CCC1(NC(=O)CCNc1ccccn1)C2 C1(O)(CNC(c2ocnc2C2CC2)=O)CCN(C(C2CC3CCCC23)=O)CC1 c1(N(C(=O)C(C)OC)CCOC)cc(OC)cc(OC)c1 C1(C(=O)NC(C(C)NC(COCCSC)=O)CO)COCC(C)O1 C1(NC(c2cnc(OC)nc2)=O)CCC2(CC1)CC2NC(=O)COCC(F)(F)F N1(C(COC)=O)CCOC2CN(C(n3ccc(-c4ccc(F)c(C)n4)n3)=O)CC12 CCC(C(=O)NC1CCC(C(N2CC(CO)C3(CCC3)C2)=O)CC1)C(C)(C)CC n1(CCC)ccnc1C(F)(F)C(=O)NCCCN(C(C1CC1C#N)=O)C1CC1 C(=O)(CC(O)CNC(=O)C(F)F)NC(C(=O)OC)(C)C1CCC1 N1(C(C(C)N(C)Cc2cccnc2)=O)CC(C)(C)OCC1NC(=O)CNC(N)=O c1(OC)c(C(=O)NC2CN(C(C3(n4cccn4)CCC3)=O)CC2C)csc1C CC(C)CC(O)C(=O)NC12CC(CNC(c3coc(C(F)(F)F)c3)=O)(C1)C2 C1(C(=O)Nc2cn(COC)nc2)CCN(C(C2COCCC2C)=O)CC1C c1(C(N(C2CN(C(=O)CCC3CC3)CC2F)C)=O)ccc(S(N)(=O)=O)cc1 Cn1c(C(=O)NC2CCCCC2NC(=O)Cn2cnc(=N)[nH]2)cnc1S C1(CCNC(C(C)NS(C)(=O)=O)=O)CCN(C(=O)CC(F)(F)F)CC1 c1(C(=O)NC2CN(C(C3C(C(=O)OC)CC3)=O)CC2C)cnc2c(c1)CCC2 C(=O)(C(C)(C)COCCOC)N(C(CC)C1CC1)C.C(=O)(CCO)NCC(C)(C)C c1(OC)cc(NCc2cc(CNC(=O)CC3CC34CC4)cs2)ncn1 CCCC(CC)CC(=O)NCC1(O)CC(NC(c2sc(CCC)nc2C)=O)C1 C1(CCNC(c2nnnn2CC2CCOC2)C2(OC)CC2)CC(F)(F)C1 C#CCC(O)C(=O)NCC1(NC(=O)Cc2ccc(C(N)=O)cc2)CCC1 c1(OCC(=O)NCC2CC(F)(CNC(C3(O)CCOC3)=O)C2)cc(F)cc(F)c1 c1(C(N(CC(C)NC(C)(C)C)C=O)=O)cnc(C2CCCO2)s1 c1(C(N2CC=CC(NC(c3ccc(C4CC4)nc3)=O)C2)=O)cnc2ccccn12 C(=O)(CC(C)(C)CCOC)N1CC(CN(C(C2C(C(=O)OC)C2)=O)C)C2(C1)CC2 C12C=CCC(C1)C(=O)N2.C(C)(C)(C(=O)NCC(C)C(=O)OC(C)C)OCCC CCC(C)C(C(=O)NCCC12CCCN1CCC2)OC.C12CCC(O1)C(=O)N2 C1(NC(c2c(C)coc2C)=O)CCN(C(=O)C(C)Oc2ccccc2)CC1F N1(CCNC(C2CCC(C(F)(F)F)O2)=O)CCCN(C(C2(CO)CC2(F)F)=O)CC1 C(C(=O)NC(C)(C)C(C)NC(=O)Cn1nccn1)(C(C)C)c1cnc(C)s1 C1(OC)(CNC(=O)Cn2nccc2C)CN(C(c2occc2C)=O)C1 C1(NC(=O)C(O)C2CC2)CC2C(NC(c3[nH]nnc3C(F)F)=O)C2C1 c1(NC)ccc(C(=O)N(C)CC2CCCN(C(c3cnoc3C)=O)C2)nc1 c1(C(N2CC(C(N)=O)(CNC(c3ncc(C)nc3)=O)C2)=O)ccc(CO)nc1C c1(C(=O)NCCCC(C)(C)NC(C2CCCN2C2CC2)=O)cccc2nsnc12 N1(C(CC(C)N(C)C)=O)CCN(C(c2cc(-c3ccccc3)on2)=O)CC1CO c1(C(N2CC(NC(CC(CC=C)(C)C)=O)(CC)C2)=O)ccc(C)c2c1CCC2 C1(C(=O)NCCCNC(=O)CCN2CCC(F)C2)C2Cc3c(Cl)cccc3C12 c1(OC)ccc(C(=O)N(CC(C)O)CCNC(=O)C(c2ccnn2C)O)nn1 C1(CCF)C(=O)N1.C(C(C(=O)NCc1cnsc1)OC)OC c1(OC)cc(C(=O)N(C(C)CNC(=O)CC2CCN(OC)CC2)C)c(F)c(Cl)c1 C1(NC(C=NOC)=O)CC2CCC1C(NC(c1ccc(C)c(C)c1N)=O)C2 N1(C(C=CCOC)=O)CCN(C(=O)C=Cc2ccc(C(=O)OC)o2)C2CC12 C1(CC(=O)NCC(C)NC(=O)CCC2(CO)CCCC2)CCC(=O)NC1 C#CCC(C(=O)OC)NC(c1ccc(-c2ccc(F)cc2)cc1)=O Cc1cc(CN(CC(C)C#N)C(c2cc(C)n(C)n2)=O)n(C)n1 C=CCC(C(=O)NCCCC1CCCCO1)NC(=O)CCCCC Cc1cc(C(N2CC(O)(CNC(=O)C(c3cncc(F)c3)C)C2)=O)nnc1C N1(CCC(=O)NCC(C)N(C(C2(c3ccno3)CC2)=O)CC)CCCCC1=O C(=O)(C1CCCc2nc[nH]c21)NC1CCCN(C(CCSCC(C)C)=O)C1C C1(NC(C2(NC(C3CC(OC)C3)=O)CC(F)C2)=O)CCC(C)(O)CC1 C1(Br)(NCC(c2ccccc2)CN)CC(F)(F)C1 C1(NC(CCCn2ncc(C)c2)=O)CN(C(=O)C(=O)NCC(F)F)CC1C1CC1 c1(OC)cnc(C(=O)NC2(C)CCN(C(=O)Cc3occc3C)C2)cn1 C1(CNC(=O)Cc2cocn2)CCN(C(C2CCC2)=O)CC1O Cc1sc(O)nc1C(=O)NC1CCN(C(c2ccn(C3CCC3)n2)=O)C1 c1(C(C(=O)NCC2CC(NC(CCCSC)=O)C2)C)ccc(N)cc1 Cc1ccccc1NC(=O)C(N1CCN(CC(F)F)CC1)C1CCSC1 C1(CN2C(=O)CN(Cc3cccc(OC)n3)C2=O)CCCC(C)(C)CC1 c1(SC)cc(C(N2CC(NC(C3CNC(=O)C3)=O)C(O)C2)=O)nn1C C1(C(=O)NC(COC)COC)CCCN(C(c2n[nH]cc2C(C)C)=O)C1 C(C(=O)NCCC1CN(C(c2csnc2Cl)=O)CCCO1)(C(C)(C)C)NC(C)=O Cc1coc(C(=O)NCC2CC(NC(c3ccn(CN4CCOCC4)n3)=O)C2)c1 c1(C(N2CCN(C(c3c(=O)ccn(C)c3)=O)C3C2C3)=O)ccc2ncccc2c1 c1(CC)ccccc1C(=O)N(C1CCN(C(c2cocc2Cl)=O)C1)CC Cc1cc(C)c(C(=O)NC(CCN(C)C(c2nsnc2O)=O)C(C)(C)C)c(O)n1 O=C(N=c1cc2ccccn2[nH]1)N1CCc2ccccc21 C1(CNC(CCc2n(C)cnc2)=O)CN(C(=O)CSCC#N)CC(C)(C)C1 C1(CNC(C(C)Cn2ccnc2)=O)CN(C(c2n[nH]cc2Cl)=O)C2(CCC2)C1 c1(C(N(C2CC(CCC(=O)N(CC(=O)NC)C)C2)C)=O)cn2ccnc2s1 N1(C(C=C(C)C)=O)CCN(C(c2[nH]nc3ncccc23)=O)C(C)CC1C C1(NC(C(c2ccc(CC)cc2)O)=O)CC2CC(C1)N(C(=O)CC1(OC)CC1)C2 C(=O)(C1=C(Cl)CCOC1)N1C(CNC(c2ncn3c2CCC3)=O)COCC1 N1(c2ccc(S(=O)(=O)N3CCC(C)(F)C3)cn2)CCC(C2CNC(=O)C2)CC1 c1(OC)ccc(Br)c(OC)c1C(N1CCC(C(=O)Nc2cncnc2Br)CC1)=O c1(C(=O)NC2N(C(C3C(C(C)C)CCC3)=O)CCC2)ccc(C=O)cc1.C1CC1 c1(NC(N2C(C=CCC)CCC2)=O)ccc(C(F)(F)F)nc1Br C1(NC(C(C)OCCCC)=O)CCCCC1CNC(C1CCNC1=O)=O c1(C(=O)Cc2cn(CC3(CNC(C(C)OCC)=O)CCC3)nn2)cccc(Cl)c1 Cc1cn(C)nc1C(=O)NCC1(NC(=O)CC2(CN(C)C)CC2)CCCCC1 c1(C(C)C)cc(C(N2CC(NC(=O)C=CC(=O)N(C)C)C(F)C2)=O)ccc1O N1(C(c2nc(C)sc2)=O)CCC(C(=O)NCC(C)(C)C#N)C(C)C1 c1(C(=O)NCCCC(C(=O)NCC(COC)O)O)ccc2nccn2c1 N1(C(COCc2c(C)occ2)=O)CC2CC(NC(=O)C(F)CC3CCCC3)C1C2 Cc1c(Cl)cc(C(N2CC3(CC3)CC2C(=O)NC2CCCC(O)C2)=O)cc1Cl c1(CC(=O)N(CCCNC(C2C(OC(C)=O)C2)=O)CCO)ccnc(F)c1F N1(C(COCc2c(C)cccc2)=O)CC2CC1CN2C(c1ccc(=N)[nH]n1)=O c1(C(N2CC(C)(NC(c3nc(C)oc3)=O)C2)=O)cccc2ccc(O)nc12 C#CCC(CC(F)F)NC(C1CCC=CC1NC(c1ccc(F)c(C)c1)=O)=O c1(NC(C2CCN(C(=O)CCC3CCC(O)CC3)CC2O)=O)nc(Cl)c(Br)cc1O C1(C(=O)NCC(O)C2(Cl)CC2)(CNC(C2CCSC2)=O)CCCO1 C1(NC(C(C)(C)CC2CC2)=O)CC2CC1CN(C(c1cc(CO)cc(F)c1)=O)C2 C(=O)(CC1=NNC(=O)C1)NC1CC=C(C(=O)N(C)C)C1 C1(NCC2(CCC(=O)NC3C(C(=O)OC)CCC3)CCCC2)CCC12CCCC2 N1(NCC=C)CCN(C(=O)C(C2CCN(C(=O)CC(C)CC)C2)F)CC1 c1(CC)ncccc1C(=O)NC(CNC(c1cccc(SC)n1)=O)C(C)(C)C C1(C(N2CC(C)C(O)CC2)=O)CCN(C(=O)Cn2ccnn2)C2CCOC12 C1(C(=O)NC(C(C)NC(=O)COC(C)(C)C(F)(F)F)C)OC2CCC1CC2 c1(Cc2cn(CC(C)NC3CC(CO)CO3)nn2)ccc(F)cc1 C1(NC(c2ccc(CC)s2)c2nnnn2CC(F)F)CCCC=C1Br C(=O)(CC(C)CC(=O)N1CC(NC(=O)COC2CCCCC2)CC(F)(F)C1)OC C1(C(=O)NCC2(C(C)NC(c3cncn3C)=O)CC2)CCC(C2CC2)C1 N1(C(C2CCC(C(F)(F)F)C2)=O)CCC2CCN(C(=O)CC3CCC(O)C3)C2C1 C1(C(N2C(CCNC(C3(CF)CC3(F)F)=O)CCC2)=O)CN=C2N=CNN2C1 c1(CCCC(N2CC(F)(CNC(CCN(CC)CC)=O)C2)=O)c(C)noc1C N1(C(C2CC(O)(CNC(C(C)OC(C)(C)C)=O)C2)=O)CCCC12CCCC2 C1(C(N2CC3CC(OCC)C3C2)=O)CC(C(C)C)=NO1.C=C1CC2(C1)C(=O)NC2 C=CC(C)(CC)C(=O)N1CCN(CCCNC(=O)COc2cccc(Cl)c2)CC1 N1(Cc2cn(C)nc2-c2ccccc2C(F)(F)F)CCC(N)C(F)(F)CC1 C1(C(=O)NCC(c2ccccn2)C)CN(C(c2cc(Cl)c[nH]2)=O)CC12CC2 c1(N2CCCC(SCC)C2)cc(=O)n(C)c(O)n1.c1(C2CNC(=O)N2)ccco1 c1(C(C)=O)ccc(C(N2CCC(CNC(C34CC(F)C3C4)=O)C2)=O)cc1F C(C(C)(C)C(=O)NCC1(O)CN(C(C2CCC2C(F)(F)F)=O)C1)N(C)C Cc1coc(C(C)(C)C)c1C(=O)NC1CC(NC(=O)CCCc2cccnc2)C1 C(=O)(CC(C)C(C)C(C)C)N1CC=CC(NC(CN(CC)CC)=O)C1 C1(C(=O)NCCN(C(=O)CCc2ccn(C)n2)CCOC)CC(O)C(OC)C1 Cc1ccccc1C1=NOC(C(=O)NC2CC(C)(NC(C3C4CCC34)=O)C2)C1 C1(CNC(c2cncc(C)n2)=O)CCN(C(c2cnc(C)s2)=O)CC1O c1(C(N2CCC(NC(CCC(C)C)=O)CC2C)=O)cc2ccc(Cl)c(F)c2[nH]1 C(=O)(CC1=NNC(=O)C1)N1C(CNC(CCCC(=O)NCCC)=O)CC(O)C1 C(CCN(C(=O)C(=O)NCC(F)(F)F)C)(C(C)(C)C)NC(C(CC)SC)=O c1(C(=O)NC(C(C)NC(c2csc(C3CC3)n2)=O)CO)nccc2n[nH]cc12 N1(C(c2cc(C)on2)C(=O)O)CCSC(C)C1C.c1(OC)ccc(OCOCCO)cc1 C1(C(N(C(C(CC)C)C(=O)NCC2(C(C)(F)F)CC2)C)=O)CC(=O)CC12CCC2 C1(N)COc2cccc(Br)c2C1.c1(OC)ccc(-n2nnnc2C2(COC=C)CC2)cc1 c1(C(C(=O)NC2CCCC2)C)c(F)cccc1F.C1(=O)CC(=O)NC2(CC2)C(C)N1 CC(C(=O)N1CC(CNC(=O)C(C)(C)CC#N)C(C)(C)C1)C(F)(F)F c1(CC)nccnc1C(N1CCC(C(C)NC(=O)Cc2cnn(C)c2C)CC1)=O C1(CCNC(c2c(C)nn(C)c2)=O)CC(F)(F)CN1C(=O)CC1C=CCCC1 C=CCCC(=O)N(C(=O)CC1CCOCC1)CC(=O)OCC.C12CC1C2=O N1(C(c2c(CC)nns2)=O)CCCCC1CNC(C1C2(CC2)C12CC2)=O N1(C(C(C)OCCC=C)=O)CCCCC(CC(=O)NCCN(C)CCOC)C1 C1(C(N(CCCCC)CCCC)=O)CC(F)CN1C(=O)CCc1ccc(OC)cc1 C1(NC(CCc2ccnc(C)n2)=O)C(C)(C)C(NC(=O)C(C)C(C)(F)F)C1(C)C C#Cc1ccc(C(N2CCC(F)(CNC(=O)CC3CC3(C)C)C2)=O)cc1C C12(NC(c3c(CC)cco3)=O)CC(CNC(=O)CC3C=CCC3)(C1)OC21CCC1 C1(C(N2CCC(OCC)C2)=O)C2CN(Cc3ccnc(SC)c3)CC12 c1(C(=O)OC)ccc(C(N2CCCC2CNC(=O)C(C2CC2)OC)=O)n1C C1(O)(C(C)CNC(c2ccc(Cl)s2)=O)CCN(C(c2cc(F)c[nH]2)=O)C1 S(=O)(=O)(c1cccc(Cc2ccc(F)cc2)c1)N1CCC(NC(=O)C(F)Br)CC1 c1(C(=O)NC2CC(NC(C3CC4(C3)CC43CCC3)=O)C2)cccc([N+](=O)[O-])c1Cl c1(CC)n[nH]c(=NCCOCCN(C(C2CCOC(C(C)C)C2)=O)CC)s1 C1(OC)CC(C(F)(F)F)N(C(=O)NC2CC(C)N(C(=O)OCc3ccccc3)C2)C1 Cc1nc2cc(C(=O)NC3CCN(C(=O)CCNS(C)(=O)=O)CC3C)cnc2[nH]1 CCC(C)CC(C(=O)Sc1cc(Cl)ccc1Cl)NC(C1NCCC1CC)=O Cc1nc2cc(Cl)cc(C(=O)N(CC(C)NC(=O)CC3(O)CCCC3)C)c2[nH]1 c1(OCC)ccc(C(=O)NC2CCN(C(=O)CCC(C)(C)C)C2C)cc1Cl O=C1CCCCC(CC(=O)NC23CC(CNC(=O)C4=C(Cl)CC4)(C2)C3)N1 N1(C(C(CC)OC)=O)CCc2nc(C(=O)Nc3onc4ccccc34)ccc2C1 N1(C(C(n2cnc(C#N)n2)C)=O)CCCC(C(=O)Nc2n[nH]cc2C(F)(F)F)C1 N1(C(CC2CCN(C(C3C(CC)C3)=O)CC2)=O)CC(C)CCC12CC2 C12(CC(=O)NC(CC3CCN(C(c4c(C)nsc4)=O)CC3)C)CCC(C)(C1)OC2 C1(C(=O)NC(C(F)(F)F)C2CC2)CN(C(=O)CCc2cscn2)CC1C1CC1 C1(N(C(=O)CC2C=CS(=O)(=O)C2)C)CN(C(c2cnnc(C)c2)=O)CC12CC2 C1(C(=O)NCC(N(C)C)C2CC2)CC(CNC(=O)CCc2nc[nH]n2)C1 c1(C(=O)NCC(CC)Nc2nnc(C3CCCC3)s2)ccccc1-c1ccc[nH]1 N#Cc1ccc(Cl)c(C(N2CCCCC(NC(C3CCC4CC34)=O)C2)=O)c1 CCC(CCCC(=O)NC1CCN(CC)C1=O)NC(=O)CCOCC1CC1 C1(C(c2nnnn2CC(F)F)NCC2(C(C(C)C)O)CC2)CC2(CCC2)C1 Clc1cccc(CCNc2ccccc2Br)c1.C12(CC1)NC2 C=C1CC2(C1)CN(C(C1C(C)CCN1C(c1cccn(C)c1=O)=O)=O)C2 C(C)(C(C)(C)C(=O)N1CC(c2cc[nH]n2)C1)ONC(C1CC(=C)C1)=O CCCCCC(O)CC(=O)NC1(C(N2CCC2C)=O)CC1(C)C C(C(C)(O)CC(=O)NC(CCN(C)C(C12CC(C(C)C)(CO1)C2)=O)C(C)C)OC c1(C(=O)NCCCC(C)NC(c2cn(C3CCCC3)nn2)=O)csc(C#N)c1 c1(-c2ccc(C(C)OC(C3CCCN(S(=O)(=O)C(F)F)C3)=O)o2)ccc(F)cc1 C(=O)(CCS(=O)(=O)C1CCCC1)NC1C2CN(C(c3c(C)c(Cl)cnc3)=O)C1C2 C=CC(CC)CC(=O)NCCCC1CCN(C(c2cnc(O)n2C)=O)CC1 N1(C(CC=C)=O)CCC2CN(c3cc(-c4ccccc4)nc(Br)c3)CC12 c1(C(N2C(C3(NC(c4cc(CCC)on4)=O)CC3)CCC2)=O)cccc(C)c1Cl c1(C(N(C(C)CCNC(=O)C(C)O)C)=O)sncc1Br CC1CN(c2ccnc(C#N)n2)CCC1CNC(C1CCC2(CCC2)O1)=O N1(C(C(C2CCC2)OC)=O)CCC(C)(C)C(C(N2C(C)CCC2(C)C)=O)C1 Cc1c(C(N2CCCC2CNC(=O)CCc2ccoc2)=O)ccn1C1CC1 N1(C(C(C)(CO)OC)=O)CCN(C)C(CNC(C2CN(C(C)=O)C2)=O)C1 C(CC(=O)Nc1conc1C)(C(C)(C)C)NC(C(C=C=C)C)=O C(=O)(C(C)(CC=C(Cl)Cl)c1ccccc1)N(CCN(C(CC(C)N(C)C)=O)C)C O(NC(=O)C1=NOC(CNC(=O)C=CC2CC2)C1)C(CC)CC C1(O)(CN(C(C(C)CN(C)C)=O)C)CCN(C(=O)C(c2ccccc2)O)C1 c1(C(N(CCCNC(C(C)N(C(C)=O)CC)=O)C)=O)cccc2ccncc12 Cc1cc(=NCc2nc(Br)n(C)n2)[nH]c(N2CCn3c(cnc3C(F)F)C2)n1 C(=O)(C1=CCS(=O)(=O)C1)N1C(C)(C)CC(CNC(=O)C(C)(F)c2ccccc2)C1 c1(CC)cc(C(=O)NCC(CC)NC(C2CC(CC(=O)OC)C2)=O)ccn1 C#Cc1c(F)ccc(NC(c2nc(C(=O)OC)ccc2C#C)=O)c1F CC1OC2(CCN(C(c3ccc4c(c3)C(N)CCC4)=O)CC2)NC1=O c1(CNC(=NCCOC)NC(C2CCC(F)(F)CC2)C)nnc2ccc(Cl)cn12 C(C(O)CN(C(=O)C(C)NC(=O)OC(C)(C)C)C)N(C(C=CC)=O)C.[nH]1cnnn1 Cc1cc(C(=O)N(C)CCN(C(=O)Cc2nonc2C)C)on1 c1(CN(C(=O)C(C)C2CCC2)CCCNC(C=C(CC)CC)=O)ccccn1 c1(C(=O)NC2(C)CC(NC(C(C)CC3CCCCC3)=O)C2)n[nH]cc1[N+](=O)[O-] C(=O)(CC1C(=O)Nc2ccccc21)NCC1N(C(C(C=CC)O)=O)CCCC1C CC1(C)CCc2ccc(Br)c(C(=O)NCC3CCN3C(=O)CCNC(N)=O)c2C1 CC(c1cccs1)=CC(=O)NCC1(O)CCN(C(C2CCC(=C3CC3)CC2)=O)C1 C(CCC(C)(C)C(=O)NC1CCN(C(C)(C)C)C1)NC(CCc1n(C)ccc1)=O C1(C(=O)NCC2CC2)CCCC1CNC(C1CCCCO1)=O C12(NC(C3N(S(C)(=O)=O)CCC3)=O)CC1CN(C(=O)CN(C)C1CC1)C2 c1(-c2ncc(OCC(N(CC)OC)=O)s2)cn(C)c2ccccc12 c1(C(=O)NCC(C)(C)CNC(=O)C(F)C(F)(F)F)cncc2nc[nH]c12 C1(C(N2CC(CCO)(NC(c3cnc(SC)s3)=O)C2)=O)CCCCN1C(C)=O c1(CC(=O)NCC2CCC(C(=O)NC3C=CC(C(=O)OC)C3)C2)ccc(O)cc1 C1(NC(C=CC(C)C)=O)CCN(C(c2csc(-c3ncccn3)n2)=O)C(C)C1 c1(OC)nc2c(cc1NC(=O)C(=O)NC1CC1C1CC1)CCC2 Cn1cnc(S(=O)(=O)NCC(N2CC3(CNC(=O)CCS(C)=O)CC2CO3)=O)c1 N1(C(c2cc(C)no2)=O)C2CCC1C(NC(c1cc(Cl)cnc1O)=O)C2 N1(C(c2c(C(C)C)ocn2)=O)CCN(C(=O)CSc2n[nH]c(O)n2)CC1C c1(C(=O)OC)cnc(N2C3CCC2C(CNC(=O)Cn2ncnn2)C3)cc1C CC(C)C(F)(F)CCNC(=O)C(F)C1CC(N2C(NC(=O)OC(C)(C)C)CC2)C1 C1(NC)CC(C)N(CCN(C(C2CCN(c3ccncc3)CC2)=O)CC)C1 N1(C(C2(C(=O)OCC)CCCC2)=O)CCN(C(=O)CC2NC(=O)NC2=O)CC1 CCCCC(C)C(=O)N1CC=CC1C(=O)N(CCO)CCOC C1(NC(C2(N(C(C(C)OCC)=O)C)CC2)=O)CC(C)CC(C)(C)C1 C1(CNC(c2c(CC)onc2)=O)C2CN(C(C3CC3CC(C)(C)C)=O)CC12 CC(CCCC(=O)N1CCC(N(C)C(c2cncnc2)=O)C1)c1ccccc1 C1(C(=O)NCC(CNC(C=NOC)=O)(C)O)CC2(CCOCC2)C1 C1(OC)CC(CCNC(C2(F)CC2)=O)N(C(c2ccoc2C)=O)C1 c12ccc([N+](=O)[O-])cc1NC(=O)CO2.c1(C(=O)OCC)ccc(C(=O)OC)nc1 Cc1cccc2c1OCC2C(=O)N(C1CCCC1Cc1ccccc1)C c1(C(=O)NC2CC(CNC(=O)CN3C(=O)C=CC3=O)C2)ccccc1C(F)(F)F n1(CCC(N2CC(C)(NC(Cc3nc(C)sc3)=O)C2)=O)c(C)cc(O)cc1=O CCC(C)CC(C)C(=O)N1CCCC(N(C)C(c2ccnn2CCN(C)C)=O)C1 N1(C(c2n(CC)nnc2)=O)C2CCCC1CC(NC(c1cnoc1C1CC1)=O)C2 C12(CN)CC(C(=O)NCc3cscc3SC)(C1)C2 c1(NC(C2(COC)CN(C(=O)C(C)CSC)C2)=O)cc(C)cc(F)c1 CC(CN1CCCCC1)C(=O)NC1CCC1NC(=O)CCc1cnn[nH]1 C(C(C)C(=O)N(C)CCN(C(=O)CC1CC(N(C)C)C1)CC(C)O)SC N1(C(CN(C(C)=O)C)=O)CC(CNC(c2ccccc2CCN(C)C)=O)C(C)C1 CN1CCC(C)(C(=O)NCC23CC2CN(C(c2cc(Cl)n[nH]2)=O)C3)C1 C1(OC)(CNC(c2cncnc2C)=O)CCN(C(=O)C(N2CCNC2=O)C)C1 c1(CC)cccc2c(C(=O)NC(CO)C(C)NC(c3nocc3C)=O)c[nH]c12 N1(C(C(CC)OCC)=O)CCN(C(=O)C(C)(C)CC2CCOC2)CC1C1CC1 CN1CC2CCCC(C1)N2C(=O)NCCC1CC2(CCO1)CC2 CCCC(F)C(=O)NCC1(n2ccc(Br)n2)CC1.C12CCC(CC1)CNC2=O C=C(C)CCN=c1[nH]c(=NCC2CC(CO)CO2)c2ncccc2[nH]1 c1(C(N(CCCNC(c2oc(C)nc2CC)=O)CC)=O)sccc1S(N)(=O)=O CC1CN(c2ncccc2S(=O)(=O)NCCCn2cccn2)CCc2ccccc21 CCCCCCCCC(=O)N1CC2(NC(c3ncccc3N)=O)CC1C2 c1(OC)c(CNC(c2cccn2C2CCCC2)=O)cccc1Cl C1(CC)CN(C(c2[nH]nc(C(=O)OC)c2OC(C)=O)=O)CCC1c1ccc(I)cc1 CC(C)(F)C(C)(F)C(=O)NC1CCCC1CNC(c1c[nH]c2ncccc12)=O S(=O)(=O)(c1coc(C(N2CCC2CNC(C2CC3COCC3C2)=O)=O)c1)NC CC1C(NC(c2cncc(-n3cnnn3)c2)=O)CCN1C(=O)Cc1ccco1 C(N=c1nc2[nH][nH]cc-2c(O)n1)C1CCCN(C(=O)CC2CC(O)C23CCC3)C1 N1(C(C(C)OC(=O)OCC)=O)CCC(O)(C(N2CC(N(C)C)CC2CO)=O)CC1 c1(C(CC)C)ccc(C(=O)N(CCCN(C(=O)CSC)C)C)c(O)n1 N1(C(C(C(C)(C)C)O)=O)CCC2(CC2)CC1C(=O)NCCn1ccnc1 C(=O)(C(C)(C)C(=O)N1CCCC(N(C)C(c2ccn(CCOC)n2)=O)CC1)NC Cc1cc(N2CCC(NC(c3nccn3C(C)C)=O)C2)nc(CO)n1 C1(CCNC(C=CCN(C)C(C2(C=C)CCC2)=O)=O)CC(C)(C)CO1 N1(C(C=NOC)=O)CC(C(=O)N(CCC(=O)NC2CC2)C)C2(CCC2)C1 c1(COC)ccccc1CC(N1CC(C)(NC(c2nnn(C)c2N)=O)C1)=O C1(NC(C(C2CC(F)(F)C2)OC)=O)CCCCC1NC(c1cccc(O)n1)=O N1(C(c2c(OC)c(Cl)ncc2)C(=O)NC2CCOC2)CCC2CCCCCC2C1 C#Cc1cc(=O)n(C)cc1NC(c1coc2ccc(O)cc12)=O c1(CNC(=O)NCCC2(F)COC2)cc(Cl)cnc1F CC1=C(C)CCCC1N=c1[nH]c(N2CC3CCC(C2)N3C)nc2ncn(C)c12 C1(C)(CNC(C2N=C(C)SC2)=O)CCCN1C(=O)CCCn1nc(C)cc1C C=CC(CC)C(=O)NCc1ncc(C(=O)NC2CCCC2C(C)C)cn1 c1(CC)csc(C(F)(F)C(=O)NCC2(O)CN(C(C3CC3[N+](=O)[O-])=O)C2)n1 C1(CC=C)(NC(C2CCCC(=O)N2)=O)CCN(C(C2CC3(CC(=C)C3)C2)=O)CC1 C1(CCC)CN(C(=O)Cc2occc2C)CCN1C(C1(S(C)(=O)=O)CCC1)=O Cc1nc(C(=O)NCCOC2CCN(C(C3CCN(C(N)=O)CC3)=O)C2)nn1C Cn1cc(C(C)(C)C(=O)NC2CCC(NC(=O)C(O)CN3CCCC3)C2)cn1 N1(C(CC2C(C)=NOC2=O)=O)CCC2CN(C(c3ccccc3S(C)=O)=O)CCC12 CC1(C)OC(=O)CC1C(N1CCC(C=CC(=O)NCC2CSCCO2)CC1)=O c1(OC)ccsc1C(=O)NCC=CCNC(=O)C(F)(F)c1ccccn1 C1(NC(C(CC=CCC)C)=O)CC(OC)CN(C(=O)Cc2ccccc2SC)C1 CC1(C)C(CC(=O)NC2CCC(NC(=O)CC3COCCO3)CC2)C1(C)C c1(C(=O)NC(CC2CN(C(C3(SC)CCC3)=O)C2)C)cncc2sccc12 C(CN=c1nc2sccc2c(NC2CCC3C(CC2)C3(F)F)[nH]1)C1CC(O)CC1 Cc1ccc(C(C)CNCC2CC(O)(C(F)(F)F)C2)cc1 c1(OC)ccc(-c2cscc2C(N2CC(O)C(F)C2)=O)nc1C Cc1cnn(C)c1CC(=O)NC1CCC(NC(c2c(C)cnn2C)=O)CC1 N1(C(CP(C)(C)=O)=O)CC(C2CCN(C(=O)COCC3CCOC3)CC2)C1 c1(C(N2CC(N3C(C)CCC3)C2)=O)cccc(S(=O)(=O)N2CC3OC(=O)OC3C2)c1 C1(N(C(COCCC)=O)C)CC2CC1N(C(=O)CCC(=O)N(C)C(C)C)C2 CC1CC(C(=O)NC(Cc2ccccc2)CO)N(C(=O)CSc2nc[nH]n2)C1 n1(CC#C)cnnc1C(=O)NC(Cc1cc[nH]n1)C(=O)N1CCC1(C)C(=O)NC Cc1ccc(CC(N2CCC(N(C)C(c3cccc(C(C)C)n3)=O)C2)=O)cc1C O(NC(=O)CCCC(C)(C)NC(C1CC(C)CCO1)=O)CC#C C1(C(=O)NCCC(C)(C)NC(=O)Cn2ccc(C(F)F)n2)CCn2ncnc2C1 N1(C(CC(C)(F)F)=O)CC(C(=O)NC(CO)C2(C)CC2)CC1(C)C CC(C)(C)C1=NOC(C(=O)NC(CC2CCC2)C(=O)NCc2cnccn2)C1 Cc1oc(CO)cc1C(=O)NCCCN1CCN(C(c2ccc(C#N)[nH]2)=O)CC1 c1(C(=O)NC(C(C)NC(c2ncc(C)c(Cl)c2)=O)C)cc2c(C)cc(Cl)cc2[nH]1 c1(CCC(=O)NCC(C)CNC(c2ccc(Br)o2)=O)ccc(F)c(F)c1 C(C(CC(C)C)C(=O)N1CC2CCN(C(=O)CC3(O)CCCCCC3)C2C1)OC C=CC(C(=O)N1CCC(OCCNC(c2ccon2)=O)C1)N(c1ccccc1)C CC(C)(CCNC(C1SCCS1)=O)C(=O)NCCCc1ncco1 c1(C(=O)NC(C)CNC(=O)C(=O)N(CC(F)F)C)n[nH]c2c1C(=O)CCC2 c1(C(c2n(CC)nnn2)NCc2cccc(C(C)(C)C)n2)c(C)nn(CC)c1Cl Cc1coc(C)c1C=CC(=O)NC(C)CCNC(=O)CN1C(=O)NC(C)(C)C1=O C1(CNC(Cc2cc(OC)no2)=O)CN(C(c2c(OC)cccc2F)=O)CCC1C N1(C(=O)NC2C(C(C(=O)OC(C)(C)C)CC)CC2)CCC(O)(C(C)(C)C)C1 CCCC(CCCNC(c1cscc1Cl)=O)NC(=O)Cc1csc(Cl)c1 C1(C(=O)NCC(=C)CCNC(=O)CSCc2n[nH]c(C)n2)CCCCC1N(C)C C12(C(=O)NCC3CC(F)(CNC(CC(=C)Br)=O)C3)CCN(CC1)CC2 C(=O)(C(C)(F)C(C)(C)F)NCC1(C(F)F)CCN(C(c2c(OC)nc(C)s2)=O)C1 CC(C)C(CC(=O)NCC1CC1NC(=O)C=Cc1cncc(O)c1)C(C)C C(C)(C)(CCCCNC(=O)CC1CC(C)C1)NC(C(C(C)C)OC)=O N1(C(c2cn(CCNC(c3c(C(C)C)noc3)=O)nn2)=O)CCSC(C)C1 CN1CCC(C(=O)NCC2CCC(NC(=O)CN(C)Cc3ccccc3)C2)C1=O N(C(=NCCc1ccc(O)cc1)NCc1ccccc1)Cc1c(C)cco1 N1(C(c2c(CCC)[nH]cc2)=O)C2CC1CN(C(=O)CCc1scnc1C)C2 Cc1cccc2c1N(C(C1CCCCN1C)=O)CCC2C c1(OC)ccc([N+](=O)[O-])cc1C(N1CC2CCN(C(=O)CCC3CCC3)C2C1)=O c1(CC)cnoc1C(=O)NC1CCC(CNC(C2(C)CC2(F)Cl)=O)C1 N1(C(CN(C(=O)Cc2nonc2C)CCOC)=O)CCC2CCCC2C1 C=C(C)CCCC(=O)N1CCC(C)C1C(=O)NCCn1ccnn1 c1(-c2nc(C3C(C)OCCC3)on2)cnc2n(c1=O)CCS2 c1(CS(N2CCC(F)(CC)C2)(=O)=O)ccc(-c2cccc(CO)c2)c(F)c1 CC(C)C(C(=O)N1CCCCC1CNC(c1cnn(C)c1Br)=O)NC=O C1(C)(C(=O)NCCCN(C(=O)CN2CCC(F)C2)C)CCCS1(=O)=O C1(C(=O)NCC2C3N(C(C4CC(=O)CC(=O)C4)=O)C(CC3)C2)CCc2nncn2C1 C1(CC)CCN(C(=O)CCC2(C)CC(F)(F)C2)C1NC(=O)C(=O)NC(C)C1CC1 C12(C(=O)NC(C)Cc3ccco3)CC1CN(C(=O)CN1CCOC1=O)C2 C1(C(=O)NCC2CCC(NC(C3(CC)CC3)=O)CC2)CCc2nncn2C1 C1(NC(Cc2ccn(CC)n2)=O)CN(C(=O)C(CNC(C)=O)C(C)C)CCC1F C1(NC(C2N(CCCC)CCCC2)=O)Cc2n[nH]cc2C(C(F)(F)F)C1 Cc1nc2cccc(C(=O)NC3CCN(CC4CCCCC45CCCC5)C3)n2n1 C1(NCCNC(c2cc(C)c(C)s2)c2n(CCOC)nnn2)CC(=O)N(C)C1 N1(C(C(=O)NC(C)C)=O)CCN(C(CNC(=O)C(C)(C)C)=O)C(C)CC1C N1(C(c2c(CC)scn2)=O)CC2CCCC2(NC(c2ccc(C3CC3)nn2)=O)C1 C1(NC(c2cc(OC)n(C)n2)=O)CN(C(C2(NC(N)=O)CC2)=O)C2(CCC2)C1 C1(CC(=O)NC(CNC(CNC(CC)=O)=O)C2CC2)CSCCO1 C1(C(N(C(C)(C(=O)NC2CC3(C2)CC3(F)F)C2CC2)C)=O)CC(C2CCC2)C1 C=CC1(C(N2CC(C(C(N3CC(=O)N(C)CC3C)=O)OC)C2)=O)CCOCC1 c1(NC2CCC(OC)C2)ncc(S(=O)(=O)NC(c2ccccn2)C)cc1Cl c1(CCCc2cn(CCCC(=O)N(C3(C)CCOC3)CC)nn2)cccc2cc[nH]c12 C(=O)(C(O)CC(N)=O)NC(CNC(c1c(C)oc(-c2ccccc2F)n1)=O)CCl C1(O)(CNC(c2ccc(Br)o2)=O)CCN(C(C2(O)COC2)=O)C1 c1(CC(N2C3CCC(C3)C2C2(C(=O)O)CC2)=O)cc(C(F)(F)F)cc(Br)c1 C=CC(C)(O)CC(=O)N1CCC(CN(c2cc(C(C)(C)C)ncn2)C)C1 CC1CCc2nc(C(N3CCCC(O)(CNC(=O)Cc4ccoc4)C3)=O)cn2C1 C1(CN(C(c2cc(C)ns2)=O)CC)CCCN(C(=O)C(c2cccc(Cl)c2)O)C1 N1(CC)CCOC(C(N2CCCC(C(C)(C)C(=O)NC3CC(CC)(CC)C3)C2)=O)C1 C(=O)(C1CCc2nnc(C)n21)NCC(CNC(C(CC)(CC)CO)=O)(C)F C(=O)(CCCCCF)NCC1C2CN(C(C(c3cccc(Cl)c3)C)=O)CC21 CC(C)CCC(F)C(=O)N1CCCC(CNC(C2CCCN2C(=O)C(C)C)=O)C1 C1(CC)CC(C(=O)NCC(n2cccn2)C)CCN1C(c1ccncc1C)=O Cc1cccc2c1OCCC2N(C)C(=O)Nc1n[nH]cc1C1CCC1 C(=O)(C(CC)C(=O)N1CC=CC1CNC(c1ccc(F)c(F)c1)=O)OCC N1(C(c2ccc(C)o2)=O)CCC(NC(=O)CCC[N+](=O)[O-])C(O)C1 C1(CC2(C)NC(=O)N(CCC=C)C2=O)CC2CN(C(=O)OC(C)(C)C)CC2C1 C12(CNC(Cn3ccc(C)cc3=O)=O)CCCC1N(C(=O)C=CC(N)=O)CCC2 C1(C(N2CC(n3cnnn3)C2)=O)CCN(C(c2cc(CO)[nH]n2)=O)CC1 c1(NC(CCNC(Cc2ccc(OC)cc2F)=O)(C)C)ncnn2c(Br)ccc12 CC(CCCNC(C1CC(C)(C(C)(C)C)C1)=O)NC(=O)C(C)(C)Sc1ccccc1 C1(CC)CCCC1C(N1CC(C)(CO)C1)=O.C(=O)(NOCCO)C1CCC1 N1(C(C(=O)N(C)C)=O)CCC2CCN(C(c3coc4c3COC4)=O)CC2C1 C1(NC(c2[nH]ccc2CNC(C2(F)CCOC2)=O)=O)CCOC1=O C1(NC(C(C)OCC=C)=O)C2CC3CN(C(=O)CSCCC(C)C)C1C3C2 C(N=c1[nH]c(=N)[nH]c(=NC2CCOC3(CCC3)C2)[nH]1)c1n[nH]c(C)c1C CC(CN=C(NCC(F)F)N1CCN(CC2CCOC2)C(=O)C1)N(C)C CC(C)C(CNC(c1cc(C2CC2)[nH]n1)=O)NC(=O)NCc1ccccc1 N1(C(C(C#C)(C)C)=O)CCCCC(CNC(=O)C(C)NC(C2CCCC2)=O)CC1 c1(OCCC(=O)NC2C3CN(C(C(CC)(F)F)=O)CC32)ccc(Cl)c(F)c1 C1(CC(=O)N(C2CCN(C(c3cnsn3)=O)C2)CC)CCCCO1 CC1CCC2CN1C(=O)CN2.C1(C(=O)NCc2nccn2C)CCCCC1F N1(C(C(CC)Oc2ccccc2)=O)CC2CCCC(C1)N2C(=O)C(F)C(C)(F)F N1(C(C(C)O)=O)CC2CC(C1)CN(C(C1CCC(C(=O)N(C)C)CC1)=O)C2 C(=O)(CCCCCS(N)(=O)=O)N1CC(C(C)NC(c2nc(Br)c[nH]2)=O)C1 c1(C(=O)NC2C(C)CN(C(=O)CCCC3CC3)C2)cc2c(cc1F)NCCC2 CC1CC(C(N2CCCC(F)(CNC(c3c(Cl)n[nH]c3C3CC3)=O)C2)=O)CC(C)C1 c1(C(N2CC3C(NC(C4C(C)C4)=O)(C3)C2)=O)cc2c(F)c(Br)ccc2[nH]1 C(=O)(N=c1[nH][nH]c2c1CN(C(=O)CSC(=N)N)C2(C)C)c1c(O)ccc(C)c1 N#Cc1c(N2CCN(C(c3ncccc3C(F)C(F)(F)F)C3CC3)CC2)cccc1Cl N1(C(c2cc(SC)oc2)=O)CC(NC(c2nc(O)c(C)s2)=O)C(O)C1 c1(C(=O)NC(c2ccc(C3CC(F)(F)C3(F)F)cc2)C)ccc2cncn2c1 C(C(C)(CC(C)C)NC(c1ccccn1)=O)NC(C1C(CC)C1)=O Cc1c(NC(C2C=CCN2C(C2CCC=CCC2)=O)=O)cccc1C1CC1 C1(C(N2CC(O)(C(C)NC(=O)C(C)C(F)F)C2)=O)CCC2(CC1)CC(O)C2 C=CCC(CC=C)C(=O)N1CCC(NC(=O)CSc2ccc3c(c2)CCC3)C1C c1(CCCC=C)ccc(C(=O)NCC2CC2NC(=O)CCN2CCCC2)cc1 c1(C(=O)NC2CC(C)(CNC(C(CC)(C)O)=O)C2)cc(C)c(O)nn1 C(CC(=O)NC(C1CN(C(C2CC(C(N)=O)C2)=O)C1)C)SC N(C(=NCCc1cn(C)cn1)NCc1ccc(F)cc1N1CCCC1)C(CC)C N1(C(CCc2c(C)ncs2)=O)CCCC12CCN(C(=O)CC1C=CCCC1)C2 C1(N(C(=O)CC2CCCO2)Cc2ccccn2)CCN(C(c2cnsn2)=O)C1 c1(C(=O)NC2C(NC(C(COC)COC)=O)CCOC2)ccc2ccn(C)c2c1 c1(C(=O)NCC(C2(O)CN(C(C3CC(OC)C3)=O)C2)(C)C)cncc(C2CC2)c1 c1(C(N2CC(C)C(NC(=O)Cn3cc(Cl)cn3)C2)=O)c(F)cc(F)cc1F c1(C(=O)NC(CN(C(C2CC3(C2)CC32CC2)=O)CC)C)cnc(C)c(N)c1 C(CC1CC1)(C(=O)NCCN(C)CC)NC(COC(CC)C)=O C(=O)(C(F)(CNC(c1nccnc1C)=O)C(C)C)Nc1cnc(OC)nc1 C1(CCNC(c2cc(CC)no2)=O)CCCCN1C(C1CC=CCO1)=O CN1CCCC(F)(C(N2CCCC(N(C(=O)C=CC3(C)COC3)CCO)C2)=O)C1 c1(C(=O)NC2CCN(C(CCC=C=C)=O)CCC2CO)cnc2ncccc2c1 c1(OC)cccc(F)c1C(=O)NC1CC(C)CN(C(c2cc(C)ccc2Br)=O)C1 c1(C(N(CCN(C(COCC(=C)C)=O)C)C)=O)ccnn1C C1(C(N2CC3C(CNC(C45CC(CO)(C4)C5)=O)C3C2)=O)CCCC2CCCCC12 C1(CNC(C2(C=C)CC2)=O)CCC12CCN(C(c1ccc(C3CC3)nn1)=O)CC2 CC(C)(CCC(=O)NOCC(O)CO)C1CN(C(C2C3CC(=O)CC23)=O)C1 c1(C(=O)NCC(C)NC(C2(C)CC2F)=O)cnc(OC2CCCC2)s1 C1(NC(C#C)=O)CCSC12CN(c1ccc(C(F)(F)F)cn1)C2 c1(OC)ccc(CN(c2ncnc(NCC(C)(C)N3CCCC3)c2C)C)cc1Cl C#Cc1cc(F)c(C(N2CC3CCN(C(C4(n5nccn5)CC4)=O)C3C2)=O)cc1F N1(C(Cc2c(C)noc2C)=O)CCC(NC(=O)C(c2ccccc2)C)CC1C CN1C(=O)CC(C(N2CC(NC(c3ccc(F)c(CO)c3)=O)C2)=O)NC1=O N1(C(C2CCN(CC)CC2)=O)CC(C2CN(C(C3(C)CCCC(F)(F)C3)=O)C2)C1 c1(CNC(c2ccc(C(N(C(C)(C)C)CC)=O)o2)=O)nn(C)c(C)c1S(N)(=O)=O N1(C(c2ccn(CC#N)n2)=O)CCCCC1CCNC(=O)CC=C(Cl)Cl N1(C(=O)CC2CCCN2C(c2ccnnc2)=O)CC2CCC(C2)C1 C1(NC(C(C)(C)N(C(=O)CC2COCC2O)C2CC2)=O)CN2CCC1C2 CN1CCC2(C1)C(=O)N2.C(C1=NOCC1)NC(=O)CCOCC(F)F N1(CC#C)CCC(N(C(=O)CCCC2CCCCC2)C)C1 CC1CC2(CC(C(N3CCC(C(F)C(N4CCOCC4)=O)C3)=O)C2)C1 CC(C)CC(C(=O)N1CCC(CC(C)(C)C)C1)N(C(=O)C(C)(C)CO)C C=C(C)CC(C)C(=O)NCC(CNC(c1nn(C)c(C)c1Br)=O)OC CC1(CNC(=O)CCCc2ccccn2)CC(NC(c2cc(Cl)cs2)=O)C1 c1(C(=O)NCc2cccc(NC(C3C(CCC)C3)=O)c2)cc(F)cc(F)c1OC c1(OCCCC)ccc(C(=O)NCCC(C)CCNC(=O)COCCSC)cc1 c1(C(=O)OCCCSc2ccccc2F)c(Cl)sc(Cl)c1Cl C12(NC(C(CC)NC(N)=O)=O)CCC(C1)N(C(=O)C(C)Cc1cnn(C)c1)C2 C1(CC(=O)N(C2CCCCC2)C2(C(=O)NCCSC)CC2)CC(O)CCO1 c1(C(N2C(C(=O)Nc3nccc(I)n3)COCC2)=O)cc(F)c(F)cc1F C1(NC(c2cc(C)oc2)=O)CN(C(c2cn3ccnc3cn2)=O)CCC12CCC2 C1(C)(C(=O)NCCCC(C)NC(CCC=C(C)C)=O)CC(C)(C)C1 N(C(=NCCC1CCC(C)O1)NCC1(C(C)(F)F)CCC1)Cc1nc(C)on1 c1(C2CC(CC(=O)NCC(C)CN(C(=O)CC3CCCO3)C)C2)ccccc1 CC#CCC(C(=O)NCC1C=CCCC1)NC(=O)C(C)S(N)(=O)=O N1(C(CC(C)F)=O)CCC2(C1)CN(C(c1ccccc1-c1nncn1C)=O)C2 N1(C(C2CC(=C)C2)=O)CCC2C1CCCN2C(c1cc(F)c(F)cc1OCC)=O N1(C(N)=O)CCC(C(=O)NC(CNC(C2CCCN2N=O)=O)CO)CC1 N1(CC)C(C)CN(C(C2(CO)CCN(C(c3ccccn3)=O)C2)=O)CC1C CC1(C)CCc2nc(CNC(N3CCOCC(C)(F)C3)=O)ccc2C1 c1(NC(c2cc(OC)ns2)C)nc(N2CCCCCC2)nc2scnc12 C1(NC(Cn2c(C)nc(C)n2)=O)CC(NC(C2CC3(C2)CC(C)C3)=O)C12CCC2 n1(CCCC)nnnc1C(CC1CC1)(CC)NCC(C)SC C1(NC(CCc2onc(C)n2)=O)COCCN(C(=O)Cc2cncs2)C1 C1(n2cc(C(C(C)C)(C)C)nn2)CCC(NC(C2N(CC(F)F)C2)=O)CC1 CC(C)(O)CC(=O)NC(C1CCCC1)CN1CCN(C(C2C3CCOCC23)=O)CC1 Cc1ccncc1C(C)NC(=O)CCc1ccc(CNC(=O)OC(C)(C)C)cc1 Cn1cnc2c(NC3CCC4(CCC4)CO3)[nH]c(=NCc3cncnc3)nc12 C12(CNC(CCSC)=O)CCCCC1N(c1cc(Cl)nc(C(F)(F)F)n1)CCC2 C1(C(=O)OCC=Cc2ccco2)CCN(C(=O)Cc2cccs2)C(=O)C1 C1(C(N(CC(C)NC(C2(O)CCCCC2)=O)C)=O)CC2CCCCCCC12 [N-]=[N+]=NCCCCC(=O)NCC1(C(=O)NC2C(O)CC2O)CC2(CC2)C1 C(=O)(C(C)(C)C(c1nnnn1Cc1ccccc1C)Nc1ccccc1C)OC C1(C(=O)NCCCCCCNC(c2cncc(C)c2C)=O)CCC([N+](=O)[O-])CC1 C(=O)(C1CCCc2c1ncn2C)NCC1(CNC(C=C(C)C(C)C)=O)CC1 Fc1cc(F)c2c(-c3nc(-c4cncs4)nn3CC3CCOC3)n[nH]c2c1F C1(NC(C(C)=CC2CC2)=O)CN(C(C2CC2c2nccn2C)=O)C2CC12 c1(C(NOCC(C(=O)OC)O)=O)n[nH]c(C(C)NC(=O)Cc2ccon2)n1 C1(N(C)C)CCCC(C(=O)NC2CC(F)(CNC(=O)C=CC3CCCN3C)C2)C1 Cc1c(NCC(C)(C)CCCN(C)C)nc[nH]c1=NCC1COCC(C)(C)O1 C1(NC(c2ccccc2Cl)C)CNCC2(CCC2)C1 c1(C(N2C3(CCN(C(C4=CCCCC4C)=O)C3)C2)=O)csc(=NC2CCC2)[nH]1 c1(CC)nc(C2CC2)sc1NC(=O)NC1(CCCCO)CC1 c1(C(c2cccc(F)c2)NC(c2cccc(I)c2)=O)cc(Cl)ccc1Cl c1(OC)cc(F)ccc1C(N1CC(CNC(=O)CCC2CC2(F)F)CC(C)C1)=O c1(OC)cccc2c1CC(c1nnc(C)o1)(N(C1CC1)Cc1cnc(C)s1)CC2 C1(NC(c2ccc(OC)s2)=O)CC2CC1CC2NC(C1CC(SC)C1)=O C1(C)(CNC(CCC)=O)COCCN(C(=O)C(c2cncc(Br)c2)OC)C1 CC1CCC(NC(=O)CC2(O)CCCCCC2)CN1C(C1CC2(C1)CC2F)=O n1(C(C)C)cc(C2CN(C(C3CCC(N)C3)=O)C2)nn1 c1(C(=O)OC)cc(Cl)sc1NC(C1(F)CN(C(C2CC2C2CC2)=O)C1)=O c1(OC)ccc(N)c(C(N2CCOCC(NC(=O)C=CSC)C2)=O)c1Br C1(C(N2C3CC(CNC(C(C(C)C)(C)C)=O)C2CC3)=O)CC2CCC1C21CC1 O=C1CCN(C(C2(C(=O)C3CC3)C=CCN2C(C2CC(=C3CC3)C2)=O)=O)CCN1 C(C(=O)NOCCO)(C1CCOC1)NC(C1CCC(=O)N1)=O.C1(C)CC1 N1(C(Cc2c(C)cco2)=O)CCC2(C1)CN(C(C1(N3CCOCC3)CC1)=O)C2 N1(C(CC2CN(C)C2)=O)CCCC(n2cc(-c3ncccc3Cl)nn2)C1 C=CCN=C(NCc1ccc(Cl)o1)NC1CC1(C)CC N1(C(CNC(c2cc(CC)[nH]n2)=O)=O)CC(O)CCC1C c1(OCC)cc(C)nc2ccc(C(N3CCCC3(CO)CO)=O)cc12 C1(CC)(CC)CC(NC(=O)C(C)(C)Oc2ccccc2)CN1C(=O)C(C)OCC N1(C(CC2CC(NC(C(CC3CCC3)OC)=O)C2(C)C)=O)CCOCCC1C C(CC(C(=O)NCCC(C)NC(=O)C(c1cccc(F)c1)(C)C)OC)OC N1(C(C2=CC(C)(C)C2)=O)CCC(NC(c2cccc(F)c2F)=O)C12CCCC2 N1(C(COC)=O)CCN(CC(C)NC(=O)C(c2cccc(O)c2)C)CC1 C1(CC)CCCCC1OCCC(=O)NCC1CCCN(C(=O)CN(C)C(C)C)C1 C1(NC(CN2CCN(C)CC2)=O)CN(CCP(C)(C)=O)CC(C)(C)C1 c12ccccc1O2.CC(C)C(CO)N(C)C(C1CCC(OC(F)(F)F)C1)=O c1(-c2nnc(N(CCc3cccc(C)n3)C)n2CCC#N)ccc(S(C)(=O)=O)cc1 N12CCC(N=C3NC(=Nc4[nH]ccc43)N(C)CCC1=O)C(C)(C)C2.C(C)(=O)NC CC1(NC(c2ncon2)=O)CN(C(=O)CC#N)C1 C=CCCCC(=O)NC1(CO)CCN(C(c2ccoc2C2CC2)=O)C1 C1(NC(=O)CCF)CCCCC1CNC(c1cccc(-c2cscn2)c1)=O C(CS(=O)(=O)C1CCCC1)C(C1CC2(N)CN1C2)=O.OC C1(NC(c2c(C)c(N)cnc2)=O)CCCC2CN(C(=O)CCc3cscn3)CC12 CN1CCC2(C1)C(=O)NCC(=O)C1CC(C1)N2.c1(C(=O)NC2CC2)ccsc1 C1(C(=O)NC2CC(F)(CNC(CCCC(=O)NCC)=O)C2)CCc2c[nH]nc2C1 n12c(nnc1-c1cnccn1)N1CCC(C1)C2.C(C(F)(F)F)N(CC)CC C1(C(=O)NC(CCC=C)C2CC2)CN(C(=O)C=Cc2cn[nH]c2)CCC1(C)C C=CCCCC(C1CC1)NC(=O)C=CCNC(=O)CC1CSCCO1 C1(C(=O)OC)C(C2CC2)CCN1C(=O)CC1CCC1.C1(=O)C(OC)CN1 C1(NC(CC2N(C(C3(C(=O)NC)CCC3)=O)CC2)=O)CCCCN(C)C1=O c1(CC(N2C(c3nc(C)[nH]n3)COCC2)C(=O)NC2CC2)ccc2n[nH]cc2c1 N1(C(CCNC(COC)=O)=O)CC(NC(C2CC(SC)C2)=O)CC(F)C1 c1(OC)ccc2c(C(=O)NCC3(C4(O)CN(C(=O)C(C)SC)C4)CC3)cnn2c1 C1(CCOC)(NC(C2CC2F)=O)CC1.C12(CC1)C(=O)N(C)C2 C1(NC(CCC(C)OCC)=O)CCSC12CN(C(c1scnc1CC)=O)C2 C1(CNC(CCc2ccc(C)s2)=O)CCCCC1NC(=O)Cn1cncn1 c1(C(N(CCN(C(C(CC)(C)F)=O)C)C)=O)cc(F)ccc1OC(F)F Cc1cc(C#N)cc(C(N2CCCC(CNC(=O)C3=CC(O)CCC3)C2)=O)n1 c1(C(=O)NCCCOCCCNC(C(C(C)C)SC)=O)cc(C)nnc1N(C)C c1(C(CCC(=O)NC2CCN(C(c3c(OC)csc3)=O)C2)=O)c(F)cccc1F C(CN=c1ccnc(NCc2ccccc2N=[N+]=[N-])[nH]1)(C(C)C)OC N1(C(C2CCN(OC)CC2)=O)CC2(C=C(C(=O)N3CCCC3C(N)=O)CO2)C1 C(C(=O)N1CC(N(C(=O)C(F)(F)C2CCCCC2)C)C1)(C(C)C)OCC(C)C N1(C(CN(CCC)C(C2CCOC2(C)C)=O)=O)CCC2(CC2)C1 CC1(NC(c2nnnn2C2CCOC2)(C2CC=CC2)C)CCSC1 N1(C(C2CC(OC)C2)=O)CCC(C)(NC(=O)CCc2cnn(C)c2C)C1 CN=c1nc(N(C2CC3(CCC3)C2C(F)(F)F)C)[nH]c(NCC2CC3C=CC2C3)n1 C(=O)(C(C)C(F)(F)F)N(CCNC(C(CC)NC(N)=O)=O)CC Cc1oc(C)c(C(=O)NCC2(CN(C)C(c3ccncc3F)=O)CC2)c1C N1(C(c2c(C)nns2)=O)CCC2CN(C(c3ccnnc3)=O)CCC2C1 Cc1nn(C)c(C(=O)NC2CC3(C2)CN(C(=O)C(O)C2CCCC2)C3)c1Br N1(C(C2C(=C)C2)=O)CCCN(C(=O)C=Cc2cc(Br)cs2)C(CO)C1 N1(C(C2(C#N)CCC2)=O)CCC2CN(C(=O)C3CCc4c[nH]nc43)CCC2C1 c1(C(N(CCN(C)C(c2cscc2F)=O)C)=O)nccc2ccsc12 C1(NC(=O)CSCc2ccccc2Cl)CCC12CN(C(C1CC=CCC1)=O)C2 Cn1ccc(=O)c(C(N2CCOC(CNC(C3CC4(CCO3)CC4)=O)C2)=O)c1 c1(C(=O)NC2CC(NC(=O)Cc3ccc(CO)cc3)C2)cnn2c1OCCC2 c1(CC)cccc(CS(C)=O)c1.C12CCC(=O)N1C(=O)NCCN(CC)C(=O)C2 C1(C(=O)NCCCn2cccn2)(CNC(C2CCSC2)=O)CC=CC1 c1(C(=O)NCC(C(=O)NCC2(CC)CCC2)O)cccc(O)c1C C1(NC(CCC(C)NC(c2cc(C)ncc2)=O)=O)CCc2nn[nH]c2C1 c1(NC(=O)NC2(c3ncc(C)[nH]3)CCOC2)ccc(Br)cc1F Cc1nc2ccc(C(=O)N(CC(CO)(CO)NC(C3SCCC3C)=O)C)cc2[nH]1 C1(CC(=O)NCC(C)C(F)F)CCN(C(C2CCCCN2C)=O)CC1 C1(CNC(Cc2cc(CC)on2)=O)CC2CCC1N2C(=O)Cn1cc(C)cn1 C1(CNC(CNC(CCCCC)=O)=O)CC(C)CN(C(=O)C(C)SCC)C1 C1(F)(C(=O)NC2CC(C(C)NC(c3cn(C)nc3C3CC3)=O)C2)CCS(=O)(=O)C1 C1(C(=O)NC(CNC(C2CC(=C)C2)=O)C)CCCCC1c1nc[nH]n1 CS(=O)(=O)CC(=O)NC1CCC(CCNC(c2ccc(CO)o2)=O)C1 c1(C(=O)NC2CN(C(C(C)Cn3ccnc3)=O)C2)ccc2[nH]ccc2n1 N1(C(C(=O)NCC2N(C(CNC3C(C=C)C3)=O)CC2)=C)C(=O)c2cccnc2C1=O c1(OC)ccnc(CN2CC3C(NC(=O)CCc4ccnc(Cl)c4)C3C2)c1 CC#CCC(C(=O)NC1CCC2(CC2)C1)NC(C1CCCC(=O)N1C)=O C(=O)(C(C)(C)CC(=O)NCCCN1CCC(NC(=O)C(C)(F)F)CC1)OCC CC(C)CC(CNC(C1CCCS1)=O)NC(=O)C(C(C)C)c1ccccc1 c1(C(N(C(CCNC(CCSCC)=O)C)C)=O)cnn(C(C)C)c1F C=CCCC(C)NC(c1conc1C(C)NC(=O)C=CC1CCOC1)=O CC(CC1CCN(C(C2C3CCCC23)=O)CC1)N=c1c(Br)c[nH]cc1[N+](=O)[O-] c1(NC(C(=O)N(CCCC)CCCO)C)cccc([N+](=O)[O-])c1 CC1C(NC(=O)CC(C)n2ccnc2)CCN1C(=O)Cc1cccc(N(C)C)c1 N1(C(C2N(C)CCOC2)=O)CC2CC(NC(C3CC(=O)NC3(C)C)=O)CC1C2 N12CCN(C)C(C1)CNC(=O)C2.C1(C(N(CC)CC)=O)Cc2nncn2C1 C1(CNC(C=CC=CC)=O)CCCN(C(C2(C#N)CC(C)C2)=O)C1 C1(NC(C2(NC(C(CC3CC3)OC)=O)CC(F)C2)=O)CCS(=O)CC1 CCCC(C(=O)NC(C)CCNC(=O)CCc1ccccc1)NC(C)=O Cc1ccc2cc(CN(c3cc(NCCn4ccnn4)ncn3)C3CCC3)sc2c1 C1(COC)CC(CNC(c2cnn(CCO)c2)=O)N(C(=O)C=CC(C)CC)C1 C1(NC(=O)C=Cc2ccco2)CC(NC(=O)CCOC2CCOCC2)CC1O c1(NC(=O)CCN2CCN(C(C3CCCC3O)=O)CC2)nccc(Cl)c1F c1(CCC)cc(C(=O)N(CC(C)NC(=O)CCCOC2CC2)C)nn1C C=CCCCCC(=O)NCC(C1CC1)N(c1ccsc1)C(=O)COCC(C)C c1(OC)cc(C(C)CC(=O)N2CC(CNC(=O)CC3CCCO3)C2)ccc1C C12(CNC(C3CC4CC4C3)=O)CCC(CC1)CN2C(=O)C=CCOCC(F)(F)F C1(c2nc(C3N=C(C)SC3)on2)CN(n2cc(C3CCCC(O)C3)nn2)CC1C C(c1ccncc1)=CC(=O)NCCC1CCN(C(C(C)NC(CC)=O)=O)C1 c1(C(=O)NCC2(c3cccc(Cl)c3Cl)CC2)ncc2[nH]ncc2n1 Cc1nn(CC(=O)NCCCCC2(NC(=O)C(c3ccccn3)C)CC2)cn1 C(=O)(C#CC1(C)COC1)NC(C(C)NC(c1sc(C)c(O)n1)=O)C Nc1cccc(Cl)c1C(=O)NC1CC1NC(C1(C(N)=O)CC1)=O.C1(O)CCCC1 c1(NC(c2ccccc2F)C)ccc(S(=O)(=O)Nc2nncs2)cc1F C(=O)(CC(F)(F)Cl)NCC(CC)(C)NC(=O)C(CO)OC c1(C(=O)NC(CN(C(=O)CC2CC(n3cnnc3)C2)CC)C)cc(Cl)c(F)cc1F C1(C#N)(C(N(CC(C)N(C)C(c2cc(Cl)ccc2F)=O)C)=O)CC2CC2C1 N1(c2snc(NC(=O)OC)n2)Cc2cnn(C3CCN(CC(C)O)CC3)c2C1 Cc1nccc(NCC2CCCC2(F)F)n1 C1(CNC(C(CC)OCC)=O)CN(C)CCN1C(c1cc(C#N)on1)=O N1(C(C2=CCCC2C)=O)CCC(C(=O)N2CCS(=O)CC2C)=C(F)C1 C(CC(=O)N(C1CCCC(C)(C)C1)C)(C(C)C)NC(C1CC(OC)C1)=O N1(C(=O)C2=CCC(NC(=O)CC3(O)CCC3)C2)CC2(CCC(O)CC2)C1 Cn1nc2c(c1C(=O)NCC1CC1NC(C1(C3CCCCO3)CC1)=O)CSCC2 C1(C)(CNC(=O)NCCCNS(C(C)C)(=O)=O)CCOC12CC2(F)F c1(C(=O)NCC2N(C(C(C(C)C)O)=O)CCC2C)ccc2nccn2c1 N1(C(c2c(C)nc(O)cc2)=O)CCC2(CCCN2C(=O)C2=NOC(C)C2C)C1 CC(C)C(O)C(F)(F)C(=O)NCCCCN(CCCNC(=O)C(C)C(C)(C)C)C c1(C(N(CCCCNC(=O)C=C(C2CC2)C2CC2)C)=O)cnc2ncnn2c1O C1(OC)CN(C(c2cn(CC(N)=O)nn2)=O)CCC1NC(C1(OC)CCCC1)=O C1(NC(CSCCCC)=O)COC2(CNC(=O)C(C)OC)CC1C2 c1(NC(C(=O)N(C(C(C)C)c2ncc[nH]2)CCN)=O)ccc(OCCCO)cc1 c1(CNCC(c2ccc(Cl)cc2)N)ccc(N2CCOCC2)nc1 c1(OC)ccc(NC(=O)NCCCOc2ccc(C#N)cc2)c(Br)n1 C(=O)(CCCCC(C)(C)C)NC1C(C)CCN(C(C(CC#C)CC#C)=O)C1 N1(C(C(C)N(CCCCCC)C)=O)CCOCC1CN(C(=O)CSC(C)C)C Cc1c(C(=O)NCC(C)N(C)C(c2ccccc2C2(C)CCO2)=O)nn(C)c1N Cc1ccc(CN2CCC(O)C(C(=O)NCc3ccoc3)C2)c(Cl)c1Cl N1(CCN(C)C)C(=O)CCC1C(N1CC(c2cccc(F)c2)(C)C1)=O CC1(C)COCC(C(N2CCC(NC(c3ccc(C#N)s3)=O)C2)=O)O1 N1(c2ncc(C#C)cn2)CC=C(CCNC(=O)C(C)Sc2nncn2C)CC1 C(=O)(CC(C)C(C)C)N1CCC(C(N)=O)(CNC(C(C(C)C)N(C)C)=O)C1 C1(NC(=O)CC2CCC3(CC2)CC3)CCc2nncn2C1 Cc1ccnc2c(C(=O)NC3CCCC3CNC(=O)CNC=O)cccc12 C(CNC(=O)CNc1ccc(C(C)(F)F)cc1)(CC(C)C)NC(C=CC=CC)=O c1(C(C)(C)C)nc(S(=O)(=O)Nc2nonc2C(=O)O)cn1CCC(=O)N(C)C N1(CC(=O)NCC(C)N(C(C2CCCC2)C=C)C)Cc2ccccc2C1 C(CN=c1nc(N2CCN(C)CC2)[nH]c(N2CCOC(CC(N)=O)C2)n1)SC CC(C)CC(C(=O)NCC1CCC(=O)N1)ONC(=O)Cc1ccco1 CC1CCN(C(=O)COCC2CCCO2)C1CNC(c1ccc(Cl)nn1)=O S(=O)(=O)(c1c[nH]ccc1=NCCC1CCCN(C)C1)NC1CCN(CC)C1 C1(C(=O)NCCc2ccc(C)cc2)CN(C(=O)Cc2cc(C)[nH]n2)CC1(F)F C1(N(CC(N2CCCC2CNC(=O)CC2(CO)CCC2)=O)C)CN(S(N)(=O)=O)C1 c1(C(N2CC(C)C(CNC(c3cc(=N)[nH]n3C)=O)C2)=O)coc(S(N)(=O)=O)c1 C1(OC(c2c(CC)nns2)=O)COc2nccnc2C1 c1(N2C3CN(C(CCCC#C)=O)C(C3)C2)ncnc2ccccc12 C1(CNC(=O)Cc2ccc(Br)cc2F)CC2(CCOCC2)CN1 C=CC(CC)C(=O)NCCOCCCNC(=O)C(C1(O)CCOCC1)(F)F N1(C(Cc2c(C)nc(C)s2)=O)CCN(C(=O)Cn2ccc(O)nc2=O)C(C)C1 C1(C(CNC(C2(CNC(C=CC)=O)CC2)=O)O)CCCCC1 Cc1nc2cc(C(=O)NC3(CNC(=O)CS(C)(=O)=O)CCC3)cnc2s1 CC12CN(C(c3cccc(Cl)c3F)=O)CC1CN(C(=O)C(F)CC1CCC1)C2 C1(N)(C)CCN(C)C1.c1(CCN(C(C(=O)NS(CC)(=O)=O)=O)C)ccccn1 N1(C(c2ccc(F)c(F)c2F)=O)CCC2CN(C(=O)CC34CCC(CC3)C4)C2C1 C12(C(=O)NCCCNC(C(C)OC3CCCCC3)=O)CCCCC(=O)N1CCC2 C1(NC(CC(C2CC2)NC(C(C)(C)Cl)=O)=O)CCOCC1F c1(CCC)cc(C(=O)NCCCC(C)(C)NC(=O)CCOC(C)=O)sc1C c1(C(=O)O)cc(C(=O)NCCC2(O)CN(C(C3(CC)CCCC3)=O)C2)ns1 N1(C(c2c(OC)ccc(OC)c2)=O)CC2CCC(C1)N2C(C1CCC(O)C1C)=O CC(C(=O)N1CCC(N(C(=O)Cc2ccc(O)cn2)CC2CC2)C1)C(C)(C)C CC1c2ccccc2CN1C(=O)C(n1cc(CSCCCO)nn1)C C(=O)(CS(N)(=O)=O)N(CCNC(Cc1cc(C)no1)=O)C1CC1 c1(C(=O)NC2CC(NC(CCc3c(C)ncs3)=O)C2)cc(=O)cc[nH]1 CCCC(C)(C)CC(=O)N1CC(OCC(N2CC(O)CCC2C)=O)C1 CCCCC(C)C(=O)N(C(C)(C)CC(=O)NCC1CCCNC1=O)C C12(C(=O)NCC3CN(C(C4CN5CCC4CC5)=O)CC3O)CCC(O)(CC1)CC2 c1(COC)ccc2c(c1)OCCN2S(=O)(=O)c1cn(C(C)C)nc1C(C)(C)C c1(CC(=O)NCCC(N2C(CC(=O)NC)CC2)=O)ccnn1C C1(C(=O)NCC2CC2)COCCC12CN(C(=O)CCc1ccccc1)C2 CC(C)C(O)CC(=O)NCC(C)C(C)(C)NC(c1ccccc1CO)=O C1(NC(C(F)(F)C2(OC)CCC2)=O)CCN(C(=O)CSC2CC2)C(C)C1 N1(C(CC(C=C)C)=O)CC(NC(c2coc(CO)c2)=O)CC2(CC2)C1 C1(C(=O)NCCN(C(c2c(COC)nn[nH]2)=O)C2CC2)CCC(C(F)(F)F)CC1 C1(C(=O)NC2CC(NC(C3C(C)OCCC3)=O)CC2O)Cc2nccnc2C1 C1(CCNC(C(CC)F)=O)CC(F)(F)CN1C(c1cc(C)cc(Cl)c1)=O C1(CC#C)(C(=O)N)CCCN1C(=O)COC(N1CCC(OC)CC1)=O.C1(O)CCC1 N12CCC3CN(CCC3C1)C(=O)O2.C=CC1CCCN1C(CC1CC1)C(=O)OC C(=O)(CCCC(C)(C)NC(=O)COCc1nc[nH]n1)N1C(CC)COCC1 C1(NC(=O)C=C(C2CC2)C2CC2)CC2(CCCN(C(=O)CC3(O)CCOC3)C2)C1 C=CCCCCC(=O)N1CCC(CCC(N2CCC(O)(COC)C2)=O)C1 C(CCN=C(NC1CCC1)N1CCC(O)C(C)C1)c1c(C)ccs1 C1(NC(=O)C(=O)NC2CC3CC2CC3(F)F)COC2(CCOCC2)C1 c1(OC)ccc(C(=O)NCCCC2CCN(C(C3CC3(F)Cl)=O)CC2)nn1 C(=O)(CCC(CC)CC)N(CCC)CCNC(=O)CN1CCCC(N(C)C)C1 C1(C(N(CC(CN(C(C2CCC(CC)O2)=O)C)O)C)=O)CCc2nccn2C1.NC C1(C(=O)NCCCN(C(C(CC)n2ccnc2)=O)CCO)CCCC2(CCC2)O1 c1(C(=O)NC2(C)CC(NC(C(F)OC)=O)C2)cnn(C)c1Cl n1(CC)cc(CC(=O)NCc2csc(C(=O)NCc3cn(C)nn3)c2)cn1 Cc1nc(C)c(CCC(N2CCOCC2CNC(=O)CC2CCCO2)=O)c(O)n1 C(=O)(CCCCCC(C)C)N1CC(CC(N2CCC(C=C)C2)=O)(CO)C1 C1(NC(C2(c3ccsc3)CC2)=O)CC(NCc2cc(Cl)ccn2)C12CCC2 Cc1nc(CO)ncc1C(N1CCCC(Cn2cc(C3COCC3O)nn2)C1)=O N1(C(c2cc(CNC(=O)C3=COCC3)sc2)=O)C2CCCC1CC2 C1(NC(C2(NC(C)=O)CCCC2)=O)CC2(CCN(C(=O)CC(C)C3CC3)CC2)C1 C(=O)(C(C)C(C)NC(c1coc(CNC(c2csc(C(C)=O)n2)=O)c1)=O)OC S(=O)(=O)(c1cccs1)N(CC(N1C(=O)CNC1=O)=O)C C1(C(=O)NOCCc2ccncc2)CCN(C(C2CC2O)=O)CCO1 c1(C(=O)NCCCC(C)NC(C=CC=CC)=O)ncnc2c1ccn2C CCC(C)C(O)C(=O)Nc1cc(COC)nc(CC)n1.C12CCC(F)(CC1)CN2.C=O c1(C(N2CCC3CN(C(c4csc(C)c4C)=O)CC32)=O)csc(N=S(C)(C)=O)n1 C(N=c1[nH]c(=NCc2nc(CO)cs2)c2sccc2[nH]1)c1nccc(CC)c1 C1(CNC(C2C(C)CCCC2)=O)CC2(C1)CN(C(c1cnc(O)o1)=O)C2 C(=O)(C1=CCC(C)(C)CC1)N1Cc2c(C(=O)NC3(C)CCC(C)C3)n[nH]c2CC1 N(C1c2ccccc2CC1O)C(=O)NCC1CCCC12CCC2 c1(C(N2C3(CCCN(C(C)=O)C3)CCC2)=O)coc2c(Cl)c(Cl)ccc12 C=CC(C)(O)C(=O)N1CCN(CCn2cc(-c3csc(C(=O)O)c3)nn2)CC1 C1(C(=O)NC(C)CNC(=O)C=CC(CC(F)(F)F)=O)CCCN1C1CCCC1 c1(CC)c(C(=O)NCCCCC(C)(C)NC(C2CC(C)N(C)C2)=O)cccc1F c1(N(C)C)nc(C(=O)N(C2CCN(C(c3cccc(F)c3Cl)=O)C2)C)[nH]c(=N)n1 C1(C2CCN(C(C3CCCOC3)=O)CC2)(NC(c2c(C(C)C)ocn2)=O)CCC1 C#Cc1ccc(CC(=O)NCC2(NC(c3nnn(C)c3N)=O)CCOC2)cc1 N1(C(C(C)(C)N2CCOCC2)=O)CCC2(CCCCC2C(=O)O)C1 c1(C(N2CC(NC(C3CC(OCC)C3)=O)C(CO)CC2)=O)c[nH]cc(Cl)c1=O C(=O)(C1=CC2(CN(C(c3cc(O)n(C)n3)=O)C2)OC1)NCc1ccc(CC)cn1 C1(CC(N2CC(COC)C2)=O)C2CCCC2N1C(=O)C(C)(C)C(C)C C1(C(C)O)COCCN1C(c1ccc(CNC(=O)C(N2CCOC2=O)C)o1)=O CON(C(=O)C1OCCOC1(C)C)C1CCC1.c1ccccc1 CC(C)CCCC(=O)NC(Cc1ccoc1)C(N1CCCC(N2CCC2)C1)=O C(C(=O)N=c1ccc2cc(C(F)(F)F)[nH]c2[nH]1)=Cc1c(F)ccc(OC)c1 c1(C(N(C(C)C)CCN(C)C(C2(S(C)(=O)=O)CC2)=O)=O)cc2ccc(F)cc2o1 c1(C(=O)NCC2CC(O)CN2C(c2cnco2)=O)oc2ccccc2c1C(F)F C1(F)(CNC(CC(C)n2cccn2)=O)CCCN(C(C2(C#N)CCOC2)=O)CC1 c1(CC)c(C(N2CC=C(CNC(=O)COCC(F)F)CC2)=O)cccc1F c1(CNC(=O)NC(c2ccccn2)CC)cnccc1C Cc1cccc(C(O)C(=O)N(C2CCC(O)(C(F)(F)F)C2)Cc2ccccc2)c1.NC c1(C(N2C3C(NC(C(C)N(C)C)=O)C(CC3O)C2)=O)c[nH]c2cc(F)ccc12 N1(C(CCOCCOC)=O)CCC(C(C)NC(=O)COc2cnn(C)c2)C1 CCCC(CC)CCC(=O)NCC1(NC(c2ccn(C)n2)=O)CC2CCC1CC2 c1(C(=O)NCC(C)CN(C(=O)C(C)(C)N(C)C)C)c[nH]c(=N)c2[nH]ccc12 C(=O)(CC1C(=O)Nc2ccccc21)N1CCC(N(C(C2(Br)CC2)=O)CC)C1 C12(NC(C=CCC)=O)CCOCC1CN(C(=O)Cn1nc(C)ccc1=O)C2 Cc1cc(C(N2CCC(NC(C3CC(CCF)C3)=O)C2)=O)c(Cl)cn1 N1(C(C(C(C)C)OCC)=O)CCCC2(C1)CN(C(c1scnc1C(F)(F)F)=O)C2 Cc1nc2cncc(C(=O)N(CCC#N)CCNC(=O)CSC3CC3)c2[nH]1 C1(CC(N2CCCCC2C(F)F)=O)CC2(C1)CN(C(c1ccc3c(c1)CC3)=O)C2 Cn1nc(C2CC2)nc1CC(=O)NCC1CCCCC1NC(=O)C(O)C1CC1 c12ccc(Br)cc1C(=O)N2.Cc1ccccc1C(=O)N(CC(=O)CC#N)CCO N1(C(c2ccc(O)nc2)=O)CCOC(C(N2CCC(O)C2)=O)C1 CC1(C)CC(C)(CNC(=O)CCC2CCCN2C(C2CCC(=O)N2)=O)C1 c1(C(N2CCCC(CCNC(Cc3cn(C)nc3)=O)C2)=O)coc2c1CCCC2 CCCC(CC1CCCC1)C(=O)OCC1C(NC(=O)OC(C)(C)C)C1 N1(C(C(C=C)(C)O)=O)CCC2CCC(Nc3ncnc(Cl)c3C(=O)OC)C1C2 C1(NC(C=CC)=O)CC(OC)C12CCN(C(=O)Cn1nc(Cl)ccc1=O)CC2 C1(CC=C)(NC(=O)CCNC(C)=O)CCCN(C(=O)C(C)n2cccn2)C1 C1(CC#C)(C(=O)NCC2C3CC2N(C(C2CC4CCCC4C2)=O)C3)CCCOC1 C(=O)(CCC(=O)OC(C)(C)C)NC1CC(C)(NC(C2CC2(C)C(F)F)=O)C1 c1(OC)cc2c(cc1CNCC1CCC3(CCC3)C1O)CC(C)O2 C1(C(=O)N(C2(CO)CCOC2)C)(COC)CC(F)(F)C1 C1(C)(CCNC(C2(OC)CCC2)=O)CCN(C(=O)CN2CCC(F)(F)C2)C1 CCS(=O)CC(=O)N1CCCC1C(C)(C)CNC(=O)Cc1cnc(C)[nH]1 CC(C(=O)NCC1(C)CC(C)(C)C1)C(C)NC(c1ccn(C2CC2)n1)=O c1(C(N2CC(C)(NC(C3CSCCS3)=O)C2)=O)ccnc(F)c1O O=S(=O)(c1ccc(N2Cc3c[nH]c(=N)nc3C2)nc1)N1CCN(S(C)(=O)=O)CC1 C(C)(c1ccccc1F)=CC(N1CCN(C(C(C)SC)=O)C(c2cn[nH]c2)C1)=O Cc1cccc(S(=O)(=O)N2CC(NC(c3nccc(Cl)c3C)=O)C2)c1 Cc1ccc(OCCC(=O)NCC(C)NC(c2cccnc2S)=O)c(C)c1 C1(NC(C(CC)C(C)O)=O)CN(C(c2cc(CC)[nH]c2C(C)C)=O)CCC12CCC2 N1(C(c2c(C)csc2)=O)CCCC2(CCN(C(C3(F)CC=CCC3)=O)C2)C1 N1(C(C2(O)CCN(C(c3nn[nH]c3C(F)(F)F)=O)C2)=O)CCCC(F)(F)C(F)C1 c1(OC)cc(Cl)cc(C(=O)N(C2CN(C(c3cnn(C)c3)=O)CC23CC3)C)c1N C=CC1(C(=O)NC(C2CCN(C(c3scc(C)c3Cl)=O)C2)(C)C)CCOCC1 CN1CCC(C(=O)NCCC(O)C2CCC2)(NC(c2ccc(=N)[nH]n2)=O)C1 N1(C(C(N2C(CC)CCC2)=O)=O)CCC(C)(CNC(C2CC2(F)F)=O)CC1 Cc1nn(-c2ccc(F)cc2)nc1C(=O)NC(C1CCCN1C(=O)C=CCO)C CC1CCN(C(=O)C=C(Cl)Cl)C1C(=O)NCCC(=O)NC(N)=O c1(C(CC(=O)NCC(C)NC(c2nc[nH]n2)=O)C)cccc(F)c1.C1CC1 N1(C(c2nc(N(C)C)oc2)=O)CC(C(N2CC(C)(C)C2C2CC2)=O)CC(C)(C)C1 C1(NC(C2(CC#C)CCCC2)=O)CN(C(=O)CC2CC(C)=NO2)CC1C C(CCC(O)C(=O)NCC1CC(F)(F)C1)NC(C1C(C(C)(C)C)CC1)=O C1(OC)CN(C)C(C)(C(=O)NCCC2(O)CN(C(c3cc(C)ccn3)=O)C2)C1 CC(C)CCN=C(NCC1CCOC1)NCC1COC(=O)N1 n1(CC)ncc(C(=O)NC2CCCC2CNC(C2(C(F)F)CC2)=O)c1Cl C(=O)(CC(C)C(=O)N(C(C)CCNC(c1ccccc1C1(C)CC1)=O)C)OCC c1(CSCC)ccc(C(=O)NC(CC(C2(NC(C)=O)CC2)=O)(C)CO)cc1 N1(C(c2ccn(C)n2)=O)CCCC2(NC(=O)Cc3cccc(CO)c3)CCCC12 c1(C(N2CCN(C(=O)C=Cc3cccnc3)C(CF)C2)=O)cccc2c1CCO2 N1(C(=O)NC(CCCC(=O)Nc2cccc(C)c2)C)CCOc2cccc(Cl)c2C1 C(=O)(C(O)C(F)(F)C(F)(F)F)NCC(C1CCN(C(CC=CC)=O)CC1)(C)O N1(C(C2CCC(C(=O)NC3(CC)CC3)C2)=O)CCc2c(O)n[nH]c2C1 N1(C(CNC(CC(C)C)CCc2ccccc2)=O)CC2CC3CC2C1C3 C1(OC)CC(CNC(C2NC(=O)CC2C(F)(F)F)=O)N(C(=O)COC(F)F)C1 C(=O)(C(F)(F)F)NC(C)C(=O)NCC1CC(NC(C2CCCN2C)=O)C1 c1(NCC2C(F)(F)CCN(C(CCCC#C)=O)C2)ncnc2ccc(OC)nc12 Cc1cc(CO)oc1C(N1CCC(N(C(=O)CS(C)(=O)=O)CCO)C1)=O c1(C(=O)NCCCN(C(COCC(=C)C)=O)C(C)C)ccc(OC)cc1 C1(CC(=O)NCC2CNCCC23CC3)(C(=O)OCC)CCCNC1=O C1(CC(C)C)C(=O)O1.c1(C2CC(=O)N2)cccc(F)c1.c1(C(C)=O)ccc(C(C)=O)s1 Cc1cccc(C(=O)NCC2OCCC2C(=O)NCCC2CC2)n1 C1(C(=O)NCCn2cnnc2)CC2(CCC2)CN1C(c1cncc(Cl)c1)=O N1(C(c2ccc(CCC)cc2)=O)CCN(C(=O)C=CC(F)(F)F)CC1C(C)C N1(C(C2(C)CC(C#N)C2)=O)CCC2(CC1)CC2CNC(C1CC1c1cccs1)=O c1(N(C)C)ccc(C(N2CCC3(CC3C(=O)NCC3(F)CC3)C2)=O)c(F)c1 C(=O)(C1=CCCOCC1)NC(c1cccc(C)c1)CNC(=O)C1=CCOCC1 C(CC(CS(=O)(=O)c1ccccc1)NC(c1ccc(N)cn1)=O)OC C(=O)(C(CO)C(C)(C)C)N(CCCNC(c1ccc(COC)o1)=O)C(C)C C1(NC(c2ccc(C)n2C)=O)CCCCC1C(N1CC(N(CC=C)C)C1)=O C1(NC(CC=C=C)=O)CN(C(c2c(C(F)(F)F)cccc2O)=O)CC12CCOCC2 c12cnn3c1CN(CC3)C2.c1(OCC)ncccc1C(=O)Nc1ncncc1Cl N1(C(C2C(NC(C)=O)CC2)=O)CCC2C(O)C(C)(C)C12 C1(CNC(=O)COC(F)F)CC2(CCC2)CN1c1cc(C(F)F)ncn1 C(C(C)C(=O)NC(C1(NC(=O)CCN2CCC(F)C2)CC1)=O)OC c1(C(=O)NCC(CO)NC(c2cc(-c3ccccn3)no2)=O)nnc(O)cc1O C1(C(N2CCCC(C)(NC(c3c(C)c(O)ccc3)=O)C2)=O)CCc2c[nH]nc2C1 C=CCC(CC(=O)NCc1cnccc1Cl)NC(=O)C(C)S(C)(=O)=O c1(CC(=O)NC(CNC(CC=C=C)=O)C2CCC2)c[nH]c2cc(C)ccc12 N1(C(C2C(C=C)CC2)=O)CCC(NC(=O)Cc2ccc(C)cc2Cl)C(CO)C1 c1(CC(=O)NC2(C)CC(NC(C(C)=C(C)C)=O)C2)cccc(Cl)c1F C1(C(=O)NCCN2CCN(C(CCC(CC)C)=O)CC2)CCn2ncnc2C1 N1(C(c2nnc(O)nc2O)N2C(CC(=O)OC)CCC2)CC2CCC2(C)C1 C1(C(=O)NC2CCCN(C(C3(C)CC3(Cl)Cl)=O)C2)CCCS(=O)(=O)C1 c1(C(=O)NCC2CC(NC(C(c3n(C)ncc3)O)=O)C2)ccc(C#N)o1 N1(C(c2cn(C)cn2)C(=O)Nc2ccc(OC)cc2C)CCn2ncc(Cl)c2C1 N1(Cc2c(-c3cccc(Br)c3)csc2)CCOC2(CCCCC2)C1 C1(NC(C(CCC)OCC)=O)CC2(CCCCN2C(c2ccsn2)=O)C1 N1(C(C2CC(=C)C2)=O)CC23CCCCC2(C1)CN(C(c1ccc(F)cc1Cl)=O)C3 c1(CC(N2C(CNC(=O)COC(F)F)CCCCC2)=O)ccc2nonc2c1 CC1CCN(C(c2cc(CNC(=O)C(C3CC3)C3CC3)no2)=O)CCO1 CC(CC(=O)N1CCC(O)(CCNC(c2cnc(O)o2)=O)C1)C(C)(C)C C1(CNC(c2n(CC)ncc2C)=O)CN(C(c2ccnnc2)=O)C(C)(C)C1 N1(C(CS(=O)(=O)N(CC)CC)=O)CCC2CC2(NC(=O)C2=C(C)CCC2)CC1 C1(C)(C(=O)NC(C)CC2CN(C(C3CCOC3)=O)C2)COC(=O)OC1 C(CNC(c1ccc(Cl)s1)=O)(C(C)(C)C)NC(c1ccc(C)s1)=O C1(C(N2CC(COC)N(C(=O)CCc3ccsc3)CC2)=O)CCCCN(C)C1=O Cc1cc(C(F)(F)F)ccc1C(N1CCOC(CNC(=O)C2=NNC(=O)C2)C1)=O C1(CNC(C(C2(C)CC2)NC(Cc2cncc(C)c2)=O)=O)CC(C(N)=O)=NO1 CC(CN1CCOC1=O)CN=c1nc(N2CCOCC2)[nH]c(-c2ccccc2)n1 Cc1ccncc1C(C)(C)C(=O)NCC(n1cc(CCC2CCOCC2)nn1)C N#Cc1cc(Cl)ccc1COC(=O)CCc1ncc(-c2cccc([N+](=O)[O-])c2)o1 C1(CCNC(C=C(COC)C)=O)CC2CCC(C1)N2C(c1csc(Cl)n1)=O N1(C(C(C)OCC#C)=O)CCC(NC(c2ccncn2)=O)C(CO)CC1 C1(CN2CCN(C(c3c(CC)cc(Cl)cc3)=O)CC2)COC2(CCCCC2)C1 C1(CC(C)O)CCN(c2nnc(-c3cnsn3)n2-c2ccccc2)CC1 C12(CC(=O)N(CC(C(=O)OC)C)C)CCC1CN(C(=O)CC1CC1OC(C)=O)C2 C(C(C(C)(C)C)NC(=O)CC=CC1CCCCC1)NC(C1C(=C)C1)=O c1(CC(=O)NCCN(C(C2(O)CCC2)=O)CC2CC2)ccc(Cl)cn1 c1(OCCC(=O)NCCCCCNC(CCCCOCC)=O)c(C)nn(C)c1C N1(CC(=C)CC)CCC(C2CCCO2)C1 c1(C(N(C2CCN(C(c3ccc(SC)s3)=O)C2)C)=O)cn(C)nc1O C1(CNC(CC(=O)NCC#C)=O)CC(C(C)(C)C)CN(C(C2(C)CC2)=O)C1 Cc1nc(NC2CC2)sc1C(N1CC(NC(C2(C)CCCCC2)=O)C(F)C1)=O c1(CC(=O)N(CC(C)NC(C(COCC)C)=O)CC)ccc(OC)cc1C N1(C(c2c(Cl)c(C)n(C)n2)=O)C2CCC1CC(CNC(C1C3CCCCC13)=O)C2 c1(C(=O)NC(CC=C)CNC(C2CC(C)=NO2)=O)nc2cncnc2[nH]c1=O N1(C(C(C)(C)CO)=O)CC(C(=O)NCC(C)(C)n2ccnc2)CCC1(C)C C1(NC(CC(C)c2cccnc2)=O)CC12CC(NC(C13CC(CF)(CO1)C3)=O)C2 N1(CCC(=O)OCCC(C(=O)OC)(C)C#N)C(=O)C2CC=CCC2C1=O C1(Cc2ccccc2)Cc2ccccc2NC1C(N1CCC(F)(C(=O)O)CC1)=O c1(SC)cscc1C(=O)NC1CCCC1CNC(c1cc(C)ns1)=O C1(CNC(C=CC(C)C)=O)CC(NC(c2cnn(CC(F)(F)F)c2)=O)C1(C)C C1(NC(c2cc(C)nn2CCO)=O)CN(C(c2cnnn2C2CC2)=O)CCC1F N1(C(C2CN(CCOC)C(=O)C2)=O)CCCC2CN(CCOC)CC12 c1(C(N2C3CN(C(c4c(OC)cccc4OC)=O)CC32)=O)nc2ccccc2s1 O=C(C1CCCc2scnc21)NC1CC2CCC(C1)N2C(=O)CC1CCCS1(=O)=O Cc1c(C(N2CCCC2C(C)(C)C(=O)NC(C)CC(F)(F)F)=O)ncn1C C1(NC(C2(C(=O)NC)CC2)=O)COCC1CNC(=O)Cn1nccn1 N1(C(C(CC)N(C(C)=O)CC)=O)CC(C(N2CCC(O)C2)=O)C2(CC2)C1 C(C(=O)N1CC(NC(c2ccncc2F)=O)C(F)C1)(C(C)(C)C)NC(C)=O CC1C(=O)CCC1CC(N1CC(CNC(=O)CCC2COC(C)(C)O2)C1)=O C1(C(N2CC(C)NC(=O)C2)=O)N(C(=O)COCC(F)F)CCCC1(C)C C(=O)(C(C)C(C)C(C)(C)C)NCCN(C(=O)C(=O)NOC)CCC N1(C(C2(COC)CC(=O)C2)=O)CC(CNC(C2CCC(=O)NC2)=O)CC12CCC2 CC1CC(CNC(c2ccc(=O)n(O)c2)=O)CN(C(c2cncnc2)=O)C1 N1(C(CCC)=O)CC(NC(=O)C2=CCCCO2)CC1(C)COC C=C(Cl)CC(C(=O)N1CC(OC)C(C(N)=O)C1)NC(c1ccc(C)nc1)=O Cn1nc(C(N2CCOCC2C(=O)NC2CSC2)=O)ccc1=O N1(C(CN(C(C(C)n2ccnn2)=O)C)=O)CCCN(C=O)CC1.C12CCC(C1)N2 Cc1ccc(C(N2CC(NC(=O)CCC(N)=O)C(F)C2)=O)nc1 c1(C(=O)NCC23N(C(c4cc(C)n(C)c4)=O)CCC2CC3)csc2c1CCCC2 C1(C(C)NC(=O)CCc2nc(C3CC3)no2)CCCCN1C(=O)CN(C)S(N)(=O)=O N(C(=NCCN1CC=CC1)NC1CCOC1)CC(c1ccccc1)OC C1(C)(C(=O)NC(C)CC2CCC2)CCCN(C(c2cc[nH]c(=N)c2N)=O)C1 c1(C(N2CC(CNC(Cc3cccc(C)c3)=O)OCC2)=O)cc(Cl)c(N)cc1Cl C(=O)(CC(C)(C)C#N)N1CCC(CN(C(Cc2c(C)scc2)=O)C2CC2)CC1 N1(C(C(C)N(C(CCOCCC)=O)CC)=O)CCNC(=O)C1CC C=CCC(CO)CN=C(NCC1CC(C)(C)CN1C(=O)OCC)NCC.C(C)(C)(C)OCC c1(C(C)=O)ccc(COCC(=O)NCC2CC(NC(=O)CC(=O)N(C)C)C2)cc1 N1(C(C(CC)N(CC)CC)=O)CC(F)(F)CC1CCCNC(C1CCOC1C)=O c1(C(N(C)CC2CCN(C(=O)CC34CCCC3C4)C2)=O)cnc2ncnn2c1O CCCCC(C)CCC(=O)Nc1cc(O)ncn1 c1(CCC)cc(C(=O)NC2(CN(C)C(c3oc(C)nc3C)=O)CC2)cc(O)n1 c1(C(N2CCN(C(c3cc(C)c(Cl)s3)=O)C3C2C3)=O)cccc2nc(O)ccc12 S(=O)(=O)(c1ccc(F)c(F)c1)N.N1(C(c2c(C)cnc(Cl)n2)=O)CCC2COCC2C1 C1(C)(C(=O)OCC)CC1C(=O)NC(C1(CN=[N+]=[N-])CC1)C1CC1 C1(C(=O)NCC(C)NC(Cn2c(=O)ccc(C)n2)=O)CNC(=O)C(C)(C)C1 CC1CN2CCN1CC2C(N1CCN(C(C2CC3CCC(C2)C3)=O)CC(C)C1)=O c1(OC)ccc(NC(=O)NCCC2CCCCC23CC3)cc1I C(CC(CC)(CC)NC(=O)Cc1cc(Cl)ccc1Cl)NC(CC(=O)NC)=O N1(C(c2cc(C)sn2)=O)CCC(C)(C)C(NC(C2CCOCC2(C)C)=O)C1 N1(C(c2c(C)nc(C)o2)=O)CC2(CC(NC(C34CCOC(C)(C3)C4)=O)C2)C1 CCC(CC)(C(=O)NCC1(O)CCN(C(c2nc(C3CC3)oc2C)=O)CC1)OC C1(NC(C2(C#C)CN(C(=O)Cc3c(C)n[nH]c3C)C2)=O)CC2CCC(C1)O2 C(=O)(C1=C(C)OCCC1)NC1(C)CCCN(C(C(CC)Oc2ccccc2)=O)C1 N1(n2ccc(C#N)n2)CCC(c2ccccc2)C(F)(F)CC1.C12(COC1)CC(=O)N2 CCC(C(=O)NCC1COCC1NC(=O)CC#N)n1ccc(C2CC2)n1 C1(NC(CCC(CC)OC)=O)COC2(CCN(C(=O)CN(C)CCOC)CC2)C1 C(=O)(C1CCCc2n[nH]cc21)NCC1(CNC(C(CC)(C)CC)=O)CC12CCC2 S(=O)(=O)(c1ccc(=NCC2COCCN2C)[nH]c1)N(C(c1cccc(C)n1)C)CC N1(C(C(C=C)CC)=O)CCC(NC(=O)CC(C)F)C2(CCC2)C1 N1(C(c2ccc(OC)nn2)C(=O)NC2(C)CC2)CCCc2ccccc2C1 C(=O)(C(O)C(C)c1ccccc1F)NCCN(C(=O)CC1(C)OCCO1)CCC N1(C(CN(C)C(N)=O)=O)CC(NC(c2cc(C3CCCCC3)on2)=O)C2CC12 N1(C(CN(C2CC2)CC)=O)CCC(CNC(=O)C(F)(F)C(C)O)C12CCC2 C1(SC)CN(C(=O)CC2(C)CCCO2)CC1NC(c1sc(N(C)C)nc1C)=O c1(COCc2ncc(C)[nH]2)ccc2ccccc2n1.c12cccc(c1)NC(=O)N2 c1(C(N2C(CNC(c3c(CC)cno3)=O)CC2)=O)ccc2cc[nH]c2n1 N1(C(c2nnn(C(C)(C)C)n2)=O)CCC2CCC(NC(=O)C=C3CCC3)C1C2 CSC1=C(C(=O)N2CCC(C(C)NC(c3cc(Br)oc3C)=O)C2)CCCC1 C1(NC(=O)Nc2n(C)nc(N3CCCC3)c2)CC2C=CC1CC2=O c1(C(=O)OCc2c(C)cc(F)cc2)nccc2ncncc12 C1(F)(C(N2CC3C(CNC(=O)CC(F)(F)F)C3C2)=O)CCCCCC1 c1(OC)cncc(C(=O)NC2CN(C(c3cc(SC)ccc3C)=O)CC2C)c1C C1(C(=O)NC2CCCC(C)(C)C2)CCN(C(c2n[nH]cc2Cl)=O)C(C)(C)C1 c1(OC)cc(N)cc(C(N2CCOC(CNC(C3CCNC3=O)=O)C2)=O)c1OC Cc1nc(C)n(CCC(=O)NCCC(C)N(C(=O)CN2CCCC(C(N)=O)C2)C)n1 C(=O)(CN=c1cc[nH]cc1)N1C(CN(C)C(c2cnc(O)s2)=O)CC(F)C1 C(C(=O)NCC(C)NC(C1CC2CCC1CC2)=O)(C(C)(C)C)OC C1(C(N(C)CCc2cccc(Br)c2)=O)C2CCC(C2)N1Cc1nc[nH]c1C(F)(F)F c1(CC(Cn2cc(Cn3c(C)ncc3)nn2)O)ccc(F)cc1 c1(SCCC(=O)N(C(C(=O)NCC(C)NN(C)C)C)C)ccc(F)c(F)c1 C1(C(N2C(C)(CNC(C(C(C)C)F)=O)CCC2)=O)COc2ccccc2O1 C1(C(N2CC(NC(C(CC=C)OC)=O)C(CCC)C2)=O)CCCCCN1C C1(NC(c2cn(CC)nc2)=O)CC(NC(C2(SC)CCC2)=O)C12CCC2 c1(C(N2CCC(O)(CC#C)CC2)=O)coc2c1CN(C(c1cnc(OC)s1)=O)C2 C(CC(C)C)(C(=O)N1CC(C)(NC(=O)CCCCCF)C1)NC(=O)OC Cc1cccc(C)c1CC(=O)NC1CN(C(=O)C(C)(C)N(C)C)CC1C(F)F N1(C(C=Cc2cc(C)no2)=O)C2CCC(C2)C1C(N1CCCCC(C)C1)=O C1(C2CN(C(C3(C)CCCC3CC)=O)C2)(NC(COCCOC)=O)CC1 c1(C(=O)NCCNC(C(C(C)(C)C)Cc2ccccc2)=O)cc2cccnc2o1 N1(C(c2ncsc2-c2ccccn2)=O)CCN(C2CCN(CCF)C2)CC1 CC1CC(C(N2CC3CCC(C2)O3)=O)CN(C(C2CCCC2O)=O)C1 C(CCC(=O)NCCC(O)CNC(=O)CC1CC1CC)COCC=C C1(C(=O)NCC2(C)CCC(NC(C(C=C)O)=O)CC2)Cc2cc(F)ccc2O1 C(=O)(CC1CCCc2cc(NC(=O)CC3CC3)ccc21)N(CC1(CC=C)CC1)CC1CC1 O=C1CCC(C(=O)NCCC2CC(NC(c3scnc3C3CC3)=O)C2)CN1 N1(C(CCCOC(C)=O)=O)CCN(C(C2CCC3CC23)=O)CC1c1cccnc1 Cc1ccc(CCC(N2CC(NC(C3(C)CCSCC3)=O)CC2C)=O)c(C)c1 C=Cn1nccc1C(N1C(C)(C)CCC1)=O.n1(-n2cc(CN)nn2)cc(C#N)cn1 C1(C(N2CCC(NCc3c(Br)ccc(OC)n3)C2)=O)Cc2ccccc2O1 N1(C(C(C)OC(C)=O)=O)CCC2(CCOC2)C(CNC(=O)COCCCOC)C1 C1(COC)CN(C(=O)C(CCC2CC2)NC(c2cc[nH]n2)=O)C1(C)C C1(NC(C2CC(SC)C2)=O)CC2CC1CN(C(=O)CC(C)C1CCCCC1)C2 CC12CN(C(C3(CO)COC3)=O)CC1(C)CN(c1ncccc1[N+](=O)[O-])C2 c1(CCCC)cc(C(=O)NCC(CNC(=O)C=Cc2cccs2)CO)c(C)o1 C1(CCC)CCCN(C(=O)C(CNC(c2ccsc2C#N)=O)N(C)C)C1 CCC(C)(C(=O)N1CCC(CCNC(c2cnccc2C)=O)CC1)C(N)=O C(CC(CC)(CC)N(C(c1ccc(-c2cc[nH]n2)cc1)=O)CC)NC(CCC)=O C1(CNC(CCCOCC)=O)CCCC(NC(=O)C(C)=C2CCC2)C1 CC1=C(C(=O)NC(C2CCN(C(c3cn(C)ccc3=O)=O)CC2)C)CCC1 c1(C(N(C2CN(C(=O)CCc3cccc(Cl)c3Cl)C2)C)=O)noc2ncccc12 c1(C(=O)NCC2(C)CCCN(C(C(F)=CC)=O)C2)ccc2c(c1)CCCCN2 CCC(O)C(F)(F)C(=O)NC1CCCN(C(=O)CC(C)c2cnn(C)c2)CCC1 c1(NC(C)=O)ccc(F)c(C(=O)N(CC(C)(C)CNC(C2CC2F)=O)C)c1 CC1CN(C(=O)C=CI)CC2(CCN(CCc3ccc4c(c3)OCCO4)C2)O1 C1(CNC(C(F)OC)=O)CCCC2(CN(C(c3ccc4c(c3)CCC4)=O)C2)O1 c1(C(=O)NC2(C(=O)NC)CC(F)C2)nc(C(C)=O)sc1C C1(CNc2ccc(C(CC)C)cc2C(F)(F)F)CC(C2CCCCC2)C1 Cc1nc(C(C)C)ccc1C(=O)NC1CCC1CNC(C1CN(C)CCO1)=O C=CCCCCCCCC(=O)N1CC2(C1)CN(C(c1cnsc1)=O)CC2CO C1(c2nc(C(C)SCC)nn2-c2cccc(SC)c2)CCOCC12CCCCC2 N1(C(c2ncnc(C)c2C)=O)CCCC2(CCN(C(=O)C(F)CC(C)C)C2)C1 C1(NC(CCCC(C)C)=O)CCC2(CCCN2C(=O)C2=NOCC2)CC1 C=CC1(C(=O)NC2CCN(C(=O)CCc3cc[nH]n3)CC2C)CCCCC1 CC(C)C(C(=O)NCC(C1CC1)N(C(=O)CN(S(C)(=O)=O)C)C)n1cccn1 N1(C(=O)CN2CCC(O)CC2)CC(C(N2CCC(CCF)CC2)=O)C(F)(F)C1 C1(N(C)C)CCc2ccccc2C1NC(c1nccc2c1CCNC2)=O Cc1coc(C(N2CCC(C(C)NC(=O)CCC3CCCC3)C2)=O)c1 C(C)(CO)(C(=O)NCCCCC(C)NC(c1cc(C)on1)=O)NC(C)=O N1(C(=O)CCC2CCCN2C(c2ccon2)=O)CCc2ccsc2C1 C(=O)(C1Cc2ccccc21)N1C(C(N2CC3CC3(CO)C2)=O)(CC)CCC1 C1(C(N2C(CNC(CC3(C#N)CCC3)=O)CC2)=O)CC2(C1)C(C(=O)O)C2(F)F C1(N(C(C=CC(C)NC(CSCC#C)=O)=O)C)CCN(C)C1=O C12CCN(C1)C(=O)C(OC)C=CC2.c1(C(C(=O)NNC)=O)cnn(C)c1 c1(C2(C(=O)NC(c3cccc(F)c3)C(=O)O)CC2)cccc(Cl)c1 c1(C(=O)NC(CC)(C)CNC(c2cccn2C2CCCC2)=O)ccncc1N N1(C(C=C(C2CC(N(C)C)C2)C)=O)CCN(C(c2nccs2)=O)CC1CCC N1(C(C(CCC)(F)F)=O)CC(C(=O)N(C)C(C)C)C(C2CC2)C1 CC(C)(C)C(O)CC(=O)N(CCc1cn(C(C)C)nn1)CC1(O)Cc2ccccc2C1.C1CC1 C1(CC(=O)NCCCOCCCNC(=O)CNc2ccccn2)CC=CCC1 C1(C(=O)NCC2CCCO2)Cc2cc(O)ccc2CN1C(c1cccnc1S)=O Cc1ncc(C(=O)NC2(COC)CCN(C(=O)C(C)Oc3ccccc3)C2)cn1 Cc1ccn(C(C)(C)C(=O)N2CCCC2C(C)(C)CNC(C2CC2C(C)O)=O)n1 c1(C(N(CC(C)CNC(=O)CCc2cn[nH]c2)C)=O)cnn2ccncc12 N1(C(c2ccc(C(C)=O)[nH]2)=O)CC2(CCN(C(C3(C)CCOC(C)C3)=O)C2)C1 C1(C(=O)NCC2CC=CCC2)(CNC(C2(N(C)C)CC2)=O)CC12CCC2 CCC(C(=O)N1CCC(C(F)F)(CNC(c2occc2C(C)C)=O)C1)C(C)(C)CC c1(C(N2CCN(C(c3c(Br)ccc(C)c3)=O)CC2)=O)cnc2c(c1)CCCO2 c1(C(N2C(CC(=O)NCC(C(C)(C)C)=O)COCC2)=O)c(O)cccc1F C1(CNC(C2C(C)C2)=O)(CO)CCN(C(=O)CC2CC3(CC3)CO2)CC1 N1(C(C2N(C)C(=O)CC2)=O)CC2CCC1CN2C(C1C2CCC(=O)C12)=O c1(C(=O)NCCCC(CO)NC(C(C)SCCCC)=O)cccc(F)c1C C=C1CCCN(C(C2C3CC4C(C3NC(C3(CC)CCNC3=O)=O)C24)=O)CC1 c1(C(CNC(=O)CC2(CN3CCCC3)CC2)NC(=O)CC2CC2)cc(F)cc(Cl)c1 C12(C(N3CC4C(CNC(C(C)CSC(F)(F)F)=O)(C4)C3)=O)C3C4C1C1C2C3C41C N1(C(c2cnc(CC)[nH]2)=O)CCC2(CC(NC(c3cc4sccc4[nH]3)=O)CO2)C1 C1(S(C)(=O)=O)(CNC(NC(CC=C)C)=NC)CC1 CC1CN(C(C2CCOC2)=O)CC2(CCN(C(=O)Cc3ccnc(O)c3)C2)O1 C(=O)(CCCC(C)(C)C)NCC(CNC(c1ccnc(OC(C)C)c1F)=O)C CC1OCCC1(C)NC(=O)COC1CCN(C(=O)CCn2ccnc2)C1 C#CC1(CNC(C2OCCC2CNC(=O)CCc2cc(C)on2)=O)CCCC1 N1(C(C=C(C)Cl)=O)CCC(C)N(C(C2CCCOC2c2ncc[nH]2)=O)CC1 N1(C(CCCCC#C)=O)CCC(C2CC2)(NC(c2cnc3[nH]cncc2-3)=O)C1 Cc1sc(C(N2CC(NC(=O)C3=CC4C=CC3C4)C(C3CC3)C2)=O)cc1[N+](=O)[O-] N1(C(C(CC=C)C)=O)CCCC(CC)C1C(=O)NC1CCC(=O)N(C)C1 N1(C(c2c(C)snc2)=O)CC2CC(NC(=O)CC3(N(C)C)CCCC3)CC2C1 C1(C(=O)NCC)CCC(C(C)C)N1C(=O)C(C)Nc1cccnc1 C1(C)(C(=O)NCC(n2cc(-c3ccc(C(=O)OC)s3)nn2)C)CCCO1 C1(CN(C(c2ccccc2)CC)C)OCCC(=O)N(C)C1Sc1ccccc1F c1(C(=O)NC2CCC(C(=O)NCCOc3ccc(C)cc3)O2)c(Cl)ccc(Cl)c1F CCC1=C(C(=O)NCCCCNC(C2CC2c2cccc(Cl)c2Cl)=O)CCCO1 C1(CC)CCOCCN1C(C1CN(C(c2nocc2C)=O)CC12CC2)=O c1(C(=O)NC(C)CNC(c2cnc(C(F)(F)F)cn2)=O)cc2n(n1)CC(O)CO2 N1(C(c2ccc(CC)[nH]2)=O)CCC(O)C(C(=O)Nc2conc2C)C1 C(CC1CCOC1)(C(=O)Nc1ccsc1)NC1CN(C(=O)OC(C)(C)C)C1 c1(C(c2nnnn2CC2CCCO2)NCCSC)n[nH]c(CC)n1.c1ccccc1 N1(C(c2c(C)noc2)=O)CCC(NC(C2CCCS2(=O)=O)=O)C(O)C1 C1(C(=O)NCC2(CC=C)CC2)CCCC(NC(=O)CN2CCC(C)CC2)C1 C1(c2n(-c3c(CC)cccc3)nnn2)(NC(c2nccs2)C)CC2(CCCC2)C1 C1(NC(CCCOc2ccc(C)cc2)=O)CN(C(=O)CC(C)C)CC1C1CC1 N1(Cc2c(C)cccc2)CC(CF)C(C#N)C1 Cc1ccccc1C(O)C(=O)NCCC(O)COCc1ccccc1.OC c1(-c2cn(C(C(N3CC(OCCCCC)C3)=O)C)nn2)ccc(=N)[nH]c1 C(C(=O)N(CCCCN(C(=O)CN1CCC(OC)CC1)C)C)(C(C)C)SCC N1(C(C=CC(C)C)=O)CCN(C(=O)CC2=NNC(=O)C2)CC12CC2 CC(C)CC(C)(CNC(C1CC1(C)C)=O)NC(=O)Cc1ccncc1 C1(CC(=O)N(CCCCN(C)C(=O)OC(C)(C)C)C)NC(=O)CNC1=O N1(C(CCc2c(C)ccnc2)=O)CCCC(CC(=O)Nc2cn[nH]c2)CC1 C(C(C(=O)N1CC=CC1CNC(=O)CCC1CCC1)C(C)(C)C)OCC=C C1(CNC(C(C)N(CC)CC)=O)CCCC2CN(C(C)=O)CC12 N1(C(C(CSC)OC)=O)CC2CCC1CC2N(C(=O)Cc1csc(C)c1)CCO N1(C(CCCC(=O)NC(C)C)=O)CCCC(NC(c2nnc(S)n2C)=O)C(F)C1 N1(C(C(C=C)(C)CCOC)=O)CCC2(CC1)CC(c1nn[nH]n1)CCO2 Cc1nc2cc(C(N3CCCC(C(C)NC(c4cccc(O)n4)=O)C3)=O)[nH]c2s1 C1(C(=O)OC)CC(C(=O)NCC(C)(C)CNC(=O)Cc2cnn(CC)c2)C1(C)C c1(OC)cncc(NC(=O)CC2(C)CN(C(=O)Cc3c(Cl)cccc3Br)C2)c1C C(C)(C)(CC(C)NC(=O)C(CCN(C)C)NC(c1ccncc1OC)=O)OC N1(C(c2n(C(C)C)nnc2)=O)CC2CCC(N(C)C(c3csc(S)n3)=O)C2C1 c1(C(=O)OC)ccc(C(=O)NC2CCCC(C(=O)NC(CO)C(C)C)C2)cc1O c1(CC(=O)N(CC(CC)NC(=O)C(O)CSC)C)cccc2ccsc12 n1(CCC(N2CCC(N(C(C(COC)O)=O)C)C2)=O)cccnc1=O Cc1ccc2c(C(=O)NC3CCCN(C(C4CC5CC5C4)=O)CC3)cnn2c1C C1(C(N2CCCC(NC(c3cc(OCC)ncc3)=O)C2)=O)CCN(CC)C(=O)C1 c1(SC)cc(C(=O)NC23CCN(C(=O)CCSCC(C)C)CC2C3)ccc1F c1(C(=O)NC(CC)(C)CCNC(=O)CN2CCCC2C)ccc(O)c(F)c1 C1(NC(C=CCC)=O)CN(C(=O)CC2C=CCC2)CC1C=C CCC(CNC(=O)C(CNC(c1cncc(NC)c1)=O)N(C)C)(CC)CO N1(C(C(C)OCCC=C)=O)CCCC2(C1)CN(C(C1CCC(OC)CC1)=O)C2 CC1=CC=C2C=CC=C1NC(=O)NC1CC2=NN=CNC1 C=CCCCC(C(=O)NCC(C)(C)SC)NC(=O)C(C)CC N#CC1(C(=O)NC2CC3CCCCC23)CC2CCC1CC2 C(=O)(C(C)(C)S(C)(=O)=O)N1CCC(OCCNC(c2c(C)ccc(CC)c2)=O)CC1 Cc1c(C(N2CCC(C)(NC(=O)C(O)C3CC3)C2)=O)cnc2ncnn12 C1(NC(C(C)SCCCC)=O)CC2(CCN(C(C3CC4C(C3)C4(F)F)=O)CC2)C1 C(=O)(C(F)C(C)(C)O)N(CCC(=O)N(CCCC(=O)OC)C)C1CC1 C1(C(=O)NCC(C)OC)CN(C(=O)CC(C)SC)CC12CCC2 c1(C(N(C(CC)CNC(=O)CSc2ccncc2)C)=O)cnc(C)c(C)c1 c1(C(N(CCCC)CCCO)=O)cncc(CNC(C2C(C)C2C)=O)c1 Cc1cc(C(=O)Nc2ccc(C)c(-c3ccc(-c4cccs4)s3)n2)cnc1Br c1(C(N(CCNC(c2cnc[nH]2)=O)CC2CC2)=O)ccncc1F C(=O)(C(O)CC(F)(F)F)NCC(CC(=O)NC(c1nc(C)on1)C)C1CC1 C#Cc1ccc(C(=O)NC(C(N2CCC(NC(N)=O)CC2)=O)C2(C)CC2)o1 C(=O)(C#CC1CCCO1)N1CCC(C(C)NC(CCC(C)C)=O)CC1 C1(CCC)CCN(C(=NC)NCc2cccc(C(C)(C)C)n2)C1 C#CC1(C(=O)NCC2OCCC2C(N2CC(OCCC)C2)=O)CCCC1 c1(C(=O)NC(CC(C)NC(CCOCC(C)C)=O)C)cc2c(Cl)nccc2o1 C(C(=O)NNC(=O)CS(C)(=O)=O)NC1C(C)CN(c2cc(Cl)nc(C3CCC3)n2)C1 N(C1c2ccccc2CC1O)C1CCN(c2cnc(Cl)nc2)CC1 C1(CC(N2C(C(CCC)C)CCC2)=O)CCN(C(=O)C=CCN2CCC2)CC1 c1(C(=O)NCC=CCNC(CCn2c(=O)sc(C)c2C)=O)cnc2[nH]cnc2c1 c1(OC)cnc(C(=O)NC2CN(C(=O)COC3CC=CC3)CC2OC)c(F)c1 c1(CNC(C(CC)n2cncn2)=O)cc(C)c(C(N2CCC(O)(CC)C2)=O)o1 C#CCC(C(=O)N(C)CCOC(F)F)NC(=O)Cn1[nH]cnc1=N C1(n2cc(-c3cn(C(C)C)nc3)nn2)CCCCC1NC(C1(C(N)=O)CC1)=O CCC(CC)CC(=O)N1CCC(N2CCN(C(C3CCN(CC)C3)=O)CC2)CC1 C=CC(C)(C)CC(=O)N1CC(C(N2CC3CC3(C(=O)OC)C2)=O)C(F)(F)C1 C1(C)(CNC(C(COC)N(C)C)=O)CCN(C(c2ccc(CC(C)C)s2)=O)C1 C1(NC(c2cc(C)on2)=O)CS(=O)(=O)CC1NC(C1(C#N)CC=CC1)=O c1(CC)ncc(CCC(N2CCC(N(C(=O)CCCOC)C)C2)=O)o1 C(C(=O)N=c1cc(-c2ccc(Cl)s2)o[nH]1)NC(=O)NC1CN(C(C)C)C1 CC(C)C(CNC(C1(C)CC1(F)F)=O)C(=O)NCCS(C)(=N)=O Cc1ccncc1C=CC(N1CCCC1C1(NC(c2nnc(C)s2)=O)CC1)=O N1(C(C2C(CC)CCN2C(=O)CC2(C#N)CC2)=O)CCOCC(CC)C1 C1(NC(C2CC(OC)C2)=O)CC2CCC(C1)N2C(c1cc(C2CCOC2)[nH]n1)=O C1(C(=O)NCCCCN(C(=O)Cn2ccc(C3CC3)n2)C)OCCCO1 CC1Cc2c(Br)ccc(Br)c2CN1S(=O)(=O)CCC1CC1 C(=O)(CC(F)(F)Cl)NC1C(CNC(c2cnc(OC)s2)=O)COC1 N1(C(C2(S(N)(=O)=O)CC2)=O)C2CCC1CC(NC(C1(CO)CCCO1)=O)C2 N1(C(CCC=C)=O)CC(NC(c2sc(C(C)=O)cc2Br)=O)CC12CCC2 C1(CC2(C(=O)NCc3cc(C)cc4c3cccc4)CC2)CC2(CCOCC2)CCO1 c1(C(=O)NC(C)C(C)NC(C2CC2F)=O)ccc(CS(C)(=O)=O)cc1 c1(C(N2CC(NC(c3cn(CC)nc3)=O)C3C2C3)=O)cc(F)c(F)cc1F C#CC1CCCCN1C(c1cnn(C2CCOCC2)c1)C(=O)NCCCSC C1(N(C)C(c2c[nH]c(-c3ccccc3)c2)=O)CN(C(C2CNC(=O)N2)=O)CC1O c1(NC(C2(O)CCN(C(c3c(C)noc3)=O)C2)=O)ccc([N+](=O)[O-])nc1 c1(C(=O)NCCN(C2CCCCC2)C(c2nc(C)sc2)=O)cccc2oncc12 c1(CC(=O)NC(C(C)(C)NC(C=CCN(C)CC)=O)C)cn(C)nc1C C12COCCC1(c1cccnc1)NC(c1ccc(Br)s1)C1CC21.C1(C)CCC1 C12(C(=O)NCC(CNC(c3ccnc(C)n3)=O)F)CCCN1S(=O)(=O)CC2 c1(NC(C2CCC(NC(CNS(CCOC)(=O)=O)=O)C2)=O)cc(C)cnc1O C(=O)(CCC(C)(C)C(=O)NC1(CNC(=O)CC2(O)CCC2)CC1)OC CCCCC(O)CCC(=O)N1CCC(C(C)(C)NC(c2cnc(C)c(C)c2)=O)C1 CC(C)CC(C)C(=O)NCCN(CCOCCO)C(C1CC1C(F)F)=O CC(C)(CC(F)F)C(=O)N1CC=CC(C(=O)NCC2(C3CC3)CC2)C1 c1(C(N2CCC(NC(C(C)N(C)C)=O)CC2C2CC2)=O)nc2ccccc2[nH]1 C1(NC(C2(C#N)C(C)(C)C2)=O)C2CC3C1C3C2C(=O)NC(CC1CC1)C1CC1 c1(NC(c2c(CC)n[nH]c2)c2nnnn2CC(F)F)cccc(S(C)=O)c1 S(=O)(=O)(c1ccc(Br)cc1)N(C(C(c1ccc(CC)s1)=O)=O)C1CCCC1 c1(C(=O)NCC2CCN(CC(=O)NC3CCC3)CC2)ccc(OC(F)F)cc1F c1(C(N2C(CNC(c3c(C)cc(F)s3)=O)C=CC2)=O)ccc(OC(F)F)c(Cl)c1 c1(C(=O)NC(CC(C)NC(c2c(C)cc(C)[nH]2)=O)C)ccc(S(N)(=O)=O)n1C C(CCSC)(C(=O)N1CC(C(N)=O)(CNC(=O)Cc2cc[nH]c2)C1)OC N1(C(CC(CCC)O)=O)C(CNC(c2ccc(N)c(O)c2)=O)CC2CCCC12 C1(CC(=O)NC2(CNC(C(C3CCCC3)OCC)=O)CC2)CCCC2(CCC2)O1 c1(C(=O)NC(CNC(C(C)C2CC2)=O)C2CCC2)ccc(C#N)c(O)c1 C1(C(N2CC(C)(N(C)C)C2)=O)C2CC(O)C(C2)N1C(=O)C#CC1CCCC1 N1(C(c2cn(CC)nc2C)=O)CC(C(N2CC(OC)C2)=O)C(C)(C)C1 c1(CNC(CC2(C#C)CC2)=O)ccc(CNC(C2(C)CCCCCC2)=O)c(F)c1 N1(C(C(CO)N(C)C)=O)CCCC(CNC(C2OCC2(C)C)=O)C1 NC1(CNC(=O)C(N2CCCC2C2CCNC2)=O)CCCCC1 n1(CCOC)cc(CN(O)C(=O)c2cccn2C2CC2)nn1 N1(C(Cc2ncc(C)s2)=O)CCCOC(CNC(=O)CCC(C)(C)F)C1 c1(OC)ncc(C(=O)NCC=CC(=O)NC2CC(CCO)C2)s1 c1(C(=O)NCC(C)(CO)NC(c2cccc(COC)c2)=O)ccc2nonc2c1 C1(CC)C(NC(c2ccnnc2)=O)CCCN1C(=O)CCc1cn[nH]c1 N1(C(CNC(C2C(NC(=O)CNC3CCC3)C2)=O)=O)CCN2C(=O)OCC2C1 C=CC(CC)C(=O)N1CCC(O)(CCNC(c2cc(F)n(C)n2)=O)C1 Cc1nn(C)c(C(=O)NCCC(O)CNC(C2CN(c3ccccc3)C2)=O)c1Cl C1(NC(C=CC(C)C)=O)CCCCC1NC(=O)C(C1CCCCC1)c1cccs1 C1(C(=O)NCCC(C(C)C)NC(=O)CC2CC(O)C2(C)C)CCn2ccnc2C1 N1(C(C(C(C)(C)C)OC)=O)C2CCC(C(=O)Nc3cc(C)cc(C)c3C)C1CC2 C(C)(CCC(=O)N1CC(OCCOC(C2CCCC2)=O)C1)SC CS(=O)(=O)c1ccccc1NC(C1CC12CCN(Cc1cccc(Br)c1Cl)C2)=O C1(CS(=O)(=O)NCc2ccc(C(F)(F)F)nc2)OCCOC12CCC2 C(=O)(CC1=CCCCC1)NCC1(C(=O)NCC=C)CCCO1 Cn1cc2cc(CC(=O)NCC3CC(CNC(=O)CC4CCC4)C3)ccc2n1 CC1CN(C(c2ccc(CC(F)(F)F)nc2)=O)CC1NC(c1cn(C)nc1O)=O c1(C(=O)NCC2(COC)CC2)cc(CNC(=O)C(F)(F)O)on1.C1(C)CCC1 c1(OC)cccc(C=CC(=O)NCC(C(C)(C)C)NC(c2ccc(OC)s2)=O)c1 C12(C(=O)NCC=CCC(C)C)CCCC1CN(C(C1C3CN(C)CC13)=O)C2 N1(C(C(CCC)C)=O)CC2(C1)CN(C(=O)C(C)(C)Cc1cnn[nH]1)CC2CO c1(CNC(c2nc(CNC(C(OC)OC)=O)oc2)=O)ccc(C(F)F)cc1 OCC1CCOc2ccc(CN3CC(=O)NCC3CO)cc21 c12nc(cc(C)n1)N2C.c1(CC)ccc(CN(C2CS(=O)(=O)C2)C)o1 CC1(CCNC(C2(CF)CC(=O)C2)=O)CCN(C(C2CC3CC3C2)=O)C1 Cc1cnn(CC(=O)N(CC(=O)NOCC(C)(C)C)C)c1 C1(C(=O)NC2(CC)CC2)CN(C(c2cnn(C)c2)=O)CCC1(F)F N#CC1CCC(CC(N2CC(NC(c3ccc(C(F)F)o3)=O)C(O)C2)=O)CC1 CC(C)(CF)C(=O)NCC1(C)CCCN1C(c1cccc(NS(N)(=O)=O)n1)=O c1(CNC(CNC(C(CC)C)=O)=O)cncc(C(=O)N(C(C)CC)C)c1 C(C(C)(C)S(C)(=O)=O)c1nnnn1C.N1(CCCC)CC(N)CC1=O N1(c2snc(CCC)n2)CC(NC(c2scnc2CC)=O)CC1C Cc1cc(C)cc(C=CC(=O)NC2COCCC2NC(=O)C(C(C)C)C(C)C)c1 C1(C(=O)NC2(C)CC(NC(c3cc(OC)c(C)nc3)=O)C2)CC2COCCN2C1 N1(C(c2ccc(S(CC)=O)cc2)=O)CCN(C(=O)C(C)C)CC(C)(F)C1 c1(C(CC(=O)NCCc2ccc(O)nc2)O)ccc(Cl)cc1 c1(C(=O)NCC2(N(C(C(C)N(CC(F)(F)F)C)=O)C)CC2)coc(C2CC2)n1 c1(C(N(CCC)CCNC(=O)C2=CCOCC2)=O)ccc2c(c1)CC1(CC1)CC2 C1(NC(c2nc(OC)c(C)s2)=O)COCCN(C(=O)Cc2ccc(Cl)cc2C)C1 c1(OC(=O)NCC2CC2c2cn[nH]c2)ccccc1Oc1ccccc1.C1(N)CC1 C1(CNC(C2CC23CCOC3)=O)CCCN(C(=O)C=Cc2ccccn2)C1 c1(C(=O)NCCC(=O)NC2CN(S(=O)(=O)Cc3ccccn3)C2)ccccc1 C1(C(=O)NCC2CCCC(NC(=O)CC3CCC3)C2)CCc2ccccc2CC1 Cc1c(C(N2CCC(C(C(C)C)NC(=O)CCC(C)C)CC2)=O)c(Cl)nn1C N1(C(CCc2nnc(CC)o2)=O)CC2(CCCC2NCc2csc(C)c2)C1 Cc1ccc2c(c1)CC(C(=O)NCC1CCCCN1C(=O)Cc1nnc(C)s1)O2 N#Cc1ccccc1OCC(=O)NCCC1CCCCN1C(C1CCC(=O)N1)=O c1(-c2onc(-c3nccc(C)c3)n2)ccc2cncn2c1 C(CNC(C1CCC1)=O)(C(C)C(C)C)NC(c1c(C)n(-c2ccccc2)nc1)=O c1(CC(=O)N(CCOCCN(C(C(=O)NC)=O)C)C)cccc([N+](=O)[O-])c1C CN1C(=O)CCCC1C(=O)NCC1CCC(NC(=O)Cc2cc(Cl)n(C)n2)CC1 C1(NC(C(CC)C)=O)CCN(C)C12CCCN(c1ncnc3cc(Br)ccc13)C2 Cc1ccc(CN2CCC2Cn2cc(-c3ccc(C(=O)O)nc3)nn2)c(C)c1 C(C)(C)(CC(F)C(=O)NCc1cncc(Cl)c1)NC(CC(CC)C)=O Cc1cnnc(O)c1C(=O)NC1CN(C(=O)CCOCC(C)(C)C)CC1C c1(OC)ccc(C(N2CC(N(C(=O)C(c3ccccc3Cl)O)C)C2)=O)cc1OC N(C1CCOc2cccnc21)(CC#C)C(c1ccc(OC)c2oc(C)nc12)=O N1(C(CCCNC(=O)Cc2cnco2)=O)CC(C(=O)NCC#C)CCC1C c1(C(N2C(COC)(CNC(C3CC3C#N)=O)CCC2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 Cc1cncc(C(N2CCN(C(=O)CNC(C3CCCC3(C)C)=O)CC2)=O)c1 [N-]=[N+]=NC1CCCC2(C(=O)NC3CCC3NC(c3ccc4c(c3)NCC4)=O)CC12 C1(=O)C(CCC(N)=O)N1C(C)C.CC(C)C(=O)N(CC(=O)N(CCCN)C)C c1(C(=O)NC2(CNC(C(COC)C)=O)CCCC2)cnc(N(C)C)nc1 N1(C(c2c(Cl)cc(C)s2)=O)CCCN(C(C2NC(=O)CC2C)=O)CC1 Cc1nnc2n1CCCC2C(=O)NCC(C1CC1)NC(c1cnnn1C)=O c1(C(N2C3CC(CNC(C(C)C#N)=O)C2CC3)=O)ccc(F)c2c1CCC2 C1(C(=O)NC(C)(CNC(=O)CC2CCOC2)CO)(COC)CCOCC1 C(=O)(C1CNC(=O)c2ccnn21)N1CC(C)(NC(C(CC)F)=O)C1 C1CCCCC(=O)N1.C1(CN(c2ccnc(C(N)=O)n2)C)(CO)CC=CCC1 C(=O)(C(C)C(C)S(C)(=O)=O)N1CCN(CC2CN(C(C(C)OCC)=O)C2)CC1 N1(C(Cn2ncc(C#C)c2)=O)CCN(C(c2ccc(OC)c(F)c2)=O)C(CO)C1 c1(OCC)nc(C(=O)NC2CC(C(C)NC(C3(C)CCCC3)=O)C2)co1 c1(C(N2CCC(C(CNC(COCC)=O)F)CC2)=O)c(F)ccc(C)c1F CS(=O)(=O)c1ccccc1C(N1CC(CO)(NC(c2cc(C3CC3)on2)=O)C1)=O c1(OCC(Cn2cc(C(CCC)NC(=O)C(C)OC)nn2)O)cccnc1 C=CCC(CC(F)F)ONC(=O)N(C1COC(SCC)C1)Cc1ccccc1 N1(C(Cc2c(C)nccc2)=O)CCN(C(=O)C(C)Oc2ccccc2)CCC1C C1(N(C(=O)C(C)(C)n2ccc(C)n2)CC)CCCN(C(c2cc(C#N)c[nH]2)=O)C1 C1(NC(c2ccc(SC)s2)=O)CCN(C(=O)C(N2CCC(C)CC2)=O)CC1C Cn1cncc(-c2cnccc2-c2nccn2CCN2CC3(C2)CC3(F)F)c1=O C1(CC)CN(C(=O)C=Cc2cnn(C)c2)CCN1C(=O)CN1CCCC1CO c1(CN(C(=O)CC(N2CC(C)(C)C2c2ccccc2)=O)C)cc(O)ncc1Br C1(NC(C(C)=CC2CC2)=O)CN(C(=O)Cc2ccc(C)s2)C2(CCOC2)C1 C1(C(=O)NCCOC(C)=O)CC(C(=O)NC(=O)CC2CC2C2CC2)CCO1 c1(C(=O)OCC)ccc(C(=O)NC(CNC(=O)Cn2cnnn2)C2CCC2)s1 CS(=O)CCC(O)C(=O)NC1CCCC1.C(CCOC(C)C)OCCO.C1(=O)CCN1 CC(N=c1[nH]c2ccc(Br)cc2o1)C(=O)NCC(C)CC1CCCC1 CC1CN(C(c2cscc2F)=O)CCC1N(C(=O)C=Cc1ccsc1)C C1(OC)(CNC(C2CC(NC(C3C4CCCCC34)=O)C2)=O)CCCCC1 c1(CCC)cc(C(=O)OC)n[nH]1.C1CCCCN2CCC(C2)C(=O)N1C C1(C)(C(=O)NC(c2n(C)nnn2)Cc2ccc(C#N)cc2)CCN(C2CC2)CC1 O=C(C1=COCCC1)NCC12CC(C1)C(NC(=O)CC1C=CCCC1)CO2 C1(NC(=O)CNC(C2(C(=O)NC3CC3)CC2)=O)CCCCC1CC(=O)O C(=O)(CCCC(C)(C)C#N)NC(C)CCNC(=O)Cc1ccc(C(F)(F)F)nc1 N#Cc1ccc(Br)cc1CN1CCC2(CC1)CC2C(N1CC2CC2C1)=O N1(C(CC(C)N(C)C)=O)CC(O)(C2(CNC(C3(N(C)C)CC(O)C3)=O)CC2)C1 CC(C)CCCCCC(=O)NC(CC(=O)N1CC=C(CO)CC1)C(F)F c1(OC)nc(N2CC3CC2CN3C(c2c(F)cccc2Cl)=O)ncc1Br C1(C(=O)NC(CN(C(c2cccc(Cl)c2)=O)CC)C)CCCC2(CC2)C1 C1(CCOC)(NC(=O)Cc2cncnc2)CCN(C(=O)C(C)c2ccsc2)CC1 C1(CNC(c2cn(C)nn2)=O)CN(C(C2COCCC2(F)F)=O)CCC1(C)C C(=O)(N=c1[nH][nH]cc1-c1cccc(SC(C)(C)C)c1)NCc1ncc(C)n1C C(=O)(C1=CSCCO1)NCc1scc(CNC(C(C)OCCCC)=O)n1 C1(COC)CC(Cn2cc(C3CC3OC)nn2)N(C(=O)CN2CCCOC2=O)C1 C1(NCC(C(C)(c2nnnn2CCO)OC)C)CCCC2CN(CC3CC3)CC12 C1(CC)C(NC(c2snnc2C)=O)CCN1C(=O)C(O)CCSC n1(CCCCCO)nc(CCCO)nc1-c1cc(C2CCOC2)[nH]n1 c1(C(C)(C)C(=O)N2CC(C(C3CC3)N(C3CCCC3F)CCO)C2)ccc(O)cc1 C1(C2CCCN(C(=O)C(c3ccc(F)cc3)(F)F)C2)(NC(C=CCOC)=O)CC1 O=C(C1=COCCC1)NC1(CCCCn2ccnc2)CC1 c1(OC)cc(C(=O)NC2CCCN(C(=O)C#CC(C)(C)O)CC2)cc(OC)n1 CC(C)C(F)(F)CC(=O)NCC1C=CCN1C(=O)CCc1ccc(Cl)s1 C(=O)(C(O)C(F)(F)F)N1CCC(C)C1C(N1CCC(C#N)C1)=O CC(C(=O)N(C)CCNC(=O)CC1CCCO1)C(C)(C)c1ccccc1 C(=O)(C1=CCCCC1C)NC1CC(C)(NC(c2c(CC)con2)=O)C1 N1(C(c2ccc(C#C)cn2)=O)CC2(CCN(C(C3CCCN3C(=O)OC)=O)C2)C1 c1(C(=O)NC2C(C)N(C(=O)Cc3cnn(C)n3)CCC2)cc2ccccc2o1 c1(C(=O)NCC=CCNC(C(n2cc(Cl)cn2)C)=O)ccc(C(F)(F)F)s1 N1(C(C2CC(C#C)(O)C2)=O)CCN(C(=O)Cc2ccsc2C)C(CC(F)F)C1 N1(C(C2(CC)CCCO2)=O)CC2C(NC(=O)CCc3cc[nH]n3)CS(=O)(=O)C2C1 C=CC(CC)CC(=O)N(CCNC(c1cc(C2(O)COC2)on1)=O)CC C(C(=O)N1CCC(C(C)(C)NC(=O)C(C)C)CC1)(C(C)C)NC(C)=O c1(CNC(C2CCCN2C(c2cccs2)=O)=O)ccnc(Br)c1 C1(NC(C)=O)CCC(NCC(=O)NC2N(C(COCC(=O)NC)=O)CC2)CC1 CC(C)C(O)C(C)C(=O)NC1CC(CC(N2CCCC2C(=O)N(C)C)=O)C1 N1(CC(=O)Nn2cncn2)CCC2CCCN(C)C2C1 N1(C(C)(C)C)CC(CNC(c2c(Br)noc2C)c2nnnn2CCC2CC2)CC1=O Cn1c(C(=O)NCC2CC2CNC(c2coc(-c3cnn(C)c3)n2)=O)nnc1S N1(C(CC2CC(SC)C2)=O)CC2(CCCC2)C1C(N1CC(O)C(O)C1)=O c1(C(c2n(CCCC)nnn2)NCc2csnc2C)cc(F)cc2c1OCC2 C(=O)(CC(C)(C)C(F)F)NCC1CC(C)N(C(=O)C#CC2CC2)C1 Cc1cc(C(=O)NC(CO)C(N2CC=C(CN(C)C)CC2)=O)c(C)cn1 c1(OCC)cncc(NC(C2(NC(=O)CCc3cnn[nH]3)CC(F)(F)C2)=O)c1 C1(CNC(C(CC=C)C)=O)C2CCCC1N(C(c1cc3c(s1)CCCC3)=O)C2 C1(C(=O)NCC)CCCCCN1C(=O)C(O)C1CN(C2(C)CN(CC=O)C2)C1 C1(c2nnnn2CCCCC2CC2)(NCC2CC(F)C2)CCCCC1CCC#N N1(C(CC2C(C)CN(C(C3(O)CCSC3)=O)C2)=O)CCc2cccc(F)c21 CCCCCC(C)CC(=O)NCCCC(O)C(=O)N1CC(C)(C)C1 S(=O)(=O)(c1cccc(N2CCCC2)c1)NC.N12CCN(C)C(C1)C(=O)OC2=O N1(C(=O)CC2CC(NC(C3C4CCCC34)=O)C2)Cc2ccncc2C1 CCC(C)C(CC(=O)NCCCC1(C)CC1)NC(C1COCC(C)O1)=O C(CCC(=O)NC1CCC(CCC(=O)NCc2cscn2)C1)OC(C)C c1(C(=O)NC2CC(NC(C(C)NC(=O)NC)=O)C2)cc(F)cs1 C1(C(=O)NCC(COC)OC)CC(C)(C)CN1C(c1cccc(CO)n1)=O C1CCCC(=O)N(C)OCC(=O)O1.C(CCC(C(=O)OC)OC)OC c1(NC(C2N(C(c3ccccc3)=O)C3C(C2)C3)=O)ccc(Cl)c(Cl)c1 c1(CNC(N2CC(OC)CC2(C)CSC)=O)cc2c(cc1Cl)CCCC2 C1(CC#C)(C(=O)O)CCCN(CC(c2c(F)cccc2Cl)O)C1.OC(=N)O N1(C(CNC(C(C2CC2)OCC)=O)=O)CCN(C(c2cc(C)nn2C2CC2)=O)CC1 N1(c2cc(N3CC(C(=O)NC)N(C)CC3)nc(C)n2)CCc2sccc2C1 c1(C(=O)NC2C(CNC(CP(C)(C)=O)=O)C2)cc(F)c(Br)cc1F c1(OC)ccc(F)c(C(=O)NC2CN(C(=O)Cc3cc(C)ns3)C2)c1 CCC(C)CCC(=O)NCC(C1CCC1)OC.C1C(C)=CC(=O)N1C Cc1cc(Br)ccc1S(=O)(=O)N1CCC(NC(=O)CC2=CCCCC2)C(O)C1 C12(C(=O)NC3CCN(C(C)C)C3)CCCC1CCN2C(=O)C=Cc1cn(C)nn1 C1(N(C)C(c2ccc(C3CC3)cc2)=O)CC2CCC(C1)N2C(=O)CCCF N1(c2snc(CCOC)n2)C2CCCC1CN(C(c1ccn3nncc3c1)=O)C2 C1(CNC(c2nnn3c2CCC3)=O)CN(C(c2cnn[nH]2)=O)CCCO1 N1(C(C2(C)CCC2)=O)CC2CCN(C(=O)CCNS(C)(=O)=O)CC2C1 CC1=C(C)CN(C(c2ccnc(CNC(C3CCC(=O)N3C)=O)c2)=O)C1 N1(C(c2c(C)nc(CO)s2)=O)C2CC1CN(C(C1CCCC1C(C)C)=O)C2 N1(CCNC(=O)Nc2ccc(-n3ccnn3)cc2)C(=O)COCC1=O c1(C(N2CCC(CCNC(=O)CC3(COC)CC3)C2)=O)n[nH]c2c1CCC2 C1(C(N2CC3(CC(CNC(C(CC)(C)O)=O)C3)C2)=O)CC2(CCCC2)CO1 CC1CCN(C(c2sccc2C#N)=O)CC1NC(c1ccc(F)c(C(F)F)c1)=O C1(N(c2c(C)nn(C)c2C)C(C2COC2C(C)C)=O)CCC2(CC1)CNC2 C(C)(C)(CC(=O)NC(C1CCOCC1)(C)C)N(C)C(c1ccc(CO)cn1)=O Cc1cc(C(=O)NC2CC(Nc3nccc(CO)n3)C2(C)C)ccn1 c1(OCC)ccc(Cl)c(C(=O)NC2CC2CNC(=O)CN2CCOCC2=O)n1 C1(C(=O)NC)(C(=O)NC2CC(C(=O)NC(C)CCN(C)C)C2)CCC1 N1(C(c2c(C)c(C(F)(F)F)n[nH]2)=O)CCN(C(=O)C(O)CC(N)=O)CC2(CC2)C1 C1(C(=O)OC)CCC(C(=O)O)N(C(=O)Cc2cnoc2)C1 N12CCN(CC1C)C(=O)c1coc(n1)CCC2=O.c1(C(C)=O)cc(C2CC2)on1 c1(COC)c(C(=O)NC(C2CCCCN2C(=O)C(C)(F)F)C)sc2ccccc12 CN1CCOCC1(F)C(=O)NC(Cc1ccccc1)C(N)=O c1(C(N2CCC(C(C)NC(C3(OC)CC3)=O)C2)=O)scc(C)c1OC c1(CC(=O)N(C2CCN(C(=O)C(C)OCC)C2)CCC)nc(C)c(C)o1 C1(C(=O)NC(c2c(C)cccn2)C)CN(C(=O)COC(C)C)C(C)(C)C1 C(=O)(C1=CC2CCCC12)NC(CC)(CNC(=O)COc1cccc(Cl)c1C)CC C12CN(N3CCN(S(=O)(=O)N(C4CC4)C1)CC3)C2.[N-]=[N+]=NC[Si](C)(C)C C1(=CC(=O)NCC2CN(C(CC(CCC)O)=O)CC2C)C2CC3CC(C2)CC1C3 C(=O)(C1CCC(=O)c2ccccc21)NCCN(CCC)C(c1ccc(F)cc1)=O c1(C(=O)NCCC(=O)NCCN(C)C(C2CCCC(=O)C2)=O)ccc(O)cc1 N1(C(COC)=O)CC(Cn2cc(C(C)CCC(=O)OC)nn2)CCC1(C)C N1(C(C2CC(=C)C2)=O)CCCCC(CNC(c2cccn(C)c2=O)=O)CC1 c1(C(=O)NC(C#C)C(C)C)ccc(C2COCCN2C(c2csc(CO)n2)=O)n1C C1(CNC(c2ccc(Cl)cc2O)=O)COCCN(C(c2ccc(Cl)cc2Cl)=O)C1 Cc1ccc(CNC(C2CC23CCN(c2nccc4nc[nH]c24)CC3)=O)cc1C#N c1(C(N2C(CNC(C(C)C)=O)C=CC2)=O)ccsc1C#N C1(C(=O)NCC(C)N(C)C(C2C3CCC23)=O)CCCN(C(N)=O)C1 N1(C(C(C)(CO)NC(C)=O)=O)CCC2(CC1)CC2NC(c1cc(C2CC2)no1)=O C1(NC(c2[nH]cc(C)c2)=O)CC(C(N2CCC(CC(C)C)CC2)=O)C1(C)C N1(C(C=C(CCC)C)=O)CCOC2(C1)CN(C(=O)Cn1ccc(=O)n(C)c1=O)C2 Cn1nnc2c1CC(C(=O)Nc1ccc(C(N)=O)nc1Oc1ccccc1)CC2 C1=C(C)NOCC=CCN(C(=O)C(C)CC)CCN(CCCN(C)C)C(=O)C(C)C1 CCN(Cc1cc(F)c(F)c(F)c1)N1CC(c2cc(C)c(C)o2)C1 C12(C(N(C3CN(C(=O)C=Cc4cccc(F)c4Cl)C3)C)=O)CC(C)(C1)OC21CCC1 c1(C(=O)NC(C=CC(=O)N(C)CCOCCO)C)ccncc1Cl c1(C(N2C(CNC(C(COC)COC)=O)CCC2)=O)cccc2ncnn12 C12(NC(=O)CSc3ccccc3)CCCC1CN(C(=O)Cn1nnc(=O)[nH]1)C2 N1(C(C)=O)CC(NC(=O)CC2CCC2NC(c2ncncc2Cl)=O)C(C)(C)C1 C(CC(C)(C)CC(=O)NCC1CN(C(=O)C(O)C2CCC2)CCC1(C)C)OC CCC(F)(CNC(=O)CNC(C1(C)CC(=O)C1)=O)CC C1(C2N(C(C3C(C)C3)C3CCC3)CCC2)CCN(C(=O)CCC(F)F)CC1 c1(OC)c(OC)cccc1NC(=O)C(N1CCCC(CNC(=O)C(C)(C)C)C1)C c1(OC)ccc2[nH]nc(CN3CC(NC(=O)CCCN(C)C)C(F)C3)c2c1 C(C(C)S(C)(=O)=O)(c1cccnc1)NC(=O)NC(=O)NC(CCC)CC Cc1cc2ncc(C(N3CC4(CC(NC(=O)C(F)(F)CF)C4)C3)=O)cn2n1 Cc1nc(O)ccc1C(=O)NCC(O)CN(C(=O)Cn1ncnn1)C C(C(C(=O)N(C)CC1CCOC1C)NC(C1CC1CC(C)(C)C)=O)OCC Cc1nn(C)c(C)c1CC(N1CC2CC(C(N3CCC(C(C)(C)C)C3)=O)(C2)C1)=O C(=O)(C(O)CC(F)(F)F)NC1(C(=O)NCC2(C#N)CCCC2)CC(CO)C1 c1(OC)ccncc1C(N1CCC(N(CCO)C(c2sc(C)nc2C)=O)C1)=O n1(CC)nc(C(=O)NCCC2CC(NC(=O)C3=COCCO3)C2)ccc1=O N1(C(c2c(C)cc(C)o2)=O)CC2CCC(C1)C2NC(C1CC2(CC(C)=NO2)C1)=O c1(C(N(CC(CC)N(C(C2CCCCN2CCC)=O)CC)C)=O)ccnnc1O c1(OC)ccc(C(=O)NNC(=O)N2CCCC2C(=O)N2CC(O)CO2)c(Br)c1 N1(C(C2N(C(CC(C=C)C)=O)CCSC2)=O)CCC2C(C(N)=O)C2C1 CC1(C)CN(C(c2c[nH]nc2F)=O)CC(C)(C)C1NC(C1CCCCC1F)=O C1(CC)CC(C)CN(C(C2CN(C(=O)COCC3CCC3)CCO2)=O)C1 c1(C(C2CN(S(C)(=O)=O)C2)N(C2CN(c3nnnn3C)C2)C)cc(N)cnc1Cl c1(SC)ncc(F)c(=NC(=O)Nc2ccc(CC(=O)NC(C)C)cc2CCC)[nH]1 Cc1cc(Br)ccc1C(c1nnnn1C1(C)CC1)NCCCOC(=N)O c1(CN2CCCC(C(=O)OC)C(OC)C2)c(F)cc([N+](=O)[O-])cc1F c1(NC(c2c(-c3[nH]cc(C#N)c3)ncs2)=O)cncc(Cl)c1Cl C1(C(=O)NCc2ccccc2C)(NC(C(CC)c2cccnc2)=O)CCOCC1 Nc1cc(C(=O)NCCCCNC(c2cnccc2Cl)=O)ccc1-n1cncn1 c1(C(=O)NC2CN(C(C(CC)OC3CCCCC3)=O)C2)ccc([N+](=O)[O-])o1 N1(C(CCCC#C)=O)CCN(C(=O)Cn2cnnn2)CC1c1ccccc1OC C1(CNC(C2CCCSC2)=O)CCC(C(=O)NCCCc2ncc[nH]2)CC1 C12CC3CCC(C1)N3C(=O)N(C)C2.c1(NC(=O)CSC(=N)N)ccncc1 c1(CC(=O)N(C(C)CCNC(C2CCC(=O)N2C)=O)C)cc(Cl)cc(Br)c1 CC1CN(C(C2CC2(C)C)=O)CC1CNC(c1cccc(C(N)=O)n1)=O C(C(F)(F)CO)N(C(CNC(=O)CCC1CCC1)=O)Cc1ccsc1 CC1CN(C(c2ccn(C)c2)=O)CCC1C(=O)Nc1cnn(C)c1C(N)=O C1(C(=O)NC(CCNC(c2c(CC)ncnc2CC)=O)C)CCCCC(C)(C)C1 c1(CC)[nH]nc(C(=O)NCC2CC(C)(C)CN2C(C23COCC2C3)=O)c1[N+](=O)[O-] c1(C(=O)NC(CNC(C(C(C)C)SC)=O)(C)CO)ccc2sccc2c1 c1(C(N(C(C)CNC(C2CCN(C)C2)=O)CC)=O)cc(C)sn1 c1(SC)ccc(OCC(=O)NC2(CNC(=O)CC3CC3(Cl)Cl)CC2)cc1 CN1CC2CCC1CN(C(=O)CC1CCCN1C(c1ccc3occc3c1)=O)C2 Cc1nc(C(=O)N(C)CCc2cccc(Br)c2)nn1-c1ccccc1 N1(C(CCc2n(C)ccn2)=O)CC2C(NC(C3CCCCS3)=O)C2C1 C1(NC(CN(C(C(CC)CC)=O)C(C)C)=O)CCC(=O)N(C)C1=O C(=O)(C1=NOC2(CCCN(C3CCC3)C2)C1)N1CCN(C(CCC)=O)CC1 c1(C(N(CC(C)O)CCNC(CC(CC)(F)F)=O)=O)ncnc2ccsc12 N1(C(Cc2nnc(C)s2)=O)CCC(C(F)CNC(c2coc(Br)c2)=O)CC1 c1(OC)cccc(C(N2CC=CC2C(=O)NCc2cncc(Br)c2)=O)c1Cl N#CC1(C(=O)NC2CN(C(c3cc(O)cc(O)n3)=O)CC2O)CC12CCOCC2 C1(C(=O)NC2(C)CC(NC(=O)C(c3ccc(F)cc3F)=O)C2)Cc2nccn2C1 C1(CNC(C2(CNCC(c3cccs3)C)CCC2)=O)C2CC3C(C2)C13 C1(C(=O)NCC2N(C(Cn3nnc(C(C)(C)C)n3)=O)CC=C2)CCOC(CF)C1 C1(NC(c2n(CCC)ncc2)=O)C=CCN(C(=O)Cc2ccco2)C1 C#Cc1cccc(C(=O)NC2CCC(NC(c3cc(C)co3)=O)C2)c1F CCC(C)C(C(=O)NCC1CCN(C(=O)Cc2nncs2)CC1)c1ccccc1 N1(c2snc(C)c2C#N)CCOC2(CCN(C(=O)C3=CCCO3)C2)C1 c1(C(C(CCC#C)=O)=O)[nH]c2ccccc2c1CC(=O)NC1CC(NCC)C1 C1(CCC(N2CC(CN(C(C3C(=C)C3)=O)C)C2)=O)CCC(=O)NC1 c1(C(C(=O)NC2(C)CN(C(c3c(C)nn[nH]3)=O)C2)C)ccc(Br)cc1F C1(C(=O)NCC(C)N(C(=O)C(O)Cc2ccccn2)C)CCC(O)CN1C c1(N2CCN(C(=O)NCC3(C#N)CC4CCC3C4)CC2)cc(F)cc2cc[nH]c12 N1(C(COC(CC)C)=O)CC2CC(NC(C3CC(C)(CC)C3)=O)CC2C1 N1(C(CNC(C)=O)=O)CC(C(=O)NCc2cnn(-c3ccccc3)n2)CC1(C)C C1(OCC)CCCC1NC(C1CCCC1NC(=O)CCc1ccccc1)=O C(=O)(CC(C)C(F)(F)F)N1C(CN(C(C2CC(SC)C2)=O)CC)CCCC1 c1(CC(=O)N(CCCOCCN(C(CCC#C)=O)C)C)cnc(Cl)cc1C N1(C(c2cc(C)c(C)s2)=O)CC(NC(=O)C(O)(C2CCC2)C2CCC2)CC1(C)C C12(C(=O)NC3CN(C(=O)CCSc4ccccn4)CC3O)CC1CCC2(F)F C(CCCC(=O)N1CCC(CCC(=O)NC(C)C(C)SC)CC1)OC c1(CCC)n[nH]c(=NC(=O)N(CC(c2ccc(F)cc2)O)C)s1 N1(C(c2c(COC)ccs2)=O)CC2(COC(CNC(n3nc(C)oc3=O)=O)C2)C1 CS(=O)(=O)c1coc(C(=O)NC2C3CN(S(=O)(=O)c4cccnc4)CC23)c1 c1(OC)cc(OC)cc(CN(C)C(=O)NCC2CCOC(=O)N2)c1 C(=O)(C(CC(N)=O)NC(=O)CCC(C)=O)NCC1CCN(CCCC)C1 c1(C(N2CCC(NC(C(CC)(C)OC)=O)C2)=O)c(C)cc(C)nc1C N1(C(CC2C(=O)NC(=O)N2)=O)C2CCC1CN(C(=O)CCC1CC1(F)F)C2 N1(C(C2(C=C)CC2)=O)CCCC(CCNC(=O)C(Cc2ccccc2)OC)C1 N1(CC(=O)NC2(CC)CC2)CCN(C(=O)Cc2cnn(C)c2)CC1 c1(OC)cc(CN2CCCC2C(=O)NC2CCCN(C(=O)CC#N)C2)c(Br)cc1O c1(CNCCN(C(=O)NC(CC)COC)CCn2cnnc2)ccccc1 C12(NC(C=C(COC)C)=O)CCC(CN(C(c3ccc(N)c(N)n3)=O)C1)C2 N1(C(CNC(c2c(C)ccs2)=O)=O)CCCCC1C1CCCN1c1ncncc1I N1(C(C2OCC(C)C2)=O)CC(N=c2nc(C3CCCC3)[nH]s2)C2(CCOCC2)C1 N1(C(COCCSC)=O)CCN(C(=O)C(C)C(F)(F)F)CC1CO C(CC1C(=O)N1)OC.C1(CC(C)C)(C(N2CCC2CN(C)C)=O)CCC1 C1(C(=O)OC)CC12CN(C(C1CC(O)CN1C(C1CC3CC3C1)=O)=O)C2 c1(NC(=O)Nc2cc(F)ccc2O)c(C2CC2)cccc1F N1(C(C=CC(CC)=CC)=O)CCCC2(NC(=O)CNC(=O)C(F)(F)F)CCCC12 Cc1cnsc1C(N1CC(C(N)=O)(CNC(=O)CC2CCC(C(F)(F)F)O2)C1)=O CCC(CC(=O)N(c1nnnn1CCc1ccccn1)C)CC(F)(F)F N(C(=NCC1CN(S(=O)(=O)CC)C1)NC(=O)CC=CCc1ccccc1)C(C=C)C N1(Cc2n(C)cnn2)CCCC2(CCN(C(C3CCCC4C3C4(F)F)=O)C2)C1 c1(C(N2CCCC(C(=O)NCc3cc(CC)on3)C2)=O)cccc(C)c1O Cc1nc(C)c(C(N2CC3CCC(C2)N3c2nnc(O)s2)=O)nc1C N1(C(c2cc3c(cc2Cl)OCCO3)=O)CC(C2CCC(F)(F)CC2)C1 C1(CNC(=O)CN2CC3CCC2C3)CC2(CCOCC2)CN1C(C1CCCC1)=O Cc1nc(=N)[nH]cc1C(=O)NC1CCCC(NC(=O)COc2ccon2)CC1 C=C=C(C)CC(=O)N(CC(C)N(C(=O)CC1CCOC1)C)C N1(C(c2c(C)cccc2)=O)CCN(C(=O)COC2CCC2)CC1c1ccccn1 c1(C(N2CCC(C)(C(=O)NCCC3CCCCO3)CC2)=O)c[nH]c2nccc-2c1 N1(C(CN(CCC)C)=O)CCCCC1CCC(C)(C)NC(=O)CC1CC2CC2C1 CC1=CCS(=O)(=NC(=O)CCCC(=O)N(C2CC2)Cc2sccc2Cl)CC1 CC1(C#CC(=O)N2CCC(C(=O)NCC3(C#N)CCC3)(CF)C2)CCCO1 C(C(C(=O)N(CCCNC(=O)CSc1cccnc1)C)c1ccccc1)SC c1(CC(N2CCC(C(C)NC(COCC#C)=O)C2)=O)ccccc1C c1(N(C)C)cccc(C(CNC(=O)CC(C)F)NC(=O)CCN2CCC(F)C2)c1 c1(C(N(C)CC2(NC(C3C(CC)C3)=O)CC2)=O)cc(Cl)cc2ccccc12 C(=O)(CS(=O)(=O)C1CC1)NCc1cn(CC(C)NC(C(C(C)C)C#N)=O)nn1 C1(C2C(C(C3CC3)Nc3n(C)ncc3)C2)C(C)(C)C1(F)F [N-]=[N+]=NC1CCC(C(N2CC3CC2C3C(N2C3CCCC2CC3)=O)=O)CC1 CC1CCC(NC(=O)C(C)(O)Cn2cc([N+](=O)[O-])cn2)CN1C(C1C=CCC1)=O C1(C(N(CCCC(=O)NC2C(OCC)COC2)C)=O)CC2C(C1)C2(F)F CC(C)C(C(=O)NCCC1CC(NC(c2ccc(C(F)F)o2)=O)C1)n1ccnc1 C1(C(=O)NCC(CCC=C)O)CCCC(NC(c2cc(O)cs2)=O)CC1 C(C(C)(CC)C(C)O)NC(C1(C)CN(C(C2CCC(=C)CC2)=O)C1)=O Cc1cnnc(O)c1C(=O)NC1CN(C(=O)CC(C)c2cccnc2)C(C)(C)C1 c1(N2CC3C(NC(CCCc4ccc(C)s4)=O)C3C2)ccc([N+](=O)[O-])c(O)n1 C1(CC(N2CCN(C(c3c(CC)occ3)=O)C(C)C2)=O)CN2CCC1CC2 c1(CNC(N2CCC(OC)C2)=O)ccc2n[nH]c(C)c2c1 c1(C(N2CC(NC(C(C)OCCC=C)=O)C(C)C2)=O)cnc(C)[nH]c1=N CCC(C)C(C(=O)N(C)CC1CCN(Cc2nc(C)c(CC(=O)NC)s2)C1)OC C1(CC#C)(CNC(C2CCCN2C(=O)COCP(C)(C)=O)=O)CCCCC1 C1(F)(CNC(c2c(C)csc2Cl)=O)COCCN(C(c2ccc(=O)oc2)=O)C1 Cc1noc(C)c1C(C)C(=O)NCC(F)CNC(=O)CCCCc1ccccc1 N1(C(c2cnc(C)n2C)=O)CCCC(CC(=O)NCC2(C(C)(F)F)CC2)CC1 C(=O)(C1=CCCOC1)N1CCC(C(C)(C)CNC(C2(C#N)CC2(C)C)=O)CC1 Nc1ncnc2c1ncn2C1CC1.C1(N2CC2=O)C(O)CC1O n1(CC)c(N2CCCC2CC2CCCO2)nnc1C1CCC(=O)N1 c1(C(N(CCN(C(c2onc(C)n2)=O)C)C)=O)cnn(-c2ccccn2)c1C N1(C(c2cc(=N)[nH]cc2)=O)CCCC12CCN(C(C13CCCCN1CCC3)=O)C2 c1(-c2ccc(OC(C)=O)cc2)c(S(=O)(=O)NC2CCOC2CO)noc1C c1(OC)cc(C(=O)NC2CCCN(c3nc(C#N)c(Cl)s3)C2)cc(Br)c1 c1(C(N2CC(CNC(C3(COC)C=CCC3)=O)C2)=O)ccc2scnc2c1 N1(C(Cc2c(C)n(C)nc2)=O)CC2CCC(C1)N2C(c1nc2c(s1)COCC2)=O c1(C(CC(=O)O)NC(=O)Cn2cc(-c3ccsc3C(=O)O)nn2)ccc([N+](=O)[O-])cc1 Cc1noc(C)c1C(C)(C)C(=O)NCC1(CNC(c2cc(Cl)ns2)=O)CC1 C(=O)(CC(O)C(C)C)NCCN(C(c1occc1Cc1ccccc1)=O)CC c1(CN(CCCNC(COCC=C)=O)C(=O)CNS(N)(=O)=O)cccc(OC)c1 C=CC(C)CC(=O)NCC1(NC(c2cnc(S)nc2)=O)CCOC1 C(=O)(C(CC)C(=O)N(CC(O)CN(C)C(c1cnc(SC)[nH]1)=O)C)OCC c1(SCC(=O)N(C2C3CN(C(C4C(C)C4)=O)CC32)C)ccc([N+](=O)[O-])cc1 C12(C(=O)NC3C4N(C(CS(=O)(=O)NC)=O)C(CC4)C3)CCCN1S(=O)(=O)CC2 CC1CC(NC(C2CC(=O)N2)=O)CCN1C(=O)CC1CCC1 c1(OC)ccc2[nH]cc(C(=O)NCC3(OC)CN(C(=O)CCC=C(C)C)C3)c2c1 C(=O)(C1CCCn2ccnc21)N1CC(N(C)C(C23CC(F)(C2)C3)=O)C(O)CC1 C1(C(=O)NCC2(CCOCC)CCCC2)(CO)CCCCC1.C(=O)(C=CSC)N n1(CCNC2(c3nnnn3C3COC3)C(CCC)CCC2)ncc(O)nc1=O CC(F)(F)CCCC(=O)N1CC2(CC(NC(=O)Cn3ccc(C(F)F)n3)CO2)C1 c1(OC)ccccc1C1CC1C(=O)NC1(CNC(=O)CS(C)(=O)=O)CCC1.C(=O)OC n1(CC(=O)NCCCCN(C(COCC)=O)C)c(C(=O)OCC)nnc1S C1(CNC(C(C)(O)c2ccccc2)=O)CCCCC1NC(=O)CN1CC=CC1 c1(CNC(CC(CCSC)O)=O)n[nH]c2c1CN(C(=O)C=CC(C)C)CC2 c1(CC)ccccc1OCC(N1CC(CNC(c2csnc2C)=O)CC1C)=O [N-]=[N+]=NC1CCC(C(=O)NCC(C2CCC2)NC(C2(CO)CC2)=O)CC1 N1(C(C2C(OCC)C2)=O)CCCC(CN(C)C(c2coc(C)c2)=O)C1 Cc1c(CNC(=O)C(C2CC2)N(C)C(C2CCO2)=O)nnn1C CC(C(=O)N1CC=CCC1)C(C)NC(C1CC(C)N=N1)=O C(=O)(C(C)C(O)C(C)CC)N1CC(OCCC(=O)N(CC)CC)C1 CCCC(C)(C)CC(=O)NC1CCN(C(c2cc3oc(Br)cc3[nH]2)=O)CC1F N1(CC)CCOC(C(=O)NC(c2cccnc2)CNC(=O)Cc2cc(C)cs2)C1 CC1CC(C(=O)NC2(CCF)CC2)CN(C(C2(O)CCCCCC2)=O)C1 N1(C(CC2CCN(C)C2)=O)C2CCC1CC(O)(CNC(=O)CS(C)(=O)=O)C2 N1(C(c2c(C)[nH]cc2)=O)CC(O)CC1C(=O)NC1(c2ccccc2)CC1 c1(C(=O)NC2CCC(NC(C3(CC)CCOCC3)=O)C2)ccc(Cl)c(F)c1 Cc1nc(Cl)ccc1CC(=O)N(C)CC1CCCCN1C(C1CCSC1)=O c1(CC(C(=O)NCC(C(C)C)NC(CCCOCC)=O)SC)ccc(OC)cc1 c1(CN2C(C(=O)NCc3cc(Br)ccc3F)CC2)sc2ccccc2c1Cl c1(CC(=O)N(C)CC2(O)CN(C(CSCCCC)=O)C2)ccnc(O)c1 c1(OC)cnc(Br)c(CNc2ncnc(N3CCCC(C)(CO)C3)c2C)c1 N1(C(c2ccc(OCC(C)C)nc2)=O)CC2(C)CC1C2C(=O)O CCCC(CNC(=O)Cc1cccnc1)C(=O)NC(C1CSC1)C C=CC1CN(C(C2C3CC2N(C(=O)Cc2cncn2C)C3)=O)CC1O N(C1c2ccccc2CC1C)C(CCC(C)S(C)(=O)=O)=O c1(C(N2CCC(NC(c3cncc4c3CCC4)=O)C2)=O)nccc2n[nH]cc12 N1(C(C2CCN(C(=O)NC)CC2)=O)CCN(C(c2coc(C)n2)=O)CC1C(C)C c1(C(=O)NC2CCCC2NC(C2CC3(CCC3)CO2)=O)cccc2c1CCC2 N1(C(c2n[nH]c(C)c2Br)=O)CC(NC(=O)CCc2ccnn2C)CC2(CC2)C1 N1(C(C(CC)CC)=O)CC(C)CN(C(=O)C(c2cccc(Cl)c2)O)CC1C C1(CNC(c2cc(C(C)(C)C)no2)=O)CCN(C(c2ccc(C#N)[nH]2)=O)C12CC2 N1(C(C=NOC)=O)CCCC2(CCCN2C(=O)CC(C)C(C)(C)C)C1 C12(NC(c3ccc4ncsc4c3)=O)CCCC1CN(C(=O)Cn1cnnc1)C2 N1(C(c2cc(C)[nH]n2)=O)CC2(CCCC2CC(=O)Nc2c(C)cccc2O)C1 c1(OC)cc(C(=O)NC2(CCNC(=O)C(C)(C)C(C)O)CCC2)cc(Cl)n1 c1(C(=O)NC2CN(C(C(C=C)O)=O)C(CO)C2)cc(S(N)(=O)=O)sc1Cl c1(CS(=O)(=O)NC2CCC2)ccc(OCc2cc(C(F)(F)F)ccn2)nn1 c1(C(=O)N(CCN(C(CCN(C(C)=O)C)=O)CC(C)O)C2CC2)c[nH]ccc1=O C=CCC(C)(C)C(=O)NCCCN(C(c1cc(C(C)C)ccc1F)=O)CC c1(CCOC)cc(C(=O)NCC2CCN(C(=O)CCC(N)=O)C(C)C2)ccc1F C(=O)(C1=CCN(C)C1)N(C(C(=O)NCCC)C)C Cn1cc(C(N2CC3CC(NC(C4CC=CCC4)=O)C2C3)=O)ccc1=O c1(C(=O)NCC2C(CNC(c3c(C)cc(C)s3)=O)C2)cc2c(s1)CCCCC2 c1(CC(=O)NCCC2CCN(C(=O)CN3CCOCC3)C2)ccc(O)c(O)c1 C1(C(=O)NCCc2scc(C)n2)CN(C(=O)C=Cc2cccc(C)c2)CC1(C)C N1(CC(=O)NCCCCCCC)CCCCC(NC(=O)CC(C)c2cnn(C)c2)C1 CCCC(C(=O)NCCN(C1CC1)Cc1cnn(CC)c1)OCC N1(C(=O)OC(C)(C)C)CCCNC(=O)CC1.CC1CCC(=O)N1C N1(C(c2c(C)cno2)=O)CCC(O)(CN(C(=O)C(C)Cc2cccnc2)C)C1 c1(CN2CCC(C(N3CCC(N(C)C)C(O)C3)=O)CC2)cccc2c1ccn2C N1(C(=O)NC2CCC(O)CC2)CCC12CCCN(C(c1c(C)cc(F)cc1)=O)C2 S(=O)(=O)(c1ccc2c(c1)C(C)(C)CC(=O)N2)N1CCC(SC)CC1 c1(C(=O)NC(CC)CN(C)C(C23CCCN(CC2)C3)=O)c(Cl)nc2ccccn12 c1(C(N2C(CN(C(=O)C(F)(F)C3=CCOCC3)C)CCC2)=O)ccc(S(N)(=O)=O)cn1 c1(C(=O)OC)ccc(-c2nc(CO)cs2)cc1O.c12cn(nn1)CC(=O)NC2 C(Cc1cn[nH]c1)(C(=O)N(CCO)OC)NC(c1ccc(CC)[nH]1)=O C12CCCCN1c1nccc(n1)OC2.C(COCCOCCO)OC c1(C(=O)NCC(CC)NC(=O)C(C)(C)C(=O)OC(C)(C)C)cc(F)cnc1OC c1(OC)cccc(CNCc2csc(CC3CC3)n2)c1Cl c1(COC)cc(C(=O)NC2C3CN(C(c4cnc(Br)s4)=O)CC23)n(C)c1 Cc1cc(NC(=O)C(O)C(C)(C)C)ccc1NC(=O)C(c1cscn1)N(C)C c1(C(=O)NC(C)CNC(c2ccon2)=O)cnc(C(=O)NC2CC2)c(Cl)c1 C1(CC(=O)NCCCC(C)NC(c2c(C)ocn2)=O)CC2CCC1C2 C(C(C)(C)C(=O)N1CC(CCO)(CNC(=O)CCNC(N)=O)C1)N(C)C CC1(C(=O)NC2C=CCCC2C(=O)NC2CNC(=O)C2(C)C)CCC(=O)NC1 n1(CCC)[nH]c(=NCCC(C)c2cccnc2)cc1C C1(C)(CNC(C=CC=CC)=O)CC(NC(C2CC(C)(C)C2)=O)CN1C(C)=O c1(NCC2(F)CCN(CCC)CC2)ncc(C#N)cc1F.C1C(=O)N1 C(c1cccc(F)c1)=CC(=O)NC1C(C)CN(C(=O)C=Cc2nccs2)C1 CC1CN(C(=O)C=CC(C)(C)NC(C2CC3(CC3)CO2)=O)CCS1=O C1(C(=O)NCC(CC)NC(=O)Cn2nc(C)oc2=O)CC(C)(C)OC(C)(C)C1 N1(C(CCNC(CC)CC)=O)CC(C)C(NC(=O)CNC(=O)C(C)(C)C)C(C)C1 c1(C(=O)NC(C(C)NC(COc2cccc(C)c2)=O)(C)C)c(C)nc(C)n1O C(CC(O)C(=O)N1CC(O)CC1C(=O)NCCc1ncon1)N(C)C C1(CNC(C=C(C)C(C)(C)C)=O)CCN(C(c2cc(CF)on2)=O)CCC1(F)F N1(C(c2[nH]cc(OC)c(=O)c2)=O)CCN(C(C2OC3CCC2C3)=O)CC(C)(F)C1 Cc1cc(Cl)c(Cl)cc1C(=O)N(C(C)CN(C)C(C1CCC(=O)N1)=O)C N1(C(C2(CC#C)CC2)=O)CCCC(N2CCN(C(c3coc(CC)n3)=O)CC2)C1 O=C(CCCCCn1cnnn1)NCC1CCN1C(C12CCC(CC1)OC2)=O c1(C(=O)NC2CC(CNC(c3nccs3)=O)C2)ccc2scnc2c1 Cc1ccc(F)c(C(=O)NCc2c[nH]ccc2=N)c1.C12(O)CCN(C1)C2 C12(C(N(C3C4CN(C(c5nccc(N)c5Cl)=O)CC34)C)=O)CCC(CC1)CO2 C1(CC(C)(C)C)CCCCN1C(=O)C(O)CC1CCCC1.C1(=O)CN1 C(C(=O)NNC(=O)c1ccc(OC)s1)C1CC(c2c(OC)nccc2)C1 c1(NC)cccc(C(=O)NC2CCN(C(C3(C(=O)N(C)C)CC3)=O)C2C)c1 C1(CCC)CN(C(=O)C(O)C2CCCC2)CC1NC(C1CCN(C)CC1)=O C(=O)(C(C)(O)CC)NC(CC)CNC(C1CC(F)C1)=O CON1CC(C(N2CC(N(C)C(C3(c4ccno4)CCOCC3)=O)C2)=O)CC1=O c1(C(=O)NC(CCNC(c2c(C)nco2)=O)(C)C)cc2n(n1)CC(F)C2 C1(C(=O)NCC2CCC(CNC(C(C(C)C)NC=O)=O)CC2)CCC(C)(C)OC1 N1(CCCNC(C(C)C2CC2)=O)CCN(C(=O)C=CC2CCOCC2)CC1 C1(NC(c2ccnc(C)c2)c2n(CCCSC)nnn2)CCCCC12CC2 Cn1c(C(=O)NC2NCC3CC23)cc(=O)n(C)c1=O C1(CC(=O)N(CCC)CCNC(c2ncc(C)o2)=O)CC(O)C12CCC2 c1(OC)ccc(C(N2CC(CF)(NC(=O)C(F)=CCCF)C2)=O)cc1C(N)=O c1(C(N(C2CC(NC(=O)CNC(=O)C3CC3)C2)C)=O)nn[nH]c1Cl C1(NC(C(C2CCOC2)NC(C2(C)ON=C(C)C2)=O)=O)CCN2CCC1C2 N1(C(C=C2CCN(C)CC2)=O)CCN(C(C2(C)CCCCC2)=O)CC1CO N1(C(C=CC)=O)CC2C3CCC(C2C1)N(C(c1cc(F)cc2cc[nH]c12)=O)C3 N1(C(c2ncc(OC)cc2F)=O)CC2CCN(C(C3SCCC3C)=O)CCC2C1 C1(CNC(C2CC2CC)=O)CCN(C(c2ncoc2C2CC2)=O)CC1 C1(N(C)C(c2cn(C(F)F)cn2)=O)CCCN(C(=O)Cc2cc[nH]c2)CC1 C1(=O)CC(C2CCCC2)N1.C1(C)(NC(C2CN(C(C)C)C2)=O)CCSC1 C#Cc1cccc(C(N2CC(NC(=O)CC3NC(=O)NC3=O)C(C)C2)=O)c1Cl C(=O)(C1=CCC(C)CC1)N1CC(C(C)C)N(C(=O)C(F)CC2CCOC2)CC1 N1(CC(=O)N(CCCN(C(=O)C=CBr)C)C)C(=O)CCC1=O C1(NC(c2c(C)nns2)=O)CCN(C(=O)CCc2ccncc2)CC(O)C1 CCC(O)C(C)C(=O)N(CCC(C)(C)NC(C1CCC(N(C)C)C1)=O)C N1(C(CCCC(C)NC(C2(C)CC(F)C2)=O)=O)CC=C(C(C)(C)C)CC1 N1(C(c2cnc(S)n2C2CC2)=O)CC(C2CCCN(C(C3CC(CF)C3)=O)C2)C1 C(=O)(C(O)C(C)(C)CC)N(CCCNC(c1cc(C(=O)OC)ccn1)=O)CCC Nc1cc2c(cc1C(N1CC3CN(C(C4(C(F)F)CC4)=O)CC3C1)=O)OCO2 N1(C(C(CC)C)=O)C2CCC1C(CNC(=O)C(C)NC(c1ccoc1)=O)C2 CCCCC(C(=O)N(C)CCN(C)C(c1c(C)oc(C)c1Br)=O)N(C)C C(CC(C(=O)N1CCN(CCO)CC1)NC(=O)Cc1cn(CC)nn1)=CC c1(NC(C(N2C(CC(=O)OCC)CCOCC2)=O)=O)ccc2ccccc2c1 N1(C(c2c(C(C)C)ccs2)=O)CCC(CNC(=O)CC(C)CN(C)C)C(F)(F)C1 N(C(=NCCF)NCC1CC2C(C1)C2(F)F)C(C#C)CCc1ccccc1 N1(C(c2cccc(C(C)C)c2N)=O)CCCCC12CN(C(=O)CC1CCOC1)C2 CP(C)(=O)C(CC(=O)N1CCOC(c2n[nH]c(CO)n2)C1)C(F)(F)F Nc1ccc(Br)cc1C(N1CC2CC1CN2C(c1c(F)cccc1Br)=O)=O C1(C(=O)NC2C(NC(C=CSC)=O)CCC2)CCC2CC2CC1 C1(NC(C=C(CCC)C)=O)(CF)CCN(C(=O)CCC2NC(=O)NC2=O)C1 C(C(O)C(C)(C)N1CC1)N(C)C(=O)NCC1CC1(F)F N1(C(C2C3(CCN(C(CCS(C)(=O)=O)=O)C3)C2)=O)CCC2(CC1)COC2 c1(NC(C2CCCO2)=O)c(F)cc(I)c(F)c1F c1(C(N2CC(CN(C(=O)CCc3c[nH]c(=N)[nH]3)C)C2)=O)cc(O)nc(N(C)C)n1 N1(C(c2c(Cl)cn(CC)n2)=O)CC(NC(=O)C2=CCSC2)CC1(C)COCC C12(CNC(c3c(C)cn(C(C)C)c3)=O)CC(NC(C3CC=CCO3)=O)(CCO1)C2 C(CCC(O)C(=O)NCC1(CF)CC1)NC(c1c(C)scn1)=O N1(C(C(C2CCCC2)NC(c2cnc(C)s2)=O)=O)CCC2C(=O)NCC2C1 Cc1nc(C)c(Cc2cn(CCN(C(C3CCC(C(=O)O)SC3)=O)C(C)C)nn2)s1 C1(C(N(C)Cc2ccccn2)=O)CC2CCC(C1)N2C(=O)CC1CSCCO1 C#CCCCC(=O)NCC1CC(F)CN1C(=O)Cc1ccccc1C(F)(F)F C#CCC(C)C(=O)N1CC(C(=O)OC)CC1.C(=O)CCSCC CC(C)C(CCNC(=O)C#CCN(C)C)NC(C1(C(F)F)CCCC1)=O c1(C(=O)NC(C)CCCCNC(=O)CCS(C)=O)cc2c(cn1)OCCO2 CC1CN(C(c2cc(Cl)ncc2F)=O)CCC1CNC(=O)C(C)NC(=O)C1CC1 Cc1cc(=NC(=O)C(=O)N(CC(O)COc2cnn(C)c2)C)[nH]o1 C1(COC)CC(CNC(c2ccnnc2S)=O)N(C(=O)CSCCC#N)C1 c1(C(=O)NC(C2N(c3nnc(C)o3)CCC2)(C)C)cccc2c1ncn2C C(=O)(CCCCC(C)(C)C)NC(C1(O)CCN(C(c2cc(C)nnc2)=O)CC1)C C(=O)(C(C)(C)CC(=O)NC12CC(CNC(C3CCC(NC)C3)=O)(C1)OC2C)OC c1(C(N2C(C)(CNC(=O)C3=NNC(=O)C3)CCC2)=O)cnn2cccc2c1 c1(NC(C(C(C)C)O)C)ccc(S(=O)(=O)NCCSC(F)F)cc1C#N Cc1cccnc1CNC(=O)C(C)N(C)C(c1ccsc1C)=O C#CC1(OC)CN(C(=O)C(C2CCCN(C(C3(F)CC3)=O)C2)C)C1 N1(C(NOCC(C)F)=O)CCC2C(O)CC12 c1(C(N2C(CN(C(CNS(CC)(=O)=O)=O)C)CC(F)C2)=O)ccc2cccnn12 CN1CC(CCO)(CO)C1.C1(C(=O)O)CCOC1C1CC1.c1(C)cnn(C)c1.C1=COC1 c1(C(=O)NCCc2nnc(C)o2)ccc2c(c1)C(=O)CCS2 c1(OC)cnc(F)c(C(N2CCCC2(C)CNC(c2cc(C3CC3)ns2)=O)=O)c1 C#CCCCCCCC(=O)N1CCC1CNC(C1(CCN=[N+]=[N-])CC1)=O N1(C(COC2(C)CN(C(=O)CC3CC4CCC3C4)C2)=O)CC2CC2C2CC12 C1(CNC(c2ncsc2C2CC2)=O)CCCN(C(=O)CC2CCSC2)CC1 c1(C(C)NC(C(c2ccccc2)NC(CNS(CC)(=O)=O)=O)=O)ccc(O)cc1 C(CC(CC)C(=O)NCC12CC(CO1)N(C(=O)CC1CCCC13CC3)C2)=CC n1(CC)c(C)cc(C(=O)NC2CCC2NC(=O)COCC2CCOC2)c1C N1(C(c2c(C)nc(CC)o2)=O)CCC(C)(C)C(NC(c2cncnc2)=O)C1 S(=O)(=O)(c1cccc(C(F)(F)F)c1Br)C(CC)NCn1cncn1 c1(CC)cc(C(=O)NCC2CCCC2NC(C2CS(=O)(=O)C2)=O)cc(N)c1 C1(NC(CC2CCN(Cc3cc(OC)c(F)cc3)C2)=O)CCn2nnnc2C1 N1(C(CNS(CC)(=O)=O)=O)CC(NC(=O)Cc2cncc(O)c2)C(C(F)F)C1 c1(N(C)C)nc(CNC(=O)NCC(c2ccccn2)C)no1 C1(NC(CN(C)C(c2ccc(Cl)s2)=O)=O)CC(CNC(=O)C2=COCC2)C1(C)C c1(CC(=O)NCCCCNC(C2CC2(F)F)=O)sccc1Br C#Cc1cncc(C(=O)NCCOC2CCN(C(=O)C(F)C3CCC3)C2)c1 c1(C(N2C(C)CC2C(N2CCCC2C(N)=O)=O)=O)ccc(C#N)c(Cl)c1 c1(OC)ccc(CC(=O)N(C)CC2CCCCN2C(=O)C2=CCSC2)nc1OC c1(C(N2CCC(C(C)NC(CCCC#CC)=O)CC2)=O)cc(F)c(O)c(Br)c1 CC1(C)C(C)(C(=O)NCCC(=O)NCC=CCl)C1(C)C N1(C(CCOCC)=O)CCCC(C)C1CNC(c1cc(O)nc(OC)n1)=O C(=O)(C(O)P(C)(C)=O)NCC12C(CN(C(c3cn(C)nc3-c3cccs3)=O)C1)C2 c1(C(=O)OC)c(C(N2CC(CNC(c3coc(C(C)(C)C)n3)=O)C2)=O)n[nH]c1C C1(NC(c2ccc(C(F)(F)F)cn2)=O)CCN(Cc2cc([N+](=O)[O-])cs2)C12CC2 C#CC(CC(=O)N(C(C)(C)C)CCC#N)c1cccs1 Cc1nc[nH]c1C(=O)NC(C1(CNC(=O)CSc2nncn2C)CC1)C c1(OC)ccc(C(N2CC=C(CNC(=O)CN3CC=CC3)CC2)=O)cc1Br CC(CC(=O)N1CCC(NC(C2COCCO2)=O)CC1)C(F)(F)C(F)(F)F n1(C=O)nc2c(n1)CCCC2.Cc1nocc1C(N1CC(CC(C)(C)CN)C1)=O N1(C(C(N2CCN(C)CC2)C)=O)CC2CC1(CNC(C1CCCCC1F)=O)C2 N1(C(C2(CC=C)CCC2)=O)CCN(C(c2cnn(C3CCC3)c2C)=O)CC12CC2 CC1CCCCC1CS(=O)(=O)NC(C1CCC2(c3ccccc3)CC12)=O c1(N(CC(O)COC)C(c2ccc(OC)cc2)CO)cnn2ccc(Cl)c(F)c12 C1(CNC(C2(CSC)CC(F)(F)C2)=O)CN(C(=O)CC(CC)C2CC2)CC12CC2 N1(C(C2CC(C#C)(O)C2)=O)CCC(CNC(C2OCC2(C)C)=O)C(C)C1 C1(C(=O)NCCC(C)N(C(=O)CC2(O)CCOCC2)C)CCC2CC2CC1 C=C(C)CC(C)C(=O)N1CCCC(NC(=O)CC2CCC(C(C)C)CC2)C1 c1(CC(=O)NC2CCN(C(c3nc(CC)oc3C)=O)C2CC)ccc(Cl)c(F)c1 N1(CCC(=O)NC(C)CC2CN(C(C3CCN3C(C)(C)C)=O)C2)CCCS1(=O)=O c1(C(=O)NCC(CC=C)NC(c2nnsc2C)=O)cnn(C)c1C(F)F C1(C(N(CC(Cl)Cl)C)=O)CCCCCN1C(c1cn(C)c(=O)cn1)=O C#CCC(C)(C(=O)NCC1CC(=O)N(C)C1)NC(=O)CN(CC)CC C1(C(=O)NC2(c3ccc(F)cc3Cl)CC2)CN=C2N=CNN2C1 CC(C1CC1)=C(F)C(=O)NCC1CC(NC(=O)C(C2CC2)C2CC2)C1 c1(CC(=O)NC2CCN(C(c3c(F)ccc(SC)c3)=O)C2)nc2ncccn2n1 c1(C(=O)NCC2C(NC(c3[nH]c(=N)sc3)=O)CCC2)cnc2ncnn2c1O c1(C(N2CC(F)(CNC(CC(C)OC)=O)C2)=O)ccc2c(c1)nnn2C c1(C(=O)NCC(C)(CNC(=O)CSc2cn[nH]c2)OC)n[nH]c(C)c1O Cc1ncc(C(=O)NC2COCC2CNC(C2(C)CCNC2=O)=O)n1C c1(C(=O)NCC2C(C)CN(C(C3(C#N)CCOCC3)=O)C2)c[nH]c2cccnc12 c1(C(N2CC(N(C)C(C3CNC(=O)N3C)=O)C2)=O)cc2cc(Cl)ccc2[nH]1 C=CCCCCCCCC(=O)NC1CN(C(C2CN(C)CCO2)=O)CC1C(F)F N1(C(COC(C)=O)=O)CC=C(CNC(C2CCN3CCC2C3)=O)CC1 CC(C(=O)N1CCC(O)(CCC(=O)NOCC2(C)CCC2)CC1)S(C)(=O)=O C1(CC(=O)NCC2C(NC(C(C)NC(=O)NCC)=O)CC2)CC(F)(F)C1 c1(OC)cc(SC)ccc1C(=O)NC1(C2CCCN2C(c2ccon2)=O)CC1 C1(C(N2CC(C(C)NC(c3ccc(CC(C)C)s3)=O)C2)=O)CC12CCOC2 Nc1ccc(C(N2CC3(C2)CN(C(c2cc4ccsc4s2)=O)C3)=O)c(Cl)c1Cl C=C1CCN(C(=O)CC23CCCC2C3)C(C(=O)NCCC(=O)N(C)CC)C1 C1(C(=O)NC2(CNC(CCc3ccc(N)cn3)=O)CCC2)CCCCC1(F)F c1(N2CCC3(CC(OC)C3)C2)cc(C)[nH]c(=NCC2CC(C)CC(C)C2)n1 C1(NC(CS(=O)(=O)NC)=O)CCCC12CCN(C(c1cc(C(N)=O)cn1C)=O)CC2 N1(C(CCCC)=O)CC2CCN(C(=O)C3=NNC(=O)CC3)CC2C1 C1(C(=O)NCCN(CC)CC)CCN(C(=O)c2ccncn2)O1 C=CCCCC(=O)N1CCCC1C(N)=O.c12ccc(cc1)NC(=O)CO2 C1(NC(CC(=O)NCC)=O)CN(C(C2CC3(C2)CC3(F)F)=O)CC2(CC2)C1 c1(N2CCCN(C(C)(C)C)CC2)nccc(=NCCc2cc(C(F)F)no2)[nH]1 N1(C(C(COC)N(C)C)=O)Cc2ccccc2C(NC(c2ccc(C#N)n2C)=O)C1 C1(C=O)CCCCN1C(C)C.c1(C(C)C)noc(CCC(N2CC(O)(C)C2)=O)n1 Cc1cccc(NC(=O)C(C)OC2CC2)n1.c12ccccc1C1(CC1)C(=O)CO2 C1(C#N)(C(=O)NCC=C(C(=O)N(CC(=C)C)CC)C)CC1C C1(CC)CCCC(NC(=O)COc2ccc(NC(c3cc(C)ccn3)=O)cc2)C1 c1(C(=O)NCC2(C)CC(NC(CCCCCN(C)C)=O)C2)occ2c1CCCC2 c1(CN(C(=O)CCCc2cccs2)CC(C)NC(C=CC)=O)ccc(C)cc1 C1(NC(c2cccc(OCC)c2)=O)CC(O)CN(C(c2cnc3n2CCC3)=O)C1 c1(C(CCNC(=O)NCC2(CO)CC(OC)C2)C)ccc(Br)cc1 N1(c2c(C#N)cnc(C)n2)CCCC(C2CCN(c3nnc(O)s3)CC2)C1 CCCCCC(O)C(=O)N1CC2CCC1C(NC(C1CNC(=O)C1)=O)C2 C(=O)(C(C(C)NC(c1oc(C)nc1C)=O)C(C)C)N1CC(CC#C)OCC1 O=C(CCCCCCCC1CC1)NNS(=O)(=O)CC1COC(c2ccccc2)C1 CC(C)(C#N)CC(=O)N1CCC(CC(=O)NCCC(N)=O)C1 O=C(CC1=CCN(C(C2CC2Cl)=O)CC1)NCc1ccc(O)cc1 C(CC)(CC)(CCNC(=O)CC1CSC1)NC(CC(CC)c1ccccc1)=O c1(C(N(C(CNC(=O)CCC2(C)CCC(=O)N2)C2CC2)C)=O)ccc(=O)n(C)c1 N1(C(C2CC(C)SCC2)=O)CCC2(CC1)CC2C(N1CCC(=C(F)F)CC1)=O c1(CC(N2C3CCN(C(c4c(C)ncs4)=O)C(C3)C2)=O)cccc([N+](=O)[O-])c1C CC(C)CC(C)(C(N)=O)NC(=O)NC1CC2CC(OC(F)F)C2C1 N1(C(C2N(C)CCCC2)=O)CCC2CN(C(=O)CSC3CCCC3)CC2CC1 Cc1ccc(CCNC(=O)C(C2CCCCC2)NC(C2CC3(CC3)CO2)=O)nc1 N1(C(CCCOC)=O)CCC(C2CC2)(CNC(c2cnc(C)c(C)c2)=O)C1 c1(C(=O)NC2(CC)CN(C(=O)CC(C)n3cccn3)C2)ccc(C2CCC2)cc1 C(C(C)CC(=O)N1CCC(C(=O)NCC(N2CCOCC2)C)(C(C)C)C1)OC C(=O)(C(=O)N=S(C)(C)=O)NCC1C(CC(N2CC(N(C)C)CC2(C)C)=O)C1 C1(CCNC(C2(CC)CCC2)=O)CCCCN1C(c1cccc(F)c1)=O Cc1cc(Cl)ccc1OCC(=O)NC1CC12CCSCC2 c1(NC(=O)C(N2CCC(=CCO)CC2)=O)cccc(C(F)F)c1Cl N1(C(C(CC(C)C)F)=O)CCN(C(=O)C2=CCCCC2)C2COCC12 C(C(CC(C)C)C(=O)N1CCC1C(=O)OC)NC(CCOCCOC)=O C1(C(=O)NC2(C)CCN(C(C(C(C)C)C3CCC3)=O)C2)CCC(C)(C)CO1 CC(C)CCC(O)C(=O)N1CCC(C(C)(C)C(=O)NCC(O)C(C)C)C1 N1(C(C(C)=O)=O)CC2CCCC1C2CNC(=O)Cc1csc(C2CC2)n1 c1(C(CC)C(=O)N2CC(C(N)=O)(CNC(c3coc(C)c3)=O)C2)cccc(Cl)c1 N1(C(C2CN(c3n(C)nnn3)C2)=O)CCN(C(c2ccc(F)o2)=O)C2COCC12 C1(C(=O)NCCCN(CC(C)C)C)CC12CCN(C(C1CCS1(=O)=O)=O)CC2 C1(C(N2C(CNC(c3ncc(OC)nc3)=O)COCC2)=O)CC2CCC(C1)O2 C(=O)(CC(C)C(C)C)N1CC(C(C)NC(COc2ccc(C(CC)=O)cc2)=O)C1 c1(C(N(C)CC2N(C(C(COC)OC)=O)CC(F)C2)=O)csc2cc(Cl)cnc12 N1(C(c2cc(C)ncc2)=O)CCC(F)C(NC(=O)C(c2cccnc2)C)C1 c1(C(N(C2CCN(C(=O)CC3CCCO3)C2)CC#C)=O)cc2c(F)cccc2[nH]1 c1(C(=O)NC2C(NC(C3N(C)CC3)=O)COC2)cc(I)cn1C CC(CCCCNC(C1CNC(=O)N1)=O)NC(=O)CC1CCC(C)(C)O1 c1(OC)ccc(C)cc1CC(=O)Nc1cccc(CNC(=O)C(F)(F)C(F)F)c1 c1(C(=O)NC(C2CCN(C(c3ccno3)=O)C2)(C)C)cncc(F)c1 N1(C(c2ncn(CC)c2)=O)CCN(C(c2cc(F)cc(OC)c2N)=O)C(C)CC1C C1(CN(C)C(c2ccccc2)=O)CN(C(=O)CC#N)CCO1 c1(NC(CC(C(C)OC)NC(c2cc(C)oc2C)=O)=O)ccc2nncn2c1 C#CC1(C(=O)N(CC(C)C#N)C)CCN(C(C2CC(=O)NC(C)C2)=O)C1 Cc1[nH][nH]c2ncnc(=NCCC(=O)NCC3N(C(C)C)CCC3(C)C)c1-2 c1(C(N2CCC(CNC(C=C(C)C)=O)CC2C)=O)ccc2cnnn2c1 N1(C(=O)CN2CC3CC3C2)CCN(C(c2ncc(F)cc2F)=O)C(C2CCC2)C1 c1(NC(C2C(NC(c3cc(Cl)cnc3F)=O)CCC2)=O)ccc([N+](=O)[O-])cc1I Cc1cc(NC(C2(C(C3CC3)Nc3ccc(CO)cc3)CC2)=O)c([N+](=O)[O-])c(C)n1 C=C1C(C(=O)N(C(C)C(=O)NCC(O)CSC2(C(N)=O)CC2)C)C1C(=O)OC C1(CCNC(=O)COCC2CC2)(C(=O)NCC(O)CF)CCCC1 C=C(C)CC(C)C(=O)N1CCC(CCNC(C2CCNC(=O)C2)=O)CC1 C(=O)(C(C(C)C)c1ccn(C)n1)N1C(CNC(CCc2onc(CSC)n2)=O)CC1 c1(C(=O)NCCCCCNC(C2CC3(CCC3O)C2)=O)cc(Cl)ccc1Cl N1(C(C23C(CN(C(c4c(C)scn4)=O)C2)C3)=O)C2C=C(c3ccccc3)CC1CC2 C(=O)(CN=c1cc[nH]cc1)NC(C)(C)CC(=O)NC1C=CCCC1 N1(C(CCN(CCCCC)C)=O)CCC(CNC(=O)CN(C)C(C)C)C12CCC2 C1(N(C(C2C(CC)C2)=O)C)CC2CC1N(C(c1c(N)cncc1Br)=O)C2 Cc1cc(C(=O)NC2CCN(C(C3CCCCN3C(N)=O)=O)CC2F)nc(O)n1 C(CCCC(CO)NC(C1(C2CC2)CCCO1)=O)NC(c1ccc(F)cc1Cl)=O C=CCCCCCC(=O)NCC1CC(NC(=O)CCOCCN(C)C)C1 c1(C(=O)NC2CCCC(CO)NC(=O)C2(CC)CSC)cnn2c(=N)[nH]cnc12 C1(C(N(CC(CC)NC(C2CC3(C2)CC(C)C3)=O)C)=O)CCN(C)C(=O)C1 C1(C(=O)NC2CCC(NC(CC(C)C)=O)CC2)Cc2nnsc2S1 C12(C(=O)OC(c3c(C)cccc3)CC(=O)NC(=O)CC(C)C)CCC(F)(CC1)CC2 C1(C(=O)NCC2C(C(=O)NCCN(CCC)CCC)CC2)CCCC(=O)N1 CCCC(CCCS(C)(=O)=O)C(=O)N1CC(NC(=O)C(CC)Sc2ccccc2)C1 C1(C(=O)NC(C2CCN(C(c3occc3C3CC3)=O)C2)(C)C)CCCN1C c12nc(co1)OC2.CC1CC(C(=O)N(C)C(C)C)C1 N1(CC(N2C(C(C)(C)NC(c3nsnc3O)=O)CCC2)=O)CC2C=CC1C2 C1(C(N2CCC(CC(=O)NCCSC(C)C)C2)=O)CCC(C)(C)OC1 c1(C(=O)OC)n[nH]c(=NC2CC23CCC(N)CC3)s1.C(=O)CS(=O)(=O)N(C)C N1(C(CCCNC(C2C(C)C3CCC2C3)=O)=O)CCCC2OCCC2C1 CC(C)(CC1CC1)C(=O)NC1CCCCC1CNC(c1csc(Br)n1)=O N1(C(c2cnc(CCC)s2)=O)CCC2CN(C(=O)CCCN(C)C(C)C)CC12 CC1CN(C(=O)CCc2cncs2)CCC12CCN(C(=O)Cn1ccnn1)CC2 N1(C(=O)NC(C)Cn2cccn2)CCN(Cc2ccc(Br)cc2)CC1 C1(C(=O)NCCN(C(C(C)CNC(=O)OC(C)(C)C)=O)C)CCCC2CC12 c1(C(c2nnnn2CCCC2CC2)NC2CC(C)C2)ccn(C2CC2)c1 C=CC1CN(C(=O)CCc2ccc(Cl)cc2)CC1NC(=O)CSC(C)(C)C c1(NC(C2CN(C(CC=C)=O)CC2C)=O)cc(C)c(OC)cc1C C(N=c1[nH]c(=NCC2CC3(CCC3)CO2)c2ccccc2[nH]1)C1C(C)(C)OCCC1 C(=O)(C(CCNC(=O)Cn1c(O)nnc1O)OC)NCC.C12(CCCC1)C(=O)O2 c1(C(N2C3CCC(CNC(C4OCCN(C)C4)=O)(C3)C2)=O)cc(F)cc(F)c1O N1(C(c2n(C)nc(C(F)(F)F)c2)=O)CCC2CN(C(=O)CCCC3CC3)CC12 c1(OC)cc(Br)ccc1NC1(CNc2ncnc(C(F)(F)F)c2F)COC1 CCS(=O)(=O)CC(=O)N(C1CN(C(c2ccccc2C(=O)NCCO)=O)CC1O)C N1(C(c2cncc(COC)c2)=O)CC(NC(=O)Cc2ccccc2Cl)CC1(C)C C1(NC(CSCCOC)=O)CC(O)CN(C(c2ccc(C(=O)OC)cc2)=O)C1 c1(C2(CN(C(C(C)(C)C)=O)Cc3cncs3)COC2)ccc(Cl)cc1 Cc1ncccc1CC(=O)NCC(C)NC(c1csc(CC2CCCCC2)n1)=O N(C(=NCC1CCOC1)NCc1ccnn1C)Cc1cnc(C)s1 C12(C(N3CC(SC)(CO)C3)=O)C(NC(c3cc(C)n(C(C)C)n3)=O)C3CC1C2C3 C(CN=C(NCC(c1cnn(C)c1)(C)C)N1CCC2(CC1)C(F)(F)C2(F)F)SC c1(OC)cc(Br)ccc1C(=O)NCC1(C(C)NC(=O)CC=C(C)C)CC1 C1(SC2(CCNC(C=NOC)=O)CC2)CC2CCC(C1)N2C(=O)OC(C)(C)C CCCC(C)(C)C(=O)N1CC2CC1C2NC(c1csc(C(F)F)c1)=O n1(CC(=O)N(C(CCNC(COCCC)=O)C)C)cc(C)c(O)nc1=O C1(NC(C2CC(=C)C2)=O)CCCCC1NC(=O)C(C1CCOCC1)OC CCC(CC(=O)OOCOC1CCOC1)N1CCN(C)CC1 CCC(C(=O)NCC(C)(CO)NC(=O)CC1CN(C(C)=O)C1)N(C)C n1(CC(C=C)O)cc(CNC(c2cc(CN(C)C)[nH]n2)=O)nn1 c1(C(=O)NC(CC(=O)N2CC(CC(C#C)C)C2)CCC)cnc2cc[nH]c2c1 c1(-n2c(-c3nc(C)sc3C)nc(CCCC)n2)ccc(C(F)(F)F)c(C)c1 c1(OCC(N2CC(NC(=O)C(c3ccc(F)cc3)O)C2)=O)cccc(F)c1Br N1(C(c2scc3c2CCCC3)=O)CC2(C1)CN(C(C1(Cl)CC1(F)F)=O)CC2CO c1(C(CN2CCC2)NC(C2(C)CC2(F)Cl)=O)ccc2c(c1)OCO2.C1(=O)CCN1 C12(C(CC)(O)C(=O)Nc3cccc(OC4CCNCC4)c3)CCCCC1OCC2 c1(C(CC(=O)NCCC(C)(C)NC(COC(CC)C)=O)C)c(C)noc1C c1(C(N(CC(CNC(c2c(C#C)cnn2C)=O)C)C)=O)cn(C)c(=O)cc1C C1(CNC(c2ccccc2)C)(NC(=O)OC(C)(C)C)CCOC1 c1(CC(=O)NC(CN(C(=O)CN2CCCCS2(=O)=O)C)(C)C)csc2nccn12 Cc1cccc2c(C(=O)NCCCC(C)(C)NC(c3cnsc3)=O)csc12 C1(F)(CNC(CC(C)(F)F)=O)CCCN(C(=O)CC2CCCCO2)C1 N1(C(c2cn(CC3CCC3)nn2)C(=O)NC(C)C)CCC2(CCCO2)C1 C(=O)(CC1=CCOCC1)NC(c1n[nH]c(-c2ccccc2)c1Br)=O N1(C(Cc2nc(=N)[nH][nH]2)=O)CC(NC(=O)C=CC2CCCC2)CC(F)(F)C1 C1(CC)C(NC(C2(C(F)F)CCCO2)=O)CCN1C(=O)CCC#N C(=O)(C(C)C(C)S(C)(=O)=O)NCC1(F)CCN(C(C(CC(C)C)(C)C)=O)CC1 N1(C(C2(COCC)CC2)=O)CCOC2(C1)CN(C(C1(CC)CCC1)=O)C2 Cc1cc(C(=O)NCCC2CSCCN2C(c2cc(=N)[nH]c(Cl)n2)=O)cc(C)c1Cl c1(CN2CCC(F)(C(N3CC4COCC4C3)=O)C2)n[nH]c2ccc(Br)cc12 C1(CC(=O)NC(C(C)NC(c2c(C)scc2)=O)C)COC(C)(C)CO1 c1(C(C=CC(=O)Nc2cc(SC)[nH]n2)=O)cccc(F)c1.C1(C(=O)OC)(CC)CCC1 C[Si]1(C)CCCCN(C(=O)C(F)C2CC(NC(C34CCC(CC3F)C4)=O)C2)C1 C1(c2nnnn2-c2ccccc2)(NCC(C=C)(C)C)CCN(C)C1C CCCC(C(O)C(=O)N(CCNC(=O)CCCOC(C)C)C1CC1)NC(=O)CC c1(C(=O)NC2(CCCNC(C=CCC)=O)CC2)cccc(OC2CCCC2)n1 C(=O)(C(C)(C)CC(C)C)NCCCC(C(N1CCCN(CC=C)CC1)=O)O C(=O)(C1CCCn2ncnc21)NC1(C)CN(c2cc(C3CC3)nc(Cl)n2)C1 C12(C(=O)NCC3(NC(c4cncc(OCC)c4)=O)CCC3)CCC(C)(CO1)C2 CC(C)CCCCCC(=O)N(C(C)C(=O)NCC(=O)NCC(C)C)C1CC1 c1(C(=O)NCC2C3CN(C(c4cccc(C#C)c4)=O)CC32)cccc2ncnn12 C(=O)(C(C)(F)C(=O)N(C)CCOCCNC(c1ccc(CN(C)C)cc1)=O)OC C1(C(=O)NCCN(C(C(CC)CCc2ccccc2)=O)C)COC2COCC2O1 CC1CN2CCN1C(C(N1CC=CC(NC(c3cn(C)c(=O)nc3O)=O)C1)=O)C2 CC(C)CCC(=O)NC(C1CCCCC1)C(C)NC(=O)CCNC(C1CCC1)=O C1(C(=O)NCc2ccc(C(N(C)CCC3CCCO3)=O)o2)CC(C)(C)CN1C C1(C(=O)NCC2(OC)CN(C(c3cncc(SCC)n3)=O)C2)Cc2cscc2C1 C1(NC(CCCC)=O)CN(C(=O)Cc2c(C)noc2C)C2(CCOCC2)C1 CC(C)(CC(=O)N1CCN(C(=O)CCc2cnc(O)[nH]2)C2CC12)C(F)F C1(C(=O)NC)CCN(C(c2cnn(CCC(C)C)c2-c2nn[nH]n2)=O)CC1 Cc1cc(=NC(=O)N2CC3C=CC2C3)[nH]n1-c1ccccn1.CC C(C)(C(CC(=O)NCCC1CC1)NC(=O)CCC)OC.C1(=O)CCN1 Cc1ccc(Br)c(C)c1C(N1CCC2(CC1)CC2C(N1CC(F)(F)C1)=O)=O C(c1cccc(F)c1)=CCC(=O)N(CC(=O)NCCC(C)N(C)C)C Cc1ccc([N+](=O)[O-])cc1C(=O)NC(C(C)NC(C1(C2CCC2)CC1)=O)C(C)C C(C(=O)N1CCCC(C(=O)NCCC(C)(C)C)C1)(C(C)C)OC c1(NCCCSCC)cc(S(=O)(=O)Nc2cc(F)cnc2Cl)ccc1C#N N1(C(CCOC(C)=O)=O)CCN(C(=O)CCn2ccnn2)C(CC#N)C1 C1(S(C)(=O)=O)(C(N2CCN(C(C3(C)CCCC3)=O)CC2C(F)F)=O)CCCC1 N(C1CCCc2ccccc21)C(C1CC2CC2N1Cc1cnc(C2CC2)nc1)=O CC(CC(=O)NOCCN(CCCF)C)C(C)(C)C1CCC1.C(C(N)=O)O C12(CNC(=O)C=Cc3cnc[nH]3)CCC(CC1)N(C(C1COCCO1)=O)C2 CC1(C)OC(=O)CC1C(=O)NCC1(O)CCCN(C(c2cccnc2CO)=O)C1 N1(C(CN(C(C)=O)C)=O)CCC(C)(C)C1CC(=O)NCCC1=CCCC1 c1(C(N2CCC3(CN(C(C4(OC)CCCOC4)=O)C3)C2)=O)cc2cccnc2o1 c1(C(=O)OCC)cccc(=NCc2coc(C)n2)[nH]1.c12cc(on1)CN2 C(=O)(CCCC(=O)OCC)N1CCC(CNC(=O)C(C)Cc2c(C)noc2C)C1 C1(CC)(CC)CC(NC(c2nccn2C)=O)CN1C(c1ccsc1)=O O=CN1CCCC1C(=O)NCCOCCNC(=O)C1=CCSC1 C(CC(CC)C(=O)N1CCCC(N(CCF)C(c2sc(F)cc2C)=O)C1)=CC c1(C(C)=O)cncc(C(=O)NCCCCNC(=O)C(C(C)O)N(C)C)c1 c1(OC)ccc(NNC(=O)NCC2CC3CCC(C2)O3)cc1Cl c1(C(=O)NCC2CC(OC)CN2C(=O)Cc2cnsc2)ccn2ncccc12 CC1(C(N2CC(C)(C(=O)NCC(O)CC3CCCC3)C2)=O)CCOCC1 N1(C(=O)OCCOC)CCC(O)(CC2COCCN2C2CCCC2)C1 c1(C(=O)NC(COC)CNC(=O)C(O)CC(C)(C)C)ccc(O)cc1[N+](=O)[O-] c1(C(=O)NC2C(NC(C3(OC)CC3)=O)CCC2)ccc2nc(C(F)(F)F)[nH]c2c1 N1(C(C(Cc2ccoc2)NC(=O)CC2CCCNC2=O)=O)CCC2C(C1)C2(F)F c1(NC(C(N2CCCN(C(=O)OC(C)C)CC2)=O)=O)cc2nc(Br)ccc2o1 CCC(C(=O)N1CC(O)(C(C)(C)CNC(=O)CNC(=O)NC2CC2)C1)OC Cc1cc(C(=O)NCC(C)CNC(c2ccc(C(N)=O)o2)=O)ns1 C(=O)(C(C)(C)CC#N)NC1CC(COC)CN1C(=O)CC(O)C(C)C c1(CC(C(=O)NC23CC(CNC(CC)=O)(C2)C3)O)cc(C)sc1C C1(NC(=O)Cc2ncc(Br)cn2)COC2(CCN(C(=O)Cn3cncn3)CC2)C1 c1(N2C(C)(C(=O)NC)CC2)cc(NCCCCCCO)nc(COC)n1 c1(C(N(CC)Cc2ccc(Br)c(F)c2)=O)cc(-c2ccc(F)cn2)cn2ccnc12 CC1=C(C(=O)N2CCN(C(=O)CNC3(C(F)(F)F)CCCC3)CC2)SCCO1 c1(C(=O)OCC)c(NC(=O)C(C2CCOCC2)N)ncn1CC1CC1 CC(C(=O)NOCCCC(=O)N(C)C)N(C(=O)C(O)C1CCC1)C C1(C(=O)NC(C=C)C2CCC2)CN(C(c2sccc2Cl)=O)C(C)(C)C1 N1(C(CC2(CSC)CC2)=O)CCC(C(C)(C)NC(c2occc2Cl)=O)C1 CC(CC(C)(C)C)C(=O)N(C(C)CN(C)C(C1(C)CC1)=O)C c1(C(N2CCCC(C(=O)NCCCCC)CC2)=O)ccc(C)c(C)c1Cl c1(C(N2C(C)(C)C(CNC(C3CCSCC3)=O)CC2)=O)scc2c1CCCC2 C1(C(=O)NC(C(=O)N(CC(C2CCC2)OC)C)C2CCCO2)CCCC1(C)C C(=O)(CCC(F)(F)C(F)F)NCCC1(O)CCN(C(CC2(C)CCC2)=O)C1 C12(C(=O)NC(C)CNC(c3nnn(C)n3)=O)CC(c3ccc(F)cc3)(C1)C2(C)C N(C1CCCc2n[nH]cc21)C(CC1(C)CCN(C(=O)CC2CC2)C1)=O CN(C1CN(C(=O)C2=CCCS2)CCc2ccccc21)C(c1cc[n+]([O-])cc1)=O C(=O)(C(CNC(c1cccc[n+]1[O-])=O)CC(C)C)Nc1c(OC)ccc(Cl)c1 Cc1cc2cc(C(=O)NCC3CC4CC4N3C(C3CCCO3)=O)c(Cl)cc2[nH]1 c1(C(c2n(C3(C)CC3)nnn2)NCCC2CCC2)cc2cc(Br)ccc2s1 C(=O)(C(C)(C)F)NCC1(C(=O)NC(C)C)CC1.C1(c2cscn2)C(=O)N1 c12nn(nc1Br)C2.C1(C(c2nnnn2C2(C)CC2)SCC)CSCCO1 CC1COCC(C(=O)NCc2c[nH]nc2C(=O)N(C2CC3CCC2O3)C)O1 C(=O)(CS(=O)c1ccc(Cl)cc1)NCC(CNC(COc1c(C)noc1C)=O)OC Cc1noc(C)c1C=CC(N1CC(NC(c2ccc(O)c(Cl)n2)=O)CC(O)C1)=O N1(C(C(C)=O)=O)CCCC12CCN(C(=O)COCC(c1ccccc1)C)C2 CC(CS(=O)(=O)c1ccc(F)cc1)C(=O)N1CC2CC1CN2C(=O)CCC(N)=O C1(C(N(CC(CC)NC(=O)C(c2c(C)noc2C)C)CC)=O)C2CC3C(C2)C13 N1(C(CC)=O)CC(C(N2CCC2CO)=O)C2(CCC2)C1 C1(C(=O)NCCC2N(C(c3n[nH]c(C)c3Cl)=O)CCC2)C2CCC3C(C2)CC13 C#Cc1cncc(C(=O)NCC2CN(C(=O)CC3NC(=O)NC3=O)CC23CC3)c1 N1(C(c2c(OC)ccc(Br)c2)=O)CCCC2C1CCN2Cc1scnc1Cl c1(OCC(=O)NCC2CCCN2C(C2C3COCC23)=O)ccc(Cl)c(Cl)c1 Cc1nc(=NCCCNC(C2(c3ccccc3)CCCCO2)=O)[nH]cc1[N+](=O)[O-] Cc1cc(C(F)(F)F)ncc1C(=O)NC(C)(CNC(C1CC1C)=O)CC(C)C N1(C(c2cccn(C3CC3)c2=O)=O)CCC2CN(C(=O)C3=NOCC3)CC2C1 N1(C(C2(C#C)CN(C(=O)C=CCCC(C)C)C2)=O)CCCCC(F)(F)C1 c1(C(N2CCC(NC(c3c(COC)[nH]cc3)=O)CC2C)=O)ccnc2[nH]ncc12 C1(NC(c2cnc(CCC)s2)=O)CC12CCN(C(C1C=CCCC1)=O)C2 C1(C(=O)NCC2CCC3CC23)CCCCN(C(=O)CC2CCC3(CC2)CC3)C1 c1(C(=O)NC(CCN(C)C(c2cc[n+]([O-])cc2)=O)c2cccs2)c[nH]cc(Cl)c1=O C=CCC(C)(C)C(=O)N1CCC(NC(c2ncccc2SCC)=O)C(O)C1 c1(C(C(=O)NCC(CNC(c2c(C)c[nH]n2)=O)C)O)ccccc1Br N1(C(C(COC(C)=O)OC(C)=O)=O)CCCC2(C1)CN(C(=O)C(O)C(C)C)C2 N1(C(c2ccn(CCC)n2)=O)CCCC(C(=O)N(CCOC)CC2CC2)C1 C1(C)CC(=O)N1.C1(C(C(C)C)C(N(CCNC(CC)=O)C)=O)CCCCC1 c1(C(c2ccsc2)N(C(C2CCN(C(C3CC3F)=O)C2)=O)CC)cccnc1 C1(C(=O)OC)CSCCN(C(c2ccc(Cl)o2)=O)C1 C(=O)(C1=NOC(CNC(c2ccc(Cl)o2)=O)C1)NC(c1nc(C)on1)C c1(CNCc2nc(-c3ccc(F)cn3)oc2)c(F)cc(I)cc1F N1CCOC(C(=O)NCCC(=O)NCC2CCCO2)C1.C1(CNC(C)=O)CCC1 Cc1ccc(C)cc1.N1(C(c2cc(C3CC3)on2)=O)CC(c2nccn2C)C1 Cc1cc(CNc2ccc(C(=O)Nc3csnc3C)c(C)c2)cc(Cl)c1 CC1(C)CCCCN(C(C2(F)CCCN(C(=O)C(C)(C)N3CCCC3)C2)=O)C1 C1(C)(C(N2CC(CCNC(C(C3CCCN(C)C3)(C)C)=O)C2)=O)CCC(F)(F)C1 N1(C(C=C(c2ccn(C)n2)F)=O)CC2CCC1CN(C(=O)C(Cl)=CCl)C2 Cc1ncsc1CCC(=O)NCCN(C)CC1CCCN1C(=O)CC1C=CCC1 CCCC(C(=O)N1CC(CNC(=O)CC2(C)CC2)C(C(F)(F)F)C1)OCC CC1(CNC(c2csnc2Cl)=O)CCC(NC(=O)CC2CCC=CCC2)C1 C1(NC(c2c[nH]cc(C)c2=O)=O)COC2CN(C(c3csc(C)c3C)=O)CC12 C1(CCC)CCN(C(=O)CC2CN(C(=O)CC3CCCC4CC34)CCO2)CC1 c1(CC(C)NC(C(=O)Nc2sc(C)c(C(F)(F)F)n2)=O)ccc(Cl)c(Cl)c1 c1(C(N2C(C(C)(C)NC(C3CCCO3)=O)CCC2)=O)cncc2c(O)nccc12 c1(NCCC(c2c(CC)n(CC)nc2)=O)ccc2ccccc2c1 Cc1oc(Cl)nc1C(=O)NC1CCCN(C(=O)CCn2cnnn2)C1 N1(C(C(COC)O)=O)CC23CCCCC2(C1)CN(C(=O)CCc1cnc(C)s1)C3 c1(C(=O)NCCCN(C(C(C)OCCC(C)C)=O)CCO)ccnn1C1CCCC1 CC1CCC(CNC(c2cc(C3CC3)n(C)n2)=O)CN1C(=O)C=CC(F)F n1(CC(=O)NCCN(C(C2CC2c2ccco2)=O)CC)nc(C)ccc1=O N1(C(C2C(C(N)=O)C2)=O)CCCC(NC(=O)Cc2ccn(CC(F)(F)F)n2)CC1 N1(C(CCCCC(N)=O)=O)CCC2CC1CN(C(=O)C1=CS(=O)CCC1)C2 N1(C(COC(CC)C)=O)CCCC1Cc1cn(CC)nn1.C(C)=O n1(C(C(=O)NCC2CCC(CNC(c3cc(SC)no3)=O)C2)C)cnc(C#N)n1 c1(C(C)C)cc(NCC2=CCSC2)n2ncnc2n1.N12CC3CC3(C1)CNC2=O CC(C)(O)CC(=O)N1CC2CC2(NC(c2ccc(N3CCCCCC3)nc2)=O)C1 C1(CC(=O)N(CC(CC)NC(=O)C(C)=CC2CC2)C)CCCCN1CC c1(C(C(=O)N(C)Cc2ccccc2)NCC(C)SC)ccc(C(F)(F)F)o1 N1(C(c2cccc(NC(CC)=O)c2)=O)CCN(C(=O)C(C)C(C)(F)F)CCC1C N1(C(C2(C#C)CN(C(=O)C(CCC)N(C)C)C2)=O)CCC2(CCCCC2)C1 c1(OC)cnc(C(=O)NCC(C(C)C)NC(c2ccnc(Cl)c2N)=O)c(F)c1 Cc1nn(C)c(C(=O)NCCCC(C)NC(C2CCCCNC2=O)=O)c1Cl c1(CCCC)cc(NC(=O)CNCC23CCC(CO)(CO2)C3)n2ncnc2n1 N1(C(c2c(OCC)ccc(F)c2)=O)CC(C)N(C(c2ccoc2)=O)CC1C C(C(C)(C)CN(C)C(C)C)NC(C(C)NS(CC)(=O)=O)=O.C(=O)(C=CI)NC c1(CNC(CCC=C(C)C)=O)ccc(CN(C(=O)CN2CCCC2CO)C)cc1 C1(CCC)(CNC(C2(F)CC2)=O)CCCN(C(=O)CC2CC(CC)C2)C1 C(=O)(C(C)CCCOC)NCCCN(C(C=C(CC)CC)=O)CCO c1(C(=O)NC2CCN(Cc3ccc(Br)s3)C2)coc2c1CCCC2 C12(CNC(CCCC=C)=O)CCC1CCN2C(=O)COc1ccc(C)cc1C C1(C(C)C)CC(C(=O)NCc2cccc(NC(=O)CCc3cncs3)c2)CCO1 N1(C(C2C(c3c(C)ccs3)C2)=O)CCC2(CC1)CCN(C(c1ccsn1)=O)CC2 Cn1cc2cc(C(N3CCCOC(CNC(C4(C)CC4(C)C)=O)C3)=O)ccc2n1 c1(C(N(C(C)C)CCNC(=O)CCC2CC2(F)F)=O)ccc2[nH]c(=N)sc2c1 C(CN(C)C(c1cc(Cl)c[nH]1)=O)(CO)(CO)NC(C(C)OCC=C)=O N1(C(CC=CC=C)=O)CC2(CC(CNC(c3cc(Cl)cnc3OC)=O)C2)C1 C1(C(N2CCN(C(c3c(C(F)(F)F)ncn3O)=O)CC2)=O)COCCC1(F)F c1(C(=O)NC(CC(C)C)C(=O)N2CCCC2CO)ccnc2cc[nH]c12 N1(C(C(C)NC(C)(C)C)=O)CC(NC(=O)CCn2cnc([N+](=O)[O-])c2)C(C)(C)C1 C1(NC(=O)CCc2cnn[nH]2)CCCN(C(=O)CC23COC(CF)(C2)C3)CC1 C1(CC#C)(C(=O)N(C(c2cccc(F)c2)CC)C(C2CCCC2)=O)CCCCC1 C12(NC(CC(CCC)C)=O)CCC(CNC(C3(F)CCCOC3)=O)(CC1)OC2 Cn1cnnc1CC(N1CCC(CNC(=O)CC2(C3CC3)CC2)C1)=O CC1(CNC(=O)C(C2CC=CCC2)NC(C2(F)CCOCC2)=O)CCCC(=O)N1 c1(C(N2CCCC3(Nc4ncnc(Cl)c4Br)CC3C2)=O)cc2ccc(Cl)cc2o1 c1(N2CCC(C)(CO)CC2)ccncc1S(=O)(=O)NC1CCCN(CCF)C1 N1(C(CC2CCN(C(COCCC=C)=O)CC2)=O)CC(=O)NC(C)C1 c1(C(=O)NC2CC(NC(C3(OCC)CCCCC3)=O)C2)cn(C)ccc1=O C1(C(=O)NC2CCN(C(c3ccc(C)nc3N)=O)C23CC3)Cc2nnc(C)n2C1 c1(CC)cnn(CC(N2CCC(NCC)C2)=O)c1.c1(C(=O)NC)scnc1Cl C(=O)(C(C)(C)C(C)NC(=O)CN1CC2CC2C1)NC(CC=CC)CO N1(C(C(C)Oc2ccc(OC)cc2)=O)CC2(C1)CN(C(=O)C=CC1CC1)CCO2 C(c1cc2ccccc2o1)=CC(=O)N(c1c(O)ncc(C(=O)OC)c1)C C12(C(=O)NC(CNC(=O)CCn3cnnn3)CO)CCCN(CC1)C2 C1(NC(c2cnc(SC)s2)=O)CC2CC1N(C(C1CC3CCC3C1)=O)C2 N1(C(Cc2c(C)[nH]nc2Cl)=O)CCCC1C1CCCCN1C(c1cccnn1)=O C(=O)(C(CNC(=O)C(C(C)C)OC1(N)CCCC1)CC=C)NCC=C CC1(CNC(c2ccc(O)cn2)=O)CCN(C(c2cc(C(F)(F)F)ccn2)=O)C1 CC1Cc2c[nH]nc2C(C(=O)NCC2(O)CC(CN)C2)C1.N(C)(C)C N1(C(C(C)OCCOCC)=O)CC2C3CCC(C2C1)N(Cc1csc(C)n1)C3 c1(NC(c2cc(OC)ncc2-c2cccc(OC)n2)=O)cccc2c(I)n[nH]c12 c1(OC)cc(C(N2CCCOC(CNC(c3coc(Cl)c3)=O)C2)=O)cc(Cl)c1 C(=O)(CCC(F)(F)F)NCC1C(NC(c2cn(C)nc2-c2nc[nH]n2)=O)C1 C(CCCC(=O)N(CCC(O)CNC(=O)CCOCC(F)(F)F)CCO)N(C(C)=O)C c1(CNC(C2CC(NC(C3(CC=C)CCOC3)=O)C2)=O)cccc(NC(C)=O)c1 N1(C(Cn2c(C)nc(C)n2)=O)CCC(C)C(CNC(c2ccc3c(c2)CC3)=O)C1 C1(NC(C(C(C)C)C)=O)COC2(CCN(C(c3ccsc3Br)=O)CC2)C1 O=C(C(Cn1cccn1)NC(=O)C(F)OC(F)(F)F)NCC(O)CO C(=O)(CC(C(F)(F)F)S(=O)(=O)Nc1cccc(C(F)F)n1)OCCC N1(C(CC2CCN(c3c(C)nccn3)C2)=O)CCC2(C1)CS(=O)(=O)CCO2 C(=O)(C(C)CC(C)CC)NCCN(CCC)C(c1nc(Cl)sc1Br)=O c1(C(N2C(C(C)(C)CNC(=O)C(=O)N3CCCC3)CCC2)=O)ccc(F)c(O)c1 N1(C(C2(C(=O)OC)C(=C)CC2)=O)CCC(CNC(C2(CCO)CC2)=O)C(F)(F)CC1 C=C1CCN(C(=O)COC(C)(C)C)C(C(=O)NC(COC)CCO)C1 C(=O)(C(O)C(F)(F)F)N1CC(C)(NC(C(N2CC(C)C2)C)=O)C1 N1(C(=O)C=CCBr)CC(C2CCCN(C(C)=O)C2)C1.C12(C(=O)OC)CC(C(=O)O)(C1)C2 c1(C(N2C3C(NC(C(CCC)OCC)=O)C(CC3)C2)=O)ccc2c(c1)CCC=C2 C(=O)(CC1=CCOCC1)NCC1C(N(C)C)CN(C(C(=CC2CCCC2)C)=O)C1 C1(C(=O)NC(C(C)NC(COCCOCC)=O)C)COCCN1C1CCCC1 N1(Cc2cnc(CC)s2)CCC2CN(C(c3ccc(F)cc3Cl)=O)CC2C1 c1(C(=O)NCCCCCNC(C(F)=C(C)C)=O)ccc2c(c1)C(=O)N(C)C2 Cc1cccc(CC(=O)NC2CC2NC(=O)C(C(C)(C)C)N2CCNC2=O)c1F C(C)(C)(CCCNC(C1(n2ccnn2)CC1)=O)NC(C=C(CCC)C)=O C(=O)(CCCC(C)NC(=O)CC1CCCC1C)NCCOCC(=C)C c1(CC(=O)NCC2CC2CNC(c2cc(C3CC3)n[nH]2)=O)cnn2c1OCCC2 C#CC1(NC(c2ccc(CNC(=O)CC(C)(C)C)nc2)=O)CCOC1 N1(C(C2(C(CC)=O)CC2)=O)CCC(CO)(NC(=O)C(c2ccc(Cl)cc2)CO)C1 N1(C(Cn2c(C)ccn2)=O)C2CCC1CC(F)(CNC(C1C(C)(C)C1(F)F)=O)C2 C(=O)(NNc1ccnc(F)c1)Oc1ccc(C#C)cc1OC(F)(F)F C1(C(=O)NC(C)C(O)C(F)F)CCN(C(=O)Cc2csnn2)CCO1 c1(C(C)=O)cc(C(=O)NC2(CNC(C3CCC3CF)=O)CCOCC2)oc1C CN1CCCCCC1C(N1CC(CCNC(C2(C)COCCO2)=O)C1)=O c1(C(N2CCC(O)(CNC(C34CC(OC)C3C4)=O)C2)=O)cc2occc2s1 c1(C(=O)NCC(C)N(C(c2ccc(C)c(C)n2)=O)CC)cc2cnccc2[nH]1 C(=O)(C1=NOC2(CCOC2)C1)NC1(CCOC)CN(C(C(C)SCC)=O)C1 c1(NC(C(C)(C)NC(Cc2cc(CC)no2)=O)=O)cnc(Br)nc1 c1(CNC2CCN(C(c3ccc(Br)cn3)=O)C2)c(C(F)(F)F)cccc1Cl C(C(C)C(C)C(=O)N1CCC(CCC(N2CCCC(C)C2)=O)C1)OC Cn1ncc(C#N)c1C(=O)NCC1(CNC(C2CCC2(F)F)=O)CCCC1 c1(C(N2CCC(NC(C(COC)O)=O)C2)=O)ccc(N)c(C(F)(F)F)n1 C(C)(CN=c1nc2[nH][nH]cc-2c(O)n1)NC(c1ncc(CC)s1)=O c1(OC)cccc2c(C(=O)NC3CC3NC(c3ccn4nnnc4c3)=O)coc12 C#CC1CN(C(C2CSC2)=O)CCN1C(C1CC1CCOC)=O N1(C(c2cc(OC)c(OC)nc2)=O)CCC(C)N(C(C2CC2F)=O)CC1 N1(CCC)CCCC(C(=O)NC2CC(CNC(=O)CN(C3CCCCC3)C)C2)C1 N1(N(c2ccccc2)C(C(c2c(OC)ccc(Cl)c2)OC)=O)CCC(F)(F)CC1C CCC(C)(CC)C(=O)NC1CC(F)CN(C(=O)Cc2cncc(Br)c2)C1 N1(C(c2c(C#N)cccc2)=O)CCC2(CC1)CN(C(C1CC1F)=O)CCC2O C(=O)(CCCC(=O)N1CCN(C)C(CNC(C2SC3C=CC2CC3)=O)C1)OCC N1(C(c2ncc(C)cn2)=O)CCN(C(=O)CC2COC(=O)N2)CC1C(F)F C1CCCCC(=O)N1C.C1(C(C2CCCOC2)=O)C2CCC(F)C12 N1(C(C2C(CC)C2)=O)CC2CC(C(=O)NCCC3CCCC34CC4)(C2)C1 c1(OC)ncnc(N2CCC(C(C)NC(=O)CCCNC(C)=O)C2)c1OC c1(C(C(=O)O)C)ccc(C)s1.c1(N(CC(C)=O)C(=O)CN(C)C(C)=O)cc[nH]n1 CC1(CNC(C2CCN(C(c3nonc3N)=O)C2)=O)CC2(CC2)C1 c1(C(N2CC(CN(C)C(C34CC(O)C3C4)=O)OCC2)=O)ccc2c(c1)CCCS2 C1(C(=O)NC2(CCCC)CC2)CN(C(c2ncncc2OC)=O)CCO1 C(N=c1[nH]c(N2CC(CO)C3(CCC3)C2)nc2c1COC2)c1ccc(C)nn1 c1(OC(C)C)ccc(Cl)c(C(=O)NCC23CC2CN(C(=O)CC2(C)OCCO2)C3)c1 Cc1nc2cc(C(=O)NC3(N4CCOC4=O)CC3)cnc2s1.C12(O)CN(C1)C2=O N1(C(C2=C(C)CCOC2)=O)CCOC2CCN(C(C3C4COCC34)=O)CC12 C1(NC(C2N(C(C(C(C)O)N(C3CC3)C)=O)CCCC2)=O)CCn2nncc2C1 C1(C(=O)NCC2N(C(c3cccc(C#C)c3)=O)CCC2C)CCc2c[nH]nc2C1 Cc1cc(N2CCCC(C)(F)C2)nc(NC2(c3ncccn3)CCC2)n1 CC1CCC(C)N(C(=O)NCCNC(c2cc(OC(F)(F)F)ccc2F)=O)C1 C1(COC)(NC(=O)C(C)Cc2cccc(F)c2)CCN(C(=O)Cn2nccn2)C1 CC(N=c1[nH]c(N(C)Cc2ncnn2C)nc2c1COC2)c1cnc[nH]1 N1(C(COCC#C)=O)CC(NC(c2ccc(=O)oc2)=O)C2(CCC2)C1 C1(C(N2CC3C(NC(c4cncc(C#C)c4)=O)C3C2)=O)CCc2n[nH]c(C)c2C1 C1(C(=O)NCC=CCNC(c2ccc(C)c(C#N)c2)=O)C2Cc3ccccc3C12 C1(CNC(C2CC(=O)NC2)=O)C(O)C(O)CN1C(c1ccnnc1O)=O Cn1nncc1CC(=O)NCC1CCN(C(c2ccc(SC)s2)=O)C1 c1(CN(C(C23CC(C(=O)NCCCSC)(C2)C3)=O)CC)coc2ccccc12 c1(C(=O)NCCCC2CN(C(c3ccns3)=O)CCO2)cc2ncccn2n1 C1(CC)CC(N(c2ccccc2Cl)C2CC2)C12CCC2.c12nc(cs1)C(C)NC2=O N1(C(c2c(C)ccc(C)n2)=O)CCC2CCN(C(c3coc(C4CC4)n3)=O)C2C1 C#Cc1ccccc1NC(N1CC(NC(=O)CC)C(C#N)C1)=O C1(N(C(=O)CC2CC2)C)CCCC(NC(c2cn(CCC3CC3)nn2)=O)C1 N1(C(c2c(C)nc(CO)s2)=O)CC(C2CN(C(C3(C)CCCOC3)=O)C2)C1 c1(C(=O)OC2CCCCC2CCC(F)(F)F)cccc(SC2CC2)c1 C(CC(C)(C)C(=O)NC1CN(C(c2ccc(C(F)F)cn2)=O)CC12CC2)OC C1(CC(C)NC(Cc2n(C)ncc2)=O)CC2CCC(C1)N2C(=O)CN1CC=CC1 c1(OC)cc(C=CC(=O)NCC2(O)CCN(C(=O)CC(C)F)C2)sn1 Cc1cc(C(=O)NCC(C)CC(=O)N(C)Cc2ccn(C)n2)ncc1N N1(C(C(CCC)C)=O)CCCC12CN(Cc1sc(OC)nc1Cl)C2 C(=O)(C1=NOC(C)C1C)Nc1ccc(C(C)C)cn1.C12(F)CCC(C1)C(=O)NC2 CC(C(CO)NC(=O)CCCc1ccsc1)NC(=O)CSC(F)F N1(C(CCn2c(C)ncc2)=O)CCC(CNC(=O)CSC2CCOC2=O)CC1 c1(C(=O)OC)cnc(NCc2ncc(C)cc2Cl)c(Br)c1 C=CCC(CC(=O)NC(c1cscn1)C)NC(=O)CSc1nc[nH]n1 c1(C(=O)NCC2CC(COC)CN2C(=O)CC(C)(C)O)cc(C)c2[nH]cnc2c1 C(CN=C(NCC1CCSC1(C)C)N1CCN2C(=O)OCCC2C1)OC c1(NC(C2CC(F)(F)CN2Cc2ncccn2)=O)cnc2[nH]ccc2c1 C(=O)(C(C)(C=C)CC)NC(CC=C)CNC(c1c[nH]c(=S)cn1)=O c1(C(=O)NCC2CC(C)N(C(C3CCNC3=O)=O)CC2)cc(F)c(Cl)c(C#N)c1Cl c1(CC)cnn(C(C(=O)NC(C)C)N(C)CCN(C)C(C)=O)c1 CC1c2c[nH]nc2CCC1C(=O)NCC12CC(CN1C(c1csc(S)n1)=O)C2 c1(C(=O)NC2CN(C(C3CC(C4CC4)C3)=O)C2)cc2n(n1)CCCC2 C1(C(=O)NCC(C)CN(C)C(c2cc(-c3ccns3)on2)=O)CCN(C)C1=O C1(NC(C2CCCN(C(CC)=O)C2)=O)CS(=O)(=O)CC1N=c1[nH]c(Cl)ncc1Cl CCCC(C(=O)N(C)CCN(C(=O)Cn1ccc(=N)[nH]1)C)NC(N)=O CC1CN(CCCCNC(=O)C(C)(C)Cc2cnn[nH]2)CCO1 N1(C(C2N(CCC)CCC2)=O)CC2CC(NC(C3CC(C)(C(=O)OC)C3)=O)CC1C2 c1(C(=O)NCC(C2CCCC2)NC(CC2CN(C)C2)=O)cncn(C)c1=O C12(NC(c3ccc(OC4CC4)cc3)=O)CC1CN(C(=O)CCCc1cccs1)C2 N1(C(c2c(C)nn(C(C)C)c2C)=O)CC(C)CN(C(=O)CCC(C)(C)C)C(C)C1 Cc1cc(C)c(C(=O)N(C2CCC(NC(c3cnoc3C)=O)CC2)C(C)C)s1 C1(O)(C(C(=O)NC(C)CCNC(=O)C=CC2CC2)(F)F)CCCCC1 C1(C(=O)NC(C(=O)N(C)Cc2onc(C)n2)CO)CCCCCCC1 N1(CCC(C)C2CCCC2)CC2(CCN(C)C2=O)C1 N1(C(c2c(C)n(C3CC3)cc2)=O)CCC(C)(NC(=O)CC2CC3C=CC2C3)CC1 N1(C(CCCC)=O)CCC(NC(c2ccns2)=O)C(c2ccccc2)C1 c1(CCC(=O)NCC2(C)CCN(C(c3c(C)n[nH]c3)=O)C2)c(F)cccc1Cl C(C(=O)N(C)CCOCCCNC(=O)CO)(C(C)C)n1ncc(C)c1 C1(CNC(N2CCC(NC(c3ccccn3)=O)CC2)=O)CC2CC(C1)C2 CC1CCN(C(=O)CCn2ccnn2)C1C.C1(=O)CN1CC1CC1 c1(C(N2CCC(CNC(CC(CC)CC)=O)C2)=O)ccc(S(=O)(=O)CCO)cc1 c1(N2CCCC(COC)CC2)nc2ccccc2nc1NCC1(CO)CC2CC2C1 CC1CN(C(=O)CP(C)(C)=O)CC1(C)C(=O)NC1CC1.N1(C=O)CCCC(O)C1 N1(C(c2cc(C)c(C)c(C)c2)=O)CCC2(CCCC2NC(=O)CN(C)C(N)=O)C1 C1(C(=O)NCC2(SC)CC2)C2CC3C(C2NC(=O)C(O)CC(C)C)C13 c1(OC)cc(Cl)c(C)cc1-c1nnc(COC(c2cc(C)ccc2F)=O)o1 c1(NC(=O)CC2CN(C(c3ccco3)=O)CCO2)c[nH]c2ncccc12 C1(NC(C(C2CC(NC(C=Cc3cc(C)no3)=O)C2)F)=O)CC2OCCCC12 n1(CC(=O)NCC(C)NC(C2CCCC(=O)O2)=O)ncn2nccc2c1=O C(=O)(CCCC(C)(C)C)NCC1CN(C(C(C)CCN(C)C)=O)CC1C(F)(F)F N1(C(CCC=CCC=C)=O)CCC(CC)C1CNC(c1ccsc1OC)=O Cc1sc(NC(=O)Cc2cc(O)ccn2)nc1C1CCOC1 C1(CC(=O)NCC2CN(C(=O)Cc3cnns3)C2)CC2(C1)CC1(CCC1)C2 c1(C(C)C)ccc(C(=O)NC2CCN(C(=O)CCCNC(N)=O)CC2C)c(F)c1 c1(CC)nc(N(C)CC2CCN(C(=O)C3=CCCS3)C2)c2ccsc2n1 C1(NC(c2ccon2)=O)CCN(C(C2CCC(F)CC2)=O)CCC1CO C1(C(N2CC=CC2CNC(C(CC2CC2)OC)=O)=O)(CCF)CCCCC1 c1(SCC)ccccc1CC(N1CCC(C)(CNC(c2occ(C)c2C)=O)C1)=O CC(C)CCC(=O)NCC1COCC1NC(c1c[nH]c(=N)s1)=O C(=O)(CCCC(=O)N1CCCC1CCCNC(=O)CSC)OCC C1(COC)(NC(c2cc(C)oc2C)=O)CCN(C(=O)C2=CCCS2)CC1 O=C(C1=CCCC1)NCCC1CCCN(C(=O)CN2OCCC2=O)C1 c1(CN(C(=O)COC(C)(C)CNC(c2cncs2)=O)C)ncccn1 c1(-c2cc(C(=O)NCC(CN(C(C(=O)NC(C)C)=O)C)C)on2)cccc(F)c1 c1(C(c2nnnn2CCC)NCCCC)cc(OCC)cc(OC)c1Br C1(NC(CCC(=O)NCC)=O)C2CC1(C)CN2C(c1cnn[nH]1)=O c1(NC(C2C(C(=O)NCC3CC3)C2)=O)cc(O)ccc1Cl.CC1(C(=O)NC)COC1 C(=O)(C(C)C(O)C(C)C)NCc1oc(C(=O)NC(CC=C)CC=C)c(C)n1 C1(O)(C(C)NC(C2(CO)CC2)=O)CCN(C(=O)C(C)(O)c2ccccn2)C1 c1(CC2(COCC(C)COC)CCCO2)ccc(Cl)c(F)c1 c1(CNC(C2C3CCC(C3)N2C(=O)CN2CCOCC2)=O)ccc(O)nc1Cl CC(CCC(=O)N1CCC1C1CCCOC1)NC(c1ccc(F)s1)=O N1(C(=O)ON2CCC(CC(=O)NC(C)C)CC2)CCOC2CNCCC12 C(=O)(CC1=CCCCC1)NCCC1OCCN(C(C(C)NC(C)=O)=O)C1 N1(C(N(CCOC)Cc2ccsc2)=O)CCCC1C(C)(F)F CC1CN(C(C2CC2C)=O)CCC1NC(=O)CCc1cncc(F)c1 c1(C(=O)NC2CN(C(c3c(C)cccc3)=O)C(C)CC2)ccc2ccccc2n1 C(=O)(CC1=NNC(=O)C1)NC(C)CNC(=O)C(c1ccccc1)c1cccnc1 N1(CCn2cc(-c3c(C)cc(F)cc3)nn2)CCCCCCC1C Cc1cc2[nH]c(C(N3CCC4(CC3)CC4CNC(=O)Cc3ccon3)=O)cc2o1 C1(CN(CC)Cc2nc(-c3ccccc3)n[nH]2)CCCCN1C(=O)OC(C)(C)C c1(C(=O)NCc2cccc(C(=O)NC3(CF)CCOC3)n2)cncc2cnccc12 C1(NC(=O)C(F)CC2CC2)CC2CCC(C1C)N2C(C1(N2CCOCC2)CCC1)=O C(C(=O)NCC(C)(C)NC(=O)Cc1cccc(OCC#N)c1)(C(C)C)OC c1(C(=O)NCC2(O)CN(C(C(CC(=C)C)NC(C)=O)=O)C2)nc(C)c(C)[nH]c1=O C12(CNC(=O)Cc3ccoc3)CCC1CN(C(c1ccccc1Br)=O)C2 c1(C(N2CC(O)(CNC(C34CC3C4)=O)C2)=O)sc(O)nc1O CC1CCN(C(=O)NC2CC3CC2C3NC(=O)OC(C)(C)C)CC1(F)F C=CCC(C)(C)C(=O)NCCN(C(=O)CNC(C1CCCC1)=O)C C1(n2cc(C(C)N(C(=O)CCc3cncnc3)C)nn2)COC(C)(C)C1 C1(NC(C2(COC)CCC2)=O)CN(C(c2ccnc(C)c2)=O)CC1OC C(=O)(N=c1ccc(N2CCOCC2)n[nH]1)NC(CCCC(=O)OC(C)C)=O CC(C)(C)CC(O)C(=O)NC1CN(C(c2c[nH]nc2-n2cnnn2)=O)CCC1F C1(CNC(c2ncnc(O)c2Br)=O)CCCCC(O)C1 C1(F)(CNC(c2cnn[nH]2)=O)CCC(NC(c2ccoc2C2CC2)=O)C1 N1(C(CSCCC)=O)CCC2CN(C(C3CN(C)CCO3)=O)C(C)C12 N1(CC(N2CC(n3cc(-c4cccs4)nn3)C2)=O)CCOCC1 C1(CC(=O)NCC(=O)NCCC(COC)O)CC=CCN1C c1(C2CC2)c(N)cccc1Cl.N12CCN(CC1)C(=O)C1COCCN1N(C)CC2 Cc1ccc(C(=O)N(C)CC2CCN(C(C3(N(C)C)CCC3)=O)C2)c(O)c1C C(CC(=O)N1CCCC1CC1CCC1)(C(F)(F)F)NC(c1c(C)occ1)=O CCCCS(=O)(=O)NCC(=O)NC1CC1CNC(=O)C(N1C(=O)CCC1=O)C N1(C(c2sc(CC)c(C)c2)=O)CCC2C1CCCN2C(C1(CSC)CC(F)(F)C1)=O c1(C(=O)NC(C2N(C(C(C=C=C)C)=O)CCC2)C)ccc2nc(CC)cn2c1 C(=O)(CCCCCCc1ccccc1)O.N1(C(=O)OC(C)(C)C)CCCC1C(=O)OC CCCCCCCC(=O)OCCOC.C1=CC(=O)N2C1CNCC2 c1(C(N2C(CCC)CN(C(=O)CSC(C)C)CC2)=O)cc2cc(Cl)sc2[nH]1 N1(C2CN(C(CN(CC)CC)=O)C2)CCN(C(=O)Cc2cc(C)no2)CC1 c1(CN2C(C(N3CCCC(Br)C3)=O)CC(O)C2)c(N2CCOCC2)ccnc1Br O=S(=O)(c1cnc(NCC2(CCO)CCOC2)c(Cl)c1)NCCC1CC=CCC1 c1(NCC(c2ccccc2)C)cc(=NCC2(C)CC2)nc2scnn12 C1(CC#C)(C(=O)N(C2CC(SC)C2)C)CCN(C(C2(C)CCCCO2)=O)C1 N1(c2nc(C)nc(O)c2)CCCC2(NC(c3cnc(Cl)cc3Cl)=O)CCCC12 c1(OC)ccc(O)cc1C(N1CCCC(NC(=O)Cc2conc2C)C1)=O C1(C)(NCCC(N2CCC(CNC(C(C)=CC3CC3)=O)CC2)=O)CC2CCC1C2 S(=O)(=O)(c1cccc(F)c1)Nc1ccc(NC(c2c(CC)cno2)=O)cc1 C1(C(N(CC(=O)NCC)C)=O)C(C)CCN(C(=O)CC2CCC(=O)NC2=O)C1C C1(C(N(CC(=O)NC)C)=O)CC(C)(C)CN1C(=O)CCn1ccnn1 N(C(=NCCC1CCOC1)NCc1cccc(Br)n1)CC(c1ccc(C)cc1)O C1(N(C)C(C2CCC(=O)O2)=O)CCCC2CN(C(c3ccnn3C)=O)CC12 c1(C(N2CCC(NC(c3cccc(OC)c3)=O)C23CC3)=O)cccc2nn[nH]c12 C1(CC)CN(C(c2cocc2C)=O)CCC1NC(=O)CCn1ccc(C)n1 Cc1c(C(=O)NC2CCC2NC(c2cnc(C(C)(C)C)o2)=O)cccc1N C1(C)(C(=O)NCC(C#C)OC)CCCN1C(c1ccc(CO)nc1)=O N1(C(C=CC)=O)CC23CCCCC2(C1)CN(C(=O)C(C)NC(C)=O)C3 C1(C(=O)NC2(CCNC(C3(C(C)(F)F)CC3)=O)CC2)CCCCO1 N1(C(c2nn(C)c(O)c2)=O)CCCC(C2CN(C(=O)C=CC3CCCO3)C2)C1 c1(C(=O)NC(C2CCN(C(c3cc(C4CCC4)[nH]n3)=O)C2)C)ccc(F)cc1Cl C1(F)(C(=O)NC(CSCC)CO)CCN(C(=O)COC(C)=O)C1 c1(N2CC(CC)CC3(C2)CCC3)ccc(S(=O)(=O)N2CCN(C)CC2C)cc1F C1(C)(CC(=O)OC)C=CCN1C(=O)CC1CC(C)N(C(=O)C(=O)C(C)C)C1 N1(CC(=O)N(CC(C)O)CCNC(c2cnc(SC)s2)=O)CCC(C)CC1 c1(C(=O)NC2(CCC(=O)NCC=CCCC)CCCC2)cc(O)ccc1F c1(OC)cnc(C(N2CC(NC(c3cccc(OC)c3)=O)CC(F)C2)=O)c(F)c1 C12(C(N3CCC(C(C)NC(c4ccc(CO)cc4)=O)C3)=O)CC3CC1C2C3O Cc1nc2sc(C(=O)NC(=O)CCCSc3ccc(Br)cc3)nn2c1I CC1(C)CCN(C(=O)CC2CC(=O)NC(=O)C2)C1CNC(=O)CC1CCC1 c1(CC(=O)NC2CC2NC(C23CC4CC2C3C4)=O)ccc(Cl)nc1 N1(C(=O)CCNc2cccc(F)c2)CCCCC1C1CCCN1CC=CCl c1(C(N2CCN(C(c3c(CC)scc3)=O)C(C)C2C)=O)cc2cc(N)ccc2[nH]1 CCCC(C)(CC)C(=O)NCc1n[nH]cc1C(N1CC2(CCCC2)C1)=O C(C(C)(C)CC(=O)NCC(C)CC(C)C)NC(c1nc(C)sc1)=O C12(CNC(C(C3CCC3)OC)=O)CCC(CN(C(=O)C=C(C)C(C)(C)C)C1)C2 c1(C(=O)NCC2CCC2NC(C23CCC(CC2)CO3)=O)nnc(O)nc1O N1(C(c2n(CC)ccn2)=O)CC2(CC2)CC1C(=O)NC1CN(C)CC12CC2 c1(CC)cc(F)ccc1C(=O)N(C(C)CNC(c1cscc1F)=O)C CCC(CCCC(=O)N1CCCC(N=[N+]=[N-])C1)NC(c1occc1C)=O c1(CSCC(=O)NCC2CCC(NC(CCCOCC)=O)C2)cccc(C#N)c1 c1(C(N2C(C(C)NC(C3(n4cncn4)CC3)=O)COCC2)=O)ccc(N)cc1C C12(CC(=O)NC(C3CCCN(C(C4C5CCN4CC5)=O)C3)C)CCC(CC1)C2 N1(C(c2[nH]n(C)c(=O)n2)=O)CC2CCCN(C(c3csc4nnsc34)=O)C2C1 c1(C(=O)NC2(CCNC(C3C(C=C)C3)=O)CC2)cc(C)nn1C1CC1 N1(C(c2cnc(C)c(N)c2)=O)CC(NC(=O)CC(O)CN(C)C)CC2(CCC2)C1 c1(CC)ccc(C(=O)NCC2CC3(CC3)CN2C(=O)C(C)(C)C2CC2)cc1CC c1(NC(C2C(CNC(c3cccc(F)c3F)=O)C2)=O)nc(Cl)cnc1Br N#Cc1ccc(C(N2CCC2CNC(C2CC(n3cnnc3)C2)=O)=O)c(F)c1 N1(C(C2=C(C)OCC2)=O)CCC(C2CC2)C1CNC(c1ccc(O)cc1F)=O c1(Nc2cccc(C(=O)NCCOCCO)n2)cc(-n2cccc2)cc(Br)c1 C1(COC)(NC(=O)C2=CCCC2)CCN(C(C2CC2CSC)=O)CC1 c1(C(=O)NCCC2(CNC(c3c(C)scc3)=O)CC2)cccc2c1OC(C)(C)C2 C(c1c(F)ccc(F)c1Cl)=CC(=O)NC1C(CNC(c2c(C)cc[nH]2)=O)COC1 C1(NC(C(CC)COC)=O)CN(C(c2cn(C)c(=O)nc2O)=O)CC12CCC2 C1(NC(c2c(C(C)C)ocn2)=O)CCC(C)N(C(C2CCC(F)(F)C2)=O)C1 CCCCC(O)CC(=O)NCCCCCNC(=O)Cc1cnnn1C c1(C(C)C)n[nH]c(CNC(=O)C=CC(C)(C)NC(c2cnsn2)=O)n1 Cc1ncc(C(=O)NC(C)(C)CCNC(=O)C(C)C2CCOC2)cc1C#N CCC(C)(C(N)=O)NC(=O)CCN(C(=O)Cc1cnccc1C)C(C)C c1(NC(c2ccc(CNC(C3N(C=O)CCC3)=O)o2)=O)ccc2c[nH]nc2c1 N1(C(C(CC)n2cncn2)=O)Cc2n[nH]cc2C1C(=O)Nc1cccc(OC)c1 N1(C(C2C(CC)C2)=O)CCN(C(=O)CCS(C)(=O)=O)C(CF)C1 CC(C)(F)C(C)(F)C(=O)NCC12CC1CN(C(=O)C(F)=CC1CC1)C2 C(C)(CCC1CC1)(c1nnnn1C1CC(F)(F)C1)NCC(C)F c1(C(N2CC(O)(CNC(C(N3CCN(C)CC3)C)=O)C2)=O)cncn(C)c1=O CCC(CC(=O)N1CCCCC1C(C)(C)CNC(=O)CN(CC)CC)C(F)F C1(NC(c2cc(COC)no2)=O)C2CC(NC(=O)COC3CC3)CC12 N1(C(CC)C(=O)OC)CCN(N2CCCCCC2C(=O)OC)CC1 N1(C(c2c(C)cncn2)=O)CCN(C(c2ccc(Cl)s2)=O)C(CF)C1 c1(-c2n(C(COC)C)nc(COC)n2)cnc(C)nc1O C(=O)(C1=C(C)S(=O)(=O)CC1)NCC1C(NC(C2CC(OC)C2)=O)CC1 n1(CC)ncc2cc(C(=O)N(C)CCN(C)C(C3(C#N)CCCOC3)=O)cnc12 Cn1c(CNCC2CC(=C3CCC3)C2)nc2cc(C(=O)OC)ccc12 c1(C(=O)NCCC(C)NC(=O)CC2CCC3CC23)cc(C(N)=O)ccc1F CCC(C)C1C(=O)N2CCC(C)(C)C2C(=O)N1C.C(C(F)F)OC CC12C3C4C1C1C2C3C41C(=O)NC1CC2CCC1N(C(c1cccnc1S)=O)C2 n1(CCC(N2CCC(N(C(C(C)C)=O)C)CC2)=O)cc(C#N)c(O)nc1=O c1(C(N(CC(C)NC(=O)C(O)CSC)CC)=O)ccccc1SC(F)(F)F CCC(C(=O)N1CC(NC(c2ccc(OC)c(Cl)n2)=O)C(C)(C)C1)C(C)(C)CC C1(NC(C(N2CCOCC2)C)=O)CN(C(c2c(C(F)F)cnn2C)=O)CCC1CO CC(C)C(C(=O)NCC(C)(C)CN(C)C(C1(C)CCCOC1)=O)NC(N)=O C(=O)(C1CCCc2nc(C)[nH]c21)NC(CCCNC(c1c[nH]c(=NCC)s1)=O)C C(CNC(=O)CC1(N(C(=O)CNC(N)=O)C)CC1)(C1CC1)SC C1(CC#C)(CNC(=O)Cc2cnsc2)CCN(C(C2CC2C(=O)OC)=O)C1 C(C)(CCCCNC(=O)C(C)(Cn1cccn1)SC)NC(CN(C1CC1)CC)=O C1(C)(C(N2CC(C(C(=O)NCCC3(CC)CCC3)O)C2)=O)CCC(=O)N(C)C1 N1(C(CC(CC)C2CC2)=O)CCCN(C(=O)CN2CCn3ccnc3C2)CC1C C(=O)(C1COc2ccc(F)cc21)NC(CC)CN(C(=O)CSS(C)(=O)=O)C c1(N(C)CC2CN(C(c3cc(C)[nH]n3)=O)C2)ccc(SC)cc1Br.C=CCO c1(CN2C3C(C(=O)NC(c4ccc(Br)cc4Cl)C)C(C3)C2)ccc2c(c1)CNC2 O=C1CC(=O)NC(C(N2CCCC(CC(N3CCCC(O)CC3)=O)C2)=O)C1 N1(C(CC=C)=O)CCC(O)(CCNC(=O)C(=O)NOCC2CCOCC2)CC1 Cc1ccccc1S(=O)(=O)CC(=O)N1CCC(NC(c2occc2Cl)=O)C1 C1(c2cn(C3CCCCN(C)C3)nn2)CC2CCC(C1)N2C(=O)Cc1ccon1 C(=O)(C(=O)N=S(C)(C)=O)NCC(C(C)C)(C)NC(c1noc2c1COCC2)=O N1(C(CCCC(CCC)C)=O)CCC2(CCC(NC(c3ccns3)=O)CC2)CC1 c1(C(=O)NCC(c2ccccc2F)NC(c2cc(C)[nH]n2)=O)ncc2[nH]ncc2n1 C1(CCOC)(NC(C2CCCO2)=O)CCN(C(C2C3CCCC23)=O)C1 c12ccccc1NC(=O)CCOC2.c1(C(C2CCCO2)NC(C)=O)ccccc1F c1(Cn2c(C(C)(C3CC3)OC3CC3)nc(-c3ccnn3C)n2)cccc([N+](=O)[O-])c1 C1(C)(C(N2CC(C)(CCC)C2)=O)CN(C(=O)COC(CC)CC)CC1C C(C(C(C)(C)C)C(=O)NCC(C)Oc1ccccc1)NC(C1C2COCC12)=O CN1CCN(C(C2CCN2C(=O)CCc2cnco2)=O)CC1=O C1(CNC(C(C(=O)NC)(C)C)=O)CC2CCC(C1)N2C(=O)C#CC1CC1 Cc1sncc1C(=O)N(C)CCN(C)C(=O)NC1(CC(=O)N(C)C)CCCC1 C1(CC)CCCN(CC(=O)NCCN2CCC(NC(=O)C(C)(C)C3CC3)CC2)C1 C1(NC(C2(N(C)C)CCCC2)=O)CC2CCC(C1)N2C(=O)CCCNC(N)=O n1(C2C(C(N(C3CCNCCC3C)CCC)=O)CCCC2)cnc2ccccc12 Cc1cc2c(C(N3C4CCC3CC(NC(c3ccn(C)n3)=O)C4)=O)cccc2o1 n1(CC)cc(Cl)c(C(=O)NC2CCN(C(=O)Cc3n[nH]cc3Br)C2)n1 C1(C)(C(=O)NCCN(C(c2nc(C(C)C)oc2C)=O)CC)Cc2ccccc2N1 CCC(C(C)(C)c1nnnn1CCCF)NCCc1ccccc1 N1(C(C2OCCN(C(c3nc(CC)sc3)=O)C2)=O)CCC12CCC(C)CC2 c1(C(=O)NCC23N(C(C(C)N4CCC4)=O)CCC2CC3)ccc2ccccc2c1 C1(C(N(C(C(CC)C)C)C)=O)C2CC3C(C2=O)C13.C12CC(C1)C(=O)N2C CCC1=C(C(=O)NC(CNC(c2cccnc2SC(C)C)=O)C(C)C)SCCO1 c12ccc(o1)CN1CCC1CNC2=O.c1(C(N(C2CC2)CC)C)ccccn1 C1(CC=C)(C(=O)NC(C2(O)CN(C(C3(C)CCCS3)=O)C2)C)CCCC1 N1(C(c2cc(C(C)=O)oc2)=O)CC2OCCN(C(c3cc(CC)c(C)s3)=O)C2C1 Cc1cc(C#N)nc(N2CCCC2C2CCN(C(=O)C(F)(F)C3CC3)C2)n1 C1(NC(CC2CC(NC(c3ccc(C(N)=O)[nH]3)=O)C2)=O)CCCCCC1O C1(S(N)(=O)=O)(C(=O)NCCCOCC(C)(C)NC(c2c(CC)ccs2)=O)CC1 c1(C(=O)NC2C(C)CN(C(=O)CC34CCC(CC3)C4)C2)cc2c(nn1)OCCS2 C1(NC(C2(C(C)C)CCC2)=O)CN(C(C2CC(C)CCO2)=O)C(C)(C)C1 CN1C(=O)CCC1C(N1CC2CC2(CNC(C2(C3CCCCO3)CCC2)=O)C1)=O c1(C(N2CCC(C(F)F)(CNC(COC(CC)C)=O)C2)=O)cncc2ccsc12 N1(C(c2ccc(O)nc2)=O)CCC(NC(C2(Br)CCC2)=O)C(F)C1 c1(OC)ccc(CNC(=O)CC(c2c(F)cccc2Cl)=O)c(OC)c1OC c1(NC(N(CC(CC)CC)CC)=O)n[nH]c2cc(O)ccc12 N1(C(C2(OC)CCCC2)=O)CCC(F)(C(=O)NCC2CCC=CO2)CC1 C12(CNC(c3cnc(SC)s3)=O)CC(CO1)N(C(c1cnoc1C(C)C)=O)C2 Cc1coc2ccc(C(N3CC=CC3CNC(=O)Nc3ccccc3Cl)=O)cc12 C1(OC)=CC=NC=CC(c2cccnc2CNC(c2cnc(C(C)(C)C)cn2)=O)=C1 c1(C(N2CCC(NC(C(COC)O)=O)C2)=O)cc(C)cc(O)n1 N1(CC2CCCN(CC(c3nc4ccccc4s3)(C)C)C2)CCn2ncc(Cl)c2C1 N1(C(CNc2ccc(C#N)cc2)=O)CCC2(C1)CN(C(C1CCC3CCC13)=O)C2 N1(C(c2n(CC)nnc2)=O)CCC(F)(CNC(=O)C=C(C)c2ccsc2)CC1 C=C=CCCC(=O)NCC1(F)CCC(CNC(=O)C(C)N2CCC2)C1 c1(C(=O)NC2C(NC(c3cn(C)nc3C(F)F)=O)CCC2)ccc2c(c1)COCO2 Cc1ncc2n1CCC(C(N1CC(C3(NC(C4COC(=O)N4)=O)CC3)C1)=O)C2 CCC(CC)(CC)C(=O)NC12CC(COC)(CN1C(=O)C(COC)OC)C2 c1(C(N2CC(CNC(c3c(OCC)nccc3)=O)C2)=O)ccc([N+](=O)[O-])cc1 Cn1nccc1C(C(=O)N1CCC1C1CCC1)NCC1CCCCO1 C1(CCNC(c2ccc(C(C)C)o2)=O)CCCN(C(C2(C)CCC(=O)C2)=O)C1 Cn1cc(C#CCNC(=O)C(CNC(C2CC2(C)C)=O)C(C)(C)C)cn1 C(c1ccco1)=C(C)C(=O)N(CC(C)N(C)C(c1ccc(C(C)C)o1)=O)C Cc1cccc(CN2CC3C(C2)N3C(=O)CCc2cnc[nH]2)c1 C1(C(CNC(C(C)C2CC2)=O)C)CCN(C(c2ccn(CN(C)C)n2)=O)CC1 C#Cc1ccc(CN2CCC(C(=O)NC(Cc3ccc(OC)cc3)CO)C2)cc1 C1(O)(C(C)NC(c2cscn2)=O)CCN(C(=O)Cc2cccnc2O)C1 C1(C(N2CC(CNC(C(C)C3CCOC3)=O)C2)=O)CC2CC(=O)C1O2 CC(C)(CCCNC(=O)CCc1nc(-c2ccco2)no1)NC(=O)C(N)=O.C1CO1 C12(C(N3CC(NC(c4nn(C)c(O)c4)=O)(CO)C3)=O)C3C4C1C1C2C3C41CO c1(CO)ccc2c(c1)nc(C1CCN(c3cc(-n4cncn4)ncn3)CC1)n2C N1(C(C(C(C)SC)O)=O)CCC(C)(NC(=O)COc2c(C)cccc2Cl)CC1 CCCCC(CC(=O)NC1CCCN(C)C1=O)NC(=O)CNC(=O)OC c1(C(N2C(CNC(CCc3ccc(C)s3)=O)CC2)=O)cnc2[nH]ccc2n1 C12(C(=O)NC(C=C)(C)C)CCN(C(=O)CCN(C)C(C)=O)CCC1C2 N1(C(CC(C)CF)=O)CCC(C2CCN(C(=O)CN(C)C(C)C)CC2)CC1 Cc1cc(C(=O)NCC23CC(CO2)N(C(=O)Cn2nccc2N)C3)ncc1C(N)=O N1(C(=O)Cc2ncc(F)cc2F)CCC2C(CCCN2C(c2ccc[nH]2)=O)C1 c1(C(=O)NC2CC(CNC(CCC(=O)NC)=O)C23CCC3)ccn2cncc2c1 C1(CC(=O)NCCC(CNC(c2c(C)occ2)=O)O)Cc2ccc(Cl)cc2C1=O N1(C(C(C2CC2)OC)=O)CCCC2(CCN(c3cc(CO)ncn3)C2)C1 CCC(CC(=O)N1CCN(C(=O)CC(C)(F)F)CC(C)(F)C1)C(C)C CCC(CNC(=O)CC(C)(O)C1CC1)(CC)NC(c1ccc(C(N)=O)o1)=O N1(C(CC(C(F)F)NC(=O)CNc2ccccc2)=O)CC2(CCC1CO)CC2 c1(C(CC)NCCOc2ccccc2F)cc(Br)c(C)cn1 N1(C(CCCC)=O)CCC(CF)(OCC)C1.c12coc(n1)CNC2=O C1(NC(CCCNC(N)=O)=O)CCN(C(c2cc(C(N)=O)c[nH]2)=O)CC1O C1(C(=O)NC(c2ccc(-c3ncco3)cc2)C)CCNC2CCOCC12 c1(C(N2CCC(F)(CNC(C3C(C)C3)=O)C2)=O)ccc2[nH]c(=O)c(=O)[nH]c2c1 C(CCCCCC(=O)NC(c1n[nH]c(C)n1)C)NC(c1ccc(C#C)nc1)=O C(C(C)(C)C(=O)NCC1CCC1(F)F)NC(Cc1c(C)ocn1)=O C1(OC)CN(C(=O)CC2NC(=O)NC2=O)CCC1NC(C1(CCOC)CC1)=O Cc1noc(C)c1CC(C)C(=O)NCC1CC(NC(c2c(C)noc2C)=O)C1 CCCC(C)(CC)C(=O)NCCCNC(c1csnc1C)=O C(C(C)N=c1[nH]c(=NCCCN2CCC(C)CC2)[nH]c2cccnc12)OCC n1(CC(=O)NCC(CN(C(CNC(CN(C)C)=O)=O)C)O)cn[nH]c1=N C12(NC(c3cc4scc(Cl)c4[nH]3)=O)CCCC1(F)CN(C(c1cc(F)n[nH]1)=O)C2 C1(N)CCC(=C(F)F)CC1.N1(CCOC)CCCC(O)(CN(C)C(C)=O)C1 c1(NC)ccc(C(N2CC(N(C(=O)C(O)CN(C)C)C)C3(CC3)C2)=O)cc1F N1(C(c2ccc(CCC)s2)=O)CC2=C(C1)CN(C(c1ncccc1Cl)=O)C2 N1(C(C2CCN(C(C)=O)CC2)=O)CC2CC(NC(C3CC4(CCC4=O)C3)=O)C(C2)C1 Cc1cccc2c1c(CNC1CC(C(=O)Nc3nccc4[nH]ccc34)C1)cn2C N1(C(CSCCC)=O)CCCC(C(C)(C)C(=O)NCC(CN(C)C)CO)C1 N1(c2nc(COCC)nc(O)c2)CCC(C2CCCN(C(c3cccs3)=O)C2)C1 C1(C(=O)NC(CC=C)C)CN(C(c2ocnc2CC)=O)CC(C)(C)C1 N1(C(C(C)=C2CC2)=O)CCC2(CC1)CN(C(c1cnc3n1CCC3)=O)C2 c1(CNC(N(c2cccc(C(N3CCOCC3)=O)c2)C)=O)ccnc(Br)c1 c1(C(=O)NCCN(C2CCCCC2)C(C2CCS(=O)(=O)N2)=O)ncc(Cl)cc1F C1(C(=O)NC2CC(CNC(=O)CC3CCCC(=O)N3)C2)CC12CCSCC2 c1(CC(C(=O)N(C(C)C)CCN(C)C(c2cnn(C)c2)C)C)ccc(Cl)cc1 N1(C(C(C)N(CC(F)(F)F)CC(F)(F)F)=O)CC2(CCN(C(=O)CC3CC3)CC2)C1 c1(C(N(C(CNC(C2CC3(CC(OC)C3)C2)=O)C)C)=O)cccc2cnsc12 c1(NC(C=CCNC(C(CC)n2cncn2)=O)=O)cccc(CO)c1C c1(CC(=O)NC(C2CCN(C(C(C)(C)OC(C)=O)=O)C2)C)ccc2c(c1)COC2 C1(NC(C2CC(OC)C2)=O)CN(C(c2ccc(F)s2)=O)CCC1C(F)(F)F CCCCCC(O)CC(=O)NC1C2CC3C1C3C2C(=O)NC1CCCC12CC2 c1(CCC(=O)NC2C(CNC(CC3C(CC)C3)=O)CC2)cc(C)no1 c1(C(=O)NC2(CCNC(C3CCCC(C)C3)=O)CCC2)ccc2[nH]ccc2c1 N#Cc1cc([N+](=O)[O-])cnc1NCC1CN(C(C2CS(=O)(=O)CC(=O)N2)=O)C1 C1(C(=O)OC)CCC(F)(CN)CC1.c12ccc(C(F)(F)F)cc1NC2=O C12(C(=O)OCC)CC(N(C)C(=O)NC3CC3C#N)(C1)C2 c1(OC)ccc2scc(CNC3CC4NCCC34)c2c1 C1(CNC(=O)CC2CN3CCN2CC3)CC2(CCC2)CN1C(=O)Cc1cnc[nH]1 C(c1ccc(C)s1)=CC(=O)NC1CCC(CC2(NC(C(COC)OC)=O)CC2)CC1 Cc1nn(-c2ccncc2)cc1C(=O)N(C(C)CNC(=O)CC1(CC#N)CC1)C Cc1cnn2ccc(C(=O)NCC3CCN(C(C4CC(=C(F)F)C4)=O)CC3)nc12 C(=O)(CCC(C(C)C)NC(=O)CCc1cnn(C)c1)N1C(CC(=O)NC)CC1 c1(NCc2nc(C)[nH]n2)nc2ccsc2c(=NC(C)Cc2cc(F)cc(F)c2)[nH]1 c1(C(N2C(CCNC(c3c(C)onc3O)=O)COCC2)=O)cc2n(c1)CCOC2 C#Cc1cnc(=NCCC2(O)CCN(C(c3cccnc3CC)=O)CC2)[nH]c1 C1(C(=O)NCc2c(CC)noc2CC)CCCN1NC(=O)C1CC1(F)F N1(CC)CCC(C(=O)NCC2(O)CN(C(c3snnc3C3CC3)=O)C2)C1 c1(C(=O)NC2CCC(CCNC(C3(CCC)CC3)=O)C2)cnc2n1CCCC2 C1(C#N)(OC)CC(C(N2CC3C(NC(=O)CCc4ccccn4)C3C2)=O)C1 c1(C(N2CCC(C)(NC(C3CCC4(CCC4)C3)=O)C2)=O)cc2n(n1)CCNC2=O O=C(C1=NOC(C(O)CO)C1)N1CC(CO)(NC(C2(C3CCCO3)CC2)=O)C1 CCC(C(=O)NCC(CNC(=O)CCc1cn(C)nn1)OC)N(C)C c1(C(=O)NC2(CC=C)CCN(C(=O)C(F)CC3CCOC3)C2)ncnc2ccsc12 CC1CN(C(c2ccc(C3CC3)c(F)c2)=O)CCN1C(=O)CN1CCCC1CO c1(C(=O)NCC2(CNC(C(C)n3ccnn3)=O)CCC2)ccc2cn(C)nc2c1 C1(C(N(CCCNC(CC(C)(C)OC)=O)C)=O)CCCCC12OCCO2 c1(CC)c[nH]cc1C(=O)NCCC1CCN(C(C2CC23CC3)=O)C1 N1(C(C(CC2CCC2)NC(C)=O)=O)CC2CCCC(C1)N2Cc1cnn(C)c1 c1(-c2cn(CC3N(C(COC)=O)CCC3)nn2)c(C)noc1C N1(C(c2c(C)noc2C(C)C)=O)CCC(O)(CNC(=O)CCC2CC2(Cl)Cl)CC1 C(CCC(=O)N(C1CCCC1N(C)C(=O)NC)C)OCCOCC=C N1(C(C=CCC)=O)C2CCC1CC(O)(CNC(=O)COCCc1ccc(Cl)s1)C2 C(=O)(C1=NOC2(CCC2)C1)NCC(C(C)C)NC(C(CC(=C)C)C)=O c12ccc3c(c1)CN(C3)C(C)C(=O)N2.CCC(=O)NCCCNC(C)=O c1(C(=O)NC(C(C)NC(c2nc(C)oc2)=O)C)cccc(OCC(F)(F)F)c1 Cc1c(C(=O)NCC2CCN2C(C2(C#N)CC3(CC3)C2)=O)cccc1S(N)(=O)=O CC1(C)COC(CC(=O)NCC2(O)CN(C(=O)CNc3nccs3)C2)CO1 C=CC(C)(C)C(=O)C(=O)OCCOCC=C.C1(CC(C)N)CN(C(=O)C=C)C1 N1(C(CCCCOCC)=O)CC2CC(C)N(C(C3CCOC3C)=O)C2C1 C(N1C(=O)Cc2ccccc21)n1nc(N(C(=O)OC(C)(C)C)CCF)oc1=O CC(C)C(CC(=O)NCC(Cl)Cl)NC(c1ccco1)=O C1(C(=O)NCCCCCNC(=O)CCc2ccncn2)CC2(C1)CC1(CC1)C2 C1(CNC(c2c(OC)cccc2)=O)CC2COCC2N1c1ncc(C)cn1 c1(C(=O)NC2CC3CC(NC(C(CCC)OC)=O)CC32)cc2cccc(C)c2[nH]1 CCC(CCC(=O)NCC(C(=O)NCc1c(O)cccc1F)N(C)C)OC N1(C(C(C)CCN(C)C)=O)CCCC(C)(NC(=O)CCOc2cccnc2)C1 C1(NC(C(c2cccs2)NC(CCCOCCOC)=O)=O)CCc2nncn2C1 c1(-c2cn(C3CN(C(C4(OC(C)C)CCC4)=O)CC3O)nn2)c(F)cccc1F C1(CNC(c2ncn(CC)n2)=O)CN(C(c2c(CO)noc2C)=O)C(C)(C)C1 c1(C(N2C(CNC(=O)CCOC3CC3)CC2)=O)cc2sc(Cl)cc2s1 C1(C(=O)NCC2CC(F)(CNC(C3N(C)C(=O)CC3)=O)C2)CN(CP(C)(C)=O)C1 Cc1cc(C(=O)NCCC2(C)CCN(C(c3cncn3C3CC3)=O)C2)ccn1 C(=O)(CCS(N)(=O)=O)N1CC(CCC)C(NC(C2(NC(=O)NC)CC2)=O)C1 CC1CCN(C(C2CC3(CCC3O)C2)=O)CC1CC(=O)NCC(C)(O)CCO N1(C(CC23CC(C)(OC2)C3)=O)CC(N=c2c(C#N)c[nH]c3ccccc23)C1 c1(C(=O)NC2(CCNC(c3c(C)ccc(C)c3)=O)CC2)cccc([N+](=O)[O-])c1 c1(C(=O)NC2CCN(Cc3nc(-c4cccs4)no3)C2)ccn2c1CSCC2 c1(OC)cc(C)cc(OC)c1C1CCCN1C(c1ccc(N2CCCC2)n1C)CO Cc1ccc(OCC(NC=CC(=O)Cn2cc(-c3c(C)noc3C)nn2)=O)cc1 c1(-c2c(CCC)cccn2)ccc(-c2nccn2C(C)(C)CO)cc1OC N1(C(=O)C(F)(F)c2cncs2)CC2CCN(C(=O)Cn3cncc3Cl)CC(C2)C1 c1(CCC)nnsc1C(=O)N(CC(C)(C)NC(C1C=CCC1)=O)C C1(C2(O)CCC2)(C(=O)NCC23C(CN(C(C(C)NC(CC)=O)=O)C2)C3)CC1 N1(c2n(C(CC=C)C3CC3)c(C3CCC(=O)N3)nn2)CCc2nc(C)ncc2C1 n1(C(C2CCCCCC2)C)nc(-c2cncs2)nc1C1CC=CC1 Cc1cccc2[nH]cc(C(=O)NCC(C)(O)CNC(C34CCCC3C4)=O)c12 c1(NC(CC)=O)cc(OC)c(S(=O)(=O)N2CCCCC2C2CCCOC2)cc1Br C(C(=O)N1CC(O)(C2CCCO2)C1)(C(C)O)NC(C(C)CC1CCC1)=O C(C(CC(=O)NOCC(=O)OC)NC1CC1)NC(C(C(CC)C)=O)=O c1(C(=O)NC2(C)CCN(C(C3CCCCS3)=O)C2)ccc(C2=NOC(=O)C2)cc1 Cc1ccc2[nH]cc(CC(=O)N(CC(C)(C)NC(=O)Cn3cncn3)C)c2c1 C1(NC(c2ccc(C#N)cc2)CC)CCC2(CCC2)CN1CCOC C1(CC)CN(C(=O)C(N2CCOC(COCC(F)(F)F)C2)=O)c2ccccc2N1 O=C(N=c1[nH]onc1C1CC1)c1sccc1NCC1CC=CCC1 N1(C(c2n[nH]c(C)c2F)=O)CCCC2(CCN(C(c3cnc(C)n3C)=O)C2)C1 c1(C(C(=O)NCC2C(C)C2)N(C)Cc2cccc(F)c2)nccc(Cl)c1Cl C1(NC(C2CC(C(C)C)C2)=O)CN(C(=O)CN2CSCC2=O)CC(C)(C)C1 N1(C(CCN(C(c2c(OCCC)cccc2)=O)CCC)=O)CCNC(=O)CC1C CON1CC(C(=O)N(C)CCNC(=O)C=Cc2cccc(C(F)(F)F)c2)CC1=O C1(C(N(CCCOC)CCO)=O)CC(NC(c2ccnc(C)c2)=O)C12CCC2 c1(OCCN(C(c2n(CC)nnc2)C(=O)NC)C)ccccc1C C(C(C)(C(C)C)NC(C1CN2CCC1C2)=O)NC(c1c(OCC)scn1)=O Nc1cc(F)c(C(N2CC3CC3(NC(c3cc(F)ccc3F)=O)C2)=O)cc1Cl c1(N(C(C(C)C)=O)C2CC2)cccc(OCC(N2CCCC(c3nccs3)C2)=O)c1 N1(C(CC2C(NC(C(C3CC3)OCC)=O)CCC2)=O)CC(N=[N+]=[N-])C1 N1(C(C(C)=CC=C)=O)CC2CC(C(N3CCCC(OCC)C3)=O)CC2C1 N1(C(c2cc(C)[nH]n2)=O)CC2CCC1CC2NC(c1ccnc(C2CC2)c1)=O N1(c2nccc(C(=O)OC(C)(C)C)c2)CCC(NC(=O)OC(C)(C)C)C(F)C1 C1(CC(=O)NC(CN(C)C(c2ccc(C3CC3)cc2)=O)(C)C)CCC=CCC1 C1(C(=O)Nc2cc(OC)cc(F)c2)CC2(CCCC(N)C2)C1 Cc1nc2ccc(C(N3CCC(C4CC4)C3)C(=O)NC3CCOCC3)cc2[nH]1 C1(CO)(NCc2cc(OC)ns2)CCN(C(=O)C(C(C)C)Sc2ccccc2)C1 C1(C(N)=O)CC(F)CN1c1nnc(C2CC2)n1C1CC1 N1(C(CC(C)(C)C)=O)CC2CCN(S(=O)(=O)Cc3cccnc3)CC2C1 N#Cc1ccc(-c2ccc(NC(c3cc(Cl)ccc3O)=O)cc2)c(Cl)c1 c1(C(N2CC(N3C(=O)CC(NC(CNC(C)=O)=O)C3)C2)=O)ncccc1O CCC(C)(C)C(C)CC(=O)NCC1(CNC(C2CCc3c(nnn3C)C2)=O)CC1 N1(C(C(C)c2ccsn2)=O)CCc2ccccc2C(NC(C2(Cl)CC2)=O)C1 N#CC1(C(N2CC(CC(N3CCC(N4CCC4)C3)=O)C3(CC3)C2)=O)CCCCC1 CC1C(NC(C2(CC3CC3)CCCCC2)=O)CCN1C(=O)CCCN1CCCCC1 c1(C(=O)NC2CN(C(c3cn(CC)nc3)=O)C(CO)C2)cc(C)c(Cl)cc1C C(=O)(C(C)(F)C(C)(C)F)N1CC=C(CNC(c2cnn(C)c2C(F)(F)F)=O)CC1 CC1(C)C(NC(CCCn2cc(O)c(C(F)(F)F)n2)c2nnnn2C2CC2)C1(C)C N1(C(=O)C(O)Cc2cnc[nH]2)CC2CCCCC2(NC(C2CN(C(N)=O)C2)=O)C1 c1(C(N2C(C)(C)C(NC(C3CC3(C)C(F)F)=O)CC2)=O)ccc2c(c1)CCCC2 c1(C(=O)NC2C3CN(C(C=CSC)=O)C2C3)ccc(C)c(O)n1 Cc1cccc(Cl)c1OCCNC(=O)NCC(CO)n1cccn1 c1(CC)cc(CC(=O)NOCC(=O)NC(C)CN(C)C)n(C)n1 CC1=NN(C)C(=O)C1CC(=O)N(CCCNC(=O)C(C)OCc1ccccn1)C N1(C(CCc2onc(CC)n2)=O)CC(NC(=O)C(C)n2cnnn2)C(F)C1 c1(-c2cc(CC(=O)NCCN(C(=O)CSCC3CC3)CC)no2)ccc(F)cc1 C1(NC(c2cnc(C3CC3)[nH]2)=O)CCN(C(c2ccoc2Br)=O)C1 C1(C(N2CC(n3cnnn3)C2)=O)CCC2CCC1N2C(=O)CCc1ccncn1 C1(N(C(=O)CCOCCOC)CCN)CCCN(C(c2nnc(S)n2C)=O)C1.CC c1(C(N2CC(C)C(CNC(=O)CCN3CCCCCC3)C2)=O)cc2occc2s1 c1(C(N2CCC(C(N(CCC#C)C)=O)C2C(C)C)=O)ccn2ccccc12 C(=O)(C(C)(C)CN(C(=O)C(F)n1ccnc1)C)NCC(CCC)C C=C(C)CC(C(=O)N1CCN(C(=O)CSC)C(CF)C1)NC(=O)OC(C)(C)C N1(C(C2CCC(NC(c3ccc(C(C)=O)[nH]3)=O)C2)=O)CC(N=[N+]=[N-])C1 Cc1nnc2n1CC(C(=O)NC13CCC1CN(C(=O)CCc1ncc[nH]1)C3)C2 S(=O)(=O)(c1cccnc1N1CN(C)C(=O)C1C)NC(c1cnc(C)s1)C c1(OC)ccnc(C(=O)NCC(O)CCNC(=O)C(O)CN2CCCC2)c1OC c1(C(=O)NC2CN(C(CC)=O)C(CC)(CC)C2)cc2nc[nH]c2cn1 CC1=CCC(C)(C(=O)NCCC(C)NC(c2ncccc2C2CC2)=O)CC1 C=C(C)C(CC(=O)N(C1CCN(C(=O)COC2(C)CCC2)C1)C)OCC CC(C)CC(C(=O)NCC#CC(N1CC(O)C(C2CC2)C1)=O)C(N)=O c1(C(=O)NC2(COC)CCN(C(=O)C(C)CSC)C2)c(N)c(C)cc2c[nH]nc12 C1(CNC)CCCN(C(c2ccc(Br)cc2)=O)C1 Cc1nc2c(o1)CCCC2CC(=O)N1CCCN(C(=O)C(F)C2CCC2)CCC1 C1(NC(COC(C)C)=O)CCC2CN(C(=O)CC3(C(F)(F)F)CC3)CCC2C1 c1(C(=O)OC)csc(C(=O)OCC(=O)NCCCC(F)F)n1 c1(C(=O)NCC2=CCCN(C(c3c(C)noc3N)=O)C2)ccc2nc[nH]c2c1F C1(C(=O)NCCCCC(C)NC(=O)C=CCF)COc2cc(F)ccc2O1 N1(C(CC(=O)OCC)=O)CCC2OCCN(C(c3cc(COC)nn3C)=O)C2C1 CC1CC(CNC(C2CC=CC2)=O)CN1C(=O)CCCn1ccnn1 c1(CC(=O)NCCC2COCCN2C(C2CC2C2CC2)=O)ccccc1[N+](=O)[O-] C(=O)(CCCCCCC1CC1)N1CCCC(NC(C(C)(C(C)C)OC)=O)C1F C#Cc1cccc(C(=O)N(C)Cc2ccc(CNC(=O)CCSC)cc2)c1F N1(C(C(C)C2CCCO2)=O)CCC(CO)(NC(c2nccc(Br)c2O)=O)CC1 C1(C(=O)NCC=C)CN(C)CCN1C(c1ccc(O)nc1)=O N1(CCc2cn(C3(NC(c4c(C)scn4)=O)CC3)nn2)CCCS1(=O)=O C(=O)(C1CCc2cn(CC)nc21)N1CC(C(N)=O)(NC(CCN(C)CC)=O)C1 CC1CN(C(C2CCN(C(=O)CC3CCCN(C)C3)CC2)=O)CCO1 N1(C(CNC(C(C)(C)C)=O)=O)CC2(C(N3CCOCC3CC(N)=O)=O)CC1CO2 n1(CC(N2CC(F)(CNC(C(C)C(C)(F)F)=O)C2)=O)ccc2cc([N+](=O)[O-])ccc12 C(=O)(C(C(C)(C)C)c1ccccc1)NC(CNC(C(=O)NCCOC)=O)C N(C(=NCc1ccc(CC#N)cc1)NC1CCN(C(=O)CCC)C1)C(CC)C C(=O)(C1=COc2ccccc2O1)N1CC(CC(C)NC(c2scc(C)c2)=O)C1 C1(C(N2CCC(CCOC)C2)=O)CC2C=CC1N(C(C1C(C)C1C)=O)C2 N1(C(C(COC)C)=O)CCCN(C(=O)Cn2cc(CN(C)C)nn2)CC1 C(c1ccncn1)=CC(=O)NC1CC(NC(CC2C(OC)CCC2)=O)C1 C1(Cn2cc(-c3ccc(CC)c(F)c3)nn2)CCCCN(C(=O)C2CC2)C1 CC(C(C)(C)C(=O)NC1(C(O)CO)CC1)NC(C1CSCC(=O)N1)=O N1(C(C(C)=CC)=O)CC(N(C(=O)CCC(=O)N(C)C)C)C(C)(C)C1 c1(OC)cccnc1NC(=O)CC=CCNC(=O)C(C)(CO)OC C1(CC(=O)NCC(C)NC(c2cc(C(F)F)on2)=O)CCCS(=O)(=O)C1 C(c1ccc(O)cc1)=CC(N1CCC(NS(=O)(=O)CCc2ccccc2)C(F)C1)=O N1(C(C(C)=C2CC2)=O)CCC(C2(O)CCN(C(c3cc(Cl)ccn3)=O)CC2)CC1 N1(C(C2CCN(C(=O)OCC)CC2)=O)CC2(CCCC2NC(C2CCCO2)=O)C1 N1(C(C=C)=O)CC2(CCN(C(C34CCC(OC)(CC3)OC4)=O)CC2)C1.C(COC)OC CC(CC(=O)c1ccc(Cl)cc1)C(=O)NCC1CCN(C(c2sccc2Cl)=O)C1 CCS(=O)(=O)CC(=O)NC1CCC(C)(CNC(c2coc(-c3ccsc3)c2)=O)C1 C1(NC(c2nccc(OC)c2OC)=O)CN(C(C2C=CCCC2)=O)C2(CCC2)C1 C(C1=NOC2CC12)(c1nnnn1-c1ccc(F)cc1)NCC1(O)CCOC1 c1(C(N2CCC(CNC(C(CC)C#N)=O)C2(C)C)=O)cc(F)c(C)cc1F c1(N2CCC(CC)(CO)CC2)ccc([N+](=O)[O-])cc1CNC(=O)C(C)CCCOC C(=O)(C1=NNC(C(F)(F)F)C1)NC1CCC(NC(C(CCC)OCC)=O)CC1 C1(OCC(=O)Nc2cccc(OC)c2)CCC(C)N(C(=O)C=CC(C)(C)C)C1 c1(NC(c2cn(CCN(C)C)nn2)=O)nc2c(s1)CCc1cc(Cl)ccc1-2 C12(C(N3CC(=O)NC3=O)C3CCC3)CCC(CC1n1cc(-c3c[nH]nc3F)nn1)C2 CC(C)(C#N)CCCC(=O)N1CCOC(CC(=O)NCCCCN(C)CCO)C1 C1(NC(c2ccccc2)=O)CCCC1NC(=O)Nc1cc(SC(F)(F)F)c[nH]1 C1(C2(C(=O)NCC(C3CC3)NC(C3CC(C)(C)C3)=O)CC2)(COC)CC1(F)F N1(C(c2cc(C)oc2C)=O)CC2CN(C(=O)C=C3CCN(C)C3)CC12 C(C(CC(C)C)NC(c1cc(C(C)(F)F)on1)=O)NC(CCCOCCOC)=O c1(C(=O)NCC(CC)NC(C2(CC)CCOCC2)=O)ccc(OC(F)F)nc1 c1(OC)ccc(OC)c(C(=O)N(CCCCNC(c2cn(C)nc2C)=O)C)c1N C1(NC(CC(CCC)O)=O)CCCC12CN(C(c1sc(C)nc1CC)=O)C2 C(=O)(C1CCCc2cncn21)NC(COC(C)(C)C)C(C)(C)C O=C1CC(=O)NC(C(N2CC(N3CC4(CN(C(=O)C5CC5)C4)C3)C(F)(F)C2)=O)C1 C12(CNC(C(C)Oc3ccccc3F)=O)CCCC1N(C(C1CCCC1)=O)CC2 c1(C(N(CC(CC)NC(C2CSCCS2)=O)C)=O)ccc(C)nc1 C1(NC(C(C(C)(C)O)F)=O)(CNC(=O)CCSC(F)(F)F)CCC(F)(F)CC1 Cn1ncc(C(=O)NC2CN(C(C3(C)CC4CC4C3)=O)C2)c1Br N1(C(CC(C)NC(N)=O)=O)CCC2(CCC(CNC(=O)CCCF)C2)CC1 C(=O)(C(C(C)C)OC(C)=O)N1CCC(CCC(=O)N(CCC#C)C2CC2)C1 C1(C2CN(C(C3(N(C)C)CCC3)=O)C2)(NC(C(C)c2cncs2)=O)CC1 C(C(C)(O)C(=O)N(CCC(C)NC(C1CC(Cc2ccccc2F)C1)=O)C)OC N1(C(C(CCC)N(C)C)=O)CC(C(=O)NCC(C)CC)CC(F)(F)C1 C1(C(=O)NC2(CCC)CCCN(C(=O)C(F)=C3CCC3)C2)CC2CCC(C1)C2O c1(C(=O)NCc2cccc(NC(CCCOCC)=O)c2)ncc(F)cc1F c1(CC)nccc(=NC(=O)CC2CN(S(=O)(=O)c3ccc(Cl)cc3C)C2)[nH]1 C1(CCNC(c2cc(CC)[nH]n2)=O)CN(C(c2ccncc2N)=O)CC(C)O1 c1(C(=O)N(C(C)CN(CC(=O)O)C)C)cc([N+](=O)[O-])ccc1Br c1(CC(C(=O)NC(CC)(C)CNC(=O)C(C)(C)OC)C)ccc([N+](=O)[O-])cc1 N1(C(C(CC=CC)C)=O)CC(CCC2CCCN2C(=O)CCC2(C)CC2)C2(CC2)C1 CC1Cc2cc(C(N3C(C)CC3(C)C)C(=O)NCc3ccccc3)ccc2O1 c1(CC(=O)NCCN(C(C2CC(C)(C)O2)=O)C2CC2)ccc2[nH]ccc2c1 N1(C(c2c(NC)nccc2)=O)CCC2(CC1)CC2C(=O)N(CCCN(C)C)C C1(CNC(C(COC(C)C)NC(c2occc2C2CC2)=O)=O)CCC=CCCC1 CC(C)C(F)(F)CC(=O)NC1(CNC(=O)C(Cc2cnc[nH]2)N(C)C)CCC1 N1(C(CCCN(C)C)=O)CC2CCC2(CCNC(=O)CSc2nncn2C)C1 CCC(C)(C)CCCC(=O)NCC1(F)CCCN(C(=O)CSC)CC1 Cc1cccc(O)c1C(=O)NC(CNC(=O)Cc1n[nH]cc1Br)C(C)C(C)C C1(NC(Cc2c(C)cccc2)=O)CN(C(C2CC(F)C2)=O)CC(C)(C)C1 c1(C(=O)NC2CCCN(C(c3c(C)snn3)=O)CC2)c(Cl)cc(Cl)nc1N C(=O)(CCC(=O)NCCC1CC(NC(C2(C)CC(C#N)C2)=O)C1)N(CC)CC c1(C(=O)NC2C(NC(C=NOC)=O)COC2)nc(C)c(C)s1 Cc1c(C(N2CCC(C)C2CNC(=O)COCCc2cccs2)=O)cccc1O c1(CSCC(=O)NCC(CC)N(C(=O)C(O)C2CC2)C)cccnc1 C=C(C)CCCC(=O)NCCC1(O)CCCN(C(=O)Cn2cc(C3CC3)nn2)C1 c1(CC)cccnc1C(=O)NCC12CC(NC(c3c[nH]c(=S)cn3)=O)(C1)C2 C(C1CCc2nccn21)NC(C12N(C(c3c(CC)ncnc3)=O)CC(C1)C2)=O c1(NC(=O)COc2ccsn2)ccnc(N2CCOCC2)c1Br n1(CC(C)O)cc(C(=O)NCC(O)CCNC(c2cccnc2C)=O)ccc1=O Cc1cc(C(=O)NC2CCN(C(C3C(C)C3C)=O)CC2F)c2[nH]cnc2c1 c1(CCC)c(C(=O)N(CCC(C)NC(C2(C)CC2)=O)C)[nH]c(C)c1C(C)=O c1(OC)ccc(C(=O)NC2CC(NC(c3n[nH]c(C)c3C)=O)C2)cc1N c1(C(N2C(CNC(C3CCC(C#C)CC3)=O)CC2)=O)cc(F)cc2cnccc12 C1(C(=O)NCC(C2CC2)N(C)C(c2ccn(C(F)(F)F)n2)=O)(COC)C=CCC1 C1(N(C(=O)C#CC2CC2)C)CN(C(c2c(Cl)noc2C)=O)CC12CC2 O=C(N=S1(=O)CCCC1)c1ccccc1Br C(C(F)C(=O)N)N(CCC)C.n1(CC2(C(=O)NC3C(COC)C3)CC2)ccnn1 C1(CC)CCC(C(=O)N(C)CCOCCN(C(=O)CC2CC=CCN2C)C)CC1 C(CCNC(=O)CN(C1CCC1)C)(C(C)C)NC(C(C)=CC)=O Cn1[nH]c(C(=O)NC(C)(CNC(=O)Cn2cnnc2)Cn2cccn2)nc1=O S(=O)(=O)(c1ccc(N2C3CCC2CC3)c(Br)c1)NCC(N1CCCC1C)C C12(C(N3C(c4c(C(=O)OC)nco4)CCCC3)=O)CCCCC1CNC2 C(=O)(CC1=CCCCC1)NCC1(C)CC12CCNCC2 CC(CC(=O)N1CCC2(CC2C(=O)NCCC(C)N(C)C)C1)C(C)(C)C c1(CNC(N2CCC(N3CCNS3(=O)=O)CC2)=O)cc(Cl)cc(Br)c1O c1(CC)cccnc1NC(C1CCC(F)(CNC(=O)CCCC2CCCC2)C1)=O C(CC(=O)NC1CC12CC2)N(C(c1nc[nH]n1)=O)CC c1(C(N2CC(NC(c3cc(CC)n(C)n3)=O)C(C)C2)=O)nccn2cnnc12 CC1CC(NC(=O)CCNC(C2CCOCC2)=O)CN1C(C1CCCCCC1)=O N1(CC(N2CCC(O)(CNC(C(CC#C)C)=O)C2)=O)C(=O)C(=O)N(C)C1=O c1(C(=O)NC(C)CCNC(=O)CNC(C2CCCC2)=O)cncn1C N1(C(Cc2cc(C)sc2)=O)CCc2sc(CNC(C3CC(O)C(F)C3)=O)nc2C1 N1(C(CS(CC)=O)=O)CCC(CNc2nnccc2C#N)C(F)(F)CC1 C1(CNC(c2ccoc2Cl)=O)CCC2(CN(C(=O)Cc3cocn3)C2)O1 Cc1csc(C(N2CC3CC3(NC(=O)CC3(C)CC3(Cl)Cl)C2)=O)c1C N1(C(c2scc(C(N)=O)c2)=O)CCN(C(=O)CNS(=O)(=O)CC)CC1CC(C)(C)C C(=O)(CCC(=O)NC=O)N(C1C2CN(C(N(C(C)C)C)=O)CC12)C.[nH]1cc(Cl)cn1 c1(OC2(C(=O)NC(C(C)NC(C(C)N3CCC3)=O)CO)CC2)ccc(Cl)cc1 c1(C(N2C(CNC(C(C=C)(C)O)=O)(COC)CCC2)=O)cn2c(n1)CCC(C)C2 c1(OC)cncnc1C(N1CC(NC(=O)C(C2CC2)OC)C1)=O c1(C(N2CC(O)(CNC(CNS(N)(=O)=O)=O)C2)=O)ccnc2c1CCC2 CCCCC(CNC(c1cccc(C(C)(C)C)n1)=O)NC(C1C(C)C1C)=O N(C1CCOc2ccccc21)C(C1N(C(CCCC(=C)C)=O)CC(O)C1)=O c1(OC)cc[nH]c(=NCCC2CCCN(C(=O)CC(=O)NCC)C2)n1 C1(C)(CC)CN(C(=O)C(N(CCCSC)CC)C2CC2)CCO1 CC1CC(C)N(C(c2coc3c2CSC3)=O)CCN1C(c1ccon1)=O CCCCC(CCC)NC(=O)CC(CNC(=O)CCn1cnc(=N)[nH]1)C1CCC1 C1(C(N2CCC2(C)CC(=O)Nc2cnoc2)=O)(OCC)CCCC1 c1(NC(C)=O)cccc(F)c1C(N1CC(CNC(=O)CSCc2csc(C)n2)C1)=O C(=O)(CC(O)C(=O)NC(C)CN(C)C(c1nc[nH]c1C(C)(C)C)=O)OCC C(=O)(C1CC(=O)Nc2c(F)cccc21)N1CCCC(NC(=O)COCC2CC2)C1 C(C1=NOC2CN(C(=O)Cn3cc(C4CC4)nn3)CC12)NC(c1c(C)ccs1)=O c1(C(N(CC(=O)NC(C(O)CO)C2CC2)CC#C)=O)ccc(F)c(O)c1 c1(-c2c(C(C)Nc3nccc4ncncc34)n(C)cn2)cnc2ccccc2c1 N1(C(CC2CCC(C)(C)O2)=O)CCN(C(c2coc(CC3CC3)n2)=O)C(CO)C1 c1(OCCC)cccnc1NC(c1ccc(CNC(=O)COC2CCC2)cc1)=O C(C(CC(F)(F)F)NC(c1occc1CC)=O)NC(c1c(CC)nn(C)c1)=O N1(C(=O)NC(c2ccc(OC(F)(F)F)cc2)C)CCC2(C1)COC(=O)N2 c1(NC)ccc(C(N2CCCCC2C(C)NC(=O)CN=[N+]=[N-])=O)cc1 C1(C(N(CCCNC(=O)CC2(C)CCOC2)C)=O)CC2(CCC2O)C1 C1(NC(C(=O)NCC2CC3CCC3C2)=O)CCN(c2ccc(Br)nn2)CC1 c1(C(N2C(CC)CN(C(C3=CN=CNN3C)=O)CC2)=O)ncnc2cc[nH]c12 N1(C(COCCCOC)=O)CCC2(CC1)CC2CNC(=O)Cc1ccnn1C c1(C(=O)NC2C(NC(C3N(C)CC(C)(C)C3)=O)CC2)ccc2oncc2c1 Cc1cccc(OCC(=O)NCC(CNC(C2(C)CC2(F)F)=O)S(C)(=O)=O)c1C N1(C(C(C2CCCOC2)C)=O)CC(n2cc(CCNC(N)=O)nn2)CCC1(C)C N1(C(C2C(=C)C2)=O)CCC(F)CC1C(=O)NOCCCC C1(C(=O)NCCCc2cccc(O)n2)CCc2nc[nH]c2C1 c1(C(=O)NC(C(CO)NC(c2ccn(CCOC)n2)=O)C)cccc2c1CCO2 N1(C(C(C)N(C(C2(COC)COC2)=O)C)=O)CCCC2(CC2)C1 C(CCCCCC(=O)NCC(C)OCCO)n1cc(-c2nccc(C)c2)nn1 CCC(C)C(C(=O)NCC1(F)CCC1)NC(=O)CCC(=O)N(C)C Cc1cnc(C(=O)NCC2CC2CNC(=O)Cc2cc(C)cc(C)c2)c(F)c1 C1(=CCNC(=O)Cn2cncn2)CCN(C(c2ccc(F)nc2)=O)CC1 C(CCNC(=O)CCN(C)CCO)(C(=O)NCc1cnn(C)c1O)OC N1(C(c2c(C)n(C)nn2)=O)CCCC(C)(C(N2CC(c3cnccn3)C2)=O)C1 n1(C2CN(C(C3(CCC=C)CC3)=O)C2)cc(C2CCN(C)C2)nn1 Cc1cc(C(N2CCN(C(C3(F)CCC3)=O)CC2C(C)C)=O)nc(O)c1 c1(C(N2CC(O)(C(C)NC(C3C(C)CC(C)O3)=O)C2)=O)cc([N+](=O)[O-])cnc1O c1(OC)c(F)cc(C(=O)NC(C)C(C)NC(=O)C(=O)NCC2CC2)c(N)c1F.C c1(OC)ccc(N)c(C(N2CC=CC2CNC(=O)Cc2ccnnc2O)=O)c1 C(C)(CCC(C)C)SC.N12CCC(C1)OCC(=O)NC(C1CC1)C2=O Cc1cc2[nH]c(C(N3CCC(O)(C(C)NC(c4occ(C)c4C)=O)C3)=O)cc2s1 C1(C(=O)NCCC(C)NC(=O)CC2(CS(C)(=O)=O)CC2)Cc2nncn2C1 CC1(C(=O)NCCCCl)CN(C(c2ccc(-c3ccncc3)o2)=O)C1 C(=O)(CCC(=O)N1CC2CC1C2NC(=O)C(C)c1cccs1)OC CC(C)(C)C(O)Cc1cn(CCC2CC(NC(C3CCC(=O)N3)=O)C2)nn1 C1(CNC(c2ncccc2CO)=O)CCCN(C(=O)C(CC2CC2)CC2CC2)C1 C(=O)(CC(C)CC(C)(C)C)NC(CC(=C)Cl)C(=O)N1CCC2C(OC)CC12 C12(C(=O)NC(C#C)C(C)(C)C)C(NC(=O)CC3CCCC(=O)N3)C3CC1C2C3 C1(C)(CNC(C(C)C2CC2)=O)CC(F)(F)CN1C(=O)Cc1ccc(C#N)cc1 C(=O)(C(C)(NC(=O)C1CC1)SC)N(CCOCCO)CC CCC(C(=O)NCC1CCN1CC)NC(=O)CC1(CC)CCC1 c1(SCC)n[nH]c(=NC(=O)OC)s1.C1(OC)CC2C1(C)C(CCC)C(=O)N2 CC(CC(=O)NCC(C)(C)CC(=O)NC1CCCC(C2CC2)C1)C(F)(F)F c1(OC)nc(C)c(C)cc1C(N1CCN(C(c2cscc2C)=O)C(C)C1)=O C1(CC#C)CN(C(c2csc(CNC(=O)C(C)CSC(F)(F)F)c2)=O)CCO1 C12(CNC(C3(C)CCN(C)C3=O)=O)CCC(CN(C(=O)CC(F)(F)F)C1)C2 CC(CC(=O)N1CC(CCCCNC(=O)Cn2ccc(C3CC3)n2)C1)CC(F)(F)F c1(CN2CC(F)CC(C(=O)NCCOCC#C)C2)cc([N+](=O)[O-])ccc1F CC1CCC(C(N2CC(NC(c3cccc(Cl)c3)=O)C(O)C2)=O)CC1 CC1CCCC1(C(N1CCC1)=O)NC(=O)CN(C)C1CC1.n1(CC2CC2)ccnn1 N1(C(c2cc(CCC)n[nH]2)=O)CC2CCCCC2(NC(=O)C(C)O)C1 Cc1cc(Br)c(Cl)cc1-c1cn(C2(C#N)CCN(c3ccc(Br)c(C)n3)C2)nn1 CC(C)C1=NOC(C(=O)NC23CC(NC(=O)Cc4ccc(CO)cc4)(C2)C3)C1 c1(C(=O)NC2(C3CCN(C(=O)CSC(F)F)C3)CC2)cc2ccccc2oc1=O C1(CC)(NC(C2CC(O)CN2C)=O)CC(C)(C)C1 C1(N(C(c2ccn(C)c2)C(=O)NC(C)C)C)CCCCC1 c1(C(=O)NC(COC)C2CC2)nn(C)c2c1CN(C(=O)C(C)(C)N(C)C)CC2 c1(CC)nc(C)ccc1NC(=O)CC(CC1CC1)NC(=O)C(C)C(F)F Cc1ccc2sc(C(N3CCC(C)C(CNc4ncccn4)C3)=O)c(C)c2c1 c1(NC23CC2CNC3)ccc([N+](=O)[O-])cn1.c1(SCC)ccccc1C(OCOC)=O C(=O)(C1Cc2ccccc21)NCC1(C)CC(F)(F)CN1C(c1ncc(F)cn1)=O N1(C(C#CC(C)C)=O)CC(=O)NCC1C(=O)NCC1(O)CCOC1 N1(C(c2c(C)cccc2F)=O)CC2CCC(NC(c3cnn(C)n3)=O)CC2C1 C(=O)(CCCCCCCCCC1CC1)NCC(CNC(CC(CC)CC)=O)CO Cc1cnc(CC2CCCN2C(C2CC2[N+](=O)[O-])=O)nc1-c1cn(C(C)C)nn1 c1(N(C(c2nc(C)on2)C)C(C2CC3CNC2C3)=O)ccccc1Cl C#CC1CCCN(C(c2coc(CNC(c3ncncc3Cl)=O)c2)=O)C1 N1(C(c2c(C)cccc2O)=O)CC(C2CN(C(C3CC3(C)C(F)F)=O)C2)C1 c1(CC(N2CCC(OCCNC(C3CC(=C4CC4)C3)=O)C2)=O)ccnc(O)c1 C(=O)(CCCC(CC)CC)NCC1C(C(N(CCCC=C)C)=O)CCCC1 C1(C(N2CC(C)(C)C2Cn2cc(C3CC4C=CC3C4)nn2)=O)(CC)CCNC1=O c1(C(=O)NCCC(C)OC)ccc(N2CCN(C(C3CC(=O)C3)=O)CC2)cc1 C1(N(C(C(CCC)NC(=O)C(CC2CC2)OC)=O)C)CN2CCC1CC2 C1(CC(=O)N(CCCN(C)C(c2ccn(CC(F)F)n2)=O)C)CC2CCC1C2 CCCC(CCCNC(=O)C(C)C1(O)CCC1)NC(=O)CN(C)CCOC CCC(CC(=O)NCC(CC1CC1)C(=O)NCc1cn(C(C)C)nn1)C(C)(C)C c1(NC2C(CNC(C(C)c3ccco3)=O)CCCC2)ncc(Br)c(O)n1 C=CCCC(F)(F)C(=O)NCC12CCC1CN(C(=O)Cn1ccc(O)nc1=O)C2 CCC(C)(C#N)C(=O)N1CC(NC(C2(N3CCCC3)CCC2)=O)CC(F)C1 N1(C(C(=O)NCCCC)C(C2CCC2)C2CCC2)CCC(C2CC2(F)F)C1 c1(-c2cn(OCC3CCC(F)CC3)nn2)c(F)cc(Cl)cc1F N1(CC)CCC2(CC2)CC1CNCc1cn(-c2ccccc2SC)nn1 c1(C(N(C2CN(C(C3CC(F)C3)=O)C2)C)=O)c(C(F)(F)F)cccc1F Cc1cc(Cl)c(C(=O)NCC2(CNC(=O)C(C)C#N)CC(F)(F)C2)cc1F C1(NC(c2ncccc2Cl)=O)CN(C(c2cc(O)nc(O)n2)=O)CC(F)(F)C1 C(=O)(CC(C=C)CCC)N1CCN(C(CCCOCC=C)=O)CC1CCC C(=O)(C1=CCCSC1)N1CC(CC(=O)NCC2(C)C(C)(C)C2)OCC1 C(=O)(C(CC)(CO)OC)NCC(CC)NC(=O)CCOC1COC1 CC(=O)C(C)(C)CC(=O)N1CCCC(C(C)(C)C(=O)NCCCc2cc[nH]n2)C1 C(=O)(C1Cc2ccc(Cl)cc21)NCCCC(C)(C)O c1(C(=O)NCC(C2CCN(C(=O)CO)C2)C)cc(S(=O)(=O)N2CCSCC2)c[nH]1 c1(NC(N2CCNCC2c2ccccc2Cl)=O)c(C(F)(F)F)ccnc1Cl C(CO)(CC(C)(C)C)NC(C(CCC)NC(C1(N(C)C)CC1)=O)=O Cc1cc(C(=O)N(C(C)C)C(C2CC2C2CCCO2)=O)n(C2CCC2)n1 N1(C(C(=O)NC(C(C)(C)C)C(=O)O)=O)CCc2ccc(Br)cc2C1 N1(C(c2ccc(C#C)c(F)c2)=O)CC2CC(C)N(C(=O)Cc3cncnc3)C2C1 C1(CC)CCC(C(=O)Nc2cncc(C(=O)NCCC3CC4CCC3C4)c2)CC1 C1CCCCCN=C2NC(=NC(=N)N2)N1CC.c1(C(CF)SC)ccccc1 C1(NC(=O)C=Cc2ccsc2)CCC2(CC1)CCN(C(=O)COc1ccsc1)C2 C1(N(C(C=C(C)C)=O)C)C2CN(C(c3occc3Cl)=O)CC12 C12(NC(CC(C(C)C)O)=O)CC3CCC(C1C2)N3C(C1CC2(C1)CC(C)(C)C2)=O NC(=O)CCCCC(=O)N1CCN(CCCNC(=O)C(C(=O)OC)C(F)(F)F)CC1 N1(C(c2ccc(Br)cn2)C(=O)NC)CCC(F)(F)C(CC(=O)OC(C)(C)C)C1 CCC(C(=O)NCC1(O)CN(C(c2cccc(SC(C)C)c2)=O)C1)n1ccnc1 c1(SC)ccsc1C(=O)NCC(C)CNC(C1(Cc2ccccc2)CC1(F)F)=O C1(NC(CSC)=O)C2CCCN(Cc3ccnn3C3CCC3)C2C1(C)C c1(C(N2C(C)CN(C(c3c(CC)scc3)=O)C(C)C2)=O)cc([N+](=O)[O-])cc(C)n1 c1(CC(N2CCC(COC)(NC(C3CS(=O)(=O)C3)=O)C2)=O)ccc(Cl)nc1C c1(C(c2nnnn2C2CCOC2)NCC2CC(=C)C2)cc(C)c(C)c(Br)c1 c1(C(N2C(C)CC(NC(=O)C(C)(C)CN(C)C)C2)=O)cc(Cl)c(F)c(Cl)c1 C1(C(=O)NCc2cc(C(=O)NCC(C=C)O)n[nH]2)C2CC3C(C2=O)C13 Cc1cc(C(=O)NC(C(=O)NCC(CO)C2CC2)C2(C)CC2)ccc1C#N C(=O)(C(C)CC(C)(C)C)NCC=CC(=O)Nc1c(C)cccc1C C1(C(N2CC(NC(=O)C(F)(F)C3CCCCC3)C(O)C2)=O)CC2CCC1CC2 c1(CN(C)C(=O)NC(CC2CC2)C2CC2)n[nH]c(=N)s1 C1(CNC(C2(OC)CCCC2)=O)C2CN(C(=O)C(F)(F)CO)CC12 C(=O)(C(F)CCC(C)(C)C)NCCCC(C)NC(c1cc(C2(C)COC2)no1)=O C1(CNC(C=CC(CC)C)=O)CC2(CC(NC(c3ccc(F)c(F)c3)=O)C2)C1 N1(C(CCOCC(C)C)=O)CC2CCCC(NC(=O)C#CC3CCCO3)(C2)C1 CC1CC(NC(c2cncnc2C2CC2)=O)CN1C(=O)C=Cc1cccn1C N1(C(C2(COC)CC2)=O)CCC(C(C)NC(c2cnc[nH]2)=O)CC1 c1(C(=O)NC(CNC(C2CC(S(C)(=O)=O)C2)=O)C2CC2)cccc2ccoc12 C1(CNC(CCc2onc(C)n2)=O)CN(C(c2ncn(C(C)(C)C)n2)=O)CC1C CC(C)(C)C(=O)c1ccc(C(=O)NCCc2cn(C(C)(C)C(=O)O)nn2)s1 C1(NC(CC(=O)NCC#C)=O)CCCC(C(=O)NC(c2ncc(C)s2)C)C1 c1(SC)nc(N(CCCN(C(c2cccc(C)c2)=O)C2CC2)C)cc(C)n1 C(=O)(C(C)(C)Cc1ccc(O)cc1)NCC(C)NC(=O)C(F)C1CCC1 C1(C(N2CCC(C(C)NC(C(C)C)=O)CC2)=O)CCC2C(C1)C2(F)F CC(CC(C)(C)C)C(=O)NCC(CNC(=O)C(C1(O)CCOCC1)(F)F)CO C1(CNC(c2n(C)cnc2)=O)CN(C(c2ncccc2Cl)=O)C2CCCC2O1 C1(NC(C(C)OC)=O)CCC(C(C)(O)CNC(=O)Cc2cccc(SC)c2)CC1 c1(C(=O)NC(CNC(COCC)=O)CC)nn(C)cc1SC Cc1ccc(C)n1CC(=O)N(C)CCC1CCCCN1C(C1CCC(=O)N1C)=O c1(C(=O)NC2CCN(C(=O)NCC3(SC)CCC3)C2)cc(OC(F)F)ccc1F CC1(C)CN(C(=O)CCCCC2CC2)CC1C(=O)NCCn1cnnc1 C(=O)(CC(CC)CC)NC(CCN(C(c1nnn(COCC)c1N)=O)CC)C.C1CC1 C1(CNC(c2cn(C)nn2)=O)CN(C(c2n[nH]c3c2CCC3)=O)CC12CC2 CC1CCN(C(c2cc(O)ccc2F)=O)CCN1C(=O)C(C)c1ccco1 CN1CC2CCC1CN(C(=O)C(c1ccco1)NC(c1ccc(C#N)s1)=O)C2 C1(NC(N(C)C)=O)CCCC2CCN(C(N3CCC(CO)CC3)=O)CC12 CC(C)C(C)C(=O)NC1CCOC1C(=O)NC(c1cscn1)C C1(C(N2CCN(CC#C)CC2)=O)CC(C)(C)OC1(C)C.N12CC(C1)S(C)(CC)CC2=O C1(NC(c2c(C)csc2)=O)CCC(C)(CNC(=O)C(=O)NC2CCCCC2)CC1 C(=O)(C(CC(F)F)N(C(=O)Cc1ccsc1C)C)NCCc1onc(C)n1 c1(CN2CCC(CNC(c3cc4ccccn4n3)=O)C2)csc2ccc(Cl)cc12 NC1C=CC(CCSC2CCNC2)C1 C1(NC(C=C(C)C(F)F)=O)CCCCC1CNC(=O)CCCc1csc(C)n1 C=C(C)C(C)(O)C(=O)NC1CN(C(=O)C(F)(F)CO)CC1O N1(C(CC(C)C)=O)CCC(C)C(NC(=O)CCC2CCCC2)C1 c1(C(=O)NCCNC(C(c2ccc(Cl)cc2)N(C)C)=O)ccc(O)c(C(N)=O)c1 c1(C(N2C(CNC(c3cc(C)no3)=O)CCC2)=O)ccc(CF)cc1 c1(NCCCCC2CN(C(c3nccc(OCCC)n3)=O)C2)cccc(Cl)c1F CC1CN(C(=O)N(c2cccc(C(C)(C)C)c2)C)CCC1C(=O)O c1(C(=O)NCC23N(C(C(C=C=C)C)=O)C(CC2)CC3)cccc2snnc12 N1(C(CCCOCC)=O)CCCC(COC)(NC(C2(N3CCC3)CCCC2)=O)C1 c1(C(=O)NC2(CO)CCN(C(C3C(=C)C3)=O)CC2)cc(F)c(N(C)C)c(F)c1 c1(CC)cc(C(=O)NCC(C)(C)NC(C2(C)CCCO2)=O)oc1CC c1(C(N2C3C(NC(C(C)OC)=O)CC(C3)C2)=O)cccc2cccc(O)c12 C(=O)(C1=CCCC1(C)C)NC1CCC(CNC(c2n(CC)nnc2)=O)C1 n1(CC)cc(C(=O)NC2CCN(C(=O)Cn3cc(CO)nn3)CC2)c(C2CC2)n1 N1(CCCCCNC(C(C2CC2)OCC)=O)CCN(C(C2(CO)COC2)=O)CC1 CCC(O)C(F)(F)C(=O)NCCN(C(=O)CCc1cc(C)nc(C)c1)CC c1(OC)cc(CNC2CCCC2C(N2CCC2CO)=O)cc(C(F)(F)F)c1I C12(C(=O)NC3(C)CC(O)C3)C(NS(C)(=O)=O)C3CC1C2C3 N1(C(C2C(C)OCCO2)=O)CCC(C(=O)NCCCOCCCO)=C(F)C1 CC1CN(C(c2cc(C3CC3)ns2)=O)CCN1C(C1CC(=O)C1(C)C)=O N1(NC(=O)CC2CC(NC(C3CC(C(=O)O)(CCF)C3)=O)C2)CSCCSC1 C(=O)(C1=NOC2(CCOC2)C1)N1CCCN(N(C(CC2CCN(C)C2)=O)C)CC1 N1(C(c2c(NC)cncc2)=O)CC(C)C(NC(c2cnn(C3CC3)c2)=O)C(C)C1 N1(C(C(C=CC)O)=O)CCC(C)(CNC(c2cn[nH]c2)=O)CC1 CCC(N=c1cc(C)[nH]c(=NCCCc2cn[nH]c2)[nH]1)c1ccc(Cl)s1 c1(C(N2CCC(CC)C2CNC(C2CCCC2(C)C)=O)=O)ccc(S(N)(=O)=O)s1 c1(C(=O)NC2CCN(C(Cn3c(C)csc3=O)=O)C2C)c(C)nn(C)c1C C1(CNC(c2n[nH]c(C)c2C)=O)CCCCN(C(c2c[nH]c(C(C)(C)C)n2)=O)C1 c1(C(=O)NCC2CN(C(=O)CCCCF)CCC2(F)F)cnc2c(n1)CCCC2 Cc1cc(C(N2CCOC(c3csc(C4CC4)n3)C2)C(=O)NC2CC2)cc(Br)c1C N1(C(C(C2CC2)OCC)=O)CCC(O)(CN(C(=O)Cc2ccc(C)cc2)C)C1 N1(C(COC2(C)CCCC2)=O)CCC(NC(=O)CSc2cccc(Cl)c2)CC1 C1(NC(CCN(C(c2c(C)nco2)=O)C)=O)CC(C)N(C2CC2)C1 CC1OCCN(C(C2CCC(=O)CC(CO)C2)=O)C1C(N1CCC2(CC1)N=N2)=O c1(N(C(=O)C(=O)NC(c2ccc(F)cc2F)COC)CC)ccc(F)c(OC)c1 c1(CC(=O)NC(C2CN(C(COC(CC(C)C)C)=O)C2)C)c[nH]c(=N)nc1O c1(NC(N(CCCC)C)=O)cc(S(=O)(=O)N(C)C(C)C)ccc1Cl O=C(C1=CCCSC1)NCC1(O)CCCN(C(=O)Cc2ccc(O)cc2F)C1 CC1(N(C)C)CCCN(c2ccnc(NCc3csc(Br)c3)n2)C1 C1(CC=C)(NC(=O)CC2CCC(C)CO2)CCN(c2nnc(C(C)C)s2)CC1 c1(OCC)ccc(Cl)nc1C(=O)NCC(C)CN(C)C(c1nnc(C2CC2)o1)=O CC1(O)CCN(CC(=O)NCC2C3CN(C(C4(F)CC=CCC4)=O)CC23)C1 C1(C(=O)NC2(CN(C)C(c3sccc3F)=O)CC2)CC2(CCC2)CCO1 C(=O)(C(C(C1CCOC1)OC)N(C1CC(O)CCO1)C)NCC C1(C(=O)NC2CC(NC(C(CCOC)C)=O)C2)CCC(=O)N(C2CC2)C1 N1(C(c2c(C#N)cccc2)=O)CCCC2CN(C(c3cncnc3)=O)CCCC12 CC(C)(C(=O)N1CCN(C(C2CCN2S(C)(=O)=O)=O)CC1CCO)C(N)=O c1(NC(=O)C(N)C2CCCC2)cc(C(N2CCCC2)C#N)cc([N+](=O)[O-])c1 C1(N(C(C(CC)SC)=O)C)CN(C(c2ccnc(OCC3CC3)c2)=O)CC1C c1(C(=O)NCC2CCCC(NC(c3cnsc3)=O)C2)n[nH]c2c1CCOC2 C(=O)(C1=CCCSC1)NCCCC1(NC(=O)CC2CCCCC2)CC1 c1(CC)ncc(C(=O)NCC2CC3CCC2N3C(c2occc2C)=O)c(O)n1 C(CC(C)C)(C(=O)N(CC(C)COCC)C)NC(C(CC#C)C1CC1)=O c1(C(=O)OCC)cccc(CN(CC(N2CCCC3CC23)=O)C)c1 N1(C(c2c(C)ccc(OC)c2)C(=O)NC)CCCC2C1CCN2C C1(NC(C(CC)(F)F)=O)CCN(C(=O)C(C)CCOC)CC1O N1(C(C(C2(C(F)(F)F)CCCC2)C)=O)CCCN(C(=O)C(C)(O)C2CCC2)CC1 N1(C(c2cccc(CC)n2)=O)CC2CCN(C(c3cc(O)cc(O)n3)=O)C2C1 c1(C(C(=O)NC(C)C(C)NC(=O)COC(C)(C)C)N(C)C)cccnc1 C(CC(C(=O)NC(C(F)(F)F)C1CC1)NC(c1csc(C)c1C)=O)=CC c1(C(N2CC(F)(CNC(CN(S(CC)(=O)=O)C)=O)C2)=O)cc(C)c(C)cn1 N(C1CCc2c(F)cc(F)cc21)C(C1CN(C(c2cc(I)c(F)cc2Cl)=O)C1)=O C1(NC(CCn2ccc(C)n2)=O)CN(C(C2CCCN(C)C2)=O)CCC1O c1(NCC(C)(C)NC(c2c(OC)cc(C)cc2)=O)ncc(C#N)c2ccsc12 N1(C(CC)=O)CCC(C(=O)N(c2cnc3ncnn3c2)CC)CC1(C)C CCC(CN(C(=O)CC1CC(SC)C1)C)NC(=O)COC(F)(F)F Cc1cnc2cc(C(N3CCCC(N(CCO)CC4CCC4(C)C)C3)=O)nn2c1 c1(NS(C)(=O)=O)cnc(CCN2CC(CN(C(C3(C(=O)OC)CC3)=O)C)C2)nc1C C1(NC(CCOCCNC(C(CCCOC)C)=O)=O)CN2CCC1(C)CC2 C1(C(=O)NCC(CC)NC(C23CCC(CC2=O)C3)=O)CC2CCCC2C1 C1(CCNC(CC2(COC)CC2)=O)CN(C(C2CCC3CC23)=O)CCCO1 C1(CC=C)(C(=O)NCCC2(CNC(=O)CC(C)n3cccn3)CC2)CCCO1 CC(C)(C(=O)NC1CCc2nn[nH]c2C1)C1=CCN(C(=O)C=CCN2CCCC2)C1 c1(C(=O)NC(CNC(C(C)N(C2CCCCC2)C)=O)C)n[nH]c2ccc(F)cc12 c1(C(=O)NCC2C(NCc3cn(C)nc3)CCC2)cnccc1CC(F)(F)F C(=O)(C1=NOC(C)C1)NC1(C)CCN(Cc2ccc(COC(C)C(=O)NC)o2)C1 CCCCC(C(=O)NC1CCCN(C(=O)CSCCC(F)(F)F)C1)C(C)C C1(NC(C=COCC)=O)CC2(CCN(C(c3ccc(OC)c(C(C)C)c3)=O)C2)C1 c1(-c2nc(C(C3CC3)OC)nn2C2CCS(=O)(=O)C2)c[nH]c(=O)c2ccnn12 N1(C(CCCC#C)=O)CCC2(CC1)CCN(C(C1(O)CCSC1)=O)CC2 N1(C(c2ccc(OC)c(C)c2)C(=O)NCC)CCC(F)(F)C(O)C1 c1(C(N2CCC(CNC(C(CC)Sc3nccs3)=O)CC2)=O)cn(C)c(=O)cn1 C1(OC)CN2CC1C1CCCN21.C(=O)CN(C)CCOCCO.C1(C=O)CCO1 C=CCCCC(c1nnnn1C1CC1)NC1CCCCC1C(=O)NCCSC Cn1cncc(C(N2CC(C(N)=O)(CNC(=O)CC3(C)NC(=O)NC3=O)C2)=O)c1=O N1(CC(=O)N(C2CCC(NC(=O)COCCCF)CC2)C)CC2C=CC1C2 N1(C(C=C(CCC)C)=O)CC2(CC(NC(=O)C(C)(C)C(C)O)CO2)C1 CCCC(F)C(=O)NCC1CCN(C(C2CC2C#N)=O)C1 C(C(C)(O)C(=O)NC(CNC(=O)Cc1scnc1-c1ccccc1)C(C)C)OC Cc1cccc(C(=O)NCC2CCCN2C(=O)C=Cc2ccc[nH]2)n1 c1(C(N(CCNC(c2cn(C3CCC3)nn2)=O)CC)=O)ccnc2cc(Cl)ccc12 CC1=NC(C(=O)NC(C)CC2CN(C(=O)C(F)=CC3CC3)C2)CS1 C=C(CCC=O)C(=O)NCCNC(=O)NC(C)C.OCC C1(N(C)C)CC(NC(C2CCNC2=O)=O)C1(C)C.C1(=O)CCN1C1CC1 c1(NC(C2CCN(C(COc3ccc(C)cn3)=O)C2)=O)nc(C)c(Br)c(C)n1 c1(C(N2C(CNC(=O)CCOC3COC3)C=CC2)=O)cccc(CSC)c1 C(=O)(C(CC(N)=O)NC(C)=O)NCC(CC)NC(c1cc([N+](=O)[O-])c[nH]1)=O N1(C(c2c(C)nccc2)=O)CC2CN(C(c3c(C4CC4)cnn3C)=O)CC(C1)O2 N1(C(CCOC)=O)CCC(C(F)CNC(c2ccccc2C(=O)OC)=O)CC1 C(=O)(CC(C)C1CC1)N1CCC(OCC(=O)NCC(COCC)O)C1 CC1(C)CCN(C(=O)Cn2ncnn2)C(CNC(=O)CC2CCCCC2(F)F)C1 c1(C(=O)NCN2CCCC(COCC=C)C2)ccc(Br)c(Cl)n1 c1ccccc1C(N(C)C)=O.C(CCC(=O)N1CCC1(C)C(=O)O)NC C1(C)(C(N(C(C)CNC(=O)COC)CC)=O)CC(C)=NO1 C(=O)(C1OCCn2ccnc21)N1C(CNC(C2(c3ccc(C)cc3)CC2)=O)CC1 N1(C(=O)CCOC2CCOCC2)CCCC2C1CCN2C(C1CC12CC(O)C2)=O Cc1cc(C(=O)NCC2CC(C)N(C(C34CSCC3C4)=O)C2)ccn1 C(=O)(C1=CC(C)(C)C1)NCC(c1cc(F)cc(Cl)c1)N(C(=O)C(O)C(F)F)C c1(OCCC)cccnc1C(=O)NCC(C)CN(C(=O)CCSC)C c1(OC)ccc(CC(O)C(=O)NC2(CNC(=O)CCc3ccon3)CCOC2)cc1 C(=O)(C1Cc2c(Cl)cccc21)N1CCCC(CCNC(CC2(C)CCC2)=O)C1 C1(NC(C2C(C)N(C)CC2)=O)CC2(CCC(NC(=O)CCC3(C)CC3)CC2)C1 CC1CCC(O)(C(N2CCC(N(C(=O)Cc3csc(NC=O)n3)C)C2)=O)CC1 c1(C(C(=O)NCCC(C)N(C(C(c2cccs2)SC)=O)C)C)ccc(F)cc1 c1(CC)nc(C)c(C(=O)NC23CC(CNC(C4CCCS4)=O)(C2)C3)o1 c1(C(N2C(CCNC(CN(CC)CC)=O)C(C)CCC2)=O)cc2ccccn2n1 C(=O)(C1CCc2ccccc21)CC1C(CC(=O)OC)C1.C1(N)CC2(CCC2)C1 c1(C(=O)NCC2C(C)CN(C(C3CC(C)(C)C3)=O)C2)c(O)nnc2c1CCC2 Cc1nc(CO)ncc1C(=O)NC(c1ccc(Cl)cc1)CO N1(c2snc(CCC)n2)CC(NC(c2cccc(CS(C)=O)c2)=O)CC(C)(C)C1 c1(C(N2CCC(C3OCCO3)C2)C(=O)NCCCC)cc2sccc2s1 c1(CCC(=O)N(C)CCOCCNC(C2CC3CCC2O3)=O)ccccc1O C1(CC(=O)NC2CCC2)CCN(C(c2scnc2Cl)=O)CC1 N1(C(C2N(C(CC(CC)SC)=O)CC(=O)C2)=O)CCOCC(C(C)C)C1 O=C(N=c1c(Cl)c[nH]cc1Br)c1ccc(NS(=O)(=O)CC2CC2)cn1 [N-]=[N+]=NCCCC(=O)NC1CC2(C1)CC2NC(=O)C(Cl)=CCl N1(C(c2cncc(Cl)c2)=O)CC2C3CCC(C2C1)N(c1ccncn1)C3 C1(NC(C2C(COC)C2)=O)(CO)CCN(C(C2(C#N)CCSCC2)=O)CC1 N1(C(CCCc2ccc(C)cc2)=O)CCCN(C(C2CC(F)C2)=O)CC1 c1(C(N(C2CCN(C(C3CC4CC4C3)=O)C2)C)=O)cccc(CCO)c1 C1(NC(C(CC)c2cnccn2)=O)CC(NC(=O)Cc2ccsc2)CC1O C(=O)(CC1OCCc2ccsc21)N(CCNC(c1c(CC)scn1)=O)C1CC1 n1(CC(=O)O)cccc(CNCc2ccncc2C2CC2)c1=O C(=O)(C1=C(Cl)CCOC1)N1C(CNC(C2CN(C)C(=O)N2)=O)CCCCC1 O=C(N=c1cc2n([nH]1)CCCC2)C1CC2(CCC2)CN1C(C1CCCC2CC12)=O C1(CNC(C2CCC(C)(C)O2)=O)CN(C(=O)CNC(=O)C2CC2)CC2(CCC2)O1 C1(NC(c2c(CC)n(-c3cccc(Cl)c3)nn2)=O)NCCC12CCCC2 Cc1cc(O)ncc1C(=O)NCC1CCC(C)CN1C(=O)C(C)SC(C)C c1(C(N(C2C(C)CCN(C(C(COC)(C)OC)=O)C2)C)=O)nc[nH]c2nccc1-2 C1(CC)CCCCC1C(=O)NCC1(C(=O)NCC(C)(C)n2ccnc2)CC=CC1 N1(C(C=C=C(C)C)=O)CC2(CCC2NC(=O)CCc2cccc(F)c2)C1 C=CC1(C2(C(=O)NCC(CNC(=O)CN3CCCC3=O)CO)CCC2)CCC1 c1(CC)ccc(CNC(=O)C(=O)NC2CC2)nc1.C12(CCCC1)C(=O)O2 N1(C(C(=O)NC(C)CCC2CCCC2)=O)CCOC(C(C)(C)C)C1 C12(C(=O)O)CCN(C1)CC2.c1(C(C)=O)cccc(CSC(C)C)c1 C1(C)(C(=O)NCc2ccc(CNC(CC(C)CN(C)C)=O)cc2)CCN(C)C1=O C(C(F)(F)CCC(=O)NCC(C)(CO)N(C)C)n1cc(-c2ccc(C)cc2)nn1 N1(C(c2ccc(NC)cc2)=O)CCN(C(=O)C(O)C(C)C)C(CO)C1 C(CC(C)C)(C(=O)NC1CC(CCNC(=O)CCC(C)C#N)C1)NC(=O)OC N1(C(CC(CC)NC(=O)CCCCCOC)=O)CC(C)(C2CCC2)C1 CN1CCN(C(C2CC(CF)C2)=O)CC1.c1(C(N2CCC2)=O)cccs1 c12ccc(CN3CCC(F)(CNC)CC3)cc1O2.C(CO)OCC CCCC(CNC(c1ccnnc1C)=O)C(=O)N1CCC(C)C1C c1(C(=O)NC(CNC(c2c(C)nn(C(C)(C)C)c2)=O)(C)C)ccc(F)c(F)c1F Cc1c(C)c(Cc2cn(CC)nn2)c(C)c(C)c1Br.c1(C)cccc(N)n1 Cc1cccc(Cl)c1C(=O)NC1(C#N)CCN(C(c2ccnc(Cl)c2F)=O)C1 C1(OC)CC(c2nnnn2C2CC2)(NCC2CCCC2C(C)C)C1 N1(C(c2n(CC)ncc2)=O)CC2CCC(C1)N2C(C1CN(S(=O)(=O)C(F)(F)F)C1)=O C12CCN(C1)CC(=O)N2.c1(C(C(=O)NCCCCCO)C2CC2)ccccc1 CCC(C#N)(CC)C(=O)N1CCOC(CCCNC(=O)C(C)CC(C)(F)F)C1 c1(C(C(=O)NCC(CO)NC(c2nc(CC)oc2)=O)C)ccc(Cl)c(Cl)c1 C1(NC(c2cccc(OC)c2Cl)=O)CN(C(=O)C#CC2CCCC2)CC(C)(C)C1 S(=O)(=O)(c1cccnc1NC(C)(C)C)N(C)C(=O)NC1CC(NC2CCC2)C1 OC1CN(c2nccc(-n3ccnc3)n2)CCC1COc1ccccn1 N1(C(C(C)OCOC)=O)CC2(C1)CN(C(c1c(C)cccc1F)=O)CC(C)(C)O2 C1(C)(CC(=O)NC(C(=O)OCC)C2CC2)CCN(C(C2CC(O)C2)=O)C1 Cc1cnc(CN(C)C(C2(NC(C3C4CCC(=O)C34)=O)CCN(C)C2)=O)cn1 c1(C(=O)NC2C(CNC(CCNC(N)=O)=O)CCCC2)cnc2cccnc2c1 C(=O)(CCC(C)(F)F)N1CCCC(N(C(=O)CN2CCCC2C)CC)C1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)NCC1OCCN(Cc2c(C)nn(C)c2)C1 C=CC(CCC)CC(=O)NCCN(C1CCCCCC1)C(c1ccc(O)nc1C)=O C1(C(=O)NC2CCN(C(C3(C)CCC3)=O)CC23CC3)Cc2cccc(O)c2O1 C1(C(=O)NC2C(C)(C)CN(C(c3cc(C(N)=O)no3)=O)C2)CNC(=O)CC1(C)C c1(C(N2C(CNC(=O)CC3CCCCO3)C(O)C(O)C2)=O)c[nH]c2nccc-2c1 Cn1nc(C(F)F)cc1C(=O)NC1CCC(NC(=O)CC2COC(=O)C2)CC1 c1(C(=O)N(CC(N(C(C(C)OCCN(C)C)=O)C)C2CC2)C2CC2)ccc(Cl)nn1 Cc1cc2ccccc2c(NCC2(c3ccccn3)CCOCC2)n1 C(=O)(CC(C)(O)C(F)(F)F)NC1CCCN(C(C(C)Sc2ncccn2)=O)CC1 C1(F)(C(=O)OC)CCCN(Cc2cc(C)cc(Cl)c2)C1 N1(C(CCCC(=C)C)=O)CCCC2C1CCN2C(c1ccn2nnnc2c1)=O c1(C(N(CCNC(Cc2cc(C)[nH]n2)=O)C2CC2)=O)cccc([N+](=O)[O-])c1O C1(NC(C(CCCC)O)=O)CCOC2(CCN(C(=O)C=CS(C)(=O)=O)CC2)C1 C(=O)(CCCC(F)(F)F)NC1C(NC(c2cc(C(=O)OC)sn2)=O)CCC1 C1(NC(C2C(C)(C)NC(=O)C2)=O)C2CC(O)C1N(C(=O)CN(C1CCC1)C)C2 C1(NC(C(CO)OC)=O)CCN(C(c2ccccn2)=O)CCC1CO Cc1cc(=O)n(C)cc1C(N1CC2CCC1CN2C(C1CCC(C(N)=O)C1)=O)=O C1(C2CCN(C(C3CC(F)C(=O)N3)=O)CC2)(NC(C(C)OCCCC)=O)CCC1 N1(C(c2nccc(C)c2)=O)CCC(NC(=O)CSCc2ccco2)C(CO)CC1 N1(C(c2ccc(OCCCC)cc2)=O)CCN(C(=O)C(O)CN(C)C)CC12CC2 C1(NC(C(CCC)OC)=O)CC2CN(C(c3cccc(C4CCOC4)c3)=O)CC12 C(C(C)(C(=O)NCCn1ncccc1=O)NC(C1CC(=O)N(C)C1)=O)SC C1(CNC(CCC=C)=O)CC(C)(C)CCC1NC(c1nn(C)cc1Cl)=O c1(C(=O)NC(CC(C)NC(C2CC(C#N)C2)=O)C)ccnc2c1CCO2 c1(N2CC(C)C(N(C)C)CC2)nc(N2CCC(F)CC2)c2c(n1)CSC2 N1(C(=O)Cc2ccsc2)CCC2CN(C(=O)Cc3ccc(Br)cc3F)CC12 C1(C2(NC(CCOCC#C)=O)CC2)CCCN1C(=O)C(F)C1CC1 C1(NC(c2occc2Cl)=O)CC2CC1N(C(=O)CCc1nnc(O)nc1O)C2 C1(C(N2CC(CNC(=O)CC3CCC(C)CO3)(OC)C2)=O)(OC)CC(C)(C)C1 c1(C2C(C)C2)ccc(C=CC(N2CC(C)(NC(c3cn(C4CC4)nn3)=O)C2)=O)o1 C(CC(C)(O)C(C)(C)CNC1CS(=O)(=O)C1)N(C)C C1(CCC)CN(C(=O)C(C)CC(C)C)CCN1C(C1CCC(C(F)(F)F)CC1)=O Nc1ccc(C(=O)NOCc2cn(C3CC4CCC3CC4)nn2)cc1OC(F)F C(=O)(CC(C)(C)C(C)(F)F)NC(C)CN(C)C(c1ccnc(C(N)=O)c1)=O Cc1cc(C(=O)NC2CC(O)CN(C(=O)CCC(C)(C)C)C2)c(C)nc1C CC(C)C(CC(=O)NCCOc1ccccc1)NC(C1CCCC1(C)C)=O Cc1nnc2n1CCC2(C)C(=O)NCC(C)(O)CNC(c1nccn1C)=O C1(NC(c2c(C)nn[nH]2)=O)CN(C(c2c(C(C)C)cnn2C)=O)C2CCCCC12 c1(C(=O)NCC(CC)NC(=O)Cc2n[nH]cc2C)ccccc1F CCC(CC)C(O)CNC(=O)C(C)(C)NC(c1cocc1C)=O N1(C(c2ccc(C(C)C)cn2)=O)CC2(CCC2)CC1CNC(=O)C(F)=CC1CC1 N1(C(C2(COC)CC2)=O)CCC2(CCC(NC(c3csc(Cl)c3)=O)C2)C1 C1(C)(C(N2CC(F)(CNC(CCCOC(C)C)=O)C2)=O)CCCC(F)(F)C1 Cc1ccc(OCCC(=O)NC(CNC(C2SCCS2)=O)CC(C)C)c(C)c1 C1(C(=O)NCCCCC(=O)N(C(CSC)(C)C)C)CCC(C2CC2)C1 C(=O)(CCCCCNC(C)=O)NCC(C)N(C(C1COC2COCC12)=O)CC N1(CC(=O)NC2CCN(C)CC2)CCCCC(N(C)C(c2ccc(F)cn2)=O)C1 c1(C(=O)NCC2C=CCN2C(=O)COc2ccsn2)ccc2occc2c1 O(NC(=O)C(CCCOC)NC(=O)C(C#N)C(C)(C)C)CC=C C1(C)(C(N2C(C(CC)C)CCC2)=O)CCCN(C(C2CCC(C3CC3)C2)=O)C1 CC(C)CCC(=O)NCC12COC(CNC(C3CCCC(N(C)C)C3)=O)(C1)C2 c1(CC(N2C(C)CCC(NC(c3cc(Cl)c(Cl)s3)=O)C2)=O)cn2ccccc2n1 c1(C(N2CCC(NC(=O)CCCCC3CCSS3)C2)=O)cnc2ccc(Br)cn12 C=C1CC(C)(C(=O)N(C2CC(C(=O)NCc3ccn(C4CC4)n3)C2)C)C1 Cc1cc(F)c([N+](=O)[O-])cc1C(N1CC2C(N(C)Cc3ccc(F)cc3)C2C1)=O Cc1cc(C#N)ccc1C(N1C(C(=O)NC2CCOC(C)(C)C2)CCC12CC2)=O C=CC(CC)CC(=O)N1CCC(C(=O)NC(c2cn[nH]c2)C)C1C(C)(C)C C1(N)C(C)(C)CN(C(C2(CC)CCC2)=O)CC1(C)C.C(C=O)=CCC Cc1nc(C(=O)NC2CC(F)(CNC(C3CN(C4CCCCC4)C3)=O)C2)[nH]c1C C1(NC(C2C(C(=O)OC)C2)=O)CC2CN(c3cc(C(F)F)nc(C(C)C)n3)CC12 CCC(CNC(c1cncc(CO)c1)=O)(CC)NC(=O)CCC(C)=O C(=O)(C(F)(F)C(C)O)NC(C1CCCC1)CNC(C1(C)CC(C)C1)=O C#CCCCC(C)C(=O)NCC1CC(C)CN(C(C2CCCCC(=O)N2)=O)C1 C1(NC(CC=C=C)=O)CCC2CCN(C(c3cc(OC)n(C)n3)=O)C12 C1(N(C(CC=C)=O)CCC)CCN(C(=O)CCCc2cnn[nH]2)C1 C1(CNC(c2occ(C)c2)=O)CN(C(c2ccc(C3CC3)o2)=O)CC1(F)CO C1(NC(C(C2CCOCC2)OCC)=O)CCN(C(c2ccc(C)c(N)c2)=O)CC1F N1(C(Cc2cnc(C)[nH]2)=O)CCC(C(C)CNC(=O)CSc2nncn2C)CC1 c1(COC)nc(C2(Nc3cnn(CC(C)C)c3)CCC2)no1 C1(NC(Cn2c(C)csc2=O)=O)CCN(C(c2csnn2)=O)CC1C(C)C c1(NC2CN(CC)C2)cc(N2CCOC(C3CCCCC3)C2)ncn1 CCC(Cc1ccccc1)C(=O)NCC(C)CN(C(=O)CCn1ccnc1)C C1(C(=O)NCC2(NC(CC3C(=O)OCC3)=O)CCCC2)OCC2COCCC12 N1(C(=O)OC(C)(C)C)CC(CC(=O)Nc2nc(C3CCOC3)cs2)C2(CC2)C1 C#CCC(CC(F)F)C(=O)NCC1CCN1C(=O)CCn1ccnc1C CC(O)C(C(=O)N(CC(=O)N=CC(=O)N(CC(F)F)C)C)NC(N)=O C1(C#N)(C(=O)NC2CC(C)N(C(c3cn(C4CCC4)nn3)=O)C2)CC12CCC2 C(=O)(C(C)(C)CC1CCOCC1)N1CC(NC)C1 C(=O)(C1=CCN(C(c2ccc(C3CC3)cc2)=O)C1)NC1CC(C)SC1 c1(CC(C)NCC2(N)CC3(CCCC3)C2)ccc2occc2c1 c1(C(=O)NCC2(F)CN(C(CC3C(C)(C)C3)=O)C2)ccc(F)c(F)c1 Cc1ccc2nc(C(N3CCN(C(C4CCOCC4)=O)C(C)C3C)=O)ccc2c1 c1(C(N(C(C(NOCCC)=O)C)CCC)=O)cc(F)cnc1O C1(NC(C2(C(F)F)CC(=C)C2)=O)CCN(CCNC(=O)Cn2ccc(=O)cc2)CC1 CCCC(O)CC(=O)NC1(CCNC(=O)C(C)SC)CC1 N1(C(COC(C)=O)=O)CCC(C(F)(F)F)C(NC(c2ccc(C)c(F)c2)=O)C1 C=CC1(C(=O)NC(c2ccccc2O)C)CCN(C(=O)C(C)C(C)C)CC1 Cc1cncc(C)c1C(=O)NCCC(C)N(C(=O)C(C)n1ccnc1)C C1(OC)CN(C(=O)CC2(C)CC2)C(C)(CNC(C2(F)CCOCC2)=O)C1 Cc1cn2c(n1)CC(C(N1CC(NC(c3cccc(C(C)(C)C)c3)=O)C1)=O)CC2 N1(C(c2cccc(OC)n2)=O)CCN(C(c2cnn(C)c2N)=O)C(C)C1C C(=O)(CCC(N)=O)N1C(C(C)NC(CCCOCC)=O)CCC1 N1(S(=O)(=O)CCNC2CCCCNC2)CCCc2cc(Br)c(F)cc21 N1(C(C(CCC)Cl)=O)CCc2cc(S(=O)(=O)N3CCC4CC(C(=O)O)C4C3)ccc21 c1(C(=O)NC2CCN(c3ncnc(C(F)(F)F)c3Br)C2)ccc(Cl)c(Br)c1 C1(CC(N2CC(C)(NC(C3C(c4ccc(C)s4)C3)=O)C2)=O)CC(=O)NC1=O C(=O)(C1CNc2ccccc21)N(CC1N(C(=O)OC(C)(C)C)CC(C)(C)OC1)CC#N c1(C(=O)NCC2CSCCN2C(c2cc(Cl)ccc2O)=O)nccc2[nH]ccc12 C(=O)(C(C)(C)C(C)C)NCC(CNC(c1c(C)oc(C(C)C)n1)=O)O N1(C(Cc2nc(C)sc2Cl)=O)CC(C)(C)CC1CNC(=O)C1=CCCCC1 N12CCC(F)(CC1)CSCCC2=O.C(=O)(C(F)(F)CC1CCCC1)N(CC)CC N1(C(c2cncc(OC)n2)=O)C2CCC1C(CO)N(C(c1csc(C)n1)=O)C2 c1(C(N(CCN(C(c2c(CC)c[nH]c2)=O)C)C)=O)cc(O)ccc1OC C1(C(=O)NC2CC2(F)F)CN(C(c2ccc(F)cc2I)=O)CC(F)(F)C1 c1(C(=O)NCCCCN(C(=O)Cc2cnc[nH]2)C)n[nH]c2cc(Cl)ccc12 C1(C(=O)NC2C(NC(c3cccc(C4CCC4)c3)=O)CCC2)Cc2nccn2C1 Cc1nn(C(C)(C)C)cc1C(=O)N(C)CC1CCCN1C(=O)CC1CCC2CC12 c1(OC)ccc(C(=O)NC2CC(C)N(C(=O)C(C)=C3CCCC3)C2)cc1O N1(C(=O)COCC(F)(F)F)CCC2(CCCN2C(c2ccncc2)=O)C1 C(CCc1ccccn1)(C(=O)Nc1cn(C)nc1OC)NC(C12CC(C)C1C2)=O Cc1ccc(C(N2CC(CF)(NC(C3CC(F)C(=O)N3C)=O)C2)=O)cc1C C(C(C)(C)CCCO)C(C1CC(CCO)(SC(C)(C)C)C1)C(=O)NC1CCOC1 c1(NC(=O)NC)ccc2c(c1)CN(C(c1csnc1C)C(=O)NC1CCC1)CC2 c1(OC)cnnc(C(N2CCC(CC(N3CCC3C3CCCCC3)=O)CC2)=O)c1 C(=O)(CC(C(C)C)C(C)C)NCCCNC(c1c(-c2ccc(C)cc2)ocn1)=O Nc1cc(F)c(CC(N2CCOCC(NC(=O)Cc3cnoc3)C2)=O)cc1F C1(NC(CCCCOC)=O)CN(C(=O)Cc2nnc(C)s2)C2(CCOC2)C1 N(C1CCCc2ccccc21)CC(=O)Nc1ccc(N2CCCC2=O)nc1 C(=O)(CC(C)C(C)(C)C)N(CCOC)CCNC(=O)C(O)Cc1ccccc1 CC1(C)CN(CCNC(=O)C(N)CC2CCCO2)CCS1=O C1(C)(CCNC(Cn2ncc(C)c2)=O)CCN(C(=O)C(F)C2CCC2)C1 c12ccccc1C2.C1(CN(C(C2C(=C)C2)=O)C)CCCN1C(=O)CCSC Cc1cc(C(=O)NCC2CCC(C(=O)NCCCn3cccc3)CC2)nc(C)c1 C(CN=c1ncc(Br)c[nH]1)(c1ccccc1F)N(C(CCCCC)=O)CCC c1(C(CCC)NC(C2CCCCCC2)C(=O)OC)ccc(OC)c(OC)c1 C(c1ccc(F)cc1)=CC(=O)NC1CCCC(N(C(=O)C=Cc2ccoc2)C)C1 C1(C)(CC)CC(NC(=O)Cc2csc(S)n2)CN1C(=O)C=Cc1nccs1 C1(CC2C(C)=CCS2)CC(C(=O)NOCc2cn(-c3ccc(Cl)cc3)nn2)=NO1 C=C(F)C1(CC(=O)NCCC2CCCN2C(=O)Cc2cc(C3CC3)no2)CCC1 N1(C(COCC(=O)NC)=O)CCC(C2CC2)C1C(N1CC2CCC2(CO)C1)=O C(=O)(CC(C)CCCCC)N1CCC(C(=O)NCC(C#C)OC)(CC)CC1 C1(CNC(c2cc(C)on2)=O)CC(F)(F)CN1C(=O)C=CC(F)(F)F N1(C(C(CC=C)CC)=O)CCc2ccc(C(=O)NCC(C)(C)F)nc2C1 c1(OC)cc(N)c(Cl)cc1C(=O)NC(C1(CNC(=O)C2=CCCC2C)CC1)C C(=O)(C(C)(C)C(F)(F)F)N1C(CO)CC(NC(COc2cc(C)cc(C)c2)=O)C1 N1(C(CCC2(C)CC2)=O)CCCC(C)(CNC(c2csc(O)n2)=O)C1 Cc1cc(C2CC2c2ccccc2F)ccc1CN1CCC1C(=O)NC(C)C C(CNC(C1CCN(C(=O)C=C(C)C(C)(C)C)CC1)=O)(CC(C)C)OC Cc1scc(C(=O)N(C)CC2(CNC(C3CC3C(C)(F)F)=O)CC2)c1Br C1(C(=O)NCC(C)NC(=O)COc2cccnc2)CC2(CCCCC2)S1(=O)=O C1(CC)CN(C(=O)CC(C)(C)OC)CCC1NC(c1snc(Cl)c1Cl)=O C(CC1=CCCCC1)NC(C1CC(N(C(Cc2c(C)noc2C)=O)C)C1)=O CCCC(C)(O)CC(=O)N1CC(CSC)C1.c12cccc(c1)CN(C)C2=O CCC(CC(F)(F)F)C(=O)NC1CCCC(NC(c2coc(C(C)OC)n2)=O)C1 c1(C(C(N2CCC(NC(c3cn(C)nn3)=O)C2)=O)O)cc(F)c(F)c(F)c1 CCCCC(O)C(=O)NCC1CCC(C(N2CCCC2)=O)O1.C12CCN(CC1)C2 C(C(C(C)C(C)C)NC(C1(C(=O)NC)CC1)=O)NC(c1n(C=C)ncc1)=O CCC(CC)(CO)C(=O)NCC1(C)CCCN(C(=O)C(c2ccccc2)C)C1 C1(NC(c2ccc(OCC)cc2)=O)(CC)CCN(C(=O)Cc2c[nH]c(=N)o2)CC1 C1(NC(=O)Cc2cscn2)CC(NC(C2CC3(CCCC3)C2)=O)C12CCC2 c1(C(=O)NCC(C)(C2CCC2)NC(C2CCNC2=O)=O)ccccc1C#CC1CC1 S(=O)(=O)(c1ccc2nc(NC3(C4CCCO4)CC3)sc2c1)N1CC=C(C)CC1 S(=O)(=O)(c1ccccc1F)N(C(CNC1CCCN(CC)C1)C)C CON(CCC(=O)N1CCC2(CNC(=O)CO2)C1)C(=O)COC1CCOC1 C(CC(C)(C)CNC(C1(F)CC=CC1)=O)NC(C(CC)n1nccc1C)=O C=CC(C)(O)C(=O)N(C)CC1(O)CCN(C(c2cc(F)n[nH]2)=O)C1 c1(NC(C(C(C)C)C2CCC2)=O)ccc2nn[nH]c2n1.C12CN(CC1C)C2=O CC(C)(C)S(=O)(=O)Cc1ccc(C23COCC(c4ccc(C(=O)O)cc4)(C2)C3)s1 C1(CC=C)CCCC1C(=O)NCCN(C(C12CC(CO1)C2)=O)CC CC(CC(=O)NCCC1CCCN(C(c2ccn(C(C)(C)C)c2)=O)C1)C(F)F c1(C(=O)NCC23N(C(c4ncc(C)nc4)=O)CC(C2)C3)cccn2nccc12 C1(NC(C2CC(CO)N(c3nnc(C(=O)O)s3)C2)=O)CCC2C(C1)C2(F)F c1(CC(=O)NCCCCCCNC(=O)C(O)C2CCCC2)ccc(O)c(OC)c1 c1(C(N2C(CNC(=O)CC3CCC(F)(F)CC3)CC(O)C2)=O)cc(O)ccc1F C(=O)(CCCN(C)C(C1CCN1C(c1cn(CCOC)nn1)=O)=O)NC1CC1.CO N1(C(CC)=O)CCC2(COCC(CNC(=O)COCCOC)O2)C1 N1(C(COCC=C)=O)CC2CC3CC2C1C3NC(c1ccc(OC)c(Cl)n1)=O CC1(C)CC(NC(=O)C(C2(O)CN(C(=O)C=C3CCCC3)C2)F)C2(CCC2)C1 c1(C(=O)NC(C(=O)NC(c2nncs2)C)CO)ccc(=N)[nH]c1 c1(C(=O)NC2CCC(C(=O)Nc3c(C)c(F)ccc3)C2)ccc2ccc(Cl)cc2n1 CCCCS(=O)(=O)CC(=O)N1CCC(Nc2cnc(C#N)cn2)C(C)C1 C(CC(C(=O)NCCC(O)CO)NC(=O)C(c1cncnc1)C)OCC c1(NC(C2CCN(S(=O)(=O)CC3CCC3)C2)=O)cc(Cl)c(F)cc1F C#CCC(CC(=O)NC1CCCC1F)NC(C1CC2(CC2)CO1)=O C1(NC(=O)NC2CC(C)(C)N(CC3CCC3)C2)C2CCC3C(C2)CC13 c1(C(C)=O)cc(C(=O)NCCCC2CCCN2C(=O)C(N)=O)n(C)n1 c1(NC(N2CC(O)CC2Nc2ccc(NC(C)=O)cc2)=O)ccc(C)cc1Br c1(C(=O)NC2(C)CN(C(=O)C(C3CCCCCC3)O)C2)cc2n(n1)C(C)CCC2 CCC(C(=O)OC)C(=O)N1CCC(C)(NCCNC(c2cnn(C)c2Cl)=O)CC1 N1(C(C2(C(F)F)CC(=C)C2)=O)CCC(CNC(=O)C(C)SCCCC)(OC)C1 N#Cc1ccc(CN2CCCC(C(=O)Nc3ccnc(C4CC4)c3)CC2)cn1 n1(CNC(CN(C2CCC2)CC=C)=O)cc(C)cn1 c1(NC(N)=O)ccc(C(=O)NC2CCCCC2CNC(c2coc(O)n2)=O)cc1 N1(C(C)C)CCC(C(N2CCCC(N(CCO)C(C3(CF)COC3)=O)C2)=O)CC1 N=c1[nH]c(N2CC3CC(NC(C4(C(N)=O)CC4)=O)C3C2)ncc1[N+](=O)[O-] Cc1nc2c(cc1NC(=O)NCC(c1cc(F)cc(Br)c1)N)c(C)nn2C C1(C2CC2)(C(N2CCCC(F)(CNC(C(C)n3cnnn3)=O)C2)=O)CCOCC1 CC(CNC(=O)Cn1ccnc1)C(=O)NCC1=CCCC1 C1(C(=O)NC2CC(C)(NC(C3(CC)CC3(F)F)=O)C2)CC(=O)NC(CC(C)C)C1 C1(NC(C(C)(C)C)=O)CCCC12N(S(=O)(=O)Cc1ccc(Cl)c(Cl)c1)CCC2 c1(C(=O)NC2CCC(C(=O)Nc3c(Br)cncc3Br)C2)cc(Cl)cc2nc[nH]c12 c1(C(=O)N(CC(C)C)C2CC2C2CN(C(=O)CC3CCCC3)C2)conc1C1CC1 N1(C(C2C(=C)CC2)=O)CC(NC(c2c(N)cncc2Br)=O)CCC1C CCC(O)C(C)C(=O)NC1CCN(C(c2cc(C)[nH]n2)=O)C1(C)C c1(C(N(CC(CN(C(=O)C(O)C(F)F)C)O)C)=O)csc2cccc(F)c12 N1(C(c2cnc(CC)[nH]2)=O)CCCC(NC(=O)C=Cc2ncc(C)[nH]2)CC1 c1(C(N2C(CCNC(c3c(C)cccc3)=O)CSCC2)=O)ncn2c1CCCC2 C(C(C)(C(=O)N(C)Cc1c[nH]nc1C)NC(=O)Cc1cc(C)on1)SC c1(C(=O)NC2CC(CNC(CC(C)(C)C#N)=O)C2)ccc2nc(S)oc2c1 C1(C(C)(C)NC(CC=CC)=O)CCN(C(c2cc(Cc3ccccc3)on2)=O)C1 c1(C(N2CCC(C)(CNC(C(F)=CC)=O)C2)=O)ccc(C(F)(F)F)cc1 N1(C(c2ncc(C)o2)C(=O)NC(CC)C)CCN(C(=O)NC)CC1 c1(C(=O)NC2C=CCN(C(c3cnc(SC)s3)=O)C2)nccc2nn[nH]c12 c1(C(N(CCN(C(C23C(C)OC(C)(C2)C3)=O)C)C)=O)cc(F)c2ccccc2c1 c1(NC(C(=O)NC(c2ccc(Cl)cc2F)C)=O)ccc(S(N)(=O)=O)s1 c1(OCC(=O)N(C2CCN(C(=O)CCCF)C2)C)ccc(C=CC#N)cc1 C1(NC(=O)CC2CCOC2)CC2(CCC(NC(=O)C3=CCCSC3)CC2)C1 c1(C(C)(F)C(=O)NC2CCN(C(=O)Cn3cc(C4CC4)nn3)C2)ccccc1F c1(C(=O)NC(C(=O)N(C2CC2)CC)(C)C2CCC2)cnccn1 C12(NC(C(N)=O)=O)CCN(C(C3(S(N)(=O)=O)CC3)=O)CC1C2 N1(C(C2CC(COC)C2)=O)CCC2CC1CN(C(=O)CC(C)(C)N(C)C)C2 c1(C(c2nnnn2C)NCC(C)CC(F)(F)F)nc2ccccn2c1Br C1(CC(=O)NCC(CNC(CC=CC=C)=O)(C)OC)CCN(OC)CC1 C(C(=O)N1CCCC(CN(C(=O)C(C)OCOC)C)C1)(C(C)C)NC(=O)OC c1(C(=O)NC(CCNC(=O)NC)C2CNC2)ccc(-c2ccccc2)nc1 N1(C(CCC)=O)CC2(CNC(C3C=C(C)CS3)=O)CC1CCO2 c1(C(N2CCC(NC(c3ccc(C#N)[nH]3)=O)(CO)CC2)=O)cc(F)c(F)cc1F c1(NCC(=O)NC(CC=C)CNC(=O)C(C)OCC2CCCO2)ccccc1F c1(C(=O)NC(C2CCCC2)CNC(C=C(COC)C)=O)cc(C)c(C)[nH]1 c1(C(C)NC(=O)C(=O)NC2CCC(N)C(F)(F)C2)nc2ccccc2n1C c1(C(N2CC(C)C(CNc3cccc(C(F)F)n3)CC2)=O)c([N+](=O)[O-])cnn1C N1(C(c2c(CC)c(C)sc2)=O)CCC2C(CCN2C(=O)CCCc2cccs2)C1 c1(C(N2CCC(NC(C3(C)C=CCC3)=O)C2)=O)cccn2c(CC(=O)O)nnc12 C1(NC(CCCOC(C)C)=O)CC(C(N2CC(C)(F)C2)=O)C12CCC2 N1(CCC)CCCC(C(=O)NCC(C)N(C(c2cnc[nH]2)=O)CC)C1 c1(-c2cn(CCCCCNC(=O)CN3CCC(CO)C3)nn2)cccc(F)c1F Cc1c(Cl)nc(NC(C2CCCC2NCc2cnc(Cl)nc2Cl)=O)nc1Cl C1(CNC(c2c(C)n(C)nc2)=O)COCCN(c2nnc(C(N)=O)s2)C1 Cc1ncnc(C)c1CC(=O)NCC12CC(CN1C(=O)C(C)S(N)(=O)=O)C2 O(CP(C)(C)=O)CC(=O)NC1CC(NC(COC(C)C)=O)C1.C1CC1 c1(C(C(=O)NCC2(C)N(C(CNC(=O)OCC)=O)CCC2)O)cc(C)cc(F)c1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC(NC(c2c(SC)cccn2)=O)CC1(C)C c1(OC)cc(=NCC2C=NN(C)C2=O)[nH]c2cc(Br)ccc12 C12(C(N3C(CN(C(C4CCCNC4=O)=O)CC)CCC3)=O)CCCN1CCC2 C1(CNC(C(C)NC(C)=O)=O)CCN(C(=O)C(C)(C)N(S(C)(=O)=O)C)CC1O c1(CC)oc(C(=O)NCC2(CCNC(C3CC4CCC3O4)=O)CC2)cc1C C1(C(=O)NC2(C(C)O)CC2)CCC2CCC1N2C(C1CCC(=O)O1)=O CC1(C)C(NC(=O)C(F)CC2CC2)CCN1C(=O)CCOCC1CC1 C(=O)(N1CCCc2nncn21)C1CCC(n2cc(SCC(=O)O)nn2)CC1 C=CCCCCCP(C)(C)=O.C(=O)C(C(C)NC(=O)NC(C)(C)C)C(C)C C=CCCC(F)(F)C(=O)NCC1CC(C)CN(C(c2cccc(F)c2F)=O)C1 C123C(C4CC1C2C4)NC3=O.CC#CCN(C(=O)COCCF)C c1(C(N2CCCC(CNC(COC(C)=O)=O)CC2)=O)ccccc1N=NN(C)C Cc1c(N)ccc(C(=O)NCC2CCCCN(C(=O)C#CC3CCCO3)C2)c1C C1(C(=O)NCC#C)CC(NC(=O)C(C)NC(=O)CC)C(O)C1 c1(C(N2CCN(C3CCN(CC)C3)CC2)C(=O)NC2CCC2)cccc(Br)c1Cl C1(NC(c2nc(C)oc2)=O)CCC2(CC1)CN(C(=O)C(C)(C)C(C)C)CCO2 C(=O)(C1CNC(=O)c2ccnn21)N1C2CN(C(CC3CC(=C)C3)=O)CC1CCC2 CCC(O)(C(=O)NC1CCN(C(c2ccncc2)=O)C1C)c1cccc(Cl)c1 c1(OC)ccc2c(c1)CC(C(=O)NCC(O)CNC(c1ccc(Cl)cc1O)=O)O2 c1(NC)ccc(C(=O)NC2CN(C(c3ccc(F)o3)=O)CC2C)cc1.OC(F)(F)F c1(C(N2CC(CC=C)(NC(=O)C=CCO)C2)=O)cc(Br)c2c(c1)nnn2C c1(CC)c(C(=O)NCC(C)(C)Cn2cc(-c3cncc(N)c3)nn2)nnn1CC CC(C)CC(CNC(C1(n2cnnn2)CC1)=O)C(=O)N1CC(=C(F)CO)C1 CC1(C)CCC(O)(C(N2CC3CC2C3CNC(=O)CCc2nc[nH]n2)=O)CC1 c1(CC(=O)NC(C(=O)NCC(C(C)(C)C)OC)C2CCCC2)cc(C)ccc1F c1(OC)ccccc1CCC(C(=O)NC1CC(F)(F)C1)N(C)Cc1ncnn1C CCC(CC(=O)N(C1(CC(=O)NCCC(C(C)C)OC)CC1)C)C(F)F c1(C(N2CC(C(C(=O)NC3(CC=C)CC3)O)C2)=O)occ2c1CCC2 c1(OC)cccc(Cl)c1C1CC1C(=O)NCC(C(C)C)NC(C1CCC(=O)N1C)=O c1(C(C(=O)NCCCSC)N(C)CC2COC(C)(C)O2)cc(Cl)cc(Cl)n1 c1(C(=O)NCC(C)NC(C2CCCO2)=O)ccc(C2CC2)cc1 CS(=O)(=O)c1ccc(N(C2(c3ccccc3C(F)(F)F)CCOC2)CCl)cc1C#N c1(C(N2CCCC(CNC(c3ccc(CF)cc3)=O)C2)=O)cc(O)ccc1F N1(C(C2(c3cccc(C)c3)CC2)=O)CCCC(F)(COC)C1.C1(=O)C(C)CN1 C1(CNC(C=C(CCC)C)=O)CCC2(CN(C(=O)C=C3CCC3)C2)O1 CCS(=O)CC(=O)NC1(C(=O)NCc2nn(C)cc2C)CCCC1 N1(C(CN(C(C)=O)C)=O)CCC(C2(O)CN(C(=O)CC(C)(C)N(C)C)C2)CC1 C(=O)(CCCCN1CCCCC1)NC(C1CN(C(c2ccsc2)=O)C1)C Cc1ccc2c(=NC(C)CN3CCC(C)C3)[nH]c(=NCCC3(C)CC3)[nH]c2c1 C(=O)(C(C)(CNC(=O)CC(C)n1ccnc1)CC)NCC1(CC)CCOC1 C1(CNC(c2nccc(CC)c2)=O)(NC(C2CCN(C)C2)=O)CCC(C)(C)CC1 C1(CC(=O)O)CC2CC1N(C(=O)COCc1cc(Cl)ccc1Br)C2 N1(C(CC(C(C)C)(F)F)=O)CCCC12CCN(C(C1CCC(=O)N(C)C1)=O)C2 c1(CNC(c2ccc(CNC(C3(C)N(C)CCC3)=O)o2)=O)cc(Cl)ccc1F C(=O)(C1=CS(=O)CCC1)N(C1CC1)CC1N(C(c2c(C)cc(SC)o2)=O)CCC1 c1(C(=O)Nc2nnc(C(=O)OCC)s2)ccncc1C.n1(C)cc(CCOC)nn1 C(=O)(CCCCCc1cccs1)NCC(CCNC(c1onc(CC)c1C)=O)(C)C c1(OCC)ccc(NC2CC2)c(C(C(C)CC(C)C)c2nnnn2C2CCC2)c1 N1(C(C(CCC)F)=O)CCCC2(C1)CN(C(c1coc(COC)n1)=O)CCO2 C1(NC(C(C)CC2CCC2)=O)CCN(C(=O)Cc2ccnc(C(F)(F)F)c2)CC1 N1(C(C2=CCN(C(C3CCCC(=O)N3)=O)C2)=O)CCc2ccccc21 c1(N(C(C=CC(=O)NC(CC#C)CC)=O)C)ccccc1O c1(C(=O)NC2(C)CC(NC(c3ccc(C)nc3C)=O)C2)ccc(S(N)(=O)=O)cn1 C1(C(=O)Nc2cc(CCC)no2)CCN(C(c2cc(C)cs2)=O)C1CC Cc1cc(NC(=O)C(C)(C2CCC2)NC(c2ccnc(C)n2)=O)c(O)c(C)c1 C1(NC(C(C)(C)O)=O)CN(c2ccn3nccc3n2)C2CCCCC12 C1(C#N)(CC(=O)NCC23C(CN(C(c4n(C(C)C)ccn4)=O)C2)C3)CCCCC1 c1(NC(CN(C(=O)CCC2OCCO2)C)=O)ccc(Br)c2ccccc12 CC1(C)CC(NC(=O)CCc2csnn2)CCN(C(=O)CC2CC3C=CC2CC3)C1 CC(C)(CC(=O)NCCC1(CNC(C2CCC3(C2)CC3(F)F)=O)CC1)CC(F)F c1(C(=O)NCCCNC(C2CCC3(C2)CC3(F)F)=O)cc2c(cc1O)CCCC2 CCC(C)CCCC(=O)NC(C(=O)N(C)Cc1n[nH]c(C)n1)C1(O)CCC1 c1(CC(N2C(CNC(c3ccn(C)c3)=O)CCC2)=O)ccccc1Br Cc1c(C(N2CC(NC(=O)C(O)Cn3cncn3)C(F)C2)=O)nn2c1CCCC2 Cc1ncccc1C(=O)NCC1CC(NC(c2cc(-c3ccc(C)o3)[nH]n2)=O)C1 C1(C(=O)NC(C2(O)CCN(C(=O)Cc3ccccc3C)C2)C)CC12CC(O)C2 C1(NC(C(C)N(CCC)C(C2CCOC2CC)=O)=O)CCN(C)CC1(C)C c1(C(=O)NCCN(C(=O)C=Cc2cnccn2)C)cccc(S(=O)(=O)CCO)c1 C1(C)(CCC(=O)N(CCCNC(c2cnc(C)[nH]2)=O)CCO)CCC(=O)N1 c1(C(=O)NCC(CC)NC(c2c(N)cc(CC)cc2F)=O)ccc(F)c(C)c1N Cc1csc(C=CC(=O)NCCN(C(=O)CC2CCC23CCC3)C(C)C)n1 N1(C(CNC(CC)=O)=O)CCC2(CC2NC(C2CN(C)CCN2C)=O)C1 N1(C(C2(CC)COC2)=O)CC2(CCN(C(c3ccc4c(c3)OCO4)=O)CC2)C1 c1(C(=O)NC2C(NC(C3C(C)CCO3)=O)CCCC2)cc2nc(F)ccc2o1 CN1CCCC(CNC(C2(F)CCCN(C(=O)C=Cc3cnn(C)c3)C2)=O)C1=O N1(C(CCC=C)=O)CCC(F)C(NC(=O)CC(=O)NCC(F)(F)F)C1 c1(C(N2C(C(=O)Nc3c(C)ccnc3Cl)CC2)=O)nccc2ccccc12 CC1CNc2c(C(=O)NC(C)(C)CN(C)C(c3cc(C#N)c[nH]3)=O)cnn2C1 N1(C(c2cn(C(C)C)nn2)=O)CCN(N2CCCC(C)C2)CC1CCO.C(=O)CO CCC(C)CCCC(=O)N1CC(OCCNC(C2(c3ccccc3F)CC2)=O)C1 c1(C(=O)NC(CCNC(C#CC2(CC)CC2)=O)C)c[nH]c2nccc-2c1C c1(CC)cc(OC)ccc1C(C(=O)Nc1ccccc1Br)N(CCCO)CC c1(C(=O)NCC(C)N(C(=O)CC2(O)CCCC2)CC)ccc(C(=O)NC2CC2)s1 N1(C(C(C)OC)=O)CCN(CC2CN(C(c3nnc(C(C)(C)C)s3)=O)C2)CC1 c1(CC(N2C(CNC(c3cc(CO)on3)=O)CC(OC)C2)=O)c(C)ncnc1O c1(C(CCNc2cccc(SCC)c2)C)csc2ccc(O)cc12 C(CN=c1[nH]c(=NCC2COC(=O)O2)c2c(F)cccc2[nH]1)(C(C)C)OC C1(NC(c2cccc(C)c2O)=O)CC2COCC(C1)N2C(=O)CC1COC(=O)C1 CC1(C)CN(C(=O)Cc2ccc(C#N)cc2F)CCC1NC(C1CNC(=O)C1)=O C(CC(=O)N1CC2C(C1)C2(F)F)(C(F)(F)F)NC(c1ccccc1C1CC1)=O CC1(C)CCCC1(C)NC(=O)C#CCNC(C1(C#N)CCOC1)=O CC1CCC(C(=O)NC2CSC2)N(C(C2CC=CCO2)=O)C1 C(=O)(CC1=NN(C)C(=O)C1)NCC1C(NC(C(C(C)O)(F)F)=O)CCC1 C1(NC(=O)C(F)=CC2CC2)COC2(C1)CN(C(C1CC3CCC1C3)=O)C2 N1(C(C(C(=O)OC)C)=O)CCC(C2CCN(C(c3ccc(CSC)[nH]3)=O)CC2)C1 Cc1ccncc1C(=O)NCC(O)CN(C)C(C1(C)CC(F)(F)C1)=O c1(C(N2C(C)CC(NC(c3cc(CC)c(O)cc3)=O)C2)=O)ccc2n[nH]cc2c1 c1(C(=O)NCC(C2CC2)NC(CCc2ccn(C)c2)=O)c(C2CCC2)cnn1C N(C(=NCCc1ncnn1C)NC1CC1(c1ccc(F)cc1F)C)CC c1(CN2CCCC(C#C)C2)cc(O)c(O)cc1O.C12CC3CCC1N3C2=O c1(C(N2CCC(CN(C(c3cc(C)on3)=O)C)CC2)=O)cc(F)c(Cl)c(N)c1Cl N1(C(CCOCCOCC)=O)CC=C(CNC(=O)Cc2cn[nH]c2)CC1 N1(C(c2ccc(OC)nn2)C(=O)NC2(C)CC2)CC2C(=O)N(C)C(=O)C2C1 c1(OC)sccc1CNC(C1(Cl)CC1C(=O)NC1CC1c1ccnn1C)=O c1(CC)cc(C(=O)N(C(C)(C(=O)NC(c2ccc(C)s2)C)C2CC2)C)ccn1 c1(N(C)Cc2cccnc2)ccnc(NCCCn2cncn2)n1 N1(C(C(CC)(C)CC)=O)CCC(C)(C)C(NC(=O)CCOc2cccc(C)c2)C1 c1(CNC(=O)NCCCP(OCC)(C)=O)cc(Br)cc2nc[nH]c12 C1(C(N(C)CC2N(C(CCCC)=O)CCCC2)=O)CCN(C)S1(=O)=O C1(C(=O)NC2CCC(C#C)C2)(NC(c2ccn(C)n2)=O)CCC(C)(C)C1 N1(C(c2csc(Br)n2)=O)CCC(O)(CNC(C2(F)CCCOC2)=O)C1 C1(C(=O)NCC2CCCS2)CC(F)CCN1C(=O)COC1CCOC1 C1(C(N2CCC(OCCNC(c3ccc(C)nc3)=O)CC2)=O)C2CS(=O)(=O)CC12 c1(OC)cccc(Cl)c1C(N1CCC(NC(=O)CC2CSCCS2)C1)=O N1(C(CCSCC)=O)CCC2(CCCC2NC(=O)CCC2OCCO2)C1 C(CCC)(C(=O)NCC(O)CNC(C1CC1C(C)(F)F)=O)=CCC CC1(C)CCC2(CC1)CC2C(=O)NC12CC(NC(c3cc4n(n3)CCO4)=O)(C1)C2 N1(C(C(CC)Nc2cnn3c2OCC3)=O)c2ccccc2CC1C C1(CC(C)NC(c2cc(OCC)n[nH]2)=O)CCN(C(=O)Cc2cnn(C)c2)CC1 c1(C(=O)NC2CCC(NC(c3c(COC)noc3)=O)C2)ccc(C)c(C)c1O C1(C(=O)NCC(C)NC(CCSCC)=O)CCc2nn(C)cc2C1 CCC(C)C(CC(=O)NC1CC1C1CCC1)NC(=O)CCCNC(C)=O CC(C)CC(C)CC(=O)NCC1CCN(C(c2cccc(C3CC3)n2)=O)C12CC2 C(=O)(CCCC(=O)OC(C)(C)C)NC1CCC(N(C(c2c(C)cns2)=O)C)CC1 N1(C(Cc2ncc(CC)[nH]2)=O)C2CCCC1CN(C(=O)C=C1CCC(C)C1)C2 Cc1ccc(F)cc1NC(=O)C(=O)N(c1ccccc1)CC(=O)O.C1(SCC)CCS(=O)(=O)C1 CC1CN(C(C2CCCN(Cc3nc(-c4ccsc4)no3)C2)=O)c2ccccc21 CC(C)(CS(N)(=O)=O)C(=O)NCCCCNC(C1CCC(C(=O)O)S1)=O CS(=O)(=O)c1cccnc1N1CCC(NC(=O)CCn2cccn2)C(F)C1 c1(C(=O)NCC(C(=O)N2CC(C)(COC)C2)(C)C)ccc2n[nH]cc2c1 N1(C(c2ccc(SC)o2)=O)CCCC(NC(c2cc(F)c(F)c(F)c2)=O)C(F)C1 c1(C(N2C(CN(C(C3CCCO3)=O)CC)CCC2)=O)c(C)sc(C)c1Br N1(C(c2ccc(CC)[nH]2)=O)C2CCCC1CCC(NC(c1ncsc1C)=O)C2 Cc1cccc(CC(=O)N(C2CC(NC(=O)CC3CCC3C(=O)O)C2)C)c1F CCCC(C#N)C(=O)N1CC(F)(F)CC1CNC(c1cc(OC)nn1C)=O C1(CNC(CNC(C)=O)=O)C2CN(C(c3cn(C(F)F)cn3)=O)CC12 c1(Nc2ccc(C(C)C(=O)OCCN(C)C)cc2)nc2c(Cl)cccc2o1 C1(C(=O)NC(C)Cc2nccs2)CCC(C)CN1C(=O)CCn1cccn1 C1(C)(C(=O)NCC2N(CC)CCC2)CCCN1C(C1CCCC(F)C1)=O c1(C(N2CC(CNC(CNC(CC)=O)=O)C(C)C2)=O)cnn2ccc(C)cc12 C1(C(N2CC(NC(C(c3c(C)ccnc3)(C)C)=O)C2)=O)COCC(=O)N1C(C)C CCCC(CC)CC(=O)N(CCCNC(=O)C(c1ccc(F)cc1)(C)O)C(C)C C(C)(N=c1cc[nH]c2ccc(OC)cc12)c1c(OC)nccc1 Cc1ccc(C)n1CC(N1CC2(NC(C3CCCC(C(F)(F)F)C3)=O)CC1C2)=O c1(C(=O)NCC(C)(O)CNC(=O)Cc2cc(Br)cs2)ccncc1Cl C(=O)(C(F)(F)CC1CCCC1)N(CCOC1CN(C(C2(C)C(C)C2)=O)C1)C1CC1 c1(C(=O)NC2CC(OC)CN(C(C3(CSC)CC3)=O)C2)[nH]cc2c1CCS2(=O)=O C(=O)(C1=CC(C)(C)C1)N(C1CCC(NC(c2c(N(C)C)nccn2)=O)C1)C C1(CC(=O)NCC(CNC(CCCOCCOC)=O)(C)O)CC2CCC1CC2 N1(C(CCCCCC)=O)CC(OC)C2CCCCC12.C(=O)(CC(=O)O)OC(C)=O c1(NCCN(C(c2ccc(C)nc2)=O)Cc2ccccc2)ncc(C#N)cc1C N1(C(CN2CC(C)(OC)C2)=O)CC2CC1CN2C(c1ccc(N)c(Cl)n1)=O C1(C)(CNC(C2(C)COC(=O)N2)=O)CN(C(=O)C=CCN2CCCC2)C(C)(C)C1 N1(C(C(CC=C)C)=O)CCN(C(c2cccc(COC)c2)=O)C(CCO)C1 N#Cc1c(Cl)nsc1NC(C1CCCC1)CNC(=O)CC1CCC(=O)N1 N1(C(CCc2nc(C)sc2)=O)CCC(O)(CN(C(=O)C(F)C2CCOC2)C)CC1 NC(=O)CCCCC(=O)N1CCC2CCCC12CNC(=O)CN1CCC(=O)NC1=O C=CC1CCCN(C(c2cc(CNC(=O)C(C)(C)C(F)F)ccn2)=O)C1 Cn1[nH]c(=N)c(Br)c1C(=O)NC1CC(C(F)(F)F)CC(C(F)(F)F)C1 N1(CC)CCCC(CC(=O)Nc2cccc(Cl)c2)C1.N12CCC(C)(C1)C2=O C1(CNC(C(CC=C)(C)C)=O)CCC12CCN(C(=O)C(C)CF)CC2 Cc1ncsc1CC(=O)N(CCNC(=O)Cn1ccc(C2CC2)n1)C(C)C n1(CCOC)nc(C2Cc3ccccc32)nc1-c1cc(C)nnc1C C1(NC(C2CN(C)C2)=O)C2CCC1N(C(=O)CCC1CCCC(=O)N1)C2 Cc1[nH]c(=N)ccc1C=CC(=O)NC1CC(NC(c2ccc(Cl)[nH]2)=O)C12CCC2 c1(CCC(=O)NC2C3CC2N(C(c2ccc(CF)cc2)=O)C3)nnc(S)nc1O N1(C(c2nccc(N)c2)=O)CCCC1C1CCCN1C(c1cc(Cl)no1)=O CC1CN(C(c2ccc(Cl)cc2N)=O)CCCN1C(=O)CSc1nc[nH]n1 N1(C(Cn2c(C)cc(C)n2)=O)CC2(CC(CC(N3CCC(F)C(F)C3)=O)CO2)C1 c1(C(=O)NCc2c(C)cc(N(C)C)cc2)cc2nncn2cn1 N1(C(C(n2cnc(C#N)n2)CC)=O)CCN(C(C2CC(C)(O)C2)=O)CC(O)C1 C(=O)(C1CCCn2cnnc21)NCCC1(NC(Cc2cc(C)[nH]n2)=O)CC1 c1(OC)n[nH]c(C(=O)NC(C)(C)CN(C)C(C2CCC(=O)N2C2CC2)=O)c1Cl c1(OCC)cc(C(=O)NCC2CC2NC(=O)CN2CCCC2)[nH]n1 C(=O)(C(CC(F)F)NC(=O)C(C)NC(N)=O)NC(CC)C(C)O CP(C)(=O)c1cnc(C(=O)NNC(=O)c2cnccn2)cn1 c1(NC(C)=O)cccc2c1C1CN(C(c3nc(C)ccc3C)=O)CC1O2 C1(C2N(C(C3(OCC)CCC3)=O)CCC2)CCN(C(=O)CC(C)CN(C)C)CC1 C1(C(=O)NC(C(CO)NC(COCCOC)=O)C)CC2CCCC12 C=C(C)CC(C)C(=O)N1CCCC(N(C(=O)CCc2ccc(Cl)c(Cl)c2)C)C1 c1(C(=O)NCCCCC2CC2)ccc(Cl)c2occc12 c1(C(=O)NC2CCN(C(C3CCC(C(=O)OC)C3)=O)C2)ccccc1C(C)O C1(N(C)CC2(C(=O)OC)CC2)CCCCN(Cc2c(C)noc2Cl)C1 C(CC(C(C)C)NC(=O)C(F)n1cccn1)N(C(CCCSC)=O)C C1(C(=O)OCC)CN(C(=O)NCc2cnc3n2CCC3)CC2(CCC2)O1 c1(CC(N2CC(C)C(CNC(c3ccc(Cl)s3)=O)C2)=O)coc2cc(F)ccc12 C1(CNC(C2(OCCO)CC2)=O)CC2COCC2N1C(=O)CCNC1CCOCC1 CC(C)CCOC(C)C(=O)N(CC(C)(C)NC(=O)COC1CCOC1)C N#CC1(C(=O)NCC2C3CN(C(=O)CCc4cncc(F)c4)CC23)CCOC1 c1(NCCOc2ccc(C#N)cn2)ccc(S(=O)(=O)N2CC=CCC2)cn1 c1(CC(N2CC3C(C(=O)Nc4cnc(Br)s4)(C3)C2)=O)cccc([N+](=O)[O-])c1 C1(CNC(C2N(C)CCC2)=O)CN(C(=O)CC2COCCN2C)CC2(CCC2)O1 CC1CCOC(C2C(C(=O)NC3CCCC3)C2(C)C)C1.C1CO1 C1(NC(C#C)=O)CC2CCC(C1)N2C(c1ccc(-c2ccccc2)nc1)=O C1(CNC(CC(=O)OCC)=O)CN(C(C2CC(C)OC2C)=O)CC1C C(=O)(CCCC(C)(F)F)NC(C1CCN(C(CSc2cccc(C)c2)=O)C1)C CC1CC(N(C(=O)CC2(NC(C3CS(=O)(=O)C3)=O)CCC2)C)CC(C)C1 CC(C)CCC(F)C(=O)NCCCCC1(NC(c2ccnc(O)c2)=O)CC1 c1(C(N2CC(C)(NC(=O)CC3CC4COCC34)C2)=O)cc(N)c(O)c(F)c1 N1(C(CC2(N(C(C3CC4(CC(C)C4)C3)=O)C)CC2)=O)CCC2(CCC2)CC1 N(C1CCCc2nc(Cl)ccc21)CCc1c[nH]c2ccc(C)cc21 C1(NC(c2ccc(COC)o2)=O)CCCC(C(=O)NC2CCCCCC2F)CC1 N1(C(=O)C=Cc2ccc[nH]2)CCC(C(N2CC3CC2CS3)=O)(CF)C1 N1(C(c2c(CNC(C=CC(CC)C)=O)c[nH]n2)=O)CCc2ccsc2C1 C#Cc1ccc(C(N2CC(CNC(C3(CCF)CC3)=O)CC2C)=O)cc1F c1(N(CC(F)Cl)C)[nH]c(=NCc2ncc3c(n2)CCC3)nc2scnc12 C1(CC(=O)NC(CCC=C)C2CC2)C2CCCC2N1C(c1ccc(C)cc1F)=O CCCCCCOCC1CCN1CC(=O)Nc1nnc(CC)s1 c1(NC(CCN(CC(N)=O)C2CC2)=O)cc(C(F)(F)F)cnc1O Cc1cc(C(=O)NC2(CNC(c3cccnc3Cl)=O)CCCCC2C)cc(O)c1 C1(CC#C)(C(=O)NC)CCCCC1.c1(CC(=O)NCCN2CC2)cn(C)cn1 c1(C(=O)NC(C)CCCNC(=O)CCCN2CCCC2)c(O)ccc(F)c1Br c1(OC)cc(CC(=O)N(CCCCNC(=O)C(C)OC(C)=O)C)ccn1 C1(NC(CS(C)(=O)=O)=O)CC2CCC1N(C(=O)Cc1ccc3c(c1)OCO3)C2 Nc1ccc(Cl)c(C(N2CCC(NC(c3nncn3C3CC3)=O)C(F)C2)=O)c1 CCC(CC(=O)OC1CCCC(OCC)C1)C1C(NC(=O)OC(C)(C)C)CCC1 O=C(CC(F)F)NC1CCCC1CNC(C1CS(=O)(=O)C1)=O c1(N(C)C)cncc(NC(=O)CC=CCNC(=O)CC2(O)CCOC2)c1 c1(CN(C(N2CCC(=C)CC2CC)=O)CCO)c(C)ccc2ncccc12 C1(CNC(c2ccc(CC)s2)=O)CC(C)N(C(c2ccc(C(N)=O)cc2)=O)C1 c1(C(=O)NC2(CNC(C3C(C)CCC3)=O)CCC2)cnc2[nH]cnc2c1 n1(OC)c(CNC(=O)C=CC(C)(C)NC(=O)CCOCC2CC2)cnc1C Cc1ccc(C)c(C(N2CC3(CC3)CC2CNC(=O)C(C)C(C)C)=O)c1O c1(C(=O)NCC(CO)NC(Cn2c(C)csc2=O)=O)cc2cccnc2[nH]1 C=Cc1ccc(C(=O)N(C2CC(NC(c3c(Cl)ccnc3C)=O)C2)C)cc1 C=C(C)CC(C(=O)NCCOCC(N)=O)NC(=O)CCc1cnco1 C1(C(C)C)CN(C(=O)NCC(C)(C)Oc2cccc(F)c2)CC1N(C)C Cc1oc2ccccc2c1S(=O)(=O)N(C(C(=O)NCCCF)C(C)CC(C)C)C Cc1cnccc1C(=O)NC1CCCC1CC(=O)Nc1cccc(CN(C)C)c1 N1(C(=O)OC)CC(CNC(=O)CC2CC(C(F)(F)F)C2)C1 N1(C(c2cc(OC)no2)=O)CCCC12CN(c1ccc(C(F)(F)F)nn1)C2 C(=O)(CCCC(F)F)N(CCCNC(=O)COC1CC1(F)F)C CC(C)(CN=c1[nH]c(=NCc2cn3ccccc3n2)[nH]c2ccsc12)CC(F)F C1(N(C(N(CC(c2ccccc2)C)C)=O)C2CC2)CC2CC2C1 c1(C(=O)NC(C)C(CO)NC(=O)CC#N)cccc(OC2CCC2)c1 C1(CC(=O)NC2CCCCN(C(=O)Cc3nc(O)n[nH]3)C2)CC2(CCCC2)CO1 N1(C(c2ccc(N)cc2F)=O)CCC2C(C1)CN2C(=O)CNC(=O)C(F)(F)F Cc1nc(CC(C)C)oc1C(N1CCC(c2cn(-c3cccnc3)nn2)C1)=O N1(C(C)=O)CCC(C2CCN(C(c3cn(CCC4CC4)nn3)=O)CC2)CC1 c1(C(=O)NC2CC(CNC(C3CC=CC3)=O)C2)sccc1Br c1(CC(C(=O)NC(CC(C)NC(c2c(CC)csc2)=O)C)C)ccccc1F c1(CN(CC=C)C(c2nc(C(=O)OC)cs2)=O)ccc(OC)c(OC)c1 N1(C(C(C2CCCCC2)OC)C(=O)NC(C)(C)C)CC2CC(O)CC2C1 c1(C(=O)NCC2(O)CN(C(C3OCC(C)C3)=O)C2)ccc2c(c1)CC2 c1(NC(CN(CC(C)C)C(=O)CN2CCC(CC3CC3)C2)=O)ccncc1N C1(C2CC2)(NC(CCNS(C)(=O)=O)=O)CCN(C(C2CCNC2=O)=O)C1 c1(C(N2CCN(c3nnc(O)s3)CC3(CC3)C2)=O)ccc2c(O)nnc(O)c2c1 N(C(=NCc1cccc(F)c1)NCCN1CCC1)CC1(CCOC)CCCC1 C1(NC(C2CC(C#C)(O)C2)=O)(CNC(c2ccc(OC)nn2)=O)CCCCC1C c1(NC(=O)OC)ccc(-c2nc(CC(N3CCCCC3CC3CC3)=O)cs2)cc1 Cn1cccc(C(=O)NC2(C(=O)NC3(C)CCCOC3)CCSC2)c1=O N1(C(c2nn(C(CC)CC)c(C)c2)=O)CC(C)CN(C(C2CSCCS2)=O)CC1C C1(OC)CC(NC(C2(CO)CC2)=O)CN(C(c2csc(-c3ccco3)n2)=O)C1 c1(C(=O)NCC(C(N2CC3C(C(N)=O)(C3)C2)=O)O)cccc2cc[nH]c12 N1(C(CCCCSC)=O)CCOCCC1C(=O)N(C)CC1COC(=O)N1 n1(CC)c(C(=O)NC2COCCC2NC(=O)C(C)C(=O)OC)cnc1O N1(C(C2(C=C)CCC2)=O)CCCC(C2(NC(c3cnc(C)c(C)c3)=O)CC2)C1 CC1CN(C(=O)COC2(C)CCC2)C(C)CN1C(=O)CN1C(=O)CN(C)C1=O c1(C(=O)NCC2CC(NC(C(C)n3cccn3)=O)C2)cc(C#N)c[nH]1 c1(C(N2CC(C(C)NC(C3C(C)C3)=O)C2)=O)csc(-c2cccnc2)n1 N1(C(CC(=O)N(C)C)=O)CCN(C(c2cnccc2Cl)=O)C(C2CCC2)C1 C1(CC#C)CN(C(c2cn(CCNC(=O)CCn3cnnn3)cn2)=O)CCO1 CCC(CC(=O)NC(C1(C(=O)NC(C)C(C)(C)CN(C)C)CC1)C)OC CC1COC(C(N2CC(F)(C(=O)N(CCCCCO)C)C2)=O)C1 N1(C(c2n(C3(C)CC3)ccn2)=O)CCC(O)(CNC(=O)CCN2CCCCC2)C1 C1(O)(CNC(c2ccn(CC)n2)=O)CCCN(C(C2Cc3nnsc3S2)=O)CC1 Nc1c(C(=O)NC2(C(F)(F)F)CCCCC2C(F)(F)F)cc(F)cc1C(F)(F)F C(=O)(C1CCc2c[nH]nc21)N1CC(N(C(C(C(C)C)SC)=O)C)C1 C1(OC)CC2(CCN(C(C3CC(O)CCN3C(=O)CC(C)O)=O)C2)C1 N1(C(=O)OC)CC(C(=O)NC2CCC(C)O2)CC(CC#N)C1 CC1CCC(NC(C2CC(N3CCCC3)C2)=O)CN1C(c1ccc(C(F)F)s1)=O N1(C(CN(C(=O)OCC)C)=O)CC2CCC1C(NC(=O)CC1CC(F)(F)C1)C2 C12(C(N(CC(CN(C(Cn3c(C)ncc3)=O)C)O)C)=O)CC(C1)C(C(F)(F)F)O2 C1(CC)CC2CCC(C1)N2C(C1CCC(CNC(c2ccncn2)=O)C1)=O c1(N(C(=O)C(C2CCN(C(C3CCSC3)=O)C2)F)CCC)ccnc(C)n1 c1(CC)nn[nH]c1C(=O)NC(C)CNC(C1(NC(N)=O)CC1)=O C(C)(CC)(CCNC(C1CC(N=[N+]=[N-])C1)=O)NC(CCOCCOC)=O N1(C(C2CC(C#C)(O)C2)=O)CCC2(NC(c3cncc(Cl)c3)=O)CCCC12 N1(C(Cc2c(C)ncs2)=O)CCOC(CCNC(c2ccc(Cl)s2)=O)C1 c1(C2(CC(=O)N(C(C)CN(C(=O)CCSC(F)(F)F)C)C)CC2)ccccc1 Cc1cc(O)cc(=O)n1C(c1nc(C2CCCC(F)(F)C2)no1)C1CCCC1 C#CCC(C(=O)OC)NC(C1CCCN(C(C2CC=CCC2)=O)C1)=O C1(C(C)(F)F)(NC(CNC(=O)OC(C)(C)C)=O)CCOCC1.N12CCCC(C1)C2=O C1(NC(CC(N2C(=O)CCC2=O)C)=O)CN(C(=O)CC2CN(C)C2)C2(CCC2)C1 c1(C(N2CCC(N3CCN(C(CCCSC)=O)CC3)C2)=O)ccnc2ccsc12 N1(C(C2C(C)C2c2ccccc2)=O)CC2CC1CN2C(c1cc(Cl)sc1Cl)=O C(CN=c1[nH]c(=NC(C)CCC2CCCO2)[nH]c2c1CSC2)c1c(C)ncs1 CC1C2=CC(=O)N(C)C(C)CN(C)C(=O)CC(COCCO)CCCCCC12 N1(C(C=CC(CC)C)=O)CCC(CN(C(=O)C(C)OCCOC)C)CC1 CCC(C#N)C(=O)N(CC(=O)NCC(CC(C)C)NC(C)=O)C(C)C c1(OC)nc2cc(NC(N3CCCC(c4nccn4C)C3)=O)ccc2o1 C(=O)(C(F)CCC(C)(C)C)N1C(C(=O)N(C)CC2CCCOC2)(CC)CCC1 CC1(C)COCCC1C(=O)NC1(C)CCN(C(C2CC3CC(=O)C2C3)=O)C1 C1(C(=O)NCCN(C(c2cc(C3CCCC3)[nH]n2)=O)CC)CCc2nnc(O)n2C1 c1(C(N2C(C(=O)NCCC3(COC)CCC3)COCC2)=O)cncc2[nH]ccc12 c12nc(nn1-c1ccc(CCC(C)C)cc1)CNC2.C(C(C)C)N(CCOC)C N1(C(C2(NC(C3C(=C)C3C(=O)OCC)=O)CC2(C)C)=O)CC(OC)C(F)C1 C(=O)(C(CC)(CC)C(=O)O)N1CCN(CC(N2C(CC)C=CC2)=O)CC1 c1(C(=O)NC2(COC)CN(C(c3cc(COC)on3)=O)C2)cc(C)ncc1C N1(C(C2NC(=O)CC2Cc2cn(CCF)nn2)C)CCCC1(C)c1ccccc1 c1(C(=O)NCC(CNC(COCCC(C)C)=O)C(F)(F)F)ccc2cnoc2c1 N1(C(CC=C=C)=O)CC2(CCC2CNC(c2cccnc2NCC(C)C)=O)C1 C(=O)(C#CC1CCCO1)NC1(CO)CCN(C(CNC(CNC(C)=O)=O)=O)C1 N1(C(C2(C)CNC(=O)C2)=O)CCCC(F)(CNC(c2sccc2C2CC2)=O)C1 N1(C(Cc2c(C)nc[nH]2)=O)CC2(CC(NC(=O)COCC3CCC3)C2)C1 N1(C(CCc2ccc(C)c(Cl)c2)=O)CCC2CCCC12C(=O)O C#Cc1cc(C(=O)NC2CC2CNC(=O)C2=C(Cl)CCC2)cc(C(F)(F)F)c1 C(C(O)C(=O)NCC(C(C)C)NC(=O)C=CC(C)C)SC C=CCC(F)(F)C(=O)NC1CCN(C(c2cc(CN(C)C)c[nH]2)=O)CC1O C(=O)(CC(C)C(C)(C)NC(c1cscc1Cl)=O)N(C(C)C)CC Cc1ccc(C(N2CCSCC2)=O)cc1Nc1ncc(Br)cc1C(F)(F)F CC(C)(COC(=O)C(=O)Nc1ccc(OC(F)F)cc1)CC#N N1(C(C(CCC)O)=O)CC(NC(=O)C(C)SC(C)C)CC12CCOCC2 CC(C)CC(CC(=O)NCC(C)(C)CN(C)C(C1CCC1C(F)F)=O)CC(N)=O c1(C(CC)NC(C2(CCNC(=O)C=CCO)CC2)=O)cn(C)nn1 C1(C(=O)NC2CN3CCC2CC3)CCC2CCC1N2C(C12CCCC1C2)=O N1(C(C2N(CCC)C(=O)CC2)=O)CC2CCN(C(C3(OC(C)=O)CC3)=O)C2C1 C(=O)(C(C)NC(C1(C(C)NC(C2CC2C(N)=O)=O)CC1)=O)NC C(=O)(CCCCN1CCCC1)C(CC)=O.C(=O)(C(C)CSC)NCC(C)NC C(=O)CCCCNC(=O)NC1(C(N(CCOCC)C)C)CC1.c1(C)ccc(C)cc1 C1(CC#C)(NC(c2cn(CCNC(C3CCC3)=O)nn2)=O)CCCCC1 CC12CCC(C(N3CCC(CNC(=O)Cc4ccc(F)cc4Cl)C3)=O)(C1)OC2 N1(C(CNC(C(CC=CC)C)=O)=O)CC(=O)NCC1C(C)C C12(C(=O)NC(C3CCCN(C(c4cnnn4C(C)C)=O)C3)C)CCCCC1C2 CCCCCC(O)CC(=O)NCC1=CCN(C(=O)Cn2ccc(=N)[nH]2)CC1 C1(C(=O)NCC2(COC)CN(C(=O)CCCc3ccc(C)cc3)C2)COCCC1C CC(CN(C)C)CC(=O)N1CCCC(C(C)(C)C(=O)NCC2CCCSC2)C1 C1(CC(=O)NCCC(=O)OC)C2CCCC2N1C(=O)Cc1cncs1 C1(C(N2C(CNC(c3cccnc3)=O)C3CCC2C3)=O)COc2ccccc2C1 N1(C(CC(=C=C)C)=O)CC(CNC(=O)Cn2ccccc2=O)C2(CC2)C1 C(C)(C(C)(C)C(=O)N1CC=CC1)NC(COCC(=O)NC)=O Cc1nc(O)ccc1C(N1CCC(C(C)NC(C2(F)CCS(=O)(=O)C2)=O)CC1)=O Cc1nc(C)n(O)c1C(=O)NC(CNC(c1ccoc1Br)=O)CC(F)(F)F c12cc(ccc1C)C(=O)C(=O)NC1CC1O2.N(CCOC)(CC)CC Cc1cnc(CCCC(=O)NCC2(F)CC(NC(=O)C(=O)N(C)C)C2)o1 C1(NC(CC2(C)CCCC2)=O)CCCCN(C(=O)CC2CCC3(CCC3)O2)C1 C1(C(N2CC(O)(C(C)NC(CSCCCC)=O)C2)=O)C(C(F)(F)F)C1[N+](=O)[O-] c1(C(=O)NCC=CC(=O)NC(C2CCCOC2)CC)c[nH]ccc1=O N1(C(c2csnn2)=O)CCC(C(F)(F)F)(CNC(C2CC2C(F)(F)F)=O)C1 C1(NC(Cc2c(C)ocn2)=O)CC(CNC(=O)CC(C)C2CC2)C(O)C1 C1(C(=O)NCC(CC=C)NC(c2ccc(NCC)cc2)=O)CCCC(C)(C)CC1 N1(C(C(=O)NCC(=C)C)CCSC)CCCC(C(C)C)(CO)C1 C1(C)(CC)CC(NC(=O)CCOC)CN1C=O.c1(N2CC(N)C2)ccccc1Cl C1(C(=O)NC(C(=O)NC)(C)C)CC2CCC(C1)N2C(=O)CC(C)P(C)(C)=O C1(NC(Cc2cc(C)n(C)n2)=O)CN(C(c2cnc(N)c(Cl)c2)=O)CCC1(C)C n1(CCN(C)C)cc(C(=O)NCCCCNC(=O)C=Cc2ccsc2)nn1 Cc1nc(C(N2CCCC2C2(C(=O)NC)CC2)=O)cs1.c1(S)cncs1 c1(C(=O)NCCC2CC(NC(CSCCC)=O)C2)cc(COC)on1 Cc1cc(C(N2CC3(NC(c4cc(CF)no4)=O)CC2C3)=O)ccc1C(F)(F)F Cc1cc(C(N2CCCC2CN(C(=O)CN(C)C(N)=O)C2CC2)=O)nn1C CC(C)C(C)(O)CNC(=O)C(CCOCCO)NC(c1ccsc1Cl)=O [N-]=[N+]=NC1CCCN(C(C2(NC(C3C4CC5C(C4=O)C35)=O)CCSC2)=O)C1 Cc1oc2ncn(C)c(=O)c2c1C(=O)OCC1=NOC2COCCC12 n1(CC)c(C(=O)NC2CCC(CNC(=O)C(C)N(C(=O)COC)C)C2)cnc1O C=CCC(C)(CC)C(=O)NCC(F)(C(=O)NCCC1CC(C)=NO1)C(C)C N1(C(C2CC2F)=O)CCC(C2CCN(C(=O)C(C3CCOCC3)F)CC2)CC1 c1(C(N(CC(C)N(C)C(C2CC3CCC2O3)=O)C)=O)cnc2c(n1)CCCC2 N1(C(c2cnc(CSC)s2)=O)CCC(NC(=O)COCc2cccnc2)C(C)C1 N1(C(=O)Nc2ccc(Oc3c(C(C)C)cccc3)cc2)CCC2(C1)CC2(F)F c1(SCC2CC(C(=O)NCCc3c(C)cccc3Br)C2)c(Cl)cc(C#N)cc1Cl c1(C(=O)Nc2c(S(C)(=O)=O)csc2)ccc2c(-c3cnn4c3SCC4)n[nH]c2c1 c1(NC(=O)NC2C(C)(c3ccccc3)CC2)cnn2ncccc12 C1(CCCNC(CCn2c(C)ncc2)=O)CN(C(=O)CC2CSC2)CCO1 c1(C(N2C(CCNC(Cc3cc(C)on3)=O)CCC2)=O)ncc([N+](=O)[O-])n1C c1(C(N2C(C)(CNC(Cn3nnc(C)n3)=O)CCC2)=O)cnc2c(c1)COCC2 N1(C(CC2N(C(c3c(CC)cno3)=O)CCC2(C)C)=O)CCC2(CC1)CC(O)C2 c1(CSCC)ccc(C(N2CC(OC)CC2CNC(=O)CC2CCCO2)=O)cc1 Cc1nc(S)sc1CC(=O)NCC1CCC(N(C)C(C2COC(=O)N2)=O)CC1 N1(C(c2c(CC#N)cccc2)=O)CCCC(F)(CNC(=O)CC2CC23CC3)C1 C1(NC(C2(NC(CC3C=NN(C)C3=O)=O)CC2(C)C)=O)CCn2ccnc2C1 c1(N(C)CC2CCC(CNC(C(C)C(C)(C)C)=O)CC2)ncnc2scc(Br)c12 N1(C(C=CCCN=[N+]=[N-])=O)CCC2(CCN(C(c3cnnc(O)c3)=O)C2)C1 C1(C(C(=O)NCC2C(CC(=O)N(C3C(C)CC3)C)C2)O)CCCCC1 Cc1ccc(O)c(C)c1NC(=O)COCCN(C)C.C1(=O)C(CC2CCC2)N1 C(CS(=O)(=O)CC(=O)N(C1CN(C(=O)C(C)(O)CC(C)C)CC1(C)C)C)OC N1(C(C(F)=CC)=O)CC(NC(=O)C(C)Sc2ccc(Cl)cc2)CC12CCC2 N1(C(CCC=C)=O)CC2CC(NC(c3cnn(CCC)c3C3CC3)=O)CC1C2 c1(OC)cnc(C(=O)NCC(C)NC(C2CC2c2nccn2C)=O)c(OC)n1 CC1C(NC(C2(C)C=CCCC2)=O)CCN1C(=O)CCc1nc(C2CCCC2)no1 C1(CC=C)(C(=O)NCC2CCC3(CC3)C2)CCCN1C(c1nnsc1N)=O O=C(C1=C(F)CN(C(=O)CC2CCCC(O)C2)CC1)NCC1CN2CCC1CC2 c1(NC(C2(C)N(C(c3nc(C)c(F)cc3)=O)CC2)=O)c([N+](=O)[O-])ccc(F)c1F C(=O)(C1CC(=O)Nc2ncn(C)c21)NC(C)CNC(=O)CC1CCCC1 C1(C)(C(=O)OCC2(CCN3C(C)COCC3)CC2)COC(=O)OC1 C(=O)(CC(C(F)(F)F)NC(c1n[nH]c(C)n1)=O)NC(COC)C(C)C C1(CC)CN(C(c2sc(C)cc2Cl)=O)CCN1C(=O)CC1CC1CF N1(C(C2(OC)CC2)=O)CCC2(CC1)CC2NC(=O)C(C(C)C)SC c1(C(=O)NCC2C(NC(c3c(C)nco3)=O)CCC2)nnc2n1CCCC2 N1(C(=O)Nc2cc(OC(CC)C)no2)Cc2ccc(C(=O)OC)cc2C1 CC1CN(C(=O)CCOCC2CC2)CC1(C)CNC(=O)CC1CCOCC1 C1(C(=O)NCCCN(CCC)C(c2cncc(F)c2)=O)CCCC(=O)N1 C(=O)(C(C)=Cn1ccnn1)NCC1CN(C(C(CCSC)O)=O)CC1(F)CO N1(C(C23C(CN(C(CC(=O)OC)=O)C2)C3)=O)CC2CCCCC2C1 c1(OC)ccc(N)c(C(=O)NC2CCN(CC(N3CCCC(N)C3)=O)C2)c1 C1(COC)(NC(c2c(C)nsc2NC)=O)CCN(C(c2ncn(C)c2C)=O)CC1 C1(F)(CNC(c2csc(-c3ccco3)n2)=O)CCN(C(C2(CF)CC2)=O)CC1 C1(NC(CC(=O)NCC)=O)CC12CCN(C(c1cc(C#N)n(C)n1)=O)CC2 C1(NC(=O)CC2CCS(=O)(=O)C2)(CO)CCCN(c2ncncc2I)C1 C(C)(C)(C(=O)N(C(C)CCNC(=O)C(n1ccc(C2CC2)n1)C)C)OC C(=O)(N=c1cc(C)nc(Cl)[nH]1)C1CCCN(c2ccc(SC)c(C(F)(F)F)c2)C1 C1(CC(=O)NCCN(C(C2(C)CC2F)=O)C2CC2)(COC)CCOCC1 N1(CC(=O)N(CCC)C)CCN(C(=O)COC(C)=O)CC1 c1(C(=O)NCC2N(C)CCN(C(C(C)c3cccs3)=O)C2)cccn2ncnc12 N1(c2n(CC)c(CCSC)nn2)CC(F)(F)CC1C N1(C(c2c(COC)scc2)=O)CC(NC(C2C3C4CCC(C4)C23)=O)CC2(CC2)C1 C(=O)(C(C)(C)CS(C)(=O)=O)NCC1(NC(C(CCOC)C)=O)CCOCC1 C1(NC(C=CC)=O)COC2(C1)CN(C(c1ccc(OC3CCOCC3)nc1)=O)C2 N1(C(C2CCSC2)=O)CCC(C(F)Cn2cc(-c3ccc(CO)s3)nn2)CC1 c1(NC(CCC(=C)Cl)=O)cc(C(F)(F)F)ccc1C#CC CCS(=O)(=O)CCNC(=O)C=CCC(C)(C)NC(C1CCOC1C)=O Cc1[nH]nc(C(N2CCC(C(C)NC(c3scnc3C(F)(F)F)=O)C2)=O)c1Cl C(=O)(C1=NOC2(CCC2)C1)N1C(C)(C)C(CNC(C2(N3CCCC3)CC2)=O)CC1 c1(NCC(=O)OCCOc2cccc(C)c2C)cc(N)nc2ccnn12 C1(C)(C(N2CCCCC(N(C(CCCC)=O)C)C2)=O)CCC(F)(F)CO1 C12(C(=O)NCC(C)NC(C3CCCN3C)=O)CCC(=O)N1CCS2 C1(NC(C2CC(NC(c3cc(COC)no3)=O)C2(C)C)=O)CCOCC1(C)C c1(CC(C)C)c(C(=O)NCC2CCCC2NC(C2(CO)COC2)=O)cnn1C Cc1cc2c(C(=O)NCCc3cc(Br)sc3Br)cccc2o1 c1(C(=O)NCC2CCN(C(C(C)n3ccnn3)=O)C2(C)C)cccc2ccoc12 N#Cc1ccc(F)c(S(=O)(=O)N2CCC(F)CC2C(=O)NNC(=O)C2CC2)c1 C1(C)(NC(C2CN(C(C)C)C2)=O)CCN(C(C2CCCC(C#N)C2)=O)CC1 CC1CCOC(C(=O)NC(CCF)C(=O)NCc2cc(C(C)C)n[nH]2)C1 CCC(CC(=O)N1CCOC(C)(C)C1)C(C)(C)C.C12CCC1C(=O)N2 c1(CC)nc(C)n(C)c1C(=O)NCCC1CCN(C(=O)C=C(C)c2cccs2)C1 C1(CNC(CC=C)=O)CCC(C)N(C(=O)C=CC(=O)Nc2cccc(F)c2)C1 C(c1ccc(O)cc1)=CC(N1CC(CNC(c2ccc(F)o2)=O)C1)=O C1(NC(CN(C(c2cc(CC)[nH]n2)=O)C2CC2)=O)CC(C(N)=O)C1(C)C c1(CCNC(C2N(CC)CC2)=O)cccc(CNC(=O)CCC2CC2(F)F)c1 C1(NC(Cc2ccc(SC)cc2)=O)CN(C(=O)CCCF)CCC1C C(=O)(CC(C)(C)NC(C1CC2CCC2C1)=O)NCCC=C N1(C(C(=Cc2ccccc2)CC)=O)CC=C(CCNC(=O)C(C)SC(=N)N)CC1 CC1(C)CN(C(C2CC2F)=O)CCC1NC(c1cscc1Br)=O c1(OC2CCN(CC3N(c4cn(C)nc4)CCCC3)C2)ccc(F)cc1F N1(C(C(CCC)OC)=O)CCCN(C(c2cc(C#N)on2)=O)C(CO)C1 C1(CCOC)CN(C(C2CCCNS2(=O)=O)=O)CCN1C(=O)CCc1nc[nH]n1 CC1(C)C(=O)CC1C(N1CCCC(NC(C2CCCN2CC2CCC2)=O)C1)=O CC1CCC=C1C(=O)NC12CCC(C1)N(C(=O)Cn1cnc(Br)c1)C2 c1(C(N2CCCC(Cn3cc(C(C=C)(C)O)nn3)C2)=O)ccc([N+](=O)[O-])cc1Cl C1(NC(=O)CC2CC(F)(F)C2)CC2CC(NC(=O)COc3cc(F)cc(F)c3)CC12 c1(C(N(C(C)CNC(=O)CN(C2CCCCC2)C)CC)=O)cccc(F)c1N c1(CC)ccc(F)c(C(=O)NC2CC(CNC(=O)C(C(C)CC)OC)C2)c1F N1(C(c2c(C)scn2)=O)CC(NC(=O)CCC2COC(C)(C)O2)CC12CCCCC2 C(C)(CCCNC(=O)Cc1ccsn1)NC(CCN(C(CCC)C)C)=O Cc1c(C(=O)NCC(C)(C(C)C)NC(=O)CCc2ncc[nH]2)ccn1CCO N1(CCNC(=NC)NCC2(C)CC2)CCCC2CCCCC12 C#CC(C)(C)C(=O)N(C)CCN(C(=O)C(C)(F)F)C C1(CS(=O)(=O)NC)CCCN(C(C2CCC(NC(=O)OC(C)(C)C)CC2)=O)C1 N1(C(C(CCC)C)=O)CCC(C(=O)OC(C)=O)C(C)C1 c1(-c2ccc(C(C)(C)C)cc2)sc2c(c1C(=O)NCc1cccc(F)c1I)CCC2 N1(C(=O)C=CC2CC2)CCC2(CCCN2C(c2cnn(CCO)c2)=O)C1 N1(C(c2c(OC)cccn2)=O)CCCN(C(c2n[nH]cc2Cl)=O)CC1C(C)C N1(C(c2n(CCOC)ncc2)=O)CCN(C(c2cc(C)c(Br)s2)=O)C2CC12 C=C(C)CC(C(=O)N(CCCN(C)C)C)NC(=O)CN(C)CCN(C)C C1(O)(CNC(CN(C2CCSC2)C)=O)CCN(C(=O)CCCn2cncn2)CC1 N1(CCC(=O)NCC2(C(F)(F)F)CCCCO2)CC2CN(c3nncs3)CC2C1 CC1CCCCN1CC(=O)NCCCN1CCN(C(=O)CN(S(C)(=O)=O)C)CC1 C=C(Cl)CCC(=O)NCCN1CCN(C(C2CC2Cc2ccco2)=O)CC1 CC(C)(C(=O)NC1CN(C(c2cnccn2)=O)CC(F)(F)C1)C(F)(F)F O=C(C1c2c[nH]nc2CN1C(=O)CCC1CCCO1)NCC(F)C1CCC1 Cc1cc(Cl)cc(C(=O)N(C2CC(NC(=O)CCC(C)(C)C)C2)C)c1O N1(C(C2(C)CC2C(F)(F)F)=O)CC2(CCOCC2)CC1CNC(=O)COC(F)F C1(C(C)C)C(NC(=O)Cn2cc(C3CC3)nn2)CCN1C(=O)Cc1c(C)noc1Cl N1(C(C(c2cccc(C)c2)C)=O)CC(O)(C2(CNC(C3CCC(=O)N3)=O)CC2)C1 N1(C(C(CNC(CCc2cc(C)[nH]n2)=O)CC2CC2)=O)CCS(=O)C(C)C1 C1(C(=O)Nc2ccc(I)o2)CCCN(CCO)CC1.CC12CCN1C2 c1(C(N2C(c3n(C(C)C)ncc3)CCC2)=O)ccc2c(c1)OCC(=O)N2 CN(C)NC(=O)CCC(=O)NC1C=CC(CC(=O)NCC2CN3CCC2C3)C1 c1(CCO)cccc(F)c1F.CON(C)C(=O)CNC(=O)C(CCOCCO)NCCO c1(C(N(C2CCN(C(CCCC)=O)C2)C)=O)cccc2c(C)[nH]nc12 c1(CNC(Cc2scc(C)c2)=O)nc(C)c(C(=O)NCCC2CC(=O)N(C)C2)o1 CC(C)(CCNC(=O)COc1ccsn1)NC(C1COC1)=O C12(CC(=O)NC3CC(C(C)NC(c4cc(Cl)c[nH]4)=O)C3)CCC(CC1)C2 C1(F)(CNC(c2c(C)cccc2N)=O)CCCN(C(=O)CCC(N)=O)CC1 C1(OC)(OC)CC(NC(C2CCN(C(=O)CN(C)S(N)(=O)=O)C2)=O)C1 N1(C(C)=O)CCCC2(C1)CN(C(=O)OCCc1ccc(C(F)(F)F)[nH]1)C2 N1(C(CC(CCC)(C)C)=O)CCCC(C2CCN(C(=O)C(C)(C)OC)C2)C1 c1(C(=O)NC2C(CNC(CCn3c(C)ncc3)=O)CC2)ccc2c(c1)CN(C)C2 C(=O)(CC1=CCN(C(=O)C(C)Cn2cccn2)CC1)NCc1c(C)nc(C)s1 C(=O)(C(F)CC1CCCC1)N(CCN(C(c1cnn(CC)n1)=O)CC)CC c1(C(=O)NCC2(C)CCN(C(C3C(C)C3C)=O)C2)cc(F)cc2ccncc12 C(=O)(C1=C(C)OCCS1)N1CC(CN2CCN(C(C3(COCC)CCC3)=O)CC2)C1 c1(CCNC(CCOC2CN(C(C(C3CCCC3)OC)=O)C2)=O)n[nH]c(C)n1 C1(NC(N(CC#C)CCOC)=O)CCN(C(=O)CC=CCC)C1 CC(C)C(CCNC(=O)CC(C)n1cccn1)NC(=O)CSCc1ccccc1 S(=O)(=O)(c1c[nH]ccc1=NCCCCCOC1CC1)NC(CCC)C Cn1cnc2c(NCc3ccns3)[nH]c(=NC3C=CCCCC3)nc12 N1(CC)CC(C(N2CC(NC(=O)C(O)C(C)C)C2)=O)CCC1=O c1(C(NCCCOC)=O)cc(N)cc(O)n1.N12CCCCC1C2=O CC1CCc2[nH]nc(C(N3CCC(C)N(C(=O)CC=C(Cl)Cl)CC3)=O)c2C1 C1(CNC(CCC=C)=O)(CO)CCN(C(c2n[nH]cc2I)=O)CC1 C1(NC(c2nc(CC)sc2)=O)(CNC(=O)CC2(O)CCCCC2)CCCCC1C Cn1cc(S(C)(=N)=O)c(CNc2n[nH]c(-c3ccc(Cl)cc3F)n2)n1 C(C(CC(C)C)C(=O)NCC(N1CCCC1)C)NC(C1(CC=C)CC1)=O C(=O)(NNC(=O)C(=O)N(c1cccc(C)n1)C)C1C(C)OCC1 C(N=C(NC1CCC1)N1CCC(C(C)(O)C(F)(F)F)CC1)c1cnn(C)n1 C(CCC(N)=O)(C(=O)N(CC(C)NC(c1cccc2oncc12)=O)C)NC(C)=O C(=O)(CC(C)C(C)C)NCC1(C(=O)NCC(C)OCCO)CC(=C)C1 N1(C(CCNC(=O)OCC=C)=O)CCC2C(CCCN2C(=O)C(C)(F)CC)C1 c1(C(=O)NC(C)C(c2ccccc2)NC(=O)CC(C)(C)F)ccccc1C#N c1(OC)ncc(Cl)c(=NCCCC(C)NC(C2(O)CC(C)(C)C2)=O)[nH]1 c1(C(=O)NC23CC(C2)N(C(c2cnns2)=O)C3)ccc(-c2cccs2)c(F)c1 c1(C(=O)NC)cccc(C(N2CC(C(C)NC(=O)C(C)OCC3CC3)C2)=O)n1 C1(CNC(C(CC)(C)F)=O)CN(C(c2ccccc2O)=O)CC(C)(C)C1 C(CCC=C)(C(=O)N(C1CC(F)C1)C)NC(COCC=C)=O C(=O)(CC1=Cc2ccccc2C1)N1CC(CCNC(C2CC3(CCC3)CO2)=O)C1 C1(CNC(C(=O)NCC)=O)COCCN1C(c1ccccc1F)=O N1(CC(=O)NC(C2(O)CCN(C(=O)C(O)C3CCCC3)C2)C)CCOCC1=O C1(C)(C(N(CC(C)N(C(=O)C(C)(F)F)C)C)=O)CCC2(CC1)CC2 C1(C2CC2)(NC(=O)CCc2cnc(O)[nH]2)CCN(C(=O)CC2CCSC2)C1 CC1(CNC(=O)C=CC2CCCO2)CCN(C(=O)CCCn2ccccc2=O)C1 Cc1cnc(C(=O)NC2(C3CN(C(C4CCCC(C)(C)C4)=O)C3)CC2)cc1C#N c1(C(=O)NC2(CCNC(c3c(C)nc(CO)s3)=O)CC2)cc2n(c(=O)c1)CCS2 C1(C(N(C)Cc2onc(CC)n2)=O)CSCCN1C(=O)Cc1ncoc1C CC1CCN(C(=O)C(C#N)=CC2CC2)CCN1C(c1nncn1C1CC1)=O N1(C(c2cnn(CC)c2C)=O)CCC(NC(C2CCOC(C)C2)=O)C(C)C1 C=CCC(CC=C)C(=O)N(CC(O)CNC(=O)C=Cc1ccnn1CC)C C1(C(=O)NC(c2ncn(C)n2)C)CC12CCN(C(=O)C(C)C(F)(F)F)C2 C(CC(=O)N(CCCNC(=O)Cc1ccc2nsnc2c1)C)(C(F)(F)F)OC c1(C(=O)NC(C2(O)CN(C(C(CC=C)CC)=O)C2)C)ccc2c(c1)NC(=O)NC2 c1(OC)cc(CC(=O)NCC2CN(C(c3cn(C)nc3C)=O)CC2C)ccc1F CC1CN(C(c2ccc(C3CCCO3)[nH]2)=O)C(C)CN1C(=O)CCCCCC#N N1(C(C=CS(CC)(=O)=O)=O)C2CCC1C(C)C(NC(C1CC(=O)NC1(C)C)=O)C2 c1(C(N2C3C(CNC(CSC)=O)(CCCC3)CC2)=O)n[nH]c2c(=O)n(C)cnc12 C(=O)(C1Cc2ccccc21)N1CC(NC(CC(=C)C)=O)C(CC2CC2)C1 N1(C(Cc2cccc(OC)c2)=O)CCC(CNC(=O)C=C(Cl)Cl)C12CC2 C(C)(CCC1CC1)(c1nnnn1C(C)(C)C)NCCC1(OC(C)C)CCC1 n1(CC(=O)N(C)CC2N(C(C(C)OCCC=C)=O)CCC2)c(C)cc(C)nc1=O C1(CC)CCC(N=c2[nH]c(N3CCCC(NCCSC)C3)nc3c2SCC3)CC1 N1(C(CNC(C)=O)=O)CCCC2CN(C(C3CCC(C(F)(F)F)CC3)=O)CC12 C1(CC(=O)NC(C2CCCN2C(C2CC(OC(C)(C)C)C2)=O)C)CCS(=O)(=O)C1 Cc1cc(=NC(=O)c2[nH]nnc2C(N2CC3(CCC3)C23CCC3)=O)[nH]o1 C1(NC(CC(C)C)=O)CC2(CCCN(C(c3cccc(P(C)(C)=O)c3)=O)C2)C1 CC1(C#N)CCCN(C(=O)CC2CCCCC2NC(c2n[nH]c3c2COC3)=O)C1 N1(C(c2ccc(F)c(C)c2N)=O)CCC(C2CCN(C(c3cnccn3)=O)C2)C1 c1(C(N(C(C)CNC(=O)Cn2nc(Cl)ccc2=O)C)=O)ccc(Cl)c(F)c1F c1(C(N2CC(C)C(NC(C3CC(C#N)C3)=O)CC2)=O)ccc2ncccc2c1F CCC(C(=O)NC(C)(C)CNC(c1ncoc1CSC)=O)OC1CCCC1 c1(OC)cc(CC(N2CCC(C(=O)Nc3cc(Cl)ncc3Cl)C2)=O)ccc1O N12CCC(CC1)CNCc1ncoc1C2C(=O)N.N1(CCOC)CCNC1=O Cc1cnccc1C(C)C(=O)NC1CCC1NC(c1c(C(F)F)n[nH]c1C)=O c1(CCNC(=NCC=C)NC2CCC(CC#N)C2)c[nH]c2ccc(F)cc12 N1(C(C2CC(NC(=O)C=CCn3cncn3)C(O)C2)=O)CCN2CCCC2C1 c1(NC2CC(NC(C3N(CC#C)CCC3)=O)C2)cc(S(C)(=O)=O)ncn1 N1(CCNC(C(CC)OC)=O)CCCN(C(=O)Cc2csc(=N)[nH]2)CC1 C12(NC(c3c(C)coc3C)=O)CCCN(C(c3cnc(C4CC4)[nH]3)=O)CC1C2 C1(C(=O)OC)CCNCCC1NC(=O)Cc1ccc(Br)cc1F c1(C(N2CCC(N(C)C3CC3)C2)=O)ccc2nc(Cl)nn2c1 CC1(NC(=O)CCc2ncccn2)CCCCC1C(N1CCCC(O)C1)=O c1(N2CCC(=C)CC2)nc(-c2cccnc2)nc(=NCCCN2CCNC(=O)C2)[nH]1 C(C(CCOC)NC(=O)C(N1CCCC1C(C)(C)C)=O)OC.C(C)(=O)O CC1(C)CN(C(=O)C2CC2)C1CCc1csc(-c2ccccc2)n1 CC(C)CCC(=O)NCCN(C1CCCC1)C(c1cc(Cl)cnn1)=O C1(C(=O)NC(CN(C(c2ccc(OCCOC)cc2)=O)C)C)CC(C)CC(C)C1 c1(OCC=C)ccc(CC(N2CCC(N(C(=O)CCCC)C)CC2)=O)cc1OC C(=O)(C1=CC2C=CC1C2)N1CC(NC(C(C)(C)Cc2cnn[nH]2)=O)(CO)C1.C=O CC(C)C1=NOC(C(=O)NC2COCC2C(=O)NCC2(Cl)CCC2)C1 c1(N2CCCC(COC)C2)cc(NCC2(C)CCCS2)nc(C(F)(F)F)n1 C1(NC(C2CC2c2ncccn2)=O)CCN(C(=O)CN2CCC2)C1 Nc1ccc(-c2nc(CCC(=O)NC3CC3)n(-c3ccccc3F)n2)cc1 N1(C(c2cc(C(C)C)n[nH]2)=O)CC(C)(C)C(NC(=O)Cn2cccn2)C(C)(C)C1 C1(C(N2CCC(C(C)(C)C)(NC(=O)C=CSC)C2)=O)(COC)CCCCC1 c1(CC(=O)N(CCCn2cc(CCOC)nn2)C2CC2)coc2ccc(OC)cc12 C1(C(N2CC(N(C(C(=O)Nc3ccc(C)cc3)=O)C)C2)=O)CC2(CCOCC2)C1 C1(OC(C)C)CCCC(c2nnnn2CC2(CC(C)C)CCC2)(NC2CC2)C1 C1(CNC(C(C)NC(C2CCCC2)=O)=O)CCCCCN1C(C1CSC1)=O CC1CCC(OCC(=O)N(CCC(C)NC(=O)CN2CCCCC2=O)C)CC1 C1(C)(C(=O)NC(C)(C)C)CC(NC(=O)CC(C)C)C1.C(C(=O)NC)N1C(=O)C1 c1(C(=O)OC)cnc(NCC(C)NC(C2(O)CCOC2)=O)c([N+](=O)[O-])c1 c1(OC)cc(C(N2CCCC(N(CCO)C(c3ccco3)=O)C2)=O)sc1Cl C(CC(C)C(=O)NC1CCCCC1CNC=O)n1cc(CCCCC)nn1 c1(C(=O)NCC2C3CCC(C3)N2C(c2cc(F)n[nH]2)=O)ccc2c(c1)CCO2 c1(C(C)=O)c(NC(C2CCCN(C(c3cc(C#N)c[nH]3)=O)C2)=O)cccc1F c1(C(=O)NC)cccc(NC(=O)CC2(O)CN(C(c3ncccn3)=O)C2)c1 C(=O)(C(C(C)(C)C)NC(C1CC1C)=O)N(CC(C)NC(CCCOCC=C)=O)C c1(C(=O)NC(CN(c2ncnc(CC)c2F)C)C)ccc2nccnc2n1 C1(NC(CCCCC)=O)CN(C(c2cccc(=S)n2O)=O)C2CCCC12 Cc1c(Br)c(C(N2CC(NC(=O)CCSCC(N)=O)C(F)C2)=O)nn1C C1(C(C)C)CCN(C(C2C3CC2N(C(=O)C(Cl)Cl)C3)=O)CC1 C1(C(=O)NCC2C(CO)CN(C(c3c(CC)cccc3)=O)C2)CCC(=O)N(C)C1 c1(OC)cncc(C(=O)N(CC(C)(C)CNC(=O)CCN2CCOC2=O)C)c1 C1(C(=O)Nc2csnc2C)(CC)CCCN(C(=O)C#CC(C)C)C1 CC1C=C(C(=O)NCC(C2CC2)NC(c2ccc(-c3ccco3)nc2O)=O)CC1 c1(C(N(C(C)CNC(=O)CN(C)C(C)=O)CC)=O)cccc(-c2nccs2)c1 c1(C(=O)NCCC2(CNC(c3c(C)scc3)=O)CC2)cccc(OCF)c1F c1(CC(COC)O)cn(CCN(C)C(c2cnc(-c3cnn(C)c3)s2)=O)nn1 c1(C(=O)OC)nn(C)cc1C(N1CCC1CNC(c1cn(CC(N)=O)nn1)=O)=O N1(C(C(CC=CC)NC(c2cc(C)nn2CC)=O)=O)CCCC(O)(CO)C1 Cc1nccc(C(C)NC(C2(C)C=CCN2C(=O)CC2CCOCC2)=O)n1 C12CC1=CC=C(Br)C=CC(C)CCN(C)C(=O)CCS2 C#CC1(C(N2CCCOC(C)C2)=O)CCN(C(C2CCC2C#N)=O)C1 CCCC(CCCNC(=O)C(C)C(F)F)NC(=O)C(=Cc1cnn(C)c1)C C1(O)(CNC(Cc2cnc(C)[nH]2)=O)CCN(C(C2CCCN2N=O)=O)CC1 C(=O)(CC(C)(C)NC(C1CC12CCC2)=O)N(CC#C)Cc1ccco1 C(=O)(N=c1ccn(C2CN(C(=O)CC#N)C2)[nH]1)NC(Cc1nc(=N)[nH][nH]1)=O c1(C(=O)NCC(CNC(C=CCOC)=O)OC)c[nH]c2cccc(C)c12 C1(C(F)(F)F)(C(N(CC(CNC(c2c(CC)nns2)=O)C)C)=O)CCCCCC1 C(=O)(C(CCOCCO)NC(=O)CCC1CCCN1C)NCC(=O)NC C(=O)(CS(=O)(=O)C(C)(C)C)NCC(C)N(C(=O)CC1(C(F)(F)F)CCC1)CC CC1C(NC(=O)Cc2cn[nH]c2)CCCN1C(=O)CNC(c1cccs1)=O c1(C(N=S(CC)(=O)C(C)C)=O)ccc(Cl)c(S(=O)(=O)N2CCCCC2)c1 c1(C(N2C(CNC(c3c(C)cncc3)=O)CC2)=O)cccc2c(C#N)c[nH]c12 c1(CC)cc(NC(C23CC2CN(C(C2CNC(=O)O2)=O)C3)=O)cc(F)c1 c1(C(=O)NCCN(C(C2CC3CC3C2)=O)CC)cc2ccc(Br)nc2[nH]1 c1(C(N2CC(C(=O)OCC3CC3)C(F)(F)C2)=O)nc2cncnc2[nH]1 N1(C(C(C)N(C)C)=O)CC=C(CNC(C2CCC(C(F)(F)F)O2)=O)CC1 c1(NCC(CNC(C(CCC)O)=O)O)cccc2sccc12 c1(C(=O)NCCCCNC(C2(COC)COC2)=O)csc2c1CCC(C)C2 Cc1ccc(-c2nc(C(=O)NCC3CCC(NC(C4C(C)C4C)=O)C3)cs2)[nH]1 N1(C(CCCCC#N)=O)CCN(C(=O)CC2CC=CCC2)C2COCC12 C1(CCNC(C2C(=O)NCC2)=O)CN(C(c2cc(C3CC3)[nH]n2)=O)CCO1 CC(C)(C(=O)NC1CC(CNC(c2nnc3n2CCCC3)=O)C1(C)C)C(F)(F)F c1(CC)cccc2ccc(C(N3CC(NC(C4CC(=O)NC(=O)N4)=O)C3)=O)nc12 C#CCCCCCC(=O)NC1CN(C(=O)C(C)C2(O)CCC2)CC12CC2 C(=O)(CCN=[N+]=[N-])N(C1CCN(C(C(C)CS)=O)C1)C.c1(CCO)ccccc1 c1cc2ncc(C3CS(=O)(=O)C(CO)C3)[nH]c-2n1 c1(C(N2C(CNC(CC(C(C)C)O)=O)C=CC2)=O)[nH]nc([N+](=O)[O-])c1Cl c1(N2CCC(CC=C)C2)[nH]c(=NCc2cnccc2Cl)nc2sccc12 CCCCC(CC)CCC(=O)NC(C)(CNC(c1cc(C#N)on1)=O)C(C)C S(=O)(=O)(c1cnn2ccc(=NC(C)c3cccc(Cl)c3)[nH]c12)NC(C)C(C)(C)C N1(C(C2CCN(C3CC3)S2(=O)=O)=O)CC2(CCN(C(=O)COCCF)CC2)C1 c1(C(C(=O)N(CCNC(=O)CC(C)O)CC)(C)C)ccc(Cl)cc1F c1(CC(=O)NC2C(CNC(c3c(C)nn[nH]3)=O)COC2)ccc([N+](=O)[O-])cc1 N1(C(Cn2nc(C)c(Cl)c2)=O)CCCCCC(NC(C2CCC(F)(F)C2)=O)C1 C(=O)(C(CNC(c1ccc(OC)cn1)=O)CC(C)C)N1CC(CC)C1 C1(C(=O)NC(C=CC(N2C(COC)CCC2)=O)(C)C)C2CCCCC12 C1(N(C(c2c(OC)c(C)cs2)=O)C)CCCN(C(=O)CCn2ccnc2C)CC1 c1(C(N2CC3N(C(C4C(C)CCO4)=O)C(CC3)C2)=O)n[nH]c2c1CC(F)(F)CC2 c1(C(N2CCN(C(=O)C=Cc3ccc(C(=O)O)o3)C2)=O)ccnnc1O C1(NC(CCN(CC)CC)=O)CC(N=c2cc[nH]cc2C#N)C1(C)C c1(C(=O)NC(CNC(c2cnc(C)[nH]2)=O)(C)CO)cc2c(o1)CCCNC2=O S(=O)(=O)(c1ccccc1C#N)N1CCC2(CN(Cc3cccc(C)c3Br)C2)CC1 c1(CC(=O)N(CCN(C(=O)COC)CCC)CC)csc(-c2nc[nH]n2)n1 c1(CC)cc(Br)ccc1C(=O)OC.C1(=O)C(C)N(C(C)C)CCCN1 Cn1c(O)nc2cc(C(=O)NCC34CC3CN(C(C3NC(=O)OC3C)=O)C4)cnc12 N12CCC(CC1c1ccccc1)C2=O.C(=O)(CC=C(Cl)Cl)NCC1C(C(C)(C)C)C1 c1(C(=O)NC2C(CC)N(C(=O)C(COC)OC)CCC2)ccc2sc(=N)[nH]c2c1 N1(C(c2cccc(N)c2O)=O)CCC2(CC=CCO2)C1 c1(OC)cc(-c2c[nH]nc2C(N2CC3CC(C2)N3C)=O)cc(OC)n1 c1(C(=O)NC2C(NC(c3cnn(CCC(F)(F)F)c3)=O)CCC2)cc2sccc2s1 C1(C(CC)NC(c2n(CCC)nnn2)CCC=C(C)C)C2COCC12 C1(O)(CN(C)C(c2ccc[n+]([O-])c2)=O)CCCN(C(C2CCCCCN2C)=O)C1 c1(COc2nc(-c3ccc(OC)cc3)sc2)cc(=O)oc2cc(O)ccc12 c1(C(=O)NCC23C(CN(C(=O)Cc4ncc[nH]4)C2)C3)ccc2cc[nH]c2c1 C1(NC(CN(C(=O)C(=O)NCC(C)C)CC)=O)CCN(CC(F)F)CC1 N1(C(c2ccc(CCCC)s2)=O)CC(C(=O)NCC(C)O)CC(F)C1 c1(C(COC)NC(=O)C(C)c2ccco2)ccc(C(F)(F)F)cn1 C12(C(=O)NC3(C)CCN(C(c4c(CC)nccc4)=O)C3)CCCCCC1OCC2 C1(C(N2CC(N(C)C3CC3)C2)=O)CN(C(C2(C)CCC(=O)CC2)=O)CC1(F)F c1(OC)cc(C(=O)NCC2(O)CN(C(c3cn(C(C)C)nn3)=O)C2)ccn1 c1(C(N2CC(C(=O)NC(C(=O)OC)C)C2)=O)ccc(C)n1C N1(C(C)=O)CCN(C(C2(O)CCOC2)=O)C(C)C1.c1(C2CC2)ccccc1Br c1(N(C(C(C)(C)C)=O)c2nc(-c3ccccc3)ns2)ccc(NS(C)(=O)=O)cc1 O=C1CC2(CCC(C(N3CCC(NC(C4(Cl)CC45CCC5)=O)C3)=O)CC2)CN1 c1(C(C)CNC(=O)NC2CC(C(=O)OC(C)(C)C)C2)cccc(Br)c1 N1(C(CC)=O)CCOC(CNC(=O)CC2CCSC2)C1 c1(C(=O)N)cc2ccncc2o1.N12CC(O)(C1)C(C)CCC2=O.C(CCOC)OC C1(c2cn(C(C3(C(=O)NC4CCC(C)C4SC)CC3)=O)nn2)(OC)CCOCC1 C(C(O)C(=O)NCC(CC)NC(c1ccc(C)s1)=O)=CC C(=O)(CC(COC)COC)N1C(CC=C)(C(=O)N(C2CCC2(C)C)C)CCC1 Cc1cc(Cl)c(C(N2CC(O)(C(C)NC(c3cnc(CC(C)C)[nH]3)=O)C2)=O)s1 C#Cc1ccc(C(=O)NCCNC(=O)CC2CCCC(C)(C)C2)nc1 c1(NC2CON(CCO)C2=O)cccn(C2CCC2)c1=O.n1(CCSC)nnnc1C1CC1 CCC(C)CCCCC(=O)N1CCOCC1CN(C)C(C1(CC)CCOCC1)=O c1(CC(=O)NC(CNC(c2cc(C)n(C3CC3)n2)=O)C)ccnc(F)c1F CN(C1CCOc2cc(F)ccc21)C(Cn1ncc(CNC(N)=O)c1)=O C1(C)(CNc2cnn(C)c2)CCC(N(C(=O)Nc2nccc(=N)[nH]2)CC)C1 c1(-c2ccc(CN(CCCN(C(C)=O)C)C)cc2)cnc2cccc(C(C)C)n12 Cn1cc2cc(C(=O)NC3CC4CC3N(C(C3CCS(=O)CC3)=O)C4)ccc2n1 C1(C(=O)NC(CN(CC)CC)C)CCCN(C(C2CCCCN2CC(F)F)=O)C1 C1(CC(=O)NC2(CCC)CN(C(=O)C=CC(C)(C)SC)C2)C=NN(C)C1=O N1(c2ccnc(C)n2)CC2CC(NC(c3cnc(C)c(O)c3)=O)CC2C1 c1(C(=O)NC(C(C)NC(c2cnc(C#N)s2)=O)C)cc2ncccc2cc1Cl CC(C)(C)CC(O)CC(=O)N1CC(CNC(c2nsnc2C(=O)O)=O)C2(CC2)C1 C(CCCC(C)(C)C(=O)NNC(=O)c1nccc2ccsc12)NC(COC)=O c1(N2CCCC(C(N)=O)(NC(c3scc(C)c3)=O)C2)ncnc2[nH]cc(C(N)=O)c12 Cc1ccc(C#N)cc1NC(=O)CC1CC(F)CN1C(=O)C(F)CC(C)(C)C C(=O)(CC(=O)N(C)C)NCCC(C)N(C(=O)CCCNC(c1cccnc1)=O)C O=C1CCC(C(N2CCC(CNC(=O)CCc3nnc(S)nc3O)CC2)=O)CN1 C(N=c1cc(C)[nH]c(=NCCOc2ccc(C)cc2)[nH]1)C1CCC(C)(CC)O1 C12CCN(C1)C2=O.C1(CCC#C)CN(C(=O)CNC(=O)CO)C1 C(C(O)C(=O)NCC(C(=O)NCc1nnc(C)s1)N(C)C)SC CCCCCCCC(=O)NC1CC(F)(CNC(c2occc2C(=O)OC)=O)C1 c1(-n2ccc(C(=O)NCCCCCNC(C(C)CN(C)C)=O)n2)ccnc(Cl)c1 C1(NC(c2c(C)n[nH]c2C)=O)CC2CC(NC(=O)CC3CCCCCCC3)CC12 C1(NC(C2(OC)CCN(C(=O)C3=CCOCC3)C2)=O)CCN(C)CC1(C)C CCCC(C#N)C(=O)NCCC1CC(NC(=O)CCC2CCCCO2)C1 C1(NC(c2n(C)c(S)nn2)=O)CCC2(CC1)CN(C(C1CCC(C(N)=O)C1)=O)C2 CC(C)CCCC(C)C(=O)NCC1(F)CCCN(C(=O)COC(F)F)C1 c1(C(N(C2CCN(C(=O)CC3CC(F)C3)CC2)CC)=O)cccc(F)c1C#N Cn1cccc(C(=O)NC2(C)CCN(C(=O)CC(C)(C)C)C2)c1=O CCC(CC)CCCN(C)C(C1CCCC1NC(c1cnc(OC)nc1)=O)=O C(=O)(CCCCO)N(C1CCCN(C(c2cnn(CCO)c2N)=O)C1)C.C1(=O)CN1 C1(C(=O)NC(CNC(=O)Cn2ccc([N+](=O)[O-])n2)CO)Cc2c[nH]cc2S1(=O)=O Cc1ncc(C(=O)NCC(C)CN(C)C(c2cnc(C(C)(C)C)s2)=O)cc1N C1(NC(c2c(C)ocn2)=O)C(C)CCN(C(c2ccoc2)=O)C1C c1(NC(C2CCCN(c3ncccn3)C2)=O)ccnc2c(Br)cccc12 Cc1cc(F)c(C(=O)NCCC2(O)CCN(C(c3cc(Cl)c(Cl)[nH]3)=O)C2)cc1F C1(C(N2CC3C(CNC(=O)CS(=O)(=O)N(C)C)C3C2)=O)(COC)CC=CCC1 N1(C(=O)C(O)Cn2cncn2)C2CCC(C(N3C4CCC3COC4)=O)C1CC2 c1(C2C(CNCCOCCOC)C2)nnnn1C C1(CNC(CN(C(=O)Cc2ccc(Cl)o2)CC)=O)CCN(C(C)C)C1 c1(CC(N2CCC(CN(C)C(C3CC(O)C3)=O)C2)=O)n[nH]c2ccccc12 N1(C(CC2(C)CC2)=O)CCNC(c2ccc(OC(F)(F)F)cc2)C1 c1(NC(C2CCCCC2OCc2ccccc2)=O)cc2cc(Br)cn2cn1 C(=O)(C(CCC1CC1)NC(c1cncc(Cl)c1)=O)NCC=CCSC c1(C(=O)NCCNC(Cc2n(C)nc(C(F)(F)F)c2)=O)ccc(Cl)c(N)c1 c1(CN(C(CC(C2CC2)NC(C2C(C)=CCS2)=O)=O)C)cccc(F)c1 C(=O)(C1=NNC(=O)C1)N(C1CCN(C(C2CC(=O)N(CC(F)(F)F)C2)=O)C1)C c1(C(N(C2CCN(CC=C)C2=O)CC)=O)cc2n(n1)CC(C)NC2=O C1(C(C)NC(=O)C(=O)NC2(C)CCC(=O)NC2=O)CCc2ccccc2C1 N1(C(C(N2C(CC)CCC2)=O)=O)CC(C)Oc2ccc(C(=O)O)cc21 C(=O)(C1=CN2CCN=C2C=C1)NCCOC1CN(C(c2noc(CC)c2C)=O)C1 C1(NC(C(C=C)O)=O)C2CCN(C(c3cc4ccsc4s3)=O)CC12 C1(NC(C2(NC(c3ccc(Cl)cn3)=O)C(C)CCC2)=O)CCC(O)C(O)C1 N1(C(C#CCNC(C(C)OCCC(C)C)=O)=O)C(CO)CCC12CCC2 Cc1cc2[nH]c(C(N3CC=CC(NC(=O)C(C)C4CCCC4)C3)=O)cc2s1 c1(CC)ccccc1C(N1C(C(=O)NC2CN(CCOC)C2)CC2CC12)=O C=CCC(CC)C(=O)N1CC(CNC(c2ccc(C3CC3)cc2O)=O)C(C)(C)C1 c1(NC(c2c(C)nn(C(C)C)c2C)=O)ccc2c(c1)N(C)C(=O)CO2 C1(CC)CCN(C(c2nn(C)cc2N)=O)C1CNC(=O)C(CC1CC1)OC C1(CC)C(C(=O)NC2(CC)CC2)CCN1C(C1CC(CF)C1)=O C1(CN(C(C2CN(C)CCO2)=O)CC)CCN(C(=O)C(=O)N(C)C)CC1 C1(C(=O)NCCN(C(=O)CN(C)C)C(C)C)Cc2c[nH]cc2S1(=O)=O N1(C(C(=O)N(C)C)=O)CCN(C2CCCOC2=O)CC1C CC(C)(C)CC(O)CC(=O)NCC1CCCCN1C(=O)CCOC1CCOCC1 CC1CCN(C(C2CC3CC3C2)=O)C1CNC(C1CNC(=O)N1)=O C1(OC)CC(C(N2CCC(OCCF)C2)=O)N(C(c2cccc(O)c2)=O)C1 C(=O)(CCCCC(F)F)N1CCCC(NC(Cc2c(C)non2)=O)CC1 N1(C(C(CSC)C)=O)CC(NC(c2ccc(C)nc2C)=O)CC12CCCCC2 N1(C(C(C)(C)C2CCCO2)=O)CC2(C(=O)NCc3cnn[nH]3)CC1CO2 N1(C(C(C2CCC2)OCC)=O)CCC(N(C)C(c2cc(CC)nn2CC)=O)CC1 CCCCC(C(N)=O)NC(=O)CONC(C1CCCN1CC)=O C1(CNC(Cn2cc[n+](C)c2)=O)CCCCN(C(c2ccc(O)nn2)=O)C1 N1(C(c2c(CC)[nH]nc2Cl)=O)CCN(C(=O)CC2CCC3CC23)CC2(CC2)C1 CC(C)C1=NOC(C(=O)N(C2CCN(C(=O)COCC(F)(F)F)CC2)C)C1 c1(N2CCC(N(CCC)C(c3ncc[nH]3)=O)CC2)nc(C#N)c(Cl)s1 c1(C(=O)NCC(C(=O)NC(c2nc(CC)on2)C)C)cc(C)c(N)cn1 C1(C(C(=O)OC)=O)CCC(NC2C(NC(C3C(COC)(CO)C3)=O)C2)CC1 c1(C(=O)NC(CC=C)CNC(=O)C(C)c2cccs2)ccc(CC(N)=O)cc1 N1(C(C(C=C)(C)O)=O)CC(NC(C2(n3cc(Cl)cn3)CC2)=O)C(C)(C)C1 C#CC1(CNC(=O)CCOCCNC(C23CCCCC2C3)=O)CCOCC1 O=C(CC(F)(F)c1ccccc1)N1CC(NC(C2C3COCC23)=O)C1 N1(C(CCCNC(=O)OCC)=O)CCCC(C(=O)N(CC)CC23CC(CO2)C3)C1 c1(N(C)C)ccnc(C(=O)NC2(C(=O)NCCS(C)(=N)=O)CC2)c1 c1(N2CC(C(C)NC(CC3CC(OC)C3(C)C)=O)C2)ncnc2cc(Br)ccc12 O=C(C(O)CC(F)(F)F)N1CCC(CO)C(NC(C2(O)CCCC2)=O)C1 N1(C(C(OC)OC)=O)CC2CC(NC(=O)Cc3c(CC)noc3CC)C1C2 C(=O)(C(O)P(C)(C)=O)N1CCC(COC)(NC(=O)CCOC2CCN(C)CC2)C1 N1(C(C2C(NC(CCc3c(C)cccc3)=O)C2)=O)CC2(C1)CC1(CCC1)C2 C(C)(C)(C(=O)NCC(COC)NC(C1CCCCC1)=O)OCC c1(NCc2c(C)ccc(OC)n2)nc(=NC(C)C(C)F)[nH]c2c1CCC2 CCCC(CCC)C(=O)NC1C=CC(CNC(C2CCSC2)=O)C1 c1(CC)noc2ncc(C(N3CCN(C(=O)C(C)C4CC4)CC3CC)=O)cc12 c1(N(C)CC2CC(F)CN2C(=O)CCc2cccc(O)c2)ccc(S(C)(=O)=O)cn1 c1(CC)ccc(C)c(Cl)c1.C12CCN(C)C1C1CCCN1C(=O)C(=O)N2 c1(CNC(c2ccc(F)cc2)c2n(C)ccn2)ncc([N+](=O)[O-])s1 CC(CC(=O)N(CC(C)(C)CNC(=O)C(CO)N(C)C)C)C(C)(C)C C1(CCCNC(COC(CC)C)=O)(NC(=O)COCCSC)CCCC1 c1(C(=O)NCCCN(C2CCCC2)C(C23CC(C)C2C3)=O)nc2c(s1)COCC2 Cc1cc(NC(=O)CN2CCN(Cc3cc[nH]n3)CC2=O)cc(C)c1Br N1(C(C2CC=CC2)=O)CCC(F)(c2cn(C3CCCC3)nn2)C1.C1CCCCS1 C12(CNC(C(COC)O)=O)CC1CN(C(=O)Cc1cnc[nH]1)C2 C1(NC(C2(N(C(c3ccc(Cl)cn3)=O)C3CC3)CC2)=O)CC2(CCC2)CO1 CC(C)C(C)(CNC(=O)CNC(c1ccoc1)=O)NC(C1CCC(F)C1)=O CCCCC(CNC(=O)CN(S(C)(=O)=O)CC)NC(c1ccc(CC)[nH]1)=O C(=O)(C#CC(C)(C)C)CCN(C)C.C1(OC)CN(C(=O)C(c2ccco2)N)C1 N1(Cc2ccc(CC)cc2)CC2(CCN(C(c3cc(F)c(Cl)c(Br)c3)=O)CC2)C1 N#Cc1cccc2[nH]cc(C(=O)NC3CCC3CNC(=O)Cn3ccnn3)c12 N1(C(Cc2nc(C)oc2)=O)CC(C(=O)NC(C)C(O)C(F)F)CC1(C)C N#Cc1c(NC(Cn2cc(C3(O)CC3)nn2)=O)cnn1-c1ccccc1 C1(C(N2CCC(CC(N3C(CC)CCCC3)=O)C2)=O)C(C)CCNC1C C1(N(C(CC2(OC)CN(C(c3cnn(C)n3)=O)C2)=O)C)CCCCCC1O Cc1cc(C(N2CCC(NC(=O)C(C(C)O)N(C)C(C)=O)CC2)=O)ccc1O c1(C(=O)NC2CC(CNC(c3c(C)nc[nH]3)=O)C2(C)C)ncc(C)cc1F Cn1nccc1CC(=O)NCC1CC(NC(=O)CC2COC(=O)C2)C1 CCC(C(=O)N1CCC(OCCCNC(C2CC2(F)F)=O)CC1)C(C)C c1(N(CCCNC(=O)NC2(CC#C)CCCCC2)C)ncc(C#C)cc1C c1(OC)ccc(CC(=O)N(C)CCNC(=O)CC2CC3CCC2C3)c(Cl)c1 CC1(C)CCCOC1CNC(C1CCC1CNC(C1CCNC1=O)=O)=O N1(CCNC(C(COC)O)=O)CCN(C(c2ccsc2-c2ccccc2)=O)CC1 C1(CNC(C(Cc2cnc[nH]2)OC)=O)CC(O)CN1C(=O)CC1CCCNC1 C1(NC(=O)CN2CCCC2CO)CCC2CC1CN2C(c1cnc2n1CCCC2)=O C1(CC)CN(C(=O)CN2C(=O)CNC2=O)CCC1NC(C1SCC=C1C)=O c1(OC)ccc(Br)c(F)c1CN1CCC1(C)C(=O)NCC1(C)CCCC1 C=C1COc2c(C(N3CC(NC(=O)CC4(N(C)C)CC4)C4(CC4)C3)=O)cnn2C1 CC1(C)CCCOC1C(=O)NCCCCNC(=O)CSc1nc[nH]n1 CCC(CC)CC(=O)NC12CCCC(NC(=O)C(C3CCCOC3)OCC)(C1)C2 C(C(CNC(c1scc(C)c1C)=O)C(F)(F)F)NC(C1C(OC)CC1)=O CC(C)(C(=O)N1CC2CN(C(c3cc(-c4ccccc4)on3)=O)C2C1)C(F)F Cc1cc(C(=O)NC2CC(F)CN(C(=O)COC(C)C)C2)ncc1Br N1(C(Cc2n(C)cnc2)=O)CCC(C(=O)NCCCCC2CC2)C(C)(C)C1 C(=O)(C1c2c[nH]nc2CN1C(c1n(C)cc(Br)c1)=O)OC(C)(C)C C1(CNC(C(CCOC)C)=O)CCN(C(=O)COCC2CCOC2)C12CC2 N(C(=NCC1CC12CC2Br)NCc1cccc(C(F)F)n1)C(C=C)C c1(CC(=O)N(CC(CC)NC(C2CC(=O)N(O)C2)=O)CC)cccc(C)c1C C(c1ccnn1C)=CC(=O)NC1(C2N(C(C3ON=C(C)C3)=O)CCC2)CC1 C1(C(=O)NCC(F)Cl)(CNC(c2ccnc(CO)c2)=O)CC12CCC2 CC(C)(C)S(=O)(=O)CC(=O)NC1CCC1CNC(c1ccc2cccnc2n1)=O Cc1cc(CCC(=O)NCCNC(=O)CC2CC3(CCC3)C2)ccc1Cl C(CC(C(=O)NCCC(F)Cn1ccnc1)NC(=O)Oc1cc(C)on1)OCC c1(CCC)cc(C(=O)NC2CCCCC2CNC(=O)C(C)n2ccnn2)nn1C c1(C(N2CCCC(CCCCNC(CC(=C)C)=O)C2)=O)ccc(C(N)=O)c(Cl)c1 c1(C(N2C(C(=O)NCCCC3(C)CC3)CC3(CC3)C2)=O)cc2ccccn2n1 C1(C(=O)NC2C(C)CN(C(=O)C(F)(F)NS(C)(=O)=O)C2)CCc2nn[nH]c2C1 C1(NC(CC2(C)CCN(C(c3ncc(CC)cn3)=O)C2)=O)CC2CCC(C1)O2 CCC(CC)(CCNC(c1ccccc1SCC#N)=O)NC(c1nc(O)c(C)s1)=O c1(OC)ccc(C)c(OC)c1C(N1CCOC(CNC(C2CC2OC)=O)C1)=O c1(C(=O)NC(C(C)NC(C(CCC)C(C)C)=O)CO)ccc2cnccc2c1 c1(C(N(CCCO)C)=O)cc(-c2ccc(C(N)=O)cc2F)cc2[nH]ncc12 C1(C)(NC(=O)NCCC(CC)(C)C)CCC(C)=C(C)C1 n1(CCNC(CC2N(C(C3N(CC)CCC3)=O)CCC2)=O)ccc(=O)cc1 c1(C(=O)Nc2ccccc2)cccc2cnnn12.CC1CCCO1.C1CCN1C c1(C(N2CCC(C(=O)NCCCN)CC2)=O)ccc(Oc2ccccc2)nc1 c1(OC)cc(CNC2CCC(CC(N3CCCC(O)C3C)=O)CC2)cc(Cl)c1 C12(NC(CCC(=O)NCCC)=O)CCCCC1N(C(=O)COC)CC2 c1(OC)ccc(C(=O)N(C)CCN(C(=O)C=Cc2cnc[nH]2)C(C)C)c(F)c1F C(=O)(C1=NOC(C)(C)C1)N1CC(CNC(c2c(C)n[nH]c2)=O)C2C1C2 Cc1ccsc1C(=O)NCC1CC(NC(c2cscc2C)=O)C1 c1(NCC(=O)NCC2N(C(c3ncn(C)n3)=O)CCOC2)ccc(F)cc1F C1(NC(c2cn(CCOC)nc2)=O)CCSC12CN(C(C1(OC)CCOC1)=O)C2 C1(CC)CCOC1C(=O)N(CCC=CC(N1CCCC1C1(C)CC1)=O)CCO Cc1ncoc1C(=O)N(C)CCOCCCN(C)C(C1(C)CC1)=O N1(C(C(C)(C)CF)=O)CCC2CN(C(=O)C(F)(F)CC3CC3)CCC2C1 c1(C(=O)NCC(CC)NC(=O)CC2CN3CCN2CC3)cccc2nc(O)[nH]c12 N1(C(C(=O)N(C)C)=O)CC2CC1CCC2NC(c1ccc(N2CCOCC2)nc1)=O N1(C(C(CC#C)C)=O)CCC(C)(N(C(=O)C(C)n2cncn2)Cc2ccsc2)CC1 Cc1cnnc(O)c1C(=O)NCC1CC1CNC(C1(C)CC=CCC1)=O C(=O)(C(CNC(=O)CCCC)CC(C)C)N(C1CC(C=C)OCC1)C c1(NCC2(c3ccc(OC)cc3)CC2)nccc(=NC2CCCC2)[nH]1 Cc1nsc(C(=O)NC2CCOC2C(=O)NC(c2ccnn2C)C)c1N C(=O)(C1=CC2(CCOC2)C1)NC(CC(=O)NCc1c(OC)nsc1)(C)C CC1(C)CN(Cc2c(F)cccc2Cl)CC(C(C)(C(=O)O)c2ccccc2)O1 C(c1ccncn1)=CC(=O)NC(C1CC(NC(=O)CC2SC(=N)NC2=O)C1)C C(C)(CCC(=O)N1CC(C)(CCC(=O)NCc2cnccn2)C1)OC c1(C(=O)O)ccc(-c2cccc(Cn3cccn3)c2)nc1 C(=O)(C(C)S(N)(=O)=O)NC(c1ccc(F)c(Cl)c1)CNC(CCC=C)=O CC1(C)C2CC(C(=O)CCOC3CN(c4nc(-c5ccccc5)ns4)C3)CC12 c1(C(N2CCC(F)(CNC(=O)C(O)C3CCC3)C2)=O)cc(O)cc(Cl)c1 C(=O)(C(C)CC(F)F)NCC1(Cn2cc(CNC(c3c(C)nns3)=O)nn2)CC1 CCC(O)C(C)C(=O)N1CCC(N(c2ncc(I)cn2)C)C1 Cc1cc(C(=O)N(CC(C)O)CCNC(c2ccsn2)=O)c(C)cc1Cl c1(NC(C(c2cncc(OCC)n2)N2CCC(C)(CO)C2)=O)ccc(Cl)cc1F CC1CN(C(c2c[nH]c(=N)s2)=O)CC(C)C1NC(=O)C(Cl)=CCl N1(C(c2cccc(C)c2C#N)=O)CCN(C(c2ccc(F)cc2)=O)C2COCC12 C(C(=O)NC1CC12CC(OCC)C2)(C(C)CC)NC(C(CC)=CC)=O N1(C(C(C)OCC=C)=O)CCC2(CC1)CC(NC(C1CNC(=O)S1)=O)C2 C(C(C)(C)CNC(=O)COCCn1cncn1)N(C(C(c1ccn(C)c1)C)=O)C N1(CCC(N2CCCC(CNC)C2)=O)C(=O)C2CCCCC2C1=O c1(OC)ncc(C)cc1NC(C1(NC(C2CC(=O)CC(=O)N2)=O)CCC1)=O C(c1cnc(O)nc1O)=CC(=O)N(C)CC1CCN(C(C(COC(C)=O)C)=O)C1 N1(CCCCNC(c2ccccn2)=O)CCCN(C(=O)C2=NOCC2)CC1 CC1CC(c2cccc(F)c2)N(C(c2ccnn2CCF)=O)C1 c1(CN2CCC3(C(C(N4CC(C5(C)CC5)OCC4)=O)C3)C2)cnc2ccccn12 c1(C(=O)NC(C(C)NC(C2CC2(C)C)=O)(C)C)cc(O)c2ccsc2c1 c1(C(=O)NCC2C(NC(c3cccc(OCCF)c3)=O)CC2)ccc(N)cc1F C1(CC)CN(C(C)=O)CCC1NC(=O)Cc1ncccc1C C1(F)(C(=O)NC(CC)CN(C(c2ccc(Br)o2)=O)CC)CCC(COC)CC1 C1(NC(CCCN(C)C)=O)CC2(CCCN(C(C3CCOC3(C)C)=O)C2)C1 C=C(Cl)CC(C(=O)N(C)CCN(C)CCO)NC(c1cc(CC)[nH]n1)=O c1(OC)cc(CNC(C)(C(C)C)c2nnnn2CCN2CCOC2=O)on1 C1(C(=O)NCC2(O)CC(NC(C3CCN(C)CC3)=O)C2)CC(C)(C)OC1=O CC#CCCCC(=O)NC1(CF)CCN(C(=O)C(C)(C)c2cncs2)C1 CC1CCOC1C(=O)NC1CC(CNC(=O)C(F)=CCCF)C1 c1(OC(C(=O)OCC2(C)CC(=C)C2)CO)ccc(F)c(F)c1 CCC(C)C(O)C(C)C(=O)N(C)CC1COCCN1C(=O)CN1CC(C)C1 N1(C(CCCSCCCC)=O)CCN(C(=O)C=CC(C)(C)C)C(CO)C1 C1(CCNC(C(F)=C(C)C)=O)CN(C(C2OC3CCC2C3)=O)CCO1 CC1CN(C(=NCC2CC2)NCc2ccc(C(C)(F)F)cn2)CCC1O N1(C(C=CCCCCC)=O)CC(NC(c2ccc(C(N)=O)c(Cl)c2)=O)CC(F)C1 Cc1c(C(N2CC(NC(c3cc(F)n[nH]3)=O)C3(CC3)C2)=O)cccc1S(N)(=O)=O Cc1cnc(CCCNC(c2cc(C(F)F)nn2C)=O)nc1 C1(NC(CCCC(=O)NC)=O)CN(C(C2CCCN2C)=O)C2CCCCC12 CC(C)(CCCN=c1ccnc(Cl)[nH]1)NC(=O)CCC=Cc1ccccc1 C12(C(=O)NCCN(C3CCC3)C)CNCC1(C(F)(F)F)C2 N1(C(CCOC)=O)CCC2(CC1)COC(CNC(=O)CSCc1csc(=N)[nH]1)C2 C1(N)CC2(CCN(C(=O)C=CC(F)(F)F)C2)C1.C12CCCN1C(=O)C21CC1.CCC c1(CC(=O)NC2C(CNC(c3ccc(CC)s3)=O)C2)c(C)nc(O)nc1O N1(C(C(=O)OCC)=O)CCCCCC1C1CCN(C(c2cnsc2C)=O)CC1 C#CCCCC(=O)NCCNC(=O)C(O)CC1=CN=CCC1.C12CC(C)(C1)NC2=O C1(NC(C2(F)C(C)OCC2)=O)CCC2(CC1)CN(c1ncc(O)cn1)CCO2 C1(CNC(COCCN(C)C)=O)CN(C(=O)CCNC(c2ccoc2)=O)CCO1 c1(C(N(CCCCNC(C(C)C2CCCO2)=O)C)=O)cc2c(O)ncnc2cn1 c1(NCC(CC2CCCCC2)N(C)C)[nH]c(=NC2CC(F)C2)nc2scnc12 N1(CC)CCOCC1CC(=O)NCC(=C1CN(C(=O)CCc2cscn2)C1)F c1(Cc2ccccc2NC(C(N2C(COCC)CCC2)=O)=O)cc(C)ncc1C N1(C(C2CCCN(C(C(=O)NCC(F)F)=O)CC2)=O)CC2(CCC(=O)NC2)C1 N1(C(c2ccc(C)c(F)c2)=O)CC2CCN(C(C3CC=CC3)=O)CC12 c1(COC)ccccc1C(N1CCC(C(C)NC(c2ccc(C#N)s2)=O)C1)=O C1(F)(C(=O)NCC2CCN(c3ccncc3)CC2)CNCC1F N1(C(C(Cc2ccccc2)OC)=O)C2CCCC1CN(C(C1CC(C)(F)C1)=O)C2 C12(C(=O)NCC(C)(O)C(F)(F)F)CCN(C(=O)Cc3cccnc3O)CCC1C2 C1(C)(NC(CNS(C)(=O)=O)=O)CC(NC(C2(c3ccccn3)CC2)=O)C1 Cc1ccc(C(N2CC(NC(=O)CSCC3CCCO3)C(F)C2)=O)cn1 c1(N2CCC(N(C3CC4(CC(C#C)C4)C3)C)CC2)ncnc2[nH]cc(C#N)c12 Cc1oc(-c2ccccc2)nc1CC(=O)N(C(C)CN(C(=O)CP(C)(C)=O)C)C CN1CCN(C2CC(Nc3nnc(SC(F)F)s3)c3ccc(F)cc32)CC1CO c1(C(N2C(CCNC(C3CC34CC(F)(F)C4)=O)COCC2)=O)ncn2c1CCC2 C1(C(N2CCN(C(c3c(C)cc(Br)s3)=O)CC2)=O)CC(C2CC2)=NO1 C1(CN(C2CCN(C(=O)OC(C)(C)C)CC2)C)CCC(C2CC2)C1 C12(C(N3CC(C)(CCC(=O)NCc4ccsc4Cl)C3)=O)CCCC(CO1)C2 c1(C(=O)OC)c(N)sc2c1CCN(c1nnnn1Cc1cc(C)ccc1OC)C2 c1(C(=O)NC(C)CN(C(=O)C(=O)NCC(F)F)C)ccc(F)c2occc12 N1(C(c2c(NC)cccc2)=O)CC2CC1CCN2C(c1ccc(C)cn1)=O N1(C(CCCOCCC)=O)CC2(CC(C(=O)N(c3csnc3C)C)CO2)C1 N1(C(C(C=C)(C)O)=O)CCC2(CCCCC2NC(c2csc(C3CC3)n2)=O)CC1 C=CCC(CNC(=O)CCCC1CC1C)C(=O)N1CC(CC2CC2)C1 c1(C(N2CCC(CC)C2)C(=O)NCCCC(=O)OCC)cnc(C(=O)OC)nc1 N1(C(C(c2cncnc2)C)=O)CC(C(=O)NC2CC2(C)C)CCC1(C)C CC1(C)CN(C(CC(C)C2CCCCC2)=O)C1c1nccn1Cc1ccccn1 c1(OC)ccc(CN(CC(C)O)C(=O)Nc2cccc(C)n2)cc1Br c1(-c2ccc(N(C3(c4ccccn4)CC4(CCC4)C3)C=O)o2)cc(F)cc(I)c1 N1(C(=O)NCCn2cnc(C(=O)OC)n2)CCn2c(nc(C(F)(F)F)c2Br)C1 C1(C(N2CC(Cn3cc(-c4cccc(C)n4)nn3)C2)=O)CCC12CCOCC2 C(CC(C(C)(C)C)NC(=O)CC1=CCCC1)N(C(C(C)OC)=O)C C=CC(C)(O)CC(=O)N1CCCCCC1C(=O)NCC(C)(CC)C(C)O N1(NC(C(C)c2cc[nH]n2)=O)CCCCC1CF.C12CCC1C(=O)NC2 n1(CCOC)nnnc1C(c1cc(OCC2CC2)ns1)NC(c1nc(C)cs1)C C1(O)(CC=C)CCCN(C(=O)CNC(CNC(c2ccccn2)=O)=O)C1 c1(NC(COC(CNC(Cc2cn(C)nn2)=O)(C)C)=O)cc(F)ccc1O c1(-c2ncn(C)n2)ccc(C(=O)OC(Cc2ccccc2Cl)C(N)=O)cc1 C=C1CCN(C(=O)C(C)C2(O)CCC2)C(C(=O)NCC(O)C2(Cl)CC2)C1 c1(C(N2CCCC(CCNc3nnc(C4CCC4)s3)C2)=O)cccc2nccn12 c1(CC)cc(C(=O)NCc2ncccc2C(=O)NC(C)(C)C(C)O)nn1C c1(C(N2CCC(C)(CNC(=O)Cc3cc[nH]c(=N)c3)C2)=O)cc(F)cnc1O c1(C(=O)NCC2CCCCCN2C(c2n[nH]cc2F)=O)nccc2ncncc12 N1(C(CC)=O)C2CCCC1CC(CNC(=O)C(c1ccc(OC)c(F)c1)C)C2 C1(NC(c2c(CNC(C3=CC(C)(CC)C3)=O)n[nH]c2)=O)CCn2nnnc2C1 C1(C(N(c2cc(-c3cccnc3)ccn2)C)=O)CCC=CCCC1N c1(OC)ccccc1C(N1CCOC(CNC(c2cn(CCO)nn2)=O)C1)C N1(CC)CCOC(C(=O)N(C(C)C(=O)NCC(c2nccc(O)n2)C)CC)C1 C1(C(=O)NCCN(C(CC(C)SC)=O)CC2CC2)CCc2[nH]nc(C)c2C1 CCC(CC)(CN=c1[nH]c2c(c(=NCC3(F)CC3)[nH]1)COC2)OC c1(C(N2CC3CCN(C(C(CC#C)(C)C)=O)CC32)=O)ncc2ccccc2c1O C1(C(N2CC3(C2)CN(C(C2CC2c2ccco2)=O)C3)=O)CN2CCCN1CC2 c1(C(N(C)CC2CCN(C(c3c(C)cc(N)cc3)=O)C2)=O)c(C)cc(F)cc1C N1(C(C(c2cncnc2)C)=O)CCC2CC(NC(C3(F)CCC3)=O)CCC2C1 c1(CCC(=O)CCN(C(CNC(C2C(C)C2)=O)=O)C)cccc(F)c1Cl.C(CSC)O C#CC1(O)CC(C(=O)NC(COC)C(=O)NCC2(C)CC(C)=NO2)C1 N1(C(c2c(C)nco2)=O)CCN(C(c2cc(F)cc(F)c2F)=O)CC(O)C1 Cc1ccc(C(=O)NCC(CNC(=O)Cn2cncn2)C(F)(F)F)c(N=[N+]=[N-])c1 c1(OC)ncccc1CC(=O)NC1(CCNC(=O)CCN2CCCC2)CCC1 CCCCCC(C(=O)N1CC2(CCN2C(c2ccc(C(F)F)cn2)=O)C1)C(C)C C1(CC(N2CC3CC3(NC(C3(Cl)CC3(F)F)=O)C2)=O)(COC)CCOCC1 C(=O)(C(O)CC(F)(F)F)N(C(C)CNC(=O)CC1CCCCCCC1)C c1(CC(=O)NC2CCC(NC(CNC(CC)=O)=O)C2)cccc(Br)c1Cl C(CCCCCCC(=O)N(CCNC(c1ccnc2ncnn12)=O)C(C)C)SC N1(C(C(C)Oc2ccccc2F)=O)CCC2(CC(NC(C3CCC(=O)C3)=O)C2)C1 c1(CC(=O)NCC(CC)(CC)NC(=O)CCc2nccn2C)c(Cl)cccc1Cl Cc1cc(C(=O)NC(C)CCCNC(=O)CC2CSCCS2)c2ncccc2c1 Cc1nc2ccccn2c1C(=O)N(CCN1CCN(C(C)(C)C)CC1)C1CC1 N1(C(c2c[nH]nc2-c2ccco2)=O)CCC2CN(C(c3cccc(Cl)c3)=O)C2C1 C(=O)(CN(C)N1CCC(C)(c2ccccc2F)CC1)OC(C)C N1(C(c2cc(C)nn2C)=O)CCN(C(c2cc(Br)co2)=O)CC1C N1(C(CN(CC#C)C(C2CCCC2C)=O)=O)C2CCC1CC1(CC1)C2 c1(C(=O)NCC(C(C)C)NC(c2ccc(Cl)o2)=O)cc(O)n(C)n1 c1(C(N(CC(C)NC(=O)C(C)CF)CC)=O)cc(O)nc2c1c(C)nn2C c1(C(N2CC(=C(CNC(c3cnc(C4CC4)nc3)=O)F)C2)=O)nnn2c1CCC2 C1(C)(c2cn(-c3cccc(C)c3)nn2)COCCN1C(c1ccc(F)c(Br)c1)=O c12c([N+](=O)[O-])ccc(c1O)N2.C1(N(CCO)C2CC2)CCCCC1 C(=O)(C(CC)C(C)(C)CC)N1CCC(C(NOCCC)=O)(CC)CC1 c1(C(N2CCC(N(CCC)C(C3CC3C(N)=O)=O)C2)=O)cc(C(=O)OC)c[nH]1 CC1CCCn2cc(C(=O)NCC3CCCN3C(c3cc(N)nc(Cl)c3)=O)nc21 C(=O)(C1=NN(C)C(=O)CC1)N(CC(CNC(c1c(OCC)nccc1C)=O)C)C N1(C(C(CCC)OC)=O)CCN(C(=O)CCSC)C(c2cc(F)ccc2OC)C1 C1(=CC(N2CC(CNC(=O)C=C3CCSCC3)C(O)C2)=O)CN2CCC1CC2 n1(C(C)C)ccc2c(N3CCCC(NCCN4CCCCC4C)C3)nc(Cl)nc12 c1(CNC(C)Cn2ccnc2-c2ccsc2C(F)(F)F)ccccc1Cl C(=O)(C1CCCc2nn[nH]c21)NCC1C(C(=O)Nc2nn(C)c(Cl)c2Cl)CCC1 C1(CNC(=O)C=Cc2nccs2)C2CC1N(C(=O)Cc1cccnc1)C2 c1(C(=O)NC2CN(C(C3N(C)C(=O)CC3)=O)C(C)(C)C2)cc(F)cc(Cl)c1O c1(CC(=O)NCC(N(C(Cn2nc(C)oc2=O)=O)C)C2CC2)cccc(F)c1Cl N1(C(C2CC3(C2)CC3(F)F)=O)CCC(F)(C(=O)NC2CCC(O)CC2)CC1 C12(C(N3CC(C)C(CNC(C4(C5CC5)CC4)=O)C3)=O)CCCCC1C2(F)F C1(C(N(CCN(C(=O)Cn2nccc2C)CC)CC)=O)CCCC(C)CC1 c1(C(N2CC(CNC(c3c(N)nc(Cl)cc3)=O)OCC2)=O)cnc2[nH]nnc2c1 c1(C(=O)NCC2(C)OCCN(C(C(CCC)C)=O)C2)nn(CC)cc1[N+](=O)[O-] C12(CC(=O)NC3C(NC(C(C)NC(c4cccs4)=O)=O)CCC3)COCC(C1)C2 N1(C(c2c(-c3cc(C)no3)ocn2)=O)CCC(C)(NC(=O)OC(C)(C)C)CC1 C1(NC(CCSC)(C)C)C2CC3C1C3C2CC(=O)OC C(CO)(C(=O)NC(C(=O)NCc1nc(C2CC2)n[nH]1)C1CCC1)OC O=C(NNc1ccccc1-c1nn[nH]n1)NCCSc1nc2ccc(Cl)cc2[nH]1 C1(O)(CCNC(c2c(CC)occ2)=O)CCN(C(c2cnc(C(C)OC)s2)=O)C1 C(=O)(C1CCCn2cnnc21)NCC(C1CCOC1)NC(=O)COCCF CCC(C)N(OC)C(=O)C1CC(NC(C2CC(C3CC3)C2)=O)C(O)C1 N1(C(C2OCCN(CC)C2)=O)CCN(C(=O)C=Cc2sccc2C)CC1C C1(NC(=O)NCCC(CC)CC)CNCC12CCOCC2 c1(OC)cccc(CNC(=O)C=CC(C)NC(=O)CCc2nc(C)no2)c1 Cc1c(C(=O)NCCC2(O)CN(C(=O)C(C)C(F)F)C2)cnn1CCC(C)C C1(C)(C(C)O)CCCN1C(C1CCCN(C(c2ccc(C(=O)CF)cc2)=O)C1)=O c1(OC)c(NC(=O)NC2(c3ncco3)CCCCC2)cc(C)cc1C c1(SC)ccc(CC(=O)NC2CC(C)N(C(=O)C=CC(C)(C)C)C2)cc1 C(C)(C(C(=O)NC(c1cncnc1)C)C(C)C)NC(C1CCN(CC)CC1)=O N1(C(c2ccc(C)o2)=O)CCCCC2(C1)CN(C(=O)C=CC1CCCC1)C2 CC1COC2(C1)CN(C(C1CN(C(=O)CSC3CCOC3)CCC1O)=O)C2 c1(C(=O)NCCNC(C(C)(O)C(F)F)=O)c(F)ccc(OCC(F)(F)F)c1F CC1CCN(C)c2ccccc2N1Cc1cc(C(F)(F)F)n(C)n1 c1(CC(=O)N(C2CCC(N(C(=O)CCn3cccn3)CCO)C2)C)csc(Cl)c1 c1(N(CCCN2CC(C(CS(C)(=O)=O)=O)C2)C)ccc(Cl)cc1Cl N1(C(C(c2cnn(C)c2)C)=O)CC2C(C(=O)NC3CCN(C(=O)N(C)C)C3)C2C1 N1(C(C(=O)NC(CNC(C(CC=C)(C)C)=O)C)C)C(=O)NC2(CCCC2)C1=O c1(C(N2C(C(CNC(CN(C3CC3)CC)=O)(C)C)CCC2)=O)cc(C)ccc1F C1(C(=O)NC2C=CC(CNC(C(c3ccccc3F)(C)C)=O)C2)CCCC(=O)O1 C=CCC(C(=O)NCC1CCC(C(N2CCCCCC2)=O)O1)OC C#Cc1ccc(C(=O)NCCCC(=O)N2CCCC2C(C)(C)S(C)(=O)=O)nc1 C1(C(=O)NC2CN(C(C=NOC)=O)CC2C)CCC2C(C1)C2(F)F N1(C(c2cc(C)sc2)=O)CC(CNC(C2C(C)C2(F)F)=O)CC12CCC2 CC1(O)CC2CC1CC2NC(=O)CC1CCCCN1C(C1OC2CCC1C2)=O CC(C)C(C)C(CNC(=O)C=CSc1ccccc1)NC(c1cnc(S)nc1)=O C(CC(=O)Nc1ccc(Cl)cc1C)(C(C)(C)C)NC(C(CCC)C)=O N1(C(C(=O)NCC=C(C)C)=O)CC(NC(C2(C(C)(F)F)CC2)=O)CC(C)C1 c1(C(N(C2CN(C(C(CC)OC)=O)C2)C)=O)cnc(C)n1-c1ccc(OC)cc1 c1(C(N(C)CC2CCCN2C(=O)CCCn2cncn2)=O)cccn2nnnc12 N1(C(CC(CCC)(C)C)=O)CC=C(C(C)(C)C(=O)NCC2CC2CC(C)C)C1 C1(CNC(c2cn(CC)nn2)=O)CN(C)CCN1C(c1c(Cl)c(C)nn1C)=O c1(SC)cc(C(=O)NC2(CN(C)C(C3C(C)(C)C3(F)F)=O)CC2)oc1C Cc1ccc2sc(C(=O)NCc3ccc(CNC(=O)C(C)C4CC4)cc3)cc2c1 C1(CC(N2CC(OC)C(N(C)C)C2)=O)C2CCCC2N1C(=O)C(O)C(C)(C)C C(=O)(C1=NN(CCO)C(=O)CC1)N1C2CN(C(C(C)OCC#C)=O)CC1CC2 C(=O)(C(F)C1CCCC1)NCCCOCCN(C(=O)CCn1cccc1)C.C(N)(=O)N c1(CCC)cccc(C(=O)NCCC2CCN(C(C3(C)CC3(C)C)=O)C2)c1 C1(OC)CC2CC(NC(c3sccc3CNC(=O)CCC3CC(C)C3)=O)CC12 N1(C(C2CCCC3CC23)=O)CCC(C2CC2)(NC(=O)C(F)(F)CO)C1 N1(C(C2N(C(COC(CC)C)=O)C(C)CC2)=O)CCC2(CCC2)C(O)C1 Cc1ccc(C(=O)N(C2CN(C(c3sccc3C)=O)C2)C)cc1N1CCOCC1 CCCC(CC)CC(=O)NC1(CCNC(C2Cc3nc(C)cn3C2)=O)CC1 N1(C2CCCC(C)O2)CCC(O)(C(=O)NCCc2cnn(C)c2)CC1 CC1(C)CC(CNC(C2C(F)(F)C23CCC3)=O)N(C(=O)C=C2CCCC2)C1 CC(C)C(C)(CNC(=O)COCCCF)NC(C1CCOC1C(C)C)=O c1(C(=O)NCC2(CC(=O)OC)CCOC2)cc2c(=O)[nH]ccn2n1 c1(C2CCN(C(C(C)(F)c3cncnc3)=O)C2)ccc(NC(=O)OC(F)(F)F)cc1 N1(C(Cc2n(C)ccn2)=O)CCCN(C(=O)NCCc2ccncc2)CC1 Cc1cc(NC(=O)C(CC2CCCC2)NC(c2cc(C(C)C)on2)=O)ccc1Cl CC(C(=O)NCC12CC(NC(c3csc(=N)[nH]3)=O)(C1)C2)C(C)S(C)(=O)=O C(CCC(F)(F)F)(C(=O)NC1CC1)NC(=O)NC(CC)CSCOC c1(C(N(CC(CC)NC(Cn2ncc(CC)c2)=O)C)=O)cc(S(N)(=O)=O)ccn1 C1(C(=O)NCC(C(C)C)NC(c2cn(CC)nc2)=O)CCc2c(n[nH]c2C)C1 C1(NC(=O)CCc2ccccc2F)CCN(C(C2CCC2CF)=O)CC(O)C1 Cc1cccc(C)c1NC(=O)C(=O)NCC(Cl)C(F)(F)F N1(CC2CC(OC)OC2OC)CCOC(C)(Cc2cccc(Cl)c2)C1 C1(C(=O)NC(C2(CNC(c3cncc(NCC)c3)=O)CC2)C)CC(S(C)(=O)=O)C1 N1(C(CCCC(=O)NC)=O)CCN(C(=O)CCNC(C2CCCO2)=O)CCC1C C1(C(=O)NCCOCCCC)CSCN1C(=O)CC1(C)OCCO1 c1(C(N2C(C)CC(NC(c3c[nH]nc3[N+](=O)[O-])=O)C2)=O)ccnc(P(C)(C)=O)c1 c1(C(=O)NCCC(=C)CNC(=O)CC2CCOC(CC)C2)cnc2c(c1)CCC2 C1(CC(=O)NCCN(C)C(c2nccnc2N)=O)CCCC(O)C1 Cc1cn2nc(C(=O)NC3CCC(CCNC(=O)COC(F)F)C3)cc(C)c2n1 c1(NCCN(C(c2ccc(OCC)nn2)=O)C)ccc(-c2ccncc2)c(C)c1 c1(C(=O)NCC(CNC(CC(C)c2cccnc2)=O)O)cc2n(n1)CCO2 C1(NC(=O)C(C2CCCO2)C2CC2)CCC(NC(=O)C(C2CCCCC2)O)CC1 C(CC(F)F)(C(=O)O)N(C)Cc1cn(Cc2ccccc2)nn1.C12CC1C(=O)N2 C1(OC)(CNC(=O)C(CO)NC(=O)C(F)(F)F)CCN(C(=O)CC(C)(F)F)C1 C12(NC(C3(C)CC3)=O)CCC(CC1NC(=O)CCn1cc[nH]c(=O)c1=O)C2 C1(NC(CC(C)(C)OC)=O)CC2CCC1N(C(=O)COCC1(F)CC1)C2 N1(C(c2c(CC)noc2)=O)CCN(C(c2occc2CC)=O)C(COC)C1 CS(C)(=O)=NCC(=O)NC1CCCN(C(C2CCCCS2(=O)=O)=O)CC1 N1(C(C2C(C)(C)C2NC(c2cc([N+](=O)[O-])c[nH]2)=O)=O)CCC2(CCC(O)C2)C1 N1(C(CCCCC#C)=O)CCC2(CC1)COCC(CNC(=O)C(C)N(C)C)O2 CC1CN(C(C2(C)C=CCC2)=O)CCN1C(=O)Cc1cn(C)nc1C(F)F N1(CC(=O)N(C2CC2)Cc2cn(C)nc2C(F)F)C(=O)NC2(CCOCC2)C1=O n1(CC(=O)NC2CN(C(C3CCC(=O)NC3)=O)CC23CC3)ccc(O)nc1=O CC(CNC(=O)CCCC1(NC(=O)C(Cl)Cl)CCC1)C(C)O CCC(CC)CC(F)C(=O)OC(C)CC(=O)NCCC(=O)NC(C)(C)C c1(C(=O)NCCOC(C)=O)ccc(CNC(=O)CC2CCCCN2C)cn1 c1(C(N(CC(CN(C(C(C(C)C)OCC)=O)C)O)C)=O)ncn2cc(Cl)ccc12 Cc1cc(Cl)ncc1CC(=O)NCCN(C)C(c1ccnn1CCN(C)C)=O c1(CC(=O)NC(CCNC(Cn2c(C)ccn2)=O)C)ccc(Br)cn1 C1(C(N(OC)C)=O)C2CCC(C2)N1C(=O)CC(F)(F)F O=S(=O)(c1cccc(N2CCC(C3OCCO3)C2)n1)NCC(O)CN1CCOCC1 CC(C(C)NC(C1CS(=O)C1)=O)NC(=O)Cn1cncn1 CC1(C)C2CC(C(=O)NC3CC(O)C3CC(N3CCOCC3C3CC3)=O)CC12 c1(C(C)NC(COCCC)=O)ccc2c(c1)CN(C(=O)CC(O)C(C)C)C2 Cc1ccc2cc(C(=O)NCC3CCN(C(=O)C(C)N(C)C)C34CC4)nn2c1 Cc1nc2cc(Cl)cc(C(=O)NC(C)CNC(C3CCCN3S(C)(=O)=O)=O)c2[nH]1 c1(CC(NC(=NC)NCCC(=O)OCC2CCOC2)CC)ccccc1OC(F)F C1(NC(CC(C)C)=O)CC2(CCC(CNC(c3cnc(C(C)C)[nH]3)=O)OC2)C1 CCCCS(=O)(=O)N(C1CCCCC1)CC(=O)NC(C)C.N12CCC(C1)CC2=O c1(C(N2CCC(CCNC(C3CCCOCC3)=O)CC2)=O)noc2ccccc12 CC1(C(=O)NCC2(O)CCN(C(c3cc[nH]n3)=O)C2)CCCC1(F)F C1(CNC(c2cnc(CC)o2)=O)CC(C)(C)CN1C(c1cc(C(F)(F)F)ns1)=O C1(C(N(CC(C)(C)NC(c2ccc(CF)cc2)=O)C)=O)CCCC(=O)N1C C1(C#CC(=O)NC2(C)CCCN(C(c3cccc(Cl)c3C)=O)C2)(CC)CC1 c1(C(N2CC3CCCC3(CO)C2)=O)ccc(S(=O)(=O)N2CCCC(O)C2)cc1 Cn1cnnc1CN(C1CCNC1)CC(=O)NC1CCCO1 O(NC(=O)C(C)(CNC(c1cc(C)cc(F)c1)=O)CC)CC=C C1(CC(=O)OC(C)=O)CC=CCC1.C1(=O)C(C)N(C(C)C)C(C)CN1CC N1(C(C(CSC)NC(C2CC(CC)(CCl)C2)=O)=O)CCc2ccccc21 C1(C)(C(=O)OC)CCC1(C)C(=O)NCC1CN(C(C2CCOC(C)C2)=O)CCO1 C1(C(=O)NCc2n[nH]cc2C2CC2)C2CN(C(=O)C=C(C3CC3)C3CC3)CC12 c1(C(N2C(C(=O)NC3(C(=O)NC)CC3)CC2)=O)cncn(C)c1=O C1(CC)CCc2nc(CC3CC3)[nH]c2C1.C12CCCN(C1)C(=O)c1csc2n1 C1(N(C(C2N(CC)CCC2)=O)C)CN(C(=O)COC2COC2)CC1(C)C N1(C(CC2C(C)C2)=O)CCC(O)(C2CCN(C(=O)C(O)C(C)(C)C)CC2)C1 c1(C(=O)OC)n[nH]c(CN(C2CCCC2)C(c2ccn(C3CCCC3)n2)=O)n1 c1(CC(=O)N(CCCC)CC(=O)NCC(CCC)NC(C)=O)ccccc1C c1(C(=O)NC2C=CC(CNC(C(CCCCC)O)=O)C2)ccc2sc(C)nc2c1 C(CNC(=O)CCc1nc(O)n[nH]1)(CCNC(=O)CC1CC1)OC C1(CNC(=O)CCCc2cccs2)CCCC(NC(=O)Cc2ccco2)C1 C1(CC(C)N(C(C(N2CC(C(C(=O)OC)OC)C2)=O)=O)C)CCC(=O)N1 C=C(C)C(C)(C)C(=O)N1CCOC(CNC(C2CCC(=O)NC2)=O)C1 c1(CCC)n[nH]c(=NC(C)C2CCN(C(c3cc(C(F)(F)F)ns3)=O)CC2)s1 C(=O)(C(F)C(C)CNC(c1nonc1C)=O)NC(CC(=O)OCC)C S(=O)(=O)(c1ccc(NCC2(CC3CC3)CCCO2)nc1)N(CC(c1nccs1)C)C C(C)(C(C(=O)N1CCC(CC(C)C)C1)NC(c1ccc(C#N)o1)=O)OC N1(C(c2c(CC)ocn2)=O)CCC2(NC(c3cnc(O)c(C)c3)=O)CC2C1 N1(C(C(C2CC2)OC)=O)CCN(C(=O)COCCN(C)C)C(CO)C1 C(=O)(CCCC(C)=O)NCC(CCCC)NC(C1(C)CC=C(C)CC1)=O C1(NC(C(COC)OC)=O)CC2CN(C(=O)C3=C(C)OCC3)CC12 c1(NC(CC2CC(CC(N3CCC(n4cncn4)C3)=O)C2)=O)cc(F)c(Cl)cc1Br CCCC(C)(CCC)C(=O)NCC1COCC1NC(C1SCC=C1C)=O C1(C(=O)NC(C(=O)NC)C2CC2)CCC(C)(C)N(C(=O)COc2ccsn2)C1 C1(F)(C(=O)NCC(C)NC(=O)OC(C)(C)C)CCN(C(=O)C(F)CC2CC2)CC1 c1(OCCN(C(c2sccc2I)C(=O)NC(C)(C)C)C)ccccc1 c1(C(=O)NC2C(OC)CN(C(c3ccco3)=O)CC2)c(F)ccc2[nH]ccc12 c1(C(=O)NCC(C2CC2)NC(c2cn(CCCC#N)nn2)=O)cc(O)ccc1F CC(C)CC(CNC(C1Cc2nccn2C1)=O)C(=O)N(C1CC(C(C)O)C1)C C=Cn1nccc1C(=O)NCC(C)NC(c1cc(-c2cccc(O)c2)ccn1)=O C1(OC)CCC12CC(C(=O)NCC1CCC1NC(=O)Cc1cncnc1)C2 C12CC(O)CN1C2=O.C(CC(=O)N(CCNC(=O)OC(C)(C)C)C(C)C)=CC=C CCC(C)CC(=O)N(CC(C)O)CCNC(=O)CN1CCN(c2ccccc2)CC1 c1(C(N2CCC(C(=O)NC3(CC#C)CC3)C2)=O)ccc(O)nc1C c1(OC)cccc2cc(C(N3CC4CC3CN(C(C3CCC5CC35)=O)C4)=O)oc12 C(C1c2ccsc2CCN1C(c1ccc(F)cn1)=O)NC(C1CCC1(F)F)=O N1(c2snc(CCCCCC)n2)CCNCC1c1cccc(C(=O)O)c1 Cc1ccc([N+](=O)[O-])c(C(=O)NCCCNC(c2nccc3ccccc23)=O)c1 CC(C)CCC(=O)NC1CCC(CNC(=O)C=CC(=O)Nc2ccccc2Cl)C1 C1(OC)CC2(C1)CC(C(=O)NC1CN(C(=O)C(C#N)C3CC3)CC1O)C2 c1(C2(C)CC2NC(=O)C(=O)NCC2C3CCC2NC3)ccccc1F C1(NC(CC2(OCC)CCC2)=O)C=CCCC1C(=O)NCC1CCSC1 c1(C(=O)NC2CC(C)(CNC(=O)CSCC(N)=O)C2)ccc(N(C)C)nn1 c1(C(N2CC(F)(C(N3CC(C)C(F)C3)=O)C2)=O)c[nH]nc1[N+](=O)[O-] c1(C(C)CN(CC)NC(=O)COc2nc[nH]n2)nc(C)no1.C1(C)COCCO1 C1(C(C)C)CN(C(C2CCCC(F)C2)=O)CCN1Cc1ncccn1 c1(C(N(C(C(=O)NCCCC=C)C)CC)=O)ccn(CC)n1 N1(C(C2(OC)CCC2)=O)CCC2(C1)CN(C(=O)Cc1ccc(C#N)nc1)CCO2 C1(C(=O)NCC(C2CCCC2)NC(C2CC(=C)C2)=O)CC=CC(O)C1 c1(C(=O)NC2CCC(NC(=O)Cn3cnnc3)C2)cccc2ccncc12 C1(C)(CC)CCC(C(=O)NC(CN(C)C)C(=O)NCC(C)(C)n2ccnc2)O1 C1(NC(C(c2ccc(C)o2)C)=O)CCCCC1N(C(=O)Cn1cc(Cl)cn1)C c1(C(=O)NCCCC(=O)NCCc2nc(C)sc2)cc(O)cc(=O)o1 CC(C)(C)C#CC(=O)N1CCC(CF)(NC(=O)CC(C)(C)c2cccs2)C1 N1(C(C(C)N(C(=O)CN=[N+]=[N-])C)=O)CCC2CC12C C(=O)(C1=CCCCC1C)NCC(=C)CCNC(=O)Cc1cccc(O)c1F C#CC1(NC(C23CCCC2C3)=O)CN(C(=O)COc2cn[nH]c2)C1 c1(C(=O)NCC(C)(C2CC2)NC(C(C)=C2CCC2)=O)cc2ncccc2s1 C(CC(C(C)(C)C)NC(c1cnnn1C)=O)N(C)C(C1CCC(=O)C1)=O N#Cc1ccccc1OCC(=O)NCCC1CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)C1 c1(C(=O)NCC(F)CNC2CCCO2)[nH]cc2c1CCS2(=O)=O c1(OC)ccc(I)c(C(N2CCCC(NC(c3ccc(Cl)nn3)=O)C2)=O)c1 CCC(C)CCC(=O)NC1CC(CC(=O)N(CC(C)C(C)C)C)C1 N1(C(c2c(CC)con2)=O)CCC(C(=O)NC(C)C2CC2)=C(F)C1 C1(C(N(CCNC(=O)C(O)c2ccsc2)CC)=O)SCCCS1 C(C(C(=O)NCCc1ccncc1)NC(=O)CCC1CC1(C)C)OCC N1(C(C#CC2(CC)CC2)=O)C(CNC(C2C3COCC23)=O)CC2COCC12 C(=O)(C(C)(C)C1=CCN(C(=O)CCc2cnco2)C1)NC(C#C)CC(C)(C)C C1(C(=O)NCC=CCNC(C(C)(C)NC(=O)NCC)=O)CCC2CCC1O2 C1(CNC(C2CC2C(=O)OC)=O)CCOC1.C(C(=O)N(C)CC)=CCC.C(=O)(CO)N CC(Cn1ccnc1)C(=O)NCCNC(=O)Cc1csc(Br)c1 CCC(C)CC(=O)C(=O)N(CC(C)C(=O)NC(C)(CSC)CO)C C(=O)(CCC(C)CC)NC(CCC)CNC(c1cc(CC2CCC2)c[nH]1)=O N1(C(C23CC(NC(c4cc(C)c(O)nc4)=O)(C2)C3)=O)CC2(CCC(=O)O2)C1 O=C(C1Cc2ccc(Cl)cc21)NCCCOCCNC(=O)Cc1cnoc1 C(=O)(C(C)(O)C(F)(F)F)N(CCN(C(c1cnn(CC(C)C)c1C1CC1)=O)C)C n1(CC(C)(C)C)nc(C2CCOC2)nc1-c1cn(CCc2ccccc2)nn1 c1(C(N2C3CN(C(c4c(OC)nc(C)cc4)=O)C(C3)C2)=O)ccc2[nH]ccc2n1 c1(N(C(C2(F)CCN(C(C)(C)CN(C)C)CC2)=O)CC)ccc([N+](=O)[O-])cc1Br c1(CC(=O)NC(c2ccccc2)CNC(C(C)N(C)C)=O)ccc(C(F)(F)F)nc1 C1(CNC(CCC#C)=O)CC(F)(F)CN1C(C1CCN1CC)=O C1(NC(C=CCN(CC(F)(F)F)C)=O)CCCN(C(c2cc(C)ns2)=O)C1 c1(C(=O)NCC(=O)N(CCCCCNC(C(CC)SC)=O)C)ccc(O)cc1 C1(NC(N2CC(OC3CCN(C(C(C)(C)C)=O)CC3)C2)=O)CN2CCN1CC2 C(=O)(CC(CNC(=O)OC)OC)N1CC(COCC)C1.C(C)(C1CC1)=CC(=O)N Cc1nn[nH]c1CC(N1CCC(C2CCCN2C(=O)C(c2cccn2C)=O)C1)=O C1(C(=O)N(C2CC2(Cl)Cl)CC2CC2)C2CCN(C(=O)CN3CCOC3=O)CC12 c12ccc(-n3cccn3)cc1[nH]c(=O)c(=O)n2CC(C(=C)C)C.CC.CC N12CCCC(C1)C(=O)NCC2.CC(C)(C)OC(=O)NCC(N)=O c1(CC)nn(C)cc1C(=O)NC(C1CCN(C(C2(Cl)CC2(F)F)=O)CC1)C(C)C CCCC(CC)CCC(=O)NCC(c1ccccc1)NC(C1CCC1(C)C)=O Cc1ccc(C(=O)N(C(C)CCNC(=O)Cn2cc(Cl)cn2)C)c(Cl)c1C Cc1cc(Cl)ccc1-n1cc(CN(C(=O)CCCCOCC2CCC2)C)nn1 c1(C(=O)NCc2cccc(C(F)(F)F)n2)csc(=NCc2sc(Br)nc2Br)[nH]1 C1(CNC(CCc2c(C)noc2)=O)CC2(CC2)CN1C(=O)CC1CNC(=O)C1 N1(C(COCCOCC)=O)CC2(CCCC2NC(C2COCCO2)=O)C1 C(=O)(CCCC(=O)NC1CCOCC1)N(CCCOCCNC(C(CC)O)=O)C CCC(C)(C(=O)N1CC(NC(=O)C(C)(C)OC)C(c2cccc(F)c2)C1)C(F)F CC1(C)C(c2ccccc2)CC(C(=O)Nc2scc3c2OCCO3)S1(=O)=O CC1CN(C(=O)C=CCN2CCCC2)CC1NC(C1CCC(C(N)=O)N1C)=O Cc1ncc(N)cc1C(=O)N(CCC(C)NC(c1ccc(Cl)[nH]1)=O)C C=CCC(COC(c1nc(CC)oc1C)=O)CO C1(NC(c2c(C)scc2)=O)CCC2(CCN(C(C3(F)CC=CC3)=O)C2)C1 c1(C(N2CC(NC(C3(CC#C)CCC3)=O)C(O)C2)=O)ccc(Br)cc1O C(=O)(CC(c1ccccc1)C1CC1)NC(C1CCN(C(c2cncs2)=O)C1)C Cc1ccn2cc(C(N3CCCC(NC(=O)C(C)CC(C)(C)C)C3)=O)nc2c1C c1(C(C(=O)NCC)N(C)Cc2cncn2-c2ccccc2)cc(Cl)cc(Cl)c1Br CC(C(C)(C)C(=O)NCC(c1ccncn1)=O)NC(=O)OC(C)(C)C n1(CC=CC2=NC(c3ccccc3)C(=O)N2)ccc(=NC2CCS(=O)(=O)CC2)[nH]1 N1(C(C(C=C)O)=O)CCC(C(C)C(=O)NC(CC)C(C)CN(C)C)CC1 CC1(C)CCN(C(C2CC2(Cl)Cl)=O)C1CC(=O)NCC(O)Cn1cccn1 C12(NC(c3cnc(OCC)s3)=O)CCCC1CN(C(c1cc(C)n(C)c1)=O)C2 c1(NC(c2sccc2Cl)=O)cnc(C(=O)Nc2c(OC)c[nH]n2)nc1 c1(OCC)ccccc1C=CC(=O)NC1CCC(OC)C1.C12CN(C1)C2=O N1(C(CC(C)OC)=O)CCC2(CCN(C(C3CC(c4ccccc4)C3)=O)CC2)C1 C1(NCc2c(OC)ccs2)CCC(C(=O)NC2(C)CCOCC2)CC1 C1(NC(c2nc(CC)oc2)=O)CCCN(C(C2CCC(=O)N2C)=O)C1C N1(C(C(CO)NC(c2c(CC)nccc2)=O)=O)CCC(O)C(C)C1 c1(C(N2CC(N(C(=O)C=Cc3ccsc3)C)C(C)(C)C2)=O)cnn2c1OCCC2 N1(OCc2c(F)cc([SH](=O)=O)cc2F)C=CNc2cc(Cl)c(Br)cc21 C1(C(=O)O)C(c2ccc(CO)cc2)C2CCC1N2CC(O)C(F)(F)c1ccccc1 c1(CCN(C)CC)cn(CCCCNC(C2CC(C)=NO2)=O)nn1 CC#CCCCC(=O)NCCOC1(CNC(=O)CN2CCCCC2=O)CCOCC1 C1(NC(CNC(C)=O)=O)CCN(C(C2CC(C)CO2)=O)CC1 C1(CNC(=O)CCCc2ccsc2)CCCC2CN(C(c3cncnc3)=O)CC12 C1(CNC(C(C)OCC#C)=O)CC2CCC(C1)N2C(C1CC2(CCCCC2)C1)=O C1(CNC(CC=C)=O)CN(C(c2nn(C)c(C)c2[N+](=O)[O-])=O)C2(CCOCC2)C1 C(C1=CCN(C(=O)NCC(c2ccc(F)cc2)C)CC1)OC N1(C(c2ncc(OCC)nc2)=O)CCN(C(=O)CSC2CCCC2)C(C)CC1C C12C=CCN(C1)C(=O)CCCOC2=O.c1(NC(C)=O)ccc(C(=O)C(C#N)Cl)cc1 Fc1cc(Cl)ccc1-n1nc(C2CCOCC2)nc1-c1ccnc(F)c1 N1(C(C(C)N(C)C(C2CCSCC2)=O)=O)CCC(C2=NOCC2)C1 c1(NC(c2cn(CCC(C(=O)NCC)O)nn2)C)ccc(OC(F)F)cn1 C(=O)(CC(C)(C)C(=O)N1CC(NC(=O)C2CC2)C(CC2CC3C=CC2O3)C1)OC C(=O)(CCCCN(C)C(C1CCN(c2ccccc2)C1)=O)NCC(C)CN(C)C Cn1c(NC(N2CCC(n3ccc(O)nc3=O)CC2)=O)nc2ccccc12 c1(C(=O)NCC(c2ccccc2)CNC(CC=CCC)=O)ccc(Cl)c(F)c1 C1(C(C)C)CN(C(C2CCCCC2CNC(C2CCOC2(C)C)=O)=O)CC(=O)N1 C(=O)(C1=C(F)CN(C(c2cnnn2C)=O)CC1)N(C1CCCNC1=O)C Cc1cncc(CCNC(C2(C)CN(C(=O)CC3OCCC3(C)C)C2)=O)n1 c1(NC(COC)=O)ccc(C(=O)NC2(CO)CN(C(=O)C(C)CC(N)=O)C2)c(C)c1 Cn1c(C(=O)NC2COC3CN(C(=O)CC4(C5CC5)CC4)CC23)cc2occc12 c1(C(N2CC3CCN(C(c4cccc(C)n4)=O)C3C2)=O)cc(C)n2ccnc2n1 C=C1CCN(C(C2CC(=O)OC2(C)C)=O)C(C(=O)NCCCOCC(F)F)C1 Cc1cncc(C(=O)NCC(F)CNC(=O)C(c2ccccc2)N2CCCC2)n1 C(N=c1nc(N(C)Cc2ccc(CO)s2)c2c([nH]1)CCC(C)C2)c1ncc(C)cn1 C12(C(=O)OCC)CN(Cc3cnc(Cl)c(Cl)c3)CC1CCCO2 CCC(CNC(=O)COCc1ccnc(O)c1)(CC)C(=O)NC(C1CCC1)C N1(C(CN(CC)CC)=O)CCCC2CCN(C(=O)CSCCC#N)CC12 N1(C(CNC(CC)=O)=O)CCC2CCN(C(=O)Cc3nccn3C)CC2C1 C1(NC(=NC)N(C)Cc2nc(C(F)(F)F)cs2)CCc2nnnn2CC1 Cc1cncc(C(=O)NC2CC(C)N(C(c3ccc(CN(C)C)nc3)=O)C2)c1 CC(C)CC(C(=O)NCCC1CC(=O)N(C)C1)NC(C1CNC(=O)N1)=O C1(C(N(C2CCOC2)C)=O)N(C(=O)CC2(O)CCOC2)CCCC1(C)C O=C(C1Cc2ccccc21)N1CC(F)(C2CC2)C1 N1(C(Cc2cn(CC)nc2)=O)CC(O)CC1CNC(=O)Cc1cnccn1 c1(N(C)C)ccc(-c2nc(Cn3cccn3)nn2-c2ncccc2Cl)cc1OC c1(CC(=O)N(CC(CNC(CCC=C(C)C)=O)C)C)nsc2ccccc12 Cc1cc(C(=O)NCC23CC2CN(C(c2ccccc2O)=O)C3)c(C)s1 CCC(F)(C(=O)OC)C(=O)NCCC(C)N(C)C(c1cnsc1C)=O CCC(N=c1nc2scnc2c(N2CCC(F)(F)C(C)C2)[nH]1)C1CCCC1 N1(CC)CC(C(=O)NC2CN(C(c3occc3C)=O)CC2O)CC1=O C1(C(=O)NC2CCC(CNC(=O)C=Cc3ccccn3)C2)CCC(C2CC2)CC1 c1(C(N2CCCC(CNC(C(CC)(C)OC)=O)C2)=O)cc2c(s1)CCS(=O)(=O)C2 C1(C(=O)NC(CC)CNC(=O)C(O)CNC(=O)OC(C)(C)C)CCSCC1 S(=O)(=O)(c1ccc(NCC2CC3CC3C2)c(Br)c1)NCc1c(C)cc(Br)cc1 c1(C(=O)NC(CNC(C(F)=C(C)C)=O)(C)C2CC2)ccc(C(C)(C)C)[nH]1 c1(C(N(CCCCN(C(C2CCN(C)CC2)=O)C)C)=O)cnc2c(c1)CNC2=O c1(OC(CCSC(C)(C)C)=O)ccc(F)cc1SCCC(F)(F)F Cn1nc(C(F)(F)F)c(N)c1C(=O)NC1(C)CC(NC(C2(C)CC(F)C2)=O)C1 N1(C(CN(C(=O)Cc2cnoc2)CCOC)=O)C(CO)CC1C N1(C(C=CC(=O)N(C)C)=O)CCN(C(C2CCC2)=O)C2CC12 C#CCCCCC(=O)NCC(C)(F)CNC(C1CCCCC1CF)=O Cc1cc(N2CCC(NC(=O)CC(F)(F)C(F)F)C2)cc(C#N)n1 c1(CC)ccc(Cc2nc(-c3cn(CC)cn3)n(CC3CC3)n2)cc1 C1(CNC(CC=CC=C)=O)(NC(c2c[nH]c(=N)o2)=O)CCCCC1 c1(C(=O)NC(C(=O)NC(C=C)(C)CC)Cc2cnc[nH]2)ccsc1C#N C1(CNC(C(C)=NOCC#N)=O)CC(O)C(O)CC1C(=O)NCC(CO)C1CC1 C1(C(=O)NC2(C)C(C)C2)C2CC1N(C(=O)Cc1ccon1)C2 C(CC(=C)C)(C(=O)OC)NC(CC#C)C(=O)OC(C)(C)C C1(NC(COC2CN(C(C)=O)C2)=O)CC(NC(c2scnc2C)=O)CC1O CCCC(C)C(C)NC(C1(CNC(=O)COCCCN=[N+]=[N-])CCC1)=O C1C(C(F)(F)F)O1.C1(C(=O)NC)CCN(C(=O)N(c2ccnn2C(C)C)C)C1 C1(C(N(CCCNC(CC=C)=O)CCO)=O)CCOC2(CCC2)C1 C1(CNC(CC(=O)OCC)=O)CN2CCCCC2CN1C(=O)CP(C)(C)=O N12CCOc3cc(ccc31)C2C(=O)NCCCC(=O)OC.C(C)C.C(N)=O C1(CNC(=O)CC2CN(C(=O)CCCn3ccnn3)C2)CC2(CC2)C1.[nH]1ccnc1 c1(NC(c2nc(Br)nn2C)c2n(CC(=C)C)nnn2)nn(CC)nc1C C1(F)(C(=O)NCC)CCN(C(=O)CCC2CC2C)C1 C1(CC(=O)NCCCCC)CCCN(C(c2sccc2Br)=O)C1 c1(C2C(NC(CN(C(C(C)=CC=C)=O)C)=O)C2)cnn(C)c1 CC(=O)CCCCC(=O)N1CCC(NC(=O)CC2COCCO2)C(CO)CC1 N1(C(CC2C(C)=NN(C)C2=O)=O)Cc2ccc(C#N)cc2C1 c1(C(=O)NCCCOCC(C)(C)NC(C2C(C)CCS2)=O)ccccc1F c1(OC)cc(O)ncc1C(N1CCC(NC(C2CCCS2(=O)=O)=O)C(F)C1)=O C1(NC(=O)Cn2nnc(-c3ccsc3)n2)CC(O)CN(C(c2cnco2)=O)C1 C12(C(=O)NC3CCC(NC(=O)CCc4ncco4)CC3)CC=CC(C1)OC2 C(=O)(C1COc2ccccc21)N1CCCC(COC)(NC(=O)C#CC(C)C)C1 C=C(C)CCC(C)(c1nnnn1CCCSCc1ccccc1)NCC1CCCO1 C1(C)(CC(=O)N(CCNC(CCC=CC)=O)C(C)C)CC(F)(F)C1 C(=O)(CC(O)C(=C)C)NC1CC(N(C(CC=C=C)=O)C)C1 c1(C(=O)NCC2(C(F)(F)F)CCCC2)ccc(Oc2ccc(Br)cc2)cn1 c1(OC)cccc(C(C(=O)NCCC(C)(C)NC(C2CCCN2C=O)=O)OC)c1 C1CC2(C1)CC(CO)CC13C2C(C(=O)OC)CCCN(C(CC)C1=O)C(=O)N3.OC c1(C(=O)NCC(C)(C2CCC2)NC(C(C)n2cncn2)=O)cccc(CO)n1 C1(NC(c2n(C)ccc2)=O)CCCN(C(c2csnc2-c2ccccc2)=O)C1 c1(C(=O)NC2CC3(CC(NC(C(CC)C(C)O)=O)C3)C2)nccc2n[nH]cc12 c1(-c2nc(C(CCC)C)nn2-c2ccc(OC)c(C)n2)cc(C)c(C)c(Br)c1 c1(OC)ccc2[nH]c(=NC3CC(NC(C4CC4C4CC4)=O)C3(C)C)sc2n1 CCCCC(CNC(c1cnc(SC)n1C)=O)NC(=O)C(C)OCC1CCCO1 C1(C(=O)NCC2(O)CCN(C(CCC=C)=O)C2)COc2ccc(Cl)cc2O1 n1(CCC)ncc(C(=O)NC23CC2CN(C(=O)CCC2CC2(C)C)C3)c1C N1(C(=O)CCc2ccon2)CCC2CCN(c3nnc(C(F)F)s3)CC2C1 c1(CN2CCC(C)C2C(F)(F)F)cccc2c1OCCC2 c1(C(=O)NCC(C)(CNC(C2(C(F)F)CC2)=O)OC)cc([N+](=O)[O-])nn1C Cc1nc2ncnn2cc1C(N1CCC(C)N(C(=O)C=CCn2cncn2)CC1)=O c1(C(C)C)n[nH]c(=NC2CC(NC(=O)C(C3CC(F)(F)C3)O)C3CC23)o1 C(=O)(C(C#N)C(C)(C)C)NC1(C)CCN(C(C2(COC)CCOC2)=O)CC1 c1(C(C(=O)NCCOCCN(N2CCCCC2)C)N(C)C)noc2c1CCCC2 C1(NC(=O)C=CC2CCOC2)CCCC12CN(C(C13CC(F)(C1)C3)=O)C2 CC(CC(=O)N1CCC(O)(CCNC(=O)CC2C=CS(=O)(=O)C2)CC1)C(F)F O=S(=O)(c1c[nH]ccc1=NC1CC2CCC(C1)O2)N(C1CCC1)C1CC1 C(C)(CCC(=O)N1CCOC(CNC(=O)CCc2nc(C3CC3)no2)C1)OC Nc1cc(F)cnc1C(=O)NCCCOCCCNC(C1CCC2CC12)=O c1(N(C(=O)NC(Cc2cccc(C)c2)CO)C(C)C)cc(Cl)ccc1C C#CC1CCC(C(N2CC(O)(CNC(C3CC(=O)N(CCC)C3)=O)C2)=O)CC1 C(C(=O)NNC(=O)C1CCCC1OC)OCC Cc1cccc(C(F)(F)C(=O)N2CCCC2CNC(=O)CN2C(C)CCC2C)c1 O=C(N=c1nc[nH]n2cccc12)c1csc(-c2cnn(CCO)c2)n1 N1(C(C=CCC)=O)CC(CNC(=O)CC2CCCNC(=O)C2)OC(C)(C)C1 c1(NC(=O)CC2CN(Cc3cnc[nH]3)C2)cc(Br)cn2ccnc12 c1(OC)cc(CO)ccc1C(N1CC=CC(NC(=O)CC2CCC(=O)NC2)C1)=O N1(C(c2nc(C(=O)OCC)sc2)=O)CCC2CCC12CNC(c1sccc1C)=O N1(C(CCc2cncc(C)c2)=O)CCC2(CCCC2C(=O)NC2(CO)COC2)C1 Cc1ncc(C(=O)NCC2CN(C(=O)C=CC3CCCC3)CCO2)cc1N C1(NC(CCN(CCC)C)=O)CCCC1NC(c1cscc1C(F)F)=O O=C(C1NCCc2ccc(Br)cc21)N1CCOC(Cn2ccnn2)C1 c1(OC)ccc(F)cc1CCC(=O)NC(C1CCN(C(C2(C)CC2)=O)CC1)C c1(C(=O)NC2C(NC(C=C(C)C3CC3)=O)CCC2)nn2c(c1C)CCCC2 CCC(C)(C(=O)NCC1CN(C(=O)C#CC(=O)N(C)C)CCC1(F)F)C(F)F C(=O)(C1Cc2ccc(F)cc21)N1C(C2CCCN(C(=O)C=C3CCC3)C2)CCC1 C(CC1=CCCCC1)C(N(C(C)CN(C(=O)C(O)Cc1cnc[nH]1)C)C)=O C1(C(=O)NCC2CN(C(C=CCCC)=O)C(C)C2)CCC(=O)CC1(C)C CC1(C)CNCC1CC(=O)NCc1csc(-c2ccccn2)n1 c1(OCCOC)ccc(CCCNC(=O)C(=O)NCCc2ccsc2)cc1 c1(CC)n[nH]c(=NCC2CCCC(NC(c3ccnn3COC)=O)C2)s1 C1(C(=O)NC2C=CC(C(=O)NC(C)CCN3CCCC3)C2)CC2CCC2C1 C(=O)(CCCC(=O)N1CCC(O)(CCNC(C2CCC2C)=O)CC1)NCC N(C)(S(=O)(=O)N(C)C)CC(CNC(C(C(C)C)F)=O)C.C(=O)C C#CC1CCCCN1C(=O)C(CCOCCO)NC(c1sccc1CO)=O C(=O)(C(C)S(=O)(=O)C1CCOCC1)NC12CN(C(C(C)(C(C)C)OC)=O)C(C1)C2 N1(C(=O)CC2CCOC2)CCC2(CC1)CN(C(C1CS(=O)(=O)C1)=O)CCO2 Cc1nc(C(=O)N(CC(C)NC(=O)Cc2cccc(C(C)C)c2)C)n(C)n1 N1(Cc2ccc(O)nc2)CCN(C(=O)Oc2c(OC)cccc2)C(CO)C1.C(C)(C)O C1(C(=O)NCC2(NC(C(COCC)C)=O)CCOCC2)CCCCN(C)C1=O C=C1CCN(C(=O)CCC(C)OCC)C(C(=O)NCC2CC(O)(CC)C2)C1 Cc1noc(N)c1C(=O)N(CC(C)CNC(C1CCN1C1CCCC1)=O)C CCS(=O)(=O)c1ccc(C(=O)NCC2CN(c3cc(O)ccc3Cl)C2)c(Cl)c1Cl CC1CN(C(C2CCCC2)=O)CC1CC(=O)NCCC1CC1 c1(CC(=O)NC2CN(C(C(CC)n3ccnc3)=O)CC2C)cc(Cl)ccc1F C1(C(=O)NCCCc2c(C)n[nH]c2)COCCN(C(c2nccnc2N)=O)C1 c1(OC)ccccc1N=c1scc(-c2sccc2C)n1CCC1CCCSC1 C1(CCCC)Cc2ccccc2N(C(=O)CCc2cn(C(C)(C)CO)nn2)C1 C1(OCC=C)CCN(C(C2CCCSC2)=O)C1 C1(C(=O)NCc2c(C(N(C(c3ncccn3)C)C)=O)occ2)CCOC(C)(C)C1 N1(C(COCCC=C)=O)CCC2C(C1)NC(=O)CN2C(=O)CCC(C)(C)[N+](=O)[O-] N1(C(CC=CC=C)=O)CCCC(CN(C)Cc2nnc(C(C)(C)C)s2)C1 c1(OC)c(C(N2CC(OC)C(NC(=O)C(CCCO)N(C)C)C2)=O)cnn1C c1(CC)cccc(NC(=O)C(=O)NCCNC2CC2)c1.N12CCC(CC1)C(=O)N2 Cn1nc(C2CC2)c2c1CN(C(=O)OCC1CCN(c3cccc(F)c3)C1)CC2 N1(C(Cc2ccn(C)c2)=O)CC2(CNC(C3CC(F)C3)=O)CC1CCO2 C1(C2CCCOC2)(NC(C(Cc2cn[nH]c2)NC(c2c(C)snn2)=O)=O)CC1 N1(C(c2c(F)ccc(C)n2)=O)CCC2CCN(C(C3(n4cnnn4)CC3)=O)CC12 N1(C(c2c(C)sc(Cl)n2)=O)CCOC2(CCC(NC(=O)C(C)(C)CC#N)CC2)C1 c1(COC(=O)COC2CCC2)ccc(OCC2(C(=O)O)CC=CCC2)cc1 COn1cnc(C)c1C(=O)NC1CC(CCNC(C2OCC3CCCC23)=O)C1 c1(C(N2CC(F)CC(NC(c3coc(O)n3)=O)C2)=O)ccn2ncccc12 Cc1cc(C(=O)NC2CN(C(C3(c4ncccc4F)CC3)=O)CC2C)ncc1Cl CCC(C(=O)N1CC(F)CC1CC(=O)NCC1CCCCN(C)C1)C(F)(F)F C1(CC(=O)NC(CCOC)CNC(c2ccc(C)nn2)=O)CCC(C)(C)CC1 c1(C(CC)NC2CN(C)C(C)C2)cc(C)ccc1OC C1(NC(C(C)NC=O)=O)CCOCC1C(N1CC(CC2CCC2)C1)=O c1(C(=O)NCC(O)CC(=O)N2CCCSCC2)ccc(F)c(F)c1 CC1CN(C(c2nnc(S)n2C)=O)CCCN1C(c1ncccc1C(F)(F)F)=O c1(CNC(Cc2cccc(NC(C(C)(C)C)=O)c2)=O)nc2cccnc2s1 Cc1cc(F)c(C(N2CC(c3cn(Cc4ccc(Cl)cn4)nn3)C2)=O)c(Br)c1 Cc1ccoc1C(=O)NCC(=O)NC1C=CCC1 c1(C(=O)NCCCNC(c2cnc(O)c([N+](=O)[O-])c2)=O)ccc2c(c1)CCC2=O c1(C(=O)NCC(C)N(C(CCC(CC)C)=O)C)ccc2nc(C(F)F)[nH]c2c1 C1(C(=O)Nc2ccccc2-n2cccn2)CCCN(C(=O)CCn2cccc2)C1 CC(C)(CNC(C1(F)CCCN(C(=O)C2=CCSC2)C1)=O)C(F)(F)F N1(C(CC(C)C(C)(C)C)=O)CCn2c(CNC(=O)CSS(C)(=O)=O)nnc2C1 CSC=CC(=O)N1CCCC1CN(C(=O)C=CSCC(F)(F)F)C C1(C(=O)NC(c2ccc(C)cc2)C)C2CCC(C2)N1C(c1ccc(F)c(Br)c1)=O CS(=O)CCC(=O)NC1CC2(C1)CC2NC(=O)CC1CC2(CC2)C1 C(=O)(CCS(C)(=O)=O)NC(C(CO)NC(C(C)C(=O)N1CCOCC1)=O)C.C(=O)C1CC1 C1(C(=O)NCC2(NC(C3CC3C(F)(F)F)=O)CCCCC2)C2CCC3C(C2)CC13 C(=O)(C(F)(F)CO)N(CCN(C(C)C)C(c1c[nH]c(=N)s1)=O)C c1(C(N2CC(C(N)=O)C(O)C2)C(=O)NCCCSC)nn(C)nc1Br c1(OC)c[nH]c(C(=O)N(C)CC2(O)CCN(C(C3CCOC3)=O)C2)cc1=O c1(C(=O)NC2CC(OCC)C2)ccn2c(-c3cc(F)cc(F)c3O)cnc2c1 c1(C(N2CCC(NC(COCCOC)=O)(CO)C2)=O)cn2cccnc2n1 N12CCC(C13CC3)Cc1cccc(c1)C2=O.C1(CC(=O)OC(C)=O)OCCC1C N1(C(c2c(OCC)nccc2)=O)CCCCC(CNC(=O)Cc2cnc(C)[nH]2)C1 N1(C(CCC#C)=O)CCN(C(c2cc(C)cc(O)c2)=O)C(CC(F)F)C1 C(=O)(CCCn1ccnn1)N(CCN(C(=O)Cn1ccccc1=O)C(C)C)C C1(C#N)(CCC(=O)NC(CC)CN(C(=O)C(c2cscn2)N(C)C)C)CCC1 C12(O)CCCN(C1)C2=O.C#CCCCC(=O)N(C1(c2ccccc2)CCC1)C c1(N(CC=C)CCO)ccc(S(=O)(=O)N2CCCC2CC2CCCN2)cc1Cl C=CC1CN(C(=O)CCCSC)CC1NC(C12CC(C)(C1)OC2C)=O c1(NC(N2CCC3(CC(C(OCC)OC)C3)CC2)=O)cnc(P(C)(C)=O)cn1 c1(C(N(C2CCCN(C(C3CNC(=O)N3)=O)C2)CC)=O)c[nH]c(=O)cn1 C(CCN=C(NCc1cocn1)NCC1CCCO1)c1nnc(C)s1 C(CNC(=O)CCN1CCN(C)CC1)(C(C)(C)C)NC(C1C(C(=O)OC)C=C1)=O c1(OCC)ccc(CC(=O)NC2CC2NC(c2cnn(CCF)c2)=O)cn1 N1(C(Cc2c(C)non2)=O)CCC(C(=O)NC(C)Cn2ccnc2C)C12CCC2 c1(C(C(C)NC(C)(C)C)NC(CNC(=O)OC)=O)ccc(Cl)cc1OC c1(C(=O)NC2C(C)(C)CN(C(=O)C3=CCCCC3)CC2)cc(C#N)c(O)nc1N C1(C2CCN(C(C3COC3)=O)CC2)(NC(C2N(CCC)CCC2)=O)CCC1 CC1CC(NC(c2c[nH]cc2Br)=O)CN1C(=O)C=CCn1cncn1 c1(C(=O)NCCCN2CCC(NC(C=CC(CC)C)=O)C2)cnc(S)n1C N1(C(C2(N(C)C)CC2)=O)CCC2(CC1)CC(NC(=O)CCC1CCCO1)C2 C12(C(=O)NCC3C(NC(C4C(C)(C(C)C)C4)=O)COC3)CC(C#N)(C1)C2 C1(C(=O)NCCC2CCN(C(CC)=O)C2)CCC2(CCCCC2)CC1 c1(C(=O)NCC2(NC(c3ccc(Br)c(O)c3)=O)COC2)c[nH]c2cccc(Br)c12 CC(C)C(C(C)NC(=O)Cc1cc[nH]c(=N)c1)NC(=O)CC=Cc1ccccc1 CC1(C)C(C(=O)NCC2(C)CCCS2)CCN1C(c1cccc(O)c1F)=O CCS(=O)(=O)c1ccc(C(=O)N=c2cns[nH]2)c(Br)c1 Cc1ncc(C(=O)NCC2CCCN(C(C3C4CCCCCC34)=O)C2)c(=N)[nH]1 C(CNC(=O)C(C)NC(C1CCCC1)=O)(C(C)C)NC(C(C1CC1)OC)=O S(=O)(=O)(c1cccc(Cl)c1Cl)N1CCC(NC(c2c(CSCC)cccc2)=O)C1 CC(C)(CNC(C1(C(C)(F)F)CCC1)=O)CC1CN(C(C2CNC(=O)N2)=O)C1 C=CCC(C)(C)CC(=O)NCCC(O)CNC(c1cc([N+](=O)[O-])nn1C)=O C1(C(=O)OC)CC(C)CCN1C(=O)Nc1cn(CCF)nc1Cc1ccccc1 C1(C(=O)NC2C(C)CN(C(=O)C=C3CCCCC3)C2)CCCC(F)(F)C1 C12(CNC(C(C(C)C)(C)O)=O)CCCCC1N(C(c1ccc(Cl)s1)=O)CC2 N1(C(c2cccc(F)c2)=O)CCN(C(C23CCCN(CC2)C3)=O)C2(CCC2)C1 C=CC1(O)CN(C(C2CC=CCN2C(=O)C(C)C2CCC2)=O)C1 c1(CN2CC3(C(C(=O)Nc4c(C(C)=O)ccc(Cl)c4)C3)C2)ccc2occc2c1 C12(NC(c3cc(Cl)ns3)=O)CCCC1CN(C(=O)CCOc1ccc(F)cc1)C2 c1(N2CCCC(COC)C2)nccc(=NCc2cc(C)cc(Cl)n2)[nH]1 c1(OC)ccc2c(c1)NC(=O)C2CC(=O)NC1(C)CN(C(=O)C(C)=C2CCC2)C1 CC(C)(C)C(CNC(c1ccc(N)c(F)n1)=O)C(=O)NCCc1ncon1 C1(NC(CSc2cn(C)nc2)=O)C2CCC1N(C(=O)CSc1ccncc1)C2 C1(CCC(N2CC(NC(C3C(CC)C3)=O)C2)=O)CCCN(CC(F)F)C1 N1(C(C(C)SCCCC)=O)CCC(C2CCCC2)(CNC(=O)C(F)COC)CC1 C1(C)(OC)CCC(NC(C2CCN(C(c3cc(F)cc(F)c3)=O)CCO2)=O)CC1 c1(CNC(=O)Cc2cnns2)ccccc1CNC(C1(Cl)CC12CCC2)=O CC(=O)C(C)(C)CC(=O)N(C1(CC(=O)NOCCF)CC1)C C1(CNC(=O)CCn2cc(CO)nn2)CN(C(C2C3CCCC23)=O)CCO1 c1(C(N2C(CNC(C3(OC(C)C)CCC3)=O)CCC2)=O)ccc2nnc(C)n2c1 C1(NC(C2C(C)C2)=O)CCOCC1NC(=O)COc1cncc(Cl)n1 CN1CCOC(C(=O)NC2CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C2(C)C)C1=O Cc1nn(C)c(C(=O)NC2CC3(C2)CC3NC(C2(N(C)C)CCC2)=O)c1Br CCCC(C)(O)CC(=O)NC(Cn1cccn1)C(=O)NC1CN(C)CC1O c1(C(=O)NC(C=C)C)cn2c(C)ccc(-c3ccc(C(N)=O)cc3)c2n1 C1(C(=O)NCCCCNC(C=CC)=O)CCCC(=O)O1 N1(C(c2cccc(OC)n2)=O)C2CCC(C2)C1C(=O)NC1CN(C)CC12CC2 CN1CCCC(CC(=O)NC2(CCNC(=O)C(O)C3CC3)CC2)C1 c1(NC(=O)CC2CCCN2C(C2(COC)CC2)=O)cccc(C2CC2)c1 N1(C(Cc2c(C)cco2)=O)CCOCC1C.C(=O)(C(CCO)C(=O)N)N(C)C1CC1 c1(C(N(C2CC(C(=O)NCCC(=O)NC)C2)C)=O)cc2ccccn2n1 N1(Cc2cc(OCC)ns2)CCCC(C(=O)NCCC2CCCO2)CC1 N1(C(c2n(CC)nc(C)c2)=O)CC2CC(NC(=O)C(=O)Nc3ncc[nH]3)C(C2)C1 c1(OCC)cccc(C)c1C=CC(=O)NC1CC1NC(=O)C(C1CC1)OC O=C(N=c1[nH]c(Br)cnc1Br)C1CC1C1CCCCC1 c1(CC)c(C2CCCN2C(C2(C(=O)OC)C(CO)C2(C)C)=O)ccnc1F CCCC(O)CC(=O)C(=O)C=Cc1cncn1C.C(C)(CN)(C1CC1)N C(=O)(C(F)C(C)(C)O)N(CC(C)CNC(c1cscc1Br)=O)C c1(N(CC(C)C(F)(F)F)C)nc(=NCCc2ccccc2Br)[nH]c2c1CCC2 c1(OC)ccc2c(c1)C(C(=O)NC1CCC(C)N(C(=O)CCOCC)C1)CCC2 c1(C(=O)NCC(C(C)C)NC(C2C(=C)C2)=O)ccc(-c2cnco2)cc1 c1(C(N2CCCCC(NC(CSC)=O)CC2)=O)cn2cccc(C)c2n1 c1(-c2cn(C3(C(C)NC(C4C(C(=O)OC)C4)=O)CC3)nn2)c(F)cc(F)cc1F C1(C(=O)NCC=CCNC(C2C(C3C(C(=O)OC)C3)C2)=O)CCc2cnnn2C1 Cc1c(C(O)C(=O)NC2CC2Cc2ccc(OC(F)F)cc2)cccc1Cl Cc1ccc(CNC(C2CC3CC3N2Cc2cnc(C)nc2)=O)c(C)c1 C1(C(=O)NCC2(NC(CC(C)(F)F)=O)CCCC2)CCn2c(cnc2Br)C1 C12(C(=O)NCC3(F)CN(C(CCCNC=O)=O)C3)CCC(CO)(CC1)CC2 c1(C(=O)NC(C(C)NC(C(CC=C)CC)=O)C)c(C)cnc(OC)c1Cl N1(C(C(C)n2cccc2)=O)CCN(C(=O)CCCCC2CC2)CC1CCN(C)C C1(NC(c2scc(C)c2C)=O)CC(C)CN(C(C2(CO)CCC2)=O)C1 C1(CC(=O)NC)CCN(C)C1=O.c1(C(=O)OC)cn(C2CC2)cn1 CCCC(F)(F)C(=O)NCC1CC(F)(CNC(=O)C(C)CC2CC2)C1 CCCC(C(=O)OC)C(=O)N1CCN(C(c2ccc(Cl)nn2)=O)C(C)C1 N1(C(CCN(CCCCC)C)=O)CCOC(C)(CNC(c2ccc([N+](=O)[O-])s2)=O)C1 Cc1ccc2c(c1)CC(C)N(CC(=O)Cc1cccc(Cl)c1)C2 C1(CC)C(NC(c2cc(C(=O)OC)no2)=O)CCCN1C(=O)COC(C)C N1(C(C2(COC)CC2)=O)CC(NC(C2CC2C#N)=O)C(c2nccn2C)C1 C=CCCCC(C)(C)C(=O)N1CC2CC1C2NC(c1cc(C)ccc1C)=O c1(CCCC(=O)NC2CN(C(C3C(=C)CC3)=O)CC2F)c(F)cccc1F Cc1nc[nH]c1CC(O)C(=O)N1CC(O)(CCNC(C2CC2(C)C)=O)C1 C1(CC(=O)NCC2CC(NC(C3CC4(CC4)C3)=O)C2)Oc2ccccc2NC1=O N1(C(c2ccoc2C(C)C)=O)CCCCC1C1CC1.CC1=CC(=O)NC1 C1(C(N(CCCCN(C)C(c2cc(C#N)c[nH]2)=O)C)=O)CC2C=CC1CC2 c1(C(N2CCC(CCOC)(NC(C3CCC(C)(C)O3)=O)C2)=O)cc(N)cc(O)c1 Cc1ccc(-c2cn(CCONC(=O)CN3CCNC3=O)nn2)c(C)c1 C1(N(C(c2cnccc2C)=O)CC)C2CN(C(n3cc(I)cn3)=O)CC12 c1(C(=O)NCC(CNC(c2ocnc2C2CC2)=O)O)ccc(=O)n2c1COCC2 CC1(C(N2CCOC(CNC(=O)CCCC(F)(F)F)C2)=O)CCS(=O)(=O)CC1 c1(C(=O)NCC2N(C(C(CSC)O)=O)CC2)cnc(C(=O)Nc2ccccc2)cn1 c1(C(=O)NCC(C2CC2)NC(C(C)OC(F)(F)C(F)(F)F)=O)cnc2n1CCS2 N1(CC(C)C)CCCC(NC(=O)CC2CN(C(c3cc(F)n(C)n3)=O)CCO2)C1 N1(c2nc(SC)nc(C(F)F)c2)CC(F)(F)CC1(C)CNC(C1(C(C)C)CC1)=O N1(C(C2N(C(C3OCCC(=O)C3)=O)CC2)=O)CCc2c(F)cccc21 C1(C(N2CC(NC(c3c(C)cno3)=O)C(C)C2)=O)C2CCCCCC12 CC1(C(=O)NC2CCCC(C(=O)N(CC3=NOCC3)C3CC3)C2)CCCC1O C(=O)(CC1=NNC(=O)C1)NC(C(C)NC(=O)C(F)C(C)(C)O)CO Cc1ccc(F)c2c1CCN(C(c1cc(Cl)c3ncccc3c1N)=O)C2 C(C)(CCC(=O)NC1(C2CCCC2)CC1)SC.C12CCN(C1)C(=O)N2 N1(C(c2cc(C)[nH]c2)=O)C2CN(C(c3cc(Cl)sc3Cl)=O)CC12 N1(C(C(F)OC)=O)CCN(C(=O)CC(c2ccc(Cl)cc2)O)C(C)C1 N12CCC(CC1)c1n[nH]cc1C2=O.C=CCC(CC(=O)OC)OC CC(C)C(CC(=O)NCCc1c[n+]([O-])ccc1O)c1ccon1 N1(C(C=CC(C)NC(CC(CC)OC)=O)=O)CC(C)C(F)(F)C1 c1(CC(CO)OC(=O)NC2CC2)ccccc1 C1(C)(C(N(C)CC2CCN(C(=O)CCCF)CC2)=O)CCC(F)(F)C1 c1(C(=O)OC)ccc(NCCNC(=O)C(F)F)cc1.c12cncc(c1)C(=O)N2 CCCCCS(=O)(=O)CC(=O)NC1CCC12CN(C(=O)C(c1cccnc1)O)C2 C1(CCC(=O)NCC(C)(C)C(F)F)CCCN(C(c2cc(CO)[nH]n2)=O)C1 CN1CC(C(N2CCCCC2C(=O)Nc2cnccc2N(C)C)=O)CC1=O N1(C(=O)NC(C=C)COC)CCOC(C)(C)C1CSC C#CCCCC(C)(c1nnnn1Cc1nnn(C)n1)NCC1(CC(N)=O)CC1 CCC(CNC(=O)C(C)=CC(C)(C)C)(CC)C(=O)N1CCC(C)C(C)C1 C1(C(N(CCN(C(=O)CC=C(Cl)Cl)C(C)C)C)=O)CC2(CO1)CC(F)(F)C2 c1(C(N(C(C)C(=O)NCC2CC2(Cl)Cl)CC)=O)n[nH]c2c1CCC2 N(C1CCc2c1ccc(F)c2F)C1CC(CCC)OCC1 Cc1ccc(F)c(CC(=O)NC2CN(C(=O)COc3cccnc3)CC2C)c1 C1(CC=C)(C(=O)N(C)CC2CCOC2)CCN(C(=O)C#CC2CC2)C1 c1(C(=O)OCC)c(NCC(C2CC2)NC(=O)CCF)nnc2c1COCC2 c1(C(=O)Oc2ccc(F)cc2)[nH]nc2c(-c3ccccc3C(F)(F)F)cccc12 c1(C(=O)NC(CCC)CNC(=O)C2=COCCC2)noc2c1CCCC2 c1(C(N2CC(CN(C(COCCOCC)=O)C)OCC2)=O)coc(S(C)(=O)=O)c1 C=Cn1nccc1C(N1CCCC(CN(C)C(c2c[nH]c(=NC)s2)=O)C1)=O N12CC(C(O)C1)NC2=O.C1(C2CCCO2)(C(=O)OCc2ccccc2)CCCC1 N1(C(c2c[nH]c(Br)c2)=O)CC2CC1CCC2NC(C12CCC(CC1)OC2)=O C1(CCc2cn(CC(=O)OC)nn2)CCN(C(C2CCC(C)CC2)=O)CC1 CC(CS(C)(=O)=O)C(=O)N1CCC(N(c2ncc(C(F)(F)F)cc2Cl)C)C1 C1(NC(Cc2cc(OC)no2)=O)CN(C(=O)CCc2c[nH]c(=N)[nH]2)CCC1C C1(C(=O)NCC(CCCC)NC(=O)Cc2cc(Cl)sc2Cl)Cc2ccccc2O1 N1(C(=O)NCCCSc2ccccc2Cl)CCN(c2ccccc2Cl)CC1 c1(C(=O)NC2C(NC(CCCCOC)=O)CCC2)cccc2nsnc12 c1(C(C(N2CCCC(CN(C(=O)Cc3ccoc3)C)C2)=O)=O)cc(F)cc(Cl)c1 N1(C(C#CC(C)(C)C)=O)CC2CC(NC(=O)CC3CCSC3)C(C2)C1 Cc1cc(CNC2CC(NC(=O)Nc3cc(CN(C)C)ccc3F)C2)ccc1F N1(C(c2n(CC)cc(Cl)c2)=O)CC(=O)NC2CN(C(=O)C(O)C3CC3)CCC12 c1(C(=O)NC(CC=C)CNC(C2COC(=O)N2)=O)cc2ncccc2s1 C(C(C)(C(=O)NCc1cn(C2CN(C(n3nc(C)oc3=O)=O)C2)nn1)OC)OC c1(CN(S(c2cccc(CC)c2)(=O)=O)CC)c([N+](=O)[O-])cnc2c(F)c(F)ccc12 C1(CC(COCC)O)CCN(CC(=O)NOCC(F)F)C1=O c1(CC(C(C)C)NC(=O)C(=O)N2CCC2c2ccccc2)ccc(Cl)cc1 C1(N(C(C(C2CCCC2)OC)=O)C)CCN(C(=O)CCn2cccn2)CC12CC2 c1(OC(=N)O)ccc2[nH]c(C)c(C(=O)Nc3cccc(NC(C)=O)c3)c2c1.CO CC(C)C(C(=O)NCC1CN(C(c2cccc(-n3cncn3)c2)=O)C1)n1cnnn1 C1(C(=O)NCC(c2cnn(C)c2)C)CN(C(=O)CN=[N+]=[N-])CCN1C c1(C(=O)NC2CN(C(C=NOC)=O)CC2O)nn(C(C)C)c(=O)c2ccccc12 C(=O)(CCN=C(NCCC1(CO)CC1)NCC1(c2cccs2)CC1)NC c1(C(=O)NC(CC(C)NC(c2nc(CCC)oc2)=O)C)ccc(N)c(Cl)n1 C1(C)(C(=O)NCC(C)N(C(=O)CCc2ncccn2)C)CCCS1 Cc1c(C(N2CC=C(CNC(C3CCN(C)C3)=O)CC2)=O)sc2nnc(S)n12 c1(C(=O)NC(CC=C)CNC(=O)CCc2nccs2)cncc(NCC)c1 n1(CC(C)O)cc(C(=O)N(CC(C)(C)NC(c2cc(CO)on2)=O)C)ccc1=O N1(C(CC2C(=O)NC(=N)S2)=O)CCC2CCC(C1)N2C(C1CC2CCCCN2C1)=O c1(C(=O)NCCC=CC=C)c(CNC(c2cscc2CC)=O)cnn1C C1(CC(=O)N(C(C(C)C)C)C)CC(F)CN1C(C1C(C#N)C1(C)C)=O C1CC12CCC2.c1(C2C(=O)N2)cnn(C)c1.C12(CC1)CC(=O)N2.CN(C)C=O N1(C(c2cc(COC)on2)=O)CCC(NC(=O)COCC(F)(F)F)CC1 N1(C(C(CC#C)(C)CC)=O)CCC2(CC1)CCN(C(=O)C(C)(O)C1CC1)C2 N1(C(CCc2cnc(C)s2)=O)CC2=C(C1)CN(C(C1CC1OC(C)(C)C)=O)C2 c1(C(N2C(C)(C(=O)NCCCc3ccncc3)C=CC2)=O)c[nH]c2cccnc12 c1(C(=O)NC(C(=O)NC(C#C)CC2CCC2)C2CCC2)cnsc1C C1(CNC(COCCC#C)=O)CCC(NC(C2(C(O)C(F)(F)F)CCC2)=O)CC1 CC#CCC(C(=O)NC(c1cccnc1)CO)NC(c1csc(O)n1)=O N1(C(COC(C(C(c2ccccc2)C)O)=O)=O)c2ccccc2CCC1C C1(NC(C=CC)=O)CC12CCN(C(=O)CC1OCCCC1(C)C)CC2 c1(C(=O)NCCN(C(CCSCCC)=O)CC(C)O)cnc2c(c1)N(C)CCO2 c1(C2C(C(=O)NC(CN(C(C=C(C)Cl)=O)C)(C)C)C2)cc(Br)ccc1C c12sccc1S(=O)(=O)N1CC3CN(CC13)C2=O.c1(CC(C)OC)ccccn1 C#CCCCCC(=O)N(C)Cc1ccc(CNC(=O)CC(C)(C)C)cc1 c1(C(=O)NC2CCCCN(C(C3CC(=C)C3)=O)C2)c[nH]c2c(OC)nccc12 C1(C(=O)NCC(=O)NCC(C)(C2CC2)OC)CCCN1C(C)C C=C1CCN(C(=O)CCOCCCNC(c2nc(Cl)cs2)=O)CC1 c1(OC)cc(C(=O)NC(C)CC(C)NC(=O)CC2(C3CC3)CC2)c(N)c(C)c1 C1(C(C)C)CCC(NC(=O)CC2CC(C)N(C(c3cnns3)=O)C2)CC1 C1(NC(C(C)N(C(C)=O)C)=O)OCCOC12CCC2.C1(N2CCNC2=O)CCC1 C1(C(=O)NC2C3CN(C(Cc4c(C)nc(C)s4)=O)CC2C3)CCC2(CCCC2)CC1 c1(NC(c2cn(C3CCCC3CO)nn2)=O)ccc(Br)c(Cl)c1Cl C1(CNC(C2(C)CC2Br)=O)CC2CCC1N2C(=O)CCn1ccnn1 C1(N(C(=O)COC2(C)CCC2)C)CCN(C(c2cnn(C(C)(C)C)c2)=O)C1 N1(C(c2cnn(C)n2)=O)CCCCC2(CCN(C(=O)CCCN3CCCC3)C2)C1 c1(C(=O)NC2CCN(C(C(COC)OC)=O)CC2F)cccc2sncc12 C1(C(N2C(C)(CC)CC2)=O)CN(C(c2cnc(C)c(C)c2)=O)CC12CCC2 CC(C)(C)CCC(=O)NC1(CNC(=O)C(=C2CCCCC2)F)CC2CCC1C2 N1(C(c2c(C)sc(Cl)n2)=O)CCN(C(=O)CN(C)C)C2COCC12 CCC(C)CCCCC(=O)N(C1CN(C(C23CC(CF)(CO2)C3)=O)C1)C Cc1nc2cccnn2c1C(=O)N(C(C)CCNC(=O)CCC(C)(F)F)C C(=O)(C(CC(C)C)C(N)=O)NCCC(C)NC(c1[nH]c2ccc(C)cc2c1)=O O=C1NCCc2c(Br)c(-n3cc(-c4cccc(OC(F)F)c4)nn3)ccc21 N(C1CCCc2ccoc21)N1C(CCSC)CC(C(=O)OC(C)(C)C)CC1.C(=O)O c1(C(=O)NCc2c(C(N3C(COC)C(C)(C)C3)=O)con2)cc(O)cc(=O)o1 n1(C(CC)CC)nc(CCc2ccccc2)nc1-c1cn(C2CCOCC2)nn1 c1(C(=O)NC(C)CCCNC(c2csc(C3CC3)n2)=O)coc2ccccc12 C1(C#N)(C(N2CCC(N(C(c3cn(CCC)nc3)=O)CCC)C2)=O)CCSCC1 C(C(C)C)(C(O)C(=O)NCc1ccc(N)c(Br)n1)OC Cc1sc(C(=O)N(CCNC(C2CC(F)(c3ccccc3)C2)=O)C(C)C)nc1O c1(OC)cccc(CN(C(C2CCCC2Nc2ncccc2O)=O)C2CC2)c1 C(N=c1nc(-c2ccccc2)[nH]c(=NCc2cc[nH]n2)[nH]1)c1cncc(CC)c1 N1(C(c2c(C)cns2)=O)CCCCC(NC(C2CCC(=O)NC2C)=O)C1 N1(C(c2c(CC)oc(C)c2)=O)CCN(C(=O)CCc2cnoc2)C(C2CCC2)C1 C1(C(C(=O)NC(c2n(CC)ccn2)C)C)CCN(C(c2cnc(=N)[nH]c2)=O)CC1 C=CCN(OC)C(=O)c1cccc(CNC(c2cccc(C#N)c2)=O)n1 Cc1cc2[nH]c(C(N3CCCC(CN(C(=O)COCC4CCC4)C)C3)=O)cc2o1 C1(NC(c2cc(C)oc2C)=O)CCC2CCN(C(=O)CC3CCC(=O)N3C)C1C2 c1(C(=O)NC(CC=C)CNC(=O)C=Cc2ccc(C)o2)c(C)cccc1F N1(C(c2nc(CCCC)sc2)=O)CC(NC(=O)CCc2ncc(C)[nH]2)C2(CC2)C1 C=Cc1ccc(C(=O)NCC2(F)CCN(C(c3cc(Cl)c(Cl)s3)=O)CC2)cc1 Cc1ccc(C(=O)Nc2nc(C(N3CCCC(C#N)C3)=O)cs2)c(F)c1 C=C=CC(C)C(=O)NCCC1CCN(C(C2CCC23CCC3)=O)CC1 c1(C(=O)NC2CCN(C(CSCC)=O)CC23CCC3)cc(F)c(F)c(Cl)c1F c1(CNc2ccc(CNC(=O)Cc3ccc(O)cn3)s2)cc(F)ccc1C(F)(F)F C1(CC(=O)NC2COCC2NC(C2(CF)CCC2)=O)CC2CC2C1 N1(C(c2cc(C)n(C)n2)=O)CC(NC(=O)CCCN(C)N=O)C2CCCC12 c1ccc2c(c1)CN(C)CC2.N1(CC)CCN(CCN(C)C)CC1.C12(CC1)C(=O)N2 N1(C(C2(N(C(CC=CCCCCC)=O)C3CC3)CC(O)C2)=O)CC2C(CO)C2C1 C(C(=O)N(C)CC1(CSC)CC1)(C(C)C)NC(=O)COc1ccsc1Cl C1(C(=O)NCC(CN(C(=O)CC(C)C)CC)(C)C)C2CCN(CC2)S1(=O)=O C1(NC(c2n(CC(C)C)ncc2)=O)(CO)CCCN(C(c2csnc2Cl)=O)C1 C1(NC(C(C(CC)C)O)=O)CCC2CCN(C(c3cnc4cc[nH]c4c3)=O)C1C2 N1(C(CC2CC(C)(C)C2)=O)CCOC(CCNC(C2CCC2(C)C)=O)C1 c1(C(=O)OC)cccc(CNC(=O)N(C2(C(C)C)CCC2)C)c1F C1(NC(c2c(NC(C)=O)cccn2)=O)CCC12CN(C(c1ncc(F)cn1)=O)C2 C1(C(=O)NCC2(C3CCC3)CC2)CCCCN(C(C2C3CCC(F)C23)=O)C1 CCCC(C(=O)NC(C1CCN(C(c2csc3nccn23)=O)C1)(C)C)S(N)(=O)=O C(C(CC(C)C)NC(c1scnc1C1CCCC1)=O)NC(C(C)=C1CCCC1)=O c1(OCC(=O)NCC2(NC(=O)C=Cc3cocn3)CCCC2)c(F)cccc1F C(=O)(C(F)(F)C(O)C(C)C)N1CCC(NC(CC(C)C)=O)C(C(N)=O)C1 C1(C(N(C(CC(=O)OC)C)C)=O)CCC(CNC(=O)C(C)C2CCCO2)CC1 c1(N(CC(C)NC(=O)CC2CCCOCC2)C(=O)C2CC2)nn(C)cc1S(N)(=O)=O c1(OC)ccc(C(C)NC(=O)C(=O)NCc2cscc2SC)cn1 C1(CC=C)(C(=O)NC(C)CC(C)NC(C2CC3(CCC3)C2)=O)CCOCC1 c1(C(N(CCCN(C)C(C2CCCC(F)C2)=O)C)=O)ccccc1OC1CC1 N1(C(C=COCC)=O)CC2CC(NC(c3c(C)cc(Br)cc3C)=O)CC1C2 N1(C(C(C)SC(F)(F)F)=O)CC2CCC2(NC(=O)C(c2ccc(N)cc2)C)C1 CCCC(C)(CC)C(=O)N1CCC(CC(N2CCCC(C)(CC)C2)=O)C1 c1(OC)ccc(C(O)C(=O)N(CCCCCNC(c2ccoc2)=O)C)cc1 C(=O)(C(C)C(O)CC(C)C)N(C(C1=C(C)CCC1)=O)C1CCN1CN1CC2CC2C1 C1(C)(C(=O)NCCC(C)CCNC(C2C3CC4C(C3=O)C24)=O)CCC(F)(F)CC1 c1(C(N(CCC(C)NC(c2cn(CC3CC3)nn2)=O)C)=O)nccn2nccc12 c1(OC)cc(C(=O)NCC2(O)CN(C(=O)Cn3ccc(O)nc3=O)C2)cc(F)c1 C1(OC)CN(C(=O)CN2CCOCC2)C(C)(CNC(c2ccc(CO)nc2)=O)C1 Cc1c(SC2CCCN(C(C34CC(n5cc(C6CC6)nn5)C3C4)=O)C2)cccc1F c1(CC)cc2c(NC3CC4OCCCC34)nc(C)nc2s1 c1(NC(C2(C)CN(Cc3ncccc3Cl)C2)C)cccnc1-c1ccccc1 Cc1ccc(C#N)cc1C(=O)NC(C)(C(=O)NC1CC(=O)N(C)C1)C1CCC1 C12(NC(CCCCN(C)C)=O)CCCN(C(c3cc(Cl)nnc3O)=O)CC1C2 C(=O)(C1Cc2ccc(C)cc21)N(C)CC1CCN(C(c2c(CC)cco2)=O)CC1 C(=O)(CC(C)(C)COC)NCC1(C(N2CCC(C(C)OCC)C2)=O)CC1 CC1CCC(C)(C(=O)NCC2CN(C(=O)C(C)(C)C3CCCC3)CC2O)CC1 c1(C(C(=O)NCC(CNC(C=CCCC=C(C)C)=O)C)C)cccc(Br)c1 C1(C(N2C(C)C(NC(=O)CC(=O)NC3CC3)CC2)=O)CCc2ccccc2C1 S(=O)(=O)(c1ccc(Cl)c(C(F)(F)F)c1)N(C1CC1F)C(c1cnc(CCCC)[nH]1)=O c1(NC(C(C2CC2)OCC)=O)ccccc1Cn1cc(CCS(C)(=O)=O)nn1 C#CCC(CC(F)F)C(=O)NCC1(C(=O)NCc2cc[nH]c(=N)c2)CCOCC1 N1(C(c2n[nH]cc2F)=O)C2CCCC1CN(C(C1CCC1C1CC(F)(F)C1)=O)C2 C1(C(=O)OC)CCC(NC(=O)N(CCCN=[N+]=[N-])CC2(O)CCCCC2)C(C)C1 c1(C(=O)NC(C2CCCCC2)CNC(CCC(=C)Cl)=O)cc2cccnc2cn1 C1(S(N)(=O)=O)(C(=O)NCCCOCCCNC(c2c(C)cn(C)c2)=O)CCC1 C#CCCCCCCC(=O)N1CCCC(C)(C)C1C(=O)NC(C)(CC1CC1)C1CC1 C#CCC(CC(F)F)NC(c1cnn(CCNC(=O)C(C)(C)C=C)c1)=O c1(CC)cccc(C(=O)NC2CC(C(N3CCC(C)(C(N)=O)C3)=O)C2)n1 Cc1ncc2cc(C(N3CC4CC3CN4C(C3CC=CCC3)=O)=O)c(O)nc2n1 c1(C(C(N2CC(O)(CCNC(C3C=CCCC3)=O)C2)=O)OC)ccccc1Cl N1(C(C(CC)n2ccnc2)=O)CCCC(C(=O)Nc2cnc(OC)nc2)(CC)C1 c1(C(=O)NCCc2cnc(NC(C3(C#N)CCC3)=O)s2)cc(Cl)cc(Cl)c1 CCC(CC(F)(F)F)C(=O)N(CC(C)NC(=O)C=Cc1cc(OC)ns1)C C(=O)(C1=CC(c2ccccc2)NC(=O)N1)NC(C)(CNC(c1cnn[nH]1)=O)CO CC1CN(C)CC(C(N2CC(F)(CNC(=O)Cc3ccnc(Cl)c3F)C2)=O)O1 C1(C(N(CCCNC(=O)C(C#N)C2CC2)C)=O)CCCCN1S(=O)(=O)CC N1(C(COC2CCN(C(C3CC=C(C)CC3)=O)C2)=O)CCc2ccc(Cl)cc2C1 c1(C(C(=O)NCC(C)N(C(C(c2c(C)noc2C)CC)=O)C)C)ccccc1F C(=O)(C#CC(C)(C)CNC(c1ccc(C#N)s1)=O)NC(C1CCOC1)C#C C1(O)(CCNC(C2ON=C(C)C2)=O)CCN(C(=O)CC(C)C2CCCCC2)CC1 c1(C(N(CCCOCCNC(C=C(C)C(F)F)=O)C)=O)ccc2oc(=N)[nH]c2c1 C1(C(=O)NC(CNC(=O)CCC2CCCC2)C2CC2)CCN(CCF)CC1 C1(NC(C(C)C2CC2)=O)CC2CCC1CC2NC(=O)C=Cc1ccco1 CC1(C)CN(C(C2C=CC(NC(C3CCNC3=O)=O)C2)=O)CCC1CO C(=O)(CC(C)(C)N(C)C(C1(C#N)CC1C)=O)N(CCCOC(C)C)C c1(C(N2CC(N3CCN(C(C(C)SC)=O)CC3)C2)=O)cc2n(n1)CC1(CC1)C2 CC1CCN(C(C2CC=CCC2)=O)CC1CNC(c1cc(Br)cs1)=O c12ccc(o1)CNC2=O.C(=O)(CC1(N(C)C)CC1)N(CC)CC1CCC1 Cc1cnc(N(CCNC(=O)Cc2cn(C)nn2)C2CC2)nc1O C1(CNC(C)=O)CN(C(c2ccnc3c2CCO3)=O)CCC12CCC2 N1(C(CN(CCOC)C)=O)CCC2C(C(=O)NC(c3ncccc3C)C)C2C1 C1(Sc2cccc(C(=O)NC(CC#CC)C)c2)CC(O)CN1C(=O)C1CC1 N1(C(c2ccc(F)s2)=O)CC2CC(C(N3CCOC(C4CCC4)C3)=O)(C2)C1 N1(C(c2c(CC(=O)OC)scc2)=O)CCCC(N(C(=O)Cc2ccns2)C)C1 O=C(C#CC1CCC1)NCC1CC1NC(c1ccc(-c2cccs2)s1)=O CC1CCCN(C(=O)C(=O)NCC2CC3CC3N2C(=O)CCN2CCCC2)C1 c1(OC)cc(C(=O)NCC(C)NC(=O)CCC(C)O)ccn1 CC1CCC(O)(C(=O)NCC(C)(C2CCC2)NC(C2CC2F)=O)CC1 n1(CC(=O)OCc2nccs2)nc2n(c1=O)CCSC2 c1(C(=O)NCCCCC2CN(C(C(C=C)(C)O)=O)C2)cc(S(=O)(=O)NC)oc1C Cc1ccc(O)c(C(=O)NC2CC(CNC(=O)CSc3c(C)n[nH]c3C)C2)c1 N1(C(C2C(C(=O)OC)C2)=O)CCC(F)(F)C(NCc2ccc(SC)s2)C1 c1(CN2CCCN(C(c3cn(C(C)C)nn3)=O)CC2)ccc2ccccc2c1Br c1(C(N(CC(C)CNC(=O)CCOc2ccccc2Cl)C)=O)cc(O)nc(O)n1 n1(CC(C)C)ccc(CC(N2CCCC2c2cn(C3CCCC3O)nn2)=O)n1 CC1CC(C2CN(C(=O)CCC3CN(C(C4CS(=O)C4)=O)C3)C2)=NO1 c1(CCC)cc(C(N2CCC(C)(NC(c3ccn(CC(C)C)n3)=O)C2)=O)c(C)o1 c1(C(N2CC(CNC(C(C(C)C)SC)=O)C2)=O)cccc2[nH]ncc12 C12(NC(c3cccc(O)c3)=O)CCCC1N(C(=O)Cc1cnc(C(F)(F)F)s1)CC2 C(=O)(CCCCCCn1cc(CCCCO)nn1)NCN1C(C)CCCCC1 CCC(COC)(CC)C(=O)NCCC1(O)CN(C(=O)C(C2CCCO2)C2CC2)C1 C1(C(=O)NCCCC2COCCO2)(CC)CN(C(=O)CN(C(=O)C(C)C)C)C1 Cc1cccc(F)c1CC(=O)N(CC(C)NC(c1cc(C#N)cn1C)=O)C CN1CCCC(C)(C(=O)NCC2CC2CC(=O)NCC23CCCN2CCC3)C1 c1(OC)ncc(C)cc1NC(C1CCN(C(=O)C(n2ccnc2C)C)C1C)=O C1(CNC(C(C)SCC)=O)CC2(CCN(C(C3CCN(C(=O)OC)CC3)=O)C2)CO1 C#CCCCCCCCC(=O)NC(CO)C(=O)NC(C=C)CO C1(N(C(CC(C)O)=O)C)C2CN(C(c3ccc(C4(C(F)(F)F)CC4)cc3)=O)CC12 N(C)(C(=NCCC(C)=O)NCC12CCCC1C2(F)F)Cc1ccc(OC)cc1C#N C1(C(=O)NCCNc2cc(Br)ncc2F)(OC)CCN(C(c2ccco2)=O)CC1 C(CC(C)C)(C(=O)NC1(CO)CCN(C(C2(C)CCN(C)CC2)=O)C1)OC CC1(C)OCCC1Cn1cc(CC(N2CCCC2n2nccc2)=O)nn1.C(=O)O C(=O)(CCCC(C)(C)NC(=O)CN(C)C)NC1CCCC(C)C1 C(=O)(C1CCc2ccccc21)NC1CCC(C(N)=O)C1.c12ccoc1COC2=O Cc1ccn2ncc(C(N3CCCC3N(CC(C)C)C)=O)c2n1 C1(C(N2C(C(C)NC(C3(CC#C)CCCCC3)=O)CCC2)=O)=CC2=NC=CS2=N1 Cc1cc(C(=O)NC2CCCCO2)n2ncc(Br)c2n1 C1(CN(C(C=CCCC(C)C)=O)C)CN(C(c2ccccc2C#N)=O)CC12CC2 N1(C(C(CC)N(CC)CC)=O)CCC2(CC1)CN(C(c1ccc(Cl)nc1)=O)C2 C(C(C)(C)CCNC(C1(NC(C2CCCCS2)=O)CCCCC1)=O)OC c1(C(=O)NC2C3CCN(C(c4ccc(-c5cccs5)s4)=O)C23)ccc(O)c(F)c1 c1(NC(CC(C(C)(C)C)=O)C(N)=O)cccc2c1C(=O)N(c1ccc(F)cc1)C2=O C(CNC(=O)CCn1cnnn1)(CCNC(C1(CC(C)C)CC1)=O)OC S(=O)(=O)(c1c[nH]c(C(=O)N(CC(C)NC(C2CCCN2C)=O)C)c1)NCC(C)C C(CCC(C)C(=O)NC1(CCCNC(c2sccc2Cl)=O)CCCC1)OC C=C1c2ccccc2C(=O)N1CCC(N1CCCC1CNC(C1OCCO1)=O)=O n1(CC)ccnc1C1OCCC1NC(=O)C(=O)NC(C1CCCOC1)(C)C N1(C(c2ccc(C)cn2)=O)CC(C)(C)CC1C(=O)NCC1CCC1C(=O)OC c1(C(=O)NCCOCCNC(=O)C(=O)NCCO)ccc2c(c1)COC2 N1(CCC(=O)NC(C(C)NC(=O)C=CC(=O)NCC(F)(F)F)C)CCC(O)CC1 Cc1ccc(O)c(C(=O)N(C(CC(C)C)C(=O)NC(C)Cn2ccnc2)C)c1 C1(CNC(C(=O)NC(C)C)=O)(CNC(C23CC(F)(C2)C3)=O)CCCC1 C1(NC(C(Br)=C(C)C)=O)C2CC1N(C(c1ccc(C)c(OC(F)F)c1)=O)C2C C1(CC(=O)NC(CC)CNC(=O)C(O)CSC)COCCOC1 N1(C(CCC(C)C)=O)CC(NC(=O)CC2CCCCC23CC3)CC12CCC2 c1(SC)ccsc1C(=O)NCC(C1CCOC1)NC(=O)C(C)OC(C)=O c1(C(N2C(CNC(c3c(C)n[nH]c3)=O)C=CC2)=O)ccc(O)nc1 c1(OC)ccc(SCC(=O)NC(C)CNC(c2ccc(CO)nc2)=O)cc1 N1(C(=O)OC(C)(C)C)CC(C(=O)O)CC12CCCCC2.c12cnc(nc1)NC2 C(C)(c1cccc(Cl)c1)=CC(=O)NCCCC(CCC)NC(=O)CCCCC(N)=O C1(CNC(c2cc(C)sc2)=O)CN(C(c2cc3n(n2)CC(F)C3)=O)CCC1(F)F CC(C)C(C)(N)C(=O)N1CCOC(C(=O)NCc2cnn(C)c2)C1 N1(C(c2c(C)nc(C)s2)=O)CCOC2(C1)CN(Cc1ncccc1C(F)(F)F)C2 c1(C(N2C(CNc3scc(C)n3)CCC2)=O)cc(C(F)(F)F)cc(N)c1 C(=O)(C1CCc2ccccc21)N1CC2(OCC(NC(c3cc(C)nn3C)=O)C2)C1 N1(C(c2n(CC)nnc2)=O)CCCN(C(=O)C(C)OCCN(C)C)CC1 CCC(C)(O)C(=O)N1CCN(C2CCCC2NC(C2(c3cc[nH]n3)CCC2)=O)CC1 N1(C(C(C)(C)OC)=O)CCC(NC(=O)CC2(C#N)CCC2)C(CO)C1 C(=O)(C(C(C)O)NC=O)N(CC(CC)NC(=O)CNS(C)(=O)=O)CC1CC1 C=C(C)CC(C)C(=O)NC1CCC(F)(CNC(=O)CCCCc2ccccc2)C1 C(CC(C)C)(C(=O)NC1(C)CCCCC1NC(=O)CC(=O)OCCC(C)C)OC C12(NC(CC3N(C)CCOC3)=O)CCC(F)(F)CC1CN(C(=O)C=CC1CC1)C2 C(=O)(C(O)P(C)(C)=O)N1CC(COC)(NC(C2CCN(C)CC2)=O)C1 C1(C(N(CC(CC)NC(=O)CC2(O)CC2)C)=O)CCCN(C(=O)NC2CC2)C1 C1(C(=O)NCCOC)CCN(N2CCCC(Cc3ncccn3)C2)CCC1 O=C1CCN(Cc2ccc(Br)cc2F)C(=O)N1CC1CC(n2cncn2)C1 N(C1CCOc2cc(F)ccc21)C(n1cc(CCN2CCC(=O)NC2=O)nn1)=O c1(CC)ccccc1-n1nnnc1C(COC)NCC(C)OC(C)(C)C Cc1nc(-c2cccc(F)c2)sc1OCc1ccc(C(N)=O)cc1 C=CCCCCC(=O)N1CC(F)(F)CC1C(=O)NC(C)CCOC(C)=O C1(NC(C2CC3CC2C3)=O)CCCCN(C(C2CCNC2=O)=O)C1 C1(F)(CN(C(=O)CNC(c2ccoc2)=O)C)CCN(C(=O)C(O)C2CCCC2)C1 c1(C(=O)NCc2cc(Br)c(Br)o2)cncc(OCC(F)(F)F)n1 N1(C(c2cc(OC)no2)=O)CCC(N(C(=O)COCC2CC2)C)C(C)C1 N1(C(c2cccc(C(C)=O)c2)=O)CC2(CCCN(C(C3(O)CCCC3)=O)C2)C1 c1(OCC)nc(C(=O)NC(CNC(=O)CN2CC3CC3C2)C(C)C)ns1 C(CCCCCC(=O)NC12CCCCC1C2)NC(Cc1nc(C)oc1)=O C1(C(NOC(C=C)C)=O)CCN(C(=O)Cc2cc[nH]c2)C1C(C)(C)C CC(=O)CCN=C(NCCCC(F)F)NC1CCCCC1.c1(C)ccccc1C(F)(F)F c1(OCC)c(C(N2CCCOC(CNC(c3cnc(F)s3)=O)C2)=O)cccc1N C1(NC(CCC(C)NC(C(N2CC(C)C2)C)=O)=O)CC(C)(C)C(C)C1.c1cccs1 c1(CS(=O)(=O)Nc2c(C)nn(CC#C)c2C)c[nH]c2cccc(Br)c12 c1(C(=O)NC2CC(C(C(=O)N(CCN(C(C)=O)C)C)F)C2)cc(N)cc(F)c1 CN1CCN(C(C(=O)OC(CNC(=O)OC(C)(C)C)=O)C2COC2)CC1(C)C C=Cc1ccc(C(N2CC(O)C(O)C2CNC(c2scnc2C2CC2)=O)=O)cc1 c1(CC)c[nH]nc1C(=O)NCCCN(CCCNC(c1cc(C(C)C)no1)=O)C c1(C(C(=O)N(CCOC)CCNC(=O)C(C)CSC)(F)F)ncccc1F C1(NC(CCOCC#C)=O)CN(C(C2CC(C)(C)CO2)=O)CC1c1cncn1C N1(C(C2C(OC)C2)=O)CC(NC(=O)Nc2cnoc2)CC1(C)C n1(CC)nc(NC(c2nnnn2C2CC2)C2CN(CC3CC3)C2)c(C)n1.CC C1(=CC(=O)N(C(C)CNC(=O)Cc2ccc(Cl)cn2)C)C2CC3CC(C2)CC1C3 C1(CNC(c2nc(CCCC)sc2)=O)COCCN(C(C2CC2c2cnc[nH]2)=O)C1 C1(C(NOCCCOC)=O)CCC(O)CN1C(C1(C)CC1)=O C1(NC(c2nc(C)sc2)=O)CC2CCC1CN(C(=O)CNc1cccc(Cl)c1)C2 c1(NC(c2c(NCC#N)cccc2)=O)nn2ccnc2s1 c1(CN(C(c2cocn2)C(=O)NCCC#N)CC)cc(OC)ccc1OC c1(CC)ccc(C)c(C(=O)NCCC2(O)CN(C(=O)CC3CC(F)C3)C2)c1 C1(CN(C(C2CCCS2)=O)CC)CCCN(C(=O)Cc2ccc(O)cc2)C1 C1(NC(C=CCC)=O)CCCN(C(=O)Cc2cncn2C2CC2)C1 c1(C(N2CC3CC(NC(C(C(C)C)O)=O)C3C2)=O)cnn2c1CC(C)CC2 Cc1cc(C(F)F)n(CC(=O)NCC2CCCCN2C(c2cnc[nH]c2=N)=O)n1 c1(CC(=O)N(CCN(C(C2CCCC(OC)C2)=O)C(C)C)C)c(Cl)cccc1Cl c1(C(=O)NCC(CC=C)NC(=O)C(C(C)C)NC(N)=O)ccc2oc(C)nc2c1 N1(C(c2cn(C(C)C)nn2)=O)CCCC12CCCN(C(c1cn(C)cn1)=O)C2 c1(OC)ccc(-c2cn(CCNC(C3CC4(CCOC4)C3)=O)nn2)cc1Cl CCCC(CC)CC(=O)NCC12CN(C(=O)COCCCC(C)C)CC(F)(C1)C2 c1(C(=O)NC2C(CNC(c3nc(CC)oc3)=O)CC2)ccc(O)c(C)c1C CCCCCCC(C)C(=O)N1CC(NC(=O)CCC(N)=O)C(CCC)C1 CC1CN(C(=O)Cc2ccc(O)nc2)CC1NC(c1ccccc1CC#N)=O C(=O)(CC(C)(O)COC)N1CC(CC=C)(NC(=O)C(n2cc(COC)nn2)C)C1 Cn1cc(C(=O)NC2CC3CC2N(C(C2CC24CC4)=O)C3)c2ccccc2c1=O C1(C(N(C)CCNC(=O)CC2C=CCCC2)=O)CCCC1S(C)(=O)=O CON(CCC(=O)N1CC=CC1COC)C(=O)C(C(=O)OC)N(C)C C1(c2ccn(C(C)(C)C)n2)COC2(CCC2)C1 C(=O)(C1=Cc2ccccc2OC1)NCCC1(C)CCN(C(c2cc(F)n[nH]2)=O)C1 C1(C(=O)NCC2CCN2C(C2CS(=O)(=O)CC(=O)N2)=O)C2CC3CC(C2)CC1C3 C1(NC(C2N(C(CC(CC)C3CCC3)=O)C(C)CC2)=O)CC2(C1)CC(O)C2 C12CCN(C(=O)O1)O2.c1(C(N(C(C)C(=O)OC(C)(C)C)C)=O)ccc(Cl)cc1 C1(C(=O)OC)CCCC1C(=O)NCC(O)CN(C)C(C1CC2(CC2)C1)=O c1(CN2CC(OC)C(NC34CCCC3C4)C2)c(F)cc(Cl)cc1Br c1(C(N(C2CCN(C(=O)Cn3nc(Cl)ccc3=O)C2)C)=O)cc2ccncc2o1 N1(C(C(C=C)C)=O)CCOC(C)(CNC(=O)C(C)=CC(C)(C)C)C1 S(=O)(=O)(c1ccc(NCCCOc2ncccn2)c(Cl)c1)NCC(C(C)O)C Cn1nc(C(N2CCC(CCNC(c3ccc[nH]3)=O)C2)=O)c(Cl)c1C(F)(F)F C12(C(N(CCN(C(c3c(CC)oc(C)c3)=O)C)C)=O)CCCN1CC(O)C2 N1(C(C(c2cccc(O)c2)(C)C)=O)CC2(CC(NC(C3CC3C(F)F)=O)CO2)C1 C1(CC(=O)N(C2CCCN(C(=O)C=CC(C)(C)C)C2)CC)CCCNC(=O)C1 C(=O)(CCC(C)NC(=O)C(c1cccnc1)O)NCC1CC(C=C)C1 N1(C(c2cc(C)nc(C)c2)=O)CC2ON=C(CNC(C34CC(C)(CO3)C4)=O)C2C1 Cc1ccc(C)c(CN(C(C)(C)C)C(c2ccc(Cl)cn2)=O)c1 C1(NC(c2c(C)nc(O)nc2C)=O)CCCC2CN(C(=O)C#CC3(C)CC3)CC12 C1(C(=O)NC2C(CC=C)COC2)(CNC(=O)C(C)O)CCCCC1 n1(C(C)(C)C)cc(C2CC2NC(=O)CNC2CC(=NC(c3cc[nH]c3)=O)C2)cn1 N1(C(C=C(C)Cl)=O)CC2CCC1CC(NC(C1(c3cc(C)sc3C)CC1)=O)C2 C1(NC(c2cc(OC)n[nH]2)=O)CC(C)CN(C(C2(CCO)CC2)=O)C1 CC1CC(C(=O)NC2CCC2NC(c2cc(Cl)ccc2F)=O)CC(=O)N1 N1(C(CN(CC#C)C(C23CSCC2C3)=O)=O)CCC(N(C)C)CC1 CC1(C)CC(C(=O)NCc2sccc2Cl)CN1C(c1ccc(CF)cc1)=O N1(C(c2c(=O)cc(C)[nH]c2)=O)CC=C(CC(=O)NC2CC(=O)N(O)C2)CC1 N1(C(CCCCOC)=O)CCC(CF)(NC(=O)CCCc2cnn[nH]2)C1.CO N1(C(C2=NNC(=O)C2)=O)CC2CC3CC2C1C3NC(c1cc(C(F)F)cs1)=O c1(NCC)ccc(C(=O)NCC(N)C(C)C)cn1 c1(C(=O)NC(C(=O)NCCC(=O)OC)C2CCOC2)ccc(OC)c(OC)c1C N(C(=NCCCCl)NCC1CCOC1)CCOc1c(Cl)ccc(C)c1 c1(CC)cc(C(=O)N(CC(C)(C)CNC(c2ccoc2C(F)(F)F)=O)C)c(C)o1 C(=O)(C1=CC2CC(C1)CC2O)N1C(CN(C(CCNC(N)=O)=O)C2CC2)CCCC1 C(=O)(C1CCCc2nncn21)NCCC1OCCN(C(C=CC(CC)=CC)=O)C1 N1(C(C(CCC)F)=O)CC(C(N2CCOC(C(C)C)CC2)=O)CCC1(C)C c1(N2CC(C)OC(C)(C(F)F)C2)nc(C(F)(F)F)nc2ncnn12 CCCC(C)(C)CC(=O)NC1CN(C(C2CCC(C)O2)=O)CC1n1ccnn1 N1(C(CCc2nnc(C(C)C)o2)=O)CC2CN(c3nccnc3C#N)CC2C1 C(=O)(CCCCC(=O)NC1CCCCC1NC(=O)C(C)C(O)C(C)C)NC Cc1c[nH]cc(Br)c1=NC(=O)OCCN(C)CCO.C(C(F)F)O N1(C(C2(C(C)C)COC2)=O)C2CCC1CN(C(=O)C(C1CC1)C1CC1)CC2 C#Cc1cc(C(=O)NC2(CC(=O)NCC3(Cl)CCC3)CC2)cc(F)c1 N1(C(CC#N)=O)CCN(C(c2ccc(OC(F)(F)F)cc2)=O)C(CO)C1 C=C(C)CC(=O)NCC1CN(C(=O)C(N2CCOCC2)C2CC2)C1 Cc1cc(NC(c2cc(C(F)(F)F)cc(-c3cnn(C)c3)c2)=O)n2ncnc2n1 C(=O)(C(C)CCCOC)Nc1cccc(CC=CC(C)NC(C=CCOC)=O)c1 Cc1cc(C)c(N2CCC(C(=O)NCC(C)(O)c3cccs3)C2=O)c(C)c1 c1(-n2ncc(NC3C(C)COC3)c2)ccc(Cl)cc1 Cn1nnc2cc(C(=O)NCC34CC(n5cc([N+](=O)[O-])cn5)(C3)C4)sc12 CC1(C)CCN(C(=O)CC(C2CC2)C2CC2)C1CC(=O)NCC1CC2(CCC2O)C1 N1(CCCn2cc(CC=C)nn2)CC(C)Cn2nc(C)cc21 Cc1cccc(=O)n1CC(C)(O)C(=O)NCCNC(=O)C(=O)C(C)C c1(C(N(CCC)CCNC(c2cnc(C3CC3)s2)=O)=O)nnn2c1CSCC2 Cn1nc(C(=O)NCc2ncc[nH]2)c2ccc(-c3ccccn3)cc12 CC(CNC(=O)CN1C(=O)CCCC1=O)C(=O)NOCc1ccc(F)cc1 CCC(C)(C)C(C)CC(=O)NCC(C1CC1)NC(=O)CCc1ccccc1 C(=O)(C(CCN(C)C)NC(=O)COc1cnn(C)c1)NCC1(CC)CC1 Cc1ccc(-c2nc(C(N3CCC(c4cn(C(C)C(=O)O)nn4)C3)=O)cs2)nc1 C1(C(=O)NCC(C)Cc2cn[nH]c2)CN(C(c2ncc(F)cc2F)=O)CC1(C)C C1(N(C(C(C)=C(CC)C)=O)C)CCN(C(c2cnn(CCC)c2Cl)=O)CC12CC2 N1(C(c2cc(CC)c(C)s2)=O)CCCN(C(c2cnc(=N)[nH]c2)=O)C(C)C1 c1(C(N2C(CCNC(CN(CCC)C)=O)CC(OC)C2)=O)ccc(F)cc1OC c1(CNC(c2c(F)cncc2Br)c2n(C(C)C)nnn2)ccc(F)c(Cl)c1 Cc1cccc2cc(C(N3CCC(NC(=O)C(F)(F)C4CC4)CC3)=O)sc12 c1(CC(C)CNC(c2ccccc2)c2nc(-c3ccccc3)no2)ccccc1I C1(c2ccc(F)cc2)(NC(C=C(C)C)=O)CCN(C(=O)CCOCC(F)F)C1 c1(C(=O)NCCCN(C(C2OCC2(C)C)=O)CC)sc2ccc(F)cc2c1C C1(CNC(C(CC)C)=O)CN(C(c2ccnc(C(N3CCCC3)=O)n2)=O)CC1O n1(CCC)cc(C(=O)NC2(C)CC(NC(=O)CNC(=O)OC(C)(C)C)C2)cn1 CC1(C)NC(=O)CC1C(N1CC(NC(=O)Cc2sc(O)nc2O)C2(CC2)C1)=O CC(C)(CC(F)(F)F)C(=O)N1CCN(C(=O)CCOCc2ccoc2)C(C2CC2)C1 c1(C(N(C(C)C(=O)NCC(C)(O)C(F)F)CC)=O)cccc(C)c1N c1(C(N(CCNC(=O)C(C)Cc2ccco2)CC)=O)c(Br)c(C)nn1C Cc1c(N)cc(C(N2CCn3ncc(CNC(=O)C(C)N(C)C)c3C2)=O)cc1N C1(C)(CNC(CSC)=O)CCCN(C(=O)C=CC(=O)NCc2ccncc2)C1 C#Cc1ccc(OC)c(C(=O)NC2CC2CNC(c2ccc(CC)c(Cl)c2)=O)c1 C(=O)(CC(C)C(C)(C)NC(=O)C(O)CC1CCCC1)Nc1cccc(C(C)C)c1 CCC(CC(=O)NC1CCC(NC(C2CC3CC(=O)C2O3)=O)C1)C(C)(C)C c1(C(N(C2CCC(NC(=O)C=Cc3cccnc3)CC2)C)=O)cc(Cl)nnc1O Cc1nn(C)c(C)c1CC(=O)N(C1CN(C(N)=O)C1)CC(C)(C)C c1(C(=O)NC2(CNC(c3cccc(F)c3O)=O)CCC2)ccn2ncc(Br)c2n1 N1(C(=O)CC2CCN(C(C3CCCCCN3)=O)CC2)CCC(F)C(F)C1 c1(OC)c(CN2CCOC(C(N3CCCC3C(F)(F)F)=O)C2)cccc1F N1(C(c2c(CC)nco2)=O)CCC(CO)(NC(=O)C=CBr)C1 c1(C(N2C(C)C(CNC(=O)CCF)CCC2)=O)nc[nH]c2ncnc1-2 c1(C(=O)OC(C)(C)C)c(NC(N2CCN(CC)C(C(C)C)C2)=O)ccc(Cl)c1Cl N1(C(CC2CC(=C)C2)=O)CCCC(CCC(N2CC(O)C(O)C2)=O)C1 CCC(CC)(CC)C(=O)N1CC(C(=O)NCC2CCCSC2)C2(CCC2)C1 C1(CNC(c2ccc(C(N)=O)s2)=O)C2CN(CCC3(CC)CC3)CC12 C(CC(=O)NC1CCC1NC(c1cccs1)=O)N(C)CCO c1(C(=O)NCCCNC(c2ccc(OC)nn2)=O)cc(O)c(F)cc1N CC1CCCN1C(=O)C(CNC(=O)CCN(C)CCO)N(C)C c1(OC)ccc(Br)c(C(=O)NC2C3CC2N(C(C2CC(C)C2)=O)C3)c1 Cc1cc(C(=O)NCC2CCC2C(=O)NCCc2ccon2)c(C)s1 c1(C(N2CC(CC=C)(NC(=O)C(O)Cc3cn[nH]c3)C2)=O)cnnc(O)c1 N1(C(C(C)NC(C)=O)=O)CC2CC(NC(C3CC34CC4)=O)C1C2 C1(C)(CNC(c2n(CC)ccn2)=O)CCC(NC(=O)CCCC2CC2)C1 Cn1c(C(N2CCC(CCNC(=O)C=CC=C(Cl)Cl)C2)=O)cc2sccc12 c1(C(=O)NCC(CC)NC(c2cccc(F)c2C(C)C)=O)ccc(F)c(F)c1F C1(C(N2CCCC2)=O)CCCN(C(CN(CCCCCC)C2CCCCO2)=O)C1 C1(NC(C2(C)C(C)C2)=O)CCCCC1NC(=O)CCCc1ccc(Cl)cc1 C(=O)(N=S(C)(=O)c1ccc(C#N)c(F)c1)c1c(C)nn2c(C)cccc21 C1(C(N(CCCCCC)C)=O)COCCC1NC(C1(C)CC1(F)F)=O NS(=O)(=O)CC(=O)N1CC(NC(=O)Cc2cccnc2)C2CC12 Cn1cc(N)c(C(=O)NCCNC(=O)CCc2ccc(OC(F)F)cc2)n1 C1(N(C(CCN(c2ccccc2)C)=O)C)CCN(C(C2CC3(CNC3)C2)=O)CC1 C1(CNC(CSCC=C)=O)CN(C(=O)C(F)(F)c2ccc(C(F)(F)F)s2)CC1C C(=O)(C(CC(C)C)CC(C)C)NCC(C1CCCC1)NC(c1n[nH]c(C)c1C)=O c1(OC)ccc(C(c2nnnn2C2(C)CC2)NC2CC23CCCCC3)c(Br)c1O N1(C(C(C2CC2)OCC)=O)CCCN(C(=O)CCCc2cc[nH]n2)CC1 Cc1nc(C)c(C(=O)NC(C)C(C)C(=O)NCC2CCC2(F)F)o1 Cc1c(F)cc(CN2CCCCC2CNC(=O)Cn2nccn2)cc1F C1(Cn2cc(CNC(C(CC)NC(C)=O)=O)nn2)CCCOCC1 N1(C(CSCCCC)=O)CC(CNC(=O)Cc2cc(F)ccc2Cl)C(C)(C)C1 CCC(COC)C(=O)NC(C(C1CCCCC1)NC(c1cnn(C)c1)=O)C(C)C c1(C2(C(=O)NC3C(NC(=O)C(F)=CCCF)C3)CC2)ccc(Br)cn1 C12(CNC(=O)CCn3cncn3)CC(NC(c3ncccn3)=O)(CCO1)C2 CC1CCCN(C(c2nnsc2C2CC2)=O)C1CNC(c1cc2ccsc2[nH]1)=O S(=O)(=O)(CCC(=O)NCC1CC2CN(C(=O)C(F)C(C)(C)O)CC12)NC N1(C(C23CC(C(=O)OC)(C2)C3)=O)CCC(NC(=O)CCCCC#N)C(F)C1 C=CC(C)C(=O)NC(CC1CCCO1)C(=O)N(C)Cc1cc(C)no1 N1(C(c2c(Cl)cc(C)s2)=O)CC2CCC1CN2C(=O)C(C1(O)CCOCC1)(F)F C1(CCOCC)(NC(C2CC(NC)CN2C)=O)CCN(c2nnnn2C)C1 C12(C(=O)NCc3c(CCNC(C(N)=O)=O)ocn3)CCOC1CCOC2 C#CCCC(O)C(=O)N1CC(CNC(c2ncn(C)c2C)=O)C1 CCCCC(C)CCC(=O)N1CCCC(CC(=O)NCC2CCC2C)CC1 C(C)(C(C(=O)NCC1(O)CN(C)C1)NC(=O)C(C)N1CC(C)C1)OC c1(C(c2nnnn2C(C2CCCC2)C2CC2)NC(CCCC)C)cc(F)cc(Cl)c1 C1(CCC)CN(C(=O)C(CCOC)OC)CCN1C(=O)CN1CCC(C(N)=O)CC1 CCCC(C)C(=O)NCC(CO)NC(=O)Cc1csc(COC)n1 c1(C(=O)NCCN(C(c2sc(F)cc2C)=O)CC)cnnc(C)c1 N1(C(CCC2C(C)C2)=O)CCCN(C(=O)Cc2ccsc2)C1C(C)C C1(CC)CN(C(=O)CCc2ncccc2C)CCN1c1nccc(SC)n1 C1(C(N(CCCNC(c2cn[nH]c2)=O)CC2CCCC2)=O)CCC(=C(F)F)CC1 N1(C(C(CCSC)NC(C2CCC(C(C)C)CC2)=O)=O)CCc2sccc2C1 N1(C(C2(SCC)CC2)=O)CCCC(NCc2cn(-c3ccccc3C)nn2)C1 CCC(CCC(=O)N(C(C)CC)CC)NC(c1nc(=O)o[nH]1)=O C#CC1CN(C(c2ccc(C)c(C)c2)C(=O)NCCCNC(=O)OCC)CCO1 C(=O)(C1=NOC2(CCOC2)C1)N(CCCNC(C1CNC(=O)N1)=O)CCO N1(C(c2ccc(=N)[nH]c2)=O)CC2=C(C1)CN(C(c1cccc(NC(N)=O)c1)=O)C2 c1(C(=O)NCC2C(NC(CN(C3CC3)CC)=O)COC2)ncc(C)cc1OC c1(CC2CC2)cc2ncccc2o1.C12(F)CC(C1)COCC(=O)NCCNC2=O CC1CC(=O)Nc2ccccc2N1C(=O)CCC(C)(C)C#N Cc1ccc(C(F)F)cc1C(=O)NC(C)CCCCNC(=O)COCCCF C(CCC(O)C(=O)NCCS(N)(=O)=O)NC(c1c(C)nccn1)=O c1(C(c2n(CCCSC)nnn2)NCc2nc(Br)sc2C)ccc(F)cc1C#N C1(NC(C(CCC)C)=O)C2COCC1CC(NC(=O)C=CC1CCCCCC1)C2 C(=O)(C1CCCc2nncn21)N1CCC(CNC(=O)C#CC2CCOC2)CC1 c1(C(=O)NCC(C2CCC2)NC(C2CN3CCN2CC3)=O)cc2cccn2cn1 c1(SCC)cncc(C(=O)NC2CC(NC(=O)C=C(C)C)C2)n1 N1(C(CCCCOC)=O)CC(C)(C)CC1C(=O)NCC1CCCN1C C1(C(=O)NC2(C(NOCCOC(C)C)=O)CCSC2)(CF)CCOCC1 C1(CC(N2C(CNC(C3(c4nc(C)[nH]n4)CC3)=O)CCC2)=O)COC(C)(C)CO1 C1(Cl)(C(=O)NCCC2CCN(C(c3c(SC)ccs3)=O)C2)CC12CCC2 C12CCC3CCC1N3C2=O.C1(CNC(C2(CC3CCC3)CC2)=O)(CO)COC1 C1(CC(=O)N(C)CC2CC(=C)C2)C2CCCC2N1C(=O)C(C)C(O)C(C)C c1(NC(CN(C2CCCCC2C(N2CCCC2)=O)C)=O)nc(F)ccc1Cl C1(C(=O)NCC(C2CCCC2)NC(C(C)Oc2ccccn2)=O)CCC(C)(C)OC1 c1(C(=O)NCCC(=O)N(c2ncccn2)C2CCCOC2)ncc(Br)cn1 N1(C(c2c(C)con2)=O)C2CCC1CN(C(c1csc([N+](=O)[O-])c1)=O)CC2 Cc1cc(C(=O)NC2(C)CCN(C(=O)C(C)(F)F)C2)cc(N)c1O c1(OC)ccc(C)c(C(=O)NCC(C2CCN(C(C3CC(CF)C3)=O)CC2)O)n1 C1(CC)CN(C(c2ccc(C)nc2)=O)CCC1NC(c1scnc1C(N)=O)=O N1(C(CCCOCC)=O)CC(C)CN(C(c2cc(=N)[nH]c(Cl)n2)=O)C(C)C1 N1(C(c2cccc([N+](=O)[O-])c2)=O)CC(NC(=O)C(F)(F)CO)CC12CCOC2 C(=O)(C(C)CS(C)(=O)=O)N1CC(CNC(CN(CCC)C)=O)C(C)CC1 N12CCC(C3CC3)C1C2.Cc1ncccc1-n1c(=O)sn1C.N12CC(O)C(C1)C2 N1(C(CC=CCC)=O)CCN(C(c2cc(C(F)(F)F)c[nH]2)=O)C2(CCC2)C1 CCC(C)(CNC(C1CCC(N=[N+]=[N-])C1)=O)C(=O)NCC(C)(C)F C1(C(=O)NCC(C)N(C)C)COCCN1C(c1cnc(C2CCC2)o1)=O C(CCCC(CO)NC(c1scnc1C1CC1)=O)NC(CNC(C(CC)CC)=O)=O c1(C(=O)NCC2COCCN(C(CC(C)(C)SC)=O)C2)c(F)cc(C)cc1F N1(C(C2C(C(=O)OC)C2)=O)CCC1c1ncon1 N1(C(c2ns[nH]c2=O)=O)CC2(CO)CC1(C(=O)NC1CCCCC1(F)F)C2 N1CCC(C)(NC(=O)C(F)(F)C(C)O)CC1.C1(Cl)(COCC)C2CCC(=O)C12CC=O c1(NC)c(C(=O)OCCC(=O)N(CC(F)(F)F)C(C)C)cccc1N N1(C(C2=NOC(C)C2)=O)CCc2[nH]nc(CNC(=O)CC3CCCCO3)c2C1 C1(CC=C)(C(=O)N(CCCO)CCC)CCN(C(c2occc2C)=O)C1 C(=O)(C(N)CCC(F)(F)F)NCC(CN(C)C)O CN1CCC(C(N2CCCCC2CNC(=O)CN2CCCNC2=O)=O)CC1 C(=O)(C1=CC2CCC=CCCC12)NC(C)(C)CNC(=O)Cc1cccc(CO)c1 C12(CNC(C=CC(C)(C)SC)=O)CN(C(c3c(C)ccnc3O)=O)CC1CCO2 CC(C)C(F)(CNC(c1cnn(C)c1N)=O)C(=O)N1CCCC(C(=O)N(C)C)C1 C1(C(=O)NC(c2scc(C)n2)C)(NC(=O)CN2CSCC2=O)CCOCC1 c1(C(=O)NCC2(C(=O)NCC3(OC)CN(C)C3)CCCCC2)cc2cccnn2c1 N1(C(C(CC2CC2)OC)=O)CC(NC(=O)C(c2ccccc2C)(F)F)CC1C CC(CC(=O)NC1(C2CCN(C(=O)CN3CCCCC3=O)C2)CC1)CC(C)(C)C c1(C(=O)NC2CN(C(c3n(CCN(C)C)ncc3)=O)C2)cc2occ(Br)c2[nH]1 C#Cc1ccc(CCC(=O)NC2CCCCN(C(c3cc[nH]c3)=O)C2)cc1 C1(CC=C)(NC(=O)CNS(=O)(=O)C2CC2)CN(C(=O)C(O)CC2CCOCC2)C1 Cn1ccc(=Nc2ccccc2NC(=O)NCC2CC(C)(C)OC2(C)C)[nH]1 c1(C(=O)NCCC2CCN(C(c3cncn3C(F)F)=O)C2)ncccc1O c1(NC(C2CC23CCCCC3)c2n(CCSC)nnn2)cn(C)c2c(C#N)cnn12 CN1CCC(C(N2CC(O)CC2C(=O)NCCC23CC(CCO2)C3)=O)CC1 c1(C(=O)NC(CCCNC(CS(CC)(=O)=O)=O)(C)C)c(Cl)cc(C#N)cc1Cl N1(C(CCC(=O)N(C)C)=O)CCCC(C)(NC(c2cc(Cl)n(C)n2)=O)C1 c1(C(C(=O)NCC2C(CNC(c3ccn(C)n3)=O)C2)(F)F)c(F)cccc1F c1(C(N2CC(CC=C)(C(=O)NCC(C)(C)N3CCCC3)C2)=O)cnc2n1CCC2 Nc1cccn(CC(N2CCCC2CCCCNC(=O)CC2CC3(CC3)C2)=O)c1=O c1(C(C)C)ccc(C(=O)NCCOCCN(CC(=O)N(C)C)C)o1 n1(CC(=O)NC2C(C)CN(C(c3cnc[nH]3)=O)CC2)ccc2cccnc12 C1(C2CN(C(c3ccsc3Cl)=O)C2)(NC(C(C)OC2CCOC2)=O)CC1 N1(C(C=CC(C)(C)NC(C(n2ncc(C)c2)C)=O)=O)CCCC(CCO)CC1 C1(C(=O)NCC(CC)OC)(CNC(=O)CCc2ccon2)CCCC1 c1(CCCC)cc(C)c(C(N2CC(NC(C3(CO)CCCCO3)=O)C(F)C2)=O)o1 C(N=C(NCC1CCOC1)N1CCC(C)(CC)C1)c1ccc(OCCC)c(F)c1 S(=O)(=O)(c1csc(C2CCCCC2)n1)N1CCCN(C)CC1 CC1C(NC(=O)CCF)CCC(n2cc(-c3ccc(Cl)cn3)nn2)N1CC(=O)O N1(C(C(C(=C)Cl)(C)C)=O)CC2OCCN(C(c3ncc(CC)cn3)=O)C2C1 c1(SCC(=O)NC2C(NC(C(C(=O)OC)OC)=O)C2)ccccc1[N+](=O)[O-] N1(C(CN(c2occc2C)C(=O)CC2CC2C(F)(F)F)=O)CCN(C(C)=O)CC1 C(c1ccc2c(c1)CCO2)=CC(=O)NCC(C)N(C(=O)C1=CCSC1)C C1(CNC(=O)C=CCO)CCC2CN(C(=O)CCc3ncccn3)CCC2C1 C(=O)(C(F)C(C)C)NC1CC(C)(C(N2CCC(CC#C)C2)=O)C1 Cc1ccc2[nH]c(C(=O)NC3CCC(NCc4ccc5ccnn5c4)C3)cc2c1 N1(C(C(C)=C2CCC2)=O)CCC(C)C1C(=O)NCCCF c1(OC)cccnc1Sc1ccccc1.C12(CN(C(=O)NC(C)C)C1)C(=O)N2 Cc1ncnc(C)c1OCC(=O)N(CCCCN(C)C(C1CCC(F)(F)C1)=O)C N1(C(C2CC(CC)C2)=O)CCCC(NC(=O)CSCC2CCCO2)C(O)C1 c1(C(=O)NC(C2CCN(C(=O)C(C)C3CC3)C2)C)cnc2ccnn2c1O N1(C(CN(C)C)=O)CCC(C(F)(F)F)C(SCCOCCNC(=O)CCC#N)C1 C(=O)(CCCC(C)(F)F)N1CCC(NC(C(C=CC)O)=O)C1 CC1CN(C(C2CCO2)=O)CC1CNC(c1ccc(-c2cnc[nH]2)cc1)=O CC1(C)CC(NC(=O)CCn2cnnn2)CN1C(c1cc(Cl)ccc1F)=O C(=O)(CCC(C)(C)OC)NC(C(=O)NCc1nc(CC)oc1)CCN(C)C c1(C(=O)NCC2N(C(C(CC)C(C)C)=O)CCC2)cc2nccc(C(F)F)n2n1 Cc1nc(C#N)ccc1NC(C1CCN1Cc1cccc(Cl)c1F)=O N1(C(c2cn(CC)nc2)=O)CCCC(C2CCCN(C(C3COC(=O)N3)=O)C2)C1 C1(NC(C(CCC)N(C)C)=O)CCCN(C(c2c(C)nn(C)c2N)=O)CC1 S(=O)(=O)(c1ccc(C(N2CCCCCC2CNC(=O)CC2CC2(C)C)=O)o1)NC N1(C(C(C=C)(C)CC)=O)CCC(C)(C)C(NC(c2cnccn2)=O)C1 C1(N(CC#C)C(c2sc(C)nc2C)=O)CCN(C(=O)COCC2CCC2)CC1 CC(C)CC(CNC(=O)C(C)(C)OC(C)C)NC(c1cccc(SC(F)(F)F)c1)=O Cc1ccc(C(N2CC3CC3(CNC(=O)Cc3c(C)noc3Cl)C2)=O)c([N+](=O)[O-])c1 C1(CNC(c2c(SC)ccs2)=O)CCN(C(=O)C(F)=C2CCCC2)C12CC2 c1(C(N(C(CNC(C2(C(=O)NC)CCC2)=O)C)C)=O)conc1C1(C)COC1 c1(CNC(=O)CCc2cccc3[nH]ncc23)nc2cnc3ccccc3c2[nH]1 Cn1ncc(C(N)=O)c1N(C1CN(S(C)(=O)=O)C1)C(C1C2CC(N)CC12)=O c1(NC(=O)CCn2cc(CCCO)nn2)nc2ccc(I)cc2s1 N1(C(c2c(CC)con2)=O)CC(C2CC2C(=O)NCC(O)(C=C)CO)C1 Nc1ccc2[nH]c(=NC3CCC(NC(C4CC45CCCOC5)=O)CC3)sc2c1 c1(COC)ccc(NC(c2cc([N+](=O)[O-])sn2)c2nnnn2C2CC2)cc1C#N c1(C(C)=O)ccc(C(=O)NCC2CC2NC(c2c[nH]cc(Cl)c2=O)=O)cc1C C(=O)(C1CCCc2c[nH]nc21)N1CC(NC(C2=NOC(C)C2C)=O)C(C)(C)C1 c1(C(N2CCOC3(CCN(C(C4CC4(F)F)=O)C3)C2)=O)c[nH]c2cc(O)ccc12 C1(C(N(CCC(C)NC(c2ccc(C)s2)=O)C)=O)COc2ccccc2O1 CCCCC(CC(=O)NCCN(CCO)C1CC1)NC(C1CC=CCC1)=O C1(N(CCCN(C)C)C)(CNCCCl)CCC(=O)CCC1 Cc1cccnc1CCC(=O)NCC(C)(C1CC1)NC(=O)CC1CCCCC1F c1(NC(N2C3CN(C(C4=C(C)OCCS4)=O)C(C3)C2)=O)nc2cccc(F)c2[nH]1 c1(C(=O)OCC(=O)Nc2ccc(C(=O)OCC)cc2)ncnc2[nH]cc(C)c12 N1(C(CN2C(=N)NCC2)=O)CCC2(CC1)CCN(C(=O)Nc1cc(Br)c[nH]1)C2 Cc1nsc(C(=O)NC2C=CCC(C(=O)NCC(C)(C)CCO)C2)c1N C1(C(N(C(COC)C)CC)=O)CCC(C)(C)N(C(=O)Cc2nc[nH]n2)C1 C1(NC(N2CC(OCCCc3onc(C)n3)C2)=O)CCOCC1C(C)C Cc1cccc2[nH]c(C(=O)NC3CN(C(=O)Cc4sc(O)nc4O)CCS3)cc12 c1(OC)cc(C(=O)N(C2CN(C(=O)CC(C)CF)CC23CC3)C)ccc1C c1(OC)ncccc1C(C)NC(=O)NCC1(N2CCC(O)CC2)CC(F)(F)C1 C123CCCC1N(CC2)CC1(CC1)C(=O)N3CC.c12cc-1cc(C)c2.C(C)(=O)OC S(=O)(=O)(c1ccc([N+](=O)[O-])o1)N(CC(=O)Nc1c(C)cccc1)C CCC(C)C(O)C(=O)NCCC1(NC(c2cc(F)cnc2O)=O)CCCC1 CC1C(NC(c2ccc(C(N)=O)[nH]2)=O)CCCN1C(=O)Cc1ccc(Cl)c(F)c1 N1(CC2OCCN(C(C3CC(CC)C3)=O)C2)CC(NC(=O)CN(C)C)CC1=O C1(C(=O)NC2(C)CCN(C(=O)CSCCC(F)(F)F)C2)CC2(CCC2)CO1 c1(C(=O)NCC2CN(C(C34CC(C)(OCC3)C4)=O)C2)ccc2ncc(=O)[nH]c2c1 Cc1cn2c(CC(=O)NC3CC3CNC(=O)Cc3ccccc3Br)csc2n1 c1(NC(C2CC(NC(c3ccc(C(N)=O)cc3I)=O)C2)=O)cc(Cl)cc(Cl)c1F c1(OC)cc2c(cc1OC)N(C(=O)NC(Cc1ccc(C)cc1)CO)CCC2 Cn1cc(Cl)c(CC(=O)NC2CCC2NC(c2nccnc2N)=O)n1 CC(C)C(C(=O)NCC=CCNC(=O)CCC1CCCN(C)C1)n1cccc1 C1(NC(CN2CC(CC#N)OCC2)=O)CCC2(CCOC2)C1 C1(N(C(=O)C=Cc2cn[nH]c2)CC#C)CCN(C(C2(C(N)=O)CCC2)=O)CC1 C(=O)(C(C)(COC)CC)NCC1N(C(=O)COC)CC(C2CCC(=C)CC2)C1 c1(C(=O)NC2(CNC(c3cc(Cl)sc3Cl)=O)CCOC2)cccc(OC2CC2)c1 c1(C(=O)NC2CN(C(CCc3c(C)cccc3)=O)CC2O)ccc2ncnn2n1 N1(C(CN(CC)CC)=O)CCC2(CC1)COC(CNC(=O)CCc1cc[nH]n1)C2 C1(N(C(c2cccc(C3(C)CCO3)c2)=O)C2CC2)CCCN(C(C23CC2C3)=O)CC1 c1(C(=O)NC(CN(C(c2cc(C3CCC3)[nH]n2)=O)CC)C)cnnn1C C1(CN(C(=O)CCCC2CCC2)C)CN(C(c2cc(C(F)(F)F)n[nH]2)=O)CCO1 CCCC(CC)CCC(=O)N1CCCC(F)(C(N2CCCC(CO)CC2)=O)C1 CCCC(C)(C)CC(=O)NC1(CO)CCN(C(c2csc(Cl)c2Cl)=O)C1 N1(Cn2ncc(S(=O)(=O)NC3CCC3)c2)CCC2(CC1)CNCCO2 N1(C(c2ccc(C(C)=O)cc2F)=O)CCCC(NC(c2csc(C)c2)=O)C(F)C1 c1(C(=O)NCC(n2cc(CCC#N)nn2)C)cn2c(n1)CCC(C)C2 C(CCC(=O)NCC(C)CNC(=O)C(c1ccccc1)n1cccc1)NC(C)=O C1(NC(CSCCCC)=O)C=CCN(C(C2(C)CC(C#N)C2)=O)C1 c1(N2CCCC(NC(c3ncc(C)cc3C)=O)C2C)nc2cccc(F)c2s1 c1(C(C(=O)NCc2ccncc2)N(CCC)CCOC)cc(Cl)cc2c1OCC2 O=S(=O)(c1[nH]c(=NCCc2nccs2)ccc1Br)NCC1CCCC12CC2 C1(CNC(CC(=O)OC)=O)CCN(C(C2CC(C(F)(F)F)(OC)C2)=O)CC1C N1(C(CNC(C(CC)CC)=O)=O)CCC12CN(C(C1(O)CCSC1)=O)C2 N1(C(CN(C(C(C)C)=O)C)=O)CCC(C(=O)N2CCCC(O)C2C)=C(F)C1 CC1OC2CCC1(NC(=O)CCCCCN(C(=O)C(F)C1CCOC1)C)C2 c1(Cn2cc(CC3N(C(C(C)OCC(F)(F)F)=O)CC3)nn2)cccc(F)c1I C1(CCO)(NC(CCN(CCCCC)C)=O)CN(C(C2(CN(C)C)CC2)=O)C1 C1(C(=O)NCc2cc(O)cc3c2CCC3)CCc2ncccc2C1 C1(NC(c2c(CC=C)cccc2)=O)CN(C(c2cccn2C)=O)CCC1(C)C N1(C(c2c(Cl)cc(C)s2)=O)CC2CCC(Nc3ccc(S(C)(=O)=O)cn3)CC2C1 N1(C(=O)CCN2CCOCC2)CC2CCN(C(=O)C(O)Cc3cnc[nH]3)C2C1 C12(C(=O)NC3CCC(N(C)C(c4cc(-c5cccs5)on4)=O)C3)CC(C1)S(=O)(=O)C2 N1(C(C(N2CCOCC2)C)=O)CCC(CF)(NC(C2CC2C(=O)NCCO)=O)C1 C1(CNC(c2c(OC)csc2)=O)CC2CCCC2N1C(c1cn2c(n1)CCC2)=O Cn1[nH]c(=NC(=O)c2cc3cc(-c4cnn(CCO)c4)ccc3o2)c2cccnc12 C1(CNC(C2CN(C(c3ccccn3)=O)C2)=O)(CO)CC12CCC2 C1(n2cc(C(C)OCC)nn2)CCCN(C(c2ccc(C(F)F)o2)=O)CC1 C1(C(N2CCC(COC)(NC(c3cccc(OC)c3)=O)C2)=O)CC2C=CC1CC2 C(C1=CCN(C(c2ccnn2CC(F)(F)F)=O)CC1)NC(c1cc(C)n(C)c1)=O c1(C(N2C(C(C)(C)C(=O)NCC3CCNC3=O)CCC2)=O)ccc(C2CC2)cc1 C1(NC(C2CCC(=O)N2)=O)CN(C(=O)COc2cc(F)cc(F)c2)CC2(CC2)C1 N1(C(C2C(CC)CCO2)=O)CCC(NC(=O)Cc2ncn(C)c2C)C(F)C1 c1(C(N(CCNC(=O)C(=O)NC2CC2)CC)=O)cc(C(F)(F)F)ncc1Cl C#CC1(C(=O)NCCC(F)F)CCN(C(=O)COc2cccnc2)C1 N1(CC(=O)N(CC)CC)CCN(S(=O)(=O)N(C)C)CC(CO)C1 C(=O)(C1CCCc2nnn(C)c21)N1CC(CNC(CCCOCC=C)=O)C1 c1(C(N2CCC(NC(c3cc(C(=O)OC)sc3)=O)C2C)=O)cccc2c1NCC2 c1(C(=O)NCC(=C)CCNC(=O)C(C(C)C)NC=O)cnc2ccccn12 C1(NC(c2ccc(CC)cc2)=O)CC2CCC1N(C(c1cccnc1)=O)C2 C1(O)(CNC(CC=C(C)C)=O)CCCN(C(C2CC(N(C)C)C2)=O)C1 C1(N(C)C(C2CCCO2)=O)CCC2CN(C(C3CCC4(CCC4)O3)=O)CC12 c1(C(N2CCCC(NC(CSCC=C)=O)C2C)=O)ccc(F)c(C)c1N c1(CCC)nc(=NC2CCC(N(C(=O)CCOC)C)CC2)s[nH]1 N1(C(c2cnn(CC)n2)=O)C2CCC1C(CNC(=O)CCc1cc(C)n(C)n1)C2 c1(C(=O)NCC(C)(C)OCCNC(c2ncc(C)nc2)=O)cccn(C)c1=O C1(CNC(=O)COC2CC=CC2)CN(C(C23CC(C2)C3)=O)CCCO1 C1(OCC)CC2(C1)CC2NC(C1CCCN(C(=O)COc2cccc(Cl)c2)C1)=O CC1CC(C)(C(N2CCCC2CN(C(=O)C2=CSCCO2)C)=O)CC(C)O1 c1(OC)ccc2occ(C(=O)NCCCC3(NC(C4(OC)CC4)=O)CC3)c2c1 C1(NC(C(C2CCOCC2)C)=O)CCC(N(C)C(c2cnc(C(F)F)nc2)=O)CC1 c1(CC)ccc(C(=O)NCC2CCN(C(c3sc(C(C)C)nc3C)=O)C2)cn1 c1(NC(C2N(C(=O)C(C)c3cc[nH]n3)CCC(=C)C2)=O)cc(C)cn(C)c1=O C1(CNC(c2cscc2C(F)F)=O)CN(C(=O)Cn2nnnc2C(F)F)CCO1 C(CCC(C)C)(C(=O)NC1CCC(C)N(C(=O)COC(F)F)C1)NC(C)=O C(CC)(C(=O)N(C(C)CN(CCCCC)C)C)=CCCC CC1CC2CN(C(=O)C(C)(C)C3CCCC3)CC2N1C(=O)CCOCCC1CC1 n1(CCCN(C(C2(CCC)CC2)=O)C)cc(C2CCN(C)C2)nn1 N1(C(CCC2CCC(C)O2)=O)CC(O)(C2(CNC(C3CCCS3)=O)CC2)C1 N1(C(c2ccn(CC)c2C)=O)CC(NC(C2CC2F)=O)CC12CCC2 C(=O)(CCC(F)F)N1C(C(N2CC(n3cc(-c4cn(C)nc4)nn3)C2)=O)CCC1 C(=O)(C#Cc1ccccc1)N1CC(C)(CNC(c2c(F)ccc(C)c2Br)=O)C1 c1(CC(=O)N(C)CCN(C)C(c2n[nH]cc2CN(C)C)=O)ccc(Cl)cc1Cl CCC(C(=O)N1CCC2CC12)N(C)C(c1csc(F)c1)=O c1(C(=O)N(C2C(CCC)CN(C(=O)Cc3ccccc3)C2)CC)cc(C)cc(O)c1 c1(C(=O)OC)ccc(C(F)(F)F)c(Cl)c1.c1(CN2CC(N(C)C=O)C2)ccc(N)o1 Cc1cccc(CCN2CCN(C(=O)Oc3oncc3C)CC2)c1 N(C(=NCCS(=O)(=O)C(C)(C)C)NCC1OCCC1(C)C)C(C=C)C n1(C(C)C)ccc(CC(=O)NCC2CC(F)(CNC(=O)C=CC3CCOC3)C2)n1 [N-]=[N+]=NC1(C(N2CCc3nocc3C2)=O)CCN(C(=O)CCC(N)=O)C1 CC(C)CC(C)C(=O)N1CCC(C2CCCN2C(=O)CC2CCC(C(F)(F)F)O2)C1 c1(C(=O)Oc2cc(N3CCS(=O)(=O)CC3)cc(F)c2)ccc2c(c1)CCC=C2 C(=O)(C(C)CC(=O)N(CCC(=O)NC(c1ncc(C)s1)C)CC1CC1)OC C1(C(=O)NC2CC(CC)(CC)N(C(=O)CC3=CCCC3)C2)CCC2(CCC2)O1 [N-]=[N+]=NC1CN(C(=O)CCC2CC2)CC1NC(c1cc2ccccc2o1)=O C1(CNC(CCNC(COC)=O)=O)CN(C(c2cc(O)cc(F)c2)=O)CCCO1 n1(CC)ccc(C(=O)NC2CC3CC2N(C(=O)CSC(C)C)C3)cc1=O C(=O)(C1=C(Cl)CCC1)NCCN(CCOC)C(C1(C(=O)NC(C)C)CC1)=O c1(CN(C2CC(O)C2)C=O)cccc2occc12 C1(CC(=O)NC2C(OC)CN(C(C3CC(C)N(C)C3)=O)C2)CCC(C)(C)CO1 c1(C(N(CC(C)CNC(=O)CC2CCC2)C)=O)ccc(=O)n(-c2cnn(C)c2)c1 c1(OC)ccc(Cl)c(C(C)NC(=O)CN(C2CCC2)C(C)=O)c1 N1(C(Cc2nc(COC)sc2)=O)CC(C)C(C)(CNC(=O)C2=CSCS2)C1 c1(OCC)ccc(C(C(=O)NC(c2ccncc2OC)C)C(C)C)cc1 C12(NC(c3c(CC)nco3)=O)CCN(C(=O)CCc3cc(C)sc3C)CC1C2 c1(C(=O)NCC(C)(F)CNC(C2CC3C(C2)C3(F)F)=O)cc2c(Cl)nccc2o1 c1(C(=O)NCCN2CCN(C(c3c(COC)scc3)=O)CC2)ncn2ccccc12 N1(C(C(CCCC)=O)=O)CC2CN(C(=O)Cc3cc(Cl)n(C)n3)CC2C1 C(C(C)C)(C(O)C(=O)N1CCC2(C1)CN(C(=O)C(F)(F)C(C)O)C2)OC C(=O)(CCCCCCCSC)NC1CCCN(C(c2ccc(SC)o2)=O)CC1 c1(C(N2CC(=O)N(CCc3cscn3)C2=O)C)ccc2c(c1)OCO2 c1(OC)cnncc1C(=O)NCCCCCN(C(=O)CC1CC2(CC2)CO1)C c1(C(CC)C(=O)NC2CCCC2NC(=O)CN2CCCC2=O)ccc(F)cc1 C1(CN(C(c2scnc2Cl)=O)CC)CCCN1C(c1ccc(C2CC2)o1)=O N1(C(c2c(CC)n(C)cc2)=O)CCC=C(C(=O)NCC2CN(C3CC3)C2)C1 N1(C(C(COCC)n2cc(-c3[nH]cnc3C#N)nn2)=O)CCCC(C)(O)CC1 N1(CCC)CCCC1C(=O)NC1(C(=O)N(CCC#N)CC)CC1 C(c1ccc(Cl)c(C)c1)=CC(N1CC(CC)N(C(=O)CCC(=O)NCC)CC1)=O N1(C(CCC(=O)NCCC)=O)CCC2(CCC2NC(=O)CC(C)(C)C(F)F)CC1 c1(OC)ccc(-c2cc(=NCC(C(=O)O)C3CC3)[nH][nH]2)c(Cl)c1 c1(OC)ccc2c(NC(C3CC3NCc3c(C)n[nH]c3C)=O)cccc2c1 C(=O)(CCCC(N)=O)N(CCCCN(C(=O)CCC1CCC(=O)N1)C)C c1(N2CCC(NC(C=CS(CC)(=O)=O)=O)C(F)C2)[nH]cnc2nc(Cl)cc1-2 c1(C(=O)NCC(C)N(C(=O)CC2OCCC2C)C)cnn(C)c1C(=O)O C1(C2CCCN(C(=O)CCc3cn[nH]c3)C2)(NC(CSCC=C)=O)CC1 n1(CC(=O)NCC(CC)NC(=O)CC(C(F)F)c2ccccc2)ccc(=O)cc1C N#Cc1c(F)cc(C(=O)NC2CC2CNC(C2(O)CCSC2)=O)cc1F C1(C(N2C(C)CN(C(=O)COCc3nc[nH]n3)CC2)=O)CCOCC12CCC2 C1(CC(N2C(CN(C(=O)Cc3cnc[nH]3)C)CCC2)=O)CC2C=CC1CC2 C1(NC(c2ccc(CCC)[nH]2)=O)CC2(C1)CN(C(=O)CCc1ccoc1)C2 C1(C2CCN(C(=O)C(CC)Nc3ccccc3)C2)(NC(c2ccc(CC)[nH]2)=O)CC1 C#Cc1cccc(C(N2CCC(CC(=O)NCC(F)(F)F)CC2C)=O)c1 N1(C(C(C)OCCOCC)=O)CCCC(CN(C(=O)Cc2c(C)n[nH]c2C)C)C1 c1(C(=O)NCC=CCNC(C(C(CC)C)O)=O)ccc(Cl)c(C(=O)OC)c1Cl CC(C)C(C)CC(=O)NC(C)(C)C(=O)NC1CC(=O)N(C)C1=O c1(C(N2CC(CC(C)NC(C3(COC)C=CCC3)=O)C2)=O)nc(Cl)sc1C(C)C c1(C(N2C(C)CC(NC(c3cnc(Cl)[nH]3)=O)C2)=O)cc(N)c(F)c(F)c1F Cc1ccnc2sc(C(=O)NC3(CO)CN(C(C4CC(C)C4)=O)C3)c(C)c12 c1(C(=O)NCC2CCN2C(C2CNC(=O)N2)=O)ccc(-n2cccn2)nc1 n1(C(C)C)nnc(C(N2CCC(CNC(=O)CC3C(C)C3(F)F)C2)=O)c1C1CC1 N1(C(c2c(COC)csc2)=O)CCC2C(CCCN2C(=O)CCCC2CC2)C1 c1(OC)ncc(Cl)cc1C(=O)NC1CCN(C(c2cnc(NC(=O)OC)o2)=O)C1 C(CN=[N+]=[N-])(C(=O)NC(C)C(C)C)NC(CN(C1CC1)CC)=O C(=O)(C(CNC(=O)C(F)CC1CCCC1)CC1CC1)NCC1(CC(N)=O)CC1 C(=O)(CCCCCF)NC(CC)CC(=O)Nc1ccccc1O C12(NC(C3CN(C(c4cc(OC)c(C)cc4)=O)CC3C)=O)CCC(O)(CC1)CC2 C1(OC)CN(C(C2CCCN(C(C)C)C2)=O)C2(CCCC2)C1 CC(C)CC(O)CNC(=O)C(CCF)NC(c1ncccc1N)=O C(CC(=O)NCCc1ccns1)(C(C)(C)C)NC(Cn1ccc(C)n1)=O Cc1cnc(C(N2CCC(CCNC(=O)CSc3cnn(C)c3)CC2)=O)cn1 C(=O)(CC1=CCCCC1)N(CC(N1CCCC(C(F)F)C1)=O)CCOC N#Cc1ccc(F)c(C(N2CC3CC2CN3C(=O)CCCN2CCCC2)=O)c1F C1(NC(c2ccc(C#C)cn2)=O)CC2CC(NC(C3OCCO3)=O)CC2C1 c1(C(=O)NC2CCN(C(Cc3c(C)scc3)=O)C2C(C)C)cc2n(n1)CCO2 C(CC)(c1ccccc1)=CC(=O)NC1C2(CCN(C(C3(CCCC)CC3)=O)C2)C1 c1(NC(N(CC2C(C)CCCC2)Cc2ccccc2)=O)nc2nccc(Cl)n2n1 C(=O)(C1CCc2c[nH]nc21)NC1C(NC(=O)Cc2ccccc2Cl)CCC1 C1(CNC(C2C(OC(C)=O)C2)=O)CN(C(=O)CC2CCCCO2)CC12CC2 N1(C(=O)C(Cl)=CCl)CCC2(CC1)CCN(C(=O)C(c1cccc(F)c1)O)C2 CN1CC(C(N2CC3CC3(C(=O)NC3C4CCCOC34)C2)=O)CC1=O N1(C(c2n(C(CC)C)ncc2)=O)CCC2(COCC)C(C1)C2(F)F Cc1cccc2c1c(CN1CC(C)(CNC(c3cnnn3C)=O)C1)cn2C N1(C(c2c(C)nco2)=O)CCC(C(=O)NCC2CC(O)C23CCC3)C(O)C1 c1(C(N2C(CNC(c3ncsc3C3CC3)=O)CCC2)=O)cc2c(cc1Cl)NCC2 N(C(=NCC1CC1)N1CCC(C)(CNS(=O)(=O)c2ccccc2)C1)C(CC)CC c1(N(C)C(=O)OC(C)(C)C)nnc2ccc(OCN=S(C)(C)=O)nn12 C1(CNC(C(C=C)(C)C)=O)CC(NC(=O)C(=O)Nc2c(F)cccc2F)C12CCC2 c1(CC)ccc([N+](=O)[O-])cc1C(=O)NCCNC(=O)Cc1sccc1S(N)(=O)=O CC(C)C(C)(C)C(=O)NCC1CN(C(c2c[nH]nc2C2CC2)=O)CC1(F)F C1(NC(CCC(C)C)=O)CC(O)CN(C(c2nn(C)c(Cl)c2C(F)(F)F)=O)C1 N1(c2ncnc(C)c2C#N)CC2CCCC(NC(C3NC(=O)C4CCC34)=O)C2C1 C=CCCCC(C(=O)NCCCNC(C)=O)NC(c1cccn1C)=O N1(C(C2CN(C)C2)=O)CCCC1CCC(=O)N(C1CC1)Cc1ccoc1 S(=O)(=O)(c1cccc(Cl)c1)NC1CCC(C(=O)NCC2CC3CCC2CC3)C1 N1(C(CCN(CCC)C)=O)CC(C)CN(C(C2(C)CCC(=O)NC2)=O)CC1C C1(C(=O)NCC=C=C)C(O)CCN1C(c1csnn1)=O Cc1ccccc1CC(N1CC2(NC(=O)CSc3ccccn3)CC1C2)=O Cn1nc(-c2ccoc2)cc1C(=O)N(C1C2CNCC12)Cc1nc[nH]n1 N1(C(c2ccc(CC)cc2)C(=O)NC2COC2)CCCC2NC(=O)C12 CCCC(CCC)=CC(=O)NCCn1ccc(C(N2CC(n3cccn3)C2)=O)c1 c1(OCC(N2CC(C)C(CNC(=O)CCC#N)C2)=O)ccc([N+](=O)[O-])cc1Br CC1CC(C(=O)NC(CNC(c2cc(-c3ccccc3F)no2)=O)CO)CN1C C(=O)(C(C)(O)CC)N(C)C(C12CC(N(CC(CC)O)C(C)=O)(C1)C2)=O Cc1c(OC)cccc1NC(=O)COC1CC2CC2C1.C=CC C1(CC(=O)N(CCSC)C)CCC(C)CN1C(=O)CCNc1ccccc1C(N)=O C1(C(N2CC(CC)C(NC(=O)C(c3ccccc3)F)C2)=O)CC(C)(C)OC1(C)C c1(C(N2CC(NC(CC(=O)NCC#C)=O)C(F)CC2)=O)ccc2nn[nH]c2n1 C=C=CC(C)C(=O)NC(C1CC(NC(C2(CCCCO)CC2)=O)C1)C Cc1noc(N)c1C(=O)NC1CN(C(=O)CC2CCCS2(=O)=O)CC1C(F)(F)F N1(C(c2c(CNC(CC3CCN(C)C3)=O)noc2)=O)CCc2nn(C)cc2C1 CC1CN(C(=O)C(C#N)CC2CC2)CC1CNC(=O)Cc1cccc(F)c1 Cc1cncc(CCC(=O)NCC=CCNC(=O)CC2CCC(C(F)(F)F)O2)c1 C(CCC(=O)NCC(CNC(=O)C(O)C1CC1)CO)OCC=C CC1C(NC(c2cc3occc3[nH]2)=O)C(C)CCN1C(C1CSCCS1)=O Cc1ccc(C(N2CCCC2C(C)NC(C23CCN(CC2)C3)=O)=O)nc1C C(=O)(C(C)C(F)F)NCc1cn(C(C(=O)N(C(C)(C)C)CC)C)nn1 N1(C(CC(C)CNC(C2(C#N)CCCO2)=O)=O)CCC2C(O)C(C)(C)C12 c1(C(=O)OC)nc(Cl)[nH]c(=NCC2(C)CCCN2C(=O)Cc2cscn2)c1OC O=C(CN=c1cc[nH]cc1)NC(C(=O)NC1CCCOC1)c1cccs1 c1(C(C)C)ncc(C(=O)N(C2CCN(C(=O)CN(C)S(N)(=O)=O)C2)C)[nH]1 N1(C(CN(C(CN(C)CC)=O)C(C)C)=O)CCC(CC(=O)NCCCO)CC1 CCCCCC(C(=O)NC1(C)CC(NC(=O)CCc2ccc(F)nc2)C1)C(C)C C1(CNC(C2C(NC(c3cnc(C(N)=O)s3)=O)C2)=O)CCNC(=O)C1 Cc1ccn(C)c1C(=O)NC1COCC1CNC(=O)CC1(C)CCOC1 N1(C(c2c(C)nc[nH]2)=O)CCN(C(c2coc(-c3ccsc3)c2)=O)C(CC2CC2)C1 c1(CC)nscc1NC(C1CCC1CNC(c1cnn(CCO)c1)=O)=O C#CC(C)(C)C(=O)NC=CCC(=O)NC(C1(COC)CC1)C c1(C(=O)Nc2c(C)nc(-c3cc(OC)cc(C)c3)s2)cc(OC)c(O)c(Cl)c1 N1(C(c2n[nH]c(C)c2O)=O)CC2(COC(CNC(=O)CCC3CCOC3)C2)C1 c1(Cn2c(-c3c(-c4n(C(CC)C)ccn4)cccc3)ncc2)cc(C#N)n(C)c1 c1(OC)cccc(C(N2CCNC(C(N3CCOC(C4CCC4)C3)=O)C2)=O)c1 C1(CC)CN(C(c2cccc(C)n2)=O)CCN1C(=O)C(C(C)C)c1cnn(C)c1 N1(C(c2cnc(C(=O)OC)s2)=O)CC2(CCCC(CNC(=O)C(C)O)O2)C1 C1(C)(CNC(C2N(C(C(CC=C)NC(C)=O)=O)C(C3CC3)CC2)=O)CCC(=O)N1C C1(C(N(CCC(C)NC(c2ccn(CCN(C)C)n2)=O)C)=O)CC2CCCC2C1 C1(C(N(CC(CC)NC(=O)CC2CCCCC2(C)C)C)=O)CC2(C1)CC(F)(F)C2 C(CC(C)C(=O)NC(CNC(c1cc(-c2ccccc2)oc1C)=O)CC)=CCC C1(NC(C2C(C(=O)NC(C(=O)OC)c3ccoc3)C2)=O)CC(N=[N+]=[N-])C1.C1(C)CC1 Cc1ccc(C(N2CC(O)(CC(=O)NCc3cccc(Cl)c3)C2)=O)c(C)c1 N1(C(CNC(=O)NC)=O)C2CCC1C(CNC(=O)C(c1c(C)noc1C)(C)C)C2 C1(C(=O)NC(C)C(CO)NC(c2cnc(C(C)(C)C)[nH]2)=O)CC(N=[N+]=[N-])C1 C1(c2cn(CC(=O)NC)nn2)COCCN1C(c1sccc1SC)=O C#CC12CCC(C(=O)NCCOC3CN(C(c4cc(C)n(C)c4)=O)C3)(CC1)CC2 N1(C(C(C)=C2CC2)=O)CCC(C)(CCNC(c2nsnc2O)=O)C1 C1(C(N2C(C(N)=O)CC2)=O)(NC(C23CCC(C2)C3)=O)CC=CC1 C(=O)(C1=C2CCCN=C2NN1)N1C(CNC(COCCCC)=O)C(C)CCC1 c1(OCC(=O)NCC2CC2NC(c2nnc(O)cc2O)=O)cc(F)cc(Cl)c1 CC1CC(CNC(c2ncc(N(C)C)cn2)=O)CN1C(C1CCCS1)=O n1(CC)nc(C)c(CC(N2CCC(CCNC(=O)C=C3CCC(C)C3)C2)=O)c1C c1(C(N(CCN(C(c2csc(Cl)c2Cl)=O)CC)CC)=O)ccc2c(n1)CCC(C)C2 c1(C(CC)C)cc(C(N2CCC(C(C)NC(=O)C(F)(F)C3CC3)C2)=O)on1 C12(CNC(C(CCC)(C)C)=O)CCCC1CN(C(c1cnc3n1CCOC3)=O)C2 C1(CNC(C=C(C)c2cnn(C)c2)=O)N(C(=O)CCC2(C)CC2)CCCC1(C)C N1(C(c2ccc(C)c(C)c2)=O)CC2CCCC(Nc3cccc(F)c3C#N)C2C1 C(C(CNC(c1nnc(S)n1C)=O)S(C)(=O)=O)NC(c1cncc(OC)c1)=O O(NC(=O)C(c1cccs1)NC(c1ccc(Cl)cc1)=O)CCCC N1(C(C2(CC)CCN(C(=O)Cc3csc(C)c3)C2)=O)CCC(F)(F)C(O)C1 CC1CN2CCN1C(C(N1CC(O)CC1CNC(=O)C(C)(C)C(F)F)=O)C2 C1(NC(C2(OC)CCSC2)=O)CN(C(=O)Cc2c[nH]nc2C)CCC1CO C1(CC)CN(C(c2ccc(-c3ccno3)cc2)C(=O)NC2(C)CC2)CC(CC)O1 C1(CC(=O)NC2(C(=O)NCc3c(C)noc3Cl)CC2)CCC2(CCC2)CO1 N1(C(C2CCCC(=O)N2)=O)CCC12CN(C(=O)C(O)CC1CCOCC1)C2 C(=O)(C1Cc2ccc(F)cc21)N(C1CN(C(C=Cc2scc(C)n2)=O)CC1O)C c1(CC(N2C3CC(NC(CC(C)SC)=O)C2CC3)=O)c(C)nc2ncnn2c1C C1(C(N2CCC(NC(c3c(C)cns3)=O)CC2C)=O)CCc2ccccc2O1 C1(C(C)NC(c2sccc2C2CC2)=O)CCCCN1C(=O)CC1(C2CC2)CC1 CCC(C(=O)N1CCCCC1CN(C)C(c1cccc2c1COC2)=O)C(F)(F)F N1(C(c2n(CC)ncc2)=O)CCC(C(=O)Nc2cc(C)cnc2OC)C(O)C1 c1(C(=O)NCC2CN(C(=O)CC3CCCCO3)CC23CC3)cnc2c[nH]nc2c1 Fc1ccc(Br)c(CSCc2nnc(-c3cn[nH]c3)n2C2CCCCC2)c1F c1(CSC)nc(-c2ccc(Cl)cc2)nn1-c1ccc(F)nn1 C(=O)(C1=NN(C)C(=O)CC1)NC(c1c(OC)cc(C)c(C)c1)c1ccc(Cl)cc1 C1(CNC(C2C(=C)CC2)=O)(CNC(=O)C(F)(F)c2cnn(C)c2)CCOCC1 C1(C(=O)NC2(C)CCC(NC(=O)COC(F)F)CC2)CCc2n[nH]cc2C1 C1(C(N(C(c2ccncc2)CC)C2CC2)=O)COc2cc(C(=O)O)ccc2O1 c1(C(=O)OC)ccc(CC(=O)NC2CCCC2NC(=O)CSC(F)F)s1 N1(C(C(C)CC(=O)c2ccccc2F)=O)CC2(CCN(C(=O)CC3CC3)CC2)C1 c1(OC)nc(N2CCCC(C)(C(N3C(C)CCC(F)C3)=O)C2)ncc1F C=C1COCC1C(=O)NCC1(CC2CCC2)CC1 c1(NC(C2C(NC(C=CC(C)C)=O)CCCC2)=O)nc(Cl)ccc1Br N1(CC(=O)NCc2cn(C=C)nc2)CCCC2C(O)C(C)(C)C12 C1(N(C)CC)CCCN(C(c2conc2C(C)NC(C2CC2Cl)=O)=O)C1 c1(C(=O)NCCc2c(C)n[nH]c2)c(CNC(C23CC(C#N)(C2)C3)=O)cnn1C C12(C(N3CC(C)S(=O)CC3)=O)CC(CCO1)N(C(c1csc(O)n1)=O)C2 c1(C(N(C(CNC(CC(=O)OCCC(C)C)=O)C)C)=O)ccc2ncn(C)c2c1 N1(C(CCC(=C)Cl)=O)CCCC(NC(c2cnc(CC)s2)=O)C1C CCCCCCCCCN1CC(C)(CC(=O)O)C1 c1(C(N(C)CC2CCCN(C(c3cc(OCC)no3)=O)C2)=O)c(C)cccc1Cl O=C1CC(O)(c2ccccc2)N1.c1ccccc1.C1(CCN)CCSC1 c1(CC(N2CC(OC)(CNC(c3cnn(CCF)c3)=O)C2)=O)cc(F)cc(Cl)c1 Cc1ccc(OCC(=O)N(C)C(C)C2CC2)c(Cl)c1 N1(Cc2ccc(COC)cc2)C(=O)CN(C(c2cccc(C)n2)C)C1=O c1(C(=O)NC(CNC(C2(Cl)CC23CCC3)=O)CO)cc2c(O)cccc2[nH]1 C12(NC(c3cc(C)[nH]c3)=O)CCC(CC1)N(C(=O)CCc1c(F)cccc1Cl)C2 Cc1ccncc1C(=O)NCC1CC(O)(CNC(c2cc(Br)no2)=O)C1 C1(O)(CN(C)C(c2sccc2CO)=O)CCN(C(c2cc(F)ccc2O)=O)CC1 C(N=c1[nH]c(=NC2CCCCCCC2)c2sccc2[nH]1)C1CCN(CCOC)C1 C(=O)(CC(C(C)(C)C)NC(C1CCC(=O)C1C)=O)NC(C(C)C)c1ncc[nH]1 C12(NC(c3cnc(C(C)(C)C)[nH]3)=O)CC1CN(C(C1CCCOC1)=O)C2 C(CN=C(NCCSC)NC1CC(OC(C)(C)C)C1)=CCC C#CCCCCC(C(=O)N1CCOCC(C)C1)N1CC(=O)NCC12CC2 C(=O)(C(O)CC1CCOCC1)NCCN(CCOC)C(c1cc(C)c[nH]1)=O Cc1[nH]nc(C(N2CCC(CC(=O)NCC(C)(O)C3(C)CC3)CC2)=O)c1Cl c1(C2(C(c3nn[nH]n3)N(CC(=O)N(C)CCO)C)CCC2)ccc([N+](=O)[O-])cc1 c1(C(=O)NC(C2C3CC4C(C3)C24)C)ccc(-n2cc(Br)cn2)nn1 c1(C(=O)NCC(c2ccc(Cl)cc2)N(C(C)=O)C)nn(C)c2c1CCC2 S(=O)(=O)(c1ccc2nc(N3CCSCCC3)sc2c1)N1CCC([N+](=O)[O-])CC1 CCCC(CC(=O)N1CC(c2cc[nH]n2)C1)NC(C1(CC)CC(C)(C)C1)=O C(=O)(CCC(C)S(C)(=O)=O)N(C1CCN(C(=O)CCCCC(=O)OC)CC1)CC C1(CC(=O)NC)CN(C(=O)Nc2ccc(C3CCOC3)cc2)CCO1 C1(C(=O)NC2C=CC(CNC(=O)C(C)Cc3ccco3)C2)(CC)CCOCC1 C1(NC(CC2CCN(C(COCCCN(C)C)=O)C2)=O)CCC(N=[N+]=[N-])CC1 CC1(C)CCc2cc(C(N3CCCC(NC(=O)CCC4CC4)CC3)=O)c(O)nc21 C1(OCC)CC(N)(C(=O)Nc2ccc(Oc3ccccc3C)cc2)C1(C)C N1(C(CNC(CCC)=O)=O)CCCC(CN(C)C)C1.c12ocnc1C(=O)NC2 C(=O)(C1CCCc2c[nH]nc21)NCC(CNC(c1cc(CC2CCC2)c[nH]1)=O)F C1(C(=O)NCCn2c(C)cc(C)n2)CC2C=CC1N(C(c1cc[nH]c1C1CC1)=O)C2 CCCCC(CNC(C1CCC(NC)CC1)=O)NC(=O)CC(C)c1ccccc1 C1(C(=O)OC)NC2CC1CC2NC(=O)NC(c1ccc(-c2nnc(C)s2)cc1)C N1(C(COCCC)=O)CCN(C(=O)CCCC2CCCO2)C(c2nccn2C)C1 C1(C2CN(C(=O)C(C)(CC3CCC3)OC)C2)(NC(C=CC(C)(C)SC)=O)CC1 N1(C(CCCCC)=O)CCC2(CCC2)C(CNC(c2c(CO)noc2C)=O)C1 CCC(CN(C(=O)C(F)C1CCCC1)CC)NC(=O)Cn1ccnn1 C1(NC(CNS(CC)(=O)=O)=O)CCN(C(c2cccc(C(F)F)c2)=O)CC1C C(=O)(C1CCC(=O)c2cccn21)N1CCC(CNC(C2CC(OC)C2)=O)C1 C(=O)(CC(C(F)(F)F)NC(c1ccccc1)=O)NCC12CC(NC(CSC)=O)(C1)C2 C1(C(=O)NC2C=CCN(C(c3cnc(SC)nc3O)=O)C2)CCc2nc[nH]c2C1 N1(C(c2cncc(C)n2)=O)CCN(C(c2cn3cnnc3cn2)=O)CC(O)C1 N1(C(CCc2cc(C)no2)=O)CCN(C(=O)C#CC2(C)CC2)CC2CCCCC12 C1(COC)(NC(=O)COCCC(C)C)CCN(C(c2cc(C(F)F)cs2)=O)CC1 c1(CC)c[nH]nc1C(=O)NCC1(C(=O)NCC2CC(SC)C2)CC=CC1 C(C(C(=O)NCc1ccc2cncn2c1)C(C)(C)C)NC(C(C)SC(C)C)=O CC(C)CCC(O)C(=O)NC(C1CN(C(c2c[nH]cc2-c2cnn(C)c2)=O)C1)C C1(CC(=O)NCC(C)NC(=O)C(C)(C)C(F)F)Oc2ccccc2NC1=O c1(NC(COC2CCN(C(C(CC)SC)=O)C2)=O)ccc(C)c(C)c1F C1(CN(C)C(c2ncc[nH]c2=O)=O)CCCN(C(=O)CC2(N(C)C)COC2)C1 Cc1nc(-c2cccc(Cl)c2)sc1C(N1CCC(NC(=O)CC(C)O)C1)=O CCC(C(=O)N(CCCCCNC(c1cc(C)ns1)=O)C)C(C)C CCC(C)C(CNC(=O)C(O)C1CN(C(=O)C(c2c(C)noc2C)(C)C)C1)OC C1(C(=O)NCCOCCNC(=O)C#CC2CC2)CC12CCOCC2 C1(NC(CC#N)=O)CCCN(C(C2(Cn3ccccc3=O)CC2)=O)CC1 C(=O)(C#CC1CCCC1)NCCC1CC(NC(C(c2cccc(C#N)c2)O)=O)C1 C(=O)(C1CCOc2ccccc21)N(CCCNC(c1ccc(OC)nc1)=O)C1CC1 C1(OC)CC(C(N2CCC2C(N)=O)=O)N(C(=O)CC2CCSC2)C1 S(=O)(=O)(c1cccc([N+](=O)[O-])c1)NC(C)C(=O)NC1CC12CCCC2 Cc1cc(S(N)(=O)=O)ccc1NC(c1n[nH]cc1-c1ccnc(C)n1)=O c1(C(N2C(CNC(C(C)(C)Br)=O)CCC2)=O)cccc2c[nH]nc12 C1(=O)C(C)C(O)C(C)CON2CCC(F)C(CC(SC)=NN(C)C=CC2=O)N1 N1(C(c2nccc(N(C)C)c2)=O)CC(C2CN(C(=O)C=CCF)C2)C1 C1(NC(COCCC(C)C)=O)CN(C(=O)Cc2n[nH]c(=N)s2)C(C)(C)C1 c1(C(=O)NCC2N(C(C3C(OC)CCC3)=O)CCC2)c(C)ccc(N)c1C C1(NC(C2CCCSC2)=O)CCN(C(C2(Cl)C3CCC(=O)C23)=O)CC(O)C1 C=CCC(CNC(=O)CCC1CCCO1)NC(=O)Cc1coc(C(F)F)n1 C1(SC)CN(C(c2ccc(=O)oc2)=O)CC1NC(c1cccc(OC(F)F)c1)=O C1(NC(C(C2CC(NC(CC)=O)C2)F)=O)CC(C)(C)OC1(C)C C(=O)(C(C)C(=O)N1CCC(NC(=O)CSc2nc[nH]n2)CC1)OC C1(c2cccc(SC)n2)CN(N(C)C2CCc3ccccc32)CCO1 c1(OC)cc(C(N2CCCC(C(=O)NCc3cocn3)CC2)=O)ccc1C(F)F c1(C(N(CC(CNC(C2CC(C)=C(C)CC2)=O)(C)C)C)=O)cccc2c1COC2 c1(CC(=O)N(C(C)C)CCNC(C2CNC(=O)N2)=O)ccc2nn[nH]c2c1 C1(C(=O)NCCCCCN(C)C(c2nnn(C)c2N)=O)CCCC12CC2 Cc1nc(NC(C2COCCN2Cc2ccc3c(c2)CCC3)=O)c(Br)cc1Br C1(C(N(CCNC(=O)CCc2cc[nH]n2)C2CC2)=O)CC2(C1)CC(O)C2 C(=O)(C1CCCc2c[nH]nc21)N(C1CCC(NC(c2n[nH]c3c2CCOC3)=O)C1)C C(c1cncnc1O)=CC(=O)NC(C1N(C(c2c(OC)cccc2)=O)CCC1)C O=C(C(Cc1cc[nH]n1)NC(C1(F)CCOC1)=O)NC1(CCF)CC1 c1(C2(CC(=O)N(C3CCCC3)CCNC(=O)C(F)C3CCC3)COC2)ccccc1 CC1CCN(C(=O)CCCN2CCCC2)C1CNC(=O)C1=CCCC1 N1(C(c2ccc(SCC)cc2)=O)CC2(C1)CN(C(=O)CCc1cnn[nH]1)CCO2 N1(C(COC(Cc2ccc(C)o2)=O)=O)CC(C)CC(C)C1 C1(NC(c2c(CC)csc2)=O)CC(C)N(C(c2ccnc(CO)c2)=O)C1 C1(CC(=O)NC(C(C)NC(CCC(=O)NC)=O)C)NC(=O)CNC1=O C1(CNC(C2CCC(=C)CC2)=O)CC2(C1)CN(C(c1csc(Cl)c1Cl)=O)C2 N1(C(C(CC)(F)F)=O)CC(C)(C)CCC1CNC(=O)Cc1ccc2cncn2c1 C1(CC(=O)NC2CCC(CCNC(CCC3(C)CC3)=O)C2)CCCC(F)(F)C1 c1(C(=O)NCCC(C)N(C(CCSCCOC)=O)C)ccc(F)c(OC)c1 C1(C(C2N(C(CCCCC3(O)CCOC3)=O)CC2)=O)CCN(C2CCCCC2)C1=O N1(Cc2ccc(OC(C)C)cc2Cl)CCc2cc(Cl)cc(Cl)c2C1C C(C(C(=O)NCC(C)N(C(c1ccnc(O)c1)=O)CC)C(C)(C)C)OCC=C c1(-c2n(CC)ccn2)ccc(NCc2n[nH]c(C)c2Br)cc1 C1(C(N(CCS(C)(=O)=O)C(C)C)=O)CCCN(C(=O)OC(C)C)CC1.C(C)(C)C c1(Cc2cn(CCCC(=O)NCC(COCC)O)nn2)ccnc(C)n1 c1(C(N2CCC(C)(O)C2)=O)cnc2ccc(C3=CC(C)(C)C3)cn12 C1(NC(C=CC=CCC)=O)CC2CN(C(C3CCN(C(=O)C4CC4)CC3)=O)CC12 C1(NC(C2(CCCC)CCCC2)=O)CC(C)CN(C(=O)CCCC(N)=O)C1 c12ccc3c(c1)CCN(C3)C(=O)c1cccc-2c1.c1(CN(C)C)cnn(C)c1 N1(C(C(C)OCC)=O)CCCC(CN(C(c2cnc(C(C)C)[nH]2)=O)CC)C1 N(S(=O)(=O)N1CC(C)OC(C)C1C)(CC=C)CCC C12(OC(c3ccsc3)=O)CC(C(F)(F)F)C1CN(C(=O)CCNC(=O)NCC)C2 C(C)(C)(C(=O)N1CC(OC(C2C(C(=O)OC)C2)=O)C1)NC.C(C)(C)OC N=c1[nH]c(=NCC(F)(F)c2ccccc2Br)[nH]c(=NC2CCC(O)C2)[nH]1 c1(C(=O)NCC(N2CCCCC2)=O)cc(NC(C2CC3C=CC2C3)=O)ccc1O c1(OC)ccc(CSN2CCC(Cc3ccccc3C)C2)c(OC)c1OC C12(CC(=O)NC3C=CC(C(=O)NC)C3)CCC1CN(C(c1cncc(F)c1C)=O)C2 CCCCC(C(=O)NC(C)CN(C)C(c1cccc(SC(F)(F)F)c1)=O)N(C)C c1(C(=O)NC(C)CN(C)C)n[nH]c2cccc(-c3cccc4nonc34)c12 c1(OC(C)=O)ccc(CC(=O)NCC2CCOC2)cc1OCCOCCN(C)C c1(C(N2CC(NC(C(CC)NC(C)=O)=O)C(F)C2)=O)cccc(F)c1O c1(OC)c(Cl)ccc(C(=O)NCC(C2(O)CCN(C(=O)Cn3nccn3)C2)C)c1F C1(C(=O)NC2C(NC(C(C)SC)=O)CC2)CCN(C(=O)C2CC2)CCC1 c1(OCC(=O)NCC(CC=C)NC(=O)CC(C)(C)C)ccc([N+](=O)[O-])c(C)c1 N1(C(C(c2cccc(C)c2)F)=O)C2CCC1C(F)C(NC(=O)C(C)C1CC1)C2 C(c1ccccc1)=C(OC)C(=O)NCC(CO)NC(c1ccc(C(C)(C)C)s1)=O C(=O)(CS(=O)(=O)C1CC1)NCCCNC(CC1CC(C(=O)OCC)C1)=O c1(C(=O)NC(c2cc(F)ccc2F)C)ccc2c(c1)S(=O)(=O)CCC2 C1(CNC(C2C(C)C2)=O)CCCC(CNC(=O)CCOc2ncccc2Br)C1 C(=O)(C(CN(C)C)NC(=O)COC(F)(F)F)NCC(C)(C)c1cnco1 CCC(C)CC(C)C(=O)NC1CCCN(C(=O)COCc2ccncc2)C1C C1(C(N(CCCNC(c2c(CCC)onc2C)=O)C(C)C)=O)CC2(C1)CC(F)C2 C1(C(=O)NCC2N(C(C3N(C(=O)NC)CCC3)=O)CCCC2)C2C3CCC(C3)C12 C1(OC)CN(C(C2CC2C2CC2)C(=O)Nc2ccccc2Cl)CC12CC2 Cc1c(C(N2CC3(CNC(=O)C(C)CO)CC(F)(C2)C3)=O)[nH]c2c1C(=O)CCC2 N(C1c2ccccc2CC1O)C(=O)Nc1nccs1 CCC(CC)C(C(=O)N1CC(NC(C23CC2CNC3=O)=O)C(F)C1)OC C1(NC(CCCC)C2CCOC2)CC2C3CCC(C3)C2C1 Cc1nn2c(c1C(=O)NC1CC(NC(=O)C(C)OCCC(C)C)C1)CCCC2 c1(C(N2C(C(=O)NC(C)Cn3ccnc3)C=CC2)=O)cc(=O)n(C)cn1 C1(CC(=O)OC)CN(Cc2cc3c(F)cccc3[nH]2)C2COCC2O1 N#CC1CCCCN1C(C1(CO)CN(C(=O)CCC(F)(F)F)C1)=O C=CC(CC)CC(=O)N1CCN(C)CC1C(=O)NCC(=O)N(C)O c1(Cn2cc(CN(C3CCC=CCC3)C)nn2)cn2c(n1)CCCC2 N1(C(c2c(C)snn2)=O)CCC(O)(C(C)CNC(=O)COc2cccnc2)C1 Cn1cccc1CCC(=O)N(CCCNC(C1CC(O)C1)=O)CCO Cc1cnc(O)n1-c1cccc(C(N2CCC(NC(=O)C=C(Cl)Cl)CC2)=O)c1 C1(CC=C)(C(=O)N(C)CCn2ccnn2)CCCN1C(=O)CCc1cn(C)nn1 N1(C(c2cc(C)nn2C)C(=O)Nc2ccc(C)cc2C)CCCC1P(C)(C)=O C(CNC(=O)CC1(OC)CC1)(C(=O)N1CC(n2ccnc2)C1)OC c1(C(N(C2CC(OC)C2)C)=O)c(C)[nH]c(-c2ccccc2)nc1=S n1(CCC)cc(Cl)c(C(=O)NC2CCCC2C(=O)OCCNC(C)=O)n1 c1(CN(C)C(c2cc(C(=O)Nc3ccns3)[nH]n2)=O)ccccc1 c1(-c2nc(C(C)C3CC3)nn2C2CCN(C)CC2)ccc(F)c2occc12 c1(C(=O)NCC=CCNC(C2C(C)C2C)=O)cc(F)c2ccccc2c1 C1(NC(CC=C(C)C)=O)CCOCC1NC(=O)CC1(O)CC1 C(=O)(C1=CC2CCC(C1)C2)N(CC(N1CC(C#CC)C1)=O)C c1(C(=O)NCC2(C(C)(C)O)CN(C(CC=CC)=O)C2)cc2c(s1)CCCNC2=O C(=O)(CCCC(=O)NC1CC(O)(CNC(=O)CC2(C)CCCO2)C1)N(CC)CC C1(NC(c2scc(C)c2C)=O)CN(C(c2ncsc2C(C)C)=O)CCC1CO C1(NC(C(COCC(C)C)F)=O)C2CC1N(C(C13CC(F)(C1)C3)=O)C2 Cc1cc(O)cc(=O)n1CC(N1CCCC1C(=O)NCCCCCO)=O C1(C(N2CC(CCNC(C(C)NC(C)=O)=O)C(C)C2)=O)CCC(F)(F)CC1 C1(NC(C(CC=C)(F)F)=O)CN(C(=O)Cn2cnnc2)C2(CCOCC2)C1 c1(CNC(C(=O)N(CC(C)(O)C(F)(F)F)C)=O)cccc2ccccc12 Cc1cc(Cl)ccc1C(O)C(=O)NCCCCCCn1cc(CCCC#N)nn1 N1(C(C2CCC(NC(CC(C(C)C)O)=O)C2)=O)CCC2CN(C)CCC12 CC(C)(CF)C(=O)NCC1CCC(CNC(=O)CCC(=O)C2CCCCC2)CC1 C(=O)(N=c1ccn(CCC2CCC(C(=O)NC)O2)[nH]1)C1C(C(=O)NC)OCC1 N1(C(CC(CC)C2CC2)=O)CCCCC(CNC(c2cccc([N+](=O)[O-])c2)=O)CC1 C(=O)(CC(C)C(C)(C)C)NC1(CCO)CN(C(c2c(CC)onc2C)=O)C1 Cc1cc(C(=O)NCC2(NC(c3cnc(O)o3)=O)CCCCCC2)c(F)cc1F C1(C(N2CCN(C(COCC(C)C)=O)CC2CCO)=O)CCn2ccnc2C1 N1(c2nnc(C#N)s2)CCN(CCNC(=O)CC2CCCCCO2)C(=O)C1 n1(CCN2CCCC(C3N(C(CC(CCC)O)=O)CCC3)C2)c([N+](=O)[O-])cnc1C N1(C(CC(OCC)OCC)=O)CCCC(F)(C(=O)NCc2cnns2)C1 C(=O)(CS(=O)(=O)c1ccccc1Cl)NCc1cn(C(C)C(N2CC(C)C(F)(F)C2)=O)nn1 N(C1CCCc2sc(Br)cc21)C(C=Cc1c(C)nn(C2CC2)c1Cl)=O c1(C(N2CCC(NC(C(CC)NC(N)=O)=O)C2)=O)cc(C)c(N)cn1 Cc1cc(F)sc1C(=O)NCC12COC(CNC(=O)CCc3nccn3C)(C1)C2 c1(C(=O)NC2CN(C(C3CCCC3)=O)C2)cc2c(Br)[nH]nc2s1 c1(C(=O)NCC2N(C(C(C)N(C)C)=O)CC=C2)cc2c(s1)CCCCCC2 c1(N2CCN(C(C)=O)CC2)nc2cccnc2c(=NCc2ccc(CSC)o2)[nH]1 C1(OC)CN(C(=O)CN2CCOCC2=O)CCC1NC(=O)CC1CCCN(C)C1 C1(C(=O)NCc2cccc(OC)c2)CN(CC2CC2c2ccc(F)cc2)CCC1O CC1CC(NC(=O)C=Cc2cncs2)CN(C(c2csc(C(C)(C)C)n2)=O)C1 Cc1ccc2cccnc2c1C(=O)NC1CC(CCNC(c2n[nH]cc2Cl)=O)C1 C(CC(C(C)(C)C)NC(=O)C(C)CC(C)C)N(C(c1nncc(OC)c1)=O)C C(C(C)(O)CC(=O)NCC(C)NC(=O)C(C(C)C)OCCc1ccccc1)OC N1(C(CN)=O)CCCC(O)(C#C)C1.C1(CC(=O)CC#C)CCOC1(C)C c1(OC)ccc(C(N2CCC(C3CCCN3C(c3cncc(O)c3)=O)C2)=O)cn1 N1(C(C)C)CCCCC1C(N1CCCC1(C)CNC(c1cccnc1)=O)=O c1(C(C(=O)NC(C#C)CC)NC(=O)C(CC)SC)c(C)cccc1Br N1(CCC(=O)NCc2scc(CNC(C3N(CC)CC3)=O)n2)C(=O)CCC1=O c1(OC)ccccc1C(CNC(=O)C(F)F)NC(c1csc(Cl)n1)=O C(=O)(C(C)(C)CCOC)NC(CNC(C1(COC)CCC(=O)N1)=O)C C=CC(CCC)CC(=O)N1CC(OCCC(=O)NCC(=O)N(CC)OC)C1 N1(C(c2cc(C)oc2)=O)CCCC(NC(=O)CCN2CCOCC2)CC1 c1(OC)nc(C(N2CC(NC(C3(C)CC(F)(F)C3)=O)C(O)C2)=O)sc1C C=CCCC(F)(F)C(=O)N1CCC(O)(Cn2cc(CC(O)C3CC3)nn2)C1 N1(C(CCCCC=C)=O)CCC2(C1)CN(C(=O)C=C1CCCC1)CC(C)O2 C1(OC)CN(C(C2CN3CCC2CC3)=O)C(C)(CNC(=O)Cc2cnc(C)o2)C1 c1(NC(=O)C(=O)NC2CCN(c3ncccn3)CC2)cccc(N2CCCC2)c1 c1(C(N2CCC(CC(N3CC(COC)OCC3)=O)C2)=O)nnc2ccccc2c1 C1(N(C(=O)NC(c2nccc(OC)c2)C)Cc2ccccc2)CC2(CCC2)C1O CC(C)C(C)(C)C(=O)NC(C)C=CC(=O)NCC(C)(C)OCCO C1(CN(C)C(c2cnc(C(C)(C)C)[nH]2)=O)CCCN(C(C2CC2CF)=O)C1 C1(C(=O)NC(c2cccnc2)C(C)C)CCc2nc(C3=COCCC3)sc2C1 c1(C(C)C)nc(NCC2CCCC2O)cc(=NCC2(n3ccnn3)CC2)[nH]1 CCC(C)(C(F)(F)F)NC(=O)CC(CNC(c1cccnc1S)=O)OC c12ccc(cc1)C(=O)N1CCC1CNC(=O)C2.C1(C(C)C)(CC)CC1NC(C)=O C(c1cnn(C)c1)=CC(=O)N(CC(CNC(C(Cc1c(C)nc[nH]1)O)=O)C)C CCCCC(C(=O)NC(C1CN(C(=O)COCC2CCCOC2)C1)C)C(C)C Nc1cc(Cl)ccc1C(=O)NC1CCCN(C(=O)C=CSc2ccccc2)CC1 N1(C(c2ccc(OC)s2)=O)CC(NC(c2c(Cl)cnn2C)=O)CC1C N1(C(CC(CC)CC)=O)CCCN(C(=O)CN2CC(=O)NC2=O)CC1CO N(C(=NCC(C)c1ccccc1Cl)NCc1cc(C)on1)Cc1c(OC)c(Cl)ccc1 C=CCCCC(=O)NC1CCC(NC(=O)C(C)Oc2ccc(F)nc2)CC1 c1(C(=O)NC(CNC(COCC=C)=O)CCCC)oc2ccccc2c1COC N(C1CCSc2ccccc21)NC(C)(Cc1ccccc1C(F)(F)F)CO C1(C(=O)NCc2ccc(C3CC3)nc2)CCn2ccnc2C1 CCC(CC)C(=O)N1CCOC(Cn2ccsc2=O)C1.n12cc(nn1)C2C1CC1 c1(CC(=O)NCC2(F)CN(C(=O)CC3CCC4(CCC4)O3)C2)ccc(O)c(Cl)c1 N1(C(C(CSC)C)=O)CCCC2(NC(c3cnc4[nH]nnc4c3)=O)CCCC12 C(=O)(Nn1cnn(C)c1=S)C1(NC(C(COC)C)=O)CCSC1 C1(NC(c2nc(Cl)cs2)=O)CCC2(CC1)CCN(C(C1CCCNS1(=O)=O)=O)CC2 C(=O)(C1=NN(C)C(=O)CC1)N(C1CCCCN(C(C2CC3CCC(C2)S3)=O)C1)C CCC(CCC(=O)N(C)CC1CN(C(=O)Cc2cocn2)CCO1)OC C1(C(=O)NC(C(CO)NC(Cc2ncc(C)o2)=O)C)(OC(C)C)CCOCC1 c1(C(=O)NCC2(F)CN(C(C(C(CC)O)(C)C)=O)C2)cc(F)c2cn[nH]c2c1 C(=O)(CCC1=CCCCC1)C(C(C(C)(C)C)CN)=O.N1CC2CC2C2CC12 O=C(C(F)C(F)(F)F)NCC1(F)CCC(NC(C2(CC3CC3)CC2)=O)C1 C(CN(C)C)(CC(C)C)NC(C1N(CC)CC1)=O.C1(C)CC(=O)N1 N1(c2nccc(NC(C(CCCC)O)=O)n2)CC2CC(CO)CC(C2)C1 C(=O)(C#CC1CCCC1)N1C(C)CCC(CNC(=O)Cc2cscn2)C1 CC1C(NC(=O)CNS(C)(=O)=O)CC2CCC1N2C(c1cc2ccc(Cl)cc2o1)=O N1(c2nnc(C)s2)CCCC2(CN(C(=O)CC(C)C(F)(F)F)CCO2)C1 C(=O)(CCNC(=O)C=C(C)C1CC1)NCCCOCCC(CC)C c1(OC)cc(OC(C#CC(=O)NC2CCOC2CNC)OC)cc(CCCO)c1.OC Cc1nc(C2CC2)[nH]c1C(=O)NCCC(C)NC(c1nc(C)c(C)[nH]1)=O N1(C(C(CCCC)O)=O)CCCC2CN(C(C3CCCCC3OC)=O)CCC12 c1(OC)ccsc1C(=O)NC1(CCO)CN(C(C2CC(N(C)C)C2)=O)C1 CCC(O)CC(=O)N1CCCC(CCNC(=O)CN2CCN(C)CC2)C1 C1(CN(c2cnn(C)n2)C)CCCN(C=O)C1.C1CCOC1 N1(C(C(C)OCC#C)=O)CC=CC1(C)C(=O)NCc1cncn1C N1(C(c2cc(CCC)nn2C)=O)CCCC(CO)(NC(c2coc(C#N)c2)=O)C1 C(=O)(C(CNC(=O)C(C)(C1CC1)OC)C(C)(C)C)NCC(CC)(C)C CC(CCC(C)(C)C)C(=O)NCCC(C)(C)CNC(C1C=CCCC1)=O CC(C(=O)NCC1CN(C(C2C3CC4C(C3)C24)=O)C1)C(F)(F)F C1(C(C)C)CN(C(=O)CCc2ccccc2)CCN1CCNc1cc(Cl)cs1 N1(C(C2C(OCC)CC2)=O)CC(C)(C)OCC1CNC(c1ncccc1O)=O N1(C(C2CC(CSC)C2)=O)CCN(CC(=O)OC)CC1.c12cccc(c1)CN2.C(C)C c1(-c2cn(CC(C)(C)O)nn2)nc(CCCO)nn1CC1CC2CCC1C2 C1(C(C(=O)NCCC(=C)C)F)CCN(C(c2cn(C(C)C)nn2)=O)C1 c1(C(=O)NC2CC3CN(C(CC(=C=C)C)=O)C(C2)C3)nc[nH]c2ncc(Br)c1-2 c1(CNc2c(C)nc(C3CCN(C(=O)OC(C)(C)C)C3)[nH]2)cnc2[nH]nnc2c1 N1(C(c2nn(C)c3c2CCC3)=O)CCC2CN(C(c3coc(O)n3)=O)CCC2C1 N1(C(c2ccc(C)cn2)=O)CC2CCC(C1)N(C(c1ccsc1C)=O)C2 C(C1=Nc2ccccc2S(=O)(=O)N1)CCOCCNC(C(C)C)=O C1(c2cn(CC=C)nn2)(NC(c2nnsc2Cn2cc(Br)cn2)=O)CCCOC1 N1(C(C(CCC)c2ccccc2)=O)CC(C(N2CC(O)C2)=O)C(F)(F)C1 C#CC1(C(N2CCC(C)(CC(=O)Nc3ccc(C(=O)OC)s3)C2)=O)CC(=O)C1 c1(C(=O)NCC(N(C(C(C2CC2)OCC)=O)C)C2CC2)cn(C2CCCCC2)nn1 C1(CNC(CN(C2CC2)CC)=O)CN(C(C2CCC3(CC3)C2)=O)CC1(F)F Cc1ncc(C(=O)NC(C)CC(C)NC(c2cccc(F)c2)=O)n1C N1(C(C(C)CF)=O)CCC2(CC1)CCN(C(C1CCCC1C)=O)C2 C(=O)(CC(C)(C)C1CC1)NCC#CCNC(c1cn(CCC=C)nn1)=O c1(C(=O)NC(c2cn3c(n2)SCC3)C)cc2ccccc2cn1 Cc1cc2nc(N3CCC(C)C3CNC(C3(C4CC4)CCC3)=O)cc(=O)n2o1 C1(C2CC2)OC(=O)NC1(C)C.C1(C(N2C(C)C(C=O)CC2)=O)CC(C)(C)CN1C C1(NC(C2CCCC(NC(C3(OC)CCSC3)=O)C2)=O)CNC(=O)C1(C)C Cc1ccc(C(=O)NC2CCC(NC(c3cccc(F)n3)=O)C2)c(F)c1F CCCCC(CNC(=O)CC1CC(C(F)F)C1)NC(C1(C)CC1C)=O Cc1ccc(C)c(C(=O)NC(C)(CNC(=O)CC2COC(=O)N2)C2CC2)n1 Cc1c(F)ccc(Cl)c1C(=O)NCC1CCN(C(=O)C(C)(C)C)C1 C1(C(=O)NCC(C)NC(=O)C(F)(F)c2cccnc2)CC=CCC1 c1(C(N2CCC(NC(C34CCC3CC4)=O)CC(O)C2)=O)cc(F)c(F)cc1O CC1(C)CCCCC1NC(=O)C(C)(CO)NC(=O)Cc1cccc(O)c1 C(=O)(C(COC)C(F)(F)F)NCC1(NC(C2CCN(CC)C2)=O)CCCC1 N1(C(CCc2n(C)ncn2)=O)CC2CC(NC(c3coc(Br)c3)=O)CC1C2 c1(OC)cc(Cl)c(Cl)cc1C(=O)NC1CC(F)(F)CC1NC(=O)CC1CCCO1 C=CCC(C)C(=O)NC(CO)C(=O)N(C(CCO)C(F)F)C1CC1 N1(Cc2cccc(CC)c2)CCc2c(Cl)cc(Cl)cc2C1C c1(CC(=O)NCC(=C)CCNC(C23CCC2C3)=O)ccc(F)cc1 c1(OC)cc(I)c(C(N2CC(C(=O)Nc3cc(Cl)sc3Cl)C2)=O)cc1OC C1(C(N(CCCC(C)C)CCO)=O)COC2(C1)CN(C(=O)C=CCF)C2 c1(CC2C(CCC)C2)ccc(OC(=O)CC(CC)SC)cc1 N1(C(COCC#C)=O)CCN(C(=O)CCCOC)CC1c1ccnc(N(C)C)n1 C1(C(N(C2CCN(OC)CC2)C)=O)CC2CCCC2N1C(c1ccc(N)cn1)=O C1(C(=O)NCCC2(C)CCOC2)CC12CCN(C(C1CNC(=O)O1)=O)CC2 C1(CC)CCCCCC1NC(NCP(C)(C)=O)=O N1(C(c2ccc(OCC)cc2)=O)CCN(C(c2ncc(Br)cc2Cl)=O)C(CC)C1 c1(C(C)(C)C)ccc(C(F)(F)F)nc1NC(=O)CC1SC(=N)NC1=O Oc1cnc(N(C2CC2)Cc2ncn(-c3ccccc3)n2)c(O)n1 c1(CSCC)cncc(C(=O)NCCC2COCCN2C(=O)CC2CCCOC2)n1 c1(C(=O)NCC(CCOC)NC(CSCC=C)=O)cn2cccnc2n1 C1(CCNC(C(C)(O)C2CCC2)=O)CCCCN1C(=O)CNS(N)(=O)=O N1(C(CCCCCC#N)=O)CCn2nc(CNC(c3cnsn3)=O)cc2C1 C1(c2ccon2)(CC(=O)NCCCN(C)C(C2(N(C)C)CC2)=O)CCC1 N1(C(CC)=O)CCN(C(c2cccc(-c3cnco3)c2)=O)C2CCCCC12 N1(C(c2c(C)ccn2C)=O)CCC2CC2(NC(=O)CCc2ccn(C)n2)CC1 N1(C(c2c(C)nn(C)c2C)=O)CC(C(=O)NCCCS(C)(=O)=O)C2(CCC2)C1 c1(C(N(CCNC(C(C=CC)O)=O)CC)=O)nnn2c1C(=O)NCC2 c1(NC(=O)NCC(=O)Nc2ccccc2)cccnc1Br C12(CNC(=O)Cc3ccsc3Br)CC1CN(C(c1cocn1)=O)C2 N1(OC(F)F)CCCC(C(=O)NCC)C1.C12CCC(CC1)NC1CC(C1)C(=O)N2 CC1CCc2c(NC(C3CN(c4nc(Cl)nc5c4COC5)CCO3)=O)csc2C1 C1(CN=[N+]=[N-])CCN(C(=O)CCNC(=O)CN2CSCC2=O)CC1 N1(C(C(C)OCC#C)=O)CCC(NC(=O)CC2CCOC2=O)C(C)C1 N1(C(c2cc(CC)on2)=O)CC2OCCN(C(c3cc4ccsc4n3C)=O)C2C1 c1(C(=O)NC(CC(C)NC(C2(NC(C)=O)CCC2)=O)C)c(C)cc(Cl)cc1N Cc1ccccc1C=CC(=O)NC1CC(C)N(C(c2cn(C)c(=O)cn2)=O)C1 C1(C(=O)OCC)CCN(C(C2CCCN2Cc2ccsc2)=O)CC1C c1(C(C)=O)cc(C(=O)N(CC(C)NC(C2CCC(=O)N2C)=O)C)c(C)o1 C=CC1CN(C(C2(c3cccnc3Cl)CC2)=O)CC1NC(=O)CNC(=O)COC C(=O)(CCCCC(=O)NCC1CC(C(=O)NCC(C)(C)CO)=NO1)OC N1(C(C2CCN(CC)C2)=O)CCC(CC(=O)Nc2cccc(C(C)=O)c2)C1CC c1(C(=O)NC(c2ccc(I)cc2)CC)ccccc1OCCc1ccc(Cl)cc1 Cc1c(C=CC(=O)N(CCCNC(c2conc2C2CC2)=O)C2CC2)cnn1C C(=O)(C(C)(C)CNC(c1ccn(CCC)n1)=O)N(C1CCCCC1)CC#C c1(C(=O)NCC(=O)N(CCCN(C(C2C(C)(COC)C2)=O)C)C)cc(C)no1 Cc1cnc(N)c(C(=O)NC2CC(C)(NC(c3ccc(C(F)(F)F)cn3)=O)C2)c1 c1(C(=O)NCC(C2CC2)OC)c(CNC(C2CCS2(=O)=O)=O)cnn1C Cc1ccc(C(=O)NCC2(C)CCN(C(c3c(C)nsc3C)=O)CC2)c(N)c1F c1(CN2CC3C(C(=O)NCCC)(C3)C2)ccc(C#N)cc1F Cc1cc(C(=O)NC(C)CCNC(c2cc(C3CCC3)[nH]n2)=O)ncc1C(F)F c1(OC(C)C)ccc2cc1-2.c1(CNC(c2occc2Br)=O)ccc(F)c(NC)c1 CCC(CNC(=O)CC(O)c1cn(-c2cnn(C3CCC3)c2)nn1)CC(F)(F)F c1(C(=O)NC2CCC(CNC(C(CC(C)C)O)=O)CC2)cn(C)c2ccccc12 C1(C2CCN(C(=O)C(C3CC3)OCC)C2)(NC(C=CCCC)=O)CC1 CC1=C(C(=O)N(CC(C)NC(c2ccc(Br)c(C)c2)=O)C)CCCC1 C1(OC(C)(C)C)CC(NCc2ncc(-c3cnn(CC(F)(F)F)c3)[nH]2)C12CCC2 C1(C(=O)NCC(CC)(C)NC(=O)C=Cc2cc[nH]n2)CCCC(=O)N1 c1(C(=O)NCC(CN(C(=O)CCF)C)O)c(S(N)(=O)=O)ncn1C C12(C(N3CCC(F)(CNC(=O)CCCCc4cnc[nH]4)C3)=O)CCCC1C2(F)F C(=O)(C1=CCOCC1)NCC1C(C)CN(C(=O)CC2CCC(C)O2)C1 N1(C(CC2CN(C)C2)=O)CCC(C2CC2NC(=O)C=Cc2cocn2)CC1 C(CCCC(=O)N(C)CC1OCCC1C)NC(C1(COC)CC1)=O C(=O)(C(C(C)CC)N(C(=O)C(C(C)(C)C)N(C)C)C)NCCN(CCC)CCC CC1(C)C(NC(=O)C(F)n2ccnc2)C(C)(C)C1NC(=O)CCc1ccoc1 C(CC(=O)NC1(C)CCCCCC1)(C(F)F)NC(C1CC(CN(C)CC)C1)=O C(=O)(C(C(C)(C)O)NC(=O)C(C)C1(O)CCC1)NC(CCC)CCO c1(C(N2CCN(C(Cc3n(C)ccc3)=O)CC2CCO)=O)[nH]nc([N+](=O)[O-])c1Cl C12(C(=O)NC(C)C(C)NC(C3CCCCN3N=O)=O)CC(C)(C1)OC2(C)C N1(c2ncnc(C)c2Br)CC23CCCC2(CN(C(=O)CC(C)CN(C)C)C3)C1 C(C(C)N=c1ccnc(N2CCC(F)(CO)CC2)[nH]1)N(CC)CC N1(C(C2(C)CCCC2)=O)CC2CCN(C(=O)C(=O)Cc3cccc(Cl)c3)C(C2)C1 C1(C(=O)NCC(=O)Nc2scnc2C(F)(F)F)COCCN1C(c1nocc1Cl)=O C1(C(N2CC(CC)C(NC(c3cc(CO)oc3C)=O)C2)=O)CCOCC1(C)C C(CNC(=O)CC(C)c1ccccc1)(CCNC(=O)CCc1cnn(C)c1)OC c1(CNCC2N(C(c3cc(Cl)c(Cl)cn3)=O)CCC2)c(Cl)ccnc1Cl C1(NC(CC2CCC(OC)CC2)=O)CC(F)CN(C(=O)CN2CCCNC2=O)C1 C(=O)(CN=c1[nH]c(N2CCN(C)C(c3ncc[nH]3)C2)nc2c1CCCC2)NC C1(C(=O)NCC(CNC(c2cnsc2C)=O)OC)(CC)CCCCO1 N1(C(C2C(C)(C)C2(C)C)=O)CC2CC(C(=O)NCCCO)(C2)C1 c1(CC(N2CC3CC3(CNCc3nccc(C(F)(F)F)n3)C2)=O)cccc(Cl)c1 Cc1ccc(C(=O)NC(CNC(=O)Cn2cc(C3CC3)cn2)C2CCC2)nc1C C12(CNC(c3c(SC)ccs3)=O)CC1CN(C(=O)C(C)(C)O)C2 C1(C)(NC(C(CC)F)=O)CCN(C(c2ccc(OC(C)=O)c(OC)c2)=O)CC1 c1(N(C)Cc2scc(C)c2)[nH]c(=NCCCn2cnnc2)nc2sccc12 c1(OC)ccc(S(=O)(=O)F)cc1N(C1CCC1)Cc1ccccc1 N1(C(C(=O)NC(C)C)=O)CC2OCC(C(N3CCC(O)C(CO)C3)=O)C2C1 C1(COC)(NC(=O)CCn2cnnn2)CCCN(C(=O)CC2CC=CC2)C1 c1(C(=O)NCC2(F)CN(C(c3c(CC)n[nH]c3)=O)C2)cc2c(C)ccc(F)c2[nH]1 CC1(C)CCCC1(C)NC(C1CCCC(NC(c2nocc2Cl)=O)CC1)=O Cc1n[nH]c(C)c1CNC(C1CCN(C(=O)C(F)CC2CCOC2)C1C(C)C)=O C1(CNC(C(C)(C)OC(C)=O)=O)CC(NC(C2CC3CC2C3)=O)C12CCC2 N1(C(C(CC#C)C)=O)C(C)C2CC1C2NC(=O)Cc1ccc(Cl)c(F)c1 C1(C(=O)NCC(CCCC)NC(=O)COCCOCCO)CC(C2CC2)=NO1 Cc1ccc(CC(=O)N(CC(O)CN(C)C(C2CCCCC2(F)F)=O)C)c(Cl)n1 C1(NC(c2cccc(OC(F)F)c2)=O)CN(C(=O)CCc2nncs2)CCC1CO c1(C(=O)NC2CCN(C(c3c[nH]nc3OC(F)F)=O)C2)cnc2ncccc2c1 C(=O)(C(O)C(F)(F)F)NC1CC(NC(Cc2nc(=N)[nH][nH]2)=O)C1 c1(CNC(c2cncc(C)n2)=O)cc2n(n1)CCN(C(C1CC3(CC3)CO1)=O)C2 C1(CNC(C2(OC)CCCCC2)=O)CCN(C(C2CCC(C)(CC)O2)=O)CC1O Cc1[nH]nc2c1CCC(NC(c1cccc3ccccc13)C)C2 N1(C(c2c(C)sc(O)n2)=O)CC(O)(C2(CNC(C3C4CCCCCC34)=O)CC2)C1 c1(OC)ccc2c(c1)CCCC2c1noc(-c2csnc2-c2cccc(OC)c2)n1 CS(=O)(=O)c1ccc(CC(=O)NCC2(F)CCN(C(c3cc(Cl)no3)=O)C2)cc1 C1(C(N2CCC(NC(COCCCCC)=O)C2(C)C)=O)CCc2cnnn2C1 c1(CCC)ccc(C(=O)NCc2ccoc2C(=O)NCC2(CC3CC3)CCC2)[nH]1 c1(C(=O)NC(C(C)NC(C(COC)(F)F)=O)CO)c(F)cc(C(F)(F)F)cc1F C1(NC(=O)C=CC2CC2)CCCC(NC(c2ccc(-c3ccccc3)cc2)=O)C1 N1(C(C2CN(OC)C2)=O)CC(C(N2CC3(CC(F)C3)C2)=O)C2(CC2)C1 CC1=CC2=C(C=N2)CN(C(c2cn3cc(Br)ccc3n2)C(=O)NCC2CC2)C1 C=Cc1ccc(C(N2C(C(=O)NCCOCC3CCCC3)CC2C)=O)cc1 CC(C)C(C)(O)C(=O)NC1CN(c2nnc(C3CC3)s2)CCC1C Cc1cccc(O)c1CNC(C1CC2CC(=O)C1C2)=O CC(C)(C)C(C#N)C(=O)NCC(O)CNC(=O)CC1CCC1(F)F CC1c2ccccc2CCN1C(=O)C(c1cccc(Cl)c1F)(F)F c1(COC)nc(NCC2(C)CCOCC2)cc(=NC2CCC3CCC23)[nH]1 C(=O)(C1=NOC(C)C1)NCCN1CCC(NC(C(CCC)=CC)=O)CC1 C1(F)(C(=O)NCCCN(C(c2ccc(C(C)=O)cc2)=O)CC)CCOCC1 n12nccc1C2.N1(CC)CCC1C(=O)N(CCCN(C(=O)CO)C)C c1(C(N(C2CCN(C(C3(F)CCOC3C)=O)C2)C)=O)ccc(C(O)CF)cc1 C1(C)(C(=O)NCCC2(O)CCN(C(C3C(C)OCC3)=O)CC2)CC2CCC(C1)S2 C12(CC(=O)NC3(CO)CN(C(=O)CNS(C)(=O)=O)C3)CCCC1C2 C1(C(N2CCC(O)(CC(=O)NC3C(C)(C)C3(C)C)C2)=O)CC2C(C1)C2(C)C Cc1ccc(CNC(=O)NCC2CCC2NC(C2CCN(CC(F)F)CC2)=O)cc1 CC1CN(C(=O)C(=Cc2c[nH]cn2)F)CCCN1C(=O)C=CCN1CCCC1 C1(NC(=O)OC(C)(C)C)CC(O)CN(C(C2(C#N)CC2C(F)(F)F)=O)C1 c1(OCC(=O)NC2CN(C(=O)CC(C3CC3)C3CC3)CC23CC3)ccc(Cl)c(Cl)c1 N1(C(C(CC=CC)C)=O)CC(NC(=O)Cc2cncs2)C(C2CC2)C1 C12CCCN(C1)C2.c1(N(C(C(=O)NC2CC2)=O)Cc2cccs2)cccc(Br)c1 C(=O)(C(CC(F)F)N(C(=O)CC1CCCNC1=O)C)NCC1C(C)OCC1 c1(C(N(CC(C)NC(=O)CC(F)(F)C(F)F)C)=O)cc(O)ccc1[N+](=O)[O-] CN1C(=O)C(=O)N(CC(=O)NCCCCCNC(C2CC3CCC2CC3)=O)C1=O CC1(C)C(C)(C(=O)NC2CCCCN(C(c3cn(C4CC4)nn3)=O)C2)C1(C)C c1(C(N2CC(NC(C3(NC(=O)OCC)CCO3)=O)C2)=O)cnc2n1CCC(C)C2 C(=O)(CC(F)(F)CC(=O)N(C1CCCN(C(C2CCCN(C(C)=O)C2)=O)C1)C)OC N1(C(C2N(C(c3cc(COC)on3)=O)C(C)CC2)=O)CCCC(F)(F)C1 c1(CCN(C(c2ccc(Cl)c(-c3nn[nH]n3)c2)=O)CC)cc2ccccc2[nH]1 N1(C(C(C)=C2CC2)=O)CCC(C(=O)NCCC(C)(O)C2CC2)C12CC2 N1(C(c2nc(CCC)sc2)=O)CC2CC1CCC2NC(=O)C=C1CC(C(C)C)C1 CCC(CN(C)C)CC(=O)NCC1(O)CC(C(=O)N(C2CCN(C)C2)C)C1 C1(N(C)C(C23CCC(CO2)C3)=O)CCCCN(C(=O)C=Cc2cncs2)C1 C(=O)(C(F)(F)C(F)F)N1CCCC(C(C)NC(c2cc(C)nnc2)=O)C1 Cc1nc(C(=O)NC2CN(c3nc(Cl)c(C#N)s3)CC2(C)C)ccc1C#N c1(C(=O)OC)cccc(NC(C2(NC(C3CCCCCC3)=O)COC2)=O)n1 c1(C(=O)O)ncnc2sccc12.C1(CN)COCCN(C(c2cccc(Cl)c2F)=O)C1 C1(CNC(C=C(CCC)C)=O)CCCC12CCN(C(C1OCCCO1)=O)CC2 C(C(C(=O)NC1(CN(C)C)CC1)C(C)C)NC(C1N(CC)CCC1)=O C1(C(=O)NC(CCCC)CNC(c2ccnnc2C)=O)CCCC2(C1)CC2(F)F C(=O)(CC(O)C(Cl)(Cl)Cl)NCC1CCCN(C(c2nc(C(C)=O)sc2)=O)C1 C1(CNC(CC(=O)N(CC)CC)=O)CC2CN(C(=O)CN3C(C)CCCC3C)CC12 Nc1ccc(C(=O)NCCC(O)CNC(=O)CCF)cc1N1CCCCC1 CCCCCS(=O)(=O)CC(=O)N1CC(NC(=O)C(c2cncn2C)O)C2CC2C1 S(=O)(=O)(C1CC2C1C2(F)F)NC(c1cccc(OCCOCC)c1)=O C1(C)(CC)C=C(C(=O)NC2CN(C(=O)Cn3cnc(C(N)=O)n3)CC2C)C1 N#CC1(CC(N2CC3C(CNC(c4ccn(CCF)n4)=O)C3C2)=O)CCCCC1 C1(CNC(c2cscn2)=O)CN(C(C2CC23CCOCC3)=O)CCC12CCC2 N1(C2CCN(C(C3(CNC(=O)Cc4ncc(C)s4)CC3)=O)C2)CCN(CC)CC1 c1(C(=O)NC(C2CCN(C(C3CC4C(C3)C4(C)C)=O)C2)C)cc2n(n1)CCCC2 C(=O)(CCCCCNC(c1nnnn1C(C)(C)C)(C)CC1CCC1)NC Cc1ccc(NC)nc1.CCS(C)(=O)=O CC1CCCN(C(C2CC=CC2)=O)C1CNC(C1C2CCCCC12)=O C(=O)(C(c1cccs1)=Cc1ccco1)NCC1(OC)CNC1 C1(=CCNC(C(C)c2ccon2)=O)CCN(C(c2cc(N(C)C)ccn2)=O)CC1 N1(C(CC(CC)OC)=O)CCCC(C)(NC(=O)CC(C)(C)c2cnsc2)C1 C1(NC(C(C)=C(C)C)=O)CC2(C1)CC(NC(c1cc(O)n(C)n1)=O)C2 c1(CC)ccc(C)cc1NC(=O)CCCCC1CCCCN1c1ncncc1C c1(CC(=O)NC23CC2CN(C(=O)C=Cc2ccco2)C3)cn2cc(F)ccc2n1 C1(NC(CC2(N(C)C)CC2)=O)CCCN(C(c2ccnn2-c2ccncc2)=O)C1 C(=O)(CC(C)C(C)C(C)C)N1CCC(C(c2nc(OC)cc(OC)n2)CC)C1 c1(C(N2C(C3(NC(c4n(CC)ccn4)=O)CC3)CCC2)=O)ccc(O)cn1 C(=O)(C(F)(F)C(O)CC)NCC1CC(NC(C2(C=C)CCCCC2)=O)C1 N1(C(c2cc(CC)c(C)s2)=O)CCCCC(NC(c2sccc2Cl)=O)C1 CC1CCC(NS(C)(=O)=O)CC1C.N12CC(C)(C1)NC1(CC1)CNC2=O c1(C(N2CCC3(C(N4CCC(=C)CC4)=O)C(C2)C3)=O)ccc(Br)c2cccnc12 Cn1nc(C2CCCCC2)cc1NC(=O)C(=O)NC1CCNCC1F C1(NC(c2[nH]cc(C(C)=O)c2)=O)CN(C(=O)C(C)(C)NS(C)(=O)=O)CC1(C)C C(=O)(CS(=O)(=O)N(C)C)NC1(C)CC(NC(C(C)NC(C)=O)=O)C1 C1(C(=O)OC)C(F)(F)C12CC(C(N1CC(NC(=O)Cn3nccn3)CC(F)C1)=O)C2 N1(CCC(=O)NC(CCCC2(OC3CNC3)CC2)=O)CCCCC1C.C=CCCO Cc1cc(C#N)nc(N2CCCC2CC(=O)Nc2nc(C)ncc2Br)n1 c1(C(N2C(CCNC(c3cc(C)c(C)s3)=O)CCC2)=O)cc[nH]c(=N)c1N C(c1ccccc1C(F)(F)F)=CC(N1CCC(N(C(C(CC)OC)=O)C)C1)=O C(CCN(C)C)(C(=O)N(C)CC1CCSC1)NC(Cc1c(C)con1)=O c1(C(N2CCCC(C)(CNC(CCC(C)C#N)=O)C2)=O)cccc2[nH]cc(Cl)c12 C=C1CCC(C(=O)NC2(C)CCN(C(=O)CC3CC4(CC4)CO3)C2)CC1 c1(C(=O)NCC2CN(C(c3cc[nH]n3)=O)C2)cnc(C2CCC2)o1.C1CC1 C=CCCCCC(=O)N1CCC(C(C)(C)C)CC1CNC(=O)CSC(C)(C)C N1(C(C(C)SCC)=O)CC2CN(C(=O)CCCCNC(N)=O)CC2C1 N1(C(c2occ(C)c2C)=O)CCCC(C)C1CNC(c1sccc1CN(C)C)=O n1(CC(=O)NC2C3CCN(C(c4cnc(N(C)C)s4)=O)C32)cc2ccccc2n1 N1(C(C(C(C)C)OC)=O)Cc2n[nH]cc2C1C(=O)N1CC(C2=NOCC2)C1 C1(CSC)CN(C(=O)CCCCC2CC2)CCN1C(=O)C=CC(C)(C)SC C(=O)(C1=CC2CCCCCC12)NCCN(C(c1c(C#N)scc1)=O)CC1CC1 CCC(C)C(C)(O)CNC(=O)CC1CN(C(=O)C(C)(C)N2CCCCC2)CCO1 c1(C(C(N2CCC(CN(c3ncc(C)cn3)C)CC2)=O)C)nc(F)ccc1Cl n1(CCC)ncc(CN2CCCCC2CNC(C2CCOC2C)=O)c1C N1(C(c2cc(N(C)C)ncc2)=O)CCCC(C)(C)C1CNC(C1CCS1(=O)=O)=O O=C(C1c2ccccc2CN1C(c1cccc(F)n1)=O)Nc1cnn(C2CC2)c1 c1(C(CCC=C)(c2nnnn2CC(F)F)Nc2ccncc2)ccc(F)cc1F C1(C(=O)NCC2CN(C(C3N(C(C)=O)CCOC3)=O)C2)CCCCC12CC2 N1(CC)CC(CNC(=O)CN(C(c2n[nH]cc2CC2CC2)=O)C(C)C)CC1=O CCC(CC)(CO)C(=O)N1CCCC(N(C(=O)Cc2cnc[nH]2)C)C1 C=CC1CN(C(=O)CCC(=O)OC(C)(C)C)CC1NC(=O)C=CC(C)(C)SC N1(C(c2ccoc2Br)=O)CCC(C(C)NC(=O)C(C2CCCCC2)N(C)C)CC1 c1(NC2CC(F)(NCC(=O)NC(=O)CC3C=CCC3)C2)ccccc1[N+](=O)[O-] C1(C(=O)NC(c2noc(C)n2)CC)CCCN1NC(=O)c1ccnn1CC N1(C(C2C(NC(CCc3nc(=N)[nH][nH]3)=O)CC=CC2)=O)CC2(CNC(=O)N2)C1 N1(C(c2cc(CCC)on2)=O)CCC(F)(C(=O)NC2(C3CCCO3)CC2)C1 c1(CC(=O)NC2CC(NC(C3C(OC)CCC3)=O)C2)sc(C2CCC2)nc1C Cc1nnc(C(=O)N(C2CC(NC(c3cc(Cn4cccn4)on3)=O)C2)C)s1 C(=O)(C1COc2ccccc21)NCC(CNC(c1c(C)noc1C)=O)S(C)(=O)=O Cc1ccc2cc(C(N3CCCC(NC(=O)Cc4ncc(C)o4)CC3)=O)cn2c1 C(=O)(CS(=O)c1ccc(Cl)cc1)NCC(CC)NC(=O)CC1CC(C)(C)C1 c1(C(N(CCCN(C(C=C(C)C2CC2)=O)C)C)=O)cc(C2CCCC2)nn1C C1(NC(C(c2ccccc2)OC)=O)C(C)(C)CN(C(C2(C)CC2F)=O)CC1(C)C C1(NC(CCCC(CNC(=O)OC(C)(C)C)O)=O)CC2CC1CC21OCCO1 c1(CNC(C2(NC(CC3N(C(C)=O)CCC3)=O)CCSC2)=O)ccc(C)cc1 N1(C(=O)CCN2CCCS2(=O)=O)CCN(C(c2ccc(Cl)s2)=O)C2(CC2)C1 C(=O)(CC(C)(C)CC)NC1CCN(C(c2c(CC)cccc2)=O)C1C O=Cc1sc(CN2CC3C(C2)N3C(=O)C=CCBr)c(Br)c1Br c1(C(N2CC(OCCF)CC(O)C2)=O)cc(Cl)c2[nH]c(-c3ccco3)nc2c1 C(CN=C(NCC(F)F)NCC(O)(C1CC1)C1CC1)c1cnc(OC)nc1 N1(C(C2N(C(C)C)CCCC2)=O)CCC(NC(C2C3CC4C(C3=O)C24)=O)C12CC2 O=C(CN=C(NC1CC1)NC1CC(c2ccc(Cl)cc2)C1)N1CCCC1 c1(CCC)cc(C(=O)N(C2CCCCC2N(C(=O)CC(C)(F)F)C)C)c(C)o1 c1(COCC(=O)NCCC(C)(C)NC(=O)CS(N)(=O)=O)ccc(F)cc1Cl C1(CNC(COC2CN(C(C)=O)C2)=O)CN(C(=O)Cc2cc(C3CC3)no2)CC1C c1(SC)cc(C(=O)NC2C3CC2N(C(=O)CSc2cccc(Cl)c2)C3)ccc1F N1(C(C(=O)Nc2ccnc(-c3ccccc3)n2)=O)CCCC(F)(F)CC1 C1(CNC(c2coc3c2CSC3)=O)CCCCN(C(C2CC2(Cl)Cl)=O)C1 c1(C(CNCCCOC)OC)cccc(Br)c1Cl N1(C(C=C(C)C(F)F)=O)CCC(C(=O)NCc2ccncn2)C(O)C1 c1(CC)noc(CC)c1CC(=O)NCC1(NC(C2CC(=O)N(C)C2)=O)CCOC1 c1(CC(C)C)c(C(=O)NC2C3CN(C(=O)CCCC#N)CC23)cnn1C CC1COc2c(C(N3CCC(NC(c4ccnnc4Cl)=O)CC3C)=O)cccc21 C1(F)(CNC(C(CN(CC)CC)F)=O)CCCN(C(c2scc(C)c2Cl)=O)C1 N1(C(C(C)c2cccs2)=O)CCOCC1C(=O)NCC(C)(C)C1(O)CCC1 C1(NC(c2ncn(C(C)(C)C)c2)=O)CC(C2CCN(C(c3cnsc3)=O)C2)C1 c1(C(=O)NCC2CC(NC(c3ccccc3SC(F)F)=O)C2)ccc(O)nn1 C(=O)(C(C)CC(F)F)NCCc1c(CNC(Cc2cncc(C)c2)=O)nco1 c1(C(=O)OC)cn(CC(=O)Nc2ccc3c(c2)c(C)nn3C)c(C)c(Br)c1=O C1(C(N2CCN(C(C3C4NC(=O)C(CC4)C3)=O)CC2)=O)CCc2nnc(O)cc2C1 CC(C)CC(CNC(C12CC(C)C1C2)=O)NC(C1COCCN1CC(F)F)=O c1(OC)cc(O)cc(OC)c1CN1CCC(C(=O)Nc2ccc(Cl)c(Br)c2Cl)C1 c1(C(N(CCN(C(C2(C=C)CCC2)=O)CC)CC)=O)ccc(F)c(N)c1 C(=O)(C(O)CNC(=O)CN1CCOC1=O)N1C(C)CC1 N1(C(CN(C)CC)=O)CCCC2CN(C(c3cc(C)c(C)o3)=O)CCC12 N1(C(CC(=C)Br)=O)CC(CC2CCCCC2)C(C(=O)N(C)C)C1 CC(C)(C)CC(=O)NCCC1CCCN1C(c1cnn(CC(F)(F)F)n1)=O C=C(Cl)C(C)(C)C(=O)N1CCN(C(=O)C#CC(=O)N(C)C)CC1 CCS(=O)CC(=O)NC1CC1NC(C1(N(C)C)CCCC1)=O Cn1nc(C(=O)NCC23CC(NC(=O)CSc4nncs4)(C2)C3)c2cc(F)ccc12 N1(C(C2C(CC)CCO2)=O)CCC(C(C)(C)C)(CNC(=O)C(C)n2ccnc2)C1 C(=O)(C(C)(C)C(F)F)N1CCCC1.CN1CCN(CCOCCN)CC1 c1(C(=O)NCC=CCCCN2CC3CC3C2)cn(CC(=O)N(C)C)nn1 N1(CC(c2ccccc2)C)CCN(C2CCN(C(=O)NC3CC3C3CC3)C2)CC1 C12(C(=O)NCCC(=O)N(C)C)CCCC1CN(C(=O)CCc1cncn1C)C2 c1(-c2n(CCCC)nc(C3CCCO3)n2)cnc(C2(CO)CC2)nc1O Cc1c(C(=O)N(C2CCCC(NC(c3occc3C3CC3)=O)C2)C)cnn1C C(C(=O)N1CC2CC2(C(N2CC(C)(C)C2COC)=O)C1)(C(C)C)SCC C1(NC(C(C=C)CC)=O)CC(C)CN(C(=O)C(c2ccc(C)s2)C)C1 C(=O)(CC(C(C)(C)C)NC(=O)CCOCCOC)N1C(C(=O)OC)C(C)CC1 CCCC(CCC)C(=O)N1CCC(NC(c2ccc(C(C)C)o2)=O)C1C(C)C C(Cn1cccn1)(C(=O)NCc1cnsc1)NC(CC1C(CC)C1)=O N1(C(c2ccc(NC(C)C)cc2)=O)CCc2nc(S)[nH]c2C1 C(CC(=O)N(CC(C)CNC(c1cnns1)=O)C)SCCCC N1(C(C(CC=C)N(C)C)=O)CC2(CNC(=O)C=Cc3ccccn3)CCC1CC2 N1(C(CCOC(CC(C)C)C)=O)CC2CN(C(=O)CC(C)(C)C)CC(C1)O2 CC1(C(N2CC=CC(NC(=O)CSCC3CCCO3)C2)=O)CCCCO1 N1(C(c2ccn(C)n2)=O)C(C(=O)NC2CCS(=O)(=O)C2)CC2CC12 C=CC(C)(C)CCCNC(=O)C(c1c(C)cccc1Br)NC(=O)C(C)OCOC Cc1cnsc1C(N1CCC(CNC(=O)Cc2c[nH]nc2O)C1)=O C1(C(C)NC(COCC)=O)CC2CCC(C1)N2C(c1cccc(Cl)c1N)=O C1(CNC(c2c[nH]nc2-c2cccs2)=O)CN(C(c2ncccc2F)=O)CCO1 C(=O)(C(Cc1cn[nH]c1)NC(=O)CCc1ccoc1)OC N1(C(c2nnn(C)n2)=O)C(CNC(=O)C(c2ccccc2Cl)O)CC2COCC12 CCC(CCc1ccccc1)C(=O)NC1CCCC1NC(C1(CO)CC1)=O c12c(cnn1C)NC(=O)C(C)N(CC)C2=O.c1(C(=O)NC)cnc(Cl)s1 Cc1ccc(CN(C(c2c(C)n[nH]c2C)C(=O)NCC2CCCO2)C)cc1Cl c1(OCC=C)ccc(CN2CCCC2C(=O)NCCc2nn[nH]n2)cc1 N1(C(C(C)SC)=O)CC2CC2(CNC(c2cccc(-c3nnc(O)n3C)c2)=O)C1 Cc1sc(=O)n(CC(N2CC(N)CC(O)C2)=O)c1C Cc1cncc(C)c1C(N1CC2CC2(CNC(=O)CCc2cnccn2)C1)=O c1(C(=O)OC)c(C(=O)NCC(C2CC2)NC(=O)C(F)=C2CCCC2)n[nH]c1C c1(C(=O)NC2CCCC(NC(c3ncn(CC)c3)=O)C2)c[nH]c2c(F)cccc12 c1(C(C(=O)NCC2CCOC2)N(c2occc2C)CCOC)cn(C)nc1C CCC(C)C(C(=O)N1CSCC1C(N1CCC(N(C(=O)CC)C)C1)=O)NC(C)=O c1(N2CCN(CC)C(C)(C)C2)nc(N2CCC(CSC(F)F)C2)nc2c1COC2 Cn1nc2c(c1C(=O)NCC1(C)CCCN1C(C1C3COCC13)=O)CSCC2 c1(CC)cc(C(=O)N(C(C)CN(C(=O)CSc2c(C)n[nH]c2C)C)C)cc(F)c1 C1(C(=O)NC2CCN(CCC)C2)CN(C(=O)C(C2CCCCC2)=O)C(C)(C)C1 C1(OC)CN(C(=O)Nc2ccc(C(F)(F)F)cc2)CC1CC(C)(C)C C1(C(N(C)CC2(O)CN(C(c3nc(CCC)oc3)=O)C2)=O)(C(F)F)CCOCC1 C(CC(C)C)(C(=O)NC(CNC(=O)C(c1ncccc1F)(F)F)C1CC1)NC(C)=O C1(CNC(C2CCC(F)(F)C2)=O)C2CCC(C2)N1C(c1ccc(C(F)F)cc1)=O C1(NC(c2[nH]n(C)c(=O)n2)=O)CN(C(C2(C)CCCOC2)=O)CCC12CCC2 N1(C(C(CNC(C2(O)CCC(C)CC2)=O)O)=O)CCCC2CC1C2(C)C c1(NC(C=C)C)nc(N(C)CC)nc2sccc12 CC(CNC(c1occc1F)=O)C(=O)N1CC(NC(C2CCCC2)=O)C1 C=CCC(C)(C)C(=O)NCC1CN(C(C2CC(C)(O)C2)=O)CCO1 CN1CCCC1(C)C(=O)NCC1(C)CCOC1.c1(NC(=O)CCO)ccccc1Cl C1(C(N(C(C)CNOC(C)=O)CC)=O)CC(C)N1C(c1cc[nH]c1C)=O Cc1c(C)c(C)c(C(=O)NC(CNC(=O)COc2ccon2)C2CC2)c(C)c1C c1(CCNC(C(C)C(=O)c2ccccc2)=O)ccc(Cl)c(F)c1 C1(NC(=O)CC(F)F)CC2CN(C(c3cc(C(F)(F)F)no3)=O)CC2C1 C(=O)(C(C(C)C)C(=O)OC)N(C)C1CC1.c12cc(on1)C(=O)N1CC(C1)CS2 CC(C)C(C)NC(=O)NC(C)CCn1cncn1 C12(C(=O)OC)CCOCC1CN(Cc1cccc(CC(=O)OC)c1Br)C2 CC1(C)C(NC(=O)Cc2sccc2Cl)CC1C(=O)NC1(CO)CCCCC1 N1(C(c2[nH]cc(C)c2)=O)CC(NC(C2CC(CN(C)C)C2)=O)C2(CC2)C1 c1(C(=O)OC)cnc(NC(C2CNCCN2Cc2cc(Cl)nc(Cl)c2)=O)c(I)c1 CCCCCC(O)C(=O)NCC(C)(C)CC(=O)N1CCCCC1C(O)CO N1(C(C2OCC(C)C2)=O)CCC(F)(CNC(c2cc(C(C)(C)C)n(C)n2)=O)CC1 c1(N2CC(NC(c3nc(SC)[nH]c(=N)c3)=O)C(C)C2)ccccc1[N+](=O)[O-] c1(C(=O)NCC(C)NC(CC(=C)C)=O)cc2ccccc2n1CC(=O)NC N1(C(CCCN(C(C(CC=C)C)=O)C)=O)CC2CCC(NC(=O)C3CC3)C2C1 c1(OC)cccc(F)c1C(N1CC(O)(C(C)NC(=O)C(C)O)C1)=O c1(CC)ccc(C(=O)NCC2(CNC(c3ncccc3C)=O)CCC2)cc1 C12(CCN(C(=O)CCNC(=O)C3CC3)C1)C(=O)N2.C1(CC)CC2C=CC1C2 C(=O)(C(F)(F)C(F)F)NCc1nc(CNC(CC2OCC(C)(C)C2)=O)sc1 C1(C(N2C(C)(C)C(CO)C2)=O)CCN(C(c2ccsc2)=O)C1(C)C C1(NC(C(CC)OCC)=O)CC2CCC1CN2C(=O)C(SC)SC C1(S(C)(=O)=O)(C(N2CCC(=CCNC(C(C3CCCO3)OC)=O)CC2)=O)CCC1 C1(NC(C2(C#N)CCCC2)=O)CCCCCN(C(=O)CC2CCCC2O)C1 c1(C(N2CCC(OC)CC2)=O)c(F)cc(Cl)cc1Br.N12CCC(F)(F)C(C1)C2=O C(N1CCOCC2(COCC3CCCCN23)C1)N1CCn2c(cc(C)n2)C1=O c1(C(=O)NCC2CC(OC)CN2C(=O)C=Cc2cnc[nH]2)n[nH]c2c1CCSC2 CCCS(=O)(=O)C(C)C(=O)N1CCCN(c2cccc(F)c2)CC1 c1(CC(C)NC(C2CCC(CNC(c3ccc(CC)o3)=O)C2)=O)ccc(C)cc1 C12CN(CC13CC3)C2=O.C1(C(=O)NCC2(C(=O)OCC)CCC2)CCC2CC12 Cc1ncc(C(N2CCCC(CNC(c3ccc(O)cc3)=O)C2)=O)n1C c1(C(=O)NC2(CO)CCCN(C(CN(C)C)=O)C2)cc2c(nc1O)CCCCC2 C1(NC(C=CC(=O)OCC)=O)(COC)CCCN(C(c2ccc(F)cc2F)=O)C1 CCC(CC)C(C)C(=O)N1CC(O)CC1CNC(=O)CC1(NC(C)=O)CC1 C1(C(N2CCC(C)(NC(=O)C3=COCC3)C2)=O)CCNc2ccccc2C1 C12(CNC(COCCC=C)=O)CCCC1N(C(c1ccon1)=O)CCC2 Cc1cccc(C(=O)NCC(N2CCN(c3ncc(F)cn3)CC2)=O)c1 c1(C(=O)NCC2CC3CCC2N3C(c2ccsn2)=O)cnn2c1OCC1(CC1)C2 N1(C(CC(CC)(F)F)=O)CC(NC(c2ccc(Cl)cc2C(F)F)=O)C(C2CC2)C1 C#Cc1ccc(C(N2CC(O)(CCNC(c3cnc(C(C)C)s3)=O)C2)=O)cc1Cl S(=O)(=O)(c1cc(C(F)(F)F)co1)NC(C)(C)C.C12CCC(O1)CNC2=O C(=O)(C(COC)COC)NC1CCC(CCC(=O)NCC(C#C)CC)C1 N1(C(CC(C)n2ccnc2)=O)CC2CCC1CN2C(c1n[nH]cc1[N+](=O)[O-])=O c1(C(=O)NC(C(=O)NC2C(OC)CCC2)Cc2ccco2)c[nH]c(=O)cn1 c1(C(=O)NCC2N(C(Cc3cncc(OC)c3)=O)CC2)c(C)nc(C2CC2)nc1C CC(C)CCC(O)C(=O)NCC1CCC(NC(c2nnc(O)cc2O)=O)CC1 c1(C(=O)NC(CNC(c2cc3c(o2)CCCC3)=O)CO)cc2c(nn1)CCCO2 CC1CC(NC(c2cnccn2)=O)CN1C(c1ccc(C2CCCO2)[nH]1)=O C1(NC(c2ccc(Cl)cc2Cl)=O)COC2(CCN(C(=O)CCN3CCCC3)C2)C1 c1(CCC)cc(CNC(CN2CC(c3cccc(C)c3)C2)=O)c(C)s1 C1(NC(=O)NCC#C)CC=C1CNC(=O)CCC c1(C(C(=O)NC2CC(CNC(C3CNC(=O)C3)=O)C2)OC)ccc(F)cc1 CC1CCN(C(c2cc(C(N)=O)c[nH]2)=O)CC1NC(=O)CN(C)S(N)(=O)=O N1(C(C(C(C)(C)O)F)=O)CC(C2CN(C(=O)CC3C=CS(=O)(=O)C3)C2)C1 c1(SCC#C)cccc(C(=O)NCC(CCOC)NC(=O)C(C2(O)CCCC2)F)c1 C1(CNC(c2c(C)nn(C)c2)=O)CC2(CCN(c3ccnc(Cl)n3)C2)CO1 CCC(C)CC(C)C(=O)NCC1(COC)CCN(C(C2CC3(C2)CC(C)C3)=O)C1 c1(C(C(=O)N(CC(C)C)CCCO)NC(=O)C(C)C2CCC2)ccccc1 N1(C(CC(=O)OCC)=O)CCCC(CO)(NC(c2cc(C)c(F)cn2)=O)C1 Cc1ccc(C=CC(=O)N(C)CC2CCN(C(C3(C4CC4)CC3)=O)C2)cc1F c1(C(N2CC3C(NC(CCCCC)=O)(C3)C2)=O)cccc2oncc12 c1(NCC(COCC)C)cc(NC(c2cccc(C)n2)C)nc(C)n1 C1(N(C)C(c2cc(C3(C)CC3)n[nH]2)=O)CCC(NC(c2c[nH]nc2CF)=O)CC1 c1(OCC)cc(Cl)ccc1C(N1CCN(C(=O)CC(C)COC)C(C)C1)=O C(C(CC(C)C)C(=O)N1CCC1C(=O)NC1(C)C2CC3C(C2)C13)OC c1(NC(C2C=CC(NC(=O)CN3CCCC(CO)C3)C2)=O)c(F)cccc1Cl C#Cc1ccc(Br)c(C(=O)N(C)Cc2ccccc2COCC)c1 N1(C(CC(CNC(c2c(OC)n(C)nc2)=O)C)=O)CCC2(CC1)CC2C#N C(=O)(C1CCc2nccn21)NC(CNC(C1ON=C(C(C)C)C1)=O)C C1(CC#C)CCCCN1C(=O)C(CC1CC1)NC(C1CCCN1C)=O C1(NC(=O)NCC(=O)NCC)CN(C(=O)C(C)NC(=O)OC(C)(C)C)C1 c1(CN(CC(=O)NC)CCOC)ccc(C(C)(C)C#N)cc1 C=C(C)C(C)(C)C(=O)NCCOCCN(C(=O)Cc1ncn(C)c1C)C N1(C(CN2C(=O)CCCC2)=O)CCC(C2(O)CN(C(c3cn[nH]c3)=O)C2)CC1 N1(C(C(C(=O)OC)OC)=O)CCC(O)CC1C(=O)Nc1ccc(Cl)cc1C(F)(F)F C1(NC(C(CC)NC(C)=O)=O)CC(C)CN(C(c2snc(O)c2Cl)=O)C1 c1(N(C(C(=O)OCC)C)CC2CC2C)ccccc1 N1(C(C)=O)CC(C(N2CCCC2(C)c2ccccc2)=O)Oc2ccccc21 c1(OC)c(NC(=O)NCCN(C(=O)CCC2CCCC(=O)N2)C(C)C)cnn1C N1(C(CN2CCC(C)CC2)=O)CC2CC(NC(c3cncc(Cl)c3)=O)C2C1 Cc1cncc(C=CC(=O)NCC2CCN2C(=O)C(C)CCCO)c1 CN1N=C(CC(=O)NC2CN(C(c3ccccc3F)=O)C3(CCOC3)C2)CC1=O C1(CNC(CN(C(=O)OCC)C)=O)CN(C(=O)C(C)SC)C1 N1(C(C(C=C)c2ccccc2)=O)CCC(C)(NC(=O)C=Cc2ccn(C)c2)C1 C1(CC(=O)NCC2CCCN2C(=O)CC2CC=CC2)CC2(CCOCC2)CO1 c1(C(N(CC(CN(C(COC(CC)C)=O)C)O)C)=O)cc2c(cn1)NC(=O)CO2 C#Cc1cccc(CC(=O)N(C2CC(NC(=O)CN3CCCCS3(=O)=O)C2)C)c1 CC1(C(N2CC=CC2CF)=O)CCCN1C(C1CC12CCCC2)=O CC1COCC(C(=O)Nc2cccc(CNC(C3CCC3CF)=O)c2)O1 C1(C(=O)NCCC(C(=O)N(CCC(=O)OC)C2CC2)O)CC2CC(=O)C1O2 C1(CNC)CCCCN1N(C)C=Cc1ccco1 c1(CNC(CCn2ncc(C)c2)=O)ccc(C(=O)N(CC(C)C(C)C)C(C)C)cc1 C1(S(C)(=O)=O)(C(N(CC(C)CNC(=O)CC2CCSC2)C)=O)CC1 Cc1c(C(=O)NCCCNC(C2CC(N(C)C)C2)=O)cccc1Cl.C1(N)CCCC1C C1(C(=O)NCC(C2CCN(C(CN(C)CC)=O)CC2)O)COCCC1(F)F C1(C(N2CCC(NC(=O)CC3(C(F)(F)F)CCC3)C2)=O)CCCCC1(F)F CN(C)NC(=O)CCC(=O)NC1CC1C(=O)N=c1cc[nH][nH]1 N1(C(C(CC=CC)C)=O)CCCN(C(=O)CSCC(=O)NC)C(C(C)C)C1 CC(CCC(=O)NCC1(O)CCN(C)C1)NC(C1(C)CC1(F)F)=O N1(C(c2occc2C)C(=O)NCC(=C)C)CCC(O)C(C(N)=O)C1 C(C)(C)(CCC(=O)NCC1(NC(c2cc(=O)cc[nH]2)=O)CCOC1)OC CC(C)CCCC(C)(c1nnnn1CC1CC1(Cl)Cl)Nc1ccc(C(F)(F)F)cc1 C1(C(N2CC3(CC(OC)C3)C2)=O)CC2(CCN1C(=O)CCC(C)OC)CC2 c1(C(N2CCC(CCC)(C(=O)OCC)CC2)=O)cc(Cl)ccc1N=[N+]=[N-] c1(CC(C)C)n[nH]c(=NCc2cn(CC3CCCCN3CC(C)C)nn2)s1 Cc1cc(NC(=O)C(C)(C)C)sc1C(=O)NCCCNC(C1CC=CCO1)=O C1(NC(c2cc(COC)oc2C)=O)CCCCN(C(=O)CCC=C(C)C)C1 C1(CC(=O)NCC(=O)OCC#C)CC(C)N(C(=O)CCc2cncnc2)C1 Cc1nc(C)c(C(N2CC(F)CC2C(=O)NCCF)=O)o1 N1(C(CC(C)C(F)F)=O)CC2CCC(CNC(c3ccc(Cl)[nH]3)=O)C2C1 CC(Cn1ccnc1)C(=O)N1CCC(C(C)(C)NC(=O)C=Cc2cccs2)C1 C1(CNC(c2c(C)nc(NC3CC3)s2)=O)CN(C(C2CCCO2)=O)CCC1C c1(C(=O)NC)cc(CNC(=O)CC2(N3C(CC(=O)NC)CC3)CC2)no1 C(=O)(CC(C)CC)N1CCC(N(C(c2c(CC)scc2)=O)C)C1 C1(CS(=O)(=O)NCCCc2c(C)ccc(Br)c2)Cc2cc(F)ccc2O1 C(=O)(C(CC1CCC1)NC(=O)Cc1ccon1)NC1CC(SCC)C1 CC1C(=O)CCN1C(=O)NC1(c2cccc(Cl)c2)CCS(=O)(=O)C1 Nc1cc(Cl)ccc1C(=O)NCCCCNC(=O)CCCOc1ccc(Cl)cc1 Cc1ccc(CCC(=O)NCC2CC2NC(c2cnc(C(C)N(C)C)s2)=O)cc1C N1(Cc2n(C)c(S)nn2)CC(NC(=O)C2=CCCC2)C(C)(C)C1 c1(CC(=O)NC(CC=C)CNC(C2CCCN2CCOC)=O)c(C)ncnc1C C1(NC(C2(COC)CN(C(c3ccc(CC)[nH]3)=O)C2)=O)C=CCCCC1 CCCCC(C(=O)N1CCOCC1C(=O)NC(C)C(=O)N(CC)CC)C(C)C C(=O)(C(CNC(c1c[nH]c(=N)c(C)c1)=O)CC=C)N(C(C=C)C1CC1)C c1(C(=O)NCC(CC)N(C(=O)Cn2cccn2)C)ccc(=O)n(CCO)c1 N1(C(C(C(CC)C)O)=O)CC(NC(=O)CCCOC(C)C)CC(C)(C)C1 N1(C(c2ccc[nH]2)=O)CCCCC1CCNC(C1(c2ccc(O)nc2)CCC1)=O N1(C(C2C(NC(CCCC#C)=O)C=CCC2)=O)CC2(CNC(=O)C2)C1 CCC(C)CC(C)C(=O)NCCC1CCCCN1C(C1CCCC2(CCC2)C1)=O c1(OC)ccc(Cl)c(C(=O)NCCC2CN(C(=O)C(C)CC3CC3)C2)c1Cl c1(OC)ccc(F)c(C(=O)NC2CC(CNC(C3CCCC3(F)F)=O)C2)c1Cl N1(C(C2CCN(C(CC)=O)C2)=O)CCCC(CC)(NC(C2CC(C)CC(C)C2)=O)C1 c1(SC)n[nH]c(=NC(=O)Nc2nc(-c3ccccc3OC(C)C)cs2)s1 N1(C(c2n(CC)ncc2)=O)CCC(NC(c2ccn(C3CCCC3)n2)=O)C(F)C1 C(=O)(CC(C)(C)CC(=O)N1CCC(NC(C2CCC(=O)N2)=O)C(F)(F)CC1)OC C=CC(C)(O)CC(=O)NC1CCC(N(C(=O)CC(C)F)C)CC1 C1(CN(C(=O)CCc2cncc(O)c2)C)CC(F)CN1C(=O)CCC(F)F n1(CC)c(C)cc(OC)c1OC.c12ccc(C(C)C)cc1N2 C1(OC)(CNC(c2cc(C)co2)=O)CCN(C(=O)C(C)(C)C2CC2)C1 N1(C(C(C)OCCCC)=O)CC2CC(N(C)C(c3sc(CCC)nc3C)=O)C1C2 CC(C)C(CCNC(c1nn(C(C)(C)C)cc1Cl)=O)NC(C1CCC=CCC1)=O n1(CC(N2CCC(CNC(c3n(C)ccc3)=O)C2)=O)nc2n(c1=O)CCCCC2 C1(NC(c2c(COC)ccs2)=O)CC2CC(NC(=O)CCC3CC3)C1C2 c1(COCCNC(N2CC3(C(C(=O)NC4CC4)C3)C2)=O)ccc2c(c1)CCO2 Cc1cc(C(=O)NOC2CN(C(=O)CNC=O)C2)cc(C)n1 c1(CCC)nccn1CC(=O)NCC1COC(CNC(=O)C(F)(F)C2CC2)C1 c1(CNc2c(OC)nsc2)[nH]c(=NC2CCC(F)CC2)nc2c1ncn2C CC(C)(C)C(CO)C(=O)NCC(C1CCC1)NC(c1cc(N)c(Cl)cn1)=O c1(CCC(=O)N(CCNC(Cc2ccn(CC)n2)=O)C2CC2)cccc(Cl)c1Cl c12ccnc(c1)C2.c1(CC)ncc(C(=O)NN2CCC(N(C)C(C)=O)C2)[nH]1 c1(C(=O)NCC=CCNC(=O)CCc2ccc(-c3ccccc3)o2)ccc(Cl)nc1 C12=CNC(=NCCNC1=O)C=C2.C1(CC(=O)N(CCOC)C)CCCS(=O)(=O)C1 CC(C)S(=O)(=O)C(C)C(=O)NCC(C)CNC(=O)C(c1ccccc1F)O C1(NC(C2N(C(C)C)CCCC2)=O)CN(C(=O)CC23CC(C2)C3)CC1(C)C C1(N(C(c2cccc(C(F)(F)F)c2)C(=O)NC)C2COC2)CCCCCC1C N1(C(C(Cn2cccn2)OC)=O)CC2CC(NC(=O)CC3CCCCC3)CC2C1 C1(O)(COC)CCN(C(=O)C(F)(F)C2(NC(=O)OC)CCC2)C1 N1(C(c2cccc(C)c2)=O)CCN(C(c2cnnc(C)c2C)=O)CC1C(C)C C1(CNC(CSC)=O)CCN(CCC2CCCS2)C1.S CCC(CC)(CO)C(=O)NC1CC(NC(=O)C(N2CCCCC2=O)C)C(O)C1 C(C)(C)(CC(=O)N(C)CCN1CCCC1=O)N(C(c1ccn(CC)n1)=O)C C1(CNC(CCSCC)=O)CC(O)CN1C(c1n[nH]cc1OC)=O c1(NC(C2CCCN(C(c3ccc(CC)nc3)=O)C2)=O)cc(C)ccc1C C1(C(=O)NCCOCC)CN(C(c2cc(Cl)cc(Br)c2O)=O)CC(F)(F)C1 C1(C(=O)NC(C)CNC(c2cc(N)ccc2O)=O)CC(F)(F)CCC1(C)C c1(C(=O)NC2CN(C(Cc3nnc(C)o3)=O)CC2C)c(C)nn(CC(C)C)c1Cl c1(OC)ccc(F)c(C(N2CCCC2CN(C(=O)CC(C)CC)C)=O)n1 CONS(=O)(=O)c1c(C(=O)NC2CCN(CCF)C2)cnn1C C(=O)(CC(O)C(Cl)(Cl)Cl)NCCCCCOC(=O)C(C)Sc1cnn(C)c1.CC C(=O)(C1CNC(=O)c2ccnn21)N1CC(O)(CNC(c2cnc(CC)[nH]2)=O)C1 c1(C(=O)NCC(CC=C)NC(c2sccc2NC)=O)cnc2cc(C)ccc2c1 C(=O)(CCCCC(=O)NCC1(N(C)C)CC1)c1ccc(C)cc1.C12CC(C1)NC2=O c1(CNCC2(F)CCN(c3cc(C(C)C)ncn3)CC2)nnc2n1CCCC2 N1(C(C2CN(OC)C(=O)C2)=O)CC2(C(=O)NCC3=CCCCC3)CCC1CC2 C1(NC(C2CCCN(CC)C2)=O)CCN(C(=O)C=Cc2cccc(F)c2)C1(C)C C12(NC(c3cc(CC)no3)=O)CCN(C(C3C=CC=CC=C3)=O)CCC1C2 C(=O)(CC(F)(F)c1ccccc1)NCC1CC(NC(C(c2cn(C)cn2)C)=O)C1 N1(C(c2c(C)occ2)=O)CC2ON=C(CNC(=O)CCC=CBr)C2C1 Cc1cc(C(=O)N(C)CC2(O)CCN(C(C3NC(=O)OC3C)=O)C2)c(N)cc1F c1(C(=O)NC2CC(CNC(c3cc(C)oc3C)=O)OCC2)ccc(F)c(Cl)c1 C1(NC(c2ccc(CCCC)cc2)=O)C2CCC1N(C(=O)C(C(C)CC)OC)C2 CC1=NOC(C(=O)N(CCCn2cc(-c3cnc(Cl)s3)nn2)C2CC2)C1 C1(NC(c2cn(CC)nc2C)=O)CCCC12CCN(C(=O)C=C1CCC1)CC2 c1(C(N2C(CN(C(c3ccc(C)s3)=O)C)CCC2)=O)cnc(Cl)cc1N C(CC1C(=O)N1)(c1nnnn1CCCSC)OC.c1(COC(C)=O)cnn(C)c1C N1(C(c2[nH]cc(-c3nc(C)sc3)c2)=O)CC2CCC2(NC(c2cccs2)=O)C1 C(CN=c1[nH]c(=NCc2ccccc2N(C)C)[nH]c2c1CSC2)N1CC(C)OCC1 C(c1cc(F)cc(F)c1)=CC(N1CCN(C(=O)NC(C(=O)OCC)C)CC1C)=O c1(C(=O)NC2C(C(C)NC(C3(O)CCC3)=O)C2)cnn(C(C)(C)C)c1Cl N#Cc1ccc(NCC(=O)NC2CCCN(C(C3CCCC3O)=O)C2)cc1 C(=O)(C(C)(C)C(C)(C)O)N1CCC(N(C(=O)CCn2ncn(C)c2=O)CC)CC1 C(C(C)(C(C)C)NC(c1cccc(CCN(C)C)c1)=O)NC(C=NOC)=O c1(C(=O)OC2CC3C=CC2C3)c(Br)c(C(F)(F)F)nc2[nH]cnc12 C1(CN(C)C(C2C=CCS2)=O)CN(C(C2(CO)CC2)=O)C1 C1(CC(=O)N(CCCOCCOC)C)CCN(C)C1=O.C1CC(=O)N(C)CCN1 O=C(CS(=O)(=O)C1CC1)NC1CN(C(c2cc3ccccn3n2)=O)CC(F)(F)C1 C1(CNC(C(C)OCC)=O)CC(O)CN1C(=O)C(C)Oc1ccccc1 C1(N(C(C(C)C)C(C)O)C(c2ccc([N+](=O)[O-])cc2)=O)CCC2(CCNCC2)CC1 c1(NC(C2N(C(c3c(COC)nn[nH]3)=O)CCC2)=O)ncc2ccccc2n1 c1(CC)cc(CC)[nH]c(=NC(CNC(C2(CF)CCOCC2)=O)C(C)C)n1 C=CCCCCCN(C(=O)CC1CC(C)N(C(c2nccs2)=O)C1)C N1(C(C(C)OC(C)(C)C)=O)CC2(CCCCN2C(=O)CCF)C1 CCC(CC)N=c1nc(N2CCC(c3cccnc3)C2)c2c([nH]1)CSC2 CC1=NNC(=O)C1CCC(N1CCCCC1C(=O)NCC(O)C(C)O)=O N#Cc1cn[nH]c1C(N1CCCCC1C1CCN(C(C2CCC(F)(F)C2)=O)CC1)=O C1(NC(C(C)C2CCCC2)=O)C2CC1CN(C(=O)C(F)=CCCF)C2 C12(NC(C(CC)SC)=O)CCCC1CN(C(=O)Cc1ccccc1CO)C2 C=CC(C)(C)CCCNC(C1C=CCN1C(=O)CCOCCCOC)=O C1(C(N2CC(C(C(=O)N(C(C#C)C3CCC3)C)OC)C2)=O)CC2(CCC2)C1 N1(C(CN2C(C)CCC2)=O)CCN(CC2CN(C(C3(Cl)CC3)=O)C2)CC1 C1(C(N2CC(CC)N(C(=O)COC(C)(C)C)CC2)=O)OCC2CCCC1C2 N1(C(C2CC(CCO)C2)=O)CCN(c2ncc(F)cn2)C(Cc2ccccc2)C1 c1(C(=O)NCC(C)(C2CCC2)NC(C2ON=C(C)C2)=O)cn2ccsc2n1 N1(C(C2(OC)CCCC2)=O)CC(NC(C2COCCN2C=O)=O)C2(CCCC2)C1 C(C(=O)NCC(C1CC1)N(C)C)(C(C)C)NC(c1c(COC)nco1)=O N1(C(C2CC(C)(OC)C2)=O)CC2CCC(C1)N2C(=O)CC(C)c1cccnc1 CCCC(C)(O)CC(=O)N1CC2(CO)CC1(C(=O)NCCOC1CCCCC1)C2 C1(NC(c2c(C)cccc2)=O)CCCC12CCN(C(c1ncoc1C)=O)C2 O=C(C1Cc2ccc(F)cc21)N1CC2CN(C(C3C=CC=CC=C3)=O)CC2C1 Cc1nc(C(C)NC(C2CCN(C(c3cc(C(N)=O)ccn3)=O)C2)=O)c(C)o1 C(CC(=O)NCC1(C2CC2)CC1)(C(F)F)NC(Cc1n(C)ncc1)=O c1(C(=O)NCCOCC(=O)NC(c2cccnc2)C)ccc(F)c(Br)c1 N1(C(C(C=C)O)=O)CC(NC(=O)Cc2nocc2C)CC(C)(C)C1 C(CCC(C)CC(=O)NC1(C2CCCCN2C(C2COC(=O)N2)=O)CC1)=C(C)C C1(C(=O)NCC2(NC(c3cccs3)=O)CCC2)CC(=O)c2cc(Cl)ccc2O1 c1(OC)cccc(CC(N2CC(n3cc(C(N(C)C)C4CC4)nn3)C(SC)C2)=O)n1 N1(C(C(CC)(C)CO)=O)CC2CCN(C(c3cccc(OC(C)(C)C)n3)=O)C2C1 C1(CNC(CCCCN(C(=O)COC(C)(C)C)C)=O)CCCCC(O)C1 Cc1noc(C(=O)NC(C)CN(C)C(C23CC(c4ccccc4)C2C3)=O)c1C Cc1nn(C)c(C)c1OCC(N1CC=CC1CNC(C1COC(=O)N1C)=O)=O CC1CCC(NC(C2CCC=CO2)=O)CN1C(C1CCCC12CCC2)=O c1(CNC(C2(COC)COC2)=O)cc(C(=O)Nc2cnn(C)c2)n(C)n1 N1(C(C(CC(C)C)(C)C)=O)CCC(C2CC2NC(C2CCCCS2(=O)=O)=O)CC1 c1(C(=O)NC2CC2CNC(C2CCCN2C2CCCC2)=O)cc2c([nH]1)CCCC2 c1(C(=O)NCC2N(C(c3c(=O)ccn(C)c3)=O)CC=C2)occ2c1CCCC2 CCC(CC)C(F)C(=O)NCCN(CC(C)O)C(=O)CNC(=O)OC N1(C(CC=C=C)=O)CC2CC(C1)C2NC(=O)CCc1cnccn1 c1(CN(C(C)C)C(=O)NC(c2cccnn2)C)ccnc(Oc2ccccn2)c1 C12CN(C(C)(CO)C1)C2=O.C(=O)(C(F)(F)c1cnn(CC2(CO)CC2)c1)N.CCO C1(NC(CCOC)=O)C(C)CCN(C(=O)CCc2cncs2)C1C N1(C(COCC(C)(C)C)=O)CC2C(C(=O)N)C2C1.c1(-c2ccccc2)csnc1Cl N1(C(C2C(C)(C(F)(F)F)C2)=O)CCCC(C)(CNC(=O)C2=CCOC2)C1 N1(C(=O)Cc2sccc2Cl)CCC2C(CCCN2C(c2cnco2)=O)C1 C(=O)(CC(c1ccccc1)SC)NCCN(C(C1(C)CC1(F)F)=O)CC C1(NC(C2CCC(CC)CC2)=O)CCN(Cc2cccc(Cl)c2Br)CC1(C)C c1(CN2CC(CNC(C3CCN(C)C3)=O)C2)c[nH]c2cc([N+](=O)[O-])ccc12 c1(C(C)C)cc(CC(N2CCC(c3cn(CC4C=CCCC4)nn3)C2)=O)on1 C12(C(=O)NCC(C)Nc3c([N+](=O)[O-])cnn3C)CC(C)(C1)OC21CCC1 C#Cc1ccc(OC)c(C(=O)NC2CC(C)CN(C(c3n[nH]cc3CC)=O)C2)c1 c1(CN(CC(=O)OCC)Cc2ccccc2)ccc(NS(C)(=O)=O)cc1 n1(CC(=O)NCC(CNC(c2nccnc2Cl)=O)OC)cccc(C)c1=O c1(C(N2C(C)CC(NC(C3CCC=CCCC3)=O)CC2)=O)cnc2ncccn12 Cc1cncc(C(=O)NC(C)CCCCNC(=O)Cc2nc[nH]n2)n1 C=C(F)C1(CC(N2CCC2C(=O)NCC(C)OC(F)F)=O)CCC1 Cc1sc(C(=O)N(C2CN(C(=O)COCC3CCOC3)C2)C)c(C)c1C C1(NC(c2cc(C)on2)=O)CC2(CCN(C(C3CC(C)CC(C)C3)=O)C2)C1 C(c1cccc(F)c1Cl)=CC(N1CCC(NC(C2C(CC)C2)=O)C1C)=O N1(C(c2cc(CC)nn2C)=O)CCC2CN(C(c3cnc4[nH]ccnc3-4)=O)CC12 C(=O)(N=c1ccn(Cc2ccccc2C)[nH]1)NCC1(OC)CCC(C)C1 c1(C(=O)NCc2ncccc2F)ccc2oncc2c1 C1(C(=O)OCC(C)CSc2ccccc2)COC2(CCC2)CO1 CCCC(CCC)CC(=O)N1CC(F)CC1CNC(=O)CCCC1CCOCC1 CC1(C)CC(COC(c2ncnc(O)c2Cl)=O)C(C)(C)O1 N1(C(CCc2n(C)ncc2)=O)CCOCC1CNC(c1n[nH]c(C(C)(C)C)n1)=O C=C(C)CC(C)C(=O)NC1CC(OCCNC(=O)C(c2ccsc2)=O)C1 c1(C(=O)NC2CC(NC(c3c(N(C)C)cncc3)=O)C2(C)C)cc(O)nc(Cl)c1 C1(CNC(c2ccc(C(F)(F)F)s2)C)CC2(C1)C(F)(F)C21CC1 N1(C(c2nccs2)=O)CC2(C1)CN(C(C1(CC3CC3)CC1)=O)CC2CO C(=O)(C(C)S(C)(=O)=O)N1CCCC(CN(C(C(n2ncc(C)c2)C)=O)C)C1 C(=O)(C(C)C(O)CC)NCC1N(C(c2cc(CCCC)oc2C)=O)CC(O)C1 CC(F)CN=c1[nH]c(=NC(C)c2ccc(Cl)c(F)c2)c2ncccc2[nH]1 N1(C(CN(C2CCOC2)C)=O)CCCC(C2CC2NC(=O)C=CCN(C)C)C1 C(=O)(C(C)C(C)(C)C)NCC1(C)CCN(c2snc(C(=O)OC)n2)C1 CCC1=C(C(=O)NC2C=CCC(C(=O)Nc3cnn(C(F)F)c3)C2)CCCO1 Cc1ccc(C(=O)NCC2(NC(=O)CCc3c(C)n[nH]c3C)CCOC2)cc1Cl c1(C(N2CCC(NCc3c(F)ccc(Cl)c3F)C2)=O)cc(F)c(F)c(Cl)c1 C1(C(N2CC(O)(CCO)C2)=O)(COC)CN(C(C23CC(OC)(C2)C3)=O)C1 CC1CC(C(=O)NC2C3CN(C(c4cc(Cl)cnc4O)=O)CC23)=NO1 c1(NC2(CNC(C=CCN(C)CC)=O)CCOCC2)ncc([N+](=O)[O-])c(=N)[nH]1 Cc1nc(C(F)(F)F)oc1C(N1CCC(O)(CNC(C2CC(C)(C)O2)=O)C1)=O N1(C(CC(CC)(C)C)=O)CC2CC(NC(=O)C(COC)OCCN(C)C)C(C2)C1 c1(CSC)c(C(=O)NC2CC(C(C)C)C2)sc2ccccc12.C12(CCC1)C(=O)N2 C1(N(c2cccc(C(CC)(C)C)c2)C)CN(C(=O)Cc2csc(C)n2)CCC1O CC1(C)C(CNC(C2(P(C)(C)=O)CC2)=O)CCN1C(c1cnco1)=O N1(C(CCC(=C)Br)=O)CCN(C(c2ccc(Cl)nc2N)=O)C(C)C1 c1(OC(C2C=CCCCC2)=O)cc(C(=O)CN2CCC(F)C2)ccc1O N1(C(c2c(C)cncn2)=O)CC(C(=O)N(C)Cc2ncco2)C2(CC2)C1 c1(C(=O)NCC(C)(C2CCC2)NC(COCCCOC)=O)ccnc2ncnn12 Cc1ccc(CN(C(CC2CCCO2)C(F)(F)F)Cc2ccccc2I)c(C)c1 Cc1nc2ccc(C(=O)NCC3(NC(c4cc[nH]n4)=O)CC3)cc2s1 c1(SCC(=O)NC2(CO)CN(C(C3CC3C3CC3)=O)C2)ccncc1 C(=O)(C1CCCc2n[nH]cc21)NCC=CCNC(c1cnc(SC)s1)=O C1(CN(C(=O)CC2CC3CCC2C3)CC)CCN(C(c2oc(C)cc2C)=O)CC1 c1(C(=O)NCC(CCOC)NC(c2cc(C)c(C)nn2)=O)cc(Cl)cnc1C CCCC(CCC)CC(=O)N1CCC(C(=O)N(CC(C)(C)C)C)(C(C)C)C1 C1(N(C)C(c2ncccc2F)=O)CCCCN(C(=O)CCn2ncn(C)c2=O)C1 c1(N2CCC(C)(CC)CC2)cc(C)c(S(=O)(=O)NCc2cc(C)cnc2F)cn1 N1(C(C2CCC(=O)O2)=O)CC(C(=O)NC2(CC3CC3)CCC2)C2(CC2)C1 CCC(C)C(C(=O)C(=O)C=CCN(C(=O)Cn1cncn1)C)NC.N(C)C C(=O)(CC(O)CC(C)(C)C)NCc1c(CNc2ncc(CC)cc2N)nccc1 Cc1cc(O)c([N+](=O)[O-])cc1C(N1CCC(C(N(C)Cc2ncccc2O)=O)C1)=O N1(C(c2cc(CC)no2)=O)CC2CCCC(NC(c3coc(C4CC4)n3)=O)(C2)C1 c1(C(N2C(CNC(CCC(C)=O)=O)CC2)=O)cc(Cl)cc(Cl)c1[N+](=O)[O-] Nc1c(C(N2CCCCC2CNC(=O)C=CC(F)F)=O)nnc2ccccc12 C(=O)(C1CCCc2c1ncn2C)N1CCOCC(NC(c2nccc(C)c2)=O)C1 c1(NCc2c(C)cncc2)[nH]c(=NCC2(C)CC2)nc2c1cnn2C c1(C(N2C(CNC(C(C3CC(F)(F)C3)OCC)=O)CC2)=O)cc(C)c(Cl)s1 Cc1c(C(=O)O)cnn1CCNC(n1cc(C(C)(C)C(=O)O)nn1)=O c1(C(=O)NC2C(NC(c3n(C)ccn3)=O)CC2)cccc2ncnc(O)c12 c1(C(=O)NC(CN(C(C(C)Cc2ccccn2)=O)C)C)ccc2c(c1)OCCN2 c1(C(=O)NCC23N(C(=O)OC(C)(C)C)CCC2CC3)ccc2nc(CO)[nH]c2c1 c1(C(=O)NCCNC(=O)CC2CCCCO2)ccc(F)c(F)c1Cl C1(C)(CC(=O)N(CCC(=O)NC(c2ccsc2)C)C)CCCC1 C1(C(=O)NCC2N(C=O)CCC2)CN(C(=O)CC2CCCSC2)CC1C1CC1 CC(C#N)CCC(=O)N1CCC(CO)(NC(=O)CCOCCN(C)C)C1 c1(OC)ccc2ncn(C)c(=O)c2c1.c12cccc(c1)CN1CC2C1 CC1CN(C(c2nccc(Cl)c2F)=O)CCC1CNC(C1(CO)CCCC1)=O N1(C(C2(C#C)CN(C(c3cnccc3C)=O)C2)=O)CCC(CC)CC1CC c1(C(=O)NCC2C(NC(C(C)(C)F)=O)COC2)ncc2ccccn12 CC1=C(C(=O)NOC(CC(C)C)C(=O)Nc2cscc2C)CCC1 c1(OCC)ncc(C(N2CC(NC(=O)C(O)CC3CC3)CC(O)C2)=O)cc1Cl C1(C(N(C)CC2(CNC(=O)CC(=O)NCC(F)(F)F)CC2)=O)CCC(C)(C)O1 C1(NC(C2CC(O)(CNC(C3CCCC3O)=O)C2)=O)CC2(CC2)C1 c1(C(N2CCC(N(C(CC3CC(=C)C3)=O)CC)CC2)=O)cnn2c(C)cccc12 c1(NC(C23CC2CN(Cc2cc(Br)c[nH]2)C3)=O)cc(Br)c(C(F)(F)F)cc1[N+](=O)[O-] c1(C(=O)NCC=CCNC(C(c2c(OC)cccc2)C)=O)ccc(=N)[nH]c1Cl CCCCC(F)C(=O)N(C)CCOCCCNC(c1cn(CCO)nn1)=O c1(NC(C2(OC(c3cnc(OCC)c(Cl)c3)=O)CC2)=O)cnn2c1CCCC2 Cc1ccnc(C(=O)N(CCCN(C)C(c2c[nH]nc2-c2ccco2)=O)C)n1 c1(C(N2C3CN(C(C4(C)CCC(=O)NC4)=O)C(C3)C2)=O)cccc2c1OCCCO2 c1(N2CCC(C(=O)OCC)CC2)cnc2c(F)cccc2n1 N1(C(COC(C)=O)=O)CC(NC(C2CCN(C3CCCCC3)C2=O)=O)CC(F)C1 C(=O)(C(C)(C)CC(C)C)N1CC(OC)CC(NC(Cc2ccc(CC)cc2)=O)C1 c1(C(N(CCCN(C(=O)CCC2CC(OC)C2)CC)CC)=O)scnc1Cl c1(NC(CC2CCN(C(C(CNC)C)=O)C2)=O)cccc(OC)c1 N1(C(CCCCN(C(c2cncc(OC)n2)=O)C)=O)CCN(C)CC1CO c1(NC(c2ccc(CNC(C3(CCF)CC3)=O)cc2)=O)ccc2nccn2c1 N1(C(c2n(C)nc(C(C)(C)C)c2)=O)C2CCC1C(CNC(=O)CCC1(C)CC1)C2 CC1=C(C)CC(C)(C(N2CCC(OCCNC(C3CCCOCC3)=O)C2)=O)CC1 N1(C(C2CC(C(C)C)C2)=O)CCOC(CCCNC(=O)C=C(C2CC2)C2CC2)C1 c1(C(=O)NCCC2CN(C(C3CC(C(F)(F)F)C3)=O)C2)conc1C1CCC1 c1(C(=O)NCC(C2CC2)NC(c2ncc(OC)cc2F)=O)ccc2nsnc2c1 c1(C(=O)OCC2C(C)C2)ccc2cc[nH]c2n1 c1(C(N2CC(C#C)(C(=O)N(CCCOC)C)C2)=O)cc2occc2[nH]1 CC12CCN(C1)C2=O.c1(C(=O)NC2CC2)cnc(NC(C2CC23CC3)=O)o1 C12(CNC(CSC)=O)CCC(CN1C(=O)CCOC(C)CC(C)C)C2 C(C)(CCC(=O)N1CC(CN(C(=O)CN(C)C2CC2)C(C)(C)C)C(C)C1)SC C(CC(F)(F)Cn1cc(CCCC)nn1)N(C(CCC=C)=O)C c1(C(N2CCC(C)C2CNC(c2c[nH]c(C(N)=O)c2)=O)=O)ccc(Cl)c(Cl)c1O O=C1CCC(C(=O)N2CCCC(O)(CN3CCC(c4cc(Cl)cc(Cl)c4)C3)C2)=NN1 c1(NC(CCN(C(C2(C)CC3(CCC3)C2)=O)C2CC2)=O)ccc2ncnn2c1 CC#CCC(C(=O)Nc1ncc(OC)cn1)NC(C1(C)CCOCC1)=O c1(C(C(=O)N(C)CC2CCN(C(=O)OC)CC2)(C)C)ccc2c(c1)OCCO2 O=C1CS(=O)(=O)c2ccc(C(=O)Nc3cccc(I)c3)cc2N1 c1(C(=O)NC2CCCN(C(=O)C=C3CC3)C2)ccc2c(c1F)NCCC2 N1(C(C(CC2CC2)ONC(c2ccc(C#N)o2)=O)=O)CC2CCCC2(CO)C1 CC1=C(C(=O)NC23CCN(C(C4CC5(CCCCC5)C4)=O)CC2C3)CCCO1 c1(OC)ccc(C(N2CC(N(C(=O)CCC3CC3(F)F)CCO)C2)=O)cc1N Cc1cc(=NC2CCC(NC3(c4ccccn4)CC3)CC2)[nH]c(C(C)(C)C)n1 N1(C(C(CCC)=CCC)=O)CCC(C)(NC(C2CC(OC)(OC)C2)=O)CC1 CC(O)CCCCCC(=O)NCC1(C)CC(F)(F)CN1C(=O)C=Cc1ccc[nH]1 c1(C(N2C(C)CN(C(=O)CC3CC=CCC3)CC2)=O)ccc2c(c1)CCCCN2 C(=O)(C1=NNC(=O)CC1)NC1CCCC(C(C)C)C1.c12sccc1NC2=O C1(SC)CCOC2(CCC2)C1.C1(COC)CN2CCN1C(=O)C1(CC1)C2=O CCC(O)C(C)C(=O)NCC=C1CCN(C(C2(C(N)=O)CCC2)=O)CC1 C1(NC(CN2CCC(OC)C2)=O)CC(F)CN(C(=O)C(C)(F)c2ccon2)C1 C1(CC=C)(C(=O)N(CCC)CC)CCN(C(=O)C(C)n2cccn2)CC1 C1(C(N2CC(NC(C(Cc3c(C)cccc3)C)=O)C2)=O)CC12CC(C)(C)C2 C1(CNC(CNC(c2n(C)nnn2)c2cnn(C)n2)=O)CC2CC(OC)C2C1 Cc1cc(=Nc2cccc(N(C3CCOCC3)C)c2)[nH]c(CC2CC2)n1 C1(C(=O)NCC2(C(=O)NC3(CC)CCCCC3)CC2)CC2CC(=O)C1O2 CC1=NN(C)C(=O)C1CC(N1CCOC(CN(C)C(c2sccc2Cl)=O)C1)=O Cn1c(O)nc2c(C(=O)NCCOCCNC(c3cocn3)=O)cc(Br)cc12 N1(C(C=CCN2C(=O)CN2)=O)CC2(C(N)=O)CCC1CC2.CCC(=O)OC.CC C1(NC(C=CC=CCC)=O)C2CCN(C(c3ccnn3C3CCC3)=O)CC12 c1(C(N(CCCCNC(c2ccccc2OC(F)F)=O)C)=O)cc(Cl)ncc1O N1(C(CC2(C)CC2(Cl)Cl)=O)C2CCC1C(CNC(C1CCC=CCCC1)=O)C2 c1(OC)ncc(C(N2CCC(NC(C3CC(=O)N(O)C3)=O)C2)=O)cc1C O=C(CCCCCc1ccccc1)NCC#CCNC(C1CCSCC1)=O C1(CNC(C2(C)CC(=C)C2)=O)C2CCCC1N(C(c1cn(C(C)C)nc1C)=O)C2 c1(C(C(=O)NCC(CNC(c2c(NC)nccc2)=O)CO)O)ccc(Cl)cc1F C1(C(N(CCCNC(c2cn(C3CC3)nn2)=O)C(C)C)=O)CCC(=O)CC1 c1(C(N2C3C(CC2)NC3=O)=O)cccn2nccc12.c1(CC)nnsc1N Cc1ccc(C(C)CC(=O)N2CCC(N(C(=O)C(C)(C)OC3CC3)C)C2)cc1 c1(CNCC(C)NC(c2cc(C(C)C)cc(C(C)C)c2O)=O)ccc2cnnn2c1 c1(NC(N2CC(C(c3ncc(C)s3)CC)NCC2)=O)cccc(C)c1Cl C(=O)(CC(N)C(O)C(C)(C)C)N1CCCC(CC=C(C)C)C1 C1(CN(C(=O)CC2(CO)CC2)C)CCCN1C(=O)C(=O)NCCCCNC1CC1 C1(CNC(C2N(C(=O)NC)CCC2)=O)CC2(CCOCC2)CN1C(C1CCSC1)=O Cc1coc(C(=O)NC2C=CC(CC(=O)NC(C)C(C)(C)C)C2)c1 C#CC1(C(=O)NC2CC(OCC(=O)Nc3cncnc3)C2)CCCC1 C(=O)(C(C)CCCC(C)=O)N1CCC(C(N2CCC(O)(CN(C)C)C2)=O)(CC)C1 C(C(O)C(CC)CC)NC(C(C)N(C(c1ccc(CCC)s1)=O)C1CC1)=O CC(C(=O)NS(=O)(=O)CCCCC1CC1)P(C)(C)=O c1(NC(c2c(C)nc(C3CCCCC3)s2)=O)ccc(F)c(-c2ccc(O)cc2)c1 CS(=O)c1cccc(NC(c2ccnn2CCF)=O)c1 c1(C(=O)NC(c2ccc(Cl)cc2)C)cc2cc(S(N)(=O)=O)sc2s1 c1(C(N2CCC(O)(C(F)(F)F)C2)C(=O)NCCC)cc(Br)cc2cccnc12 c1(C(N2CCCC(NC(COC)=O)CC2)=O)ccc2c(c1)C=CS2(=O)=O C1(C(=O)NCCN(CC)Cc2nn(C)cc2C(=O)O)CCC2C(C1)C2(F)F C1(N(C(C2CC(C)(F)C2)C(=O)NC(C)(C)C)C)CCC(C(N)=O)C1 C(=O)(C(C)(CC)CO)N1CC(OC)C(C(=O)N(C)CCc2cccs2)C1 C1(C(=O)NC2CC(=C)C2)C2CCC(C2)C1C.O1NC(=O)C(C)Cc2ccn(n2)C1=O C(=O)(C1CCCc2sccc21)NCC1C(C)(C)CCN(C(C2(N(C)C)CC2)=O)C1 C1(C(=O)NCCN(CCC)C(C2CCCC(F)C2)=O)CCCC1S(C)(=O)=O c1(C(=O)NC(CNC(C2N(C)CCOC2)=O)(C)CO)cc2c(F)c(F)ccc2s1 C1(CC(=O)NC(C(C)NC(C2(CCCC)CC2)=O)CO)CCCC(C)(C)CC1 C(=O)(C(CSC)C(C)c1ccccc1)NC(CNC(C(CC)=CC)=O)CC(C)C C=CC1(C(N2CC(COC)C2)=O)CCN(C(=O)C(c2cnn(C)c2)=O)C1 Nc1ccc(C(=O)NCC2(NC(C3CC(F)(F)CS3)=O)CC(F)(F)C2)c(F)c1 Cc1nnsc1C(=O)NCC(=O)NC1CCCC1C(N)=O c1(C(N2C(CC)C(NC(c3ocnc3C)=O)CC2)=O)cccc(O)c1Cl Cc1c(N2CCSC(C)CC2)ncnc1NC1CCCC(OC(F)F)C1 CC1OC2CCC1(C(=O)NCC(c1cccc(C3CC3)c1)NC(C1(O)CC1)=O)C2 C1(F)(CNC(c2ccccc2Cn2cccn2)=O)CCN(C(C2CC2F)=O)C1 C1(C(=O)NCC2(CNC(C3CCCC3C)=O)CCC2)(OCC)CCOCC1 N1(C(CCC2CCC(C)O2)=O)CCCC12CCN(C(c1cnoc1)=O)CC2 N1(C(C)=O)Cc2nccn2CC(N(C(=O)C(C)(C)C)CC2(Oc3ccccc3)CC2)C1 N1(c2c(Br)cnc(OC)n2)CCN(C(c2ccc(C(F)F)c(Cl)c2)=O)CCC1C c1(C(C)NC(=O)C(F)OC(F)(F)F)nocc1C(=O)NCC(C)N=[N+]=[N-] C1(C(N(CC(=O)NC2CC2)C2CC2)=O)CC2C=CC1O2 c1(C(=O)NCC2(CNC(C(C(=O)OCC)SC)=O)CC2)ccc(C2CC2)cc1Cl C1(NC(C(C)SC)=O)CC2CC1CN(C(C1CC1Cc1ccccc1)=O)C2 CC1=C(C(=O)N2CCC3CCC23c2nnc(C(C)C)o2)SCCO1 N1(CC(C)O)CCCC2C1CCN2C(=O)Cc1noc2ccc(F)cc12 CC(CC(N)=O)C(=O)NCCC1CCN(C(c2cn(C)cc2C(F)(F)F)=O)CC1 c1(C(N2CCC=C(C)C2)=O)c(NC(=O)Cn2ccc(C3CC3)n2)cccc1F c1(C(=O)NCC2CC(C(=O)NCCC(C)OC)C2)c[nH]c(=N)o1 c1(C(N2C(C(=O)Nc3ncc(Br)c(I)n3)CC(C)C2)=O)ccc(F)cc1[N+](=O)[O-] c1(C(N2CC3C(CNC(c4ccnnc4O)=O)C3C2)=O)cc2c(Cl)ccnc2s1 C=CCCCCCCC(=O)N1CCCCCC1C(=O)NCCn1nncc1C Cc1ccc(C(N2CC=CC(NC(=O)CC3CCC=CCC3)C2)=O)cn1 C(CCC(C)C)(C(=O)N1CCC(O)(CNC(=O)CCC2CCC(O)CC2)C1)OC N1(C(c2c(C)cco2)=O)CC2CCN(C(c3nc(Br)c[nH]3)=O)CC2C1 c1(C(N2CC(C)C(NC(C(COC)OC)=O)C(C)C2)=O)c[nH]c2nc(Cl)ccc12 c1(C(N2CC(NC(C3CCC(CC)CC3)=O)(CO)C2)=O)cc2c(s1)CCOC2 c1(C(=O)NCC(CNC(c2nc(CCC)oc2)=O)C)sc(C)nc1C CC(C)C(CN(C)C)C(=O)N1CCC1CNC(=O)C(C)(C)c1cccs1 c1(OC)cc(CN2CCC2(C)C(=O)Oc2ccc(F)cc2)ccc1O C1(C(=O)NCC(CC(C)C)(C)NC(c2ncn(C)n2)=O)CS(=O)(=O)CC12CCC2 C1(CC(N2CC(OCCNC(c3cccnn3)=O)C2)=O)CCCC2(CC2)C1 C(CCC(O)C(=O)N1C2COCC1C2)NC(=O)COC1CCCC1 CC1CCc2onc(C(=O)NCC3(C)CCN(C(c4cn[nH]c4)=O)C3)c2C1 N1(C(c2n(CC)ncc2)=O)CCC(C)C(NC(c2sccc2C2CC2)=O)C1 N1(C(C(C=CCCC)O)=O)CC=CC(NC(=O)CCSc2csc(C)n2)C1 c1(C(N(C2CN(C(COCC(C)C)=O)CC2F)C)=O)n[nH]c2ccc(Cl)cc12 N1(C(C(N)CCSC(F)(F)F)=O)CC(F)(F)C(F)(F)C1 c1(C(C2CCC2)NC(C(CC)Oc2ccccc2Cl)=O)c(C)cccc1C N1(C(CC(=O)OCC)=O)CCC2CC(C1)CN(C(c1cc(C)nnc1CC)=O)C2 c1(C(N(C(C)CNC(=O)C(C(C)(C)C)OC)CC)=O)c(C)ncnc1O c1(NC(C2C3(CCN(C(c4c(C)cc(F)cc4)=O)C3)C2)=O)cc(F)cnc1C#N N1(CC(C)C)CCC(C(=O)NCC(C)(C2CC2)NC(=O)CCC2CCCO2)CC1 c1(C(=O)NCC(C)(O)CNC(C2CCn3cnnc3C2)=O)cnn2c1OCCC2 N1(C(=O)NC2CCCCC2)CCOC2(CCCOC2)C1 C#Cc1cncc(NC(=O)CC2COCCN2C(C2CN(C)CC(C)O2)=O)c1 c1(C(=O)NC(c2ccc(-c3ccccc3)cc2)C(C)C)nnc2ccccn12 c1(OC)nc(C)sc1C(=O)NCC1(CO)CCN(C(=O)C(C)(C)NC(C)=O)C1 c1(C(N2C(C(=O)NCC(=O)NC)CC(C)(C)C2)=O)cc2cccnn2c1 c1(CC)ncc2c(n1)CCC(C(=O)N(c1ncccc1Cl)CCC#N)C2 c1(-c2cn(C3CCC(C(N4CCCC(CC)C4)=O)C3)nn2)cc(C)c(C)cc1C C1(COC)CC(CNC(=O)Cn2cnnc2)N(C(=O)CCCc2cccnc2)C1 Cc1nocc1NC(=O)C(=O)NC(Cc1ccccc1)C(=O)N1CCCC1 N1(C(C(CC)O)=O)CC2CN(C(C3CCC3)=O)CC12 C(CC(C(=O)NCCC(F)Cn1cc(C(C)C(O)C2CCC2)nn1)OC)OCC c1(CNC(=O)Nc2cnn(CC(F)(F)F)c2)cccc(Br)c1O C(N=C(NCC(F)F)N1CCC(OCC(N)=O)C1)C1(C(=O)OCC)CCCO1 C1(C(=O)NC(C(C)(C)NC(c2c(CC)occ2)=O)C)CCC(C(N)=O)CC1 C1(CNc2nccc(=NCc3cn(C(C)C)nn3)[nH]2)CCC2(CCOCC2)CO1 Cc1ccccc1C1(C(N2CC(N(C)C(c3cccc(C(C)C)c3)=O)C2)=O)CC1 CCC(C)C(C(=O)NCCCn1ncnn1)N(C(=O)Cc1cc[nH]n1)C CC1N(CCCC2CNC2)CC12CCC2 C1(CNC(=O)CC2CCC3CC3C2)CC2(CCC2)CN1C(c1occc1Br)=O N1(C(C2(C)CCCC2O)=O)CCOCC(CNC(c2cc(CC3CC3)on2)=O)C1 c1(C(N2CC(NC(C3CC(OCC4CC4)C3)=O)C2)=O)cc(C2CCCC2)no1 c1(C(=O)NC2C(CNC(c3cc(CC4CC4)on3)=O)C2)ccccc1OC(F)F Cc1cc(C(=O)NC(C2CCN(C(C3(C)CCCC3)=O)C2)C)cc(N)c1 C(CC(C(C)C)NC(C1CC(C)N(C)C1)=O)NC(C(c1cc(C)sc1)(F)F)=O C1(NC(C=COCC)=O)(CNC(=O)Cn2cc(C(F)F)cn2)CC2CCC1C2 C(=O)(C1CCCc2cccnc21)NC1C(O)CCN(C(C(C)(C)C(F)(F)F)=O)C1 C1(C2CCCC2)(C(=O)NC2CN(C(c3cc(C)c(C)nc3)=O)C(C)(C)C2)CCC1 C(=O)(C1c2c[nH]nc2CN1C(=O)C1=CCCCCC1)NCC(CCOC)O O=S(=O)(C1CCCC1)NCc1cccc(C(F)F)c1 n1(CCNC2CCC(CC#N)C2)cc(Br)ccc1=O c1(CN2C(C(=O)Nc3ncc(C(F)F)cn3)C(O)CC2)cc(Cl)cc(Cl)c1O N1(C(C2CCCC2C)C(=O)NCCC(=O)OC)CCC(C(=O)NC2CCCC2)C1 CC(C)C(CNC(=O)CCC1CCCN1C)NC(=O)CSc1n[nH]c(O)n1 CCCCCCC(=O)N1CCC(C(=O)NCC2CCN(C)C2)C1(C)C N1(C(CN(C(CC)=O)CC)=O)CCC2(CC1)CC2NC(=O)C=Cc1scnc1C Cc1cc(CC(N2CC(CN(C(=O)CNc3nc(C)cs3)C)C2)=O)cc(C)c1 c1(C(=O)NC2CN(C(C3CC=CCC3)=O)C3CC23)ccc2nc(S)oc2c1 n1(CC(=O)NCCc2c(CNC(C=CC(N)=O)=O)nco2)nc(Cl)ccc1=O C1(NC(c2cccc(CC)c2O)=O)CCC2(CC1)CC2NC(=O)CC(F)(F)CC CCCC(CC1CCCC1)C(=O)NCCCCCNC(C1CCCN1C1CC1)=O N1(CC)CN(c2nnc(CC(C)(C(C)C)c3ccc(C)cc3)n2C)C(C)CO1 N1(C(C(C)OCC#C)=O)CCC(C(C)NC(=O)CCc2nncs2)C1 c1(OC)cc(C(C)NC(C2OCCC2F)=O)ccc1OC(F)F C1C(CC(=O)O)NC(=O)N1.Cc1ncsc1CCOC(c1nn[nH]n1)C N1(C(=O)C(F)C2CC2)CCOC(CNC(C2(CF)CCC2)=O)C1 c1(-c2nc(-c3ccc(OCC)cc3)nn2C2CCC=CCCC2)nnc(O)cc1O N1(C(C2CCC(F)(F)C2)=O)CC2CN(Cc3ccc(I)cc3O)C2C1 c1(C(N(C(C)CNC(C2(c3cc[nH]n3)CC2)=O)C)=O)cc2c[nH]cnc-2n1 C1(C(=O)NC(C(C)NC(CCCNC(C)=O)=O)CO)CC2OC1C1CC21 C(=O)(C(O)CC(C)(C)C)N1C(CNC(C=CC(CC)=CC)=O)CCCC1 Cn1c(NC(c2cc(Cl)cc3cccnc23)=O)nc2c1CCN(CC(F)(F)F)C2 C1(C(=O)NC2C(NC(Cn3nc(C)n(C)c3=O)=O)C2)CC(C(C)(C)C)=NO1 N1(C(C2(CNC(C3(SC)CSC3)=O)CC(=C)C2)=O)CC(C)N(CC)C(C)C1 C(c1ccco1)=C(C)C(=O)NC1COCC1CNC(C1(CCN(C)C)CC1)=O c1(C(=O)NC2CN(C(CC(CC)C3CC3)=O)CC2O)ccc(C(F)(F)F)nc1C Clc1ccnc(N2CCCN(c3ccc(Br)cn3)CC2)c1Br C1(NCCN=C(NCC(CC)C)NCC)CCc2cc(OC(C)=O)ccc2C1 N1(C(C2C3CNC(=O)C32)=O)CC(C2CN(C(=O)CC34CCCN3CCC4)C2)C1 c1(CCNC(C(C)SC)=O)ccc(CNC(=O)C(C2CCCCC2)O)cc1 N12CCCC(CC1)CNC(=O)CC2=O.c1(C(=O)NCC(F)(F)F)ccc(C2CC2)o1 C1(NC(CC(=O)OCC)=O)CCN(C(=O)CC(C)N2CCCC2=O)C(C)C1 C1(C(N(CCOCCNC(C(=O)NCC)=O)C)=O)CC12CCOCC2 C(=O)(C1=NOC2(CCOC2)C1)NCC(C)CNC(=O)Cn1ccc(C(F)(F)F)n1 c1(Cc2nnc(CNC3C(NC(=O)OC(C)(C)C)CCC3)s2)ccc(F)cc1 C1(C(=O)NC2(C(=O)Nc3cnn(CC4CC4)c3)C(C)CCC2)CCOCC1(C)C c1(C2(NC(=O)NC)CC2)ccccc1.C(=O)(C(C)CC1CCCO1)N.C1(=O)CO1 C12(NC)CCC(C(=O)NCC3(CNC(c4c(C)ocn4)=O)CC34CCC4)(CC1)C2 C1(NC(c2nc(CC)sc2)=O)CC1C1CCN(C(=O)CC2=CCN(C)CC2)CC1 c1(CNC(C)=O)nnc2n1CCN(C(=O)C1=COCC1)C2.C1(C(C)C)C(=O)N1 c1(C(=O)NC2(C)CC(NC(=O)CCc3ccc[nH]3)C2)cc2cc(Br)ccc2s1 C1(N(C(C(C(C)C)SCc2ccccc2)=O)CC2CC2)CCOCC1(C)C N1(C(Cc2c(C)cco2)=O)CCC(C(C)NC(c2cn(CC3CC3)nn2)=O)CC1 C(CCC(=O)N1CC(=O)N(C)C(=O)C1)(C(C)C)NC(C1(OCC)CC1)=O CC1CCCc2nc(C(=O)NCC3=NOC4CN(C(C5CN(C)C5)=O)CC34)cn21 C1(C)(C(=O)NCCNC(N(C(C2CCC2)C)C)=O)CNC(=O)N1 C(=O)(C1CCC(=O)Nc2ccccc21)NC(CNC(C(C)C)=O)(C)C C1(C(N(C)Cc2c(C)ncs2)=O)CC(C)(C)CCN1C(C1CC1F)=O C(=O)(C(C)CCCC(C)C)N1C(C(N(CCCC)C)=O)C(CC)CC1 C1(NC(c2ccc(C)[nH]2)=O)CN(C(c2cc(C(C)(C)C)n[nH]2)=O)CC2(CC2)C1 C1(NC(C)=O)COCCN(C(=O)C(Cc2ccncn2)NC(=O)OC(C)(C)C)C1 C(=O)(C(O)C(F)(F)F)NCC1CCN(C(c2nccc(N)c2)=O)CC1 C1(N(C(C(C)(C2CCC2)NC(c2cccnc2O)=O)=O)C)CCCCCC1O c1(C(=O)NCC(CNC(C(CC)(C)C)=O)C)nn(-c2ccccc2)c2c1CCCC2 CC12CC(C(N3CC(NC(c4cccs4)=O)CC3(C)C)=O)(C1)C(C)(C)O2 Cc1oc(-c2cccs2)nc1C(=O)NCC(C1CC1)NC(c1csc(C(C)C)n1)=O C(=O)(C(O)CCCc1ccccc1)NC(c1ncc[nH]1)C C=CCC(CC=C)C(=O)OC(=O)CCc1nc(NC)no1 C1(NC(=O)NCCN2CCN(CC3(C)CC3(F)F)CC2)C2CCC(F)(F)C12 c1(NC(C2CC(=C)CN2Cc2cc(Br)cc(I)c2)=O)cc(O)nc(=O)n1CC CC1(C)CCCC(O)(C(=O)NC2CC3(C2)CC(CNC(=O)CN2CCC2)C3)C1 C1(F)(CNC(COCC=C)=O)CCN(C(=O)C(F)(Cl)c2ccccc2)CC1 c1(NC(=O)CCCN2CCCC2)ccc(C(=O)NC2(CC3CC3)CCCC2)cn1 Cc1cc(=NCC(CNC(=O)CC(O)CNC(N)=O)C(F)(F)F)[nH]c(Cl)n1 N1(C(CCC(=O)OCC)=O)CC(C(C)(C)C)CC(COCC)C1 C(=O)(C(C)C(O)C(C)C)NCCC(CNC(=O)Cc1cnns1)OC N1(C(c2nccnc2OC)=O)CC(C(N2CCC(F)(CF)C2)=O)C(F)(F)C1 N1(C(CCC)=O)CCN(CCCO)CC1.c1(C(=O)NCCC(=O)O)ccc(Cl)cc1 Cc1ccc(C(N2CCN(C(=O)C(c3cnccn3)C)CC2C(C)C)=O)nc1F C1(C(=O)NCCOC(CC)C)CN(C)CCN1C(=O)COCc1nc[nH]n1 N1(C(C(C)O)=O)C2CCC(C2)C1C(N1CCC(CNC(=O)C(C)C)C1)=O CCCCC(O)CC(=O)NCC1CCC(NC(c2sc(N(C)CC)nc2Cl)=O)C1 N1(C(CN2CCN(C(C3(OC)CCC(C)C3)=O)CC2)=O)Cc2nc(C)sc2C1 CC1CCN(CCC(=O)NC2CCCC2NC(=O)CCc2nccs2)CC1 c1(CNC(=O)Oc2ccccc2)cccc(C#N)c1.CC1=CC(=O)OCC1 Cc1ccc(O)c(CNC(c2ccc(CNC(=O)C(C)c3ccco3)cc2)=O)c1 Cc1noc(C(=O)NCC(C2CCCN2C(=O)CN(C)C)(C)C)c1C c1(CNC(C2(CC=C)CCN(C(C3CC=CCC3)=O)C2)=O)ccc(F)c(O)c1 c1(C(N(C2CCCC2CCCF)C)=O)cccc(C(C)(C)C)n1 c1(OCC(=O)NC(C)CC(C)NC(C2(n3cnnn3)CC2)=O)cccc(F)c1 c1(CC)csc(CCC(N2CC(C)(NC(=O)C(C)Cc3ccco3)C2)=O)n1 C1(O)(C(N2CC(OCCNC(C3CCC3)=O)C2)=O)CC2CCC1C2.C1(CN)CC1 c1(CN(C(=O)CC2CC3(CC3)CO2)C)ccc(CNC(C2CCSC2)=O)cc1 Cn1nc(C(=O)NC(CNC(=O)Cn2cnc(C(F)(F)F)c2)CO)c(Br)n1 C(C(C)N=c1[nH]c(=NCCCN2CCCC2=O)[nH]c2c1SCC2)n1c(C)ncc1 C(=O)(C1=Cc2ccccc2C1)NC(CCN(C)C)C(=O)NCCS(C)(=O)=O c1(OC)cc(C(C)N(CC(=O)N(c2ccc(OC(C)=O)cc2)C)C2CC2)ccc1O N1(C(C2(CCOC)CCCC2)=O)CCCC(NC(C2(CF)CC2)=O)C1C C1(NC(c2cncc(OC)c2)=O)C2CCN(C(c3nccn3C)=O)CCC12 Nc1cc(F)c(F)cc1C(N1CC(CF)OC(C(F)(F)F)C1)=O.C12CN(C1)OC2=O C(=O)(C(=O)N=S(C)(C)=O)NCC1C(C)CN(C(C2CN3CCC2CC3)=O)CC1 C(=O)(CCCS(C)(=O)=O)N1CCN(C(C2(c3c(OC)cccc3)CC2)=O)CC1CO CC(C(=O)NCC1C2CC1N(C(=O)CN1CC3CC3C1)C2)C(F)(F)F c1(NC(C2C(O)CCN(C(c3c(C)nc(Cl)cc3)=O)C2)=O)cnc(C#N)c(Br)c1 c1(N(C)C)cc(C(=O)NCCNC(C2(n3ccnn3)CC2)=O)cc(C#N)c1 c1(C(=O)NCC2CC(OC)CN2C(c2ccc(C)cn2)=O)c(C)ccnc1C N1(C(C2C(NC(=O)OC(C)(C)C)C2)=O)CCN(C(=O)C(O)C(F)(F)F)C(CCO)C1 C(=O)(C#CC(C)(C)O)N1CC(C(C)NC(c2cnc(Cl)s2)=O)OCC1 C1(SCC)CCN(C(=O)C(C(=O)Nc2ccc(NC(C)=O)cc2)NC(C)=O)CC1 C12(NC(C(CC(C)C)N(C(c3c(OC)cncn3)=O)C)=O)CC1COC21CCC1 C(C(O)C(=O)NC1CC1C(F)(F)F)NC(CCNC(COC)=O)=O C(c1ccc(F)cc1)=CC(N1CCCC(CN(C(CCC=C=C)=O)C)C1)=O C1(CNC(c2ccc(C)[nH]2)=O)CCCC2(CN(C(=O)C(F)=CCCF)C2)O1 C1(C(=O)NC2CC(O)C23CCC3)CCc2nnnn2CC1 N1(C(CCOC(C)C)=O)CCCN(C(c2cccnc2Cl)=O)CCC1 c1(C(N2CCN(C(c3cnc(Cl)[nH]3)=O)CC2)=O)cc(C(F)(F)F)nc(C2CC2)c1 c1(C(=O)NCC(C2CC2)NC(C(CC)C(=O)OC)=O)ccc(Cl)c2ccccc12 CC(C)(CC(F)(F)F)C(=O)N1CC(O)(CCNC(c2ccn(CC#N)n2)=O)C1 C(=O)(C1=NNC(=O)C1)NCc1c(N(C)C)ccnc1.N12CCCC1C2=O C12(CC(N3CCN(CCCNC(C4CC(CC)C4)=O)CC3)=O)CCC(CC1)CC2 c1(C(CNC(c2ccccc2-c2ccncc2)C)O)ccc(-n2cnnc2)cc1 N1(C(c2n(CC)ncc2Cl)=O)CCC(C(C)C)CC1CNC(C1CC(F)(F)C1)=O N1(C(c2cc(C(C)C)on2)=O)CC2CCC1C(NC(=O)CCc1cn[nH]c1)C2 c1(COC)cccc(C(N2CC3C(Nc4ncccn4)C3C2)=O)c1C CCC(C)(C)C(C)CC(=O)NC1(CNc2ncc3ncnc-3[nH]2)CC1 Cc1cc(CNC(C2COC(CNC(=O)C(C)(C)c3ccsc3)C2)=O)ccn1 N1(C(C2CC2[N+](=O)[O-])=O)CCCN(C(c2cccn(C3CCC3)c2=O)=O)CCC1 Cc1ccc(Cl)c(O)c1C(=O)NCC1CC1CNC(C1CC2(C1)CC1(CC1)C2)=O C1(NC(CCN(CCC)C)=O)CC1C1CCCN(C(c2cc(C)nc(O)n2)=O)C1 N1(C(c2c(C)cncc2)=O)CCCOC(CNC(=O)C=Cc2ccsc2)C1 Cc1ccc(C(=O)NC2CN(C(C3(n4cccn4)CC3)=O)CC(F)(F)C2)c(F)c1F c1(C(CNC(C2OCC2(C)C)=O)NC(C=CC)=O)ccccc1F CN(CCCC(=O)NCc1nnc(O)nc1O)N=O CCC(CC(=O)NCCCCCCN(C)C)NC(=O)C(C1CCOC1)OC C1(C(N2C(C)CCC2)=O)CC2CCCCCC12.N1(C(=O)C2CC2)CCC1 c1(C(=O)NC23CCN(C(=O)Cc4cnns4)CC2C3)nccn2ccnc12 N12CCN(C)CC1C(=O)NCCn1nncc1C2=O.C1(CC)C2CCCCCC12 C12(NC(C3C(C)C3)=O)CC3CCC(C1C2)N3C(c1cc(C#N)ccc1Cl)=O c1(C(=O)NC2C(CC)CN(C(c3cc(SC)oc3C)=O)C2)ccc(F)c(O)c1F N1(C(c2nc(C)oc2C)=O)CC(C(=O)NCc2nc(C3CC3)n[nH]2)CCC1C c1(C(=O)NC(CNC(c2c(O)ccc(C)c2)=O)C)cn2cc(Cl)cnc2n1 CC1(C)CC1(NC(=O)CCOC1CC(C(=O)NCC2(F)CC2)C1)CO CCC(C)CN=c1cc(C)c(OC(F)(F)F)n[nH]1 O=C(C1CCCn2ccnc21)NC1CC2(CCN(C(C3CC3(F)F)=O)CC2)C1 c1(CC(N2C(C(=O)NCc3ncc(F)cn3)CC(O)C2)=O)ccccc1[N+](=O)[O-] c1(OCC)cc(C)nc(CO)n1.C1(N2C3(COC3)C2)CCOC(C)C1 C1(C(C)NC(=O)C(F)(F)c2nccn2C)CCN(C(=O)C(O)CC2CC2)CC1 N1(C(C2CC(=O)NC2)=O)CC(NC(c2cccc3ccsc23)=O)C(N=[N+]=[N-])C1 c1(COC)ccc(C(=O)NCC(CCOC)NC(c2ncoc2)=O)s1.C1CC1 c1(C(=O)NCC2CC2)cccc(O)n1.S(=O)(=O)(C1CC1)NC.C12(CCC1)C(=O)NC2 c1(C(=O)NCCN(C(C(C(=O)OC)C)=O)C)c[nH]nc1S(N)(=O)=O C1(C(=O)NCC2(SC)CC2)CCC(C)CC1.C12(C)CN(C1)C2=O Cc1cnc(CCNC(C2C=CC(NC(C3CCSC3)=O)C2)=O)cn1 C(=O)(CCCCN(C)C)NCC(CC=C)NC(=O)C(F)(F)C1(OC)CCC1 Cc1ccccc1CCC(=O)NCCN(C(=O)C(C)(C)Oc1cccc(Cl)c1)C C(=O)(CC(C)(C)CCOC)N(C1(C)CCCC1C)NC(C=CCC)=O c1(C(N(CCC(C)NC(c2nc(C)oc2)=O)C)=O)cnc2n1C(C)CCC2 N1(C(CN(C)C)=O)CC=C(CNC(C2CC(=O)N(CCCC3CC3)C2)=O)CC1 CC(C)C(=O)NNC(=O)c1ccc(-n2cc(C(N(C3CC3)C(C)C)C)nn2)cc1 c1(NC2CC(N(C(C)C(=O)Nc3ccccc3C#N)C)C2)ncnc2[nH]cnc12 Cc1ccc(-c2cccc(CN3CCOC4CCCNC34)n2)c([N+](=O)[O-])c1 C1(CC)CNC(=O)CN1C(=O)CC1CCN(C(=O)C(CC)N(C)C)C1 N1(CC(N2CCCC2Cn2cc(C3CC3)nn2)=O)CCOCC1CC1CCC1 N#Cc1ccc(-c2cncc(NC(c3ccsn3)=O)c2)nc1 c1(CNC(CC2(C)CN(C(c3cc(Cl)cnc3F)=O)C2)=O)cccc2ccoc12 C1(C(=O)NCC(C)CNC(=O)Cc2ccsc2)CC2CCC2C1 C(CCSC)(C(=O)NC(CCNC(c1c[nH]nc1C1CC1)=O)C(C)C)OC C1(NC(Cc2ccc(C)cc2)=O)CC(OCCNC(=O)COC(F)F)C12CCC2 C(=O)(CCCC(=O)NCC(C)(C)NC(c1c[nH]nc1Br)=O)NCC c1(NC(C2N(Cc3cc(C)n(C)n3)CCSC2)=O)c2c(nn1C)CCC2 c1(C(=O)NC2(CCCNC(C3CCCS3)=O)CC2)ccnc(CO)c1 C1(N(C(C2(NC(c3ccc(C)s3)=O)CCSC2)=O)C)CCN(C)C(C)C1 N(C1CCOc2c(Br)cccc21)C(CN1C(=O)C(C2CC2)CCC1)=O CC1CC(NC(c2ccc([N+](=O)[O-])[nH]2)=O)CN(C(c2ccccc2)=O)C1 C1(C(N(CCNC(c2cc(COC)on2)=O)C)=O)CCN2CCC1C2 C(=O)(CCC(C)(F)F)NCCN(CCC)C(c1cc(Br)cnc1O)=O C1(CNC(c2cocn2)=O)CCCC12CCN(C(C1CC3CCC1O3)=O)CC2 N1(C(C(C(C)(C)O)F)=O)CCC2(CCCN2C(=O)COCC(F)F)CC1 C(C(C)(C(=O)NC1CCCN(C(=O)C(F)F)C1)OC)OC N1(CCCC(=O)NC(c2cn(C3CCOCC3)nn2)C)CCCCC1 C1(OC)CN(C(=O)C=CC(C)N)C2(CCCC2)C1 Cc1cccc(S(=O)(=O)N(C2CC2c2ccccc2)Cc2nnn(C(C)(C)C)n2)c1Cl c1(OC)c(F)cc(CNC(=O)C(c2cccc([N+](=O)[O-])c2)C)cc1F Cc1c(Cl)cc(C(=O)NC2CCC(C(=O)Nc3ncc(F)cc3Cl)CC2)cc1Cl c1(C(=O)NCC(CC=C)NC(=O)CC(C)COC)cc(C(F)F)ccc1F N1(C(c2nc(COC)sc2)=O)CCCC2(NC(=O)C=CSC)CC2C1 C(CC(C(C)(C)C)NC(=O)C=CC(F)F)N(C)C(C1CCCOC1)=O C1(NC(N2CCCC(C)C2)=O)CC12CCN(C(C1(CC3CC3)CCC1)=O)CC2 C1(CNC(=O)OC(C)(C)C)CC(NC2CCC=CO2)C2CC12 c1(C(=O)NCCC2CC(NC(c3csc(Cl)c3)=O)C2)coc2c(F)cc(Cl)cc12 Cc1ccc(OCC(=O)N(C)C)c(C)c1.C12CCN1C(=O)C(=O)NC2.C1CN1 C(=O)(C(CC(F)F)N(C(=O)C(O)CC1CCCC1)C)NCCc1ncc(C)o1 C(CC1c2ccccc2CCN1c1nnc(C#N)s1)NC(C(C)(C)O)=O c1(NC(C(C(C)O)NC(C2C(C(=O)OC)CC2)=O)=O)cccc(C#N)c1 c1(C(=O)NCC2CC(NC(c3nc(C)c(Br)cc3)=O)C2)cc(Cl)c(Cl)cc1F N1(C(CC2(N(C(c3c(C)ocn3)=O)C)CC2)=O)CC2CN(C)CC2(C)C1 N1(C(c2c(C(=O)OC)c[nH]c2)=O)CCN(C(=O)Cn2cncc2C)C(C2CC2)C1 CCC(O)C(C)C(=O)N(c1ncc(I)cn1)C1CCCNCC1 Cc1[nH]nc2cc(C(N3CCC(C)(NC(=O)CCc4ccccc4)C3)=O)ccc12 C=CC(C)(C)CC(=O)NCC(C1CCCC1)NC(C1CCC(F)(F)CO1)=O c1(-n2cc(C(C)NC(c3c(CC)scn3)=O)nn2)cc(Cl)cc(Cl)c1 N1(C(C(N)Cc2cocn2)=O)CCCCC1c1ncc(-c2ccccc2)[nH]1 N1(C(C2CCCC2CNC(C2(n3cncn3)CC2)=O)=O)C(CO)CC2COCC12 Cc1cc(C(=O)N(C2CCN(C(=O)C=Cc3cccc(Cl)c3)C2)C)cc(C)n1 C12(CNC(C(CCCC)O)=O)CCC(CNC(=O)C(C3CC3)SCC)(CC1)OC2 c1(OC(C)C)ccc(C(O)C(C)NCC(n2nccn2)C)cc1 N#CC1CCC(C(N2CC(F)(C(N3CCOC(CC(N)=O)C3)=O)C2)=O)CC1 c1(C(=O)NC2CN(C(c3c(C)snc3)=O)C(C)C2)cc(O)c2ccoc2c1 C1(NC(c2cncnc2)=O)CC(O)CN(C(c2ccc(-c3ccccc3)o2)=O)C1 c1(CCNC(=O)NC(CCC)C2CC2)c(Cl)cccc1Cl CC(C)CC(=O)NC1CC1CNC(c1cnoc1)=O N1(C(C(CCC)CCC)=O)CCCCC2(CCN(C(c3cnoc3)=O)C2)C1 Cc1cc(C)c(NC(=O)C(N2CC3CN(C)CC3C2)COC(C)(C)C)c(C)c1 N1(C(C2CCC(N(C)C)C2)=O)CCN(C(c2csc3nccn23)=O)C(C2CC2)C1 CC1CNc2c(C(N3CCN(C(C4(N5CCOCC5)CC4)=O)CC3)=O)cnn2C1 C1(CC=C)(NC(c2cc(C)nn2C)=O)CCN(C(=O)C(C#N)C2CC2)C1 CC1CC(NC(=O)CC23COCC(C2)C3)CCN1C(C1CCCN1C)=O CC1CC=C(C(=O)NCCC23CCC2CN(C(=O)Cn2cc(Cl)cn2)C3)CC1 Cc1cc(C(=O)NCCN(C(C2CC(C(C)C)C2)=O)C(C)C)c(C)n1-c1nccs1 N1(C(COCCCOC)=O)CC2(C1)SCCC2NC(c1cccc2nnnn12)=O c1(NC(C2CCCCN2C(c2cc(O)nc(Cl)c2)=O)C)ncnc2scc(Br)c12 c1(CNC(N2CC3C(F)(F)C3C2)=O)cncc2ccsc12.c12c[nH]nc1CN2 C1(C(=O)NCC2CN(C(C3(C)CCCO3)=O)CC2O)CC2(CCC(F)(F)CC2)C1 C(C(C)C)(C(O)C(=O)N1CC(C(C(=O)N(C)Cc2occc2C)OC)C1)OC CC(O)C(C)(C)C(=O)NCC=C1CCN(C(c2ccoc2)=O)CC1.C1(N)(C)CC1 C1(CNC(c2c(C)n[nH]c2)=O)C2CN(C(=O)C(=O)C(C)C)CC12 c1nc(=NCCOCCO)[nH]c2ccccc12.N(C1Cc2ccccc21)CCOC c1(C2C(CC)CC2)nc(-c2ccc(C(F)(F)F)cc2)nn1CCOC C(=O)(C(CC)(CC)CCC)NCCCC1(CNC(CC(C=C)C)=O)CCCC1 c1(OC(C)C)cccc(C(=O)NCCC(C(C)C)NC(=O)CC2COC(=O)C2)c1 N1(C(C(CCC)=CCC)=O)CCOCC(CNC(c2cccc(OC)n2)=O)C1 NCCC(CN1CC(Nc2ccc(OC(F)(F)CF)cc2)C1)CO C(=O)(C(F)(F)F)NCC(=O)N(C1CCN(C(C2(C)CCC2)=O)C1)C n1(CC)cc(Cl)c(NC(=O)C(N)C(C)OCc2ccccc2)n1 N1(C(N(c2sncc2Br)C)=O)CCCC(c2cccnc2)C1 CCC(COC)C(=O)NCC(C)(C(C)C)NC(c1cc(CC(C)C)[nH]n1)=O c1(OC)ccc(C(C)C(=O)NC(C2CCCN2C(C2SCCS2)=O)C)cc1F c1(C(=O)NC2C(CN(C)C(C3(O)CCCC3)=O)CCC2)ccnn1CC(F)F Cc1cc(CNC(C2CN(C(=O)CSCC(N)=O)CC2(C)C)=O)nnc1C c1(C(=O)NC(c2ccccc2F)CNC(CCC=C)=O)ccc(OC)c(Cl)n1 c1(C(N2CC(NC(C3(COC)CC3)=O)C(F)CC2)=O)c(Cl)ccc(O)c1Cl c12cccc(c1)N2.O=C(C(F)=C1CCCC1)N(C(=O)CN(CC(F)(F)F)C)CCF C1(NC(CN(C)C)=O)CCN(C(c2ccc(N)c(Cl)c2O)=O)CC1(C)C c1(C(=O)NCC2N(C(c3cncc(N)n3)=O)CCC2)cc2occc2s1 Cc1nc(F)ccc1-c1cn(CC(=O)NC2CC23CCOCC3)nn1 c1(C(N2C(CNC(=O)CN3CSCC3=O)CC2)=O)ccc(Cl)cc1F Cc1cccc(NC(=O)CN2CCN(CC(F)F)CC2)c1 C(=O)(CCCCCn1cnnn1)N(C1CC(NC(C2OC3CCC2C3)=O)C1)C Cc1cnn(C)c1CC(=O)NCCCC(C)NC(c1cnsn1)=O C1(CNC(CCNC(COC)=O)=O)CC2CCC1N2C(c1cc(Cl)cs1)=O C1(NC(CNC(CCC#C)=O)=O)CCC2(CC1)CN(C(=O)C(C)CO)CCO2 C(CCCC(=O)N(C(C)CCNC(C1CCC12CCC2)=O)C)N(C(C)=O)C C1(N(C(C(C)CF)=O)C)CC(N=c2cc(C#N)nc(C(C)C)[nH]2)C1 C1(C(=O)NC(c2ccncc2)C)CCCC12CCN(C(=O)C1=CCCCO1)C2 C1(=CCNC(c2cn(CC)nc2)=O)CCN(C(=O)C(C)C2CCCC2)CC1 c1(CCNC(C(=O)N(CCF)Cc2cccc(OC)c2)=O)cc(F)ccc1Cl c1(OCC)cc(CCC(C(=O)NC)N(C)CCC2CCC(N)C2)ccc1O C1(C(NOCC(=O)OC)=O)CN(C(c2ccn(C)c2)=O)CC1(F)F c1(CC(=O)N(CC(C)(C)NC(=O)CC2CC3CCC2C3)C)ccc2sccc2c1 c1(CC)cccc(S(=O)(=O)N2CC3CN(C(c4cccnn4)=O)CC3C2)c1 c1(C(=O)NCc2occ(C(=O)NC3(CC)CCCC3)c2)cn(CCF)nc1C c1(C(=O)NCCN(C(=O)Cc2ccccc2CC)CCC)ccnnc1O C1(NC(CC(C)N(C)C)=O)Cc2nccnc2CN1C(=O)CCc1ccccc1 N1(C(C2CCN(CC)C2)=O)CC(F)(F)CC1C(N1CCC(C)(O)C1)=O c1(N2C(CNC(c3c(OCC)cccc3)=O)CCCC2)nc2ncc(Cl)cc2o1 C1(C(N2CC3CCC(C(N4CCCCCC4CO)=O)(C3)C2)=O)Cc2ccccc2C1 N1(C(C2(CC(C)C)CCC2)=O)CCC(C(C)(C)NC(=O)C=CC=C(Cl)Cl)CC1 C(=O)(C1=CN(C(=O)OC(C)(C)C)CC1)NCC(CCNC(C(CC)CC)=O)O C12(CNC(CS(=O)(=O)NC)=O)CCCCC1N(C(c1cc(OC)n[nH]1)=O)CCC2 Cc1cc(NC(=O)C(CO)NC(C2(C)CCOCC2)=O)cnc1O c1(CNC2C(C)CN(C(=O)C(C)(F)F)C2)c[nH]c2cccc(C#N)c12 CC1CC(C(=O)NCCN(C)C2CC2)CN(C(=O)Cn2cnnc2O)C1 c1(CC(N2CCC(CNC(c3[nH]cc(CC)c3)=O)C2)=O)cccc(CC)c1 c1(C(C(=O)NCC2(CNC(CCSC)=O)CC2)C)cc(C)cc(F)c1 Cc1[nH]nc(Cl)c1C(=O)NCC1(C(N)=O)CN(C(C2CCO2)=O)C1 C(CC(C)C(C)(C)C)NC(C1C(CNC(C(c2ccn(C)c2)C)=O)CCO1)=O C1(CCC)CCCCC1N=c1[nH]c(=NCCC2CC2)c2sccc2[nH]1 Cc1ccsc1C(=O)NC(C(=O)NCC(C)C)c1ccco1 c1(C(C(=O)NCCNC(C2(CNC(=O)C(F)F)CC2)=O)(F)F)nc2ccccc2s1 c1(SC)nc(O)nc(C)c1C(N1CCCC(NC(C2C=CCC2)=O)C1)=O C1(CNC(C2(C(F)F)CC(=C)C2)=O)C2CN(C(C3CCC=CCC3)=O)CC12 C1(C(=O)NCc2cccc(C)c2)CCC2CCC1N2C(c1noc(C(C)C)n1)=O N1(C(C2CN(CCC)C(=O)C2)=O)CCN(C(=O)Cn2cnc(=N)[nH]2)CC2(CC2)C1 C(=O)(N=c1cc(-c2ccc(Br)cc2)[nH][nH]1)C1CCC(CC)O1 C(C(C(=O)NC1CCC(C(C)O)CC1)C(C)(C)C)NC(Cc1c(C)ccs1)=O c1(CC(=O)OCCOCCn2cc(Br)c(O)nc2=O)cc(F)c(Cl)cc1Cl C(C)(C(=O)NC1CC(N(C)C(c2cnoc2-c2ccoc2)=O)C1)(C1CC1)OC CCC(C)CCC(=O)NCC(C)(C)CNC(c1cc(C2CCC2)ccc1F)=O C1(C(N2C(CNC(c3cc(O)ncn3)=O)COCC2)=O)CC12CCCCC2 C12(C(N3CCC(N(C(CC=C(C)C)=O)C)C3)=O)CC1COC2(C)C C(=O)(CN=c1cc[nH]cc1)N1C2C(NC(C=CC)=O)(CCC2)CC1 C=C(C)C1OCCC1C(N1CCCC1C(=O)N(CC)Cc1cccc(C)c1)=O C1(CC(=O)N(CCCC)C2CC2)CN(C(=O)OC(C)(C)C)C(C)(C)C1 C1(N(C)C)CCC(C(N2CCC2C(=O)NCC2CCC2(F)F)=O)CC1 N1(C(c2cc(NCc3cc(OCC)ncc3)cn2C)=O)CCOC(C#N)C1 N1(C(CCNC(=O)OCC)=O)CCC(C2CC2)(NC(=O)CCCOC)C1 N1(C(CC(=C)C)=O)C2CCC1C(C)C(NC(c1ccn(CCC)n1)=O)C2 N1(CC)CCC(NC(=O)CCC2CCN(C(C3CC3C(F)F)=O)CC2)C(C)C1 CC1CCCCN1CC(=O)NC1(NC(C2CCC2C(C)(C)C)=O)CCOCC1 C1(C(N(C(C)C(=O)NC2(CC(=O)OC)CC2)CCC)=O)CCCC(=O)C1 C(=O)(C1=CC2(CCOC2)C1)N1CCC(C)(CNC(C2=C(C)CCC2)=O)C1 c1(OC)ncc(C=CC(N2CCN(C(C34COCC(C3)C4)=O)C(C)C2)=O)cn1 c1(N2CCC(C)(O)C2)cc2c(I)cnc-2[nH]n1.C=O CC(C)C(O)CC(=O)NC(C)(C)CC=CC(N1CC(C(=O)N(C)C)C1)=O c1(C(=O)NCC2(OC)CN(C(C3CCCC(C)O3)=O)C2)cccnc1C(F)F C=CCC(CNC(=O)C(C)(C(C)C)OC)C(=O)N(CC(C)(C)O)C c1(CCOCC(C)SC)ncco1 C1(C(=O)NCC(=C)Cl)CCC(C2CC2)N1C(c1cc(C)co1)=O N1(C(C=Cc2cnc(C)s2)=O)CCCC(NC(c2c(CO)noc2C)=O)C1C c1(CCCC)ccc(C(=O)NC(C)C(C(C)C)NC(=O)Cc2cncn2C)cc1 C1(=O)C(C(=O)N)CNCC(CC)N1.C1(CSC)CC1.C(C)(C)(C)OC(NC)=O CCCCC(CC)CC(=O)NC(CCCNC(c1ccon1)=O)c1ccccc1 C#Cc1cc(C(N2CC(C)CCC2CNC(=O)C(C)(F)F)=O)cc(Cl)c1 N1(C(c2c(C)n[nH]c2C)=O)CCN(C(=O)Cc2ccc3nn[nH]c3c2)C2CCC12 c1(COC)cncc(C(=O)NC(CCN(C(C2(OC)CCOC2)=O)C)(C)C)c1 c1(CNCC2CC(OC(CC)C)CC2OC)ccc(C(=O)OC)nc1 CCN=C(NC(C1CCCN(C)C1)C1CC1)NCC1CC1c1ccccc1 c1(C(=O)NC(C(C)C)CNC(=O)C(C)CC(N)=O)cc(F)cc(Cl)c1N N1(C(c2cc(COC)no2)=O)CC2CCCC(C1)N2C(C1CCOC(=O)CC1)=O C1(C(=O)NCC2C3CN(C(C4CC(=C)C4)=O)C2C3)CCc2nnc(C(C)C)n2C1 c1(C(N(C(CNC(C(C)=CC)=O)C2CC2)C)=O)ccccc1Sc1nc[nH]n1 Cc1cncc(C(=O)NCCSCC(=O)NCC2CC(C#N)C2)n1 C1(C(=O)NCCOCCCC)CCCCCCN1C(C1CC=CC1)=O C1(CC=C)(NC(c2nccn2C)=O)CN(C(=O)Cn2nccc2C)C1 c1(C(N2CC(NC(=O)CC3NC(=O)NC3=O)CC(C)C2)=O)cccc2scnc12 Cc1ncc(C(N2CCC2CNC(C2C3CCN2CC3)=O)=O)c(O)n1 c1(C(N2CC(N(C(C3N(S(C)(=O)=O)CCOC3)=O)CC)C2)=O)cnc2[nH]cnc2c1 Cc1c(NC(C2CC2NCc2cc(O)cc(F)c2)=O)cccc1Cl Cn1ccc2cc(C(N3CC4CN(C(c5cccc(Cl)c5F)=O)C4C3)=O)ccc12 C(=O)(CN=c1ccc(C#N)c[nH]1)NC1(CO)CCCN(C(c2cc(C)ns2)=O)C1 C(C(=O)NCCn1cc(C(=O)Nc2cccc(F)c2O)cn1)(C(C)(C)C)N(C)C c1(CC)nc(C)cc(=NCC2CCN(C(=O)Cc3c(C)nn(C)c3C)C2)[nH]1 N1(C(c2cnn(CCF)c2)=O)CCCC(CCC(N2CCC(CC3CC3)CC2)=O)C1 C(=O)(CC(C(F)F)NC(C1CC1C)=O)NCCC1C(C)(C)OCC1.OC(=N)O c1(OC)ccccc1C(=O)NC1CCOC1C(N1CCSCC1C)=O C1(CNC(=O)Cn2[nH]cnc2=N)CCN(C(c2ccc(Br)o2)=O)C12CC2 O=C(C1=CCCCCC1)N1CC(CC(F)C(=O)NCC=Cc2ncc[nH]2)C1 c1(-c2cn(CC3N(C(CCCc4ncc(C)s4)=O)CCC3)nn2)cncc(Cl)c1 c1(C(N2CC(OCCNC(CCc3n(C)ccn3)=O)C2)=O)ccccc1Cl C1(NC(c2c(C)ocn2)=O)CCCCN(C(c2cc(OC(F)F)n(C)n2)=O)C1 c1(OC)ccc(CNCC2CC(OC)C2)c(Br)c1OC S(=O)(=O)(c1ccc(NCCC(F)F)nc1)NC(c1nc(C)oc1C)C c1(CC)ccc(F)c(C(=O)NCC(O)CNC(C2(C)CC(C3CC3)=NO2)=O)c1F N1(C(c2c(C)cc(Br)c(F)c2)C(=O)NCCC#N)CCN2CCCC2C12CCC2 C(=O)(C1CCCc2ncnn21)N1CCC(NC(CCCCCC=C)=O)C12CCC2 c1(COCCNC(=O)NCC2(F)CCOC2)ccccc1Cl Cn1[nH]c(=NC(c2ccccc2)C2CC3(CC3)C2)c([N+](=O)[O-])c1C(=O)O c1(CN(C(=O)CSCC2(C(=O)NCC)CCCNC2=O)CC)ccc(F)cc1 c1(OC)cccc(OC)c1CN1CC(O)CC1C(N1CCS(=O)(=O)CC1)=O CC(C)CCCC(C)C(=O)NC(C(=O)NCCOC1CC1(F)F)C1CC1 N1(C(c2c(C)noc2C)=O)CC2CN(C(C3CCN3S(C)(=O)=O)=O)CC2(C)C1 CC(C)C(N)C(=O)NCC(=O)Nc1n[nH]c(C(C)(C)C)n1 CC1=C(C(=O)NCC(C)CNC(C2(F)CCOC2C)=O)Cn2ncnc2N1C Cc1nc(C(C)C)[nH]c(=NC(C)C2CCCCN(C(=O)CC3CCCO3)C2)c1Br C1(CC(C)(C)C)CN(C(c2ccc(CCN)cc2)=O)CCN1Cc1cccnc1 CC1(C)CCCN(C(=O)CSC(F)F)C1CNC(c1csc(C2CC2)n1)=O c1(CNC(C(CSC)(C)NC(=O)CCOC2CCC2)=O)ccc(C)c(C#N)c1 N1(CC(=O)NC2C(NC(C(C(C)C)F)=O)CCCC2)C(=O)NC2(CCCC2)C1=O CC1=C(C)CC(C)(N(C(=O)CC2C3CCC(C3)N2C(=O)C(C)(C)O)C2CC2)CC1 C1(CC=O)CCCCC1(F)F.C1(CN(C(=O)C(C)OC)C(C)C)CCCCO1 c1(C(=O)NCC2CC3(CN(C(C4C(C)C4)=O)C3)C2)cc2n(n1)CCNS2(=O)=O C1(N(C2(C(N(C)OCC(F)(F)F)=O)CCC2)CC=CC)CCC=CCC1 C1(NC(C(C)(C)N2CCCC2)=O)CC2CC(NC(C3(C)CCC(=O)NC3)=O)CC12 C(=O)(CCC(C)(C)[N+](=O)[O-])N1C(CNC(C(c2ccccc2)C)=O)CC(C)(C)C1 C1(C(=O)NCC(CNC(CC2N(C(C)C)CCC2)=O)(C)F)CC2(CCCC2)CO1 C1(C(=O)Nc2c(C)cc(Br)c(N)c2)CCc2c(nnn2C)C1 n1(CC(=O)N(C)CC2CCN(C(C(COC)(C)O)=O)CC2)cnc([N+](=O)[O-])c1 C1(C(=O)NC(CNC(C2=CC(C)(C)C2)=O)(C)C2CC2)CNC(=O)CC12CCC2 C(=O)(C#CC1(CCC)COC1)N1CCN(C(C2C(=C)C2)=O)CC1CC c1(CC)c(-c2nc(COC)no2)sc(C)c1Br.N12CCCC(C1)C2=O C1(C)(CNC(C(COCC)n2cc(-c3cncnc3)nn2)=O)CC2(CCC2)C1 CC(C)(C)C(CNC(=O)CCCC1CCCC(=O)N1)NC(=O)Cn1nccn1 N1(C(C(C)NC(CC)=O)=O)CCC(C)CC1C(=O)Nc1ccccc1CC C=CCC(C(=O)N1CCN(C(C)CNC(c2ncccc2O)=O)CC1)OC c1(OC)cc(C(=O)NC(C)CCNC(c2ccccn2)=O)on1 N1(CC(N2CC(OCC(=O)NC(c3cscn3)C)C2)=O)CCOCC1=O C(=O)(CCC(C)(F)F)NCC(CNC(c1csc(Cc2ccccc2)n1)=O)OC c1(C(N(C(CCNC(COC(C)=O)=O)C)C)=O)cc(=O)c(C)c[nH]1 CC1(C)C2CC1C(=O)N2.c1(CN(C(c2cnns2)=O)C2CC2)ccc(F)cc1 c1(N2CCCCC(NC(CCC#CC)=O)C2)ncnc2cc(C(C)C)nn12 S(=O)(=O)(c1ccccc1Cl)N1CC(C(N2CCC(C)(C#N)C2)=O)C(F)(F)CC1 C(C(=O)NCc1cc(C(=O)NCC2(CO)CCC2)n(C)n1)(C(C)C)SC N1(C(C2CCN(C(CNC(C)=O)=O)C2C(C)C)=O)CCCNC(=O)C1 C#Cc1cn(C)nc1C(=O)NCCCOCCNC(c1cnc(C(F)F)nc1)=O C1(CC(F)F)C(=O)N1.CCC(CC=O)SC.C1C(=O)N1C.C(C(F)F)N c1(C(=O)NC2CCCC2NC(C2C(F)(F)C23CC3)=O)c(F)ccc(F)c1F C(C)(C(CO)NC(c1cc(-c2ccccc2)[nH]n1)=O)NC(C1(CSC)CC1)=O c1(C(N2CC(C)C(NC(=O)Cc3nccs3)C2)=O)nc2ccccc2nc1O C1(O)(CNC(Cc2cccc(OC)c2OC)=O)CCCN(C(=O)CC(C)F)CC1 N1(C(C(C2CCC2)OC)=O)CCCN(C(c2c(F)cc(Cl)cc2F)=O)CC1CO c1(COC)cc(C(=O)OCCCCn2ccnc2)ccc1O CC(CC(F)F)C(=O)N(CCNC(C1(C2CCCO2)CC1)=O)C1CC1 N1(C(CC2CCC(=O)O2)=O)CCN(C(c2ccc(F)o2)=O)CC1CO N1(NC(=NCC)NCCC2CCCCO2)CC2CCC(C(N)=O)(C2)C1 N1(C(c2cncc(N)c2)=O)CC2(CCCC(CNC(=O)Cn3ncnn3)O2)C1 CCC(COC)(CC)C(=O)NCC(C)CN(C)C(c1cccc(C2CC2)c1)=O C=CC1(CC(=O)NCC2(O)CN(C)C2)CN(C(C2(NC(C)=O)CC2)=O)C1 N1(CC)CC(NC(=O)CNC(c2c(C)nn(C)c2N)=O)CCC1=O c1(C(=O)NC2(C(C)O)CC2)c([N+](=O)[O-])cnn1C c1(C(=O)NCC2N(C(C(CC)N(CC)CC)=O)CC(OC)C2)cncc(Cl)c1C c1(CC(=O)N(C2C3CN(C(C(CC(=C)C)C)=O)CC32)C)cc(F)c(F)cc1F C(C(N=c1[nH]cnc(Cl)c1Br)C1CC1)NC(Cc1n2c(nc1)C(C)CCC2)=O c1(NC(C(COCC)NC(c2cnsn2)=O)=O)cncc(C)c1 C#Cc1ccc(C(=O)NC(CC=C)C(=O)N2CCCC2(C)CO)cc1 CCC(C)(C)CCCC(=O)NCCC(Cc1ccccc1)NC(=O)CC(C)C(F)(F)F C1(NC(c2nc(CC)oc2)=O)CCCCCC1C(=O)NCC(c1ccnn1C)O c1(C(N2C3C(C(=O)NC(C(C)C)(C)C)C(C3)C2)=O)cc(O)ncc1F NC(=O)CC(O)C(=O)NC1CCC1C(N1CCN(C2CC2)CC1)=O C(C(CO)(CO)NC(c1cc(C(C)=O)c(C)o1)=O)N(C(C(C)=CC)=O)C C(=O)(C1=CCCCC1)NC1C(C)CN(C(=O)CN2CCCCC2C)C1 CN1CCN(C(=O)C(O)C(C)(C)C)CC1CNC(c1ccnn1C1CCC1)=O c1(CC)cc(C(=O)N(CCCNC(C2CCNC2=O)=O)CC)cc(C)c1 CN1CC(CC(=O)N(C(C)(C)C)CCc2ccccc2F)C(O)C1 N1(C(c2c(C)n(C)nn2)=O)CCC2CC2(NC(C2SC3C=CC2CC3)=O)CC1 n1(C(COC)C)nc(-c2ccnc(OC)c2)nc1CCN1CCCC1=O c1(C(=O)NC2CN(C(=O)CCC3CCCC(O)C3)C2)cc(-n2ccnc2)ncn1 C(c1cc(C)cc(C)c1)=CC(=O)NC1(C)CN(C(CC(CC)(F)F)=O)C1 N1(C(C(C)n2ccnc2)=O)CC2CCN(C(=O)C(C)O)C2C1 Cc1c(C(=O)NC2CC(CCNC(=O)C(O)CN(C)C)C2)nn2ccccc12 CC1CCC=C1C(=O)N(CCCNC(=O)C=CCN1CCCC1)C1CC1 C1(C(N(CCC(C)NC(C(C)NC(CC)=O)=O)CC)=O)CC2(C1)CC(C)(C)C2 N1(C(C)=O)CCN(C(=O)C(C)NC2CC(Nc3ccccc3Cl)C2)CC1CF N(C1CCc2ccccc21)C(N1Cc2ccc(N3CCOC3=O)cc2C1)=O c1(C(=O)NCC2C(OCC)CN(C(=O)C(F)CC)C2)cnc2c(cnn2C)c1 CCCC(C#N)C(=O)NC(c1ccccc1)CNC(c1csc(C)c1)=O N1(C(C(=O)NC(CC)CN(C(=O)C=CSC)C)C)CCCCCC1 C(=O)(CC(C)C(C)C)N1CC(CNC(C(C=C)(C)C)=O)C1 C1(NC(CCSCCCC)=O)CCCN(C(c2ccncn2)=O)C1C CC(C(C)(C)NC(=O)CC1CCCN1C)NC(=O)Cc1csc(CC(F)(F)F)n1 C1(COC)CC(CN)N(C(=O)C(CCCl)N(C)C)C1 c1(CC(=O)NC2C=CCN(C(C3C(C)C3C)=O)C2)ccc2c(c1)NC(=O)C2 C1(NC(c2cc(CNC(c3c(CC)nco3)=O)no2)=O)CC12CCCCCC2 C(=O)(C1=C(C)OCCS1)N(C1CC(C(N2CCC(CCC#C)C2)=O)C1)C N1(C(c2nc(CC)oc2)=O)CC2CS(=O)(=O)CC2(NC(c2cnncc2O)=O)C1 CON=CC(=O)N(CC(C)(C)CNC(=O)C(C)Cc1ccnn1C)C c1(C(=O)Nc2ccc(C(=O)Nc3cccc(Cl)c3O)nc2)cc(Cl)c(Cl)cc1F C1(O)(CNC(C2C(CC)C2)=O)CCN(C(C2(OCc3ccccc3)CCSC2)=O)C1 c1(C(N(C)CC2CCN(C(=O)CCC(C)(C)F)CC2)=O)c[nH]c2c(F)cccc12 N1(C(C)=O)CCC(CCC(=O)N2CCC2)C1.C1(CCc2ccco2)CCCN1C C(CN=C(NCC(F)F)N1CCC(c2nc(O)n[nH]2)CC1)OCCSC Cc1noc(C2CC2)c1C(=O)NCC(O)CNC(c1sccc1C(F)F)=O N1(C(=O)Cc2nc(Cl)cs2)CCC2(CC1)CN(C(c1ccc(F)nc1F)=O)C2 Cc1ccnc2nc(C(=O)NC3CC(N(C)C(C4CC4(F)F)=O)C3)nn12 C1(C)(C(=O)NC2CC(NC(c3nc(C(C)(C)C)[nH]n3)=O)C2)CCNC1=O C(=O)(C1=C(Cl)CCC1)NCC1(C(N2CCC(O)CC2CC)=O)CC(=C)C1 O(NC(=O)C(O)C1CN(C(c2cccc[n+]2[O-])=O)C1)Cc1cn(C)nc1 c1(NC(C2CN(C(C(C)(C)O)=O)CC(F)C2)=O)cc(F)c([N+](=O)[O-])cc1Br CC(C)CC(C)CC(=O)NC(C)(C)CCNc1ccc(C#N)nc1 c1(OC)cccc(COC(=O)C(O)CCn2cc(-c3cccc(C)c3)nn2)c1 CN=c1[nH]cc(C(=O)NCC2OCCC2C(=O)N(C)Cc2cnnn2C)s1 N1(C(C2CCCN2C(c2cnn(CCF)c2)=O)=O)C2CCC1CC2 C1(NC(CC(CC)N(C(C(CCC)NC(C)=O)=O)C)=O)COCC(C)(C)C1 C1(C(=O)NC(COCC)C(C)C)C=CCCN1C(=O)CCOC c1(C(=O)NCC(C(C)C)NC(c2cncn(C)c2=O)=O)ccc2ccncc2c1 C12(OC)CCC(C(=O)NC3CCCC(Cn4cc(C5CCCCO5)nn4)C3)(CC1)C2 c1(OC)ccccc1C(O)C(N1CCN(CCNC(C2CC2(F)F)=O)CC1)=O c1(-n2c(C)ncc2)ccc(C(=O)NC2CC(NC(=O)C(Cl)(Cl)Cl)C2)cc1 C1(CC(N2CC(C(=O)NCC3CC3(C)C)(COC)C2)=O)C=NN(C)C1=O Cc1cc(C#N)c[nH]c1=NC(=O)C1CCCN1C(=O)COc1ccncc1 S(=O)(=O)(c1ccc(Cl)cc1)N(c1ccc(N2CCOCC2)cc1)C(=O)CCC1CC1 c1(C(N2CC3C(CNC(C=CC(CC)C)=O)(C3)C2)=O)nccn2cc(C)nc12 c1(N(S(c2ccc(C)c(Cl)c2)(=O)=O)C(C)C)ccc2nc(C)c(=O)n(C)c2c1 C1(C(=O)NCC(C)CC2CCC2)CC(C)(C)CCN1C(c1c[nH]ccc1=O)=O O=C(N=c1[nH]c(=O)c2ccccc2nc1NS(=O)(=O)c1cccs1)C(=O)O c1(OC)cc(CN2CCC2(C)C(N2CC3C(C2)C3(F)F)=O)cc(OC)c1O N1(C(CCC)=O)CC=CC1(C)C(=O)N(C)C(c1nccs1)C c1(C(N2CCCC(N(C(=O)C(C)CC3CC3)CC)C2)=O)ccc2c(Cl)nccc2c1 c1(C(N(C2C3CN(C(C(CC)C)=O)CC32)C)=O)cc(C)c2ncccc2c1 c12ccc(OC)c(c1)N2.c1(OC)ccc(C2CCN(CCn3cccn3)C2)cc1 c1(C(N2CCC(NC(CCOCC#C)=O)C(F)C2)=O)cnc2scc(C)n12 CCC(C)CC(=O)C(=O)NC1(C)CCC(NC(c2cc(C)[nH]n2)=O)CC1 C#CCC(C(=O)N(CCCNC(=O)CCc1ccncc1)C1CC1)C1CC1 C12(NC(c3ncc(Cl)nc3Cl)=O)CCCC1N(C(C1(F)CCC1)=O)CC2 N1(C(C2(CC)CC2)=O)CC(CCNC(c2cc(C3(C)CC3)on2)=O)OC(C)C1 N1(C(C2CC(=C)C2)=O)CCCC(N(C(c2ccccc2OC(F)F)=O)CC)C1 C(=O)(CCC(C)CN(C)C)NC1C=CC(CC(=O)NCc2nnn(CC)n2)C1 Cc1cc(C(=O)NC2CCN(C(=O)CC3CC4CC4C3)CC2O)cc(Cl)c1 CCC(CC(=O)NC1CC(N(C(=O)CCc2ncc[nH]2)C)C1)SC C12(CNC(COC(C)=O)=O)CC(NC(C3CCC4(CCC4)OC3)=O)(C1)C(C)(C)O2 C1(NC(C=C(C)CNC(=O)CN2CCSCC2)=O)CC=CCC1 c1(C(N2CC3(CN(C(CNC(C(C)(C)C)=O)=O)C3)C2)=O)cc2c(s1)CCOC2 C(=O)(N1OC2CCC1CC2)CCC1CCN(C(c2ccc(C)o2)=O)C12CC2 CS(=O)(=O)C1(CC2CCC(NC(=O)Nc3cn(C4CCOC4)nn3)CC2)CC1 C1(C(=O)N(C2CCC2)C2CC2)(CNC(COCCCCC)=O)CCCCC1 c1(NC(C23CC(NC(=O)NC(C)C)(C2)C3)=O)cccc(-c2cnccn2)c1 O=C(C1=CC(O)CCC1)NCC1CCCC1NC(c1c(O)cccc1F)=O C#CC(C)(C)C(=O)NCCC1(O)CCN(C(C2(CC(F)F)CCC2)=O)C1 c1(C(=O)NC(CNC(C2(CC#C)CCCO2)=O)(C)C)cnc(C(F)(F)F)nc1 N1(C(c2ccn(C(CC)CC)n2)=O)CC(NC(=O)C2=CC(C)(CC)C2)CC(F)C1 CC(C)CC(O)C(=O)N1CCC(NC(c2cc(-c3cnccn3)[nH]n2)=O)C(O)C1 n1(CC)ncc(C(=O)OC(C)(C)C)c1NC(=O)OCCc1ccoc1C c1(C(N2CCN(C(c3ccc(C)cc3N)=O)C(C)C2)=O)cnn2cc[nH]c(=O)c12 N1(C(c2c(C)nccc2)=O)CCC(NC(C2(F)C(C)(C)C2(C)C)=O)C(C)(C)C1 c1(CCC(=O)NC(C=CC(=O)N(CCCC)C2CC2)C)nnc(C)n1C C(=O)(C1=NN(C)C(=O)CC1)OC(c1cc(C)n(-c2ccc(Cl)cc2Cl)c1C)=O CC(CC(=O)N1CC2(NC(=O)Cc3ccc(Br)s3)CC1C2)C(F)(F)F N1(C(CC=C(C)C)=O)CC(C)(CNC(=O)CSc2cc(F)cc(F)c2)CC1(C)C Cc1cc(F)c(C(N2CCCCC2)CN2CCC(C(N)=O)CC2)c(F)c1 Cc1cc(C)cc(C2=NC(=Cc3cccc(OC(F)(F)F)c3)C(=O)O2)c1 C(Cc1cc[nH]n1)(C(=O)NCCCc1cccnc1)NC(c1cccnc1)=O c1(C(=O)NC2CC(CCNC(c3snc(C)c3N)=O)C2)cnc2c(c1)CNC2=O c1(C(=O)NCC(N2CCN(CC(=Cc3ccccc3)F)CC2)=O)ccccc1Cl c1(C(=O)NC2C(CO)CCN(C(C=C3CCN(C)C3)=O)C2)cnc2n1CCOC2 CCCC(C)(CC)C(=O)N1CC2CCCC2(CNC(=O)CCc2cn(C)nn2)C1 c1(C(N2CC(C)CC(NC(C3(CC#C)CCOC3)=O)C2)=O)cccc2c1OCC2 Cc1cc(CNc2ccccc2-n2cncn2)ncc1Cl CC1CCCCN1CC(N1CC(F)(C(=O)NCCC2CC(O)C2)C1)=O c1(CC(=O)NC23COC(C2)C(NC(C2CC(=C4CC4)C2)=O)C3)cccc(Cl)c1F CC1CN(C(=O)CCC(=O)Nc2c(F)cccc2F)CCN1C(=O)CCC(N)=O Cc1ccc(Br)c(C(N2CCCCC(NC(c3cc(=O)n(C)o3)=O)C2)=O)c1N C1(NC(N2CCN(c3cccc(C(F)(F)F)n3)CC2)=O)CC1C1CCCCC1 c1(C(=O)NC23CCCN(C(C(C=C)(C)C)=O)CC2C3)cnc2ccccc2n1 C1(C(=O)NC(C2N(C(COC)=O)CCOC2)C)CCc2ccccc2C1 c1(-c2cn(C3C(NC(CN(C)C(N)=O)=O)CCC3)nn2)cc[nH]c(=N)c1 C1(C(=O)NC2CC(C(N(C)C)=O)C2)CCCCC1C(N)=O C(C(F)(F)F)OCCO.C(=O)(CC1CC1)N(CCNC(=O)CSC)CC CN1C(CNC(=NCC2CCCOC2)NCC2(C3CC3)CC2)CCS1(=O)=O C(=O)(C(CC(F)F)C1CCC1)NC(CNC(C1(C(CC)=O)CC1)=O)C1CCC1 C1(F)(CNC(C(F)=C(C)C)=O)CCN(C(=O)CC(C)c2ccccc2)C1 c1(C(=O)NC(C)C(C)NC(c2cnc(N)cn2)=O)cc2c(F)c(Cl)ccc2[nH]1 C(=O)(C(C)C(C)(F)F)N1CC(N(C(CCCc2ccc(OC)cc2)=O)C)C(O)C1 c1(CN(CC(CNC(C(C(=O)OC)OC)=O)C)C)ccc([N+](=O)[O-])cc1OC c1(CN2C(C(N3CCC(Br)C3)=O)C3CCC2CC3(F)F)ccc([N+](=O)[O-])cc1F C12CC3(C1)CN(C3)C(=O)C(CC)N2C.C(=O)(CSC(F)F)NC N1(C(c2c(C)nns2)=O)CCC(F)(C(=O)Nc2ccnc(C#N)c2)CC1 CCC(C(=O)Nc1ccc(OCC(C)(C)C)o1)OCOCCCOC c1(C(N(C2CN(C(c3nnc(O)cc3O)=O)CC2O)C)=O)ccnc(F)c1N N1(C(Cn2ncn(C)c2=O)=O)CC2CCCC2(CNC(=O)CC2CCNC2=O)C1 CC1(C)CCOC1CC(=O)NC(C)(CNC(C12CCC1CC2)=O)Cn1cccn1 c1(CC)noc(C)c1C(=O)NCC1CCCCC1NC(C1CC=C(C)CC1)=O CCCCC(C(=O)N1CC2CC1CC2O)NC(c1cnc(Cl)n1C)=O C(c1nc2ccccc2o1)=CC(=O)NCC#CCNC(c1nnc(C)s1)=O C1(N(CCOC)C(=O)NCc2ccnc(N3CCCC3)n2)CNC2CCCCCC12 N1(C(CCC(C)(C)NC(CSCC#C)=O)=O)CC(C(N)=O)OC(C)(C)C1 CCC(C)CCNC(=O)CCNC(=O)OC.C12(C)CCN1C(=O)C2 c1(OC)cc(OC)nc(C(=O)NC2CC(NC(C3CCCC4CC34)=O)C2)c1 N1(C(C(CCC)NC(c2ccc(OC)cc2)=O)=O)CCOC(C)(C)C1 c1(C(N2CC(C(C)NC(c3ncn(CC)c3)=O)C2)=O)cc(Cl)ccc1Cl C1(C(=O)NC(C)C(CO)NC(c2cc(O)cc(=O)o2)=O)CCc2nncn2C1 C1(CC=C)CCN(C(=O)C(CNC(=O)C(C(C)C)OC)CC2CCCC2)C1(C)C c1(CCNCC2C(SC)CCC2)nccc(C)c1Br.c12cn(nn1)C2 S(=O)(=O)(c1cnc(NCc2cnn[nH]2)c(Cl)c1)N(C(CC)CC)CCO c1(SC(C)(C)C)cccc(C(=O)NC(C)(CSc2ccccc2)CO)c1O n1(CCOC)cc(C(=O)NCC(C)NC(C2(C)CCCC2(F)F)=O)c(=O)cc1C C1(NC(C(N(C(CCOCC#C)=O)C)C2CC2)=O)CCC=CCCC1 N1(CC)CC2CC(N=c3ccc(C#N)c(OC(c4c(CC)cno4)=O)[nH]3)CC1C2 Cc1c(C(=O)NC2CN(C(c3cnn[nH]3)=O)C(C)(C)C2)cccc1Cl O=C(CCCn1ccnn1)NC1CCCC1CNC(C1CC1F)=O N1(C(c2nccc(CC)c2)=O)CCOCC(NC(c2c[nH]nc2C(F)(F)F)=O)C1 C1(C(N(CCCNC(c2ncn(CC)c2)=O)C)=O)CCCC(C#N)C1 c1(C(=O)OC)n[nH]c(C)c1S(=O)(=O)Nc1cccc(Oc2cccc(Cl)c2)c1 c1(C(=O)NC(CC=C)CNC(=O)C(F)n2ccnc2)ccc(C(F)(F)F)cc1F c1(OC)c(F)ccc(C(=O)NC2CCC3CC2CN3C(C2COC(=O)N2)=O)c1F CCC(CCCC(=O)NC1(C)CC2CCC1C2)NC(=O)C1=C(Cl)CCCC1 C(=O)(C(C)C(C)CC)N1CCN(c2nccc(CNC(C(F)=CCC)=O)c2)CC1 c1(CC)cc(CC(=O)NCc2csc(CNC(=O)Cc3cc(C)on3)n2)no1 C(=O)(C(COC)C(F)(F)F)N1CC(CNC(C=CC=CC)=O)C2C1C2 C(C(CO)(CO)CO)SCc1c(C)sc(Br)n1 CC(C)CC(CNC(=O)Cc1ccsn1)NC(c1ccc(C(N)=O)cn1)=O c1(NS(=O)(=O)CCC2COCCO2)ccc(CC(O)CO)cc1 c1(C(=O)OC)ccc(C(=O)NCCC(C)NC(C2CCC(C)O2)=O)cc1F C1(OC)C(OC)CN(C(c2ccccc2CO)=O)C1CNC(=O)C1=NOCC1 C(=O)(C(C)S(N)(=O)=O)NCCCN1CCN(C(CCNC(C)=O)=O)CC1 c1(CCC(=O)N(CCC)CCNC(C2(F)CCOC2C)=O)cccc2c1OCO2 C1(N(C(=O)CC2CC=CC2)C)CCCN(C(c2cccnc2C(F)F)=O)CC1 N1(C(CCCC=C)=O)CCN(C(c2cn(C(F)F)cn2)=O)C(c2ccncc2)C1 CC1CC2(CC(C(N3CC(CCNC(C4(c5ncccn5)CC4)=O)C3)=O)C2)C1 C(CC(N)C(=O)N(CCCc1cn[nH]c1)C1CC1)OC Cc1nn(CC(N2CCN(C3CN(C(C4COCCN4C)=O)C3)CC2)=O)c(=O)o1 C1(CNC(CCC(=O)NC)=O)CN(C(C2(SC)CCC2)=O)CC12CCOCC2 C1(Cn2cc(CSC)nn2)CC(O)CN1C(=O)COc1cccc[n+]1[O-] CN1C(=O)c2ccc(NC(C3CCCCN3)=O)cc2S1(=O)=O c1(OC)ccc(CCCC(=O)NCC2CCN2C(=O)C(C)C#N)cc1 C1(CNC(C2(C(N)=O)CCC2)=O)COCCN(C(C23CC=CC(C2)OC3)=O)C1 Cc1ccc(C(N2CCCC(NC(=O)CC3CC(O)C3(C)C)C2)=O)c(Cl)c1 C(=O)(CCCCCC#N)N(CCc1n(C)ccn1)C1CC1.C1(=O)CC(CC2CC2)N1 C1(CC(N2CC(O)(C(C)NC(c3cnn(CCF)c3)=O)C2)=O)C(C)(C)C1(C)C Cc1cc(N)c(C(=O)N(C)CC2COCCN2C(C2CCNC(=O)C2)=O)cc1C C1(C(N(CCC(C)NC(c2c(C)cc(C)o2)=O)C)=O)CC12CC(F)(F)C2 c1(C(=O)NC(CNC(CC=CC=C)=O)CCOC)cc2ccc(F)cc2o1 Cc1cccc2c1NCCC2C(=O)N(C1CC1)CC1CN(C(C2CCC(C)C2)=O)C1 Cc1ccccc1C(=O)NC1CCCC(NC(C2(C)CC2(F)Cl)=O)C1 C(=O)(CCC(C)(C)NC(C1CC(=O)N(CC)C1)=O)N(C(CCCC)C)C c1(N2CC3CC(NC(CC4N(C)C(=O)CC4)=O)C3C2)ncnc2ccccc12 C(=O)(CC(O)C(C)C)N1CCC(CC=C)(NC(=O)C=CC2CCCN2C)C1 C1(CNC(c2nc(NC(C)=O)sc2)=O)C2CCCC1N(C(c1cncc(C)c1)=O)C2 Nc1cc(C(=O)NCC(CO)NC(c2ccc(CO)nc2)=O)ncc1F c1(C(N(C2CC(NC(CC(C)F)=O)C2)C)=O)ccc(-n2cccn2)nc1 Cc1cc(N(C)C)ccc1NC(C1CC(O)CN1C(=O)C(N1CC2CC2C1)C)=O C1(C(=O)NCCOCCCN(C(=O)C(C2CC(F)(F)C2)O)C)CC(=O)NC(=O)C1 N1(C(COCc2c(C)ncs2)=O)CC2CN(C(C3CCN(C)C3=O)=O)CC2C1 C12(CC)CC(C(=O)NC(C)(C)CCNC(=O)C(C(C)C)n3cnnn3)(CO1)C2 C1(C(N(CC(C)N(C(COCC=C)=O)C)C)=O)CCn2nccc2C1 C1(C)(CC)CC(C(=O)NCC(CNC(=O)C(F)(F)C2(OC)CCCC2)OC)C1 N1(C(CSCC)=O)CC2CCN(C(=O)COCc3ccco3)C2C1 C(=O)(C1CCCc2ncnn21)NC1CCC(CCNC(CC(=O)OC)=O)C1 N1(C(CCCOCC=C)=O)CC2CCCC2(NC(c2ccc(CSC)o2)=O)C1 C1(NC(CN(C)C(=O)OC(C)(C)C)=O)CC(F)CN1C(c1ccco1)=O c1(OC)cccc(C(=O)NC(C)CCCCNC(C2COC3CC2C3)=O)c1C CCC(C)(C)C(c1nnnn1C1COC1)NCc1cc(-c2ccccc2)cs1 CCC(C)(CNC(c1cnc(C)cc1C)=O)C(=O)NC1CCC(F)(F)C1 N1(C(CCC(C)NC(c2ccon2)=O)=O)CCC(O)C1(C)C N1(C(c2cc(C3CC3)cnc2Cl)=O)CCC2(CCOC2=O)C1 C=C1CC(C(=O)NC)(C(=O)OC)C1.C1(CC)(N)CN(C(C2CCC(C)O2)=O)C1 c1(C(=O)NC(CCN(C(C2(C#C)CC2)=O)C)C(C)C)ccc2ccccc2n1 C(C(C)(C)CC(=O)N1CCCC1CNC(C1CC1CN(C)C)=O)OC(C)=O c1(CC(=O)NCCN(C(C(C)CC2CC2)=O)C2CC2)ccn2cncc2c1 Cc1cc(C(=O)N(C(C)CNC(c2cnn(CCO)c2C)=O)C)c2nccn2c1 N(C(=NCCCCl)NCC(c1cccc(F)c1)(C)C)CC1(CC)CCCCCC1 c1(SC2CC2)cccc(NC(c2onc(CC)n2)c2nnnn2C(C)C)c1 C1(N(C(C(C)N(C(c2c(COC)cco2)=O)C2CC2)=O)C)CC(O)C1(C)C c1(C(=O)OC)ccc2c(c1)NC(=O)CN2C(c1n[nH]c(CC2CCCO2)n1)=O c1(C2CCC(C(=O)NC(c3ccco3)COC)C2)ccc(Cl)cc1 N1(C(c2c(COC)ccs2)C(=O)NCCSC)CCS(=O)CC(C)C1 c1(C(N2CCCC(NC(C3CC4CC3CC4O)=O)CC2)=O)ccc(F)c(F)c1F n1(CC)nccc1C(=O)OCCc1csc(OC)n1 N1(C(C(CCCCC)O)=O)CC(C2CCCN(C(=O)CC3CC4(CCC4)C3)C2)C1 C(=O)(C(C(C(=O)O)N1CCCOC(CN)C1)c1ccccc1)Nc1ccc(C)cc1 C1(C(N(CC)Cc2ccoc2)=O)CC2(CCN(C(=O)CC3CCC(=O)NC3)C2)C1 C1(C(F)F)(CNC(c2sccc2I)=O)CCN(C(c2ccn(C3CC3)n2)=O)C1 N1(C(C(C(C)C)SC)=O)CC(NC(c2cn(C)nc2C(F)F)=O)CC2(CCC2)C1 C1(CCOC)(NC(c2cc(C)c(C)o2)=O)CCN(C(c2cc(C)co2)=O)C1 C1(=O)C(C)O1.CCCCN(CCCO)C(C)CO c1(OCCCC(=O)NCCCNC(C2C(C)C2)=O)ccccc1F c1(C(C)C)ncc(C(=O)NC2CC2CNC(=O)CCc2nccs2)o1 C1(n2ccc(C(=O)NC(C)CN(C)C)n2)CCNCC1.c1(COC(C)(C)C)cccs1 CC1(NC(c2scnc2C2CC2)=O)CCN(C(C2CC2(F)F)=O)C1 C(c1ccc2[nH]ccc2c1)=CC(=O)NCC1(O)CN(C(CC(CCC)O)=O)C1 c1(C(N(CCC(C)NC(C23CC(F)(C2)C3)=O)C)=O)cc(C(F)(F)F)ns1 c1(C(N2CC3(CC2CO)OCCO3)=O)nc2cncnc2nc1O c1(C(=O)NCC2C(NC(C=C(C)C3CCCCC3)=O)CC2)nn(C)c2c1CCC2 N1(C(c2nc(C)sc2C)C(=O)NC2CCCC2)CCCC2CCCC12 C1(NC(c2ccc(C)o2)=O)CC(O)CN(C(=O)COCC2CCC2)C1 C(c1cccc(Cl)c1)=C(C)C(N1CC(NC(C23CC(C)C2C3)=O)C(C)C1)=O CCCCCCC(=O)NC(C)C(C)(C)C(=O)NCCC1CCOC1(C)C c1(C(=O)NC23CCCN(C(C=C)=O)CC2C3)cc2c(O)cccc2n1C C1(OCC)CN(C(=O)C(=O)C(C)C)CC1C(=O)NCc1ccc(CC)cn1 C1(NC(=O)Cc2n[nH]cc2Br)CN(C(=O)CC2OCCO2)CCC1O C1(CNC(COC(C)=O)=O)CC(F)(CNC(=O)C(F)=C2CCCC2)C1 N1(C(CC2(C)CC2)=O)C2CCC1C(CNC(=O)C(F)(F)SC13CC(C1)C3)C2 C1(C)(C(=O)NCc2c(C(N(C(CC#C)C)C)=O)n[nH]c2)CC=CCC1 C(=O)(C(Cc1ccccc1)NC(=O)COCCc1cn(C(C)C(=O)O)nn1)OC C(CCCCC(=O)N1CC(N(CCO)C(c2c[nH]nc2-c2cccs2)=O)C1)N(C)C N1(C(CCC2CNC(=O)N2)=O)CCC2C(NC(c3ccc(Cl)cc3)=O)C12 C1(NC(CC(=C)Br)=O)CN(C(=O)C(C)(C)OCC)CC1C C(=O)(CC(C)(C)CNC(=O)OC(C)(C)C)NCC1CCN(C(COC)=O)C1 Cc1nccc(C(=O)NCC2(C(N3CC(SC(F)F)C3)=O)CCCC2)n1 Cc1cccc(-n2nccc2-c2nc(-c3cc(C)nn3C)no2)c1 C(=O)(C1CCCc2nn(C)cc21)N1CC(NC(CC(CC)C(F)F)=O)C1 C=CC(C)(CC)C(=O)NCC(C)(C)NC(C1CCN(C(c2ccoc2)=O)CC1)=O C(CO)(CCCCNC(c1cccc(C)c1-n1cccc1)=O)NC(C(C)SC)=O n1(CC(=O)NCCN(C(C2(O)CCCC2)=O)CC)ccc(=O)n(C)c1=O c1(C(=O)NC(CC(=O)N(CC(O)C2CCC2)C)C)nnc(O)nc1O c1(C(C(=O)NC2(CNC(C(C)O)=O)CCC2)C)ccc(Cl)cc1 N1(C(C(=O)OC)C)CCN(C(=O)C(c2cccc(F)c2)O)CC1 CC1COCCN1C(c1ccc(NC(c2cn(C(C)(C)C)nn2)=O)cn1)=O c1(C(C)NC(=O)N(c2ccccc2OC2CCCC2)C)nc2ccccc2s1 C1(NC(CC2CCN(OC)CC2)=O)CC2(CCC(CNC(=O)COC(C)=O)OC2)C1 O(S(=O)(=O)c1sccc1Br)c1c(C)ccc([N+](=O)[O-])c1 C123CC(CCO1)N(C2)C3=O.C1(CC(C)(C)C)CCCN(C(C2C3CCCC23)=O)C1 N1(C(C2C(C)C2)=O)CC=C(CCNC(c2cn(C3CCOC3)cn2)=O)CC1 C1(NC(C(CC)CC2CCCC2)=O)CN(C(=O)CN2CCSCC2)CCC1O c1(C(=O)NCCC(C)(C)NC(c2cnc(C(C)O)s2)=O)coc2c1CCCC2 C1(C(=O)NC(c2ccccn2)CC)(CC)CCN(C(C2CCCSC2)=O)C1 N1(C(c2snc(C)c2N)=O)CC2(CCC2)CC1CNC(=O)C(C)CS(C)(=O)=O N1(C(C2(C)CC2(F)F)=O)CCC(C)(CNC(C2(C)CC2(F)Cl)=O)C1 NC1CC2CCC1CN(C(=O)NCc1cc(F)c(F)c(F)c1F)C2 N1(C(CSCCCC)=O)CCC2CN(C(c3cnn(C4CCC4)n3)=O)C2C1 CCC(C(=O)NCCC1(O)CCN(C(c2cc(F)ccc2Cl)=O)CC1)C(C)O N1(C(C(CC(=O)OC)C)=O)CCC2CCCC12C(=O)NCCOCCCF C=CC(C)CC(=O)NC1CC1CNC(c1c(Br)noc1C)=O C(=O)(CC(C(F)F)CCC1(C(N(OC)C)=O)CC=CC1)NC(C1CCCO1)=O c1(NC(=O)NC(C2Cc3ccccc3C2)C(C)C)ccc2ncnn2c1 C1(CCNC(CCCOCCC)=O)CSCCN1C(=O)C=CC1CCCO1 C1(CNC(=O)C=CCc2ccccc2)CN(C(=O)CCC2CCCC2)CC1(F)F c1(SC)ccc(C(N2CC(NC(=O)C(O)CCn3cncn3)C(SC)C2)=O)cc1 C12CCCCCN1C(=O)COC2=O.C(=O)(C(F)(F)F)NCC(=O)OC1CCOC1 c1(C(=O)NCCC2N(C(CC3C(CC)C3)=O)CCC2)c(Cl)ccc2ccncc12 c1(C(N2C(CCNC(=O)CNC(=O)C3CC3)CCCC2)=O)ccc(F)c(F)c1F C=CC(CC(=O)N(C)CCNC(=O)COC(F)(F)F)c1ccccc1 [N-]=[N+]=Nc1ccc(C(=O)NC2(CNC(=O)C(F)CC3CCCC3)CCCC2)nc1 C(=O)(C(C)C(C)(C)C)N1CC(CCC=C)(C(=O)NCc2cn(C)nn2)C1 CCCCCC(C)CC(=O)NCC(C)(C)CC(=O)N1CCCC(C)CC1 c1(C(C(=O)N(C(C)CC)CCC2CC2)N(CCCC)CCCC)ccn(CC)c1 Cc1cc(C(=O)NC2CCCN(C(=O)CCc3ccccc3C)C2C)nc(O)n1 c1(C(=O)NC(CNC(c2nc(C)sc2)=O)C2CC2)[nH]c2cccc(F)c2c1C C1(C(=O)NC2CCCC2O)(CC)CCN(C(=O)CC2CCN(C)C2=O)CC1 N1(C(Cn2cc(CCC3CN(C(CC)=O)C3)nn2)C)CCN(C)CC1.CCS C1(C(=O)NCC2C(COC)C2)CN(C(=O)C(C)NC(C)=O)C(C)(C)C1 c1(OC)cc(C(N2CCC(NC(=O)C(F)n3cccn3)C2)=O)c(C)cc1Br c1(C(=O)NCC2(C(F)F)CCN(C(CSC)=O)C2)ccc2nnnn2c1 N1(C(c2cccc(CC)c2F)=O)CCN(C(=O)C(C(C)(C)C)OC)CC(C)C1 N1(CCCOC)CCC(=O)N(CCc2cc3ccccc3o2)C1=O C1(C(N(C2CCN(C(=O)CCc3cnoc3)CC2)C)=O)CCCC(F)C1 C(=O)(CCCCC(F)F)NC(C)CN(C)C(c1ncc(Cl)cc1O)=O Cc1cc(S(N)(=O)=O)sc1C(C(=O)NC)NCC1CCCN(S(=O)(=O)C(F)(F)F)C1 C=CC1(NC(=O)C(O)C2CN(C(C3CN(C(C)C)C3)=O)C2)CCCCC1 C1(CNC(C(C)CC2CCC2)=O)CC2(CC2)CN1C(c1ccnc(Cl)c1N)=O c1(COC)cccc2c1CN(C(=O)NCC1(F)CCN(C(=O)OC(C)(C)C)C1)CC2 C(=O)(C#CC1CCCOC1)NCC1(F)CCN(C(C(CC(C)C)C)=O)CC1 N1(C(C(CC)O)=O)CC2CC1C2NC(c1ccc(CNC(c2cccs2)=O)o1)=O C1(CNC(C(CC)(C)C)=O)C(C)CCCN1C(c1cc2ccsc2s1)=O C1(NC(c2cc(COC)on2)=O)C2CC1N(C(c1ccc(CO)cn1)=O)C2C Cn1ccc(C(=O)NC2C=CCN(C(c3cc(=O)c(Br)c[nH]3)=O)C2)cc1=O CC(CCCCNC(C1CCCCC1O)=O)NC(=O)Cc1cocn1 C1(C(C)(C)C)C(=O)N2CCCC2C(=O)NC1.C1(CSCC)CCCC(CO)C1 Cc1ccc(C(=O)NCC(C23CCC(CC2)C3)NC(=O)CSC(F)F)cc1F N1(C(c2cc(SC)oc2C)=O)CCC(O)(CNC(C2CC(C(C)C)=NO2)=O)CC1 N1(C(c2c(C)cn(C(C)C)c2)=O)CC2(C1)CN(C(=O)C(C)(C)CF)C2 c1(C(N2CC(O)(CN(C(C=CC(=O)OC)=O)C)C2)=O)cc(Br)ncc1N(C)C c1(C(=O)NCC(C2CCCC2)NC(C2CC(C)(C)C2)=O)cn2cnnc2cn1 C(CC(O)CC(=O)N(C1COCC1n1cc(C(C)(C)N)nn1)C1CC1)SC.CSC CC12COCC1(C)CN(C(C13CCCC1CCN3C(C1C3CC4C(C3)C14)=O)=O)C2 C1(=CCCC(C)=CC(N2CCC2CC(=O)OC)=O)CCOCC1.CO N1(C(CC(C)NC(C2C3CCC(=O)C23)=O)=O)CC2CC=CCC2C1 C(C(CC(C)C)NC(c1ccc(CNC(=O)CNS(C)(=O)=O)s1)=O)OC N1(C(C(c2cccc(OC)c2)O)=O)CC(NC(c2ccc(F)cn2)=O)CC2(CC2)C1 C=Cc1cnn(C)c1C(=O)NC(C1CCCC1)CNC(c1cnc(OCC)s1)=O N1(C(c2c(C)cco2)=O)CCCC(O)(CNC(=O)C=Cc2ccccn2)CC1 CC(C)(C)C(CNC(=O)CC1CC=CCC1)NC(c1scnc1C1CCCC1)=O N1(C(c2cn(C)nc2)=O)CCC(C2CC(NC(c3cncc(C#N)c3)=O)C2)C1 C1(CC(=O)NC(CNC(C2(OC)CCOC2)=O)C(C)C)CC2CCC(C1)N2C N(C(=NCCC(C)=O)NCCC1(C)COCCO1)CC1(OC)CCSC1 c1(CC(N2CC(O)(C(C)NC(=O)CC=CC(C)(C)C)C2)=O)cc(Cl)n(C)n1 N1(C(C(C)CN(C)C)=O)CCN(C(=O)Cn2cnc(C(N)=O)n2)CC(O)C1 C1(C(N(CC(C)NC(c2cscc2Br)=O)C)=O)CCOC2(CCC2)C1 CCN=c1cc(Nc2cccc(N(C)C)c2)[nH]c(=NCC(C)SC)[nH]1 C1(C)(NC(C2N(CCC)CCC2)=O)CCC(NC(=O)C(C#N)CCC)CC1 c1(NC(C2CCC(C(=O)NC(C)C#N)C2)=O)cccc(C(C)(C)C)n1 c1(OC)cc(N)[nH]c(=NCCOCCCNC(C)=O)n1.C(=O)(C(C)CSC(F)(F)F)O CN1CCC(O)(CCNC(C2CSCCN2C(C2CC3CCC(C2)O3)=O)=O)CC1 C1(CC(N2CC(NC(=O)C(F)(F)c3nccs3)C2)=O)CCCCC1(F)F c1(SC)cccc(C(=O)NCC(CNC(c2cnn(C(C)C)c2N)=O)OC)n1 c1(NS(C)(=O)=O)ccccc1C(=O)NC1C=CC(C(N2CCC(F)CC2)=O)C1 c1(OCCNc2c(C(=O)OC)c(F)ccc2)ncccc1S(C)(=O)=O C(=O)(C(O)C(O)C(=O)N(C)CCOc1cc(F)ccc1F)OC C(=O)(CCCCC(C)(C)C)N1C(C(=O)NCC(=C)C)CC2(CC1)CC2 C(=O)(C(F)(F)CO)NCCN(C(CC=C=C)=O)CC1CC1 C(=O)(CCN=C(NCc1n[nH]cc1Br)N1CCCC(OC)(OC)C1)NC C(C(C(C)C(C)C)NC(c1cn(Cc2cccs2)nn1)=O)NC(C=CCC)=O c1(CC(=O)NCC(CCCC)NC(=O)C(C#N)=C(C)C)ccc(Cl)c(Cl)c1 c1(C(N(C(C)CNC(c2cn(C)[nH]c2=N)=O)C)=O)cc(F)c(F)cc1F C1(NC(c2ccc(CC)c(C(F)F)c2)=O)CC1C1CCCN(C(=O)C(C)(C)Br)C1 N1(C(C)=O)CCN(C(c2ccn(CC(F)F)n2)=O)CC1c1cn[nH]c1 C#Cc1cccc(CCCNC(C2CNC(=O)C2)=O)c1 CCCCC(C)CCC(=O)NC1CC(CO)N(C(=O)C(c2cccc(C)c2)=O)C1 C1(NC(c2cc(CC)on2)=O)CCC(O)CN(C(C2CCC(C)(C)C2)=O)C1 c1(C(=O)NC(CNC(C2C(C)CCCC2)=O)(C)C)nc[nH]c2nccc1-2 N1(C(C2CC(=C)C2)=O)CC(CNC(C2(c3cc[nH]n3)CC2)=O)C(C)C1 C1(C)(C(N(CCN(C(=O)CCC2CC2(F)F)C)C)=O)CCC(=O)N1 C1(NC(C2(CC)COC2)=O)CCC2(CCN(C(c3nnn(C(C)(C)C)n3)=O)C2)C1 C1(N2CCC(CC#C)C2)CCN(S(=O)(=O)C(F)F)C1=O C=Cn1nncc1C(=O)NCC1(C(=O)NCc2cc(Cl)ccn2)CC(C)(C)C1 C1(N2CCN(C(C3CC(C)OCC3)=O)CC2)CC2CCCNC1C2 C1(C(N2CCOC3CNCC23)=O)CCN(C2=CCS(=O)(=O)CC2)CC1 N1(C(CSCCC)=O)CCC2CN(C(=O)Cc3cc(F)ccc3Cl)C(C)C12 CC1CCN(C(C23CC(C(C)(F)F)(C2)C3)=O)C(C(F)(F)F)C1 C(=O)(CC(C)(C)CC(C)=O)N1CCC(N(C(C2(C)CCCCCC2)=O)CC)C1 c1(C(=O)NCc2cccc(NC(CC(CC)OC)=O)c2)ccc(C)c(OC)c1 N1(C(c2c(C)[nH]cc2)=O)CC2CC(C(=O)NCC(c3nccs3)C)(C2)C1 N12CCN(CC1)CC2.c1(C(=O)NC(c2cc(C)sn2)=O)cc(Br)n(C)c1 CC(CC(=O)N1CCCC1CCNC(c1cnn(C2CCC2)n1)=O)P(C)(C)=O CS(=O)C=CC(=O)N1CCC(C)(NC(=O)COc2nc(Br)cn2C)C1 N1(C(c2c(C)nn(C)c2C)=O)CCC(C2CC2)(CNC(C2OCC2(C)C)=O)C1 C(CCN(C(=O)Cc1ccns1)C)(C(C)C)NC(c1cc(C(C)C)no1)=O C(=O)(CCC(C)(F)F)N(CCC(N)C(=O)OC)Cc1ccc(Br)cc1 Cc1ccc(-c2ccc(CNC(=O)CCN(C)C)nc2)c(C#N)c1 CC(CCC(=O)NC1(CO)CCN(C(c2ccccc2-n2ccnn2)=O)C1)N(C)C c1(C(=O)NCCCN(C(=O)Cc2ccc(C)s2)CC)cc(C(C)=O)ncc1F c1(N2CCC(N(C)C)(C(=O)OC)CC2)nc(C)nc(C)c1C.C(C)(CN(C)C)N Cc1cc2[nH]c(C(N3CC4CN(C(c5cc(Cl)ccc5C(C)C)=O)C4C3)=O)cc2s1 C1(CN(C(CCSC)=O)C)CCN(C(=O)CC2C=CCCC2)CC1 C(=O)(CC(C)(C)C(=O)OC)NCC(CC)(C)NC(=O)CC1(COC)CCCC1 Cc1ccncc1C(N1CCCC(C(C)(C)C(=O)NC(C(C)(C)O)C2CC2)C1)=O c12cc(nn1-c1ccccc1)CN1CC(C1)C(=O)N2.c1(C(=O)O)cc(Cl)c(Br)s1 c1(OC)cccc2c1CCCC2N=c1ccnc(NCC2CN(C3CC3)C2)[nH]1 C#CCC(C(=O)N1CCN(C2CC2)CC1)NC(=O)CN1CCOC1=O C1(C(=O)NC(CCC)CNC(C2(SC)CC(CO)C2)=O)CCN(C)C1C c1(C(=O)OC)ccc(C(=O)NC2CCN(C(C3CCCO3)=O)C2C(C)C)cc1Cl N1(C(C(c2cn(C)nc2)NC(=O)CSc2cn[nH]c2)=O)CCCC(F)(F)C1 C(CN=c1nc2c(cnn2C)c(NCCN(C(C)C)CC)[nH]1)OCCC N1(C(C(CC=C)C)=O)CCC(NC(=O)CC(C)(C)C)CC(O)C1 c1(CCC)ccc(OC)c(NC(=O)Nc2c(C)nn(C3CC3)c2Cl)c1 C1(N(C)CC2CN(C(CC(C)c3ccncc3)=O)C2)CC(F)C(=O)N1 C=CC(CC)CC(=O)N1CCN(C(=O)CC2COCCOC2)C(CC)C1 c1(CC)ccccc1C(=O)NCC1CCCC1NC(=O)Cc1cnns1 N#CC1(C2CCCC2)CCN(C(C2CC3(CC(OCc4ccccc4)C3)C2)=O)CC1 C(C(CC(C)C)C(=O)NC1(C(=O)NOCC(C)(C)C)CC(F)(F)C1)OC c1(C(N2CCC3CN(Cc4cncc(O)c4)CCC23)=O)ccc2ccncc2c1 CCC(CCC(=O)NCC1(C(C)C)CCCC1)NC(c1n[nH]cc1Cl)=O C(=O)(CCC(C)(F)F)NC(c1cccc(Cl)c1)CNC(CCn1ncc(C)c1)=O C1(C(=O)NC2CN(C(C(c3ccncc3)C)=O)C(C)C2)CCCC2CCCCC12 C(C(CCO)N=c1[nH]c(=NC(C)CCSC2CCCC2)c2ccccc2[nH]1)N(C)C C1(NC(CCNC(C)=O)=O)CCCCC12CCN(C(c1c[nH]c(C)c1)=O)C2 C(=O)(CCS(=O)(=O)CC(C)C)N1CC(CN2CCN(C(C(C)SC)=O)CC2)C1 C1(C(=O)NC(C(=O)NC)C)COCCN1Cc1cnccc1C(F)(F)F C(=O)(CCCC(=O)NC1CCN(C(C2CC(c3ccccc3)O2)=O)C1C)NC C1(C(=O)O)(CCc2cc(OCF)ccn2)CN(C(=O)CC(=O)NCCO)CCO1 N1(c2cn(C)nc2)CCCC(NC(=O)C(=O)NCC(N2CCCOCC2)=O)C1 C1(NC(C23C(NC(CCO)=O)C4CC2C3C4)=O)CC2(C1)CC(C(C1CCCO1)=O)C2 C12(COC)CC(NC(=O)CSC(F)(F)F)(CN1C(C1C3CCCC13)=O)C2 c1(C(=O)NC(c2onc(C)n2)C)coc2c1CN(C(c1c[nH]nc1Cl)=O)C2 C1(C(=O)OC(C)(C)C)(CSC2CC(C(=O)O)CN2OC)CCC(=O)N1 N1(C(c2n(C)cnc2)=O)CC2CC(C(N3CCn4cncc4C3)=O)C(C2)C1 c1(C(=O)NC2CN(C(C=NOC)=O)C(C)CC2)cnc2sccn2c1=O CC(CF)CC(=O)NCC1(O)CCN(C(=O)CNC(=O)NC2CC2)C1 c1(-n2cc(CC)nn2)cnn(C)c1CNCc1nc(C(=O)O)c(C)o1.C1C(=O)NO1 N1(C(C(CCC)=CCC)=O)C2CCCC1CN(C(=O)CC1CCC(O)C1)C2 N1(C(CC(CCC)NC(C2CC(C)C2)=O)=O)CCC2(CCOC2)CC1 C1(C)(CC)CCC(C(=O)NC(C)(C)C2(NC(C34CC(CO)(C3)C4)=O)CC2)C1 c1(C(=O)NCC(CNC(Cc2c(C)cc(C)s2)=O)O)cnn2c1S(=O)(=O)NCC2 C(C(=O)N1CCC(CCCO)C1)(C(C)C)OC c1(CCN(C)CCN2CCCC2)cn(C)nc1-c1cccc(Cl)c1 N1(C(c2cn(CC(C)C)nn2)C(=O)NCCCOC)CCC2(CCOC2)C(C)C1 C(=O)(C1=NOC(c2ccccc2)C1)NC(CNC(c1c(C)occ1)=O)CO CC1CC(=O)NCC1C(N1CCC(C)(C)C1CNC(=O)CCc1ccsc1)=O CCCCC(C)(F)C(=O)N1CCC1CNC(=O)C=Cc1ccnn1C Nc1cnc(Cl)cc1C(N1CCCCC(NC(c2ccc(O)cc2F)=O)C1)=O C1(C(=O)NCC2(SCC(=O)NC3(CCCF)CC3)CCOC2)CCCOCC1 C(=O)(CCC(F)(F)F)N1CCC(C(C(=O)NC2C(C)NC(=O)CC2)(C)C)C1 C12(C(=O)NC(CC=C)CO)CCCC1N(C(C1CCN1C)=O)CC2 c1(C(=O)OCc2ncc(-c3c(OCCCC)cccc3)cn2)c(C)ccnc1Cl C1(C(=O)NC(c2ccncc2)(C)C)CCCN(C(=O)CC2CCC(=O)C2)CC1 C1(C(=O)NCCNC(CN(C)Cc2ccc(Cl)cc2)=O)CCCC(F)C1 C(=O)(CCCC(C)NC(C1CCSCC1)=O)NCC(C1CC1)OC CCC(CC)(CO)C(=O)N1CCn2ncc(CNC(c3ccoc3)=O)c2C1 c1(C(=O)NC(CC(=O)N(CCC(C)O)C)C)ccnc(OCCCC)c1 C1(C(=O)NCC2(F)CN(C(C3C(C)(C(C)C)C3)=O)C2)CCC2(CC1)CC2(F)F c1(CNC(c2ccncc2)=O)ncnn1C.C1(=O)CCC2(CCC2)N1C C1(C(N(CCC#C)CCO)=O)CCCN(C(=O)CCc2ccc(OC)nc2)C1 N1(C(CN(CCOC)C)=O)CCCCC1C(C)NC(=O)Cc1nc[nH]n1.CO C1(NC(C2C(OCC)C2)=O)(CNC(c2nc(O)c(C)s2)=O)CCCCCC1 C12(C(=O)NCC3N(C(Cc4c(C)n[nH]c4)=O)CC(O)C3)CCN(CC1)CC2 c1(C(N2CCN(C(=O)CC3CCCCC3O)C3CC23)=O)cc2c(F)cccc2s1 N1(C(C2C(C)=C2)=O)CCC2(CC1)CCN(C(=O)CCCn1c(O)nnc1O)CC2 Cn1nc(C(N2CC(NC(c3nncs3)=O)C(C3CC3)C2)=O)c2c1CCSC2 CCC(C)(C#N)C(=O)N1CCC(OCCCNC(=O)C(C)NC(C)=O)CC1 CCCC(C)(CC)C(=O)NCCC(=O)NC1CC2OCCCC12 c1(C(N(C2(CC(=O)NCCOC3CC3(F)F)CCC2)C)=O)cncnc1S c1(C(C)Nc2cc(N3CC(C4CCCC4)C3)ncn2)ccc2c(n1)OCCO2 c1(C(c2nnnn2C2CCOC2)NCC(NOCC)=O)cccnc1F c1(C(=O)NC2(C)CCN(C(c3nc(C)oc3)=O)C2)ccc(F)c(C)c1Cl Nc1c(C(=O)NC2CN(C(=O)CC3CCOCC3)CCC2O)ccnc1Br N1(C(C(C)=C2CCCC2)=O)CC(CNC(c2nc(Cl)oc2C)=O)C(F)(F)C1 c1(OCC)ccc(NC(=O)CO)c(F)c1.c12ncccc1OCC1CCN1C2.OC C(=O)(C#CC(C)(C)CNC(=O)CC1(C)CCC1)N1C(C=C)CCC1 C(=O)(CCC1=NNC(=O)CC1)NC1(C)CCN(C(C2OCC(C)C2)=O)CC1 C=CCC(C)(C)CC(=O)NC(CNC(C1(OC)CCSC1)=O)CCOC C(=O)(CS(=O)(=O)CC(=O)NC1(CO)CCN(C(c2cn(C)c(C)n2)=O)C1)OC c1(COC)cccc(C(=O)NC(C(N2CCCC2c2ncc[nH]2)=O)C2CCCO2)n1 CC1CC2(CCN(C(C3(C)CC3C)=O)CC2)CN1C(=O)C(N1CCNC1=O)C N1(C(C2ON=C(C(C)(C)C)C2)=O)CCC2(CC1)CC(CNC(C1CCCC1)=O)C2 CCCCC(O)CC(=O)N1CC(NC(C23CCC(C2)C3(C)C)=O)C(C)C1 CN1CCC(NC(C2CCC(NC(=O)Cn3ccnc3)C2)=O)C1 C1(O)(C(=O)NCC)CCN(C(c2ccc(OC)cc2Br)=O)CC1 Cc1cc(C(N2CCCC(CC(=O)Nc3ccc(Cl)c(C)c3)C2)=O)cc(O)n1 CC(C)(C)S(=O)(=O)CC(=O)N1CC2CN(C(c3cn(C4CC4)cn3)=O)CC2C1 N1(C(c2ccc(CC)[nH]2)=O)CCC(C)(CNC(=O)C(c2cnccc2C)(C)C)C1 CC1CC(CNC(=O)N(C)C(c2cccc(Cl)c2)C)CCS1 C1(C(=O)NCCCC(CO)NC(=O)CC2(OC)CCCC2)(CC)CCCCC1 C(=O)(CC(C)(C)CCOC)N1CCCC(CC)C1C(=O)NCC1CC2CCC(C1)C2 C1(C)(C(=O)NC(C(C)NC(=O)CCC2(C)CC2)CO)CC=CCC1 Cc1c(C(=O)N(C)CC2CCN(C(c3cnn(C(C)(C)C)c3)=O)C2)cccc1F C(=O)(C1=CCCN(C(=O)C(CO)C(F)(F)F)C1)N(C(C)C(C)(C)O)C C(C(F)(C(=O)NCCOC1CCC1)C(C)C)NC(C(CC=C)CC)=O c1(C(N2CC(O)(NC(C3N(C(C)=O)C(=O)CC3)=O)C2)=O)ccnc2ncsc12 c1(N(C)Cc2cscn2)nc(N(C)Cc2nc(O)cc(O)n2)c2c(n1)CCS2 c1(CCCC)cn2c(C(N3CCC(C(=O)O)C3)=O)cccc2n1 c1(OC(C)C(=O)NCC(C)(C)NC(=O)Cc2cccc(F)c2)ccccc1C#N C1(C(=O)OCC)CN(C(=O)Nc2ccccc2Oc2cccc(F)c2)C2CC12 C1(C(N(C)Cc2nc(C)[nH]n2)=O)CC2C=CC1N(C(c1nnc(S)n1C)=O)C2 CCC(CC)(CCNC(c1ccc(=O)oc1)=O)NC(C1CCC(C)(C)C1)=O [N-]=[N+]=NC1CCCN(C(=O)C=CC2CCCN2C(C2CC(N=[N+]=[N-])C2)=O)C1 N1(C(C2CC(C)(O)C2)=O)CCCC2CCN(C(=O)C=C3CCC3)CC12 C1(C(=O)NCC(C)=CC(N2CCC23CC(O)C3)=O)CC1C1CCCC1 N1(CC=C)CCC(NC(=O)CN(C)C(c2cccc(F)c2)=O)CC1 C=C(C)CC(C)C(=O)N1CC2CC1C2NC(=O)C(O)CC c1(C(=O)NC2C(NC(c3cc(C(=O)OC)sc3C)=O)CCC2)cc(O)nc(C)n1 C(C(=O)NCC(C)N(C(=O)CC1CCC=CCC1)C)(C(C)O)NC(=O)OC N1(C(c2cc(SC)nn2C)=O)C2CCC1C(NC(c1cnc(CC(C)C)[nH]1)=O)C2 c1(CCC(=O)NC2C(NC(Cn3c(C)nnn3)=O)CC2)cccc(F)c1Cl C1(C)(C(=O)NCCC2(CNC(C(c3cn(C)nc3)O)=O)CC2)CCCCO1 C1(C(N2CCN(c3cncc(F)c3)CC2)=O)(ON)CCCCC1 C1(CNC(C(CC)OC)=O)CCCCCN1C(=O)CCC1(C#N)CCC1 C1(C(=O)NC(CCNC(c2ccsc2)=O)C(C)C)(CC)CCC(F)(F)CC1 Cc1c(N2CCCC2C(=O)OC(C)(C)C)cc(Cl)cc1S(N)(=O)=O N1(C(c2scc(C)c2)=O)CCC(NC(c2cc(Cl)sc2Cl)=O)CC1C c1(CNC(CC)=O)cccc(C(N2CC3C(C(=O)NC(C)C=C)C3C2)=O)c1 c1(CC)ccc(F)c(C(N2CC(=CC(=O)NCC(=O)NC3CCC3)CC2C)=O)c1 N1(C(=O)OC(C)(C)C)CC2(C)CC1(NC(=O)OCCCc1ccncc1Br)C2 N1(C(c2c(C)noc2)=O)CCN(C(=O)CC2CCC(=O)NC2=O)CC(C)(F)C1 c1(NC(CNC)CO)ccc(OC(F)(F)F)cc1.C1(C(C)C)CO1 Cc1cc(C(=O)NCC(F)(F)F)ccc1NCC1CC1CNC(=O)C(C)(C)C#N N1(CCC2(NC(CC=C=C)=O)CC2)CCN(C(c2cnccc2C(N)=O)=O)CC1 c1(CC)ccc(C(N2CC(O)(C(F)C(=O)NCC3CCCCS3)C2)=O)[nH]1 c1(CCOC)n[nH]c(=NCC2(O)CCN(C(C34CCC(C3)OC4)=O)CC2)s1 N1(C(c2noc(CC)c2C)=O)CC(NC(=O)CCS(C)(=O)=O)CCC(O)C1 C1(CNC(C=C(CNC(C)=O)C)=O)CCN(C(=O)Cc2ccc(Cl)cc2)CC1CO CCCCCCC(=O)N1CC2CC1(CNC(C1COC(C)C1)=O)C2 C(=O)(C1CCCc2nc[nH]c21)NC(c1ccc(OC)cc1)CNC(=O)CO Cc1ccc(CN=C(NCC2CCC2)NCC2CCCC(C(F)(F)F)O2)cc1 C1(C2(O)CN(C(=O)CC(=O)N(C)C)C2)(CNC(c2c(SC)cc(C)cc2)=O)CC1 C1(C(=O)NCC2CCN2C(C2(C3CC3)CC2)=O)CCCCC1C1CC1 C1(C)(C(=O)NCCC2CC(OC)C2)CC(O)CN1C(c1ccc(C)o1)=O C=CCC(C)(C)CC(=O)NCCCNC(=O)Cc1ccn(C(C)C)n1 c1(Cn2cc(CC(N3CCC(C(=O)O)C3)=O)nn2)cn(CCN2CCOC2=O)nn1 Cc1nc(C(N2CCCC(NC(C3CC(O)CN3C(=O)N(C)C)=O)C2)=O)sc1C N1(C(C2(C)CC2)=O)CCC=C(C(=O)NCC(C)O)C1.C(C(C)O)SC C1(NC(C2CC(OC)C2)=O)CC2CCC1(CNC(c1oc(C)nc1C)=O)C2 c1(C(=O)NC2CCC(CNC(CC=C(C)C)=O)C2)cc2c(o1)CCCC2 c1(OC)cc(CN2CC(C)(CC(=O)NCCc3ccccc3C)C2)ccn1 N1(C(C(n2cc(Cl)cn2)C)=O)CCC2(CCCN2C(c2cc(Cl)ccc2O)=O)C1 N1(C(C(C(C)C)C#N)=O)CCc2sccc2C1CNC(c1cc(F)cc(F)c1)=O c1(C(=O)NC(C)Cn2cc(-c3cc[nH]c(=N)c3)nn2)ccc(-c2nc(=O)o[nH]2)cc1 c1(OC(C(=O)NCC(CC=C)NC(c2ccncc2)=O)C)cccc(SC)c1 C1(CC)CCN(C(c2cn(C)nn2)=O)C1C(=O)N(C1CCN(C(C)=O)C1)C C(C)(CCCC(C)C)NC(C(COCC)NC(C1CC(C#C)(O)C1)=O)=O C#CCC(C)(C)NC(=O)CN(C(=O)C(C1CC1)C1CC1)CC(C)C c1(NC2C(C)CN(C(c3ccc4nsnc4c3)=O)C2)ncccc1[N+](=O)[O-] c1(C=O)nc(Cl)ccc1OCCOC.C1(C(CSCC#C)=O)CCCN1N(C)C c1(CC)cc(C(=O)NC2CCC(N(C)C(C3CSCN3CC)=O)C2)ccc1O N1(C(c2ccnc(CC(C)C)n2)=O)C2CCC1C(NC(=O)C(F)F)C2 c1(C(=O)NCC(C)NC(=O)C(C)C(F)F)cc(Cl)ncc1N c1(C(=O)NC2CCN(CCOCC)C2)ccnc(-n2ccc(C)n2)c1 N1(C(CC(OCC)OC2CC2)=O)CCC(C(=O)N2CCSCC2)=C(F)C1 c1(CC(=O)NC(C2CCCC2)CNC(c2cnn(C(C)C)n2)=O)cccc(Cl)c1 c1(C(=O)NCCN2CCCN(C(=O)C(O)C(F)(F)F)CC2)ccc2nc[nH]c2c1F C(=O)(C1=C(Cl)CCOC1)NC(C(N1CCCC(C)(O)C1)=O)C1(C)CC1 N1(C(=O)CC2CCCN2C(c2cnsn2)=O)Cc2ccnn2CC(F)C1 C12(C(N(C3CCCC(O)C3)C)=O)CC(CN(C(=O)C(c3cnn(C)c3)=O)C1)C2 C(=O)(CS(=O)(=O)NC1CC1)NC(C)(CNC(=O)Cc1cnoc1)Cn1cccn1 c1(Cc2cn(CCC(N3CCC(CCC(=O)NC)C3)=O)nn2)ccc(F)cc1Cl C(CCCCN=c1cc(C)nc(N2CCOCC(C(=O)OC)C2)[nH]1)SCC c1(OC)c(NC2CC(NC(c3nn(C)cc3Cl)=O)C23CCC3)ncnc1C N1(C(COCCCCC)=O)CCN(C(C2CCCN2C2CCC2)=O)CC1 c1(C(=O)NCC(c2c(OC)cccc2)(C)C)ccc2cc(N)ccc2c1 C1(C(=O)NCC2CCC(CNC(C3(CSC)CC3)=O)CC2)CS(=O)(=O)CCO1 C1(OC)CN(C(=O)Cn2nccc2C)C(C)(CNC(=O)C(F)=C(C)C)C1 Cc1ccc(C(=O)NCC(C)CNC(=O)CC2=CCOCC2)c(N)c1Br c1(NC(N2CC(C)C(n3cc(C(C)(C)S(C)(=O)=O)nn3)C2)=O)cccc([N+](=O)[O-])c1F Cc1ccc(C(=O)NC2(CCCNC(C3CCN(C(=O)C4CC4)C3)=O)CC2)cc1 c1(NC(=O)NCC2CCC(C(F)F)CC2)ccc2ccc(Br)c(Cl)c2n1 N1(C(n2cccc2)=O)CCCC(C2CCCN2C(=O)CCC2CCC2)C1 N1(C(CCOCCOC)=O)CCN(C(c2cncs2)=O)CC1C1CCC1 Cc1cc(N)cnc1C(=O)NCC(CO)NC(c1ccc(CN(C)C)nc1)=O C1(NC(=O)C2=CCCCO2)CN(C(=O)C=CSc2nc[nH]n2)CC2(CC2)C1 C1(C(=O)NCC2(NC(c3nccc(C)n3)=O)CC(OC)C2)CCC2(CCC2)CC1 C1(C(=O)NC2C(NC(C=CCOC)=O)CCCC2)CC(F)(F)CCC1(C)C C1(CC(=O)NC(CNC(CCCC2(C)N=N2)=O)(C)CC2CC2)CC2(CCC2)C1 c1(C(=O)NCC2C(C(N(C3CCC3(C)C)C)=O)OCC2)ccsc1C#N Cc1cnc(C(=O)NCC(C)NC(c2cc3occc3n2C)=O)cc1C#N CCC1C(=O)Nc2ccc(C(=O)NCC(F)CNC(=O)CC3OCCO3)cc21 C(=O)(C(CCC(N)=O)N=[N+]=[N-])N1CCC(CNC(C2(C(=O)OC)CC2)=O)C(O)C1 C1(C(=O)NCC(C)N(C(c2ccnc(OC)n2)=O)C)CCc2nn[nH]c2C1 C1(C(=O)NC2CCN(C(C3(S(N)(=O)=O)CC3)=O)C2)Cc2c[nH]cc2S1(=O)=O C1(CCC)C(=O)NCCN1C(C1CN(C(c2cc(Cl)n[nH]2)=O)CC1CC)=O Nc1c(C(=O)NC2C3CN(C(C4CC5CC4C5)=O)CC23)cccc1Cl C1(CC(=O)N(C)CC2CCN(C(=O)Cc3nc(=N)[nH][nH]3)C2)CCC(F)(F)CC1 C(=O)(C(C)(C)n1ccc(C)n1)N1CC(NC(C(C)=CC2CC2)=O)C1 C(N=c1ncc(I)c[nH]1)C1OCCCN(C(c2cnn3c2OCC3)=O)C1 c1(CC(N2C(CNC(C(C(C)C)OC)=O)CC(OC)C2)=O)c(C)cccc1F N1(C(CS(CC)=O)=O)CCC(C2(NC(=O)Cn3cc[n+](C)c3)CC2)CC1 c1(CC)nn(C)c(Cl)c1C(=O)NCCC(C)N(C(=O)Cc1cc(Cl)ccc1F)C N(C(=NCCN1CCOCC1)NCC1(C(F)(F)F)CCSCC1)C1C(O)CCC1 CCC(O)C(C)C(=O)N1CC2CC1C2CNC(c1ccc(C(N)=O)c(Cl)c1)=O C1(C(N(C)CC2CCCCC2O)=O)COCCN(C(N)=O)C1 c1(C(N2C(C)CN(C(=O)C(F)n3ccnc3)CC2)=O)cccc2c1nc(O)n2C N1(Cc2cc(C)n(C)n2)CCC(C(=O)Nc2ccc(F)c(C(N)=O)c2)C(O)C1 N1(C(C2C(OC(C)(C)C)C2)=O)CC(CNC(=O)CC2CCC(=O)O2)C2(CC2)C1 C1(NC(c2ncc(OCC)nc2)=O)CS(=O)(=O)CC1NC(c1ncn(C)c1C)=O CC(C)CN=C(NCC1CCCCN1C(C)C)N1CCC2(CCOCC2)CC1 N1(C(C(C)(C)n2cc(CCSC3CC3)nn2)=O)CCC2NCCC12 C1(CNC(CNC(COC)=O)=O)CCCCC1N.C1(CCO)CCN(C(C)=O)CC1 C1(C)(CC(=O)N(CC(=O)NC(C)(C)CN(C)C)CC#C)CCOCC1 c1(C(=O)NC2C(CNC(CCSc3nc(C)[nH]n3)=O)CC2)cnc2ncccn12 C(=O)(C1=CCCC1C)NCC1(OC)CN(C(c2ccnc(C3CC3)n2)=O)C1 N1(C(C)C(c2ccc(Br)cc2)=O)CCCCCCOCC1 C#CCC(C)C(=O)NCCCN1CCC(NC(=O)C(c2ccccc2)OC)C1 c1(C(C(=O)NC2CCN2CC(F)F)OCCCF)ccccc1 c1(C(=O)NCC(CC)NC(=O)Cc2cn(C)nn2)cc(F)c(F)cc1OC(F)F C1(c2nnnn2CC(F)F)(NCCc2c(OCC#C)cccc2)CC(C)N(C)C1 N1(C(C(CC=C)C)=O)CCC=C(C(=O)N2CCC(N3CCCC3)C2)C1 N1(C(C=C(C)c2ccccc2F)=O)CCC2(C1)CN(C(C1CSC1)=O)CC(C)O2 c1(CC)cc(C(=O)N(CC(=O)NCC2(C)CCN(C)C2)C(C)C)ccn1 c1(C(N2CC3CN(C(c4ncccc4Br)=O)C3C2)=O)c(F)cccc1F C(CC(C)(C)C)(C(=O)N(C)CC1CC1(F)F)NC(c1cc(C)nc(C)n1)=O Cn1[nH]c(=NC(=O)C(=O)N2CCCC(OCCCO)C2)cc1Cl c1(OCC(=O)NCC(C)(C)NC(c2coc(Cl)c2)=O)ccccc1Cl CC1(C)CCCN(C(C23CC(CN2C(=O)C2=NOCC2)C3)=O)C1 CC(C)(CCCCNC(=O)Cn1cnc(C(N)=O)n1)NC(C1COCC1(C)C)=O c1(C(=O)OC)conc1C(C)NCc1cn(C)nn1.c1(C=O)ccn(C)c1 CCCC(CNC(C1(CC)CCC1)=O)OCC c1(C(N2CCCC(NC(C(CCC)OCC)=O)C2)=O)ccc(S(=O)(=O)NC)o1 Cc1c(C(=O)NC2CC(NC(c3cscn3)=O)C(O)C2)cccc1N C1(CNC(C(C)=O)=O)CCCCN1C(C1CC(c2ccc(F)cc2)(F)C1)=O CC(F)(F)C(F)C(=O)NC1CCC(C(=O)NCCC=CBr)C1 CC1CCC(O)(CNC(=O)C(CC(F)F)NC(=O)COc2ccccc2)CC1 N1(C(CSCCC)=O)CC2CC1CC2NC(=O)C(F)(F)c1ncccn1 C1(CNC(C(C2CC2)OCC)=O)CCN(C(=O)C=CCN2CCCC2)C1C C(=O)(CC(C)(C)CC(F)F)N(C)CCNC(C12CCC(CC1O)C2)=O Cc1ccc(C(=O)NCC2CCCN2C(c2cnc[nH]2)=O)[nH]1 CC1CCCC=C1C(=O)NCCc1ccc(Br)cc1Cl c1(CC)conc1CC(N1CC(C(O)C(=O)NCc2occc2C)C1)=O C(=O)(C(C)(O)CC(C)C)NC1CC(CNC(c2cc(C)c(CO)cn2)=O)C1 N1(C(CSCCOC)=O)CCCC12CCN(C(=O)CC(C)N1CCCC1=O)C2 N1(C(c2c(C)cccc2)=O)CCN(C(=O)C=Cc2ccc[nH]2)C(C)C1C c1(C(=O)NCCC2C(C)CN(C(C3CC34CC4)=O)C2)c(F)ccc(Cl)c1O N1(CCC)CCCC1(C(=O)NC1COCCO1)CCF C1(C(=O)NCC2(NC(CC3CCCC(C)C3)=O)CCOCC2)CC(=O)NC(=O)C1 C1(CN(C(=O)C(C2CCC2)C2CCC2)CC)CCN(C(=O)C#CC(C)C)CC1 N1(C(C=C(C)c2ccco2)=O)CCN(C(C2CCC(O)CC2)=O)CC(CO)C1 c1(CNC(CN(C)CC)=O)cn(C2CN(CC3(C#N)CC3C)C2)nn1 c1(C(=O)NC2C(CNC(CCCNC(=O)OC)=O)CC2)nccnc1N c1(C(=O)NC(C2(O)CN(C(c3cc(C4CC4)[nH]n3)=O)C2)C)ncccc1O CC1OC2(C(=O)NCC(C)(CO)NC(=O)C=CCN3CCOCC3)CC1C2 C(C(C)(O)CC(=O)N1CC(=O)CC1C(N1CC(CO)CC(C)C1)=O)OC CC(C)CC(C(=O)NC1COC2(CCC2)C1)NC(=O)CN1CCCCC1=O C12(CNC(=O)CCCc3ccc(F)cc3)CCC1CCN2C(c1cocn1)=O c1(OC)ccc(I)cc1NC(C1CC(F)CN1C(c1[nH]ccc1C)=O)=O C=CC1(C(=O)NC2CC=C(C(=O)N3CCC(O)C(CO)C3)C2)CCOCC1 CCCCCCC(=O)N1CC(C(O)C(=O)N(C2CCN(CC)C2)C)C1 S(=O)(=O)(c1cc(Cl)ccc1Cl)NC1CCN(C(C23CC(C(F)(F)F)(C2)C3)=O)C1 c1(SC)ccc2c(c1)C(NC(=O)CCc1c(F)cccc1Cl)CCO2 Cn1cc(N)c(C(=O)NC2CC(F)(CNC(c3cncc(C4CC4)c3)=O)C2)n1 n1(C(CC)C)nnnc1C(CCSC)NC1CC(OC)C1.C1(O)CCCC1 C(=O)(C1=CCCOC1)C(CCc1ccc(C(N)=O)nc1)=O.C1(N)CC(F)(CN)C1 C1(CNC(C2(CC)CCNC2=O)=O)COCCN(C(=O)CCCc2cccs2)C1 N1(C(Cc2cc(CC)nn2C)=O)CCN(C(C2(OC)CC(COC)C2)=O)CC1C C1(C(=O)NC2COC(C3CCNCC3)C2)CCc2nnc(-c3ccc(F)cc3)n2C1 N1(C(=O)OC(C)(C)C)CCC2CCN(C(=O)NCCc3ccc(O)nc3)CC2C1 C1(CN(C(C(C)NC(C)=O)=O)C(C)C)CN(C(=O)OC)CCS1.c1ccccc1 c1(C(=O)NC2(CCNC(CC3C(CC)C3)=O)CCC2)cnc2ccnn2c1C C(CC(CCC)NC(=O)CCCC1CC1)OC.C(=O)(C(O)COC)N c1(C(N2CC(C(C)(C)O)(CNC(C3C(OCC)C3)=O)C2)=O)cccc2nc(O)oc12 CC1CN(C(c2cnn(C)n2)=O)CC1CNC(=O)CCC(=O)c1cccc(F)c1 CCC(C)C(C(=O)N(CC(=O)NC1CCCC(C(C)C)C1)CC)N(C)CC C(CO)(CCCCNC(c1cn2ccnc2s1)=O)NC(=O)CC1CCS(=O)(=O)C1 CC1(C)C[Si]2(CCCC2)CN(C(=O)C(N2CCCC3(CCCOC3)C2)=O)C1 CCCC(C(=O)N1CC2CC1CN2C(c1cc2n(c1)CCOC2)=O)C(C)C C(=O)(C1=C(C)C(C)(C)OC1=O)NC(CCNC(c1cccc(OC)n1)=O)(C)C c1(C(N2CC(OC)(CNC(c3cn(C(C)C)nc3C)=O)C2)=O)occ2c1CCC2 c1(C(=O)NC(C)CNC(=O)CSC(F)F)cc(CC2CC2)on1 Cc1ccccc1C(F)(F)C(=O)N(C)CCNC(c1cncc(N)c1)=O Cc1cccc2[nH]c(C(=O)NC3CC3CNC(c3ccnn3CC(F)F)=O)cc12 C(=O)(C1=C(Cl)CCOC1)NC.C12(CC(C(F)(F)F)(NC(CC)=O)C1)C(=O)NC2 CC1(C(=O)NC2CC(=O)N(CCO)C2)CCCN1C(=O)Cn1cccc1 Cc1ccc(F)c(CC(=O)NC(CNC(=O)COCc2nc[nH]n2)C(C)(C)C)c1 N1(C(=O)CC2CC(CF)C2)CCN(C(c2c[nH]nc2O)=O)CC1 C(=O)(C(C)(C)C(F)(F)F)NCC1(F)CC(NC(c2c(C)n(C3CC3)nc2)=O)C1 c1(OC)cccc(C)c1C(N1CC(Cc2cn(-c3ncccc3F)nn2)C1)C c1(C(=O)NC2C(C)N(C(=O)Cc3ccccn3)CC2)ncnc2c1c(Br)cn2C CCC(C#N)(CC)C(=O)NCC=CCC(=O)N(C)Cc1ccn(C)n1 Cc1ccc(-c2cc(C(=O)NC3CCC(NC(=O)C(O)C4CC4)C3)no2)c(C)c1 N1(C(=O)NC(c2cncc(Br)c2)C)CCCC2(C1)OCC1CC21 C(CN=C(NC(C)C)NC1CCCN(c2nnc(C)n2C)C1)OCCOC C=CC(CC)C(=O)NC1CC=CCC1C(N1CCC(O)(CC)C1)=O N1(C(C(CC(C)C)C(N)=O)=O)CC2(C)CN(C(c3nscc3N)=O)CC2(C)C1 N1(C(COCCCC)=O)CCC(N=[N+]=[N-])(C(=O)N(CCCO)CCO)C1 c1(C2C(NC(=O)NC(CC3CCCCC3)C(=O)O)C2)ccc(F)nc1 CC(C)(C)CCC(C(=O)OC(C)(C)C)N(C1CCC12CCCCC2)C.C1C(=O)O1 C#CCCC(O)C(=O)N1CCN(CCNC(=O)CNS(C)(=O)=O)CC1 CC(C)(CCS(C)(=O)=O)C(=O)NC1CCC1CNC(C1C2CC3C(C2)C13)=O C1(CNC(C2C(C)CC=CC2)=O)CC2CN(C(=O)C3CC3)CC12 N1(C(C2CCC(OC)C2)=O)CC2CCC1CC2NC(C1CCCN(C(C)C)C1)=O CCCCCC(O)C(=O)NCC1CCN(C(=O)Cc2ccc(Cl)c(OC)c2)C1 N1(C(Cn2c(C)c(Cl)cn2)=O)CC2CCCC(NC(=O)Cc3ccns3)C2C1 Cc1cn2c(n1)CC(C(=O)NCCCCCCNC(=O)C(F)(F)C(O)C1CC1)C2 C1(CC)CCC(C(=O)NC2CCC(C(=O)NC3CC3(C)C(F)F)CC2)CC1 C1(C2CCN(C(C3CC3NC(=O)C3CC3)=O)C2)(NC(C(C(C)C)OCC)=O)CC1 N1(C(CS(CC)(=O)=O)=O)CCCCC(C2CN(C(=O)C(C)(COC)CC)C2)C1 C1(NC(C2(C(N(C(C)C)C)=O)CC2)=O)CN(C(=O)C#CC2CC2)C(C)(C)C1 c1(C(N2CC(CNC(C3CCC(C)CC3)=O)CC2(C)C)=O)cc(S(N)(=O)=O)cs1 C1(C(N(C2(CN(C)C)CC2)C)=O)CN(C(=O)CCc2nc(O)n[nH]2)CCO1 Cc1ccc(C(N2CCC(N(C)C(N)=O)CC2)C(=O)Nc2ccccc2)cc1C CCCCCCC(CC)C(=O)NC(C)CCCNC(C1(N(C)C)CCCCC1)=O C(=O)(C(F)CC1CN(C(=O)C(C)c2ccsc2)C1)N(CC(C)OC)C N1(C(C2CC(C(=O)OC)C2)=O)CCC(NC(c2csc(C3CC3)n2)=O)C(F)C1 C(=O)(C1=CCCC(C)(C)C1)N1CCCC(NC(CCCCCCC#C)=O)C1C N1(C(C(C)Sc2ccccc2Cl)=O)CCCC(NC(=O)CC2CSC2)CC1 c1(C(N(C2C(O)CCN(C(c3c[nH]c(=NC)s3)=O)C2)C)=O)ccc2cncn2c1 N1(C(CCCSC)=O)CC(C)(C(N2CC(CO)CC2CO)=O)CC1(C)C c1(C(N(C)CCNC(=O)CC2(C(F)(F)F)CC2)=O)cc2ccccc2cc1N C1(NC(CC(=C)C)=O)CCN(C(=O)CCCc2cc(C)ccc2C)CC(C)(C)C1 N1(C(CCN(CCCCC)C(C)C)=O)CCCCC(NC(c2cncnc2)=O)C1 CCC(CCCC(=O)N(C(CC1CC1)CO)C)NC(=O)CN(C)C(C)=O c1(OC)ccccc1N(C)Cc1cc(C2CCCN2)[nH]n1 N1(C(c2c(CNC(c3c(C)n[nH]c3)=O)cco2)=O)CCCCC(C)(C)C1 N1(C(c2cc(C)nc(C)c2)=O)CC2CCCC2(CNC(C2COC(=O)C2)=O)C1 Cc1cc(N)cnc1C(=O)NCC1CCC(C(=O)NCC2CC3(CCC3)CO2)C1 C1(CNC(CCC=CCC=C)=O)CC(F)(F)CN1C(=O)C(F)C(C)C CCCC(CNC(=O)CCn1cccc1)C(=O)NCC(C)(O)CCC N1(C(c2cc(C)nnc2)=O)CCCC12CCN(C(c1c(C)cccc1F)=O)CC2 c1(C(N2C3C(NC(CCN(C(CCC)C)C)=O)C(C3)C2)=O)c[nH]cc(Cl)c1=O CC1CCC(C(=O)Nc2ccc(F)cc2)CN1C(C1CCC(O)C1)=O C(=O)(C1=CCCCC1)N1C2(C(=O)NC3(CO)CC(OC)C3)CC(C1)C2 N1(C(C(CC)C)=O)CC2(CO)CC1(C(=O)N(C)Cc1ccncn1)C2 c1(C(=O)NCC2N(C(CC=C)=O)CCC2C)c(C(F)(F)F)cccc1Cl N1(C(C2C(C)(CC)C2)=O)CCC2(CC1)C(NC(c1nccc(C)n1)=O)CS2(=O)=O C1(NC(CCC=CCC=C)=O)CCN(C(C2CCCCC2(C)C)=O)CC1CO C1(NC(c2n[nH]cc2CNC(c2cnnn2C2CC2)=O)=O)C2CCCCCC12 C1(NC(COCC)=O)CC2(C1)CC2NC(=O)CCCN=[N+]=[N-].C12CCN(CC1)C2=O c1(C(=O)NC(C2CC(CCC(CC(=O)NC)C3CC3)C2)=O)c[nH]c(C#N)c1 C1(NC(C2CN(C3CCCC3)C2)=O)CCN(CC(F)F)CC1.C12(CCC1)C(=O)N2 C=CC(CCC)CC(=O)NCC1=CCCN(C(C2CC3(CSC3)C2)=O)C1 c1(C(=O)NCC(C)N(C(c2ccsc2C(F)F)=O)CC)ccc2nc(S)oc2c1 C1(NC(C(CSC)O)=O)CCCCN(C(=O)CC(O)C2CCCC2)C1 C1(CC(C)NC(c2csc(C3CC3)c2)=O)CCN(C(C2(C#N)CCCC2)=O)CC1 N1(C(c2cc(CNC(C(C)C)=O)ncc2)=O)CC2CCN(C(C)=O)C2C1 C12(NC(C(CC)(C)O)=O)CCCC1N(C(=O)COc1ccccc1Br)CC2 C1(C(=O)NCC2(C(N)=O)CN(C(c3c(C)scn3)=O)C2)CCSC(C)C1 C(=O)(CCCCC(C)(C)C)NCCCC(CCC)NC(=O)C(F)(F)C(F)(F)F Cc1cc(C)c(C#N)c(NCCNC(=O)CCC2CCC2)n1 c1(CN(C2CCN(C(C(CCC)C)=O)C2)C(C2(CF)CC2)=O)cc(F)cc(F)c1 C1(C(CNC(=O)OC(C)(C)C)CNC(=O)CCF)CCCCC1 C1(NC(C(C=CCCC)O)=O)COCCC1NC(=O)Cc1ccsc1C CC(C(C)C(=O)NC1CCCC1CF)NC(=O)C=Cc1cn(C)nn1 C1(CC(=O)N(C(C)C)CCN(C)C)CCCN1C1CCCCC1.C12(F)CC(C1)NC2 C1(CN(C(=O)CC2CCCCN2C(c2ccnnc2)=O)C)CCC(C)(C)CO1 c1(C(=O)NCC(C)N(C(=O)C(C)(C)C(N)=O)C)nc(C(F)(F)F)n2c1CCCC2 Cc1nn(C(C)C)c(C)c1NC(C1CC(F)CN(Cc2ccnn2C)C1)=O C1(CC(=O)NCCCN(C(=O)Cc2ccc(F)cc2)CC)CC2(CCC2)C1 C1(CCNC(Cc2c(C)scc2)=O)CN(C(c2ccc(Cl)cc2)C)CCS1(=O)=O CC1CC(C)(C(=O)NCCCN2CCC(NC(C3CC(F)(F)C3)=O)C2)C1 C1(NC(C2CN(C(C(C)OCC)=O)CC2(F)F)=O)CCCCCC1(C)C C(=O)(C#CC1CCCCO1)NC1CN(C(c2cc(OC)ncn2)=O)CC(O)CC1 c1(-c2cnc(C)nc2)ncn2c1CN(C(c1cnc(Cl)c(F)c1)=O)CC2 C1(NC(C2(C#C)CCC2)=O)CCCC(NC(=O)CCNS(=O)(=O)C(F)(F)F)C1 c1(C(N2CC(F)CC(NC(C3CC(=C)C3)=O)C2)=O)ccc2nc(Cl)nn2c1 Cc1cn2c(n1)C(C)N(C(c1sc(C)cc1Br)C(=O)NCc1nnn(C)n1)CC2 c1(N2C3CC(=C)CC2CC3)nc2c(c(=NC3CCn4cnnc4C3)[nH]1)CCCC2 CC1CN(C(C2CCCSC2)=O)CCN1C(c1ccc(C2CCCO2)[nH]1)=O c1(C(N2C(C(C)NC(C(C(=O)NC)(C)C)=O)CCCC2)=O)nc2ccccc2s1 CC1CN(c2nnnn2-c2ccccc2)CC(C)S1=O.c12ccc(cc1)OCC2 c1(C(=O)NC(C2CCN(C(C=C(CCC)C)=O)C2)(C)C)cc2c([nH]1)CCOC2 C1(F)(C(C2CC2)NC(c2c(OC)c(Cl)ccc2)=O)CC(N=c2nc[nH]cc2C#N)C1 Cn1c(O)ncc(NC(=O)NCC2CC3CCC2CC3)c1=O C(=O)(C1=C(Cl)CCCC1)NCCCNC(C(c1n(C)ccc1)=O)=O CC(CCN=C(NCC1CCCCO1)NCC(c1cccs1)C)C(F)F CCC(CCC(=O)NOCc1ccco1)NC(=O)CCc1csnn1 Cc1cc(C)cc(S(=O)(=O)NC2CCC3(C2)CN(C(c2cnsn2)=O)C3)c1 O=C(CC(C(F)(F)F)N1CCCCC1)NC1CC1CNC(=O)C(F)F N1(C(C(c2ccn(C)c2)C)=O)CC2(CC(C(N3CC(N(C)C)C4(CC4)C3)=O)CO2)C1 C(=O)(C1=CS(=O)CCC1)N1CCCC(CNC(c2ccccc2C(F)F)=O)C1 CCCC(CCCNC(=O)CCCC(C)C)NC(=O)CC.C(C(F)(F)F)=CC C(CCC(C(=O)NCCOCCO)NC(C1C2CCC(C2)C1C)=O)CCN=[N+]=[N-] C(=O)(CC(F)(F)C(F)(F)F)NCCCCC1CCN(C(CSC(C)C)=O)CC1 CC1(C)CC(CCN2CCC(c3cc(Cl)ccc3I)CC2)CC(C)(C)N1 C1(NC(c2cc(C3CC3)no2)=O)CN(C(=O)Cc2nnc(O)s2)C2CCCCC12 n1(CC(=O)NCCCC2(NC(c3c(SC)snn3)=O)CC2)ncc(C)cc1=O Cc1c(C(=O)NCC(F)CNC(c2cnoc2CC(C)C)=O)cnn1C N1(C(=O)C(N2CC3CC2CC3O)=O)CCC(O)C(C2CCCC2)C1 n1(CC)c(=O)nc(O)c2cc(C(N3CCN(C(=O)CC4CC4)CC3C)=O)cnc12 c1(C(N2C3(CN(C(c4scc(CC)n4)=O)C3)CC2)=O)nc2ncccn2n1 C1(C(=O)NCc2c(C3CN(C(CC(C)(C)SC)=O)C3)ocn2)Cc2ccccc2S1 c1(C(N2CCC(CCNC(C=C(CC)C)=O)C2)=O)cc(C(C)C)n(C)c1C C1(CCC)CN(C(=O)C(CC(C)C)NC(N)=O)CCN1C(=O)CCCCSC C1(NC(C(c2cnc(C)o2)C)=O)CCCC1(C)C c1(C(=O)NC2C(NC(c3cnc(C)[nH]3)=O)CC2)ccc(Cl)cc1Cl CC(CC(F)F)C(=O)NCC1=CCN(C(c2ccccc2-c2nc[nH]n2)=O)CC1 C(=O)(CS(=O)c1ccc(Cl)cc1)N(CCC)CCNC(=O)C(F)CC C(=O)(CCCCC(=O)N1CCCC(CNC(C2(C)CCC(F)(F)C2)=O)C1)OC N1(C(c2cc(COC)oc2C)=O)CCOCC(F)(CNC(c2cnccn2)=O)C1 C1(C(=O)NC2CC(NC(Cc3nn(C)c(Cl)c3)=O)C2)C2CCN(CC2)S1(=O)=O C1(NC(=O)OCC)CC2CCC1N2C(=O)NCC1CN(C)CCO1 C1(C(=O)NCCC(C)(C)NC(=O)Cc2nc(=N)[nH][nH]2)CCCCC1N1CCCC1 C1(C2CC2)(C(=O)NCC(=C)F)CN(C(C2CC(C)(F)C2)=O)C1 C(=O)(C(O)CC(C)(C)C)N1CC2(CC(CC(=O)NC(COCC)C)C2)C1 Cc1c(C(N2CCC(CO)(NC(C3CC3C(N)=O)=O)C2)=O)csc1Br CCC1=NOC(CN(CC#N)C(N2C(CC(=O)OC(C)(C)C)CCC2)=O)C1 n1(CC(=O)NC2CC(C)(C)CN(C(C3(O)COC3)=O)C2)[nH]cc2c(=O)ncnc1-2 N1(C(CSC(C)C)=O)CCCC12CCN(C(=O)C(C)NC(C1CCCO1)=O)CC2 c1(C(N2C(CNC(c3c(OC)ccs3)=O)CCC(C)C2)=O)cnn2c1NCCC2 C1(C(=O)NCC2N(C(C)=O)CCC2)CCN(C(=O)CNC=O)C1C(C)C C1(NC(C2(N(C)C)CC2)=O)CCCN(C(C2CC(c3ccccc3)O2)=O)C1 c1(OC)cc(C)sc1C(=O)NCC(C1CC1)NC(c1ccc(C(N)=O)[nH]1)=O c1(OC)c(-n2cc(CN3CCN(C(C4CNC(=O)N4)=O)CC3)nn2)cccc1Cl O=C(C1CCc2ccccc21)NCC1CCCN(C(C2(n3ccnn3)CC2)=O)C1 N1(C(c2c(F)cc(C)c(F)c2)=O)CC2COCC(C1)C2NC(=O)CSCC(C)C Cc1cc(=NCc2cc(F)ccc2Cl)[nH]cc1S(=O)(=O)N1CC(O)CC(C)C1 C1(C#CC(=O)NOC(CO)C(C)C)(NC(CC)=O)CCCC1 S(=O)(=O)(c1ccc(C#N)c(NCC2CCCOCC2)c1)NC(CCC=C)C Cc1ccc2c(c1)SC(C(=O)NCCC(O)CNC(c1sccc1C)=O)C2 c1(C(=O)NCC2(C)CC(NC(C3(C4CC4)CCC3)=O)C2)cnc2[nH]ccc2n1 c1(C(c2ccc(Cl)cc2)C(=O)S(CC2C(C)(C)OCC2)(=O)=O)cccc(Cl)c1F C1(C(=O)OC)COC(C)(C)CN1C(=O)C(C)CC1CCC1.CCCCC(=O)NC CC(C)C(O)C(F)(F)C(=O)N1CC(O)(CCNC(c2ncc3ccccn23)=O)C1 N1(C(C(C(C)C)NS(C)(=O)=O)=O)CC=C(CCNC(=O)CC2CCOC2C)CC1 c1(OC)cccc(C(=O)NCC2CC(C)N(C(C3(CO)CCCO3)=O)C2)n1 C1(C(N(CC(C)N(C(=O)C=CCn2cncn2)CC)CC)=O)CCN(C)S1(=O)=O C#CCCCC(=O)N1CC(NC(C23CC(CCC)(C2)C3)=O)C(C)C1 c1(C(=O)NCC(C(C)C)NC(C2C(OC)CCCC2)=O)cnc2sc(C)cn12 N1(C(CCCC)=O)CCCC(C(=O)NCCN(C(c2[nH]nnc2C)=O)CC)C1 C1(CC(=O)NCC23C(CN(C(CCN(S(C)(=O)=O)C)=O)C2)C3)CC(C)(C)OC1=O C1(COC)(NC(=O)C(C)n2cnnn2)CCCN(C(c2csc(=N)[nH]2)=O)C1 C=C=CC(C)C(=O)NC1(CNC(c2coc(C(=O)OC)n2)=O)CCOCC1 c1(NCC)ccccc1C(N1CCNC(C(=O)NCCc2ccccc2)C1)=O c1(COC)cc[nH]c1C(N1CC(CCCCNC(=O)C(c2ccccc2)C)C1)=O N1(C(C(CC=CC)NC(=O)C(=O)Nc2ncc[nH]2)=O)CCCCC(C)C1 c1(C(=O)NCC2(NC(Cc3ccc(C)o3)=O)CCOC2)cnn(C)c(=O)c1 c1(C(N(C)CC2(O)CN(C(=O)CCOC3COC3)C2)=O)ccc(F)cn1 C1(=CCNC(=O)C(Cl)=CCl)CCN(C(C2(F)CC2)=O)CC1 C(=O)(C(CNC(C1CC(=O)CS1)=O)OC)N(C(CC#C)C)C C(=O)(C1CNC(=O)c2ccnn21)N1CCC2(CCN(C(CC3(C)CCC3)=O)C2)C1 c1(C(COC)NC(=O)C(=O)NC(c2ccc(OC)cc2)C2CC2)cc(F)cc(F)c1 C1(C(=O)NCCN(C(c2nccc(OC)c2OC)=O)CC)CCCC1S(C)(=O)=O CCC(C#N)(CC)C(=O)NC(c1ccc(CNC(c2ccc(CC)[nH]2)=O)cc1)C c1(CCNc2c(C3CCN(C(=O)OC(C)(C)C)C3)n[nH]c2)ccc(F)c(F)c1 c1(CNC(=NCCc2c(OC)ccc(Cl)c2)NCCF)cc2cc(F)ccc2o1 C12(C(=O)NC(C(=O)OCC)CO)CCC(CN(C(=O)CC(C)F)C1)C2 C1(NC(c2n(CC)nnc2)=O)CN(C(=O)CC(C)(C)C)Cc2nccn2C1 C1(CC(=O)NCCCC2CCCOC2)CN(C(c2cccc(F)c2)=O)CCO1 C1(C(=O)NC(C)CC2CN(C(C3CC3(C)C(F)F)=O)C2)CC(F)C(=O)N1 c1(C(N2CCCN(C(C(C=C=C)C)=O)CC2)=O)c(C)cc(F)cc1C C1(CC)CN(C(=O)CCc2cn(C)nn2)CCC1NC(C1(O)CCC(C)CC1)=O C(C(C)C=O)OC(C)Cc1ccccc1.n1(COC)cc(C)nn1 CCC(O)C(F)(F)C(=O)NCc1ncoc1CCNC(=O)C(c1cnn(C)c1)C C(C(C)C)(C(O)C(=O)N1CC(C)C1C(=O)NCC(C)(O)C1CC1)OC N1(C(c2cc(CNC(C(C)=CC=C)=O)[nH]n2)=O)CCOC(C)C1C N1(C(C(C)CNC(c2cnn(C)c2Cl)=O)=O)CCC2(CC=CCO2)C1 C(=O)(C1CCc2ccc(OC)nc21)N1CC(OCCNC(COC)=O)C(CO)C1 CCCS(=O)(=O)CC(=O)N1CCC(C(C)(C)CNC(C2CC2C)=O)CC1 c1(O)ccccc1C(=O)NOCC1CC1(F)F.c1cccc(Br)c1 N1(C(c2cc(C)nc(C)c2)=O)CCCC2(C1)CN(C(=O)CN1CCCCC1=O)C2 N1(C(c2cc(C)cc(Cl)c2)=O)CC(NC(=O)CC2CC(=O)C2)CC12CCOC2 N1(C(CCCOCC)=O)CCC(C(=O)NC2CC2C2CC2C)C1(C)C CC(CCN(C)C)C(=O)NC1C2CN(C(=O)Cc3cnnn3C)CC12 C1(C(N(C(C)C)CCN(C(=O)CCCS(C)(=O)=O)C)=O)CN2CC3CC2(CO1)C3 CCC(C(=O)N1CCOC(C(=O)N(CC(O)(CC)CC)C)CC1)C(C)C c1(NC(CCN(C)CC2C(C)OCC2)=O)cccc(OC(F)F)c1 C1(C(=O)NCC(=O)OCC)CCC(C)(C)N(C(=O)C(C(C)C)SCC)C1 c1(CNC2C(C(=O)NCC(C)OC)C2)cccnc1.C12(COC1)N(C)C2 c1(COC)cc(C(=O)NC2(CF)CN(C(C3CN(C)C(=O)N3)=O)C2)n(C)c1 Cc1cc(F)c(C(N2CC3CC3(NC(c3csnc3C)=O)C2)=O)c(Br)c1 Cc1nn(C)c(C)c1CCCNC(=O)COC(=O)CNc1ccncn1 CC(CC(=O)N1CCN(C(=O)CCc2cnn[nH]2)C(CC2CC2)C1)C(F)F c1(NCC(S(=O)(=O)NC)C)nc(N2CC(=O)NC3(CC3)C2)nc2ncn(C)c12 C1(N(C(=O)C(F)=C(C)C)CCC)CCN(C(C2CCCC2SC(F)(F)F)=O)C1 CC1=C(C)CC(C)(NC(=O)CCC2(C)CN(C(C3(C)COCCO3)=O)C2)CC1 C1(C(=O)NCc2cn(CC=C)nn2)CCOCCN1C(=O)C(CC)NC(C)=O C12(NC(=O)CCCCN3CCCC3)CCOCC1CN(C(=O)C(F)F)C2 N1(C(c2c(OC)cc(C#N)cc2)=O)CCC2CCC(NC(=O)CC3CC3C)C1C2 C=CCC(C(=O)NCCC1CN(C(c2ccc(OC)nc2Cl)=O)C1)C(C)C C1(C(N2CCC(N(C(Cc3cc(OC)no3)=O)C)CC2)=O)CCC2CC2CC1 c1(OC)ccc(C(=O)NCCC2CCCN2C(C2COC(C)C2)=O)c(Cl)c1 C(=O)(CC(CNC(=O)C=C(C)C1CC1)C(F)F)NC(COC)(C)C c1(C(=O)NCC(C)CNC(C2CC3C=CC2C3)=O)c[nH]c(=O)cn1 N1(C(CC2CCCC(C)O2)=O)CCCC2C(NC(=O)Cc3cncs3)C(C)(C)C12 C1(CNC(=O)NCCCSC(C)(C)C)CCCC2(CC2)C1 C1(O)(C(=O)NCc2ccc(C(C)NC(CSC)=O)cc2)CC2(CCOCC2)C1 N1(C(CCOCCOCC)=O)CCC2(CC2)CC1C(=O)NCC1CCC(C)(C)C1 N1(C(c2c(CC)cns2)=O)CCCN(C(=O)CCc2cccc(C#N)c2)CC1C C1(CC(=O)N(CCOCCN(C(=O)CC2CCCSC2)C)C)COCCO1 C(=O)(C1CCCc2ncccc21)NCCNC(c1c(C)nn(C(C)(C)C)c1C)=O C=C(C)CCC(=O)NC(C)CCCCNC(=O)C(N1CCSCC1)C c1(OCC)cccc(Br)c1C(c1nnnn1C1CC1)NC1(CF)CC1 C12CC(=NO1)c1ccc(cc1)N2.CCCCCCCNC(=O)CCC(=O)OC C1(CNC(C(C)(C)N2CCC2)=O)CCC2(CN(C(=O)C(F)OC(F)(F)F)C2)O1 CCCCC(C)(F)C(=O)N1CC2(C(=O)NC(C)CN(C)C(C)C)CC1CO2 n1(CC)cc(Cl)cc1C(N1CCC(C)(NC(c2cnc(C3CCOC3)s2)=O)C1)=O C#Cc1ccc(C(=O)NCc2cc(C(N3CC(O)CC3C)=O)on2)cc1C c1(OCC)c(CNCC2(C(=O)Nc3ccc(C)nc3)CC2)cccc1C C12(C(N(C(c3ccccc3)CNC(=O)CCCF)C)=O)CCC(C1)C2 N1(C(C2(CSC)CC2)=O)CCC(CCN(C(=O)CCc2cc(C)sc2C)C)CC1 C1(C(=O)NC2(CC(=O)OC)CC2)CCCN(C(C2CC2C2CCCCO2)=O)C1 C1(NC(C(CC)(C)O)=O)CCC(C)N(C(C2CCC(C(=O)OC)C2)=O)C1 C1(CNC(C=CSC)=O)CC2(CCN(C(c3cccn4cnnc34)=O)C2)CO1 Cc1nc2cc(C(=O)NC3CC(O)CN(C(=O)CC4CC5(CC5)C4)C3)ccc2s1 c1(C(=O)NC2CCCN(C(C(CCOC)C)=O)C2C)ccc(C)c(Cl)c1N CC1=C(C(=O)N2CCCC(CNC(C3CC34CC(C)(C)C4)=O)C2)CCCO1 C1(CCCC)CCCN(C(C2(C)CN(C(=O)C(F)C3CCCC3)C2)=O)C1 c1(C(N(CC(C)NC(C2CC2(C)C)=O)CC)=O)cccc2c1ccn2C(C)C c1(C(=O)NCCC2OCCN(C(C(CC)C#N)=O)C2)cccc(=O)n1C Cc1ccc(SCCC(=O)NCC2COC(CNC(c3coc(C)c3)=O)C2)cc1 N1(C(C(COC)NC(c2csc(C)n2)=O)=O)CCC(F)(F)C(CO)C1 C1(C(=O)OC(C)(C)C)CCN(C(C2(C)CCC2)=O)C2CC12.C1CCC(=O)N1C CCC(C)C(C(=O)N1CC2CC2(CNC(c2ccco2)=O)C1)c1ccccc1 C1(C(N(C2CCN(C(C)=O)C2)CC)=O)CCc2ccccc2O1.C12CC(C1)NC2=O CCCCCC(C)CC(=O)N1CCN(C(c2ccc(CCC)[nH]2)=O)C(C2CC2)C1 C1(NC(c2cn[nH]c2)=O)CN(C(C2CC3CCC2O3)=O)CCC12CCC2 C1(C(=O)NCc2c(C)n(C)nc2)C2CCC(C2)N1C(=O)CC1CCCSC1 CCC(C)C(O)C(C)C(=O)NC1C(CCNC(=O)OC(C)(C)C)C1(F)F C(CC1CC1)(C(=O)NC)NC(C(C)=CC(=O)OCCc1ccsc1)=O C1(CC(=O)NCC2(F)CCN(C(CCSC)=O)C2)CCOCC1(C)C CCCC(C)C(=O)N1CC(C)C1CN(C(=O)N(C)C)CCC c1(C(=O)NC2C(CNC(=O)Cn3cccn3)COC2)cc2c(cn1)OCCC2 CC1C(NC(=O)C(F)(F)CO)CCCN1C(=O)C=Cc1cccnc1 N1(C(CC2CC(=C)C2)=O)CC(NC(=O)CC2CC3CC3C2)C(CC2CC2)C1 CCCC(C(O)C(=O)Nc1ccc(OCC)nc1)NC(=O)CC(C)C Cn1cc(C(=O)NCC2CC3CC2CN3C(=O)CCOC2CC2)cc1S(N)(=O)=O C1(NC(C(CCC)(C)C)=O)CC2CCC1C(NC(=O)Cc1ccn(C(C)C)n1)C2 Cn1c(C(=O)N(C2(C(=O)NCC3C=CCOC3)CC2)C)nnc1S C12(C(N3CC4CC4C3)=O)CCC(CNCC3CCCCO3)(CC1)CC2 CS(=O)(=O)c1cc(C(=O)NC2CCC(CNC(c3cnc(O)o3)=O)C2)co1 C1(CC(N)=O)CC(O)CN1C(=O)CC1(NC(C2C3CC(=O)CC23)=O)CCC1 C1(NC(C(C)C#N)=O)C2CC(NC(c3cccc(OCC(F)F)c3)=O)CC12 c1(C(=O)NC(CCCC)CNC(c2ccn(C3CCC3)n2)=O)cc2cn[nH]c2cn1 Cc1cccc(Cl)c1C(=O)NC1CCCCC1CNC(c1ocnc1C1CC1)=O c1(C(=O)NCC(CC(=O)NCC(F)(F)C(C)C)OC)cnc(O)c(C)c1 N1(C(C(CCC)NC(C23CCC(C2)C3)=O)=O)CC(N(C)OC)C1 CCC(CNC(c1ccnnc1C)=O)(CC)C(=O)NCc1ccnn1C(C)C c1(-c2c(C(F)(F)F)ccc(C#C)c2)ccc2c(c1)CN(Cc1nn(C)nc1C)C2 c1(CC)oncc1C(N1CC(C(C)NC(=O)Cn2cnnc2)C1)=O C1(C(=O)NC(CC)C(N)=O)C=CCCN1C(C1CC(F)C1)=O Cc1cn2nnc(C(=O)NCCC(O)CNC(C3(CC4CC4)CC3)=O)c2c(O)n1 N1(C(C(C=C)(C)C)=O)CCC2CN(C(c3cc(Cl)ccc3OCC)=O)CCC2C1 c1(OC)c(C(=O)NC2CCCN(C(=O)CCC3C(=O)ON=C3C)C2)cccc1F C1(C(N2CC(CC)C(NC(C)C)C2)=O)CC2COCC2C1.C12(CCC1)C(=O)N2 C(=O)(C1SCc2cccnc21)N(C1CCN(C(c2ccc(F)c(CO)c2)=O)C1)C c1(C(N(C(CCNC(c2nc(C)n(C)c2C)=O)C)C)=O)cc2c(nc1N)CCC2 c1(C(C(F)(F)F)OC(C(c2ccc(OC)cc2)C)=O)cc(Cl)ccc1Cl C1(F)(CC)CCCN(C(c2cc(C(F)(F)F)ccc2F)C(=O)NC(C)C)C1 O(NC(=O)C(C(C)CC)C(C)C)CC(=C)C.C1(=O)C(C2CC2)N1 C12(CNC(C(CC=C)C)=O)CC(CNC(=O)C(O)C(F)F)(C1)C(C)(C)O2 c1(C(=O)NCC(C)NC(=O)C(C(C)O)N(C)C)nn(C(F)F)cc1Cl Cc1nn(C)c(C)c1C(=O)NCC(O)CNC(C1(C(C)C)CCCO1)=O C1(NC(c2cscc2Cl)=O)CCN(C(=O)Cn2cc(C3CC3)nn2)CC1 C1(S(=O)(=O)c2ccccc2)(c2onc(-c3ccc(OC)cc3)n2)CC1 C1(NC(c2c(COC)noc2)=O)CCN(C(=O)CC2CC3(CCC3)CO2)CC1C C1(NC(C2CCCN(C)C2)=O)CN(C(C2CC(CC3CC3)C2)=O)CCC1F CC(C)C(C(=O)N1CC(C(C(=O)N(CC(C)(F)F)C)N(C)C)C1)n1cnnc1 C12(NC(c3cn(C(C)C)nc3O)=O)CCN(C(C3(CF)COC3)=O)CC1C2 C(=O)(CCCF)N(C)CCN(C)C(C1CC(CNC(=O)OC(C)(C)C)C1)=O N1(CC(=O)N(CC(C)N(C(=O)C(C)c2ccco2)C2CC2)C)CCP(C)(=O)CC1 c1(C(N2C3C(N(C(c4cnc(C)[nH]4)=O)C)CC(C3)C2)=O)ccc2ncn(C)c2n1 O=C1CC2COC(C(N3CCC(c4ncccn4)C3)=O)CN2C1 C(=O)(CCCC#N)N1CC(C)(NC2CC(c3ccccc3)CCO2)C1 N1(C(CC(OCC)OCC)=O)CCN(C)C(C(=O)NC(C)(C)CCF)C1 C1(CC(=O)NC2C(NC(C3(OCC)CCOCC3)=O)COC2)CCCC(C)(C)C1 C(C)(CCCCNC(c1sc(CN(C)C)nc1C)=O)NC(C1C(C(=O)OC)C1)=O C1(CNC(C(c2ccc(F)cc2F)C)=O)CN(C(=O)CCC(F)(F)F)CCN1C N#Cc1cncc(NC(c2cc(CNC(c3ccncc3Cl)=O)cs2)=O)n1 C(CC(C)CC)(C(=O)N1CCCC1CN(C)C)NC(C(C=C)CC)=O C(C(O)(CNC(C1CC(=O)CN1C(C1(C)CC=CC1)=O)=O)CO)OC C=CC1(CC(=O)NCC(CC)NC(c2cc(C(C)C)ccc2O)=O)CCCCC1 C(C(C)C(C)C(=O)N1CCC(CF)(NC(c2ccc(Cl)nc2C)=O)C1)OC C1(NC(C(C)NS(CC)(=O)=O)=O)CCC2CC1CN2C(=O)CC1CCCCC1 c1(C(=O)NC2(CCOC)CCN(C(c3ccncc3N)=O)C2)cc(C)nnc1O CCCC(C)CC(=O)N1CC(CC)(NC(C2CCC23CCC3)=O)C1 N1(C(C(CC)O)=O)CCCC(NC(=O)C(c2ccccc2C(F)(F)F)(F)F)CC1 C1(NC(c2cc(CNC(CNC(=O)OC)=O)no2)=O)CN2CCC1C2 C(=O)(C(C)(O)CC(F)(F)F)NCCC1N(C(CN(C(C)=O)C)=O)CCC1 N1(CCC(N2C(CNC(c3cnc(CC(C)C)s3)=O)C=CC2)=O)CCNC(=O)C1 C1(c2n(CCOC)nnn2)(OC)CCOCC1NC(c1nncs1)C C#CC1CCCN(C(=O)C(c2cn(C)nn2)NC(c2ccccc2F)=O)C1 C1(OCC(=O)NCCNC(C(C)C)=O)CCN(C(C2CCC(O)CC2)=O)CC1 c1(C(=O)NCC(C2CCCN2C(C2CCS(=O)CC2)=O)(C)C)cncc(F)c1 C(=O)(CC(F)(F)CC(=O)OC)NC(CNC(c1c(OCC)c(F)ccc1)=O)C C1(NC(c2ccc(C)s2)=O)CC(CC(=O)NCc2ccncc2F)C1(C)C N1(C(c2cc(CSC)on2)=O)CCC2(CCC2NC(=O)CC(C)SC)CC1 c1(CC(=O)NC2C3CN(C(C=CC=CC)=O)CC2C3)ccc2c(c1)CC(C)O2 n1(CC)ccnc1C=CC(=O)N(CCNC(=O)CC1CCC(C#N)C1)CC1CC1 C1(CC(=O)NCCC(CNC(CSCC=C)=O)OC)CCn2cncc2C1 N1(C(CC=C=C)=O)C2CC=C(C(=O)NCCn3ccnc3C)C1CC2 Cc1c(C(=O)NCC2CC2CNC(=O)C(C)(F)F)sc2[nH]cnc(=S)c12 CC(CC(=O)N1CC2=C(C1)CN(C(=O)CC1CCC3CC13)C2)C(F)(F)F C1(CCNC(c2[nH]cc(CC)n2)=O)CN(C(=O)CCc2cncc(F)c2)CC1C C1(C(=O)NCC(O)CCNC(C2(Br)CC2)=O)CC2CCC1O2 N1(C(CNC(C2(C(C)C)CCC2)=O)C)CCCC1C.C(CC=O)CC#C Brc1nc(CNC(c2nnnn2CCC2CC2)C2CC3CC3C2)cs1 N1(C(CCCSC)=O)CCC2C(C1)NC(=O)CN2C(c1cc(C)ncn1)=O Cc1cccc2[nH]c(C(=O)N(C)CC3CCCN3C(=O)CCOCCOC)cc12 C1(C(N(C(C)CNC(c2occc2Br)=O)C)=O)CCCCC(F)(F)C1 C1(NC(CN2CC(C)C2)=O)C2CCN(C(=O)C(C3CCCO3)N(C)C)CC12 C(C(C)(O)C(=O)NCCCNCC=CCNC(=O)CC(=O)N(C)C)OC C1(O)(CC(=O)N(CCCNC(C(F)=C(C)C)=O)C(C)C)CCCN(C)C1 c1(C(N(CCCNC(C2CC(C)(C)C2C(F)(F)F)=O)C)=O)cc2sccc2[nH]1 CC1CN(C(=O)C(F)F)CC(C)N1C(=O)CC1CCCCC(=O)N1 CC(CN(C)C)CC(=O)NC1CCC(NC(C2(CN(C)C)CC(F)(F)C2)=O)C1 c1(C(CNC(c2c(CC)n(-c3ccc(F)cc3)nc2)=O)(C)C)ccc(F)c(F)c1 C1(C(N2CCC(C(C(C)C)NC(c3cscn3)=O)CC2)=O)Cc2nnc(C)n2C1 c1(C(=O)NCC2(N(C(COCCOCC#C)=O)C)CC2)nccc2ncccc12 c1(C(=O)NCCN(C)C(C2CCC(F)(F)CC2)=O)ccc2c(O)nc(S)nc2c1 c1(CSCCN(C(CSC)=O)C)cc2ccccn2c1 C(CN=c1[nH]c(=NCC2CCCC23CCC3)[nH]c2c1CSC2)N1CCC(C)(F)C1 Cc1nsc(N)c1C(=O)NC1CC(F)(CNC(c2sc(C(C)C)nc2C)=O)C1 N1(C(Cn2ncc(CC)c2)=O)CC(O)CC1(C)C(N1CCCC(CCO)CC1)=O c1(CNC(CSC)=O)ccc2c(c1)CCN(C(=O)C(C)(C)F)CC2 C(CCC)(C(=O)N1C(C)CCC1)=CCC.C(C(C)(C)C)NC.C(=O)(CN(C)C(C)=O)N c1(C(=O)NC2(C)CCN(C(c3cnc(CC(C)C)s3)=O)C2)ccc(F)c(F)c1 N1(C(=O)CS(=O)(=O)C2CC2)CCOC2(C1)CN(C(C1CC1Cl)=O)C2 Cn1cc(S(N)(=O)=O)c(C(N2CC(CNC(=O)C(O)C3CCC3)C(C)(C)C2)=O)n1 N1(C(C2(C)CCCCC2)=O)CC(NC(C2CC(C(F)F)C2)=O)CC(O)C1 C1(NC(CCC(C)N(C)C)=O)CN(C(=O)COc2ccsn2)CC12CCOCC2 C(=O)(C#CC1CCCC1)NCCC(=C)CNC(=O)CC1CCc2ccccc2C1 CC(C)C(C(=O)N1CC2C(C1)C2(C)C)C(C)NC(=O)CN1CC=CC1 N1(C(c2cn(CCOC)nc2)=O)CCN(C(c2ncn(C(C)C)n2)=O)C(C)C1C C1(C(=O)NC(C2CCCN2C(=O)C(c2cc(Br)co2)=O)(C)C)CCCCCC1 Cc1ccc(C(=O)NCCCC2(NC(c3cc[nH]c(=N)n3)=O)CC2)cc1Br C1(C(=O)NCC(F)CNC(c2cc(C3CCC3)no2)=O)(OC)CCSC1 CC1CCN(C(C23COC(C2)C3)=O)CCN1C(=O)CC1OCCO1 C12CCC(CC1)C(=O)N2.N1(C(CC2(C)CC2Br)=O)CCC(c2cn(CCO)nn2)C1 C1(NC(C(C)C)=O)CC2(CCC(NC(=O)C(C)C3CCCC3)CC2)C1 C1(NC(C2CCCN(C)C2)=O)C2CCC1CN(C(=O)CCc1ccsc1)C2 c1(C(=O)NC(CC#C)(C)C(=O)N(CC(C)(C)CO)C)cc(C#N)ccc1N C(=O)(C1(C)COc2ccccc21)NC1CC(NC(C2(OCC)CCSCC2)=O)C1 Cn1[nH]c(C(N2CCCC2C2(NC(c3cccnc3N)=O)CC2)=O)nc1=O C1(C(=O)NC23CC(NC(c4nn(CC)nc4Br)=O)(C2)C3)CCc2nccn2CC1 n1(CC(=O)N(CCNC(C2(CC)COC2)=O)C2CC2)nccc1C C12(C(=O)NC(C)C(=O)NCCF)CC(C)(CN1C(=O)CC1(C)CCCC1)C2 c1(C2(C)CC=CC2)nc(CC2CCOCC2)nn1-c1ccc(F)nc1 C1(C(C(=O)NC(C2(C)CC2)CO)(C)C)CCCN(C(=O)Cc2cncs2)C1 c1(NC(C2C(NC(c3ncc(OCC)nc3)=O)C2)=O)ccc(OC)nc1Cl N1(C(C)=O)CCN(C(=O)Nc2ccccc2)CC1NC(c1ccno1)=O c1(NC(=O)OC)cc(C(=O)N(C)CCNC(=O)C(C(C)C)N(C)C)ccc1F c1(C(=O)OC)nn(C)c2c1CN(C(=O)C(=O)N(C1CCCN(C(C)C)C1)C)CC2 C1(CNC(CCOC(C)C)=O)C2CC2CN1C(=O)CSc1nncn1C(C)(C)C N(C1CN(C(=O)C(C)=C2CC2)CCc2ccccc21)C(c1ccn(CC=C)n1)=O c1(C(=O)NC(CN(C(C(COC)(C)O)=O)C)(CO)CO)cc(C)c(C)[nH]1 c1(CCCNC(C(=O)NC(C)C(N)CO)=O)ccc(O)cc1 N1(C(c2n[nH]c(C)c2Cl)=O)CCCC(F)(CNC(=O)COc2cnn(C)c2)C1 C1(OCC)COCCC1C(N1CCOC(CNC(c2cccnc2)=O)C1)=O C(CCCCCNC(=O)COC1CCOC1)NC(C1(N(C)C)CC1)=O CC(C)(C)C#CC(=O)N1CCCCC(CNC(C2(S(C)(=O)=O)CC2)=O)C1 N1(C(C2CCN(C(c3c(C)cns3)=O)CC2O)=O)CCCCCCC1C CS(=O)(=O)c1ccc2c(c1)CCN2C(N1C2CCCC1COC2)=O CC(F)(F)CCC(=O)NCCC1CCN(C(c2cnc(N(C)C)o2)=O)C1 c1(NCC(=O)NC(CC)CNC(c2ccc(C(N)=O)o2)=O)ccc(F)c(Cl)c1 C12(NC(c3c(OC(C)C)nccc3)=O)COCCC1CN(C(=O)CC(C)(F)F)C2 CCCCCCN(CC(=O)NCC(C1CC1)NC(=O)Cc1cscn1)CC(F)F c1(CNC(CC2(C)CC2)=O)ccc(CNC(C2CCC2C(F)F)=O)nc1 C(C(=O)OC(C)(C)C)(C(=O)N1CC(CNC(C2CCCN2S(C)(=O)=O)=O)C1)OC N1(Cc2cnc(-c3ccccc3)s2)CCC2C1CCN2CC1(CBr)CC1 c1(C(=O)NCC2(F)CCN(C(c3[nH]cc(C)c3)=O)C2)ccc2cc[nH]c2c1F C1(C(=O)NC2CN(CC)C2)(SC)CCN(C(=O)C(c2cccc(F)c2)F)CC1 c1(C2N(C(=O)NCC(=O)Nc3cc(C)c(Cl)cc3)CCC2)nc2ccccc2[nH]1 c1(C(=O)NCC(=O)NC2(C)CC(NC(C(C)NC(C)=O)=O)C2)cccc(F)c1 C(=O)(CCC(C)(C)C#CC)N1CC(C(C(=O)NC2CC(OCC)C2)O)C1 N1(C(CC(CC)(F)F)=O)CCC(NC(c2cc(OC)ccc2N)=O)C(CO)CC1 C1(=O)C(C(C)O)N1.C(COC)(CO)C(=O)CN.C1(=O)CN1.C(C)(=O)OC Cc1cc(O)ncc1C(=O)NC1CCCN(C(=O)C(C)(C)c2ccno2)CC1 c1(CCC)cc(C(N2CCCC2C(=O)Nc2cnn(C(F)F)c2)=O)n[nH]1 C1(NC(=O)CC23CCCC2C3)CN(C(c2cncnc2)=O)CC1F C#CCCCCC(=O)N1CCC2C(NC(c3cnc(C)s3)=O)C2C1 Cc1cccc(C(F)(F)C(=O)N(C)Cc2cccnn2)n1 CCCCC(C(=O)N(CCCC)CCO)NC(=O)CCn1ccnn1 C(=O)(CN=S(C)(C)=O)NCC(=O)NCC(C)(C)NC(=O)CCSC(F)(F)F N1(C(c2cc(C)[nH]n2)=O)C(CNC(C2CC3C(C2)C3(F)F)=O)CC2COCC12 C1(C(=O)NC)CCC(F)(F)CC1.C12CC(C(O)C1)NC(=O)CN(CC)CC(=O)N2 c1(-c2cn(CC(N3CCOC(Cn4cncn4)C3)=O)nn2)cc(Cl)c(Cl)cc1Cl c1(C(=O)NC2C(CNC(C(C)Oc3cccnc3)=O)C2)nncc2c1CCCC2 CC1(CNC(=O)CCc2cc(Cl)no2)CCCN(C(C2(C3CCC3)CCC2)=O)C1 C(=O)(C1=CC2C=CC(C1)C2)N1C(CC(=O)NC(CCCCN(CC)CC)=O)CCC1 C1(N=[N+]=[N-])(C(N(C(C#C)C)C)=O)CCN(C(c2cc(C(N)=O)co2)=O)C1 C(=O)(C(C(C)C)NC(=O)C(F)=C(C)C)NCC(CC=C)NC(c1ccccc1)=O C1(C(C)C)CN(C(=O)Cc2cn[nH]c2)CCCN1C(=O)C(O)Cn1cncn1 C1(CC(N2CCCC(CNC(c3oc(C)c(Br)c3)=O)C2)=O)CCC(C)(C)CO1 CC1CN(C(=O)CN(C(=O)OC2CCCO2)Cc2ccccc2)CC(C)S1 Nc1cc(F)cc(C(=O)NCC2CC3CN(C(=O)CC4CCC5CC45)CC23)c1F N1(C(C(C)OCC#C)=O)C2CCC(C(=O)NCc3ccc(C)nc3Cl)C1CC2 c1(C(=O)NC2C(C)CN(C(=O)CC3CCCOC3)CC2)ccc([N+](=O)[O-])c(O)c1 Cc1ccc(CO)c(F)c1.N1(C(CC(O)CO)=O)CC(C(=O)O)(Cc2ccccc2)C1 N1(C(C(C)Cn2cncn2)=O)CCC2(CC1)CC2C(N1CCC(C)(O)CC1)=O C1(NC(c2cncc(NC(C3CCCN(CC)C3)=O)c2)=O)CC2(CCCC2)C1 C1(C(F)F)(CNC(Cc2cc(CC)no2)=O)CCN(C(C2CCCCC2O)=O)C1 CCCC(O)(CCC)CC(=O)NCC(C)(O)CNC(C1OCCOC12CCC2)=O N1(C(CCc2n(C)cnn2)=O)CC2CCC(C1)N2C(c1ccn(C2CC2)n1)=O Cn1cc(C(=O)NCC2CN(C(c3cc(F)cs3)=O)CC2(C)C)c(O)nc1=O CC(CCCCNC(=O)C(C)(C)C1(C)CC1(F)F)NC(c1cnn(C(F)F)c1)=O CN1CC(C)(C)CC1C(=O)NC1(C)CCN(C(=O)CCCCC2CCCCC2)C1 N1(C(CCSCCC)=O)CC(C(=O)NCCCOCCO)CCC1(C)C C(c1c(Cl)cccc1Cl)=CC(=O)NCC1CCCN(C(C(CC#C)C)=O)C1 N1(C(CC2CN(C(C)=O)C2)=O)CC(C)(C)CC1CNC(=O)Cc1cc(F)ccc1O c1(NC(=O)NC2CN(C)NC2=O)cccc2nccnc12 N1(C(C(COC)(C)C)=O)CC2CC(C(=O)Nc3cnn(C(C)C)c3C)(C2)C1 C1(CNC(C(COC)OC)=O)COCCN(C(=O)CCC2CCC(=O)C2)C1 c1(C(N2CC(CNC(c3ccc(OC)o3)=O)C(C)C2)=O)nn(C)c2c1CSCC2 C1(CN(C)C(C2COCCO2)=O)CCCN1C(=O)CN1CCCC1=O C1(CC(=O)NC2CC3CC3C2)CCCN(C(=O)CCn2cccn2)C1 C(C(=O)NC1CC(CO)N(C(c2n[nH]cc2Cl)=O)C1)(C(C)C)OCC(C)C c1(OC)cc(Cl)c(C(=O)NC2CC2NC(=O)OC(C)(C)C)cc1Cl Nc1ccc(C(N2CCN(C(C3CC3C(N)=O)=O)C3CCC23)=O)c(F)c1F CON(CCC(=O)N1CCc2nn[nH]c2C1)C(=O)C(C)COC(C)=O c1(CC)cc(C(=O)NCCCN(C(=O)COCCF)C2CC2)n[nH]1 c1(C(=O)NC(C(C)C)(C)CNC(=O)CC2CCC(=O)N2C)n[nH]c2c1CCC2 C(c1nccs1)=CC(=O)N(C1CCN(C(=O)Cc2cnnn2C)C1)C Cc1c(N(C)CCc2ccc(Cl)cc2)ncnc1N1CCOCC(C)C1 CC1(C)CCCC(c2noc(-c3ncc(-c4cc(Cl)ccc4C(F)(F)F)o3)n2)C1 C(=O)(CS(=O)(=O)CC1CCCO1)NC1C(NC(C2C(C)OC(=O)N2)=O)C1 Cc1ncnc(C(=O)NCC2C(O)C(O)CN2C(=O)C=Cc2ccncn2)c1C c1(CC)ncccc1C(=O)NCCNC(=O)CNC(C#N)CC C=CCC(CC(C)C)C(=O)NCCCNC(C1(CC)CCOCC1)=O c1(C(=O)NC2CC(N(C(C3N(C)CC(C)(C)C3)=O)C)C2)ccnc2c1cnn2C C(=O)(C1=NNC(=O)C1)NCC1C(NC(CC(C)N(C)C)=O)C1 CC(CN(C)C)CCC(=O)N1CCC(C(C)(C)NCc2ncc(CO)[nH]2)C1 C12(CC(=O)NCCn3cc(C(=O)NCCc4ccco4)nn3)COC(C1)C2 Cc1csc(=NCC(=O)N(C)CC2CCCN(C(C3CC3C)=O)C2)[nH]1 C1(C(=O)NCc2ccc([N+](=O)[O-])o2)CN(C(c2ccc(Cl)o2)=O)CCC1O C(=O)(C(CC1OCCO1)Nc1ncc(C(C)(C)C)o1)OC C1(C(C)(C)C)CC(C(=O)N2CCCC(CCNC(=O)C(O)CC3CC3)CC2)=NO1 c1(CC(C(=O)NCC(CC)NC(c2nccc(C(F)F)n2)=O)O)cccc(Cl)c1 CC(C)(CNC(C1CCCCO1)=O)CNC(=O)Cn1ccc(C(F)(F)F)n1 CON(C)C(=O)CNC(=O)CN(CCOC)C(C1CC(=O)C1(C)C)=O c1(C(C)C)nc(=NC2(CNC(=O)CC3CC4CCC3C4)COC2)s[nH]1 C(C(C(=O)N1CC2CCCC2C1)C(C)(C)C)NC(C(COC)(F)F)=O C=CCC(CC=C)C(=O)N1CC(NC(=O)CCN2CCC2)CC1CO c1(N2CC(CCOC)(NC(=O)CC3CC3C)C2)c(F)cc(C(=O)O)cc1[N+](=O)[O-] c1(CNC2(C(=O)OCC)CCCCN2)ccc2c(c1)CCN2CC C1(NC(C2c3cnc(s3)N2C)=O)CCCCC1C.N1(CC(C)N(C)C)CCOCC1 c1(OC)ccc2c(N3CCOC(C(CC)CC)C3)nc(=NC3COCC3)[nH]c2c1 N1(C(C2CC(O)CCN2Cc2cc(O)ccc2F)=O)CCN2CCCCC2C1 C1(c2nc(CCCSCC)nn2C2CCOC2)Cc2ccccc2S1 C1(NC(c2c(N)cc(Cl)cc2)=O)CCSC12CN(C(=O)C(C1(O)CCCC1)F)C2 CC(C)CS(=O)(=O)CCC(=O)N(C)CC1(NC(=O)CC2CCOCC2)CC1 c1(CSC)cc(C(=O)NCC2COC(CNC(=O)Cc3nncn3C)C2)sc1C C1(C(N(C(C(=O)NC(COC)C2(C)CC2)C)C2CC2)=O)CC(F)CN1C C(=O)(C1=NOC(C)C1)N(C)CC1CCCN(C(c2c(CC)sc(=N)[nH]2)=O)C1 Cc1c(C(=O)NC(C)CCNC(=O)CSC(C)C)csc1Br C=C1CCN(C(=O)C(CN(C)C)C(C)C)C(C(=O)NCCc2nccs2)C1 C1(C(N(C(C(=O)NCCCCF)C2CN(CC)C2)C)=O)CCOC(C)(C)C1 C1(C(N(C)Cc2nnc(C)s2)=O)CCC(C)N1C(c1cn(CCO)nn1)=O CCC(C)C(O)C(=O)N1CC(CN(C)C(c2ccnc(SCC(F)(F)F)c2)=O)C1 C(C(O)C(=O)NC(C)CNC(C1CC(O)(C(F)(F)F)C1)=O)=CC c1(C(=O)NCC2(C(N3CC(OC)(CO)C3)=O)CCC2)ccc2n[nH]cc2c1 C(=O)(CCCC(C)C)NC1(CNC(c2cn(CCOC)nc2)=O)CC1 C1(OC)CCCN(NC(=O)C2CC(=O)Cc3ccccc3C2)C1 c1(C(N(CC(CC)NC(=O)C(C)CC(N)=O)CC)=O)cc2nc(C)[nH]c2cc1F CC1CCCCC1C(N1CC(CCNC(c2nccnc2N)=O)C1)=O C(=O)(C(O)CC(F)F)NC(CSC(CN(C)CC)C)=O c1(C(=O)NC2CC(NC(c3c(C)nn(CCO)c3)=O)C2)cc2c(nn1)CCCO2 CCC1=C(C(=O)N2CC(CNC(=O)CC3CC(=O)NC(=O)C3)CC(C)C2)SCCO1 Cc1c(C(N2CCOC(CCNC(=O)C(C)(O)C3CCC3)C2)=O)ccc(Cl)c1Cl Nc1cc(C(=O)NC2CN(C(c3scnc3C(F)(F)F)=O)C2)cc(O)c1 Cc1cc2sc(=O)n(CCN3Cc4cc(Br)ccc4C3)c(=O)c2cc1F C1(O)(C(C)NC(=O)CCNC(=O)CO)CCN(C(=O)C(c2nc(C)cs2)C)C1 C12(NC(c3cnn(CC)n3)=O)CC1CN(C(=O)Cc1ccsc1Cl)C2 c1(C(=O)NC(C2CN(C(CN3CCC(C)CC3)=O)C2)C)cccc2nc(O)oc12 N1(C(C(CC)Cc2ccccc2)=O)CC(NC(c2cnoc2)=O)CC(F)C1 CC1(C#N)CCN(C(c2cnc(C3CC3)nc2)C(=O)NNCC#N)C1.C1(C)CCOC1 C(CCNC(=O)C1CC1)(C(C)(C)C)N(C(C(=O)NC(=O)NC)C)C N1(C(Cc2c(C)cccc2)=O)CCCC(NC(=O)C(c2ccnn2C)C)CC1 c1(NC(CC2CCN(C(C(C)CCl)=O)CC2)=O)cccc2sccc12 C1(NC(c2cccc(F)c2)=O)CC2C1CCN2C(c1cc(-c2ccccn2)no1)=O CCC#CCN=c1[nH]c(=NCC(C)C2CCCC2)[nH]c2c1COC2 n1(CC)cc(Cl)c(C(=O)NC2CCN(C(C3CCC4CC34)=O)CC2)n1 N1(Cc2c(OC)nsc2)CC2CCC1CN2C(=O)CC(C)C(C)C C=CC1(CC(=O)N(C)Cc2cc(C)nn2C)CN(C(C2CCC(OC)CC2)=O)C1 N1(C(=O)NC(C2CCC2)C)CCC(OCCCCc2ncc[nH]2)C1 c1(OC)ccc(OC)c(-n2nnnc2C2(NCC3CC(F)(CF)C3)CC(CF)C2)c1 C1(NC(=O)C#CC2CC2)CCCC12CN(C(=O)CCc1nnc(C3CCCC3)o1)C2 c1(OC)ccc(C(=O)NCCOCCCNC(=O)CN2CCSCC2)c(F)n1 c1(CC)nn(C)cc1CNC(c1cncc(-c2cc(O)n[nH]2)n1)c1ccccc1 c1(OC)cncc(C(=O)NCCCC2CN(C(C3CC3C3CCC3)=O)CCO2)n1 C(=O)(C1CCCc2nc[nH]c21)NC1(CF)CCN(C(c2cncc(N)n2)=O)C1 Cc1cc(=NC2CCc3n[nH]c(C)c3C2)[nH]c(=NC(C)c2cccs2)[nH]1 c1(ONC(c2ccc(Cn3cc(Br)cn3)o2)=O)cc(Cl)cc([N+](=O)[O-])c1O CCCCCCC(=O)NCC(CC(F)(F)F)NC(=O)C(C)ONC(=O)OC(C)(C)C c1(OC(C(=O)NCC(CC)NC(c2coc(Cl)c2)=O)C)ccc(F)cc1Br c1(C(N2CC(CCC=C)(C(=O)NC3CC(=C4CC4)C3)C2)=O)cccc(CO)c1 Cc1cccc(C2(CN3CCC(C(N4CCCC4CCO)=O)C3)CCC2)c1 C1(O)(C(N(C)CCC2CCC2)=O)CCN(C(=O)C(CC=CCl)c2ccccc2)CC1 N#Cc1cc(S(=O)(=O)NC(c2ccc(C(F)(F)F)cc2)=O)ccc1Br C1(CNC(C2CCC(=C)CC2)=O)CCN(C(=O)CCC(=O)NC)CC1O N#CC1CC1C(=O)OC(CCCl)c1cccs1.C1C(=O)O1 C1(C(N2C(CCC(=O)NCCCCOC(C)=O)CCC2)=O)CCN(C)C1=O N1(C(CCC2CC(OC)C2)=O)C2CCCC1CC(NC(=O)Cc1ccn(C)n1)C2 c1(C(N(CC(C)CNC(C2CCC(F)(F)CC2)=O)C)=O)ccnc2ccccc12 C1(NC(CCC=C=C)=O)CS(=O)(=O)CC1NC(c1cc(-c2csc(C)n2)c[nH]1)=O N1(CCF)CCN(N2C3CCC2CC(c2ccsc2)C3)CC1 c1(C(=O)NC(CNC(c2c(C(=O)OC)coc2)=O)(C)C(C)C)ccc(Cl)cc1C Cc1nc2nccc(N3CC(CNC(C4CCc5ccnn5C4)=O)CC3C)n2n1 C(=O)(C1=NNC(=O)C1)N1CC(NC(C(C)Oc2ccccc2Cl)=O)C1 c1(C(=O)NC23C(CN(C(C(C(C)C)(C)O)=O)C2)C3)ccc2nnc(S)n2c1 C1(C(N(CCCNC(Cn2c(C)cnc2)=O)CCO)=O)CCC(=O)N1C CC(C(=O)N1CCCCCC1CNC(c1cc(Br)ccn1)=O)S(C)(=O)=O c1(N(C(CNC(c2c(CC)[nH]cc2)=O)C(=O)NC)CC)cnc2[nH]cnc2c1 S(=O)(=O)(CC(=O)NCC1CCN1C(=O)C(C)OCCN(C)C)NC c1(C(=O)NC2C(C)CN(C(c3ccc(Cl)c(N)c3)=O)C2)ccc2c(c1)CCCCS2 CC1=C(C(=O)NC2CC3CCC2(NC(C2C=CCCC2)=O)C3)CCO1 C1(C(=O)NCCC(C)CC(=O)O)CCCC2(CCNCC2)O1 c1(C(N(C(CNC(CCCOCC=C)=O)C)C)=O)cccnc1SC(F)(F)F N1(C(c2[nH]cc(C#N)c2)=O)CC2(C1)CN(C(=O)C(C1CCOCC1)O)C2 C1(NC(C(C)(C)NC(C=COC)=O)=O)CC2(CCN(C(C3(SCC)CC3)=O)C2)C1 N1(C(=O)NC2CC3C(NC(C4CC4Cl)=O)C3C2)CCc2ccccc21 c1(CNC(C(CCCC)OC)c2nnnn2CC2CC2)cc(Cl)c(Cl)cc1Cl CCC(C)CCC(=O)NC12CCC(CC1NC(c1ccc(-c3ccco3)o1)=O)C2 C1(N(C)CC)CN(C(c2cc(F)ccn2)C(=O)NCCCF)CC1C N1(C(COCCCC)=O)CCCC(N2CCN(C(=O)C(O)c3cnc[nH]3)CC2)C1 C1(C(=O)NCC(CNC(C(n2c(C)ccn2)C)=O)(C)C)CCc2ccccc2O1 C=C1CC(C)(NC(c2coc(CNC(=O)C(C3CCC3)OC)n2)=O)C1 Cc1cccc(NC(c2ccc(CN3CCOCC3)c(F)c2)=O)c1[N+](=O)[O-] C1(CCNC(Cc2nc(C)[nH]n2)=O)COCCN1C(c1cnn(C(C)C)c1Cl)=O C1(C(=O)NCc2n(CC)nnc2C)CCC(C)(C)N(C(C2CCCC(=O)N2)=O)C1 N1(C(c2ccc(C(N)=O)cc2)C(=O)NCC=C)CCC2(C1)NC(=O)N(C)C2=O N1(C(C(CCSC)O)=O)CCC2C(CCN2C(=O)CSc2ccc(C#N)cc2)C1 C1(NC(CCC(=O)NCCC)=O)CCCCN(C(C2(C#N)CC(C)C2)=O)C1 C(C(C)(C)CC(=O)N(CC(O)C1CCC1)C)NC(Cc1cn(CC)nn1)=O O=C(C(O)CC(O)CO)NCCCc1ccco1 N1(C(C2CCCN(C(c3cc(SC)oc3)=O)CC2)=O)CCC(O)C(C)(C)C1 c1(NC)cncc(C(=O)NC2CCN(C(=O)C(C)Cc3c(C)noc3C)C2)c1 C1(NC(=O)C(O)CCC(F)(F)F)CCCC(NC(c2csc(Br)n2)=O)C1 N1(C(c2cccc(C)c2C#N)=O)CCN(C(C2CCCCS2)=O)C2CCCC12 N1(CCNC(C2C(c3ccccc3)(C)C2)=O)CCCN(C(=O)C2=CCOC2)CC1 N1(C(CCOCC)=O)CCC(C(C)(C)C)(CNC(=O)C(C)(O)CC)C1 c1(C(N(C2CCN(C(=O)COCC(F)(F)F)C2)C)=O)cccc2nn(C)nc12 CCC(C)C(CC(=O)Nc1ccc(Cl)c(C)c1)NC(c1cc(Cl)ns1)=O C1(C(N2CC3CCN(C(CCOC)=O)CC32)=O)Cc2ccccc2NC1=O c1(NC(C(C)NC(=O)NC2CC2)=O)cccc(CNC(c2cc(Cl)ccn2)=O)c1 c1(C(N(C2CCN(C(=O)C(C)C3CCC3)C2)CC)=O)cc2ccccc2oc1=O C12(CNC(CCSC)=O)CC(NC(c3ccc(C(C)C)cc3)=O)(CO1)C2 N1(C(CN(C(CC)C)C)=O)CCC(O)(CO)C1.C(=O)(COCC)N(C)C(C)C C#CCCC(C(=O)N(C1CCCC1)C)N(C(=O)C(C)C(=O)OC)C C(=O)(CCCCCCNC(=O)CC1CCCCCC1)NCC(C)(C)C1CCCO1 N1(C(c2[nH]cc(C(=O)OC)c2)=O)CCCC(C)(CNC(c2cnnn2C)=O)C1 C(=O)(C(CCC)NC(=O)NCc1ccc(OC)nc1)NCC=C N1(C(C(C)N(C(=O)CCc2ccncn2)CCC)=O)CC2CC1CS2=O C1(O)(CNC(C(C2CCN(C(Cc3cc(CC)no3)=O)C2)C)=O)CCOCC1 CCC(C)CC(=O)C(=O)N1CC2CC2(NC(=O)C(C)C(C)C)C1 CC(CC(C)NC(c1ncsc1C1CC1)=O)NC(=O)CC(C)F C1(CC(=O)NCC2(O)CCN(C(c3cnc(O)c(Cl)c3)=O)C2)CCS(=O)(=O)CC1 N1(C(c2cn(CC)nc2)=O)CCn2ncc(CNC(C3CC(O)C(F)C3)=O)c2C1 C1(CCNC(c2c(CNC(CCn3ncc(C)c3)=O)occ2)=O)CCCC2CC12 C1(OCC=C)CCN(C(=O)C(=O)N(C)CC2CC2C)C1 c1(CC(C)NC(=O)Cn2cc(C(N3CCOCC3)C3CC3)nn2)nncn1C.C(C)=C N1(Cc2nc(C)sc2)CCOC(CNC(=O)CCc2ccncc2)C1 N1(C(C=C(C)C(C)(C)C)=O)CCC(C2CC2)C1C(=O)N.C(=O)(CCCF)N1CC(O)C1 c1(CC(=O)NCCCCN(C)C(C2CC3CCC3CC2)=O)c(Cl)cccc1Cl c1(OC)cc(C(c2nnnn2C2CCC2)Nc2ccc(O)nc2)ccc1C#N C1(NC(=O)C=CC(F)(F)F)CNC(=O)CN1C(=O)CCC1(N(C)C)CCCC1 C1(NC(c2cn(C)nc2O)=O)CCCCN(C(=O)C=CSCc2ccco2)C1 C1(C)(C(=O)NC2(COC)CC2)CN(C(=O)CC(C)C2CCCO2)C1 CN1CCc2cc(C(N3CCC(NC(c4cnns4)=O)CC(O)C3)=O)sc2C1 N1(C(C2CC(=C)C2)=O)CCOC2(CCCN(C(=O)C(c3cnn(C)c3)C)C2)C1 Cc1nc(C(N2CCC(NC(c3c[nH]c(=N)o3)=O)C(C)C2)=O)c(C)n1C1CC1 C(=O)(C(C)(C)CC(C)(C)C)N1CCC(CC(=O)NCCc2cc(C)ns2)CC1 CC1N(C(=O)COCc2cn(CC3CCCC4(CC4)C3)nn2)CC(C)OC1(C)C c1(CC(=O)NC(C2CCOC2)CNC(c2cnc(SC)s2)=O)cc(F)ccc1C C1(C)(C(=O)NC2C(CCC)C2)CCCN1C(c1cc(CC)no1)=O N1(CCC(=O)N(c2ccc(OC)c(OC)c2)C)CCS(=O)(=O)CC1CC(N)=O C1(C(N2CCN(C(c3cnn4c3OCC4)=O)CC2)=O)(OC)CC2CCC1C2 c1(NC(CC)CNC(c2ccc(OC)c(C(C)C)c2)=O)c(Cl)cccc1[N+](=O)[O-] CCC1c2ccsc2CCN1Cc1c[nH]cc1Br c1(C(N2CCCC(CNC(CC3C=NN(C)C3=O)=O)C2)=O)nccc2[nH]ccc12 N1(C(CSC)=O)CCOC2(CCCN(C(c3cn(CC4CCC4)nn3)=O)C2)C1 C(=O)(N=c1cc(C)n(C)[nH]1)c1c(F)ncc(-c2ccc(OC)c(F)c2OC)c1 C1(C(=O)NCCCn2cc(-c3c(C)ocn3)nn2)CSCC(=O)N1 N#CC1(F)CCN(C(=O)CC2CCCN(C(c3sccc3Cl)=O)C2)C1 c1(C(c2cn(C)nn2)NC(c2c(OC)cncn2)=O)ccc2ocnc2c1 C1(C(CNC(C(N2CCC(OCCOC)C2)=O)=O)(C)C)CCCNC(=O)C1 C1(NC(C(C)OC2CCOC2)=O)CCN(C(C2(CN(C)C)CC2)=O)CC1C Cc1cncc(C(=O)NCCCNC(C2CCN(C)C(=O)C2)=O)c1Cl C1(CN(C(CN(C(CN(C)C)=O)C)=O)C)CCCN1C(=O)COC1CCOC1 Cc1n[nH]c(C)c1S(=O)(=O)NC1CCN(Cc2ccc(Cl)cc2Cl)CC1F C=CCC(F)(F)C(=O)NC1CCCC(n2cc(C(=O)ON(C)C3CC3)nn2)C1 Cc1c[nH]cc(C(N2CCC(F)(CNC(=O)CN(C3CCCC3)C)C2)=O)c1=O C(=O)(CS(=O)(=O)CCOC)NC(CC)CCC(=O)NCC(C)(O)COC c1(C(=O)NCC(C(=O)NCC(C=C)O)C(C)C)cccc2[nH]ccc12 CC#CCC(C)N=c1nc2scnc2c(NCCC2(CO)CC2)[nH]1 N1(C(C=CC)=O)CCN(C(c2ccc(C(C)=O)cc2)=O)C(c2ccncc2)C1 C12(CNC(C=C(C)C3CC3)=O)CCCC1N(C(=O)CC1CCCCO1)CC2 C1(C(=O)NCC(CC)C#N)CCC(C)N1C(=O)CC1C=NN(C)C1=O N1(C(CSC(C)C)=O)CCCC(C2CN(C(=O)CN3CCC(C)C3)C2)C1 C1(CCC)(NC(c2nnsc2C)=O)CCCN(C(c2[nH]c(C3CC3)nc2C)=O)C1 Cc1cc(C(N2CC(CC(C)Nc3cc(C(=O)O)cc(C)n3)C2)=O)nc(C)c1 N1(C(C2N(C)CCC2)=O)CCOCCC1C(N1C2CCC1COC2)=O N1(C(C(CC#C)C)=O)CC2(C1)CN(C(c1c[nH]cc1C(F)(F)F)=O)C2 c1(C(C)=O)cc(C(N2CCC(C)(CNC(=O)Cn3nccn3)CC2)=O)cc(C)c1 CC(C)CC(C)CC(=O)N1CC(CNC(c2cc3cnccc3o2)=O)C(O)C1 CCCCC(=O)NC1CCC(CNC(c2cc(-c3ccco3)on2)=O)C1 CCC(CC)C(C(=O)N1CC(O)(C(C)NC(C2CC(CF)C2)=O)C1)OC C1(C(N2CC(OC)C2)=O)CC(OC)CN1C(=O)C(CO)OC CC1OCCC1(F)C(=O)NCCC1(NC(=O)CC2(C)CCCC2)CC1 C1(CC(=O)N(CCNC(C2(C3CC3)CC2)=O)CC2CCCC2)CC2CCC1O2 N1(C(C2C(OCC)C2C)=O)CCC2(COC(CNC(C3CCCOC3C)=O)C2)C1 N1(C(CC[SH](CC)C2CC2)=O)CCN(C(C2(n3cncn3)CC2)=O)C2CCCC2(C)C1 c12cccc3c1CN(C3)C2.c1(CCCC)cnc(NC)s1 N1(C(=O)CN2CCN(CC(F)(F)F)C2=O)CCN(C(C2CCCC2)=O)C2CC12 N1(C(c2cc(C(=O)OCC)no2)=O)CCN(C(=O)CCc2cncs2)CC1C C1(OC)CC(C(=O)Nc2c[nH]nc2C#N)N(C(=O)CCC(C)OC)C1 c1(OC)ccc(CN=C(NCc2ccc[nH]2)NCC2CCCCC2)cc1F C(=O)(C(C)C(O)C(C)C)N1CCCC(CC)C1C(=O)NC1CCN(CC2CC2)C1 C(CCC(=O)N1CCC1C(=O)NCC(=O)NCCOC)OCC C1(NC(C(C)OCOC)=O)CN(C(=O)CSc2cccc(C)c2)C(C)(C)C1 C(=O)(C(C)(C)c1ccccn1)NCC(CNC(C1(CC#C)CCC1)=O)OC c1(OC)ncc(Cl)cc1NC(=O)CNC(c1ncnc(O)c1F)=O C1(C(N2CCC(F)(c3cn(CCCCF)nn3)C2)=O)CCc2ccccc2O1 C1(CC(=O)NC2(C)CCN(C(=O)CCNC(=O)CO)C2)CCc2ccccc2C1 c1(C(N2CC3(CC(NC(c4c(OC)cccc4I)=O)C3)C2)=O)ccc(C#N)cc1F CC1(C)CN(C(=O)CCSc2ccc(Cl)c(Cl)c2)CC1NC(=O)COC(F)F Cc1ccc(Cl)c(N)c1C(=O)NC1CCCC1CNC(C1CC(n2cccn2)C1)=O c1(C(=O)NCC2N(C(CC(C)c3ccncc3)=O)CC=C2)ncccc1O C(=O)(C1=C(Cl)CCCC1)NC1C(NC(c2ncc(C)c(C)c2)=O)CCC1 C1(NC(C(CC)(C)CC)=O)CCN(C(C2(OC)CCC2)=O)CCC1CO C1(CNC(C2(OC)CC2)=O)CN(C(=O)C(c2cccc(Cl)c2)(F)F)CC1C N1(C(=O)OC)CC(Oc2csc(-c3cccc(F)c3F)n2)CCC12CC2 N1(C(C2N(Cc3ccc(CC)cc3)CCC2)=O)CCCC2(CCN2CC)C1 N1(C(CC2(C=C)CCC2)=O)CCCN(C(=O)C(C)C2CCCO2)CC1CO N1(C(CCCCC)=O)CCC2(COC(CNC(c3snc4ccccc34)=O)C2)C1 N1(C(c2cc(C)oc2C)=O)CC(C2=NOCC2)C1.N12CCCC1(C)c1cn(nn1)CC2=O Cc1ccn(C)c1C(=O)NCCCN(C(=O)C(N1CCCC(O)C1)C)CCO C1(CC(=O)NCCC2N(C(CCC(=O)N(C)C)=O)CCOC2)CCCC(C)(C)O1 c1(NC(c2c(Cl)cncc2Cl)c2n(C(CC)C)nnn2)cc(C(=O)OC)cc(F)c1 Cn1cc(C(N2CC(NC(=O)CCCC#N)CC23CCOC3)=O)c2cccnc12 c1(C(N(CC#C)C)=O)coc(CNC(=O)C(C)C#N)n1 N1(C(=O)OC(C)(C)C)CCCC1C#CC(=O)N1Cc2cccc(C(F)(F)F)c2C1 N1(C(CC2(OC)CC2)=O)CC(C(=O)NCCCN2CC=CC2)C(C)C1 c1(C(=O)NC2CC(CC(=O)NC3CC(C)SCC3)C2)cnn2cccc2c1 c1(C(=O)NCC2(NC(C3CC(C(C)(C)C)C3)=O)CCCC2)cncc(Br)c1 CC1CN(C(=O)CC2CCCO2)CCC1C(N1CCC(F)(CF)C1)=O C1(NC(=O)CCn2cncn2)CN(C(C2CC(n3cnnc3)C2)=O)C2(CCOC2)C1 CC(CCCN=c1[nH]c(=NCc2csnc2Br)[nH]c2ccsc12)c1ccccc1 [N-]=[N+]=NC1CN(C(c2ccnnc2)=O)CC1NC(c1cccc2c1NCC2)=O C1(C(=O)Nc2c(C)ccc(C#C)c2)CCCN1NC(=O)C=CC=CC=C C1(=O)C(C2(C(C(F)=CCC)=O)CC(COC)C2)CN1 C(=O)(C1CCC(=O)c2cccn21)NCCC1CCCN(C(CCCC#N)=O)C1 Cc1ccc(C(=O)NCCC(C)NC(C2CCN(C)S2(=O)=O)=O)c2c1CCC2 C1(C(N(C2CCCN(C(c3nnc(S)n3C)=O)C2)CC)=O)CCC=CCCC1 C1(NC(c2cn(COC)nc2C)=O)CN(C(=O)Cc2cc[nH]n2)C2(CCOC2)C1 c1(C(=O)NC2CN(C(C(C)c3ccco3)=O)C(C)(C)C2)cccc2c1CCC2 Cn1nc(C(N2CC3C(NC(c4cccnc4O)=O)C3C2)=O)c2c1CCSC2 c1(CCC(=O)N(C2CCN(C(c3coc(C(F)F)n3)=O)C2)C)ncc(F)cn1 C1(NC(C2C3(CC(C)(C)C3)C2)=O)CN(C(=O)CCn2cnnn2)CC2(CC2)C1 N1(C(c2nccc(C)n2)=O)CCN(C(c2occ(C)c2C)=O)CC2(CC2)C1 N1(C(c2c(CC)cncc2)=O)CC2CC(C)N(C(=O)C(C)NC=O)C2C1 n1(CC)cnnc1CC(=O)NCC(C)(C1CCC1)NC(=O)CNc1ccccn1 N1(C(CSC)=O)CC(O)(C(C)NC(C2CCCN2c2ncccn2)=O)C1 c1(OC)cc(OC)c(C(=O)NC(C2(O)CN(c3nccc(C)n3)C2)C)c(CO)c1 C1(NC(c2cnc(CC)s2)=O)CN(C(=O)C(N2CCCC(C)C2)=O)CC1C c1(CC(C(N2C(C)CC2CO)=O)C)ccc(O)cc1 C(=O)(C1CCCc2nc[nH]c21)N1C(CN(C(C(=O)NC(C)C)=O)C2CC2)CCC1 CCC(C)(CC)C(=O)NCC1(O)CSC1.C1=CCNC(=O)C1 C12(C(=O)Nc3c(C)nc(F)cc3)COCC1CN(C(c1cc(CO)ccn1)=O)C2 C1(C(C)NC(=O)NC(CNC)(C)COC(C)(C)C)CCCCCC1 CCC(CC(F)F)C(=O)N(C1CCN(C(=O)CC2CCS(=O)(=O)CC2)C1)C c1(C(=O)NC(CC(C)NC(=O)C(O)Cc2cnc[nH]2)C)cc(F)cc2nn[nH]c12 c1(NCC(N2CC(=O)N(C)C2=O)N2CCCC2)cc(O)nc(=O)n1C S(=O)(=O)(c1ccc(NCC(C)Oc2ccccc2)c(C#N)c1)N(C(C=C)C)C c1(NCCN(C(c2ccc3c(c2)COC3=O)=O)CC)cccc2c(C)ccnc12 CCC(C(=O)NNC(=O)NC(c1ccc2ccccc2c1)C)n1cccn1 C1(CC(N2CC(C)N(C(=O)CCCF)CC2)=O)Oc2ccccc2NC1=O CCC1=C(C(=O)N2CC(CNC(C3(F)CCOCC3)=O)CC2(C)C)CCCO1 Cc1cccc(C(F)(F)C(N2CCC(CCNC(C3CCOC3C)=O)CC2)=O)n1 CC1(C)CCC1CCCNC(=O)C(C)(O)C1CCOCC1 C(=O)(C1=NNC(=O)C1)N(CCNC(CCc1nc(C)c(C)o1)=O)C(C)C Cc1nc(C(=O)NCCCCCCNC(c2ccccc2)=O)cn1C C12(NC(C3CCC3)=O)CCC1CN(C(c1ccc(Cl)s1)=O)C2 c1(C(N(CC(O)CN(C)C(C2CC23CCC3)=O)C)=O)cc2c(o1)CCCC2 C12(CNC(C(C)SC)=O)CCC(CC1NC(c1ccc(Br)cn1)=O)C2 CC1CCC(C(N2CC3CCCC2C3)=O)CN1C(C1CC2(CC2)C1)=O C(=O)(CCC(=O)C(C)(C)C)N1C(C(N2CC(COC)C2)=O)CC1C C1(N2CCC2=O)CCC(=O)NC1=O.CC(CCC(=O)N(C)CCO)N(C)C c1(C(N(c2cccc(C)c2)SCCC)=O)cccc(-c2ccc(C(C)=O)cc2)c1 C(=O)(C(F)(F)CCn1ccnn1)NC(C1CCN(C(C=NOC)=O)CC1)C c1(C(N2CC(N(C(=O)C(c3cnn(C)c3)O)C)C2)=O)nnc(O)cc1O c1(NC(=O)Nc2ccc(Cl)cc2C(F)F)c[nH]c2cccc(Br)c12 CC1CC(NC(=O)CCc2cncnc2O)CN1C(=O)COCCCF N1(C(C(C)CCC(C)(C)C)=O)CCOC2CCN(C(=O)CSC(F)(F)F)CC12 C(=O)(C#CC1CCOCC1)N(C)CCNC(C1(C#N)CC=CC1)=O c1(OC)ccc(Cn2c(C)cc(NC(c3cccc(SC)c3)=O)c2C)c(F)c1Br C=CCN=c1[nH]cc(C(N2CC(NC(=O)COC3CCCOC3)CC23CCC3)=O)s1 CCCCCC(O)CC(=O)NCC(C)(CO)NC(=O)Cn1cccc(C)c1=O c1(-c2cn(CCCCNC(C3(C)CS(=O)(=O)C3)=O)nn2)ccc(Cl)c(F)c1 C1(C)(NC(C2(NC(C)=O)CCCC2)=O)CCN(C(C2(C#N)CCCC2)=O)C1 N1(C(CCSC)=O)CCCC(CNC(c2cn(C)nc2-c2cc(C)no2)=O)CC1 n1(CCC)cc(C(=O)NCC(C)(C)CCNC(=O)C2=C(Cl)CC2)c(C)n1 C(=O)(CC(C(C)OC)NC(c1ccc(OC)s1)=O)N1CC(COC)OCC1 CCCCC(C)C(=O)NCC1CCCN(C(c2cc(C(=O)OC)sc2C)=O)CC1 c1(C(=O)NC(CNC(c2oc(C)c(CO)c2)=O)CO)ccc(C)c2cccnc12 c1(CSCC#C)cccc(C(=O)NCC2CC(O)CN2C(=O)C2=CCCC2)c1 Cc1ccsc1C(=O)NCC1(C(C)NC(=O)CC2(O)CCC2)CC1 C(=O)(CC1=CCCC1)N1C(C2(NC(C3CC4CCC3C4)=O)CC2)CCC1 C12(C(=O)NC3CCN(C(C(CC)N(C)C)=O)CC3F)CCC(CC1)C(C)O2 C(C1c2ccccc2CCN1C(C1CC(=O)CO1)=O)NC(c1c(CC)nns1)=O n1(CC)nccc1C=CC(=O)NC1CC1NC(c1ccc(CN(C)C)nc1)=O C1(CC)(CC)CC(NC(=O)C(O)C2CCC2)CN1C(=O)CCc1cnn(C)c1 c1(C(=O)NCC(=O)NCCNC(C2CC2(Cl)Cl)=O)ccc2cc[nH]c2n1 C1(NC(C(C)=C2CCC2)=O)CCN(C(c2coc(-c3ccsc3)c2)=O)CC1F c1(OC(F)F)cccc(CSCCCNC(C(N2CC(CC)C2)=O)=O)c1 c1(C(N(C2CCCC(NC(CCCOC)=O)C2)C)=O)ccn2ccsc12 N1(C(c2cccc(C(F)(F)F)n2)=O)CCC2CCN(C(C3CCC3)=O)C2C1 c1(C(C(=O)NCCCC)N(C2CCCC2O)C(C)C)cccc(S(N)(=O)=O)c1 c1(C(C2CCC2)NC(c2nnnn2CCCF)C)cc(C(F)(F)F)cc([N+](=O)[O-])c1 C1(N(C(c2c(Cl)cn(CCC)n2)=O)C)CCN(C(c2cc(Cl)n(C)n2)=O)CC1C Cc1ccc(OCCCNC(=O)C(C)n2cccn2)cc1C C1(C(=O)NC2C(C)CN(C(=O)C(O)Cn3cncn3)C2)CCCC(=O)N1C C1(NC(C(C)(F)c2ccon2)=O)C2CC3C1C3C2C(=O)NCC1CC2CCC1O2 C#CCCCC(C(=O)NCC1CCOC1)N1CCC(C(O)C#C)CC1 C1(CNC(C(CC=C)NC(=O)OC(C)(C)C)=O)CC2(C1)CN(C(=O)CC(C)CC)C2 c1(-n2cc(CN3CCN(C(C(CO)N(C)C)=O)CC3)nn2)cc(F)ccc1F N1(CCCc2cccc(-c3c(Cl)cn(C)n3)c2)CC(C)(C)OCC1COCCCO C12(CC(=O)NC3(C)CN(C(C4CCCCC(=O)N4)=O)C3)CCCN1CCC2 c1(CCCC(=O)N(CC(C)NC(=O)C(=O)NC2CC2)C)ccc(F)cc1F C1(NC(C(=Cc2ccccn2)C)=O)CCCCN(C(=O)C(N2CCOCC2)C)C1 c1(C(=O)NCC2CN(C(c3onc(C)c3C)=O)C(C)C2)ccc2ncncc2c1 CCC(CC(=O)N1CCCCC1CC(N1CC(CF)(CO)C1)=O)C(C)C N(C(=NCCCCC#N)NCC(=O)NC(C)C)Cc1ccc(SC)cc1 c1(CC)cc(C(F)(F)F)ccc1C(N1CC(NC(=O)C(O)C2CCC2)C(C)C1)=O C=C(C)CCCC(=O)NCCC1CCC(NC(C2CCC(C)O2)=O)C1 O=C(C1=CCCCCC1)NC1C(CNC(C23C=CC(CC2)C3)=O)CCC1 CC(F)CN=c1[nH]c(N2CCCC3(CCCCC3)C2)nc2c1CSC2 c1(C(N2CCCC(O)C2)=O)nccc(F)c1Cl.C1(N(C(C)C)C)CN(C=O)C1 C1(C(=O)OC)CC12CCCN(C(c1ccc(CCCC#N)cc1)=O)C2 CC(C(=O)NCC(CNC(c1ccnc(-c2ccccc2)c1)=O)CO)C(C)(F)F Cc1ccc2[nH]c(C)c(CN3CCC(C)C(OC(=O)C(C)C)C3=O)c2c1 c1(C(=O)NCCN(CCOCC)C(C2CC2C(=O)OC)=O)cccn1C C1(CC2(C(N(CC(C)NC(=O)CCn3cncn3)C)=O)CCC2)CCCCO1 C(=O)(CC(C)CC(=O)N1CCC(NC(c2coc(Cn3cccn3)c2)=O)C12CC2)OC c1(NC2CC(O)(CNC(CCn3ncc(C)c3)=O)C2)ncc([N+](=O)[O-])c(C)n1 C1(CNC(c2n(C)ncc2C2CCC2)=O)CCN(C(c2cc[nH]n2)=O)C12CCC2 c1(CC)ccnc(C)c1.c1(C(N2CCN2C)=O)cc(-c2cnccn2)[nH]n1 c1(CC)[nH]c(C(=O)NC2CC(F)(CNC(c3cnc(C(C)OC)s3)=O)C2)nc1Cl c1(OC(CC(C)C)c2cn(C3CCCC3)nn2)ccc(C)cc1.C(=O)C(C)CO c1(C(=O)NCCN2CCN(C(CCCCC=C)=O)CC2)cccc2ncc(Br)cc12 N1(C(c2c(CCC)nco2)=O)CCC(C)C1CNC(=O)CCc1ccc(F)cc1 C1(OC)CC2CC(NC(=O)CCN(C(c3cc(C)cc(C)n3)=O)C3CC3)CC12 S(=O)(=O)(c1cc2ccccc2s1)N1CC(NC(c2cccc(Br)n2)=O)C(F)C1 C(=O)(C1=NOC2(CCN(Cc3ncccc3F)C2)C1)Nc1c(OC)cc(F)cc1 C1(C(=O)NCC(CC(C)C)NC(CCn2c(C)ncc2)=O)CCOC(=O)CC1 C(c1c[nH]c(=N)c(C)c1)=CC(N1C2C(NC(CCCC)=O)CC(C2)C1)=O N1(N2CCC3(CC3)C2)CC(CO)C(C2CC2)C1.CC(C)(C)OC=O c1(C(N(CCOC)CCNC(C23CC(C)C2C3)=O)=O)cnc2[nH]cncc1-2 c1(NC(=O)OC(C)(C)C)ccc(C(=O)NCC#CCC2CCCC2)nc1N Cc1cc(Br)c(C(=O)NC2CC(C)CN(C(=O)CC3CC3)C2)cc1F c1(C(=O)NC2CC(C)(COC)N(C(=O)C(C)=C3CC3)C2)cc(C)[nH]c(=NC)n1 C1(CN(C)Cc2nn(C)cc2-c2cccc(C(=O)O)c2)C=CCCCC1 CCC(C)(C)C(C)NC(c1nc(C)sc1C)c1nnnn1C(C)(C)C c1(C(=O)NC(CNC(C)=O)CC)cn(C(C)C)nn1 c1(NC(N2CC(OC)C2)=O)ncc(NC(c2ccco2)C2CC2)c(=N)[nH]1 CS(=O)(=O)c1ccccc1-c1cn(Cc2ccc(C3(N)CC3)cc2)nn1 C1(C(=O)NC(COC2CCN(C(c3cnc(C)nc3)=O)C2)=O)CC(C)CC(C)C1 N1(C(N(C)Cc2nc(CCC)on2)=O)CCC2(CCC2O)CC1 c1(C(=O)NCC2(CNC(C3(C)CC3)=O)CCC2)ccc2c(c1)NCCC2=O C1(C(N)=O)CCC(C(=O)NCC2CCCN2C(C2C=CCCC2)=O)C1 c1(C(=O)OC)cccc(Cl)c1C(=O)NC1CC(F)(CN(C)C(C2(OC)CC2)=O)C1 CN1CCCC(CC(=O)NCC2CCC(NC(=O)CN3CCCC3=O)CC2)C1 C1(C(=O)NCC2CCC(CNC(=O)C3=CCCC3)CC2)CCc2nccn2C1 N1(C(C(=O)N(C)C)=O)C2CCC1CC(F)(CNC(C1CCn3nnnc3C1)=O)C2 N1(C(CCOCC#C)=O)CCCC2CN(C(c3c(C)nc(Cl)nc3Cl)=O)CC12 N1(C(C2C(C)CC2)=O)CC2CC(NC(c3nc(C(F)(F)F)cn3C)=O)C1C2 N1(CC(CC)CC)CCC(c2nnnn2C)(NC2CC2c2cccc(F)c2)C1 CC(CC(=O)NCC1CCCC1NC(c1ccc(CN(C)C)s1)=O)n1cccc1 CCC(C)C(O)CC(=O)N1CCC(C)CC1C(=O)NCCC(C)(C)C1CC1 c1(-c2nn[nH]n2)c(N)cc(C(=O)NCCCCCCOC)cc1F C12(NC(C#CC(C)(C)C)=O)CN(C(c3cnn[nH]3)=O)CC1CS(=O)(=O)C2 N1(C(c2ccc(NC)cc2)=O)CCC2(CC1)CCN(C(c1cnc(SC)s1)=O)C2 C(c1ccccc1)=CC(=O)NCCN(CC(C)O)C(c1cc(Cl)c[nH]1)=O C(CC(C(=O)N(CC(Cl)Cl)C)NC(=O)CSC(F)(F)F)SC C1(CNC(=O)CCF)CC2CCC1N2C(=O)C(F)=C1CCCC1 C1(CC)(NC(c2cccc(C)c2Cl)=O)CCN(C(c2cc(N)nc(Cl)c2)=O)CC1 c1(CN(C(=O)C(O)CNC(C2(CN(C)C)CC2)=O)C)ncc(Cl)cn1 CCC(C(=O)NCCNC(c1cc(CO)[nH]n1)=O)N(C1CCC1)CC.OC C(=O)(C1CCc2c[nH]nc21)NC1CCC(N(C(=O)CCC2CC2(Cl)Cl)C)CC1 c1(CC)ccc(SC2(CN3CCCC(C4(C)OCCO4)C3)CC2)cc1 c1(C(=O)NCC(C)N(C(=O)C(C)O)C)cc(C2CC2)ccn1 c1(C(=O)NCC2CC(O)CN2C(=O)C=CBr)cccnc1Cl CC(C)(CC(F)F)NC(C1C=CCCN1C(=O)CCn1ccnc1)=O C(=O)(CC(CCCC)NC(=O)CCCC1CCCC1)NCC1C(CCC)C1 CC1(C)CNCC(C(=O)NC(C(F)(F)F)C2CCOC2)O1 CCCCC(CNC(=O)C(C1(O)CCC1)NC(=O)CC1OCCCO1)CC C1(NC(CC2CCCN(C)C2)=O)CN(C(=O)CC2CC3(CC3)C2)CC2(CCC2)C1 CCCC(C)(CC)C(=O)N1CCN(C(c2cn(CC)nn2)=O)C(CO)C1 N1(C(C2(C)CC=C(C)CC2)=O)CC=C(CCNC(c2csc3cncn23)=O)CC1 C1(NC(F)F)CN(C(=O)CCOC2CCCC2)CC1O.C(C)(C)(C(=O)N)NC(CC)=O C1(CNC(C2CC23CC3)=O)CN(C(=O)Cc2ccc(Cl)s2)CC12CC2 Cc1oc(-c2ccccc2)cc1CCc1nc(CO)nn1CCF N1(C(c2ccc(CC)nc2)=O)CC2CC(NC(C3(C(N)=O)CC3)=O)C2C1 Cc1nn(C)c(=O)c(C(=O)NC2CN(C(=O)CN3C(=O)CNC3=O)CC2C)c1C N1(C(C(CNC(=O)CC2CCC2)N(C)C)=O)CC2(C1)CC2(F)F C1(OC)CS(=O)(=O)C2CN(CC(C3CC(O)C3)=O)CC12 C(=O)(CCCC(=O)O)NC1CCC(n2cc(CCCOC)nn2)CC1 C1(CNC(C(CC)C)=O)C(C2CC2)CCN1C(c1ccc(CC(C)C)cc1)=O c1(CCC(=O)N(C)CC2C3CN(C(c4cncs4)=O)CC23)ccc2ccsc2c1 C1(NC=O)CC2(C1)CC(CNC(=O)C(=O)N(C)C)C2.Cc1sc(CC(C)N)nc1O N1(C(c2nc(N(C)C)oc2)=O)CCCC(C2CN(C(C3(F)CCC3)=O)C2)C1 N1(C(C23N(C(CCC=C(C)C)=O)CCC2C3)=O)CCN2C(=O)OCC2C1 C(CCCCC(=O)NCC1CCN(C(=O)CCCOC(C)=O)C(C)C1)OCC c1(C(=O)NC2CCC(CCNC(C3(OC)CC3)=O)C2)ncc2ccccc2c1O N1(C(C(CCN(C)C)NC(C(CCCC)O)=O)=O)C(CO)CCC12CCC2 CC1CN(C(C2CC23CCN(c2nccc(-c4cccnc4)n2)C3)=O)CCC1=O C1(C(=O)NC(C)(C)C=C)CC=CC(n2cc(C3(O)CC3)nn2)C1 C1(NC(c2c(C)scc2)=O)COC2(CCCN(C(c3cnnc(O)c3)=O)C2)C1 c1(OC)cc(CN2CC(C)(CNC(C3CC4C=CC3C4)=O)C2)c(Br)cc1O N1(C(=O)Nc2nnn(C)n2)CC2CN(N3C(NC(=O)OCC)CCC3)CC2C1 Cc1ccn2cc(C(=O)NC3(CNC(C4CC45CCCC5)=O)CCCC3)nc2c1 c1(C(=O)NC(COCC)CO)cc(CNC(c2[nH]ccc2CC)=O)no1 CC1=NOC(C)(C(=O)NCCN(C)C(C2CCC(F)(F)C2)=O)C1 C12(NC3CCN(C(=O)NCCOC(C)=O)CC3)CCCCC1C2(F)F c1(C(=O)NC(CC)CN(C)C(C2COCCO2)=O)cc2sc(Cl)cc2[nH]1 C1(NC(C2(OC)CCSC2)=O)CN(C(=O)C2=CCCO2)CC2(CCC2)C1 C1(COC)CN(S(=O)(=O)Cc2ccc(F)c(Cl)c2)CCC1CO CCC(CC)C(C)C(=O)NC1CCCC1CNC(=O)C=CC(=O)OC(C)(C)C c1(C(=O)NC2(C)CCCN(C(CN(C)C(N)=O)=O)C2)ccc(F)c(O)c1F CC#CCC(CO)NC(=O)C=CC1CCCN1C(=O)CC1(COC)CC1 CC(C)C(C(=O)OC(C)(C)C)C(=O)N1CC=CC(NC(C2C(C)(C)C2(C)C)=O)C1 C1(NC(Cc2ccc(NC(C(C)n3ccnn3)=O)cc2)=O)CCCC(C)C1 O=C(CCCC1CC1)NC1(CCNC(=O)CNC(C2CCCCC2)=O)CC1 Cc1n[nH]c(C)c1CC(C)C(=O)N(CC(O)CN(C(=O)Cc1cn[nH]c1)C)C c1(C(=O)NCCOC2CN(C(=O)CSC(F)(F)F)C2)ccc(O)c2ncccc12 C12(CC)CN(C(C3CCC(F)(F)CC3)=O)C(CNC(C3(N(C)C)CCCC3)=O)(C1)C2 c1(NC(C(CC2CC2)NC(N)=O)=O)ccc([N+](=O)[O-])nc1 Cc1c(C(=O)NC(c2cccnc2)C2CCCCC2)cnc(O)c1Br CC1=C(C(=O)NCCC2CCCCN2C(c2scc(C)c2Cl)=O)CCC1 c1(C(N2C(C)C(NC(C3CCC3)=O)CC2)=O)ccccc1S(C)=O.C(C(C)(C)C)C1(C)CC1 C1(C(N2CC(CNC(CN3C(C)CCC3)=O)OCCC2)=O)CCn2c(O)nnc2C1 C1(NC(c2ccc(OC)nc2)=O)COCCN(C(=O)CN2CCCS2(=O)=O)C1 C1(C(=O)NC2CCCC2)CC2CC(C1)N(C(=O)COC(=O)CCCC(F)F)C2 Cc1ccc(CCN(C(=O)Cc2cccs2)C(C)C)nc1 S(=O)(=O)(c1ccccc1Cl)NC(C(C)O)C(=O)N(CC(N1CCCC1)=O)C c1(C(N2CCCC(C)(NC(=O)CC3CCCC(=O)N3)C2)=O)ccc2occc2n1 CC1CCC(CCNC(=O)NC2(C)CS(=O)C2)O1 C(=O)(CCCCN(C)C(C)C)NC(c1ccccc1)C(C)NC(c1cnc(C)o1)=O N1(C(C2(OC)CCSC2)=O)CC2COCC(C1)C2NC(c1cn[nH]c1)=O CC(C)(C(=O)NCCN(C(C1C=CCC1)=O)C1CC1)C1CCOC1 Cc1c(C(=O)NCCCCNC(=O)C(C)CC2CC2)cnn1-c1nccs1 N1(C(CC2(C=C)CCOCC2)=O)CC2CCC(NC(C3CC(C)(N(C)C)C3)=O)(C2)C1 C(=O)(C1=CC2CCCCCC12)NC1CC2(CCN(C(C(COC)(C)C)=O)C2)C1 C1(NC(C2C(OCC)C2)=O)CCC(NC(c2cnccc2C(C)(C)C)=O)CC1 C(=O)(C1=NOC2(CCC2)C1)N1C(CNC(CC(C=C)C)=O)C(C)CC1 N1(C(c2c(C)snn2)=O)CC2CC2C1CNC(=O)CC1CCCCC1 C1(CN2C(C)CCCCCCC2)CCc2cnn(C)c2C1 C12(NC(C(C)Sc3scc(C)n3)=O)CCCC1CN(C(=O)C1=NNC(=O)CC1)C2 C1(C)(C)CCCNC(=O)C2C(C2)C(=O)N1.c1(CCC)ccccc1NC(=O)CC CC1(C)CC(NC(c2ccoc2C(F)(F)F)=O)CN(C(C2(CF)COC2)=O)C1 C1(CN(C)C(C2(CO)CN(C(c3ccsc3)=O)C2)=O)CCCCO1 C1(NC(CC2(C)CC2)=O)CCC2(CCN(C(=O)COCC3(F)CC3)C2)C1 N1(C(c2occ(C)c2C)=O)CC(NC(=O)C(c2cc(F)cc(F)c2)C)C(C)(C)C1 N1(C(C(=O)N(C)C)=O)CC(NC(c2cccc(C(C)(C)C)c2N)=O)C2(CC2)C1 C1(CNC(C2CCC=CCCC2)=O)CCCN(C(=O)Cc2cccc(F)c2)CC1 C1(C(C)NC(C(N2CCC(n3cc(COC)nn3)C2)=O)=O)CC2(CCC2)C1 c1(N2CCCC(C=C)C2)nc(=NCc2cc(C)ccn2)[nH]c2c1CCC2 C1(NC(C(C(C)C)NS(C)(=O)=O)=O)CCCCN(C(=O)C2=NOC(C(C)(C)C)C2)C1 N1(CC(=O)NCC2(CNC(c3ccn(C)c3)=O)CC2)CCCC(C(N)=O)C1 c1(CC(N2CCCCC(NC(C(C)C(C)(C)C)=O)C2)=O)cccc2cnccc12 Cc1cc(=NC(C)c2c(Br)cnn2C)[nH]c(=NC(C)CF)[nH]1 c1(C(=O)NC(C2CCOC2)CNC(CNC(N)=O)=O)ccc(O)c(OC(F)F)c1 c1(OC)ccc(C)c(C(=O)NC2CCN(CCC(C)C)C2)c1.C1(=O)CCC(C)O1 N1(Cc2ccc(CS(C)=O)cc2)CCC2(COC(CNC(=O)CNC=O)C2)C1 N1(C(CCOCCOC)=O)CCCC(N(C(=O)C=Cc2nc(C)co2)C)CC1 CCCCC(CC(=O)N(C)Cc1ccccc1C)NC(=O)CC1CC2(CC2)CO1 N1(C(=O)CSC(F)(F)F)CCC2C1CCN2C(c1ccnc2ccnn12)=O c1(C(N(CCOCCCNC(C2(C)CC(=C)C2)=O)C)=O)ccnc(C(C)C)n1 C1(NC(C2C(C=C)OCC2)=O)CCC12CN(C(c1ccn(C3CC3)n1)=O)C2 C1(C(=O)NCCCCCCNC(c2cncnc2)=O)CCc2nnc(O)n2C1 C1(C(=O)NC(C2(O)CN(C(c3cn(CC=C)nn3)=O)C2)C)CC2CCCC12 C1(C2(C)N=N2)CCN(C(C23CC(NC(=O)C(C)(F)F)(C2)C3)=O)C1 N1(C(c2nc(C(=O)OC)sc2)=O)CC2(C1)SCCC2NC(c1[nH]cnc1C)=O N#CC1CCCCC1NC(C1C2CC1N(C(c1cccc(F)c1F)=O)C2)=O C1(NC(=O)CC2(N(C)C)CC2)CC(C(N(CCC)CCN(C)C)=O)C1 CC(C)C(O)C(C)(C)C(=O)NC1CCCCCCC1NC(=O)CC1CCCCO1 N1(C(C(C=C)CC)=O)CCCC(OCCNC(=O)C(c2ccccc2)F)CC1 c1(CC(=O)NC2(CCNC(c3cc(OC)ns3)=O)CCCC2)ccc(C)cc1Cl Cc1nn(C)c(C)c1C(=O)NCC1CCCN(C(=O)CN(c2cnccn2)C)C1 C1(CC)C(C(=O)NC(C)(CNC(=O)CCC2CC2)C(C)C)CCN1C C1(CNC(Cc2cc(C)cc(C)c2)=O)CCN(C(=O)CC(F)F)CC1(F)F c1(C(=O)NCC2CC(CNC(c3cn(CC=C)nn3)=O)C2)cc(C)nnc1O C(=O)(CC1CCCc2ccccc21)N1C2C(CNC(CCOCC)=O)C(C2)C1 CN1CCN(C(C2CC=CC(O)C2)=O)CC1C(N1CCC2C(O)CC12)=O C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C=CC(N1CCC(CCCC)C1)=O)(C)C c1(C(=O)NCCC2(CNC(CN3C(C)CC(C)C3)=O)CC2)ccccc1S(C)=O c1(OC(C(=O)NCC(CNC(C(C)C(F)F)=O)O)(F)F)ccc(Cl)c(F)c1 C12(C(=O)NC(CC)CC(=O)N3CC(CCO)C(C)C3)CC(C)(CCO1)C2 C1(CC)CCN(C(=O)C(C)=C2CCC2)C1C(=O)NCc1nn(C)c(=O)o1 CC(C(=O)CN1CCCC1c1cn[nH]c1)c1ccccc1 C=CCC(CNC(c1cncnc1)=O)C(=O)NC1(CO)CC(C)(C)C1 C#CCC(C)(C(=O)NC(CC(N)=O)C(=O)OC)NC(C1CCOC1C(C)C)=O C1(NC(C2CC=C(C)CC2)=O)CCCC2CN(C(=O)C(C)C3(O)CCC3)CC12 c1(N2CCC(n3cc(N(C(CC(=O)NC)C)C)nn3)C2)nc(Cl)nc2c(C)n[nH]c12 N1(C(CC(=C)Br)=O)CCC2(CC1)COCC(CNC(=O)CN1CC=CC1)O2 Nc1ccc(C(=O)NCCCCC2CCN(C(C3CC34CCC4)=O)CC2)nc1Cl C1(NC(C2CC(C(C)C)OCC2)=O)CCC(C)N(C(=O)CO)C1 O=C(C#CC1CCCO1)NC1CCC(CNC(c2cnc3scnc3c2)=O)CC1 C1(CNC(Cc2scc(C)n2)=O)C2CN(C(c3c[nH]nc3C(C)(C)C)=O)CC12 C(=O)(CC(C(F)F)NC(C12CCN(CC1)CC2)=O)N(CC(O)C(F)(F)F)C C=CC(C)(O)CC(=O)NC1(CO)CCCN(C(=O)Cc2ccc(C)cc2)C1 C1(C(=O)NCC2CN(C(Cc3c(C)ccs3)=O)CC2O)CCc2nc[nH]c2C1 C1(CCC=C)CCCN1C(C1CCN(C(C2CCCCC2)=O)C1)=O N1(C(=O)C=C2CCCC2)CCC(C2CCCN2C(C2CC2Br)=O)CC1 C(=O)(CCCCN(C)C(C)C)NCC(C(C)C)NC(c1cn(CC(N)=O)nn1)=O N1(C(C2(CC(C)=O)CC2)=O)CCCC(F)(CNC(=O)C(C)(C)F)CC1 CC1(C)C(C(N2CCC(OCC(N)=O)C2)=O)CCN1C(C1SCCCS1)=O N1(CC(=O)NC2(n3cncn3)CN(C(=O)C=Cc3cnccn3)C2)CC=C(Br)CC1 C1(NC(C2C(C(=O)OC)C2)=O)CC2CCC1N2C(C1CCCN1C(C)=O)=O C(=O)(C1=C(C)OCCS1)N1CCCN(C(C(C2CCOCC2)OCC)=O)CC1 S(=O)(=O)(c1ccc(Br)cc1NCC1CCCC(OC)C1)NCCOC(NOCC)=O C1(C(=O)NCC(C2CC2)NC(C2(C)CSC2)=O)CCC2(CC1)CC2(F)F Cc1nc(C2CC2)ccc1C(=O)NCC1(CN)CC1.c1(C(n2ccnn2)=O)ccco1 C1(NC(C(CC2CC2)OC)=O)CN(C(=O)Cc2nc([N+](=O)[O-])n[nH]2)C(C)(C)C1 C=CC(C)(C)C(=O)N1CCC(CNC(C2CCCCN2S(C)(=O)=O)=O)CC1 CC(C)CCC(F)C(=O)NCC(C)CC(N1CC2(CCCC2)C1)=O C1(NC(c2cnc(C)c(C)c2)c2n(CCCSC)nnn2)CCC2(CCC2)C1 CCC(CC)(CO)C(=O)NCC1CN(C(c2csnc2Cl)=O)C2CCN1C2 C1(CNC(c2c(C)csc2)=O)CN(C(=O)COc2ncccn2)CCC1(F)F C1(N(C(C(c2ccccc2F)OCC)=O)C)CCCC(NC(C2(OC)CC2)=O)C1 Cc1cccc(N(C(C)C)C(C)C)c1NC(c1ccc(C#N)cc1)=O c1(C(=O)NCC2(CCNC(C3COC(C)(C)O3)=O)CC2)n[nH]c2cc(Cl)ccc12 N1(C(C(C)OC)=O)CC2(C1)CN(C(C1(C)CC3CCC(C1)S3)=O)CC2CO C1(NC(C(C)n2ccnc2)=O)CC(C)(NC(=O)C(O)Cc2cn(C)cn2)C1 C1(C(=O)NCC(CC(C)C)NC(CN(C(COC)=O)C)=O)CN2CCC1CC2 c1(CNC(C2C(C)C2)=O)nc2c(s1)CN(C(c1ccc(Cl)s1)=O)CC2 c1(C(=O)NC2CN(C(C(CC=C)C)=O)CC2O)ccc(-c2cccnc2)nc1O C1(C(N(CCNC(=O)C(O)C(C)(C)CC)CC)=O)Cc2cc(Cl)ccc2O1 N1(C(C(CC)SC)=O)CCC2(CC1)OCCCC2NC(c1cc(F)cc(F)c1)=O C1(CC(=O)NCC(C)N(C(=O)Cc2cn(C)cn2)C)OCCC1(C)C Cc1cc(C)n(CC(N2CCC(C(C)C(=O)NCc3cn(C)nc3C)CC2)=O)n1 N1(C(c2ccc(C(=O)OCC)[nH]2)=O)CCC2CN(C(=O)CC(C)CF)CCC12 C12(C(N(C)C)=O)CC3CCC(C1C2)N3Cc1cn(C2COC(C)(C)OC2)nn1 N1(C(C2CCN(C(CC=C)=O)CC2O)=O)CC(=O)N(C)CC1C(=O)OC C(C(=O)NC1(CCNC(C2CC(O)C(F)C2)=O)CCCC1)(C(C)C)OC C#Cc1ccc(C(=O)NC2CN(C(=O)CC3=CCCC3)CC2CC2CC2)cc1F c1(C(N2CCC(N(C(=O)CC3CCCC3C)CC)C2)=O)nccc(C)n1 c1(C(=O)NCC2C(CNC(c3c(COC)noc3)=O)C2)oc(S(N)(=O)=O)cc1C C(=O)(C(C)C(O)C(C)C)N(CCC)CCNC(c1cc(OC)nc(C)c1)=O c1(CC)n[nH]c(=NCC(O)COC)s1.c12cc(c(OCC(F)(F)F)c(Cl)c1)N2 O=C(O)CC(CCNCC1(C(F)(F)F)CCOC1)c1ccc(F)cc1 C1(C(=O)NCC2CN(C(=O)C(O)Cc3cccc(F)c3)C2)C2CCCCCC12 CC(=O)C(C)(C)CC(=O)NCc1occc1C(=O)NC1CC1C1CCCC1 C1(C(=O)NCC(CNC(C2(n3cnnn3)CCOCC2)=O)O)CCCS(=O)(=O)C1 C1(=CC(=O)NC(CNC(=O)C(F)CC2CC2)C2CC2)CCOc2ccccc21 C1(F)(C(=O)NCC2(C)CCCO2)CCN(C(C2CCC(O)CC2)=O)C1 C1(C(=O)NC(CN(C(CC2CC(OC)C2)=O)C)C)COC(=O)O1 Cc1nccc(=NCC2CCCN(C(c3cnn(C(C)C)c3CC(C)C)=O)C2)[nH]1 N1(C(c2cc(C)cs2)C(=O)N(c2ccccc2Br)CCCC)CCOC(C)(C)C1 n1(COC)ccc(C(N2CC(C(C(N3CCCC3C(N)=O)=O)OC)C2)=O)n1 N1(C(C(CC(=O)OCC)C)=O)CCN(C(C2CC3CCC2C3)=O)CC(C)C1 C1(C(=O)NC2(CC)CC2)N(C(=O)C=Cc2cc[nH]c2)CCC1(C)C N1(C(c2cc(SC)nn2C)=O)CCN(C(C2CCCN2N=O)=O)CC(O)C1 C(C(CN(C)C)CC(=O)N1CCC(F)(F)C1)NC(C)=O.N1CCCC1CC=O Cc1ccc(F)cc1C(=O)NC(C)CCC(=O)NCCN1CCCC(O)C1 C1(CC)CN(C(C2(c3ccccc3)CC2(F)F)=O)CCC1N=c1[nH]nc(CO)s1 C1(C(N2CC(OCCNC(C3(CC)CCCC3)=O)C2)=O)CCc2cnc(C)n2C1 c1(OC(CNC(c2nnc(-c3cccnc3)o2)C)C)ccccc1F c1(C(C)OC)nc(-c2cnn(C(C)C3CC3)c2)nn1C1CCN(C)CC1 C(CC(C)(C)CC(=O)NCCCNC(C1CC1(C)Cc1ccccc1)=O)OC C1(CNC(C=C(C)C)=O)CC(O)C(O)CC1C(N1CC(C)(CO)CC1(C)C)=O C1(NC(C2(OC)CCCC2)=O)CC(CNC(c2cncc(CO)c2)=O)C1(C)C c1(N2C(CNC(C3CCN(C)CC3)=O)CCC2)nccc2c1C(=O)OC2(C)C CN(S(=O)(=O)N1CCOCC1C)C1CN(C(=O)OC(C)(C)C)C1 C(=O)(C1=NN2CCCN=C2N1)N(CCN(C(C)C)C(c1cncnc1)=O)C N1(C(C)=O)CC(CNC(=O)CC2CCC(C)(C)CO2)C2(CCC2)C1 n1(CC)ncc2cc(CC)ccc12.C1(C(=O)OCC2CN2)Cc2ccccc2O1 c1(OC)ccc(C(=O)NC2CC2CNC(=O)CC(C)N(C)C)c(OC)c1 c1(C(N(C)CC2(NC(C3CC(C(C)C)C3)=O)CC2)=O)cccc2c1C(=O)CC2 CN1CC(CCNC(=O)CC2(C(=O)NCc3cnns3)CCC2)C1 CC1(C)C(C)(C)C1(F)C(=O)NC1COCC1NC(=O)CCC1CCOC1 C1(CC#C)(NC(C2CC(CNC(c3c(C)[nH][nH]c3=N)=O)C2)=O)CCCOC1 N1(C(c2c(OC)cnnc2)=O)CCC(NC(C2OCCC2(C)C)=O)C(C)(C)C1 O=C(C(F)(F)CC1CCC1)NC1CCN(C2CCN(C(=O)C(O)C3CC3)C2)CC1 C(C(C(=O)NCCC(C)COC)NC(=O)COC1CC=CC1)OC C(=O)(C1=CCCS1)NC(C(C)NC(C1CCCN1c1ccccc1)=O)CO c1(CNC(C(=O)NCCC(C)(C)SC2CCCO2)=O)ccc(OCC(F)F)cn1 Cc1nn2c(C)cccc2c1C(=O)NCC(O)CNC(=O)CS(=O)(=O)C(C)(C)C C1(CNC(CCN(CCC)C)=O)CCC(C)CN1C(c1cc(Cl)cs1)=O Cn1cnc(C#N)c1C(=O)NCC=CCNC(c1cnn(C2CC2)c1)=O CC(C(=O)N(CC(O)CN(C(=O)C=Cc1ccc(Cl)nc1)C)C)S(N)(=O)=O c1(C(=O)NCC2CCN(C(=O)CN3CCCC3=O)C2)cc2c(O)ncnc2cn1 C1(C(N2CCC(CN(C)C(C3CC=CCC3)=O)C2)=O)CCN(CCO)C(=O)C1 C1(C(N(C2CCCN(C(c3ccc(C(F)F)o3)=O)C2)C)=O)CC(=O)N(C2CC2)C1 C1(C(=O)NCC(CC)Oc2ccccc2)C2CN(c3ncccc3C)CC12 c1(CC(N2CC(O)(CNC(=O)CC3CCCC3(F)F)C2)=O)cc(C2CC2)ccc1Cl CCC(c1ccc(OC)cc1)=CC(N1CCN(C(C2CC2C(F)F)=O)CC1C)=O Cc1cnc(CC(=O)NC(C)CN(C)C(C2CCN(C3COC3)C2)=O)s1 C1(C(N(CC(=O)NCCc2ccc[nH]2)C2CC2)=O)CCCN1C1CC1 CCC(C(=O)OC)C(=O)NCC(C)N(C)C(C1CCOCC1(C)C)=O C1(C(=O)OCc2ccccc2)(CC)CN(N2CCCC(OC)CC2)C1 C1(C2CC2)(C(=O)OCC)CC1NC(c1ccncc1F)=O N1(C(C2CC(F)CN(C(c3occc3C3CC3)=O)C2)=O)CCN2CCOCC2C1 C(CC(C)(C)C(=O)NOC1CC2CCC1C2)NC(C1(C)N(C)CC(O)C1)=O c1(NC(C2C=CCN2C(c2cnccn2)=O)=O)c(O)cccc1Br C12(NC(C=CC)=O)CC(C)(C1)OC21CN(C(=O)C(C)(O)C(C)C)C1 C1(F)(CNC(c2cc(C)n(C(C)(C)C)n2)=O)CCCN(C(=O)CC2CCOC2)C1 CS(=O)(=O)CC(=O)NCCCOCCNC(=O)CCNC(C1CCCO1)=O CC(C)CCCCCC(=O)N1CC(C(=O)NCC2CC23CCOCC3)C(C)(C)C1 C(=O)(CCCC(C)(C)C)N1C(C2CCCN(C(C(C)N=[N+]=[N-])=O)CC2)CCC1 N1(C(CSCCC#N)=O)CCC2CCN(C(=O)CCCC(F)F)C2C1 C(C(CC(=O)NCc1ccccc1O)NC(c1cnoc1C(C)C)=O)OC C1(NC(C(F)=CC)=O)CCC(NC(=O)Cc2cncn2C2CC2)CC1 C(=O)(C(C(C)(C)C)NC(=O)CC1CCC(=O)C1C)N1CC(C)(C)C1C1CC1 c1(C(N2C(CC)C(NC(C34CCC3C4)=O)CC2)=O)cc2c(C)cc(Cl)cc2[nH]1 N1(C(C(CN(C)C)NC(=O)CC(C)(C)C(F)F)=O)CCc2c(cnn2C)C1 C1(COC)COCCN(C(=O)CNC(C2CC(N(C)C)C2)=O)C1 C1(CC(NOCC(=C)C)=O)CCCN(C(c2cc(Cl)cs2)=O)C1 N1(C(c2c(F)ccc(OC)c2)=O)CCCC12CCN(Cc1ccccc1)C2=O C(=O)(C1=NOC2COCC12)N1C(C(=O)NCC(CSC)(C)O)CCOCC1 C1(C(C)NC(c2csc(Cl)c2)=O)CCCN(C(=O)CCc2ccccc2O)C1 c1(SC)nc(CC2CCCCC2)nn1C1CCN(CCCCOCCO)CC1 c1(C(CNC(=O)NCCN(CCC)C(C)C)CC)cccc(Br)c1 CC1(C)CC(C(N2CCCC(C(N3CC=CC3)=O)CC2)=O)CNC1=O C1(NC(C(C)NC)=O)CN(C(c2csc(-c3ccc(OC)nn3)n2)=O)CC1C c1(CNC(C(c2cccc(F)n2)N(C)CC2(CCO)CCC2)=O)ccccc1Br CCC(O)C(C)C(=O)N(CCCNC(c1cccc(N)n1)=O)CCO C(C)(C)(CCNC(C1(SC)CN(C(=O)CC(C)O)C1)=O)SC c1(OC)cc(C(N2CC3C(C2)N3C(c2ccccc2N(C)C)=O)=O)cc(Br)c1 N1(C(C(C(CC)CC)C)=O)CCOC2CN(C(C3CN4CCC3CC4)=O)CC12 C=C(Br)CC(C)(C)C(=O)N1CC(NC(C2CCOC2)=O)C(SC)C1 N1(C(c2scc(C)c2Cl)=O)CCC2ON=C(CNC(=O)CS(=O)(=O)C(C)C)C2C1 CC1(C(=O)NCC2(C(=O)NCC3CNC(=O)C3)CC2)CCCO1 c1(OC)ccc(N)c(C(N2CCC(C)(CNC(c3nnc(S)n3C)=O)C2)=O)c1 c1(CN(CCCNC(=O)C(=O)NCCC2CCCO2)CC)cccc(Cl)c1 C(=O)(N(CCC(=O)NC1CCCC1CF)OC)c1n(CC)cnc1 C12(NC(c3cncc(C)c3)=O)CCC(C1)N(C(=O)C(Cl)=CCl)C2 C(C(CC)CC(C)C)NC(c1c(Cl)noc1C)c1n(CCC)nnn1 c1(CCCC)cc(C(=O)NCCCCCNC(=O)CC2CCCN2N=O)sc1C N1(C(C(CCN(C)C)NC(=O)Cc2cccnc2O)=O)CCC2(CNC(=O)N2)C1 N1(c2c([N+](=O)[O-])cn(C)n2)CCCC(C2CCCN(C(C3CC3(Cl)Cl)=O)C2)C1 CCCCC(C(=O)NC(CN=[N+]=[N-])C(=O)NCCc1cccnc1F)C(C)C CCC(CNC(C1CCC2(CCC2)C1)=O)(CC)C(=O)N1CCOCC(CO)C1 c1(OC)cc(Cl)c(Br)cc1C(N1CC2(CNCCO2)C1)=O CCCC(CC(=O)NCC=CCl)NC(=O)C(C)NC(C)(C)CC C(c1cccc(Cl)c1)=CC(N1CC(C)C(CNC(=O)CNS(=O)(=O)N(C)C)C1)=O Cn1cnc2[nH]c(C(=O)NC3CCCC(NC(c4cc(Cl)ns4)=O)C3)cc12 C(C)(C(CC(=O)NC(CO)C(C)(C)CO)NC(=O)C(C)(O)C(C)C)OC CC(CNC(=O)CC1NC(=O)NC1=O)CC(=O)NC(C)Cc1cnc[nH]1 C1(NC(c2c(C)c(C3CC3)on2)=O)CC2(C1)CC(NC(c1ccc(CO)o1)=O)C2 C(=O)(C(C)CCCC(C)C)NC1C(CNC(C(CCC)NC(N)=O)=O)COC1 c1(C(N2CCC(N(C(CNC(CC(C)O)=O)=O)C)C2)=O)cccc2c1CCCC2 N1(C(c2ncn(C)c2)=O)CCC2(NC(C3CCC3)=O)CCCC12 C1(NC(C2CC(=C)C2)=O)C2CC1N(C(c1ccc(CCC)cc1)=O)C2 C(=O)(C(C(C)(C)C)N1CCCNC1=O)NC(CNC(CCC(=C)Cl)=O)C(C)C c1(CCC(=O)NCCNC(c2nnc(-c3ccccc3)o2)=O)c(Cl)cncc1Cl c1(C(N(CC(C)NC(C2C(C(=O)OC)C2)=O)C)=O)ccc(C2CC2)nn1 N1(C(C(CC=C)NC(C)=O)=O)CC2CN(C(c3ccc(OC(F)F)nc3)=O)C2C1 C(CCC(C(=O)NCC(F)(F)F)NC(C1CCCSC1)=O)OC c1(C(N2C(C)CC(CNC(CC(=O)NCC#C)=O)C2)=O)nccc2ncccc12 C1(C2CCN(C(=O)CCCc3cnn[nH]3)C2)(NC(=O)CC2CCCC23CC3)CC1 Cc1c(C(C)(C)NC(C2OCCC2C)=O)nnn1C.C(C)(C)(C)OC(N1CC1)=O C(=O)(C(=O)C(C)CCC)NC1C(OC)CN(C(=O)C(=Cc2cnc[nH]2)C)CC1 c1(NCc2cc(C)no2)cccnc1C(=O)Nc1ncccc1F c1(CNCC(N2C(C(=O)Nc3cccc(Cl)c3)CCC2)=O)ccc([N+](=O)[O-])c(Br)c1 c1(C(C)=O)cc(=NC(=O)COC(c2ccnn2C2CCC2)=O)cc(C)[nH]1 N1(C(C(COC)OC)=O)CCC=CC1C(=O)NCC1CCNC(=O)C1 C1(C(=O)NC2CC(CCNC(CC(C)(C)C)=O)C2)CCC2(CC1)CC2(F)F N1(C(C(C)NC(C)=O)=O)CC(F)(F)CC1C(=O)Nc1ccc(C)c(C(F)(F)F)c1 c1(C(=O)NCCCCNC(C2OCCN(C)C2)=O)ccccc1N=[N+]=[N-] C(=O)(CCC(C)NC(C1(C(=O)OC)CCCS1)=O)N(C)Cc1cnc(C)s1 C=CC(C)CC(=O)NCc1nnn(C)c1C(=O)N(C)CC1CC1C N1(C(COc2cn(C)nc2)=O)CCC2CN(C(C3CC3F)=O)C2C1 C1(OC)(CNC(c2cc(CF)on2)=O)CN(C(=O)CCc2nncn2C)C1 c1(OC(C)C(=O)NC2CN(C(=O)CC3CCCO3)CC2C)ccc(F)cc1 N1CCN(C)CC1C.c1(C(=O)OC)ncnn1CC(=O)OC C1(NC(c2ccc(C)nc2)=O)CCN(c2nccc(Br)n2)CCC1CO N1(C(C=CCOC)=O)CCCC2(CNC(c3[nH]nnc3C3CC3)=O)CC12 Cc1cnc(NC2CCOCC2C)c(S(=O)(=O)NC(c2ncc(F)cc2F)C)c1 c1(C(N2CC(CC)C(NC(=O)C3=CCCC3)CC2)=O)c(C)nc2ccccn12 c1(COC(C2C(C(=O)Oc3c(C)n(C)nc3)CC=CC2)=O)ccc(F)c(Cl)c1 Cc1ccc(C(=O)NCc2nc(C(=O)NC3CC4(CC4)C3)co2)c(C)n1 n1(CC=C)nnnc1C(C)(CNC(C)=O)NCC1(C(F)(F)F)CCC1 C1(CC(C)NC(c2cc[nH]c2)=O)CCN(C(c2cscc2C2CC2)=O)CC1 N1(C(C2COCC(C)O2)=O)CC2(C(N3CC(F)(C#N)C3)=O)CCC1CC2 c1(-n2ncc(C(CC)NC(=O)NCCC3CC(C)C3)c2)ccc(Cl)cc1 Cc1ccc(C)c(C(=O)NCC2CC(CNC(c3cncc(Cl)c3Cl)=O)C2)n1 C(=O)(CC(C(C)C)CCNC(=O)C=CCCC)N1CC(CC#C)OCC1 C1(NC(c2cc(C)cc(O)n2)=O)C2CC3CN(C(=O)C(C)CC(C)(C)C)C1C3C2 C#CCC(C(=O)N1CCCC1CN(C(c1cc(CO)[nH]n1)=O)C1CC1)C1CC1 Cc1nc(C)c(C(=O)N(C2CC(NC(=O)Cn3cnc(=N)[nH]3)C2)C)[nH]1 C(CCN=c1nc(N2CC=C(C(F)(F)F)CC2)c2nccn2[nH]1)c1cc(C)no1 Cc1ccc(CC(=O)NCCC(C)N(C(=O)CC2CCOC2)C)s1 N1(C(c2c(CC)nc(C)n2C)=O)CCN(C(=O)Cc2ccc(C)s2)C(C)CC1C c1(OC)cccc([N+](=O)[O-])c1C(N1CCC(CN2CC(OC)C(F)C2)C1)=O C(CCN(C)C(c1sccc1F)=O)(C(C)(C)C)NC(C(C)CO)=O C1(C(=O)NCCC(C)(C)N(C)C)CC(NC(c2cc(Cl)ns2)=O)C1(C)C N1(C(c2c(SC)ccs2)=O)CC2CCC1C(NC(c1cn(C)nc1C1CC1)=O)C2 N1(C(c2c(CC)noc2)=O)CC(F)(F)CC1NC(=O)CC(C)OC C1(CCCNC(Cc2n(C)nnc2)=O)CCN(C(C2(C)CC2F)=O)CC1 c1(CNC(CCCC(OC)OC)c2n(CCC)nnn2)cc2ccncc2s1 CCC(C)CC(=O)N(C1CC1)CC1CCCC1NC(c1csc(C)n1)=O c1(SC)ncc(C(N2CCN(C(C34CC(C3)C4)=O)C(C)C2)=O)c(Cl)n1 Cc1cc(C(=O)NC2CCN(C(=O)CP(C)(C)=O)C2c2ccccc2)nn1C(C)C C1(CC)COCCC1(c1nnnn1CCC1CC1)NCC(C)(C)C(C)(C)C C1(NC(C2CN(S(=O)(=O)C(F)(F)F)C2)=O)CN(C(=O)CC(Cl)Cl)CC12CCC2 C1(=CCNC(=O)Cc2cnc(C3CC3)[nH]2)CCN(C(C2CC2C(F)(F)F)=O)CC1 c1(CN(C(C2(CNC(C3(C)C(C)C3)=O)CCCO2)=O)C)cnc(C)cn1 C(C)(C(=O)N1CCC(C(C)(C)NC(=O)Cc2ccc(C)c(Cl)c2)C1)(C(C)C)OC c1(C(N2CCCC(c3nncs3)C2)C(=O)NC)ccc2c(c1F)CCC2 c1(C(=O)NC(C#C)CCC)ccc(CC(C)(C)C(N)=O)cc1 C1(NC(C2(SC)CCC2)=O)CCCC(CNC(=O)CSc2nccn2C)C1 CCC(C)(C)CN=c1[nH]c2c(c(=NC3CCC4(CCC4)CC3)[nH]1)COC2 CCC(C)(O)C(=O)N1CC2(NC(=O)CCN3CCC(OC4CC4)C3=O)CC1C2 C1(C(=O)NCCC(=O)N(CC)CC)CC12CCN(C(c1cc(F)c[nH]1)=O)C2 CCC1=C(C(=O)NC2CCC2NC(=O)Cn2cc(C)cn2)SCCO1 N1(C(c2n(COC)ncc2)=O)CC2(CC2)CC1CC(=O)NCC1CC=CC1 C=CCC(C)(CC)C(=O)N1CCC(CCNC(c2ncncc2N)=O)C1 Cc1ccncc1C=CC(=O)NC1(C)CCCN(C(c2[nH]cnc2C)=O)C1 N1(C(C2C(C)(C)CC2)=O)CC2(CC(NC(c3ccc4c[nH]nc4c3)=O)CO2)C1 n1(C(C)CC(=O)N2CC(N(C)C(C3CC3(F)F)=O)C2)cnc2ccccc12 C1(CNC(c2c(C)[nH]nc2-c2ccccc2)=O)CCN(C(C2CC2F)=O)CC1O c1(C(N2CCCC(N(C(=O)COC)CC)C2)=O)cc(C)c(C#N)cn1 c1(C(=O)NC2CCCN(C(CCc3c(C)nccc3)=O)C2)nccc(Cl)c1C c1(C(C)NCC2CCC(F)C2)cc(F)c(O)c(F)c1 CC(C)C(C(=O)N1CC(NS(=O)(=O)CCc2ccccc2)C(F)C1)c1ccc(F)s1 N1(C(CC(CC)C)=O)CCC2(CC1)CN(C(=O)C(C)Cc1ccccc1)C2C(C)C CN=C(NCCc1ccc(C)cc1)N1CCC(F)(C#N)C1 c1(C(N2CC(NC(c3cnn4c3CCC4)=O)C(O)C2)=O)cc(F)cc2cc[nH]c12 c1(C(=O)NC(COCC)(C)C)conc1C(C)NC(c1ncoc1CC)=O C1(C(N2CCC(N(C(C3(C)C(C)C3)=O)C)C2)=O)CC2(CSC2)C1 c1(C(=O)NC(C2CCCN(C(CN(CCOC)C)=O)C2)C)cccc(C)c1C#N C12(CNC(C(=O)N(C)C)=O)CCC(CNC(c3nn(C)c(Cl)c3Br)=O)(CC1)CO2 C1(F)(C(N2CC(C)(NC(c3cccnc3)=O)C2)=O)CC2CC1(c1ccccc1)C2 N1(C(C(C(C)C)=O)=O)CCCCC(C(=O)NCc2cnc3n2CCC3)C1 C=CC(C)(O)CC(=O)NCc1ccc(CNC(=O)CCP(C)(C)=O)cc1F N1(C(C2C(C)C(=O)C2)=O)CC(CC(=O)NCCOC(=N)O)C2(CC2)C1 c1(C(N2CC(CNC(C3CC(=O)NC3)=O)C(F)(F)C2)=O)c(F)ccc(F)c1Cl C#CCC(O)C(=O)N1CCC(CNC(c2c[nH]c(-c3ccc(OC)cc3)n2)=O)C1 n1(CC)cnc2c(NCC(C)C(F)(F)F)[nH]c(=NCc3ccc(Cl)o3)nc12 c1(CN(C(CCN(C(=O)CC2CC(C)=NO2)CC=C)=O)CC)nnc(C)n1C N1(C(CC(CC=C)(C)C)=O)CCc2nc(CNC(=O)CC3(C(F)F)CC3)sc2C1 c1(CC)cccc(C(N2CC(CNC(c3cc(O)nc(Cl)c3)=O)C(O)C2)=O)c1N c1(C(=O)NC2C3CC2N(C(=O)COCCF)C3)cccc2c1OCCO2 c1(C(=O)OC)cc(F)cc2c1CCN(C(C(=O)NC1CCOC1)C1CC1(C)Br)C2 C1(C(=O)NC2(C)CC2C)CCC(CN(C(c2cc(OCC)no2)=O)C)CC1 N1(C(C=COCC)=O)CC2(COC(CNC(C3OCCCO3)=O)C2)C1 C1(C(N(CCC)CC)=O)CC(NC(c2cccc(OC)c2C)=O)C12CCC2 CCCC(C)C(=O)N1CC2CC1C2C(=O)Nc1cccnc1Cl c1(C(=O)NC(CNC(C(C)OCC#C)=O)C)ccc(Br)cc1N(C)C N1(C(CN(CCOC)C)=O)CCCC(C2CCN(C(c3c[nH]c(=N)s3)=O)C2)C1 c1(C(N(C)CCOCCCNC(=O)CS(C)(=O)=O)=O)ccc2c(c1)NC(=O)C2=O c1(NC(NOCC(N2C(C3C(C)C3)COCC2)=O)=O)ccc(C#N)cc1 C1(C(=O)NCC2CCCN2C(C2CCCCC2(F)F)=O)Cc2ccccc2C1 c1(C(=O)NC(C(C)NC(=O)Cc2n[nH]c(=N)s2)(C)C)nccn2nccc12 Cc1ccc(C)c(OCC(=O)NCC2(NC(=O)Cc3n[nH]c(=N)s3)CCOC2)c1 n1(CC(=O)NC2CCN(C(=O)C(F)=CC3CC3)CC2F)ccc2ccccc12 Cc1ccc(=O)n(CC(=O)NC2CCN(C(c3cccc(Br)c3C)=O)C2)n1 C1(F)(CNC(CC(C)F)=O)CCCN(C(C2CC3CC(=O)C2C3)=O)C1 C(=O)(C1=CCCOC1)NCCCC1N(C(CCSC)=O)CCOC1 C(C(C)(C)C(=O)NCc1coc(C)c1)NC(C1CCC(CC)C1)=O Cc1cn2c(n1)CC(C(N1CC(CNC(=O)Cn3ccsc3=N)CC1(C)C)=O)C2 c1(OC)cc(C)c(C(N2CCC(NC(=O)C(C)(C)C)C(OC)C2)=O)c(C)c1 C(=O)(C(CC(F)F)C1CCC1)NCC12COC(C(=O)Nc3ccn(C)n3)(C1)C2 C1(C(=O)OC(C)(C)C)CCCC2(C1)OCCO2.C12CC(C13CCC3)NC(=O)N(C)C2 N1(C(C=C(CC)CC)=O)CC(F)(C(N2CCC(OCCO)C2)=O)C1 c1(C(=O)NCC(C(=O)NC)c2ccccc2)ncc(C(F)(F)F)cc1Cl c1(C(=O)NC(CC)CN(C(=O)CC2CC(CF)C2)C)cnc(C(C)C)s1.C(C)C N1(C(Cc2nc(C)sc2)=O)CCc2ccccc2C1CCNC(=O)COC1CC1 N1(C(C(C2CC2)OCC)=O)CC(NC(c2cnoc2C2CCC2)=O)CC(C)(C)C1 c1(C(=O)NCC(CN(C(COCCC#C)=O)C)(C)C)nnn(C)c1CCC c1(C(=O)NC(C2CCCC2)CNC(C2CC2(F)F)=O)cncc(Cl)n1 N1(C(c2cnc(OC)s2)=O)CCC(C)(CNC(=O)Cc2ncccc2C)C1 C(COC)(CC(=O)N(CCCCC(=O)NC)C)NC(C=CC=CCC)=O c1(C(=O)NCCC2CCN(C(CN(C)CC)=O)C2)ccc(C(F)C(F)(F)F)cc1 c1(C(N(C2CCN(C(c3ccc[nH]3)=O)C2)CCC)=O)cccc([N+](=O)[O-])c1 C1(NC(=O)NC2CC2C2CCCNC2)CCc2nnnn2CC1 C1(NC(C2CCN(C(C3CNC(=O)N3)=O)C2)=O)CCCN(O)C1=O CC1(C)C(C(N2CCC3(CCC3)C2)=O)CCN1C(=O)C1=CCCCC1 CCCCC(CC)CC(=O)N1CC(NC(=O)COC(C)=O)C(c2cncn2C)C1 C1(NCc2ccc(C(=O)OC)o2)CCOC(CSC(C)C)C1 c1(C(N(C2CCCN(C(N)=O)C2)C)=O)cc(C(C2(F)CC=CCC2)=O)ccc1Cl C(=O)(CCC(=O)N1CC(NC(C2CC2c2nncs2)=O)C(O)C1)NCCC N1(C(c2[nH]cnc2C)C(=O)NC(CC)C)CCC(O)(CC)C1.c12ccc(o1)C2 N1(C(C(=O)NCC2(F)CC(NC(C3ON=C(C)C3)=O)C2)C)CCOCC1=O c1(C(CC)NC(=O)NCCC2CC(O)C2)nocc1C C(=O)(CCCCCC(C)C)N1C(NC(C(CCC)CCC)=O)CC(OC)C1 c1(C(N(CCNC(c2cn(CC=C)nc2)=O)CC)=O)c(SC)nc(O)nc1C C1(NC(C=NOC)=O)CCC2(CCCN(C(c3scnc3Cl)=O)C2)C1 C12(C(=O)O)CCCC1(C(=O)NC1CCCN(c3ccccc3)C1)C2 N1(C(c2cn(C)nc2)=O)CCC(N(CCO)C(C2CCSC2)=O)CC1 N1(C(CC2CCN(C)CC2)=O)CCN(C(=O)CC2CCOC2)C2CCCC12 C1(C(N2C(C)CNC(=O)CCOCC2)=O)CC(N(C)C)C1.C(C(C)C)OC C#CC(C)(C)C(=O)NC1CCCC(N(C)C(c2ncsc2NC)=O)C1 C(=O)(CC(C)(C)CNC(c1cccc(CO)c1)=O)N1CCN(CCOC)CC1 C1(C(N2CCN(C(C3C(=C)C3)=O)C(C)C2)=O)C2CCC1(C)C2(C)C C1(C(=O)NCC(=O)N(C(C)C(=O)NC2CC2c2cnc[nH]2)CCC)CCCC1 C(=O)(C1CN(C)C(=O)c2ccccc21)N(C1CN(C(C2CC2C(C)(F)F)=O)C1)C Cc1cncc(C(=O)NCC2CC2NC(=O)CCc2cccc(O)n2)n1 N1(C(c2cccc(CC)n2)=O)CCCC12CCN(C(=O)C(C)c1ccco1)C2 CCCS(=O)(=O)CC(=O)N1CC2C(CNC(C3CCCN3C(=O)OC)=O)C2C1 C1(CCOC)(NC(C2CCC2(OC)OC)=O)CCN(C(c2cc(C)c(C)o2)=O)C1 c1(C(=O)N)ccc(Oc2ccccc2Cl)nc1.CC1CN1C.C(C)(C)(C)OC C1(C2CCN(C(=O)CC3SC(=N)NC3=O)C2)(NC(Cc2ccc(C)s2)=O)CC1 N1(C(C(CCSCC)NC=O)=O)CCCC(NC(C2COCCN2C=O)=O)CC1 C1(C(C)(C)C)CCCN(S(=O)(=O)NCc2ccc(Cl)o2)C1 CCCCCCCCN(CC(C)CNC(C)=O)C(C1(C)CC2CC2C1)=O c1(C(N2CC(C)N(C(c3sccc3CN(C)C)=O)CC2)=O)cnn2cccc2c1 C1(NC(CN(CCC)C)=O)CCC(C)(C)CC1CNC(c1ccsc1CC)=O C(C(C)C(C)C(=O)N1CC(C(O)C(=O)Nc2csc(C)c2)C1)OC C1(C)(CNc2cc(N3CCCC(C)C3(C)C)nc(CO)n2)CCOC2(CCC2)C1 CC(C)(CC(=O)N1CC(CNC(c2ccc(O)c([N+](=O)[O-])c2)=O)C1)CC(F)(F)F N1(C(C(C)Br)=O)CCCC2(CCN2C(=O)Cn2ccnc2)C1 S(=O)(=O)(c1ccc(F)cc1)N1CCC(CC(=O)NCCc2cnc(C)s2)C1 C1(C(=O)NCC)COCC2(CCNC2)O1.c12cc(ccc1F)CCOC2=O C1(C(=O)NC(C)CCCCNC(=O)CCn2cnnn2)CCC2(CCC2)C1 CC(C)CCC(=O)N1CC2CC2(NC(=O)C(C)CCOc2ccccc2)C1 c1(N2CC(CC)OCC2)ccc(S(=O)(=O)NC2CC3(C2)CC32CCC2)cc1C#N C1(N(C)C(C2(C)CC3CC3C2)=O)CCCN(C(=O)C=CC=C(Cl)Cl)C1 c1(OC)ncc(Cl)c(C)c1C(N1CCCOC(CCNC(=O)C(C)SC)C1)=O c1(OC)cc(C(=O)NC(C)CC(C)NC(=O)C(=Cc2ccco2)C)cc(F)c1F N1(C(c2ccc(CC)[nH]2)=O)CC2CC(O)C1C2NC(C1(COC)C=CCC1)=O C(CCC(C)C(=O)NC1(CC(=O)NCC2Cc3nccn3C2)CCC1)OC C1(CNC(c2ccc(-n3nccn3)cc2)C)CC12CCSCC2 c1(C(=O)NCc2onc(-c3ccc(C(=O)OCC)cc3)n2)ccc(F)c(Cl)c1F c1(C(=O)NCC2CC2NC(=O)Cn2ccc(C(F)F)n2)ccc(OC(F)F)cn1 c1(C(N2C(C(C)NC(CCC(=C)Cl)=O)CCC2)=O)ccc2ccccc2c1 S(=O)(=O)(c1cccc(=NCC2CCCC(C)(C)CC2)[nH]1)NC(CCCC=C)C CCC(CC)CCCC(=O)N1CCC(OCC(=O)NCCC(C)N(C)C)C1 C12(NC(c3ccc(OCC)nc3)=O)CCCC(NC(c3cn(C)nc3C)=O)(C1)C2 C1(NC(C2CC3(C2)CC3F)=O)CC2(C1)CN(C(c1csc(-c3cn[nH]c3)n1)=O)C2 C#CCC(C)(CNC(C1CSCCN1C(c1cncs1)=O)=O)CO C1(C(=O)NC(C)CN2CCOCC2)CN(C)CCN1C(c1cnn(C2CC2)c1)=O c1(C(=O)NC(CC)(C)CNC(=O)CCN2CCC2)ccc(F)c(OC)c1 N1(C(C(=O)NC2Cn3c(COC)nnc3CC2)=O)CC(C)(C)C(O)C(C)(C)C1 Cc1ccccc1-c1nsc(N(C2CC(NC(=O)CC3CCNC3=O)C2)C)n1 Cc1cnc(CC(C2CCC2)NC(=O)C(=O)NC(C)C(F)(F)F)nc1 N1(C(c2cccc(-c3nc(=O)o[nH]3)c2)C(=O)NCC=C)CCC(C#N)CC12CC2 n1(CC(=O)NC2C(NC(C3(C=C)CC3)=O)CC2)cc(S(C)(=O)=O)cn1 C1(C)(CNC(C2C(C(C)C)C2)=O)CC(NC(=O)CCN2CCOCC2)C1 C(=O)(C(CO)C(C)(C)C)NCC1(CC(=O)NCC(C)CC(F)(F)F)CC1 c1(C(=O)NC(CNC(C(C(C)(C)C)O)=O)CO)ccc2ccccc2c1F C(=O)(CCC(F)(F)Cn1cc(CO)nn1)N(C)CCSC(=S)SC(C)(C)C CN1CCCCC(C(=O)NCC2C3CCC(C3)N2C(c2cc(CO)[nH]n2)=O)C1=O C(=O)(C1=Cc2ccccc2OC1)N1C(CNC(C2CCC(C)(O)CC2)=O)C=CC1 N1(C(c2cncc(C)n2)=O)CCC2(CCCN2C(=O)C(CO)C(C)C)CC1 c12csc(c1)C(=O)NC2.c1(C(=O)NC2C(OCC)CC2)ncnn1C(C)C C1(n2cc(-c3cncc(OC)c3)nn2)CON(C(=O)C(C(C)C)NC=O)C1 N1(C(C(C(C)(C)C)NC(C=CC(C)C)=O)=O)CC2CCC(C1)C2O c1(CN2CCN(CC)C2=O)nc2ccc(C)cc2[nH]1.c1(NC)cnc(OC)n1C CCCCC(O)CC(=O)NCCC1CC(F)(F)CN1C(c1cnc(Cl)c(C)c1)=O c1(C(=O)NCC(C)CN(C(=O)C(C)N2CCCC2)C)cccc2c1CCO2 C1(NC(CN(c2ccnn2CC(F)(F)F)C(C)=O)=O)C(C)C1(F)F CC1NC(=O)CCC1NC(C1(CCNC(=O)CC2CC3(CC3)CO2)CCC1)=O NC1(C(=O)NC(c2ccncc2)CO)CCC2CCC12 c1(CCC(=O)NCC2CC(NC(c3ccn(COC)n3)=O)C2)cc(C)nn1C c1(CNC(=O)NCc2cc(C)c(-c3ccccc3Br)s2)cccc2nn[nH]c12 N1(C(c2c(CC)nccn2)=O)CCN(C(C2CCCC23CC3)=O)CCC1C Cc1c(Br)ccc(C(=O)NCCC(C)NC(C2CCC(F)(F)C2)=O)c1F C1(CN(C(C2N(C(CC3(OCC)CC3)=O)CC=C2)=O)C)CCCCC1O c1(NC(c2c(CNC(C3(C)CC4CC4C3)=O)noc2)=O)cnc2ccccc2c1 N1(C(CSCC)=O)CCN(C(C2(c3ccccc3)CC2(F)F)=O)CCC1C C(C1C(=O)N1)N(C)C.C1(CNC(=O)OC(C)(C)C)CCCS1 c1(NC(C)=O)cc(C(=O)NOCC(=O)N(CC(C)C(C)C)C)c[nH]1 C1(CNC(c2c(C)n[nH]c2)=O)CCN(C(C2CCSC2)=O)C12CC2 N1(C(CSC)=O)CCOC(CC(=O)NC2CN(C)CC2C)C1 n1(CC(=O)NCC2CC(NC(C=C(CC)C)=O)C2)cc(Br)c(=N)[nH]1 N1(C(c2cc(C)c(F)cc2)=O)CC(O)(C2CCN(C(C3CCCSC3)=O)CC2)C1 N1(C(C2C(C)C2C)=O)C2CCC1CN(C(=O)CN(c1ccccc1)C)CC2 CCCCC(C(=O)N(CCCCNC(c1[nH]ccc1C)=O)C)N1CCCS1(=O)=O C1COCCN(C(C2(C)CCC(=O)N2)=O)C1.C(=O)(CCC(=O)NC(C)C)NC CC(C)C1C(=O)N2C(CC2C)C(=O)NC1C.c1(C(N)=O)cnc2ccccn12 c1(NC(C2N(Cc3ccc(C(=O)OC)cc3)CC(O)C2)=O)cnc(Br)cc1C C1(NC(c2ccc(Cl)nc2O)=O)COCCN(C(C2(C3CCCO3)CC2)=O)C1 c1(C(C)C(=O)NCCNC(c2cnc(C(C)O)s2)=O)ccc(S(C)(=O)=O)cc1 C(C(C(=O)N=c1ccn(C(C)C)[nH]1)NC(c1cnc(C2CC2)o1)=O)OCC CCC(C#N)C(=O)NCC1CC(NC(C2CCS2(=O)=O)=O)C1 c1(CNC(=O)NC2C(C(=O)OC)CCOC2)ccnc(Cl)c1F N1(C(CNS(N)(=O)=O)=O)CCC(CC2COCCN2C(=O)Cc2ccoc2)CC1 c1(CNC(=O)NC2(C)CCSC2)cc(Cl)ccn1 Cc1c[nH]c(C(=O)NC(C(=O)NCC(F)(F)C(C)C)C2CCCO2)c1C C1(CC(=O)NCCOCCNC(c2n(C=C)ncc2)=O)CCC2(CCOCC2)CO1 c1(OC)ccccc1N1CC(C(=O)NC(c2cccc(Cl)c2)CO)CC1=O CCC(C)(C)C(=O)C(=O)NC1CCCN(C(c2cnoc2-c2ccco2)=O)C1 C1(NC(C2COCCOC2)=O)CCOCC1NC(C1(c2cccnc2)CC1)=O c1(N2CC(CNC(CCC(C)SC)=O)OCC2)ncnc2c(C)csc12 N1(C(CCN(c2ccncc2)C)=O)CCOC(CNC(c2csc(Cl)c2)=O)C1 C1(N(C)C(c2ccc(CO)cc2)=O)CN(C(C2(CO)COC2)=O)CC1(C)C c1(C(C)=O)cc([N+](=O)[O-])ccc1NC(C)CC(C)NC(=O)CCc1ccnc(Cl)c1 C(=O)(C(CC(F)F)NC(c1cc(C(C)C)no1)=O)N1CCC(CC(C)C)C1 C1(N(C(=O)CCc2ccco2)C)CCC(NC(C2(O)CCOC2)=O)CC1 N1(CC(C)CC(F)(F)F)CCC2CCC(C1)N2C(c1cccs1)=O c1(NC(c2c(C)cc(C(N3CCC(OCCSC)C3)=O)o2)=O)cc(Cl)ccc1C c1(C(=O)NCC2(CNC(C(CC)OC)=O)CC2(F)F)csc2c1CCCC2 C(CCC(C)C(=O)N(CCCC(=O)NC1(C(O)COC)CC1)C)OC c1(NC2CCCC(CNC)C2)nccc(=NCCS(=O)(=O)C(F)(F)F)[nH]1 C(C(=O)NCC(F)CNC(c1cnn(C2CC2)c1Cl)=O)(C(F)(F)F)OC(C)=O N1(C(Cc2cc(C)on2)=O)CC2CC(C1)CN(Cc1cn3c(C)cccc3n1)C2 CCC(C(=O)NC(c1ccns1)C)NC(=O)COCCOC c1(C(N2CCN(C(C3(C)CCCCO3)=O)CC2)=O)cc2n(n1)CCCNC2=O c1(C2C(C(=O)NCCC3(CNC(CC=C=C)=O)CC3)C2)ccncc1C CCC(C(=O)NC(CO)CCCNC(c1cc(CO)n(C)n1)=O)C(C)(C)CC C1(NC(CC(C)c2ccncc2)=O)CN(C(=O)CC2CSC2)CC1C(F)F CC1(C)CC(NC(c2cc(Br)c[nH]2)=O)CN(C(c2coc3c2C(O)C3)=O)C1 N1(CC(=O)NCC(=O)N(c2sccc2Br)C)CCCC2(CCc3ccccc32)C1 c12ccccc1C(c1nnnn1C)NC2CCO.c1(CC)cccc(C(C)C)c1 N1(C(c2cc(C)c(Cl)cc2C)=O)CCC2(CCC2)C(CNC(=O)C(C)C2CC2)C1 C1(NC(C(C)O)=O)CCN(C(=O)Cn2nnc(C(C)(C)C)n2)C1C c1(C(=O)OCC)c[nH]cc1C(=O)NC1CCC(NC(=O)CC(=O)N(C)C)C1 C(=O)(C(C)CC(C)C)NCCOCCOCCNC(c1cc(COC)[nH]n1)=O C1(OC(C)C(N2CCC(O)(CNC(=O)CCc3ncco3)C2)=O)CCCCCC1 c1(C(N2CC(CN(C(C3CCCN(CCC)C3)=O)C)C2)=O)c(C)cccc1F c1(C(N2CCC(NC(c3coc(C(F)F)n3)=O)C2)=O)ccccc1C(F)F C1(C(=O)OCC)C(O)CCN1C(C1CC1CNC(C1CCC(=O)N1CC)=O)=O N1(C(CCC(C)O)=O)CC(O)CC1CNC(C1CC=CCC1)=O N1(C(C2(NC(c3cocn3)=O)CCCCC2)=O)CC(C2CCCCC2)C1 C1(NC(CSc2cc(OC)ncc2)=O)CC(F)CN(C(=O)CC2(NC(C)=O)CC2)C1 N1(C(CCC)=O)CCc2ccccc2C(NC(c2cccc(C(=O)O)c2)=O)C1 Cc1snc2sc(C(N3CCC(CNC(C4CCCC(C(N)=O)C4)=O)C3)=O)cc12 Cn1c(C(=O)Nc2ncc(Cl)cc2Cl)cc2cc(Cl)ccc12 N1(C(=O)OC(C)(C)C)C(C(=O)N=c2nc(C3CCC3)[nH]s2)CCC12CCC2 c1(C(=O)NCCCN(C(=O)C=CSC)CC)csc(Cl)c1 C1(Nc2snc(CC)n2)CCCC12CN(C=O)C2.c1(C(=O)OC(C)(C)C)cnoc1 c1(C2CN2C(C2CC2OC(C)(C)C)=O)ccccc1.C(=O)(CCC=CC(C)C)NOC.C(=O)CN.CC.OC C1(C)(C(=O)NCC2N(C(c3c(CC)nco3)=O)CC2)C=CCCC1 C1(C(N(CC(CC)NC(c2ccno2)=O)C)=O)Cc2nnsc2S1 C1(NC(C=CCNC(CC2C(C)CCO2)=O)=O)CC2CC1OC(=O)N2 C1(OC)CC(O)CN(C(=O)CCN(C(=O)CCNC(=O)CO)CC2CC2)C1 CCC(O)C(C)C(=O)N1CC(N(C)C(c2ccc([N+](=O)[O-])s2)=O)C1 CS(=O)(=O)CCCC(=O)N1CC2C(CNC(=O)CCOc3ccc(Cl)cc3)C2C1 c12ccc3scc-1c3c2.N1(C(=O)Nc2ccc(Br)cc2)CCCC2CCCCC12 N1(C(c2c(CC)c[nH]n2)=O)CCCCCC1C(=O)NC1CCCN(C)C1=O C1(C(=O)NCCNC(c2ccc(C(C)F)cc2)=O)C2CC(=O)CC(=O)C12 Cc1cc(O)c(C(=O)NC2CC3CCC2N3C(=O)COc2ccsn2)cc1Br C(C(=O)N1CCN(CCn2cc(-c3ccc(F)nc3)nn2)CC1)(C(C)C)OC(C)=O c1(NC(N2CCC(OCCOC(C)C)CC2)=O)nc(F)ccc1Cl N(C(=NCc1ccccc1OC(F)(F)F)NCC(C)(O)C1CCC1)CCSC.C1(C)CC1 CN1CCC(C)(NC(=O)CCN(C(C2(C)COC(=O)N2)=O)C2CC2)C1 N1(C(C(C)(C)C2CC2)=O)C2CCC1CC(CCNC(=O)CC1CCCC1)C2 N1(C(c2ccc(C=C)cc2)=O)CCCN(C(=O)C2=C(CC)OCCS2)CC1CO c1(CC)c[nH]c(C(=O)N(CC(C)NC(C2CC2c2ccccc2)=O)C)n1 N1(C(C(C)OCC=C)=O)CCOCC1CC(=O)Nc1ccc(O)cc1 c1(N2CCCC(CNC(CN(C3CCSC3)C)=O)C2)cc(C(C)(C)C)nc(Cl)n1 Cc1cc(CNC(C2CCN(C(=O)C(C)c3cc[nH]n3)C2)=O)on1 c1(C(=O)NC(C2CCN(C(C3C(OC)C3)=O)CC2)C)cc2n(c1)CCOC2 c1(C(N(CCCCN(C)C(C2CCC3CC23)=O)C)=O)c[nH]nc1OCC(F)F C(=O)(C1=C2CCCN=C2NN1)NC(CC)CNC(c1cc(Cl)c(F)cc1OC)=O C1(C(=O)NC(C)C(=O)N2CCCC2)CC=CCN1C(=O)C(C1CCCCC1)F C(=O)(C1CCc2ccccc21)N1CC2C(NC(=O)C3=CCCOCC3)(CCC2)C1 C12(CNC(C3(Br)C(C)C3C)=O)CCC(CC1)N(C(C1CCOC1)=O)C2 c1(OCCC)ccc(CNC2COCC2(C)C)c(C)c1 C1(NC(c2cc3n(c2)CCCC3)=O)CCN(C(=O)C=C2CCCC2)CCC1CO c1(OC)cc(C)c(NCCOC(C)C)cc1Br Cn1ccnc1S(=O)(=O)NC(C1CCCC1C(c1ccccc1)=O)=O C1(OC)CN(C(=O)CCc2cccnc2F)CC1NC(=O)Cc1ccns1 Cc1cc(C(N2CCC(N(C)C(c3cc(CC(C)C)[nH]n3)=O)CC2)=O)cc(F)c1 c1(C(N2CCCC(NC(CS(N)(=O)=O)=O)C2)=O)nccc2occc12 C=Cc1ccc(C(=O)NCC2(NC(c3cc(C)cc(O)n3)=O)CC2)cc1 C1(CNC(COCCCC)=O)C2CCN(C(=O)CC(C)c3ccco3)C12 c1(C(=O)NCC2(C)CN(CCC3CCS(=O)(=O)C3)CCO2)cc2c([nH]1)CCOC2 N1(C(c2c(OC)n[nH]c2)=O)C2CCCC1CN(C(=O)C(=Cc1ccncc1)C)C2 c1(C(N2C(CC)CN(C(=O)CCSC)CC2)=O)sc2ccccc2c1CC C1(NC(=O)CNc2ncccn2)CC12CCN(C(C1CC1C1CCCO1)=O)CC2 c1(C(N2CCC(Cc3nn[nH]n3)C2)C)c(F)cccc1Cl Cc1cc2cc(C(=O)NCC(C)(O)CNC(c3nc(O)c(C)s3)=O)ccc2[nH]1 C=CCC(CC(=O)NC1C(O)CC1O)NC(=O)CC(C)n1cccc1 C1(CC)CCN(C(C2CC23CCOC3)C(=O)NC2COC2)C(C)(C)C1 Cc1ccc(C(=O)NC2CC(C)(CNC(C3CCNC(=O)C3)=O)C2)c(F)c1F c1(C(N(CCNC(C2CCC(c3cc[nH]n3)O2)=O)CC)=O)ncc(F)cc1N C#CCC(CC(F)F)C(=O)NCC(C1CCN(C(=O)C=CCCCC)CC1)(C)C c1(C(N(C)CC2N(C(C(Cc3c(C)nc[nH]3)O)=O)CCC2)=O)ccc(C#N)[nH]1 c1(CC)conc1CNC(=O)C(C1CC1)NC(c1cc(Cl)ns1)=O CS(=O)(=O)CC(=O)NCCC1(O)CCN(C(c2cc(C(N)=O)ccn2)=O)C1 C12(NC(CC(C)(C)F)=O)CCCCCC1N(C(c1ccc([N+](=O)[O-])s1)=O)CC2 c1(C(N2CCC(NC(C(CC)N(CC)CC)=O)C2)=O)sc2ncnc(N)c2c1C N1(C(C(COC)(C)O)=O)CC=C(CC(=O)Nc2ccc(C(C)C)nc2)CC1 c1(SCC(=O)NCCOCCCN(C)C(C2(C)CC2Br)=O)ccncc1 c1(C(=O)NCC2N(C(C(=O)N(C)C)=O)CCOC2)cnc(OC(C)(C)C)c(Cl)c1 Cn1ncc(C(=O)NC(C)(C)C=C2CCN(C(=O)C(Cl)=CCl)C2)n1 C1(C(=O)NC(CNC(c2c(C)n(C)c(C(C)C)c2)=O)C(C)C)CCCC(C)(C)CC1 Cc1cncnc1C(N1CCCC1C(C)(C)NC(C1CCN(C)C1=O)=O)=O N12CCC(CC1)NC(=O)C2=O.Cc1ccn(CCC(N2CC(C)(N(C)C)C2)=O)n1 c1(C(N2C(CNC(c3c(C)snn3)=O)CC(O)C2)=O)ccc2ncccc2c1 N1(C(C2C(NC(COC3(C)CCC3)=O)CCCC2)=O)CC(O)(C2CC2)C1 C1(NC(C(c2ccnn2C)C)=O)CCC12CN(C(c1ccc(Cl)cc1F)=O)C2 CC1CN2CCN1C(C(N1CCCC(Nc3nccc(C(F)F)n3)C1)=O)C2 c1(C(N2CCC(N(C(=O)CC3CCC(C)C3)CC)C2)=O)ccn(CC)c1C N1(C(C(C(C)O)N(C)C)=O)CCOCC(C)(CNC(=O)CCN2CCCC2)C1 c1(C(N(c2c(C#N)ccs2)C2CC3CNC2C3)=O)cc2ncsc2[nH]1 n1(C(C)(C)C)ccc(C(=O)NCCNC(=O)C(O)(C2CC2)C2CC2)n1 O=C(CCCN=c1nc(N2CCC3CC3C2)c2ccccc2[nH]1)NCC(F)F CC1(C(=O)NCCC2CCCCN2C(c2cc3occc3s2)=O)CCCC1(F)F C(N=c1[nH]c(=NCC2CCSC2)c2sccc2[nH]1)c1c(C)csc1 C=CCC(CC(C)C)C(=O)N1CCC(C)C(NC(=O)COC2COC2)C1 Nc1c(C(N2CCOCC(F)(CNC(c3ccncn3)=O)C2)=O)ccc(Cl)c1F C(=O)(CC(C)CNC(=O)C(C1CCOC1)NC(c1[nH]ccc1C)=O)OC C1(NC(CCNS(C)(=O)=O)=O)CCN(C(c2ccc(=N)[nH]c2Cl)=O)CCC1(F)F CCC(C)(O)C(=O)N1CCN(S(=O)(=O)CC)CC1.N12CCN(CC1)S(=O)(=O)CC2 C1(N)CCc2nnc(C3CCCCC3)n2C1.O=C1CN(C=O)CCCN1 c1(C(=O)NCCC(C)C)ccc(S(=O)(=O)N(CCO)CCN(C)C)cc1.CCO C1(C)(C(=O)NC2C=CCN(C(c3c(C)nc(N(C)CCO)s3)=O)C2)CCCC1(F)F N1(C(CCOC2CN(C(c3cc(C)no3)=O)C2)=O)CCN(C)C2(CCC2)C1 c1(NC)cc(C(=O)NC2(C)CN(C(c3cnc(C(C)(C)C)o3)=O)C2)cc(Cl)n1 c1(C(N)=O)csc(NC(=O)Nc2ccnn2C2CCCOC2)n1 CC(C1CCCCC1)=CC(=O)NCC1C2CN(C(=O)C(=O)NCC3CC3)CC12 Cc1cc(C(=O)NC(C)(C)C(C)NC(=O)Cc2ccccc2F)cc([N+](=O)[O-])c1 N1(C(C(CC)NC(C)=O)=O)CCC(C(F)C(=O)NC2(CO)CCCCC2)CC1 N1(C(COC(C=CS(C)=O)=O)=O)CC(C)Oc2ccccc21.C1(C(=O)NC)CCCO1 CC1CC(N(C(Cc2cnc[nH]2)=O)CCO)CCN1C(=O)COCc1nc[nH]n1 C1(NC(C2CCC3CC23)=O)CC2CCCC(C1)N2C(c1[nH]cc2c1CCCC2)=O C(=O)(C(CCC1CCCC1)N1CCC(C(O)C(F)(F)F)C1)NC(C(=O)OCC)C CC1CN(C(C23CCN(C(=O)C=C4CCC4)CCC2C3)=O)CC(C)(C)C1 c1(-c2nnc(N3CC(CO)OCC3)n2C)ccc(OC(CNC(=O)OC)C)cc1 C1(NC(CCC)=O)CC2CN(C(c3cc(C(C)C)on3)=O)CCN2C1=O c1(-c2nc(CCNC(=O)OC(C)(C)C)sc2)coc2cc(Cl)ccc12.C1(=O)CCO1 Cc1ccc(Cl)cc1C(N1CC(O)(CN(C)C(c2cn(C3CC3)nn2)=O)C1)=O C1(C(=O)NCc2c(CC)nn(C)c2)CC(C23CC(C2)C3)CN1 C1(C(N(CC(C)(C)C(=O)N2CCC(CO)C2)C)=O)C2CCC(F)(F)C12 C(=O)(C1CCCc2cncn21)N1CC=C(CNC(C2(COC)CCCC2)=O)CC1 N1(C(C(CC(C)C)N(C(CCn2ncc(C)c2)=O)C)=O)CCCCC(C)(C)C1 c1(C(N2C(C(=O)OCC)C(Cc3ccccc3)CC2)=O)cc(N(C)C)ccc1N c1(C(=O)OC)nsc(=NCCCCNC(C2CCN(C)C2=O)=O)[nH]1 C1(C(=O)NCCCC(C)NC(c2cc(CO)[nH]n2)=O)CN2CCN1CC2 N1(C(C2(C)CCCCCC2)C(=O)NC(C(=O)OC)C)CCCC(C)(C#N)C1 c1(NC(C(=O)NCCC(CC)O)=O)cccc(OCCN(C)C)n1 C=CCC(CC)C(=O)NCCOCCC(=O)NC(CO)CC(F)(F)F C1(C(=O)NCC)CCCN(C(=O)NC2CCCN(c3ccnn3C)C2)C1 N1(C(C=CCOC)=O)CC(C(=O)NC2(N3CCOCC3=O)CC2)C(F)C1 CC(C)(C)C(CO)NC(C1C=CCN1C(c1occc1Br)=O)=O N1(C(CCC2(C)CN(C(C3(OC)CCCC3)=O)C2)=O)CC2CCC(C1)C2COC N1(C(C=C(CC)CC)=O)CCOCC(NC(C2CC(CF)C2)=O)C1 C1(C(N2CCCN(C)CC2)=O)CNC(=O)CN1C(=O)CCOCC(F)F c1(C(N2C(C)CN(C(=O)C(F)=CCCF)CC2)=O)ccc2ccccc2c1F c1(OC)ccc(NC(C23CC(CO2)N(C(c2ccccn2)=O)C3)=O)cc1C N1(C(C)=O)CCCCC1C(=O)NCCCN(C(C1(C)COC(=O)C1)=O)C1CC1 C12(NC(C(C)OCCN(C)C)=O)COCCC1CN(C(=O)C(C)(C)CF)C2 C1(C(=O)NC2(CO)CN(C(c3cscn3)=O)C2)CCCCC1F c1(C(=O)NC2(CNC(CN3CCC(C)C3)=O)CCC2)cn2c(n1)CCCC2 C1(C(=O)OC)CN(C(=O)C(c2cc(OC)cs2)N)CCN1CC CC(C)C(CO)C(=O)N1CCCC(C(C)NC(c2ccc(F)nc2F)=O)C1 C12(CC)CC(CNC(=O)C3CC3)(CN1C(=O)C(C)Sc1n[nH]c(C)c1C)C2 c1(OC)cc(CNC(=O)NCCc2cc(O)nn2C)c2ccccc2n1 Cc1nc(C(N2CCC(O)C(NC(c3cc(F)ccc3F)=O)C2)=O)c(=O)[nH]c1C n1(CC#C)c(C)cc(C(N2CC(NC(=O)OC(C)(C)C)C(C(F)F)C2)=O)c1C c1(C2CC(C(=O)NC(CC(C)NC(c3c(C)cc[nH]3)=O)C)C2)ccc(O)cc1 c1(OC)ccc(F)c(CNC(C2(NC(C34CC5CC3C4C5O)=O)CC2)=O)c1 c1(OC)ccc(F)c(CN2CCC2C(=O)NC(c2cccc(Cl)c2)C)c1 C=CCC(C)(O)C(=O)NCc1ncccc1C(=O)N(CC(=C)C)C C1(C(=O)NC(C)(C)CNC(=O)CCCn2ccnc2)CC(c2ccccn2)=NO1 C1(C(=O)NCC(C)(CO)NC(=O)CC2CC2)CC2CCC1CC2 c1(-n2cc(C(C)NC(c3cc(Br)c(Br)o3)=O)nn2)ccc(S(=O)(=O)N(C)CCO)cc1 C1(C(=O)NCCC2CC(F)(F)CN2C(=O)C=C(Cl)Cl)(OC)CC2CCC1C2 c1(NC2C(CC)CN(C(=O)C3=CCCS3)CC2)ccc(C)cc1[N+](=O)[O-] C(C(CC)(CC)NC(=O)CC(C)C)NC(C1C(COC)C1)=O.C1(=O)CCN1 Nc1c(F)cc(C(N2CC3(CC(NC(C4(CC(F)F)CCC4)=O)C3)C2)=O)cc1F c1(C(N2C(C)CN(C(c3c(C)ncs3)=O)C(C)C2)=O)ccc2[nH]ccc(=O)c2c1 C1(CN(C(c2cnn(CC)n2)=O)C)CN(C(C2CCCCO2)=O)CC12CC2 Cc1ccc(CN(C(C)C(=O)N(CCCNC(=O)CSCC(F)(F)F)C)C)cc1 c1(CC)ccc(C(=O)NC(C)CCCCNC(C2CC2(C)CC)=O)c(C)n1 C1(CNC(C2(SCC)CC2)=O)CC2CN(C(C34CCC(C3)C4)=O)CC12 C12(CNC(C(CC)(C)OC)=O)CCC(CNC(C3ON=C(C)C3C)=O)(CC1)OC2 C1(OC)CN2CCCC2(C(=O)NCCCn2cnc3c2CCCC3)C1 C1(CNC(CCc2nc(C)sc2)=O)C(C)CCN1C(=O)CN(C)C(C)C N1(C(c2c(C)n(C)nc2)=O)CC2CCC(C1)N(C(c1ccn3cnnc3c1)=O)C2 C1(C(N(CCC(C)NC(=O)CCNC(=O)C=CCl)C)=O)CCc2nn[nH]c2C1 C(CNC(c1cc(C2CC2)[nH]n1)=O)(C(C)(C)C)NC(C1C(C)C1C)=O C1(CNC(CC(C)CNC(C2(C)CCCC2O)=O)=O)CC2CCC(C1)C2 N1(C(C(c2cccnc2)OC)=O)CCC2(CCN(C(C3CC3C(C)C)=O)CC2)C1 C12(C(N(C(C)CCNC(C3CCCOCC3)=O)C)=O)CCC(N(C)C)(CC1)CC2 C1(C(=O)NC2C=CCN(c3nc(SC)nc(Cl)c3)C2)C2Cc3cc(Cl)ccc3C12 CCC(CCCC(=O)N1CCN(C)C1C)NC(=O)CCCCNC(C)=O C=CC(C)CC(=O)N1CC(OC)C(OC)C1CNC(c1cc(O)nc(O)n1)=O c1(OC)ccc(OC)c(C(=O)NCCN(C(=O)CC(F)(F)Br)C)c1 N1(C(c2c(CC)csc2)=O)C2CCC1CC(C(=O)NCC1=CCCOC1)C2 c1(NC(=O)Nc2ccc(OC(C3CCC3)C)cn2)cccc(F)c1I c1(C(=O)NCC(CC(C)C)NC(C(CC#C)C)=O)cnn2cc(OC)ccc12 CC12CC(C(N3CCC(NC(C4CC5(CC5)CO4)=O)C(F)C3)=O)(CCO1)C2 CC1(C)C(NC(=O)Cc2cnsc2)CC1CNC(c1cnc(O)s1)=O N1(C(C2CCCCC2F)=O)CCN(C(=O)NC2(c3ccccc3)CC2)CC(O)C1 CCC(Cc1ccccc1)C(=O)NCC1CC(O)CN1C(=O)CNS(C)(=O)=O C1(CN(c2ccc(Cl)cc2)CC)CCCN1NC(=O)C1CC1 c1(C(=O)NCC2(NC(CC(C)(F)F)=O)CCCCC2)ccc(Cl)c2ccccc12 N1(C(CCC(=O)NC)=O)CC(C)CN(C(c2[nH]nc(OC)c2Cl)=O)C(C)C1 C=C1CCC(C(=O)NC(C(=O)NC2CC(n3ccnn3)C2)C(C)C)CC1 N1(C(Cn2c(C)ncc2)=O)CCC(C)(C(N2CC(N3CCOCC3)C2)=O)C1 N1(C(Cn2ncc(C#C)c2)=O)CCCC1C1CCCCN1C(c1nocc1C)=O c1(C(=O)NC(CC2CN(C(C(C)OC)=O)C2)C)ocnc1C C1(C(N(CCOCCNC(C#CC(C)C)=O)C)=O)CCC(C)(C)OC1 c1(C(C(=O)NCCC(C)NC(c2c(C)ncnc2)=O)C)ccc(F)c(F)c1 N1(C(C2=C(C)OCC2)=O)CC2(NC(c3cc4ccncc4[nH]3)=O)CCCC2(F)C1 c1(CC(=O)NC2C(CNC(C3(OCC)CCCC3)=O)C2)cccc(C(F)(F)F)n1 c1(CCNC(c2c(C)cnn2C)c2nnnn2C(C)(C)C)ccc(Cl)c(F)c1 CCC(CCC(=O)NC1CCSC1)NC(=O)Cc1ccco1 CC1(C)CC(CNC(c2cc([N+](=O)[O-])cs2)=O)N(C(C2CCCCO2)=O)C1 C1(C(=O)NC2CC(C(=O)Nc3cccc4c3OCO4)C2)CCn2ccnc2C1 Cc1nc(C(C2CC2)NC2CC2C)sc1-c1ccccc1 C(C#N)(C1CC1)N(C(C)C1CC1)CC1CC1 c1(COC)cc(O)ccc1[N+](=O)[O-].c12cc(nc(C)n1)N1CC(CO)(C1)NC2=O C(=O)(C(C)(O)C(C)C)NCC(CCCC)NC(c1cccc(C(N)=O)c1C)=O c1(CNC(C(C)N(C(=O)C(O)CC2CCCC2)C2CC2)=O)cccnc1 N12CCC(C(O)C1)C2=O.C1(OCCOC)CCCCC1NC(=O)Cc1cc(C)cs1 C(N1CCCC(CC(=O)N(C)C)C1)N1CCCC(C(CC)(C)O)C1 Cc1c(C(N2CCC(NC(c3c[nH]nc3-c3cccs3)=O)C2)=O)csc1Br N1(C(Cc2cc(C)on2)=O)CCCCC1CCNC(C1(C(F)F)CCCC1)=O C=CC1(C(=O)NC2CCC(NC(C3CCCN3C(C)=O)=O)C2)CCCCC1 C(CNC(=O)CCN1CCCC1)(CNC(=O)C(C)ONC(=O)OC(C)(C)C)OC CC(C)CC(C(=O)NC1CC12CC(NC(=O)CC1CC1)C2)N1CCCCC1=O c1(C(=O)NC)ccccc1OC(CN1CCCC1c1cncn1C)C(=O)O C1(O)(C(=O)NC2CCSCC2)CCN(Cc2csc(Cl)c2)CC1 CCC(C)(C)CC(=O)NC1C2CCN(C(=O)Cc3c[nH]nc3O)C12 C(=O)(CC(C(=O)NC1CCCC(NC(C2(CCO)CC2)=O)C1)NC(C)=O)OC c1(C(N2CC(C(N(CCC(N)=O)C)=O)C(O)CC2)=O)cc(Cl)cc(Cl)c1O CC(C(CO)NC(c1cc(Cl)ns1)=O)NC(=O)CC1CCSC1 c1(C(=O)NCC(C)(C)NC(c2ccc(COC)o2)=O)c(Br)ccc(F)c1C C(CCC(=O)NC1CCCC1CCO)(C(C)C)NC(C(CCCC)O)=O C1(C)(C(=O)NCCC(C)(C)NC(c2n(C)cc(C#N)c2)=O)CC(C(F)(F)F)=NO1 c1(C(=O)NCc2cn(CCN(C(CSCC)=O)C)nn2)ccc(CC)c(Cl)c1F c1(OC)cc([N+](=O)[O-])ccc1CNc1cc(C(N2CCC3(CC3)C2)=O)n(C)c1 C1(O)(CNC(C(N)=O)=O)CCCN(C(=O)CN2C(=O)C=CC2=O)C1 C(=O)(C(F)(F)c1ccccc1)NC1CC(CNC(=O)CC2CCCC2)C1 C1(NC(CC2(CC)CC2)=O)CC2CCC1(CN(C)C(c1cn(C(C)C)cn1)=O)C2 C=CC(CC)CC(=O)NC(CO)C(=O)N1CCC(CC(C)(C)C)C1 Cc1cc(CNC(=O)C=CC(C)N(C(=O)CC2CCCO2)C2CC2)cc(C)c1 C1(C(N(C)Cc2ncnn2C)=O)CCCCN(C(=O)C(O)C(F)(F)F)C1 N1(C(CCC=CC)=O)CC(C(=O)Nc2cccc(Cl)c2C)C(F)(F)C1 C1(C(=O)OCC)CC(F)(CNC(=O)C(=O)NCC2(C(C)(C)C)CCC2)C1 Cc1ncnc(C)c1OCC(=O)NCC(C)(CO)NC(c1cc[nH]c1C)=O C1(C(N2CCCC(NC(CCCOCCC)=O)C2)=O)CCCC(C)(C)O1 N1(Cc2c(CC)cccc2)CCCC2(CCN(C(=O)C(C)n3cncn3)C2)C1 C1(SCC)(NC(=O)C(=O)NCC2CC2)CCCC1.C12CN(C1)C(=O)C2 c1(C(N2C(C(N3CC(COC)C3)=O)CCCC2)=O)c[nH]c(=N)c(C)c1 N1(C(C(=O)NCC(F)F)=O)CCC2(CC1)CC2C(=O)NCC1C=CCC1 CC1(C)CN(CC2CCC(F)(F)C2)CC1NC(=O)CCc1ccco1 c1(CC)nc(=N)[nH]cc1C(N1CC=CC1CNC(c1ccc(C2CC2)cc1)=O)=O C(=O)(C(C)(O)C(C)C)N(CCCN(CC(c1ccccc1)N(CC)CC)C)C n1(CC(=O)OC)cc(C(=O)N(Cc2ccc(C)o2)OC)c(C#N)n1 C1(NC(C2CC(C#N)(OC)C2)=O)CCCC12CN(C(c1cn(C)cn1)=O)C2 C1(C(=O)NCCCc2ccccc2C(F)(F)F)CC(C2CC2)=NO1 c1(C(=O)NC2CCC(CNC(=O)COc3ccon3)C2)c(F)cncc1Cl c1(C(N2C3CCN(C3)CC2)=O)cccc(C)c1O.Cc1nnc(CC=CCCO)s1 CC1C(NC(c2ccc(Cl)cc2F)=O)CCCN1C(=O)CN1C(=O)CN(C)C1=O N1(C(C(C)NC(C)=O)=O)CCC(C)C(NC(c2csc(Cl)c2)=O)C1C C1(=O)CC(=O)NC(C2CC2)C1=O.c1(C(C)N)ccnn1CCc1ccccc1 N1(C(C(C2CCC2)OC)=O)CCC(CC(=O)NCC2CCNC(=O)C2)CC1 C1(C(=O)NCC2N(C(C3OCCC(=O)C3)=O)CCC2)CCCCNC1=O CC#CCCC(=O)NC1CCOCC1NC(C1CCCOC1)=O C1(C#N)(C(=O)NC2(C)CCN(C(COCCOCC#C)=O)C2)CCOCC1 CC(C(=O)NS(C)(=O)=O)N(CCC#N)CC1CC1 c1(C(=O)NC2C(CN(C(COCCN(C)C)=O)C)CCC2)cc2n(n1)CCC2 C1(COC)CC(CNC(=O)Cn2cc(Cl)cn2)N(C(C2CNC(=O)C2)=O)C1 C1(CC)CN(C(=O)CC(=O)NCC(F)(F)F)CCN1C(c1cc(COC)on1)=O C1(NC(C(F)=CC)=O)CN(C(=O)CCc2ccc(C)cc2Br)CC12CCC2 C(CCCC(=O)NC(CSC)C(=O)NCC(c1ncc[nH]1)CO)OCC N1(C(=O)NCC2CCCCC2)CC2CCN(S(=O)(=O)CCBr)C2C1 N1(C(Cc2ccc(CCC)cc2)=O)CC(NC(=O)CC2CCSC2)C2(CC2)C1 c1(-n2ccc(C(=O)NCC3CC(OC)CN3C(=O)CC(C)F)n2)c(F)cccc1F c1(N(CC(=O)NCCCF)CCC)ccccc1 c1(C(=O)NC(CC=C)CNC(c2nsnc2O)=O)cc2cc(F)ccc2s1 C(=O)(C1Cc2c(Cl)cccc21)N(C1CCCN(C(=O)CC=CC(C)(C)C)C1)C Cc1nc(C(=O)NCC(C)NC(=O)C2=CCCC2)c(C)s1 c1(N2CCC(N(C)C)CC2)nc2c(c(=NCC3CC(C)(C)CCO3)[nH]1)COC2 CC(C)CCC(O)C(=O)N(CC(C)(C)CNC(c1ncccc1C(F)F)=O)C C=CCCCCC(C(=O)NCC(=C)C)N1CCN(C2CCC2)CC1.CC=C C(=O)(C1=C(Cl)CCC1)N1C(CN(C(C(c2cc(C)oc2C)C)=O)C)CCC1 c1(NC(CSC)C(=O)NC2CC2)ccc(F)cc1.C1(C)C(=O)OC1=O C#CCC(C(=O)OC)NC(=O)C(C)(C1CC1)N(C)C(c1ccn(CC)n1)=O CC1CC2(CC(NC(=O)C(C)C(C)NC(C3(C(N4CCCCC4)=O)CC3)=O)C2)C1 C1(NC(=O)CCSCC2CCCO2)CC2CC(NC(c3cccnc3)=O)CC2C1 c1(C(N2CCC3(CC2)CN(c2nnc(C4CC4)s2)C3)=O)nccc2ncncc12 C(CCC(C)C)(C(=O)NC1(C)CCOC1)NC(C=NOC)=O c1(C(=O)NC(CO)C(N2CCC=C(Cl)C2)=O)cnn2ccccc12 C1(C(N2CCC(N(C(CN(c3ccccc3)CC)=O)CC)C2)=O)C2(CC2)C12CC2 CC1=C(C)CC(C(N2CCCC(C)(C(=O)NC3CC4CCCC4C3)C2)=O)CC1 C1(CN(C(C2CCCC(F)C2)=O)CC)CCCN(C(c2cc(CC)no2)=O)C1 C1(NC(c2cc(C)ncc2)=O)CN(C(c2cnc(C(C)C)[nH]2)=O)CC2CCCC12 N1(C(c2cn(CCC)nc2)=O)CC(C)C(NC(c2c[nH]nc2C)=O)C(C)C1 C12(CNC(C(C)NC(c3ccoc3)=O)=O)CCC1CN(C(c1ccc[nH]1)=O)C2 N1(C(c2nc(N(C(C)=O)C)sc2)C(=O)N=Cc2ccco2)CCC(CCO)C1C N1(C(Cc2cc(COC)on2)=O)CC2OCC(NC(C3(C)CCCC3O)=O)C(C2)C1 Cc1nc2cc(C(N3CCN(C(c4cnn[nH]4)=O)CC3C(F)F)=O)cnc2[nH]1 CC(C)(CNC(c1cc(CO)[nH]n1)=O)CCNC(=O)CC1CCCOCC1 N1(C(CC2C(C)(C)C2)=O)CCCCCC(NC(c2coc3c2CSC3)=O)C1 OC1(C(F)(F)F)CCC(n2cc(C(CC(=O)O)C3CC3)nn2)CC1 c1(CC(=O)N(C(CN(C(c2c(C)ccnc2)=O)C)C)C2CC2)cccc(C)c1Cl C1(NC(CN(C(=O)CCOC(C)C)CCC)=O)CSCC1C C(C)(CO)(C(=O)N(CCCCCCNC(c1cc(C)n(C2CC2)n1)=O)C)OC C(CC(O)C(C)C)NC(C1(CCO)CN(C(C(C)OCCOC)=O)C1)=O N1(C(c2c(C)nns2)=O)CC2CC(N(C)C(c3ccc(C(C)C)cc3)=O)C1C2 CC(C)C(C(C)NC(=O)C#CC(=O)N(C)C)NC(c1cccc(N(C)C)n1)=O c1ccc(SC(C2CCCC2)Cc2csc(CCN3CCOCC3)n2)cc1 N12CCCN(C(C(C)C)C1)C(=O)c1ccc(n1C)C2=O.C1(C(=O)OC)(OC)CC1 N1(C(C(C2CCN(C(C3CCC(C)O3)=O)C2)(C)C)=O)CCOC2C(O)CC12 C1(CNC(C2(CC=C)CCC2)=O)CN(C(C2CC=CC2)=O)CC(C(F)(F)F)O1 C12CN(CC(F)(F)F)C(=O)CC(CCC)C(Br)=CC=CC(F)=C1CC(=O)N2 N1(C(Cn2ccc(C)n2)=O)CCC(C)(CNC(c2c(C)nn(C)c2C)=O)CC1 c1(C(N(CCC(C(C)C)NC(CCC(=C)C)=O)C)=O)cnc(C)c(CC(C)C)c1 Cc1cc(C=CC(=O)NCC2CCC(NC(=O)C(O)C3CCC3)CC2)c[nH]c1=N O=C1NC2CC(CC3CCN(Sc4ccc(F)cc4)C3=O)(OC1)OCCO2 C1(NC(c2cc(C3CC3)on2)=O)C2CC(NC(C3CC(CO)(CO)C3)=O)CC12 C1(NC(C(=O)NCC(c2ccn(C)n2)C)=O)CCc2nccn2C1 c1(C(=O)NC2CCCC(N(C)C(c3coc(O)n3)=O)C2)c(F)c(N)cc(Cl)c1F N1(C(CC(C)=O)C)CC(O)CC2(CCCC2)C1 CCC(C)CCCC(=O)NC1(C(=O)NC(CO)C2CCC2)CC1 C(c1cnc[nH]1)=CC(=O)NCC1CC(NC(=O)CCC2CCCC2)CO1 c1(C(=O)NCc2c(C)ccc(C)c2)cc(F)c(-n2ccnc2)c(F)c1 C1(C(=O)NCCCN(C(=O)CC2(C)CC2)C(C)C)COC(CCC(=O)OC)C1 C1(CNC(C(CC)CC)=O)Cc2ccccc2CN1C(=O)Cc1cccc(Cl)c1 c1(OC)cc(CC(=O)NCCCC(C)NC(c2cnc(S)[nH]2)=O)ccc1Cl C1(C2CCCN(C(c3ccco3)=O)C2)(NC(=O)C=Cc2ccoc2)CC1 c1(C(N2C(CN(C(=O)CCCOC)CC)CCCC2)=O)cncc2nc(C)[nH]c12 C(N=c1ccc(-c2ccc(CSC)cc2)c[nH]1)c1ccc(OCCC)c(OC)c1 N1(C(C2(CCC)CCC2)=O)CC2C(C(N3CCC(F)(CO)C3)=O)C2C1 CCCC(C(=O)N1CCOC(CC(=O)NCCc2cscn2)C1)NC(C)=O N12CC(=O)N(C1=O)CC1CCCN(C1)CC2.CN(C)CC1CC1 C1(CCNC(C(CC)OCC)=O)CCCCN1C(c1cncc(C)n1)=O C1(O)(CNC(C(CC(=C)C)C)=O)CCCN(C(=O)CN2CC(C)(C)C2)CC1 C(=O)(C(O)CC(C)C)N1CC(CC=C)(C(=O)NC(c2n[nH]c(CC)n2)C)C1 c1(C(=O)NC2CCCCN(C(=O)CCCCF)C2)cc(C2CC2)nc2ccnn12 C12(C(N3C(C(=O)NC(C(=O)N(CC)CC)C)CC3C)=O)CCCC1C2(F)F c1(CN(C(CC)C)CC(=O)N(C)Cc2ccccn2)cnc2c(c1)COC2 Cc1cccc(Cl)c1C(c1nnnn1C1COC1)NC1(c2ccccc2)CC1 C1(C(=O)NCCOCCNC(CCOCC)=O)CN2CCN1CC2 C=C(C)C(C)(O)C(=O)N1CCN(C(=O)CCc2nc[nH]n2)C(C)C1 C1(CC)CC2(CCC2)CN1C(c1cscc1-c1cccc(OC)c1)=O C1(C(=O)Nc2cccc(NC(C(C)n3cccn3)=O)c2)CCc2nccn2C1 CCC(CC)(C(=O)NCC(C1CC1)N(C)C(C1(C)CC1F)=O)c1ccccc1 C1(CNC(C(COC)(F)F)=O)CN(C(c2coc(C)n2)=O)CC12CC2 c1(C(=O)NCCN(CC(C)O)C(c2c(COC)scc2)=O)c(C)[nH]c(C)c1C c1(C(=O)NCCC(C)(C)NC(c2cc(O)ncn2)=O)ccc(O)cc1Cl c1(C(=O)NCC2N(C(C(C)=C(CC)C)=O)CCC2)cc(O)n(C)n1 c1(C(C)C)n[nH]c(=NC(C)(CNC(=O)Cc2c(F)cccc2F)Cn2cccn2)s1 C1(CC=C)(NC(C2CCCC2O)=O)CN(C(C2(NC(C)=O)CCC2)=O)C1 C1(CC)CCCC(NC(=O)C(C2CCCCC2)O)CC1.C12(C)CN(C1)C2=O C1(CCCC)CN(C(=O)CCOC2CC2)CCN1C(c1ncccc1CO)=O C1(N(c2cc(O)c(C)o2)CC)CCCC(c2ccccc2)CC1.c1(C)cn(CC)nn1 C(=O)(C(=O)C(C)(C)C)N(C1CC(C(=O)NCCN(C)C)C1)C.CCO Cc1ccc(S(=O)(=O)N2CCN(C(c3cccc(C(F)F)c3)=O)C3CC23)cc1C C1(CC(=O)N)CC=CCC1.O=C(CCN1CCC1)NCCCCCO C1(C2CCC2)(C(N2CCN(C(CCCC)=O)CC2)=O)CC1(F)F C(CC(F)F)(C(=O)NCc1ncoc1CC)NC(c1c(CC)cno1)=O CCC(C)(C)C(C)CC(=O)N1CCN(C(c2cnc(O)c3cncn23)=O)C(C)C1 C1(N(C(=O)CCN)CC)CCN(C(=O)C(C)N2CC(C)C2)CC1.OC c1(C(=O)OC)cnccc1C(=O)NCCC1(C)CCN(C(C2CCCCN2C)=O)C1 C1(NC(c2c(C)scc2)=O)CCCCC1NC(C1(c2cccc(F)c2)CC1)=O c1(C2C(Nc3cc(NCCc4nc(C)on4)ncn3)C2)cc(Cl)cc(Cl)c1 N1(C(CN(S(C)(=O)=O)C)=O)C(CNC(C2(C)CC=CCC2)=O)CC2CCCCC12 c1(OC)cc(CN2CCC(C(C)NC(=O)Cn3cc(Cl)cn3)CC2)cc(Br)c1 C1(C(N2CCCCC2)=O)(OC)CCN(c2ccncn2)CC1 C1(NC(=O)CC2CC2C2CC2)CC2CC(NC(c3ccccc3O)=O)CC12 c1(C(N2CC(O)(C(C)NC(=O)CCCCO)C2)=O)cccc2c1CCCC2 c1(CC)c(F)c(-c2noc(-c3cc(C)n(CCOC)c3C)n2)cc(F)c1F C1(CC)CCN(C(c2cncc(OC)c2)=O)C1C(=O)N(C)CC1(N(C)C)CC1 c1(C(=O)NCC(CNC(c2c(C(C)C)noc2)=O)C)nccnc1-n1ccnc1 c1(CCC(N2CCC(CNC(C(CCOC)C)=O)C2)=O)ccc(O)c(F)c1 N1(C(CC(=O)OC)=O)CC(CNC(=O)C(F)C2CCOC2)CC(C)(C)C1 N1(C(CC(CC)O)=O)CCC2(CCCC2C(=O)Nc2cc(O)c(C)cc2C)C1 N1(C(CC(COC)(C)C)=O)CCC2(CCCCN2)CC1 C(C(CO)(CO)NC(c1csc(C#N)c1)=O)N(C)C(c1cscn1)=O C1(O)(CNC(c2[nH]cc(CC)c2)=O)CCN(C(C2(C(F)(F)F)CC=CC2)=O)C1 Cc1cc(C2(C(=O)N(C(C)CNC(c3cnn(C)c3)=O)C)CC2)on1 C12(C(=O)NC(C3CN(C(c4cnc(Cl)c(Cl)c4)=O)C3)C)CC=CC(C1)OC2 N=c1[nH]c(C(=O)NC2CC(NC(=O)C(O)C3CC3)C2)c(-c2ccccc2)s1 Cc1cccc2[nH]c(C(=O)NCCN(C(=O)C(C(C)C)SC(F)(F)F)C(C)C)cc12 c1(CC)onc(C)c1C(=O)NC1(CCNC(=O)C(N2CCCC(C)C2)=O)CC1 CC1CCOC1C(=O)NCc1cnn(CCO)c1.C12CCCC1CC(=O)N(C)C2 c1(C(N2CCN(C(=O)C(O)CF)C(CCO)C2)=O)ncnc(Cl)c1C1CC1 C(C)(C(CC(=O)NC12CC1COC2(C)C)NC(=O)CC(=O)N(C)C)OC c1(N(C(CCNC(CSCC)=O)C)C)ncnc2sc(C)c(C)c12 C1(CN(C)C(=O)NCC(C)(C)CN2CCCC2)CC(CN)CC1O CC(C(=O)NCCCCN(C(=O)C(C)OCCN(C)C)C)c1cc[nH]n1 c1(OC)ncc(Cl)cc1C(=O)NCC(C)(O)CNC(=O)CCNC(=O)C=CCl C(=O)(CCCCCCC(=O)OC)N1C(CNC(c2n(CCC)ncc2)=O)CCC1 Cn1c([N+](=O)[O-])cnc1C(N1CCCN(C(=O)CC2CCC(C)(C)CC2)CC1)=O c1(OCC)ncc(C(=O)NC(C(=O)NCCC2COC(C)(C)C2)C2CCC2)cn1 N1(C(CC(=O)NCC#C)=O)CCC2CN(C(=O)C(C)(COC)CC)CC2C1 c1(OC)ccc(NC(=O)C(=O)NC2CC(CC(=O)OC(C)(C)C)C2)c(C)c1 N1(C(c2ccc(CCC)[nH]2)=O)CCC(C)(C)C1C(N1CCSC(C)C1)=O c1(C(N2CCN(C)CC2)C)nccc(C(=O)NC(C2CCC2)=O)n1 Cc1c(N(C(=O)CN2CCCCC2CC(n2cncn2)=O)C(C)C)cccc1Cl c1(CC)noc(CC=O)c1N1CC(NC(=O)CSCC2CC2)C(SCC)C1 c1(C(=O)NCC2N(C(C(C)(C)N(C)C)=O)CC2)ccc(=O)n(-c2cnn(C)c2)c1 C1(CNC(C(=O)NCC(F)(F)F)=O)CC(O)CN1C(c1coc(Cl)n1)=O C1(C#N)(CC(=O)NC(C2CN(CC3C(C(=O)OC)C3)C2)C)CCCCC1 C1(N(C)C(c2cncc(C(F)F)c2)=O)CCCN(C(c2cscc2C(F)F)=O)CC1 Cc1cc(C(N2CC(NC(=O)CCS(C)(=O)=O)C2)=O)cc2nn[nH]c12 C1(N(C(c2cc(CC)[nH]n2)=O)C)CCCN(C(=O)C(c2ccccc2F)(C)C)C1 c1(NC)ccccc1C(=O)NC(C1CCCN1C(C1CCCC12CC2)=O)C c1(C(=O)NCCN(C(C2(N3CCOCC3)CC2)=O)C2CC2)ccn2cccc2c1 C(CCC)(C(=O)NCCCC1(NC(=O)CC2CCN2C(C)=O)CC1)=CCC c1(C(N2C(CNC(c3n(CC)cnn3)=O)CC(OC)C2)=O)cc(CO)ccc1Cl C#Cc1ccc(CC(=O)NC(c2ccccc2)C(=O)NCC(C)C(F)(F)F)cc1 C1(NC(C2N(C(C3CCN(CC)CC3)=O)CCC2)=O)CC12CCOCC2 c1(C(C(=O)OC)N(C)C(c2cc(OCC#N)cs2)=O)cccc(OC)c1 C1(C)(SCC)C=C(C(=O)N2CCN(CCNC(=O)CCF)C(CC(F)(F)F)C2)C1 Cc1cnnc(O)c1C(=O)NCCCCC(C)NC(C1CCC(=O)NC1)=O c1(C(=O)NC(C)CCCCNC(=O)COCCN(C)C)cn2ccnc2s1 C1(F)(CNC(C2(C)CCCCC2)=O)COCCN(C(C2(C)CCCOC2)=O)C1 c1(C(N2C(C(=O)NCc3cn[nH]c3)CC(F)C2)=O)ccc2c(c1)CCCS2(=O)=O C1(C(=O)NCC(C)CCCO)CCCN1NC(=O)CN1CCCCCC1 O=C(CC(=O)N1CC(CC2CC2)C1)NC(C1C(c2ccccc2)C1(F)F)=O CC1(C)CC(C(N2CCOCC2C2CC2)=O)CCN1C(c1cc(Cl)c[nH]1)=O c1(C(=O)OC(c2c(OC)ncc(C(=O)OC)c2)=O)c(C)cnc2ccccc12 CC1CCC(CCNC(=O)C(F)CC2CN(C(=O)CNC(=O)C3CC3)C2)O1 C1(CC(=O)N(CC(C(=O)NC)C)C)CCCN(C(=O)CC2CNC(=O)O2)CC1 C(C(F)(F)C(=O)NCCC1CN(C(=O)CC2C=CCCC2)CCO1)OC C1(C)(NC(CCC(=C)Br)=O)CCCN(C(c2ccc(C(C)C)cc2O)=O)C1 c1(CCNc2cccc(NC(N(C)C)=O)c2)nccn2c(CO)nnc12 C1(NC(c2cccc(O)c2F)=O)CC(NC(C2(C(F)F)CC2)=O)C12CCC2 C1(CC#C)(C(=O)NCC(C2CCN(C(=O)CC#N)CC2)F)CCCCO1 C1(NC(=O)C(F)OC(F)(F)F)CN(C(c2ccc(CF)cc2)=O)CC1F Cc1cc(OCC(=O)NCCCCCNC(C2(O)CC2)=O)cc(C)c1 N1(C(c2oc(CC)c(C)c2)=O)CCCC2C1CCCN2C(=O)CCCCC(N)=O N1(C(C2N(C(CC(=O)OCC)=O)CC(O)CC2)=O)CC2CCCC(O)C2C1 c1(C(N(C)C)=O)ccccc1C(=O)NCC1CC(NC2(CC(F)(F)F)CC2)C1 C1(CC(=O)NCC2(O)CCN(C(C(C(C)C)F)=O)C2)CCCNC(=O)C1 CCCC(C)(CC)C(=O)NC(C)CNC(c1cnn(-c2ccc(Cl)cc2)c1C)=O C12COC(C(F)(F)F)CN1C(=O)COCC(=O)C2=O.C1(F)(CO)CC1.C(CF)N N1(C(COCC=C)=O)CCN(C(c2cn(CC=C)nn2)=O)CC1.C1(=O)CN1 c1(C(=O)NC(CNC(C(F)=C(C)C)=O)C2CCC2)cc(=O)n2ccsc2n1 CC1CC(NC(=O)C=Cc2ccc(Br)cc2)CC(C)N1 C1(C(CNC(C)=O)NC(C2(C#C)CC2)=O)CCCCC1 C1(NC(C=COCC)=O)CCCN(c2ncncc2C)CC1 C1(CNC(C#CC(C)(C)C)=O)CC2(CN1C(c1ccc(C#N)[nH]1)=O)CC2(F)F c1(OC)cc(C(N2CC(CNC(=O)CN3CCCNC3=O)C3CC23)=O)ccc1F C(=O)(C(F)(CC)C(=O)OC)N(C1CCN(C(COCC=C)=O)CC1)C c1(C(C)C)nnsc1C(=O)N(C1CCC(NC(=O)CCc2nccs2)C1)C C12(NC(C(C(CC)C)O)=O)CC(CO)(C1)OC21CN(C(=O)CN2CCCC2=O)C1 c1(C(N2CC(C(C)NC(C(CC)(CC)CO)=O)C2)=O)cccc2[nH]cc(C#N)c12 N1(C(c2cc(CCC)oc2C)=O)CCN(C)C(CNC(c2c(C)coc2C)=O)C1 C1(CCCC)CN(C(=O)CCN2C(=O)CCC2=O)CCN1C(c1cc(Cl)no1)=O N1(C(Cn2cccc(C)c2=O)=O)CC(O)(C2CCN(C(C3(N(C)C)CC3)=O)CC2)C1 CC1CN(C(c2cc(Cl)ccn2)=O)CC(C)N(C(=O)CC2CC(=O)C2)C1 C(=O)(C(CCC1CCC1)NC(c1ccc(O)cc1)=O)NCCC(C)(C)OC C=CCC(CCCCC)C(=O)N(C1CC(NC(C2CCCN2C)=O)C1)C C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CC(NC(C2C(c3n(C)ccc3)C2)=O)C1 C1(NC(CC2(CC)CCC2)=O)CS(=O)(=O)CC1NC(=O)CCc1cnccn1 Cc1cc(=O)c(C(N2CC(F)CC2CNC(c2cnccn2)=O)=O)c[nH]1 C1(C)(C(N(C)Cc2scc(C)n2)=O)CCCN(C(c2cnnc(O)c2)=O)C1 C(=O)(C(C(C)C)C(C)C)N(CC(CNC(C1CCCN(C(CC)=O)C1)=O)O)CC CCC(CO)(C(=O)N(C)CCOCCNC(c1ccc(C)c(C)c1)=O)OC C(=O)(C1=NNC(=O)CC1)NC1CN(C(COC2(C)CCCC2)=O)CC(O)C1 CC1(C(N2CC(CNC(=O)Cn3nnc(=O)[nH]3)C(O)C2)=O)CCCS1(=O)=O C#CCCCCCC(=O)NC1CCCC1(C)CN(C)C(C1CCCN(C(N)=O)C1)=O c1(CC)ccc(C)cc1NNC(=O)C1(c2cncnc2)CCCC1 C(=O)(C1=CC(O)C(C(c2ccc(OC)cc2SC)=O)C1)OC C1(C(=O)O)(C(N2CCC2c2cn(C3C4CC5C(C4)C35)nn2)=O)CC2(CCC2)C1 C(=O)(C(C(C)C)NC(=O)C=Cc1ccncc1)NC(C(=O)OCC=C)(C)C N1(C(CN(C(C(CC)=CCCC)=O)CCOCN(C)C)=O)CCC(F)(F)C(O)C1 C(CN=c1nc(C2CCOCC2)[nH]s1)(c1ccccc1F)C(=O)C=CC1CCC1 C1(C(N(C2CCN(C(C3CCCC3O)=O)CC2)CC#C)=O)CC12CCCCC2 N1(C(c2nccc(C)c2N)=O)CCC2CN(C(C3C4CCC3CC4)=O)CCC12 Cc1nc2ccc(C(=O)NC3CCN(Cc4c(O)ccc(F)c4Br)C3)cc2o1 C1(CC)CCCN(C(C2C=CCN2C(=O)CCCOCCOC)=O)C1 C=C(C)CC(C(=O)N1CCC(C)(CO)C1)NC(c1cnc(=N)[nH]c1)=O C1(CNC(C(C)OCC)=O)(COC)CCN(C(c2cnnn2C)=O)C1.C(C)(C)(C)S CCC(C)(CNC(C1(NC(=O)C(C)CSC)CCCC1)=O)NC(=O)OC(C)(C)C N1(CC(=O)N(C(C2CCCCC2NC(=O)C2CC2)=O)C2CC2)CCC(F)CC1 C1(C)(CNC(C(CC2CN(C(CCC3(C)N=N3)=O)C2)F)=O)COC(=O)N1 Cc1cc(C(=O)NCC2CCCCC2C(=O)NCCS(C)(=O)=O)nc(O)c1 c1(C(N2CCOCC2CC2CCOC2)C(=O)NCC)cc(C(F)(F)F)cc(F)c1 N1(C(c2c(Cl)cc(C)nc2)C2CC2)CCC(N=c2cc(Cl)nc(C3CC3)[nH]2)CC1 C1(NC(c2cc(N(C)C)no2)=O)CC(CNC(=O)CC2CCC(=O)NC2)C(O)C1 c1(NC2CC(OC)C2)ccc(S(=O)(=O)NCC2CCN2N(C)C)cc1Cl C=CC(C(=O)NCC1CC(C(=O)N(C(C)CC(C)C)C)C1)OC c1(NC(C(=O)N(CCCC)C(C2CCS(=O)(=O)C2)CO)=O)ccccc1OC N1(C(c2c(SC)cn(C)n2)=O)CCCOC(CNC(=O)CCCn2cccn2)C1 C=Cc1cc(C(=O)N(CCN(C)C)Cc2ccc(C#N)cc2)cc(F)c1 c1(C(=O)NC(CCNC(C2N(C(CCC)=O)CSC2)=O)C)onc2ccccc12 C(=O)(CCCCCN(C)C)N(CCCNC(c1cnn(CC)n1)=O)C(C)C N1(C(c2ccsc2)=O)CC(O)(C2CCN(C(C3CCCS3(=O)=O)=O)CC2)C1 c1(C(=O)NC2CCN(C(CC(C)c3ccco3)=O)C2(C)C)cc(N)cc(O)c1F C1(NC(c2cncc(C#N)c2)=O)CN(C(c2cnccn2)=O)C2(CCCCC2)C1 c1(C(N(CC(C)NC(c2c(Cl)cc(C)nc2)=O)C)=O)cc(N(C)C)cc(C#N)c1 C(CC(C)C)(C(=O)N1CC=CC(NC(C2CC(=O)N(OC)C2)=O)C1)NC(C)=O C1(C2CC2)(C(=O)NCC(CNC(c2c(C)ccnn2)=O)CO)CC=CC1 CC1(C)CC(O)CN1C(C1CC(F)CN1C(C1CC1c1ccccc1)=O)=O c1(OC(c2c(OCCCC(=O)NCC)scc2)=O)cccc([N+](=O)[O-])c1 n1(C(C)C)nc(C(N2CCC(C)C(NC(C3CC(C(F)F)C3)=O)C2)=O)ccc1=O C1(C(N(C)CC2CC(=C)C2)=O)CCC2CCC1N2C(c1coc(C)c1)=O n1(C2CN(C(C3(C)COC3)=O)C2)cc(CNC(c2cnn(CC(F)F)n2)=O)nn1 N1(C(CN2C(C)CCC2C)=O)CCN(C(=O)CNc2cccc(Cl)c2)CC1C c1(CC(N2CCN(C(C(CCSC)O)=O)CC2)=O)c(F)c(F)cc(F)c1F c1(C(N2CC3CC2CO3)=O)c(C)cc(Cl)cc1Br.C1(C(C)=O)CC1C=O N1(C(c2scc(S(=O)(=O)NC)c2)=O)CC2(CCN(C(=O)CCN(C)C(C)=O)C2)C1 c1(NC)cccc(C(N2CC(CNC(C3COC(=O)N3)=O)(COC)C2)=O)n1 N1(CCC(=O)NCC2(C(C)(C)O)CCC2)CCCc2ccccc21 C1(OC)CCC(C)(C(=O)NCC(C)(C)OCCNC(=O)C(C)O)CC1.C1(C)CC1 CC(C(=O)NC(CNC(c1ncoc1C1CC1)=O)CO)C(C)(C)c1ccccc1 CCCC(CC(=O)NCC(F)Cl)NC(c1c[nH]c(C)cc1=O)=O c1(C(=O)OC)[nH]c2ccc(F)cc2c1CN1CCC(C(N2CCC2CO)=O)C1 C1(CNC(CN(C2CC2)CC)=O)CN(C(C2CCCC2CF)=O)CCO1 c1(OC)nc(Cl)ccc1C(=O)NC1CC1NC(=O)Cc1cc(C)n(C)n1 C(=O)(C1CCOc2ccccc21)N(C)CCOCCNC(c1nc(Cl)sc1Cl)=O CC(C)C(CCN(C(=O)CCn1cnnn1)C)NC(=O)C(C1CCCCC1)F C(=O)(C(CC(F)F)NC(C1CCOC1)=O)NCCc1cnc(C)o1 C(CCC(C)CC(=O)N1CC(NC(c2cc3n(n2)CCC3)=O)C2(CCC2)C1)=C(C)C C(C)(CN=c1[nH]c2c(c(=NCC3CC4(CC4)CO3)[nH]1)CCC2)c1ncc(C)s1 C#CCCCCC(=O)NCC(C)NC(=O)Cc1cccc(C(F)F)c1 Cc1cc(C(=O)NCC(O)C(=O)NC(C)COC(F)(F)F)c(C)n1C c1(N(C2CC2O)C)ncc(S(=O)(=O)N2CCCN(CC(C)O)CC2)cc1Cl C(=O)(C(CCN(C1CCCC1)C)NC(=O)CCc1nncs1)N(CCC)CCC n1(CCOC)nnnc1C(C)(CCN1CCOCC1)NCC1CCCOC1 c1(C(=O)OC)ccc(NC(C2(C)CCN2Cc2sccc2Br)=O)c(F)c1 c1(C(N(C2CCN(C(c3cc(F)cnc3Cl)=O)C2)C)=O)ncnc2c1cnn2C O=C(C(CC(F)F)C1CCC1)NC1CC(NC(=O)CC2CCCCC2O)C1 c1(CC(=O)NC2CCC(CCNC(CNC(CCC)=O)=O)C2)ccc(C)c(Cl)c1 CCCCCCCCC(=O)NC1C=CC(C(N2CCOCC(CO)C2)=O)C1 C1(NC(C2C(C)CC2)=O)(CNC(=O)CS(=O)(=O)N2CCN(C)CC2)CCCCC1 c1(C(=O)NC(C)CN(C(=O)CNC(C2CCCC2)=O)C)coc2ccc(O)cc12 C1(NC(c2n(C)ncc2)=O)(CNC(=O)CC2CCCS(=O)(=O)C2)CCCCCC1 C1(CC(=O)OC)(NC(=O)C(CCCF)OC)CCC(C)(C)C1 c1(C(=O)NC2(C)CCCC2NC(C2CC(F)(F)C2)=O)noc2c1CCCCC2 N1(C(c2c(CC)ccs2)=O)CCCC(O)(CNC(C2(C)CC3CC3C2)=O)CC1 c1(C(N2CCC(CN(c3nc(SC)nc(C)c3)C)C2)=O)nccc2cccnc12 CC1CN(C(=O)CNC(N)=O)CC1CNC(c1coc(Cl)n1)=O C(=O)(C(O)CCNC(=O)C(c1ccccc1)NC(c1sncc1C)=O)OC CCC(C)CCC(=O)NCCCCCCNC(c1[nH]c(O)nc1C)=O N1(C(CC(CNC(CNC(=O)OCC=C)=O)(C)C)=O)CCC(=C(F)F)CC1 c1(SCC)cccc(C(N2CCC(N(C(=O)C(C)Cc3ccccc3)C)C2)=O)c1 c1(C(=O)NCCCCC(C)NC(Cn2c(C)nc(C)n2)=O)cc2ccccc2o1 Cc1cnc(O)c(CNC(=O)C(F)C2CC(NC(=O)CNS(N)(=O)=O)C2)c1 CC1(NC(=O)CCCNC(N)=O)CCCN(C(C2CC3CCC2CC3)=O)C1 c1(C(=O)NCCNC(C2CC3(C2)N=N3)=O)noc2cc(Cl)ccc12 C(C1=NOC2CCCC12)NC(C1C(C)(C)N(C(=O)CCCC(=O)C2CC2)CC1)=O C(=O)(CC(C)(C)C(C)(F)F)N.Cc1ccc(C(C2COC2)C2CC2NC(CS)=O)cc1 CC1CCCC(CC(=O)NCCC2(C(=O)N(CC(O)C(F)(F)F)C)CC2)O1 C1(NC(COCCSC)=O)C(C)(C)C(NC(=O)CCn2cncn2)C1(C)C C1(C(=O)NC(CCC)CNC(=O)Cn2nc(C)oc2=O)CCc2nnc(O)n2C1 C1(CNC(C(CCC)OCC)=O)CCCCCN1C(=O)CSC1CC1 N1(C(c2c(C)[nH]nc2Br)=O)CCN(C(c2ccoc2C)=O)C2CCCCC2C1 C(C(C)(C)COCC(C)C)NC(C(C)SC(C)C)=O.c1(CC=O)ccn(C)n1 C1(NC(C2CC(CC(=O)OC)C2)=O)CCC(N(C)C(c2oc(C)nc2C)=O)CC1 c1(OC)nc(C)cc(=NCC2CCN(C(c3ccncc3Cl)=O)CC2)[nH]1 C1(CNC(c2cn(CCC)nn2)=O)(CNC(c2cnc(N)cn2)=O)CC12CCC2 c1(OC)ccc(C(=O)NCC2CCN(C(C3CCC34CCC4)=O)C2)nn1 c1(C(N2C(CCCC)CCC2)=O)cccnc1CNC(=O)CCOCC(F)F c1(C(=O)NCC2N(C(c3cc(CC)no3)=O)CC(F)C2)cccc2c1CCN2 O=C(CC1=CSC2=NCCN12)NCC1(F)CCCN(C(=O)CSc2n[nH]c(O)n2)C1 C1(C(N2CC(O)C(C3CC3)C2)=O)CCN(C(=O)CC2CSCCO2)C12CCC2 C1(CNC(c2n(CC)ncn2)=O)CC2(CO1)CN(C(C1CC(=O)NC(=O)N1)=O)C2 Cc1cc(O)ccc1C(=O)NCC(N1CCCC(CCC(=O)N(C)C)C1)=O CC1(C)CC2(CC2C(=O)NCCC2CCCN2C(=O)CCc2cncnc2)C1 Cn1cc(C(=O)NC2CC3CCC2N3C(=O)C(C)(F)F)c2ccccc2c1=O C1(O)(CN(C(C2(CCCC)CC2)=O)C)CCCN(C(=O)Cc2ncc(C)s2)C1 Cc1ccc(NC(=O)C(CNC(C2(C)CCCNC2=O)=O)CC2CC2)cc1C#N N1(C(C(CC)OCC)=O)CC(C(=O)N(CCCN2CCCC2)C)C(C)(C)C1 C(=O)(CCCCC#N)NC(c1cncc(F)c1)CNC(CCCCC=CCC=C)=O c1(CCC(=O)N(C)CCn2cc(CS(=O)(=O)C3CC3)nn2)cccnc1Br Cc1ccc2c(C(=O)NCC3COC(=O)N3)nc(=NCC3C4COCC34)[nH]c2c1 C=CCCC(CC(C)C)C(=O)NCC1(CNC(C2(C#N)CC(=O)C2)=O)CCCC1 c1(C(N2CC(NC(C(C)SCC)=O)CC2(C)C)=O)cnn2c1CCCC2 N1(C(CCc2c[nH]c(=N)[nH]2)=O)CC(NC(c2cn(C3CCCC3)nn2)=O)C2CC12 CC(C)(CC(=O)N1CC(C(F)(F)F)C1CNC(=O)C=CC(F)(F)F)C(F)F CC(=O)CCCCC(=O)N1CC(OCCNC(C2CC(C)N(C)C2)=O)C1 C(C(C(=O)NCC1(F)CC(NC(=O)C(C)(C2(C)CC2)OC)C1)OC)OC CCCC(C(=O)NC1COCC1NC(c1ccc(F)c(F)c1F)=O)C(C)C c1(C(N2CCC(NC(C3C(OCC)C3)=O)C2)=O)ccc(C2CC2)c(F)c1 C1(C(=O)NC(CCC)C)CCC(O)CN1C(=O)C1=C(C)CC1 N1(C(CCCOCC=C)=O)CCCCC12CC(NC(C1CSCN1CC)=O)C2 C1(NC(CC(C)C(F)F)=O)CCCC12CN(C(c1ccnn1CC(F)F)=O)C2 C1(CNC(C(C)OCC#C)=O)CCC(C(N2CC3CC2C3)=O)C1 c1(C(CC)N(CCCC)Cc2nnnn2CC(=O)OCC)c(Br)cnn1C N1(CC)CC(C(N2CC(NC(=O)CC(C)n3cc(Br)cn3)C2)=O)CCC1=O C1(CC)CCCC1(C)C(=O)NC(C1CN(C(=O)CCC2CC(F)(F)C2)C1)C N1(C(=O)C2=CCC2)CCN(C(=O)C=CCF)C(c2ncc[nH]2)C1 N1(C(CCC(CC)NC(C(CC)SC)=O)=O)CC(O)CC12CCCC2 c12coc(c1)CNC2=O.C#CCCCOCC(=O)NC1CC1(C)C(C)C c1(C(N(C2CC(CNC(COC)=O)C2)C)=O)ccc(=O)n(C)c1 Cn1cc(S(N)(=O)=O)cc1C(=O)NC1(CCNC(=O)CC2CCCC(O)C2)CC1 N1(C(C(C)NC(N)=O)=O)CC(NC(=O)C(F)(F)CO)C(CC2CCCC2)C1 CCC(C)(CNC(=O)CC(C)CNC(c1cc(C(C)C)on1)=O)C(N)=O c1(C(N2CCOCC(NC(C3C(C)C3(F)F)=O)C2)=O)cn(C)c2ccc(F)cc12 C1(F)(C(N(C(C(C)SC)C)C)=O)CCCN(C(=O)C(C(C)(C)C)OC)C1 c1(CC(N2C(CCNC(COC)=O)CCC2)=O)ccc(F)cc1Cl c1(C(N(CC(CC)NC(c2ccc(CO)s2)=O)CC)=O)cnc(C2CCOC2)s1 C12(C(N(C3CCN(C(=O)CCc4ccccn4)C3)CC#C)=O)COCC1C2 C1(C(N(C)CC2CCCN(C(C3CC(C#C)(O)C3)=O)C2)=O)CCCCCN1C CCCC(C(=O)N(CCCNC(=O)C=Cc1ncco1)CCC)OCC CCC(CNC(=O)C(c1cscn1)NC(C1(COC)CC1)=O)OC(C)=O CC1(CNC(c2ccc(CCF)cn2)=O)CCCC1NC(=O)CC#N C(CC(O)C(=O)N(C1CN(C(C)C)C1)C)NC(C(C)C1(O)CCC1)=O CCC(CC(F)F)C(=O)N(CCCCCNC(=O)CCc1ccco1)CC N1(C(CC(C)CF)=O)CCN(C(c2ccc3nccnc3n2)=O)C2CCCC12 C(CCCCN=c1[nH]ccc(=NCC2CCCC2O)[nH]1)c1n(C)ncc1 C12(C(=O)Nc3cccc(C)c3C)CCCC1CCN2C(=O)CNc1ccccc1 N1(C(C=C=C(C)C)=O)CC(=O)NCC1C(=O)NCC1COC(=O)N1 C12(C(N3CC4C(NC(C5(C)CC5Br)=O)C4C3)=O)CCC(F)(CC1)CC2 N1(C(C2(CC)CCC2)=O)CC2CC2(CNC(c2ccsc2)=O)C1 C(=O)(CCCCC(C)(C)C)NC(CSCC)C(=O)N(CCC1CC1)CC C(=O)(C(C)(O)CC)N(C1CCN(C(COCCOC)=O)C1)C N1(C(CC2CC(=C)C2)=O)CC(NC(c2c(OC)cccc2O)=O)CCC1C N1(C(C2C(C)(C)CCCC2)=O)CCOC(C)(CNC(=O)CCCCCF)C1 C1(C(C)C)CCN(C(=O)CCC2CCCN2C(C2CC2C2CCC2)=O)CC1 c1(NC(CSCC(=O)NC2CCN(C(C=COCC)=O)C2)=O)ccc(F)cc1 C1(NC(C2CCC(C)O2)=O)CC=CCC1C(=O)NCCS(N)(=O)=O N#Cc1nn(CC(F)F)cc1OCC1(F)CCN(C(=O)C(c2ccccc2)O)C1 c1(C(=O)NCCCN(C(C)C)C(C2CC(F)C2)=O)ccncc1OC(F)F CC12CC(C(N3CC4CC4(CNC(=O)CCC(F)F)C3)=O)(C1)C(C)(C)O2 N1(C(c2c(N)nccc2)=O)CCCC(NC(=O)CC(c2ccc(F)cc2)O)CC1 C1(NC(C(CSC2CC2)NC(C2CC3CC(=O)C2O3)=O)=O)CCCC(C2CC2)C1 N1(C(CCc2ccn(C)n2)=O)CC2CC(NC(=O)Cc3cn(C)nc3Cl)C1C2 CCCC(C(=O)N1CCCC1(C)CNC(=O)CNS(=O)(=O)N(C)C)N(C)C C(=O)(C1=COc2ccccc2O1)N(C(c1c(CC)csc1)C(=O)OC)CC1CCC1 N1(C(C(CCC)F)=O)CCN(C(c2csc3cncn23)=O)CC1CCOC C(=O)(C(F)CC(C)(C)NC(c1ccc(C(F)F)o1)=O)NCc1n(CC)c(C)nc1 N1(C(c2c(CC)nns2)=O)CCCCC(N(C(=O)CC2CCCC2O)C)C1 C1(CN(C(c2cnsn2)=O)CC)CCCN(C(c2cncc(C(C)=O)c2)=O)C1 N1(C(c2cccc(Cl)c2)=O)CCN(C(=O)NCc2cc3sccc3s2)C2CC12 C(C(CNC(=O)Cc1ccns1)C(F)(F)F)NC(c1ccc(COCC)cc1)=O N1(C(C=CCC)=O)CCN(C(c2sccc2C)=O)CC1CC1CC1 c1(C(N(CC(N2CC3CCC3(C(F)(F)F)C2)=O)C)=O)n[nH]c2ccc(Br)cc12 O=C(C#CC1CCOC1)N1CC(C(=O)NCC(N2CCCC2)=O)C2(CCC2)C1 c1(O)ccccc1[N+](=O)[O-].C1(OCCCNC(=O)NC2(OCN)CC2)CC12CC2 N1(C(c2scc(C#N)c2)=O)CC(NCc2ccc(-c3ccncc3)o2)C(F)(F)C1 c1(CS(=O)(=O)NCCS(CC)=O)c(Br)ccc2c1OC(F)(F)O2 c1(C(=O)NC2N(C(C(CC)(O)c3ccccc3)=O)CC=C2)cnn2cnnc2c1 CCCCC(C)C(=O)N(CCCNC(=O)COc1ccc(Br)nc1)CC c1(CC(=O)NCC23CCN(C(C(C)(C)C)=O)CC2C3)ccc(F)cc1[N+](=O)[O-] N1(C(C(C)(C)C(F)(F)F)=O)CC2CCCN(C(=O)C(O)Cc3ccccn3)C2C1 c1(NC)cc(Cl)ccc1C(N1CCC(C)(C)C1CNC(=O)Cc1ccnn1C)=O C1(OC)CCCC(C(=O)NC(C2CN(C(c3ccccc3O)=O)C2)C)C1 C1(CNC(CCCCCC#C)=O)(CO)CC12CCN(C(=O)C(C)(Cl)Cl)CC2 C12(C(N(CCCC)C(C)CC)=O)CC(CN(C(C3CC(C)(C)C3)=O)C1)C2 c1(CNC2CCC(N(C(C3CN(CC)C(=O)C3)=O)C)CC2)cnn2c1CCCC2 C(C(C)(C)C#CC(=O)N1CC(N(C)C2CC2)C1)NC(c1cc(C)c(F)cn1)=O c1(COCC(=O)N(C2CC(C(=O)NC(C(O)CO)C3CC3)C2)C)ccncc1Cl C=CC(C)CCNC(=O)CCC1CCCN1C(=O)C(=CCCC(C)C)NC(C)C Cc1ccc(CC(=O)OCC2OCC3CCC2C3)c(F)c1F C(=O)(C1=CNC2=NCCC2=C1)C(C)CN(C)C(C1CC(c2ccccc2)O1)=O c1(SCC)ccc(C(=O)NCC2CN(C(=O)Cc3cn[nH]c3)CCO2)cn1 N1(C(c2ccc(CC)o2)=O)CCN(C(=O)CC(C)CN(C)C)CC1C(C)(C)C c1(C(=O)NCC2C(NC(C(C)CO)=O)CCC2)cc(C#N)c2n1CCCC2 CCCCCCC(C)C(=O)N(CC(N1C2CCCC1CC2)=O)C(C)C CC(C(O)C(=O)NCC1CCN(C(=O)C=CI)C1)c1ccccc1 c1(C(N2CC(C)C(N(C)C(c3cc(Cl)no3)=O)CC2)=O)n[nH]c2ccc(F)cc12 C12(C(=O)NCC(CCNC(c3ccn(-c4cccnc4)n3)=O)O)CC(CCO1)C2 N1(C(C(C(C)C)SCC)=O)CC2CN(C(c3cc4cccnc4o3)=O)CCC12 N1(C(C(CC)F)=O)CCC(NC(c2cncc(C(=O)N(C)C)c2)=O)C(O)C1 C=CCC(CC)C(=O)N1CCN(C(c2ccc(CCO)cc2)=O)CC1 Cn1cnc(NCC2(C)CCCN(C(=O)CCC3CCCOC3)C2)cc1=O C1(NC(C(C2CC(NC(=O)CCc3ccco3)C2)F)=O)CC(C2CCC2)C1 N1(C(c2c(C)n(C3CCC3)nc2)=O)C2CCC1CN(C(=O)CC1CSCCS1)C2 NS(=O)(=O)c1ccc(C(=O)NCC#CCNC(c2cc(COC(C)(C)C)on2)=O)s1 CCCCCCCCC(=O)NC(CC)CCCC(=O)NC1CCCC1C#N c1(C(N2CC(C)N(C(C3CCS(=O)(=O)C3)=O)CC2C)=O)cc2ccoc2cc1F c1(C(N2CCC(C#C)CC2)=O)c[nH]c2cc(-c3cccc4c3OCO4)cnc12 c1(OC)nc(C)cnc1C(N1CC(CNC(c2cc(C)ncn2)=O)C(C)C1)=O C#CCC(C)(CC)C(=O)NCC(CCC)NC(c1[nH]nc(OC)c1Cl)=O CC(C)(CCC(=O)N1CC(NC(=O)C(O)CC2CCOCC2)CC1(C)C)[N+](=O)[O-] CC(C(=O)OC)C(=O)N1CCC(N2CC(C)(NC(=O)CC3(C)CC3)C2=O)CC1 C(C(=O)NC1COCC1NC(c1nn(C)cc1Cl)=O)(C(C)C)OC Cn1nc2c(c1C(N1CC3CCC1(CNC(=O)COCCF)CC3)=O)COCC2 c1(C(N2CC(CNC(c3cnco3)=O)C2)=O)cccc(OC2CCC2)c1 c1(-c2c(OC)c(C#N)ccc2)ccn2cc(C(N3CCC3C(N)=O)=O)nc2c1 N1(C(c2n(CC)cc(Cl)c2)=O)CC2CCOC2(CNC(C2CCOC2)=O)C1 c1(C(C(=O)NCCCC(=O)NC)N(C2(CCOC)CC2)C)cc(Cl)cc(Cl)c1Br c1(OCC)cc(C(=O)NS(=O)(=O)CC2C=CCC2)ccc1F C1(C(=O)NCC2CCCCCN2C(=O)C2=CCCCC2)CC2CCC(C1)C2 c1(C(N2CCOC(CCCC)C2)C(=O)NCC(=C)C)cc(F)cc2c1CCC2 N1(SC2(C(N(CCN(C)C)C)=O)CC2)CC(NC(=O)Cn2cnnc2O)CC1=O C12CCN(C)C13CCCN(C3)C2=O.c1(OC)ccc(C2CC2)cc1C(F)(F)F C1(CC)(CC)CC(NC(c2cc(C(F)F)on2)=O)CN1C(=O)CCc1nccs1 C=CC(C)(C)C(=O)N1CCC(CC(C)NC(=O)CC2OCCC2(C)C)CC1 C(CCCCNC(c1cc(-c2ccn(C)n2)[nH]n1)=O)OCC C12(CNC(C=CC=CC)=O)CCCC1N(C(c1cn3c(n1)COCC3)=O)CCC2 C1(NC(Cc2cc(C)on2)=O)CCCC(C(=O)NC(C)(C)CCO)CC1 C1(NC(C2CC3COCC3C2)=O)CC2(CCN(C(c3cc(CCO)on3)=O)C2)C1 N1(C(=O)C=CC=C(Cl)Cl)CC(F)(CNC(C23CC(c4ccccc4)C2C3)=O)C1 C(CC(C)SC)(C(C)C)(c1n(C(CC)C)nnn1)Nc1ccc(F)c(C(F)F)c1 C12CN(C3(CCOCC3)C1)N2c1csc(C2(O)CCOCC2)n1.C=CCC.c1(C)ccccc1 C(=O)(C1=NOC(C)C1C)NC(CNC(c1c(C)ncnc1C)=O)C C1(NC(c2nccc(C)n2)=O)CN(C(c2cnccc2Br)=O)CC1S(C)(=O)=O C1(NC(c2cncc(C#C)c2)=O)CC(C2CCN(C(c3ccco3)=O)CC2)C1 C1(CCN(C)C)CCCN(C(c2cc(Br)no2)C(=O)NCC(F)F)C1 c1(C(=O)NCC(N(C(C(C)c2cc[nH]n2)=O)C)C2CC2)cncc2ccccc12 Cc1ccc2occ(CC(=O)NCC3COC4(CNC4)C3)c2c1 C(=O)(C#CC1CCCCO1)NC1CCC(NC(CCCc2n[nH]c(=N)s2)=O)C1 C1(C(=O)NC(CC2CN(C(c3cc(C)c(N)cn3)=O)C2)C)C2(CCC2)C12CCC2 N1(C(CCCCCC)=O)CCCC2(C1)CN(C(C1(C(=O)N(C)C)CC1)=O)C2 C1(C(=O)NC2C(NC(CNC(N)=O)=O)C2)CCC=CCCC1 C1(C(C)C)CCCCN1C(=O)CC1C=CC(NC(=O)C(C)CC2CCC2)C1 C1(NC(c2c(OC)ncc(C)c2)=O)C(C)(C)C(NC(=O)C(C)CC(C)C)C1(C)C N1(C(CN=S(C)(C)=O)=O)CCC2CCCN(C(c3nccc4[nH]ccc34)=O)C2C1 N1(C(C2=C(C)OCCC2)=O)CC23CCCC2(C1)CN(C(=O)C(F)C(C)C)C3 C12COCCN1C2.C1(C(=O)NCCOCC#C)CCC1C(=O)NCC(F)F C(=O)(CC(C)(C)C(F)F)N(CCCNC(c1onc(OCC)c1Br)=O)C N1(C(C(c2ccoc2)NC(C2CC3(CC3)CO2)=O)=O)CC2COCC(C2)C1 C1(C)(C(N(C2CCN(C(CC(C)(C)OC)=O)CC2)CC(C)C)=O)CCNC(=O)C1 c1(C(=O)NCC)cc(OCC(N2CC(COCC#C)C(O)C2)=O)cc(=O)o1 c1(C(N(CCCCNC(C(C)n2cccc2)=O)C)=O)ccc(Cl)cc1Cl C(=O)(CC(CC(C)C)NC(c1sncc1C)=O)N1CC(OC)C(OC)C1 c1(CCNC(C)Cc2nccn2C)cc(O)ccc1Br C=C(C)C(CC(=O)NC1CN(C(C2(CC)COC2)=O)CC12CC2)OCC CC1C(NC(c2ccc(N)cn2)=O)CCCN1C(c1ccc(C2CC2)cc1)=O N1(C(COCCCC)=O)CCCCC1C(C)NC(=O)Cc1nc(C)c(C)o1 C1(CNC(c2ccc(CC)s2)=O)CN(C(C2CC23CC3)=O)CCO1 c1(CC)cccc(C)c1NC(=O)C(C1CCC(C)CC1)N1CCCC1C C1(NC(C2(C)CCCCO2)=O)CN(C(=O)CCc2ncc[nH]2)CCC1C(F)(F)F CCCC(C(=O)NCCOC1CCN(C(=O)C(c2ccccc2F)O)C1)C(C)C c1(CC(=O)NC2C(NC(C(C(C)O)N(C)C)=O)CCC2)ccc(S(N)(=O)=O)cc1 C(C)(CO)(C(=O)NC(C1CCN(C(C2CCCCC2)=O)C1)C)OC C1(C)(OCC(=O)N(C(CO)C2CC2)CC)CN(C(=O)Cc2nc[nH]n2)C1 c12nnc3n1CCCC3C(=O)N2.C(=O)(C#CC(C)(C)O)N1CC(CC)C1 N1(C(C(C(C)C)Cc2ccccc2)=O)CC2CCC1CN2C(=O)C(O)CN(C)C N1(C(C2CCN(S(C)(=O)=O)C2)=O)CCC2C(NC(C3CCOCC3)=O)C12 c1(CC(=O)NCC(N(C(c2c(C)cno2)=O)C)C2CC2)cc(Cl)ccc1Cl C(=O)(CCC(=O)NCC(C1(O)CN(C(=O)CCNS(C)(=O)=O)C1)(C)C)NC Cc1cc(C(N2CCSCC2)C(=O)NCC(F)F)n(C)n1 c1(CN2CCC3(C(C(=O)NCc4cccnc4O)C3)C2)cccc2ccccc12 CCC(C)N(CCO)N(C)CCN1CCCCC1 C1(CNC(CCCOC)=O)CN(C(=O)CC2CC3CCC(C2)C3)CC1(F)F N1(C(c2c(C)coc2)C(=O)O)CCOCC1(C)c1cn(CC(=O)NCCO)nn1 C1(CC(=O)OC(=O)C(C)C(=O)OC)CCCC(C)(C)C1.C1(C)CC(=O)N1CC Cn1cc(-c2cc(C(=O)NC3CCC(NC(c4ccoc4)=O)C3)n[nH]2)cn1 c1(C(=O)NC(c2cccnc2)C(=O)NC(C=C)C)c[nH]c(=NC)o1 CC(C(=O)NC1CCC1NC(=O)CCCN1CCCC1)C(C)c1ccc(F)cc1 c1(CC(=O)NCC2C(NC(Cc3c(C)cc(C)s3)=O)C2)csc2sc(C)cc12 c1(C(=O)NCCC2N(C(C(CSC)O)=O)CCC2)ccc(C(F)(F)F)c(F)c1 c1(C(N(CC(C)(C)CNC(C2CCCS(=O)(=O)N2)=O)C)=O)cccc2c1OCC2 c1(C(C(=O)N2CC(n3cc(C4(C5CC5)CC4)nn3)C2)O)ccc([N+](=O)[O-])cc1 N1(C(C(C=CC)O)=O)CCN(C(c2cc(O)nn2C)=O)CC12CC2 CC1=CCN(C(=O)C(CCN(C)C)NC(c2c[nH][nH]c2=N)=O)CC1 Cc1cnccc1-c1cc(CNC(=NCc2ccccc2)NC2CCCC2)[nH]n1 c1(NC(CCOCCNC(CCC=CC)=O)=O)cc(C)ccc1CO C1(c2n(C(C(=O)OC)C)nnn2)(NCc2cnc(Br)n2C)CC2CCCC12 n1(CCCN(C)C)nc2c(cc1=O)C1(CC2)OCCO1 c1(C(N(CCNC(C2(CO)CC2(F)F)=O)CC)=O)cnn(C(C)(C)C)c1Cl C1(CC=C)(NC(c2c(C)coc2C)=O)CCCN(C(c2cccnc2)=O)C1 C1(CNC(CCOCC)=O)CCCC2CN(C(=O)C(C)(C)CO)CC12 c1(C(=O)NCCN(C(C(=O)NCc2cccc(C)c2)=O)C)cnn2ccn(C)c12 C12(NC(C(C(CC)C)OC)=O)CCCCCC1N(C(c1oc(C)nc1C)=O)CC2 CS(=O)(=O)C1CCC(NC(=O)NC2CCCCC(=O)CC2)C1 C1(C(N2C3C(C(=O)OCC)C(C3)C2)=O)CN(C(=O)CC2CCC=CCC2)CCO1 Cc1ccccc1CCC(=O)NC(C)C(C)(C)NC(=O)CC1CCOC1 c1(C(=O)NCC(CC(C)C)NC(CCCC(C)=O)=O)c(F)cc(C)cc1F C1(C(=O)NC(C=C)COC)CCCCCN1C(c1ccnc(C)n1)=O C1(NC(c2n(CC)cnn2)=O)CS(=O)(=O)CC1NC(C1CC(SC)C1)=O N#CC12CCC(CNC(c3ccc(OCC4CCCCC4)cc3)=O)(CC1)CC2 N1(Cc2cc(OC)c(O)cc2Cl)CCC2(CCCN(C(=O)CCN(C)C)C2)C1 c1(CNC(Cc2cn(CC)nn2)=O)nnn(C)c1C(=O)NCC=C(C)C(C)C N1(Cc2n(CC(=O)OC)ncc2)CC(C(=O)NC2(C(C)(F)F)CC2)CC(F)(F)C1 c1(C(=O)NC2C(NC(C3(CC)COC3)=O)CCC2)nc2c(C)cccn2c1Br CCCC(C(=O)NC1CN(C(=O)CCC2CC(OC)C2)CCC1O)C(C)C C(=O)(CCCCCC(C)(C)C)N(CC(C)(C)CNC(=O)CN1CCCCC1C)CC C12(C(=O)NC(CCNC(c3c(CC)[nH]nc3Cl)=O)C(C)C)CCN(C1)S(=O)(=O)C2 C=CC(C)(O)CC(=O)NCC(C1CCN(C(=O)COCc2nc[nH]n2)CC1)O Cc1nc(Cl)c(NC(c2n[nH]cc2NCc2ccc(F)c(F)c2F)=O)c(Cl)n1 C#Cc1cncc(C(N2CCCC(CC(=O)NCC3(C=C)CCC3)C2)=O)c1 C1(C(=O)NC(C2CCN(C(C3CC(F)C3)=O)C2)C)CN(C)CCO1 C1(NC(c2c(C)ocn2)=O)CCC(CNC(C2(C(C)(C)O)CC2)=O)CC1 C12(CNC(c3c(C)oc(C)c3C)=O)CCC(NC(=O)C(C#N)C3CC3)(CC1)CO2 c1(C(=O)NCC2CCCCN2C(C2CC3C(C2)C3(F)F)=O)ccc([N+](=O)[O-])nc1 C1(NC(C2(C#C)CC2)=O)CCCC(CNC(c2cc(Br)cn2CC)=O)C1 N1(C(CCC2CCN(C(C3(C#N)C(C)(C)C3)=O)C2)=O)Cc2cccnc2C1 N1(C(C(C)NC(CC(C)N(C)C)=O)=O)CC(O)(C2CC2)C1 c1(OC)sccc1COCN(C)CCSc1ccccc1 CC(C)(C)CC(O)C(=O)N(C1(CNC(=O)CC2CCC2C2CC2)CCC1)C1CC1 C1(C(F)(F)F)(NC(COCCCn2cc(CCC(=O)OC)nn2)=O)CC(F)(F)C1 C12(C(N3C(CC#C)(C(=O)O)CCC3)=O)CCC(OC)C1C2 C1(C(C)C)(C(=O)NC2CC3(C(=O)O)CC23)CCCN1C(c1cccs1)=O C1(C(CC)O)CCCCN1C(=O)C(C1CC1)N(C(=O)CCc1ccsc1)C c1(CNc2cccc(CCc3ccc(C(=O)OC)o3)c2)[nH]c(C)c(C(=O)O)c1C N(C1CCc2cc(C)ccc21)N1CCN(Cc2ccc(OC)cc2OC)CC1.C(C)C C(N=c1ccc2ncc[nH]c-2n1)C1OCC(CNC(C2CC23CCSCC3)=O)C1 N1(C(C(C)c2ccsc2)=O)CC2CC2(CNC(c2ccc(F)s2)=O)C1 N1(C(c2ccc(CC)cn2)=O)CCN(C(=O)CCc2cnc(O)[nH]2)CC1CF N1CC2(CCCC2)c2ccc(Br)cc21.N#Cc1cc(S(=O)(=O)N)ccc1C(F)(F)F CC1CC2CN(c3ncnc4c3ncn4CC(O)CCCCO)CCN2C1 N1(CC(=O)OC)CCc2cc(C(N3CCN(C(C)(C)CO)CC3=O)=O)ccc21 Cc1cc(C(N2CCC(NC(=O)C(C(C)O)N(C)C)C(O)C2)=O)cc2nc[nH]c12 N1(C(c2cc(C)c(Br)s2)=O)CCC(F)(C(=O)NC2CC2(F)F)CC1 Cc1nc2cccnc2n1CC(N1CCC12CCCCC2)=O c1(C(=O)NC2C(CNC(CNC(CC)=O)=O)CCCC2)cc(C)c2[nH]cnc2c1 c1(C(=O)NCC(CO)NC(C2N(C)CCC2)=O)cc(N2CCCC2)ccn1 N(C(=NCC(C)c1nccs1)NOCC=C)C1CCC(NC(C)=O)CC1 C1(COC)CN(C(c2c(O)cccc2O)=O)CCN1C(c1cnc(Cl)cc1Cl)=O c1(OC)cc(C2N3CCC2CC3)cc(Br)c1.C(CCN)SC c1(CN(C)Cc2ccc(Br)s2)cc(F)ccc1O N1(C(C=COCC)=O)CCOCC(NC(=O)C(C)(C)C(C)O)C1 CCCC(CC(=O)NOC(C)C(=O)OC)NC(=O)C(C)=C(C)C CCC(C(C)(F)F)NC(C1CN(C(C2(C#N)CCC2)=O)CC1F)=O C1(NC(C(C2CN(C(=O)OC3CC3)C2)O)=O)CCC(NC(c2ccoc2)=O)CC1 c1(OCOC)ccc(S(=O)(=O)NCc2ccc(C)cn2)cc1.N12CCCC1C2 C(=O)(C(C)S(C)(=O)=O)N1CC(OCC)(CNC(c2cc(CC)[nH]n2)=O)C1 N1(C(c2c(C)cccc2O)=O)CC2CC(NC(c3cc(Cl)cc(Cl)n3)=O)CC2C1 C(=O)(CCC(C)CC(=O)OC)N1C(CNC(C(C)=C(CC)C)=O)CC1 N1(c2c(C(C)=O)cccn2)CCC2(CC1)CC2(C)C(=O)NCc1sc(C)nc1C CCCC(CC1CCCCC1)C(=O)N1CCC(NC(=O)CCCSC)C(O)C1 c1(C(=O)NC2CN(C(CC(C(C)C)O)=O)CC2O)cc2ncccc2[nH]1 C(=O)(CC(C)(C)C(F)(F)F)N1CC(Cn2cc(C(C)(C)OC(=N)O)nn2)C1 N1(C(C2CC(C)N(C)CC2)=O)CC2CCC(N=c3[nH]c(C(F)F)nc(=N)[nH]3)C2C1 c1(C(=O)NCC(C)(C)NC(C2(C)CC2(Cl)Cl)=O)ccc(Cl)cc1 C1(NC(C(N2CCSCC2)C)=O)CC2CN(C(C3CN(C)CCO3)=O)CC12 c1(C2(NC(=O)C(N3CCSCC3c3nccs3)=O)CC2)cccc(C(F)(F)F)c1 C1(CC)CN(C)CCN1S(=O)(=O)c1nccs1.C(CC(C)C)(C(=O)N1CCCC1)N C(=O)(C1CCCc2cccnc21)N(CC(C)NC(c1cc(C)cc(F)c1N)=O)C CC(C)(C)CCCC(=O)NCC12CCC(CC1)N2C(=O)C(C1CCOCC1)F C1(CCC)CN(C(C2CC(F)(F)C2(F)F)=O)CCN1C(=O)CN1CCSCC1 c1(C(C(=O)NCC=C)N(CC(F)(F)F)CCC)cc(Cl)c(Br)c(Cl)c1 C1(c2cn(CCN(C)C)nn2)C2CN(C(=O)CC3OCCCO3)CC12 C1(C(N(C(C)C)CCNC(=O)Cn2nccn2)=O)CN(c2ccccc2)CCO1 C(=O)(CC(C)(C)COC(C)=O)NCCCCC(=O)N1CC(CCC#C)C1 N1(C(C2CCC(=O)N2)=O)CC(NC(c2ncccc2Br)=O)CC1C1(CO)CC1 Cc1ccc(C(N2CC=CC(NC(C3(C)CCN(C)C3=O)=O)C2)=O)nc1F C=C(Cl)CC(C(=O)NCCC1CC(=O)N(C)C1)NC(=O)CC1CCCCN1C n1(CC)nc(CCOC)nc1-c1ccc(Cn2ccnc2)s1.C12CN(C1)C2 CC(C)C(C(=O)N1CC2CC2(CNC(C2(C(C)C)CC2)=O)C1)n1cccc1 Cc1nc(CO)oc1C(=O)NCCN(C(c1cccc(CS(C)=O)c1)=O)C(C)C CC(C)C(C(=O)N1CCN(CCCNC(=O)CC(C)F)CC1)N(C)C C(CC(=O)N(C)CCCC(=O)NCCCNC(=O)C(F)C1CCC1)C.CO N1(C(C(c2cccc(C(F)(F)F)c2)C)=O)CC(NCc2csc(Cl)c2)C2(CC2)C1 N1(CCOC)CC(C(=O)NCC2CC2CNC(c2coc(Cl)n2)=O)CCC1=O c1(CNC(C(C2CN(C(C(C)SC(C)C)=O)C2)O)=O)ccc(F)cc1O C#CC1COCCN1C(=O)C(C)N(C(=O)Cc1cn(C)nc1C)C1CC1 N1(C(C2CCC(CC)O2)=O)CC2CCC(C1)N2C(=O)CC1CCOCC1(C)C c1(NC(=O)OC)noc(CCC(=O)NC)n1.C(C(=O)OC)(C1CCC1)OC Cc1c(C(=O)NC2(CCNC(C3CCC3)=O)CC2)ccc(F)c1F Cc1c(C(N2CC(CNC(c3ccco3)=O)CC2C)=O)cnn1C(C)(C)C O=C1CN(C(=O)Cn2cnnc2)C(C(=O)NC(C2CCOC2)CO)CN1 C(CCC(=O)N1CC(=C(F)CNC(c2ncsc2C2CC2)=O)C1)N(C(C)=O)C C1(CN(C(c2c(C)scc2)=O)C)CC(F)CN1C(c1cn(CC(F)(F)F)cn1)=O N1(CCNC2C(C)CN(C(=O)Cc3cnn(C)c3)CC2)CCc2sccc2C1 c1(C(=O)NCC2(C)CCCN2C(=O)CC2CC3CC3C2)c(N)cc(Cl)cc1F n1(CC)nccc1C(=O)NCCOCCN(C(=O)CC1(O)CCOC1)C C1(C(=O)NC2(CN(C)C)CC2)CN(C(c2ccncn2)=O)CC1C(C)C C(C(=O)N1CC(N(C(=O)Cc2nncs2)C)C1)(C(C)C)N(CC)CC N1(C(c2nc(C)oc2)=O)CC2CCC1CN(C(c1cnc(C)nc1)=O)C2 C1(n2cc(CNCCS(=O)(=O)CC(=O)O)nn2)COc2ccccc2C1 C1(C(=O)NCc2ccccc2O)CC=CCN1C(C1CCCCC1O)=O Cc1cnc(C(=O)N(C2CN(C(C3CCC(CCO)CC3)=O)C2)C)cn1 c1(C(N2C(CN(C(c3ccc(COC)o3)=O)C)CCCC2)=O)ccc(F)cc1N C12(CNC(CNC(C(CC)C)=O)=O)CC(CO1)N(C(=O)Cc1cc(CC)on1)C2 C1(C(=O)NC(CNC(C=C(CCN(C)C)Cl)=O)C2CC2)CCC2CC1CO2 C1(NC(CC2(N(C)C)CC2)=O)CCN(C(=O)Cc2cc[nH]n2)C1C c1(CC)ncc(C(=O)NCCNC(c2cc(C)sn2)=O)cn1 C(=O)(C#CC1CCCO1)NCC1N(C(c2cc(CCCCC)[nH]n2)=O)CC(O)C1 C1(NC(C2N(CC)CCOC2)=O)CCN(Cc2ncn(C)n2)CC1O C(CCC(=O)N(CC(C)NC(=O)CCCN1CCC1)C)OC(C)=O c1(C(=O)NC2C(NC(CC(C)CF)=O)CCC2)c(F)ccc(F)c1Br c1(C(N2CC(C)C(CNC(=O)CCCn3ccnc3)C2)=O)ccc(F)c(Cl)n1 C1(C(=O)NCC(CNC(c2ccc(-c3ccco3)s2)=O)O)CC(C2CCC2)C1 Cn1nc(C(=O)NC(CC2CCCC2)C(=O)NC2CCC(N(C)C)C2)cc1O c1(OC)ccc2cc(C(=O)NCC3CC3CNC(=O)CCC(C)OC)[nH]c2n1 C1(C(=O)NCCC(C)CCO)(CC)CCCN(C(C2CC3CC(=O)C2O3)=O)C1 c1(C(=O)NC2C(CC)CN(C(c3oc(C)nc3C)=O)CC2)ccc(S(N)(=O)=O)[nH]1 C(=O)(C(C)(O)C(C)C)N1CCC(COC)(NC(=O)CNC(c2ccncc2)=O)C1 C1(C(=O)OC)CCCC(OC(=O)NCC(C)(C)Cc2ccc(C3CC3)cc2)C1 CCC(C)(COC)C(=O)N1CCC(c2nnc(CNC(=O)C=CC=C(Cl)Cl)s2)CC1 CN1N=C(C(=O)NC2CN(C(C3CC3c3ccn(C)n3)=O)CC2O)CCC1=O c1(CC(=O)NCC2(NC(CC=C=C)=O)CC2)ccc(Cc2cccc(F)c2)cc1 C(=O)(C=CS(C)=O)C(C(COC)OC)=O.C1(N)COCC1SC O=C(CCCCc1cnn[nH]1)NCCCCNC(C1CCC(NC(N)=O)CC1)=O C1(C(C(=O)NCC(CC)NC(=O)Cn2ccc(C(F)(F)F)n2)C)CCCCCC1 c1(C(N2CCN(C(c3cccnc3)=O)CC2CC(F)F)=O)ccc2cccnn12 c1(C(N2CCC(CN(C(=O)C(C)(C)c3ccnn3C)C)C2)=O)cnc[nH]c1=N c1(NC(CC(C)NC(C2CCCC2)=O)=O)cc(=O)n(-c2ccccc2)n1C C1(C(=O)NCC(C)(C)NC(=O)CSCc2ccccn2)Cc2c[nH]cc2S1(=O)=O Cc1n[nH]c(C)c1CC(N1CC(NC(=O)CCc2nc(C3CC3)no2)CC1C)=O C(C(C(=O)NOCC(C)O)NC(C1CC(C)=NO1)=O)OC(C)C c1(CC)ncc(CNC)s1.C1(N2CCSCC2)(C)CCCC1 N1(C(CCC(C)SC)=O)CCCC(F)(CNC(c2ncccc2C2CC2)=O)C1 c1(CC)cc(C(=O)NC2CCN(C(C3CCC4(CC3)N=N4)=O)CC2C)ccc1F C1(CO)C(C)N1CC1CCOC1.C(C(=O)OC(C)(C)C)OC c1(C(=O)OC)cc(F)ccc1NC(=O)Cc1cccc(N)n1 c1(C(N2C(C)CC(NC(C3CCC4CC34)=O)CC2)=O)cc2ccc(F)cc2s1 Cc1nc(C(C)(C)C)[nH]c(=NC2CC(NC(=O)Cn3cc(C4CC4)nn3)C2)c1C C1(C(=O)NCC2CCC(CNC(c3ccns3)=O)CC2)CN2CCC1CC2 N1(C(C(CC)(C)O)=O)CCC2(CC1)CN(C(=O)CC1CC1C)CCO2 C1(C(=O)NCCc2ncn(CC)c2)C2CC3C(C2NC(=O)CCC2CC2)C13 N1(C(CCc2cc(C)on2)=O)CCC2CCCC12C(=O)NC1CCC2(CC2)C1 c1(C(=O)NCC2C(C)C2)cc2cc(Br)[nH]c2[nH]1 c1(CC)onc(C)c1C(=O)NCc1ccc(C(=O)NCC2CCOCC2C)o1 c1(C(N2CCC(F)(C(=O)NCCN3CCCCC3=O)C2)=O)ccc(SC(F)F)cc1 C12(CNC(=O)COC(F)(F)F)CCC(CN(C(=O)CC3CCC34CCC4)C1)C2 c1(N(C(CC)CO)C)ccc(S(=O)(=O)NCCCNN2CCCC(C)C2)cc1Br c1(OC)cc(C(=O)NC2CC2C(=O)Nc2cc(Cl)c(Cl)cn2)c(F)cc1Br N1(C(C2C(CC)N(C)CC2)=O)CCC2CCN(C(=O)C(C)OC)C2C1 C(=O)(CC(CCc1ccccc1)C(F)(F)F)NCCC1(NC(C=C(C)C)=O)CC1 C1(C(=O)NC(C)CN(C)C)CC2CCC(C1)N2C(=O)CCC(C)CN(C)C C(=O)(C1=NNC(=O)CC1)C(C(CCSC1CCCCC1CN)NC(C)=O)=O.C(N)(=O)N N1(C(CCOC)=O)CCCN(C(c2sc(CO)nc2C)=O)C(c2ccccc2)C1 c1(C(N2CCC(C)C2CNC(C2CC(F)(F)CS2)=O)=O)cccc(F)c1F C1(OC)CN(C(=O)CC2NC(=O)NC2=O)CC1NC(C1(CO)CCCC1)=O c1(OC)ccc(S(N)(=O)=O)s1.c12coc(c1)C(=O)OC2 CC1=NOC(C)(CNC(=O)C(C)(C)CN(C(=O)C(C)OCC2CC2)C)C1 C1(CC(=O)OCC)CN(C(=O)C(c2ccc(F)cc2)COC)CCN1CC(F)F CC(CCCCNC(C1CC(=O)N(C(F)(F)F)C1)=O)NC(C1(F)CC1)=O N1(C(C(C)OCCC(C)C)=O)CCC2CC1CN2C(c1cnc(C(F)(F)F)s1)=O N1(C(C=Cc2cn(C)nc2)=O)CC(NC(=O)C2=CC(C)(C)C2)CC12CCCOC2 c1(CCC(=O)Nc2n(C)ccn2)ccc(S(=O)(=O)N2C(C(=O)O)CCC2)cc1N C(=O)(C(C)CCCC(C)=O)NCC1OCCN(C(CC(CC)C)=O)C1 N1(C(c2nc(C)sc2C)=O)CCC2CCC12CNC(c1ccncc1Cl)=O C=C(C)C(CC(=O)N(CC(C)C(N1CCC(C)(N(C)C)C1)=O)C)OCC N1(CCC(=O)NCCn2cc(CNC(C(CC)(C)O)=O)nn2)CCP(C)(=O)CC1 c1(OC)ccc(C(=O)NC2CC2CNC(C2Cc3nccn3C2)=O)c(Br)c1F c1(N(CC(N2CCCC(NC(C(C)P(C)(C)=O)=O)C2)=O)C)ncnc2[nH]cnc12 C12CCCN(CC1)CCc1n[nH]cc1C(=O)NC(=O)C2.C1(CCO)CCS(=O)CC1 N1(C(CCN(C)CCO)=O)CCCCCCC1C(=O)N(CC1=CCCCC1)C1CC1 c1(C(=O)NC2CCCCN(C(CCC(=O)NC)=O)C2)c[nH]c2cc(C)ccc12 c1(C(N2C(CNC(C(COC)OC)=O)C(C)CC2)=O)cc2[nH]ccc2s1 Cc1cc(CCC(=O)NCCc2cc(C(N3CCCC3C(C)(C)O)=O)no2)on1 c1(C(=O)NC2CC3(CCN(C(=O)CSC4CC4)C3)C2)cc(Cl)c(F)c(Cl)c1 N1(C(CC2(N(C(C)=O)C3CC3)CC2)=O)CCCN(C(=O)C2=CCCC2C)CC1 N1(C(CC2(N(C)C)CC2)=O)CC(NC(c2cnc[nH]c2=N)=O)CC12CCOCC2 Cc1cccc(O)c1C(N1CC2CC(C1)N2C(C1CCCC(C)(C)C1)=O)=O C1(CC(=O)NC2CCCC(C(=O)O)C2)CCCCN1Cc1ccccc1 Cc1nc(C2CC2)ncc1C(=O)NCC1CCCC1NC(c1cnc(N)c(F)c1)=O NS(=O)(=O)CC(O)CNC(=O)NCc1ccc(N2CCCCC2=O)cc1 c1(OC)c(C(=O)N(C2CN(C(c3coc(O)n3)=O)C2)C)cc(Br)cc1F C1(C)(N)CCN(C(=O)C(N)=O)CC1.CC(C(=O)NCC(F)(F)F)NC(N)=O c1(C(=O)NC2CCC(C)(CNC(=O)CCSC(F)(F)F)C2)cc2c(s1)CCC2 c1(NC(N(C)Cc2ccc(CSc3nc(C)on3)o2)=O)ccc(Br)cc1 Cc1nscc1CC(=O)NCC1(C)CN(C(=O)CC2CCC(C)C2)C1 N1(C(CC2(CSC)CC2)=O)CC2CN(C(c3cc4cn[nH]c4cn3)=O)CC2C1 c1(C(=O)NC2CN(C(C3C(C(=O)OC)CC3)=O)CC2C)cc2cccc(C)n2n1 C1(O)(C(C)NC(c2cnc(CCC)s2)=O)CCN(C(c2[nH]c(C)nc2CC)=O)C1 c1(CC)nc(C)c(C(=O)N(C2CCN(C(=O)C(C)(CO)OC)C2)C)s1 Cc1cn2nnc(C(=O)NC3(CO)CN(C(C4CC#CC4)=O)C3)c2c(O)n1 C1(C)(OCC)CCCN(C(=O)CC2CCN2C(C2CCS(=O)CC2)=O)C1 c1(C(N(C2CCN(C(CCC=CCC)=O)C2)C)=O)ccc(C2CC2)c(Cl)c1 c1(CC)ccc(C(=O)NCCCC(C)(C)NC(C23CCCC2C3)=O)c(N)c1 N1(C(C(C)C2CC2)=O)CCC2CN(C(=O)C(n3cc([N+](=O)[O-])cn3)(C)C)CC12 C1(C(=O)NC2C3CCCOC23)(NC(C2=CC(C)(C)C2)=O)CC2CCC1CC2 CCC(C(C)C)C(C(=O)NCC1CCOC1)N(C1COC1)C.C1CCOC(=O)C1 CCC(CN(C)C)C(=O)N(CCC(=O)NC(c1ccccc1)CO)C1CC1 c1(C(=O)OC)cc(C(N2CCOC(CNC(c3nc[nH]n3)=O)C2)=O)ccn1 c1(OC)ccc(Cl)cc1C(N1CC2CC1CC2C(=O)NCc1ccc(F)cc1)=O C(=O)(CCCC(=O)N(C)C)N1CC(N(C(C(C)C2CCCC2)=O)C)C1 C1(C(C)C)CN(C(=O)COC2COC2)CCC1NC(=O)CC(F)F C1(C)(CNC(C2(C(N)=O)CCC2)=O)CN(C(c2cc(N)c(F)cn2)=O)CCO1 N1(C(CCOC)=O)CC2OCC(NC(c3ccc(Br)cc3Br)=O)C2C1 N#Cc1ccc(Br)cc1CN1CCSC(C(=O)Nc2cc(Br)cc3cn[nH]c23)C1 C(C(CNC(C1(n2cccn2)CCC1)=O)CO)NC(c1cccnn1)=O C1(CC(=O)NC(C2CCN(C(c3cccnc3O)=O)CC2)C)CC(C)(C)CO1 c1(OCC)nccc(C)c1C(=O)NC(CNC(=O)C(F)CC)CO C1(C)(C(=O)NCCn2ncc(C)c2)CCN(C(=O)C(O)Cn2cncn2)C1 C1(OC)CC(CNC(C2(F)CCOCC2)=O)N(C(C2CCCS2)=O)C1 N1(C(CCCNS(C)(=O)=O)=O)CCCC12CCCN(C(c1ccc(=O)oc1)=O)C2 c1(COC)cc(NC(=O)OC)no1.C1(C)CC(C)NC(=O)CC2(CCC2)C(=O)N1 N1(C(=O)C(C2(O)CCCCC2)N(n2ccnc2)CC2CCC2)CCCC(CF)C1 N1(C(CCC2N(C(c3c(CC)c[nH]c3)=O)CCC2)=O)CCOC(C2CC2)CC1 N1(C(c2c(CC)nns2)=O)CC(CNC(=O)C(CC(C)C)OCC)OC(C)(C)C1 N1(C(COCCN(C)C)=O)CCCCC1C(=O)NC1(CO)CCCCC1 Cc1nc2cc(CNC(=O)NCC3C=CCCCC3)ccn2n1 C1(NC(Cc2nnc(C)o2)=O)CCCCN(C(=O)Cc2[nH]cnc2C)C1 C1(NC(=O)COC(N(C(C(=O)NC)CC2CC2)C)=O)CCN(C)C1=O c1(NC(C(C)OCCN(C)C)=O)ccnc(C(=O)NC(Cc2cnc[nH]2)CO)c1 CC1(C(N2CCN(C(=O)CC3CC4(CCC4)C3)C(CO)C2)=O)CC2CCC(C1)S2 Cc1cc(C)c(NC(N2CCC3(CC3)C2)=O)cc1C Cc1cccc2c1OCC(NC(=O)NC(C)Cc1ccccc1OC(F)(F)F)C2 C1(CNC(C2(CC(C)C)CC2)=O)CCN(C(=O)CC2CCSCC2)C12CC2 CC1(C)C(C(=O)Nc2cccc(F)c2)CCN1C(c1ccncc1)=O C1(=O)CCNCC(=O)OCCO1.c1(C(N(CC(F)(F)F)C)=O)ccco1 c1(OC)cccc(CCC(N2CC3C(CNC(C4(C)CCC4)=O)C3C2)=O)c1 c1(C(=O)NCC2CCC(NC(C3CC=CCO3)=O)C2)ncccc1F N1(C(Cc2c(C)con2)=O)CC2CC(NC(=O)C3=CCCSC3)CC2C1 c1(CN2CC3(C(C(=O)NCc4cccnc4Br)C3)C2)c(F)ccc(F)c1Cl C#Cc1cc(F)c(C(=O)NCC(C)NC(C23C=CC(CC2)C3)=O)cc1F c1(C(=O)NC(C2CCCN2C(C23CC(F)C2C3)=O)C)cccc(-n2ccnn2)c1 N(C)(C(=NCc1ccc(C(C)(C)C)s1)Nc1cccs1)CC1CC(OC(C)C)C1 CON(Cc1ncc[nH]1)CC1CCCCO1 Cc1ccc(N(C)C(c2sccc2CNC(C2CCCO2)=O)=O)cc1F Cc1c(CNC(C2(c3ccccc3)CC2(F)F)=O)cccc1Cl C(=O)(C(CNC(C1CCN1C)=O)CC1CCCC1)N(CCN(C)CCO)C C=CC(C(F)(F)F)NC(=O)C(Cc1ccco1)NC(=O)Cn1cccn1 c1(OC)cc(CC(N2C(C)C3CC2C3NC(C2(CO)CC2)=O)=O)cc(Cl)c1 C1(F)(C(N(CCC(C)NC(c2ccc(NC)cn2)=O)C)=O)CCC(C)(C)CC1 Cc1nc(NCCN2CCN(C(C3C(C)CC3C)=O)CC2)c(C)c(O)n1 c1(CC(=O)NC(C(=O)NCCOC)C2CCCC2)cnn(C(C)(C)C)c1Cl N1(C(C2N(C(C3N(C)C(=O)CC3)=O)CC(O)CC2)=O)CC(C)(C)OC(C)(C)C1 C1(N(C)C)CCCN(N2CCN2CCN2CCCC2C)C1 C(=O)(CC(C(F)(F)F)c1ccccc1)OC(C(=O)N(CCC)C(C)C)O CC1OC2(C(N3CCCC3(C)COC(=O)Nc3ccccc3)=O)CC1C2 N1(C(COCC)=O)CCN(c2ccccc2CNC(=O)CC2CCC(=O)N2)CC1 C1(NC(CC(=C)C)=O)CCC2(CC1)CN(C(=O)COCc1nc[nH]n1)CCO2 N1(C(c2cc(CC)ncn2)=O)CC2C3C=CC(O3)C2C1.C12CCC(C1)CC(=O)N2 Cc1ncccc1-c1cn(CC2CCCC2NC(=O)Cc2cnn(C)c2)nn1 C(=O)(CCCCCC(C)C)N(CCN(C(c1c(C)cc(C(=O)OC)o1)=O)C)C(C)C C12CC13CCN(N1CC(C(O)C1)SC2)CC3.c1(OCC)ccccc1 N(C(=NCC(CO)C(C)C)NCC(F)F)C(c1cnn(C)c1)C C1(NC(CC(CC)SC)=O)C2CCC1N(C(c1cccnc1SC(C)C)=O)C2 C1(CNC(c2n(CC)ncc2)=O)C(C)CCN1C(c1nc(C)cs1)=O Cc1cc(F)cc2c(=O)c(C(=O)NCC(CO)NC(=O)C=CC3CC3)c[nH]c12 N1(C(c2coc(Cl)n2)=O)CCC(CNC(C2(CC(F)F)CC2)=O)C(F)(F)CC1 N1(C(CCOC)=O)CCCC(C)(OCCCNC(C(CC)CN(C)C)=O)C1 CCCC(CCC)C(=O)NC1CCN(C(=O)Cc2csc(C3CC3)n2)C1(C)C c1(C(=O)NC2(C(F)(F)F)CC2c2ccccc2)ccc2c(c1Cl)OC(F)(F)O2 C1(CNC(C2CC3CCC2C3)=O)CCCN(C(C2CCC(CF)C2)=O)CC1 C1(NC(=O)CCOCCOCCO)CCN(C(=O)C=CC2CCCC2)C1 O=C(N=c1[nH]nc(-c2ccccc2)s1)c1ccc(=O)n(-c2ccc(I)cc2)c1 C(C(C(=O)NC1CC(C(F)F)C1)C(C)C)NC(c1c(CC)n(C)cc1)=O CCC(CNC(=O)C(C)=CC1CC1)(CC)C(=O)NC(c1ncccc1F)C Cc1cc(C#N)ccc1NC(N1CC(CNS(=O)(=O)c2cnoc2C)C1)=O CC1CN(C(=O)C(F)=CC2CC2)CCC1NC(=O)CCCc1ccccc1Cl c1(OC)cc(Cl)c(Cl)cc1C(C)NC(=O)NCc1ccccc1-c1n[nH]c(C)n1 C#Cc1ccc(NC(C2CCOCCN2C(c2ccoc2CC)=O)=O)c(C)c1 CC(C(C)(C)C(=O)NC(c1nc[nH]n1)C1CC1)NC(C1CC=CC(O)C1)=O C1(CNC(C(CC)SC)=O)CN(C(c2ccccc2OC2CC2)=O)CC1O C1(C(N(CCCNC(=O)CCC2CCCN2C)C)=O)CCCC(F)(F)CC1 C1(C(=O)NCC(C(C)C)NC(c2csc(O)n2)=O)Cc2cc(Br)cnc2C1 c1(C(N2C(CNC(C3C(CCC)C3)=O)CC(F)(F)C2)=O)c2c(nn1C)CCOC2 C(CCC(C)(C)C(=O)NC1CC=C(C)CC1)NC(C(CCC)C#N)=O c1(N(C2(CO)CNC2)C(C=Cc2cnc(C)s2)=O)ncc2c(n1)CCC2 c1(N(C(C)C)C)ccc(SCc2ccc(F)nc2)c(N)c1 CCCC(C)CC(C(=O)NCC)N1CCN(C(=O)CCC(C)=O)C(C)C1 N1(C(c2cc(C)oc2C)=O)CC(C)OC2(CCN(C(c3nccs3)=O)C2)C1 c1(C(N(CC(CC)NC(=O)CSCCC#N)C)=O)nn(C2CCCCC2)cc1C C(CCNC(=O)C(O)CCc1ccccc1)(C(C)C)NC(C(C1CCC(C)O1)=O)=O C1(OC)CCC2CN(C(=O)NC(C)C(c3ccc(Br)cc3)C)CC12 Cc1cc(C(N2CCCC2CCCNC(c2ccc[nH]2)=O)=O)nc(Cl)c1 N1(C(C=CSC)=O)CCCN(C(=O)C2=NOCC2)C(C)C1.c12cn(nn1)C1CCC21 C1(NC(c2cn(CC)nn2)=O)CC2(C1)CC2C(=O)NC1CCCC(C)C1 c1(C(=O)OC)ncc(S(=O)(=O)NC2CCN(S(C)(=O)=O)C2)n1C c1(OC)cc(C(C)(C)NC(C2CCCC2n2cc(COC(C)C)nn2)=O)sn1 N1(C(CC(C)n2cccc2)=O)CC(NC(c2ccc([N+](=O)[O-])o2)=O)CC1(C)C C(=O)(C#CC1CCCCC1)N1CCN(C(C2C(C)(C)C2)=O)CC1CCO C(=O)(C#CC1(C)CCCO1)N(C(=O)C(C)OC(Cc1c(C)n[nH]c1C)=O)C(C)C C1(C)(NC(CC2(N(C)C)CCC2)=O)CC(NC(C2(c3ccncc3)CC2)=O)C1 N1(C(C2C(C=C)C2)=O)CCCN(C(=O)Cc2n[nH]c3ccccc23)CC1C CC1CC(NC(c2ncncc2F)=O)CN1C(c1cnc(-c2cccs2)s1)=O c1(C(=O)Nc2ccc(OCF)cc2)ccc2cc(O)c(C(=O)Nc3ccsc3)cc2c1 N1(C(C=CC)=O)CCC(CNC(=O)C(C)(C)C2CCCCO2)C(C)C1 c1(C(N2CCC(C(=O)O)(COC)C2)=O)cc2ccccc2n1C C12(NC(C(CCSC)OC)=O)CCCC1N(C(c1cc(F)cc(F)c1)=O)CCC2 Cc1nc2cncc(C(=O)NCC3(CNC(=O)C(C)C(C)C)CCCC3)c2[nH]1 c1(CC(=O)NCC23CCCC2CN(C(=O)CC2CCC2)C3)c[nH]c2cccnc12 c1(C(N2CC(CN(C(c3c(OCC)scn3)=O)C)C2)=O)ccc(I)cc1O N1(C(CC(C(C)C)O)=O)CCC2(C1)CN(C(=O)CCc1cccs1)CCO2 N1(C(CC(=C=C)C)=O)CCCC(O)(CN(C(=O)CCc2cnccn2)C)C1 C1(CC(N2CC(CNC(C(C)(F)F)=O)C2)=O)CCC2(CCC2)CO1 Cc1ccc(OCC(=O)NC2CCC2CNC(=O)CC2CC2)cc1 c1(C(=O)NCC23CC(NC(C(C=C=C)C)=O)(C2)C3)cccc(N)c1O C1(C(N(CC(O)CNC(c2ccc(C#N)s2)=O)C)=O)CC12CCCCC2 N=c1[nH][nH]c2ccc(C(N3CCCC(c4cccc(C(=O)O)c4)C3)=O)cc12 c1(OC)ccc(SCCC(=O)NCC2CC(C)N(C(c3oncc3C)=O)C2)cc1 N1(C(C(C)S(N)(=O)=O)=O)CCC(C(=O)N2CCCC(C)(C#N)C2)=C(F)C1 CC1(C)CCOC1CC(=O)NC1CC(NC(=O)CC2CCCCCC2)C(O)C1 c1(C(=O)NC(C(C)NC(C(C)NS(CC)(=O)=O)=O)(C)C)cnc(=N)[nH]c1 Cc1ccc(Cl)cc1N1CCN(Cc2cn(CCc3cncnc3)nn2)CC1 C(=O)(CCC(F)(F)Cn1cc(-c2ccc(Br)cc2OC(F)(F)F)nn1)NC(C)C N1(C(c2c(C)nc(O)[nH]2)=O)CCCN(C(C2CCCO2)=O)CC1C(C)C CC(C)CC(C(=O)NC12CCN(CC1)C2)N(C(=O)C(C)NC(N)=O)C C1#CCCC(O)CCCCC1=O.OCCN c12cccc(c1)C(=O)N1CCCCC1N2.N1(CC)CCC(CN(C)C)CC1 C1(NC(C=NOC)=O)CCN(C(=O)CC(C)N2CCCC2=O)CC1 C1(CC(=O)N(C)CC2OCCC2(C)C)CCCN(C(C2CCN2C)=O)CC1 Cc1nc(C(=O)NC(C)(C)CNC(=O)C(C2CCOCC2)F)c(C)n1C C(CCC(C)C(=O)NC1CN(C(=O)C(F)CC2CCOC2)CC1(C)C)OC N1(C(C2N(C(C(CC(C)C)OC)=O)C3CCC2C3)=O)CCc2ccsc2C1 N(C1c2ccccc2CC1NC(C1CCN1C1CC1)=O)C(C(C)(C)C1CCOC1)=O c1(C(N2C(C)CN(C(c3c(C)ccs3)=O)C(C)C2)=O)cnc2cnc(Cl)cc2c1 S(=O)(=O)(c1cnn(C)c1)NC(C(CSC)O)C.C(C)(C)(C)SC C(=O)(N1CCC(C(=O)NCC23CCCC(CO2)C3)O1)c1cc(COC)ncc1 c1(C(=O)NC2(CO)CCCN(C(CC(CC)C)=O)C2)nc2cccnc2s1 c1(CN2CCC(C)C(NC(c3ccc(F)c(Cl)c3)=O)C2)cn(C)c(=O)nc1O n1(CCC(=O)N(C(C)CN(C)C(c2nc(Cl)cs2)=O)C)cnc2sccc2c1=O N1(C(C(CCCC)O)=O)CCN(C(C2CCN(S(N)(=O)=O)CC2)=O)C2(CCC2)C1 c1(C(N2C(C(=O)NCCC3CCCCCC3)CC(=O)C2)=O)cncc2[nH]ccc12 CCC(Cc1cccc(C)c1)C(=O)NC(CNC(=O)C(F)=CCCF)CO N1(C(C(C)=CC)=O)CC(C)(CNC(=O)Cn2cc(C(F)(F)F)cn2)CC1(C)C c1(CC(=O)N(CC(CC)NC(=O)CC(F)(F)C(F)F)C)ccc2[nH]ccc2c1 N1(C(C(CCC)C)=O)CCN(CCN(C)CCNC(C)=O)CCC1C C1(NC(CC2COCC(C)O2)=O)CCN(C(c2ccnc(SC3CC3)c2)=O)C1(C)C C1(Nc2snc(C)c2C#N)CCC2CN(C(c3sccc3F)=O)CC12 C(=O)(C1=CCC(NC(=O)CSC2CCC2)C1)N(CCCF)C c1(OC)c(I)cc(NC(N2CCC(CC3CCCC3)C2)=O)cc1I n1(CC(=O)NC(CN(C(C(C)OCOC)=O)C)C)ccnc1C Cn1c(C(N2CC3CC(NC(=O)CCCc4ccncc4)C2C3)=O)cc(Cl)c1Cl S(=O)(=O)(c1cccnc1NCCc1ccco1)NC(c1nc2c(s1)CCC2)C c1(C(=O)NC2(C)CC(NC(CCC=C)=O)C2)cccc(N2CCCCC2)c1 c1(CCC(N2CCCC(C(=O)NCc3cc(OC)no3)C2)=O)ccc(Cl)c(Cl)c1 CN1CCCC12CN(C(C1(C)CCCN(C(C3C4CC5C(C4)C35)=O)C1)=O)C2 C1(O)(CNC(CN2C(C)CCC2)=O)CCN(C(=O)C=CCF)C1 C(CC(C)C(=O)NC(c1cnn(C)c1)C(=O)NCc1n[nH]c(C)n1)=CC c1(C(N2CCN(C(COC)C)CC2)=O)ccc([N+](=O)[O-])cc1C C1(C(N(C2CCCC(NC(=O)C=CC(=O)N(C)C)C2)C)=O)CC(C)(C)CCO1 N1(C(C(c2ccc(C)cc2)=O)=O)CCC(NC(=O)C(C)(C)c2ncco2)C(F)C1 c1(C(N2C(C(C)C)CN(C(=O)C=CC3CCCC3)CC2)=O)cc2c(o1)CCCC2 c1(C(=O)NCCC2N(C(c3c(N)nccc3)=O)CCOC2)cc(F)cc(F)c1 c1(OC)c(F)cc(C(=O)NCCC(O)CNC(c2sccc2C)=O)c(N)c1F c1(CC)cc(C(=O)NC(CNC(=O)C(F)F)CC)c(C)nn1 N1(C(C2(CC)CCCN(C(C3OC4CCC3C4)=O)C2)=O)CCC12CCCCC2 c1(SC)ccc(N)cc1C(N1CC(CNC(=O)C=Cc2ccc(C)o2)C(C)C1)=O c1(C(N2CCC(F)(C(N3CCCC(O)C3)=O)CC2)=O)occc1C1=CCNCC1 c1(C(N2CCC(CNC(c3c(F)ccc(C)n3)=O)C2)=O)cc2c(nn1)CCCO2 C(CC(C(C)(C)C)N(C(=O)CCOCCC)C)NC(CCC=C=C)=O N1(Cc2cccc(OCC)c2O)CC2(CCC(C(=O)NC(C)C#N)O2)C1 c1(C(=O)OC)cc(NCCNC(=O)C(C)CN2CCOCC2)cn1C C1(CC)CCCC(CNC(C2C3CCC2(c2cscn2)C3)=O)C1 N1(C(CC=C)=O)CCOC2(CCC(NC(c3ccc(S(C)(=O)=O)cc3)=O)CC2)C1 Cc1noc(Cl)c1CC(=O)N(C(CNC(C1CCCC(=O)O1)=O)C1CC1)C c1(C(N(CCCCN(C(CC2CC(OC)C2)=O)C)C)=O)cc(C(C)(C)C)n(C)n1 c1(C(=O)OCCC23COC(Cc4ccc(CO)cc4)(C2)C3)cccc2scnc12 C(=O)(C1CCCc2ccnn21)N1C(CNC(c2c(CC)onc2)=O)C=CC1 c1(NCC(=O)N(CC(C)C)Cc2cn[nH]c2)ccc(-c2cncc(N)c2)cn1 c1(OC(C(=Cc2cn[nH]c2)C)=O)noc2c1CC(C)CC2 C12(CNC(N(CCCC)Cc3ccccc3)=O)CC(CN1C)C2 C1(C(N2CC(C)(CC=C)C2)=O)CCOCCN1C(C1CC(SC)C1)=O C(=O)(C(C)(C)S(=O)(=O)C1CC1)N1CCCC(NC(C(CCC)NC(C)=O)=O)C1 N1(C(C(C)(C)OCC)=O)C2CC1CN(C(C1CC13CCOC3)=O)C2 c1(C(=O)Nc2cc(CCOC)no2)[nH]c2ccccc2c1CSC c1(C(N2CC(CCNC(=O)Cc3cncc(F)c3)C2)=O)noc2ncccc12 c1(C(=O)NCCCCC(CO)NC(CC(C)OC)=O)cccn2cnnc12 S(=O)(=O)(CC(=O)NC1CCCC1C(N1CCC(CO)CC1)=O)NC C1(OCC)CCN(C(=NC)NCc2cc(OC)ccc2Br)C1 C12(NC(Cc3ccn(C)n3)=O)CC1CN(C(c1csc(Cl)n1)=O)C2 c1(C(N(CCN(C(=O)C(O)c2cnc[nH]2)C)C)=O)nncc2c1CCCC2 C1(NC(C)=O)CC2(CCC(CNC(c3cscc3C)=O)OC2)C1 N1(C(CC(C)OC)=O)CCC2(CC1)OCCCC2NC(=O)CNC(=O)CN(C)C C1(C(=O)NCCCCC(N)=O)C2CC(O)C(C2)N1C(=O)C1=CCCOCC1 c1(COC)ccccc1C(N1CC2CC2(NC(=O)C2=COCC2)C1)=O C1(NC(=O)Cn2cnc(Br)c2)CCCN(C(=O)C(F)(F)C(F)F)CC1 C#CCCCCCCCC(=O)NC(C)(CNC(C1(O)COC1)=O)C(C)C Cc1nc(C(N2CCC2CNC(=O)Cc2ccno2)=O)n[nH]1 c1(-c2cn(C(C(=O)OC)C)nn2)ccccc1CNC(c1cc(Br)n[nH]1)=O C1(CCNC(COC(CC)(C)C)=O)CCCN(C(C2CCO2)=O)C1 CN1CCC(CCNC(C2(NC(C3SCCS3)=O)CC2(C)C)=O)CC1 C1(C(N(CC=C)CCc2ccccc2)=O)COC2(C1)CN(C(=O)NC1CC1C)C2 c1(C(N2CCC(OCCNC(C3SCCS3)=O)C2)=O)cc(O)cc(F)c1 C1(CC=C)(NC(c2ccc(Cl)nc2)=O)CCN(C(c2cncc(C)c2)=O)C1 CC1(C)CC(CNC(=O)Cc2ccn(C(F)F)n2)CN1C(c1c[nH]ccc1=O)=O O=C1C=C2CN(C(=O)C(N)Cc3csc4ccccc34)CCC2S1 N1(C(C2C(=C)CC2)=O)CCCC(O)(CCNC(c2ccccc2OCC)=O)C1 C12(C(=O)NC3C(NC(C(C(C)(C)C)O)=O)CCC3)CC3CC(C1)CC(F)(C3)C2 c1(-c2onc(COc3c(CC)ccc(F)c3)n2)cc(F)cc2cc[nH]c12 N1(C(CCC2C(C)C2)=O)CCC2(CC(NC(c3ncc[nH]c3=O)=O)C2)C1 c1(C(=O)NCC2C3N(C(CC(CC)SC)=O)C(CC3)C2)c(N)cc(F)cc1Cl c1(NC(C2CCN(C(c3cccc([N+](=O)[O-])c3)=O)CC2)=O)cccn2nccc12 C#Cc1cccc(OCC(=O)NCC2CC2CNC(c2cnnn2C(C)C)=O)c1 c1(C(=O)NC(C(C)NC(=O)CCCn2cccc2)(C)C)cc2c(s1)CCCC2 C1(C(=O)NCC(C(=O)NC)(C)C)CCN(C(c2n[nH]c(=N)[nH]2)=O)C12CCC2 C1(CC(=O)NC(CC)Cn2cncn2)CCN(C(=O)CC(C)(C)C)CC1(C)C N1(C(c2nc(OC)sn2)=O)CCN(C(=O)CCc2nc(O)n[nH]2)C(CSC)C1 c1(C(=O)NCC2(F)CN(C(CNC(CN(C)C)=O)=O)C2)cc2cc(F)cc(F)c2o1 CC1CN(C(C2CCSC(C)C2)=O)CCN1C(=O)Cc1cccc(C(N)=O)c1 CC1CC(F)(F)CCN1C(C1N(C(c2ccc(F)c(O)c2)=O)CCC1(C)C)=O N1(C(CC2C(NC(COCCC#C)=O)CC2)=O)CCCCC(OC)C1 N1(C(c2cc(C)n(C(F)F)n2)=O)CCCC(C)C1CNC(C=CCN(CC#C)C)=O c1(C(c2nnnn2C)NC(C=C)CC)ccc(OC(F)F)c(F)c1F C(CC)(CC(=O)N(CC(C)N(C)C(C)=O)C)N(C(C=CCCC=CC)=O)C C1(CC(=O)NCC2(NC(C3CC3F)=O)CC(F)(F)C2)CC2(CCC2)C1 C(=O)(C1=C(Cl)CCC(C)C1)NCCN(C(CC(C)OC)=O)C1CC1 N1(C(COCCNC(C(COC)OC)=O)=O)CCC(SC)CC1 c1(C(N(C(C(=O)OC)C)C2CC2)=O)sc(-c2cnccn2)nc1C N1(C(CCCOC)=O)CC(NC(=O)C(COC)NC(=O)OC(C)(C)C)CC1(C)C N1(C(c2cnn(C(F)F)n2)=O)CCC(C2CCCCN2C(C2CCOC2)=O)CC1 N1(C(c2c[nH]c(=N)s2)=O)CCOC2CN(C(=O)Cc3ccc(Cl)cc3Cl)CC12 C(=O)(C(C)CC(F)(F)F)N1CCN(CC(C)NC(C(CCOC)C)=O)CC1 C(=O)(C=CSc1nc[nH]n1)N(CCCCN(C(=O)CCN(S(C)(=O)=O)C)C)C CC1SCCCC1C(N1CCN(C(=O)CC2(C)CCC2)CC1)=O N1(C(c2c[nH]c(=NC)s2)=O)CCC2(CC2C(N2CCCC(C)(CCO)C2)=O)C1 C(=O)(C(C)(CO)NC(c1cccc(OC)c1)=O)NC(C#CCC)(C)C N1(C(CCN(C(=O)CC(C)(C)OC)CC=C)=O)CCC(F)CC1 C(CNC(=O)Cc1ncc(C)s1)(CC(C)C)NC(C(C)NC(CC)=O)=O C(CCC(=O)N1CCNC(=O)C2(COC2)C(C)S1)OCCCC.C1CC(C)O1.CC C1(C(=O)NC2(CO)CCN(C(C(CCOC)OC)=O)C2)CC2(C1)NC(=O)NC2=O c1(C(N2CCC(C(C)NC(C(CC(C)C)=O)=O)C2)=O)cn2cccnc2n1 CN1CCN(Cc2cccc(-c3coc(C#N)c3)c2)CC(F)(F)C1 Cc1cc2ccc(C(=O)NC3CC3CNC(c3cnnn3C3CC3)=O)cc2o1 C(C(O)C(=O)N(CCNC(=O)NC1CC1)C1CC1)=CC.C(C)(C)(C)CO C1(N(CC#C)C(C2(n3cc(Cl)cn3)CC2)=O)CCN(C(C2(CC)CCCO2)=O)CC1 Cc1cc(C(=O)NCC(C(C)C)NC(=O)CC2CC=CCN2C)c(C)n1C C1(NC(C(COC)OC)=O)CC2(CCCCN2C(=O)CC2CCCNC(=O)C2)C1 CC(C)CC(C(=O)NC1CC(NC(C23CC(C)(CCO2)C3)=O)C1)C(N)=O C1(C#C)(C(=O)N(C2(CC#C)CCCCC2)C2CC2)CCN(C(=O)C=CC(F)F)C1 C1(C(N(CCOCCCN(C(=O)CN2CCNC(=O)C2)C)C)=O)CC2CC(=O)C1C2 c1(C(=O)NC(C(C)NC(=O)C(CO)NC(N)=O)(C)C)sccc1-c1ccccc1 c1(CC(=O)NCC(O)CNC(C2CC2C2CCOCC2)=O)ccc2c(c1)CCO2 CCC(C(=O)NC1CCCN(C(=O)CCn2ccnc2)CC1)C(F)(F)F N1(C(C2CCC(C)(CC)O2)=O)CC2CC(C1)CN(C(C1(O)CCSCC1)=O)C2 C12(CNC(c3ccnc(-c4ccccc4)c3)=O)CC(CN1C(=O)CC1CCC1)C2 c1(CNC(C=NOC)=O)cnc(-c2cn(CC3(F)CCNC3)nn2)nc1 N(C(=NCc1ccc(F)cc1)N1CCCC(C)C1)C1CCN(S(CC)(=O)=O)C1 N1(C(C(C)O)=O)CC(NC(=O)Cc2ccn(-c3ccc(Br)cc3)n2)C2CC2C1 C=C(Cl)CC(C(=O)NCc1ccc(Cl)o1)NC(=O)CC1(O)CCC1 N1(C(CCNS(C)(=O)=O)=O)CCN(C(=O)CS(C)(=O)=O)CC(CO)C1 N1(C(c2ccc(OC)c(Br)c2)=O)CC(C(=O)O)C2(C1)CN(C(=O)CC(C)O)C2 C1(CCC(=O)NCCC(=O)NC(COC(C)C)CO)CCN(C)C1 c1(C(N(C2CCN(C(CCC(C)CN(C)C)=O)C2)C)=O)cccc2nc[nH]c12 CC1(C)C(CC(=O)NCC(F)(F)CO)CCN1C(C1CC2(CC2)CO1)=O C#Cc1ccc(C(N2CC3CC3(NC(c3cn(CCC)nc3C)=O)C2)=O)o1 C(CN=C(NCC(Br)=C(C)C)N1CCC(C(C)C(=O)NC(C)C)C1)OC C(C)(C)(C)NC(=O)NC.C1(N(CC(C)C)C)CC(CN)C1.C(C)(C)(C)C(=O)O CC1(C(N2CCN(C(=O)CCOCC(F)F)CC2)=O)CC2C=CC1C2 CC1=C(C(=O)NCCCNC(=O)C#CC2CCOC2)CCCC1 c1(OCC)ncccc1C(N1CC2CC2(NC(=O)CC(C)C2CCCC2)C1)=O Cc1cccc2c1CN(C(C1(NC(=O)CNc3ccccc3)CCN(C)C1)=O)C2 C1(NC(=O)Nc2cccnc2)CCCCN(C(=O)C(F)CC2CCCC2)C1 c1(C(=O)NCCCC(C)NC(C2(C3CC3)CCOCC2)=O)cncc2nc[nH]c12 c1(C(N(C)CC2CN(C(Cc3cnc(C)o3)=O)C2)=O)c(Cl)nn(C)c1Cl N1(C(CC(=O)NCC)=O)CCCCC(NC(c2cn(C)nc2COC)=O)CC1 C12(C(=O)NC(C)CC(C)NC(=O)Cn3nnc(C4CC4)n3)CCCC(C)(C1)OC2 C(C(CCO)NC(=O)CC1(C)CCN1C(=O)C1CC1)N(C)C CC(C)(O)C(C(=O)Nc1cncc(F)c1)NC(=O)CCn1ccnc1 CCCCC(C)C(=O)NCc1ccc(C(=O)NCC2CC(C3CC3)=NO2)s1 c1(C(=O)NC2CC(NC(C3CCN(C)C3)=O)C2)cccc2c1nnn2C n1(CC(=O)N(C(C)CNC(=O)Cc2ccnn2C)CC)nnc(-c2cccs2)n1 C12(C(=O)NC3C(NC(c4ccc(COC)cc4)=O)CCCC3)CC=CCN1CCC2 c1(C(N2C(C)(C(N3CCC(OC4CC4)C3)=O)CCC2)=O)n[nH]c2c(Br)cccc12 c1(SC)cc(Br)ccc1ON1CCCC(n2cc(Cn3nccc3C#N)nn2)C1 C1(CNC(C2(C)CCCOC2)=O)Cc2ccccc2CN1C(=O)CCn1cnnn1 CC1(CNC(=O)Cn2[nH]cnc2=N)CCCN(C(C2(C(F)F)CCCO2)=O)C1 C(C)(C(C)(C)C(=O)NC(C1CCCC1)C)NC(C1CC(C#N)(OC)C1)=O NS(=O)(=O)c1n[nH]cc1C(=O)NC1C=CCN(C(=O)CCF)C1 CC1OC2(C(N3CCC(CN(C(=O)C(C)OC(C)(C)C)C)CC3)=O)CC1C2 C1(C(N2C(CNC(C(COC)C)=O)COCC2)=O)CCOC(C)(C)C1 Cc1csc(=O)n1CCC(=O)N(CCCN(C(=O)CC1CCOC1)C)C N1(C(CCOCCSC)=O)CCN(C(=O)Nc2cnn(C)c2)CC1C1CCCC1 C12(C(=O)NCC3CCCN(C(c4nc(C(C)C)sc4)=O)C3)CCOC1CCOC2 CC(C(=O)NC1(CO)CN(C(c2sccc2Cl)=O)C1)C(C)C(C)(C)C c1(OC)ncc(Cl)cc1C(=O)NC(C)C(C(C)C)NC(=O)CN1CCCNC1=O C(CC(O)C(=O)NC1COCCC1NC(=O)CCc1cnc(O)[nH]1)SC c1(CCCOC)ccc(Cl)c(F)c1.n1(CCCSC)c(N2CC3CCCC23)nnc1C C=C(CNC(=O)C=CC(C)(C)SC)CCNC(=O)C(O)Cc1cnc[nH]1 C(=O)(C(CNC(=O)C=Cc1ccncc1)C(C)(C)C)NC1C(CC(C)(C)C)C1 C1(C(N2CCC(OCCSCC(=O)NC3CCCO3)CC2)=O)OCC2CCCC12 C1(CC(=O)NC(C(C)NC(CC2N(C(C)C)CCC2)=O)(C)C)CCCOCC1 C1(C(C)=O)C(C(=O)N(C)CCN(C)Cc2cn(C3CCOC3)nn2)C1(C)C c1(OC)cncc(C=CC(=O)NC(CNC(=O)CN(C)C(C)=O)CC(C)C)c1 c1(C(=O)NC2C(NC(C3CCC(C)(F)CC3)=O)C2)c[nH]c2ccc([N+](=O)[O-])cc12 C#CCC(C)(C(=O)N(C)CC1(C#N)CCC1)NC(=O)C(CN(C)C)C(C)C N1(c2nc(CC(C)C)on2)CCC(O)(C(=O)NCC(C)(C)C2CCCC2)CC1 C(C(CC(=O)NCCc1cccc(O)n1)C1CCC1)NC(Cc1cc(C)sc1)=O c12ccc(c(C(F)(F)F)c1)[nH]c2=O.C(=O)(COC)N(CCOCC)CC C(CC(C)C)(C(=O)NC(CO)C1(O)CC1)NC(C(C=C)C)=O N1(C(C(C)(C)C2CCCC2)=O)CCC(O)(CNC(=O)Cc2ccc(C(C)=O)s2)C1 c1(C(N(CC(C)O)CCNC(c2cc(COC)[nH]n2)=O)=O)cncc2c1CCC2 C1(CC)C(C(=O)NC(C23CCC(CC2)C3)C)CCN1C(c1cnc(C)s1)=O C1(NC(CCCOCC=C)=O)CC2CC1CN2C(=O)CCCc1csc(C)n1 C12(C(N(C)CCNC(=O)CCc3nccs3)=O)CC(CN1C1CC1)C2.C1CCCO1 c1(O)ccc(C2(C(CCC)=O)CC2)cc1.c1(CC2CCCN2C)ccc(CSC)cc1 c1(C(=O)NC23CC(CNC(c4n(CC)ccc4)=O)(C2)C3)ccc2nnc(C)n2c1 C1(S(C)(=O)=O)(C(=O)NCC(CN(C(C2CCC(C)S2)=O)CC)(C)C)CC(O)C1 C1(C(N2CCC(C(C)NC(CC=CCC)=O)C2)=O)CCC(NC(C)=O)CC1 C=CCCC(C)(C)C(=O)N1CCCC(C(=O)NOCc2ccccc2F)C1 C1(NC(COCC(=O)NC)=O)CN(C(C2(CSC)CCC2)=O)CCC1C C1(NC(c2scc(OC)c2)=O)CCN(C(=O)C(c2ccccc2)C2CC2)CC1 N1(c2c(C)cccc2)CCCC(NC(c2cccc(CN)n2)=O)C1=O CCCC(C(=O)N(c1ncc(COCCO)s1)CC)COc1ccc(OCC)cc1 C1(C(N2CC(CC(=O)OC)C2)=O)(NC(C2CCCOC2C)=O)CCN(C)C1 C(=O)(CC(C)P(C)(C)=O)NCC(C)NC(C1(C)CC(=O)N(C)C1)=O C(=O)(C1=CCCCO1)N1CC(CNC(C(C(C)C)n2cccc2)=O)C(O)C1 Cc1ccn2nc(C(=O)NCCCN(C(=O)CSc3ccc(F)cc3)C)nc2n1 c1(COCCCNC(C(C)C2CCCO2)=O)nnn(C)c1C(=O)NC1CCCC1 Cc1csc(C)c1C(N1CCC1CNC(=O)C=CCn1cncn1)=O CC(C)C(C(=O)NC1(C)CCC1)NC(c1ccco1)=O.n1(CC(=O)N)ncnn1 N12CCCC(CC1)NC(=O)C2.O(COCCOC(C)C)CC C1(C)(Nc2nccc(CC)c2)CCCN(C(=O)C(C)S)C1 c1(CCC(=O)NCC(C)CN(C)C(c2cnn3ccsc23)=O)cc(F)ccc1F CCC(C(=O)N1CCC1CC(=O)NC(c1cc(C)on1)C)C(F)(F)F C(CC(F)(F)F)N(C)CCOCCC(=O)Nc1nccs1 N1(C(c2ncc(OC)nc2)=O)CCCC(NC(c2cncnc2)=O)C(F)C1 Cc1cc(C)c(C(=O)NCCN2CCN(C(C3CCCN3C)=O)CC2)o1 S(=O)(=O)(c1ccc(C)c(C(=O)OC)c1)n1c(CC)nnc1N1CCCc2n[nH]cc21 Cc1ccc(C(C)NC(=O)C(C)(C)C2CCN(C(C3CCN(C)C3)=O)C2)nc1 C(=O)(C1=CNC2=NCCC2=C1)NC1C2(CC(NC(C3(C)CC(=C)C3)=O)C2)C1 Cc1cccc(CCC(N2CC3CC3(NC(c3ccn(C4CCC4)n3)=O)C2)=O)c1 C1(CNC(C2(CC)CC2(F)F)=O)COCCN(C(=O)C(C)(C)c2nccs2)C1 C1(N2CCCCC2)(C(=O)NC(C2CCOC2)C)CCN(CCCN(C)C)CC1 N1(C(C2(C#C)CC2)=O)CCC(=CCNC(=O)CSC2CCCO2)CC1 C(C(C)(COC)C(=O)N1CC2CC(C1)C2NC(c1cc(COC)on1)=O)OC c1(N(C2CC3CC3C2)C(N2CC(C(C)(C)C#N)C2)=O)ccc(F)cc1 N1(C(CCN(C(CCOCC)=O)CC)=O)CCC(C(F)(F)F)C1 c1(NC(N(CCC(N2CCC(C3CCCCO3)C2)=O)C)=O)ccccc1Cl c1(C(=O)NC(CNC(c2c(C)csc2)=O)C2CCC2)cnc2c(c1)NCC2 C#CCC(C)(C(=O)NCCS(=O)(=O)NC)NC(=O)COC1(C#C)COC1 C1(OCC)CCN(C(=NCc2ncc(C(F)F)cn2)NCC2CCC2)C1 Cc1cc(C(=O)NCC(CO)NC(=O)CCCc2cnn[nH]2)c(C)cc1Cl N1(C(C(=O)Nc2ccc(CN(C(C)=O)C)cc2)=O)Cc2ccccc2C(CO)C1 c1(SCC)cnccc1C(=O)NC(CNC(=O)C(F)n1ccnc1)C(C)C N1(c2ccnc(C(CC)C)n2)CC(C)(C)CCC1CNC(=O)C(C)CC1CCCC1 c1(N2CCC(C(=O)NCCCNC(=O)CN3CCCC3)CC2)ccc(F)cc1F N1(C(C2(OC)CC2)=O)CCC2(CCC(NC(=O)Cc3scnc3C)C2)CC1 C(CCCC(=O)NCCN(C(=O)Cc1cc(C)on1)C)NC(C)=O c1(CC)cccc(C(=O)N(CCC(C)NC(c2ccc(C3CCOC3)s2)=O)C)n1 c1(OCC(N)=O)cccc(C(=O)Oc2ccc(C(F)(F)F)cn2)c1 C1(CCNC(c2c(C)c[nH]n2)=O)CCN(C(C2CC2F)=O)CC1 N1(C(c2c(OC)n[nH]c2)=O)CCC2(CC1)CC2(CO)CNC(=O)CC(C)CF C12(CNC(=O)CC3C=CCC3)CC(NC(c3ccc(-c4cccs4)[nH]3)=O)(CO1)C2 Cc1ccc(C(=O)NC2(CNC(C3CN(C(C)C)C3)=O)CCCCC2)c(N)n1 C#CCCCC(C)C(=O)NC(CNC(=O)CS(=O)(=O)NC)CC(C)C C1(C(N2CCC(CCNC(c3scnc3Cl)=O)C2)=O)CCC(CO)CC1 C1(N(C(c2n(C)ncc2)C(=O)Nc2cc3ccccn3c2)C(=O)CN)CCC(C2CC2)CC1 c1(C(N(CCNC(c2cnc(CCC)s2)=O)C)=O)c(C)oc2ncnc(O)c12 N1(C(CC(C)NC(C2CN(C)CC(C)O2)=O)=O)CCC2(CCOC2)CC1 C(=O)(C(C#N)C(C)C)NC1(C)CCN(C(c2cnc(CCCCC)s2)=O)C1 C1(NC(C(=O)OCC)=O)CCC(N(C)C(c2noc(C)n2)=O)CC1 C12(NC(C3(O)COC3)=O)CCC(CC1)N(C(C1CCC1c1cccc(Cl)c1)=O)C2 c1(C(=O)Nc2cc(Br)c(C)c(Br)c2)n[nH]c2cccc(-c3ccccc3O)c12 c1(COC)ccc(C(=O)NCC2(F)CC(NC(c3n[nH]cc3F)=O)C2)o1 c1(CC)cc(C(=O)NCC=CCNC(=O)C(F)(F)C(C)O)cc(O)n1 C1(CC#C)CCN(C(C(=O)N(C(C)CC)C2CC2)C(C2CC2)OC)CC1 C1(C(=O)NCc2cnc(C)s2)CCC(NC(=O)CCCCNC(N)=O)CC1 c1(C(=O)NCC2C(NC(c3nc(COC)sc3)=O)CCC2)c(C(F)F)n[nH]c1C c1(C(=O)NC(CNC(c2c(CC)noc2)=O)CO)cccc2c(C)ccnc12 C12(CNC(c3ccc(NC(c4nocc4C(=O)CO)C)o3)=O)CC(CO)(CO1)C2 Cc1c(F)cc(C(N2CCN(C(c3cocn3)=O)CC2CO)=O)c(F)c1F Cc1[nH]nc2c1CC(C(N1CCCC(C)C1CNC(c1csc(O)n1)=O)=O)CC2 n1(C2(C)CC2)nnnc1CNC(CC(N)=O)C1CCC1 N1(C(C2C(C)(CC)C2)=O)CC(O)(CCNC(=O)C=C(Cl)Cl)C1 c1(C(N2CCN(C3CN(C(C4CC(F)C4)=O)C3)CC2)=O)cc2sccc2cn1 Cc1nccc2c(=O)c(Oc3cc(-n4cc(C5CC5)nn4)ccn3)c[nH]c12 C12=NC=CC(=NC(C)CC3CC(=C)CC(CC3)N1)N2.SC(F)(F)F CC(CSc1ccccc1)C(=O)NCC(C)CNC(=O)COCP(C)(C)=O c1(NC(c2c(C)nc(OC)s2)=O)c([N+](=O)[O-])ncn1C.C12CCC(CC1)NC2=O c1(CN2CCC(CC(=O)NC(c3ccc(Br)cn3)C)C2)ccc(Br)c(F)c1O C(=O)(C(O)CC(O)CO)N1CC(C=C)(CC(=O)NCc2cn(CC)nn2)C1 c1(C(=O)NCC(COC)NC(c2cnc(O)c(F)c2)=O)ccn2c1CCCC2 CCCC(CCCNC(=O)Cc1csc(C)c1)NC(=O)CCC(=O)N(C)C CCCCCC(C)(CC)C(=O)N1CC(CNC(c2cncc(NC)c2)=O)C(O)C1 N1(C(=O)NC(c2ccc3ccoc3c2)C)CC2(CCCCC2)CC1CO CCCC(O)CC(=O)OC(c1cc(C)cc(Br)c1)C C(=O)(C(O)CCCNC(c1snnc1C)=O)N(C1CC1)CC c1(SC)cc(C(=O)NC2CCC2NC(c2nccn2C)=O)c(C)o1 N1(C(C2(C3CCCO3)CC2)=O)CC2CC(NC(=O)CCc3nccs3)CC2C1 c1(C(N2CCN(C(c3c(C)n[nH]c3)=O)CC2C)=O)cnc2ccnn2c1C(F)F C(=O)(C1CCCc2nc(C)[nH]c21)N1C2CN(C(C(CCCC=C)(C)C)=O)C(C2)C1 c1(C(C(=O)NCc2ccc(C)cc2O)C)cn(C)c2ccccc12 CC(CO)(CCF)NC(c1coc(CNC(C2CC(F)(F)C2)=O)n1)=O C12(C(=O)NC(C)CNC(C3CC(=O)N(C4CC4)C3)=O)CCCCN1CCC2 C1(CNC(CC(C)SC)=O)CN(C(c2ccc(OC(C)C)nn2)=O)CCN1C c1(OC)c(Cl)nc(NC(C2CCC2NS(=O)(=O)CC2CCC2)=O)nc1Cl C1(C2CN(C(=O)C(C)C(C)C)C2)(NC(c2cccc(OCC(C)C)c2)=O)CC1 c1(NC(C2(C(N(C)C)=O)CC2)=O)cccnc1C(=O)N(CC(O)C1CC1)C c1(CC)cnccc1C(=O)OC(C)(C)C.c1(CC2C(=O)N2)cccc(C)n1 C1(C(=O)NCCNC(c2cnc(CC)nc2C)=O)CCCN2CCCCC12 c1(OCC(=O)NCCNc2ccsc2-n2cnnn2)ccc2c(c1)CCC(=O)N2 C(=O)(C(Cc1cn(C(C)C(=O)NC2CCOC2=O)nn1)CC(F)(F)F)OC c1(-c2c(F)ccc(C)c2)cnc2cc(C(=O)NCc3csc(C(C)C)n3)ccn12 CCCCC(O)C(C)C(=O)N1CC2(CCCN(C(C3(CC)CCOC3)=O)C2)C1 c1(C2C(C(CC=C)=O)C2)cccc(C#N)c1.CC(CCNC(=O)CC1CCCC1)N Cc1cc(Br)nc(Cl)c1NC(=O)CC1CC2(CC2)C1 C(CC(CNC(=O)C(F)(F)c1cccnc1)OC)OC.C12CC1OC2CSC.OCC C(C(CC1CCCC1)C(=O)N(CCCC(F)(F)F)C)NC(COCCCOC)=O C1(C(=O)NC2CCCCN(C(CNC(CC(C)C)=O)=O)C2)CN(CP(C)(C)=O)C1 Cc1ccc(C#N)c(N2CCOC(C(C)NC(C3(C)CC=CCC3)=O)C2)n1 C1(C(=O)NC23CC(CNC(C4CN(C)CC(C)O4)=O)(C2)C3)CCc2n[nH]cc2C1 C1(NC(C(CCOC)C)=O)CN(C(=O)Cc2ccc(Cl)nc2C)C2(CCC2)C1 C1(CC=C)(NC(=O)COC)CC2CCC(C1)N2C(=O)CC1CC1(Cl)Cl c1(NC(C=CCC(C)(C)NC(C2CCCC2C(F)F)=O)=O)ccc(O)c(Cl)c1 c1(C(N2CC(CNC(C(C(C)C)SCC)=O)C2)=O)cc(F)cc(N)c1N C1(NC(c2csc(C3CC3)n2)=O)(CO)CCN(C(=O)C=Cc2cscn2)C1 N1(CCOC)CC(C(=O)NC2CCC2NC(=O)CN2CCN(C)CC2)CC1=O CC1CN(C(=O)CC2CCN2C(C2C=CCS2)=O)CC1(F)F c1(C(N2CC3CC(NC(c4c(C)onc4Cl)=O)C3C2)=O)ncc([N+](=O)[O-])n1C C(C)(CC(C)(C)C)(c1n(CC=C)nnn1)NC(c1ccn(C)c1)C C(C1=CCN(CCc2ccccc2)CC1)NC(C1CCC(SC)CC1)=O C1(C)(C(=O)Nc2cc(CC)c(C)cc2)CN(C(=O)CC2(C)OCCO2)C(C)(C)C1 CCC(C)CCC(O)CC(=O)NC1(NC(=O)CN2CCc3ccccc32)CCC1 N(C(=NCCCCl)NCc1cnnn1C)CC(c1ccccc1Br)OC CCC(CCCC(=O)N1C(C(=O)OC)CC1C)NC(c1c(C)cnn1C)=O C(=O)(C1CCOc2ccccc21)NC1CC(NC(c2c(C)csn2)=O)C1 c1(CN(CCCOC)C(c2cc(C3CCCNC3)no2)=O)ccccn1 c1(OC)ccc(C(=O)NCC2COCC2NC(C2(F)CC2C)=O)cc1N N1(C(C2CCC(C(=O)OC)C2)=O)CC2CCC1CN2C(=O)Cc1cc[nH]n1 C1(C(N(CC(=O)NCCCC(=C)Cl)C2CCC2)=O)CCCCCC1 N1(C(C(CC)SC)=O)CC(CNC(c2cocn2)=O)C(O)C1 Cc1nccc(C(=O)NC2(C(N3CCC3C3CCCC3)=O)CC2)c1C c1(CN2CCC(NC(C3N(C)CCOC3)=O)C(C)(C)C2)ccc2ccn(C)c2c1 N1(C(c2cc(C(CC)C)no2)=O)CC2(CC(NC(c3ccc(F)s3)=O)CO2)C1 Cc1ccc(C)c(CNC(C2CN(C(=O)CSc3nncs3)CC2O)=O)n1 C1(CNC(c2c(C3CN(C(C4CCC(=O)C4)=O)C3)ocn2)=O)C2CCCCCC12 C#Cc1ccc(C(N2CC(CNC(C3(C)CCN(C)C3=O)=O)C(O)C2)=O)c(C)c1 CC1(NC(c2nc(Br)cnc2N)=O)CCCN(C(C2(F)CCCCC2)=O)C1 C(C(C)C(C)C(=O)NC1CN(C(C2CCC(=O)NC2)=O)CCC1C)OC C(=O)(C1CCCc2scnc21)N(C1CCCC1)CCNC(=O)C=CBr c1(CSC)cc(C(=O)N(CC(O)CNC(c2ccc(O)cc2F)=O)C)ccc1F C1(C(N2CC(N(C(c3nccc(C)c3)=O)C)C2)=O)CCCN(S(N)(=O)=O)C1 CCCCCCC(=O)N(C1CCN(C(=O)C(C)n2cccn2)C1)CCC CCC(CCCC(=O)N=c1cc2n([nH]1)CCCC2)NC(C1CCCSC1C)=O C(=O)(CC(O)CC(C)(C)C)NCCN(C(c1c(C)noc1C(F)(F)F)=O)C1CC1 C1(CC(=O)NCC(C2OCCCO2)(C)C)CN(C(=O)OC(C)(C)C)CC2(CCC2)O1 C12(NC(Cc3c(C)nn(C)c3)=O)CCCCC1CN(C(C1CC1C)=O)C2 CC(C)CC(O)C(C)C(=O)N1CCC(OCC(N2CCC(OC(N)=O)CC2)=O)C1 C1(CC(N2C(C(C)C)CC(O)C2)=O)CCCN(C(C2(C)CC(F)C2)=O)CC1 C1(F)(C(=O)O)CC(N(C(CN(C)C)(C)C)C)C1.C(C)(C)(C)O C1(NC(C2C(=C)C2)=O)CCN(C(=O)Cc2csc(=N)[nH]2)C(C)C1 C(N=c1[nH]c(CO)nc2ccccc12)C1(OCC)CC2CCCC2C1 C(CC(C(C)C)N(C)C(c1ccc(OC(F)F)cn1)=O)NC(C1C(C)C1)=O N1(C(c2c(SC)ccs2)=O)CCC(NC(=O)CC2CC3CCC2O3)C(F)C1 c1(C(C(=O)N(CCC)CCNC(C2CC2C2CC2)=O)O)cc(Cl)cc(Cl)c1 C(=O)(C1=NN(C2CC2)C(=O)CC1)N(C(=O)C(C)CS(C)=O)CCCC(C)C c1(C(=O)NCCC(C)NC(C2(CS(C)(=O)=O)COC2)=O)csc(C(C)(C)C)c1 C1(O)(C(=O)NC2CCN(CCC)CC2)CCN(C(C2CC3CCC2O3)=O)CC1 N1(C(CS(CC)(=O)=O)=O)CCC(C(=O)N(CC(O)C2CCC2)C)C(C)(C)C1 c1(CC)ccc(OC)cc1C(=O)N(C)CCNC(=O)C(CC1CCC1)OC N1(C(C2(C#N)CC2)=O)CCCCC1C1CCCN(C(=O)CCN2CCCCC2)C1 c1(OC)ccc(NC(c2cnn(C3CC3(F)F)c2)C(=O)NC2CCOCC2)cc1 c1(C(=O)NCC(C)NC(CCc2cccc(OC)n2)=O)cncc(P(C)(C)=O)c1 CC1(F)CN(C(c2cncc(C#N)c2)=O)CCN(C(C2CCS(=O)(=O)C2)=O)C1 c1(C(=O)NC(CN(C(c2cc(C)ns2)=O)C)C)ccnc(-n2cccn2)c1 C(CCCC)(C(=O)NCC1(C)CCC(O)CC1)NC(c1c(CC)cc[nH]1)=O c1(CC)oc(C(N2CCCC2CNC(c2cc(C)c(C)o2)=O)=O)cc1C c1(C(=O)NCC2N(C(c3ccc(C)nc3N)=O)C3C(C2)C3)cn2nc(C)sc2n1 C1(CNC(C(CC=CC)C)=O)CN(C(=O)CC2(O)CCOCC2)C2(CCC2)C1 C12(C(=O)OC)CNCCC1CN(C(C(C)C(c1ccc(C)c(F)c1)=O)=O)C2 Cc1nc(NCCN2CCC3CC23)cc(NCC(C)Cn2cccn2)n1 S(=O)(=O)(c1ccc(Cl)cc1)NCCC(N1CC(C)CC(NC(CC)=O)C1)=O C1(C(N2CC(NC(C)=O)C2)=O)CN(C(=O)C(C)=C2CCC2)CCN1C N1(C(C(OC)OC)=O)CC2(CCOCC2C(N2CCOC(C)(C)C2)=O)C1 C12(C(=O)NCCCN(C(c3c(C)nn(C)n3)=O)C)CCCCN1CCC2 c1(CC2N(C(=O)NCC3C(C)C3C)CCC2)cccc2ccccc12 c1(C(=O)NC(COC)C2(C)CC2)cccc(CNc2cc(Cl)n[nH]2)n1 c1(C(N2CCC(n3cc(COC4COC4)nn3)C2)=O)cc2cccn2c(O)n1 CCCCC(O)CC(=O)NC1(C)CCN(C(c2ncn(C(C)(C)C)n2)=O)C1 c1(C(N2CC(CO)CC(C(C)(C)C)C2)C(=O)NCCC)cc(Br)cnc1OC C1(CC(=O)N(C)CCc2ccccc2)CCCN(C(=O)C(F)F)CC1 CC(C(=O)N(CCCNC(=O)CSc1nc[nH]n1)C(C)C)c1ccco1 C(=O)(C(=O)NCCNC(C1(Br)CC1)=O)NCCSCC#C c1(C(=O)Nc2c(NC(c3c(C)nsc3)=O)nc(Cl)cc2)cc(F)c(F)cc1Cl CC1(C)CN(C(c2ncc(F)cc2F)=O)CCC1NC(=O)CC1COCC1(C)C Cc1cccc(C(N2CC(CC(=O)NC3(c4cccc(Cl)n4)CC3)CC2C)=O)c1Cl CCCCC(O)C(C)C(=O)NCC(C)CN(C)C(c1cc(OC)n[nH]1)=O CC(C)CC(C)CC(=O)NC1(C)CC1.C1(C(=O)NC(C)(C)C)CCC(C(=O)O)CC1 C1(C#N)(CC(=O)N(CCCN)CC)CCCCC1.C1(C(=O)CC)C=CCC1 C1(NC(C2C(=C)CC2)=O)CC2(CCN(C(=O)C(CC(C)C)N(C)C)CC2)C1 c1(C(=O)NC(CNC(C=C(C)C(F)F)=O)C2CCC2)c([N+](=O)[O-])cnn1C C(=O)(CC(COC)NC(C1CCCN(C(C)=O)C1)=O)NCC(COC)(C)C c1(CCCCC)cc(C(=O)NC2CCC(NC(C3(COC)CCCC3)=O)C2)n[nH]1 N1(C(C=C(C)C)=O)CCCCC1C1CCCN1CC.C(COC(=O)C1CC1)N N1(C(=O)OC(C)(C)C)CC2CC(Nc3nncn3-c3ccccc3)C2C1 n1(CC(=O)N(C)CCOCCNC(=O)CN2CCSCC2)cnc2ccccc12 C1(CNC(C=C(COC)C)=O)CCN(C(=O)CN2CCOCC2)C12CC2 C123CCCC1N(CCC2)C(=O)c1cocc1C(=O)OC3.C(C)(C(=O)N)SCC.COC c1(CNC(C2C(C(=O)OCC)C2)=O)n[nH]c2c1CN(C(c1cscc1C)=O)CC2 C1(NC(C2C(C)C2)=O)CN(C(=O)CCc2ccsc2Br)CC2(CCC2)C1 c1(C(=O)NCCCC(C)NC(C2CCCS2)=O)ccc(Br)cc1 C=CCC(C(=O)NC(CCOC(C)C)C(=O)NC1CCN(C(N)=O)CC1)OC C1(CNC(CCOC(C)=O)=O)COCCN1C(c1cccnc1)=O C1(C(C)NC(c2cc(CNC(C=CC=CC)=O)on2)=O)CC2(CCC2)C1 c1(CC)onc(C)c1C(N1CSCC1C(=O)NC(c1ncc(C)o1)C)=O C1(COCCN(C)C(C2CCN(C(C3(COC)CC3)=O)C2)=O)CCCC(=O)C1 C1(NC(CC=CCC)=O)CCN(C(C2CCOC2CC)=O)C1C1CC1 Cc1nn(-c2ccccc2)nc1C(=O)NC(C1CCCN1C(=O)C(C)O)(C)C c1(C(=O)NC2CN(C(C(CO)NC(N)=O)=O)CC2C(F)F)cc2c([nH]1)CCCC2 C1(C(C(=O)NCC2(F)CCOC2)=O)CCS(=O)(=O)CC1 C1(c2nc(COC)nn2-c2cccc(Br)c2)CCc2ccc(F)cc2C1 C1(C(=O)NC(CN(C(c2[nH]cc(CC(C)C)c2)=O)C)C)CC2(C1)CC21CCC1 N1(C(CC2ON=C(C)C2)=O)C2CCC1CC(C(=O)NCCC1CCCCO1)C2 C(N=c1[nH]c(=NCC2(C)CC2Br)[nH]c2c1CSC2)C1(OC(C)C)CCCC1 N1(C(c2cc([N+](=O)[O-])c[nH]2)=O)CCC2CCC(C1)N2C(C1CCC(F)C1)=O C(=O)(CC1CC(=O)c2ccccc21)N1CC(C)(NC(CSCCC)=O)C1 c1(NC(CCN(C(CC2ON=C(CC)C2)=O)C(C)C)=O)cc(C)c(O)c(C)c1 Cc1cc(NC(C2CN(C(C3CC34CCCC4)=O)CC2F)=O)cc(O)c1 C12(NC(CN(C)S(N)(=O)=O)=O)CCOC(CNC(c3cccc(F)c3)=O)(C1)C2 c1(C(=O)Nc2ncc(C)cc2O)cc2c(s1)CCN(c1ncnc3cnccc13)C2 N1(C(C(C)NC(C2CCCCC2)=O)=O)CCc2nocc2C1 Cc1ccc(F)c(C(N2CC3CC3(NC(=O)CCCn3c(C)csc3=O)C2)=O)c1 N1(C(CC(CC)c2ccccc2)=O)CCN(C(c2ccon2)=O)C2CCC12 N1(C(c2ccc(SC)s2)=O)CC2CCC1C2NC(C1CC1C(N)=O)=O C1(O)(NC(CSCCCC)=O)CCCN(C(c2[nH]c(=N)sc2C(F)(F)F)=O)C1 N1(C(CC(=O)NC)=O)CC2C(C(=O)N(C)N(C)C)C2C1.C1(CN)(C)CC1 C1(NC(c2cc(CC)on2)=O)CC(N(C(C2CC(=C3CC3)C2)=O)C2CC2)C12CCOCC2 c1(C(=O)NC23C(NC(C(CCC)(C)C)=O)CC(CC2)C3)cc(F)c(F)c(F)c1 Cc1ccc(Br)c(C(N2CCN(C(=O)C(C)n3ccnc3)CC2C#N)=O)c1F c1(C(N2CCCCC(CNC(C3C(C)(C)OCC3)=O)C2)=O)cnn2ncccc12 c1(NC2CC(OCC)C2)nc(C(=O)OC(C)(C)C)ccc1[N+](=O)[O-] CCCC(C)(C)C(=O)NC1C2CC(NC(C3CCC(SCC)CC3)=O)CC12 c1(SCC)nccnc1C(=O)NCCC(C)NC(c1ccc(F)cc1)=O CC1CN(C(=O)Cc2cncc(O)c2)CCC1NC(c1ccn(CC(F)(F)F)n1)=O C(=O)(C(F)C(F)(F)F)NCC(CNC(C12CC(C1)C2)=O)O C(=O)(C1=C(C)CCCC1(C)C)NC(CNC(c1ccc(C#C)cn1)=O)C(C)C CC(CN(C)C)CCC(=O)NC(C1CCCN1C(=O)C=Cc1cncn1C)(C)C CCC(=O)CCC(=O)NCc1cc(C(=O)NC2CCOCC2F)cs1 O=C1CC(C2CCCN(C(=O)C(=O)Nc3ccc(N4CCCC4=O)cc3)C2)CN1 C#Cc1cn(C)nc1C(=O)NCC1CN(C)CCN1C(=O)C(C)=C1CC1 c1(NC(C(C(C)C)NS(C)(=O)=O)=O)c(I)cnn1C N1(C(CC(C)(C)OC)=O)CC2CC(O)C1C2NC(c1ccc(Br)s1)=O c1(C(C)(C)C)c[nH]c(C(=O)NCCOCCn2cc(C3C4COCC34)nn2)c1 C#CCC(C)(C(=O)NC(C)(C#N)CC)NC(=O)CN(C)C(C)=O Cc1cc(C(=O)NC2CN(C(=O)Cn3nccn3)CCC2F)nc2ccccc12 C1(NC(C(C2CCCCC2)C)=O)CCC(N(C)C(C2CC2F)=O)CC1 c12cccc(c1)CONC2=O.C(C(O)C(F)(F)F)C(N1C(CCCC)C=CC1)=O C(CC1CCC1)(C(=O)NC(C1CCC1)C1CC1)NC(C1(CC=C)CCC1)=O C(=O)(CC(O)CNC(C1(COC)CCC1)=O)N1CC(CC=C)C1 C(=O)(CCC(=O)C(C)(C)C)NCC1(CNC(C2C(C)(CC)C2)=O)CC1 N1(C(c2cc(CC)c(C)s2)=O)CCCCC(NC(=O)C(C)NC(=O)OC(C)(C)C)C1 C(=O)(CCCCC(F)(F)F)N1C(CC)CC(NC(c2cccc(F)c2O)=O)CC1 C12(NC(c3n(CC)ncc3Cl)=O)CCC(CC1NC(c1cn(C3CC3)cn1)=O)C2 c1(NC(c2ccc(NC(c3cccc(Cl)c3I)=O)nc2)=O)ncc(Cl)cc1I C1(C2CC2)(NC(C(CC=C)OCC)=O)CCN(C(=O)CCC2CCCCC2)C1 n1(CC)ncc(Cl)c1C(=O)NC(CN(C(=O)C(F)CC1CCOC1)C)CC C1(C(=O)NCC(c2ccccc2)NC(CC(=O)N(C)C)=O)(CCF)CCOCC1 C=CCC(CC(=O)NC(C)CNC(=O)C(CCCC)N(C)C)N.C(C)(C)(C)SCCC CC1c2ccccc2CC12CCN(Cc1c[nH]nc1C(F)(F)F)CC2 N1(C(CCN(C(=O)CC2CC2)C)=O)CCCC(CO)(CNC(=O)Cc2cccs2)C1 CS(=O)c1ccc(CC(N2CCCC(CNC(=O)Cn3ccnn3)CC2)=O)cc1 C1(C(N2CCC(C)(NC(c3ccc(COC)o3)=O)C2)=O)CC2CCC1CC2(F)F c1(CC)cc(OC)c(COC)cc1OC.c12sc(nc1C)CNC(=O)C2C.CC N1(C(CN(C(COC)=O)C)=O)CCC2C(C1)CN2C(c1cncc2c1CCC2)=O C1(N(C(C2C(CNC(C3C(C(C)C)OCC3)=O)CCC2)=O)C)CC2CCC1CC2 C1(c2c(CCC(=O)O)c[nH]n2)CCCCN1Cc1ccccc1C(F)(F)F N1(c2cc(OCC)ncn2)CCC2(CC(C(=O)NC3CN(C)C3)=NO2)C1 c1(CC(=O)NCCC(C)NC(c2c(C)cnnc2O)=O)cnc2c(C)cccn12 c1(C(=O)NCC(C)(C)NC(CCC2CCCN(C)C2)=O)cccc2c1C(C#N)C2 CC(C)(C)CC(O)CC(=O)NC1CC2CCC(C1)N2C(C12CC(C)(CCO1)C2)=O C(C(=O)NC1CSC1)(C(C)C)NC(c1c(COC)noc1)=O CN(C)NC(=O)CCC(=O)NC1CC1CNC(c1c[nH]nc1F)=O CCC(C)(CCNC(c1ccc(CCF)cc1)=O)NC(=O)CC1COCCN1C C1(CC)CCCN(C(=O)C(CCC2CCC2)NC(=O)CC2CC(F)(F)C2)C1 c1(C(N2C(CN(C(C(C(CC)O)C)=O)C)CCCC2)=O)cc(C)cc2c1OCC2 C1(=CC(=O)NCC(=O)N(C(C2CCC2)=O)C2CC2)CCN(C(=O)Cc2cnns2)CC1 C1(C(=O)OC)CCCN(C(c2c(F)cc(C(F)(F)F)c(F)c2F)=O)CC1(F)F c1(C(=O)NCC2CN(C(C(C)(C)C)=O)CC23CCC3)cc2c(nc1O)CCOC2 CCCCCCOCC1(F)CC(C(=O)NC(=O)CCSCC(N)=O)C1 c1(C(=O)NC2N(C(C(c3ccc(OC)cc3)CC)=O)CC2)cc(S(N)(=O)=O)c[nH]1 C1(NC(c2n(C)ncc2)=O)C2CC3C1C3C2C(N1CCOC(CCF)C1)=O Cc1cn2c(n1)CCC(C(=O)NCCN(C(=O)CCCn1c(O)nnc1O)CC)C2 c1(C(C(=O)NC2CCN(C(=O)OC)CC2)N(CC=C)C)ccc(Cl)c2c1CCC2 c1(C(N2CC(O)(CCNC(C3CCCCC3O)=O)C2)=O)ccc2ncncc2c1 C1(CNC(=O)CCc2cnc[nH]2)CC(F)CCN1C(=O)CC1CCCOCC1 CCCC(C)(C)C(=O)NCCC1CC(NC(=O)CC2CCC(C)O2)C1 C1(C(=O)NC2(C)CC(NC(=O)Cn3cc(C4CCC4)nn3)C2)CC2C=CC1O2 CC(C)C(C(=O)NCc1nc(=O)o[nH]1)C(C)NC(c1ncc(F)cn1)=O C1(O)(CC(N2CCC(C(C)NC(=O)CC3CCCC34CC4)C2)=O)CCCCCC1 N1(C(C(=C)F)=O)CCC(C)C1c1cn(Cc2oncc2OC)nn1 Cc1ccc([N+](=O)[O-])c(OC2CCCN(C(CON)=O)C2)c1 N1(C(C(n2nnnc2C2CC2)C)=O)CCN(C(c2coc(Cl)c2)=O)C2CCCC12 C=CCN=C(NCC(O)COC(C)(C)C)NC1CC1NC(=O)OC(C)(C)C c1(C(N2CC3CN(C(Cc4cn(CC)nc4)=O)C3C2)=O)cc(Cl)cc(C#N)c1 C=CCCCC(=O)N1CC(O)(C(F)C(=O)NC(CCC)C(=O)N(C)C)C1 S(=O)(=O)(c1cnc(N2CCCC(CS(N)(=O)=O)C2)c(Cl)c1)N(CC(CCC)C)C N#Cc1ccc(NC2CCN(C(c3cnc(N(C)C)c(Cl)c3)=O)C2)cc1 N1(C(C2CN(C)C(=O)C2)=O)CCCC(CO)(NC(=O)CCc2ccc(F)cc2)C1 C123CCC(CC1)(C2)N3.N1(C(C(N2CC(NC(=O)OC)C2)=O)=O)CCC(C)C1 C1(C(N2CCC(CN(C(C3(OC(C)C)CCC3)=O)C)C2)=O)COCC2(CCC2)O1 Cc1cccc(NC(=O)NC2CCCCC2NC(=O)NCC2(C(F)(F)F)CC2)c1 Cc1c(C(N2CC3CN(C(=O)C(C)(C)CO)CCC23)=O)cc(Br)cc1[N+](=O)[O-] C1(C(=O)OC)CC12CN(C(C1CCC(NC(=O)Cc3cc(C)cs3)C1)=O)C2 c1(C(=O)NC(CC)CNC(c2[nH]c(O)nc2C)=O)c(O)cc(=O)n2c1COCC2 c1(N2CCCCC(CO)C2)nc2c(c(=NCCSC3CCCC3)[nH]1)COC2 C(C(C)(C)C(=O)NC1CN(C(c2cc(Br)oc2C)=O)CC1C)SC N1(C(COC2C(C)CCCC2)=O)CC2(CC2)CC1CNC(c1ccc(C(N)=O)[nH]1)=O CCC(C(=O)N1CC(CC(F)C(=O)NC(CN(C)C)C(C)(C)C)C1)C(F)(F)F C1(C(=O)NCCN(C(C)C)C(c2ccc3nn[nH]c3c2)=O)OCCOC12CCC2 c1(C(=O)NCCCN(C(C2C(=C)C2)=O)C)cc(-c2ccncc2)no1 N1(C(C(CC#C)C)=O)CC(NC(c2cc(CC)nc(C)c2)=O)C(C2CC2)C1 C1(NC(CCCOC(C)=O)=O)CN(C(C23CC4CC2C3C4)=O)CC1(C)C C1(N(C(=O)C(C)(C)c2ccns2)C)CCN(C(C2CC3(C2)CC3F)=O)CC1 c1(C(C)C(=O)NCC2CCC2NC(c2cc[nH]n2)=O)ccc(Cl)s1 CC1CCN(C(c2nscc2Br)=O)C(C)C1NC(C1CCCOC1)=O c1(C(=O)NC(c2cccc(C)c2)CNC(C(C)(C)OC)=O)cc(F)c(F)cc1Cl c1(CC)nc(C(=O)NC(C)CC(C)NC(=O)Cn2ccc(Br)n2)c(C)o1 C(=O)(C1=NNC(=O)CC1)NCC1(CNC(c2ccc(C)c(O)n2)=O)CC12CCC2 N12CCCC(C1=O)C(=O)O2.Cc1ccccc1CNC(=O)Cc1[nH]cnc1C#N N1(C(C2(CC)CC2)=O)CCC2(CC(C(N3C4CCC3(CO)CC4)=O)C2)C1 C(c1cccc(Cl)c1)=CC(N1CC2C(NC(C(CSC)(C)C)=O)(C2)C1)=O C(=O)(C#CC1CCCOC1)NC1CN(C(CCN(S(C)(=O)=O)C)=O)CC1C C1(CNC(C(C)Oc2ccc(F)cc2)=O)OCCCC1(C)C C12(C(N3CCC(O)(CC)C3)=O)CCCC1CCN2C(=O)Cn1cccn1 C1(O)(C(C)NC(C(C)NC(COC)=O)=O)CCN(C(=O)CC(C)(C)SC)C1 C1(C(=O)NC2(CC=C)CCC2)CCOC1CCC.C(=O)(C(CO)N)NC(N)=O C=Cc1cc(C(=O)NCC2CC2CNC(c2c(C#N)cnn2C)=O)cc(F)c1 N1(Cc2n(C3CC(Nc4cccc(C(C)C)c4)C3)nnn2)CCC(S(N)(=O)=O)C1 CC(C)(C)C(CO)C(=O)NC1CCCN(C(=O)CCn2ccccc2=O)CC1 N1(C(C2N(S(C)(=O)=O)CCC2)=O)CCCOC(CNC(C2(O)COC2)=O)C1 N#Cc1cccc(NC(=O)C(C2CC=CCC2)NC(=O)CC2CC(=O)NC2=O)c1 C1(NC(c2c(N)nc(Cl)cc2)=O)CCN(C(c2nscc2N)=O)CCC1CO Cc1ccc2ncc(C(=O)NCC3CN(C(=O)CC(O)CC(C)C)C4CC34)n2c1 c1(C(=O)NCC(CCNC(C2C(=C)C2)=O)OC)cc(=O)c(O)c[nH]1 Cc1cnccc1C=CC(N1CCC(C(C)NC(=O)CC(C)C2CC2)C1)=O C(=O)(CS(=O)(=O)C1CC1)N(CCC)CCNC(C1CCCCC12CC2)=O c1(C(=O)NCC(C(=O)NCC(C(=O)OC)OC)C)ccc(O)nc1 c1(OC)cc(CN2CCC(C)(NC(=O)Cc3ccccn3)C2)cc(F)c1F C1(O)(CC)CCCN(C(=O)Cn2cc(-c3cc(C(=O)OC)sc3C)nn2)CC1 c1(CNC(=O)CCCc2ccccn2)cccc(NC(=O)CC2CCCCC2)c1 N1(C(c2nccc(N(CCCC)C)c2)=O)CCC12CCNCC2 N1(C(C=Cc2cccc(N)c2)=O)CC(C2CN(C(C3CC34CCCOC4)=O)C2)C1 C1(OC)CCCN(C(=O)C(c2ccnn2C)NC(C2C3CCC(F)C23)=O)C1 C1(CNC(CCSCC)=O)COCCN(C(C2CC2C(C)O)=O)C1 C1(CNC(=O)CO)CC2(CCN(C(=O)C(O)c3ccsc3)CC2)C1 N1(C(=O)C(c2ccc(F)c(Cl)c2)O)CCC2CN(C(=O)C=CI)CC2CC1 CP(C)(=O)c1ncccc1C(=O)Nc1ccccc1.C1C(=O)NOC1 c1(N(C)C(C2CCCN(CC(F)(F)F)C2)=O)ncc(Br)c(O)n1 c1(C(=O)NCC(C)(C2CC2)NC(C(F)=C(C)C)=O)ccc2nn[nH]c2c1O N1(C(C2(CCOCCOC)CCC2)=O)CCC(NC(C)=O)C1 C1(C(=O)NC(CN(C(C=CC(C)(C)SC)=O)C)(C)C)CN2CCCC1C2 C12(NC(CSc3n(C)nnn3)=O)CCCC(CN(C(C3(C)CCCOC3)=O)C1)C2 C(=O)(C1CCc2ccccc21)N1C(C(N(C)Cc2onc(C)n2)=O)CNC(=O)C1 C1(O)(C(C)NC(c2c(C)ncs2)=O)CCN(C(c2cccc(C)n2)=O)C1 C1(N(C(=O)OC(C=C)C)C2CC2)CC(c2ccccc2)CCC1=O C1(C)(C(=O)NCCN(C(COCCCC#C)=O)CC2CC2)CCCNS1(=O)=O C1(C(=O)NC2CC3CC(NC(c4csc(S)n4)=O)CC32)CCc2ccccc2O1 c1(C(C(N2CCCC(NC(CC=C=C)=O)C2)=O)O)cc(F)cc(F)c1 N1(C(C2(C)N(C(C=NOC)=O)CCC2)=O)CCOCC2(CCC2)C1 C1(C)(CCC)CCCN(C(C2CC3(C2)CN(C(C2CC2(C)C)=O)C3)=O)C1 C(CNC(C1CC2C=CC1C2)=O)(CC(F)(F)F)NC(c1ccc(Cl)cc1F)=O Cc1ccc(C(=O)NCCCCNC(c2n[nH]cc2C2CC2)=O)c(F)c1 c1(CCNc2ccccc2)cccc(Br)c1Cl.N12CCC(C1)CN(C)C2=O c1(C(N2CC(NC(c3sc(CC)c(C)c3)=O)C(OC)C2)=O)cc(F)cc(C)c1N CC1(O)CCC(C(=O)NCCCCCCNC(c2ncoc2C2CC2)=O)CC1 N1(C(Cn2nc(C)oc2=O)=O)CCOCC(NC(C2(CS(C)(=O)=O)COC2)=O)C1 c1(SCCC(N2C(C)(C(=O)O)CC2)=O)ccc(F)cc1F.c12cncc(c1)S2 C(=O)(CS(=O)(=O)CC1CCCO1)NC1C(OC)CN(C(C2CC(C)(O)C2)=O)C1 Cc1c(C(=O)N(C)CC2CCCN2C(c2cnc(C3CCC3)o2)=O)cccc1F c1(NCC(C2CC2)OC)cc(Br)ccc1S(=O)(=O)NCCc1ncccc1F N1(C(=O)CC2(O)CCC2)CCCN(C(c2cccc(CO)c2)=O)C(CO)C1 c1(OC)ccc(C(=O)NCC(C)(C)CNC(=O)C(C)C(C)O)c(Br)c1 C(CC(=O)NC1CC=C(C(C)C)CC1)(C(F)(F)F)NC(CCCN(C(C)=O)C)=O c1(C(=O)Nc2cc(Cl)nc(Cl)c2Cl)ccc(-c2ccns2)c2cc[nH]c12 c1(C(=O)NCC(CC(C)C)NC(C2CC2C)=O)cccc2nonc12 n1(C(CC)C)ccc(=NC(=O)C2CC(F)CN2C(c2cc(CO)ccc2F)=O)[nH]1 N1(C(c2cc(N)c(N)nc2)=O)CCN(C(=O)CC2CCSCC2)CC(CO)C1 c1(C(CN)NC(C(=O)NCC(C)CO)=O)ccc(-c2ccnn2C)cc1 CC(C)C(C(c1nnnn1C1CCCC1)NCCc1ccn(C)n1)C(C)C Cc1ccc(O)c(C(=O)NCC(C)C(F)C(=O)NCc2ncoc2C(C)C)c1 C(=O)(CC(=O)NC(C1(CSC2CC2)CC1)=O)NCC(COC)F Cc1sc(C)c(C(=O)NCC2CCC(C)N(C(=O)CCCOC(C)C)C2)c1C#N c12cc(O)nc(n1)CCN2.c1(NC(C2(O)CC2)=O)ccc(-c2cccnc2)s1 C1(CCNC(C2CCC(C(F)(F)F)O2)=O)(OC)CN(C(C2CN(C)C2)=O)C1 Cc1ccc(SCC(=O)NCC(C)N(C(=O)CSC2CC2)C(C)C)cc1 C(=O)(C(CC(C)C)C(C)C)NCC(C(=O)NC(CCC(C)C)CO)CC1CC1 c1(C(=O)NC(C2N(C(c3ccc(C(=O)OC)o3)=O)CCC2)C)ccc(Cl)c(C)c1 C1(CNC(c2nc(C(C)OC)oc2)=O)CCN(C(=O)CN2C(=O)CNC2=O)CC1 N1(C(C(C)NC(C)=O)=O)CC(N(C(=O)CCC(=O)N(C)C)C)C(C)(C)C1 C(=O)(C(C)CC(F)(F)F)NC(CN(C(c1cnn(C(C)C)c1N)=O)CC)C c1(C(=O)NCC2CCN(C(CC(CC)CC)=O)CC2C)coc2ccc(C)cc12 C1(C(=O)NC2CC(Nc3ccn4nccc4n3)C2)CCCC2CCCCC12 N1(C(C2(OC)CC2)=O)CC2ON=C(CNC(=O)Cc3cccc(F)c3F)C2C1 C=C(C)CCC=O.C(C(C)(C)CN)N(C(=O)C(CN(C)C)N(C)C)CC c1(C(C)C)cncc(C(=O)NCC2CN(C(=O)C(N3CCSCC3)C)CC2C)c1 C(C)(C(O)C(=O)N1CC(NC(=O)Cc2ccc(-n3cnnn3)cc2)C1)SC c1(C(=O)NCC(CC=C)NC(C2(C(C)(F)F)CC2)=O)cnc2[nH]cc(C)c2c1 C(c1ccc(Br)s1)=C(C)C(=O)OC1CCC(=O)C1C c1(N2CCCC(NC(c3cc(C(F)(F)F)ccn3)=O)CC2)nc2c(F)cccc2o1 CC1(C)C(C(=O)NCC2(O)CN(C(C3CC3(F)F)=O)C2)COc2ccccc21 C(=O)(C1=CC2CCCC12)N(CC)CC1CCN(C(c2cncnc2)=O)CC1 c1(C(=O)NC(CCNC(CCCC)=O)C(C)C)c(Cl)ccc(F)c1F CC1(C)CCC(C)(NC(=O)C(C)(C)C2CCCN2C(=O)CCc2nncs2)C1 Cc1c(C(N2CCOC(CC(N3CCC(CF)CC3)=O)C2)=O)cnn1C C1(C(=O)NCCCOCC)C2CC3C(C2N(C(C2CC4C=CC2O4)=O)CC)C13 Cc1ccc(C(=O)NCC2(C(=O)NC(c3ccco3)CO)CCCC2)cc1 C1(C(=O)NC(CNC(Cc2scc(C)c2)=O)CO)CCN(C)S1(=O)=O C1(C)(COC)CC(NC(c2ccsc2C)=O)CN1C(c1ccnc(C(C)C)n1)=O c1(C(=O)NC(CN(C)C(c2ccc[nH]2)=O)(C)C)ccn2ncccc12 c1(C(N2CC(C#N)N(C3CC3)CC2)=O)cc2cccc(-c3cncs3)c2s1 c12ccc(cn1)C(=O)NC2.c1(CCCCC)cn(CCOC2(C)CCC2)nn1 N1(C(C)C)CC(C(=O)N(CC(C)NC(=O)C(C)(C)c2ccn(C)n2)C)CCC1=O C(=O)(C1CCCn2cnnc21)N(CCN(C(=O)Cc1sccc1C)CC)CC C12(c3cn(CCCN(C(C4CCC(C)C4)=O)C)nn3)CC(C1)S(=O)(=O)C2 C1(CC(=O)N(C(C)C)CCNC(=O)CC2(C)CCOC2)COC(C)(C)C1 CC1OCCC1(C)C(N1CC(NC(c2ccncc2F)=O)C(O)C1)=O N1(C(C(C(=C)C)(C)C)=O)CCC2(C=C(C(=O)NCCC(O)C3CCC3)C2)C1 C1(C(N2CC(C(C)NC(c3ncoc3C3CC3)=O)OCC2)=O)CC(=O)NC1(C)C N1(C(c2cnc(C(C)(C)C)s2)=O)CCCN(C(C2(CCF)CCC2)=O)CC1 CC1(C)CC2(CC2C(=O)NC(C)(C)COCCCNC(C2CC2C2CC2)=O)C1 c1(CCCC(=O)NCCC(O)CNC(=O)CCn2cncn2)cccc(F)c1 C(=O)(C1=C2CCCN=C2NN1)N1CC(CNC(CCCCC)=O)C2(C1)CCC2 c1(C(N2CC(C(C(=O)N(C3CCCCC3)CC)O)C2)=O)nnc(O)nc1O CC1(C)C(CNC(c2cnc(C(N)=O)nc2)=O)CCN1C(C1C2CC3C(C2)C13)=O Cc1cccc(C(N2CC(C)CC2C(=O)N(C2CC2C)C)=O)n1 C(=O)(C(O)CCCNC(C1COCCO1)=O)N1C(C)(CCO)CC1 C(CCCCCC(=O)NCC(F)CNC(c1c(O)cccc1F)=O)SC N1(C(c2ccc(CNC(=O)CCc3ccc(Cl)cc3)cc2)=O)CCn2nccc21 C1(C)(C(=O)N(CC)CC2CC2)CN(C(C23CSCC2C3)=O)C(C)(C)C1 Cc1cc(C(=O)NCC(C2CC2)NC(C2CCC(F)(F)CC2)=O)cc(C)c1C#N N1(C(c2cc(OC)nn2C)=O)CC(NC(C2CCCCN2C)=O)C2(CCC2)C1 C(c1cc(C)cc(C)c1)=CC(N1CC(COC)(NC(C2COC(=O)N2)=O)C1)=O C1(C2=CCCCC2)c2n(nnn2)-c2cccc(c2)N1.Oc1ccc(C2CC2)cc1 N1(C(C(C2CCOC2)OC)=O)CCN(CC(N2CCN(C3(C)CC3)CC2)=O)CC1 C12(NC(=O)C=Cc3ccsc3)CCCC1N(C(c1cc(C(F)(F)F)n[nH]1)=O)CC2 C1(CNC(C(C=C)O)=O)C2CN(C(=O)CSc3cccc(C(F)(F)F)c3)CC12 N12CCC(O)(CC1)C2(C)C.CC(CN)C(=O)Nn1cc(C2(O)CCOC2)nn1 C1(NC(c2cc(C(C)C)nn2C)=O)CN(C(c2c[nH]ccc2=N)=O)CC12CCC2 c1(N(C)C)ccc2[nH]c(C(=O)NCC3(O)CCN(C(C4CC4F)=O)CC3)cc2n1 N1(C(CSCC)=O)CC(CNC(=O)C(C(C)(F)F)c2ccccc2)C2CCCC2C1 c1(C(N2CC(CCCC)C2)=O)ccc(P(C)(C)=O)nc1 N1(C(CC(CC)(C)C)=O)CCCN(C(c2ncoc2C2CCCCC2)=O)CCC1 N1(C(C)C)CCCC(CC(=O)NCCCCNC(c2c[nH]cc2C(C)(C)C)=O)C1 C(=O)(CCC(C)(C)C)NCCC1(NC(C=CC=CC)=O)CC1 C(=O)(CC(C)(C)C(C)(F)F)NC1(C)CCN(C(C2CCCC3CCCCC23)=O)C1 C#CC1CC2CCC1N(C(=O)CC1CC(C)N(C(=O)Cc3cnc(C)s3)C1)C2 S(=O)(=O)(c1ccc(OC(F)F)cc1)NC(C1CNCCO1)C(=O)NCCC Cc1csc(C(=O)N(CC(O)CN(C)C(C2CC2(F)F)=O)C)c1Cl N1(C(C(CC)CC(F)F)=O)CC(C)CN(C(c2ccc(C)c(F)c2)=O)C(C)C1 C1(C2CCOCC2)(C(=O)NC2C(NC(C(COC)N(C)C)=O)COC2)CC1(F)F N1(C(CNC(CCC)=O)=O)CC(NC(=O)Cc2nncn2C)CC2(CC2)C1 c1(C(CC)OC(C(C)OCCCC)=O)ccc(F)c(Cl)c1 C(=O)(CS(=O)(=O)CCC)NCC(=C)CCNC(C1(Cc2cccc(F)c2)CC1)=O CC1(C)CN(C(C2CCC(=O)NC2)=O)CC1C(=O)NC1CCCC1N=[N+]=[N-] n1(CCC)ccc(CNC(C2CCCC2CNC(=O)Cc2cc(CC)on2)=O)n1 C(C)(C)(CC(=O)N(CCCOCCNC(=O)C(O)CN1CCCC1)C)OC c1(C(=O)NCC2(NC(C(COC)OC)=O)CCOCC2)sc(C)c(C)c1Br C1(CNC(c2cnc3sccn23)=O)CCCN(C(=O)CN2CCCCC2)CC1 CN1CC=C(CC(=O)NCC2CCN(C(C3CCO3)=O)C23CCC3)CC1 c1(-n2cc(CCNC(c3nc(OCC)sn3)=O)nn2)cnc2ccc(F)cc2n1 C#CC1(C(=O)NC(c2ncnn2C)C)CCN(C(=O)CC(F)(F)F)C1 c1(C(N2C(CNC(C(CC)N3CCCC3=O)=O)C=CC2)=O)cc(Cl)c(C)cn1 C1(C(=O)NC(C2(C)CCCC2)C(=O)OC)NCCC1(C)C c1(C(=O)NC2C3CCN(C(C=CC)=O)C32)cc2sccc2n1CC(=O)OC Cc1ccn(C)c1C(=O)NCCCOCCCNC(=O)C(C(C)C)n1cccc1 CC(C)S(=O)(=O)CC(=O)NCC1CN(C(C2CC(C)OC2C)=O)CC(C)(C)O1 Cc1cccc(NC(c2ccc(F)c(-c3cccc(OCC(C)C)c3)n2)=O)c1I N1(c2snc(C)n2)CCCC(CO)(NC(C2CN3CCC2CC3)=O)C1 c1(C(=O)NCCCC2CCCCN2C(=O)CC2CC(F)C2)ccc2occc2n1 N1(C(CCSC)=O)CC=CC1C(N1CC(C)(CF)C1)=O c1(OC)ccc(C(N2CC3CC2C3NC(C2CCCS2)=O)=O)cc1N C(CCN(C)C)(C(=O)N1CC(CC)(CC)C1)NC(CCC=O)=O C1(C(N(C)Cc2cccnc2)=O)CC2CC1CC2NC(C1(CF)CCOCC1)=O C1(C(N(C)CC2(O)CN(C(C3CC(CCC)C3)=O)C2)=O)(C(C)C)CNC(=O)C1 c1(CC(=O)N(CCC)CCNC(c2ccnn2C)=O)ccc(C)c(F)c1 c1(CCC(=O)NC(CN(C(CSC)=O)C)C)ccc2cccnc2c1 C1(CNC(C2(CNC(CSCC#C)=O)CCCC2)=O)CCC(C)(C)CC1 c1(N(CCN(C)C(c2coc(C3CCOCC3)n2)=O)C)c([N+](=O)[O-])cnn1C c1(OC)cc(C(=O)N(CCCCN(C)C(C2OC3CCC2C3)=O)C)cc(N)c1O N1(C(c2c(O)ccc(OC)c2)=O)CCC(NC(c2ccc(F)o2)=O)C(C)(C)C1 Cc1ncsc1C=CC(=O)NCC1C=CC(NC(=O)COc2cccc(O)c2)C1 Cc1ccc(C)c(C(N2CCC(F)(CNC(C3(c4ccsc4)CC3)=O)CC2)=O)c1 C(C)(C)(CCCC(=O)NCC1C(C)(C)C1(C)C)NC(CC(C=C)C)=O N1(C(Cc2c(C)cco2)=O)CCN(C(C2OCC2(C)C)=O)CC1C(C)C c1(OC)ccc2cc(C(=O)NCC(O)CCNC(c3ccsc3)=O)[nH]c2n1 C1(C(=O)NC2C=CC(CNC(=O)CCCc3csc(=N)[nH]3)C2)C2CCCCCC12 C(c1ccc(Cl)cc1F)=CC(=O)NC1(CF)CCN(C(=O)CC2CCOC2)C1 C1(NC(C=C(C)C)=O)CCC2CN(C(=O)C=Cc3cncc(Br)c3)CCC2C1 c1(CC)ncoc1C(=O)N(C(C)CCNC(c1cc(C(C)C)[nH]n1)=O)C c1(CNC(C2C(CCC)C2)=O)ccc2c(c1)CN(C(=O)CC1COCC(C)O1)C2 N1(C(CCc2cnc(C)[nH]2)=O)CC2COCCC2(NC(=O)CC2CC23CC3)C1 C(c1ccncc1)=CC(=O)NC1C=CCN(C(=O)C=Cc2cocn2)C1 C12(C(=O)NC3CN(C(CC4C(CC)C4)=O)CC3O)CCC(C)(C1)OC2 C1(c2n(CC)nnn2)(NC(C2CC2(Cl)COC)=O)CCN(CC)CC1 c1(C(N2C3CN(C(CN(C)C)=O)CC32)=O)ccc(Cl)c(I)c1 C(=O)(C(C(=O)N(CCCNC(=O)Cc1c(C)ncnc1C)CC)C(C)(C)C)OCC N1(C(CC=CCCC)=O)CC2CCCCC2(CNC(=O)CCCOCCCC)C1 Cc1cc(C(N2CC(CCNC(=O)Cc3cncnc3)C2)=O)c(Br)c(C)c1 C1(C(=O)NCCN(C(CC)C)C)CC(O)(CNC(c2ccon2)=O)C1 Cc1cn(C)nc1C(=O)NCC1CCCCC1NC(C1(c2cc[nH]n2)CCC1)=O N1(C(Cc2onc(C)n2)=O)Cc2n[nH]cc2C1C(=O)NCCC1CC(C)C1 N1(C(C)C)CC(C(=O)NCC(O)CNC(=O)COCc2nc[nH]n2)CC1=O Cc1ccc(F)c(C(=O)NCC(O)CCNC(c2nc(Cl)c(Cl)s2)=O)c1 c1(CC)ccc(C(=O)NC2CCC(F)(CNC(=O)C(F)CC3CCC3)C2)c(C)n1 c1(C(C)C)cc(C(=O)N(CC(C)NC(=O)Cn2cnc(Br)c2)C)on1 C1(NC(C(Cc2cc[nH]n2)NC(c2cn(CCC)nn2)=O)=O)CCOCC1F c1(C(N2CCC(C3CC3)(CNC(C3(OC)CC3)=O)C2)=O)ccc(C)cc1[N+](=O)[O-] N1(C(Cc2cccc(C#C)c2)=O)CCC(CCNC(=O)CC(C)C)C(F)(F)C1 C1(NC(C2C3COCC23)=O)C2CN(C(=O)CCN3C(=O)C=CC3=O)CC12 C1(C(N2C(C)CCC(CNC(C3CC3Br)=O)C2)=O)C2CCC1(C)C2(C)C C=CC1OCCC1C(=O)NC(C)CN(C(c1sc(C)cc1C)=O)CC c1(CC(N2CCN(C(CC(C)C)=O)C3C2C3)=O)cc([N+](=O)[O-])ccc1O c1(C(=O)NC2CCC(NC(C3(C#C)CC3)=O)CC2)nnc2c(F)cccc2c1O c1(C(N2C(C)CN(C(c3nc(Cl)cs3)=O)CC2)=O)cc(P(C)(C)=O)ccn1 C12(C)CCC(CC1)NC2=O.c1(C(=O)NCC2CC(C(=O)OCC)C2)cc(Cl)cs1 C1(CC(=O)NCC(C)(C)NC(c2cn(C3CCOC3)cn2)=O)CCCNC(=O)C1 C1(S(C)(=O)=O)(C(N2CCC(CCC(=O)OC)CC2)=O)CC(C(F)(F)F)(OC)C1 c1(NC(=O)NC(c2ccccc2)OC)ccc(CNCc2nc(C)c(C)o2)cc1 c1(CC(=O)NCc2ccc(I)nc2)ccc(-c2ccccc2C(F)(F)F)c(F)c1 n1(CC)nc(C)c(C(c2nnnn2C)NCc2ccc(C3CCC3)cc2)c1C c1(NC(=O)NC2CCCC(Br)CC2)cc(Br)cc2c1OCC2 c1(OC)cc(CC(=O)NC(C)Cn2nc(C)c(C(=O)O)c2C)cc(Cl)c1 N1(C(C2OCC(C)(C)C2)=O)CCC2(CC1)CN(C(=O)CC(F)F)C2 C=C(C)CC(C(=O)NCCN(C)CCOC)NC(C1CCCCC1O)=O C1(CC2N(C(c3c(CC)occ3)=O)CCC2)COCCN1C(=O)NC=O C(=O)(C1=C(c2ccccc2)SCCO1)NCC1(C(C)NC(CCC=C)=O)CC1 N1(C(c2ccc(C)c(Cl)c2)=O)CCCN(C(c2cc3c[nH]cnc-3n2)=O)CC1C C1(NC(CSCC(=O)OC)=O)CCC(C)N(C(=O)CCc2nc(C(F)(F)F)n[nH]2)C1 C1(NC(Cc2ccn(CC)n2)=O)CS(=O)(=O)CC1NC(=O)C(=O)C(C)(C)C c1(C(N(CCNC(=O)CC2COCCO2)C2CC2)=O)cc(C(F)(F)F)ccc1O c1(CC(N2C(CNC(c3c(COC)noc3)=O)CCC2)=O)c(OC)cccc1F O=C1CN(C(=O)C(F)C2CC(NC(C3(CCO)CC3)=O)C2)CCN1 C1(NC(C(CSC)(C)NC(c2ncc(F)cc2C)=O)=O)CC2CC1C(O)C2O c1(C(=O)NC2C3CN(C(=O)Cn4cccc4)CC23)cnc2cc[nH]c2c1 C1(CC(=O)NC)CN(C(=O)C(CO)OC)CCN1C(c1cc(O)ncn1)=O C1(C(=O)N(CCCNC(c2cc(C)nn2C)=O)CCO)(OC)CCCC(C)(C)C1 CS(=O)(=O)C1CN(C(=O)CCC2OCCO2)CC1NC(C1CC(C2CC2)=NO1)=O Cn1ccc2c(C(N3CC4CC(NC(c5ccc[nH]5)=O)C(C4)C3)=O)ncnc12 CC1(NC(=O)CC2COCCO2)CCN(C(=O)CC2CC3(CC3)C2)C1 C1(CC)(NC(=O)CCF)CCN(C(C2CCC3CC3CC2)=O)CC1 CON1CCC(=O)NC2(CC1=O)CCCCC2C.C1(COC)CC(F)(F)CO1 C1(CN(C)C(c2ccnn2C)=O)CC(O)CCN1 N1(C(CCC#C)=O)CCCCC1CC(=O)NCCOCC(F)F c1(C(=O)NCCC2N(C(c3c(CC)nco3)=O)CCCC2)cccc(S(C)=O)c1 C1(CNC(c2c(C)cc(O)nn2)=O)CC2CCC(C1)N2C(=O)CCc1ncc[nH]1 Cc1c(C(=O)NC23CCN(C(=O)CSc4cccs4)CC2C3)[nH]c2c1CCCC2 C1(COC)CN(C(c2cn[nH]c2)=O)CCN1C(=O)CCc1cccnc1C c1(C(C)(C)NC(=O)NC2CC(C3CC3)C2)cc(Br)ccc1F CC1(C)CC(C(=O)NC2CCCC(O)C2)(CNC(=O)Cc2ccco2)C1 O=C(CCCCCCCBr)Nc1cnn(Cc2ccccc2)c1.C12CN(C1)C2=O CCC(C)C(C(=O)N1CCCC(NC(=O)Cc2ccc(Cl)cc2Cl)C1)OC Cc1ccc(C(=O)NCC(C(C)C)NC(=O)CCc2ccnc(C)n2)nc1 N1(C(=O)C(F)F)CCN(C(c2csc(-c3ccccc3)c2)=O)C2(CCCC2)C1 C1(C#N)(CC)CCN(C(C2(CF)CCN(C(c3ncccn3)=O)C2)=O)CC1 N#Cc1sccc1C(=O)NCCN(C(=O)C(F)=CCCF)C1CCCC1 C1(C(=O)NCC2C=CC(NC(CC(CCSC)O)=O)C2)Cc2ccccc2C1 C(CC)(C(=O)NC(CC1CCC1)C(=O)N(C(C)CN(C)C(C)=O)C)=CCCC N(C(=NCc1nc(C(C)(C)C)co1)NCC1CCCCO1)CCC#C CC(C)C(CCNC(=O)COCC)NC(=O)CCC1CCCCCC1.C(=O)(C(C)(C)F)N C1(C(=O)NC2CCC(NC(C3CCCN(C)C3)=O)C2)C2CC3C(C2=O)C13 C1(CC(=O)NC2CCC(CNC(C(C)n3cnnn3)=O)C2)CCCC(C)C1 N1(C(c2c(C)cncn2)=O)CCOC(C)(CNC(=O)CC(F)F)C1 N1(C(C(C=C)O)=O)CC2CCC1C1CN(C(c3c[nH]cc(Cl)c3=O)=O)CC21 c1(C(=O)OCC)ccc(C(=O)NCCCNC(=O)CC(CC)SC)nc1 C=CC(C)(CC)C(=O)OCc1ccnc(C)c1O C1(N(C(CCOC2CN(C(c3c(CC)cco3)=O)C2)=O)C)CCOC(C)C1 c1(SC(C)C(=O)NCC(O)CNC(=O)CCn2cncn2)ccccc1C#N c1(C(N2CC(CC=C)(NC(=O)Cc3cncnc3)C2)=O)ccc(OCC)c(N)c1 N1(C(=O)CC2CCN(Cc3nc(Br)cs3)C2)CCC(c2ncc(Cl)cn2)CC1 c1(CCC(=O)NC2C(C(=O)NOc3ncccn3)C2)cnc2ncccn12 O=C1NC(=O)C(CC(N2CCCCC2CC(N2CC(C=O)C2)=O)=O)N1.C1CC1 CCCC(CC)CCC(=O)N1CCC1CNC(c1ccc(C)c(OC)c1)=O C(c1cnccn1)=CC(=O)NCC1C2CN(C(C3CCC(=O)N3)=O)CC12 N1(CC#N)CCN(c2ccc(Br)cn2)CC1.Cn1cc(C(C(F)(F)F)NC(=O)N)cn1 c1(C(C2CC2)NC23CC(C(N(C(C)C)Cn4cccn4)=O)(C2)C3)cc(Cl)c(O)cc1F C1(C(=O)NC(C2CCOCC2)(C)C)C2CC3C(C2NC(C2CC(CC4CC4)C2)=O)C13 C=C1CC2CCC(C1)N2C(C(=O)NC1CC1)C(C)Cc1ccccc1 C(C(C)(C(=O)N1CCC(C(C)C)CC1)NC(=O)Cc1ncn(C)c1C)SC C(=O)(C(C)(C)CC(C)C)NC(CCCC)CNC(=O)C(C)(C)NS(C)(=O)=O c1(C(=O)NC2CN(C(C(CO)N(C)C)=O)CC2(C)C)cc2c(nn1)CCOC2 N1(C(CN(C(c2c(C#C)cn(C)n2)=O)C)=O)CCOC2CCCCC12 N1(C(c2cc(C)sc2C)=O)CCC2(C1)CN(C(=O)C(C)NC=O)C2 C1(NC(C(CN(S(C)(=O)=O)C)C)=O)CCCCN(C(=O)Cc2cscn2)CC1 C1(NC(Cc2cncc(C)c2)=O)CCN(C(c2cn(CCO)nc2C)=O)CC1F C1(C(=O)Nc2scc(C#N)n2)C2C(CN1C(c1cscn1)=O)C2(C)C c1(C(=O)NC2CCN(C(CSC)=O)C2C2CC2)noc2c1COCC2 C=CC1(C(N2CC(c3nncs3)C2)=O)CCN(C(c2ccnnc2)=O)C1 C(CC(C(C)(C)C)NC(=O)CCCF)N(C)C(c1cccc(NC(N)=O)c1)=O C(=O)(C(O)C(C)C)N1CCC(CC(=O)NCc2cnn(CC)n2)C1 N1(C(C(COC)NC(=O)COc2cccnc2)=O)CC2CC(CO)C(C2)C1 C1(NC(CCC(C)OC)=O)CCC2(CC1)CC2NC(=O)CCN1C(=O)CCC1=O C1(C(C)NC(=O)CCC2CCC(=O)N2)CN(C(c2ccn(CCF)n2)=O)CCO1 C(N=c1[nH]c2cc(C)ccc2o1)C1(NC(c2cc(C)nc(C)n2)=O)CCCC1 CN=c1ccc(C(=O)N(CC(=O)NCC2CCCOC2)CC(C)C)c[nH]1 c1(C(=O)NC2(CNC(c3cn(CC(C)C)nc3)=O)CCC2)sccc1C#N C(c1ccn(C)c1)=CC(=O)N(CCC(N1CCC1(CC)CC)=O)CC#C Cc1cc(=NCc2nc(-c3ccco3)n[nH]2)[nH]c(=NCCc2ncc(C)o2)[nH]1 C1(n2cc(CCC(C)O)nn2)CN(C(=O)Cc2c(I)cnn2C)CC1C C1(C(N(C(CCNC(c2c(C)nc(C(F)(F)F)o2)=O)C)C)=O)C(F)(F)C12CCC2 Cc1ccc2c(C(=O)NC(C3CCN(C(c4c(C)coc4C)=O)C3)C)coc2c1 CCC(CC)CC(=O)N(CCC(=O)NCC1CCN(C)C1=O)CCO C1(NC(CCC2OCC(C)(C)C2)=O)CCC2CN(C(=O)C3=CCCSC3)CC12 N1(C(CC2(C=C)CC2)=O)CCC(C(F)F)(CNC(=O)Cn2cnccc2=O)C1 C1(CCOC)(NC(c2cc(Oc3ccc(Cl)cc3)n[nH]2)=O)CCN(C(C)=O)CC1 Cc1cc(C(N2CCOC(CN=c3cc(Cl)c(O)n[nH]3)C2)=O)ccc1S(N)(=O)=O C(C)(CCC(=O)N1CC(CNC(C2CCN(c3ncccc3Cl)C2)=O)C1)OC c1(C(=O)NC(C)(C)CNC(C2CC2C2CC2)=O)cccc(Br)c1 CC1(C)CN(C(C2(C)COC(=O)C2)=O)CCC1NC(=O)C=C(Cl)Cl C(=O)(C(O)CC[S+](C)C)Nc1ccc(C2(C(=O)OC)N(C(CC)=O)CCC2)cc1 C1(CC(N2CCC(OC)C2C)=O)C2CCCC2N1C(=O)COC1CCOC1 N1(C(C23CCC(C(=O)OC)(C2)C3)=O)CCN(C(C)=O)C2CC12 C12(C(=O)NC(CC(C)NC(c3coc(C#N)c3)=O)C)C3CCC(CC13)C2(F)F C#Cc1ccc(Cl)c(C(N2CC(CC(C)NC(c3ccncc3OC)=O)C2)=O)c1 c1(C2CCCN(C(c3ccc(F)cc3Cl)=O)C2)nc2ccc(F)cc2o1 c1(OC)c(C(=O)NCCCn2cc(CC3CCOC3)nn2)cccc1F c1(N2CC(NC(C(C)(F)F)=O)CC3(C2)CC3)nccc(C(N)=O)c1[N+](=O)[O-] c1(C2C(C(=O)N(c3ccccc3)c3ccccc3)C2)cccc(Cl)c1 N1(C(C2C(NC(CCC#CC)=O)COC2)=O)CCC(F)(C#N)C1 Cc1coc(C(=O)NCCOC2CCN(C(=O)CC3CCC(=O)NC3)C2)c1C C1(C(C)NC(=O)Cc2ccsn2)CCCN1C(=O)C(c1cnn(C)c1)O c1(NC(=O)NCCC(=O)NC2NCC(C)C2)ccccc1Br C1(C(=O)NCC(C2CCC2)NC(c2cnc(OC)s2)=O)CCOC(=O)CC1 CC(C)C(O)C(C)C(=O)NC1(CNC(=O)C(C)(C)C(F)F)CC1 c1(NC(C2CCN(C(=O)NCCCC)CC2)=O)ccc2occc2c1 C1(C23CC(C)(C2)C3)CC(F)(SCCNC(C(C2COC2)OCC)=O)C1 c1(C(N(C(C)CNC(C2CCC3(CCC3)C2)=O)C)=O)cccc2[nH]ncc12 C1(CC(=O)NCC(C)(C2CC2)NC(COCC)=O)CCC(F)(F)CO1 CCCCC(CC)CC(=O)N(CCNC(=O)COC(F)F)CCOCCO C(N=c1cccc(S(=O)(=O)N(C)CC2CC2C)[nH]1)c1cc(OC)c(Br)cc1 C12(NC(COCC)=O)CN(C(=O)CC3CCC4(CCC4)O3)CC(F)(C1)C2 C1(=CC(N2CC(NC(C(C=C=C)C)=O)C(C)C2)=O)CCCCCC1(F)F Cn1nc(C(F)(F)F)cc1C(=O)N(C(C)(C)C)CCC.N12CCCC(C1)C2 C1(NC(c2ccc(C)c(C)n2)=O)CCCC12CN(C(=O)Nc1cccc(Cl)c1)C2 N1(C(c2c(CC)csc2)=O)CC(NC(C2(C)CC(O)C2)=O)CC1C c1(C(N2CC(NC(C3(F)CCOC3)=O)C3CC3C2)=O)cc(Cl)c2[nH]c(O)nc2c1 C(=O)(CC(C)C(C)C(C)C)NC1CC(NC(C=Cc2c(C)ncs2)=O)C1 c1(C(N(CCN(C(c2ccc(C)nc2)=O)CC)CC)=O)ccnn(C)c1=O c1(C(=O)NCCCCN2CCCC2)csc(CNC(C2(O)CCSC2)=O)c1 N1(C(c2n[nH]c(C)c2Cl)=O)CCC2CCN(C(=O)C(C)(C)CN(C)C)CC2C1 CCC(C)(CNC(c1n[nH]cc1C)=O)C(=O)NC1COCC(C)(C)C1 c1(OCC(=O)NC2CCC(C)(NC(C3C=CCC3)=O)CC2)ccc(C#N)c(Br)c1 C1(C(NOCCC(=O)OC)=O)(NC(c2ccc(C)nn2)=O)CCc2cc(Br)ccc2C1 C(C(C)C(=O)N(CCCNC(=O)Cc1cncn1C1CC1)C1CC1)OC C1(O)(Cn2cc(CSC(C)C(=O)O)nn2)CCCC(C)(C)C1 c1(CNCC(n2cc(Br)cn2)C)ccc(C(=O)OC(C)(C)C)nc1 N1(C(CCN(C)C)=O)Cc2[nH]nc(-c3csc(C(F)(F)F)c3)c2C1 c1(Nc2nccc(=NCC3(OC)CC3)[nH]2)cc([N+](=O)[O-])cnc1C c1(SC)ccc(-c2nc(C3CC(C)CS3)n(-c3c(C)noc3C)n2)cc1 c1(C(N2CC=C(C(=O)NCC(C(CC)C)C)C2)=O)c[nH]c2cnccc12 CCC(CC(=O)NC1CC(NCC(=O)OC)C1)C1CC1.N12CCC(=CC1=O)CC2 C12(C(=O)NCCC(C)N(C(C3=C(C)CCCC3)=O)C)CCC(C1)c1ccccc12 C1(NC(CC(CC)(F)F)=O)CN(c2nc(Cl)ncc2[N+](=O)[O-])C2CCCCC12 c1(CC(=O)NCC(CC=C)NC(c2ccc(C)cc2F)=O)cc(F)cc(F)c1 c1(OC)nccc(Br)c1C(N1CCCC1CNC(=O)C(C)c1cncs1)=O c1(C(=O)NCCC(C)N(C(CSCCCC)=O)C)ccc(C)cc1OCC Cn1c(C(F)(F)F)nnc1NOCc1nccn1CC(F)(F)F N1(C(C(C)c2cc[nH]n2)=O)CCC(C)(NC(=O)CCOCC(F)(F)C(F)F)CC1 N1(C(c2cnc(C)[nH]2)=O)CCC2C(CCCN2C(c2cccc(F)c2C#N)=O)C1 C1(NC(c2c(C)nc(C)s2)=O)C2CC3CN(C(=O)C#CC4CC4)C1C3C2 N1(C(Cn2ncc(CC)c2)=O)CCC(C)C(CNC(c2nscc2C)=O)C1 c1(C(=O)NCC2N(C(c3c(CC)cns3)=O)CC(F)C2)cnc2c(cnn2C)c1 N1(CC)CCOCC1C(=O)NCCC(C)(C)NC(c1cscn1)=O c1(C(N2C(CN(C(=O)C(C3CC3)OC)CC)CCC2)=O)cnc2ccc(F)cc2c1 c1(CNC(=NCCC)NC(C)CC(=O)NC(C)(C)C)ccc2nnn(C)c2n1 N1(C(C2CCCN(C(COC)C)CC2)=O)CCC(C2CCN(C)C2)C1 CC(CN(C)C)C(=O)NCCCCC1CCN(C(=O)CCNC(=O)CO)C1 N1(C(c2cnn(CCOC)c2C)=O)CCC(CNC(=O)CCS(C)(=O)=O)CC1C C1(NC(c2c(OCC)scc2)=O)CCN(C(c2cncc(Cl)c2Cl)=O)CC1C c1(CC(=O)N(CC(CN(C(=O)CSC2CCCC2)C)O)C)ccc(Cl)s1 C1(CC#C)(C(=O)N(C2CC3CC3C2)C)CCN(C(c2n[nH]cc2OC)=O)C1 c1(OC)cnnc(C(=O)NC(C)(C)CC(=O)N2C(CO)CC2CO)c1 C#Cc1cccc(C(=O)NC(c2cccnc2)C(=O)N(C)Cc2ccco2)c1 N1(C(C(C2CCOC2)OC)=O)CCC(CF)(NC(=O)C2=CCCS2)C1 N1(C(c2c(C)cco2)=O)CCN(Cc2nccs2)C2CC12 C1(NC(c2cc(C)sc2C)=O)CCN(C(C2(CO)COC2)=O)CC1O c1(CC(=O)NC2(CN(C(=O)Cc3cnnn3C)C)CC2)c(F)cccc1Cl CC(C)C(F)C(=O)N(CC(=O)NC1CC(C)(C)C1)C(C)C c1(NC(C2(C)CCN(Cc3ccsc3)CC2)=O)cc(F)cc(C#N)c1 C1(C(N2CC(CCCCNC(C(N)=O)=O)C2)=O)CCCC2(CCC2)C1 C1(C)(C)CC(F)C(=O)N1.C[Si](C)(C)CCCc1cn(CC2(O)CCC2)nn1 c1(CC)ccc(C(C)=CC(=O)NC2CCN(C(=O)CC(COC)COC)C2)cc1 N1(c2ncc(CCC)cn2)CCC2(CNC(C3(CO)CCCO3)=O)CCCCC12 c1(OCC)cc(CN2CCCC(N(C)C(c3cccc(C)n3)=O)C2)ccc1Cl N1(C(C(CCNC(C(C(CC)C)C)=O)(C)C)=O)CC2CCCC(C2)C1 CC(C)CCCCC(=O)NC1CN(C(=O)CCc2cccn2C)CC1C1CC1 CCCC(O)C(=O)NC1CCN(C2CCN(C(=O)NC3CC4C=CC3C4)C2)CC1 CC1CC(CO)CN(C(c2conc2CNC(=O)CN2CC=CC2)=O)C1 N1(C(CN(C2CCC2)C)=O)CCN(C(=O)CCc2ccc(F)cc2Cl)CC(O)C1 C1(C(N(CC#C)C(C)C)=O)CCN(C(=O)C=CC=CCC)C1 c1(N(C)C(C2(n3cc(N)cn3)CC2)=O)cc(F)c(C(=O)O)c(F)c1 C12(NC(C(C3CCC3)OC)=O)CC(CNC(C3CCC=CCCC3)=O)(C1)OC2C Cc1cc(CNC(=O)Cn2cncn2)oc1C(=O)NCC1(C(C)C)CCCC1 N1(C(C2CCN(C)C2)=O)CCC12CCN(C(c1ccccc1Cl)=O)CC2 C1(NC(C=C(C)C)=O)CC(F)CN(C(=O)Cc2cc(Cl)cc(Cl)c2)C1 c1(NC(N2CCC(C(N3C(C(C)C)C(C)(C)C3)=O)CC2)=O)cccc2oncc12 C=CCC(CC(F)F)C(=O)NCC1(CN(C(=O)C=CCC)C)CC1 C(C(=O)N=c1ccn(C(C)(C)C)[nH]1)OC(C(C(CC)C)c1ccccc1)=O c1(C(C(=O)NCC(F)F)N(C)Cc2c(C)noc2C)cc(Br)cc2cccnc12 C(c1ccc(F)cc1)=CCC(=O)N.N1(C(C2(CC=C)CC=CC2)=O)CCN(C)CC1 c1(C(=O)NC(C)CN(C)C(c2ncoc2C2CCCO2)=O)cc2ccccc2o1 C#CCCCCCNC(=O)C=C(C)CNC(C1CC1C1CC1)=O c1(CC)cccc(F)c1NC(=O)NC12CC1CN(C(c1cncc(C#N)c1)=O)C2 CS(=O)c1ccc(CC(=O)NC2CCC2NC(c2ccccc2O)=O)cc1 N1(C(C(C)OCCCCCC)=O)CC=CC(NC(C2CCC2=C)=O)C1 C(=O)(C(C)CCN(C)C)N1CC(CC=C)(NC(c2oncc2COC)=O)C1 C(CNC(=O)C=CC1CC1)(CC(=O)N1CC(CC(N)=O)C1)OC Cc1cc(Cl)ccc1C(=O)NCC1(O)CCN(C(C2(N(C)C)CCCSC2)=O)C1 c1(CC)ccc(C(=O)NCC23CC2CN(C(c2oc(CC)cc2C)=O)C3)c(Cl)c1 C1(C(=O)NCC(CO)OCC)CC12CC(NC(=O)CCNC(C)=O)C2 C1(C(=O)NC(C2CN(C(C(CC)(C)C)=O)C2)C)CCOCC12CCCC2 N1(C(c2ccc(C(C)=O)nn2)=O)CC2=C(C1)CN(C(=O)CC(F)(F)C(F)F)C2 c1(C(=O)NCCN(C(C2(C)CC2C(F)(F)F)=O)CC)ccc(C(F)F)cc1 C(=O)(C(C)S(N)(=O)=O)NCCCC1N(C(C(CC)OC)=O)CCCC1 [N-]=[N+]=NCC(=O)NCc1cc(C(=O)NCC(c2ccco2)O)co1 C1(C(N2CCC(CC=C)(NC(c3scnc3CC)=O)C2)=O)CC2CCC(C1)C2 Cc1nc2c(C(N3CCC(NC(=O)CCNC(N)=O)CC(O)C3)=O)cccc2o1 C1(F)(C(=O)NCC2(C)CN(C(c3cccc(Br)c3)=O)C2)CCOCC1 N1(C(c2cc(C)[nH]n2)=O)CCC2(CC1)CC2C(=O)NCCS(C)(=N)=O c1(CC)ccccc1C(N1CC(C(=O)N(C2CCCC2(C)O)C)C1)=O C1(C#N)(C(=O)NCc2ccc(CNC(C(C)(C)OCC)=O)cc2)CCSCC1 c1(C(C)(C)C)nocc1C(=O)NC1CCN(C(c2cccnc2)=O)C1 N1(C(C(COCC)NC(C(F)=CCC)=O)=O)CC(C(=O)NC)CC(C)C1 c1(C(C)N(C(C=CC=CC)=O)C(C2CCCN2CCN=[N+]=[N-])=O)ccc(F)cc1 C(=O)(C1=CNC2=NCCC2=C1)N1C(CNC(C2C(CC)CCO2)=O)COCC1 O=C(CCCOC1CCC1)NC(CNC(=O)Cc1cccnc1)C1CC1 CC(C)(CC(=O)NC1CN(C(c2cc3cn[nH]c3cn2)=O)CC1CO)CC(F)F c1(CC(N2C(CN(C)C(C3CC4CCC3C4)=O)COCC2)=O)cccc(F)c1F Cc1nn(C)c(Cl)c1C=CC(=O)NCC(CNC(c1nccn1C)=O)CO c1(CC(=O)NCC(C2CCCC2)NC(C=COCC)=O)ccc(F)c(F)c1 C1(C(N(CCN(CC(NN(CC)C)=O)C)C)=O)CCCCCC(=O)C1 C1(C(=O)NCC2(CNC(CCCCC#C)=O)CCC2)CCC2(CC1)OCCO2 Cn1cc(Cl)c(CC(=O)NCCC2(C(=O)NCC(CO)C3CCC3)CC2)n1 C1(NC(c2c(CC)noc2)=O)CCC2CCN(C(=O)C(N3CCNC3=O)C)C1C2 C12(NC(c3cc(CC)no3)=O)CCCCC1N(C(=O)CCc1ccc(C)s1)CC2 C=CCC(CC(=O)NCC12CC=CC(C1)OC2)NC(C12CCC(C1)C2(C)C)=O C12(C(=O)NCC(C)N(C(=O)CSCCC#N)C)CC(C)(C1)OC21CCC1 c1(CC)cc(C(=O)NC2CC3(C2)CC3NC(c2csc(CO)n2)=O)cc(N)c1 c1(CCn2c(C3(N(C)C)CCCC(C)C3)nnc2C(=O)NC)ccc2c(c1)OCO2 c1(NC(C2CC23CCSCC3)=O)ccc2cc(-c3ccccc3)[nH]c2c1 c1(C(C)NCC(O)CO)cccc(S(=O)(=O)NCc2ccc(Cl)c(Cl)c2F)c1 CC(C(=O)NCC1CC2CN(C(=O)CC3OCCC3(C)C)CC12)C(C)(C)C Cc1ccsc1C=CC(=O)NCC1(CCCNC(=O)Cn2cnnc2)CCCC1 c1(CC(N2CC(N(CCO)C(c3cccnc3)=O)C(F)C2)=O)c(F)cccc1F c1(NC)cncc(C(N2CC(CCCCNC(C3CC(C)C3(C)C)=O)C2)=O)c1 c1(CCC(N2C(C(=O)Nc3ccc(F)cc3O)CCC2)=O)ccccc1[N+](=O)[O-] N1(C(COC)=O)CCC(NC(=O)C(C(C)C)n2cnc(C)c2)C(C)(C)C1 C1(COC)(NC(c2cc(O)nn2C)=O)CCN(C(=O)Cc2cc(C)nn2C)C1 C12(CC(=O)NC3C(NC(CCN(CCC)C)=O)CCC3)CCCN1CCC2 C1(C(=O)NCC2CN(C(c3n[nH]c(C(F)(F)F)n3)=O)CC2O)CC2CCC1CC2 CC1CCCC(CC(N2CCC2CNC(C2(CC(F)F)CCC2)=O)=O)O1 C(=O)(CCC(C)(C)C)NC1C=CCN(C(c2c(CC)cno2)=O)C1 N1(C(=O)C=Cc2ccc(Cl)s2)CC2(CC(NC(=O)C(F)(F)CO)CO2)C1 Cc1cc(C(=O)NCC(C(C)C(C)C)NC(C2CCS(=O)(=O)N2)=O)ncc1Cl Cc1cc(=NCCCCS(N)(=O)=O)[nH]cc1S(=O)(=O)NCCC1(CO)CC1 N1(C(Cc2cccc(OCC)n2)=O)C2CCC1CN(C(=O)C(C)NC=O)C2 n1(CC)ncc2cc(C(=O)NCCCN(C(=O)C(C)(C)O)C(C)C)cnc12 CCCC(C)(CC)C(=O)NC1CCC(C(N2CC(=O)NC(C)(C)C2)=O)C1 C1(CC=C)(C(=O)N(CCCn2ccnc2)C2CC2)CCN(C(=O)C(F)C2CCC2)C1 Cn1nnc2c1C(C(=O)N1CCC1CNC(=O)Cc1cccc(F)c1)CCC2 C12(NC(=O)Cc3csc(S)n3)CC(CNC(C3CC3c3cccnc3)=O)(C1)C2 CC(C)C(C)(CNC(=O)CN1C(=O)CNC1=O)NC(=O)C(O)CF c1(OCC)ccc(C(=O)NC(CO)C(C)c2ccccc2)c(C)c1 c1(C(N2CCCC(N(C(c3csc(C)c3C)=O)CC)C2)=O)c(OC)ccnc1O C(CCCC(=O)NC1CC(n2ccnn2)C1)NC(C(CC)SC)=O C1(C(N(C(CNC(c2cn(CC)nc2C)=O)C)C)=O)CC2(C1)CC(F)(F)C2 C1(O)(CC=C)CCN(C(=O)CC(COC)NC(=O)C(O)CCSC)CC1 c1(CN2CC(C(=O)Nc3ccccc3)SCC2)c(Cl)cccc1I N1(C(Cc2cccc(COC)c2)=O)CCN(C(=O)Cc2n[nH]c(C)n2)C(C)C1C c1(C(=O)NCC(CNC(=O)CC2CC2C(F)(F)F)OC)cc2c(s1)CN(C)CC2 N1(c2cc(C)c([N+](=O)[O-])cn2)CC2C3CCC(C2C1)N(C(=O)CN1CCOC1=O)C3 C1(OC)CC(CNC(=O)CCC2CCOC2)N(C(=O)Cc2cc[nH]c(=N)c2)C1 c1(C(N2CC(F)(Cc3ccc(Cl)cc3)C2)=O)ccnc(OC2CNC2)c1 c1(CC)cc(F)ccc1C(=O)NCCCC1CN(C(c2[nH]ccc2C)=O)CCO1 C1(CC(=O)NCC(CNC(c2c(C(C)C)con2)=O)(C)F)CC=CCN1C C(C1c2ccccc2CN1C(=O)CCC(N)=O)NC(c1c(C)n2c(s1)cnc2)=O C12(NC(C=Cc3n(C)ncc3)=O)COCCC1CN(C(=O)Cc1cccs1)C2 N1(C(c2c(CC)cco2)=O)CCN(C(c2coc(Cl)n2)=O)C(C)CC1C C1(C(N2C(CNC(CC(CCC)O)=O)(COC)CCC2)=O)CC2(CCCC2)CO1 C(C(O)(C(=O)NCCCNC(=O)Cc1nc(F)c(F)cc1F)C(F)(F)F)N(C)C c1(CC(=O)NCCC(C)NC(C(C)OCC)=O)cc(OC(F)F)ccc1F C1(C(N(C(C)(C)CC(=O)NCCC(O)C(F)F)C)=O)C2CN(C)CC12 N1(C(C(C)OCC2CC2)=O)CC2(CNC(=O)C3=CS(=O)CCC3)CCC1CC2 c1(CCC(=O)N(CC(CC)NC(C2C=CCC2)=O)C)nc(CSC)no1 CCCCC(COC)N=c1nc2scnc2c(N2C3CCC(C3)C2CO)[nH]1 C1(CNC(C(C)OCC=C)=O)CN(C(c2cnc(N(C)C)s2)=O)CC1O c1(C(N(C)CC2CCN(C(=O)C=Cc3ccco3)C2)=O)noc2c1COCC2 C(=O)(CS(N)(=O)=O)NCCCN(C(C1C(C(=O)OC(C)(C)C)CCO1)=O)CCO c1(C(=O)NCC2CCN(C(C(C)SCC)=O)C2)n[nH]c2c(C)cccc12 N1(C(=O)C2CC2)CCN2CCCCC1C2.c12ccoc1CNC2=O c1(-c2nc(CCSC)nn2-c2cccnc2C)cccn2nnnc12 N1(C(COC2CN(C(C(C#C)(C)C)=O)C2)=O)CC2(CCN2C)C1 S(=O)(=O)(c1ccccc1F)NCCSCC(N1CC(C(=O)OC)OCC1)=O C(=O)(CC(C)CCCCC)N(C1CCC(NC(CCCCC#C)=O)CC1)C N1(C(C=CSC)=O)CCCC(N2CCN(C(=O)COCC3CCCC3)CC2)C1.OC n1(CC(=O)NCC(C)(C)CNC(C2(CC3CC3)CCC2)=O)cc2ncccc2n1 N12CCC(C)(C1)CC=CC2=O.C(C(C)(C)CSC)NC(CC1CC(=C)C1)=O C1(C(=O)Nc2n(C)nc(C3CC3)c2)CCCN(Cc2cc[nH]c3nccc2-3)CC1 C1(C(=O)NC(C(=O)NCC2(COC)CCCO2)CC2CCC2)C2CN(C)CC12 c1(-c2n(Cc3cc(OC)ns3)c(N(C)C)nn2)nn(C)c(=O)c2ccccc12 Cc1cn2c(n1)CCC(C(=O)N(C1CCN(c3ncnc(Cl)c3F)C1)C)C2 c1(CCNC(N2CCC(c3cncs3)CC2)=O)ccc2cc[nH]c2c1 N1(C(CNC(C(CSC)C)=O)=O)CCOC(NS(C)(=O)=O)C1 c1(C(=O)NCC(CC)NC(c2nncs2)=O)ccccc1SC(F)F O=C1NCC2(CCN(S(=O)(=O)CC3CCC(F)C3)C2)O1 CN(CCc1ccc(C(N)=O)cc1)N1CCc2[nH]nc(N(C)C)c2C1 O=S1(=O)CCC2(CCN)CCN2N1CC1C(COCC(F)(F)C(F)(F)F)C1 CC1=CCN(C(C2CC(C)N2C(=O)Cc2ccc(F)cc2)=O)CC1 CC(C(=O)N1CCC(C(N2CCC(O)C2)=O)O1)c1ccsc1 c1(OC)ccc(C(=O)NC2CN(c3cncc(C#N)n3)CC2C)c(I)c1 c1(OC)cc(OC)c2sc(=NCc3cccc4ccccc34)[nH]c2c1.c1(C)ccccc1 C1(NC(CNC(=O)NC)=O)CC=C(C(=O)N2CCC(C)(N(C)C)C2)C1 n1(C(C)C(=O)NC2CCC(N(C(=O)CO)C)C2)cnc(C#N)n1 C1(C)(NC(c2nnc(CC)s2)=O)CCCN(C(c2cc(CO)[nH]n2)=O)C1 C1(CNC(C=C(COC)C)=O)COCCN1C(c1ncc[nH]1)=O C1(C(N(C(C)C)CCNC(=O)C(c2ccccn2)N(C)C)=O)OCCCC1(C)C C1(NC(C(n2c(C)ccn2)C)=O)CCN(C(=O)CCC(=O)NC2CC2)C1C1CC1 C1(C(=O)NC(CCCC=C)C2CC2)CCC2CCC1N2C(c1ccccc1C)=O C(=O)(CC(O)CC(C)(C)C)NC1(C(N2CCSCC(C)C2)=O)CC(O)C1 Cc1cc(F)ccc1C(F)(F)C(=O)NCC1CCCCN(C(=O)C(O)C(C)(C)C)C1 c1(C(=O)NC2CC3CC(NC(=O)C=CCF)C3C2)ccc2scnc2c1 c1(N2C(CCCCC(=O)NC)CCC2)cc(C(N2CCCC2CO)=O)ccc1O.CO Cc1noc(Cl)c1CC(=O)NC(C)CC(C)NC(=O)Cc1ncc(Cl)s1 C1(NC(c2ccc(COC)o2)=O)CCCC12CN(C(=O)CN(C)C1CC1)C2 c1(CC(=O)NCC(CNC(CC(=C)C)=O)O)ccc(S(C)(=O)=O)cc1 C(=O)(CC(C)C(F)(F)F)NC1C(CC)CN(C(c2nccnc2C(=O)OC)=O)CC1 C1(CC=C)(NC(C2CCCOCC2)=O)CC2CCC(C1)N2C(C1CC1OC)=O C12(NC(C(C3CCN(C(c4cc(Cl)ncn4)=O)C3)C)=O)CCC(CC1)CC2 c1(C(=O)O)ccc(S(=O)(=O)N(C2(c3ccccc3)COCCO2)CCO)cn1 C1(C(N2CCCC(O)(CCNC(C3C(OCC)C3)=O)C2)=O)CN2CCCC2CO1 c1(C(N(CC(CNC(CCN(C)CC)=O)O)C)=O)c(C)c(C)nc2ccccc12 N1(C(C2C(CC)C2)=O)C2CCCC1CN(C(c1c(Cl)noc1C)=O)CC2 NC(=O)CCC(=O)N1CC(F)CC1CCNC(C1CCNC(=O)C1)=O C1(NC(C(CC2CCC2)N(C)C)=O)CCCCC1NC(C1(CO)COC1)=O C(=O)(C(COC)CC(C)C)N(CCCNC(c1c(C)nc(CCC)s1)=O)CC c1(C(N2CC(CC)C(NC(C3(C)CC=CC3)=O)C2)=O)cccc(Br)c1Cl C(=O)(C1=C(Cl)CCC1)N1C(CC(=O)NCCc2n(CC)ncc2)CC(F)C1 C1(C(N2CCC(CCNC(C(CC)=CCCC)=O)CC2)=O)CC2COCC(C1)C2 N1(C(c2c(C)nc(Cc3cccc(Br)c3)o2)=O)C2CCC1CN(C)CC2 C1(C(=O)NCC(CC(C)C)NC(C2(C)C(C)(C)C2(C)C)=O)CCCC(C)(C)C1 Cc1cc(C(N2CC(CC(C)NC(C3CC(F)CN3C)=O)C2)=O)c(C)cc1C C1(C(=O)NC(C#C)C)CC(O)CN1C(=O)C(C(C)C)N(CC)CC c1(C(=O)NCC2C(NC(C3C(OC)CC3)=O)COC2)cncnc1C N1(C(COCCN(C)C)=O)CCOC(C)(CNC(C2CCC(C)(C)CC2)=O)C1 c1(C(N(C)CCNC(C2CCCC2P(C)(C)=O)=O)=O)ccnc2c1cnn2C Cc1nn(C)c(C)c1C(=O)C(N1CCN(C(C2CC(=O)NC=CC2)=O)C(C)C1)=O c1(CC)nnc(N2CC(C)(C)CC2CNC(=O)CN2CC3C=CC2C3)nc1CC C12(NC(c3c(C)nn[nH]3)=O)CCCN(C(=O)C(C)(C)C)CC1C2 C1(NC(=O)CSC(F)(F)F)CN(C(=O)CCc2ccoc2)C2(CCCOC2)C1 CC(F)(F)C(C)(C)C(=O)NC1CCOC(C(N2CCC(F)(F)C(O)C2)=O)C1 Cc1cc(F)c(F)cc1C(=O)NC1CN(C(c2cc(Br)cs2)=O)CCC1F c1(C(N(C2CCCN(C(c3nc(C)[nH]n3)=O)C2)CCF)=O)cnn2c1OCC2 c1(C(N2C(CCNC(C(C(C)C)C)=O)COCC2)=O)ncc(Cl)cc1Cl C(=O)(C1=CCN(C(c2coc(C(N)=O)c2)=O)CC1)NCC1CCC(C)(C)CC1 c1(C(N2C(CC)CN(C(C3(C)CCN(C)C3=O)=O)CC2)=O)cnn2ccn(C)c12 c1(C(=O)NC2CC(F)(CNC(C3C(OCC)C3)=O)C2)ccc(F)c(O)c1 Cc1c(NCc2ccc(N(C)C)c(F)c2)nc[nH]c1=NCC1(C)CC1(F)F N1(C(c2c(C)scn2)=O)CCC2(CC1)CC2NC(c1ccc(Br)o1)=O C1(C(N(C2C(C)(C)C2(C)C)C)=O)CCN(C(c2cocn2)=O)CC1O N1(C(C(CCSC)O)=O)CCCCC(NC(=O)CCc2ncnn2C)C1 C(=O)(CC(C(C)(C)C)NC(c1cc(C)c(O)nn1)=O)N1C(CCC)CCCC1 C12(C(=O)NCC(C3CCCC3)NC(CCC(=O)N(C)C)=O)CCCC(CO1)C2 C(CCCC(=O)N1CC(C)C(C)(C(=O)NC(CO)CCC2CC2)C1)(OC)OC C1(NC(CSCC)=O)CC(C)(CNC(C2(N(C)C)CC2)=O)C1 N1(Cc2c(C(C)C)[nH]cc2)CCC(=O)CC1C1CC1 C1(NC(c2c(Cl)ncc(C)c2)=O)COC2(CCN(C(c3c(C)coc3C)=O)C2)C1 C1(C(=O)NCC2(NC(c3ccc(N)c(Cl)c3)=O)CC2)Cc2cc(Cl)ccc2O1 Cc1ccc2c(=NCC(C)CCO)[nH]c(N3CCC4(CCC4)C3)nc2c1 N1(C(c2c(C(C)C)onc2)=O)CCC2(CCCN(C(=O)CC3C=CCCC3)C2)C1 c1(C(N2CCCC(NC(CCC=CC(C)C)=O)(CO)C2)=O)cnc2[nH]cnc2c1 c1(-c2cccc(CN)c2)cc(O)c2ccc(-c3ccc(C)c(F)c3)cc2c1.Cc1cnc(Br)cc1N N1(C(c2n(C=C)nnc2)=O)CCC(O)(CNC(c2nc[nH]c2C(F)(F)F)=O)CC1 C1(C(=O)OC)C(NC(=O)NC)C2CCCCC12.n1(CC)nnnc1C c1(C(N(CCC)CCNC(c2cccc(C3CCC3)n2)=O)=O)cccc(Cl)c1N N1(C(C(CC)C)=O)CCC(C)(CNC(c2ccsc2Cc2ccc(O)cc2)=O)C1 CC1=NS(=O)(=O)NC(C)=C1CC(=O)NCC1(CNC(C23CCCC2CC3)=O)CC1 c1(OCC=CC)ccc(F)c(NC(C2CC(NC(=O)CC=C(C)C)C2)=O)c1 Cc1ncc2c(C(N3CC4C(NC(c5occc5Cl)=O)C4C3)=O)cccc2n1 N1(C(C2CCCC2O)=O)CCC2CCN(C(C34CC=CCN3CCC4)=O)CC2C1 CC(C)CS(=O)(=O)CCC(=O)N1CC(C)CN(C(C2CCCC(C)C2)=O)C(C)C1 N1(C(Cc2c(C)nsc2)=O)CCCCCCC1C(N1CCN(C)C(C(C)C)C1)=O c1(C(CCC)OCC)nc(-c2ccc(Br)cn2)nn1-c1ccnnc1 c1(C(N2C(CNC(c3c(CCC)n(COC)nn3)=O)CC2)=O)ccn2ccsc12 c1(C(=O)NCC2CN(C(C(n3cc(Cl)cn3)C)=O)C(C)C2)cnc(N)c(Br)c1 c1(NC2CC(C(C)C)C2)ccc(S(=O)(=O)Nc2sc(Br)cc2F)cc1Cl c1(C(N(CCCNC(C(C#C)(C)C)=O)C(C)C)=O)ccc(S(=O)(=O)NC)o1 C=C1CC(C)(C(=O)N(C)C(C23CC(C(N4CCC(N(C)C)C4)=O)(C2)C3)=O)C1 N1(C(C2C(C=C)CC2)=O)CCN(C(c2c(C)sc(C)c2Br)=O)CC(C)(C)C1 CC(O)C(C(=O)Oc1ncccn1)NC1CCCC(NC(=O)CNC(N)=O)CC1 c1(C(N2C(CC(=O)NCC3C4CCCC34)C=CC2)=O)cnn2c1OCC2 N1(C(C(CO)OC)=O)CC2OCCN(C(=O)C(n3ccc(C(F)(F)F)n3)C)C2C1 C(N=c1cc(NC(=O)CN2C(C)CCC2C)nc(C)[nH]1)C1(CC=C)CCCC1 C1(NC(Cc2nc(C)sc2)=O)CCC2(C1)OCCO2 N1(C(c2cccc(C)c2F)=O)C2CCC1C(C)C(NC(c1snc(O)c1Cl)=O)C2 Cc1ccc(C)c(C(N2CCN(C)CC2CNC(c2nc(C)sc2C)=O)=O)c1 c1(C(N2CC(C)(NC(=O)CSC(F)F)C2)=O)ccc2c(c1)NC(=O)CN2 CCC(C)C(O)CC(=O)NCC(CNC(C1CC(=O)N(C)C1)=O)OC C=CCC(F)(F)C(=O)NCCC1CC(NC(c2cccc(-n3cnnn3)c2)=O)C1 C(=O)(C(CNC(=O)C(C)CC(F)(F)F)C(C)(C)C)N1CC(C(=O)NC)C1 c1(OC)ccc(CC(=O)NC2(CO)CCCN(C(c3cccn3C)=O)C2)c(Cl)c1 N1(C(C(COCC)C)=O)CC(CC(=O)NCCCOCC(C)(C)C)CC1(C)C C(C(C)(O)CC(=O)N1CC(CNC(=O)C=Cc2ccc(Cl)nc2)C(C)C1)OC N1(C(c2c(CC)nccn2)=O)CCC(C(N2CCC(C)(CC)CC2)=O)C1(C)C C(=O)(CCC(C)(C)C)CCn1cc(C2N(C(C(CC#C)C3CC3)=O)CC2)nn1.N(C)C CC1CN(C(=O)CC2(O)CCOCC2)CC(C)N(C(C23CC4CC2C3C4)=O)C1 C1(NC(c2cncc3ccsc23)=O)CC2CCC(C1)N2C(C1C2CCCC12)=O CCC(C)C(O)C(=O)NCC(O)CNC(=O)CC(C)N1CCCC1=O c1(OC)ccc(S(=O)(=O)N2CCC(NC(=O)CCCSc3ccccc3)C2)cc1 c1(C(N2C(C)(CC(=O)NCC(C(C)(C)C)OC)CC2)=O)ccc(=O)n(C)n1 CC1Cc2cc(S(=O)(=O)N3CCc4c(Cl)ccc(Cl)c4C3)cc(Cl)c2O1 CC(C)C(C)(O)C(=O)N1CCC(C(C)(C)C)(CNC(c2ncccc2CO)=O)C1 N1(C(CCN(C2CCCCC2)C)=O)C(CNC(C2CCC2(F)F)=O)CC2CCCC12 C1(NC(CN(C(CC(=O)OC)=O)CC2CC2)=O)CCOC(C)C1 C1(C(=O)Nc2cccc(C(C)C)c2)CC(F)CN(C(c2cnnc(O)c2)=O)C1 C1(O)(CC(=O)NC(CCNC(C(CCC)N(C)C)=O)C)COC(C)(C)C1 Cc1ccc(C(=O)NCCC2CC(NC(c3ccc(N)c(Cl)n3)=O)C2)c(=O)n1C c1(C(N2CCN(C(CC(C)(C)SC)=O)CC2)=O)cnc2c(F)ccc(F)c2c1 C1(NC(c2c(CC)nns2)=O)CN(C(=O)C(C)(C)c2ccncc2)CCC1C CC(CN(C)C)C(=O)NCC1(NC(=O)CCCF)CC(OCc2ccccc2)C1 C1(NC(CCC=CC)=O)CCN(C(c2cc(C(=O)OC)c[nH]2)=O)CCC1CO N1(C(CNC(C(C2CN(C(c3nccs3)=O)C2)OC)=O)C)CCOC1=O Cc1ccc(CNC(=O)NC(c2ccc(Br)s2)C)cc1SC1CC1 c1(C(=O)NC(C(C)C)CNC(C23CCCC(CO2)C3)=O)ccc2c(c1)OCCO2 c1(C(N2C(C)CC(NC(C3CCCCS3)=O)C2)=O)cccc2nc(C(F)F)[nH]c12 Cc1cc(C(=O)NC(C2CCN(C(c3nccc(C)n3)=O)C2)C)cc(O)n1 N1(C(=O)NC2COC(C3CCCCC3)C2)C2CCC1c1cc(F)ncc12 c1(C(=O)NC2CC(O)CN(C(c3csc4nccn34)=O)C2)ccn2cnnc2c1 Cn1ncc(C(N2CCCCC2CN=c2ccnc[nH]2)=O)c1S(N)(=O)=O Cc1cnnc(C(=O)NC2C3CC2N(C(c2cn(C4CC4)cn2)=O)C3)c1 Cc1nc(CO)ncc1C(=O)NCC1(O)CCN(C(C2(C)C=CCC2)=O)C1 CC1CC(NC(=O)C=Cc2ccoc2)CN(C(=O)C(c2ccccc2)OC2CC2)C1 C1(NC(C(C)SC(C)C)=O)CN(C(c2ccnn2CCF)=O)Cc2nccn2C1 CCC(C)C(O)C(=O)NC1CC(CNC(=O)C(C)(C)N(S(C)(=O)=O)C)C1 CCC(F)(F)CC(=O)N1CC2CC(NC(=O)Cc3ccc(C(N)=O)cc3)C1C2 c1(NC(N2CCCC(OCCN(C)C)C2)=O)cccc(NCCCC)c1 C(C1=CCCOC1)NC(CC1(C)CCN1C(=O)CC1CCC1)=O N1(Cc2c(F)ccc(I)c2)C2CCCC1CC(N=c1ccnc(N3CCC3)[nH]1)C2 C(=O)(CCCCNC(c1cc(C2(C)CC2)on1)=O)NCCN(CCC)C(C)=O C1(NCCC(C(=O)NCCOC)C)CCCN(c2ccccc2Cl)C1=O C1(C(C)C)CCC(C(N2CCCC2C(C)NC(=O)CC2CC2(Cl)Cl)=O)CC1 C1(CNC(C(CCC)OCC)=O)CCC(C)(C)CN1C(=O)CCC(C)(C)C c1(C(N2CCC(CNC(COCCC)=O)C2(C)C)=O)cnc(O)c2cnccc12 C#CCC(CC(=O)N1CC=CCO1)NC(c1cnc(Cl)s1)=O C1(NC(CC2CCC(C)O2)=O)CCC2(C1)CN(C(c1cn[nH]c1)=O)C2 c1(C(=O)NC(CNC(C(COC)NC(C)=O)=O)CC(C)C)cccc2ncnn12 N1(C(CC(C)NC(c2cn(C3CC3)cn2)=O)=O)CCC(C(N)=O)CC1 c12cnc(c(Br)c1C)C1C(CCCC1)NC(=O)C2N(CCOC)CC c1(C(N2CC3C(C)(NC(CC=C)=O)C3C2)=O)cn(CCOC)c(C)cc1=O S(=O)(=O)(c1cccnc1)N1CC(NC(c2sc(Br)cc2F)=O)C2(C1)CC2 C1(CNC(CCCCC(C)C)=O)CC2(CCN(C(=O)Cn3cnc(=N)[nH]3)C2)CO1 C1(OC)CN(C(=O)CCc2cccnc2F)CC1NC(=O)CCc1cc(C)no1 C1(NC(C(C)N(C(C)=O)C)=O)CC(CNC(=O)Cc2nc(C3CC3)n[nH]2)C(O)C1 C(C)(C)(C(=O)N1CCC(Cc2cn(-c3cccnc3)nn2)C1)SC C1(NC(C(c2cscn2)N(C)C)=O)CCCCN(C(c2cncc(Cl)c2)=O)C1 N1(C(C(C=C)O)=O)CC2CCC(C1)C(NC(=O)C(c1ccc(Cl)cc1)(C)C)C2 C1(NC(C(C)Oc2ccccc2)=O)C2CN(C(C3CC(C(F)F)C3)=O)CC12 c1(-c2c(C(NC3C(c4cn(CCC(C)(C)C#N)nn4)C3)=O)c[nH]c2)c(F)cccc1F CC1CCCC(CNc2cc(CNC(=O)CC=CCc3ccccc3)[nH]n2)O1 CN=c1ccc(C(=O)NCC2CN(C(c3csc(COC)n3)=O)CC2C)c[nH]1 c1(C(N2CC(C)N(C(=O)COC3CC3)CC2)=O)nc(S(N)(=O)=O)c2ccccn12 CC1(C)CCCC(C(N2CCCC2CNC(c2cc[nH]c(=N)n2)=O)=O)C1 c1(C(C(=O)NC2C(C)CN(C(c3ccc(Cl)s3)=O)CC2)=O)cc(F)c(F)c(F)c1 C1(CCC)CCCCC1N=c1cccc(S(=O)(=O)NCC2(CO)CC=CC2)[nH]1 c1(NC(C2N(C(C3(C#N)C(C)(C)C3)=O)CC(=O)C2)=O)ccc(O)c(Cl)c1 c12c(cccc1F)C(=O)N2.C1(NC(C=C)=O)CC(N(C(=O)CCC2CCCO2)C)C1 c1(C=O)ccc(N)cn1.N1(N(CCCC)CCCC)CCCCC1C(F)(F)F N1(C(CSSC)=O)CCC2(NC(=O)Cc3nc(C)sc3C)CCCCC12 C12(C(=O)NCC=CCCC)CCC(CC1NC(=O)CC(C)F)C2 Cc1cc(C(=O)NC2CCCC2CNC(=O)C2=COCCO2)c(C)n1C(C)C C(=O)(C#CC1CCC(=O)CC1)N1CCC(C)N(C(c2cncc(Cl)n2)=O)CC1 C(C(C)(O)C(C)C)NC(CC(C1CC1)NC(c1c(C)nco1)=O)=O c1(C(N2CC(NC(C3CC(=O)N(O)C3)=O)(CF)C2)=O)ccc(F)cc1O C1(F)(CNC(C(C)(F)F)=O)CCCN(C(c2cnc(-c3ccccn3)s2)=O)C1 Cc1[nH]nc(-c2cn(Cc3ccnc(Br)c3)nn2)c1Cl.N12CCCC(C1)CC2=O CC1(C)CCC(C)(C(N2CC(O)(CNC(C3CC4CCCCN4C3)=O)C2)=O)CC1 N1(C(C2CCC(=O)C2)=O)CCN(CC(=O)NC2CCC3(CC3)C2)CC1 c1(C(=O)NCCC(C)NC(c2cc(CCC)n(C)n2)=O)c(N)cc(OC)cc1F Cc1sc(N)c(C(=O)NC(C)C(C)NC(c2cccc(OCCOC)c2)=O)c1C N1(C(C(C(C)C)CNC(c2cccc(=O)o2)=O)=O)CCC(F)(F)C(O)C1 c1(C(=O)NC2C(C)N(C(c3ccc(C(N)=O)[nH]3)=O)CC2)ccc(N)c(Cl)c1 C1(NC(C)=O)CCN(C(=O)NC2(C(=O)NCCC(=C)CSC)CCCCC2)CC1 c1(-c2cncc(CCC(=O)NC)c2)ccc(C(CO)NCCCn2ccnc2)cc1 C(=O)(CC1=CCN(C(=O)CC(C)n2cccn2)CC1)NCC(c1nccs1)C N1(C(c2ccc(OC)cc2)=O)CCCC(C2CCN(c3nncs3)C2)C1 c1(NCCN(C)C(c2coc(C3CCC3)n2)=O)cnc(C#N)cn1 N1(C(CC(=O)NC2CC2)=O)CCC(NC(=O)CC2CCCC2)C(F)C1 C12(C(N(C(C)C3CC3)C)=O)CCC(CN(C(c3cc[nH]c3C3CC3)=O)C1)C2 C(=O)(CCCCC(=O)OC)NC1C(CC)N(C(=O)Cc2cn3ccsc3n2)CC1 C12(CNC(C=CC(C)C)=O)CCC(NC(C34CSCC3C4)=O)(CO1)C2 c1(C(=O)NCc2ncc(C)s2)cccc(S(=O)(=O)NCCc2cnn(C(C)C)c2)c1 Cc1cc(C(=O)Nc2cc(O)nc(Cl)c2)ncc1-c1c[nH]nc1C C1(CCC)CC(C(=O)NC2(CO)CCN(C(c3ccc(CO)nc3)=O)C2)CCO1 c1(OC)cc(C(=O)NC(CO)C(C)NC(=O)C(C(C)O)NC(C)=O)ccc1OC N1(C(c2ccc(C)o2)=O)CCC(NC(=O)CN2CC3CCC2C3)C12CCCC2 N1(C(C2CCC(OC)CC2)=O)CCC(O)(CN(C(=O)CCSCC(N)=O)C)CC1 C1(CCNC(CCNC(=O)NC)=O)C(C)CCCN1C(c1ccc([N+](=O)[O-])[nH]1)=O C(C(CC)(CC)C(=O)N=c1ccn(C(F)F)[nH]1)NC(C=CCC)=O c1(C(=O)NC2CN(C(=O)CC3CC(O)C3(C)C)CC2C)c(C(C)=O)n[nH]c1C C1(C(COCCN(CCCOC)C(=O)Cc2cocn2)=O)(C(=O)N)CCC1.C=CC c1(C(=O)NC2CCC(CNC(c3cc(C)oc3)=O)C2)cc(Br)cnc1N c1(C(N2CCCC(CCNC(c3ccc(F)nc3)=O)C2)=O)cc(Br)c(O)c(Br)c1 C(CCNC(c1cnn(-c2ccccc2O)c1)=O)(C(C)C)NC(C(C)SC)=O c1(C(=O)NCC2(C)CN(C(=O)CC3CCCOC3)CCO2)ccc2c(c1)OCC2 C(=O)(CCCCC#N)NC(CC=CC)C(=O)N1CCC(=C)CC1 c1(C(=O)NCCCC(C)NC(c2cn(CC=C)nc2)=O)c(C)[nH]c2ncccc12 c1(C(N2CCC(CC=C)(C(=O)NCC3(C(C)C)CC3)C2)=O)cc(C)ncc1C C#Cc1ccc(C(=O)NC2CCC(NC(=O)CN(C)C(=O)OCC)CC2)o1 CC1(C)CN(C(c2cnoc2C2CC2)=O)CCC1NC(=O)CCc1cn[nH]c1 C1(NC(c2cccc(OC(F)F)c2F)C)CC2CCCCC12 N1(C(c2cnc(C)s2)=O)CCC2C(CCN2C(c2cc(Br)cc(C)c2O)=O)C1 c1(C(=O)OC)c(C)nn(CC2CC(OCC)C2)c1C(F)F N1(C(c2cc(Nc3c(C)c(Cl)ccc3)cn2C)=O)CCC(O)C(C)(C(=O)N(C)C)C1 C1(NC(c2cc(CS(C)(=O)=O)on2)=O)CCN(C(c2coc(O)n2)=O)C1C1CC1 c1(C(=O)NC2(CC=C)CCN(c3cc(Cl)ncn3)C2)cccc(Cl)c1F C(C)(C)(CCNC(c1ocnc1C)=O)NC(CN(NC(C)=O)CC)=O.C(C)(C)C C#CC1(NC(=O)CC(C(C)OC)NC(=O)CC2(O)CCOC2)CCCCC1 N1(CC(C)C(C)C)CC(NC(C2C(C(F)(F)F)C2[N+](=O)[O-])=O)CC2(CCOCC2)C1 Cc1ccc(CN=c2ccnc(NCCCCCCCCO)[nH]2)cc1[N+](=O)[O-] Cc1nc(C2CCCC2)sc1NCC1(CO)CC(=O)N1 c1(NC)ccc(CC(C)C(=O)NC(c2cnn(C)c2)C2CCCC2)cc1 c1(-c2cc(C(=O)NS(=O)(=O)CCC3CCCC3)on2)ccc(Cl)cc1 C12(CCOCC1)N(C(=O)COCC(=O)OCC)C2.n1(COC)ccc(C=O)n1.N C(=O)(CC1=CCCC1)NC(C(C)NC(C(C)OCC1CC1)=O)(C)C N1(C(C(C2CCCC2)OC)=O)CCCC12CCN(C(c1c[nH]c(=N)nc1O)=O)C2 CCC(C)C(C)C(=O)Nc1cnn(C2CCN(c3cc(O)nc(C)n3)CC2)c1 C(=O)(C(C1=CCCSC1)N1CCC(CC(C)C(F)(F)F)CC1)NC(CC)C Cc1cc(C(=O)NCCCC2CCCN2C(=O)C2=CCCSC2)c(C)cc1Cl Nc1cc(F)cc(C(=O)NC2CCCN(C(=O)CC=C(Cl)Cl)CC2)c1F N1(C(c2c(C)[nH]c(C(F)(F)F)c2)=O)CC(O)(C2(CNC(=O)COC3CC3)CC2)C1 N1(C(c2n3cc(C)sc3nc2)=O)CCOC2(CCN(c3nnn(C)n3)CC2)C1 c1(N(C(N2CC(c3nc(C)[nH]n3)C2)=O)C)cc([N+](=O)[O-])ccc1O C#CC1(O)CN(C(=O)CCC2CCCCN2C(=O)CN(C)CC)C1 C1(CNC(C2CC(OCC)C2)=O)CC2(CC2)CN1C(=O)Cc1cccnc1O C=CC(C)(CC)C(=O)NCC(F)CNC(=O)CCCOc1ccccc1F c1(SC(C)C)ccc(C(N2CCOC(C(=O)NCC(C)(C)C)C2)=O)cc1 C1(C(N2CC3(C2)CN(C(C24CCCC2CCC4)=O)C3)=O)CCCNS1(=O)=O C(=O)(C(C)S(N)(=O)=O)N(CCN(C(=O)C(c1ccc(C)cc1)C)CC)CC N1(C(C2C(=C)C2)=O)CCCC1CN(C)C(c1c[nH]nc1F)=O c1(SC)ccc(OC(C)C(=O)NC2CC(C)(NC(=O)CC3CCOCC3)C2)cc1 C1(SC)CN(CCNC(C2CN(C(C)=O)C2)=O)C(C)(C)CO1.CO c1(OCC)ccc(F)c(C(N2CCCC(NC(=O)CC3CC(F)(F)C3)C2)=O)c1N c1(C(N2CCN(C(c3cnn(C)c3F)=O)CC(O)C2)=O)cc2c(s1)CCCCC2 C(=O)(CCCCCNC(=O)CC1CCN(C)C1)NC(c1ccsc1)C C(=O)(CCCCCCCC1CC1)NC1CCCC(NC(C2CCN(C)CC2)=O)C1 c1(CC)ncncc1C(=O)NC(CC(=O)N1CC(C)(F)C1)C1CC1 C1(NC(C=C(CC)CC)=O)CC2(CCC(NC(=O)CN3CCCC(O)C3)CC2)C1 C(C(=O)NNC(=O)NCCC(CO)N1CCCCC1)c1cc(C)no1 c1(C(=O)NCCC(C)NC(COCCOCC)=O)ccc(C)c(S(C)(=O)=O)c1 c1(C(N(CC(C)CNC(=O)Cc2cc[nH]n2)C)=O)cn(C)c(-c2ccccn2)n1 C1(NC(c2c(CC)n(CC)nn2)=O)CCN(C(=O)CC2=CCCC2)C(C2CC2)C1 C1(C)(CC)C=C(C(=O)NCCCCCNC(=O)C(C)(C)Sc2ccccc2)C1 c1(CNC(C23CC(NC(c4cc(OC)nn4C)=O)(C2)C3)=O)ccncc1OC(C)=O Cn1cc2cc(C(=O)NC3(C)CC(NC(c4ccc5ocnc5n4)=O)C3)ccc2n1 c1(OCC)nc(Br)cnc1NC(C1CCC(CNC(c2nc(Cl)sc2Cl)=O)CC1)=O c1(C(=O)NCC2C3CN(C(C4N(C)C(=O)CC4)=O)CC32)cnn2cc[nH]c12 c1(C(N2CC(CNC(C3N(C)C(=O)NC3)=O)C2)=O)cn2ccccc2n1 C1(C(N2CCC(NC(Cn3cc(C)c(C(F)(F)F)n3)=O)C2)=O)CCCCC(=O)N1 c1(CC(=O)NCC(CNC(C2CC(CCC)C2)=O)OC)ccccc1 C#Cc1cc(F)c(C(=O)NCC(C)(C(C)C)NC(=O)CC(C)C(F)(F)F)c(F)c1 C1(C(N(CCNC(=O)CSc2nnc(S)s2)CC2CC2)=O)C2CCC(=O)C12 C(CCC(C)C(=O)NCC1CCCN(C(c2nncs2)=O)CC1)OC N1(CC)CCN(CC(=O)NC2CC(CCNC(=O)Cn3nc(C)oc3=O)C2)CC1 C(=O)(C(C)(C)CC(C)(C)C)N1CC(NC(CN(C)CCO)=O)C(O)C1 Cc1ccc(CCCN(CC(O)Cc2ccccc2)C)cc1 c1(C(N(CCC(C)NC(C2CCCC2O)=O)C)=O)cccc2nc[nH]c12 CC(C)(C)CC(O)CC(=O)NCc1ncoc1CCNC(C1(C2CC2)CC=CC1)=O CCC(CC)(CC)C(=O)N1CC(N(C)C(c2ccc3nncn3c2)=O)C(F)C1 CC1CCCCC1(C)C(=O)NCCCCC(=O)N(C)CCc1ccccc1 C12(NC(c3ccn(COC)n3)=O)CC3CC(C1)CC(NC(=O)CS(C)(=O)=O)(C3)C2 C1(O)(C(C)NC(C(COC)O)=O)CCN(C(=O)COc2ccccc2Cl)C1 c1(CC)conc1C(=O)NC(C)C(c1ccccc1)NC(=O)CC1(CC)CCC1 CC(C)C(O)CC(=O)NCC1CC(C)(C)CN1C(c1cc(Br)n(C)n1)=O C12(NC(CCCN(CCC)CCC)=O)CC(CN1C(C1CCCN1CC)=O)C2 C(CC(CC)C(=O)NC12CC(C(=O)NCC3OC(=O)CC3(C)C)(C1)C2)=CC C12CN(C1)C(=O)CN(C1CC1C)C(=O)C(=O)N2.C(C)(C)(C)OC(=O)NCC C1(CNC(c2ccc(C#C)o2)=O)CN(C(=O)CC2(OC)CCC2)CC2(CCC2)O1 S(=O)(=O)(c1cc([N+](=O)[O-])ccc1C#N)NC1CCC(c2n(C)ccn2)C1 N1(C(C2(OCC)CCC2)=O)CCCC(NC(=O)CCCN2CCCC2)C1 c1(OC)cc(N2CCC2CO)c(CNC(C(C(C)(C)C)C2CC2)=O)cc1Br Cc1nc(C(=O)N(CC(O)CN(C)C(C2CC=CCO2)=O)C)[nH]c1C CC1ON=C(C(=O)N2CCCN(C(c3nccc(Cl)c3F)=O)CC2CO)C1C C(C)(C(C)(C)C(=O)NC1CC(CCF)C1)NC(C(C)c1cccs1)=O c1(C(N2CCC(F)(CNC(CCC=CCC=C)=O)C2)=O)cc(F)cc([N+](=O)[O-])c1 c1(C(=O)NCC2C(NC(CCCCC)=O)C2)coc(S(=O)(=O)N2CCOCC2)c1 c1(OC)ncccc1NC(=O)CCC1(C)CC1.C1(=O)CC2(CC2)N1C.N(C)C.N Cc1nc(C(N2CCC(N(C(=O)CCCc3n[nH]c(=N)s3)C)C2)=O)nn1C c1(OCC)ccc(NC(=O)CSC2C(CC(=O)NC(C)CNC(C)=O)CC2)cn1 N1(Cc2cnc(OC)c(Cl)c2)CCC2(CCC(Nc3nccc(I)n3)CC2)CC1 C(=O)(CCP(C)(C)=O)N1CC(CCCCNC(C(CC)OC2CCCC2)=O)C1 c1(C(=O)NC23CC(C(=O)Nc4cncnc4)(C2)C3)cc(F)c(F)cc1I Cc1noc(C)c1C=CC(=O)NC1CC2(C1)CN(C(=O)CCc1nncs1)C2 CCCCC(CC)C(=O)N1CCCC1CNS(=O)(=O)c1ccc(C)s1 C12(CNC(=O)CCc3ccc(CO)cc3)COCCC1CN(C(=O)CC1CC1)C2 N1(C(c2c(F)ccnc2Cl)=O)CC2CC(C1)CN(C(c1ccc(O)cc1F)=O)C2 CN1CCN(C(=O)CC(=O)NC2CC2)C(CNC(=O)C=C(C2CC2)C2CC2)C1 CC(O)C(C(=O)NC(CN(C)C(C1CN(C(N)=O)C1)=O)(CO)CO)N(C(C)(C)C)C c1(OC)c(Cl)cc(C(=O)NC2CC(NC(c3nccn4ccnc34)=O)C2)cc1Cl C#Cc1cccc(CC(=O)N(CC(=O)NCCN2CCC3CC23)C(C)C)c1 n1(C(C)C)ccc(C(=O)NC2CCC(NC(=O)CC3CCSCC3)C2)n1 N1(C(Cn2ccc(C(N)=O)n2)=O)CC2CCC(NC(C3(CO)CC3)=O)CC2C1 N1(C(C(C=C)OC)=O)CCC2(CC1)CN(C(=O)C(C)CCCC(C)C)C2 c12nc(cs1)CC(=O)N1CCCC1CN2.c1(CC(=O)N(CCN(C)C)C)ccon1 c1(C(N(CC#C)CCF)=O)cc(CNC(C2OC3CCC2C3)=O)ccn1 C1(NC(C(CC)OC)=O)CCCCC1NC(C1(F)CCCCC1)=O C=Cn1nncc1C(N1CCC(C(C)C(=O)NCc2ccc(F)cc2)C1)=O C1(OC(c2cccc(C3CCCCC3)c2)=O)COC2(COC2)C1 N=c1nc(N2CCOC(c3nccs3)C2)[nH]c(NC2CSCCS2)n1 C1(NC(CC2C(OCC)COCC2)=O)CC2CC1CN2C(=O)CC(C)OC c1(C(=O)NC2CC2C(=O)Nc2ccc(F)c(Br)c2)cc(O)nc(Cl)c1 N1(CC)CCCCC1C(=O)NC(C)CCNC(=O)CSCc1cccs1 C1(C(N2CC(C(C)NC(CN(CCC)C)=O)C2)=O)CCc2c(ncn2C)C1 C1(C(N2CCCCC(N(C)C(C3CC(C#N)C3)=O)C2)=O)CCCN(S(N)(=O)=O)C1 c1(C(=O)NCCCCCCNC(C23CCCCC2C3)=O)cn2c(n1)SCC2 c1(C(=O)NC2CC3(C(NC(CC(C)C4CC4)=O)C3)C2)cc2n(n1)CCNC2=O C1(C(N(CCN(CC)CC)C)=O)CCN(C(=O)CC2CC=CCC2)CC1(C)C CN1CCOC(C(=O)N(CCC(C)(C)NC(=O)CC2(O)CCC2)C)C1 c1(C(N(CC(C)NC(C(c2cccc(Cl)c2)C)=O)C)=O)ccc2c(c1)CCOC2 N1(C(C2C(CC)CCN2C(C2CC(=O)N(C)C2)=O)=O)CCCN(C)C(=O)C1 N1(C(C(CC)n2ccnc2)=O)CCC2CC12C(N1CC(n2cnnn2)C1)=O C1(C(N(C)CC2CCN(C(c3nc(OC)oc3)=O)C2)=O)COCCC1(F)F C(=O)n1ccc2c1CCN(C(=O)CSc1cnc(O)[nH]1)C2.CCO [SH](=O)(=O)C1CCC1.C(C(F)(F)F)N(C(C1CCCC1)=O)CCO N1(C(C(C)(C)OCC)=O)CCC2(CC1)COCC(CNC(=O)C(C)(C)N(C)C)O2 N1(c2ncc(-c3ccc(SN)s3)cn2)CCc2ccccc21.Cc1cc(C2CC2)ccc1Cl C1(C(=O)NCC(CC)NC(=O)C(=O)Nc2ccccc2NC)(CC)CC=CCC1 C1(NC(CS(=O)(=O)NCC)=O)CC1C1CCN(C(c2c[nH]nc2C(C)C)=O)CC1 C(=O)(C(C)(C)CCCNC(c1coc(CO)c1)=O)NC1CCCC(C#C)C1 c1(CN(C2CCCN(C(c3nc(C(C)C)cs3)=O)C2)C(C)=O)cccc(Br)c1 CN1CCn2nc(C(=O)NCCC3CN(C(c4cnnn4C)=O)C3)cc2S1(=O)=O c1(CNC(COCCC#C)=O)cc(C(=O)OC)on1.C12(CCC1)C(=O)NC2 c1(C(N2CCC(C(=O)NCC(C)C)CC2)=O)cc(C(F)(F)F)ccc1F c1(C(N2C(CCOC)CCC2)C(=O)NC(C)(C)C)ccc2c(c1)C(C)C(C)O2 C12(CCNC(CC(C)O)=O)CCC1CN(C(=O)C(C)(C)C(C)C)C2 N(C1CCc2c(Cl)cccc21)C(=O)NNC(=O)c1c[nH]c(C(=O)O)c1 c1(C(N2CC=CC(C(N(CCCCCCC)C)=O)C2)=O)nc(C)ccc1F N1(C(CC(C)F)=O)CC2CCC(C1)C(NC(c1cc(N(C)C)ccc1N)=O)C2 c1(NCC(N2CC(CCCCNC(=O)CCc3cnoc3)C2)=O)cccnc1 C1(Cc2cn(CCN(C(C(COC)NC(C)=O)=O)C)nn2)CCCCN1C c1(OCC(=O)NCCNC(C(c2ccc(F)cc2)CC)=O)ccc(Cl)c(Cl)c1 c1(C(=O)NCC2CC(NC(=O)CCCn3cccn3)C2)cccc2cnsc12 C(CCCC(C)(C)C)NC(CCC1N(C(C(c2cncnc2)C)=O)CCC1)=O c1(C(N(CCCNC(=O)CSc2ccc(Cl)s2)C2CC2)=O)ccc2c(c1)NCC2 C(=O)(C1=C(C2CC2C)N(Cc2ccccc2)C(=O)NC1c1c[nH]c(C)cc1=O)OC C12(C(N3CCN(C(CC(=O)NCC#C)=O)C4(C3)CC4)=O)CCOC1CC(=O)NC2 C1(NC(c2cc3ccoc3cc2F)=O)COC2(CCCN(C(=O)C3CC3)C2)C1 C1(C(=O)NCC(=C)CCNC(c2nn(C)cc2C)=O)CCCC12OCCO2 N1(C(c2ccc(OCC)c(C)c2)=O)CCCC2CN(C(=O)C=C(Cl)Cl)CCC12 N1(C(c2c(CC)nco2)=O)C(CNC(=O)CC(C(F)(F)F)OC)CC2CCCCC12 c1(C(=O)NCC(CNC(c2c(C(F)(F)F)nc(C)o2)=O)O)c[nH]c2nccc(Cl)c12 CCC(C)CC(=O)C(=O)N(CCC(=O)NC1(OC)CCCCC1C)CC1CC1 N1(C(CN(C)CC)=O)CC(C(=O)Nc2cncc(C)c2)CCC1(C)C c1(C(=O)NC(CNC(C(C)SC)=O)C2CCC2)ccc(F)cc1OC(F)F c1(C(=O)NCC(CC)NC(C2(C3CC3)CCCO2)=O)cncc(Br)c1 C1(C)(C(N2CCC(OCCNC(c3c(CC)scc3)=O)C2)=O)CC(C)=NO1 N1(C(C(F)=CCOC)=O)CCC(C)(NC(c2cc(C(C)(C)C)n[nH]2)=O)CC1 Cc1cccc(CC(=O)N(CC(C)N(C(=O)C(F)CC2CC2)C)C)c1 C1(CN(C2CC2)C)CCC12CCC2.c1(CC)ccc(-n2cncn2)cc1 N1(C(C(C)(C)NC(c2ccnnc2)=O)=O)CCCC(C)(O)C1 C1(O)(CCNC(C2CCCSC2)=O)CN(C(C2CC3CC3C2)=O)C1 N1(C(CCNC(=O)NC)=O)CCC2(NC(C3OCCCO3)=O)CCCC12 c1(C(N2CCCC(C)(CNC(c3ccn(CC)n3)=O)C2)=O)sc2sccc2c1Cl C12(NC(c3nn(C)c(O)c3)=O)CCCC1N(C(C1(O)CCSC1)=O)CC2 N1(C(CC2N(C(c3ccc(CC)o3)=O)CC2)=O)CCc2ccccc2C1 C(CNC(=O)C(C)n1cncn1)(CC(=O)Nc1cnc(C(C)C)nc1)OC c1(NC(C23C(CN(C(c4c(C)noc4N)=O)C2)C3)=O)ccc(=O)n(CCO)c1 CCC(C)(C)CC(=O)N1CCC1C(=O)NC1(C)CC1(C)C C1(C(N2CCCC(C)(CNC(C3(C)CC3)=O)C2)=O)CCc2nnnn2C1 C#Cc1ccnc(C(=O)NC2(C(=O)NC3CCC3C)CCCCC2)c1 N1(CCC(=O)OCC2CCCN(C(=O)OC(C)(C)C)C2)CCc2c(O)n[nH]c2C1 CCCC(C#N)C(=O)NCC1CN(C(=O)CC(=O)Nc2nccs2)CC1O c1(C(=O)NCC2C(NC(c3cc(C)ns3)=O)CCCC2)cc(Cl)ncc1N c1(C(N2CC(O)(C(C)NC(=O)CC3CC(O)C3(C)C)C2)=O)cccc2ncnn12 C(=O)(C(C(C)(C)C)c1ccccc1)NC1CCN(C(CCc2cnc(C)s2)=O)C1 N1(C(=O)NC2CCN(C(c3ccccc3)=O)CC2)CCc2c[nH]nc2C1 C1(C(=O)NCC(C)NC(C23CCC(F)(CO2)C3)=O)CCC(=C(F)F)CC1 c1(C(=O)NCC2(CCNC(c3c(C)noc3N)=O)CC2)sc(C)c(Br)c1C c1(N(C(=O)CNCCNC(=O)Nc2cccs2)C)cccnc1 c1(N2CC3CC(NC(C(C)CO)=O)CC3C2)nc(Cl)nc2sccc12 Cc1c(F)ccc(C(=O)NC2CN(C(c3cnc(Cl)nc3)=O)CC23CC3)c1F c1(C(C(=O)NCC2CCCO2)N(C(CC)C#N)CC)cn2c(F)cccc2n1 c1(CC)c(C(=O)NC2CCC2NC(=O)Cn2cc(C(=O)NC)nn2)cccc1C N1(C(C(C2CCCC2)NC(c2cccc(O)n2)=O)=O)CCC2CCCC2C1 C1(C(=O)NCCCOCCN(C(COCCOC)=O)C)CCCCC(=O)N1 C(c1ccccc1Cl)=C(C)C(N1CCOC(CNC(=O)CN2CCC(F)C2)C1)=O C1(CNC(C(C)O)=O)CCC(C)(C)CN1C(c1ccncc1F)=O c1(OC)cccc(O)c1C(N1CC(NC(=O)C(F)=C2CCC2)C1)=O N1(C(C2COCC(C)O2)=O)CCC(C(=O)NCC(c2ccsc2)C)C(O)C1 n1(C(C)C)cccc(NC(=O)CC2CSCCN2Cc2ccc(Br)s2)c1=O c1(N2CCCC(C(=O)NC)C2)nc2c(c(=NC(C)c3cc(C)oc3C)[nH]1)COC2 C1(CCNC(C2C(C(N)=O)COC2)=O)CN(C(=O)C=Cc2ccncn2)CCO1 c1(C(=O)NC2CCCN(C(c3c(Cl)ncc(N)c3)=O)C2)cc2n(n1)CCCC2 N1(C(=O)NC(C2(O)CC2)C)CCOC(C)(C(C)(C)C)C1 c1(CC(=O)NC2CC(CNC(C(c3c(C)nn(C)c3)C)=O)C2)ccc(C#N)nc1 Cc1c(-c2ccc(CN3CCC(=O)N3C(C)C)cc2)nn(C)c1Br C(C(CC(C)C)NC(=O)CC1C=CCCC1)NC(C(Br)=C(C)C)=O C1(N(C(CC=CC=C)=O)C)CCCN(C(=O)CCNC(=O)NC)CC1 c1(C(N2C(C)C3CC2C3NC(C2CCC2)=O)=O)ccnc(P(C)(C)=O)c1 C1(CC)NC(=O)C2(CCN(C(c3cc4c(s3)CCCC4)=O)CC2)NC1=O C1(CNC(N2C(c3ccc(C)o3)CCC2)=O)CC12CCSCC2 c1(CN2C(C)CCC(NC(C3CCS(=O)(=O)C3)=O)C2)ccc(C#N)c(Cl)c1 c1(C(=O)NCC2(NC(c3ncc[nH]3)=O)C(C)CCCC2)cc(F)cc2ccoc12 C(CCC(=O)N1CCCC1CNCc1cccnc1)=C(C)C C1(C(N2CC(OC)C(NC(c3cc(CC4CC4)on3)=O)C2)=O)CCCC1C1CC1 C1(NC(CN2CCS2(=O)=O)(C)C2CC2)(CO)CCN(C)C1.C(C)(C)(C)OC(=O)OC C1(C#N)(C(=O)NCC(C)CNC(=O)Cc2c[nH]nc2O)CC(F)(F)C1 CN=c1ccc(C(N2CCC=C(CNC(=O)CNC=O)C2)=O)c[nH]1 N1(C(c2sc(C)c(O)n2)=O)CC2CCC(NC(c3ccsc3)=O)CC2C1 C(=O)(C1Cc2ccccc21)N1C(CNC(C(c2ccc(CC)s2)=O)=O)COCC1 C1(O)(CNC(c2ccc(C3CC3)s2)=O)CN(C(c2cn(-c3ncccn3)cn2)=O)C1 Cc1ccc(Cl)c(C(=O)NCCCCCNC(c2nc3sccn3c2C)=O)c1N C(=O)(CC(C(F)F)CC(=O)O)N1C(C(C)C)C(C)(C)C1.c1(C(=O)C(CCF)CC)cscc1Cl C(=O)(C1=NOC(COC(=O)C(C2CC2)OC(=O)CCc2ccc(Cl)cc2)C1)OC c1(CCn2cc(CNC(c3cccc(C)n3)COC)nn2)nc2ccccc2s1 c1(C(=O)NCC(C)(C2CC2)NC(C2CC(OC)C2)=O)c(C2CC2)nc2sccn12 CN1CCCC12CN(C(=O)COC1(C)CN(C(=O)C(F)CC3CCOC3)C1)C2 N1(C(c2cnn(C(C)C)c2)C(=O)NCCOC)CCN(C2CC2)C(=O)C1 CC(C)(CC(=O)N1CCCC1C1(C)CC1)NC(=O)Cc1cnsc1 [N-]=[N+]=NCCCC(=O)NC1CCC(NC(=O)Cn2cnc([N+](=O)[O-])n2)C1 c1(C(=O)NCCC(C)NC(c2cnc3n2CCC3)=O)cnc2n1CCCCC2 Cc1cc(C(=O)NC2CC(F)(CNC(c3csc(O)n3)=O)C2)cs1 C1(C(=O)NC(C2CN(C(=O)CCF)C2)C)Cc2c(Br)cccc2O1 C1(CNC(c2nc(C(C)OCC)sc2)=O)CC2(CC2)CN1C(=O)Cn1ncnn1 Cc1cc(Cl)c(CNC(c2ncn(C)n2)=O)c(Br)c1 c1(C(=O)NC(C)CCN(C)C(C2(CC(F)(F)F)CC2)=O)cc(F)c(F)c(F)c1 C(c1ccncc1)=CC(=O)NC(C1CC(O)CN1C(=O)C(N1CCSCC1)C)C N1(C(N2CCCN(CC(F)(F)F)CC2)=O)CCCC1C1CCCO1 Cc1nc2c(NC3CCCCN(C(C4C5COCC45)=O)C3)ncnc2[nH]1 C1(N(CC(CC=C)OC)C(c2ccsc2)=O)CCN(C(=O)C=NOC)CCC1(F)F c1(NC(c2cccc(NC(c3cc(Br)no3)=O)c2)=O)cccc(CCO)c1F Cc1cc(C(N2CC(N(C(=O)CC3CCC4CC3C4(C)C)C)C2)=O)cc(N)c1O Cc1nn(C)c(C)c1CC(C)C(=O)NCC=CCNC(C12COCC1C2)=O C1(C(=O)NC2CN(C(CCC#CC)=O)CC2CO)CCCCCCC1 C(CCN=c1[nH]c(N(C(C)CN2CCOCC2)C)nc2c1CCCCC2)OCC Cc1c(C(N2CC3CC3(NC(=O)C(F)CC3CC3)C2)=O)cnn1C(C)C(C)C C1(CCNC(C(CCC)OC)=O)CN(C(c2ncccc2N)=O)CCS1(=O)=O N1(C(CCCN(C(C(C)n2ccnn2)=O)C)=O)CCOCCC1C1CC1 N1(C(CC2CC(=C)C2)=O)CCN(C(=O)CC2OCCCC2(C)C)CCC1C N1(C(C=CCCC)=O)CC(C)(C)CC1CNC(c1ccc[nH]1)=O C1(O)(CNC(C(C)(C)c2cscc2Cl)=O)CCCN(C(c2ccc(F)cc2)=O)C1 c1(C(N2C3CN(C(=O)Cc4cccc(Cl)c4)CC32)=O)c(O)ccc(Br)c1O c1(C(=O)NC(CNC(c2cn(CC=C)nc2)=O)C(C)(C)C)ncc(F)cc1N CC1CN(C(=O)CCCc2cccs2)CC1(C)CNC(c1ncoc1C(C)C)=O c1(C(=O)NCC(C)N(C(=O)Cc2cn3ccsc3n2)C)ccn2ccccc12 C1(CC)C(NC(c2cnc(C)s2)=O)CCN1C(=O)Cc1cncn1C c1(C(N2CCC(C)(NC(c3conc3C3CC3)=O)CC2)=O)cccc2c1CCO2 C1(C(=O)OCC)(NC(COC)CCOC)CCCCC1.N12CCC(CC1)CC2=O C1(O)(CCNC(C2C(C)C2)=O)CCN(C(=O)Cc2cnccc2Cl)CC1 c1(C(=O)NCC(CCOC)NC(=O)CNC(C)=O)cccc(-c2nc(C)cs2)c1 N1(C(c2scc(C)c2)=O)CCC(N(C(=O)C(C(C)C)n2cnnn2)C)CC1 C1(C(N2CCCC(NC(c3c(C)csc3)=O)CC2)=O)CCC2(C1)CC2(F)F C1(C(=O)OC(C)(C)C)CC(C(N)=O)N(C(=O)NCC2(CN)CCOC2)C1.CO c1(N2CCC(N(C(=O)C=CC=C(Cl)Cl)C)C2)ncncc1I Cc1nc(CSCC(=O)N(CCC(C)NC(=O)Cn2ccnn2)C)cs1 C1(C(N2CCC(NC(=O)NC)C2)=O)CC2CC2N1C(c1ccc(C#N)s1)=O N1(C(CN(C)C(=O)C2CC2)=O)CCC(F)CC1C(=O)NCc1cncc(O)c1 CC1C(NC(C2CC(CNC(=O)CCNC(N)=O)CCO2)=O)CCCC1C c1(CNC(C(=O)OCC)CC2CC2)cc(C#N)ccc1Cl CCCCCCCCC(=O)NCC(CC1CC1)C(N1CC(C)=CC(C)C1)=O C(C)(C)(CCCO)NC(c1cc(CNC(C(C)=CC(C)(C)C)=O)[nH]n1)=O CS(=O)c1ccc(CC(=O)NC2CC2CNC(c2cccc3nc[nH]c23)=O)cc1 C1(C)(C(=O)NC(C(C)C)CNC(C2(Cl)CC23CCC3)=O)CCC(C)(C)CC1 c1(C(N(C2CCN(C(=O)CC3(CO)CC3)C2)CC)=O)cn(CCC(C)C)nn1 N(C1CCCc2c1cnn2CCO)C(c1n(C(CC)(C)C)nnn1)C1CC1 c1(CNC(=O)NC2CCC(OC3(C)CCOCC3)C2)c(N)cccc1F C1(NC(C2C3CC2N(C(c2cc(O)cs2)=O)C3)=O)CCOCC1CO C1(C(=O)NCC23CCC(C2)NC3)C2Cc3cc(Br)ccc3C12 c1(C(N2CC(CC)C(NC(c3cn[nH]c3)=O)C2)=O)cc(Br)cn(CC)c1=O c1(C(=O)NCC2C3CN(C(CC(C)(C)OC)=O)CC32)ccc(F)c(F)c1C CC1CC(C(=O)NCC(C)(C)OCCNC(C2CC2(Cl)Cl)=O)C1 N1(C(C(C)C2CC2)=O)CCCCC(N(C)C(c2cc(-c3ccccn3)ns2)=O)C1 CCC(F)(F)CC(=O)N1CCC(N(C)C(c2cnn(CC(C)C)c2)=O)CC1 c1(CNC(C(C)OC(C(c2cnn(C)c2)C)=O)=O)cc2c(s1)CCC2 C12(C(N3CC(NC(c4cn(C)c(=O)cn4)=O)C3)=O)OCCCC1C2(F)F C1(O)(C(=O)NCC(C)C)CCN(C(=O)C(C)(C)CCl)CC1 N1(C(CC(=O)NCC)=O)CCC2(CC1)CC2CNC(C1CCOC1)=O c1(OC)cccc(F)c1C(=O)NCCNC(=O)C(O)C(C)c1ccccc1F Cc1cc(C(=O)NCC2CN(C(=O)CC3CN(C)C3)CC2O)oc1C c1(C(=O)NC(C)CCCNC(C2CC(=C3CC3)C2)=O)cccc(CC2CCC2)c1 Cn1nc(CNC(=O)Cc2ccco2)cc1C(=O)NCC(C)(O)CCO C(CN=c1c(C#N)c[nH]c2c(F)c(F)c(F)cc12)C1(NC(C(COC)C)=O)CC1 c1(C(=O)NC(c2ccnn2C)CNC(CCC2N(C)CCC2)=O)ccc(Br)c(F)c1 c1(CC(N2CC3C(NC(C(C(C)C)O)=O)(CC3)C2)=O)cc(Cl)cc2c1OCC2 c1(CCNC(CN(C(C2CC(n3ccnc3)C2)=O)CC)=O)ccnn1C c1(C(N(CCCCNC(CCN(C)CCO)=O)C2CC2)=O)nsc2ccccc12 c1(CNCC(C)(C)C)nnnn1CC1(c2ccccc2)CC1.c1(-c2ncco2)ccc(Cl)s1 c1(OC)ccc(CC(O)C(=O)Nc2ncoc2-c2cc(C)no2)cc1 c1(CC(=O)N(C2CCN(C(C(c3cc(C)sc3)(C)C)=O)C2)C)nc(C)c(C)s1 N(C1CCN(Cc2ccccc2)c2ccccc21)C(C(CCC)C)=O C1(C(=O)N(C)N(C)C(c2ccon2)=O)(CC)CN(C(=O)OC(C)(C)C)C1 CC1CN(C(C2CCCC(=O)O2)=O)CCN1C(=O)CC1NC(=O)NC1=O N1(C(CC2(OC)CC2)=O)CCC2C(NC(=O)CNC(C3CCC3)=O)CC12 CC1CCCC(CNC(C2CC(N(C(=O)Cc3ccoc3)C)C2)=O)CC1 c1(CC(C)(C)C)ccccc1C(=O)NC(CNC(C1CC1C(C)(C)C)=O)CO N1(C(c2nn(C)c(Br)c2)=O)CCC2CN(C(=O)Cc3cccc(F)c3)CC12 c1(C(N2CC(CCSC)(NC(COC(CC)C)=O)C2)=O)ccc2c(n1)CCCN2 N1(C(=O)Cc2csc(S)n2)CCCC(NC(C2(F)CCCC2)=O)CCC1 C1(CC)(NC(=O)NC2CN(C(=O)CC3CCCCC3)CC2O)CCOCC1 N1(C(C2CCN(C(C)=O)C2)=O)CCC2(NC(=O)C3=COCCC3)CCCCCC12 Cc1c(C2CCCC2NCc2cc(C3CC3)on2)cnn1C c1(C(=O)NC2(C)CC(NC(c3ccsc3C(F)F)=O)C2)ccc(O)nn1 c1(C(=O)NCCCC2(NC(=O)CC3CC3)CC2)cccc(F)c1 c1(C(=O)NC2(CC=C)CN(C(c3cn(CCOC)nc3C)=O)C2)nccnc1C Cc1nc(-c2ccsc2)n[nH]1.C1(=O)C(C2CCCO2)NC(=O)COCCCN1 C1(C)(C(=O)NC2(C)CN(C(C3CC(C)(C(=O)OC)C3)=O)C2)CCCC1(F)F C1(CC(=O)N(CC(C)N(C)C(C23CC(C2)C3)=O)C)(N(C)C)CCC1 C1(C2CCN(C(c3cnn4cc[nH]c34)=O)CC2)(NC(c2ccc(C)nn2)=O)CC1 c1(CC)cccc(CC(N2CC(c3cn(C(C4CCC4)=O)nn3)(C(N)=O)C2)=O)c1 Cc1ccc(CCC(=O)NC2CC(F)(CNC(C3CCCC(C)C3)=O)C2)cc1C c1(C(N2CCC(CNC(C3(O)CCC(C)CC3)=O)CC2)=O)n[nH]c2ccccc12 CC(C)C(O)C(F)(F)C(=O)N1CC(C(=O)N(C)Cc2ccon2)C(C)C1 C1(CC)CN(C(C2(CF)CC2)=O)CCC1CNC(=O)C(C)OCC(C)C C(=O)(CN=c1[nH]c(C)cs1)NC(CN(C(c1cc(CSCC)on1)=O)C)(C)C c1(C(N2CC(N(C)C(c3coc(Br)n3)=O)C(O)C2)=O)cccc2nn[nH]c12 c1(C(=O)NCC(CNC(c2cc(Cl)c[nH]2)=O)F)c(F)ccc2ccncc12 c1(C(=O)NC2CCN(C(c3ccc(COC)s3)=O)CC2)c(O)cc(O)cc1O n1(CCCF)c(N(CCF)C2CC2)nnc1-c1ccc(CN2CCCC2)o1 CP(C)(=O)c1ccc(C(=O)NC2COCCN(C(=O)COc3cn[nH]c3)C2)o1 c1(C(c2nnnn2CCSC)NCC(=O)OCC)ccc(F)c(OC)c1 c1(C(c2n(CCC)nnn2)NCC(CSC)OC)nc2cc(Br)ccc2n1C c1(CCSC)cn(C)nc1C(C)C.N12CC(C1)NC(=O)C2=O N1(C(c2cnc(OC)c(C)n2)=O)CCCC12CCCN(C(c1cc(C)ns1)=O)C2 CCC(C)C(O)CNC(C1(CNC(c2cc(COC)ccn2)=O)CC1)=O c1(C(N(CCN(C)Cc2c(C)ccnc2Cl)C)=O)cc2ccccc2o1 c1(C(N(CCNC(c2n(C=C)nnc2)=O)CC)=O)cc(N)c(Cl)cn1 CC1CC(C(N2CCCC2CN(C(=O)CCCCc2ccccc2)C)=O)C1(C)C C(=O)(CCCCN(C)C)NCc1scc(C(N(CC(CC)C)C)=O)c1 CCCC(C(=O)N1CCC(OCC(N2CCC(O)C2)=O)CC1)NC(C)=O c1(NC(c2c(OCC)cccn2)=O)c(-c2ccc(O)nc2)ccc2c1OCO2 Cn1cc(Cl)c(C(=O)Nc2nc(CCOCN)cs2)n1 c1(C(=O)NC2CCC(NC(c3c(C(C)C)csc3)=O)C2)cc2ccsc2s1 C1(F)(C(=O)NCCCC)CCN(C(c2cc(C)nn2CCC)=O)C1.OC c1(CC(N2C(CNC(CCC#C)=O)C(C)CC2)=O)ccc([N+](=O)[O-])cc1OC C(=O)(C(C)(CO)NC(=O)Cc1csnn1)N(CCC)CCN(C)C CC(C)(CNC(C1(C)CCC(=O)N1)=O)CCNC(=O)COCC1CCCO1 C(=O)(CCC(C)(C)C#N)N1CCC(C)C(NC(=O)CCc2nnc(C3CC3)o2)C1 C1(C(C)C)N(C(c2cc[nH]c(=N)c2)=O)CC12CCN(C(=O)C=CCF)CC2 c1(CC)cc(C(=O)NC(c2ccc(OC(F)F)cc2C)C)ccc1Br N1(C(CCC(=O)NC)=O)CC(C2CN(C(c3sc(=N)[nH]c3C)=O)C2)C1 C(=O)(C(F)C(C)CNC(c1cnn(C)c1C#N)=O)N(CC)CC1CCCC1 N1(C(N(CCOCC)Cc2cc(F)ccc2F)=O)CCN(C2CC2)CC1C N1(C(C(CC)C#N)=O)CC(=O)NC2CN(C(c3cccc4c[nH]nc34)=O)CCC12 c1(C(=O)NC(C2CCCN(C(C(C=C)(C)C)=O)C2)C)ccc(OC)c(Cl)n1 c1(C(N(C2CCN(C(c3cc(F)n(C)n3)=O)C2)CC)=O)ccc2c(c1)nnn2C C(CC(=O)N(CC(O)C(F)(F)F)C)(C(C)OC)NC(C1(CC=C)CCCC1)=O C1(NC(C(C)OCC=C)=O)C2CN(C(=O)C(N3CCC(O)CC3)C)CC12 N1(C(Cc2cccc(C(=O)OC)c2)=O)CC2CCCC(N=c3nc[nH]s3)C2C1 c1(C(N(C2CN(C(c3cnc([N+](=O)[O-])n3C)=O)C2)C)=O)nccc2ncccc12 c1(CN(CC(N2CCCCCC2)C)C(=O)NO)nnc2n1CCCC2 c1(OC)ncnc(C(N2CCN(C(=O)Cc3ccc(F)cc3)CC2CF)=O)c1F C(CC(C(=O)N1CC(=CC)C1)NC(C1CC(CF)C1)=O)OC C(=O)(C(CCS(C)=O)N(C)C)N(C(C)C)CCNC(=O)CC1C(C)(C)C1(C)C C(CCC(C)(C)NC(C1CN(C)C(=O)N1)=O)NC(C(C)Cc1ccncc1)=O N1(Cc2nc(C)c(C)o2)CC(=O)N(Cc2ccccc2OC(F)(F)F)C1=O N1(C(C(c2ccccc2)C)=O)CCC(F)(F)C(CNC(=O)C2=COCCO2)C1 c1(C2CCN(C(c3cccc(N(C)C)c3)C(=O)NC3CC3)C2)ccc(Cl)cc1F c1(CC(C)C)ccccc1C(=O)NC(CNC(=O)C(C)(C)c1cc[nH]n1)C1CC1 N1(C(CNC(c2ncn(CC)c2)=O)=O)CC(F)(F)CC1CO CC1(C)COc2cc(CNC(=O)CCCc3ccc(N)cc3)ccc21 CC(C)CC(CNC(=O)C(C)C1CCCC1)C(=O)NCCC(O)C1CCCC1 Cc1cnn(CCC(=O)NC(CN2CC(C(C)Nc3csc(C4CC4)n3)C2)=O)c1 N1(C(CSCCC)=O)CCCOC(CNC(=O)CN2C(=O)CCC2=O)C1 c1(CC(C(=O)N(C2CCCN(C(=O)CCCC3CC3)C2)CC)C)c(C)noc1C Cc1ccc(-n2nnc(C(=O)NC3CC3CNC(C3(OC)CC3)=O)c2C)c(C)c1 C1(CNC(C2(SC)CCC2)=O)CC2COCC2N1C(c1nn(C)c(=O)cc1C)=O CC1CCC(CC(=O)NCC(N2CCN(C(c3ncccc3F)=O)CC2)C)CC1 C1(C(=O)NC(c2cccc(C)n2)C)(CNC(Cc2cnc(C)s2)=O)CC(C)(C)C1 c1(OC)cccc2[nH]c(C(=O)NC(CNC(C3COC(=O)N3)=O)C(C)(C)C)cc12 Cc1ccc(C)c(C(=O)NCC(C)(CO)NC(c2c[nH]nc2OCC(F)F)=O)n1 N1(C(c2c(CC)n(C)nc2)=O)CCC2(CC2)CC1C(=O)NC(C)CC C1(NC)CN(C(=O)C(C)(C)O)CCC12CCC2.c1(Nc2cccc(C=O)n2)nn(C)c2c1CCC2 C=CCC(CC=C)C(=O)N1CC(C(N2CC=C(C)CC2)=O)CCC1(C)C N1(CCCCC=C)CCc2ccccc2C1CNC(C1CC(C)(C)C1)=O c1(C(c2ccccc2OCCc2ncccc2F)=O)cc2c(s1)C1CCC2C1 C1(C)CC(O)CN1C.C(=O)(CCC(C)=O)N(CC(=O)NCCOC)C(C)C CC1=C(C(=O)NC2CC2NC(=O)C(O)Cc2cccc(C)c2)CCCC1 c1(C(C)NCCCC2(O)CCNCC2)cncc(N2CCCC2)n1 C1(NC(c2cnc3ccsc3c2)=O)COC2(C1)CN(C(c1cnco1)=O)C2 c1(CC(=O)NC(C)CN2CCCCC2)c(O)cccc1F C1(CNC(CSCC#C)=O)CN(C(c2ccn(CCC)n2)=O)CC12CC2 c1(C(N(CCOCCN(C(C(F)OC)=O)C)C)=O)cnn2c1OCC(F)C2 c1(C(=O)NCC(CNC(c2[nH]c(CC)c(Cl)n2)=O)O)c(O)ccc(Cl)c1F c1(C(N(C2CCN(C(=O)CCC(C)OC)C2)CC)=O)cnn(C)c1C#N C12(CNC(c3ccnn3C(F)(F)F)=O)CC(NC(=O)C(C3CCCCC3)O)(C1)C2 c1(C(N2CC(C(C)(C)O)(CNC(c3c(C)ncs3)=O)C2)=O)scc2c1CCCC2 CC1(C)CC(C(=O)NCCCC2CN(C(C3CCC(=O)O3)=O)CCO2)CCO1 N1(C(c2c(C)cccc2C)=O)CCC2(CNC(C3(O)CCC3)=O)CCCCC12 N1(C(c2ncn(C)n2)C(=O)NCC)C2CCCC1COC2 N1(C(c2c(CNC(C3CC=CCC3)=O)cco2)=O)CC2COC(=O)C2C1 C1(c2nnc(CNC(c3cn(C(C)C)nc3Br)=O)s2)CCCCN1CC C(C(=O)NNC(=O)NCC1C=CCCC1)Sc1cccc(C)c1 CC1CCC(=O)N(CC(=O)NCC2CN(C)CCN2C(C2(O)CCC2)=O)C1 CCC(C)(C(=O)NC(C)CCCNC(C1(n2cnnn2)CCCCC1)=O)OC C12(CNC(C(C)(C)N(C)C)=O)CCCCC1CN(C(c1cc(CO)n(C)n1)=O)C2 c1(C(=O)NC(CN(C(=O)C(F)=C(C)C)CC)C)csc2ccc(F)cc12 N1(c2nccc(C(=O)OC)n2)CCC(NC(C2C3C=CSC23)=O)C1(C)C c1(N(CC(CC)OC(F)(F)F)C)ccc(OC(C2CC3CCC2O3)=O)c(Cl)c1 C(C)(C)(CCCN=[N+]=[N-])NC(C1OCCN(C(C(C)SC(C)C)=O)C1)=O Cc1cccc(C(C(=O)Nc2ccccc2C)N(C)CCC2CC2)n1 N1(C(C(=O)OCC)CC2(OC)CC2)C(C(=O)Oc2ccc(F)cc2)CCCC1C N1(C(C(C2(O)CCCCC2)CC)=O)CC2=C(C1)CN(C(=O)C=CC1CCCO1)C2 Cc1cccc([N+](=O)[O-])c1C(=O)NC1CCCCN(C(C2CCC2C(N)=O)=O)C1 C1(CNC(COC)=O)C(CNC(c2cnn(CC(C)C)c2)=O)C1(F)F C(=O)(CCCCC(C)(C)C)NC(C)C(CO)NC(C1CC12CCOCC2)=O C1(CNC(c2c(C)ccc(N)c2)=O)CN(C(=O)CN(C)C2CC2)C2(CCC2)C1 c1(C(=O)NC(C)CNC(=O)CC2CCCCC(=O)N2)ccc2c(c1)C(=O)CCC2 c1(C(=O)NC(CC2CN(C(c3n(CCC)ncc3)=O)C2)C)nc[nH]c2nccc1-2 C1(C(=O)NCc2c(N(C)C)nccc2)CCC(C)(F)CC1 CCCC(CCC)CC(=O)NCC(C)(C)CNC(c1cc(F)ccc1F)=O C12C3CN(CC13)C(=O)C1(CCC1)CNC2=O.c1(CCOCC)cnccc1Cl CC1CCc2onc(C(=O)NC3CCN(C(=O)C#CC4CCCOC4)C3)c2C1 CCC1C(=O)NC1=O.c1(C(=O)OC)ccccc1N1CC2CCC1C2 C1(C(=O)NC(C)C)(OC(C)(C)C)CCOCC1.CC1C(C)N(C)C(=O)N1.C1(=O)CN1 CC(C)C(C(=O)NCc1ncccc1C(=O)NCC1(C)CC1(F)F)N(C)C N1(C(C(C)(C)c2sccc2Cl)=O)CCCN(C(C2(CO)CC2)=O)CC1 c1(N2CCC(C(C)(C)C)(CNC(C=C(C)Cl)=O)C2)nc(Cl)nc2sccc12 N1(CCC(N2CC(NC(c3n(C)cnc3)=O)C3C(C2)C3)=O)Cc2ccccc2C1 C1(NC(c2cnn(CC)n2)=O)CC(NC(=O)Cc2cc(F)cc(F)c2)C12CCC2 C1(CNC(CCCc2c(C)ccs2)=O)CCN(C(c2cnsn2)=O)CC1C N1(C(c2cnc(C(C)C)s2)=O)CC2CC3CC2C1C3NC(=O)CN1CCCC1C N1(C(C(C)NC(COC)=O)=O)CC(C2CN(C(C3(C)CCC(F)(F)C3)=O)C2)C1 Nc1cc2[nH]c(O)nc2cc1C(=O)NCCNC(c1ccsc1C(F)(F)F)=O c1(C(=O)NC2CN(C(C=COCC)=O)CC2C#N)c(OC)ccc(Br)c1C c1(OC)ccc(CC(N2CC(NC(C3CC(C)(F)C3)=O)C3(CC3)C2)=O)c(C)c1 NS(=O)(=O)C1(C(=O)NCC2(CNC(=O)CC(F)(F)Cl)CC2)CCCC1 C1(C(N(C2CCN(C(=O)CC3COC(=O)C3)CC2)CCOC)=O)CCCCN1C CC1CC(C(N2CCC(O)(CN=c3[nH]nc(C(N)=O)s3)CC2)=O)CCS1(=O)=O C(=O)(C(F)(F)C(C)O)NCC(CNC(C1(C(C)(F)F)CCOCC1)=O)OC C(CCC(C(=O)Nc1ccc(Cl)cn1)NC(C1CCN(C(=O)OC)C1)=O)OC c1(-c2cnc(NC(c3nc(Cl)ccc3F)=O)s2)c(F)cc(C(O)C2CC2)cc1F C1(NC(C2CC(=O)NCC2)=O)COCCN(C(=O)Cc2nc([N+](=O)[O-])n[nH]2)C1 Cn1cncc1CC(=O)NCC1OCCC1C(N1CC(O)(c2cnn[nH]2)C1)=O Cc1nc(CO)oc1C(N1CC(NC(=O)C(O)C2CCC2)C(n2cccn2)C1)=O c1(C(=O)NCCCN2CCN(C(c3n(C)cc(Br)n3)=O)CC2)cc(F)cnc1O CC1CN(C(c2cccc(C3(C)CC3)c2)=O)CCN1C(C1CCOC(=O)N1)=O c1(C(N2CCC(NC(C(n3ncc(C)c3)C)=O)(CO)C2)=O)cccc2cnsc12 c1(CNC(CCCN(C(C2(SC)CC2)=O)C)=O)ccc(O)c(F)c1 C1(CC)(CC)CC(NC(=O)C(C)O)CN1C(=O)C=C(C)C c1(C(=O)NC2(CC=C)CN(C(=O)CCOCC3CC3)C2)cc(SC)cc(Cl)c1 n1(CC)nc(C)cc1C(=O)NC(CCOC)C(=O)Nc1cnn(C)c1C(N)=O C1(C)(CC(N2CCN(CC(C)NC(COC(C)C)=O)CC2)=O)CCS(=O)(=O)N1 N1(C(c2n(CC)ccc2)=O)CC(F)(F)CC1CCNC(C1CC1(F)F)=O C1(NC(=O)C=C(C2CC2)C2CC2)CN(C(=O)CC23CCCC2C3)CC2(CCC2)C1 c1(C(=O)NC(CC)CN(C(=O)CC2COCCO2)C)[nH]c2cc(Cl)ccc2c1C O(N(CC)C(=O)C1(NC(=O)CC2CCCC2O)CCN(C)C1)CC C1(N2C(=O)OCC2)CCCN(C(C2(n3cc(-c4ccc(O)nn4)nn3)CC2)=O)C1 CC(C(=O)N1CCCC(NC(=O)Cc2c(F)cccc2Cl)C1)C(C)(F)F C=CCC(CC)C(=O)N1CC2(CO)CC1(C(=O)NC1CCCC3CC13)C2 c1(C(C)NCC(CO)N(C)C)cccc2ccccc12 C1(OC(c2cn(CCOC(=N)O)nn2)C)CCC2(CCCCCC2)O1 N(C)(C1CCc2cc(Cl)ccc21)C(CCCCCC)C(=O)NCC N1(C(C23C(NC(C4C(C)(C)COCC4)=O)CC(CC2)C3)=O)CC(C)(C2CCC2)C1 C1(CN(C)C)COCC1NC(C1COCC1NC(=O)CN1CCOC1=O)=O C1(CC(=O)NCC2CCC(C)CC2)CCN(C(c2cccc(O)c2F)=O)C1(C)C C1(NC(c2cn(CC)nc2)=O)CC(F)CN(C(=O)CCCCc2cnn[nH]2)C1 N1(Cc2ncc(-c3cn(CC)nc3)cn2)CCc2ccc(Cl)c(Cl)c2C1 C1(NC(Cc2cn(CC)nc2)=O)CCN(C(c2cc(OC)cnc2F)=O)CC1O N1(C(C(CSC)O)=O)CC(CNC(c2cc(Br)n(C)c2)=O)CC(C)(C)C1 O=C(C(O)C(F)(F)F)NC12CC(C(=O)NCc3cnns3)(C1)C2 c1(C(=O)NCCOC2CCN(C(C(C)CC3CCC3)=O)C2)ccnc(Cl)c1O c1(-c2ccc(-c3c(C)onc3)cc2)ccc([N+](=O)[O-])o1.C12CN(CC1O)C2 C=C1c2ccccc2C(=O)N1CCC(=O)NC1CCCN(C(=O)CC(C)CF)C1 N1(C(Cc2c(Cl)cn(C)n2)=O)CC2CC(C1)CN(C(=O)C#CC1(C)CCCO1)C2 CCC(C)C(C(=O)NCC1CCN1C(=O)Cc1cccc(Cl)c1F)N(C)C C1(C(=O)NCc2c(C)csc2)CN(C(=O)CC2CCCSC2)CCO1 C1(N(C)C2CC2)CN(C(=O)CCN(C(=O)CCc2ccc[nH]2)CCCO)C1 C#CC1CCN(C(=O)C(=O)NC2CCN(CCC(F)(F)F)C2)CC1 C(CC(C)C(=O)N1CCCC(N2CCN(C(C3CCC(C)(C)C3)=O)CC2)C1)=CC C1(C(N2CCC(C)C(CNC(=O)Cn3cc(N)cn3)C2)=O)C2CCCCCCC12 C1(C)(CNC(C2(CNC(CCOCCC)=O)CCCO2)=O)NC(=O)NC1=O C1(CNC(C2CCC(CO)CC2)=O)CCN(C(C2(CF)COC2)=O)CC1 Cc1ccc2c(c1C)OCCC2NS(=O)(=O)c1cccnc1N(CCCF)C c1(C(=O)OC)coc2ccc(OC)cc12.c12ccc(F)cc1C1CCCN1C2=O c1(SCC(=O)N(C(C)CN2CCCCC2)CCC)cc(OC)nc(F)c1 c1(CNC(c2cccc(C)c2CN(C)C)=O)nc2c([nH]1)CNCC2 C#CCCCC(N)C(=O)Nc1ccccc1CN C(=O)(C(C)S(=O)(=O)Cc1noc(-c2cccc(C(CC)OC)c2)n1)OC N1(C(CC(=O)C(C)(C)O)=O)CC2CCCCC2(Oc2ccc(C)cc2C)C1 c1(-n2c(C3(C4CCCC4)CCN3)nnn2)c(C)cccc1C.CCCC C1(CC=C)(C(=O)NCC2(CO)CCOCC2)CCCN1C(c1cocn1)=O N1(C(C2N(C(CN(CCC#C)C)=O)CC2C)=O)CCCC(C2CC2)CC1 N1(C(c2ncc(C)c(Cl)c2)=O)CCN(C(c2cnccc2Cl)=O)CC(C)(F)C1 C(=O)(C(C(C)C1CCOC1)N(C1(C)CCCO1)C)NCC(C)C C1(C(=O)NCC2(C)CN(CCc3ccno3)CCO2)CCc2c[nH]nc2C1 CC(=NOCC#N)C(=O)N1CCC(C(C)(C)C(=O)NCC2=NOCC2)C1 N1(C(CC(C2CC2)NC(c2ccc(CC)s2)=O)=O)CCC2CCC12 S(=O)(=O)(c1ccc2nc(O)oc2c1)N1CC(NC(c2ccno2)=O)C(F)(F)CC1 CCS(=O)CC(=O)NCC1CCN1C(=O)C(F)(F)C1(Oc2ccccc2)CCC1 c1(CC)nc[nH]c1C(=O)NC1CCCC1NC(C1CCCN1C)=O N1(C(c2cnc(CC3CCOCC3)o2)=O)CCCCC2CCCC12 CC1(C#CC(=O)N2CCN(C(=O)C=Cc3cnc[nH]3)CC2CO)CCCO1 C1(C(N(CCCN(C)C)CC)=O)CC(=O)CN1C(=O)Cc1cnnn1C C1(CNC(C2C3(CC(OCC)C3)C2)=O)CCC2(CCC2)CN1C(=O)C=CC1CC1 C1(C)(C(N2CC(CNC(C3C(C)(C(F)F)C3)=O)C2)=O)C2CC3CC(C2)CC1C3 C(=O)(CCC(=O)NCCCNC(=O)Oc1ccccc1)OCC c1(COC)cc[nH]c1C(=O)NCCN(C(=O)CCc1nc(C)cs1)CC(C)O c1cc2nc(N3CCN(CC4CCC4)CC3)[nH]c2cn1 C12(C(N3CC(C#C)(N(C)C)C3)=O)CCC(C1)C2(C)C.c12cc(nn1C)CNC2=O N1(C(C(CC)(F)F)=O)CCN(C)C(C(=O)NCC2CCS(=O)(=O)C2)C1 c1(OC)cc(C)c(Br)cc1C(N1CCOCC(NC(=O)C(O)C2CC2)C1)=O N1(C(C2OCCN(C)C2)=O)CCOCC(F)(CNC(c2cc(CCO)on2)=O)C1 C1(CC)CN(C(C2CCCCCC2)=O)CCC1NC(c1c(SC)cccc1F)=O Cc1c(C(=O)N(CC(C)NC(c2cnc(O)c(F)c2)=O)C)nn(C)c1Br N1(C(CCC=C)=O)CCOC2(C1)CN(C(c1ccoc1CC(N)=O)=O)C2 c1(C(=O)NCC2OCCCN(C(CC(C)C(F)F)=O)C2)n[nH]c2c1CCOC2 CC1N(C(=O)NC2CCC3(CC2)CC3CO)CCCC1(C)C C1(CNC(CCCN(C)C(C2CC(F)(CF)C2)=O)=O)CC2(CCC2)CO1 CC1COC2(C1)CN(C(=O)CC1CCCCC1NC(C1CCNC(=O)C1)=O)C2 C1(CC(N2CCC(CCNC(c3n(C=C)ncc3)=O)C2)=O)CCCS(=O)(=O)C1 N1(C(c2csnn2)=O)CCC(C2CCCN(C(C3CCCC34CCC4)=O)C2)CC1 N(C1c2ccccc2CC1O)C(C1CC12CCN(Cc1ccccc1I)CC2)=O S(=O)(=O)(c1cccc(=NCc2nccn2C)[nH]1)NC(C)CS(C)=O CN(CC(=NCCCN1CCCC1)NC1CCCC1)CCN1CCCC1=O C1(CC(=O)N(CC(CC)NC(=O)COc2ccc(Cl)nc2)CC)COC2CC1C2 C(=O)(C(O)C(C)CC)N(CCCNC(c1cc(CC(C)C)on1)=O)CCC c1(N(CCC)CC)ccc(C(N2CC3CC3(CNC(=O)C(C)(Cl)Cl)C2)=O)cn1 C(N=c1[nH]c(=NCC2CC2C2CC2)[nH]c2c1COCC2)c1nnn(C)n1 CCC(C(C)C)C(C(=O)NC1CCCC1)N1CCOC(CC2CC2)C1 c1(N2CC(CC)(CC)S(=O)CC2)nc(=N)[nH]c(=NC2CCCc3ccccc32)[nH]1 C1(OC)C(NC(C2(C)CN(C(C3CC=CCC3C)=O)C2)=O)CC12CCC2 c1(NC=O)ccc(C(C)C)nc1.C(C(=O)NCC1(CC)CCC1)(C1CCOC1)OCC c1(C(N2CCCN(C(C3C(C)CC3C)=O)CC2)=O)csc(S(N)(=O)=O)c1 C1(NC(CC(C)(C)C#N)=O)CCC2CCN(C(c3c(O)cc(F)cc3F)=O)C1C2 c1(N(C2CCN(C(c3onc(C(=O)NC)n3)C)C2)CC)cccc(F)c1[N+](=O)[O-] C(=O)(CCC(C)(C)[N+](=O)[O-])N(CCC(=O)OC)CC#C.C1CNC(=O)N1 c1(C(N2C(C3(O)CN(C(c4c(Cl)cn(C)n4)=O)C3)CCC2)=O)nnc(Cl)cc1N c1(SCC)cccc(C(N2CCC(O)(C(C)NC(=O)Cc3nccn3C)C2)=O)c1 C1(C)(C(N(CCN(C(c2ccnc(NC)c2)=O)CC)CC)=O)CCC(C)=C(C)C1 N1(C(C2(COC(C)(C)C)CCCO2)=O)Cc2ccccc2CC1C(F)(F)F C12(NC(C34CC(C(C)NC3)C4)=O)CC3(C)CC(C)(C1)CC(F)(C2)C3 C1(C(=O)NCCCCCNC(c2cc(C)c(C)nc2)=O)CCCC1S(C)(=O)=O Cc1c(NC(C2CCCC(C)(C)C2)c2nnnn2C2CC2)cccc1C#N Cn1nc([N+](=O)[O-])c(Cl)c1C(=O)NCC(C1CC1)NC(c1ccc2ocnc2n1)=O CON(CCC(=O)NCC1(C)CCN(C)C1)C(=O)CC(C)(C)C(C)=O c1(N(c2nc(C)sc2)C)ccccc1CC(=O)C1(C(=O)N(C)C)CC1 O=C(CC(C(F)(F)F)c1ccccc1)NC(c1nc[nH]n1)C1CC1c1ccccc1 c1(C(=O)NCC2CCCN(C(=O)CN3CCOC3=O)CC2)[nH]nc2ncccc12 Cc1c(C(=O)Nc2cccc(NC(=O)C(O)CC(N)=O)c2)oc2ccc(F)cc12 C1(C(=O)NC2C(O)CCN(C(CN(C(C)=O)C)=O)C2)CCc2ccccc2C1 C1(NC(C2(OC)CCOCC2)=O)CC2CC1CC2C(N1CC(c2ncc[nH]2)C1)=O c1(OC)ccnc(Cl)c1CN1CC(C(=O)NCC2(O)CCOCC2)CC(F)C1 CCCC(C)C(=O)NC(Cc1ccccc1Br)C(=O)NCCC12CCCC1C2 CC(C(=O)N1CCC(N(CCO)C(C2CCC2(C)C)=O)CC1)C(F)F N1(C(C2(Cl)C(C)(C)C2)=O)CC(CO)C2(CCN(C(=O)C=C3CCCC3)CC2)C1 N1(C(c2cc(SC)n(C)n2)=O)CCC(NC(C2C=CCCC2)=O)C(O)C1 N1(C(C2CC(CC)C2)=O)CCCC1CCCNC(=O)CC1(N(C)C)CCC1 C(C)(C(C)(C)CN(C)C)NC(=O)NC1C(CC(=O)OCC)CCC1 c1(C(N2CCC(NC(c3ncon3)=O)C2)=O)cc2n[nH]cc2cc1Cl c1(NC(CN(CCOC)C)=O)ccc(Cn2cc(-c3ccccn3)nn2)o1 C1(NC(=O)CCc2cncc(F)c2)CCN(C(C2C=CCC2)=O)C12CCC2 c1(C(N2CCOCC(NC(C=CC(C)(C)C)=O)C2)=O)cccc2nsnc12 c1(C(=O)NCC2C(NC(C(C)(C)OCCC)=O)C2)cnn2c1CCC2 c1(SC)cccc(C(=O)NCC(CO)NC(c2ccc(C)n2C)=O)c1 C(=O)(C1CCc2ccc(C)cc21)NCC(CCOC)NC(=O)C(C)CC(F)F N1(C(c2c(C)n(C3CCC3)nc2)=O)CC(C)C(C)(CNC(c2cc(F)cs2)=O)C1 O=C(CC1=NNC(=O)C1)NC1CCCC(CNC(=O)Cc2csc(NC=O)n2)C1 c1(C(N2C(CNC(C(CC)C(=O)OC)=O)C=CC2)=O)[nH]c2ccccc2c1C C1(C(=O)NCC2C3N(C(COCC#C)=O)C(CC3)C2)CC2CCCN2C(=O)N1 C1(C)(C(=O)OCC)CCCCN1C(c1c(Cl)c(C)nn1CC1CC1)C(=O)NC C1(NC(c2n(C(C)C)ccc2)=O)CN(C(=O)CCN(C)CCO)CC1C c1(OC)ccc(CC(O)C(=O)N2CCC2CNC(c2sccc2Cl)=O)cc1 C1(CC)CN(C(c2cccnc2O)=O)CCN1c1ncnc(-c2ccccc2)c1C N1(C(C(OC)OC)=O)CCC(F)(F)C(NC(=O)Cc2cc(F)cc(F)c2)C1 c1(CCC)nsc(N)c1C(N1CC(CC(C)NC(=O)Cn2cc(CC)cn2)C1)=O c1(SCCNC2CCNC2)cc(C)c(OC)c(C)c1.C(=O)(CCc1cnc[nH]1)C(C)=O C1(CNC(c2c(C)sc(Cl)n2)=O)CC2CCCC2N1C(=O)C#CC1CCCO1 C=CCCCCCCCC(=O)N1CC(O)CC1CNC(=O)COCC(F)(F)F c1(CCC(=O)NCCCCN(c2nnc(C(C)C)o2)C)ccc(S(C)(=O)=O)cc1 O=C(C1=CSCS1)NCCCNC(c1cc[nH]c1)=O N1(C(c2cscc2Br)=O)CCC(N2CCC(F)(CO)C2)C2(CC2)C1 C(C)(C(C)NC(C1(CCNC(=O)CCC2(C)N=N2)CCC1)=O)SC CCCS(=O)(=O)C(C)C(=O)Nc1nc(-c2cccc3c(Br)cccc23)cs1 c1(C(=O)OC)ccccc1CC(N1CC=CC(NC(c2cncnc2CC)=O)C1)=O C1(C(=O)NCC2CC2C(=O)NCCC(O)C2CCCC2)CC2(C1)CC21CC1 c1(C(N2CC(C(=O)NCCC(C=C)C)OCC2)=O)cccc(NC(=O)OC)c1OC N1(C(c2cnc(CC3CCC3)s2)C(=O)NC(C(=O)OC)C)CCCSCC1C1CC1 Cc1cc(Cl)c(C(=O)NCCCCNC(C2(Cl)CC23CCC3)=O)cc1C C(=O)(C(C)(C)CCCF)NCC(CC=C)NC(=O)CC1CC(=O)NC1=O c1(CN2CCCC(C#C)C2)c(Br)ccc(OC)c1O.c12cccc(c1)NC2=O Cc1nc(C(C)(C)C)sc1C(=O)N(C)C.C1(=O)C(C)N1 c1(C(N2CCC(C)(C(N3CCCC(F)C3)=O)C2)=O)cc(C2CC2)ccc1Cl C1(SC)CN(C(CCC2CC2)C(=O)NCc2nocc2Br)C2(CCC2)C1 CC1(C(N2CCC(O)C(C(=O)Nc3ccc(F)nc3)C2)=O)CCC(O)CC1 C1(NC)CCCN(CC(c2nnc(-c3ccccc3)n2C2CC2)O)C1 C(=O)(C1=C(C#N)CCC1)NC1(CC=CC(=O)NC(COC)C2CC2)CC1 c1(OC)ccc2c(c1)OC2(C)C.N12CC(F)CC1C2=O.C(C)(C#N)NC(C)=O N1(C(c2cccc(N)c2)=O)CC2COCCC2(NC(c2cc(C3CC3)[nH]n2)=O)C1 c1(C(=O)NCCC2CN(C(C(C(C)O)C)=O)C2)cc2nc(F)ccc2o1 C(N=c1[nH]c2ccccc2[nH]1)c1cccc(N(CCN(C)C)C)n1 C1(C(=O)NC2(CCC(NOCCCOC)=O)CCCC2)CC(C)CC(C)C1 c1(CCNC(c2n(CC)ncn2)c2nnnn2C(C)CC)cc(C)n(C)n1 c1(C(N2CCCC(C(=O)NCCCC3CCCCC3)C2)=O)c(O)ccc(F)c1F C1(CNC(c2cc(C)c(C)nn2)=O)CC2(CCC2)CN1C(c1ncc[nH]c1=O)=O c1(CC(=O)NCCCCCN(C(CCC=C(C)C)=O)C)ccc(F)c(F)c1F C1(C(=O)OCC)(CNC(=O)CN(C)C(c2cc(Cl)cs2)=O)CCCC1 c1(OCC=C)cccnc1C(=O)NC1(CO)CCN(C(c2cc(C)oc2C)=O)C1 Cc1cc(C2CCC2)ncc1C(=O)NCCOCCN(C)C(C1CCC(C)C1)=O N1(C(CC2(C(=C)F)CCC2)=O)CCOC(C(=O)NC(c2cnn(C)c2C)C)CC1 CCC(C)CCC(=O)NCC1(C(N2CC(C(C)(C)C)C2)=O)CC12CCC2 N1(CC)CC2(CN(C(C3C4CCN(C(c5c(C)nn(C)c5N)=O)CC34)=O)C2)C1 c1(C(=O)NCC(C)(C)NC(CNC(CN(C)C)=O)=O)cnc(C(C)C)n1C C(CCCCCC(=O)NCC1CCCSC1)NCc1c(Cl)cc(C)nc1 CC1CCN(C(c2csc(-c3nc[nH]n3)n2)=O)CCN1C(C1CCCN1C)=O c1(OC)ccc(-n2cc(C3CCN(C(=O)CC4OCCC4C)CC3)nn2)cc1C C1(C(N2CCN(C(=O)COC(C)C)C(C(F)(F)F)C2)=O)C2C=CC(CC2)C1OC C1(CSc2nc(CCC(=O)N)on2)CCC2(CCOCC2)CO1 c1(C(N2CC(C)C(NC(=O)Cc3ccc(Cl)s3)C2)=O)ccc2c(c1)C(=O)C(=O)N2 C1(CCNC(CCC(=O)NC)=O)CC(F)(F)CN1C(c1ccc(C(N)=O)cc1)=O C#CC1(O)CCN(C(CCCCC2CN(C(C3CCC4CC3CO4)=O)C2)=O)CC1 CC1(C)CN(C(=O)CC2CCCO2)CCC1C(=O)NCc1ncccc1F C1(C(N2CCC(CNC(C(CCSC)OC)=O)C2(C)C)=O)CCOC2(CCC2)C1 C1(CCC)CC(C(=O)NCCCCCCNC(C2(C#N)CC(C)C2)=O)CCO1 CC1=CCC(C)(C(N2CC(NC(C3CCCN3N=O)=O)CC(O)C2)=O)CC1 C(=O)(C1=CCCSC1)NC(CNC(Cc1c(OC(C)C)cccc1)=O)C c1(CC(N2CC(CCNC(C(C)NC(COC)=O)=O)C2)=O)c(Cl)cccc1Cl N(C1CN(C(C2CCCCCC2)=O)Cc2ccccc21)C(C(CC)C(C)C)=O c1(OC)ccc(CC2CCCCN2Cc2cnccn2)cc1F C=C=CC(C)C(=O)Nc1cccc(SC2CCOC2)c1 n1(CC)ncc2c(NCC(C(C)(C)C)NC(=O)CCC3CCC(=O)N3)ncnc12 C12(CNC(CCOCC)=O)CN(C(C3CCC4CC34)=O)CC1CCO2 C(=O)(C1=CC2(CCOC2)C1)NCC1C(C)CN(C(c2ccc(C#N)c(Cl)c2)=O)C1 C1(C(N(C)C)=O)CCCCC1C(N(C1CCN(S(C)(=O)=O)C1)C)=O N1(C(C(C)CO)=O)CCC(N(C(=O)Cc2cccs2)C)CC1 c1(SCC2CCCC(OC)C2)cc2ccc(O)cc2oc1=O c1(-n2c(C(CC)OC3CCCCC3)nc(-c3cccnc3)n2)ccc(C)c(F)c1 c1(CC)cc(C(N2CCC(CO)(NC(=O)Cc3nnc(C)s3)CC2)=O)ccc1O CCCC(CC)CCC(=O)NC(CC1CC1)C(=O)N(C)CC1COC(=O)N1 C(C(=O)NOCC(=O)O)CCC#C.C1(CCNC(=O)CCc2ccc[nH]2)CCOC1 N1(C(N2C(C(N3CC(N4CC(F)C4)C3)=O)CSC2)=O)CCC(F)(CF)C1.N1CCCC1 c1(C(N2C3CC(CNC(Cc4nc(C)sc4)=O)(OC3)C2)=O)ccc(C)c(F)c1F C1(NC(c2c(C)nsc2)=O)CCN(C(C2CCC(C)CC2)=O)CC(O)C1 N1(C(c2c(C)cc(F)nc2)=O)CCC2CCC(C1)N2C(=O)CSCc1cccs1 Cc1cnc(C(=O)NC2(CCNC(=O)CC3(C)CC3)CC2)cc1Br c1(C(N2C(C(=O)NC)CCC2)=O)cnc(CNC(=O)C(C)n2cncn2)nc1 c1(CC(N2CCC(OCCNC(C3C(=C)CC3)=O)C2)=O)ccc(Cl)nc1C c1(C(N2CC(NC(c3cc(CC)ncc3)=O)C3(C2)CC3)=O)ccnc2ccsc12 C(C(=O)N=c1ccn(C2CN(C(=O)Nc3ccc(C#N)cc3)C2)[nH]1)=CCC=C N1(C(c2ncn(Cc3nc(C)no3)n2)C(=O)NCC=C)CCC(C(C)(C)C)CC1 C1(COC)CCCN(C(C2C3CN(Cc4cnc(C5CC5)nc4)CC23)=O)C1 C1(CNC(c2c(C)cns2)=O)C2CN(C(c3cc(C(C)C)n(C)n3)=O)CC12 c1(N2C(C(=O)Nc3ccc(CC)cc3O)CCCC2)nc(O)c2ccccc2n1 c1(OC)ccc(N)c(C(=O)NC2CCN(C(c3ccnn3C)=O)C2C)c1 Cc1cc(N2CCC(COC(=O)Cn3cc(Cl)cn3)C2=O)ccc1Br c1(CN2CC(COC)C2(C)C)cnc2ncccn12 N1(C(c2nc(C(C)NC(C(COC)C)=O)oc2)=O)CCC(N(C)C)C(C)C1 N1(C(CCCCC=C)=O)CC2OCCN(C(=O)Cc3ccc(F)cc3F)C2C1 CC1(C)C(NC(C2CC3C=CC2C3)=O)CC1CNC(C1CCC=CCC1)=O N1(C(C(CNC(=O)C(C)(O)C(C)C)(C)C)=O)CC2CC(NC3CCN(SC)C3)C2C1 C12(CNC(=NCC)NCC3CCCC3NC(=O)OC(C)(C)C)CCCN1CCC2 C=CCCC(CC(C)C)C(=O)NCCC1CCCCN1C(c1cnc(OC)s1)=O C1(NC(C=CCOCCOC)=O)CCSC12CN(C(C1CCOC(C)C1)=O)C2 N1(C(CC(CN(C)C)O)=O)CC2(C)CN(C(c3nc(=O)n(C)[nH]3)=O)CC2(C)C1 C12(CNC(CCOC)=O)CCCC1N(C(=O)Cc1conc1C)CCC2 c1(C(N(CCCCNC(c2scc(C)n2)=O)C)=O)c(C)coc1C1CC1 O=C(CCC1=CCCCC1)N1C(CC(=O)NC2CC3(CC3)C2)C2CCCC12 CC(C(=O)NCC(O)CNC(c1ccc(-c2nnc[nH]2)cc1)=O)S(N)(=O)=O N1(C(c2cc(OC)n(C)n2)=O)CCN(C)C(C(N2CC(O)(CCO)C2)=O)C1 CC(C)CC(C(=O)NCC1(O)CN(C(=O)C(n2ccc(Br)n2)C)C1)C(C)C.C=O C1(NC(c2nc(CC)oc2)=O)CCN(C(c2csnc2C2CC2)=O)C1C(C)(C)C C1(C(=O)NC)CCN(C(=O)CCC2(NC(=O)C(C)(Cl)Cl)CCC2)C1 Cc1ccc(Cl)c(O)c1C(=O)NCC(C(C)(C)C)NC(=O)C(C)SC(C)C c1(C(N(C(C)C(=O)N)C2(CC(N)=O)CC2)=O)ccc(CC2CC2)cn1.C(C)(C)C n1(CC)ccnc1C=CC(=O)NC1CC2(C1)CC2NC(C1CCS(=O)(=O)N1)=O N1(C(=O)NC(CC)CSCC(C)(C)C)CCOC(CC(=O)OC)C1 C1(CCC(NOCC#C)=O)CCCCN(C(c2ncc(F)cc2N)=O)C1 C=CC1(C(=O)NC2CC23CCC3)CCN(C(=O)CC(C)n2cccc2)CC1 N1(C(c2cc(CC)c(C)s2)=O)CCN(C(c2cnc(C)cc2Cl)=O)C(CCO)C1 CC1(CNC(C2(C3CCC3)CC2)=O)COCCN(C(c2ccc(N)c(O)c2)=O)C1 C(=O)(C(CC(C)C)NC(c1cc(C(N)=O)co1)=O)N(C)CC1N(CC)CCC1 N1(C(C2(CC)CC2)=O)CCC2(CC1)CN(C(=O)C=Cc1nccn1C)CC2CO CC(C(C)NC(=O)C(c1cscn1)OC(=O)CC)NC(=O)COC(C)(C)C N1(C(Cc2nc(C)sc2)=O)CCCN(C(C2CC(S(C)(=O)=O)C2)=O)CC1 C(c1ccccc1C)=CC(=O)NCC(CN(C(C1CCCC(OC)C1)=O)C)C C(=O)(C(C)Cc1cnc[nH]1)N(CCN(C(COC)=O)C)C C1(C)(CNC(C(c2ccc(C)s2)C)=O)CCCC1NC(C1C2CCCCC12)=O C(C)(N=c1[nH]c2c(c(=NCc3ccnc(CO)c3)[nH]1)SCC2)c1nc(C)oc1C c1(CN2CCCC(C)(CNC(c3cc(O)no3)=O)C2)ccc(F)cc1C#N C1(NC(C2(CC#C)CC2)=O)CCN(C(=O)CCOC(C)=O)CC1=O c1(C(=O)NCC(C)N(C)C(C2CCC=CCC2)=O)cncc2nc(O)[nH]c12 CC(CN1CCC(O)CC1)CN=C(NCC1CCOC1)NC1CCCC1 N1(C(c2nc(C)oc2)=O)CC2CC1(CNC(c1c(-c3cccs3)noc1C)=O)C2 c1(C(=O)NCCCCCCCn2cc(C3CCC3)nn2)cnn2c1OCC(F)C2 c1(NC(C(C)N(C2CCN(Cc3ccccc3)C2)C)=O)cc(F)c(Cl)cc1F C(=O)(C1=C(F)CN(C(C2CCCC2F)=O)CC1)NC1CC(C)(O)C1 c1(C(N2CCC(NC(CCc3c(C)ncs3)=O)C(O)C2)=O)ccnc2[nH]ncc12 c1(C(=O)NCC(CNC(c2nc(C)nc(O)c2)=O)F)cc(Cl)cc(Cl)c1O N1(C(C2(COCC)CC2)=O)CC(NC(c2cc(O)ccc2C)=O)CC(F)(F)C1 C(=O)(C(CNc1coc(C)c1)CC(C)C)OCCCSCC C(=O)(C(F)(F)C(F)(F)F)NCCC1CN(C(c2c(CCC)n[nH]c2)=O)CC(C)O1 c1(C(=O)NCCCCNC(c2c(COC)onc2)=O)n[nH]c(C)c1C c1(C(C)=O)cnc2sc(C(N3CCCS(=O)(=O)CC3C)=O)c(C)c2c1 C1(C(=O)NC(C2CCN(C(c3c(CC)n(C)nn3)=O)C2)(C)C)CC12CCOCC2 Cc1cnc(C(=O)NCC(c2ccccc2F)NC(c2cnn(C)c2Cl)=O)cn1 c1(NCCN(C)CCO)cc(O)cc(F)c1 N1(C(C(c2ccccc2F)OC)=O)CCC12CN(C(=O)CN1CC3CCC1C3)C2 N1(C(c2c(C)ccs2)=O)CCCC12CCCN(C(=O)C1=CCC(C)CC1)C2 c1(C(=O)NCCc2cn(C(CC=C)CC)nn2)cccc2c1C(=O)NC2=O N1(C(C(C)(C)CC2CC2)=O)CC2(CC(C(N3CC4(CC4)CC3CO)=O)C2)C1 C(=O)(CC(C)(C)O)N(C(CNC(C1NC(=O)CC1C(F)(F)F)=O)C1CC1)C c1(OC)cc(CNC(=O)NCC2CCC(CO)CC2)c(NS(C)(=O)=O)cc1I c12c(F)cc(cc1F)N(CC)CCCNC2=O.C12(C(=O)OC)CC3CC1C2C3O N1(C(c2nn(C(C)C)nc2Br)C(=O)NCCSC)CC(C)CC(C)C1 c1(NC(CNC(CCCOC(C)C)=O)C(C)C)cncc(Cl)n1 Cc1ccc(NC(c2ncoc2CNC(C2(C)CC(=O)N(C)C2)=O)=O)c(C)c1 C1(C#N)(N(C(=O)C(c2ccccc2F)NC(=O)OC(C)(C)C)C)CCOC1 N1(CC(CCCC)C)CCN(CC(=O)Oc2ccc(F)cc2)C(=O)C1 c1(C(=O)NC(CCCC)CNC(=O)C(C)COC)cc(CO)ccc1OC c1(N(C2CCN(C(c3c[nH]nc3-c3ccsc3)=O)C2)C)ncccc1S(C)(=O)=O c1(C(=O)NC2CN(C(CC(CC)CC)=O)CC2C)ccc(F)c2cnccc12 Cc1cncc(C(=O)NCc2cn(C3CCCN(C(=O)CO)C3)nn2)c1C Cc1cc(C(=O)NC(C)CCCNC(c2cnc(C3CC3)o2)=O)nc(C)c1 C1(c2ccccc2)(NC(C=COCC)=O)CCN(C(C2C=CCCC2)=O)CC1 c1(CC(=O)N(C(CNC(CCCOCC=C)=O)C)C)cccc(Br)c1F C(CC1C(=O)Nc2ccccc21)NC(c1nc(Cl)sc1Cl)c1n(CCOC)nnn1 CC1(C)CC(C)(CNC(c2ccn3cncc3c2)=O)CN1C(=O)C=C1CCC1 CCCC(C(=O)N1CCC1CNC(C1CC(=C2CC2)C1)=O)NC(N)=O C1(COC)C=CCCN1C(c1n[nH]cc1CNC(=O)CCc1ccccc1)=O C1(C2CCN(C(=O)CC3CC4CC4C3)C2)(NC(CSCCN(C)C)=O)CC1 c1(OC)ncc(C(=O)NCCC2CCC(NC(C3(F)CCCC3)=O)C2)s1 N1(C(C(C)OC2CCCC2)=O)CC(C(=O)NC2CCCCCC2)C(C2CC2)C1 c1(C(N(C2CCCN(C(C3CC=CCC3)=O)C2)C)=O)nc2n(c1C(C)C)CCCC2 C1(CC)CN(C(=O)C(=O)NC(C)C)CCC1NC(C1(c2cc(C)ccc2C)CC1)=O c1(NC(CCCCNC(c2nc(CCC)oc2)=O)C)[nH]c(=O)n(C)c(=O)c1C#N C(C(C(=O)N(C)CC1CCCO1)C(C)(C)C)NC(c1n[nH]c(C)c1C)=O C1(CC(=O)N(C(=O)CCCc2cccs2)C2CC2)CCCN(CC(c2nccs2)=O)C1 N1(C(c2cc(C)oc2)=O)CCC(O)(C(C)NC(=O)C=CSc2nc[nH]n2)C1 c1(OC(C)C)ccc(OC2CCN(C(=O)C(=O)NC3(C(=O)O)CCOC3)C2)cc1 C1(C(N)=O)CCN(C(=O)C(Cc2ccco2)NC(c2ccsn2)=O)CC1 Cc1ccnc(C)c1C(N1CC(O)(c2cn(Cc3ccno3)nn2)C1)=O N1(C(C2CCC(=O)N2)=O)CCC2C(CCN2C(=O)CCc2ccc(O)c(F)c2)C1 C(=O)(C(CC(C)C)C(C)C)N1CCC(OCCNC(Cc2cc(C)[nH]n2)=O)C1 C1(C(=O)NC(C2CCN(c3nc(Cl)c(C#N)s3)CC2O)C)Cc2cncn2C(=O)N1 c1(NC(C(=O)NC)C2CC2)nccc(=NCC23CC(C(F)F)(CO2)C3)[nH]1 c1(-c2cn(-n3c(C)c(C(=O)NC(C)C)cn3)nn2)cnn2c1NCC2 c1(COC)ccc(S(=O)(=O)N2C3CN(C(=O)CN(CCO)CCO)CC23)n1C c1(C(N2C(CNC(c3c(CC)scn3)=O)CCCCC2)=O)cn2cccnc2n1 C1(NC(c2cc(C(N)=O)[nH]c2)=O)CN(C(C2CCC3(CC3)C2)=O)CC1O n1(CC)ncc(NC(=O)CCOC2CCOCC2)c1C.C12CC(C1(C)C)NC2 c1(OC)ccc(Br)cc1C(C1CC1)NC(=O)CN1CC(C)OC(C)C1 C1(C(N2C(c3cccc(NC(C)=O)c3)CCCC2)=O)CCC(C)(C)OC1 C1(C(=O)NCC2C=CC(NC(=O)CCC3(C)CC3)C2)(OC)CCSCC1 N1(C(C2C(C(=O)OCC=C)C2)=O)CCCC2(C1)CN(C(=O)CC1C=CCCC1)C2 N1(C(C2CC(OC)(OC)C2)=O)CC2CC(NC(=O)Cc3[nH]cnc3C)C1C2 C(=O)(C1CCCc2nccn21)NC1CCC(C)(NC(CC(=C)Br)=O)CC1 C1(C)(NC(C=C(COC)C)=O)CCN(C(=O)CC2CC3C=CC2CC3)CC1 C(=O)(C(C)(F)C(C)(C)F)N1C(C2CCN(C(C(c3ccccc3Cl)C)=O)C2)CCC1 C(C)(C(=O)NCC#CCNC(=O)CC12CCCC1C2)(c1ccccc1)N(C)C C1(NC(CCCCCC)c2nnnn2C2CCCC2)COc2ccc(Br)cc2C1 C(=O)(C1=CC2CCC=CCCC12)N1CCCC(CN(C)C(c2cncc(Cl)n2)=O)C1 N1(C(c2cc(C)sc2C)=O)CCCN(C(c2c(C)nn3ccccc23)=O)CCC1 Cc1nn2cc(C(=O)N(CC(N3CCCCC3)=O)CC3(C)CCC(C)C3)nc2s1 C1(C(N(C2(CC(=O)NC3CCC(OC)C3)CC2)C)=O)CCCC(O)C1 Cc1csc(=O)n1CCC(=O)NC(C)(C)CNC(C1CC=CC1)=O C(=O)(C(=O)C(C)(C)C)NCC(C1CCCN(C(=O)Cc2cccs2)C1)(C)O C1(CC)CN(C(=O)C(c2cc(C)ccc2F)=O)CCN1C(c1cccn1C)=O c1(OC)cc(C(N2CCC3CC3(NC(c3nccn3C)=O)CC2)=O)c(N)c(C)c1 N1(CCC)CCCC(C(N2CCC(NC(=O)C(C)(Cl)Cl)C2CCOC)=O)C1 C(CCC(N)=O)(C(=O)N1CCSC(C)C1)n1cc(CSC(C(=O)OC)C)nn1 c1(C(=O)NC2C(CNC(Cc3nc(C)sc3)=O)CCC2)cnn(C)c1S(N)(=O)=O N1(C(C(CC(C)C)C)=O)CCCN(C(c2cc3oc(Cl)cc3[nH]2)=O)CCC1 N1(C(C(C)OCC2CC2)=O)CCN(C(=O)Cc2cnn(C)c2)CC2(C)CCCC12 Cc1cc(S(=O)(=O)NCCC(C)C(F)F)c(C)cc1C(F)F c1(C(=O)NCCC2(NC(Cn3c(C)c(Cl)cn3)=O)CC2)ccc(C(N)=O)c(Cl)c1 N1(C(C2(OC)CCCOC2)=O)Cc2nccn2CC(NC(c2occc2C)=O)C1 c1(C(N2C3CC(NC(c4c(C)nc(C(C)C)s4)=O)C2CC3)=O)nn(C)c2c1CCC2 C(=O)(C1=CNC2=NCCCN12)NCCC1(O)CCN(C(C(CC)(C)CO)=O)CC1 N1(C(=O)Cc2cccc(F)c2)CCCC2(CCN(S(=O)(=O)c3ccoc3)CC2)C1 C#CC(C)(C)C(=O)NCC(C(C)(C)C)NC(=O)CCC1CCCCO1 c1(CC)nnc(C)cc1C(=O)NC1CCCC1NC(=O)C(N)=O N(C1COc2ccc(Br)cc21)CC(N1CC(C)OCC1)=O C12(C(N3CC(CN(C(=O)CC4CCCC4)C)C4(C3)CC4)=O)CCC(F)(CC1)CC2 c1(C(CNC(C(C)OCC)=O)NC(c2cn(CC(F)F)cn2)=O)ccc(C)cc1 c1(C(=O)OCC)c[nH]c(=NC2CC(CNC(=O)C(C)(C)CC3CC3)C2)cn1 c1(C2(C(C)NC(C34CC5CC3C4C5O)=O)CCC2)ccc2c(c1)CCC2 N(C(=NCc1ccsc1)N1CCN2C(=O)OCC2C1)CCC(=O)NC(C)C C(CC(CC)C(=O)N(CCCC(=O)NCCN(C(C)CC)C)C)=CC Cn1cc(C(F)(F)F)cc1C(=O)NCCc1ccccc1C(=O)O Cn1cc(F)cc1C(=O)NCCC1CCCN(C(c2ncccc2Cl)=O)C1 c1(OC)cc(Br)cc(F)c1C(N1CCC(CC(=O)NCc2ccc(Cl)c(F)c2)C1)=O Cc1c(C(=O)NC2(CCNC(=O)CC3CCCCC3F)CCC2)ccn1C1CC1 c1(C2(O)CN(Cc3n(C)cnn3)C2)cccc(F)c1C(=O)Nc1ccccc1 c1(C(=O)OCC)ccc(F)c(Cc2nc(-c3ccc(Cl)cc3)n[nH]2)c1 C1(NC(C)=O)CCCN(C(=O)CCc2cnc(C)o2)CC1F Cc1ccc(CC(C)C(=O)NCCCN(C(=O)Cc2ccc(C)o2)C(C)C)cc1 C(=O)(C(O)CC(C)C)N1CCC(N(C(C)(C)C)C(c2nc(COC)oc2)=O)C1 C1(NC(c2c(C)ocn2)=O)C(C)(C)C(NC(c2cccn3cnnc23)=O)C1(C)C N1(C(c2c(F)ccc(C#C)c2)=O)CCC2(CCC(C(=O)N(C(C)C)C(C)C)O2)CC1 C(=O)(C1=CCC(NC(=O)CCC(=O)C2CC2)C1)NCC(CO)OC(C)=O c1(Sc2c(C(=O)NC(C3CCCO3)CC)cccc2)ccc(Cl)cc1 c1(C(=O)NCC2C(NC(C3(C)CCC(C)C3)=O)CCC2)c(O)cccc1F Nc1cnccc1C(N1CC(F)CC1CNC(c1cnsn1)=O)=O CCC(CC)(C(=O)OC(C)(C)C)C(=O)NC1CC(NC(=O)C(CO)NC(N)=O)C1 CC1(CNC(=O)CC2CC3C=CC2CC3)CCN(C(=O)CC2CCCSC2)CC1 c1(C(=O)NCC23C(CN(C(C4C(OC)CCC4)=O)C2)C3)ccc(=O)n(C)c1 N1(C(COCCSC)=O)CC(C(=O)NC2CCCC2CCO)CC12CCC2 C1(C(N2CCN(CC#C)C(=O)C2)=O)CC12CCN(C(c1c(Cl)cccc1Br)=O)CC2 Cc1cc(C(=O)NCCCCCN(C)C(c2cn(Cc3cnns3)nn2)=O)c(C)o1 c1(CN2CCC(=CC(=O)Nc3ccncn3)CC2)c(O)cccc1F CC(C(=O)NC1(CCNC(=O)CC2CC23CC3)CC1)S(C)(=O)=O Cc1nc(C(N2CCCC2C2(N(C(=O)CC3CCC(=O)N3C)CC)CC2)=O)nn1C c1(N2CCC3NC(=O)OC3C2)nccc(=NC2CCN(c3ncccn3)C2)[nH]1 N1(C(C2CCCCN(C(CCC(C)CN(C)C)=O)C2)=O)CC2CCC(CO)(C2)C1 c1(C(N(C(C)CNC(C23CC(N(C)C)(C2)C3)=O)C)=O)cn(C)nc1-c1cccs1 c1(C(=O)NC2CN(C(C3C4COCC34)=O)CC2CC2CC2)ccn2nncc2c1 CC(C#N)CCC(=O)NC1(CNC(C2CC3C(C2)C3(F)F)=O)CCCCC1 C1(CN(C(=O)CC2CCC2)Cn2cc(C3CCCC3O)nn2)(C)CC12CCC2.C1CC1 N1(C(COCCCC#C)=O)C2CCC(C2)C1CC(=O)NCCc1cc[nH]n1 C(=O)(C1=Cc2ccccc2C1)N1CCC(CNC(C2CS(=O)(=O)C2)=O)C1 N1(CC(C)C)CCCC(C(=O)NC2CCC(CNC(=O)C(C)c3cccs3)C2)C1 C(=O)(C(O)C(C)(C)C)NC(CC#C)C(=O)NC1CCCCC1CC=C C12CCN(CC1)CCN2.c1(CC)cc(COC)on1 C1(NC(c2c(C)noc2N)=O)CC2CCCC(C1)C2NC(C1C=CCC1)=O N1(C(c2ncn(CC)n2)=O)CC(NC(=O)CCc2n[nH]c(=N)s2)CC12CCOC2 N1(C(COCC)=O)CC2(C1)C(NC(=O)COCCC1CCCC1)CCS2(=O)=O C1(CC=C)(NC(C2CC2C)=O)CCN(C(C2CC(OC)(OC)C2)=O)C1 CC12CC(C(=O)NCC3CC4(CC(NC(=O)Cc5cscn5)C4)C3)C(CO1)C2 c1(C(N2C(CCNC(C(C)C)=O)CSCC2)=O)cccc2c1C(C#N)C2 CC1=C(c2cc(C(=O)N(C)CCO)c3ccccc3c2)CCCC1 c1(CC(=O)NCC(COC(C)C)O)cncc(F)c1 C#CCCC(C(=O)NCCOC1CCN(C(C)=O)CC1)NC(=O)CC=C(Cl)Cl C1(C(N(CCNC(=O)Cc2occc2C)CC)=O)COc2ccc(Br)cc2C1 CC(C)(O)C#CC(=O)N1CCC(NC(=O)Cc2cc(C3CC3)no2)C1(C)C c1(NCc2ccc(C)o2)cc(N2CCC(C(F)(F)F)C2)nc(C)n1 Cc1nc(NC2CCCCC(P(C)(C)=O)C2)cc(=NCCC2CC2)[nH]1 C(=O)(CCCCC(C)(C)C)N1CCCC(C(N(C2CCN(CC)C2)C)=O)C1 C1(Cl)(C(=O)NCCCN(C(=O)C=Cc2ccccc2C)CC)CC2CCC1O2 Cn1cc(S(N)(=O)=O)c(C(=O)NC2(C)CN(C(C34CCCCC3C4)=O)C2)n1 C1(C)(C(=O)NCc2c(C(=O)NC(c3ccccn3)CC)n[nH]c2)CCC(C)C1 c1(C(=O)NCC(C)(CO)NC(c2ncn(C)n2)=O)cc(Br)cn2ncnc12 N1(C(c2nc(C(C)C)sc2)=O)CCCC2CN(c3nnc(C(F)(F)F)s3)CCC12 C(=O)(CC1=NN(C)C(=O)C1)NCC(C)N(C(C1CC1CF)=O)CC N1(C(c2cnc(C)s2)=O)CC2CC(C1)CN(C(=O)Cn1cc(C#N)cn1)C2 c1(C(=O)Nc2c(N(C(=O)CC34CC(C3)C4)C)cccc2)cc(C#N)ccc1F C1(C(=O)NCC(C)NC(=O)CCc2cn[nH]c2)CC12CCc1ccccc12 C1(C(N(C(C(=O)NC(CCOC)(C)C)C2CC2)C)=O)CCN(C)C(=O)C1 c1(CC(=O)N(CCCN(C)Cc2cc(C3CC3)sn2)C)cc(F)ccc1F n1(CCC)ccc(C(=O)NCC(C)(CO)NC(c2ccsc2C)=O)n1 c1(CN2CCCC(C(C)NC(c3cc(O)nc(Cl)c3)=O)C2)ccccc1[N+](=O)[O-] c1(CN(C)C)ccoc1C(=O)NCC(F)CNC(=O)CN1CC2CC2C1 C1(CCOC)CN(C(C2CNC(=O)O2)=O)CCN1C(c1ccsc1OC)=O c1(C(C(=O)N(CCNC(c2c(C)occ2)=O)C(C)C)C2CC2)ccc(F)cc1 C1(OC2C(C(=O)OC)NCC2)(OC)CCC(C(F)F)CC1 N1(C(=O)COC2CCOC2)CCC2(CC1)CCN(C(C1CCCC(CF)C1)=O)C2 C1(C#N)(C(N2CC(F)(COC)C2)=O)CCN(C(c2ccn(-c3ccccc3)c2)=O)C1 c1(C(=O)NCC2C(OC)CN(C(C(CCC)OCC)=O)C2)nc(C)ccc1C c1(NC(C)CC(C)O)nccc(=NCCC2SCCS2)[nH]1 N1(C(C2C(CCC)CCC2)=O)CC(CNC(c2ccnc(CC)n2)=O)C(CC)C1 C1(C(=O)NCCCOC=C)(NC(=O)C=NOC)CC12CCC2 C1(CNC(COCCOCCOC)=O)CN(C(=O)CC(C)F)CC1C c1(C(N2CC(N(C(c3cc(C)n(C(C)C)n3)=O)C)C2)=O)ccc(S(C)=O)cc1 Cc1cc(C)n2nc(C(N3C4CCC3C(F)C(NC(=O)C3=CCC3)C4)=O)cc2n1 CCCCCCCC(C(=O)Nc1c(C)cccc1C)N1CC(O)CCC1C c1(C(=O)NC(CCC)C(N2CCC(C)(C)C2C)=O)cnn2ccc(Cl)c(F)c12 c1(C(N2C(CNC(C(CC(CC)C)C)=O)CC2)=O)cccc2c1C(=O)CCN2 CC(C(F)(F)C(F)(F)F)=CC(=O)N(CC(C)(C)NC(C1CC(C(C)C)C1)=O)C N12CCN(C(C3CC3)C1)C(=O)CCOC(C)C2=O.c1(OCSC)cc(F)ccc1F CCCCC(CN=c1ccc(C#N)c(C)[nH]1)NC(=O)COC1CCC1 N1(C(CC)=O)CCCC(C(=O)NCC(O)CNC(c2cnn(C3CC3)c2)=O)C1 C=C1CCN(C(=O)CC2CC3(CC3)C2)C(C(=O)NC2CN(C)CC2O)C1 C#CCC(CC(F)F)C(=O)N1C(CCC(=O)N(CC2CCCCC2)OC)CC1 C12(NC(CN3C(C)CCC3)=O)CCOC(CNC(c3cc[n+]([O-])cc3)=O)(C1)C2 Cc1cc2[nH]c(C(=O)NC3(C)CN(C(=O)CC4CC4c4ccccc4)C3)cc2o1 C1(N)CC(C)N(NCCCC#C)C1.c1(C)cnn(C(C)C)c1 C=CCC(CC=C)C(=O)N(C(C)CN(C(=O)C(c1ccc(O)cc1)C)C)C CCCCCCC(C)C(=O)N1CCC12CN(C(C1CCC=CCC1)=O)C2 c1(NC(=O)CCNCCC2CCNCC2)c(F)cc(F)c(F)c1N1CCOCC1 C1(CCC(=O)NC2CCOCC2F)CCCCN1C(c1ccsc1Cl)=O CC(F)(F)CCC(=O)NC1CC1CNC(=O)CC1CCS(=O)(=O)C1 C(=O)(C(F)(F)C1=CCCCC1)NCC(CO)NC(c1[nH]cc(C(=O)OC)c1)=O C1(CCC=C)(C(=O)NC(CCC)C2CCC2)CN(C(=O)C=Cc2cncs2)C1 C1(CNC(C(C)NC(=O)NC)=O)CN(C(=O)CCCN(C)C)C2(CCCCC2)C1 O=C(CSc1cccc(Cl)c1)NNC(=O)NC12CCC(CC1)CC2 N1(C(C(CC#C)(C)CC)=O)CCC(NC(=O)Cc2cnc(C)[nH]2)C(F)(F)CC1 C(=O)(CN=c1cc[nH]cc1)NC(CNC(c1nc(OC)c(C)s1)=O)C(C)C(C)C Cn1cnc(Cl)c1C(C(=O)NCCOC1CC1)N(C)CCC1(C)CC1 c1(C(=O)NCC2N(C(C(C(CC)O)(F)F)=O)CC2)cnc2c(F)cccc2c1 N1(C(C2(C)CN(C(C3CN(OC)C(=O)C3)=O)C2)=O)CCC2(CC1)CC2C#N CC(CC(=O)N(C1(C(C)O)CC1)C)NC(C1CCOC1)=O C(=O)(C(C)(C)C(N)=O)NC1C(OC)CN(C(=O)COC2(C)CCCC2)C1 C1(CNC(C(CC#C)(C)CC)=O)CN(C(c2cncc(C)n2)=O)CCC12CCC2 C1(O)(CC)CN(C(=O)CCC2CC(NC(c3ccc(C)[nH]3)=O)C2)C1 C1(C(=O)NC(CC=CC(=O)NCC(C)C(F)F)(C)C)CCC(=O)N1C N1(C(C=C(CCC)C)=O)C2CCC1C(C(=O)NC13CCCC1OCC3)C2 c1(C(N2CCN(C(=O)C=CCO)C(CF)C2)=O)cc2cc(Br)ccc2[nH]1 C1(CC=C)(NC(c2ccnn2CC)=O)CCN(C(=O)C(COC)N(C)C)C1 C(N=c1[nH]c(=N)[nH]c(=NC(C)C2CC2)[nH]1)c1c(C)coc1C N1(CC)CCOC2CN(S(=O)(=O)CCCCl)CC12.c12cc(F)c(c(F)c1)C(C)N2 C(=O)(C1CCc2ccccc21)NCc1cn(C(c2c(C)cc(Br)s2)C)nn1 Cc1ccc(OCCCCC(=O)N(CCNC(C2CC2(F)F)=O)C2CC2)c(Cl)c1 C(=O)(CCCCN(C)C)NCC1(C)CC(NC(CC2CC(=C)C2)=O)C1 C1(C(=O)NCCCCCNC(C2(C)CC(=C)C2)=O)Cc2cc(OC)ccc2O1 C1(NC(C(Cc2cnc[nH]2)NC(c2n(CCC)ncc2)=O)=O)CCCC12CC2 c1(C(N2CCC(CO)(COC)CC2)C(=O)NCCC)cc2nccc(Cl)c2s1 N1(C(c2c(C)snc2)=O)CCC(C)(CCNC(c2cscn2)=O)CC1 C1(C(N2C(C(=O)NC3(C(=O)OC)CCCC3)C(C)C2)=O)CN(C)CCN1C N1(CC(N2C(C(C)NC(COCCCOC)=O)CCCC2)=O)CCCCS1(=O)=O c1(OCC(=O)NC2(C)CC(C(=O)NC3C(C)CCCC3)C2)ccc(F)c(F)c1 c1(CC)ccc(C=CC(=O)NCC2C(C)CCN2C(C2CC(C)OC2C)=O)o1 C(=O)(CCCC(C)(C)C)NCCn1cc(C(=O)NCCC(C)(C)C(N)=O)nn1 C#CCCCCCC(=O)NC1CC2CCC1CC2NC(=O)CC(C=C)CC CCCC(C(=O)NCC1(O)CC(CNC(C2CC3(CCC3)C2)=O)C1)S(N)(=O)=O N1(C(CCC)=O)CC2C(C1C(=O)NCC(c1cccc(OCC)c1)O)C2(C)C C1(C(N(CCCNC(C2CC2F)=O)C)=O)CC(Cl)(Cl)C1 N1(C(COc2c(C)ccc(C)c2)=O)CC2CCC1C(NC(=O)C=CC1CCC1)C2 N1(C(Cc2onc(C)n2)=O)CC(C)CC1C(N1CCC(Br)C1)=O C1(NC(=O)CCc2ccon2)CC(O)CN(C(=O)C(c2ccc(Cl)cc2)(F)F)C1 CN1CCc2cc(C(=O)OCC3CC3N(C(=O)COC3CCOC3)CCO)ccc21 c1(CC)nccc(C)n1.O1NC(=O)C2(CCC2)CNC(=O)C1 C1(C(=O)Nc2ccccc2-c2ccnc(C(F)(F)F)c2)CC2(CCOC2)C1 N1(C(C2C(CNC(C=CC(C)(C)SC)=O)CC2)=O)CC(O)CC12CCCC2 N1(C(CCOCCOC)=O)CC(C(=O)NC)CC(C)(C)C1.C1CCCNC(=O)N1 O=C(C1CCCn2ccnc21)NC1C2CCN(C(C3(CF)CC3)=O)CC12 CC1(C#CC(=O)NC2(C3CCCN3C(c3coc(C(F)F)n3)=O)CC2)CCCO1 N1(C(C(C(C)C)OC)=O)CC2CCCC1C2CNC(c1csc(O)n1)=O c1(OC)cnc2[nH]c(C(=O)NC(C)C(C)(C)NC(=O)C(F)=C(C)C3CC3)cc2c1 c1(CC)ccc(C(=O)NCCCN(CCCCNC(=O)CC2CCCC2O)C)cn1 C(=O)(CC(C)(C)O)NCCCC(C)NC(=O)COCc1ccnn1C N1(C(CC2(C)CCC2)=O)CCC(CO)C(NC(=O)Cc2cncc(C#N)c2)C1 N1(C(CC=CC=C)=O)CCOCCC1C(=O)NCC1=C(C)CCC1 C(=O)(CCC(C)CCCCC(=O)OC)NC1CC(F)(CCC)C1 Cc1onc(-c2cccs2)c1C(N1CC(F)(CNC(c2snc(O)c2Cl)=O)C1)=O C1(COC)(CNC(C2C=CCC2)=O)CCCN1C(c1n[nH]cc1Br)=O C(C(C(=O)NC1(CNCC)CC1)n1cc(CO)nn1)OC(C1CNC(=O)N1)=O Cc1cccc(C(N2CCC(C(F)C(=O)NCCCN(C)C(C)C)C2)=O)n1 C1(C)(C(N2CCC(CNC(Cc3c(C(C)C)cccc3)=O)C2)=O)CCCS1(=O)=O C1(N(C)C(C2(CNC(c3ccc(CC(C)(C)C)o3)=O)CC2)=O)CCCC1C(N)=O C1(CC(=O)NCC(C)=CC(=O)N(C)C(c2nc[nH]n2)C)CCN(C)C1 C(=O)(C(CC(C)C)NC)NC(C1CN(CC)C(=O)C1)=O.C1(CC(=O)NC)CC2CCC1O2 N1(C(CC2CN(C)C2)=O)C2COCC1CC(NC(c1ccc3[nH]ccc3c1)=O)C2 CC(F)(F)C(F)(F)C(F)(F)F.C(c1nc2ccccc2o1)N1c2nc(no2)C1 C1(NC(c2nc(C)n(C(F)F)c2)=O)CS(=O)(=O)C2CN(C(=O)C(C)CO)CC12 N1(C2CN(C(C)=O)C2)CC(CNC(=O)C(C)(O)c2ccccc2)CC1=O c1(C(N(C2CCCC2)CCNC(COCCC#C)=O)=O)cc(C)ccc1F C(c1ccccc1)=CCCCCCn1cncn1.N1(CC(=O)N)CCC(C(=O)C2CC2)C1 CC(C(C)(C)C(=O)NCC(C)(C)CN(C)C)NC(C1CCCC(=O)CC1)=O c1(C(=O)NC(CCN(C(c2ccc(SC)o2)=O)C)C)ccncc1F c1(N2CCCC(C(N3CCC(=O)NC3=O)=O)CC2)cc2ncc(Br)cn2n1 C1(C(=O)NCC2(C)CC(CN)C2)CCCC(C(F)F)C1 C(=O)(CC(CN(C)C)C(F)F)NCCOC1CCN(C(C#CC(C)C)=O)C1 C1(C(=O)NC(CC)C(N)=O)CC(C)CN1C(c1snc(C)c1N)=O c1(C(N2CCOC(C(=O)NC(C)C)C2)C(=O)NC(CC)C)cc(S(C)(=O)=O)cs1 N#Cc1ccc(C(=O)NCCC2CCN(C(=O)C=Cc3cncs3)C2)nc1 C(=O)(C(C)(C)CCNC(C1CC2CCCC2C1)=O)NC(C(=O)OC)C CC1(NC(=O)C2=CCNC2=O)CCCCC1C(=O)NCCc1ccns1 N1(CCCCCCOC)CC2C3COCC3C2C1 Cc1cc(Br)sc1C(=O)NC1CCOCC1NC(=O)C(C)Cc1ccco1 C(CC(C(=O)OC)NC(C1CCCN1C(=O)C(C)NC(=O)NC)=O)=CC N1CC(OCC(=O)NC)CC1COC1CCCCC1.C1(=O)CCCN1.Cc1ccon1 C1(O)(CN(C(COC(C)C)=O)C)CCN(C(=O)CSC2CCOC2=O)CC1 c1(C(=O)NC2(CF)CCN(C(C3(C(F)(F)F)CC3)=O)C2)cccc2nsnc12 Cn1c(=O)n(C)c2cc(CNC3CN(C(=O)C(O)C(C)(C)C)CCO3)ccc12 Cc1occc(=O)c1OCCOC1CCN(C(=O)CC(F)(F)F)CC1 CC1CN(C(=O)CCCC(F)F)C(C)CN1C(c1cc(C(F)(F)F)c(Cl)cn1)=O C1(NC(c2cc(CC)nn2C)=O)CCCN(C(=O)C(C(F)F)c2ccccc2)C1C c1(C(=O)NC23C(CN(C(c4cc(C)no4)=O)C2)C3)cc2ccccn2c1 C(C(C)(CC(C)C)NC(c1nn(C(F)F)cc1Cl)=O)NC(c1c(C)ccn1C)=O c1(C(=O)NC2C3CCN(C(=O)C=Cc4ccc(F)cc4)C23)ccc2n[nH]cc2c1 C1(C(=O)NCCN(C(c2c(OC)cccn2)=O)CC2CC2)CCC(C)(C)OC1 c1(C(=O)NC(CC)CN(C)C(c2sccc2Br)=O)c(C)ccnc1O CC(=O)CCCC(C)C(=O)NCC(C)=CC(=O)NCCO.C12(CC1C)C(=O)NC2 N1(C(c2n(CC)ncc2)=O)CCC(NC(=O)C=Cc2cn(C)nn2)C12CCC2 C1(C)(C(N(C(C(=O)N(C)Cc2cccnc2)C2CC2)C)=O)CCC(=O)CC1 C1(NC(CCC#CC)=O)CC2CN(C(c3cscc3C(F)(F)F)=O)CCN2C1=O N1(C(C2CCCC(NCc3ccc(OC)cc3OC)C2)=O)CCCC(C)(O)CC1 c1(OC)ccc(Br)cc1-c1cn(CC(C)(C)NC(C2CC2C(=O)C2CC2)=O)nn1 C1(NC(C(C)NC(C)=O)=O)CN(C(=O)Cc2ncco2)CCC1C C1(NC(c2cc(CC(C)C)[nH]n2)=O)CCC(C)N(C(c2ccsc2Cl)=O)C1 CCC(C)(C#N)C(=O)NCC1(C(N)=O)CN(C(=O)CC2(C)CCOCC2)C1 c1(C(=O)NC(CN(C(C2(C)CCC(=O)C2)=O)CC)C)c(C(F)(F)F)noc1C N1(C(C(CCC)NC(N)=O)=O)CC(NC(=O)C(F)=CC2CC2)C2(CC2)C1 C1(CNC(=O)CN2CCCC2)CC2CC2N1C(=O)CC1CC1(Cl)Cl N1(CC)CCOCC1C(=O)NC(CNC(c1oc(C)nc1C)=O)CO c1(OC)cc(C(N2CCC(N3CCCC3)C2)C(=O)NCC2CC2)cc(Cl)n1 c1(C(=O)NCC(C)NC(=O)Cc2nnc(S)nc2O)cc2ccccc2oc1=O C1(c2nc(-c3cccc(C)n3)nn2CC2CC2)CC(c2cccc(F)c2)=NO1 N1(C(C(c2ccoc2)NC(c2c(C)nc(C)o2)=O)=O)CCN(C)CC(C)C1 Cc1noc(C(N2CCCC(C(C)NC(C3(C)CCCC3)=O)C2)=O)c1C N1(C(c2c(C)cnn2C)C(=O)NC(C(=O)OC)C)CCCC(C)(C(=O)OC)C1 C1(NC(c2ccc(C3CC3)o2)=O)CCN(C(=O)Cc2cnns2)C12CCC2 CCCCC(C)CCC(=O)N1CCOC(C(=O)Nc2scc(C)c2C(N)=O)C1 N1(C(C=Cc2cc(C)no2)=O)CC2(CC(CNC(c3cncc(F)c3)=O)C2)C1 c1(N2CCC(O)(CN(C(=O)Cc3ccoc3)C)CC2)ncc(S(C)(=O)=O)cc1Cl N1(C(C=Cc2ncn(C)c2)=O)CC2CC(NC(c3cccc(C4CC4)n3)=O)C2C1 C(=O)(CCCS(N)(=O)=O)NCC1CC(CNC(Cc2cccc(C)c2C)=O)OC1 N1(C(C(C)NCCc2cscn2)=O)CCC2C(CCN2C(=O)OC(C)(C)C)C1 c1(OC)cnc(Cl)c(CN(C2CCN(Cc3ccc(C(=O)OC)cc3Cl)C2)C)c1 C12(COC)CCC(NC(c3cnc(CNC(=O)CC4CC4)nc3)=O)(CC1)CC2 Cc1cc(C(=O)NC2CCC(CCNC(=O)Cc3nc[nH]n3)C2)sc1Cl c1(-c2n(C(C)CN(C)C)nc(-c3ccccn3)n2)cnc2n1CCC2 Cc1sc2ncnc(NC(C)CCNC(c3cc4ccc(F)cc4s3)=O)c2c1C C(=O)(CC(F)(F)CS(C)(=O)=O)NCC(C1CCN(C(=O)CCS(C)=O)CC1)C N1(C(CCOCC)=O)CCC2C(NC(C3CCCN(C)C3)=O)CC12 Cc1oc(C2CC2)nc1C(=O)NC1COCC1NC(C1CC=CCC1C)=O N1(C(CC(C=C)C)=O)CCC(O)(CCNC(C2CCCS(=O)(=O)C2)=O)CC1 N1(C(C2C(C=C)C2)=O)CCC2(CC1)CC2CNC(c1ccoc1)=O N1(C(C=CC(CC)C)=O)CCC(CNC(=O)C(C)OCCC(C)C)C12CC2 n1(CC)c(C)cc(C(N2CCC(F)(CNC(=O)C3=COCCO3)C2)=O)c1C N=c1[nH]c(C(F)(F)F)ccc1C(N1CC2CC2(NC(=O)CC2CSCCS2)C1)=O CC1C(C)N(C(c2ccc(CO)cc2)=O)CCN1C(c1ccncc1Cl)=O c1(C(N2CC(C(C)NC(C3CC(F)C(=O)N3)=O)C2)=O)ccc(F)c2ccncc12 Cc1ccc2c(CC(=O)NCC(C)(C)NC(C3CCCC(=O)O3)=O)coc2c1 CCC(CC(C)C)C(=O)N1CC(CF)(NC(=O)CN2CC=CC2)C1 C1(C(=O)NC2(COC)CN(C(C3(C(=O)NC)CC3)=O)C2)CCC(C)(C)C1 c1(C(=O)NCCSCc2cn(C(C)C)nn2)ccc2nnn(O)c2c1 C1(C(=O)NCCCSC)CCCCCCN1C(=O)CC1CCCC12CC2 C1(=CC(=O)NC23CCN(C(Cc4n(C)ccn4)=O)CC2C3)CCCCCC1(F)F N1(C(c2nc(C)oc2C)=O)CCC2C(NC(c3ccc(F)c(CO)c3)=O)C2CC1 C1(NC(=O)Nc2ccc(CO)c(OC)c2)CCc2c[nH]nc2C1.C1C(C)N1CC c1(CC(=O)NC2(CN(C(C(CC)C)=O)C)CC2)coc2cc(OC)ccc12 Cc1cc(=NCCC2(N(C)C)CCC2)[nH]cc1S(=O)(=O)NCC1CCCO1 C1(COC)CCN(C(=NCCCCl)NCc2cc(NC(N)=O)ccn2)C1 c1(C(=O)NC(C23CCC(CC2)C3)CNC(C(C)c2ccsc2)=O)ccc(Cl)cn1 C12(CNCc3nc(C)oc3)CCC1CN(CC(C)C)C2.c1(C=O)cc2n(n1)CCC2 CCCCCC(O)C(=O)NCCCC1(NC(=O)Cc2ccc(C)nc2O)CC1 n1(CCC)ccc(C(C(=O)NCC2CCCO2)N(C(C)C(C)n2cncn2)CC)c1 c1(C(=O)NCC2CN(C(C3N(CCCC)CCOC3)=O)C2)cccc(O)c1F CN1CCCC1CCC(=O)NCC(C)(C)NC(c1cc(-c2ccccn2)no1)=O c1(CC(N2CCN(C(c3nc(C)c(C)s3)=O)CC2CO)=O)ccc2c(c1)CCO2 C1(NC(CCCNC(=O)OC)=O)CCOCC1NC(c1cc(C#N)cs1)=O N1(C(CC2C(C)(C)C2)=O)CCCC(C2CN(C(c3c(F)ccnc3F)=O)C2)C1 N1(C(CC(=O)OCC)=O)CC2(CCCC2NC(=O)CC(c2c(C)n[nH]c2C)C)C1 CCC(C)C(C)CNC(=O)C(C)(CO)NC(=O)CN1CCOCC1=O Cn1cc(C=CC(=O)NCC(C)(C)CCNC(=O)C(F)CC2CCCCC2)cn1 c1(C(=O)NC(c2ccccc2)C(N2CC(F)(F)CC2CO)=O)cccc(O)c1Cl CC(=Cn1ccnn1)C(=O)NC1COCC1NC(=O)CCC(C)(C)C#N C1(CNC(C2(CCC=C)CCCC2)=O)CCC(C)CN1C(c1ccns1)=O C1(CCNC(c2c[nH]c(=NC)o2)=O)CCCN(C(C2CC2c2cccs2)=O)C1 c1(C(C)C)nc(NC(C)CC#N)cc(=NC(C)c2ccc(-c3ccncc3)cc2)[nH]1 c1(C(C)NC2(c3nnnn3C(C)(C)C)C(CC)CC2)cc(F)ccc1F Cc1ccc(C)c(SC2(C(=O)NC3CC(=O)N(C4CCCCC4)C3)CC2)c1 C1(NC(CC2(N(C(C3(CC)CCCC3O)=O)C)CC2)=O)CC2(C1)CC(C)C2 C(=O)(C(C)(C)C1CCCC1)NC1C(CNC(CCOC)=O)C1 c1(C(=O)NC(CNC(=O)C#CC2CC2)C2CCC2)ccc2ocnc2n1 Cc1ccnc(CC(C(=O)O)NC(c2ccccc2Cc2cnn(CC)c2)=O)c1 C(c1ccc(=N)[nH]c1)=CC(=O)N(C1CCN(C(C(C)N(C(C)=O)C)=O)CC1)CCO C(C(=O)NC(C)(C)C)(C1=CCCCCC1)N1CCCC(CC=C)C1 N1(C(C(Cn2cncn2)NC(c2cc(C3CC3)on2)=O)=O)CCCCCCCC1 N1(C(c2c(C)cccc2O)=O)CCC2(CO)CN(C(=O)Cc3cnns3)CC2C1 c1(CC)ccc(C(OCP(C)(C)=O)C)nc1.n12cc(nn1)NC(=O)NCC2 N(C1CC(F)(F)c2ccccc21)C(c1cc(C(=O)OC)n(C)n1)=O S(=O)(=O)(c1cc(Cl)c(F)cc1F)N1CCC(C(N2CCC(CO)C(O)CC2)=O)C1 c1(C(=O)NC(C2(O)CN(c3snc(CCOC)n3)C2)C)ccc2cnccc2n1 C(=O)(C(O)CCCc1ccccc1)NCC(C)CNC(=O)Cc1ccc(F)cc1 C(=O)(C1=NN(C(C)C)C(=O)CC1)OCc1snc(CC)n1 N1(C(c2n(CC)nnc2)=O)CC2C3CCC(C2C1)N(c1ncc(C)c(C)n1)C3 C1(NC(c2nccc(C)n2)=O)CC2CC1N(C(=O)CC1C(C)(C)C1(C)C)C2 C1(NC(c2cccc(C#C)c2)=O)CCCC2CN(C(=O)C(C)S(N)(=O)=O)CC12 CCC(CO)(C(=O)NCC(C)CN(C)C(c1ccn(C2CCC2)n1)=O)OC c1(C(C(=O)NC23CC(C2)N(C(C2(CCF)CCC2)=O)C3)O)ccc(F)c(Cl)c1 C(=O)(C1=CS(=O)CCC1)NC1C(NC(C2CCC(C(CC)=O)CC2)=O)CCC1 O=C(C1CCCc2scnc21)N1CCOC(C(=O)NCC23CCC(CC2)OC3)C1 Cc1cc(S(=O)(=O)NCC2CCN2C2CCCC2)sc1Cl C(=O)(C1c2cncnc2CN1C(=O)C(CO)OC)OC C1(CC(N2CC(C(C)NC(c3cc(OC)ncn3)=O)C2)=O)NC(=O)CN(C)C1=O C1(CNC(COCCCCCC)=O)CCC2CN(C(=O)C(O)COC)CC12 N1(C(c2ccn(C(C)C)n2)=O)CC(NC(C2(c3cc[nH]n3)CCC2)=O)CC(O)C1 c1(CNC(C2(NC(C3N(C)C(=O)CC3)=O)CCCCC2)=O)nn(C)c(=O)n1C c1(N(CCOCC)C)nc(=NC)nc(NC(C)COC(F)(F)F)[nH]1 C1(CCNC(C2(F)C(C)C2)=O)CSCCN1C(c1cncc(N(C)C)c1)=O N1(C(c2cccc(CC)n2)=O)CCC2(CCN(C(=O)C=CC3CCCO3)CC2)C1 C1(C(N2CC(CN(C)C(c3cc(C(C)(C)C)oc3C)=O)C2)=O)NC(=O)OC1C C1(NC(C2(c3cc(C)no3)CC2)=O)CN(C(=O)CC2CCCCC2C)CC1(C)C C(=O)(C(C)(C1CC1)NC(c1ccn(CCF)n1)=O)NC1(C(=O)OCC)CC1 N1(C(CSCC)=O)CCN(C(c2cc3cnc(Cl)cc3s2)=O)C2CCCCC2C1 N1(C(CSCCCC)=O)CCC(F)C(NC(=O)C(C2CC2)SC)C1 CCCCC(C)C(=O)N1CCCC(O)(CNC(c2cc(C)n(C)c2)=O)C1 C(=O)(C(C(C)(C)C)N(C)C)NC1(C2N(C(c3cccc(SC)n3)=O)CCC2)CC1 c1(C(=O)NC2C(N(C(COC(CC)CC)=O)C)CCCC2)cnc2[nH]cncc1-2 C#CCCCCC(=O)N1CC2C(NC(c3ncsc3C3CC3)=O)C2C1 c1(C(=O)OCC)[nH]c(C)c(C(=O)OC)c1NC(c1ccc(I)c(C)n1)=O C(c1ccccc1Cl)=CC(=O)NCC(C)NC(c1cnn(C)n1)=O c1(CN2C(C(=O)Nc3cc(O)nc(CO)n3)CC2)ccc([N+](=O)[O-])cc1 C=C=CC(C)C(=O)N(C1CN(C(=O)C(C)Nc2nc(C)cs2)C1)C C(=O)(C(C#N)C(C)(C)C)NCC(C)NC(C1(O)CCSCC1)=O N1(C(c2c(C)coc2)=O)CC2(C)CC1(C(=O)NCCC13CCCC1C3)C2 N1(C(C(C=C)OC)=O)CCC(O)(CNC(=O)C(C)(C)C=C)CC1 C(=O)(C(C)(O)C(F)(F)F)NCCC1CCCN(C(CCC=C(C)C)=O)CC1 c1(C(N2CC(NC(=O)C(F)(F)C3CC3)C(C3CC3)C2)=O)ccc2nnc(O)n2c1 c1(C(=O)NC2C(CNC(C3CCCN(CC)C3)=O)C2)coc(S(=O)(=O)C2CC2)c1 c1(NCC2CCCOC2)ccc(S(=O)(=O)NC2CCN(S(C)(=O)=O)CC2)cn1 c1(C(=O)NC2CCC3(C2)CN(C(c2ccccn2)=O)C3)c(Br)cc(Br)c(O)c1Br CCCCC(O)C(C)C(=O)NCc1ccc(C(=O)NOC(C)(C)C(=O)OC)cn1 C1(O)(CNC(C=C(C)Cl)=O)CCN(C(=O)CSCc2ccccc2)C1 c1(CC)cccc(C(N2CCC(NC(c3cnn(C)c3Cl)=O)CC2C)=O)c1F C1(CNC(c2c(OC)ccc(C)c2)=O)CC2(CCN(C(=O)CC3C=CCC3)CC2)C1 c1(CC(=O)NCC(C)CNC(=O)C(F)(F)CO)ccc2nc(O)[nH]c2c1 c1(C(N(C2CCCN(C(C3CCC3CF)=O)C2)CC)=O)c[nH]c2cc(O)ccc12 Cn1[nH]c(=NC(c2cc(Br)no2)c2nnnn2-c2ccccc2)cc1C(F)(F)F C(=O)(C1Cc2ccccc21)N(CC(C)O)CCNC(c1c(C)sc(Br)n1)=O c1(C(=O)Nc2c(OC)c(Br)cc(C)c2)cscc1C1=C(C)OCCC1(C)C c1(OC)ccc(CC(=O)NC2CC(NC(=O)CSCc3ccccn3)C2)nn1 CC(C)CC(C(=O)NC1CCN(C2CC2)C1)ONC(=O)CCc1ccccc1 c1(CC)c(C(=O)NCC2(C)CCCN2C(=O)CC2C=CS(=O)(=O)C2)cnn1C O=C(C1=CC2(CCN(C(C34CCCCC3C4)=O)C2)C1)N1CC(OCF)C1 n1(C(C)C)ccc(C(=O)NC2C(C(=O)NOCc3nc[nH]n3)C2(C)C)n1 Cc1cccc(C(O)C(=O)NC(CCN(C)C(c2snnc2C)=O)C(C)C)c1 C1(NC)CCNC12CC2.O=C(CC(F)(F)F)Oc1ccc(Nc2ncccn2)cc1 C1(NC(c2ccsc2)=O)CC2CC1CN2C(c1cnc(C2CCOCC2)s1)=O C12(CN3C(CNC(CC(C)(O)C4CC4)=O)CCCC3)C3C4C1C1C2C3C41C C=CC1CN(C(=O)CC2CN(C(c3nc(Cl)cs3)=O)CCC2C)CCO1 c1(C(C)C)ccc(CN(c2ccnc(NC3CCN(CC(F)(F)F)C3)n2)C)cc1 c1(C(N2C(CN(C)C(c3ccc(Cl)s3)=O)COCC2)=O)nncc2c1CCCC2 C12(C(N3CC(CC=C)(NC(c4cncc(C)c4)=O)C3)=O)CCC(=O)N1CCS2 c1(C(N(CC(C)CN(C(=O)CN2CCCC2)C2CCC2)C)=O)ccc(Br)c(N)n1 CC1=C(C)CC(C)(C(N2CCC(CCNC(=O)C(O)C(F)F)CC2)=O)CC1 c1(C(=O)NCC2(NC(C3(C#N)C(C)C3)=O)CCC2)ccc2sc(=N)[nH]c2c1 C1(NC(C(n2c(C)ccn2)C)=O)COCCN(C(c2ccc(CO)cc2F)=O)C1 C(=O)(C(F)C(=O)NCC1(NC(C2CC(C(N)=O)C2(C)C)=O)CC(F)(F)C1)OCC CC1C(NC(=O)CC2CCCS2(=O)=O)CCN1C(C12CC(C1)C(C(F)(F)F)O2)=O CCC(C)C(C(=O)NCCC(O)CCO)NC(C1CCN(C)C1=O)=O c1(C(N2C3C(NC(C4(CC#C)CCOC4)=O)C(C3)C2)=O)cc2c(F)cccc2[nH]1 C1(NC(=O)Cn2nccn2)CC(CO)N(C(c2c[nH]nc2Br)=O)C1 S1(=O)(=O)c2ccc(cc2Br)N1.CCC(C)CC(C)CCN1CCC(F)(CF)CC1 c1(C(=O)NC(C2CCOC2)CNC(c2c(OC)c[nH]n2)=O)cc(Cl)cc(Cl)c1 CN=c1[nH]c(=NCc2cnc(C(C)C)s2)[nH]c(=NCC2(C)CC2(F)F)[nH]1 c1(CC(C)C(=O)NCC2(CNC(=O)Cc3cccnc3O)CC2)ccc(Cl)cc1 c1(C(=O)NC(C(=O)NC2(C=C)CCCC2)CC2CCCC2)c[nH]c2nccc-2c1 CC(C(F)C(=O)N1CC(CNC(=O)C2=NOCC2)OC(C)(C)C1)C(F)(F)F c1(C(N(C)CC2(O)CCCN(C(CC=C)=O)C2)=O)cc2c(ccn2C)s1 c1(-n2ccc(C(=O)NCC(CO)NC(C3C(OC)C3)=O)n2)cccc(C)n1 CC1(C(=O)NC2CC(F)CN(C(c3cc(O)ncn3)=O)C2)CC(C(F)(F)F)=NO1 c1(NC(=O)NC2CCCC2c2nncn2C)nccn1CCSCCC=C c1(CCC)nnsc1C(=O)NCCCN(CCCNC(=O)C(F)(F)C1CC1)C C1(C(N(c2ccc(F)cc2)C)=O)CC2CCC(C1)C2N c1(N2CCN(C(C3(S(N)(=O)=O)CCC3)=O)CC2)cccc2cc[nH]c12 N1(C(C(C)c2ccsn2)=O)CCCCC2(C1)CN(C(C1CC=CCC1)=O)C2 c1(CC(=O)NC2(C)CN(C(C3(C)CCCC3)=O)C2)cc(Cl)c2c(c1)OCCCO2 C(C(CCNC(=O)C(C)(C1CCC1)NC(=O)C(C)CSC)OC)OC C1(NC(C2CCC2)=O)CCCCC12CCN(C(=O)C=Cc1cnc[nH]1)C2 N1(C(C2(NC(C=CCC)=O)CC(F)(F)C2)=O)CCN(CC2(O)CCC2)C(=O)C1 N1(C(COCC)=O)C2CCC1C1CC1(NC(c1nc(C3CC3)cs1)=O)C2 C1(CC(=O)N(C(C)CNC(c2cnn(C)c2N)=O)CC)CCCC(F)(F)C1 C(=O)(C(CC1CCC1)NC(C1CC2CC2C1)=O)NC(C(=O)OC(C)C)C N1(C(C23CC2CN(Cc2cccc(Br)c2)C3)=O)CCN2C(=O)OCC2C1 N1(c2ncnc(OC)c2C)CC2CCN(C(c3ccc(I)o3)=O)C2C1 N1(CC(=O)NCCc2cccs2)CCC2CC(C(N3CCOC4CNCC34)=O)C2C1 c1(C(N2CC3C(NC(Cc4n[nH]c(=NC)s4)=O)C(C3)C2)=O)cc2c([nH]1)CCOC2 Cc1cc2[nH]c(C(=O)NC3CCC(CNC(=O)Cc4csc(Cl)c4)CC3)cc2o1 C12(NC(CCOCC#C)=O)CCC(C1)N(C(=O)Cc1c[nH]nc1C)C2 C1(NC(CC(C(C)C)O)=O)CC(O)(C2CCN(C(=O)CCc3cnoc3)CC2)C1 N1(C(C(N2CCNC2=O)C)=O)CC(C(=O)N(C2COCC2(C)C)C)CC1(C)C C1(C(=O)NC(Cn2cc(C(C)O)nn2)C)CC12CCOc1ccccc12 N1(C(C=Cc2ccc(C(N)=O)o2)=O)CC2COCCC2(NC(=O)CCC(F)(F)F)C1 c1(C(=O)NCC2(CNC(c3ccc(C)o3)=O)CC2)ccc2ccnc(Cl)c2n1 N1(N2CCC(Oc3ccc(OCCC)cc3)C2)CCc2nc(C=O)sc2C1.CC Cc1ccc(F)cc1CCNC(=O)C(=O)Nc1ccccc1CN Cc1cc(C(=O)N(C2CCC(NC(=O)CCCC3CCCCC3)C2)C)ns1 c1(C(=O)OC)ccc2cc1N2.C1(C)CN(C(=O)C2CC2)C2CC12.C1(O)CC1 C=CCC(CC)C(=O)N1CC2CC2(NC(C2C3CCC2(c2ccccn2)C3)=O)C1 c1(C(C)(C)C)ccc(C(=O)NC2CC(NC(N)=O)C2)cn1.c12ccccc1OC2 n1(-c2cccc(OCC)c2)nc(C2CCOc3ccccc32)nc1CC1=CCCC1 c1(C2C(C(=O)Nc3c(C(C)C)ccc(F)c3)C2)cccc2ccccc12 C(N=c1[nH]c2c(C)nn(C)c2c(=O)n1C)c1ccc(OCC)cc1OC N1(C(CSC)=O)CC=C(CNC(=O)C(O)C(F)(F)c2ccccc2)CC1 N1(C(CCc2c(C)noc2C)=O)CC(C)CN(C(C2CC(C)(O)C2)=O)C(C)C1 Cc1sccc1NC(=O)COC(=O)CCCN1CCCCC1 C1(NC(c2cc(CC)c(CC)o2)=O)CCN(C(=O)COCC2CCC2)CC1F c1(CCC)cc(C(N2CC(NC(=O)C(c3cccc(Cl)c3)O)C(C)C2)=O)n(C)n1 c1(C(N2CCCC(N(C(CC(COC)C)=O)CCO)C2)=O)cnc(N(C)C)c(Cl)c1 C1(CNC(CCC2CCN(C(COCC(=C)C)=O)C2)=O)CCOCC1(C)C Cc1c(C(=O)NC23CC(NC(=O)COCC(F)F)(C2)C3)nn(C)c1N C(=O)(C1=CC2CCCC12)NCc1scc(CNC(CCOCC(C)C)=O)n1 C(=O)(CCCC(C)NC(c1c[nH]c(=NC)o1)=O)NC(c1cccnc1)CC Cc1noc2cc(C(=O)NC3(CN(C(=O)Cn4cccnc4=O)C)CC3)ccc12 C(=O)(C(F)(F)CCc1ccccc1)NCC(C(C)C)NC(c1cnn(CC)n1)=O C1(NC(C2CCC(C)(C)C2)=O)CCCCCN(C(c2cnc(S)[nH]2)=O)C1 CC1CCN(c2ncc(C(F)F)cn2)C1CNC(=O)CC1CC2(CC2)C1 C(=O)(CCCCCC(C)C)NC(CNC(c1cc(OCC)cc(=O)o1)=O)C1CC1 c1(C(=O)NCC(CC)NC(=O)C(C)C2CCC2)c(C#N)ncn1C C12(N(CCCN(C)C)C(=O)COC3CCCCCC3)CC3CC(C(=O)N1)C2C3 S(=O)(=O)(c1cc(C(F)(F)F)ccc1F)NC1CCC(NC(C(C)O)=O)C1 CCC(CCCC(=O)N1CC2CC1CN2CC)NC(=O)CC1CCOC1 C1(NC(COC)=O)C2CCC1N(C(=O)C(c1cc(C)ccn1)(F)F)C2 C1(CN2CC(NC(=O)NC(c3c(C)ccc(C)c3)C)C2)COc2ccccc2O1 N1(C(c2nc(C(NC(=O)CN3CCOC3=O)CC)oc2)=O)CCCC(C2CC2)CC1 CCC(C)CCCC(=O)NC1CC(C)(NC(=O)CC2COCCN2C)C1 N1(C(c2ccc(CC)cc2)=O)CCCCC(NC(=O)C(=Cc2cn(C)cn2)F)C1 c1(C(=O)NC23CCN(C(CCC=CCC=C)=O)CC2C3)ccc2nc(C)nn2c1 C1(C(N2CCCC(CN)C2)=O)CC2CCN(C(c3cccc(O)n3)=O)CC12 C1(CN(C(C2(C(C)C)CCC2)=O)C)CCCCN1C(=O)C=C1CCN(C)CC1 Cc1ccnc(C(=O)N(C)Cc2cccc(CNC(c3ccn(C)n3)=O)c2)c1 C(=O)(C1=CC(O)C(NC(=O)Cn2cnnc2)C1)NCC1(C)CCCC(=O)N1 C12(NC(Cn3c(C(C)C)nnn3)=O)COC(C1)C(NC(c1ccc(=O)oc1)=O)C2 c1(CNC(C(c2cccs2)SC)=O)ccccc1CN(C(=O)Cc1cnc[nH]1)CC c1(OCC)ccc(C)cn1.N1(C(COC)=O)CCC(N(C(=O)CCCOC)CC)CC1 C1(NC(CC2(C=C)CCC2)=O)COC2CN(C(=O)CNS(C)(=O)=O)CC12 C1(NC(COCC)=O)C2CC(NC(C3CN(C(CC(=C)C)=O)C3)=O)CC12 c1(C(=O)OC(c2ccon2)C)cc(-c2ccncc2)no1 C1(CNC(c2c(C)n(C3CCC3)nc2)=O)CCN(C(=O)CCC2(C)CC2)C1(C)C c1(C(CNC(CCC#CC)=O)NC(=O)C(O)C2CCCC2)cc(F)cc(Cl)c1 N1(C(COC(CC)C)=O)CCC(C(C)C(=O)NCCN(C)C2CC2)C1 C1(O)(CCNC(CCCC=C)=O)CCCN(C(=O)CSc2cc(C)ccc2C)C1 C(CCCC(=O)NCC(CC(C)C)NC(=O)C(C)CSC(F)(F)F)(OC(C)=O)OC c1(-n2c(C(C(C3CCOCC3)C)NCC(=O)N(C)C)nnn2)ccc2c(c1)CCC2 C1(NC(C2C(C)(Br)C2)=O)CN(C(=O)C=CC=C(Cl)Cl)CC2(CC2)C1 c1(C(C)=O)c[nH]c(C(=O)NCC(F)CNC(c2cnc(CC(C)C)[nH]2)=O)c1 c1(C(N2CC(NC(c3ccc(C)c([N+](=O)[O-])n3)=O)C2)=O)cc(Br)cc([N+](=O)[O-])c1 Cc1nc(CO)oc1C(N1CC(CO)C(C)C1)=O.C(C)(C(C)(C)C#N)N1C(=O)C=CC1 N1(C(Cc2n[nH]c(=NC)s2)=O)CCCC(NC(c2nc(C)oc2C)=O)C1C C1(NC(C2CN(CC)C2)=O)(CNC(=O)C2=C(C)CCC2)CCCCC1C C1(C(=O)NCC2(CNC(C(CCSC)O)=O)CC2)CSc2ccccc2O1 C(=O)(C1=CCCOC1)NCC1(C)N(C(C2C=C(C)CS2)=O)CCC1 N1(C(c2ccc(OC)c(O)c2)=O)CCC(NC(C2CC(F)C2)=O)CCC2(CC2)C1 O=C(CN=C(NCc1ncccc1F)NC1CC1)NC(=O)CCC(F)(F)F n1(CCCNC(=O)CCc2nccs2)cc(C2CCCCO2)nn1 Cn1cc2c(n1)CC(C(=O)NCCC1CC(NC(=O)CCc3cn[nH]c3)C1)CC2 C12C3CCCC1CN(C3)C2=O.N1(C(C)=O)CCC(C(=O)NC2CNC(=O)C2)CC1 CCC(CC(=O)N1CCCCC1)SC.C1(=O)C(OC)N1C.C(C)(=O)OC c1(C(=O)NCCC2CN(C(C3(Br)CC3)=O)C2)cc2ccccc2s1 c1(C(=O)Nc2cc(O)nc(SC3CC(C(=O)OC)C3)n2)cccc2nccn12 c1(OC)cccnc1C(N1CCCC1CCC(C)C)=O.c1(C2C(=O)N2)ccccc1 C1(CNC(COC(CC)C)=O)CN(C)CCN1C(=O)Cn1cc(C(=O)OC)cn1 CCCCCCCCOC(=O)C=CC(N1CCC(C)C1CNC(C1CC=CC1)=O)=O CCC(C(C)(C)O)NC(c1cccc(CNC(c2cccc(O)n2)=O)n1)=O C1(CNC(C(C)OCCCC)=O)CN(C(c2ccc(C(C)(C)C)o2)=O)CC1C C(=O)(C(C)CC(C)(C)O)NCC=C(C)C(C)C CC(C)CCCCCC(=O)NCC1CCN(C(c2cnc(C(F)(F)F)cn2)=O)C1 c1(OC)ccn2ccnc2c1C(N1CC2CC1C2NC(C1CC1C1CCCO1)=O)=O C12CCN(C1)NC(=O)CC2.C1(C2(CC(=O)OC)CC2)CCNC1=O C1(N(C(C=CCNC(C=C(C)C(F)F)=O)=O)C2CC2)COCCC1O N1(C(CC(C(=O)OC)(C)C)=O)CCCC1C1CCCN1C(c1cn(C)nc1Cl)=O Cn1ccc(=O)c(C(=O)NCCC2(C)CCN(C(=O)CCC3CC(F)(F)C3)C2)c1 c1(C(N2CC(N(C(=O)Cc3cn(C)nn3)C)C(O)C2)=O)n[nH]c2c1COC2 CCC(CNC(=O)CCN(C(C1OC2CCC1C2)=O)C1CC1)C(C)(F)F N1(C(C)NC(c2ccccc2)=O)CCCC2(CCN(N(C)Cc3nccs3)C2)C1 c1(CC(=O)NC2C(C)CN(C(=O)C(N)=O)CC2)ccc2c(c1)CCO2 C1(CC)(NC(C2CCCN(C)C2)=O)CCCN(C(=O)C(C)S(N)(=O)=O)C1 Cc1nccc(CSCCC2CC2(Cl)Cl)c1Cl CC(CCCCNC(=O)COc1ccccc1)NC(c1nscc1Br)=O Cc1cc(-c2cn(CCC3CC(NC(c4sccc4N(C)C)=O)C3)nn2)cc(Cl)c1 Cc1cc(C(=O)NC2CCCCC2NC(C2CC2F)=O)c(Cl)cc1Cl C1(CNC(CN(c2ncccn2)C)=O)CN(C(=O)CC2NC(=O)NC2=O)CC1(F)F CCCCCCCCCC(=O)N1CC2CC(NC(=O)CC(C)(C)C(F)F)CC2C1 Cc1cc(=O)n(C)cc1C(N1CC(CNC(c2cnsc2C)=O)CC1C)=O C1(CNC(CCCOCCOCC)=O)CN(C(=O)C(F)(F)C2CC2)CC1(C)C N1(C(C2C(C(C)(C)O)C2)=O)CCCC2(C1)CN(C(=O)CC1(O)CCC1)C2 c1(CC)c(C(=O)NCC(C(C)C)NC(c2[nH]ccc2C)=O)cnc2ncnn12 c1(C(=O)NCCCNC(c2cc(C(=O)OC)oc2C)=O)cc2[nH]ccc2s1 C1(C(N2CCC(NC(CC=CCCCCC)=O)C2)=O)CC(=O)NC1(C)C CCC(Cc1ccc(N)cc1)C(=O)NCC1(NC(=O)C(C2CC2)OC)CCCC1 CC1CN(C(c2cc(O)cc(Cl)c2)=O)CCCN1C(c1coc(C(N)=O)c1)=O c1(C(=O)NCC(CNC(CN(C2CCCC2)C)=O)F)ccc(Cl)cc1C(F)(F)F c1(C(N2CC(CNC(c3ccn(CC)n3)=O)OCC2)=O)ccc([N+](=O)[O-])c(O)c1 C1(CCC)CN(C(=O)C(O)CC(C)C)CCN1C(c1nnc(S)n1C)=O c1(CNCC2(O)CCC(C)C2)c(O)nc2ccccc2c1Cl c1(C(=O)NCC2(F)CCCN(C(C(CC)F)=O)C2)ccnc2c1nnn2C c1(NCCN(OC)C)cc(S(=O)(=O)NC(c2ccccc2Cl)CO)ccc1C#N CC(C)CC(C(=O)NCC(=O)NC1CC=CCC1)NC(=O)CN1CC=CC1 c1(N(C)C)nnc(-c2ccccc2)n1C1CCC1.C12CCN(C1)C(=O)N2 c1(C(=O)Nc2ccc(CO)s2)cccc(Cl)c1O.c12ccc(nc1)c(=O)[nH]2 c1(OCC(C)C)ccc(NC(C2CCCN(C(=O)C=CCBr)C2)=O)c(F)c1 N1(C(C(C)c2cccs2)=O)CC(NC(c2cccnc2OC(F)F)=O)CC1CO Cc1cnccc1C(C)C(=O)NCC(CO)NC(c1ncoc1C(C)C)=O CC(C)CCC(O)C(=O)N1CCC(C)(CC(=O)NC2CCN(C(N)=O)C2)C1 CCC(O)C(C)C(=O)N1CC2CC(CNC(=O)CSCc3ccncc3)C2C1 C(=O)(C(F)(F)CCCNC(=O)OC(C)(C)C)N(Cc1cn(C)nc1)C(=O)O c1(NCC(CCN(CCCC)CCC)OC(F)(F)F)ccc(Br)cc1 C1(C(N2CC(O)(CC(C)C)C2)=O)CCC(O)CN1C(=O)C#CC1CC1 C=CCN(OC)C(=O)C1CCCC1NC(=O)CC1C=CCCC1 C(=O)(CC1C(=O)Nc2c(F)cccc21)NCCN(C(C(CCC)C#N)=O)C N1(C(c2ccc(N)c(Cl)n2)=O)CC2CCCCN2CC1CNC(=O)C=C(Cl)Cl n1(CCC)ncc(C(=O)NC(C2CCCCN2C(C2CCCCC2)=O)C)c1C O=C(C(F)C(F)(F)F)N1CC(C2CN(C(=O)C=CCn3cncn3)CCO2)C1 N1(C(c2c(NCC)cccn2)=O)CC(NC(C2CN(C)C2)=O)CC(C)C1 C1(N(C(=O)C=CSc2nc[nH]n2)C)CN(C(=O)CC2(C)CCCO2)CC1(C)C CC1C=C(C(=O)NCCC2(CC(=O)NCCCCCC)CCC2)CC1 N#Cc1cc(C(=O)NCC2CCC(CNC(=O)Cc3cc[nH]n3)CC2)c[nH]1 C(CCC(=O)N(O)Cc1cn(Cc2conc2C2CCC2)nn1)OC C1(NC(CCc2ccn(C)c2)=O)CN(C(=O)CC2CCCO2)CC1O CC(C)C(C(=O)N1CC(CNC(C2CC2F)=O)C1)NC(c1ccccc1)=O C1(C(N2CCC(C)(CNC(=O)C(c3ccccn3)O)C2)=O)CC1C1CCCCC1 C1(C(N2C(CC)(CC)CC2)=O)CCCN(C(=O)COC2CCC2)C1C n1(CC)c(CNC(=O)CC(C)CNC(=O)CCC2CCC2)cnc1C c1(C(N2CCC(O)(CCSC)C2)=O)sc(OC(OC(F)(F)F)=O)cc1C C1(CN(C(c2cccc(C(N)=O)n2)=O)CC)CCCN(C(=O)CNS(N)(=O)=O)C1 CCC(C)C(C(=O)N(CCC(=O)NC(c1nn(C)cc1O)C)CCO)OC C1(C(=O)NCC(C(=O)NCC2(CCC)CC2)N(C)C)CCCC(C)(C)C1 c1(CCn2c(C(=O)NC(COC(C3C(C(N)=O)C3)=O)=O)ccn2)ccc(Br)cc1 C1(C(N(C(C)C(=O)N(C)Cc2ncc[nH]2)CCC)=O)CCOC1C(C)C c1(C(N(CC(CC)NC(c2ccc(CF)cc2)=O)CC)=O)nccc(OC)c1C C1(C(=O)Nc2c(OC)cccc2)CCCN1NC(=O)CC(C)(C)O C(CCC1CCC1)(C(=O)NCC1CCC1C(=O)O)NC(C1(OC)CCC1)=O N1(CC)CC(C)C(c2nnnn2CCCC2CC2)(Nc2cc(OCC)cc(C)c2)C1 c1(C(N2CCC(N(C(=O)CCCC#N)C)C2)=O)cccnc1C(F)F Cc1ccn2cc(C(=O)NC3CCC(NC(=O)C(C)C4CCCC4)CC3)nc2c1 N1(C(CCC)=O)CCC(OCCNC(=O)CNc2cncn2-c2ccccc2)C1 C1(C(N(c2ccc(O)cc2)C)=O)C2CCN(C(=O)CC3OCCO3)CC12 Cc1ccc(CC(N2CCC2CNC(c2cc(C(F)(F)F)no2)=O)=O)c(C)c1 C(=O)(C(O)CC(C)(C)C)N1CCC(C(C(N2CCC(C)CC2)=O)C)CC1 CC#CCCCC(=O)NC1CC1NC(=O)CCOC1CCOCC1 Cc1nn2ncccc2c1C(=O)NCCCc1ccc2[nH]ccc2c1 c1(CC(=O)NCC2CC(NC(C(N3CC(C)C3)C)=O)CC2O)cccc(F)c1F CC1CC(CNC(=O)COCC2CCOCC2)CN1C(c1sccc1Cl)=O C(CS(=O)(=O)C1CCCC1)c1nc(CCC(C)S(C)=O)nn1-c1nccs1.CC C(CCCC(C)NC(C1(CCF)CCOCC1)=O)NC(C1C(C)C1(F)F)=O C1(C(=O)NCc2n(C)ccc2)CCCC12CN(C(=O)CC1OCCOC1(C)C)C2 C12(NC(C=Cc3cn(C)nn3)=O)CCCC1N(C(c1coc(C(F)F)n1)=O)CC2 c1(C(C(=O)NC(C)C)N(C)Cc2cc(Br)cnc2F)nn(C)c2c1COCC2 N1(C(C(CC)C#N)=O)CCC(C2CC2)(CNC(=O)Cc2cccc(COC)c2)C1 C=CC(CCC)CC(=O)NCC1(CNC(C2(CF)CC2)=O)CCCCC1 C1(NC(c2cc(C)cc(F)c2)=O)CN(C(C2CC(N=[N+]=[N-])C2)=O)CCC12CCC2 c1(C(N2CCC3(N(C(CC(CC)CC)=O)CCC3)C2)=O)nccc2ncncc12 C=CCC(CC=C)C(=O)NCC1CCCC(NC(c2ccc(F)c(Cl)c2)=O)C1 N1(C(CSCCCC)=O)CC2(CCC2)CC1C(N1CC2CC2(C(=O)OC)C1)=O N1(C(C(n2ncc(C)c2)C)=O)CCN(C(=O)CCC(=O)N(C)C)CC(CO)C1 C1(C(=O)NCC(C2(O)CCN(C(c3cccs3)=O)C2)C)(CC)CNC(=O)C1 c1(SC)c(C(=O)NC2CC(NC(c3ccnnc3C)=O)C23CCC3)cccc1F C1(NC(c2c(C)cc(C)o2)=O)CCCN(C(=O)CCSC2CCCC2)CC1F CS(=O)(=O)c1ccc(O)c(NC(=O)C(=O)NCc2ccccc2F)c1 Cc1cc(N)nc(C(=O)NCC2(N3CCOCC3)CCCC2)n1 CC1(CNC(=O)COCCF)CN(C(c2ccc(-c3ccccc3)o2)=O)CCO1 N1(C(C(C(C)O)(C)C)=O)CC2COCC2(C(=O)N(C)Cc2nc[nH]n2)C1 c1(C(=O)O)cccc(S(=O)(=O)N2CC3CCC2CN3S(=O)(=O)CC2CCC2)c1 C1(C(=O)NCC2CCN(C(CS(C)(=O)=O)=O)CC2)CCC2(CCOCC2)O1 c1(OC)nc(C(N2CC(CNC(=O)CN3CCCS3(=O)=O)C(O)C2)=O)cc(O)n1 C1(C(N2CCC(NC(CP(C)(C)=O)=O)C2)=O)CC(c2cccc(F)c2)=NO1 c1(C(=O)NCC(C)N(C)C(C2COCCN2C2COC2)=O)cncc(N(C)C)c1 N1(c2n(CC)c(CCC(C)(C)c3ccccc3)nn2)CCn2cnnc2C1C CN1CCCC(C)(C(=O)NCc2c(C(=O)O)n[nH]c2Br)C1 C=C=C(C)CC(=O)NC1CC1CNC(=O)CC1CC(n2cnnc2)C1 C1(NC(=O)Nc2cccc(OC)c2Br)(C)CCCC2(CCCCC2)C1.C(C)(=O)N C#CCC(C)(C(=O)NCCC1CC1)NC(C1CC12CCC2)=O C=C(Br)CN=C(NCc1ccc(OCC(F)F)cc1)NC1CCC1 C1(CN(C)C(c2cncc(C(F)(F)F)n2)=O)C2CN(C(=O)C=CS(C)=O)CC12 C(=O)(C1=C(Cl)CCCC1)NCC1ON=C(C(=O)N(C)Cc2c(C)nsc2)C1 N1(C(c2n(COC)ncc2)=O)CCCC(NC(c2cc[nH]c2C)=O)C1 C(=O)(CC1=C(C)NS(=O)(=O)N=C1C)N1CC(NC(C(CCCC)OC)=O)(CO)C1 c1(NCC2CCN(C(=O)CC(c3ccc(F)cc3)O)C2)nc2ccc(Cl)cc2s1 C(=O)(CC(C)C(F)(F)F)NC1C(c2ccc(N(CC)CC)cc2)N(C)CCC1 C(=O)(C1CCCn2cnnc21)C(=O)Cc1ccc(Cl)s1.C1(C=O)(CN)CCCC1 Cc1cc(OCC(=O)N(CC(C)NC(c2cnc(N(C)C)o2)=O)C)cc(C)c1 C(=O)(C(C)(C)CCOC)NCC(CCCC)NC(c1cc(C(C)C)n(C)c1C)=O CCN=c1[nH]c(C)c(C(N2CC(NC(=O)Cc3ccn(C(F)F)n3)C(C)C2)=O)s1 C(=O)(C=CS(F)(F)(F)(F)F)N1CC(CNC(c2cccc(NC)n2)=O)C(C)C1 N1(C(c2cn(CC)nc2C)=O)CCN(C(=O)Cc2nc([N+](=O)[O-])n[nH]2)CC(O)C1 C1(CC)C(NC(=O)CCc2nncs2)CCCN1C(=O)Cc1ncoc1C c1(NCCS(=O)(=O)NC)[nH]c(=NC(C)CN(C)C(C)C)nc2sccc12 Cc1nc([N+](=O)[O-])cn1CCC(=O)NC(CNC(=O)C(C)(F)C(C)(C)F)CO C(=O)(CCN1C(=O)CCc2ccccc21)Nc1c(C)nn(C)c1 c1(OC)nc(Cl)c(C(=O)NC2CC(C)(CNC(c3ccn(CCF)n3)=O)C2)s1 c1(SC)cc(C(=O)NC(CCNC(c2ccoc2C)=O)C(C)C)ccc1N CC(C)C(F)(CNC(c1c[nH]c(C#N)c1)=O)C(=O)NCC1CCCNC1=O C1(CNC(C2CC2C(=O)OCC)=O)CCC(CCNC(C(C=CC)O)=O)CC1 c1(CN(C)CC2CCCN2C(=O)C(C)(C)NS(C)(=O)=O)ccc2c(n1)CCC2=O Cc1ccc2c(c1)C(NC(=O)Nc1ccc(Nc3ccc(Br)c(Cl)c3)cn1)CC2 N1(C(C(C)OCCC=C)=O)CC2CCN(C(=O)CC3CCC3)C2C1 C1(CNC(CCCOCCOCC)=O)CN(C(C2(C#N)CC2)=O)CC1C N1(CC(=O)NCC#CC#CCO)CCN(C(C2CCC(=O)O2)=O)CC1 c1(CC(=O)NCC(CC)(CC)NC(=O)CSC)ccc(S(=O)C2CC2)cc1 Cc1c(C(=O)NCCC2(CNC(=O)C(C)(C)COC(C)C)CC2)cccc1F.OC N1(C(c2cc(C)c(C)nc2)=O)CCN(C(C2CCC(C)(F)CC2)=O)C2COCC12 N1(C(C2(C)CCCN(C(C=NOC)=O)C2)=O)CCC2(CCC(N(C)CC)CC2)C1 Cc1nc(C(C)(C)C)c(C(=O)NCCC(C)CCNC(=O)Cc2cccs2)s1 c1(-c2cn(C(C)C(=O)N3CC(NC(=O)C(F)(F)F)C3)nn2)c(Cl)cc(Cl)cc1Cl C1(CC(N)=O)COCCN1C(=O)C(=O)c1ccco1.n12cc(nn1)C2 c1(CN(c2ncc(SC)cn2)C2CNCC2C#N)cc(Br)cc(Cl)c1O C1(NC(=O)CC2CCC23CCC3)CC2CCC(C1)N2C(c1[nH]ccc1C1CC1)=O C1(NC(C(C=C)O)=O)CC1C1CCN(C(C2CCC(C)(F)CC2)=O)CC1 O=C(C1=CC2CC=CCC12)NC1CC(CO)N(C(=O)CC2CCOCC2)C1 CCC(CC(=O)NCCCC(C)NC(c1c[nH]ccc1=O)=O)C(C)(C)C N1(C(CC(CCC)C)=O)CC(C)CN(C(c2cnc3c[nH]nc3c2)=O)C(C)C1 C(=O)(CCC(=O)NCC1CC1CC(N1CC(O)CC1CO)=O)NCCC N1(C(c2c(C)c(O)cc(N)c2)=O)CCC2(CCC2CNC(C2C(C)C2C)=O)CC1 CC1=C(C)CC(C(=O)NCC2CCC2C(=O)NCc2ccc(C)cc2C)CC1 c1(C(C(C)NC(=O)NCC2CCN(C(C)(C)C)C2=O)O)c(F)cccc1Cl c1(N(C(c2cn(CCF)nn2)C(=O)NCC(F)F)C)ccc2c(c1)CCC(C)(C)O2 c1(CN2CC(Nc3n(Cc4c(C)ncs4)nc(C)c3)C(F)C2)cnc(Cl)c(F)c1 c1(C(N2CC(CNC(C3C(CCC)CCC3)=O)(OC)C2)=O)c(C)cc(F)cc1C c1(C(N2CC(C3CCN(C(C4C(C)C4)=O)C3)OCC2)=O)cccn2nccc12 Cc1ccc(O)c(C(N2CCC(NC(c3ccn(C)c3)=O)C(CO)C2)=O)n1 C1(CCN2C(NC(C(C)(C)NC(C)=O)=O)CCC2)CC2(CCC2)C1 C(CO)(CCCNC(=O)C(C)n1ccnc1)NC(COCC(=O)NC)=O CC1(CNC(C2CC2F)=O)CC(F)(F)CN1C(c1ccc(-c2ccccn2)o1)=O C(=O)(N1CCC(C(N)=O)O1)C1(N(C(Cc2c(C)ocn2)=O)CC(C)C)CCC1 c1(CN(C)C(C2CCCC(=O)CC2)=O)cc(Cl)c(Br)cc1F C1(C(=O)NCC2(O)CC(NC(=O)CC3C=CCCC3)C2)CCC2(CCCC2)CC1 N1(C(C2C(CC)CCC2)=O)CC2C(CC(=O)NCC(C)(C)OCCO)C2C1 C1(C(N2CC(NC(c3cncc(C)c3)=O)CC2(C)C)=O)CC2(COCCO2)C1 c1(C(=O)NCC(N(C(C=CCCC)=O)C)C2CC2)cc(N2CCCC2)ncn1 C(CC(=O)NC(C(O)CO)C1CC1)(CC(C)C)NC(c1c(C)cc(O)cn1)=O C12(C(NOCC(CC)C)=O)CCC(NC(c3ccon3)=O)(CC1)C2 N1(C(C(=C)Cc2ccccc2)=O)CCC(C)C(NC(C2(CO)CCCCO2)=O)C1 N1(CC(=O)N(c2cnn(C3CCOCC3)c2)C(CC)(C)C)CCc2cc(C)cc(C)c2C1 C1(NC(c2n(C)cc(Br)c2)=O)CC2CC1N(C(C1(C)CC3CC3C1)=O)C2 c1(C(N2CCCC(CCNC(c3ccnc(C)n3)=O)C2)=O)ccc(=N)[nH]c1Cl C(=O)(C1=CCC2CCC1N2C(C1(SC)CCC1)=O)NC(C(CCC)C)C C1(F)(C(=O)NC2CC(CNC(C3CCCOC3)=O)C2)CC=CCC1 c1(CNC(C(CNC(C2CC2Cl)=O)N(C)C)=O)ccncc1Cl C12(CNC(c3cn(Cc4ccccc4)nn3)=O)CCC1CCN2C(C1CCC1)=O N1(C(C(=O)N(C(CCC)C)CCOC)=O)CC(C)(C)OC2(CCOC2)C1 C1(C2CC2)(CNC(c2nc(C(C)C)oc2)=O)CCN(C(=O)CC(C)(O)C2CC2)C1 C1(C(N(CCCN(C)C(c2nccnc2)=O)C)=O)CCCC(C(N)=O)C1 c1(-c2n(CC=C)nc(CCN3CC(C)OC(C)C3C)n2)ccc2ncccc2n1 c1(C(=O)OC)ccc(C(=O)NCCN(C(C2CC(C)(F)C2)=O)C(C)C)c(F)c1 N1(C(C=Cc2c(C)n[nH]c2)=O)CCC2C(CCCN2C(=O)CN2CCN(C)CC2)C1 C1(C(=O)NCCC(CC)(CC)NC(CSCCCC)=O)CCCCN(C)C1=O C1(NC(C(C)(C)C2(C)CC2(F)F)=O)CCCN(C(=O)COC(F)F)CC1 c1(CC(N2CC(CNC(C3(C)CCO3)=O)C2)=O)ccc(F)c(Br)c1 C1(C(=O)NCCCCNC(c2c(C)oc(CO)c2)=O)CCc2ccc(F)cc2O1 C(C(C)(O)C(=O)N1CCC(CNC(C2CCC(C(C)(C)C)CC2)=O)CC1)OC C1(C(=O)NCC2CC(CNC(COCCOCCOC)=O)C2)CCS(=O)(=O)N1C C12(C(N3C(COC)CC(O)C3)=O)CCC(CC1)N(C(=O)CC(C)C)C2 N1(C(c2cncc(NC)c2)=O)CCC(C)C(CNC(=O)C(C)(C)c2ccns2)C1 N1(C(c2c(OC)c(Br)cc(Cl)c2)=O)CCC2C1CCCN2C(c1ccncc1)=O C1(CCNC(C(C)NC(=O)NC)=O)CCCN(C(=O)Cc2cc(Cl)n(C)n2)C1 N1(C(c2c(C)ccs2)=O)CC(F)(F)CC1CNC(=O)CCc1ccc(Br)cc1 C(N=c1[nH]c(=NCC2(CF)CC23CCOCC3)c2[nH]ccc2[nH]1)c1nc(=N)s[nH]1 N1(C(CC(C)(C)C)=O)CC2CCC1CN2C(c1cnc(N)c(Br)c1)=O c1(OC)cccc(Br)c1NC(=O)CC(c1ccc(OC)c(Cl)c1)NC(C1CC1)=O CC(C)C(C(=O)N1CCCC(C)C1)NC(=O)CSCC(N)=O C(=O)(C1=CC2(CCOC2)C1)N1CC2(CN(C(C3(C)CC3(F)F)=O)C2)C1 c1(C(CC)N2C(C)C(=O)N3CC(O)(C3)C2)ccc(C)cn1.c1(C2CC2)ccccc1 C#CCC(CC(=O)N1CCC(OC(C)C)CC1)NC(=O)CCc1cccs1 CCCCC(C)C(=O)N(CC(C)(C)CNC(=O)C(O)CCSC1(C(=O)OC)CC1)C c1(OC)ccc(C(C)(C)C(=O)NC2CCCC2NC(C2CC2(C)C)=O)cc1 c1(C(=O)NC2CCN(C(C(C)CC(N)=O)=O)CC2C(C)C)scc2c1OCCO2 CN1CCC(NC(=O)Nc2cc(F)cnc2Cl)CC1=O C(=O)(C1=CC(C)(C)C1)NCC(C)NC(C1(OC)CCOC1)=O CN1CCCC1C=CC(=O)NCC1CCCN1C(=O)Cc1ccc(C2CC2)cc1 C1(C(=O)NCCC(=O)NCCCC)CC(C(=O)OC)C12CCNCC2 N1(CC2(C(=O)N)CCCC2)CC2CCN2C1.C12(CC1)C(=O)N2C.CO c1(C(N2CCCC(NC(C(C)C#N)=O)CC2)=O)cc(Br)cc2cccnc12 n1(CC(=O)OC)ncc(S(=O)(=O)NC(=O)Cc2csc3ccc(C)cc23)c1OC C(=O)(C(C)C(F)(F)C(F)F)NCCC1(OC)CN(C(=O)CSC(F)(F)F)C1 C1(CC(N2CCCC(N(C(=O)C=C3CCC3)C)C2)=O)CCC2(CCOCC2)CO1 c1(C(=O)NC(C2CCN(C(C(C)OCC)=O)C2)C)cnc2ccoc2c1 c1(C(N(C)CC2OCCN(C(C(CC)(C)C)=O)C2)=O)c(Br)nc2n1CCCC2 C=CCC(CC)C(=O)N(C)CC1CC(F)CN1C(C1CCN(CC2CC2)CC1)=O Cc1ccc(C)n1CC(=O)NCC1CCC(NC(=O)C=C2CC2)C1 C1(NC(CC2CC(CC)C2)=O)CC2CCC1(CNC(=O)CCC(C1CC1)OC)C2 S(=O)(=O)(c1ccc(=NCC2CC=CC2)[nH]c1)N(C(CCC)C)C CN1CCC2CCN(C(C3CCN(C(=O)COCC4CCC4)C3)=O)C2C1 C(c1cccnc1C)=CC(=O)NCC(c1cccc(C)c1)NC(CC(=C)C)=O C#Cc1ccc(C(=O)NC2CCCC2C(=O)Nc2cnn(CC)c2)nc1 N1(C(Cc2cc(C)on2)=O)CC(NC(c2sccc2Cl)=O)C2(CCCC2)C1 N1(C(c2ccn(C)c2)=O)CCC(NC(C2CCO2)=O)C(CO)CC1 C(c1ccc(Cl)nc1)=CC(N1C(C)CC(CNC(c2cc(O)ncn2)=O)C1)=O N1(C(C(C)C2CCCO2)=O)CC(C2CN(C(c3ccc(CC(N)=O)cc3)=O)C2)C1 c1(C(C(=O)NCCC)N(c2ccccc2C#N)C)ccc(F)c(Cl)c1 C1(OC)CN(C(c2c(C)cccc2O)=O)C(C)(CNC(c2sccc2F)=O)C1 c1(C(C)CC(=O)NCCC2CCN(C(C3(F)CCC3)=O)C2)ccc(F)cc1F C(=O)(C#CC1(C)CCCO1)NCC1(OC)CCN(C(C2CCCCCC2)=O)C1 C1(F)(C(=O)NCCN(CC(C)C)CC)CCN(C(C2CC(C)CO2)=O)CC1 c1(C(C)C)cc(C(N2CC(O)(C(F)C(=O)NCc3nn[nH]n3)C2)=O)on1 NC(=O)CC(C(=O)NCCSC(F)F)NC(c1cc(CO)[nH]n1)=O C=Cn1nncc1C(=O)NCC(CC)NC(C1(C)C=CCCC1)=O C1(O)(C(C)NC(c2c(C)cnnc2)=O)CCN(C(C2CC2C)=O)CC1 C1(CNC(C2(CC#C)CCOC2)=O)CN(C(C2CCS(=O)(=O)N2)=O)CCC1(F)F O=C(CC(C(F)F)C1CC1)NCC1(O)CN(C(=O)COC(F)F)C1 C=CC(C)(O)CC(=O)N1CCCC1C1(NC(c2ncc(Br)cc2F)=O)CC1 C(=O)(CCCC(=O)NC1CCC1C(=O)N(C1CCOC1=O)C)OC C(=O)(C(F)(F)C1=CCOCC1)N1C(CNC(c2n(C)nc(OC)c2Cl)=O)C=CC1 C1(C(=O)NC(C2CCCN2C(c2ccncc2O)=O)C)CC12CCSCC2 c1(OCCC(=O)NCC2C(NC(C3(Cl)C(C)(C)C3)=O)CC2)ccccc1Br N1(CC(=O)NCc2c(NC(C)=O)cccc2)CCCN(C2CCOC2=O)CC1 c1(OC)noc(C(=O)NCC2(C)CCN(C(=O)CC(C)C3CCCO3)C2)c1Br C(=O)(C(C)C(O)CCCC)NC1C(CNC(C2(CCC=C)CC2)=O)CCCC1 C(=O)(C1=NNC(=O)C1)N(C)CCC1CCN(C(c2cnccn2)=O)CC1 N1(C(C(=O)N(C2CCCCN2)CCOC)=O)CCc2cccc(Br)c2C1C N1(C(C(CSC)NC(=O)C=Cc2cccnc2)=O)CC(=O)N2CCCC2C1 CC1(C)COCC(C(N2CCOC(CNC(=O)Cc3csnn3)C2)=O)O1 C1(C(N(CC(F)F)CCC)=O)CCCCN1C(C1CCCC(CF)C1)=O CC(CCCCNC(=O)CC1(C)CC1(F)Cl)NC(=O)CC1(N(C)C)CCC1 c1(CC(=O)NC2CCN(CCNC(C(C)OC)=O)C2)cc(C)c(Br)c(C)c1 N1(C(C2CC(C)(CC)C2)=O)CCCC(CNC(=O)C(C)CSc2ccccc2)C1 C(C)(C)(CC(=O)NC12COC(CO)(C1)C2)NC(C1(CC)CCOC1)=O c1(C(=O)NC(C)CCNC(=O)CCC2NC(=O)NC2=O)cccc2nc(S)oc12 c1(CN(C(C(N2C(CC)CCC2)=O)=O)CC)ncccc1O.C1(=O)CN1.C(C)(=O)N C1(NC(c2c(CC)ocn2)=O)CC2CC(C1)N(C(=O)Cc1cc(C)no1)C2 N1(C(C2C(C)C2)=O)CCC(C)(C)C(N(C(C23CC(CO2)C3)=O)Cc2ccccc2)C1 Cc1cc(C(=O)N(C(C)CNC(C2CC2F)=O)C)c2[nH]cnc2c1 c1(OC)ccc(C(N2CCC(C)(NC(C3CC(C(C)C)=NO3)=O)CC2)=O)c(Cl)c1 c1(CC)ncnc2[nH]cc(C(=O)NCCCN(C(=O)CO)C)c12 N1(C(c2cc(C)cc(C)n2)=O)CCC(C)N(C(C2CCCN2N=O)=O)CC1 C(CCCC(=O)N1CCC(CC=CC)C1)N(C(CC=CCC)=O)C c1(CC(N2CCC(OCc3ccc(Cl)nc3)CC2)=O)cccc2c1CCC2 N1(C(Cc2c(C)nn(C)c2)=O)CCC(NCc2ccc(C(C)(C)C)cc2)C(C)C1 C1(CC(=O)NC23CC(NC(c4cccc(C(=O)C5CC5)c4)=O)(C2)C3)CC2(CC2)CO1 C1(F)(C(=O)NCCCN(CC)CC)CCCN(C(C2CCCOCC2)=O)C1 c1(NC(C(c2ccoc2)SCC#N)=O)cccc(OCC(F)(F)F)c1 c1(N2CCC3(C(C(N4CCCC(Br)C4)=O)C3)C2)ncc2cn[nH]c2n1 C1(CC=C)(NC(C2CC(=O)N2)=O)CCCN(C(=O)C(CCC)N(C)C)C1 c1(C(=O)OC)cc(Br)c(Cn2cc(C3CCCOC3)nn2)s1.N12CC(C1)C2C N1(C(CC(COC)C)=O)CCCCCCC1C(=O)NCCC1(C)CCOC1 CC(C(=O)NCC1(CN(C)C(c2cnc(O)c(F)c2)=O)CC1)S(N)(=O)=O N1(C(CN(S(CC)(=O)=O)C)=O)CC(O)C(O)C1CNC(c1cccnc1O)=O C#CC1CN(C(C2CCCN(C(=O)CS(=O)CC)C2C)=O)CCN1C C1(NC(=O)NCC(N(OC)C)=O)COCCC1(F)F N1(C(COCCC#C)=O)CC(COC)CC1CNC(C1CC(=O)N(CC=C)C1)=O Cc1ccccc1C1(C(=O)NCC2(O)CCN(C(=O)C3=NOCC3)C2)CC1 N1(CCOC)CC(C(=O)NC(C)CC(C)NC(C2CCOC(C)C2)=O)CC1=O C1(C(N(C(C(=O)NCCc2ncc(C)o2)C)C2CC2)=O)COCC1(C)C CC(C)C(C#N)C(=O)N(CCCN(C)C(C12CCCN(CC1)C2)=O)C c1(COC)cccc(C(N2CCSCC2CCNC(c2ccnnc2C)=O)=O)c1 C1(NC(C#CC2(C)CC2)=O)CCCC12CCN(C(=O)C=CCF)C2 CC(O)(CC(=O)NCCCN(C(c1coc(C(F)(F)F)n1)=O)C1CC1)C1CC1 c1(C(=O)NC2CCCN(C(c3c(OC)csc3)=O)C2C)cn(C)c(=O)nc1O CCC(C)CCC(=O)NC1(COC)CN(C(C2CNC(=O)OC2)=O)C1 N1(C(C2CN(C(N)=O)C2)=O)CCC(CC(N2CCC(O)C2)=O)CC1 C12(CC1(C)C)OC(c1ccccc1)CN2.C(C)(C)(C)COCC N1(C(COC(CC)CC)=O)CC(C)N(C(c2ccnn2C(F)F)=O)CC1C N1(C(c2[nH]cc(SCC)c2)=O)CC2(CCC(NC(=O)C(CC)OC)CC2)C1 C1(C)(C(=O)NCC2N(C(Cc3n(C(C)C)cnn3)=O)CC(F)C2)CCN(C)C1=O C(CC(=O)NCC1CCOC1)(C(F)F)NC(C(C)N(C)C)=O C1(NC(C(C)C2CCCO2)=O)CCCCN(C(c2snnc2C2CC2)=O)C1 N1(C(c2nc(CC)on2)C)CCCC2C(NC(=O)Cc3csnn3)C(C)(C)C12 Cn1ncc2c(NC3CCc4ccccc43)nc(N3CCCC(C(F)F)C3)nc12 N1(C(C(C)=CC)=O)CCCC1C1(NC(=O)C(F)n2ccnc2)CC1 C1(CCC)CCCC1C(N1CC(F)(C(=O)NCC(O)COCCOC)C1)=O C(=O)(C(C)(O)CCSc1ccccc1)N(C(C)C(O)C(F)(F)F)CC c1(C(Cn2c(=O)c2=O)=O)ccc(SC(F)F)cc1.C1(CC(C)N)CCCC1 c1(N(c2c(C(C)(C)C)occ2)C(C2CC3CNC2C3)=O)ccc(F)c(F)c1 c1(NCC(c2ccc(F)cc2)(C)F)ncnc(-c2cccs2)n1 C1(C(=O)NCC=CCNC(C=CC=C)=O)CCCCC1CN(C)C C(=O)(CCCCCCCS(C)(=O)=O)N1CC(C(C)NC(C(CC)F)=O)C1 C#Cc1ccc(C(=O)NC(CCC)CC(=O)NCC2=NOC(C)C2)nc1 c1(C(N2C(C(C)NC(=O)C(=Cc3c[nH]cn3)F)CCC2)=O)cnc2cc[nH]c2c1 C=C=C(C)CC(=O)N(CCCN1CCC(NC(=O)C=CI)C1)CC N1(C(Cc2c(C)ccnc2)=O)CCN(C(c2cc[nH]c(=N)c2)=O)C(C)CC1C c1(C(C(=O)NCC(CC(C)C)NC(=O)C(C(C)C)N(C)C)C)nc(F)ccc1Cl N1(c2nc(Cl)nc(C)c2F)CCC(C2(NC(=O)C(F)CC3CC3)CC2)CC1 C(CN=c1[nH]c(=NCCc2ccc(C)nc2)[nH]c2c1CC(C)CC2)N1CC=C(C)C1 O=C(C1=CCCCO1)NC(CNC(c1cc(C(F)(F)F)cnc1O)=O)C1CCC1 c1(CN=C(NC(C=C)C)NCc2cnco2)nc2c(s1)CCCCC2 C(c1cncnc1O)=CC(=O)NCCN(CCC)C(c1ccsn1)=O N1(C(C23CC(CC)(OC2)C3)=O)CC2(CCN(C(c3cccc(CO)c3F)=O)C2)C1 C=CC1COCCN1C(C12CC(CO1)N(C(=O)C=Cc1ccccc1C)C2)=O C1(NC(C(c2c(C)cccc2)(F)F)=O)CCN(C(c2cnn[nH]2)=O)CC(C)(C)C1 CC(CCc1ccccc1)CC(=O)NCC1(C)CCCN(C(=O)C2=CCC2)C1 c1(C(=O)NC(CCCNC(COCCCOC)=O)C)c(F)ccc2c1OCC2 c1(C(N2C(C(=O)NCC(O)Cc3ccccc3)C(O)CC2)=O)ccc(Cl)c(I)c1 N1(C(CCC(C)SC)=O)CCN(C(c2ncoc2-c2ccccc2)=O)C(CO)C1 C1(NC(C2C3COCC23)=O)CCC2(CCN(C(c3cnc(Cl)[nH]3)=O)CC2)C1 Cc1ccncc1C(C)NC(=O)C(c1ccco1)NC(=O)Cc1ccc[nH]1 Cc1sc(-c2nc[nH]n2)nc1C(=O)NCC1CC(NC(=O)C=CS(C)=O)C1 c1(C(N(C)CC2CCN(C(=O)CCc3ccc[nH]3)C2)=O)nc(O)nc(O)c1F CCC(CC)C(C)NC(=O)C(CC1CCCC1)NC(C1CS(=O)(=O)C1)=O N1(C(CN(C(=O)OCC)C)=O)CC(NC(=O)Cc2nocc2SCC)C(C)(C)C1 N1(C(C2CCN(OC)CC2)=O)C2CCC1CC(CC)C2 C(C(=O)N1CCC(C(C)(C)CNC(=O)C(O)C(C)C)CC1)(C(C)C)N(CC)CC N1(C(C2(OC)CCSC2)=O)CCN(C(c2cn(C)c(=O)n2C)=O)C(CC2CC2)C1 C1(F)(C(=O)NC(C)CNC(c2cnc(-c3ccccc3)[nH]2)=O)C(C)(C)C1(C)C C12(CNC(CCCN(C)C)=O)CCC(C1)N(C(=O)C1=CCOC1)C2 Cc1snnc1C(=O)N(C)CCOCCN(C)C(c1coc(C(F)(F)F)n1)=O C(=O)(C(C(C)C)N(C(=O)CCN(C)CC)C)N(C(C)C=O)CCCC.S(C)(=O)(=O)N C1(C)(OC)CC(NC(=O)Nc2cn(CC3CCCC(=O)C3)nn2)C1(C)C C1(C(F)(F)F)(C(=O)NCCNC(CN(C)C(C2CC2F)=O)=O)CCCCC1 O=C(C1=NNC(C(F)(F)F)C1)NCC1(CNC(c2cc(O)cc(O)n2)=O)CCC1 N1(C(CCCSCC)=O)CCOCC(NC(=O)CN2CCC(C(C)O)CC2)C1 c1(NC(C2(C)CN(C(c3ccc(C#N)c(O)c3)=O)C2)=O)cccn2nccc12 c1(OC)ccc(CC(=O)N(CCCNC(C2(F)CCCC2)=O)C)c(F)c1 c1(OCC#C)ccc(C(=O)NCC(C)(C)NC(=O)CSCC(N)=O)cc1 FC1CC(N=c2[nH]c3c(c(=NCCn4ncc(Br)n4)[nH]2)CCCCC3)C1 c1(SCCOC(C(C2CCCN(C(=O)OC(C)(C)C)C2)C)=O)cccc(O)c1 C(=O)(CCCC(C)(C)C)NC(C(C)C)CNC(=O)C(n1cnc(C#N)n1)C N1(C(C(F)=CCC)=O)CCC2(CC2NC(=O)Cn2nnc(C3CC3)n2)C1 C1(CNC(CCSCC)=O)CN(C(C2CC3OC2C2CC32)=O)C2CCCC2O1 c1(CC)n[nH]cc1C(=O)NC(C(=O)NC1C(C)C1C)c1ccoc1 CC(O)(CC(=O)NCC(F)CNC(=O)CCc1ccc(Cl)cc1Cl)C(F)(F)F C(CC(C)C)(C(=O)N1CCN(C(c2cnc(Cl)[nH]2)=O)CC1C)NC(C)=O Cc1ccc(C(=O)NC2(CO)CCCN(C(c3cccnn3)=O)C2)c(C)c1 N1(C(CCC=C)=O)CCOC2(CCCN(C(C3(S(N)(=O)=O)CCCC3)=O)C2)C1 N1(C(C(C)NC(=O)OCC)=O)CCCC(C)(CNC(c2ncsc2NC)=O)C1 c1(C(=O)NC2CCC(F)(CNC(CCOCC(C)C)=O)C2)scc2c1CCCC2 C(CCC(C)C(=O)N1CCCC(CO)(CNC(=O)COC2CC(F)(F)C2)C1)OC CCC(CC)CCC(=O)NC(C1CCCN1C(=O)C(C)c1cc[nH]n1)(C)C C#CCCCC(=O)N1CC(C=C)(CN(C)CCC)C1 c1(OC)ccnc2c(NS(=O)(=O)CC3CC(C)CN3)cccc12 C12(C(=O)OCC)CC1CN(Cc1cn(-c3ccccc3Br)nn1)C2 C=C(C)C(C)(C)C(=O)N1CC(CC(C)NC(c2cc(C)c(N)cn2)=O)C1 c1(OC(C(=O)N(CCCN(C)C(C2(O)CCSCC2)=O)C)F)ccc(Cl)c(F)c1 c1(C(=O)NC(C2CCN(C(c3nccnc3O)=O)C2)C)cc(Cl)c2n[nH]cc2c1 N1(C(C(=O)NC(C(=O)OC)CCC2CCC2)C)C(=O)c2cccc([N+](=O)[O-])c2C1=O N1(C(CCC)=O)CC(CNC(c2cccc(CCO)c2)=O)OCC1C(F)(F)F CC1C(C)N(C(=O)CC2CC=CC2)CCN1C(c1[nH]nc2ncccc12)=O N1(C(C(C(C)O)NC(C)=O)=O)CCC2CN(C(=O)CC(F)(F)F)CC2C1 C1(C(=O)NC(c2cccc(C(F)(F)F)c2)CC)CCc2n[nH]c(C)c2C1 c1(C(=O)NC(CNC(=O)C=CC=C(Cl)Cl)C2CCC2)coc2c1CS(=O)(=O)C2 Cc1csnc1C(=O)N(C1CCCC1)CCNC(=O)C(n1ccnc1C)C c1(C(=O)NC2CCC(C(=O)O)O2)cc(F)ccc1-n1cccn1 Cc1cc(=NCCOc2ccc(C#N)cc2)[nH]cc1S(=O)(=O)N(C)CC(F)(F)F C1(CC(N2C(C(CNC(CCSCCCC)=O)(C)C)CCC2)=O)C(C)(C)C1(F)F c1(C(N2C(C(C)NC(C3C=CCC3)=O)CCCC2)=O)cc(O)nc(O)n1 Cc1cc(C(N2CCOCC2C2CCCC2=O)=O)c2ncccc2c1Br c1(C(=O)NC2CC3(CC(NC(C4C(CC)CCC4)=O)C3)C2)cc2cn[nH]c2cn1 C(CCCC(=O)NC(C)Cc1cc(C)[nH]n1)NC(c1c(CC)noc1)=O c1(C(C)=O)ccc(CC(=O)NC2(C)CC(NC(=O)CN3CCC(C)CC3)C2)cc1 c1(CN(C)C(C2CC(F)CN2Cc2cncs2)=O)ccc(O)cc1 C1(C(=O)Nc2cncc(CO)c2)CC(F)(F)CN1C(c1occc1Br)=O C1(C(N(C2CCN(C(c3sccc3C(C)C)=O)C2)CC)=O)CCC(C)C1 c1(C(=O)O)ccc(C2CCN(C(C3COCCN3CC(F)F)=O)C2)cc1 c1(CNC(C2C(CC)N(C(c3cc(COC)no3)=O)CC2)=O)ccc(F)c(C)n1 C(=O)(C#CC1(C)COC1)NC(CN(C(C1NC(=O)CC(C)C1)=O)C)C N1(C(C2CCC(=O)O2)=O)CCOC(CCNC(c2cn(CC(F)(F)F)nn2)=O)C1 C1(O)(CNC(c2n(CC=C)ccn2)=O)CCN(C(c2cc(C)ncc2C)=O)CC1 N1(C(CCCNC(c2ccc(OC)cc2)=O)=O)CC2CCCC(CO)(C2)C1 S(=O)(=O)(c1ccc(NCC(O)C(C)C)cc1Br)NCc1c(C)nco1 c1(CCC(=O)NCCN(C(c2cn(CCC)nc2)=O)CCOC)ccccc1C CC1c2ccccc2CCN1C(c1ccc(F)c(Cl)c1)C(=O)NC1CCCC1 N1(C(c2cc(C)[nH]n2)=O)CCN(C)CC1CNC(C1(Oc2cnn(C)c2)CC1)=O C1(NC(c2c(SC)cccn2)=O)CC2(C1)CC(NC(C1CN(C(C)C)C1)=O)C2 c1(SC)cc(C)c(C(=O)NC2CC(NC(C3CC3(F)Cl)=O)C2)s1 C1(N(C2CN(C(c3cnc(CC)s3)=O)C2)C)CCN(C(=O)COC(C)C)CC1 c12ccc(o1)C(=O)N1CC(C1)C(O)C(=O)NC2.C1(CC)CC(CC)C1 c1(CC)sc(C(=O)NC2CCN(C(=O)CC(C)c3ccncc3)C2C)cc1CC Cc1ncnc(N2CCC2CN2CCOCC2)c1Br.C12CCC(CC1)C(=O)NC2 c1(C(=O)NCC2CN(C(c3c(C#C)c[nH]n3)=O)C3C2C3)cc2cccnc2[nH]1 C1(C(=O)NCCCC(C)NC(c2c(CC)n(CC)nn2)=O)CCC2(CC1)CC2 N1(CCNC(C(C)OCC)=O)CCN(C(C2(F)CC2c2cccc(C)c2)=O)CC1 c1(C(=O)OC)nn2c(=O)cc(CNC3CCCCCN3C=O)nc2s1 c1(CC(N2CCC(NC(C(CC)C)=O)C(C)C2)=O)ccc(C)c(F)c1F c1(NCc2cn(CCCN(CC)Cc3nc(C)no3)nn2)cccc(C(N)=O)c1 C1(CNC(C(CC)F)=O)CN(C(c2cc(C#N)n(C)n2)=O)CCN1C c1(C(=O)NCC(CCC)NC(C2(C)CCOC2)=O)cc2cnccc2[nH]1 C1(NC(C=Cc2ncc(C)[nH]2)=O)CC2CC1N(C(=O)C(=O)NCC(F)F)C2 c1(CC(=O)NC2C(C(=O)NC(C(C)C)CCO)CCC2)cc(F)cc(F)c1 c1(C(=O)NCCOCCN(C(C2CC(OC)C2)=O)C)csc2c1CCC(C)C2 CCC(CC)(CC)NC(=O)NC1CCN(CC2CCC2)CC1 N1(C(c2cc(C)on2)=O)CC(C(=O)NCC(O)Cn2cccn2)C(C(C)C)C1 CC1Oc2ccccc2OC1C(=O)NCC1CCCN1c1ccn2nccc2n1 N1(C2CN(C(=O)C(F)CC3CN(c4nccc(C)n4)C3)C2)CC(C)CC1=O.CO c1(C(=O)NC2(CNC(c3c(CC)nccn3)=O)CCOC2)c(OC)ccnc1F N1(C(C(N2CCN(C)CC2)C)=O)CC2CCC(C1)C2NC(C1CCC(O)CC1)=O C=CC(C)CC(=O)N1CCC(N(C)C(C2(N(C)C(=O)OC(C)(C)C)CC2)=O)CC1 N1(C(CN2CCCC(NC(C)=O)C2)=O)CC(NC(=O)CN(C)C)C2(CCC2)C1 c1(CCC)c(C(=O)NC2CCC(NC(c3csc(C)n3)=O)C2)cnn1CCO N1(C(c2cc(C)n(CC)c2C)=O)CCCN(C(c2cc(C#N)c[nH]2)=O)CC1C C(=O)(C1=NNC(=O)C1)NCC(CN(C(=O)C(C)(C)c1ccccn1)C)O C(=O)(CCCCC(N)=O)NC(C(C)NC(c1n(CC=C)ccn1)=O)CO C1(O)(CNC(c2c(C)nc(CC)s2)=O)CCN(C(=O)C(F)=CCCF)CC1 C1(C(=O)NCC(CNC(c2c[nH]nc2C2CCC2)=O)O)CC12CCC(F)(F)CC2 c1(CC(=O)NC(CC(=O)N(C(CC)CO)C)CC)csc2nc(C)cn12 N1(C(C2C(C)(C)CC2)=O)CC2CCCC(NC(=O)C3=NNC(=O)CC3)(C2)C1 N1(C(C2(C)CC2)=O)C(CNC(c2ccn(C3CC3)n2)=O)CC2COCC12 c1(C(=O)NC(CNC(c2ccn(C)n2)=O)CC(F)(F)F)ccc2nnnn2c1 c1(CNC(N2CCC2c2cccc(F)c2)=O)cc2cc(Cl)ccc2o1 c1(C(=O)NC(C)CCCCNC(c2ncccc2O)=O)ccc2c(c1)OCC2 c1(OCC)cc(C(N2CC(NC(=O)CC(=O)OC)CC(O)C2)=O)cc(F)c1 C(=O)(C(C(C)(C)C)NC(=O)C(CNC(C1(CSC)CC1)=O)C(C)C)NC C(C)(C)(CCCNC(c1nn(CC)cc1Br)=O)NC(COCC=C)=O c1(C(=O)NC2(CNC(c3ccc(CO)nc3)=O)CCC2)ccc2occc2n1 CCCC(C(O)C(=O)NC1CC2CC1C(O)C2O)NC(=O)C=CC1CCOCC1 CC1OCCN(C(=O)C2=CCN(C)C2)C1C(=O)Nc1cncnc1 N1(Cc2cc(C)ns2)CC2(C)CN(C(c3coc(Cl)n3)=O)CC2(C)C1 C1(CC(=O)NCC2CCCCN(C(c3cnco3)=O)C2)CCn2cncc2C1 C1(NC(C(CCC)Cl)=O)CCC2(CCCN(C(c3ccc(OC(C)=O)nn3)=O)C2)C1 O=C(CC=CCOC1CC(OC(F)(F)F)C1)NCC(O)CN1CCC1 Cc1cn2cc(CC(N3CCC(C)(NC(c4c(Cl)sc(C)c4C)=O)C3)=O)nc2s1 Cc1ccc(C(N)CC(=O)NC(c2c(C)noc2C)C)cc1C C1(CNC(CC2N(CC)CCC2)=O)CN(C(c2ccc(C#N)cn2)=O)CCN1C C(=O)(CCCCC(C)C)N1CC(NC(CCC(CC)C)=O)(COC)C1 CCCC(CC)C(C(=O)NCCCOC)N1CCC(C(=O)OC)C(C)(C)C1 C(CC)(C(=O)N(C)CC1CCCN1C(=O)C(=O)NCCC(N)=O)OCC C1(CCNC(=O)Cn2cc(C3CC3)cn2)(Nc2nnc(O)s2)CCOCC1 C1(NC(c2ccc(COC)s2)=O)CN(C(c2cc(C(C)(C)C)no2)=O)CC1OC N1(C(C(C)SC)=O)CCC(C(C)CNC(c2n[nH]cc2C(F)(F)F)=O)CC1 C1(C(N2CC(N(C(=O)Cn3cnc(C#N)n3)C)C2)=O)CN(S(N)(=O)=O)C1 CC1C(NC(c2ccc(CC(N)=O)cc2)=O)CCCN1C(=O)CC(C)(C)F Cc1cc(C(=O)NNC(=O)NC2(C)CCCCC2O)ccc1N C1(C(=O)N(C(C)(C)C)CC)CNC(=O)CN1c1cc(C)nc(C)n1 C(=O)(C(C)(C)C1=CCSCC1)NC1C(NC(c2c(C)csc2)=O)COC1 C=CC(C(=O)NCC1(C(C)(C)O)CN(C(=O)CC(C)OC)C1)OC C(=O)(C1CC(=O)c2ccccc21)NC(C(C)C)CCN(C)C(c1ncccn1)=O C#CC1CCCN(C(C23CC(CN2C(c2cnn(C(F)F)c2)=O)C3)=O)CC1 C12(C(N3C(c4ccc(COC)o4)CCC3)=O)CCC(CC1)CO2 C#Cc1ccc(C(=O)NC2CCCC2NC(=O)Cc2ccc(OC)cn2)nc1 c1(OC)ccc(C(=O)NC2CC3CC(NC(c4c(C)csc4Cl)=O)C2C3)c(F)c1 N#Cc1c[nH]cnc1=NC1CCCC2CN(C(c3ncsc3Br)=O)CC12 C(CCC1CCC1)(C(=O)NCCC(C)(C)C)NC(c1cc(CC)[nH]n1)=O c1(C(=O)OC)ccnc(N(C)CC2CN(C(=O)C(Cn3cccn3)OC)C2)c1 CCC(C(=O)N1CCC(C(=O)NCCC2CC2)O1)N(C)C C1(C(=O)OCC)CCN(C(=O)CCN(C(=O)Cn2cnnn2)C)C1CC C1(CNC(C(C2CC2)OC)=O)CCC2(CN(C(c3cnn(C(C)C)c3C)=O)C2)O1 C1(CNC(C(CC)C)=O)CN(C(=O)Cc2cnccc2C)CCCO1 [N-]=[N+]=NC1CCCCC1NC(C1CCN(C(c2cc[nH]n2)=O)C12CCC2)=O C1(NC(C2CCNCC2)(C)C)CCCC(c2ccccc2)CC1 C(=O)(C1=CNS(=O)(=O)N=C1C)N1CCC(NC(CC=CC=C)=O)C1 C1(NC(c2c(C)scc2)=O)CC2(C1)CC2C(N1CC(CO)C(CO)C1)=O c1(CN2CC3CN(C(c4c(C)cc(F)cc4)=O)CC32)ccc(F)c(C#N)c1 CCCCC(F)C(=O)NC1CC(CC(N2CCC(SCC)C2)=O)C1 CCC(C#C)N(C(C(=O)NC(C)(C)CC)c1ccsc1)C CCCCCCC(C)C(=O)NC(CCF)C(=O)NCc1ncsn1 CCC(CNC(C1CC12CCCC2)=O)(CC)NC(=O)C(=CC1CCCCC1)F c1(C(=O)NCC2CC(=O)N(CCCNC(C3(C(=O)NC)CC3)=O)C2)cc2n(n1)CCO2 C1(OC)CCC(C(N2CCN(CCNC(=O)CCCn3ccnn3)CC2)=O)CC1 C(C)(C(CO)NC(=O)CCOCC1CCCO1)NC(CCNC(=O)NC)=O c1(C(=O)NC2(C)CN(C(C3CCC(CC)O3)=O)C2)cccc2c(C)ccnc12 CP(C)(=O)C(c1cccs1)NC(=O)COC(=O)NC1CC1 CCC(CC)(CO)C(=O)NC1CC(C)(NC(=O)C(C)OCCN(C)C)C1 Cc1cn2ccnc(-c3nc(C4CC4)nn3-c3ccc(Br)nc3Br)c2n1 c1(C(N2C(CNC(C(CC)(C)OC)=O)CC2)=O)ccc(F)c(C)c1Cl CCCCCCCC(=O)N1CC(CCNC(=O)C=C2CCN(C)C2)C(C)C1 C1(NC(CCCOCC=C)=O)CCN(C(c2ccc(Cl)c(C#N)c2)=O)CC1(C)C CC1(C)CCCOC1c1nc(C(=O)NC2CC(=O)N(c3ccccc3Cl)C2)cs1 O=C(CC1CS(=O)(=O)c2ccccc21)N1CCC(C(C2CCCCC2)=O)CC1 C1(C(=O)NCC(C(CC)(C)C)=O)CCC2(CC1)NC(=O)NC2=O c1(C(=O)NC(CNC(c2c(C)nc(CO)o2)=O)C)cc(N(C)C)ccc1F C(C)(CCC(=O)N1CCC1C1CCOCC1)NC(Cc1c(C)occ1)=O CC(C)C(C)(O)C(=O)NCC1(C(=O)NCC2CCCCCC2)CC=CC1 c1(C(C(=O)NCCC2CC2)NCc2n(C(C)C)cnn2)ccc(OC(F)F)cc1 Cc1ccc2[nH]c(C(=O)NC3CCN(C(=O)C=CBr)CC34CCC4)cc2c1C Cc1c[nH]cc1C=CC(=O)NC1CCCCC1NC(=O)Cn1cc(C#N)cn1 C(F)(F)(C(F)C(F)(F)F)OC(C1CC1CNc1ccccc1NC(N)=O)=O c1(OC)ccnc(C(=O)NC2CC(N(C)C(c3nc(C)ns3)=O)C2)c1 C(=O)(CCCCC(=O)NOCCOC(C)=O)N(C(C(CC)CC)C)C(C)(C)C c1(NC(=O)NC2CN(C(C3CC3F)=O)C2)ccccc1N1CCOCC1 CC(CC(C)NC(C1CN(C(=O)CCc2ncccn2)CCN1C)=O)C(F)F C1(C2CCN(C(=O)C(F)(F)C(O)C3CC3)CC2)(NC(Cn2c(C)nnn2)=O)CC1 n1(C(C)C)cc(C2OCCC2C(=O)NCCC2CN(C(=O)CSC3CC3)C2)cn1 Cc1cc(CC(=O)NCC(C)CNC(=O)C=CCCc2ccccc2)ccc1O c1(N(C)C)ccc(Br)c(C(=O)NC2CC(N(C(=O)Cc3cncn3C)C)C2)c1 CC1(C)CCCCC1C(=O)NCC1CC(NC(C2CC(F)C(=O)N2)=O)C1 C12(CNC(C3C(C)(C)CC3)=O)CC(CO1)N(C(=O)C(F)(F)C1CC1)C2 c1(C(=O)NCC2CCCCN2C(=O)COCc2cccs2)cc2ccnn2cn1 C1(COC)C(C(=O)Nc2nc(C(=O)OC(C)(C)C)co2)CCN1C S(=O)(=O)(c1c[nH]c(C(N2CC(NC(C3(O)CCOC3)=O)CC2(C)C)=O)c1)N(C)C C=CC1(C(=O)NC2CCCC2C)CCN(C(=O)CNC=O)CC1 c1(C(N2CCn3nnc(CO)c3C2)C(=O)NCCSC)nn(C)c2c1CCCC2 c1(C(C(=O)N(CCC(=O)N(CC)CC)CCO)O)cncn1C C1(CN(C(=O)CNc2ccccc2)C)CC(F)CN1C(c1ccn(CCN)c1)=O Cc1cc(C(=O)NCC2CCN(CCCNC(C34CC3C4)=O)C2)oc1C C1(C(=O)NCC(CC2CC2)OC)(CC)CCN(C(c2ncncc2Cl)=O)CC1 C#CCCCCCCCC(=O)NCC(C)NC(c1c(C)cc(C)nc1C)=O C1(NC(C(C)SCCCC)=O)COC2C(NC(=O)CCC(F)F)COC12 N1(C(C(CCC)OC)=O)CCN(C(=O)Cc2nncn2CC)CC1CCC C1(NC(C=NOC)=O)CC2CN(C(C3CCC(CC(C)C)CC3)=O)CCN2C1=O c1(CNC(C2(C)N(C(C)=O)CC=C2)=O)nnc2n1CCS2 Cc1ccc(N)cc1C(=O)NCC(C1CC1)NC(c1cc(F)cs1)=O CC(CS(C)=O)C(=O)NCCCN(CCCCNC(=O)CC1(O)CCCCC1)C CCCCC(CC)CCC(CNC1(C)CCC(C)(C)CC1)CC Cc1cc(C(=O)N(CCC(=O)Nc2ccc(F)cc2)C(C)C)nc(C)c1 C12(CNC(c3c[nH]ccc3=O)=O)CC1CN(C(=O)C=CBr)C2 N1(C)CCC(CC(=O)NC)C1.C(C(COC)NC1CC1C=O)OC Cc1nc(C(=O)OC2CC3(C2)CC3C(=O)OC(C)(C)C)nn1C C1(CC(=O)OC)CC(=O)NC1=O.C(C(CCO)C1(CC)ONC(=O)C2CCC21)OC N1(C(C(=O)NCCOCC(F)(F)F)=O)CCCCCC1n1ccnn1 c1(-c2ccc(C)o2)nc(C2C=CC=CC=C2)n(-c2ccn(C)n2)n1 c1(C(N2CCC(CCNC(COC)=O)CC2)=O)cc2nc(C)[nH]c2cc1F N1(C(C(CC)CCOC)=O)CCN2CCN(C(=O)Cc3csc(C)c3)CC2C1 C1(NC(C(C)NC(N)=O)=O)CCCN(C(c2ccnc(F)c2Cl)=O)C1C C(=O)(CCCN1CCCC1)NCC1(C(C)NC(c2cc(Cl)cs2)=O)CC1 N1(C(C(C)SCC)=O)CCOC2(CCC(NC(c3cnns3)=O)CC2)C1 c1(N2C(CNC(C3CCCNS3(=O)=O)=O)CC(F)C2)ncnc2cc(Br)sc12 S(=O)(=O)(c1ccc(C(=O)N(C)CC2CCCN2C(c2cnc(SC)s2)=O)o1)NC N1(C(Cc2nc(C)[nH]n2)=O)CC2(CCN(C(C3CCN(C)S3(=O)=O)=O)C2)C1 C(=O)(C1=C(c2cc(OC)ccc2F)N(C)C(=O)N(C)C1c1ccc(F)cc1)OCC N#Cc1ccccc1CN1CC(NC(C(F)(F)F)C2CCCOC2)CC1=O C1(C(=O)NC(CC)CN(C(c2ccco2)=O)CC)CCCCN1CC(F)F c1(C(=O)NC2C(CNC(c3c(CC)occ3)=O)COC2)cn(C2CC2)nc1C c1(CC(=O)NC2CC3CN(C(c4nccs4)=O)CC3C2)ccn2cncc2c1 N1(C(C=C(CCC)CCC)=O)CC(O)CC1(C)C(N1CCCOC(C)C1)=O C(=O)(C(F)C(F)(F)F)N(C1CCN(C(=O)CC2CCCCC2N)CC1)CC#C N1(CC)CCCC1CN(C(=O)C(C)(C)NC(=O)COCC1CCOC1)C C1(N2CC(C=CN(CC=C)C(C)=O)C2)Cc2ccccc2C1O Cc1c(C(=O)Nc2[nH]cnc2C(N)=O)cccc1I.C12CCN(CC1)C2=O CCCC(C(=O)NC(Cc1cc[nH]n1)C(=O)Nc1c[nH]nc1C)OCC N1(C(c2cn(CCC)nc2)=O)CCCCC(CNC(C2CC23CCSCC3)=O)C1 C(=O)(CCCS(C)(=O)=O)N(CCC#N)CC.c12ccc(cc1)NC(=O)N2CC c1(CNC(C2CCCC(CC(F)(F)F)C2)=O)nc2c(s1)CCN(C(=O)CO)C2 N1(C(C(Cc2ccoc2)NC(C(CC)COC)=O)=O)CC2CC2C2CC12 n1(CC)cnc2nc(=NCC3CSCCS3)[nH]c(NCc3c(F)cccc3Cl)c12 C12(OC(F)(F)F)CC(C1)CC1(CC1)Cn1cc(nn1)CNC2=O.C1(O)CCC1.CO c1(CC)oc(C)cc1C(N1CC(NC(C2(C)COC(=O)C2)=O)C(CC2CC2)C1)=O N(C1CSCc2ccc(Br)cc21)C(Cc1sc(CC)c(C)c1)=O c1(C(=O)NC2CC(NC(C3CCC(=C)CC3)=O)C2)cc2ccc(F)cc2o1 c1(C(=O)NCCC2CN(C(CCCSC)=O)CC2C)n[nH]c2ccc(F)cc12 c1(OCC)ccc(C(F)(F)C(=O)NCC2CC(NC(=O)Cc3nc[nH]n3)C2)cc1 c1(CC)cccc(C(N2CCC(CNC(C3CCS(=O)(=O)N3)=O)C2)=O)c1N N1(C(c2c(NCC)scn2)=O)CC(C)N(C(c2csc(COC)n2)=O)CC1C N1(C(C2C(C(=O)NCC(C)(C)C)C2)=O)CC(C#N)C2(CCC2)C1 CC1(C)CC(CNC(C2(n3cncn3)CC2)=O)CN(C(=O)CC2COC(=O)N2)C1 N1(C(c2c(Cl)cnc(CC)n2)=O)C2CCC1CN(C(=O)CC1COCC1(C)C)C2 C1(C(N2CCC(N(C(C(C)OCCC#C)=O)CCOC)C2)=O)CN2CCN1CC2 c1(C(=O)NC(CC)CNC(=O)CC2CCC(C(F)(F)F)O2)c(C)cccc1C c1(CN(C(CN(C(=O)Cc2cncs2)CC#C)=O)C)cn[nH]c1 c1(CCC(N2CCC(N(C(C(C=C)O)=O)CCC)C2)=O)cc(F)cc(F)c1 C1(NC(c2cc(C(F)F)ncn2)=O)CCN(C(=O)C(F)(F)C2(O)CCCC2)CC1F c1(C(C(N2CCC(CNC(CC(C)F)=O)C2)=O)(C)C)ccc(C(C)(C)C)cc1 c1(C(=O)NCCCN(C2C3CC4C(C3)C24)C2CC2)cc2cccn2cn1 Cc1cc(N2CCN(C)C(C(C)(C)C)C2)nc(=NCC(C)(C)C)[nH]1 N1(CC(=O)NC(CC)(C)CNC(=O)Cc2cnn(C)c2)CCC(CO)CC1 c1(NC(c2c(CC)cccc2)c2nnnn2CCCF)ccnc(P(C)(C)=O)c1 C=C(Cl)CCC(=O)NCC1(F)CC(CNC(c2cnc(CC)s2)=O)C1 N1(C(C(C)N2CCCC2)=O)CC2CC2(C(=O)NCCC2CCOC2(C)C)C1 Cn1c(C(N2CCCCC2CC#N)C(=O)NCC2CCOC2)cc2ccsc12 C1(CNC(CCOCC(C)C)=O)COCCN(C(C2CCC2(C)C)=O)C1 N1(C(C2(C)CC=CCO2)=O)CCCC2(C1)CN(C(=O)Cc1ccc(O)cn1)C2 c1(SC)nc(C(=O)NCCCN(c2ccccc2)C)c2ccccn12 c1(OC)nc(C)sc1C(=O)NCC1(O)CC(C(=O)N(C)C(C2CC2)C2CC2)C1 C1(NC(c2ccc(O)c(Cl)n2)=O)CCC2(CC1)CN(C(c1n(C)ncc1)=O)CCO2 CC1C(NC(C2CCCO2)=O)C(C)CCN1C(C1CC(C)(C)CN1C)=O c1(C(N(CC(C)NC(CC2(COC)CC2)=O)C)=O)ccc2c(c1)S(=O)(=O)NC2 c1(C(N2CC(NC(CC(C)C)=O)C(F)CC2)=O)ccnc2ncccc12 CS(=O)(=O)C1(C(N2CCCCC2CNCc2cn(C3CCCC3)nn2)=O)CC1 c1(C(=O)NCCN(C(=O)CC(C)N(C)C(C)=O)CC)c[nH]c(C)c(Br)c1=O C1(COC)CC(CNC(c2ns[nH]c2=O)=O)N(C(=O)COC2(C)CCCC2)C1 C1(N(C)C)CN(C(=O)COC2CCN(C(C3CC(=O)CCO3)=O)C2)CC12CC2 C1(CNC(C2CCN(Cc3c(C)nc(C)o3)C2)=O)CC12CCOc1ccccc12 c1(C(N2C(C(C)NC(c3nc(C)oc3C)=O)CCC2)=O)cnc2c[nH]nc2c1 c1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)N2CC(C)C2)cnn2c1N(C)CC2 C#CCC(C(=O)NCC1CC1)NC(c1ccc(OCC2CCCCC2)cc1)=O C1(C(=O)NCCCN(C(=O)COCC(F)F)C)CC(C)(NC(=O)C(F)(F)F)C1 c1(C(=O)NCC(CN(C)C(C2CNC(=O)C2)=O)O)cc2nccnc2[nH]1 C(=O)(C1=NN(C)C(=O)CC1)NC1CC(CCC(=O)NC2CCN(CC)CC2C)C1 c1(C2(C(=O)NCC(C3CCCCN3C(=O)CCF)O)CCC2)cccc(O)c1 c1(C(=O)NC2CC(O)(CNC(c3cnc(C4CC4)o3)=O)C2)cnc2c(c1)CCC2 C1(CC)CN(C(=O)COCCC(C)C)CCN1C(c1ccc(Cl)cc1F)=O C(=O)(C1=CCCCC1)Nc1c(C(=O)NCC2(C)CCCC2O)nc(C2CC2)o1 C=C(F)C1(CC(N2CCOC(CC(=O)N(C)Cc3nnc(O)o3)C2)=O)CCC1 N1(C(CNS(NC)(=O)=O)=O)CC=C(CCNC(=O)C(O)Cn2cncn2)CC1 CCC(CO)C(=O)N1CCCC1C1CCN(C(=O)CN2CCCCC2=O)C1 C(CCCCCN(C(=O)CCF)C)NC(c1cc(COCC)on1)=O c1(C(N2CCC(OCCNC(C3(Cl)CC3(F)F)=O)C2)=O)ccc2c(c1)OCCO2 C1(C(=O)NC2CCN(C(c3ccnc(C)n3)=O)C2C)CC1C1CCCCC1 C(CN=c1nnn(C)[nH]1)(c1ccccc1)NC12CC(NC(CC3(C)CC3)=O)(C1)C2 C1(NC(CC2N(CC)C(=O)CC2)=O)C2CC3CN(C(C4CC(SC)C4)=O)C1C3C2 c1(-n2cc(CN(C(CN(C)C3CC3)=O)Cc3ccccc3)nn2)cc(F)cc(Cl)c1 C12(NC(CCN(C(Cc3c(C)occ3)=O)CCCO)=O)CCN(CC1)CC2 c1(CNC(c2cc(CNC(c3c(CC)c[nH]c3)=O)no2)=O)ccnnc1O c1(OC(C)C)ccc(NC(=O)NC(CC2CCCO2)C(F)(F)F)cc1C#N CC1CN(C(=O)CC2CCCCO2)CC1CNC(c1cncn1C)=O C1(C(C)C)C(C(=O)N(C)Cc2ccsc2)CCN1C(=O)Cn1ncccc1=O Cc1cc(C(=O)NCC(C)(C(C)C)NC(C23CC(CN2C2CC2)C3)=O)cc(N)c1Cl C1(C(=O)NCCCCNC(C2CCN(CC)C2)=O)Cc2cc(Cl)ccc2C(=O)O1 N1(C(CCCC#C)=O)CCC(NC(C2CC(C(F)F)C2)=O)CC(O)C1 c1(C(CC)C)ccc(F)cc1.C1(C(=O)NCCCN2CC2)OCCC1C(C)C C1(NC(CCC2(C#N)CCOCC2)=O)CCCCCCC1NC(=O)CCCF N1(C(c2c(NC)nsn2)=O)CCCC(NC(c2nc(Cl)ccc2F)=O)CC1 C1(CNC(COCC)=O)CC2(CC2)CN1C(c1cc(C)n(CC)n1)=O c1(C(N2CCC(N(C(=O)COC3CC=CC3)CC)C2)=O)cc([N+](=O)[O-])c[nH]1 C1(NC(CCOCC)=O)C2CN(C(c3c(C)noc3C(F)(F)F)=O)CC12 S(=O)(=O)(c1ccc(N2CCC3(CCC3)CC2)nc1)N1CC(C)CS(=O)CC1 CC1CC=C(c2ccc(Br)nc2C(=O)N=c2[nH][nH]c3ccccc23)CC1 C1(C(N2CC(C)N(C(c3ccn(CC#N)n3)=O)CC2)=O)CCc2cn(C)nc2C1 Cc1nc(CO)sc1C(=O)NC(C1CCCN1C(=O)CCC1CCCCC1)C C(=O)(C1CCCn2ccnc21)N1CCC2(CCN(C(CSCC(C)C)=O)C2)C1 C1(C(=O)NC2(C=C)CCCC2)CCN(C(=O)C2(C)CC(C#N)C2)O1 CC1CCN(C(c2cnccn2)=O)C1C(=O)NCCN1CCCNC1=O CC(C)(O)C#CC(=O)NCC1(C)CCN(C(C2CCN2C(=O)OC(C)(C)C)=O)C1 CCCN=C(NCCc1cccc(C)c1C)NCc1cc(Cl)cn1C N1(C(C(c2ccncc2)C)=O)CCC(C(=O)N(C(CO)C2CC2)C)C(C)C1 C1(CC=C)(NC(c2cc(=N)[nH]c(Cl)n2)=O)CCCN(C(=O)C(CC2CC2)OC)C1 C(C1CCCN1C)=CC(=O)NC(CCOC)CNC(=O)COCCOC C(C)(CC)(CCNC(=O)Cc1nocc1C(C)C)NC(C1N(CC)CC1)=O c1(C(C(=O)NC2CCN2C(=O)Cc2ccccn2)F)cccc(C(F)(F)F)c1 CC(C)C(CC1CCCCC1)C(=O)NC1C=CC(CNC(=O)C2=CCCCO2)C1 C1(NC(C(C)NC(CC)(C)C)=O)CN(C(=O)C(C)C)CC1S(C)(=O)=O c1(OC)nccc(C(=O)NC2CCC2CNC(=O)Cc2ccc(C)o2)n1 C1(NC(C(C)CC2CCCC2)=O)CC=CCC1C(=O)NCCCOC1CC1 CC(O)CCN=c1[nH]c(=NCc2ccc3c(c2)COC3)c2cccc(F)c2[nH]1 c1(CN(CCC)C)ccc(C(=O)NCCOc2ncoc2C)o1.c12cn(nn1)C2 C1(C)(CC)C=C(C(=O)NCCc2ccc(CNC(c3cccc[n+]3[O-])=O)cc2)C1 N1(CCN(CCOC)C)CCN(C(=O)COC)CC1=O.[nH]1cc(C2(C)CCCO2)nn1 CC(C)C(CC(=O)NC1(CCCNC(=O)C2=CCCS2)CC1)c1ccccc1 N1(C(C2ON=C(C)C2)=O)CCC(F)(CNC(=O)C(C)Cc2cnn(C)c2)C1 S(=O)(=O)(c1ccc(NCc2ncccc2F)c(C#N)c1)NC(CCC)C(C)(C)C CC1CCC=C1C(=O)NCC1(C(=O)NCCNC(=O)CO)CC1 C(C(=O)N=c1cc(C)n(C)[nH]1)(C1CCC(C(=O)NOCC)O1)C1CCOC1 Cc1cccc(CCCC(=O)NCC2CC(NC(=O)CC3CC(C)OC3C)C2)c1 CNS(=O)(=O)N1CCC(C(=O)NC2CCN(C(=O)Cc3csc(C)c3)C2C)CC1 C1(NC(C(n2ncc(C)c2)C)=O)CC2(C1)CC2C(N1CCC(C(C)(C)O)CC1)=O C1(C2CCCN(C(c3cc(Cl)n[nH]c3=N)=O)C2)(NC(C(C)NC(N)=O)=O)CC1 C1(NC(C2C(C)CCOC2)=O)CCN(C(c2coc(C(N)=O)c2)=O)CC(C)(C)C1 C1(C(=O)NCC2(NC(c3cc(C)sc3)=O)CC2)CC(C)OC(C)C1 N1(C(C(CC=C)N2CCOCC2)=O)CC2CCCC2(N)C1 C1(C#N)(C(N2CCC(C)(CCNC(Cc3ccc(C)cc3)=O)C2)=O)CCSCC1 N1(C(c2cccc(I)c2)=O)CC2(CCN(C(c3cc4cnccc4[nH]3)=O)C2)C1 N#Cc1sccc1C(=O)NC1C(NC(=O)CCF)CC1.C1(C=O)CCCC1 N1(C(C(C)NC(CC)=O)=O)CCCC(F)(CNC(=O)CC2COCC2(C)C)C1 CCCC(O)CC(=O)N1CC(CNC(C2CCCCN2C)=O)CC1C N1(C(c2ccc(CC)nc2)=O)Cc2n[nH]cc2C1C(=O)NCCCCCCSC C(=O)(C(C)P(C)(C)=O)N1CC(C(N)=O)(CNC(c2nccnc2CC)=O)C1 c1(C(=O)NC2CC(=O)NC2)sccc1S(=O)(=O)NC1CCCC1CO c1(CCC)nc(=NC(C)(C)CNC(=O)CN2CC3CC3C2)s[nH]1 C1(CC(=O)N(CC(CN(C)C(c2nnc(CO)s2)=O)O)C)CCCC(F)(F)C1 N1(C(C(C)OCC=C)=O)CCCN(C(=O)CC(C)(C)C#N)C(c2ccccc2)C1 C1(CC(=O)NC2CC(CNC(C3(COC)CCCCO3)=O)C2)CCCCCCC1 c1(C(=O)NCCCNC(C)=O)cncc(F)c1 N1(C(CN(C)CC)=O)CC(N=[N+]=[N-])CC1C(=O)N(C)Cc1cncnc1 c1(C(=O)NC2C(NC(C(CC)CC(F)F)=O)CC2)cc2c(OC)ccc(F)c2[nH]1 c1(CC)c(NC(C2(O)CN(C(=O)Cn3c(C)c(C)sc3=O)C2)C)ncnc1Cl C12(C(=O)NCCOCC(C)(C)C)CCCC1CCN2C(c1nncs1)=O c1(C(N(CC(CC)NC(=O)C(C)CC2CC2)CC)=O)cc2c(Cl)cncc2s1 c1(OC)cc2ccccc2cc1CN1CC(NC(c2ccc(Br)cc2)=O)C1 N1(C(c2c(OC)ccnc2F)=O)CC(C)(C)OCC1CNC(=O)C(O)C(F)(F)F C(=O)(C(C)CC(F)F)NCc1cc(C)c(C(=O)NCCC(O)C(C)C)o1 c1(C(N2CC(OC)C(NC(=O)Cc3ccccc3)C2)=O)ccc([N+](=O)[O-])cc1F CCCC(CCCNC(c1csc(CC(C)C)n1)=O)NC(=O)CC12CCCC1C2 C(=O)(C1Cc2ccc(F)cc21)N1CCN(C(C(=O)NC)C)C(C)C1 c1(OC(C(=O)N(CC(CN(C(C=C(C)C(C)C)=O)C)O)C)C)ccc(F)c(Cl)c1 CCCCCC(C)(CC)C(=O)NCC(CCOC)NC(c1cc2ccccc2o1)=O CC(C)(C)CC(C)(C)C(=O)NC1CN(C(C2Cc3ccccc3S2)=O)CCC1F c1(NC(=O)C(C)C)ccc(O)cc1.C1(NC(C)=O)CCN(C(=O)Cn2cnnn2)C1 CC(c1ccccc1Cl)=CC(=O)NC(C)CN(C(=O)CCn1ccc(=N)[nH]1)C C(=O)(C1CCC(=O)c2cccn21)NC1CC(C)N(C(C2CCC(C)(C)C2)=O)CC1 C1(C(N(C(C)C)CCN(C(=O)CC2CC3CC3C2)C)=O)CCN(C)S1(=O)=O N(C(=NCC1CC1Cc1ccccc1)NC1CCN(S(=O)(=O)C(F)F)CC1)CC c1(C(=O)NCC2C(NC(c3ccn(C)c3)=O)C2)nn(C)c2c1CC(F)(F)CC2 C1(C)(CNC(c2n(C(C)C)ccn2)=O)CC(F)(F)CN1C(C1CC1C#N)=O CCC(CCOC)NC(C1(NC(=O)CC2CCC(=O)C2)CSC1)=O CC1CC(NC(c2ccnc(-c3ccco3)c2)=O)CN(C(C2(O)COC2)=O)C1 CN1N=C(C(=O)NCC2CCN(C(=O)CC3CCC(C)(C)O3)C2)CCC1=O CC(C)CC(CNC(=O)C(C)C#N)C(=O)NCCCc1cccs1 c1(C(N(C2CCN(C(c3ccns3)=O)C2)C)=O)cccc(C(F)(F)F)n1 C(C(CC(=O)NCC1CCCCC1)NC(C1(C#N)CCOC1)=O)OC N1(C(=O)NCC=CC(C)C)CC(C)(C)C1c1nccn1C.N12CC(C1)C2=O N1(C(c2ccc(N3C(COC(C)(C)C)CCC3)o2)=O)CCOCC1C(C)(C)C C1(NC(N2CC3C(CC(C)C)(C3)C2)=O)CC(C)(C)OC1(C)C N1(C(CC2C(C)OCC2)=O)CC(C2CC2C(N)=O)C1.N12CC(C)(C1)CC=CC2=O c1(C(N2C(CNC(c3c(CC)c[nH]n3)=O)CCC2)=O)cnn2cc(OC)ccc12 CCC(C)(C)C(C)CC(=O)NC1COC2(C1)CN(C(=O)C(C)n1ccnc1)C2 C(C(C)(C)CNC(C12CC(N(C)C)(C1)C2)=O)N(C(=O)C(C)n1ccnn1)CC C(=O)(CC(C(F)F)n1ccnc1)NCC(=O)NCC(C)CNC(c1ccccc1)=O c1(CC)ccc(C(=O)NCC(C)(F)CNC(C2(C(C)(C)O)CCC2)=O)c(O)c1 C(=O)(CCCCCCS(N)(=O)=O)NCC1(NC(c2c(C)occ2)=O)CCCC1 C(c1ccco1)=CC(=O)NCC(=O)NC1CC1.C1CC(=O)NCCCN1C c1(NC2CC(=C)C2)nccc(=NCCc2ccc(OC)cc2C)[nH]1 N1(CC2N(C)CCC2)CCN(C(C2CC=CCC2c2ccccc2)=O)CC12CC2 C1(C(C)(C)NC(=O)CNc2cn[nH]c2)CCCN1C(=O)CC1CCC1 c1(C(=O)NCC(CC)NC(=O)C=C2CC2)csc(Cl)c1 c1(NC2CC3(CN(C(CC=C)=O)C3)OC2)ncnc2[nH]nc(C)c12 c1(C(N2C(C(N3CCC(C(F)(F)F)C3)=O)CCCC2)=O)ccc2c(c1)CCC2 C(=O)(C(F)(F)C(C)(C)O)NCC#CCNC(c1onc(CC)c1C)=O N1(C(C(C#N)C2CC2)=O)CCN(C2CCN(C(=O)Cc3csc(C4CC4)n3)C2)CC1 c1(CNC(c2c(CC)noc2)=O)ccc(C(=O)NC(CC)(CC)CO)cc1 C=C(C)CC(=O)NCCCN(C(C1CNC(=O)C1)=O)CC1CCCC1 N1(C(C(C)NC(=O)N(C(C)(C)C)CCO)=O)CCCN(CCc2cccs2)CC1 C(=O)(C1=NN2CCC(C)N=C2N1)NCC1(NC(C(C(CC)(C)C)O)=O)CC1 C(C)(CCC(=O)N(C)CC1(C)CCCC1)NC(C(CC)C1CCC(=O)N1)=O C1(NC(c2ccc(OC)cc2C)C)CCCC12CCNCC2 C(=O)(C(C)(C)S(=O)(=O)C1CC1)N1CC(CNC(CC=CCC)=O)(OC)C1 C(CNC(=O)Cc1ccc(O)cc1)(CC(=O)NC1COC(C2CC2)C1)OC N1(C(C(C=C)C)=O)CCC(C)(C(=O)N(CCCF)CC2CC2)CC1 N1(C(c2ncnc(C)c2C)=O)CC2CC(NC(=O)CCOCCN(C)C)C(C2)C1 c1(C(C(=O)NCCN(C(CCC#CC)=O)C(C)C)C)ccc(Br)cc1C N1(C(CCC=C)=O)CCC(CCNC(=O)CSC(=N)N)CC1 CN(C)S(=O)(=O)N1CCC(NC=O)C1.C1(C)C=CCN1C(=O)Cc1cnc[nH]1 C1(OC)CN(C(=O)CSCc2nc[nH]n2)C(C)(NC(=O)CC(C)(C)C#N)C1 CC1(C)CCCOC1CC(=O)NC1CC(NC(=O)CC2CCC=CCC2)C1 Cc1c(C(=O)NCC2CC(NC(=O)CC3CCCO3)C2)cnn1CCC#N C1(NC(C2(CNC(c3ccc(Br)cc3)=O)CCC2)=O)C2CCCCC12 c1(C(=O)OCC)ccc(C(N2CCCCC2C(=O)NCCNC(C)=O)=O)nn1 N1(C(C2CC3C=CC2C3)=O)CCCN(C(C2COC3(CCC3)C2)=O)CC1 Cn1cccc(C(N2CCC(C)(CCNC(=O)CC3(O)CCC3)C2)=O)c1=O N1(C(C(C)CNC(=O)C(=O)C(C)(C)C)=O)CCCC2(CCCC2)C1 c1(C(C(C)C)C(=O)NC2CCCCC2NC(c2cocn2)=O)cccc(C#N)c1 C1(OCC#C)CCN(C(C2CCCC2NC(=O)CC(C)n2ccnc2)=O)CC1 N1(C(Cc2cc(C)on2)=O)C2CCC1C(C)C(NC(C1(F)CC1)=O)C2 C=CCC(F)(F)C(=O)NCC1CN(C)CCN1C(=O)Cc1cc(Cl)ccc1Cl O=C(C1=NNC(=O)C1)N1CC(O)(CCNC(C2CCCC2)=O)C1 Cc1ccc(O)cc1CNC(=O)CN(c1cncc(F)c1)C(C1CCCC1)=O Cn1c(COCC(N2CCOCC2CNC(C2CNC(=O)N2)=O)=O)nnc1S C1(NC(C(C2CC(F)(F)C2)OC)=O)CC(F)CN(C(=O)CC2C(C)(C)C2(C)C)C1 C(=O)(C(C)(C)CCS(C)(=O)=O)N1CC2C(NC(c3cnc(OC)c(C)c3)=O)(C2)C1 Cc1cnn2cc(C(N3CCC(CCNC(=O)C(C)CC(C)(C)C)C3)=O)cnc12 c1(C(=O)NCC2CCCC(NC(C3C(=C)C3C(=O)OC)=O)C2)cccc(Cl)c1C Cc1nc(C(=O)NCCC2CN(C(c3nncn3C3CC3)=O)C2)c(C)o1 c1(NC(C2(C#C)CN(C(=O)CC3CC(OC(C)(C)C)C3)C2)=O)cc[nH]c(=NC)c1 c1(OC)ccc(C=CC(=O)NC2CCN(C(=O)CN3CCCC3=O)CC2)c(C)c1 Cc1ccc(Cl)c(C(N2CCN(C(=O)CC3(N4CCCC4)CC3)CC2CO)=O)c1 C1(N(C(C2CN(C)C(=O)N2)=O)C)CCCCN(C(=O)C=Cc2nccs2)C1 C(CNC(C1C(C)C1C)=O)(CCNC(c1cnoc1C)=O)OC c1(C(N2CC=CC(NC(c3cccc(C(C)C)n3)=O)C2)=O)cccc2ncsc12 N1(C(c2cnc(C(C)C)s2)=O)CCC(CN(C)C(C2CC3(CC3)C2)=O)CC1 CCC(O)C(C)C(=O)N1CCC(C)(CNC(c2cc(=O)n(C)o2)=O)CC1 CCCC(CCC)C(=O)NC(C)C(CO)NC(=O)COCC1CCOCC1 c1(CC)c(C(=O)NCC2CC(C)N(C(C34COC(CF)(C3)C4)=O)C2)cnn1CC C(CS(=O)(=O)CC(=O)NCCC1CCN(C(C2CCOC(C)C2)=O)CC1)OC N1(c2nccc(N3CCCC(CCOC)C3)n2)CCN(C)c2ncccc2C1 C(N=c1ncc(Cl)c[nH]1)C1C(NC(=O)CCc2cccnc2Cl)CCCC1 c1(CCC(N2CC(C(N)=O)(CNC(C=CCOC)=O)C2)=O)ccc(OCC)nc1 Cc1ccc(C(N2CCOC(C(=O)Nc3cnc(F)c(C)c3)C2)=O)cc1C N1(C(c2c(CC#N)cccc2)=O)CC2CC1CN(S(=O)(=O)Cc1ccccc1)C2 C1(C(N2CC(O)(C(C)NC(c3nncc(C)c3)=O)C2)=O)CCCC12CCC2 N1(C(C(ONC(COC(CC)(C)C)=O)C)=O)CCC2(CCC2)CC1 N12CC(CC(C)C1)C2=O.C(C(CNC(N)=O)CO)NC(C1(NC(C)C)CC1)=O N1(C(CCCC#CC)=O)CC(C)(CNC(=O)C(C)OCCOCC)CC1(C)C C=C(Cl)CC(C(=O)NC(C(C)(C)O)C1CC1)NC(=O)Cn1ncccc1=O C1(NC(CC(=O)NCC)=O)CC2CN(C(=O)CC3(CS(C)(=O)=O)CC3)CC2C1 c1(C(=O)N(C(=O)C2CC2)C(C2(C3CC3)CC2)=O)cccc(O)c1.C12(CCC1)NCC2 C1(C(=O)NC2CC23CC(NC(C2(O)CCSCC2)=O)C3)COc2ccc(F)cc2C1 c1(C(=O)NC2C(C(=O)NC(C=C)C)CCC2)ccc(F)c(C)c1Cl N1(S(CC)(=O)=O)CCCCC1C(=O)N(C1CC(C)C1)C(c1cn(C)c(C(F)F)n1)=O C1(C(=O)N(CCCC(=O)NC)C2CC2)CCC(C(C)C)N1C(=O)C#CC(C)C C1(CNC(c2cc(C)sc2)=O)CN(C(c2nn(C)cc2Cl)=O)CCC1C C1(NC(CC(=C)C)=O)CCN(C(=O)CCn2c(C)csc2=O)C1C C(=O)(N=c1ccn(CC(N)=O)[nH]1)C1N(C(C(C)SCCCC)=O)CC(F)C1 N1(C(CCC)CC(C)C)CCC2(CC1)CC2C(=O)NC(C)C(N)c1ccco1 c1(C(=O)NCC2CC2CNC(=O)C(F)n2ccnc2)cc(F)cc(Br)c1F C1(C(=O)NC(CC)C(N)=O)CCCN(C(c2cc(C(C)C)no2)=O)C1C O=C(N=c1cnc(NC2CCS(=O)(=O)C2)c[nH]1)c1cc(OC(F)F)ccn1 C1(CNC(C2C(C)(C(F)F)C2)=O)C2CN(C(C3(C)CCOC3)=O)CC12 N1(C(CCN(CCCCC)C)=O)CCC2CN(C(c3nnc(S)n3C)=O)CC2C1 C1(C)(C(=O)NC(c2cccc(C(F)(F)F)c2)C(=O)NCCC(=O)OC)CCN(C)C1 CCC(CC)C(C)C(=O)NCCN1CCC(NC(C2(CF)CC2)=O)CC1 C(N=c1[nH]c(=NCC2CC3CCC3C2)[nH]c2c1SCC2)C1(OCC)CCSCC1 CC(C)C#CC(=O)N(C1CC(NC(=O)CCCSCc2cccnc2)C1)C c1(CCN2CC(C)OC(C)C2)nnc2n1CCCCC2.C12(C=O)CCC(CC1)N2 c1(CN2CCN(C(C(=O)NC3CCC(OC)CC3)C)CC2)cnc(O)c(Cl)c1 c1(C(=O)NC2CC(NC(C3(COC)CC3)=O)C2)cnn2c1OCC2 c1(C(N2CCCCC(N(C)C(C3COC(=O)C3)=O)C2)=O)cccc2oc(O)nc12 N1(Cc2c(C)c(Br)cc(F)c2)C(=O)C2CC(C)(C)CN2C1=O C12(C(N(CC(C)O)CCNC(C(C(C)C)n3ccnc3)=O)=O)CCCC1C2(F)F C1(NC(c2c(CC)ncs2)=O)CC2CCC1N2C(c1ccc(CCOC)cc1)=O C1(C(=O)NCC2(CNC(C(CC)n3ccnc3)=O)CCCC2)CC(NC)CCO1 c1(CC(N2CCCC(CN(C(C(=O)N(C)C)=O)C)C2)=O)cccc2ncccc12 C(=O)(C1CCn2cc(C(F)(F)F)nc21)NCC(CCNC(CC=C)=O)O CCCC(C(=O)N1CC(C)CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CC1C)S(N)(=O)=O C(C1=Nc2ccccc2S(=O)(=O)N1)N.C(C(O)CNC)OCC C(=O)(C1=NOC2(CCOC2)C1)NC1CCN(C(c2c(NC(C)=O)c[nH]c2C)=O)C1 C1(N(C(=O)CCn2ccnn2)C)CCCN(C(C2CCCC2(F)F)=O)C1 C(=O)(CS(=O)(=O)C1CCCC1)N1CC(NC(C(CSC)(C)C)=O)C2C1C2 C1(CCNC(C2(CC)CCC2)=O)CN(C(=O)C(C)OCOC)CCO1 C=CCC(F)(F)C(=O)NCC1N(C(C2CC2CF)=O)CCC1(C)C C#Cc1cccc(NC(C(=O)NC(C)(C)C)C2CCOC2)c1 C(=O)(C(CCF)NC(=O)C(C)=CC(C)(C)C)N(CCCO)CC C1(CC(N2CC(C(C)(C)O)(CNC(CCN(CCC)C)=O)C2)=O)C=CS(=O)(=O)C1 c1(C(C(=O)NC(CC(=O)OC)C2CCCC2)Br)cc(F)cc(F)c1 C(=O)(C1=CCN(C)C1)N1CCC(C(C)C(=O)NCCOCC2CC2)CC1 c1(C(=O)NC(C)(CNC(c2ccc(F)c(Cl)c2)=O)CO)cc(F)c(N)c(F)c1 c1(OC)cc(OC)c2c(c1)C(NC(N1CCN(C(=O)C3=CCC3)CC1C(C)C)=O)CC2 C1(NC(CCCOC)=O)CN(C(C2CC3(CC(OC)C3)C2)=O)CC12CCC2 c1(C(=O)NCC2C(NC(c3c(C(C)C)ocn3)=O)C2)sccc1S(C)(=O)=O N1(C(Cc2ncc(C)s2)=O)CCC2CN(C(=O)CC3CCC(C)(C)CC3)CC12 Nc1cc(C(=O)NCC2(O)CN(C(c3c[nH]nc3-c3cccs3)=O)C2)cnc1N C(=O)(C(C)CS(C)=O)NCc1cccc(CNC(c2n(C=C)nnc2)=O)c1 C(CCC(C)C)(C(=O)N1CCC2(CC(CO)C2)C1)NC(C(C(CC)C)O)=O c1(C(=O)NC2(CCNC(C3C(C)(C)C3(C)C)=O)CCC2)cc2c(cn1)CCCC2 C(=O)(C(CC)n1cncn1)NCCC(C)N(C(CCCCCC)=O)CCOCCO C1(C(N(CC(CC)OC)C)=O)(NC(=O)C(C)Cc2ccco2)CCCC1 c1(NC(C2N(c3ncnc(C)c3Br)CC(O)C2)=O)cnc(Cl)c(Br)c1C c1(C(=O)NCC(CC)(C)NC(=O)C=Cc2cccs2)cnnc(C2CC2)c1 c1(C(CC)NC(c2cnn(C)c2C)c2nnnn2C(C)(C)CC)c(OC)cccc1Cl C1(OC)(CNC(C2CC(n3cc(C4CCCCO4)nn3)C2)=O)CCCOC1 C(CCCCC(=O)N1CC(NC(N2CCCCC2)=O)CC(O)C1)NC(N)=O CC(C)CCC(C(=O)N(C)CCc1cnc[nH]1)NC(=O)C=Cc1ccc[nH]1 C1(NC(C(C)(F)F)=O)CC(NC(=O)COC2(C)CCCC2)C12CCC2 C1(C)(NC(C(COC(C)C)(C)C)=O)CCN(C(C2CCCC2O)=O)CC1 C1(O)(CC)CCCN(C(=O)C(C)C2CCC2)C1.C1(=O)CCN1C(C)C C1(NC(c2c(C)scn2)=O)CC(F)CN(C(c2cnc(C3(C)OCCO3)s2)=O)C1 N1(C(COC(c2cnccn2)=O)=O)C2CCC1CC(NCc1ccc(Br)nc1F)C2 C1(CCN(C)C(C2CCC2(F)F)=O)CCN(C(=O)C=CC2CCC2)CC1 Cc1ccc2[nH]cc(C(=O)NC(C3(O)CN(C(=O)CC4CCCC4)C3)C)c2c1 C=CC1OCCC1C(=O)NCC=C1CCN(C(=O)C=Cc2ccco2)CC1 c1(OC)ccncc1C(N1CCC(C(C)C(=O)NCC(COC)CO)C1)=O c1(C(N2CCC(O)(CNC(CCC(=C)Br)=O)C2)=O)cc(Cl)cnc1C C12(CC(CO)C1)C(=O)N2.n1(C(C(=O)N(C)CC2(OC)CC2)C)ccc(C)n1 C1(CN(C)C(C2(CC(F)F)CCC2)=O)CN(C(C2CC(F)C2)=O)C1 c1(C(=O)NCC2N(C(c3scc(OC)c3)=O)CCC2)ccc2nccnc2c1 C(=O)(C(C)(C)CNC(=O)C(C)(C)C1CCN(C(=O)CC(C)SC)C1)NC N1(C(c2ccc(OC)c(O)c2)=O)CCN(C(c2sccc2C)=O)C(C#N)C1 c1(C(CSC)NC(C(=O)NC2CCN(CC)C(C)C2)=O)cc(Cl)nc(Cl)c1F C1(NC(CSCC)=O)(CNC(c2cc(C(C)(C)C)c[nH]2)=O)CCC12CCC2 N1(C(Cc2c(C)noc2)=O)CCCC2C1CCN2C(=O)CC(O)C(C)C C(=O)(C(C)(CNC(C1CCN1C(C)(C)C)=O)CC)NC1CC(CC)C1 O=S(=O)(c1ccc(=NCc2nc(C(F)(F)F)cs2)[nH]c1)NCCN1CCCCC1 c1(COC)ncc(C(N2CCC(C(=O)OC)C2)C(=O)NC2CCCC2)[nH]1 N1(C(CCSCC(N)=O)=O)CC2CC1CN2C(=O)CCC1CC1(F)F Cc1cc(F)c(C(=O)NC2C3CC2CN(C(C2(C)C=CCCC2)=O)C3)cc1F Cc1cc(C(=O)N(CC(C)NC(c2nc(C)ccc2Br)=O)C)c(O)c(C)c1 c1(OCC)cc(C(C(=O)NCCC#N)N(C2CC2)Cc2ccccc2)cc(F)c1 N1(C(CNC(C(C)(C)SC)=O)C)CCN(C(=O)C(C)N(C)C)CC1 CS(C)(=O)=NCC(=O)N1CCC(CNC(c2csnc2Br)=O)C1 C1(NC(c2cncc(N3CCCC3)c2)=O)CCC2CN(C(=O)CCCF)CC2C1 CCC(CC(=O)NCC(C)(C)CNC(=O)CN1CSCC1=O)C(F)F CC(C(=O)N1CCC(NC(c2ccc(F)c(C(F)(F)F)n2)=O)CC1C)C(C)(F)F C1(=CC(=O)NCC#CCNC(c2cc(C)no2)=O)CCC(C)(C)CC1 C=CCC(C(=O)NCC=CC(=O)N(C(C)C(CO)SC)C)N(C)C(C)=O C(=O)(C(C)(O)NC(=O)NC(C(C)OC)=O)NCCOC(C)(C)C.C(CN)O c1(C(=O)NCCNC(=O)C(N2CC3C(CO)C3C2)=O)ccc2cc[nH]c2c1 N(C1CCc2ccccc21)C(C)Cn1cc(CCC(=O)CCO)nn1 CC1(C)CCOC1CNC(=O)C(CO)NC(C1(O)CCCCC1)=O c1(OC)cc(F)c(F)cc1NC(C1CCN(Cc2ncco2)CC1)=O N1(C(CCC)=O)CCC(C)N(C(=O)C(C)CC(F)(F)F)CC1.c1(C(=O)CN)c[nH]cc(C)c1=O C1(CNC(c2ccc(CC)o2)=O)CC2(CCN(C(=O)Cn3nnc(C)n3)C2)CO1 Cc1ccc(NC(=O)COC2CCN(C(c3cc(O)ncc3F)=O)C2)c(C)c1 C=C=C(C)CC(=O)NC(C1CCN(C(c2cccc(-c3nc[nH]n3)c2)=O)CC1)C Cc1cc(C)c(C(N2CC3C(CNC(C4(CC(C)C)COC4)=O)C3C2)=O)cc1N C12(C(N3CC(C(C)NC(=O)CCCNC(N)=O)OCC3)=O)CCCC1OCC2 c1(C(N2C(CNC(=O)CC3CCCOC3)CC(F)(F)C2)=O)cnn2ccncc12 C1(C(N(C(C)(C)C)C)=O)CC2CC(C1)N(CCC(O)CCc1ccccc1)C2 C1(CC(=O)N(C(CNC(C2CCOC(C)(C)C2)=O)C2CC2)C)CCCCC1(F)F N1(C(C(C)(C)CO)=O)CC=C(CCNC(=O)CN2CCOCC2=O)CC1 C(=O)(CC(C)(C)c1ccccc1)NCC(C)NC(C1OCCOC1C)=O C(=O)(C1=NN2CC(C)CN=C2N1)N1CC(CO)(CNC(C(C)=CC)=O)C1 c1(C(=O)NC(CC)CNC(=O)CSC2CCOC2=O)ccc(C)c(Br)c1 N1(Cc2ccnc(SC)n2)CCC(C)C(NC(=O)C(C)Cc2cnn(C)c2)C1C C1(C(=O)NC(C2CCCN2C(=O)COCCSC2CCCC2)C)CNC(=O)C1 C(=O)(C(C)S(=O)(=O)C1CCOCC1)NCC(c1ccccc1)SC C1(C)(C(=O)NC)CCN1C(=O)C(C1CCCO1)NC(=O)CC1CC1.C1CCC1 N1(C(CC(CCC)O)=O)CCOCC(F)(CNC(=O)C=CCN(C)CC)C1 C1(OC)CCC2(C(=O)NCc3cn(C4CN(CC5COCCOC5)C4)nn3)CCC12 C1(C(=O)NCCCC2CCC(C)O2)C2CC1N(C(c1sccc1CO)=O)C2 C1(C)(C(N(CCCC)C)=O)C=CCN1C(=O)CCNC(=O)NC C(=O)(C(F)(F)C(F)F)NC1(CC=C)CCN(C(c2ncncc2OC)=O)C1 C1(N(C(C=COCC)=O)C)CN(C(c2cc(O)cs2)=O)CCC1C C1(N2C(F)C2=O)CCCN(C(c2cc(-n3ccnc3)ccn2)=O)C1.C1(COC)CC1 N1(C(c2nccc(C)n2)=O)CC(CNC(=O)CN2CCOCC2=O)C(F)(F)C1 c1(N2CCCC(NC(Cn3c(C)ncc3)=O)C2)ncnc2c1CCO2 C12(CC(N3CCCC(N(C(c4csc(C)n4)=O)CC)C3)=O)CCC(C)(C1)OC2 c1(C(N2CCCC(NC(C3(C(C)(C)C)CCC3)=O)CC2)=O)cc2ccncc2s1 C1(C(=O)NC2CN(C(C(CC)Sc3nc(=N)[nH][nH]3)=O)C2)CCC(C)(C)OC1 C(=O)(CS(=O)c1ccc(Cl)cc1)N(CC(=O)NC1CC(n2cnnc2)C1)C1CC1 N1(C(c2c(CC)nccc2)=O)CC2(C)CC1(C(N1CC(c3nncs3)C1)=O)C2 c1(CCC=CC(=O)NCCN(C)C(C2(C#N)CC2)=O)ccccc1 CC(C)CCC(C(=O)NCC1=CCCOC1)NC(C1(N2CCOCC2)CC1)=O Cc1cnc(C=CC(=O)NCCC(C2CN(C(=O)CC(C)C)CCO2)O)[nH]1 CC(C)(O)C(C)(C)C(=O)NCC(=O)NC1(C)CCOC1 C(=O)(C(C(C)CC(C)(C)C)N1CC(C(=O)OC)C2(CC2)C1)NCC=C N1(C(C2(C)CC=CCC2)=O)CCCC(CNC(c2ncsc2C2CC2)=O)CC1 c1(OC)cc(C(N2CC(n3cc(CCC(C)C)nn3)C2)=O)cnc1OC(C)C C(C(COC)CC(=O)NCCn1ccc(C(=O)N(C)C(C2(C)CC2)C)c1)OC c1(OC)cc(CNC(=O)C(C)n2cncn2)cc(C(C)=O)c1O Cc1ccc(C(=O)NCCC(C(C)C)NC(c2cnn(C3CCC3)c2)=O)cc1C CCCC(CC)CC(=O)N1CC=CC(NC(=O)Cc2ccnc(OCC)c2)C1 N1(C(CC(C)OC)=O)CCC2CN(C(c3c(Cl)nc4ccccn34)=O)CC2C1 Cc1c(C(=O)N(CC(C)(C)NC(=O)CC2(C)CCC2)C)c(C(F)F)nn1C C=C1CON(C(=O)C2CCCC(NC(=O)C(C3CCC3)OCC)CC2)C1 c1(C(=O)NC(CC)CNC(C2(C)CCCC2O)=O)noc2c1CC(F)(F)CC2 Cc1[nH]nc(C(N2CC(Cc3nc(-c4ccncc4)no3)C2)=O)c1Br Cc1ccc2c(c1)SC(C(=O)NC1(C)CCN(C(=O)Cc3sc(C)nc3C)C1)C2 Cc1nn(C(C)C)cc1C(N1CCOC(CCNC(=O)CCCN(C)C)C1)=O C(C(=O)NNc1cccc2ncccc12)Nc1c(S(=O)(=O)N(C)C)cccc1 c1(C(C2CCC2)NC2(NC(C)C)CCC2)cccnc1 c1(OC)ccc2[nH]c3c(c2c1)CCN(C(=O)NC1(C#N)CC1)C3 c1(C(=O)Nc2ccc(-c3c(C)ccc(CO)c3)nc2C)cc2cc(Br)ccc2s1 C1(CNC(c2cn(C)nc2)=O)(CNC(c2[nH]cnc2C#N)=O)CC12CCC2 c1(N2CC(N(C(c3cc(C)no3)=O)C)C2)ncnc2sc(C(C)C)cc12 C=C(Cl)C(C)(C)C(=O)N(CCC(C(C)C)NC(c1ccc(N)c(O)c1)=O)C c1(C(=O)NCC2(OCC)CN(C(=O)CCSCC(N)=O)C2)cccc(Cl)c1F C1(NCC#CCNC(C2(NC(=O)COC(F)F)CCC2)=O)CCC2CC12 C(=O)(C(C(=O)N1C2CCC1CC(CNC(=O)CCCC(C)C)C2)C(C)C)OCC C1(C(=O)OC)(C(=O)NCCCSC2(C(c3ccccc3)=O)CC2)C=CCC1 C12(CNC(Cc3cncc(C#N)c3)=O)CCCC1CN(C(=O)CC(F)(F)Cl)C2 c1(C(=O)NC(CC)CNC(c2cc(OC)n(C)n2)=O)ccc(CO)c([N+](=O)[O-])c1 N1(C(CNC(CCC)=O)=O)CC(N(C)C(c2ccc(OC)nc2F)=O)C2(CC2)C1 c1ccc(C(F)F)cc1.c1(N(CC(O)COCCO)C)ccc(I)cc1 C1(C(N(C2CC2)Cc2n(CC)ncc2)=O)CN(C(=O)C(C#N)CC)C2(CCC2)C1 C1(C(CC)NC(=O)CCC(=O)N(C)C)CCC(C)(OC)CC1 CCCCC(CC)C(=O)NC1(CCC(N2CC(C)(O)C2)=O)CCCC1 N1(C2(CC(=O)NC(C)CNC(=O)Cn3cncn3)CC2)CCS(=O)(=O)CC1 C1(CNC(C(c2ccncc2)C)=O)CCN(C(=O)CCCC2CC2)CC1C1CC1 N1(C(c2c(COC)cco2)=O)CCC2CN(C(c3ccc(=O)n(C)n3)=O)CC12 N1(C(=O)CCOCC(F)(F)F)CC(NC(c2n(CC)nnc2)=O)CC(O)C1 N1(CN(C)CCCl)CC2CCC1CN2CCO C12C3CN(CC13)C2=O.c1(C(=O)NC(c2nc(C)[nH]n2)C)cnc(CC2CC2)nc1 N1(C(C2N(C(C=CCC)=O)C3(CC2)CC3)=O)CCCN(C)CC1C C#CC1CN(C(C2CC(C)(C)C2)=O)CCN1C(=O)CCCSC N1(C(C2CC(=C)C2)=O)CC(C2CCCN(C(c3cnc(C4OCCO4)s3)=O)C2)C1 C1(CC(=O)NC(c2nc(C)oc2C)C)C2CCC(C2)N1C(C12CCC(CC1)CO2)=O C(=O)(CC(C)C(C)C(C)C)NC12C(NC(c3[nH]c(C)c(CO)c3)=O)CC(CC1)C2 Cc1cc(C(=O)N(CCCNC(=O)CS(=O)(=O)N2CCOCC2)C(C)C)oc1C Nc1cc(C(=O)NC2CCCC(NC(=O)C([N+](=O)[O-])C3CC3)C2)cc(O)c1.C1(C=O)CC1 C1(C(=O)NCC(C)N(C)C(c2ccc(OC(C)(C)C)cn2)=O)CN2CCN1CC2 N1(C(C2C(O)CCN(C(C(OC)OC)=O)C2)=O)CCn2nccc2C1 c1(C(=O)NC(CNC(C(CC)(C)C)=O)CCOC)c[nH]c2cc(F)ccc12 C(C(C)C(F)C(=O)Nc1cc(C2CCCC2)no1)NC(C(=O)NC(C)C)=O C12(CNC(C=CC(C)NC(=O)Cc3cscn3)=O)CCC(CC1O)C2 C1(C(N2C3CC(CN(C(CSC)=O)C3)C2)=O)Cc2cc(C)c(C)cc2O1 c1(OC)c(CC(=O)NCC(C(C)(C)C)NC(=O)CC2C(C)C2(F)F)cccc1F C1(F)(C(N2CCC(N(CCC)C(C3CN(C(N)=O)C3)=O)C2)=O)CCN(C)CC1 Cc1csc(CNC(N2CC(N3CCCC3)C2)=O)c1Cl CCCC(C(=O)N1CCN(C(c2[nH]ccc2C)=O)CC1)N1CCCS1(=O)=O Cc1nn(C)c(N)c1C(=O)NCCCN(CCO)C(C1CCCCC1O)=O N1(C(CSCC=C)=O)CC(C)(C(N2CC(N3CCNC3=O)C2)=O)CC1(C)C C1(N(C(CCCNC(c2n(CCC)ncc2)=O)=O)C)COC(C)(C)C1 Cc1nc(NCc2cscc2C)cc(=NC(C)c2ccc(F)cc2F)[nH]1 CCC(CC(=O)OC(C)C(=O)NC1CCOC1)C(=O)O c1(C(=O)NCC(CNC(c2n[nH]c(C)c2C)=O)O)cnc2c(c1)CCCC2 c1(CSCC(=O)NC(CNC(C(CC)OC)=O)(C)C2CC2)ccsc1[N+](=O)[O-] C(=O)(CCCCN=[N+]=[N-])NC(C(=O)NC1C=CC(C(=O)NC)C1)C(C)C N1(C(C(C)(C)c2cccs2)=O)CC2(C1)CN(C(c1n[nH]c3c1CCC3)=O)CC2CO C1(NC(C2CC(C)(O)C2)=O)CN(C(c2cccc(N)n2)=O)CCC1CO C(N=c1[nH]c2c(c(=NCCSC)[nH]1)CCCC2)C1N(C(NS(N(C)C)(=O)=O)=O)CCC1 C1(CNC(c2c(C)scc2)=O)(NC(=O)C(F)(F)c2nccs2)CCC(C)(C)CC1 Cc1cc(F)ccc1NC(N1CCC(NC(C2(C)CNC2)=O)CC1)=O N1(C(C2CC(C#C)(O)C2)=O)CCCC(O)(CNC(C2(c3cccnc3)CC2)=O)C1 C1(C(C#C)C)CCN(C(=O)CN(C(=O)C=CCOCCOC)C2CC2)CC1 c1(C(=O)NCC(C)N(C(C2CC2c2cncs2)=O)CC)cc2cncn2c(O)n1 C1(NC(C(CCCC)O)=O)C2CC3CN(C(=O)CN4CC(=O)NC4=O)C1C3C2 C1(CNC(c2c[nH]c(CC)c2C)=O)CCC2(CN(C(=O)CCC(CC)OC)C2)O1 C(=O)(C1CCCc2sccc21)NC(C)(CNC(=O)Cc1cn[nH]c1)C1CCC1 N1(C(C2CC(OC)C2)=O)CCN(C(=O)CCNC(c2ccncc2)=O)C(CF)C1 N1(C(C2CC=CC(NC(C(C)N(CC)CC)=O)C2)=O)CCOCC(O)C1 c1(C(N2CCC(CCN(C)C)C2)C(=O)NCCC)cnc(N(C)C)cc1Cl C12(Cc3cc(OC)c(OC)nc3)CC3CC(C(=O)N1)C2C3.c12cn(nn1)CCCC2=O c1(OCC)ccncc1NC(=O)CC1CC(C)N(C(c2coc(C)c2)=O)C1 N1(C(CCCC=C)=O)CCC(C(F)(F)F)C(NC(c2cncc(O)c2)=O)C1 C1(NS(CCOCC)(=O)=O)CCC2(CCN(C(=O)Cc3ccn(C)n3)CC2)C1 c1(CC(=O)NC2CC2C(C)(C)NC(C=CCN(CC)CC)=O)cc(C)cc(C)c1 c1(CCCNC(=O)C(N2CCCC2CC2CCOC2)=O)ncc(Br)cn1 c1(C(NNC(=O)c2cc(Br)c[nH]2)=O)ccc2c(c1)Cc1ccccc1-2 N1(CCC(N2CCC3CN(c4cncc(Cl)n4)C3C2)=O)Cc2ccccc2C1 N1(C(C2N(C(C(C)SC(C)C)=O)CC3(CC3)C2)=O)CC2CSCC(C2)C1 C(=O)(C(C)C(CC)CC)N(C)CC1(CNC(C2CC(CC)OCC2)=O)CC1 C1(C(=O)NC2C(CC(=O)N(CC=C=C)CC(=C)C)COC2)CC2CCC(C1)O2 c1(CN(C)C)ccc(C(=O)NC2CC2NC(c2cc(C3(C)CC3)n[nH]2)=O)[nH]1 c1(C(N2CC(NC(CC(C)F)=O)C(S(C)(=O)=O)C2)=O)ccc2c(c1)NC(=O)C2 N1(C(C(C2CCN(C(C3CCC4(CCC4)C3)=O)CC2)C)=O)CC(O)CC(C)(C)C1 C12(NC(C3N(C)CC3)=O)CCCC1N(C(C1(Oc3ccccc3)CC1)=O)CCC2 N1(C(c2cc(OCC)ns2)C(=O)NC2COC2)CCC(S(=O)(=O)NC)C1 c1(C(=O)NC2CC(CC(=O)NCC3C(C)(C)COC3)C2)ccc2cc[nH]c2c1 c1(NC(Cn2cc(-c3cc(OC)c(C)cc3)nn2)=O)c(CO)nn2c1CCC2 N1(C(c2nc(CC)oc2)=O)CC(NC(c2csc(C3CC3)n2)=O)CCC1C Cc1cc(F)c(C(=O)Nc2c[nH]nc2C(=O)Nc2cc3ccccc3[nH]2)cc1Br c1(NC(=O)NCC2CC(C)(C)C23CC3)nc2ccc(Cl)cn2c1F CC(CC(=O)NCC(O)CNC(C1(O)COC1)=O)C(F)(F)F c1(-c2cccc(CC)c2)cnc2ncc(C(=O)NC(C)C3CC3)n2c1 C(C(=O)N1CCC(C)C1c1cn(CCCOC2CCC2)nn1)(C(C)C)SC CCCC(C#N)C(=O)N1CCN(C2COCC2NC(=O)Cn2nnc(=O)[nH]2)CC1 C1(CNCC2(CO)C(C)C2)CCCCS1.c12nnnn1C2NC(=O)OC(C)(C)C Cn1cc(C(N2CC3CC(NC(=O)COC4CC4)C2C3)=O)c(=O)c2c1CCCC2 c1(OC)ccccc1C1(CNC2CCCN(C(c3ccco3)=O)C2)CC1 N1(C(C(=O)NCC(C)C)CC2CCCC2)CCCC(CC(F)F)(CO)C1 N1(C(CC(CC(C)C)C)=O)CCOC2(CCN(C(=O)C(C)(C)CO)C2)C1 C1(C(N2CCN(C(CC(C)OC)=O)CC(C)(F)C2)=O)=CN2C(=CC(F)=C1)N=CC=C2 C1(COC)CC2(CCC2)CN1C(CCC1CC1C)C(=O)NC1CCC1 C1(NC(c2ccc(CNC(COCCOCC)=O)o2)=O)CCCC2(CCC2)C1 c1(CSCCOC(=O)CC2CCCC2)c[nH]c2ccccc12 N1(C(C2C(C(C)C)(CC)C2)=O)CC2CCCC(C1)N2C(c1coc(C)n1)=O C1(COC)CN(C(c2cccc(O)c2C)=O)CCN1C(c1cncc(C)c1)=O C12(NC(C(C)N(CC)CC)=O)CCC(CC1)N(C(C1C(C)C1C)=O)C2 C1(NC(C=CC(CC)C)=O)CC1C1CN(C(=O)CCCC(=O)N(C)C)C1 S(=O)(=O)(CCC(=O)NCC1CCCN1C(=O)C=Cc1ccnn1C)NC c1(C(N(CCOCCNC(C(CC)C#N)=O)C)=O)ccnc2c1nnn2C N1(CC(N2CCCCC(CNC(=O)CC3CCCOC3)C2)=O)Cc2ccccc2C1 C1(C(=O)NC(C2CN(C(c3cnc(O)s3)=O)C2)C)CNC(=O)CC1C C1(C(N(C(CN(C(c2c(C)ccs2)=O)C)C)C)=O)COC2(CCC2)C1 c1(CC(=O)NCCN(C(c2cn(CC(N)=O)nc2)=O)C2CC2)ccc(O)c(F)c1 c1(CCNCc2cc(OC)cc(Cl)c2)cc(C#N)ccc1F C1(NC(CCCOC(C)=O)=O)CCCCN(C(=O)Cc2cc(F)ccc2C)C1 C1(NC(C(CCC)(C)CC)=O)CCC2(CCN(C(=O)Cc3nonc3C)C2)C1 c1(C(N(C2CCCCN(C(C3(C)CCC3)=O)C2)C)=O)ccc2nc(O)sc2c1 CC1(C)C(C(N2CC3CC2CN3C2CC2)=O)CCN1C(c1cccnc1)=O Cc1cc(Cl)ccc1OCC(=O)NC1CC(C)(NC(C2CC2C(F)(F)F)=O)C1 C1(C(N2CCOCC(C)(CNC(C3CC(=C)C3)=O)C2)=O)Cn2c(C)nnc2CN1C C1(C(=O)NC(C2CN(C(CCC(=O)NCCC)=O)C2)C)CC12CCCCC2 N1(C(CCOCCOC)=O)CC(CN(C)C(c2csnc2Cl)=O)C2(CC2)C1 C1(NC(CCOC)=O)CC2CN(C(c3cnc4cc(C)ccn34)=O)CCN2C1=O c1(C(=O)NCC2C(NC(C(C)N(C(C)=O)C)=O)C2)cc2cc(F)ccc2[nH]1 c1(C(=O)NC2CCN(C(c3ccco3)=O)CC2O)nc2ncccn2n1 CC1CN(C(=O)CN(CC(C)N(C)C)C)CC1(C)C(=O)N(CCO)CCO C12(N(C3CCN(CC)C3)C(=O)C(c3ccccc3)OC)CCC(NC(C)=O)(C1)OC2 N1(C(CC2C(C)=NNC2=O)=O)Cc2[nH]nc(C(=O)NC(c3cnn(C)c3)C)c2C1 c1(C(=O)NC(C(=O)NCc2cc(C)nc(O)c2)CN(C)C)cccc(C#N)c1C C1(C(N2CCC(CNC(C3(CCC)CC3)=O)C(C)C2)=O)CCC2(CC1)OCCO2 Cc1cnc2c(C(N3CC4CC4(C(=O)Nc4cccnc4I)C3)=O)cnn2c1 C#Cc1cccc(C(=O)NC2CCC2NC(=O)C(C)CC(N)=O)c1F Cn1nc(C(N2CCC3(NC(=O)Cc4cnc[nH]4)CCCC23)=O)c2c1CCSC2 c1(NC(C2CCCC(NC(c3c(F)cncc3F)=O)C2)=O)cncc(F)c1I C(=O)(C1=CNS(=O)(=O)N=C1C)N1CCCCCC(NC(CCCOC(C)=O)=O)C1 O=C1CN(CC2CCN(S(=O)(=O)C3CC3)CC2)C(=O)N1CCSc1ccco1 C1(CC)CN2CCCC2CN1C(=O)NCCN1CCCC(n2ccnc2)C1 n1(CC)ccc(C(N2CCCCC(NC(C3CCOC(=O)N3)=O)C2)=O)cc1=O C(=O)(C1=CS(=O)(=O)CCC1)NC1(COC)CN(C(=O)CC2CC(O)C23CCC3)C1 CC1(CNC(C2CC23CC(O)C3)=O)CCN(C(C2(N3CCCC3)CCC2)=O)C1 C1(C(N(CCCNC(C2CCCOC2)=O)C)=O)C2CCC1(c1cncs1)C2 c1(CC(C(=O)NC2CN(C(C(C)(C)OC)=O)CC2O)O)ccc(OC)cc1 N1(C(C2CCCN(C(c3sccc3I)=O)CC2)=O)CC2CCCCC2C1 c1(OC)ccc(C(C)NC(=O)NC(C)C(O)C(=O)OC(C)(C)C)c(F)c1 c1(N2CCC(COC)(OC)C2)ccc(S(=O)(=O)NCCc2ncnn2C)cc1Cl CCC(C)CCC(=O)NC(C)CCCCNC(=O)CN(C1CCCC1)C C1(O)(C(C)(C)C(=O)NCC2CCN2C(c2ccc(F)o2)=O)CCCCC1 N1(c2ncc(C)cn2)CC2(CC2)CC1CNC(=O)Cc1cnoc1 C1(C(=O)NC2(CCNC(C(CC)(C)CO)=O)CCC2)CCc2nncn2C1 CCCCCC(C)(C)C(=O)NC1CCCC1NC(c1oc(C(F)(F)F)nc1C)=O Cc1nc(SC(C)C)cc(N2CC3C(CNC(=O)COC4CCCCC4)C3C2)n1 C1(NC(c2cncc(N)c2)=O)CC(NC(=O)Cc2cnns2)C12CCC2 C(=O)(CS(=O)CCC(F)(F)F)N1C2C(CNC(C(COC)C)=O)C(C2)C1 C1(Cl)(C(=O)NC(c2ccc(C)c(Br)c2)C)C2CCCC(=O)C12 c1(C(N2CCC(N(C(=O)CC3CC(C)(C)C3)C)C2)=O)c[nH]c(=O)c(C(F)(F)F)c1 c1(CC(=O)N(CCCNC(C2CC3CC3C2)=O)C)ccc(C#N)cc1F C1(C(=O)NC(CNC(c2cnccn2)=O)C2CCC2)CC2CCC1O2 CC(C)CCCCC(=O)NCCC1CN(C(c2scnc2C(C)C)=O)CCO1 c1(C(c2nnnn2C2CCC2)NC2C(Br)C2)cc2ccccc2o1 Cc1occc1CC(=O)NCC(CCn1cccn1)NC(=O)CO N1(C(C2OCCN(C(CC(C)C3CC3)=O)C2)=O)CC2(CCC2O)C1 N1(C(CC(C)(C)C#N)=O)CCCC2(NC(=O)CCCCO)CC2C1 C1(C(=O)NC2CN(C(CCCOC(C)=O)=O)C(C)(C)C2)CCn2c(O)nnc2C1 c1(OC)ccc(C(N2CCCC2CN(C)C(c2conc2C(C)C)=O)=O)cc1O N1(C(C)(C)C(=O)NCCC2CN(C(C3(O)CC3)=O)CCO2)CCC(O)CC1 C12(c3nc(C(C)C)nn3-c3cccc(F)c3)CCC(c3ccccc3)(CC1)C2 CC1C(NC(=O)CCCCN2CCCC2)CCCN1C(=O)CSC(=N)N C12(C(N3CC(C(C)NC(=O)CC4CC5(CCC5)CO4)C3)=O)CCC(C1)C(C)(C)O2 Cc1ccccc1CN(C)CC1CN(C(c2ccc(=O)oc2)=O)C1.c1(C(=O)O)ccc[nH]1 c1(C(C)(C)C)conc1C(N1CCC1CNC(=O)C=CBr)=O C(=O)(CCCS(C)(=O)=O)NCCCCCNC(C1(C)CCN(C)CC1)=O c1(C(N2C(C(=O)NC3CC(SC)C3)CCC2)=O)cc(C)sc1N C12(NC(=O)CSCC(F)(F)F)CC(CO)(C1)OC21CN(C(=O)C2=CCSC2)C1 C1(C(=O)OC)CC(NCc2ccc(CCl)cc2)CCO1.c1(C=O)cccc(OCF)c1 O=C1CC(NC(=O)C(CCC2CCC2)NC(c2csc(Cl)c2)=O)C(=O)N1 c1(C(=O)N(c2ccc(I)c(C(=O)O)c2)CCO)cc(S(=O)(=O)N2CCOCC2)c[nH]1 S(=O)(=O)(c1cc(Cl)cc(Cl)c1)N1CC(CNC(c2cc(Cl)nc3n[nH]cc23)=O)C1 C1(CC(=O)N(CCNC(CCNS(CC)(=O)=O)=O)CC2CC2)CCC(C2CC2)O1 N1(C(C2(c3cnccn3)CC2)=O)CC(n2cc(NCCSCC)nn2)C(C)C1 CC(C)(C#N)CCC(=O)N1CCC(CF)(NC(c2csc3c2CCCC3)=O)C1 c1(C(=O)NCC2(O)CN(Cc3cccc(C)n3)C2)c(C)cc(Br)cc1Cl c1(C(N2CCC(C)(C(N3CCC(C#C)CC3)=O)C2)=O)n[nH]c2c1CCCC2 c1(C(=O)NC2C(C)CCN(C(=O)CC3CC4(CC4)CO3)C2)ncc([N+](=O)[O-])n1C N1(C(c2c(C)n(CCO)cc2)=O)CCC2CC1CN2C(=O)CCP(C)(C)=O C(N=c1[nH]c(C)cc(=NCCCCc2ncc[nH]2)[nH]1)c1c(C)cc(C)cc1 CCC(CC)C(F)C(=O)NC1CC(NC(c2coc3c2COC3)=O)C1 C1(c2c(OCC)scc2)NC(=S)N(CC(C)C)C(C(C)(C)C)=C1C(=O)OC c1(OC)c(CC(N2CCCC(O)(CNC(=O)CC(C)(C)O)C2)=O)cccc1C#N c1(C(C(=O)NCc2ccc(F)cc2)N(C)Cc2cn(C)nn2)cc(Cl)cc(Br)c1 c1(CNC2CC(C(=O)Nc3ncc[nH]3)C2)cc2c(cn1)OCCC2 c1(SCCC(=O)NCCCCCCNC(C(COC)C)=O)ccc([N+](=O)[O-])cc1 C1(NC(C2CCC3CC3C2)=O)CC2CN(C(=O)COc3ccsn3)CC2C1 N1(C(c2cc([N+](=O)[O-])on2)C(=O)NCC(C)C)CCC2(CCCCC2)CC1 n1(CC(N2C(C)CC(NC(=O)Cn3cnnc3)C2)=O)ccc2cc(F)ccc12 c1(OC)cc(CC(=O)NC23CC(NC(=O)CC4(C)CCOC4)(C2)C3)ccc1O c1(NC(=O)NCCOCCOCC#C)ccc(Br)cc1Br c1(C(=O)NC(C2(CNC(c3cnc(C)o3)=O)CC2)C)cnc2n1CCCC2 C1(C(=O)NCCC(C)N2CCC2)N(C(=O)CCc2cscn2)CC12CCCC2 CC1C2CCC(C2)C1CO.C1CCCCC(=O)N2CCC(C2)C(=O)N1C C(=O)(C(C)(C)C(C)(C)O)N1CCCC(NC(C(C)(C)CC2CC2)=O)CC1 Cc1cc(O)nnc1C(N1CCCC1C(=O)OCC1CC2(C1)CC(C)C2)=O CC1CCN(CC(N2CC3CC3(CNC(=O)Cc3cc(C(C)C)n[nH]3)C2)=O)CC1 c1(SC)ncc(Br)c(=NC2CC(CC(N3CCCCC3C)=O)C2)[nH]1 c1(C(=O)NCC(c2ccccc2)N(C(C)=O)C)nncn1C1CC1 c12nnc(COCC)n1CNC2.C1(CC)CN(Cc2cnc(C)nc2)CCO1 C1(NC(C2C=C(C)CS2)=O)CC(CNC(=O)C=CC2CCCO2)C1(C)C Cc1c(C(N2CCSCC2C(=O)Nc2ncc(CO)cc2Br)=O)cccc1I Cc1nnc(CN2CCC(C(F)(F)F)C2C2CC2)n1C S1(=O)(=O)c2ccc(c(Cl)c2)CN1CC.c1(OCC)ccccc1.N(C1CC1)C(C)C1CC1 CC#CCC(C(=O)N1CCC(N2CC(O)C2)C1)NC(C1CCN(CCC)CC1)=O c1(C(=O)NCC(F)(F)F)cc(F)cs1.n1(CC(=O)N2C3CC3C2)cccn1 c1(C(N2CCC(NC(c3c(C)cc(F)cc3)=O)(CF)C2)=O)n[nH]c2c1COCC2 N(S(=O)(=O)N(C)C)c1cn(CCN(C)C(c2c(C(=O)N(C)C)cnn2C)=O)nn1 C1(C(N(CC(C)CNC(C2CCC(=O)O2)=O)C)=O)CCn2c(O)nnc2C1 C1(C(N2C(C)C(NC(c3occc3Cl)=O)CC2)=O)CCc2nnnn2C1 N1(C(C)=O)CCC(C)(C(=O)NCC#CCNC(c2cc[nH]n2)=O)C1 CC(C)C(CC(=O)NCCC(C)N(C)C(c1cnc(S(C)(=O)=O)s1)=O)C(C)C Cc1[nH]c(C#N)cc1C(N1CC(C(F)C(=O)NCc2ccc(CO)cc2)C1)=O c1(CC(=O)N(CC(CC)NC(=O)Cc2cn[nH]c2)C)coc(C(F)F)n1 N1(CCCCCCC)CC2CN(C(c3cccc(F)c3C)=O)CC2C1 N1(C(C2(C)CCOC2)=O)CCCCC(C(=O)NCc2nccs2)C1 C1(NC(C=CC(CC)C)=O)CC2CCC1N2C(c1ccc(OCC)c(O)c1)=O C(CC(=O)N1CCC12CC(O)C2)(C(F)(F)F)NC(C1(C#C)CCCCC1)=O N1(C(C=CC(CC)C)=O)CCC=C(C(=O)NCC2CC2[N+](=O)[O-])C1 C(CCCCC(=O)NC(CC(C)C)C(=O)NCC1CN(C)C(=O)O1)=CC Cc1ccnc(C(=O)NC(CO)C(C)NC(C2CC23CCOCC3)=O)c1F C1(CC(=O)N(CC#C)CCF)N(C(=O)CN2CC3CC3C2)CCC1(C)C C1(CNC(COCC(=O)NC)=O)CCCCC1C(N1CC(c2cc[nH]n2)C1)=O N1(C(CCC(C)NC(=O)C(c2ccnn2C)O)=O)CCOCC(O)C1 C#Cc1ccc(C(=O)NC(C)C(C)NC(c2c[nH]c3ccncc23)=O)c(F)c1Cl Cc1cc([N+](=O)[O-])cc(C(=O)NCC2CN(C(c3cnns3)=O)CCCO2)c1Cl Cc1ccc(C(=O)N(C)CC2CCCN(C(C3(C)CC4CC4C3)=O)C2)c(N)c1F C1(CCC)CCCC1NC(=O)CC=CCNC(c1sccc1C)=O C(CCCCCNC1C(C#N)C1(C)C)N(C(CN(C)Cc1ccccc1Cl)=O)C Cc1csc(CC(=O)NC2CCC(CNC(c3n[nH]cc3F)=O)C2)c1 n1(C(C)C)cnnc1CC(=O)NCC1CCCN1C(c1cnn(C(F)(F)F)c1)=O Cc1cnc(C(N2CCCCC(N(C(=O)C3=CCCC3C)C)C2)=O)c(C)c1 Cc1ccc(-c2sccc2C(=O)NCCC(C)N(C)C(c2cc[nH]n2)=O)s1 C1(CNC(=O)CC2CSCCS2)C2CCCC1N(C(C1CC13CCC3)=O)C2 C=C(C)C1CN(C(=O)CC(c2cccc(F)c2)C)CCO1 c1(C(=O)NN2CC(C(=O)NC)CC2(C)C)ccnc2cc(C(=O)O)sc12 c1(C(N(CC(O)CNC(=O)CC2CC2)C)=O)ccc(NC(c2ncccn2)=O)cc1 c1(NC(C(CC(F)F)NC(C(CCC)OCC)=O)=O)cc(C#N)ccc1C c1(C2N(C(CC(=O)NCCC)Cc3ccc(Br)cc3)CCC2)cccc(C)c1C N1(C(c2cn(C)nc2I)C(=O)NC2CC2)CCc2cc(F)cc(Cl)c2C1 C1(NC(C2CCC(C(=O)NC3CC(OCC)C3)C2)=O)(CO)C2CCCC12.C=O C1(NC(NCC(C(F)(F)F)Cl)=NCc2ccco2)CCC2(C1)OCCO2 c1(C(=O)NC23C(CN(C(COCC(=O)OC)=O)C2)C3)cccc2c(C)ccnc12 c12ccc(nc1)OC(=O)C(=O)N2C1CCNC1=O.C(CF)OC N1(C(CC2(CSC)CC2)=O)CCC2(CC1)CN(C(c1ncccc1C(C)=O)=O)C2 FC1(F)C2CC(NCC3CC(n4cccn4)C3)CC12 n1(C(CC)C)nc(C2CC2)nc1-c1cc(Cl)n(C)n1 C(=O)(CCCCCO)N(C)CC1N(C(C(C)NC(C)=O)=O)CCC1 CCC(C(=O)OCC(=O)NC(=O)NCC)c1ccccc1 N1(C(C2(COC)CC2)=O)CCCC(O)(CNC(c2ccnc(OC)c2)=O)CC1 CCCCC(O)C(C)C(=O)N1CCC2(C)CC1(C(=O)NCC1(OC(C)=O)CCC1)C2 c1(CC)ncccc1C(=O)N(C1CCC(NC(c2cc(C)n(C(F)F)n2)=O)C1)C CC1(CC(=O)NCC(CO)NC(c2ccccc2)=O)CC1(F)F c1(C(=O)NC2C(NC(c3n[nH]c4c3COCC4)=O)C2)c[nH]c2nccc(Cl)c12 C(=O)(C(F)(F)CCn1cc(CCO)nn1)NC(C)CCN(C)C S(=O)(=O)(c1ccc(C#N)c(NCc2n[nH]c(=N)s2)c1)N1CCC(C)(C)C1 C(=O)(C1=NN(C)C(=O)CC1)N1CC(CC(C)NC(c2ccc3nc[nH]c3c2)=O)C1 CC(C)(CC(F)C(=O)NC1CCCCC1)NC(=O)CCc1cscn1 c1(C(=O)OC)ccnc(N2CC3(CN(C(C4(O)CCOC4)=O)C3)C2)c1[N+](=O)[O-] C1(C(=O)NCC2CCC(NC(c3nnc(C(C)C)s3)=O)C2)CC12CCSCC2 C=CCCCC(C(=O)NCC1(O)CCOC1)NC(=O)CC1CCOC1C C1(C(N(CCNC(C2CC(C)(O)C2)=O)CC2CC2)=O)CCN(C(=O)C2CC2)CC1 c1(C(=O)NCC(CNC(C(C=C=C)C)=O)OC)n[nH]c(CC)c1[N+](=O)[O-] C1(CNC(CC2CC(=C)C2)=O)CCC(C)(C)CN1C(=O)CN1CCCC1C CC(CCC(=O)N1CCC2CC12)NC(=O)CC1CCCN(C)C1 C(C(C(=O)N1CC2CCC(C1)C2O)C(C)(C)C)NC(c1c(C)occ1)=O C1(O)(CNC(C(C)n2cccn2)=O)CCN(C(c2cnc(C(F)F)nc2)=O)C1 C1(NC(C2CCN(C(C)=O)C2)=O)CCN(C(c2sccc2Cl)=O)C1(C)C C1(NC(CN(C(=O)C=Cc2cccc(C)c2)CCC)=O)CN(C)C(=O)C12CC2 C1(CC(=O)NCC(CNC(c2c(C)n(C)cc2)=O)(C)C)CC(F)(F)C1(F)F C(C(CNC(C1CCCOC1)=O)C(F)(F)F)NC(c1cc(C)sc1Cl)=O C1(C(=O)NC(CNC(C2CN(C(C)C)C(=O)CC2)=O)C)CCCCC1P(C)(C)=O N1(C(C(C)Oc2cccc(C)c2)=O)CC2(C)CN(C(C3CC3(F)Cl)=O)CC2(C)C1 N1(Cn2cc(Br)cn2)CCN(CC(=O)N(C2CCCCC2)CCN2CCCC2)CC1 Cc1cc(=O)n(-c2noc(-c3ccc(F)cc3Cl)n2)c2ccccc12 C(N=c1nc2ncn(C)c2c(NCC2CCS(=O)(=O)N2C)[nH]1)c1ncn(C)n1 Cc1ccc(O)c(CC(=O)NCC2CCC2NC(=O)C2CC2)c1 N1(C(CN(C)CC)=O)CCC(C(C)NC(c2ccc(COC)o2)=O)C1 C(=O)(C1=NOC(CC2(O)COC2)C1)NC1CC(NC(C2CC23CC3)=O)C1 C#Cc1cnn(CC(N2CC(O)(C(C)(C)CNC(=O)CCF)C2)=O)c1 c1(OC)ccc(-c2cn(C3CN(C(c4cc(C#N)nn4C)=O)C3)nn2)c(F)c1 CC(C)CCC(C(=O)NCCn1ccnn1)NC(C1CC12CCCCC2)=O c1(C(C(=O)NC2CCOC2)N(C)CCC2(C)CC2)cn(C)nn1 C12(CNC(c3scc(C)c3)=O)CCC(CN(C(c3c(C)cnn3C)=O)C1)C2 CC(CCC(F)(F)F)NC(C1COCCC1NC(c1cccc[n+]1[O-])=O)=O Cc1ccc(C(C)C(=O)NCCC2(NC(c3ccncc3)=O)CCC2)o1 C(=O)(C(Cc1ccco1)NC(=O)CCC1CCCO1)NCC(C)CF N1(C(C2CCCC(=O)CC2)=O)CCC(C2CN(C(=O)CCc3cc[nH]n3)C2)CC1 c1(N(c2ccccc2)C)nc(=NCC2CC3(C2)CC(C)(C)C3)[nH]c2c1SCC2 C(=O)(CC(F)(F)C(C)C)NC1CC2(C(NC(C(CC)(C)C)=O)C2)C1 C(C)(C)(CC(=O)N(CCNC(c1cc(C)c(C)o1)=O)CCc1ccccc1)OC C=CCC(CC(C)C)C(=O)NC(C)(C)CN(C(=O)C(=O)Nc1cccc(C)c1)C CCCN=C(NCc1ccsc1)NCC1(Cl)CCOCC1 Cc1nc(F)ccc1NC(=O)CCCCN(C)C(C1CC(C)C1)=O C(C)(C)(C(C)CC(=O)NCc1ccnn1CN(C)C)NC(CCNC(COC)=O)=O CCCC(C(=O)N1CCCN(C(=O)Cc2csc(Cl)n2)CC1C(C)C)C(C)C C1(O)(CNC(CN(CCC#C)C)=O)CC(NC(=O)C(F)=C(C)C2CC2)C1 CCC(F)(F)CC(=O)N1CCC(C)C(NC(c2cnc(COC)s2)=O)C1 CC(CCCCNC(c1nn(C(C)(C)C)cc1Br)=O)NC(c1ccon1)=O C(C(CO)CC(C)C)NC(C1C(CC)CCN1C(=O)CSCC(=O)OC)=O Cc1c(N(C(=O)CCC(N)=O)C)cc(-c2ccccc2)n1C1CC(C(F)(F)F)C1 c1(-c2n(C(CC)C)nc(-c3cccs3)n2)nccc(C)c1Br c1(NCCC(=O)NC)cc(NC2CC3CC3C2)nc(C)n1 c1(C(C)C)nn(C)cc1C(=O)NCC(C(C)C)NC(c1occc1C1CC1)=O c1(SCC(=O)NCC(CC)C(=O)CCn2ccnc2C)nnnn1C1CCCCC1 CC1(C)CCCC(N2CC(=O)N(CC(CC(F)(F)F)C3CCCO3)C2=O)C1 c1(CC(=O)NC2CC(C)(NC(C3CC=CC3)=O)C2)noc2ccccc12 C1(C(N(CCCNC(=O)CCC2CCC(=O)N2)C)=O)C2CC3C(C2)C13 C1(CN(C(C(=O)NCCC)=O)CCCO)CCCN2CCCCC12 N1(C(c2cn(CC)nc2)=O)CC(C(N2CCSCC2C2CC2)=O)C(C)C1 C=CC(C)CC(=O)N1C(C(=O)Nc2cccc(N(C)C)c2)CCC1C1CC1 C(=O)(CCCC(=O)NC(C)C(C)NC(c1cnc(N)cn1)=O)NCCC N1(C(C2CCC(C(=O)OC)C2)=O)CC=C(C(=O)N2CCCC(OCC)C2)C1 N1(CC(COC(COC)C)O)CC(NC(c2c(Cl)csc2Cl)=O)CCC1C C(=O)(C(C)(C)C(F)(F)F)N1CC2(CC(CC(=O)NC3CN(C(C)C)CC3C)C2)C1 C(=O)(C1CCCc2n[nH]cc21)NC1C=CCN(C(c2n(CC)ccn2)=O)C1 N1(C(COCC)=O)CC(CNC(c2cccc(F)c2SC)=O)CC1(C)C C(CNC(=O)CCc1scnc1C)(CC(=O)N1CC(C)C1(C)C)OC C=CCC(C)(C)CC(=O)N1CCC(C(=O)N(C(C)CCO)C)C12CC2 N1(C(C(=O)NCCNC(C)=O)=O)CCCC(C)(CNC(=O)CC(C)(C)F)C1 N1(Cc2cnc(OC)nc2)CCC(=O)N(CC2COC3(CCC3)C2)C1=O c1(C(=O)NC2C(C)N(C(C3CCNC3=O)=O)CCC2)nccc2ccncc12 c1(OC)ccc(C)c(OC)c1C(=O)NCc1c(C(F)(F)F)cccc1F C1(NC(C=CC2CCN(C(CC(=O)N(C)C)=O)CC2)=O)CCN(C)CC1C#N N1(C(C(CSC)(C)C)=O)CCC2CN(C(=O)CCCC(C)C)C2C1 C1(NC(=NCC)NCCC2CCCN2C)CCc2nnc(N(C)C)n2C1 c12ccccc1NC2.C1(C(=O)NCC(CO)SCC)CCOC(C)C1 C1(NC(C=CCN(C(Cc2ncc(CC)[nH]2)=O)C)=O)CC2CCC1O2 n1(CC(=O)NC(Cn2cccn2)C(=O)NCC2(O)CCC2)c(O)nnc1O C(CS(=O)(=O)c1ccccn1)N(C(c1cc(OC)c(OC)cc1Br)=O)CC c1(C(=O)NC2C=CC(CNC(Cc3c(C)noc3Cl)=O)C2)ccc(O)c(F)c1 c1(CC)ccc(CCNC(C2C=CCC2)=O)cc1.c12n[nH]cc1C(=O)NC2 c1(NC(N2CC3(CCCC3)C2c2ccco2)=O)ccc2ccnn2c1 C1(NCc2c(N3CCCC3)sc(C(=O)OCC)c2C)CC2(CCOC2)C1 Cc1cc(C(=O)NC2CCC(C(=O)NC3(Cc4ccccc4)CC3)C2)cc(C)n1 N1(CC)CC(C(N2CC(O)(CNC(=O)C(C)CN(C)C)C2)=O)NC1=O Cc1cc(S(N)(=O)=O)sc1C(=O)N(C(CC(=O)O)C(=O)O)C.c12cn(nn1)CC2 C(=O)(C#CC1CCOC1)N1CC(N(C(c2c(SC)snn2)=O)C)C(O)CC1 N1(C(CCn2ccc(C(=O)OC)n2)=O)C2CCC1C(NC(C1CCCO1)=O)C2 C1(CNC(=O)NCC(C(F)F)N2CCOCC2)CC12CCOCC2 C1(NC(c2cc(CC)[nH]n2)=O)CC2CN(C(c3csc(CO)n3)=O)CC2C1 c1(CCC)onc(C)c1C(=O)NC1CC1CNC(C1(C)CC2CC2C1)=O C1(CC)(CC)CCC(NC(=NCc2ccco2)NCC2CCN2C)CC1 O=C(CS(=O)(=O)c1cccc(F)c1)NCC1(CCNC(=O)COc2ccon2)CC1 N1(C(CC2(C)CCCO2)=O)CCC2CCN(C(=O)C=CI)CC2C1 N1(C(c2csc(C#N)c2)C(=O)NCCSC)CCCC12CCS(=O)(=O)CC2 c1(-c2cc(C(=O)NCCCN(C(C3(CC)CCC3)=O)C)on2)cccc(F)c1 C1(C(=O)NC(C(C)C)C)(NC(=O)CCSC(F)(F)F)CCOCC1 C(=O)(C1CCCc2n[nH]cc21)N1C(CNC(c2ccc(C(F)F)cc2)=O)CC1 c1(OC)ncc(NC(C2(C)CCCN2C(C2CNC(=O)C2)=O)=O)cc1Br c1(C(=O)NC(C2CC3CCC2C3)CC)ccc(F)cc1Br CC(CC(=O)NC1(CN(C(=O)CC2NC(=O)CNC2=O)C)CC1)C(C)(C)C N1(C(C)C)CC(NC(N2CCN(CC(C)O)C(CCO)C2)=O)CCC1=O c1(C(N2C(CNC(=O)C=Cc3cccnc3)CCC2)=O)cccn2nccc12 c1(C(N(C2CCN(CCCN(S(C)(=O)=O)CC)C2)CCC)=O)c(C)[nH]c(C(C)=O)c1C CCCS(=O)(=O)C(C)C(=O)NCCCNC(=O)Cc1noc2ccc(O)cc12 C(CC(C)(C)CC(=O)NCC1(NC(c2nc(Cl)c(Cl)s2)=O)CCOC1)OC C(CC(=O)N1C2CCC1C(CNC(=O)C=CC(F)(F)F)C2)(C(F)(F)F)OC C(CC)(C(=O)N1CC(O)(CCNC(=O)C(C)OC)C1)=CCCC C1(OC)CCN(C(=O)NC2(C(=O)OC)CC(=O)C2)CC1(C)C C(=O)(C1=C(Cl)CCC1)N(CCCNC(c1cnc2n1CCS2)=O)CCO c1(C(=O)NC2C(NC(=O)CSCC3CCCCO3)CC2)cccc([N+](=O)[O-])c1Cl C(C)(CO)(C(=O)NCC12CC(NC(=O)CC3SC(=N)NC3=O)(C1)C2)OC C1(C(N)=O)CCN(C(=NCc2ccco2)NCC23CC4CC2C3C4)C1 C=C(C)CC(C(=O)N1CCN(N(C(=O)C(C)n2cnnn2)C)CC1)OCC1CC1 N1(C(=O)C(c2ccccc2F)n2cnnc2)CCC(=C(F)F)CC1 Cc1cc(C)c(C(N2CCCC2C2CCN(C(=O)CC3(O)CCCC3)C2)=O)o1 N1(C(COCCCC)=O)CCCC2CCN(C(c3nnsc3C)=O)CC12 O=C(CCC(F)F)N1CCN(C2CCC(NC(=O)C(F)OC(F)(F)F)CC2)CC1 C(C(=O)NC(C)C(C)C(=O)Nc1cc(O)ccc1C)(C(C)(C)C)OC C12(NC(CCC)=O)CC(C)(C1)OC21CCN(C(c2sc([N+](=O)[O-])cc2Cl)=O)CC1 C1(NC(C(CSC)C)=O)CCC2(CCN(C(=O)CN3CCCC3C)C2)C1 O=C(C1=CCCN(C(c2ccc3occc3c2)=O)C1)NC1=C(O)OC=CC(Cl)=C1 C1(CNC(=O)CC2CC3(CC3)C2)CN(C(c2ccnn2CC2CC2)=O)CCCO1 CCCC(C(=O)N(CC(C)CC)C(C)C)NC(c1ccc(F)cc1)=O C(=O)(C1=CCCC1C)N1CCC(N(CC(C)C)C(c2c(C)cns2)=O)CC1 CC(CCNC(=O)C(CCC1CCC1)NC(=O)CN(C)C)CC(C)(C)C C(=O)(CC1=CSC2=NCCN12)N1CCC(NC(C2N(C(C)=O)CCCC2)=O)CC1 c1(C(N(C2CN(C(C(N3CCOCC3)C)=O)C2)C)=O)ccc(Cn2ccnc2)o1 C1(C(=O)NCCNC(c2c(C#C)ccc(F)c2)=O)Cc2nn[nH]c2C(C)C1 N1(C(C2N(CC)CCC2)=O)CCC2(CCCN(Cc3cc(F)ccc3C)C2)C1 C1(C)(C(=O)Nc2cn(CC)nc2)CCCN(Cc2ccc(OC)nc2Cl)C1 N1(C(CN(C)C)=O)CCCCC1CCNC(=O)C(O)COCc1ccccc1 C1(S(C)(=O)=O)(C(N2CC(C(C)NC(=O)CC3CCCCC3F)C2)=O)CCCC1 CC1(C)C(C(=O)NC2CCN(C(=O)Cc3cncnc3)C23CC3)CCS1(=O)=O C1(O)(C(=O)NCC2CN(CC3CCC3)C2)CC(CNC(=O)CCC2CC2)C1 n1(CC(=O)NC2CN(C(CC(CC=C)(C)C)=O)CC2F)c(=O)oc2ccccc12 C12(NC(CC3C(C)C3)=O)CCCCC1N(C(c1nc3ccccc3o1)=O)CC2 c1(OC)cc(C(=O)NC2CCC(C(=O)NCC3CCCOC3)C2)cnc1Cl c1(C(N2C(CN(C(C(CCC)F)=O)CC)CCC2)=O)ccn2ccnc2c1 n1(CCC#C)c(N(C)CC2CN3CCC2CC3)nnc1C1CCCc2c[nH]nc21 C=C(C)CC(=O)NCc1ccc(C(N2CC(CC3CCC3)C2)=O)s1 C=C1CC2CCC(C1)N2C(C1C2CCC(C2)C1NC(=O)CC1CCCC(=O)N1)=O N1(C(c2cc(C(C)C)no2)=O)CC2(CC2)CC1CNC(C1CCCO1)=O N1(C(CC(C2CC=C(C)CC2)C)=O)CC2CCC(CNC(=O)CCS(C)(=O)=O)(C2)C1 c1(C(C)CC(=O)NC(CO)C(C)NC(C2(CC3CC3)CCC2)=O)ccccc1F C1(C(N(CC(C)SC)C)=O)CCN(C(c2cc3n(n2)CCC3)=O)CCO1 C(=O)(CS(=O)(=O)C(C)(C)C)NCC1CN(C(CCSCCCC)=O)C(C)(C)C1 c1(CC)cccc(N(C(=O)C(CC2CC2)NC(=O)CC2(C#N)CC2)C)c1 C1(NC(c2cc(C)oc2C(F)(F)F)=O)CC2CC1N(C(=O)CCSC(F)(F)F)C2 N1(C(c2c(O)ccc(NC(=O)CN3CCC(O)C3)c2)=O)CCC2(CC1)OCCO2 CC1C(NC(c2c[nH]c(=N)o2)=O)CCCN1C(C1CCOC(C)(C)C1)=O Cc1ccc2c(=NCCc3c[nH]c4ccccc34)[nH]c(N3CCOCC3)nc2c1 Cc1cn(C(C)C)cc1C(N1CCCCC1CNC(c1ccccc1F)=O)=O C1(C(=O)NC2C3CN(C(c4c(C)n[nH]c4)=O)C2CC3)Cc2ccccc2S1 Cc1cc(C(=O)NC(C)CCCNC(=O)CN2CC(F)(F)C2)on1 c1(SC)ccc([N+](=O)[O-])c(C(=O)NC2CC(NC(=O)C(C)(C)c3cnsc3)C2)c1 C(C(C)C(=O)NOCC=CCC)NC(=O)C(COC)CC CC(C)CC(C(=O)C(=O)CCOC1CCC1)c1ccccc1.C1(CN)CC1N N1(C(c2cc(C)[nH]n2)=O)CCCCC(NC(=O)CSCCc2ccccc2)C1 C(CC(C)(C)C(=O)N1CCOC(CCNC(C2COCCO2)=O)C1)OC C1(NC(C)=O)CC(F)(F)CC1NC(c1c(C(=O)NCCOC(F)F)cccc1)=O CS(=O)CCCCC(=O)NCC1(NC(C2CCOC2(C)C)=O)CCCCCC1 C=C(C)C1OCCCC1C(N1CCN(C(c2coc(Cl)c2)=O)C2CCC12)=O Cc1c(CN2CCCC(C(=O)NC(c3ccccc3)C#N)C2)cccc1Br C1(C(=O)NC2CC(CCC(=O)N(C3CCC(C)C3)C)C2)C2CCCC(=O)C12 C12(C)C=C(C(=O)N3CCC(CC)(CC3)N1C(=O)CC)C2.C1(OCC)CCC1 n1(CCC)cc(Cl)c(C(=O)NCC2CC(NC(=O)CSc3ccc(C)cc3)C2)n1 N1(C(C(C)C2CC2)=O)CCN(C(=O)C(N2CCCCCC2)C)C(C)C1 C1(F)(CNC(c2c(CC)nco2)=O)COCCN(C(=O)CN2CCC(C)(O)C2)C1 N1(C(c2c(C)cno2)=O)CC2(CCC(CNC(C3CCC3)=O)O2)C1 N1(C(c2ccn(C)n2)=O)CC2CC(C1)N2C(c1ccc(C2CC2)o1)=O c1(C(N(CC(CC=C)NC(C2CC2c2ccccn2)=O)C)=O)cn(CC)nc1C C(C1c2ccccc2CN1C(C1C2CC3C(C2)C13)=O)NC(=O)CN1CCCC1CO C=C1CC2(C1)CC(C(=O)N(CCC)CCNC(=O)CC(C)COC)C2 c1(C(=O)NC2CN(C(C(C(C)C)NS(C)(=O)=O)=O)CC2O)cc2nc[nH]c2cn1 CC1Oc2ccccc2C1c1cc[nH]c(=N)c1C(N1CCCC(C2(CO)CC2)C1)=O c1(OC)cccc(C(=O)NC(C)(CSC)C(=O)NCC2CC2Cl)c1 CC1(C)CCC(CNC(C2CC3CCC(C2)C3)=O)N(c2ncnc3[nH]cnc23)C1 c1(C(=O)NC2CCC(CCNC(Cn3ncc(C)c3)=O)C2)nnc(O)nc1O C(=O)(C(CCNC(=O)C=Cc1ccncc1)OC)N(CC)CC c1(C(=O)NCC2(F)CCN(C(c3nn(C)c(O)c3)=O)C2)ccc2cccnc2n1 C(CCOC)(C(=O)N(CC(C)O)C)NC(c1c(CC)noc1)=O n1(CC)cc(C(=O)N(C2CC(NC(=O)CC3CC(O)C3(C)C)C2)C)c(C)n1 C1(C(=O)NCC2CCN(C(COCCSC)=O)C2)Cc2cc(C)ccc2S1 C(=O)(CC(F)(F)C(F)F)N(CCCCCCNC(=O)Cn1cc(C#N)cn1)C C1(NC(=O)C(=O)Nc2cccc(NC(C)=O)c2OC)CC2(COC)COC1C2 CC(N=c1[nH]c2c(c(=NC(C)c3cncs3)[nH]1)CSC2)c1cnc2n1CCCC2 C1(COC)(CNC(c2c[nH]nc2C2CCCO2)=O)CN(C(=O)CC2OCCC2C)C1 C(=O)(C#CC1(C)CCCO1)NC(CCC)C(O)C(=O)NC1CCC(C)CC1 c1(OC)nc(C)c(C(N2C(C(N3CCC(O)(C(F)(F)F)C3)=O)CCC2C)=O)s1 N1(C(C2C(C)C2)=O)CC(NC(c2cn3ccnc3s2)=O)CC12CCCOC2 C1(C(=O)NC(c2cccc(F)n2)C)CCN(C(c2cc(F)c[nH]2)=O)CC1 c1(C(N(C(C)CN(C)C(c2ccoc2Br)=O)C)=O)noc2c1CCCC2 Cc1nn(C)c(C)c1C(=O)NCCCC(C)NC(=O)CC1CC1(C)C C1(C(N(CCCN(C(CC2C(C)CCO2)=O)C)C)=O)CCc2nn[nH]c2C1 c12ccc(F)c(c1)C(=O)N2.c1(NC2CCN(S(C)(=O)=O)C2)ncc(Br)cn1 N1(C(c2cc(OC)ns2)=O)CC2CCCC2(C(N2CCN(C)C(C)C2)=O)C1 C1(CC)CN(C(=O)CCC=Cc2ccccc2)CC1NC(c1c[nH]c(=NC)o1)=O Cc1cc(C(C)NC(c2ncoc2SC2CC2)c2nnnn2-c2ccccc2)no1 c1(CNC(C2N(C(CC3(CC)CCC3)=O)CCC2C)=O)ccc(OC)c(O)c1 c1(CC(=O)NC(C23CC4CC(CC(C4)C2)C3)C(F)F)ccc2c(c1)CCCC2 N1(C(C(N2CCC(C)C2)=O)=O)CCN(C(C2C(F)(F)C23CCC3)=O)C2(CCC2)C1 c1(C(N2CCC(NC(CC=C)=O)(CF)C2)=O)cc(C)c(C)nn1 c1(C2CCCN(C(c3cc4ccsc4[nH]3)=O)C2)nc2ccc(F)cc2o1 c1(C(N2C3CC(NC(C(C)(C)OC)=O)CC2CC3)=O)oc2ccc(C)cc2c1C CC1CN(C(=O)C(C2CCCO2)Oc2ccccc2)CCN1C(c1ccncn1)=O c1(OC)nc(Nc2ncn(CCn3ccccc3=O)n2)nc2[nH]cnc12 c1(OC)c(C)cc(C(N2CCC(O)(CNC(C34CCC3C4)=O)C2)=O)cc1Cl c1(NCCCC2CCCC(=O)C2)ccc(S(=O)(=O)NC2CCCCC2)cc1F CCCC(CC(=O)NC1(C)CCC(NC(=O)CN(C)C2CC2)CC1)NC(C)=O c1(C(=O)NC2C(C)N(c3ncnn4cccc34)CC2)nc2ccc(Cl)nn2n1 c1(C(C(=O)NC2CC(NC(c3c(C(C)C)cco3)=O)C2)C)cccc(O)c1 C(=O)(CCCC(=O)NC1(CN(C)C(c2ccc(C)s2)=O)CC1)NCC C1(C(N2CC(C)C(CC(=O)NCCn3ncnn3)C2)=O)CC2CCC1CC2 c1(C(N2CC3CCN(C(CC(C)(C)C)=O)CC3C2)=O)csc2c1CCCCCC2 N1(C(CCc2cccc(C)c2)=O)CCN(C(c2cc(C)cs2)=O)CC1CO Cn1cnc2cccc(C(=O)NC3CC(F)(CNC(c4cccc(N)n4)=O)C3)c12 C1(N(C)C)CCN(C(C2CC2NC(c2cccc(CCO)c2)=O)=O)CC1 CC(CCNC(=O)OC(C)(C)C)C(=O)OCc1cnn(C)c1 CCCCC(CC(=O)NCC1C2COCC12)NC(C1(C(C)(C)O)CCC1)=O n1(CCC(=O)NC2CN(C(C3CC3CF)=O)CC2CO)nc(O)c2c1CCCC2 Cc1ccc(F)cc1C(=O)NCC(=O)NCC(c1ccccn1)C CN(C)NC(=O)CCC(=O)NC1CC(NC(C23CCCC(C)(C2)OC3)=O)C(O)C1 c1(OC)cc(C(=O)NC2CC(C(=O)NCC3CCN(C)C3C)C2(C)C)n(C)n1 N1(C(C=CCC)=O)CCC(CC(=O)NCC(C)S(C)(=O)=O)C1(C)C C1(CNC(C=CSC)=O)CC(C)CCN1C(=O)COc1cccc(F)c1 c1(OC)ccc(F)c(-c2cn(CC(N3CC(C(=O)O)C(C)(C)C3)=O)nn2)c1 c1(OCC(N2CCN(C(C3(O)CCCC3)=O)C3CC23)=O)cccc(Cl)c1Cl N1(C(C2C(OC)(OC)CC2)=O)CCc2c(-n3cnnn3)cccc21 N1(C(=O)NCCCCCCC#C)CCC(C)C2CCCCC12 C(=O)(C(=O)CC(C)C)N(C(CC(=O)NCC(C(=O)NC)C)(C)C)C C(CC(CNC(=O)CN1CC2CC2C1)NC(C1(C2CCCO2)CCC1)=O)OC C1(C(N2CC(O)(C(C(=O)N(CC#C)C(C)C)F)C2)=O)CC=CCN1C c1(OCCC)ccnc(CNC(C)(C(C)CC)c2nnnn2C2CC2)c1 c1(OC)nc(C)ccc1C(=O)NCC(=C1CN(C(=O)C=CC(C)(C)C)C1)F c1(C(N2C(C)CCC(CNC(C3CC(C)(C)C3)=O)C2)=O)c(O)cc(Cl)cc1Cl c1(NC(C(=O)N(CC(C)O)CCF)=O)cccc(Cl)c1OC(F)F CC1CN(C(c2cnc(N(C)C)o2)C(=O)NCCC2(C)CC2)CCN1C1CC1 c1(CC(=O)NCC2(NC(c3csc(CC4CC4)n3)=O)CC2)ccccc1F CCCCC(CN(C(=O)C(CNC(=O)C(CC)(CC)OC)N(C)C)C)CC C(=O)(CC(C)C(F)F)N1CCC(CCN(C(C(c2c(C)noc2C)C)=O)C)CC1 N1(C(C(C=C)(F)F)=O)CCC(C(F)(F)F)C(NC(=O)OC(C)(C)C)C1 c1(C(C(CS)C(=O)NC(CC)C)CC(N)C)cc(S(=O)(=O)N)ccc1Br C1(C(C)C)CCC(C)CC1NC(N1CC(C(F)(F)F)CC1CO)=O N1(C(C(c2cccs2)OC)=O)CC2CCC(C1)N2Cc1cnsn1 C1(COCCNC(CN(C)CC)=O)CC2CCC(C1)N2C(=O)CC(=C)Br c1(OC)ccc(Br)c2[nH]c(C(N3CC=CC3CNC(=O)C(C)C)=O)cc12 c1(C(N2CC3C(NC(C(C)OCCOC)=O)(C3)C2)=O)cc(C)nc2ccnn12 N1(C(Cc2ccc(SCC)cc2)=O)CC(NC(=O)C(F)C2CCC2)CC12CCC2 N1(CCC(=O)N(C2CCCC2)CC(=O)NC2CC(C3(C)N=N3)C2)CCCC1=O CCCCCC(O)CC(=O)N1CCC(NC(c2ncnc3c(C)csc23)=O)C(C)C1 c1(CC(=O)NCc2ccc(C(N3CCC(O)C3)=O)[nH]2)nccc2ccccc12 C(=O)(CC(C)C(F)F)NCC1OCC(CNC(c2c(C)onc2Br)=O)C1 C1(NC(C=CCOC)=O)CC2CC(C1)N(C(=O)CSc1ccc(F)c(F)c1)C2 C#CCC(CC#C)C(=O)NC1CN(C(C2(CC=C)CCCC2)=O)CC1(C)C c1(C(=O)NC2COCCN(C(c3c(C)nc(C)[nH]3)=O)C2)nn(C)c2c1CCCC2 c1(C(=O)NC(C2CN(C(c3cccc(Cl)n3)=O)C2)C)cccc2cccnc12 C12(C(N3CCN(C(c4ccccn4)=O)CC3)=O)CCC(O)(CC1)CC2 CC1CN(C(=O)Cc2ccns2)CC1(C)C(=O)NC1CN2CCC1CC2 Cn1nc(C(=O)NCC(c2ccccc2)OCC(F)(F)F)c2c1CCCC2 C#CC1(C(=O)NCc2ncn(C(C)C)n2)CN(C(c2cc(Cl)c[nH]2)=O)C1 C(=O)(C1CCc2ccccc21)N1CC(C(=O)NC(C#C)C(C)C)C2(C1)CCC2 N1(C(C(F)=CCC)=O)CCCCC1CCCNC(c1cc[nH]c(=N)c1)=O C1(CC(=O)NC2(CO)CCN(C(=O)C(F)=CCCF)C2)CC2(C1)C(F)(F)C21CC1 C1(CNC(C(CC)OC)=O)CCC(C(N2CC3CC2(CO)C3)=O)CC1 Cc1cc(C(=O)NC(C)CNC(=O)CCc2cc(C)ccc2C)cc(Cl)c1 N1(C(=O)CN2CSCCSC2)CCCC12CCN(C(C1C3CC4C(C3)C14)=O)C2 C(C)(CNC(c1ccoc1C)=O)(C(=O)N1CCCCC1C)OC C#CCC(CC(=O)NC(C)(CC)CCC)NC(C1CCOC1C(C)C)=O c1(C(N2CCCC(O)(CN(C(c3nc(C)sc3)=O)C)C2)=O)c[nH]c2cccnc12 c1(-n2cc(CNC)nn2)cccc(CO)c1.C=CCCC(=O)N1C(C(=O)OC)CC1C C1(NC(c2c(C)cc[nH]c2=N)=O)COC2(CCN(C(=O)CSC(C)C)CC2)C1 c1(OC)cc(CN2CCC(C(c3ccccc3)O)CC2)c(N)c(Br)c1 N1(C(CSC(C)C)=O)CCC(C)(C)C1C(N1CCCC(C(F)F)C1)=O CC1CCCN(C(=O)CCN(S(C)(=O)=O)C)C1CNC(c1c(F)cncc1Cl)=O N1(C(c2cncc(CNC(C(C(C)OC)O)=O)c2)=O)CC(N(C)C)CC1(C)C c1(C(=O)NCC(CC)(C)NC(C23CCC2C3)=O)ccc(Cl)cc1F n1(CC)ncc2c(C(=O)NC3(CNC(C4CC4C)=O)CCCC3)cc(C)nc12 CC1CC(C(=O)O)CCN1C.N12CCC(CC1)CNC(=O)C2 N#Cc1cc(N2CCC3CCN(C(=O)CC4=NNC(=O)C4)C3C2)ccc1[N+](=O)[O-] C1(C(N2CC=CC(C(=O)NCC3(SCC)CC3)C2)=O)C2CCCCCC12 CC(=O)CCCC(C)C(=O)NCc1nc(C(N2CCN(C3CCC3)CC2)=O)co1 C=CCCCCCCCNC(N1CCCC1C(=O)OC(C)(C)C)=O CC1(CNC(=O)CC2CCN(CC(=O)OC(C)(C)C)CC2)CCOCC1 N1(C(c2c(C)onc2)=O)CC2CC(NC(c3n[nH]c4c3COCC4)=O)CC2C1 c1(CCCC(=O)NC2C(C(=O)NCCOCCCC)COC2)c(F)cccc1F c1(NC)cccc(N=[N+]=[N-])c1.C(CCC(=O)N1CC2(C1)CCC(=O)N2)C1C(C)C1 C(C(=O)NCCSC)(C1=NOC2COCC12)N1C(CCC#C)CCC1 CC1(NC(C2(c3cccnc3)CC2)=O)CNCC1(F)F.n12cc(nn1)C2 c1(N2CCC(CCNC(c3ncn(C)n3)=O)C2)c([N+](=O)[O-])cnn1C C1(CNC(c2c(C)scn2)=O)C2CC2CN1C(=O)CC=C(Cl)Cl C1(CNC(C(C=C)(C)O)=O)CC(C(=O)N2CC(CCOC)C2)=NO1 C1(C)(CNC(C(C)Sc2ccccc2)=O)COCCN(C(=O)Cn2cccc2)C1 N1(C(c2c(CC)nns2)=O)CCCC(CNCCC(N2CCOCC2)=O)C1 CC#CCC(C(=O)N(CC(F)F)C)NC(=O)CC(C)CC1CC1 N1(C(c2c(C)cn(C)n2)=O)CCC2(C1)CN(C(C1(c3ccnc(Cl)c3)CC1)=O)C2 c1(CC(=O)NCCC(C)NC(=O)C(c2cccc(Cl)c2)O)nsc2ccccc12 CC1CN(C(C2(C)CC3CCC2C3)=O)CCC1NC(c1ccc(Cl)s1)=O N1(C(C2(CCC)CCC2)=O)CCC2CC2(NC(=O)CN(c2ccccc2)C)CC1 c1(C(=O)NCC2OCC(C(=O)NCCCCC(=O)NC)C2)ccc(C)cc1O C1(C(=O)NC(CN(C(c2c(COC)cc[nH]2)=O)C)C)CC(C(C)C)=NO1 C1(OC)CN(C(=O)CC2CNC(=O)C2)CC1NC(c1c(C)coc1C1CC1)=O c1(CN(C2CCN(C(COCC)=O)C2)C(c2ccccc2)=O)ccc(F)cc1 C1(C)(C(N2CC(CCC)C(NC(c3cnn(CC)c3N)=O)C2)=O)CCCC1(F)F CC1CCCN(C(N2C3C(OC(C)(C)C)C(CC3O)C2)=O)c2cc(F)ccc21 C(=O)(C(Cc1cnco1)NCC)NC(CCOC)C Cc1ccc(C(=O)NC2CCOCC2NC(c2csc(-c3ncc[nH]3)n2)=O)cc1 N1(C(CN(C(COC)=O)C)=O)CCC(CCNC(c2sccc2F)=O)C1 c1(N(CCCCCC=C)C)nc(NC2CCCCCC2F)c2sccc2n1 C1(=O)CC(C)CN(C2CC2)CCN1.C(C(C)(C)C)OCCCOC CCC(C(C)(F)F)NC(=O)CCN(C(c1cn(CC)nn1)=O)CC1CC1 C1(=O)C(O)C(C(C)C)N1.N1(C(c2cn(CC)nn2)=O)CCC(O)C(CO)C1 C1(Cn2cc(CCC(=O)OC)nn2)CC(F)CN1C(c1occc1C(F)(F)F)=O c1(C(=O)NC)ccc(C(=O)NCC(C)CNC(c2cc(C#N)c[nH]2)=O)cn1 N1(C(c2c(OCC)ccs2)=O)CC(CCNC(=O)CCCCC2CC2)OC(C)C1 Cc1ccc(C(=O)NC(C)CNC(=O)CC2CCCC(C)(C)O2)cc1F N1(C(c2ccnc(OC)n2)=O)C2CCC1C(F)C(NC(=O)CC1COCCO1)C2 N1(C(CNC(CC)=O)=O)CCC(C(=O)NC2C=CC(CN(C)C)C2)C12CC2 Cc1cc(C(N2CCC(CCNC(=O)C(c3ccnn3C)O)CC2)=O)nc(O)c1 N1(C(c2cc(C)sc2N)=O)CC2CCCC2(NC(=O)CC23CCCC2C3)C1 C(N=c1[nH]c(=NCc2ccsc2Cl)[nH]c2cccc(F)c12)C1CCCC(C)CC1 C12(C(N3CCN(CCNC(=O)CNC(C4CCC4)=O)CC3)=O)CCCC1CCC2 Cc1ccc(-c2ccc(CN3CCN(S(=O)(=O)C(C)C)CC3)s2)c(C(F)(F)F)n1 c1(C(=O)NC(CNC(c2ccc(OC)c(Cl)n2)=O)CO)c[nH]c2cc(Cl)ccc12 c1(C(N)=O)cc(Cl)ccc1C(=O)N(CCNC(c1c[nH]cc1C1CC1)=O)C1CC1 Cc1ccc(C(=O)NCCOC2CN(C(C3C4CC4C4CC34)=O)C2)cc1N Cc1noc(C)c1CC(N1CCCC(CN(C2CCS(=O)(=O)C2)C)C1)=O C(CCCC(N)=O)(C(=O)NCc1cc(O)nc(Cl)c1)N1CC(O)(CN(C)C)C1 C1(C(=O)NC(CN(C(COC(CC)C)=O)C)(CO)CO)CCCCC12CC2 Cc1cc(NC(=O)C(C)(C)C(C)O)ccc1NC(=O)CCC1CC1(F)F N1(C(C2CC=C(C)CC2)=O)CCCCC(CNC(c2cc(C3(C)CC3)no2)=O)C1 C1(C(=O)NCC(=O)N(CC(CNC(C(C)(C)OC(C)=O)=O)O)C)CCCCCC1 C(=O)(CCC(=O)NN(C)C)NC(C)CCCNC(=O)C(C1CCCCC1)O N1(C(C2C=C(C)CS2)=O)CC(NC(=O)CCCn2cccn2)C2CCCC12 N1(C(C2(C#C)CC2)=O)CCCC2(C1)CN(C(=O)CC(C)P(C)(C)=O)C2 C1(F)(CNC(c2cc(C)c(C)s2)=O)CCCN(C(=O)COC(C)(C)C)CC1 CN=c1ccc(C(=O)NCC2CC2CNC(c2cnn(C3CC3(F)F)c2)=O)c[nH]1 C(=O)(c1nn(C2CCCC2)c(=O)[nH]1)N1CC(N(C)C(c2cnsn2)=O)C1 c1(OC)ccc(Cl)cc1CC(N1CCC(CCNC(C2CC2CCOC)=O)C1)=O C1(NC(C=Cc2cnc(C)s2)=O)CCN(C(=O)C(C)N(C)C)C(C)C1 c1(C(=O)NC2CN(C(CN3CC(C)(OC)C3)=O)CC2F)ccc(O)nc1C C(=O)(CC(F)(F)C(F)(F)F)NC(C1(O)CN(C(C23CCC(C)(CO2)C3)=O)C1)C CCC(CCC(=O)N1CC(C(=O)NCc2nc(C)c(C)s2)C2(CC2)C1)OC c1(-n2cc(CC3(F)CN(C(c4nc(C(C)=O)sc4)=O)C3)nn2)c(F)cccc1F Cc1nn(C(C)C)cc1C(=O)NC(C)CCNC(c1ccc(CC(C)C)o1)=O C=C(Br)CCC(=O)NC1CCC(NC(=O)CCc2cc(C)on2)CC1 N1(CC)CCCC(C(=O)N(C(C)CNC(c2[nH]ccc2-c2cccs2)=O)C)C1 Cc1cn2cc(C(=O)NC3CCCCN(C(C4(C)CC5CCC4O5)=O)C3)nc2s1 c1(-c2c(F)cc3c(c2)CCOC3)ccc(-c2cncc(-c3cscn3)c2)c2c1OC(F)(F)O2 CC12CN(C(=O)C=Cc3cnc[nH]3)CC1CN(C(=O)CC1CCCCC1(F)F)C2 c1(C(=O)NCC(CNC(C(C)OC)=O)O)cnc(C(F)(F)F)c(C)c1 CCC(CC)(CC)C(=O)N1CCC(C2CCCN2C(=O)Cc2cccnc2C)C1 c1(NC(c2ccc(CNCc3cc[nH]c3)nc2)=O)cc(Cl)cnc1O O=C1Cc2ccc(C(=O)NCC3CN(C(c4ccnc(F)c4)=O)C3)cc2N1 n1(CC)nccc1C(=O)NCC(C1CC1)OC.C1(=O)CC=CCN1C CN1CCC(CC(N2CCCC2CNC(=O)CC2CC3(CCC3)CO2)=O)C1=O CCCCCCC(C)C(=O)N(CC(C)CN)C c1(C(N2CC(NC(c3[nH]c(CC)c(Cl)n3)=O)C2)=O)csc2nccn12 c1(C(=O)NCCCN2CCC(NC(c3nc(COC)oc3)=O)C2)ncncc1Cl C1(NC(C(C)OCCCC)=O)CCCN(C(C2CC2(F)F)=O)C1 c1(C(C)C)cccc(C(=O)NCC(O)CNC(=O)C(F)=C2CCC2)c1N N1(C(COCC=C)=O)CCCC(CNC(c2cn(C3CCOC3)cn2)=O)C1 Cc1ccc(CC(=O)NCC(C)(C)NC(=O)C=CC=C(Cl)Cl)o1 C(=O)(C1=CCCC1(C)C)NCC1(O)CCN(C(C(C2CCCC(=O)N2)C)=O)CC1 C(=O)(C1=CN(C)S(=O)(=O)N=C1C)N(CCN(C(c1cncnc1)=O)CC)CC Cc1cc(C(=O)NCCC2CCC(NC(c3snc(C)c3N)=O)C2)cc(O)n1 c1(NC(c2c(CNC(COCC(=O)NC)=O)cc[nH]2)=O)cnc(C)c(C)c1 c1(C(=O)NCC(N(C(=O)C(F)n2cccn2)C)C2CC2)cccnc1C(F)F CC1CCC(NC(=O)Cc2cccc(O)c2F)CN1C(c1cc(C#N)c[nH]1)=O c1(CNC(C)=O)ccc(C(=O)NCCCNC(=O)CSCC(F)(F)F)o1 C1(CNC(=O)CSc2cn[nH]c2)C2CCN(C(=O)CCC3CCOC3)CC12 c1(C(=O)NCCCN(C(C2CCC(F)C2)=O)C2CC2)cc(F)c(Cl)cc1Cl c1(NC(C2N(C(c3c(C)ccnc3)=O)CCC2O)=O)ccc(Br)c(C)c1C C(C)(C)(C(=O)NC1(C(=O)NC(C)C)CC1)N.C1CCNC(=O)N1CCC.CCF c1(CNCC(NN2N=C(C)C2)=O)cc([N+](=O)[O-])cc(Br)c1O CCCCC(O)C(C)C(=O)NCCCN(C(=O)CCc1cccc(OC)c1F)C N#CC1CCCCC1NC(=O)C(N1CCCC(c2cccs2)C1)=O Cc1cc(Cl)cc2[nH]c(C(=O)NC3CN(C(=O)CC(C)F)CC3(C)C)cc12 C1(CNC(C(F)=CCC)=O)CCC(F)(CNC(c2cn(CCCC)nn2)=O)CC1 N1(Cc2c(C(=O)OCC)scn2)CC2(CNC(c3c(C)n[nH]c3C)=O)CC1CO2 N1(C(C(C(C)C)OC)=O)CC2CCCC1C2CNC(=O)CC1CCC(O)C1 C12(NC(C3(C)CCCCCC3)=O)CCCN(C(=O)CCC3CC3)CC1C2 C(c1ccc(OC(C)(C)C)cn1)=CC(=O)NC1C=CCN(C(CSC)=O)C1 C1(C(N2CC3(CN(C(c4ccc(F)c(F)c4)=O)C3)C2)=O)CCc2nn[nH]c2C1 C12(CNC(C3CCOC3C3CC3)=O)CCCC1N(C(c1cncc(Cl)c1)=O)CC2 c1(CC(C)=CC(=O)NC2(C)CN(C(c3cnc(O)[nH]3)=O)C2)cnc2c(c1)COC2 Cc1cc(F)c(C(N2CCCC(N(C)C(c3cnnn3C)=O)C2)=O)c(F)c1 C1(C(=O)NC(CC)CNC(c2cncc(C(=O)N(C)C)c2)=O)COCCN1C=O N1(C(C(CC)C#N)=O)CC2(CCC(CNC(=O)CC3SC(=N)NC3=O)O2)C1 N1(C(c2cc(OC)c(Cl)s2)=O)CCC(NC(c2nnn3c2CCC3)=O)C(F)C1 C1(CNC(=O)CCF)CCN(C(=O)C=Cc2cccnc2)C12CC2 C1(CNC(c2n(C(C)C)cnc2)=O)CC(C)CN(C(=O)C(c2ccnn2C)O)C1 C1(NC(c2c(C)n(C3CC3)nc2)=O)CCN(C(c2nc(C3CC3)cs2)=O)CC1C N1(C(C(CCNC(C(CC)=CCCC)=O)O)=O)CC(C)C(C)C1C C(=O)(C1COc2ccccc21)N1CCC(NC(c2ccc(Cl)[nH]2)=O)(CF)C1 C1(CC(N2CCC(NC(C34CC(C)(OCC3)C4)=O)C2)=O)COCC2(CCC2)O1 O(C1CCc2c1ccc(Br)c2F)C(c1cc(O)ncc1Br)=O C1(C(C)NC(=O)CCN2CCCC2=O)CC(F)(F)CN1C(=O)CCCC(N)=O C1(CNC(CCCCC=C)=O)CN(C(=O)CNC(C)=O)CCC12CCC2 Cc1ccc(C(=O)NC2CCC2NC(=O)CCCC2CCC2)c(C)n1 O=C1NC(=O)C(CCNC(N2CC(CN3CCOCC3)C3(CC3)C2)=O)N1 CC1CN(C(=O)CC(C2CC2)C2CC2)CCCN1C(c1scnc1C1CC1)=O N1(C(CC(C)SC)=O)CCC2CCC(NC(=O)C(C)(C)c3ccno3)C12 N1(C(CCCC(=C)C)=O)CCC2CCN(C(=O)C(Cc3ccsc3)NC=O)CC2C1 C12(C(N3CCC(NC(c4cc(C(C)(F)F)n[nH]4)=O)C3)=O)CCC(CC1)OC2 N1(C(C2(COC)CC2)=O)CC(C(N2CC(CN=[N+]=[N-])C2)=O)C2(CCC2)C1 c1(CC(=O)NCC2(NC(C(C)NC(=O)NC)=O)CCOC2)nc([N+](=O)[O-])n[nH]1 C(=O)(C1Cc2ccccc21)NCC1C=CC(NC(CC2CCN(C)CC2)=O)C1 N1(C(C2C(OC)CCC2)=O)CCN(C(c2ccnc(C)c2)=O)CC1C c1(C(N(CC(=O)NC(C2CCCC2)CC)CC2CC2)=O)cc(C)sn1 C(CN=c1cc[nH]cc1S(=O)(=O)C(C)(C)C)N(CC)CC1CC(F)(F)C1 c1(OC)cccc2c(C(N3C4CCC3CN(C(=O)CN(C3CCC3)C)C4)=O)n[nH]c12 c1(C(C(=O)N(C(C)C(=O)N(C)CCF)C(C)(C)C)N(C)C)ccnn1C c1(CC)c(C(N2CC(CNC(c3cnc(C)o3)=O)(OC)C2)=O)cccc1F Cc1nc(C)c(C(=O)NC2CC3CC2N(C(c2cnc(Cl)cc2N)=O)C3)nc1C c1(C(N(CC(=O)OC)CC#C)=O)cc(C)no1.C12CC(C1)NC(=O)C2 CC(C)C(CCN(C(=O)CCC(N)=O)C)NC(=O)CN1C(=O)NCC1=O C1(C(=O)NCC2(OC)CN(C(=O)COCc3ccncc3)C2)CC(C)OC1C C#Cc1ccc(F)cc1C(=O)NC(C1CN(C(=O)C(CCC)OC)C1)C CS(C)(=O)=Nc1ccnc(C(=O)NCC2CN(C(C3CCCCS3(=O)=O)=O)C2)c1 CC1CN(C(C2CN3CCC2CC3)=O)CCC1N(C)C(C1(S(N)(=O)=O)CCC1)=O c1(C(=O)NC(C2CCN(C(=O)CCn3cnnc3O)C2)(C)C)csc(=N)[nH]1 N1(C(Cn2nnc(=N)[nH]2)=O)CCC2(CCCN(C(=O)COc3ccccc3)C2)C1 C1(NC(C2(NC(c3nccn3C)=O)C(C)CCC2)=O)COCC1N=[N+]=[N-] CC1CN(CC)CC2(CCNC2)O1.C(F)(F)(C(F)(F)F)n1ncc(NC(=O)C(C)O)c1 C(N=c1nc2scnc2c(N2CCC(N(C)C)C(C)C2)[nH]1)c1c(C)nco1 c1(C(N2CCCC(C)(CNC(C(C=C)(C)C)=O)C2)=O)snc2ccccc12 CN1CCC(C)(C(N2CCC2CNC(=O)Cc2c[nH]nc2O)=O)C1=O c1(NC(C(N2CCN(CC)CC2)=O)C)ccc(Br)cc1[N+](=O)[O-] CCCC(C(=O)NCC1CCCN1C(C1C=CC=CC=C1)=O)NC(C)=O c1(CNC(C2CC(F)CN2C(c2ccc(F)cc2Br)=O)=O)cccc(F)c1Br CCCCC(O)C(=O)N(C)CC1CCCN(C(=O)C(CC)CO)C1 C1(NC(CCc2scc(C)n2)=O)CC2CCC(C1C)N2C(c1cc(C#N)c[nH]1)=O C12(CNC(C#CC(C)C)=O)CCC1CCN2C(=O)C(F)=C1CCCC1 C1(CC)CC(C2CCCCC2)CN1C(CC(=O)NC1CCCC1)C(=O)OC Cc1cc(C(=O)NCC2(NC(=O)CC(F)(F)c3nccs3)CCCC2)cc(N)c1 N1(C(C2CN(C(C)=O)C2)=O)CC(N(C)C)CC(NC(c2c(C)nn(C)c2F)=O)C1 CCCCCC(O)CC(=O)NC(COC)C(=O)NOCCN1CCCC1=O c1(C(=O)NCC23CC2CN(C(C2CCSC2)=O)C3)cccc2[nH]nc(O)c12 C#Cc1cc(F)c(C(=O)NCC2CN(C(C3(F)CC=CC3)=O)CC2(C)C)c(F)c1 CC(C)CC(C)(CO)NC(C1CC1CNC(c1n[nH]c(=N)[nH]1)=O)=O Cc1n[nH]c(C)c1CC(=O)N(C1CCN(C(=O)Cc2cscn2)C1)CCO C1(ONC(C2CCC(COOC)O2)=O)CCC(C(=O)Nc2c(C)n[nH]c2C)CC1 C1(C)(C(N2CC3C(C(=O)Nc4ccc(C(=O)OC)nn4)C3C2)=O)CC2(CCC2)C1 C(C(=O)N(CCCN(C)C(C1CC1c1cncs1)=O)C)(C1CCOC1)OCC Cc1ccc(N)c(C(N2CC(CCCCNC(C3CC(NS(C)(=O)=O)C3)=O)C2)=O)c1 N1(CCNC(C(c2cccs2)NC(CC=CCC)=O)=O)CCOC(C)C1 C12(C(NOCC(=C)Cl)=O)CC(CCO1)N(C(C1CCC1)=O)C2 C(=O)(CC(C(=O)N1CCC12CN(C(=O)CC1CC=CCC1)C2)N(C)C)OC C1(CNC(c2ncn(CC)c2)=O)CN(C(C2(C)CC(C)C2)=O)CCC12CCOC2 CC1CN(C(=O)CCn2cccc2)CCCN1C(c1cnn(C)c1C1CC1)=O c1(C(=O)NCCC2CN(C(C3(C)CC4CCC3C4)=O)C2)cc2ccccc2cn1 c1(OC)ccc(OC)c(OC)c1NC(N1CC2(CC2)CC1C(=O)OC(C)C)=O N1(C(C2(C)CCC(=O)N2)=O)CCC(C)(C)C(NC(C23CCOC(C)(C2)C3)=O)C1 c1(OCC)ccc(C)cc1NC(=O)CC1N(C(=O)CC(F)(F)F)CCC1(C)C N1(C(c2conc2C)C(=O)NCCOC)CC(CS(C)(=O)=O)OC(C)C1 C1(NC(c2coc(C(F)(F)F)c2)=O)CN(C(=O)COC2CCOC2)C2(CCC2)C1 C(=O)(C1=C(Cl)CCC1)NCC1N(C(c2cccc(C(N)=O)c2)=O)C2C(C1)C2 c1(C(=O)NCC(CCOC)NC(=O)C(CN(C)C)N(C)C)cccc(CS(C)(=O)=O)c1 Cc1ccc(F)cc1C(N1CC(C(F)(F)F)C(CNC(=O)COC2CCC2)C1)=O c1(CNC(C(c2ccco2)NC(C(C)=CCC)=O)=O)c(C)cccc1F N1(C(c2scc(C)n2)C(=O)N(CCCF)CC(F)F)CCN(C2CCCC2)CC1 c1(C(=O)NC(c2nnnn2CCC2CC2)c2cccs2)ccc(CN(S(C)(=O)=O)C)s1 Cc1cc([N+](=O)[O-])ccc1NC(=O)C(=O)NCCc1ccccc1N1CCCCC1 C1(NCC(C2(OCC)CCOCC2)C)C(C)CCCC1C c1(C(=O)NCC2(O)CC(NC(C(CCC)N(C)C)=O)C2)c[nH]c2cc(Cl)ccc12 C#Cc1cccc(N(C)C(C2CC(=O)CN2C(=O)CN2C(=O)CNC2=O)=O)c1 c1(C(N(C)CC2CCN(C(=O)CCc3nccn3C)C2)=O)ccc2occc2n1 N1(C(C(C)NC(COC)=O)=O)CCC(N(C(C2CN(C3CCOC3)C2)=O)CC)C1 N1(C(CN(CC#C)C(C2CCC(F)CC2)=O)=O)CCn2nc(C)nc2C1 N1(C(C(=O)NC2CC2)=O)CCC2(CCN(C(c3cnc(O)s3)=O)CC2)C1 CCC(C)(CC)C(=O)NCC(C(C)(C)C)NC(=O)Cc1nc([N+](=O)[O-])n[nH]1 c1(C(=O)NCC)ncnc2sccc12.c1(C(N2C(CC)C2)=O)csc(COC)n1 Cc1cc2c(C(=O)N(CC(C)N(C(=O)C(C)CC3CC3)C)C)nccn2n1 N1(C(C2CCC(C)(F)CC2)=O)CC2CC(NC(C3CN(C(=O)C4CC4)C3)=O)CC2C1 c1(C(N2CC(N(C)C(c3ccc4c(c3)OCC4)=O)C2)=O)c[nH]c2cc(Cl)ccc12 N1(C(CC)=O)CCC2CCN(C(c3cn(C4CCOCC4)nn3)=O)C2C1 N1(C(CN(CC(C)(C)C)C)=O)CCCC(N(C(=O)CC2CC3CC3C2)C)CC1 Cc1cncc(CC(=O)NCC2CN(C(C3COC(=O)N3)=O)CC2O)c1 c1(NC(C2CN(S(=O)(=O)c3ccccc3Cl)C2)=O)nc2cccc(Br)c2s1 C=C(C)C(O)CC(=O)N(C1CCCN(C(c2ocnc2C)=O)C1)CC C(CCCCC(=O)N(C)C)N1CCCC(CCC(=O)NC2C(C)CCC2C)C1 c1(C(=O)NCC2(O)CCN(C(C3(C)CC=CCC3)=O)C2)ccnc2ncccc12 c1(C(N2CC(CNC(c3cc(COC)[nH]n3)=O)(OC)C2)=O)cc(F)ccc1F C1(NC(c2c(CC)ncs2)=O)CC(C)CN(C(=O)C(C)n2cccc2)C1 N1(C(c2ncn(CC)n2)=O)CCCC2CCN(C(c3cnn4c3CCC4)=O)CC12 N1(C(c2c(OC)ccnc2)=O)CCC2(CC1)CCN(C(c1ncc[nH]1)=O)CC2 c1(C(=O)NC(CC)CN(C(c2csc(CO)n2)=O)CC)n[nH]c2c1CC1CC21 N1(C(c2nn(-c3ccccc3Br)cc2Cl)=O)CC2(CCOC2=O)C1 CC(CC(=O)N1CC(NC(c2cc(Cl)n(C)n2)=O)C2CCCC12)CC(C)(C)C C1(C(N2CCC(CCNC(CCC#C)=O)C2)=O)C2CCC(=O)C12 C(=O)(CC(O)C(C)CC)NCc1c(C(=O)NC(C#CCC)(C)C)n[nH]c1 Cc1[nH]c(=N)ccc1C=CC(N1CCCC(NC(=O)C(F)CC(C)C)C1)=O Cc1cccnc1C(=O)NCC1CN(C(c2cc(Br)sn2)=O)CCO1 C=C(C)CCC(=O)NC1CCCC1NC(c1cn(CCO)nn1)=O CC1(C)CCOC(C(N2CCCC2C(=O)NCC2CC2(C)C)=O)C1 O=S(=O)(c1c[nH]ccc1=NC1CCCCCC1)NCC(c1ccccc1)F c1(C(N2CCC(C(C)NC(CC=CCC)=O)C2)=O)ncc(C)cc1F N1(CCC)CC(C(=O)N(C2CCN(C(C3(C)COC3)=O)C2)CCO)CC1=O N1(CC(N2CCC(CCNC(c3c(C)n(C)nc3)=O)C2)=O)C(=O)CCCC1=O N1(C(CCCOC(C)=O)=O)CC23CCCC2(C1)CN(C(c1c(Cl)cnn1C)=O)C3 c1(C(=O)NCCC(C)NC(C2SCCCS2)=O)coc(CC2CC2)c1 C(=O)(C1=C2CCCN=C2NN1)N1C(C)CCC(NC(CC(C)C)=O)C1 N1(C(c2c(C)ccnn2)=O)CC2CN(C(=O)C(c3ccnn3C)O)CC2C1 CC(CC(N)=O)C(=O)NC1CC(CCNC(c2cc(C(F)(F)F)ccc2F)=O)C1 C1(COC)CN(C(c2cc(C)nn2C)=O)CCN1C(=O)CC1(C(=O)OC)CC1 C(C(=O)NCC=CCl)(C(C)(C)C)NC(CCC(C)OC)=O CN1CCOCC1CC(=O)N(CCNC(=O)Cn1ncnn1)C1CC1 N1CCc2nc(N3CC4C(C)(C)CC4C3C(=O)O)ncc2C1.N1CCOCC1 Cc1nc(C(=O)NC(C2CCCC2)CNC(=O)CCOCCC2CCCO2)cs1 CC1OC2(CNC(=O)C=Cc3cc[nH]n3)CC1(NC(=O)C(C1CC1)N(C)C)C2 N1(C(c2c(CC)c[nH]c2)=O)CCOCC1C(=O)N(c1cc(C)ncn1)CC c1(C(C2(COC)CC=CC2)NCC(c2nnnn2C)C)cc(C(C)(C)C)on1 c1(CC)cc(C(=O)NC(CNC(C2(c3oncc3C)CC2)=O)C2CC2)ccc1O n1(CC(=O)NCC(CNC(CC(CC)SC)=O)O)cccc(O)c1=O Cc1ccccc1C(=O)NC1(C(N2CC(C(=O)O)C(C)C2)=O)CSC1 c1(C(=O)NC(C(C)NC(c2nc(OC)cc(OC)n2)=O)C)cc2c(s1)CCOC2 c1(C(=O)NC2CN(C(c3cccc(OC)c3)=O)C3C2C3)cnc2ncccn12 C1(OC)CCCCC1N=c1ccnc(COCC2CC2)[nH]1.c12ccc(cc1)[nH]2.C1C(=O)O1 Cc1cc(Cl)c(Cl)cc1C(=O)NC1CCCN(C(=O)COCC2CC2)C1 c1(C(N2CC(CNC(c3nc(CC(C)C)sc3)=O)C2)=O)cccn2ccnc12 C(=O)(C(C)CCC(C)(C)C)N1CCC(CC=C)(NC(c2oc(SC)cc2C)=O)C1 c1(CCC(=O)NCC23C(CN(C(c4cnn(C)n4)=O)C2)C3)ccc(F)c(F)c1 N1(CC)CCOC(C(=O)NC2CCC(C(=O)OC)CC2)C1.C12COCC1C(=O)N2 C1(NC(C(C=C)C)=O)CCCN(C(=O)C2=CCCC2)C1CC c1(OC2CCC(C)CC2)ccc2cccnc2c1.c12cn(nn1)CC1CCCN1C2=O c1(C(N(C(C)CNC(=O)CN2CCC(C)(C)C2)C)=O)cccc2c1NCCC2 C1(NC(C(c2ccccc2)N(C)CC)=O)CN(C(c2cnsc2)=O)CCC1C CCC(C(=O)OC(C)(C)C1CCC1)C(=O)N1CCC(NC(c2ccccc2)=O)C1 Cc1ccc([N+](=O)[O-])c(CNC(=O)C(=O)Nc2ccc3nnn(C)c3c2)c1 Nc1cc(C(N2CC(NC(c3scc4c3OCCO4)=O)C2)=O)cc(F)c1O C1(CC)CN(Cc2ccc(O)nc2Cl)CCN1C(c1ccc(I)cc1)=O CN1N=C(C(=O)N2CC(NC(=O)CC(O)C(Cl)(Cl)Cl)CC23CCC3)CCC1=O Cc1cc(C)cc(C=CC(=O)NC(C2CCN(C(c3ccc[n+]([O-])c3)=O)C2)C)c1 c1(NC(c2ccc(C)cc2Cl)c2nnnn2C2CCC2)ccc(C#N)cc1O C1(CN(C)C(C2(CCNC(c3cnnn3C)=O)CCC2)=O)CC2C=CC1C2 c1(C(=O)NCCCCC(C)NC(CCC)=O)cncc(OCC(F)F)n1 Cc1cc(C(N2CCC3(NC(c4cncs4)=O)CC3C2)=O)cc(C)c1Cl N1(C(C2CCSCC2)=O)CC2CCN(C(C3(CF)CC3(F)F)=O)CC2C1 CC(C)(C)CCC(F)C(=O)NCC1CCCC1NC(=O)CC1CCSC1 N1(C(c2nnc(OCC)s2)=O)CCC(C)C(CNC(=O)CCCC(N)=O)C1 c1(OC)cccc(C(=O)NCCNC(=O)Cc2cccc(SCC#N)c2)c1 C=CCCN=C(NCC1COC(=O)O1)NC1CCC(OC(F)F)CC1 Cn1cnc2nc(=NCCC3C4CCCOC34)[nH]c(NCc3ccc(F)cc3)c12 C(=O)(CC(F)(F)F)NCC1(C(=O)OCC)CCC1.C1C(C)(CO)N1 C1(CNC(=O)Cc2c(F)cccc2Cl)C2CCCC1N(c1nnc(C(N)=O)s1)C2 c1(CC(N2C(C)C(NC(=O)COCCF)CCC2)=O)ccc2c(c1)CCC(=O)N2 c1(C(N(CCC2CCN(C(C(C)OC)=O)CC2)C)=O)ccc(P(C)(C)=O)cn1 CCCCCN(CCC#N)C(=O)NC1CCC1CO C12(NC(C3CC(=C4CCC4)C3)=O)CCC(C(=O)NC(C3CCCO3)CO)(CC1)C2 c1(CNC(C2CN(C(=O)CCOCC3CC3)C2)=O)ccccc1.C1(C(F)(F)F)(O)CC1 c1(OC)ccc(Br)c(C(=O)NC2CC3(C2)CN(Cc2cc(F)cc(F)c2)C3)c1F C1(NC(C2C(CC)OCC2)=O)CCCC12CN(c1cc(C)nc(C(C)C)n1)C2 Cc1ccc(C#N)cc1CCCNC(c1cc(N(C)C)ccc1Cl)c1nnnn1C O=C1CNc2ccc(S(=O)(=O)Nc3cccc(-c4ccccn4)c3)cc2N1 C1(NC(C2(C)CC(NC(C3CC4CC3CC4O)=O)C2)=O)CC2CCCC2C1 C(C)(CC=O)NC(C)(C)CCNC(=O)C=CCOCC.C#CCN(CC=C)C C(=O)(CCC(=O)NC(CNC(C1CC1C(=O)OC)=O)C(C)C)NCC N1(C(C(=O)NC2CCN(C(CCC=C)=O)C2)=O)CCC(C(C)(C)C)C1C1CC1 c1(CC(N2C(C)CN(Cc3cc[nH]n3)CC2)=O)cc(F)c(F)cc1Br c1(CN2CC(NC(c3c(C)ccnc3)=O)(CO)C2)c(O)ccc2ncccc12 n1(CC(=O)NC2(CNC(C(C)SC)=O)CCC2)nc(C)c2cccnc12 C(=O)(C1=CC2(CN(C(C3(CC4CC4)CC3)=O)C2)OC1)NCC1(O)C(C)OCC1 Cc1onc(-c2ccccn2)c1C(=O)NC(C)CNC(c1ccsc1C)=O C(CCCCCN(C(=O)CC1CCOCC1OCC)C)NC(C(C)=CC)=O C1(C)(C(=O)NC)CCN(c2nnc(C(C3(F)CCCCC3)O)n2C)C1 c1(OC)ccc(C)cc1C(=O)N(CCNC(=O)CCc1cnoc1)CC1CC1 C1(NC(C2(C)CCOCC2)=O)CC2(C1)CN(Cc1ccc(Br)c(Br)c1)C2 C1(C(=O)NCC2CC(C)(C)N(C(c3cc[nH]c(=N)c3)=O)C2)CC2CCC1C21CC1 c1(C(=O)NC2(C)CCN(C(CN(c3ccccc3)C)=O)C2)cc2sccc2[nH]1 C(=O)(C(C)(C)C(N)=O)NCCC1N(C(c2c(C)nc(COC)s2)=O)CCC1 C1(CNC(C=CC(C)NC(C2C=CCCC2)=O)=O)CC12CCOCC2 c1(C(=O)N(C2C(CNC(c3nc(C)n(C)c3)=O)CCCC2)C2CC2)cnn2c1OCCC2 c1(CN(C(C(C)N(C(c2cccnc2)=O)C2CC2)=O)C)ccncc1F C(C)(C)(CCCNC(=O)C(C)NC(C12CSCC1C2)=O)OC c1(C(=O)NC2C(CNC(C(c3c(C)cccc3)C)=O)C2)cnc(CC2CC2)nc1O c1(C(N2CCN(CC(C)(C)NC(C3C(=C)C3)=O)CC2)=O)cc(C)[nH]c(=NC)n1 Cc1onc(C2CC2)c1C(=O)NCC1CC(NC(=O)CCC(=O)N(C)C)C1(C)C C1(C(=O)NC2(COC)CN(C(=O)C(C)=CC(C)(C)C)C2)CCCC(C(F)(F)F)C1 C1(NC(C(CC)(CC)CC)=O)CCC2(CCN(C(C3CCC(=O)O3)=O)C2)C1 c1(CC(=O)NCCC2COCCN2C(C2CC2CF)=O)cc(F)ccc1F C1(NC(c2cc(CC)n(C)n2)=O)CC2CCC1CN2C(c1csc(O)n1)=O c1(NCC(c2ccccc2)OC)ncnc(N2CCCC(C)CC2)c1C C1(C)(CNC(c2c(CC)occ2)=O)CCCN1C(C1CC(C)(C)C1)=O C1(CC#C)CCN(C(C2(CNC(=O)CCC3(C)CC3)CCCO2)=O)CC1 c1(C(=O)NC2CCN(C(C(C=CC)O)=O)C2C)cncc([N+](=O)[O-])c1 c1(C(=O)NC2C(NC(c3ccc(CCC=C)cc3)=O)C2)cnc2c(C)cccn12 C1(C(=O)NCC(CC)NC(c2cc(OC)ccc2N)=O)CCOC(C)(COC)C1 S(=O)(=O)(c1c(F)cc(C#N)cc1F)N(c1noc(C)n1)CC N12C3CCC1CC(C3)C2=O.C(C(=O)N1CC(C=O)C1)(C(C)C)OC c1(C(=O)NC(CCNC(C(Cn2ccc(C)n2)C)=O)(C)C)cnc2c[nH]nc2c1 N1(C(c2c(OCC)c(F)ccc2)=O)CC2=C(C1)CN(C(c1cc(CF)on1)=O)C2 c1(C(N2CCC(CNC(c3ccncc3Cl)=O)C2)=O)cc(Cl)cc(Cl)c1 C(CCCCCCCO)=CC(=O)NC1CC(NC(C2(F)C(C)OCC2)=O)C1 c1(NCCC2(NC(C#CC(C)C)=O)CCCC2)ccc([N+](=O)[O-])c(OC(F)F)c1 C(C)(C)(CCC(=O)NCc1ccc(C)cc1F)NC(CSCCCC)=O C(=O)(C1=CCN(C(=O)C2=C(C)CC2)C1)NCC(COC)O C1(CNC(C(C2CCOC2)NC(C2C(=C)C2)=O)=O)CC2CCC(C1)C2 N1(C(C(C=C)O)=O)CCC(C)N(C(c2cc(SC(F)(F)F)c[nH]2)=O)CC1 C1(N=[N+]=[N-])(C(N(C2(C#C)CC2)C)=O)CCN(C(C2COCCO2)=O)C1 CCC(C(=O)NCC1CCC(F)(CNC(=O)CSc2ccccn2)C1)C(F)(F)F CCCC(C)(O)C(=O)NC(CNC(c1nccnc1Cl)=O)C(C)C c1(CC)noc(C)c1C(=O)N(C1CC(NC(=O)CC2CCC23CCC3)C1)C c1(C(=O)NC(C)CCNC(=O)CNC(C2CCCC2)=O)ccc2ccoc2c1 c1(OCC)ccc(F)c(C(=O)NCCNC(c2nnc(O)cc2C)=O)c1N c1(C(N2CC(CCC)C(C(N3CCCCC3C)=O)C2)=O)cccc(C)c1F C1(O)(CC(=O)NC(C(=O)OC)C2CC2)CCN(Cc2ccnc(Br)c2F)CC1 n1(CC)ccc(C(N2CCCC(NC(c3ccc([N+](=O)[O-])s3)=O)C2C)=O)cc1=O c1(CC(C)C(N2CCCC2(C)CNC(=O)C(F)=C2CCCC2)=O)ccccc1Cl CC(=O)CC(C)(C)C(=O)NCc1noc(C(N)=O)n1.C12(CCCC1)C(=O)N2 C(=O)(C(C)(C)S(=O)(=O)c1ccc(Cl)cc1)NCC(CC=C)NC(=O)CNS(C)(=O)=O c1(C(N(C(=O)NC(c2nccc(C)n2)(C)C)C)C)ccc(Cl)cc1Cl c1(CN2CCCC2)ccc(C2CC2)cc1.C12CCCCN1C2=O CN1CC(NC(C2(C)CCN(C(N)=O)C2)=O)CCC1=O.C12CC1CC2O C1(CNC(C2C(OCC)CC2)=O)CCC2(CC2)C(=O)O1.OCC CS(=O)(=O)c1ccsc1C(N1CC2(C1)SCCC2NC(c1ccnnc1)=O)=O c1(CCN(CC)CC)nc2c(c(=NCC34CCC(C(N)=O)(CC3)CO4)[nH]1)COC2 CC1(C(=O)NCCN(C(c2nsnc2O)=O)CC2CC2)CC1(F)Cl C(=O)(NNC(=O)C(=O)NCC(c1ccc(F)cc1F)=O)C1CN(C)C(=O)N1 C1(C(=O)NCC#CCNC(C2COCCN2CC(F)F)=O)CCn2nnnc2C1 N1(C(C(C=C)O)=O)CCOCC(NC(=O)C(C2CCCCC2)OC)C1 c1(C(=O)NCCOC2CN(C(c3c(C)snn3)=O)C2)cc2cc(Cl)ccc2[nH]1 C(C)(C)(CCCC(=O)N1CCC(F)(F)CC1C)NC(CC1CN(C(C)=O)C1)=O C1(C)(C(N(CC(C)O)CCNC(=O)C(C)c2cc[nH]n2)=O)CC=CC1 c1(C(=O)NCc2cn(CCNC(C3(C)CCCO3)=O)nn2)ccnc(OCF)c1 C1(C)(CC)CC(NC(c2cccnc2-c2nnc(O)n2C)=O)CN1C(=O)C=C(C)C C(N=c1[nH]cnc2ccc(OC)cc12)C1(O)CN(C(C(COCC)N=[N+]=[N-])=O)C1 C(=O)(CC(O)CNC(=O)COC1CC1)NCC(C)(C1CC1)NC(=O)OC CCC(C(=O)N1CCC(NC(c2cnc(C(C)(C)C)[nH]2)=O)C(C)(C)C1)C(F)(F)F c1(NC(c2cc(CNC(C3C(OC)CCCC3)=O)oc2)=O)c(C)nn(C)c1C S(=O)(=O)(c1cccc(Cl)c1)N1C(COC(c2ccc(F)nc2)=O)CCC1 Cn1ncc(S(C)(=O)=O)c1C(=O)NCCCOCCCNC(=O)CCCF c1(CNC2CCN(C(Cc3c(C)cccn3)=O)C2)ccc(F)c([N+](=O)[O-])c1 C(=O)(C#CC(C)(C)CNC(C1C2CC3C(C2)C13)=O)N(CC(CC)CC)C Cc1ccc(F)c(C(=O)NC(C)C(C)NC(c2nn(C)cc2Cl)=O)c1O c1(OC(c2c(C)nc(-c3cnn(C)c3)o2)=O)ccc2ccccc2c1I Cc1cc(C)c(NCCCc2ccc(OC(F)F)cc2)cn1 CC(CCC(=O)NCC(C)(C1CC1)NC(c1cc(F)n(C)n1)=O)N(C)C N1(C(c2ccc(Br)cc2)C(=O)NC(C(=O)OC)C)CCC(O)(CC#N)CC1 c1(C(=O)NCC(=O)OC(c2ccc(Cl)c(Cl)c2)C)cccc(C#N)c1I c1(C(=O)NC23C(CN(C(C(C)OCC(C)C)=O)C2)C3)cc2c(Cl)nccc2s1 N1(C(CCNC(c2ccco2)=O)=O)CC2CC(NC(C34CC(F)(C3)C4)=O)CC2C1 C1(OCC#C)CCN(C(=O)NCc2cc(C)sc2-n2cccc2)CC1 C(=O)(C(C)CC(N)=O)NCC1(F)CC(NC(C(CC#C)O)=O)C1 C(C(C)C(F)C(=O)N1CC(C(N)=O)C1)NC(CC(CSC)O)=O CCC(C(=O)N1CCCC(NC(c2c[nH]c(=N)nc2C)=O)CC1)C(C)(F)F c1(C(N(CC(=O)NC2CC(CC)OCC2)CCC#N)=O)cc(F)ccc1F C=C1CCC12CC(C(N1CCCCC1CCNC(C1SCCCS1)=O)=O)C2 N1(C(CC2CC(C)C2)=O)Cc2occ(C(=O)NC3(C)CCOC3=O)c2C1 C(C(=O)N1CCCCC1C(C)(C)C(=O)NCC(CC(C)C)SC)(C(C)C)OC c1(C(N2C(CNC(C(CC)COC)=O)CC(F)C2)=O)ccc(N)c(F)n1 c1(C(=O)NCc2scc(C(=O)NC(c3cccnc3)CC)c2)ncc(N)cc1C N1(C(CC(=O)NCC2(F)CC(NC(=O)CC3CCOCC3)C2)=O)CCCCC1 C1(CC(=O)NCC2(OC)CN(C(=O)C(F)CC3CC3)C2)CCS(=O)(=O)C1 C1(C(=O)NCC(CC)O)CC(NC(c2cn(CCOC)nn2)=O)C1(C)C C1(C(N(C)CC2(NC(C(Br)=C(C)C)=O)CC2)=O)CC2(C1)CC1(CC1)C2 C12(CCN(C(=O)NC)C1)C(=O)N2.C1(NC(C(C2CCCC2)OC)=O)C2CCCC12 Cc1nn(CC(=O)N(CCNC(C2CCC(F)C2)=O)C(C)C)c2ncccc12 CC(C1CCCCC1)=CC(N1CC2CC2(NC(C2C(Cl)(Cl)C23CC3)=O)C1)=O C1(CC(N2CCC(C3N(C(CCCC=C)=O)CCC3)CC2)=O)CCC2(CC1)CC2 C12(C(N3CCN(C(c4cncc(OCC)c4)=O)CC3)=O)CCC(CO)(CC1)CC2 C=C1COCCN(C(C2COCC2NC(C2CCCN(C)C2)=O)=O)C1 Cc1nn(CCC(N2CC(C3(NC(C4CC4C(N)=O)=O)CC3)C2)=O)c(C)c1C c1(C(=O)NC2C(NC(C3(c4cc(C)no4)CC3)=O)CC2)ccccc1S(C)(=O)=O Cn1cccc(C2CC2C(=O)NC2(c3cc(=O)n(CC(F)F)[nH]3)CC2)c1=O Cc1nc([N+](=O)[O-])cn1CC(N1CCCC(C)(NC(=O)CCc2cnoc2)C1)=O N1(C(Cn2c(C)cc(C)n2)=O)CCC(C)C(NC(=O)NC(c2ccon2)C2CC2)C1 C(=O)(NN=c1cc[nH]c2ccccc12)NCCC(CCC)O c1(C(=O)NC2C(CNC(=O)CC3CCOCC3)CCCC2)cc2n(n1)CCO2 C1(C(NOCCOC)=O)(NC(=O)CC2CCCC23CC3)CC(F)(F)C1 C(=O)(C1=NNC(=O)CC1)NCCCCC1CN(C(c2c(CCC)nsc2N)=O)C1 c1(CCCNC(=O)CO)ccccc1.CN1CC(C(=O)NCCCNC(C=CC#N)=O)C1 C1(C(N(CC(C)O)CCNC(c2ocnc2C(F)F)=O)=O)CC2(CCC2=O)C1 C1(NC(c2ccc(OCC#C)cc2)=O)CN(C(=O)Cc2cccnc2)CCC1F N1(C(c2c(CNC(C(CSC)O)=O)ocn2)=O)CC(O)(C2CC2)C1 C12(COC(C(c3ccccc3F)(C)C)=O)C(=O)C3CC1C2C3 c1(COC)cc(C(=O)NC(c2nocc2C(=O)NC2CCSC2C)C)n[nH]1 N1(C(C(C)CS(C)=O)=O)CCC2(CC1)CN(C(=O)Cc1cccs1)CCO2 C1(N(C2CCCC3CC23)C(C2CCC(OCCO)CC2)=O)CCC2(CC1)CNC2 c1(-c2cn(C(C(N3CCCC(C(=O)NC(C)C)C3)=O)C)nn2)cc(O)ccc1Cl N1(C(C2N(C(CCC)=O)CCC2)=O)CCC(C)(C)C1CNC(=O)C(CC)C(C)C C=CCCC(C(=O)NCc1nc(C)c(C)o1)n1cc(CCCNC(N)=O)nn1 N1(C(c2cc(C(C)C)on2)=O)CCN(C(C)C)C(c2ccncc2)C1 N1(C(C(CC#C)(C)C)=O)CC=C(CCNC(C2CCCCC2C2CC2)=O)CC1 C1(C)(CC(=O)NCC2N(CCC)CCC2)CCCN(C(=O)C(=O)N(C)C)C1 N1(C(CSC(C)C)=O)CCCCC1CCN(C(=O)CCc1cncn1C)C N#Cc1ccc(O)c(C(N2CCCC(CO)(NC(=O)C=CI)C2)=O)c1 N1(C(CCc2n(C)ncn2)=O)CCC(F)C(NC(C2CCC3(CC2)CC3)=O)C1 N1(C(C(CCOC)(C)C)=O)CC(O)(C2(NC(C3(OCC)CCCCC3)=O)CC2)C1 Cc1cc(C(=O)NCCNC(=O)CCN(CC(F)(F)F)C)n2ncc(C#N)c2n1 c1(C(=O)NCC(CN(C(=O)C(C)(C)OC)CC)(C)C)cc2cc[nH]c(=O)c2s1 c1(OC(C)C(N2CCC(NC(c3c[nH]c(Br)c3)=O)C2)=O)ccccc1F C1(C(=O)NC(C)CCN2CCCC2)(NC(c2n[nH]cc2Cl)=O)CC(F)(F)C1 N1(CC(=O)NN(C(C(C)(C)CC2CC2)=O)CC2CC2)Cc2ccccc2C1 c1(C2(C(=O)NC(CC(C)NC(C(C)(C)OC)=O)C)CCC2)ccccc1F CN(C1CCc2c(F)cccc21)Cc1cn(-c2ccc(C(=O)O)cn2)nn1 Cc1onc(CC(N2CCN(C(=O)C=C3CCCCC3)C(C)C2)=O)c1C#N N1(C(CCC(C)NC(C2CCCC(CF)C2)=O)=O)CC2(CCOC2=O)C1 c1(OCC)ncc(C(=O)N(C2CCN(C(=O)CC3(OC)CCC3)CC2)CC)cn1 CCCC(C)CC(=O)N1CC(c2ocnc2CNC(C2CN(C)C(=O)N2)=O)C1 c1(OC(C)C)cccc(C(=O)NCn2cc(CO)nn2)c1.c12cc(ncn1)N2 c1(C(=O)NCC2(COC)CN(C(C(CCC)C)=O)C2)ccc2cnoc2c1 C1(NC(CCCOCC)=O)CC=C(C(=O)NC2CCCOC23CC3)C1 c1(C(=O)NC2(CNC(c3c(C(C)C)c[nH]n3)=O)CCOC2)scc2c1OCCO2 c1(C(=O)NCC(CCCC)NC(c2c(C)c[nH]c2CC)=O)ccc(Cl)c(C#N)c1 N1(C(CC2N(CC)CCC2)=O)CC2CC(C1)CN(C(=O)Cc1ccn(CC)n1)C2 c1(CC)cccc(C(N2CC(Cc3cnn(-c4ccccc4)c3)C2)=O)c1F C1(CC#C)(C(=O)NC(c2cnccc2C)C)CCN(C(=O)C(C)C2(O)CCC2)C1 N1(Cc2n(C)ncc2Br)CCn2cc(C(N3CC4CNC(=O)C4C3)=O)nc2C1 C=C=CCCC(=O)NCc1nc(C(=O)NC(C2(O)CCCC2)(C)C)co1 c1(CC(=O)NCC2C(C)(C)CCN2C(=O)Cc2ccon2)ccc2occc2c1 C1(C(N(C)CC2(O)CCOC2)=O)CC(NC(C2CCCSC2)=O)C(O)C1 N1(C(C2CC(C)N2C(=O)C(=O)O)=O)CCC(OC(C2CC2c2ccccc2)=O)CC1 N1(C(COCCNC(C2CC(C)N(C)C2)=O)=O)CCOC2CCCC12 C1(C(N(CC#C)CC=C)=O)CCC2(CC2)N1C(=O)CC1C(=O)NN=C1C CC(C(C)C(=O)NCCCCN(C)C(c1nn(C)c2c1CCC2)=O)C(C)(C)C N#Cc1ccc(C(N2CCC(CNC(=O)C(F)(F)CC3CC3)C2)=O)cc1O c1(CC)nc(C)sc1C(=O)NCC1C2CN(C(C3(N4CCCC4)CC3)=O)CC12 Cc1ccc(CNC(=O)C(Cn2cccn2)NC(c2ccc(CO)s2)=O)cc1 N1(C(c2c(C)ncc(Cl)c2)=O)CC2CC(NC(=O)C=Cc3ccnn3C)CC2C1 c1(NC(C2CN(Cc3cccc(O)n3)CCC2O)=O)cnc(O)nc1O C1(C(=O)NC)CC(C)(C)CN1C(c1ccc(C2CC2C)o1)C(=O)NC1CC1 N1(C(c2c(C(C)C)ncs2)=O)CC2CC1CC2N1CCC(c2ccccc2F)C1 C=CCCCC(C(=O)N(C)CCN(C)CCO)NC(C1(OC)CCSC1)=O S(=O)(=O)(c1ccc(C#N)cc1[N+](=O)[O-])NC(c1c(F)ccc(OC)c1Cl)=O n1(CC(N2CC(N(C(c3c(C)con3)=O)C)C2)=O)c(C)cc(O)cc1=O N12CCC(C)(C1)C2=O.C1(C(=O)OC)(OCC)CC1 N1(C(C(C)CNC(=O)CCc2nccn2C)=O)CCC(CO)(CO)C1 C1(c2n(C)ccn2)CN(C(c2ccc(Cl)o2)=O)CCN1C(=O)C1=C(Cl)CCC1 C(=O)(C1Cc2ccccc21)NC1CCN(C(c2cn(C3(C)COC3)nn2)=O)C1 C1(CC(N2CC(N(C(CCc3n(CC)ccn3)=O)C)C2)=O)CCCCN1C C=CC1CN(C(=O)Cc2cn(C)nn2)CC1NC(=O)CNC(=O)NC CC1(C)CCC(CC(=O)NC2CC(CCNC(c3ocnc3C3CCC3)=O)C2)C1 C1(C(C)(C)NC(c2ncn(CCC)n2)=O)CCN(C(c2ccn(CC)n2)=O)CC1 C1(C(=O)NC2(C(=O)NC(C3CCOC3)C#C)CCC2)CCC(C)CC1 Cc1ccc2nsnc2c1NC(=O)Cc1ccc(C(F)(F)F)cc1[N+](=O)[O-] C12(C(=O)NC34N(CC(=O)NCCCCCC5CC5)C(CC3)CC4)CCCN(CC1)C2 N1(C(C2N(C(c3cc(OC)n[nH]3)=O)CCCCC2)=O)CCC2(COC(C)C2)C1 N1(Cc2ncc(OCCOC)[nH]2)CC(NC(=O)Nc2ccccc2)CCC1=O c1(C(=O)NC(C2CCCCN2C(=O)C2=CCCCO2)C)cncc2cnccc12 C(=O)(C(C)(C)C(O)C(C)C)N1CCC(N(C(=O)C(=O)C(C)C)CC)C1 N1(C(C2CN(CCC)C(=O)C2)=O)CCN(C)C(CNC(=O)C(C)C(C)C)C1 C1(C(=O)NCC(CC=C)NC(c2coc(CCC)n2)=O)CCc2nc[nH]c2C1 C12(NC(=O)CCC3CC3)COC(CNC(c3cnoc3CC3CC3)=O)(C1)C2 C1(OC)(CNC(=NCC2CCC2)NC2CCS(=O)(=O)C2)CCCCCCC1 c1(NC(C2C3(CCN(C(c4cc(C(C)C)on4)=O)C3)C2)=O)ccc(Br)cc1C#N O=C(C(CC(F)F)C1CCC1)NC1CN(C(c2ccc(F)s2)=O)CCC1CO C1(N(C(=O)Cc2conc2C)CC)CCCN(C(c2nc(C)oc2C)=O)C1 CC1(C)CN(C(c2c[nH]c(=O)c3ccnn23)=O)CCC1Cc1nn[nH]n1 C1(N(C)C(C2CCC3(CC3)C2)=O)CC2CC1N(C(=O)CCc1cc[nH]n1)C2 c1(C(=O)NC2C3CN(C(CC(CC)C)=O)C2CC3)coc2c1C(=O)CCC2 C(=O)(C1CCCc2n[nH]cc21)NCCC1CC(NC(C2(C)CCC(F)(F)C2)=O)C1 C1(C(=O)NCC2CC(OCC)C2)CCC(C)CN1C(=O)C(C)Cn1cccn1 c1(OC(C)=O)ccc(C(=O)NC(C)CCN(C(=O)C(F)C2CCCC2)CC)cc1N C1(CN(C(CCOC(c2ccc(C)cc2)=O)=O)C)COc2ccccc2O1 C(C(C)C(=O)NCC1(F)CC(NC(=O)Cn2cnc(=N)[nH]2)C1)OCC c1(C(N(C)CC2(NC(c3c(CC)nn(C)c3)=O)CC2)=O)ccc(C)c(C)c1 C1(CNC(C2C(c3ccc(N)cc3)OCCC2)=O)(CO)COCC2COCCN12 N1(C(C2(C)CN(C(CCC(C)OC)=O)C(C)(C)C2)=O)CC2OC(=O)N(C)C2C1 c1(CC(=O)N(CC(C)NC(=O)C(N2CCOC2=O)C)C)cccc(F)c1Cl c1(CC)cscc1C(N1CC(F)(C(=O)NC23CCCC2C3)C1)=O c1(C(C2CC2)NC(COCCCOC)=O)cc(O)ncc1C(=O)NC1CC1 c1(CNC(COC)=O)cc(C(=O)NCC2CC3C=CC2C3)n(C)n1 c1(C(N2CC(C(N(CCCF)CC)=O)C(C)(C)C2)=O)cccn2nccc12 N1(C(c2cn(CC)nc2C)=O)CCCC1C1CCCN1C(C1CCCC1OC)=O CC1(CNC(C2CCS(=O)(=O)C2)=O)CCCN(C(C2CC3(C2)CC3F)=O)C1 C1(C(=O)OCCN(CC#N)CC)CCCC1(C)CNC(=O)CSC(F)F c1(C(N2C(C)CC(CNC(c3cscn3)=O)C2)=O)ncnc2c1CCCC2 c1(NCC(=C)Br)ccc(S(=O)(=O)NCC2(C)CC3CC3C2)c(Cl)c1 c1(CC(=O)NC(C)C(C)NC(C2(CO)CCOCC2)=O)ccc(Br)cc1C#N C(=O)(CC(F)(F)C(F)F)N1C2CCC(CNC(c3cncc(CO)c3)=O)(C2)C1 c1(CCC(N2CCC(O)(CNC(C(COCC)(C)C)=O)C2)=O)ccc(F)cc1Cl C1(C(=O)NCC(C)CNC(=O)CCC(=O)c2cccs2)CNC(=O)CC1C c1(OCC)nc2ccc(C(=O)N(C)CCN(C)C(c3scc(C)c3C)=O)cc2[nH]1 Cc1sccc1C(N1C(CC(N2CCC(C3CCCO3)C2)=O)CCC1)=O c1(CCC(N2CCN(C(CCS(C)=O)=O)C(C(F)F)C2)=O)cnc2n1CCCC2 c1(C(=O)NCC(C(=O)NC2(COCC)CCC2)O)cc(C)cc(F)c1 C(=O)(C1=CCCCCC1)NCC12CC(NC(c3ccc(C#N)o3)=O)(C1)C2 c1(C(=O)NC2(CC=C)CN(C(=O)C(C)(O)C=C)C2)cc(Cl)c2ccccc2n1 c1(NC2CCC(C(N(C)CCOCCNC(c3ccno3)=O)=O)C2)ccccc1Br C1(CNC(c2c(COC)noc2)=O)CN(C(C2CC(C)(C)C2)=O)CCCO1 c1(C(=O)NC2CCC(F)(CNC(C3CC34CCC4)=O)C2)c[nH]cc(F)c1=O c1(CC(C)=O)c(CN2CCCC2C=CC2CC2)oc2ccccc12 CC1(NC(c2cccc(Cl)c2Cl)=O)CCCN(C(c2cnsc2)=O)C1 C1(CC)CCN(C(c2cnc[nH]c2=N)=O)C1C(=O)N(C)CCC1CCCCC1 c1(COC)cccc(NC(N2CCC(CSc3cccc(OC)c3)C2)=O)c1 C(=O)(C1=C2CCCN=C2NN1)NC1C(CNC(Cc2c(C)nc(C3CC3)s2)=O)C1 C1(NC(C(=O)Nc2ccc(C)cc2)=O)(NC(=O)C2CC2)CCCC1C N1(C(C2CCC(C)C2)=O)CCC2CCN(C(C3CCC4CC34)=O)CC2C1 C(=O)(CCCCNC(C)CC1CCCO1)NCCCN(CCC(C)C)C N1(C(C(C(CC)C)O)=O)CCC2(CC1)CCN(C(C1CSCN1C(C)=O)=O)CC2 N#CC1(C(=O)NCC2CCC2NC(C2CC(n3cnnc3)C2)=O)CC=CC1 C1(NC(c2c(CC)nn(C)c2)=O)COC2(C1)CN(C(=O)CS(=O)CC)C2 CC#CC1CN(C(=O)C(C)(C)CN(C(=O)CCOCC2CC2)C)C1 C1(C(F)F)(OC)CC(C(=O)NCC(CNC(=O)C(O)Cc2ccccc2)OC)C1 c1(C(=O)NCC2(NC(c3c[nH]nc3C3CCOC3)=O)CC2)cnn(C)c1.C1CC1 c1(C2(C)COC2)nocc1C(N1CCCC1CNC(c1sccc1C(F)F)=O)=O N1(C(C2CN(CC)C(=O)C2)=O)CCOC2(CCN(C(=O)CCC3CCCO3)C2)C1 C1(O)(CNC(c2ccnc(O)c2)=O)CCCN(C(c2[nH]nnc2C2CC2)=O)C1 C1(CCC)CCC(NC(C2(n3cc(-c4n[nH]cc4C)nn3)CC2)=O)C1 c1(CCC)cc(C(=O)N(CC)CC2CCN(C(=O)C(F)(F)C3CC3)CC2)ccn1 C1(NC(c2cnc(C)n2C)=O)CCN(C(C2CC2(F)F)=O)CC(C)(C)C1 C(=O)(C(O)C(C)(C)C)NCc1ccc(N2CCN(C(C(CC)O)=O)CC2)cc1 CC1CCN(C(=O)CCNC(=O)CO)C1CNC(c1ncsc1C1CC1)=O N1(C(c2ccn(C(C)C)n2)=O)CCC2(CCCN(C(=O)CCCF)C2)C1 C1(CNC(c2cnsn2)=O)CCC2(CCC2)CN1C(=O)C=C(C1CC1)C1CC1 N1(C(c2cccn2CC)C(=O)NCC(=C)C)CCCC1C1CCCCO1 C(N=C(NC(C)C)N1CCC(C(N)=O)C1)c1cccc(C(=O)NC)c1 C1(C(N(CCN(C(c2ccc(C)c(C#N)c2)=O)C)C)=O)CC2CCCCCCC12 C(C(C(C)C(C)C)NC(=O)CN(C)Cc1ccccc1)NC(C(C)(C)SC)=O c1(C2C(N(C)C)CCC2)nc2nn1C2.c1(Cn2cccn2)ccc(Cl)s1 CC1CCCC(C(N2CC(NC(=O)C(N3CCCC(O)C3)C)CC2C)=O)CC1 CCCCN=C(NCCS(=O)CC(F)(F)F)N1CCN2C(=O)OCCC2C1 C1(O)(CNC(c2cncs2)=O)CCN(C(=O)COCCc2cccs2)C1 c1(OC)cc(C(N2CCN(C(=O)C(C)O)CC2C(F)F)=O)c(N)cc1F N1(C(CONC(C=CCC(C(=O)NC)C)=O)=O)CCc2sccc2C1CNC c1(SCC(=O)NC(C(CO)NC(C2(C#C)CCC2)=O)C)ccc(C)c(C)c1 C1(NC(C(C)C)=O)CC2(CCCN(C(c3nc(Cl)c(Cl)s3)=O)C2)C1 c1(OC)cc(CN(C)Cc2cc(-c3ccccc3C)cn(C)c2=O)ccc1OC n1(CC)nccc1C(N1CCCC1CN(C(=O)C(C1CCC1)OC)C1CC1)=O c1(C(=O)NC2CC(CNC(=O)CCCCN3CCCC3)C2)scc2c1OCCO2 c1(C(N2CC(CCC)N(C(c3occc3C)=O)CC2)=O)ccc2occc2n1 c1(C(N(C)CCC2CCCCN2C(c2ccsc2)=O)=O)cccc(C#N)c1 N1(C(C2CCN(C)C2)=O)CCC2(CC1)CCN(C(=O)CCCCc1cnc[nH]1)C2 N1(C(=O)CC2CCC2)CCCC2CN(C(C3(CO)COC3)=O)CC12 N1(C(c2nc(CC)oc2)=O)CCCCCC1CNC(C1CC=CCC1C)=O C1(CNC(c2cn(CCC)c(C)n2)=O)CN(C(C2CC(C)(C)CO2)=O)CC1(F)F C1(c2ccccc2)(CNC(C(=O)N(C(C2CCOCC2)C)C)=O)CCOC1 c1(C(=O)NCCC(CNC(C(CC)COC)=O)O)nsc2ccccc12 C1(NC(C(C)OC2CCCC2)=O)CCN(C(C2CC2CC(C)(C)C)=O)C1C c1(C(N2CCCC(CNC(C3C(C)C3)=O)CC2)=O)c(Br)ccc(N)c1F N1(c2nc(C)nc(=N)[nH]2)CCC2(CCCN(C(c3cnn4ccncc34)=O)C2)C1 n1(CC)nc(C(N2CCOC(C(=O)Oc3snc(C(C)=O)c3C#N)C2)=O)cc1C C(=O)(C1=CCCCCC1)NC(CC1CN(C(C2C(C)C2C)=O)C1)C c1(CCNC(C(C2CCCO2)NC(C(C)C)=O)=O)ocnc1CO N1(C(C=CCC(C)C)=O)CCC(OCCN(C(=O)C(F)(F)CO)c2ccccn2)CC1 C1(CCOC)CN(C(C2CN(S(C)(=O)=O)C2)=O)CCN1C(c1cc(C)ns1)=O C(=O)(C(F)(CNC(C1(C(C)C)COC1)=O)C(C)C)N1CCN(C(CC)C)CC1 CC1(C(N)=O)CCN(c2cc(NCC3CC3Cl)ncn2)C1 C#Cc1c[nH]nc1C(N1CC(NC(C2CCC23CCC3)=O)CC1CO)=O C(CC(C(=O)NCc1cscn1)NC(C1C(C)(C)C1(F)F)=O)N(C)C CC(C)(CCC(=O)OC(C1CC12CN(Cc1ccccc1)C2)=O)[N+](=O)[O-] N1(C(CCCCC=C)=O)CC2CCCCC2(NC(C23CCC(C)(C2)OC3)=O)C1 N1(C(C=CC)=O)CCC(NC(c2cccc(Cl)c2)=O)C(CO)C1 N1(C(=O)COC2(Cc3ccc(F)cc3)CC2)CC(NC(c2cscn2)=O)CC(O)C1 c1(C(=O)NC2(C)CCN(C(C(C)(C)N(C)C)=O)C2)cc(F)ccc1O C12(NC(c3cc(F)ccc3Cl)=O)CCC(C(=O)Nc3ccsc3)(CC1)CC2 c1(C(=O)NCCC(C)NC(=O)Cn2cnc(Br)n2)cc(N)nc(Cl)c1 C1(NC(=O)C2=CCCCO2)CC2(CCCN(C(=O)CCn3ccnn3)C2)C1 N1(C(C2(NC(=O)Cc3cncnc3)CCN(C)C2)=O)CC(C2(C)CC2)C1 C1(NC(c2ccc(CNC(c3c(OC)scc3)=O)cc2)=O)CCC2(CCC2)C1 c1(CC)nc(Cl)c(F)c(=NC(C)CNC(=O)C(C)C(C)C)[nH]1 C(=O)(C(F)(CNC(=O)CC(C1CC1)C1CC1)C(C)C)N1CC(OC)C(OC)C1 C1(C(CC)NC(=O)NC(c2cccc(OC(F)(F)F)c2)C)CCC(F)(F)CC1 C(=O)(C(C(F)(F)F)OC(C1CCN(S(=O)(=O)CC)C1)=O)OCC N1(C(C(C)C2CCCC2)=O)CC(C)CN(C(=O)C(F)=CC2CCCC2)C(C)C1 C12(C(=O)NC3C(NC(C(CCC)(C)C)=O)CCC3)C3C4C1C1C2C3C41C(=O)OC c1(C(N2CCC(CSC)C2)=O)ccc(-n2cc(CCC(=O)O)nn2)cc1 S(=O)(=O)(c1cccc2c1OCO2)N1CCC(N2C(=O)NC(=O)CCC2)CC1 C1(CC)CC(C(=O)NOCCO)CCN1C(=O)C#CC1CC1 C1(NC(CCCN2C(CC3(CNC(=O)OCC)CCCO3)CC2)=O)CN(C)CCO1 N1(C(CCSCC)=O)CCCC(CN(C)C(C2CC(=O)N(C(C)(C)C)C2)=O)C1 C1(C(=O)OC)CCC2(CCC2)N1C(c1c(O)nnc(C)c1C)=O c1(C(N(C2CCCN(C(c3cc(C)n(C)c3)=O)C2)CC)=O)cc(Cl)c(F)cc1C c1(C(=O)NCC2CC(C)N(C(C3CCSC3)=O)CC2)c(F)ccc(Cl)c1F C1(NC(C2(C)CCOCC2)=O)CCC12CN(C(=O)CNC(c1ccccc1Cl)=O)C2 c1(C(N(CC(CNC(C2CC(C(C)C)C2)=O)C)C)=O)[nH]c2ccc(Cl)cc2c1Cl C(=O)(C(O)CC(C)C)NC(CCOCC)C(=O)NCC1(CO)CC=CC1 c1(OC)ncc(C(=O)NC2CC(C)N(C(=O)COc3cccc(F)n3)C2)c(C)n1 C1(NC(C(C)C(C)(F)F)=O)CCC2CCN(C(c3n[nH]cc3C3CC3)=O)C1C2 C(CCC1CC1)(C(=O)NCc1cccnn1)NC(C(C)OC1CCCC1)=O c1(C(C)NCC(C2CCOC2)C)ccc(N2CCCCC2)cc1 CC(C)CCCC(C)C(=O)NC(CCC(=O)N1CCC(C(F)(F)F)C1)C(C)C c1(-c2cn(SCCNC(C[SH](C3CCCC3)CC(C)=O)=O)nn2)ccc(C)c(O)c1 O(NC(=O)C1=NOC(CNC(C2(CCF)CCC2)=O)C1)CCOCC C(=O)(C1CCCc2scnc21)C(C1CCCCN1C(N)=O)=O.C12(OC)CC(CN)(C1)C2 N1(C(=O)Nc2c(C)ccs2)CCn2ncc(-c3cccc(N4CCCC4)c3)c2C1 N1(C(C2(S(C)(=O)=O)CC2)=O)CC2CCN(C(c3cc4ncccc4[nH]3)=O)C2C1 C1(C)(CC)CCC(C(=O)N(C)CC2(O)CN(C(c3ccco3)=O)C2)O1.C1(=O)CN1 Cc1ccc(F)c(C(N2CC(NC(c3[nH]ccc(=O)c3C)=O)CC(C)C2)=O)n1 Cn1cc(C(N2CC(N3CCN(C(C4C=CC=CC=C4)=O)CC3)C2)=O)ccc1=O C1CCN(C(c2ccc(C(=O)O)nn2)=O)CC1.C1(COCC)CCN(C(C)C)C1 C(=O)(C1=C(C)OCCC1)NCC(C)N(C)Cc1ccc(NC(C)=O)nc1 C=CCC(CNC(c1ccc(C)nc1C)=O)C(=O)N1CCC(C(=O)NC)CC1 c1(C(=O)NC2CC(NC(c3cccc(OCC)c3)=O)C2)cnc2ncccn12 C(F)(c1ccccc1)=CC(=O)NCC(C1CCCCC1)NC(C1(CC)CCCO1)=O c1(C(=O)NCC(C(C)C)NC(CSCCOCC)=O)cc(C(F)(F)F)cc(Cl)c1 C(=O)(C(C)(F)C(C)(C)F)NCCC1(NC(Cc2n[nH]c(=NC)s2)=O)CCC1 C1(OCC)COCCC1NCc1ncc(-c2ccccc2CO)cn1.C1C(=O)O1 c1(C(=O)NCC2N(C(CC)=O)CC(O)C2)ccc(N)c2cnccc12 C1(N(C)C(c2cnc(C3CCCO3)s2)=O)CN(C(C2CC(O)C2)=O)CC1(C)C C1(NC(C2(OC)CC2)=O)CN(C(=O)CCc2ccc(N)cn2)C2(CCC2)C1 C1(C(N(C2CN(C(=O)C(Cc3ccsc3)C3CC3)C2)C)=O)CCS(=O)(=O)N1 C12(NC(C3C(NC(C4CCN(C)C4)=O)CCC3)=O)CCCN(CCC1)C2 C1(CN(C(=O)Cc2ccnn2C)C)C2CN(C(c3cc(N(C)C)ccn3)=O)CC12 C(N=c1cc(F)nc[nH]1)C1N(C(Cc2c(CC)c(F)ccc2)=O)CCC1 CC(C)CC(=O)NC1(C(=O)N(CCCCN(C)C(C2CCC2C)=O)C)CC1 c1(C(N2C(CCNC(C3CCCC4(CC4)C3)=O)CCCC2)=O)ccc(O)nc1Cl CC1CN(C(=O)C(C)(CO)N(C)C)CC1(C)CNC(c1[nH]ccc1C1CC1)=O c1(C(=O)NCC(CO)NC(c2c(C)[nH]cc2)=O)ccc(Cl)cc1[N+](=O)[O-] N1(c2c(C)cc(C(F)(F)F)cc2)CC(OC(C)(C)C)CC12CCOCC2 N1(C(CCc2n(C)ncc2)=O)CC(C2CC2)(C(=O)NCC2CCCC(C#N)C2)C1 C1(NC(=O)CC2(C#N)CC2)CCN(C(c2ccc(CO)s2)=O)C1.CCCCSC(F)F C1(CC(=O)OC(c2cscc2F)C)CCCN(C)C1 CON(CCC(=O)NCC1CC(O)CCO1)C(=O)C(C)(C)COC c1(C(N2CCC(CNC(CCC=CC)=O)C(C)C2)=O)cc2ccccc2cc1F C1(C(CC)C)CCN(C(=O)CCN(CCO)C(C2CC(=O)CCO2)=O)CC1 Cc1ccc2c(c1)C=C(C(=O)N1CCCC(O)(CNC(c3cnn[nH]3)=O)C1)CO2 CC(C)CCCCC(=O)NC(C)C(C1CCCCC1)NC(=O)CN1CSCC1=O C(C)(CC(C)C)(c1n(C(CC)C)nnn1)NCc1cnn(CC)c1C(F)(F)F C12(C(=O)NC(C(CO)NC(Cc3nc(C)oc3)=O)C)CCC(CC1)C2(C)C N1(C(CC(=C=C)C)=O)CCCC2C(NC(c3cc(CC)no3)=O)C(C)(C)C12 N1(C(c2ncn(C(C)C)c2)=O)CC2CC1C1CC21 c1(C(N2CCC(C(=O)NCc3cnco3)CC2)=O)cc(Br)ccc1[N+](=O)[O-] C(=O)(C(F)(F)C(F)(F)F)N1CCCC(CNC(=O)Cc2cc(F)ccc2Cl)C1 C1(NC(C2CCN(CC)C2)=O)CN(C(=O)C(C)(C)CF)CCC1(C)C N1(C(C(C)(C)OC)=O)CC(Nc2ccc(N3CC(O)C3)nc2)C(C)(C)C1 C=CC(C)(C)C(=O)N1CCC(C(C(C)C)NC(=O)C(C2CCOCC2)F)CC1 C(CCCCC(=O)NCc1nc(CNC(C23CCCCC2C3)=O)cs1)OC N1(C(C2N(C(CSCC#C)=O)CC(=O)NC2)=O)C2CCCC1COC2 c1(COC)cccc(C(=O)N(CCC(C)NC(c2ccc(C(F)(F)F)s2)=O)C)c1 C1(CC(N2CC(C(C)NC(Cc3cc(C(C)C)no3)=O)C2)=O)NC(=O)NC1=O CCCC(CNC(C12CCCC1C2)=O)C(=O)N1CCOCC(C(=O)OC)C1 c1(C(=O)NCCC2CCC(NC(c3c(C)con3)=O)C2)c[nH]cc(Br)c1=N C#CC1CC(NC(=O)CC2(N(C)C(c3occc3C(C)C)=O)CC2)C1 C1(CCOC)CN(c2ccnc(N3CCOC(CS(N)(=O)=O)C3)n2)CCO1 C1(C(N(C)CC2CCCN2C(=O)CCc2ncccn2)=O)CCc2ccnn2C1 C1(C(N2CC3C(CNC(C4CCCN(C)C4)=O)(C3)C2)=O)CN2CCCN1CC2 N1(C(c2cnn[nH]2)=O)CCC2CCC(C1)N2C=O.N1(C(N(C)C)=O)CC(C(=O)N)C1 C(CC(=O)NNC(=O)C(C)Nc1cccc(C)n1)c1cccc(OC)c1 N1(C(c2c(CNC(c3c(C)ccc(C)n3)=O)cco2)=O)CCC(C2=NOCC2)C1 C(C)(C(O)C(=O)NC1CC(F)(CNC(c2cc(C(C)C)nn2C)=O)C1)OC C1(NC(C(c2c(C)n[nH]c2C)C)=O)CC12CCN(C(=O)C(C)N=[N+]=[N-])CC2 N1(C(C2CN(C(=O)CN3CCNC3=O)CC(C)O2)=O)CCn2nccc2C1 C(c1c[nH]c(=N)c(C)c1)=CC(=O)NCC1(F)CC(CNC(C(CC)(C)OC)=O)C1 C1(NC(CSCC(C)C)=O)CC(NC(c2ccncc2N(C)C)=O)C(O)C1 N1(C(COC(CC)C)=O)CCOC2(C1)CN(C(=O)C=Cc1cc(C(=O)OC)co1)C2 C1(CC2(CC(C)(F)F)CC(O)C2)CCN(C(=O)OC(C)(C)C)CC1C(C)(C)C c1(C(N2CCC(OCCNC(C=CC(C)(C)C)=O)C2)=O)cnc(N)c(Br)c1 C(CC(C)C)(C(=O)N1CCC(OC)C1(C)C)NC(c1c(C(=O)OC)cncn1)=O C(CC(C)C(=O)N1CCN(c2ccc(NC(=O)C=CCO)cn2)CC1)=CC c1(C(=O)NC2CC2)c(N(C2CCCOC2C)CCOCC)nc(C)nc1Cl CC(C)(C)C(C)(O)C(=O)NC1CCC(NC(=O)CCc2cncc(F)c2)CC1 C(C(O)CC(=O)NCCN1CCC(NC(=O)CC2OCCO2)CC1)N(C)C c1(C(=O)NC(c2nnnn2C2CC2)C)[nH]ccc1CNC(=O)C1CC1 c1(CNC(=O)NC(C(=O)OC)C(C)C)cc2cc(C)c(C)cc2o1 c1(CC(N2CCCN(C(=O)CC3C=CCC3)CC2)=O)c(F)c(F)cc(F)c1F c1(C(N2C(CN(C(=O)C(F)(F)CO)C)COCC2)=O)[nH]c2ccccc2c1C#N C1(CNC(C2C(CC)C2)=O)COCCN(C(=O)C=Cc2cccs2)C1 c1(C2C(C(=O)NC3CC(C4N(N=O)CCC4)OCC3)C2)ccc(F)c(Cl)c1 n1(CC)nc(C)c(C(=O)NCCC2CCCN(C(c3cnns3)=O)C2)c1Cl N1(C(C2(OC)CCC2)=O)CC2(CCC(NC(=O)CSc3ccc(F)cc3)CC2)C1 C=CC(C)(C)CC(=O)NC1CC2(C(N3CC(C(N)=O)(OC)C3)=O)COC1C2 C1(C(=O)N)CC2(CCO1)CC2.C(C)(C)(CC(=O)NCCC1(CO)CC1)OC c1(C(N2CC3C(CCNC(C(C)=C(CC)C)=O)(CC3)C2)=O)cnn2c1OCCC2 C1(CCC(C)C)CCCN(C(=O)CC2CNCCO2)C1 c1(C(c2n(C(CC)C)nnn2)Nc2cnn(CCO)c2)cc(I)cn1C C12(C(N3CCC(CC(=O)OCC4CCC4)CC3)=O)COCC(C1)C2 c1(C(N(CC(C)N(C(c2cn(CC)nc2)=O)C)C)=O)c(O)cccc1Cl c1(OC(CC)C(=O)NCC(F)CNC(C2(CCO)CC2)=O)cccc(C)c1 c1(NC(C2CCC(F)C2)=O)ccc2cc(C3CCCCC3)[nH]c2c1 c1(NC(C)=O)ccc(C(=O)NC2CCCC2CNC(c2cc(CO)[nH]n2)=O)cc1 c1(C(N(CC(C)(C)NC(c2cc(C)nn2C)=O)C)=O)cc2cccc(F)c2s1 C12(CC=O)CCC(CC1)CC2.O=C(C(O)Cn1cncn1)NC1CCOC1C1CC1 c1(NC(C(=O)NC(CCCN(CC(=O)OCC)C)C)=O)c(F)cccc1Br C1(NC(C2(C)CC=CCO2)=O)CCCCN(C(=O)Cn2cnc(C(F)(F)F)n2)C1 C1(S(C)(=O)=O)(C(=O)NCC(CNC(c2c(N(C)C)nccc2)=O)O)CCCCC1 CCC(CC)C(C(=O)NC1CC=C(C(=O)N2CC(C)(OCC)C2)C1)OC N1(N(C(C)C)CC)CCC(C=O)CC1C.C(=O)(C(CN(C)C)C(C)C)N.C1C=CC1 c1(C(=O)NCC2CC(O)(CNC(C3(C)CC=CC3)=O)C2)ccc(S(C)(=O)=O)s1 CC1OCCOC1C(N1CCC(O)(CNC(=O)CCCNS(C)(=O)=O)C1)=O CC(C)CC(CNC(=O)CC(C)C1CCCO1)C(=O)N1CCOC(CCO)C1 C1(C(=O)NCCNC(=O)COCCOc2ccsc2)CCN(C2CCC2)C1 N1(C(c2ccc(CC)[nH]2)=O)CC(Nc2snc(Cl)c2C#N)C(C)(C)C1 N1(C(Cn2c(C)nnn2)=O)CCCCC1CN(C)C(C12CCC(C1)C2)=O C=CCC(CC(C)C)C(=O)NC(CCSC)C(=O)NCC(=O)OCC N1(C(c2cc(C)sc2)=O)CC2CC3CC2C1C3NC(c1cn2ncccc2n1)=O c1(C(N2CC(CNC(c3scc(C)c3)=O)C3C2C3)=O)ccc(Cl)c2cccnc12 C#Cc1cc(F)c(C(=O)N(CCNC(=O)C(CC(C)C)OC)C2CC2)c(F)c1 C(=O)(C(C)(C)CC#N)NC1CC(NC(C(C)c2ncco2)=O)C1 CCC(CC)CCCC(=O)N(C(CC)CC(=O)NC1CCOC1C)C C1(CC)CCCCC1OCC(=O)N(C)CC1CCCN(C(=O)C(C)(C)CO)C1 N1(C(CNC(=O)Cn2cccn2)=O)CC(C(=O)OCC)CC1C CCC(C(=O)NC1CCN(C(=O)CSC2CCOC2=O)CC1)C(C)(C)CC c1(C(=O)NC(C)CSC(F)F)csc(CNC(C2CCC(F)C2)=O)c1 N1(C(C=CCCC)=O)CC2CC(NC(c3ncc(C)cc3C)=O)CC2C1 C1(CC)C(N(C)NC(C2CNC(=O)N2)=O)CCN1C(=O)C=CCc1ccccc1 n1(CC(=O)NCC23CCC(CN2C(=O)C(F)F)C3)ccc2ccccc2c1=O Cc1ccc(C(=O)NC2CCCC2NC(c2cn(-c3cccnc3)nn2)=O)o1 C(CCCSc1cccc(Br)c1)(C(=O)O)NC(=O)NCCC(=O)OC C1(C(=O)NOC2CCCC2)CC(F)CN1C(=O)Cc1cccc(F)c1 C#CC(CNC(=O)C(=O)NCC(C)COc1ccccc1)CC Cc1nc(C(N2CCC2CNC(=O)CC2CCOC(C)(C)C2)=O)c2ccccn12 c1(NCc2ccc(C#N)cn2)cc(C#N)c(Cl)cn1 C1(NC(c2cc(CNC(Cc3n(C)nnc3)=O)nn2C)=O)CCOC(C)(C)C1 C(CC(C)(C)c1ccccc1)=C(C)Cl.N1(C(C)=O)CCCCC1 CC(CNC(c1ccc(CF)cc1)=O)CC(=O)N(C)CCN(C)CCO c1(CNC(CC=CC)=O)ccc(O)c(OC(c2cnc(SC)nc2)=O)c1 C1(NC(C2CC(=O)OC2)=O)CC2CN(C(=O)CC3(O)CCCOC3)CC12 c1(CC)ccccc1C1(C(N2CCC(N3CC=CC3)C2)=O)CCCC1 C1(C(=O)NCCOCCN(C)C(C23COCC2C3)=O)CN2CCC1CC2 C(=O)(C1CNc2ccccc21)NCC1(CCNC(C(c2ccnn2C)C)=O)CC1 C1(NC(=O)CC23CCCC2CCO3)CCN(c2c(OC)cccc2)CC12CCC2 c1(C(N2CCN(C(c3cnc(OC)s3)=O)C3C2C3)=O)ccc2c(c1C)CCC2 c1(C(N2C(C3(NC(CCNC(COC)=O)=O)CC3)CCC2)=O)c(C)csc1Cl C1(NC(C(c2ccc(C)s2)C)=O)COCCC1NC(=O)C1=CSCS1 C1(c2n(CC(C)CO)nc(-c3ccsc3)n2)CC12CCCc1ccccc12 CC(C)C(CCNC(=O)Cn1nnc(C2CC2)n1)NC(c1ccns1)=O c1(CC)c(C(=O)N(CC(O)CN(C(=O)CCC2CCC(=O)C2)C)C)cccc1C Cn1nc(C(N2CCN(C(=O)COCC3CCCO3)CC2)=O)c(Br)n1 c1(C(=O)NC(C)CCNC(C2CN(CC(F)(F)F)C2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 C(=O)(C1=CN=C2N=CNN2C1)NCC1(O)CC(CNC(C2CC=C(C)CC2)=O)C1 c1(C(C)C(N2CCC(N(C(=O)C(=O)NC)CC3CC3)CC2)=O)ccc(Cl)c(Cl)c1 C1(C(N2CCC3(NC(CN(C(C)C)C)=O)C(C2)C3)=O)Cc2cc(F)cc(F)c2O1 c1(C(=O)NC(C(=O)NC(C=C)C(F)(F)F)CCF)cc(O)cc(F)c1 N1(C(C(C)C)=O)CCC(C(F)(F)F)C(NC(c2ccccc2-n2ccnc2)=O)C1 C1(C(=O)NCC(C(=O)OC)O)CC(NC(=O)C(C)C(C)C)C(O)C1 c1(C(N2CCC(NC(Cc3nc(CC)sc3)=O)C2)=O)cnc2sc(C)cn2c1=O C(=O)(C(CNC(=O)CCS(N)(=O)=O)C(C)C)NC(C(=O)OC)CO C1(NC(=O)C2=CCOC2)CCCC(CC2C(C(C)(C)C)C2)C1 C=CC1CCCN(C(C2CCN(C(C3(C)CC(C#N)C3)=O)C2)=O)C1 c1(NC(C)CCNC(=O)C(N2C(C)CCC2C)C)nc(Cl)nc2[nH]c(O)nc12 N1(C(c2[nH]cc(CC(C)C)c2)=O)CCC2(NC(=O)C(O)CC(C)(C)C)CCCC12 N1(C(c2cc(C)nn2C)C(=O)NC2CCCC2)CCN(C(CSC)=O)C(C)C1 CCCCC(C)(F)C(=O)NCC1CCCN(C(c2cnncc2C(F)(F)F)=O)C1 N1(c2ncc(SCC)cn2)CCN(C(c2cc(C)on2)=O)C(C(C)C)C1 C1(NC(C=CCC2(NC(c3ccc(C)cn3)=O)CCC2)=O)CC(CSC)C(O)C1O C#CCCC(O)C(=O)NC1CC2CC1N(C(=O)CCc1cc(C)no1)C2 C1(C(=O)NC(CNC(C(C(C)C)OC)=O)CO)COC2(CCC2)C1 C12(C(N3CC(C)C(CNC(c4cc[n+]([O-])cc4)=O)C3)=O)CC(C)(CCO1)C2 N1(C(C2(OC(C)=O)CC2)=O)CC(F)(CNC(C2CC2(C)Br)=O)C1 C1(NC(c2ccncc2Cl)=O)CCCC2CN(C(C3CCCC4CC34)=O)CC12 Cc1c(C(N2CC(NC(c3cccc(CCO)c3)=O)C(O)C2)=O)cncc1N C1(NC(c2cccc(-n3cnnn3)c2)C)CC2CCC(C1)N2 N1(c2n(CC=C)c(CCO)nn2)CC2CC(F)(C2)C1 C12(NC(C(C3(C)CC3)NC(=O)C(C)(C)C)=O)CCN(CC1)C2 c1(C(N2CC(NC(C3N(C(=O)NC)CCC3)=O)C(F)C2)=O)cccc(C)c1C#N N1(C(CSc2ccc(OCC)cc2)=O)CCC(C2CC2)(C(=O)NC2CC23CC3)C1 C1(c2nnc(N3CCC(C(F)F)CC3)n2CC#N)(NC(C)(C)C)CCCCC1 c1(C(=O)NCC(C(C)(C)C)NC(c2cnn[nH]2)=O)cc(F)ccc1C1CC1 c1(C(=O)NCC(CO)NC(c2cc(CC)ncn2)=O)n[nH]c2ccc(OC)cc12 c1(OC)cc(C(=O)NCC(C)CNC(=O)C(COC)N(C)C)ccc1S(N)(=O)=O c1(C(N2CCCC(F)(CNC(C3C(C)C3)=O)C2)=O)cc2c(OC)cc(Cl)cc2[nH]1 c1(Cc2ccc(CNC(=O)NCC(CCOC)O)cc2)nnc2n1CCCC2 N1(S(c2n(C)ncc2C)(=O)=O)CCCOCC12CC2.c1(CCCC2CC2)ccccc1 C12(NC(C(N)=O)=O)CN(C(c3occ4c3CCCC4)=O)CC1CS(=O)(=O)C2 c1(N(CC(=O)N(CC(C)C)CC(C)O)C(C2CCCC2F)=O)ccc(F)cc1 C1(C#N)(NC(C(C)C)=O)CCN(C(=O)CC(c2ccc(F)cc2)C)C1 C#CCC(C)(CC)C(=O)N1CCCCCC(NC(=O)CSCCCC)C1 c1(OC)cnccc1Cc1cn(C2CCCN(C(c3ccc(C)nn3)=O)C2)nn1 c1(C(=O)NC(C2(C(C)(F)F)CC2)C)ccc(C2CC2)o1.C(CC(C1CC1)C1CC1)NC c1(C(=O)NC2C(CNC(c3cccc(CC)c3)=O)C2)coc2c(OC)cccc12 C=CC1(C(=O)NC2CCCCC2CNC(C2CC23CCC3)=O)CCOCC1 c1(C(N(CCOCCN(C(=O)C2=CCOCC2)C)C)=O)c(N)cc(Cl)nc1Cl c1(OC)sccc1C(=O)NC1COCC1NC(=O)CSc1nnnn1C C1(NC(C2CCCN(C(CCC(=C)Cl)=O)C2)=O)C(C)CCCC1C C(=O)(C(CNC(=O)C(C#N)CCC)CCC)NC(CC=C)C1CC1 CC(CCCCNC(c1nnsc1C(F)F)=O)NC(C1C=CCCC1)=O CCCCC(=O)N1CSCC1C(=O)NCC=CCNC(C1CC1F)=O c1(C(CCCCNC(=O)NC(C(=O)OCC)(C)C)=O)c[nH]c2ccccc12 CCC(CC)C(F)C(=O)N(CCC(C)(C)NC(c1cnncc1C)=O)C C1(C(C)NC(c2cn(CC3CC3)nn2)=O)CCCCN1C(c1cc[nH]n1)=O C12(C(=O)NC3CN(C(c4cc(C)c(C)s4)=O)CC3F)CCCN1S(=O)(=O)CC2 N=c1nc2cc(C(=O)NC3CC(NC(=O)CCc4cccc(O)n4)C3)ccn2[nH]1 N1(C(C(CCCOC)C)=O)CCC2CC2(NC(c2cc(C3CC3)on2)=O)CC1 c1(N(C2CCCNC2)C(C2CCCN(C)C2)=O)ncnc2c1cnn2C C(=O)(CC(C)C(=O)N1CCCCC1CC(=O)NCC1CC1C1CCC1)OC c1(C(=O)NCC2CC(NC(c3c(N)nccc3)=O)C2)cc2cc(F)c(F)cc2[nH]1 C1(C(=O)NCC(CC)N(C)C(c2ccc(SC)cc2)=O)CCC=CCC1 C1(NC(CCc2cc(C)n(C)n2)=O)CN(C(c2cn[nH]c2)=O)CCC1CO C1(NC(CCN(C(CC)CC)C)=O)CCN(C(=O)CCCCCF)CC1O C1(N(C(C(C)OCCCC)=O)C)CCCN(C(c2cc(C)c(C)[nH]2)=O)C1 N1(C(c2c(C)nc(O)[nH]2)=O)CC2CN(C(C3CC(O)C3)=O)CC2(C(F)(F)F)C1 c1(C(=O)NCC2CN(C(c3c(C)[nH]cc3)=O)C(C)C2)cc(C2CC2)nc(Cl)c1 c1(C(=O)NC(c2ccccc2)C(C)C)ccc(CNC(c2cc(O)n(C)n2)=O)cc1 Cc1c(Br)ccc(NC(=O)CC2CN(C(c3cccc(Br)n3)=O)CCO2)c1C N1(C(C(c2ccc(OC)cc2)=O)=O)CC2CCC2(CNC(c2cc(O)cs2)=O)C1 C1(C(N2C(CNC(C(c3ccccc3F)(C)C)=O)CC2)=O)CCCC(C2CC2)O1 c1(C(=O)NCCCN(C)C(C2(C)CCCCO2)=O)ccc(C(C)(F)F)nc1 c1(C2N(C(C3C(C)C(=O)NC3)=O)CC2)ccc(Cl)c(Cl)c1 c1(CCNC(c2csc(CNC(=O)C(F)OC(F)(F)F)n2)=O)ccncc1F CCCCC(CC(=O)NCC=CBr)NC(=O)CC1CCC(=O)NC1 c1(C(C(C)=O)=O)cc2c(s1)CCCCC2.c12cc(oc1C)c1cccc(c1)[nH][nH]2 N1(C(C(CC=CCC)C)=O)CC(CNC(c2cccc(N)c2NC)=O)C(C)(C)C1 CC1(C)CC(C(=O)NC2COC3(CCN(C(=O)C(F)(F)CO)C3)C2)CC(C)(C)C1 C1(CNC(CN2CC(C)C2)=O)CC2CCC1N(C(=O)CCc1ccc(O)nc1)C2 CC(C)(C)CC(O)CNC(=O)C(CCC1CCC1)NC(=O)CCc1cncs1 c1(OC)cc(CC(N2CCC(NC(c3cnc(Cl)s3)=O)C23CC3)=O)ccc1O c1(N2CCC(C)(F)C2)ccc(S(=O)(=O)NCC(C)(F)C(C)(C)F)cc1Cl N1(C(c2cc(C)[nH]c2)=O)CCCCC1CNC(=O)CN1CCC(C)C1 N1(C(C)=O)CCC(c2cn(CCCC(=O)N3CCCC3C3CC3(F)F)nn2)C1 C1(NC(=O)CCn2cncn2)CN(C(c2sccc2Cl)=O)CCC1O N#Cc1cc(CNCC2CCCN2C2CCCC2)ccc1Cl C1(=CC(=O)NCC(C2CCCCC2)NC(C(CCC)OC)=O)CCC(C)(C)CC1 c1(C(=O)NC(CCCC)CNC(c2ccc(Cl)nc2)=O)cccn2ccnc12 c1(C(N2CCC(NC(C3(C#C)CC3)=O)(CO)C2)=O)cc(Br)cnc1C N1(C(C2(C(N)=O)CC2)=O)CC(CCNC(c2ccc(C3CC3)nc2)=O)OC(C)C1 c1(C(=O)NC(CN(C(c2nsnc2O)=O)CC)C)ccc(O)c(N)n1 C1(CC(N2CCCC(N(C)C)C2)=O)CC2(C1)CN(C(C1CCOC(=O)CC1)=O)C2 N1(C(C=CC)=O)C2CCC1(CNC(c1c(-c3cccc(F)c3)noc1C)=O)CC2 CN(C)S(C)(=O)=NCc1cccc(C(=O)NCC2COCC(C)N2)c1 N1(C(C(C2C(CC)C2)OC)=O)CCCC(OCCN(C)C)C1 C=CC1(C(N2CCC3(CCO3)C2)=O)CCN(C(=O)CC2CC3CC3C2)C1 C1(C(=O)NCC2C3CN(C(=O)C=Cc4cc[nH]c4)CC23)CN2CCCC1C2 N1(C(C(OC)OC)=O)CC(C(=O)NCCn2nncc2C)C2(CCC2)C1 Cc1nc(C2CC2)oc1C(=O)NCC=CCNC(=O)CC(C)(F)F CC1CC2CC(C(N3CC=C(CNC(=O)CC4CCS(=O)(=O)C4)CC3)=O)(C2)O1 Cc1nc2c(F)cccc2cc1-c1nc(C2CC=CCC2)nn1CCS(N)(=O)=O C1(N(C(=O)CNc2ccsn2)CC)CCCN(C(=O)C(F)CC2CC2)C1 CC1=CCCN(C(=NCC2CCc3ccccc32)NCCN(CCN(C)C)C)C1 c1(C(N2CC3C(NC(C(CC)O)=O)CC(C3)C2)=O)coc2c(C)cccc12 Cc1noc(N)c1C(N1CC(CNC(=O)C(C)CC2CCC2)C(O)C1)=O N1(C(CCCc2c(C)[nH]c(=N)s2)=O)CCC(C)(C)C1CNC(c1ccccc1)=O CC1CCN(CC(C)NC)CC1.C1(C=O)C2CCN1CC2 c1(OC)cccc(NCC(N2CCC(N(C(=O)C(C)CSC(F)(F)F)C)C2)=O)c1 C1(F)(CNC(c2ccnnc2)=O)CCC(CNC(C2CCN(C3CC3)C2=O)=O)C1 N=c1nc2ncc(CNS(=O)(=O)c3ccccc3C(F)(F)F)nc2c(I)[nH]1 n1(C(C)C)ccc(C(=O)NCCC2(NC(=O)CC3(CS(C)(=O)=O)CC3)CC2)n1 CCC(O)C(C)(C)C(=O)N1CCCC(NC(c2ccc(OC(F)F)cn2)=O)C1 c1(C(=O)NCC2CC(NC(C3CC(SC)C3)=O)C2)cnc(N(C)C)c(Cl)c1 C#Cc1ccc(F)c(C(=O)NC2CCCCCN(C(c3scnc3Cl)=O)C2)c1 c1(C(N2C3CCC2CC3)C(=O)NC2CCCC2)cccc(C2CC2)c1 C1(C(N2C(CCC)CN(C(=O)CC3=CCCC3)CC2)=O)CCC(=C(F)F)CC1.C1CC1 c1(OC)ccc(C)c(C(=O)NCC(O)CN(C)C(C2C(C)(C)C2(F)F)=O)c1 C(C)(CCCCNC(c1n[nH]c(C)c1Br)=O)NC(CC(=O)OC)=O C1(C#N)(C(N2CCC(C)(CNC(C3CC4(CC4)CO3)=O)C2)=O)CC2C=CC1C2 N(C(=NCc1nc(C(C)C)no1)N)CC1(OC)CC1.C#CC1CC1 c1(Sc2c(=N)[nH]ccn2)nc2cc(F)c(F)cc2[nH]1 n1(C(C)C)cc(C(=O)N(C)CCN(C(=O)CC(C)C2CC2)C)c(Br)n1 Cc1cccnc1C=CC(=O)NC1(C)CC(NC(=O)CN2CC3C=CC2C3)C1 c1(OC)ccc(CC(=O)NC2(C)CCN(C(=O)C(C)CC(N)=O)C2)c(Cl)c1OC CCC(C)C(O)CC(=O)NC1(CCNC(=O)CCn2ccnc2C(C)C)CCC1 O=C(C1CCCn2cnnc21)NC1CC2CCC(C1)N2C(=O)C1=CS(=O)CCC1 C(=O)(C#CC1(C)CCCO1)NC(C1N(C(Cc2cccc(OC)n2)=O)CCC1)C CC1N(C(=O)COC2(C)CN(C(=O)CN3CCCCC3)C2)CCCC1(C)C c1(C(=O)NC(CC)(C)CNC(=O)COC(C)C)ccc(OC)c(F)c1N CCCC(C)CC(=O)N1CC(C2(NC(c3cc(C4CCCC4)n(C)n3)=O)CC2)C1 C(N=C(NCC(F)F)N1CCC(CC#N)CC1)c1c(C)cn(C)c1 N1(C(c2c(C)n(C)cc2)=O)CCC(CNC(C2CC2c2cccnc2)=O)C(O)C1 C1(OC)CCC12CC(C(=O)NCC(CNC(=O)C(C)NC(C)=O)OC)C2 c1(C(N(C(CC)CC)CC(C)C)=O)cn2c(n1)C(=O)CCC2 C1(C(N(C(C2CCOCC2)C)C)=O)CN(C(C2OCCC2(C)C)=O)CC1C1CC1 C1(=CC(=O)NCCC2(CNC(=O)Cc3cnns3)CC2)CCSCC1 CC1CN(C(=NCCc2ccc(OC(F)F)cc2)NCC2(C#N)CCC2)CC1C C(N=c1nc(N2CCC3(CC3)C2)c2c([nH]1)CCOC2)c1cc(OC)no1 N1(CCC)CCC(NCC)C1C(C)C.c12ccn(c1)C2c1nnnn1C CC(C(=O)N1CC(CC(C(NC(=O)CCc2cn[nH]c2)=C(C)C)C)C1)n1cnnn1 C1(OC(C(C(=O)OC)N)C2CC2)CC(S(C)(=O)=O)CNC1c1ccccc1 C(=O)(C(C)(C)CCOC1CCCC1)N(C1CCSC1)CC(=O)NCCOC C1(CN2CC(C(N(C3CCC4(CC3)CC4)C)=O)C2)CC(C(C)(C)C)=NO1 C(=O)(C1CCc2ccccc21)N1CC(OCCNC(CC2(C)CC2(Cl)Cl)=O)C1 c1(CC)c(N2CC3CC(NC(=O)C(C)(C)C4CCCCC4)C3C2)ncnc1Cl Cc1cc(CC(=O)NCC2C(O)C(O)CN2C(C2CC3(CC3)CO2)=O)ccc1Cl C1(C)(NC(CCCOc2ccc(C)cc2)=O)CCCN(C(=O)Cc2ccco2)C1 CCCS(=O)(=O)CC(=O)N1CCC(C)(NC(c2cc(CN(C)C)on2)=O)C1 C#CCCCCCC(=O)N1CC2CC(C(N3CC(O)(C4CCC4)C3)=O)C(C2)C1 C1(C(=O)NCc2c(C)n(C)nn2)CCN(C(c2ncncc2Cl)=O)CCO1 Cn1c([N+](=O)[O-])cnc1C(=O)NCC(F)CNC(c1csc(C2CC2)n1)=O C(=O)(C1=COCCO1)NCC(CC)NC(=O)CC1CCN(C)C1=O c1(C(=O)NC(C)CNC(=O)CC2CCC(=O)N2)cccc2scnc12 c1(C(=O)NC2C(NC(C3CC(C)(C(C)(C)C)C3)=O)COC2)cccc2[nH]ccc12 N1(C(CCCc2ccc(C)s2)=O)CCC(C)C1CNC(=O)C(F)OC(F)(F)F c1(C(N2CC(CC)CC(C)C2)C(=O)NCCCC)nc2ccccc2n1CC C1(NC(Cc2ccn(C)n2)=O)CCCC12CN(C(c1ccc3n[nH]cc3n1)=O)C2 C1(NC(C(=O)NCC2(S(C)(=O)=O)CC2)=O)CCCCN1Cc1ncccc1Cl c1(C(N2CCN(C(=O)C(F)=CCCF)C3C2C3)=O)cc2cc(F)ccc2[nH]1 c1(NC(C2OCCN(C(CC(n3ccc(C)n3)C)=O)C2)C)cnc(O)cc1C CS(=O)(=O)c1ccc(-c2ncsc2C(=O)Nc2cccc3nonc23)cn1 C1(C(=O)NC(C2CN(C(=O)Cc3cccnc3Cl)C2)C)CC12CCOCC2 Cc1cc(C(=O)NC(C)(C)C(C)NC(c2cc(F)cc(F)c2)=O)cc(C)n1 N1(C(C(COC)(C)O)=O)CCN(C(c2ccoc2Br)=O)C(c2ccnn2C)C1 C1(NC(CCCOC(C)=O)=O)CCC2(CC1)CN(C(C1CCCCC1C)=O)C2 C(c1ccc2ncccc2c1)=CC(N1C2CCC(NC(C3CC34CC4)=O)(C2)C1)=O CCC(CC)C(F)C(=O)NC(C1CCCCC1)C(=O)NCc1cc(Cl)no1 N1(c2c3ncn(C(C=C)CCO)c3ncn2)CCC(S(=O)(=O)C(C)C)C1 c1(NC(Cn2ncc(C)c2)C)cc(=NC(C)c2c(C)n[nH]c2C)[nH]c(C(C)C)n1 C(CC(CC)C(=O)NCC1(C)CCCN1C(c1csc(C)c1N)=O)=CC C1(CNC(C(C2CCCC2)OCC)=O)CC2COCC2N1C(C1CCC(=O)C1)=O N1(C(CC23C(CN(C(C4(C)CCC4)=O)C2)CC3)=O)CCC2(CCCO2)CC1 Oc1[nH]c(=NCC2CCC=CO2)nc(N2CCC(C3CC3)C2)c1Cl C12(NCCNC(N3CCCCC3c3ccco3)=O)CCC(O)(CC1)CC2 S(=O)(=O)(c1c(O)cccc1F)NC1CN(C(c2ccc(C(=O)OC)cc2)=O)C1 CCCC(CC)C(=O)N1CCN(C(c2coc(C3CCC3)n2)=O)C(C2CCC2)C1 c1(S)cccc(Cl)c1.CC12CC1C2=O.C(C(=O)NCCCNC(=O)CSCCO)N N1(C(C23N(C(c4c(C)oc(CO)c4)=O)CC(C2)C3)=O)CCCC(N=[N+]=[N-])C1 N1(C(c2ccc(CC)c(C#N)c2)=O)CCC2(CC1)CC(C)N(C(C1CC1C)=O)C2 c12cc(ccc1C#N)S(=O)(=O)N2.c1(NC2C(OC(C)C)COC2)cccc(F)c1 CN1CCC(C2(C(N3CCCC3CNC(C3Cc4ccccc4O3)=O)=O)CC2)CC1 N1(C(c2cncc(SC)c2)=O)CCN(C(c2cnoc2C)=O)C(c2cn[nH]c2)C1 c1(C(=O)Nc2c[nH]c(OCC3CCCCO3)c2)ccc2sc(Br)cc2c1 N1(C(C2CCC(N(C)C)C2)=O)CC2(CCC2)CC1C(N1CC2CNC(=O)C2C1)=O C#CCCC(O)C(=O)NC(C)CN(C)C(C1CN2CCC1CC2)=O CC1CN(C(c2cccnn2)C(=O)NC2CCCC2)CCCO1 CC1CCC(NC(=O)CN2C(=O)CNC2=O)CN1C(c1cccc(C2CC2)c1)=O CCC(CC)CC(F)C(=O)NCC1CC(C)N(C(=O)C(C2CCOCC2)=O)C1 c1(C(N2C(CC)CN(C(C3(OC)CCC3)=O)CC2)=O)cc2ccc(Br)cc2s1 C1(N(C)C(c2cc(C(N)=O)co2)=O)CCCC(NC(C2(C)CC2(F)F)=O)C1 CC1COCCCN1C(=O)CC1(NC(C2CNC(=O)C2)=O)CC1 CC1(C)CN(C(C2CN(C(=O)CCc3c[nH]c(=N)o3)C2)=O)CCC1CO C1(NC(=O)Cc2cc(Br)cs2)CCN(C(=O)Cc2cncnc2)CC1F c1(NCc2c(CC)noc2CC)nccc(=NCCC2COCCO2)[nH]1 c1(C(N2CC(SC)C(O)C2)C(=O)NC(C(=O)OC)C)ccc(I)cc1 CC1CC2CNCCN2C1.C12(CCSC1)C(=O)N2.C(=O)(CO)NCC1CC1 c1(OC)ccc(C(F)(F)CNC(=O)N(C)Cc2nnc(-c3cccs3)o2)nc1 C1(NC(c2ccoc2)=O)(CO)CN(C(C2(C3CCCCO3)CCC2)=O)C1 C1(CC(=O)NC(CSCC)C(=O)NCc2ccc(CO)o2)CCC(O)C1 N#CC1(C(=O)NCc2nc(CNC(=O)CC3CC=CCC3)cs2)CCCOC1 c1(CC)cc([N+](=O)[O-])c(C(N2CC3C4C=CC(O4)C3C2)=O)c(O)c1 N1(C(c2c(C)cncc2)=O)C2CCC1CC(NC(c1c(C)ncn1C)=O)C2 O=C(CN=c1ccnc(N2Cc3ccccc3C2)[nH]1)N1CCCc2nccn21 N1(C(C(CCC)CC(C)C)=O)CCCCC2(CCCN2C(c2ncnn2C)=O)C1 CCCC(C(=O)NC1CC(CNC(=O)Cc2cc(C(F)F)nn2C)C1)NC(C)=O C1(C(=O)NC(C2CCCC2)CNC(c2cc(OC)n[nH]2)=O)CC(C)(C)OC1(C)C N1(C(C(=O)NCCSC)C2CC2C)CCC2(CCN(C)C2=O)C1 CC1CCCC(n2cc(C(N3CCC3COCSc3ccccc3)C)nn2)C1 C1(CNC(CC(=C=C)C)=O)CC2(CCN(C(=O)C(C)(C)C3CC3)C2)CO1 N1(CCNC(C2C(CC)C(=O)C2)=O)CCN(C(C2CC2C)=O)CC1 C#CC1(O)CCN(C(C2(COC)C=CCN2C(=O)C(C#N)CC)=O)CC1 c1(CCC)cc(C(=O)N(C2CCN(C(=O)C(C)CF)C2)CCO)nn1C C(CC(=O)NCC1(CN(C)C)CC1)(C(C)(C)C)NC(C1(C=C)CCCC1)=O Cc1ccc(F)c(CC(=O)NCC2(C(N3CCOC(CC4CC4)C3)=O)CC2)c1 CCC(C)C(C(=O)OCc1ccn(C(C)C)n1)N(C)C(c1ccccc1C)=O N1(C(C2(F)CCN(C(C=CCOC)=O)CC2)=O)CCCCC(C)(C)C1 N1(NCc2cccc(OCC=C)c2)CCCC1C1CCCO1 CC1ON=C(C(=O)NC2CC(F)CN(C(=O)C(C)(C)C(=O)N(C)C)C2)C1C C1(CNC(=O)C=CI)CCCC2(CN(C(=O)CCN3CCC(F)C3)C2)O1 c1(OC)nc(C)c(S(=O)(=O)N2CCCC2C(N2CCOC(CO)C2)=O)s1 N1(C(C=Cc2cc(C)no2)=O)CC2(C=C(C(=O)NCC(F)Br)CO2)C1 C12(C(=O)NC3C(NC(CC(C=C)(C)O)=O)COC3)CC(CO)(C1)OC21COC1 C(C(CNC(C1CCCC1)=O)C(F)(F)F)NC(=O)Cc1ccns1 c1(C(=O)OC(c2ccc(Cl)cc2)CCCC)n[nH]c2c1CCSC2 C(CC(=O)NCC(C1CCCCC1)NC(c1ccsc1C)=O)(C(C)C)OCC N1(C(Cc2n(C)cnn2)=O)CCC2(NC(C3CC4(C3)CC4F)=O)CCCC12 c1(OC)ccc(CN2CCC(C)(C(=O)Nc3nnc(Br)s3)C2)c(Br)c1O c1(C(=O)NCC2(F)CCC(NC(C3(C)C(C)CCC3)=O)C2)nc(Cl)ccc1F n1(CCC(=O)OCCC2CC(C(=O)OC(C)(C)C)C2)ccccc1=O c1(C(=O)NC(C)CNC(=O)CNc2cccc(C#N)c2)cc(Br)cnc1O C(=O)(C(CC(C)C)C(C)C)NCCN(C(C=CCOC)=O)CCCN(C)C N1(C(COCC=C)=O)CC(C)(C)OCC1CNC(c1cnn(-c2nccs2)c1)=O N1(C(C(C)N2CCCC2)=O)CCC(C(C)(C)C(=O)N2CC(O)(CCO)C2)C1 CC1CCN(CC(N2CCCC(CNC(C3CC3Br)=O)C2)=O)CC1 C(=O)(C1CCc2c[nH]nc21)N1CC(O)(C(C)NC(c2cnc(C(C)C)s2)=O)C1 C1(C(=O)NC2C(CNC(C3C(C(=O)OC)C3)=O)CCCC2)CCc2c[nH]nc2C1 n1(CC)cc(CC(=O)NC2(CNC(c3sccc3C(C)C)=O)CCCC2)cn1 CCC(CN(C)C)CC(=O)NC1CCN(C(=O)COCCc2ccccc2)C1 C(=O)(CCC1=CCCCC1)N1CCN(C)CC1C(N1CCC(CO)C(O)C1)=O N1(C(C2(N(C(c3ccc(C)cn3)=O)C3CC3)CCC2)=O)CC(C)C(F)(F)C1 N1(C(c2c(OC)cccc2)=O)CCC(C)(Cn2cc(CC(O)C(C)C)nn2)CC1 C1(NC(C=Cc2scc(C)n2)=O)CCN(C(C2CC2c2ccccn2)=O)C1(C)C N1(C(c2c(C)c3c(s2)cccc3)=O)CC2CCN(C(C3(F)CCOC3)=O)CC2C1 C12(C(N3CCC(NC(C4CCN(C)C4=O)=O)(CF)C3)=O)CNC(=O)C(C1)C2 C12(NC(=O)NCC(CC=C)OC)CCCCC(NC(=O)OC(C)(C)C)(C1)C2 C1(CCOC)CN(C(c2ccc(N)cc2O)=O)CCN1C(=O)C(C)n1ccnn1 CCCS(=O)(=O)C(C)C(=O)NCC1CC2CCC1N2C(=O)C(C)(C)F c1(CCC)ccc(C(=O)NC2CCC2NC(=O)C(C)(C)n2cnnn2)cc1N c1(C(=O)NC2CCC(NC(CC3CC(C)C3)=O)C2)ccccc1-n1cncn1 C(CC(=O)NC(C)(C)CCNC(c1csc(O)n1)=O)(C(N)=O)NC(C)=O Cc1ccc2c(C(=O)NC3CN(C(C4CC(O)CN4C)=O)C(C)(C)C3)csc2c1 N12CCN(CCC1C)C2=O.CC(C(C)(F)F)C(=O)OC(C)(C)C CCCC(C(=O)NC(C)(C)CN(C(=O)CC(C)N(C)C)C)C(C)C CCC(CC(F)(F)F)NC(C1CCC(CNC(c2oc(CO)nc2C)=O)CC1)=O C1(C(=O)NC)CN(C(=O)C(=O)NCCSC)CCN1C(=O)CC1CCCCO1 CC1CN(C(=O)Cc2cc3ccccc3o2)CCCN1C(c1c[nH]ccc1=O)=O N1(C(c2cncc(C#N)c2)=O)C2CCC1CC(NC(C1CCC(C3CC3)C1)=O)C2 C1(CC)CC2CCCC(C1)N2C(=O)NNC(=O)c1nc(-c2ccccc2)cs1 N1(C(c2cc(C)ns2)=O)CCC(C2CCCN(c3ccc(C#N)nc3)C2)CC1 N1(CC(=O)NCC(C)(F)CNC(=O)CCCN2CCOC2=O)CCC(O)CC1 Cn1ccc(C(=O)NCC2C(NC(CCC3CC3)=O)CCC2)n1 Cc1cccc2c1nc(NC(=O)NCC1(C(F)(F)F)CCN(C)C1=O)n2C N1(C(Cc2c(C)nc(C)s2)=O)CCOC2(CCN(c3ccc(C#N)nc3)CC2)C1 C(CN(C)C)(C(C)(C)C)NC(CC(C)NC(=O)C=Cc1cn[nH]c1)=O N1(C(CN(C)C)=O)CCCC(O)(CC(=O)NC2(C)CCCC2)C1 N1(C(c2cc(C)oc2)=O)CC2CC1CN2C(=O)CCC1CCCCC1 C1(C(N(C2CCN(C(=O)CSC)C2)CC#C)=O)COCCN1S(=O)(=O)CCC Cc1c(C(=O)NCCCCCN(C(=O)CCC(=O)C2CC2)C(C)C)cccc1F C(C(C)(C(=O)NCC(C1CCN(C(=O)CC2CCC23CCC3)CC1)(C)C)OC)OC n1(CC(=O)NC2CCC2NC(=O)CCC2CC(F)(F)C2)cc(C#N)cn1.CC(C)C CN1CCN(CCNCC2CCCC2NC(c2cnn(CCN(C)C)c2)=O)CC1 N12CCN(CC1)C1CCCN(C1)C(=O)N(CCOC(C)C)CC2.C(CO)O c1(C(=O)NCC(F)CNC(c2cccc[n+]2[O-])=O)ccc(C2CC2)c(Cl)c1 CCCC(CCCO)C(=O)N(C(CNC(=O)Cc1cc(OC)no1)C1CC1)C n1(CC)cc(CN(c2noc(CC3CC3)n2)C)c2ccccc12 C1(NC(C2(C)CC(=C)C2)=O)CC(F)CN(C(c2ccc(N(C)C)cn2)=O)C1 N1(C(CC(=O)OCC)=O)CC2CCC(C1)N2C(=O)CC1CCC(O)C1 c1(CC(CCC)NC2CNC2C2CC2)cccc(I)c1 c1(C(=O)NC2CN(C(C(CCC)C)=O)C2)ccc2ccncc2c1 c1(C(N2CCC3C(C(=O)NC(CC)(C)CO)C3C2)=O)cc2ncccc2[nH]1 CC1=NOC(CC(=O)NC2CC(C)(NC(c3sccc3C3CC3)=O)C2)C1 C1([Si](C)(C)C)(CNC(CCN(C(=O)CCn2ccnn2)C(C)C)=O)CC1 c1(SCC(=O)N(C(C)Cc2ccccc2)CC)ccc(F)cc1 Cc1cccn2c(CC(N3CC4CC3CC4NC(C3CC3C(N)=O)=O)=O)cnc12 c1(C(N2CCC(NC(c3c(C)nns3)=O)C23CCC3)=O)cc2ccc(F)cc2o1 c1(OCC(=O)NCC2CCC(NC(c3cnn[nH]3)=O)C2)cccnc1Cl O(NC(=O)C(CNC(=O)C(C)(C)NCC)CC(C)C)CCOC(C)=O C=CCC(CC(=O)NCC(C)C#N)NC(=O)C=CCN1CCCC1 N1(C(c2ccc(C(C)(C)C)s2)C(=O)NCCCOC)Cc2ccccc2CC1C C1(NC(=O)CC2CCOC2)CN(C(c2ccc(F)cc2O)=O)CC12CCC2 N1(C(C2C=CCN(C(C(C)(O)C3CCC3)=O)C2)=O)CCCC12CCOC2 CN1CCCC(CNC(=O)C(=O)NC(c2cnn(C)c2)C2CCCO2)C1 c1(C(=O)NC2CC(CNC(=O)COCCOCCO)OC2)cc(CSC)on1 c1(C(N2CCC(COC)C2)=O)cc2n[nH]cc2cc1-c1cccc2cn(C)nc12 C1(Cc2cc(NC(C3(OC)CCC3)=O)cc(Cl)c2)CCn2c(Br)cnc2C1 Cc1cc(C)c(C(=O)NCCN2CCCN(C(C3CNC(=O)N3)=O)CC2)c(C)c1 c1(C(N2CC(NC(c3cnc(C)[nH]3)=O)C(O)C2)=O)cc2n(n1)CCNS2(=O)=O C1(NC(c2nccc(C)n2)=O)CCC2(CC1)CN(C(c1cnns1)=O)CCO2 C1(CNC(c2ccn(-c3ccccc3)n2)=O)CCCC1NC(C1CCCC1O)=O C12(CNC(N3CCC(c4csc(Br)n4)C3)=O)OCCCC1C2(F)F N1(C(c2cc(OC)ncn2)=O)C2CCC(C2)C1CNC(c1ccc(C)c(C)n1)=O C(CCN(C(=O)C(O)C(F)F)C)(C(C)C)NC(c1[nH]cc(CSC)c1)=O C(=O)(C(O)CC(F)(F)F)N(CCC(N1CCCC(OC)C1)=O)CCOC Cn1nc(C(=O)NCC(N2CCN(C(C3(C)CC3)=O)CC2)=O)c(Br)n1 COn1cnc(C)c1C(=O)N(C)CC1(NC(=O)COc2ccsc2)CC1 C(C(F)(F)Cl)N(C(=O)C(=O)NC(c1nccs1)c1ccco1)C Cc1c(C(=O)NCCC2CC(NC(C3CCCCO3)=O)C2)cnn1CC(F)(F)F C1(C(=O)NC2CC(F)(CNC(CCOCCCOC)=O)C2)NC(=O)OC1C c1(OC)ccc2cc(CNCc3ncsc3Br)nnc2c1 C#CCC(O)C(=O)NC(Cn1cncn1)C(=O)NCC1CC=CCC1 C1(CN(S(C)(=O)=O)C)CN(C(c2ccn(CCF)n2)=O)CC1O.C1CC(=O)N1 c1(C(N2CC3C(CNC(C(=O)NCC)=O)C3C2)=O)cc(Br)n2ccccc12 CCC(CC(=O)N1CC(CNC(c2cccc(N)c2F)=O)CC1C)C(C)C N1(C(c2ccc(C(N)=O)[nH]2)=O)CCC2(C1)CN(C)C2.CC1C=CC(=O)N1 CC(=O)C(C)(C)CC(=O)N1CCC(C(=O)NCC2C3CCCOC23)CC1 C(=O)(C(CC)C(C)(C)CC)N(CC(C)NC(c1ccc(C#N)[nH]1)=O)CC N1(C(C(CC=C)NC(C)=O)=O)CC2(CCC(CNC(c3n[nH]cc3CC)=O)O2)C1 CCC(CN(C)C)C(=O)N(CC(O)CN(C(=O)C(C)(C)NS(C)(=O)=O)C)C C1(CNC(C2CCSCC2)=O)C2CCCC1N(c1ncc(F)cn1)C2 S(=O)(=O)(c1ccc2nc(N3CCC(OCC(N)=O)C3)sc2c1)N1C(C)CCC1 c1(C(=O)OC)oc(C)nc1CNC(C)C(N)=O N1(Cc2ccccc2)CCCN(N2CCC3(CCO3)C2)CC1 Cc1ncc([N+](=O)[O-])n1CC(=O)N(CC(C)(C)NC(c1cncc(N)c1)=O)C CC1(C)CN(C(c2ccnnc2)=O)CCC1C(=O)NCCC1CCOC1 CC1CCC(C(N2CC3(CC3)CC2C)=O)N(C(C2C3CCCOC23)=O)C1 CC(C)(C)C1=NOC(CNc2nccc(NCCCC(F)F)n2)C1 c1(C(CCNC(c2nnnn2C2CC(F)(F)C2)C)OC)ccccc1Cl c1(CN(C(C(CCOC)(C)C)=O)C)cnn2c1CN(C(C1CCCO1)=O)CC2 C(=O)(C1CCNc2ccccc21)N1CCC(CNC(CCC=C(C)C)=O)C(C)C1 CCC(F)(F)CC(=O)NCC1CCN(C(C2CC2c2cccnc2)=O)C1 c1(N2CCCCC(CC)C2)nc(=NCC2CC2)[nH]c2c1CSC2 N1(C(CC2(OC)CCC2)=O)CCC(C(C)CNC(c2ccsn2)=O)CC1 C(=O)(C(O)CCS(C)=O)NCCCCNC(c1[nH]cc(C(C(C)C)=O)c1)=O Cc1cccc2c1OC(C(N1CCC(=CCNC(C3C(C)C3(F)F)=O)CC1)=O)C2 CN1CCN(C(C2CC(NC(c3csc(Cl)n3)=O)CCO2)=O)CC1 c1(C(N)=O)cc(C(N2CC(NC(=O)C(=O)C3CC3)C3(CC3)C2)=O)ccc1O C12CCC(CC1)Cn1cc2nn1.Cc1conc1CC(N1CCC(CC2CC2)C1)=O C1(C(=O)NC(CCCC=C)C)CCC(O)CN1C(=O)CC1(OCC)CCC1 c1(N2CCC(N(C(=O)C=Cc3nccs3)CC)C2)nnc2c(c1C#N)CCCC2 c1(C(=O)NCCNC(CCNC(=O)OC)=O)nc(Cl)ccc1Cl C1(CNC(C(C)O)=O)(CNC(=O)Cc2ncc(Cl)s2)CC12CCC2 C(=O)(CCNC(c1ccon1)=O)NC(=O)CSCOCC(C)C1CC1 CC1CN(C(c2ccon2)=O)CCC1N(C)C(c1cc(C(F)(F)F)on1)=O c1(CC)[nH]nc(C(N2CCC(CCC(=O)NCCOc3ccn(C)n3)C2)=O)c1C CCCCC(C)(F)C(=O)N1CC(CC(=O)N(CC(=C)Cl)C)C2(CC2)C1 c1(C2N(C(CC(CC(C)C)O)=O)CCC(C(=O)O)C2)ccc(O)c2ccccc12 C#CCC(O)C(=O)N1CSCC1C(N1CCCC1C(N)=O)=O c1(NCCC)nc2ccc(S(=O)(=O)c3cccnc3N3CCCC3)cc2s1 C=C=CCC(=O)NCCCN(C(=O)C(C)CN1CCCCC1)CCO c1(C(=O)NCCC2(OC)CN(C(c3[nH]cnc3C)=O)C2)cc(C)cc(F)c1 CC1CN(C(=O)CSCc2ccccn2)CCC1NC(c1c[nH]c(=O)cn1)=O N1(C(C(COC)Cl)=O)CCc2c(C(N3CCC4CCCC34)=O)csc2C1 N1(C(C(C)(CO)NC(C)=O)=O)CCC(C2CN(C(C3(C)CCSCC3)=O)C2)CC1 C1(NC(CN(C)CCO)=O)CC(=O)N(C2CN(C(=O)CP(C)(C)=O)C2)C1 C1(NC(=O)C(=O)NC(Cc2ccccc2)C2CC2)CCn2cncc2C1 N1(C(C2C(C)CCS2)=O)CCC(CO)(CNC(c2cnn(C3CC3)c2)=O)CC1 N1(C(CC)C(N)=O)CCc2ccccc2C1CNC(=O)CSC1CCCCO1 C(=O)(CC(C)P(C)(C)=O)N1C(CNC(CC2CC(CC)C2)=O)C(C)(C)CC1 C1(CC)CN(C(c2cnnn2C)=O)CCC1NC(=O)CCc1ccccc1Cl CCCC(CCC)C(=O)Nc1cccc(CNC(c2ccccc2C(C)=O)=O)c1 c1(C2C(CC)C2)cccc(C)c1.n1(C(CC)C)nnnc1C1c2n[nH]c(n2)CN1 C(C)(C)(CCC(=O)NC1CS(=O)(=O)CC1NC(c1ccc(Br)cc1)=O)OC C(=O)(CC(C)C(F)(F)F)NCC1N(C(c2c(C)nc[nH]2)=O)CCCC1 CC(F)(F)C(C)(C)C(c1nnnn1C1CCOCC1)NCCc1ccncc1 N1(Cc2ccc(OC)c(OC)n2)CCC2(CCC(OC)C2)C1 c1(C2(C(=O)NC3CC(CNC(c4sccc4Cl)=O)C3)CC2)ccc(OC(F)F)cc1 C1(C(=O)NCC2CC(NC(CCOCC(C)C)=O)C2)CCC(CCO)CC1 N1(C(CC(CC)C)=O)CCCC(O)(CNC(c2ccc(C)cc2)=O)C1 C1(CC(=O)N(CC(C)NC(=O)CC(C)N2CCCC2=O)CC)CCCC(=O)C1 c1(CC(=O)NC2C(CNC(c3ccn(C(C)C)n3)=O)CC2)cccc(F)c1 CCCCC(O)C(C)C(=O)N1CCC2CC12C(=O)NCC1CN(C(C)C)C1 Cc1cc(Cl)ncc1CC(=O)NC1(CF)CCN(C(=O)C=CC2CC2)C1 C1(C(N2CCC(N(C(CN3CCN(C)CC3)=O)C)C2)=O)CCCCCS1(=O)=O CCC(C)C(C(=O)NCC(C)C(C)(C)C)NC(=O)Cc1ccc(C)s1 C12(NC(C3CCC(=O)C3)=O)CC3CCC(C1C2)N3C(c1onc2c1CCCC2)=O c1(NC)cc(C(=O)N(C)CC2(F)CC2)cc(Cl)n1 N1(CCN(C(C)C)C(=O)NCC(F)(F)F)CCN(CC2CCCCO2)CC1 Cn1nccc1C(C(N1CCCC1C1(C)CC1)=O)NC(=O)CC1CCCO1 C(=O)(CC(C)(C)CC)NC(CC1CN(C(c2nc(CCC)sc2)=O)C1)C Cc1ccc(C=CC(N2CC(NC(=O)C3=CCCC3)C(C)C2)=O)o1 c1(C(=O)NC(C)CNC(=O)C(C)(C)C)cccc(S(=O)(=O)NC(=O)C2=CCCS2)c1 CC1CCCN(C(c2coc(C(F)F)n2)=O)C1CNC(=O)C(C)(C)n1cnnn1 C=C(C)CC(C)C(=O)NCCOC1CCN(C(=O)CC2(CS(C)(=O)=O)CC2)CC1 c1(C(N2CCC(N(C(=O)CN3CC4CC4C3)CC#C)CC2)=O)ccc(C#N)n1C C1(c2cccc(Cl)c2)(C(=O)NC(C(C)NC(C=C(COC)C)=O)CO)CC(F)(F)C1 C1(C(N(CCCOCCN(C(COCC=C)=O)C)C)=O)CCC2CC12 C(C(CNC(C1CCC=CCC1)=O)C(F)(F)F)NC(C1C(C)(C)COC1)=O C(=O)(CC1c2ccccc2CCN1C(C)=O)N1CCC(N(C(CC=C)=O)C)C1 C(CC(=O)N1CCC1CNC(=O)CC(=O)OC)(C1=CCCC1)OCC CC(CNC(=O)C(C)(C)C(N)=O)N=c1nc[nH]n2cccc12 c1(CC(=O)NC(CNC(C#CC(=O)N(C)C)=O)C)c(C)nc2ccccc2c1C C1(C(=O)NCC2CC(F)(CNC(C3CC(O)(CC#C)C3)=O)C2)CCC(C)CC1 C1(C(=O)NCCC2ON=C(C)C2)(NC(c2ccccc2F)=O)CCN(C)C1 C(=O)(C1=NN(CCO)C(=O)CC1)N(C(CNC(C1(CC#C)CCOC1)=O)C)C N1(C(c2n(CC)ncc2)=O)CCC2(CC1)CC(NC(=O)C(C)C1(O)CCC1)CO2 N1(C(C(C(C)C)OC)=O)CC2CC(NC(=O)CCOC3CC3)C1C2 N1(C(c2ccc(C)o2)=O)CCC2(CCC2)C(CNC(C2(C)CCOC2)=O)C1 Cc1c(C(N2CCOC(CN(C(=O)CCS(C)=O)C)C2)=O)cnc2nncn12 C#CCC(C(=O)NCc1n[nH]c(C)n1)NC(=O)CC1CC(O)C1(C)C CCS(=O)(=O)CC(=O)N(C)CCN(C)C(c1cnc(Cl)s1)=O C1(NC(C(C)(C)C)=O)CN(C(=O)CCc2ccccn2)CC1C1CC1 Cc1[nH]nc2c1CC(C(=O)N(CCNC(c1c(Cl)cnn1C)=O)C1CC1)CC2 c1(C(=O)NCC2(CNC(C3(F)CCCC3)=O)CC2)n[nH]cc1F c1(C(N2CC(CNc3nc(SC)c(C)cn3)OCC2)=O)ccc2oc(O)nc2c1 c1(NC(C2CCCCN2Cc2ncccc2Br)=O)cccc(Br)c1O c1(CNC(C(CC=C)NC(C23CCC(OC)C2C3)=O)=O)nc(O)ccc1C C(=O)(C(C)(C)CC(F)(F)F)N1CCC(O)(C(C)C(=O)NCc2ccco2)C1 [N-]=[N+]=NC1(C(=O)NCC2(F)CCC2)CCN(C(=O)CC(C2CC2)C2CC2)C1 c1(C(=O)NCc2ccc(CN(C)C(C3CCOC3)=O)cc2)cc(S(N)(=O)=O)c[nH]1 Cn1nccc1C=CC(N1CC2C(CNC(=O)CCc3cn(C)cn3)C2C1)=O N1(C(CCCOC(C)=O)=O)CC=C(C(=O)NC2CCC(C3CC3)C2)C1 c1(CC)nc(=N)[nH]cc1C(=O)NC1COCCC1NC(c1cnc2n1CCS2)=O c1(C(N2CC(NC(C(C)(C(C)C)NC(C)=O)=O)C(O)C2)=O)c(F)cc(C)cc1F C1(CNC(c2nc(OC)c(C)s2)=O)CN(C(C2(CC(F)F)CC2)=O)CCCO1 C1(NC(CCCC=C)=O)CC2CCC1N(C(=O)C(C)CCCC)C2 c1(C(=O)NCC(C(=O)OC)C2CCOC2)ncc(C)c(-c2ccccc2)n1 N1(C(c2ccc(NC)cc2)=O)CCCC(N(C(=O)C(C)Cn2cccn2)C)CC1 c1(CSC)ccncc1CNC.N1(C(C(=O)N)=O)CCC(C(C)(C)C)CC1 C1(CNC(C(C)OC)=O)CN(C(c2ccccc2C)=O)C2CCN1C2 C1(C(N(CC(=O)NC(c2cnc(C)s2)C)CCC)=O)OCCOC1C c1(C(N(C(CC(CNC=O)O)=O)CCCCC(F)F)=O)n[nH]c2c1COC2 C1(C(N(CCC)CCC)=O)(OC)CCN(c2ccc(Cl)cc2OC)CC1 N1(C(=O)C2=CCCCC2)CC2CCC(C1)N2C(=O)COc1ccc2c(c1)OCO2 CCCC(O)CC(=O)N1CC(NC(C2CCCC3(CC3)C2)=O)C(C)(C)C1 CC1CN(C)CC1N=c1ccc(Br)c(S(=O)(=O)NCc2cccc3cnccc23)[nH]1 N1(C(c2ncccc2Br)C(=O)NCCCC)CCc2sc(S(N)(=O)=O)cc2C1 C1(C(=O)NC2(CC)CCC2)CCN(C(=O)C2CC(F)(COC)C2)O1 Cc1[nH]nc(C(=O)NC2CCC2CNC(C2(C(N)=O)CC2)=O)c1Br C(c1ccc2nc(N=S(C)(=O)c3ccccc3)ccc2c1)=CCCC C1(COC)(NC(=O)CC2CCC(=O)N2C)CCN(C(=O)C2=CC(C)(CC)C2)CC1 N1(C(C(C(=O)OC)OC)=O)CCC(CNC(c2cc(C)co2)=O)C(F)(F)C1 N1(C(CNC(c2c(C)ocn2)=O)=O)CCN(C(c2cccs2)=O)CC1.C1(C)(C)CC1 c1(C(=O)NCC(COC)NC(=O)C=CC(C)(C)SC)csc(C(F)F)c1 c1(C(=O)NC23CC(CNC(c4c(C)nn(C)c4Cl)=O)(C2)C3)coc(S(C)(=O)=O)c1 Cc1c(S(=O)(=O)N(Cc2cccc(Br)c2)CC2CCCC2)sc(C(=O)O)c1Cl C1(CC(=O)NCCCOC(C)C)CCN(C(C2CS(=O)(=O)C2)=O)C1 N1(Cc2c(C)nc(C)s2)CCC(NC(c2ccoc2C)=O)CC1C C12(C(N(C3CC(C(N)=O)C3)C)=O)CCCC1CN(C(c1nocc1Cl)=O)C2 c1(C(=O)NC2CC3CN(C(CC(C=C)C)=O)C2C3)nc[nH]c2nccc1-2 c1(N(CC(=O)NC2(CC#C)CCC2)C(=O)OC(C)(C)C)cccc(F)c1[N+](=O)[O-] N1(C(c2cn(C)nn2)=O)CCC2(CC1)CCN(C(c1ccnn1CC(F)F)=O)C2 Cc1ccc2c(ccn2CCC(=O)N(CC(C)N(C(=O)CC(C)C(F)F)C)C)c1 Cc1ccc(CC(=O)NCCC2(NC(=O)COC(F)F)CCCC2)c(Cl)n1 c1(CC)cccc(CC(N2CC(NC(C3(NC(N)=O)CC3)=O)CC2CO)=O)c1 c1(C(C)=O)cnc(N2CCCOC(CNC(=O)COC3CCCOC3)C2)c(C)c1 CC1(CNC(=O)C(F)OC(F)(F)F)CCCN1C(=O)CCNc1ccccc1 N12CCOC(C1)C2=O.C(C(C)(C(C)C)NC(=O)CCC=C(C)C)NC(C)=O C1(C(C)Nc2nc3c(o2)CCSC3)CCc2ccccc2C1 C(C)(C(=O)NCC(=C1CN(C(c2occc2Cl)=O)C1)F)(C1CC1)OC Cc1nn2c(C(=O)NCc3ccc(CNC(C4CC4C)=O)cc3)c(C)nc2s1 c1(C(C(=O)NCCC(C)(C)NC(C2(C)CCC(=O)N2)=O)O)cc(F)c(F)cc1F C1(NC(Cc2ccn(C)n2)=O)CN(C(C2CCOC2)=O)CC1n1cccn1 CCCCCC(C)CC(=O)N(CCC(=O)NC1CCN(C2CC2)C1=O)C(C)C CCCCC(O)C(=O)NC1CC(S(C)(=O)=O)C1.C12CCC(F)(C1)CNC2=O C12(NC(C(CNC(C3CC(C#N)C3)=O)O)=O)CCCCC1OCC2 c1(NCC(CN(C)C)(F)F)nccc(N2CCC(C(N)=O)CC2)n1 C(C(O)CCC1CC1)N(C1COC1)C(C1CCN(c2ccccc2)C1)=O N1(C(C2CCN(S(C)(=O)=O)CC2)=O)CCCN(C(=O)CC2CCCC2O)CC1 C1(CNC(CC2ON=C(CC)C2)=O)CCN(C(c2cc(C)oc2C)=O)C(C)C1 C(CCC(C)(C)C)(c1ccn(C)n1)NC(C(=O)NC(c1onc(C)n1)C(C)C)=O O=S(=O)(c1ccc(N2CC=C(c3cccs3)CC2)c(Cl)c1)N1CCOC12CCC2 C(=O)(CC(C)C(F)(F)F)NC1C(CC)N(C(c2nc3sccn3c2C)=O)CC1 C(CCCCCc1ccccc1)c1ccc(CNC(=O)NCC(C)(O)CO)cc1 Cc1cccc(C(=O)NC(C2CCCN(C(c3c(C)coc3C)=O)C2)C)c1F N1(C(C(C2CCCC2)OC)=O)CCOCC(NC(c2ccc(O)nc2Cl)=O)C1 N1(C(C2(CCNC(CCCC#C)=O)CCC2)=O)CCOC(C)C1C N1(C(CCSC)=O)CC(NC(=O)C2=CCCC2(C)C)CC12CCCCCC2 N1(C(CCNC(=O)C(F)F)=O)CCN(Cc2ccc(N(C)C)cc2)C(C2CC2)C1 C(=O)(C(C)(C)CCNC(C1CC1(C)C(C)C)=O)NCC(C#C)CC1CC1 C(C1CCC(C)CC1)=C(C)C(N1CCC(C(C)NC(C2CCC(C)O2)=O)CC1)=O C1(CNC(CCCC)=O)CC2CCC(C1)N2C(c1conc1C1CCC1)=O N1(C(CCSCC)=O)CC2CS(=O)(=O)CC2(NC(C23CCC(F)(CC2)CC3)=O)C1 c1(OCC)ccc(C(N2CCCC2CNC(C23CCC2CC3)=O)=O)cc1Cl C(=O)(C(C(C)(C)C)NC(=O)CC1COCCO1)NCCN(CCOC)C c1(C(=O)NCC(C)(O)CNC(C2CCC(F)CC2)=O)cc(Cl)c2n[nH]cc2c1 CC#CCC(C(=O)NC1CC1C1CCC1)NC(=O)CC1CC(OC)C1 CC1C(C(=O)NCC2(C)NC(=O)NC2=O)CCCN1C(c1cc(C#N)cs1)=O c1(CC)cc(F)ccc1CC(=O)NCC1CN(C(=O)Cc2ccc(F)c(F)c2)C1 C1(CC)CN(C(=O)CC2(c3ccsc3)CC2)CCC1NC(C1(Cl)CC1)=O CC(C)C(C(=O)N1CC(NC(c2ccc(C(F)(F)F)[nH]2)=O)C(C)C1)n1cncn1 c1(OC)ccc(F)c(CN2CC(C(N3CCC(O)(c4ccc(C)cc4)CC3)=O)C2)c1 N1(C(c2cccc(CC#N)c2)=O)CCC(O)C(C(N2CCC3(CC3)C2)=O)C1 C(c1ccccc1)=CCN(C(C)(C)CCOC)C(C1(CCC)CCCCC1)=O C1(NC(=O)CN2CCC(OCc3ccccc3)CC2)CC2CNCC(C1)C2=O C1(CC(C2CC2)CN(C2CCCC2N)CC)CNCCC1C N1(C(C2(C(C)C)CCN(C(c3cnc(C(C)C)o3)=O)C2)=O)CCCC(C(N)=O)CC1 C1(C(N2CC(OC(=N)O)C2)=O)(CC)CCCN(C(C2CC(C)CC(C)C2)=O)C1 S(=O)(=O)(c1cccc(C#N)c1)NCC(=O)NC1C2N(C(CC(C)C)=O)C(CC2)C1 C(=O)(C(F)(F)C(F)(F)F)NC(CCN(C(C(C1CCCO1)OC)=O)C)C c1(C(=O)NCC(CCOC)NC(=O)C(c2cncn2C)O)ccc2nn[nH]c2n1 Cc1cc(CCCC(=O)NCC2CCCCN2C(=O)CC(C)(C)C2CC2)c(C)s1 c1(OC)ncc(-c2cc(CNC(c3cccc(C)c3)=O)ccn2)cn1 C1(OC)CCC2(C(=O)NCC(C)NC(=O)C(C)NC(=O)C3CC3)CCC12 C12(NC(c3cncc(Cl)n3)=O)CCCC1CN(C(C1CCC=CCCC1)=O)C2 c1(C2C(C(=O)NCC(C3CCC3)NC(C(C)n3cnnn3)=O)C2)cccnc1 c1(C(=O)NC(CC)CNC(=O)C(CC)N(C)C)c[nH]c2ccc(F)cc12 Cc1cc(NC(=O)CC2(O)CCNC2)n(C2CS(=O)(=O)C2)n1 Cc1ccc(S(=O)(=O)CC(C)NC(C2C3Cc4ccc(Br)cc4C23)=O)cc1 N1(C(C(C)NC(CC)=O)=O)C(CC(N2CC(N(C)C)C(C)C2)=O)C2CCCC12 c1(C(C)NCc2sncc2Br)cc2ncccc2o1 c1(C(N2CCCC(N(C(CC3ON=C(CC)C3)=O)C)C2)=O)onc2c1CCCC2 C1(CNC(C(CC)=CC)=O)CCCCN(C(=O)C2=NOCC2)CC1 C1(CC(=O)N(C(C)C)C)CCCN(C(c2cc(CO)on2)=O)C1 C(=O)(C1=C(Cl)CCOC1)N1CC(C)=C(C)CC1.c1(C(C=O)O)ccnn1C.c1ccccc1 C(c1ccc(Cl)nc1)=CC(N1CC(CNC(c2cscn2)=O)OCC1)=O N1(CCCNC(C2CC(CNC(C(C)N3CCCC3)=O)C2)=O)CCOC1=O Cc1cc(C(N2CCCC2CCCNC(=O)CCCSC(C)(C)C)=O)nc(C)n1 C1(NC(C(C(C)O)(C)C)=O)CCN(C(c2cscn2)=O)CC(O)C1 C(CC(C)C)(C(=O)NC1CCCC1CC(=O)NC(C)(CO)C1CCC1)OC N1(C(c2ccn(CC)c2C)=O)CC(CNC(C2CC=CC2)=O)CC1(C)C C1(C(=O)NC2CN(C(C3C(C)OC(=O)N3)=O)C2)CCCC(=O)N1C N1(C(c2ccc(C#C)nc2)=O)CC(C(=O)NCCN2CC=CC2)CC12CCC2 C(=O)(CCCCCCCCCO)NC(C(C)C)(C)CNC(c1ocnc1C1CC1)=O c1(C(=O)NC2CCCN(C(C=C(C)c3cccs3)=O)CC2)nccc2occc12 C#CC1(C(=O)NCCc2cnc(C)[nH]2)CCN(C(=O)C2=CCCC2C)C1 CCCC(O)CC(=O)NC1(C)CCN(C(C2CC2(F)F)=O)C1 c1(SC)ccc(NCc2cccnc2Cl)c(Br)c1 C1(NC(C2C(CC)C2)=O)C2CC3CN(C(c4ccnc(C)c4)=O)C1C3C2 c1(C(N(CCOC)CCNC(C2CCCC2(C)C)=O)=O)cc2scc(Cl)c2[nH]1 C(c1cccnc1)=CCNC(C1(NC(C(C)SCC)=O)CC(CO)C1)=O Cc1c(CC(=O)NC2CN(C(=O)C(C)(O)C=C)CC2C)cccc1[N+](=O)[O-] c1(Cn2cc(C(c3nccc(C)c3)(C)CN)nn2)ncc(Cl)cc1F c1(C(N(C2CCN(C(c3cc(CC)on3)=O)C2)CCC)=O)c[nH]nc1Br C1(C(=O)NCc2ccc(C(=O)NC(C)CCC3CCCC3)o2)CC(F)C(=O)N1 c1(CNC(CC2(C)N(C(C(C)=CC3CC3)=O)CC2)=O)ncccc1C(N)=O C1(NC(CONC(c2c(C#N)ccs2)=O)=O)CCCCCCC1O C(=O)(CCC(CC)OC)NC1CCC(C(=O)NC(C=C)C(F)(F)F)C1 c1(CCC(=O)NCC(CNC(C(c2cncc(F)c2)C)=O)O)c(F)cccc1F c1(OC)cc[n+]([O-])c(C(=O)NCCC2CCCCN2C(c2cnc[nH]2)=O)c1 c1(C(=O)NCCNC(=O)CCOCC(F)F)cccc(NC)n1 N1(C(C(c2c(Cl)cccc2Cl)C)=O)CC2CCC1C1CN(C(C3CC(O)C3)=O)CC21 c1(C(N(C)CC2CC2)=O)ccc(O)nc1.C1(Nc2ccccc2)CC(=O)N(C2CC2)C1 N1(C(=O)OC(C)(C)C)CCN(C(=O)CCc2cnc(C3CC3)o2)CC1C1CC1 c1(C(=O)NCC(CC=C)NC(=O)CCc2cccnc2C)cn(C)nc1Br C1(CNC(c2cnc(CCCC)s2)=O)CN(C(C2NC(=O)OC2C)=O)CC1O C12(CNC(CCOC)=O)CC1CN(C(=O)Cc1noc(C)n1)C2 C12(C(N3CCC(N4CCN(C(c5cc[nH]c5)=O)CC4)C3)=O)CC3CC1(CO)CC3C2 Cc1cn2cc(C(=O)NCCOCCNC(C3CCCC4(CC4)C3)=O)sc2n1 C12(CNC(Cc3cn(C)nc3)=O)CCCCC1N(C(C1COC(=O)N1)=O)CCC2 Cc1ccc(C(=O)NCCN(C(=O)CC2CCCN(C)C2)C2CC2)c(O)c1 C1(C(=O)NCCN(CCOC)C(c2cc(C)cnn2)=O)CC2(CCC2)CO1 c1(OC(C)C)cnc(=NCC2C(C)CCCN2C(C2COCCO2)=O)[nH]c1 C=CC(C)C(=O)NCC(C1CCC1)NC(=O)CCCc1n[nH]c(=N)s1 C(=O)(CC(C)(O)C(F)(F)F)NCCCN(C(C(C(=O)OCC)F)=O)C C1(NC(c2ccc(OC)c(Cl)n2)=O)CCC2(CC1)CC2NC(c1cscc1Cl)=O N1(C(=O)Nc2cc(NCc3ccccc3)ncn2)CCC2COCC12 c1(CNC2C=CC(C(=O)Nc3cc(OC)nnc3)C2)ccc(F)c([N+](=O)[O-])c1 N1(C(C2CC(OC)C2)=O)CC(CNC(c2cnc(Br)s2)=O)CC12CCC2 c1(CC(C)C(=O)N(C)CC2(NC(C3CCS(=O)CC3)=O)CC2)ccc(Cl)cc1 C(=O)(C(CC(C)C)C(C)C)NCCN(C(C1OCC2COCCC12)=O)CC c1(OC)cc(C(=O)NC2CN(C(=O)C(N3CCCC(O)C3)C)C2)c(Cl)cc1Cl N1(C(c2c(C)nc(O)cc2)=O)CCC2(CC1)CC2C(N1CCC(C(C)C)C1)=O N1(C(C2CCN2C(C2COCCO2)=O)=O)CCOCCC1 C1(NC(C(c2ccc(C(N)=O)nc2)C)=O)CCC(C)N(C(c2ncc[nH]c2=O)=O)C1 c1(OC)cc(C(=O)NCC2CCC(NC(c3nocc3Cl)=O)CC2)ccc1C#N CCC(C)CC(C(=O)Nc1cccnc1C)NC(c1cnc(C)o1)=O C12(C(N3CCC(C)(CCO)C3)=O)CCCC1CCN2C(C1CC(F)C(=O)N1)=O C1(NC(COc2cccc(C)c2)=O)C(C)CN(C(=O)Cc2sccc2C)CC1C C(=O)(CC(CN(C)C)C(F)(F)F)NC1C2(CN(C(CC(=O)N(C)C)=O)C2)CC1 C1(NC(C(C(CC)CC)C)=O)CCN(C(=O)COC2CCCOC2)CC12CCC2 N1(C(C2CCC(CCC)CC2)=O)CCCC(C)C1CNC(=O)C(C)SC N1(C(CCC=C=C)=O)C2CCC1C(C(=O)NCC1(SC)CC1)C2 Cc1cc(F)cc(C)c1C(=O)NCC1CCC(C)N(C(=O)C(F)=C2CCCC2)C1 C(N=c1cc(NCCCOC(=O)N(C)C)nc[nH]1)C12CC(C(=O)OC)(OC1)C2 C(=O)(CCC(C)N(C)C)N(CC(C)(C)C)CC(=O)NCC(CC)CC C1(NC(CCn2c(C)ncc2)=O)CC(F)CN(C(=O)C(C2CCOCC2)=O)C1 c1(CC)ccc(Br)cc1C(=O)NC1CC2CC1N(C(C1CCOC1)=O)C2 C(CCN(C)CC)(C(=O)N(c1ncccn1)C)NC(COCCCC#C)=O C1(C(N2CCC(CNC(c3ccc(C(F)F)cc3)=O)C2)=O)CC2(C1)CC2F CCCC(C(=O)NC1(C2CCN(C(C3OCC4CCCC34)=O)C2)CC1)C(C)C c1(C(=O)NC2CN(C(CC(=C)Br)=O)C(C)CC2)cc2ccccc2nc1O c1(C(=O)NC2CCCN(C(c3cccc(C(=O)OC)c3)=O)C2)cn2c(n1)SCC2 c1(C(N2CC(C(C)NC(c3ccc(C)[nH]3)=O)C2)=O)cnn2c1NCCC2 C(=O)(CCC(C)CC)NC(CC#CC)C(=O)N(CC(=O)NC)CCC c1(N2C3CC(CC(NC(C4CCSC4)=O)C3)C2)ncnc2cccc(Br)c12 C(=O)(C(C(C(C)C)C(C)C)N1CCC2(CCC2)CC(CO)C1)NCCCC N1(C(CC(C(C)C)C)=O)CCC2(C1)CN(CC(N)=O)CC(C)O2 c1(C(=O)NCC(C)N(C)C(c2ccon2)=O)ccc(C#N)[nH]1 C1(S(C)(=O)=O)(C(N(C(C)CNC(=O)CC(C)C(F)F)CC)=O)CCC1 c1(C(N2C(CNC(C(C)O)=O)CC3(CC3)C2)=O)cc(F)c(O)c(Br)c1 C12C=CCC(C1)C(=O)N2.c1(CNC(CN(C)CC)=O)cnn(CC2CCCC2)c1 c1(C(N(CC(C)NC(C2C(=C)C2)=O)CC)=O)cc2cc(Br)cn2cn1 C1(O)(C(=O)NC2CC(C)(CNC(CCCSCC)=O)C2)CCC(C(F)(F)F)CC1 C(=O)(C(CNC(C1(CC)CC1)=O)OC)NCC(=O)NCC=C N1(C(c2c(C)nsc2)=O)CCN(C(=O)CC2CCC3(CCC3)O2)C(C2CC2)C1 C1(NC(CCOCCOC)=O)CCN(C(=O)Cc2ccccc2O)C12CCC2 N1(C(CC(CC)C2CC2)=O)CC(C(=O)NCC(C)(F)F)CC1(C)C c1(OC)cc(OC)cc(N(C)C(c2cn(-c3cccc(Br)c3)nn2)=O)c1 CC1CN(C(C2(CO)CCCO2)=O)CC1(C)CNC(=O)CC(C)(C)O C(=O)(C(O)CCCNC(c1cn(C)c(C)n1)=O)NCc1cccc(CC)c1 n1(CC)nc(C)c2cc(C(=O)NCCNC(=O)C(=O)N(C)C)sc12 c1(C(C(=O)NCC(C)(O)C2CCC2)NC(C(CCOC)C)=O)c(C)cccc1Br CCC(C)C(=O)NCCC1(C2CCCN2C(=O)C(n2cc(C)cn2)C)CC1 c1(C(=O)NCC2(CNC(C3(C)CC4(CC4)C3)=O)CCC2)cncc2c1CCCC2 C1(NC(C(C)N(C)C)=O)CCCOC12CCN(C(c1csc(F)c1)=O)CC2 c1(C(=O)NCC(CC)NC(c2ccn(C(C)(C)C)c2)=O)cnn(CC(F)(F)F)c1 C(=O)(C1c2ccccc2CN1C(c1nc[nH]c1[N+](=O)[O-])=O)N(C)C.C1(=O)CN1 c1(N(CCN(C(C(C(C)C)SCC)=O)C)C)cc(C)nc(C(C)CC)n1 C1(OC)CC2(C1)CN(C(=O)C(C)N(C)C(C1(C#N)CC=CC1)=O)C2 c1(C(=O)NC(CC)CN(C(C2CCCCN2C(C)=O)=O)CC)cc(C)ccc1Cl C=CCC(CC(=O)N(C1CC(O)C1(C)C)C)NC(=O)CC1CC1(C)C C1(C(=O)NCCN(C(C(C)C2CCC2)=O)C(C2CCCC2)C)C(F)(F)C12CCC2 N1(Cc2ccc(Cn3cc(CC(=O)OC)nn3)cn2)CCOCCC1=O N1(c2ncn(C)c(=O)c2Br)CC2CCC1C1CN(C(=O)C=CC(N)=O)CC21 N1(C(c2cc(C)[nH]n2)=O)CCC(CCNC(c2cnn(C)c2Cl)=O)CC1C CCCCCC(O)CC(=O)NC(C1CCCCC1)CNC(c1ccnc(C)n1)=O c1(C(N2CC(C(C)NC(c3c(C)cnnc3)=O)OCC2)=O)ccc(O)c(F)c1F N1(C(N(CCN(C(=O)C(C)C(C)C)CC)C)=O)CC=CCC1 Cc1ccc(F)c(OCC(=O)NCC2(C)CCCN2C(c2cscn2)=O)c1 c1(CNC(=O)C=CCNC(c2[nH]ccc2C2CC2)=O)cc(C(F)F)[nH]n1 c1(NCCC(CC)C)cc(NCC2CC3(CC3)CO2)ncn1 CCC(C)(C#N)C(=O)N1CC(OCCNC(C2CC3CCOC23)=O)C1 C1(COC)(NC(C2CC23CCC3)=O)CCN(c2ccccc2)CC1 c1(CCC)ccc(C(=O)NCC2C3CN(C(c4ocnc4C4CC4)=O)CC23)cc1 C1(NC(CC=C)=O)CCS(=O)(=O)C12CN(C(=O)Cc1cc(C)[nH]n1)C2 C1(NC(CC2(CC)CCC2)=O)CCCN(C(=O)C(=O)NOC)C1 C1(C)(C(=O)OC)CCCN(C(C2CCN(c3ccncc3)C2)=O)C1 C1(=CC(=O)NCC(N2CC(OC(=O)N(C3CCC3)C)C2)=O)CCOCC1 c1(C(N2CCC(N(CCC)C(c3ncccc3O)=O)C2)=O)cnn2cccnc12 c1(C(=O)NCCC2N(C(CCC=CC)=O)CC(OC)C2)cnn2ccsc12 C12CC3CC(C3C1)C(=O)OC2.c1(C(=O)OCC)cc(C2CC2)[nH]n1 C1(OCC#C)CCN(C(C2CCN(C(=O)CC(C)C=C)C2C)=O)CC1 C1(NC(C(C=CCCC)O)=O)C(C)(C)CN(C(=O)CC2CSC2)CC1(C)C N1(C(CCn2c(C)cc(C)n2)=O)CCC2(CC1)CC2NC(c1ccc(F)cn1)=O C1(CNC(C=CCCC)=O)CCC12CN(C(c1ccc(-n3cnnn3)cc1C)=O)C2 c1(CC(=O)NCC2(NC(=O)CC3CCCC(=O)N3)CC2)ccc2cnccc2c1 N1(C(C(C)CNC(C2CC3CC(=O)C2C3)=O)=O)CC(C2=NOCC2)C1 c1(N2CCN(CC(=O)Nc3cccc(Br)n3)CC2)ncnc2sccc12 N1(C(C2(N(C)C)CC2)=O)CCC2(CC1)CC2NC(c1cc(C)c(SC)c(C)c1)=O N1(C(C=C=C(C)C)=O)CCC(C)CC1CNC(=O)Cc1cc(C2CC2)no1 Cc1ccc(C(N2CCCC(CCNC(c3nonc3N)=O)CC2)=O)c(C)n1 c1(C(C(C)NC(c2cccc(C)c2)C(=O)OC)=O)ccc2c(c1)CCC2 C(=O)(C(C)CC(=O)OC)NC(C(=O)NCCSCC#C)Cc1cn[nH]c1 c1(C(C(=O)Nc2ccc(F)cc2)N(C2CCN(CC)CC2)C)cccc(SC)c1 C1(C(=O)NCc2ccc(Br)c(F)c2)CN(Cc2ccnc(Cl)c2F)CC(F)(F)C1 C1(C(=O)NC2C(CNC(COCC(=C)C)=O)COC2)C2CC3C(C2=O)C13 Cc1csc(C(N2CC(CC(F)C(=O)NC3(C)CC3C)C2)=O)c1C CC1CCN(C(C2CCCN(C(=O)C(F)=CC3CC3)C2)=O)CCS1 Cc1c(C(=O)NCC2=CCN(CCN3C(=O)CCC3=O)CC2)nc2sccn12 c1(C(=O)NCC=CCNC(CC)=O)ccc2c(c1)CCCCC2=O c1(C(C(N2CC(C)C(NC(=O)C(F)(F)CN(C)C)C2)=O)(F)F)cccc(Cl)c1Cl c1(COC)cc(C(=O)N(CC(C)N(C(=O)CSCC(C)C)C)CC)no1 C1(COC)(CNC(C2CCCOC2C)=O)CCCN1C(c1nonc1N)=O c1(OC)nccc(C(=O)N(C)CC2CCCN(C(C3CC3(C)C)=O)C2)c1Cl N1(C(c2ccc(C(C)=O)s2)=O)CCCC(NC(=O)CC2CCCNC(=O)C2)CC1 c1(C(N2CCC(N3CCC(O)C3)C2)C(=O)NCCOC)c(C2CC2)cnn1C C=CCC(C(=O)NCc1occc1C(=O)NCC(CCC)CCO)C(C)C C(CO)(CCCCNC(=O)C(F)F)NC(C1CCCN(c2ncccn2)C1)=O N1(C(C(COC)C)=O)CCCC(C)(NC(=O)Cc2cnn(C3CC3)c2)C1 c1(C(N2CCC(O)(C(C)NC(C(CC)SC)=O)C2)=O)cccn2cc(C)nc12 N1(C(c2ccn(C)c2)=O)CCC2CN(C(c3ccnc(F)c3F)=O)CC12 N1(C(c2cc(C(C)C)[nH]c2C(C)C)=O)CCN(C(=O)COC2(C)CCOCC2)C2CC12 C1(=CC(=O)NC2C=CC(C(=O)NCC3CC3c3cccnc3)C2)CCCCC1 CC1CN(C(c2nc(C(F)(F)F)no2)=O)CCC1NC(=O)COC1CCCC1 C(C(N=c1[nH]ccn2nnnc12)c1ccccc1)N(C1CN(S(C)(=O)=O)C1)C N1(C(CCCC)=O)CCCC(Oc2cc(NC(=O)C(O)C(F)(F)F)n(C)c2)CC1 C1(C(=O)NCCCN(C(C(C=C=C)C)=O)CCC)CC2COCC2C1 Cc1nc(C(N2CCCC2CN(C(=O)CCOC(C)C)C2CC2)=O)ccc1C#N C1(CN(C(CC2CC(OC)C2)=O)C)CCN(C(C2CCC2)=O)C1 CC(C)S(=O)(=O)CC(=O)NC1(CF)CCN(C(=O)C=Cc2cccn2C)C1 C1(OC)(CO)CCCN(C(C(=O)NCC2CCCO2)C(C)CC2CC2)C1 C12(NC(C(C)NC(CC)=O)=O)CCOCC1CN(C(C1CC3(CCC3)CO1)=O)C2 c1(C(N2C(C(=O)NCCC(C)N3CCCC3)CC=CC2)=O)ncn2c1CCC2 N1(C(C2(OCC)CC2)=O)CCCC(CN(C(c2csc(CO)n2)=O)C(C)C)C1 c1(CC(N2C3C(NC(C4C(C)=C4)=O)C(C3)C2)=O)c(C)nc2ncnn2c1C c1(NC(C2C(CC)CCC2)=O)ncnc2ccc(O)cc12 c1(C(N2CC(C(COCCOCCOCCOC)=O)OCC2)=O)nc(Cl)ccc1Cl.OC Cc1nc(NC(=O)C(=O)N(CC(F)CC2CC2)C)nc(Cl)c1Br c1(CC(=O)NC2CC(CCNC(=O)C(Cl)=CCl)C2)cccc2nsnc12 c1(C(=O)NC2(CF)CCN(C(C3CCOC3)=O)C2)sc2cccnc2c1Cl C=CCC(C)(C)CC(=O)NCCOCCCN(C(=O)C(C#N)C1CC1)C.C(C)(=O)N N1(C(CN(C2CCCCC2)C(C)=O)=O)CCC2(NC(=O)C(C)C3CC3)CCCC12 N1(CC(=O)N(C)CCNC(=O)CN2CCCCCC2=O)CC(=O)N(C)C1=O.C1CC1 c1(C(N(C2CCCCN(C(c3c[nH]c(=N)s3)=O)C2)C)=O)cn2cccc(Cl)c2n1 C1(CNC(C(COCC)n2cc(CC(O)C3CCC3)nn2)=O)CCC(=O)NC1 CCCS(=O)(=O)CC(=O)NC1(C2CCCN2C(C23CCC(CF)(C2)OC3)=O)CC1 CN1CC=C(C(=O)NOCC(=O)NCC(C)(C)CCCO)C1 O=S(=O)(c1ccc(NCC2CCC(O)C2)cc1Cl)NCCCN1CCOCC1 CN=C(NCC1CCC(c2ccccc2)O1)N1CCC2(CCOCC2)C1 CCCCCCCCC(C(=O)NC1CC1)N1CC2CCC1C(O)C2O c1(CC)onc(C(N2CCC3C(NC(=O)Cn4ncn(C)c4=O)C23)=O)c1C C1(NC(C2(NC(C(c3cncnc3)C)=O)CSC2)=O)CCOC2(CCC2)C1 CC(O)C(C)(C)C(=O)NCC(O)CNC(=O)Cc1nncn1C c1(C(N2CC(CC(N3CCC(=C)CC3)=O)C2)=O)ccc(Br)c(F)c1F C1(C(=O)NCC2N(C(c3cccc(C)c3C)=O)CCOC2)CCn2nnnc2C1 C1(Cn2cc(C(C(C)C)O)nn2)N(C(C2(c3ccccn3)CC2)=O)CC1(C)C CC1CC(C(N2CCOCC(C(=O)O)C2)=O)CCN1C(C1CCCC1)=O C1(C(N(C2CC(C)(O)C2)C)=O)C(CNC(c2csc(F)c2)=O)C1(C)C C1(c2n(CCCSC)nnn2)(NCCC(C2CCOCC2)O)CCC2COC1O2 C1(C(=O)NCCCCNC(c2c(C(C)C)cccc2)=O)CCC(=O)N(C(C)C)C1 c1(N(CCCn2cncn2)C(C2CCC2)=O)ccc(-c2cnsc2)cc1 c1(C(=O)NCCC2(NC(C(C(C)C)OCC)=O)CCC2)c(CC)nn(C)c1Cl C(=O)(CC(C)C(C)(C)C)N1CC2C(CNC(COc3ccc(CC)cc3)=O)C2C1 c1(N(CCC)C(C2CN(C)CCO2)=O)ccnc(Br)c1 C(C1COC(C)(C)O1)=CC(=O)NC(CNC(c1cc(CCC(C)C)[nH]n1)=O)(C)CO C1(CC(=O)NCCc2n(C)cnn2)CCCCN1C(=O)C=CC1CCCCC1 c1(C(=O)NCCCN(C(c2cc(Br)c[nH]2)=O)CC)c[nH]nc1F N1(C(C(C)(C)SC)=O)CCCN(C(=O)CC2OCCC2(C)C)CCC1 CC1CCCN(CCN(C(=O)CSC2CCCCO2)C2CCC2)C1 C(C1c2ccsc2CCN1C(c1nccc2n[nH]cc12)=O)NC(C=CSC)=O c1(C(=O)NC(CNC(C2C(C=C)CC2)=O)(CC)CC)cc([N+](=O)[O-])ccc1SC C(=O)(CCS(=O)(=O)C(F)(F)F)NCCCNC(c1c(C)cccc1F)=O N1(C(C2CCC(C)S2)=O)CC2(CC(NC(=O)CC3(C)CCCCC3)C2)C1 C1(CC)CN(C(=O)C(O)C(C)(C)C)CCN1C(=O)CSC(C)C c1(CNC(N)=O)cccc(CC2(C(=O)NCC)CC2)c1.C1(C(=O)N)(CCO)CC1 c1(C(=O)NC2(C3CN(C(C4=C(C)CC4)=O)C3)CC2)cnc2c(C)nsc2c1 c1(C(N2CC(CN(C(C3C(CCC)C3)=O)C)C2)=O)csc2ncnc(O)c12 C1(OC)CC(CNC(c2c(F)cnn2C(C)C)=O)N(C(=O)C(CC(C)C)SC)C1 C1(NC(c2cccn(C)c2=O)=O)CC2CC1N(C(c1cc(C(C)(C)C)c[nH]1)=O)C2 C(CCC)(C(=O)N1CCCC1C(C)C)=CCC.c1(C(=O)NCC)cnc(Br)s1 CCCC(CCC)=CC(=O)NC(c1cn(C)nn1)C(N1CC(C#N)(CCF)C1)=O Cc1cc2c(C(=O)N(CCCN(C)C(C3CCC(O)C3)=O)C)cccc2o1 C1(C(=O)NCC(C)(CO)NC(c2c(C)ocn2)=O)CCN(CC2CC2)CC1 C1(C(=O)NC2CCC(C#N)CC2)(CC)CCN(C(C2CC(F)CN2C)=O)CC1 N1(C(C2(CC)COC2)=O)CCC(NC(c2cc(C(C)C)ccc2F)=O)C(C)(C)C1 C(CC(C)C)(C(=O)NCC1(F)CCN(C(=O)C(C)=C2CC2)CC1)NC(=O)OC c1(N2C(CCNC(c3cncc(Cl)c3)=O)CSCC2)ncnc2cc(Br)ccc12 N1(C(Cn2nc(C)oc2=O)=O)CC(N(C)C(C2CC3CC(=O)C2O3)=O)C2(CC2)C1 C(CCC(=O)N(CC(C)N(C(=O)CSCC(C)C)C)C)N(CC=C)CCC C(=O)(C1=CCS(=O)(=O)C1)NCC1OCCN(C(C(F)(F)C2(OC)CCC2)=O)C1 Cc1cc(C(=O)N2CC(n3cc(C(N4CCOCC4)CCO)nn3)CO2)ccc1N c1(C(=O)NCCCN(C(CCCCN(C(C)=O)C)=O)C)ccc2occc2c1 CCCC(CCCNC(c1cn(C)cc1CC)=O)NC(=O)Cc1nnc(C)o1 c1(OC(CNC(C2CN(C(C)=O)C2)=O)C(=O)NC(C)C)ccccc1F C#CC1(C(N2CC(F)(CO)C2)=O)CCN(C(=O)C(CC2CCC2)OCC)C1 N1(C(c2c(CO)occ2)=O)CC(CO)C2(C1)CN(C(=O)CN1CCCC1CC)C2 C(=O)(CC(O)CC(C)(C)C)NCc1ccc(C(N2C3(CN(C)C3)CC2)=O)o1 c1(N(C(C2CCN(Cc3cccc(OC)c3C)C2)=O)C)nccc(S(C)(=O)=O)n1 c1(N2CCC(OC)C(F)C2)ncnc2c1cnn2C(Cc1ccccc1)C(N)=O C12(CNC(c3cnc(CSC)s3)=O)CCC1CN(C(=O)CCc1cccn1C)C2 C1(C(=O)NC2C(CC)CCC2)C2CC3C(C2NC(C2(C)CCCS2)=O)C13 C1(C(=O)NCC2C(NC(C3(OC)CCCCC3)=O)C2)CCc2ncc(C)n2C1 C1(C(=O)NCC2CCCCN(C)C2)(NC(CSCC(C)=O)=O)CCCCCC1 C(=O)(CCCCCCN=[N+]=[N-])NC(CNC(C1N(C)CCOC1)=O)C(C)(C)C N1(C(C2(C)N(C(c3n(CC#C)ccc3)=O)CC=C2)=O)CCn2c(C)nnc2C1 c1(CS(C(COCC=C)CO)(=O)=O)ncnc2sc(C)c(C)c12 c1(-n2ncc(C)c2)ccc(NC(=O)C(N2CCNC(=O)C2C(C)C)=O)c(C)c1 c1(OC)c(Cl)ccc(Cl)c1C(=O)NCCC(C)NC(=O)CCS(C)(=O)=O N1(C(C(C)OCCC=C)=O)CCC(C(F)F)(OCCOCCC(=O)NCC)C1 c1(NC(C)=O)ncc(C(=O)N(CC(C)CNC(=O)CC(C)c2ccncc2)C)o1 C1(CC)Oc2cc(C(C)C(=O)NC(CC(C)C)c3ccccn3)ccc2NC1=O CC(C)C(F)(CNC(c1cnn(C)c1Cl)=O)C(=O)NCCCC(=O)NO C(=O)(C1CCc2ccccc21)N1CCC2CN(C(C3=NNC(=O)CC3)=O)CC21 c1(C(=O)NCCC(=C)CNC(=O)Cc2c(C)n[nH]c2C)cnc2c(c1)nnn2C c1(C(=O)NCC2C(NC(c3c(C(=O)OC)cncc3)=O)C2)ccc(C)c([N+](=O)[O-])c1 C1(NC(CC(=O)NCC)=O)CC(C)CN(C(=O)CCc2ccc(F)nc2)C1 CC1C(=O)CCC1CCNC(=O)CCN(C(=O)NCC1CC1)CCO C(CC(C(=O)N1CC(C)=C(C)C1)NC(=O)Cc1cc(C)cs1)OC C12(CNC(c3cnc(OC)nc3)=O)CN(C(c3cn[nH]c3)=O)CC1(C(F)(F)F)C2 C(C(=O)NCCN1CCN(C(=O)C(F)(F)C2CC2)CC1)(C(C)C)n1cc(C)nc1 N1(C(C=Cc2n(CC)ncc2)=O)CCN(C(c2ccc(C(F)F)s2)=O)CC(CO)C1 S(=O)(=O)(c1cccc(C#N)c1)NC(C(=O)N(C(CNC(CCC(=C)Cl)=O)C)C)C C12(CNC(C(C)C3CC3)=O)CN(C(c3ccc(Cl)cc3Cl)=O)CC1CCO2 C(=O)(C(C(C)(C)C)NC(c1cncc(N)n1)=O)NCCNC(COC(CC)C)=O C1(CN(C(N(c2ccccc2F)CCOC)=O)C)CCN(c2ccccc2)CC1 N1(C(C(CC)C(C)O)=O)CC2(CCCN(C(=O)C(c3ccccc3Cl)(F)F)C2)C1 C1(NC(C2(CC=C)CC2)=O)CCCC1(C)CNC(=O)Cc1cnco1 CN1CC(C(N2CCN(Cc3cn(CC4CCOC4)nn3)CC2)=O)NC1=O CC(CC(=O)NCCC1(NC(c2cc(N)ccc2Cl)=O)CCCC1)C(F)F c1(O)ccc(Cl)cc1F.C(=O)(C(CCC)OC(C)(C)C)OCCN(C(CCC=C)=O)CC CC1C(NC(=O)CCCN2CCCCC2)CCN1C(=O)Cc1coc(C(F)F)n1 N1(c2snc(COC)n2)CC(CNC(=O)Cc2c(F)cccc2F)CCC1C C(=O)(CC(CNC(=O)Cc1ccc(C)nc1)OC)Nc1cn(CC)nc1 COn1cnc(C)c1C(=O)NCCC1CC(NC(c2c(C)noc2N)=O)C1 C(=O)(C1Cc2ccc(F)cc21)NC1CC(C)N(C(=O)CC(C2CC2)C2CC2)CC1 C1(C)(C(N2C(CCNC(C(CC)CCOC)=O)CCC2)=O)CCCCCCC1 N1(C(c2c(N)cc(C(F)(F)F)cn2)=O)CCC(C2(CNC(=O)CCF)CC2)C1 c1(CNC2(N3CCN(C(=O)CO)CC3)CC2)cn2ccccc2n1 Cc1ccc(C=CC(=O)NC(CNC(C2CC2c2cccc(F)c2)=O)C(C)C)s1 C12(CNC(CCC(C)C)=O)CCC(C1)N(C(C1CCCN1C)=O)C2 C1(CCNC(C)=O)CN(C(C(=O)N(c2ccccc2)C(C)C)c2ccco2)CCO1 C1(CN(C(=O)CC2(CNC(C3CC(C)(O)C3)=O)CC2)C)CCCCC1n1ccnc1 C(=O)(CC(C)P(C)(C)=O)NCC1C2CN(C(C(C(C)C)NS(C)(=O)=O)=O)C1C2 n1(CC)ncc2cc(C(N3CC(C(N)=O)C(CCO)C3)=O)cnc12 C1(C(=O)NC2CCCN(C(c3c(CC)nco3)=O)C2)CC(F)(F)CCC1(C)C Cc1cc(CC(N2CC(CCNC(C34CC(O)C3C4)=O)C2)=O)sn1 CCC(C)C(O)C(=O)NCC1CC(CNC(c2nnn(C3CCOC3)c2C)=O)C1 O=C(C1=CCCOCC1)N1CC2(NC(=O)C(O)CN3CCCC3)CCC1CC2 C=C(Br)CCC(=O)N1CCCC1C(C)(C)NC(=O)CN1CCCC1CO N1(C(CCCCCC=C)=O)CCCC(C2CCN(C(C3SCCCS3)=O)CC2)C1 c1(OC)nccc(=NC(=O)C(F)CC(F)(F)C(=O)OC(C)(C)C)[nH]1 C1(SC)CCN(C(=NCCF)NCC2CC2)C1 N1(C(C(C=C)(C)O)=O)CCC2C(CCCN2C(c2ccc(C(C)=NO)cc2)=O)C1 Cn1cnc2cc(C(=O)NCC3CCCCN3C(=O)C3=COCCC3)ccc12 c1(C(N2CC(CNC(C(C3CC3)OC)=O)C2)=O)ccc2nc(C(F)F)[nH]c2c1 N1(C(C(C)(F)F)=O)CCCCC(NC(c2cccc(N(C)C)c2)=O)C1 N1(C(c2cnccc2Cl)=O)C2CCC(C2)C1C(N1CC(F)(F)C1)=O c1(C(N(CCNC(C2(n3cncn3)CC2)=O)CC)=O)cn(C2CC2)nn1 N1(CC(=O)NCCN(C(=O)Cc2cnn(C)c2)CCC)CCCC1CN(C)C C1(C(N(C2(CF)CCN(C(C3CCC3(OC)OC)=O)C2)CC)=O)CC2(C1)CC(O)C2 C(=O)(C(CC(C)C)SC)OC(C=CCNC(c1cncc(NC=O)c1)=O)=O c1(C(=O)NCC(N(C(=O)CSS(C)(=O)=O)C)C2CC2)cc(C2CCCO2)n(C)n1 C1(O)(CNC(C(C)OC)=O)CCCN(C(=O)Cc2cnc(C)[nH]2)C1 O=C1CCCCC1OC(=O)NNC(c1ccccc1Br)=O C1(C(N(CCCC)C(C)CC)=O)CCC2(CC2)N1C(c1nccc(C)c1N)=O c1(CC)nnc(C)cc1C(=O)NCC1(OC)CN(C(C2(O)CCC2)=O)C1 C#CC12CCC(C(=O)NC3CCN(C(c4cc(C)c[nH]4)=O)C3)(CC1)CC2 Cc1cnn2c1CN(C(=O)CC(CNC(=O)CCCF)C1CCC1)CC2 c1(CC)nnc(O)c(C(N2CCC3(NC(=O)C=CCOC)CCCC23)=O)c1CC c1(C(=O)NCC(C(=O)NCC2(C(C)(C)OC)CC2)O)ncn(C)c1C CC(C)(O)C#CC(=O)NCC1CCCN1C(c1cc(Cl)no1)=O C1(C(=O)NCC(CN(C(c2cncc(NC)c2)=O)C)C)C2(CCC2)C12CCC2 c1(CC)ccc(C(N2CC(CNC(c3cnoc3CC(C)C)=O)C2)=O)[nH]1 c1(CC(N2CCC(=CCNC(C3CCC4CC4CC3)=O)CC2)=O)ccc(F)c(Cl)c1 C(=O)(CC(C)CF)NCC(CCOC)NC(c1oc(CC(C)C)nc1C)=O N1(C(C(CCF)NC(C(C)n2ccnn2)=O)=O)CCCN(C)CCC1 c1(C(=O)NC2C=CC(CNC(=O)COCCOCCO)C2)cccnc1O N1(C(C(CC=C)NC(C)=O)=O)CCN(C)CC1CNC(c1ccnn1CCF)=O CCCN=C(NCC1CCC(=O)NC1)N1CCC(c2ccccc2COC)C1 N1(C(CNC2CC(NC(CCc3c(C)ncs3)=O)C(O)C2)=O)CCS(=O)(=O)CC1 c1(C(=O)OC)ccc(C(=O)NC(c2c(SC(C3CCCO3)C)scc2)=O)o1 c1(OCC(C)C)ncccc1C(=O)NCC(C(C)C)NC(C1C=CCC1)=O C1(OCC)(CNC(c2cnc(C3CC3(F)F)s2)=O)CCCS(=O)(=O)C1 c1(C(C)C)cc(N2CCC(C)C(NC(=O)Cc3c(O)ncnc3O)C2)nc(Cl)n1 c1(C(=O)Nc2ccc(C(F)(F)F)cn2)ccc(=NCc2cccc(I)c2)[nH]c1 C1(F)(C(N(OCC(=O)O)C)=O)CCN(C(=O)CN2CCCC2)C1.C(c1ccccc1)=CC C1(C(=O)NCC(=O)NCC(=O)N(C)Cc2cncn2C)CCCN(C)C1 CCCCC(C)(C)NC(C12CC1CCN2C(c1csc(C)c1)=O)=O c1(OC)cc(CN=c2ccnc(NCCN3CCOC3=O)[nH]2)cc2cccnc12 Cn1c(C(N2CCC(C)(CCNC(c3csnn3)=O)C2)=O)cc2occc12 c1(CC)ncc(C(=O)NCC(C2(O)CN(C(=O)C(F)=C(C)C)C2)(C)C)s1 C1(NC(C=CC=CC)=O)CCN(Cc2nc(-c3cc(C)oc3C)no2)CC1C N1(C(C(CC)(C)F)=O)CCC2(CC1)CN(C(c1cncc3c[nH]nc13)=O)C2 c1(C(=O)NCc2nccc(NC(c3c[nH]ccc3=O)=O)c2)ccc(O)cc1O c1(OC)ccccc1C=CC(N1CCCC(NC(c2ccc(Cl)cc2)=O)C1C)=O N1(C(C)=O)C2CCCC1CC(NC(C1CCC3(CCC3)CC1)=O)C2 C1(C(N(CCCOCCNC(C(C)=C2CCCC2)=O)C)=O)CCC(C)(C)OC1 Cc1cc(O)ncc1C(=O)NCC1CCN(C(C2CCCCC2(C)C)=O)C12CC2 N1(C(C(C)=C2CCC2)=O)CC=C(CNC(=O)C(c2cnccc2C)(C)C)CC1 C1(C(N2CCC(NC(CCOCCOC)=O)CC2)=O)CCc2nn[nH]c2C1 C1(C(=O)Nc2c(C)n(C3CCC3)nc2)CC(c2ccc(F)cc2)=NO1 CC(C)C(C)(O)C(=O)N(C1CCCN(C(=O)CC(C)(C)c2ccc(F)cc2)C1)C c1(NC(c2n(C)ncc2)C(F)F)nc2ncc(Cl)cc2o1 N1(C(CC=CCC)=O)CC2(C(=O)NC)CC1CCO2.N12CCC1C2=O N1(C(C2C(C)CCS2)=O)CCN(C(=O)C=Cc2ccccc2F)C2(CCC2)C1 C1(O)(CNC(CCCOCCOCC)=O)CCCN(C(c2cc[n+]([O-])cc2)=O)C1 c1(CC(c2n(C)nnn2)(C)Nc2cccc(Cl)c2)ncc(Cl)n1C C1(C(N(C)CC2CC2(F)F)=O)CCN(C(C23CC(C2)C3)=O)C(C)(C)C1 N1(C(c2c(C)ccnn2)=O)CC2CC1CCC2NC(C1CCC(C)O1)=O N1(C(C2(CC)CCCN2C(c2cccnc2)=O)=O)CC2CCC2(OC)C1 C1(C(=O)NCC(CCOC)NC(=O)Cn2ccc(C)cc2=O)COCC(C)(C)O1 CC(C)(C(=O)N1CCC(C)(C(=O)NCC(Cl)=CCl)C1)C(N)=O N1(C(c2c(SC)cc(F)cc2)=O)CCC2CCCC(C1)N2C(=O)C(=O)N(C)C c1(C(N)=O)cncc(C(=O)NCCN(c2nc(C(F)F)ns2)CC2CC2)c1 C=C(C)C(C)(C)C(=O)N1CC(OCCNC(=O)Cn2nc(C)ccc2=O)C1 C12(NC(CCC(=O)NCC)=O)CCCC1N(C(=O)CCc1cnco1)CC2 N1(C(C2(CCCC)CC2)=O)CCC2(C1)CN(C(c1cn(C(C)(C)C)nn1)=O)C2 C1(CNC(=O)CNC(c2cccs2)=O)CN(C(=O)CN2CC=CC2)CCC1CO CN1CCC(C(N2CCN(CCCNC(=O)Cc3cccc(O)c3)CC2)=O)C1=O C1(CNC(CCCOCCC)=O)CC2(CCC2)CN1C(c1csc(C)c1N)=O c1(CC)cccc(C(=O)NC(CCOC)C(=O)N(CC(C)(C)CN(C)C)C)n1 C1(C(=O)NCCC(=O)NC(C2CCCCO2)(C)C)CC2CC1CC2O CCC(CC)CCC(=O)N1CC2(CCCC2NC(=O)C=C2CCC(C)C2)C1 C1(COC)CC(CNC(=O)CC2OCCO2)N(C(c2nocc2C(C)C)=O)C1 c1(C(=O)NCCOC2CCN(C(c3cc(Cl)ccc3O)=O)CC2)n[nH]c2c1CCC2 N1(C(c2c(C)ocn2)=O)CCC(O)(CNC(=O)CNc2ccccn2)C1 O=C(N=c1[nH]c(Cl)ncc1O)C1CN(C(c2cc(F)c[nH]2)=O)CCC1(F)F N1(C(c2cccs2)=O)CCN(C(C23CCC(CO2)C3)=O)CC1c1ccccc1Cl C1(NC(C=C)=O)C2CCC1N(C(=O)CCC=C(C)C)C2 c1(C(=O)NC(CCCNC(CCc2cnc(C)s2)=O)C)ccc(C(C)C)nc1 C(=O)(C1=CCCCCC1)NCC1(CNC(C2CC3C(C)(C)C3C2)=O)CC12CCC2 N1(C(CNC(=O)OC)=O)CCN(C(=O)CC2CCC(F)(F)CC2)CCC1C C(=O)(C(CNC(c1ccsc1C#N)=O)(CC)CC)N1CCC(C)(CN(C)C)C1 c1(C(N2CCC(C)C2CNC(C2CC23CCC3)=O)=O)ccc2ccnc(O)c2n1 c1(C(=O)NC2CC(C)(NC(C=Cc3c(C)cccc3)=O)C2)nsc2ccccc12 N1(S(CCC(=O)OC)(=O)=O)CCC2C(CCN2C(c2cc([N+](=O)[O-])ccc2Br)=O)C1 C(=O)(CS(=O)(=O)C1CC1)N(C1CCCN(C(=O)Cc2ccns2)C1)C CC(C)(CC1CC1)C(=O)NCC1CCCC1C(=O)NC(C1CCC1)C1CC1 C12(C(=O)NC3CC4(CCCO4)C3)CCCC1N(C(c1cccc(F)c1O)=O)CC2 c1(C(=O)NCC2(O)CCN(C(C3(C#C)CCC3)=O)C2)ccc(C)nc1C C1(C(=O)NCCCCCOC)CCN(C(c2cccc(F)c2O)=O)C12CCC2 Nc1cccc(C=CC(=O)NC2(CNC(=O)CC3CCC(=O)NC3)CCCC2)c1 N1(C(c2c(O)ccc(OC)c2)=O)CCC2(CC2)CC1C(=O)Nc1cnc(Cl)nc1 C1(N(C)C(c2cc(C(F)F)n(C)n2)=O)CCC(CC(F)(F)F)CC1 N1(C(CS(CC)=O)=O)CCN(C(=O)C2=CCCCO2)CC1CC(F)(F)F N1(C(C(C2C(C)C2)NC(=O)CCC2CCOCC2)=O)CC2(COC(=O)C2)C1 C(=O)(CCS(C)(=O)=O)NC(C)CCN(C(=O)CCc1nnc(C(F)F)o1)C c1(C(=O)Nc2ccc(SCC#N)cc2)cccc2nc(C3CCCO3)[nH]c12 N1(C(c2ccc(C)c(N)n2)=O)CC2CCCC(CNC(=O)CC3CC34CC4)C2C1 Cc1cn2nnc(C(=O)NC(C)CCN(C)C(C3(C)CC3C)=O)c2c(O)n1 Cc1nc(C(N2CCCCC2CCNC(C23CC(C2)S(=O)(=O)C3)=O)=O)cc(O)n1 N1(C(CN(C2CC2)CC)=O)CCOC2(CCCN(C(c3cnc(Cl)cn3)=O)C2)C1 N1(C(c2ccoc2C)C(=O)NCC(C)C)CCCC(P(C)(C)=O)C1 CCCC(C(O)C(=O)N1CCCC(CCC)CC1)NC(C1C2CCCC(=O)C12)=O c1(COCCCNC(C(c2cn(C)nc2)O)=O)nnn(C)c1C(=O)NCC1CC1 C1(CNC(CC(CC)NC(=O)CC2(O)CCCC2)=O)CCCC(C#N)C1 Cc1ccn(CC(C)C(=O)N(C)CCN(C)C(C2CCCC2c2nc[nH]n2)=O)n1 CC1CCn2ncc(C(N3CCC(NC(=O)Cc4ccc(C#N)nc4)C3)=O)c2C1 Cc1cc(C(=O)NCC(C)NC(C2CCN(c3nncs3)CC2)=O)cc(N)c1O C(=O)(C(F)(F)C(O)C(C)C)N1CCCNCC1.Cc1ccc(-c2c[nH]nn2)s1 C1(C(=O)NC2C(NC(C3C=C(C)CS3)=O)CC2)C2C3CCC(C3)C12 c1(C(=O)NC(CN(C(=O)COC2CCOC2)CC)C)cc(C2CC2)cc(F)c1 c1(C(=O)NC2CN(C(c3cc(CC)n(CCO)n3)=O)C2)cc(Cl)c(O)c(Cl)c1 C1(COC)CN(C(c2cscc2C#N)=O)CCN1C(=O)C=Cc1nc(C)cs1 C(=O)(C(O)Cn1cncn1)N(C(CN(C(C(C)OC1CCCC1)=O)C)C)C N1(C(=O)CCC2CC2)CCN(C(c2ccn(CCF)n2)=O)C2CCCCC2C1 CC1(C)CN(C(C2C3COCC23)=O)CC(CNC(c2c[nH]nc2C2CC2)=O)O1 C1(OC)CN(C(c2csc(F)c2)=O)CC1C(N1CC(C(C)C)C1C(C)C)=O N1(C(c2cn(CCCC)nn2)=O)CCN(C(C2CC2CC)=O)C(COC)C1 c1(OCc2c3cccc(C(C)C)c3[nH]c2)cccc2c(O)ncnc12 c1(C(N2CCNC(c3ccco3)CC2)=O)cc(C2CC2)cc(F)c1F C12(C(N(C)Cc3cnc(C)s3)=O)CCCC1CCN2C(=O)CC1C=CCCC1 C1(C2CCC2)(CNc2ccc(-c3cc(NCc4ccc(Br)o4)on3)cc2)CCC1 c1(C(=O)NC(C(C)NC(c2c(C)cc(OC)nc2)=O)(C)C)cccc2c1CCN2 CC(CC(N)=O)C(=O)N1CCOC(CN(C(=O)C=CCCCC(C)C)C)C1 C1(C)(NC(C2(CCCC)CC2)=O)CN(C(C2C3COCC23)=O)C1 Cc1ccccc1C=CC(=O)NCC(C)(C)OCC(=O)NC1CC12CC(O)C2 C1(C)(OC)CCCN(C(=O)C(C(C)C)NC(=O)C(C2CC2)SC)C1 C12(C(=O)NCc3nc(CCN)on3)COCC1CN(c1ncc(F)cn1)C2 C1(S(=O)(=O)NC(C)(C)C)(C(N2CCN(C(c3c(CC)c[nH]c3)=O)CC2)=O)CCC1 c1(C(=O)Nc2c(C(=O)NCC(C)O)cc(F)nc2)cccc(S(C)(=O)=O)c1 C(=O)(CCCCCN(C)C(c1cc(C)n(CCO)n1)=O)NC(C(COC)C)C C1(NC(c2c(C)nc[nH]2)=O)C2CC3CN(C(c4ccc(C(C)O)cc4)=O)C1C3C2 C(C(C)(C)CN1CCCC1)N(C)Cc1cc(-c2cccs2)on1 c1(C(N2CCCC2c2cn(CCCCCCF)nn2)=O)cc(C(F)(F)F)ccc1Br c1(C(=O)NCC2N(C(C3C(C#N)C3)=O)CCC2)cc(S(N)(=O)=O)c(Cl)o1 Cc1cc(N2CCC(OC(C)(C)C)CC2)nc(C)n1.C1(C)C(=O)NCN1C C12(NC(c3cnc[nH]3)=O)CCCC1CN(C(c1ccc(-c3ccco3)o1)=O)C2 N1(C(C#CC(C)C)=O)CCC(C2CC2)(CNC(C2CCC(F)CC2)=O)C1 C1(C)(NC(CCCOCCOC)=O)CCCN(C(C2CC3CC2C2CC32)=O)C1 c1(OC)ccc(C(=O)NCC2CC2NC(c2sccc2C)=O)c(Cl)c1 CC(C)(CCCNC(c1cc(N)cc(F)c1)=O)C(=O)N1CCC(CF)C1 C1(C(N2CC(C(F)(F)F)C2)=O)(OC)CCN(C(=O)CC(C)C)C1 c1(CNC(=O)C(=O)NC2CC2)ccc(C2CCCOC2)cc1.C1CC(=O)N1 N1(C(c2c(CC)nco2)=O)CCC2CN(C(=O)C(C)Oc3ccc(Cl)cc3)CC12 C1(NC(C2N(CC)CCCC2)=O)CCCC12CCN(C(c1ccoc1)=O)CC2 C(=O)(C(COC)C(F)(F)F)N(CCCNC(C(CCC)OC(C)=O)=O)CCO Cc1ncnc(O)c1CCC(=O)NC(C)CN(C)C(C1CCC2(CC2)C1)=O c1(C(=O)NCC(C(C)C)NC(c2ccccc2-n2cnnn2)=O)ccc(O)nn1 C=CC(C)CC(=O)N1CC2CC2(CNC(=O)CCc2nnc(C3CC3)o2)C1 C12(C(N3CCC(C(C)C)C3)=O)COCC1CN(C(=O)C(C1(O)CCCC1)F)C2 c1(C2C(C(N3CC(C)(CC(N4CCOC(C#N)C4)=O)C3)=O)C2)cc(Br)ccc1Cl Cc1nccc(C(N2CC(CC(=O)NC(c3snnc3C)C)CC2C)=O)n1 c1(C(N2CCC(NC(COCCC)=O)C2)=O)cnn(C(C)(C)C)c1Cl n1(CCC=C)cc(C(N2CC(CNC(c3coc(N(C)C)n3)=O)(OC)C2)=O)nn1 CC(N=[N+]=[N-])C(=O)N1CCCCC1CCC(=O)NCC(C1CC1)C1CC1 C1(NC(CC2(C)CC2(F)F)=O)CCN(C(C2(CF)COC2)=O)CC1 N1(C(C2(COC)CC=CC2)=O)CCN(C(c2cc(C)c(N)cn2)=O)C(CF)C1 C1(F)(CNC(c2c(CC)ncnc2)=O)CCN(C(c2csc(Cl)n2)=O)CC1 c1(C(=O)NCC2(CO)CC2C(F)(F)F)cnn(-c2ccccc2)c1Br c1(C(=O)NC2CC(NC(=O)CC3CCCCCO3)C2)ccc(F)c(OC(F)(F)F)c1 CC(C)(O)CC(=O)N1C(C(=O)NCc2cncc(Cl)c2)CCC1C1CC1 CON(CCC(=O)NC1CCOC1C)C(=O)CC1C=NN(C)C1=O N1(C(C(C)=C2CCCC2)=O)CCCC(F)(C(N2CCC(C)(CO)C2)=O)C1 c1(C(N2CC(NCc3c(C)cncc3)CC2(C)C)=O)ccc([N+](=O)[O-])cc1 c1(OC)ncc(Cl)cc1C(=O)NCCCNC(=O)CN1CCC(F)(F)C1 n1(CC(N2C3CCC(NC(C(C(CC)O)C)=O)C(C3)C2)=O)ccc2ccccc12 C1(NC(c2c(CNC(C3C(C(C)C)OCC3)=O)c[nH]n2)=O)CC2C(C1)C2(F)F c1(CCC)ccc(CC(N2CC=CC(NC(=O)C(C)(C)OCC(C)=O)C2)=O)cc1 C1(C(N2CCC(N(CC(C)C)C(c3c(C)nco3)=O)CC2)=O)CCC(C)(C)CO1 Cc1cc(C(N2CC(CNC(=O)C=CCN3CCCCC3)C(C)C2)=O)c(C)o1 N1(C(c2nccc(C)c2N)=O)CC(NC(=O)C(Cl)=CCl)CC12CCCC2 CC(C)(C(=O)NCC1CN(C(c2cc(CN3CCCC3)on2)=O)C1)C1CCCO1 N1(C(CC2(COC)CCCC2)=O)CCN(C(c2ccccc2SC)=O)C(C)C1C Cc1cccc(CNC(C2(CNC(=O)CCc3nccs3)CC23CCC3)=O)c1O N1(C(C2CC(F)(F)C2)=O)CCN(CC2CN(C(C3(C(F)(F)F)CC3)=O)C2)CC1 c1(C(C(=O)NCCC(C)(C)NC(CC(C)OC)=O)C)cnn(C)c1C(F)(F)F c1(OCC)c(C(N2CCC(n3cc(C(C)(C)CC4CC4)nn3)C2)=O)c(C)nn1C C1(CCNC(CC=C=C)=O)CC(F)(F)CN1C(C1CC(OCC2CC2)C1)=O C1(C(N2CCCC(C(C)NC(c3cnc(CC)nc3)=O)C2)=O)CCC(O)C(=O)N1 C12(C(=O)NCC3CN(C(N)=O)C3)CC(CN1C(C1CC=CCC1)=O)C2 C(C1(C)CCCc2ccccc21)N(C(c1ccnc(F)c1)C(=O)NC)CC=C C12(CC(=O)NCCOCCC=C)CCC1CN(C(C1(Cl)CCCCC1)=O)C2 c1(CNC(Cc2cnc(C)s2)=O)cncc(C(=O)NCC2CCN(C)C2)c1 C(CCN=[N+]=[N-])N(C(=O)C(F)C1CC(NC(C2CCC2C#N)=O)C1)C c1(C(=O)NCC2(C)CCN(C(c3n(CCC)ncc3)=O)C2)n[nH]c2ccccc12 c1(C(c2ccccc2)NC(c2cccc(Br)c2F)=O)ccc(C2=CCCC2)cc1 c1(C(=O)NC2C(F)CCN(C(C(=O)NCC(F)F)=O)C2)nc2ccc(Cl)nn2n1 c1(C(=O)NC2C=CCN(C(C3CC(C#C)(O)C3)=O)C2)cccc(S(N)(=O)=O)c1 N1(C(C2(CC#C)CCN(C(C3C(C)(C)C3(C)C)=O)C2)=O)CCCCCCC1C c1(C(=O)NC(C)C=CC(=O)N(C)Cc2ccn(C)n2)cc[nH]c(=N)n1 C(=O)(CC(CC)C1CCC1)NCC(CC=C)NC(=O)C=NOC N1(C(C)C)CC(C(=O)NCC(C)CNC(=O)C2=CSCCO2)CCC1=O C12CCOCC1C(=O)N2.c1(-n2ncc(C(=O)NC3CC(CF)C3)c2)ccccc1Cl N1(C(CCC(C)SC)=O)CCCN(C(C2(N(C)C)CCC2)=O)CC1 CCC(O)C(C)(C)C(=O)NC1CN(C(C2CCC(=O)C2)=O)CC1F C(CN=c1cc(C#N)nc(C)[nH]1)(c1ccccc1)NC(c1cc(C)cc(F)c1)=O c1(C(N2C(C)CC(NC(c3c(C)ocn3)=O)C2)=O)ccn2nccc2n1 C=CCC(C(=O)NC1COCC1C(=O)NC1COCC1C(=O)OCC)OC N1(C(c2cc(C(C)(C)C)on2)=O)C2CCC1C(CNC(C1(CF)CCC1)=O)C2 Cc1ccccc1C(=O)Nc1cn(Cc2nccn2C)nn1 CC1CC(NC(=O)CCc2cncnc2)CCN1C(C1CC2CCC1C2)=O Cc1cc(F)sc1C(=O)N(C)CCN(C)C(C1(O)CCCC1)=O c1(C(N2CCC(OCCNC(C(C#C)(C)C)=O)C2)=O)nn(C)c(C)c1Br N1(C(CC(C)c2ccco2)=O)CCC(F)(CNC(c2ccnn2C(F)F)=O)C1 C(=O)(C(C)(F)C(=O)NC1CCN(C(c2ocnc2C)=O)C1)OC C1(F)(C(N2CC(CN3C(=O)CC(CNC(=NC)NCC)C3)C2)=O)COCCOC1 C1(C(N(C2CCC2)CC#C)=O)CCC(C)(C)N(C(=O)C(C2CCCCC2)=O)C1 C(C1CCCN1C(c1cncs1)=O)=CC(N1CCC(N2CC(O)C2)C1)=O CCCCC(C(=O)N(CCC(N1CCC(CC)(OC)CC1)=O)N(C)C)N(C)C C(CC(C)(C)SC)=CC(=O)N(N(C(=O)CCCOC)C(C1CCCC1)C)C C1(OC)C(NC(=O)C(F)CC2CN(C(C3(N(C)C)CC3)=O)C2)CC1O N1(C(C=C(CCC)C)=O)CC(CO)C2(C1)CN(C(=O)CC1(OC)CCCCC1)C2 c1(C(=O)NCCN(CCC)C(c2cc(C)[nH]c2C)=O)c(C(F)(F)F)noc1C O(NC(=O)CC(CCNC(=O)C(CC)n1cncn1)C1CCC1)CC=CC Cc1cc(CC(=O)NCC2COCC2C(F)(F)F)cc(C(F)(F)F)c1 N1(C(C(C)N(CC)CC)=O)CCCC(CCNC(C2CC(O)C2)=O)C1 N1(C(c2cnc(C(C)(C)C)s2)=O)CCC2C(CCCN2C(C2(C)CC2(F)F)=O)C1 C1(NC(=O)CC2CC2(Cl)Cl)CN(C(=O)COc2cccc(F)c2)CC12CCCC2 C1(NC(=O)CCc2cscn2)CCC12CN(C(=O)C(c1ccccc1F)O)C2 c1(OCC(=O)NC2CCC(CNC(CCC(=C)C)=O)CC2)cc(F)ccc1F c1(C2C(C(=O)NC3C(n4cc(CCC(=O)O)nn4)CCC3)C=CC2)ccccc1 C1(NC(CSCC#C)=O)CCCCC1CNC(c1cn(C(C)C)cn1)=O N1(C(c2ccc(N(S(=O)(=O)CCCl)CCO)cc2O)=O)CCC2(C1)CC2(F)F C(CCCCC(=O)NCC(C)(C)CN(C(=O)Cc1cc(C)ns1)CC)=CC c1(N2CC(C)NC(=O)C2)nc(N2CCC(CS(N)(=O)=O)C2)nc2c1CCCCC2 N1(C(c2c(N)cc(Cl)nc2)=O)CCCC2(NC(c3cccc(F)c3F)=O)CC2C1 Cc1cc(N2CCCCC(CNC(C3CCCNC(=O)C3)=O)C2)n2ncnc2n1 C1(N(C(C)C(=O)N2CCCC2)C)CCCCN1C(c1ncccc1F)=O C1(CC)CC(C(=O)NCCC2(NC(c3nnn(C(C)C)c3C)=O)CC2)CCO1 C12(C(=O)NC3CCN(C(CCc4nc(C(C)C)on4)=O)C3)CCC(C)(C1)OC2 c1(C(N2CCC(C)(C(=O)Nc3nc(CC)c(C)s3)C2)=O)cc(C)c(Br)cc1C C(=O)(C(C(C)C)N(C(c1cnc(OC)cn1)=O)C1CC1)N(CC(CCC)C)C C1(C(C)C)(C(=O)NCC2CC(NC(=O)C=Cc3ccsc3)C2)CNC(=O)C1 N1(C(C(C)NC(CC)=O)=O)CC(C(=O)NC2C3CCCC2COC3)CC12CCC2 c1(SC)ccccc1C=CC(N1CCCN(C(c2ccsc2)=O)CC1)=O O=C1OCCC2CN(C(C3CCN(CCc4c[nH]c5cc(Cl)ccc45)C3)=O)CC12 Cc1c(Cl)ccc(C(N2CCC(O)C(NC(c3cscc3F)=O)C2)=O)c1N c1(CN)nccc(Cl)c1F.C1(NC2(c3n(CC)nnn3)CCC2)CCC(CO)CC1 CCCC(C)CC(=O)NCc1ncoc1C(=O)NC1C(O)C2CCOC12 C1(C(=O)NC(CC=C)(C)C(F)F)N(C(C2(NC(N)=O)CC2)=O)CCCC1(C)C Cc1cc(CN(C)CC2CCCN2C(C2CCC(C(=O)C3CC3)CC2)=O)ccn1 c1(C(=O)NCCC2N(C(COCCOC)=O)CCOC2)cccc(O)c1Cl N1(C(c2c(CC)nc[nH]2)=O)CCC2(CC1)CC(C)N(C(=O)CC1CCOCC1)C2 N1(C(CC(=O)OC)=O)CCC(CN(C(=O)C(C)NC=O)C)CC1 c1(NC(=O)NC(C2CCCCCCC2)C(=O)O)cc(F)ccc1OC(F)(F)F c1(C(=O)OCC)nc(N2CCC(C)(NC(=O)Cn3cccn3)C2)sc1C C1(C(N2CCC2COC)=O)CN(C(c2occc2C)=O)CC12CCC2 C1(CNC(=O)C(C)(C)N(C)C)CC(C)(C)OC(C)(C)C1.CC1CC2CCN1C2=O C(=O)(C(C)CC(N)=O)N1C(CC=C)(C(=O)N(C)Cc2ccn(C)n2)CCC1 c1(CSC(C)C(=O)OC2CN(C(=O)C3CC3)C2)ccncc1N1CCOCC1 Cc1ccc(C2SCCN2C(C2CCCN(C(=O)C(C)S(N)(=O)=O)C2)=O)cc1C N1(C(C2(CC)CC2)=O)CCOC(C(N2CCCC(C(C)(C)C)C2)=O)CC1 C(C(C(C)C(C)C)NC(C1C2CC3C(C2)C13)=O)NC(C1C(C)=C1)=O c1(C(=O)NC23C(CN(C(CCCCCSC)=O)C2)C3)nc2cnccc2nc1O c1(CN2CCC(C(=O)NC(c3ccno3)C)C(O)C2)cc(Cl)c(Cl)cc1F C(CN=C(NC1CCOC1)NC1CC1C(F)F)n1c(C)ncc1 C1(CC)C(C(=O)NCC2(C(=O)NC3CCCC3OC)CCCCC2)CCN1C C1(NC(C(C)=C2CCCC2)=O)CC2(CCCCN2C(C2CCS(=O)(=O)C2)=O)C1 c1(NC(C2C(C)N(C(=O)C(=O)C3CCCC3)CC2)=O)ccc2ccoc2c1 n1(CC(=O)N(C(C)CCc2cccs2)CCO)cc(C(C)(C)C)nn1 CC1CN(C(=O)CCCF)CCCN1C(=O)Cc1cn[nH]c1 c1(CCC)sc(C(=O)NCCCN(C(C)C)CC2CCOC2)cc1Br C1(CNC(=O)NC(CC=C)CC)C2CCCC(=O)C12 c1(C(=O)NCC(N(C)C(C2(CO)CCCO2)=O)C2CC2)cnc(S)nc1 C1(C(=O)NCC(C(C)C)(C)O)CC12CCN(C(=O)C(C)(C)n1cncn1)CC2 CCCCC(O)CC(=O)N1CCCC(NC(c2ccc(SC)o2)=O)C1 C1(N(C)C(C2(O)CCOC2)=O)CCCN(C(C2(c3ccnn3C)CC2)=O)CC1 C(=O)(CCC(=O)C(C)(C)C)NC(C(=O)NCCC(CC=C)(C)C)CCC1CCC1 c1(C(=O)NCC23CCC2CN(C(C2(CF)COC2)=O)C3)nc2c(s1)COCC2 c1(C(=O)NC2CCC3CCN(C(CCSCC)=O)C32)c(C)c2cnccn2c1C Cc1cc(Br)ncc1C(N1CCOC(CO)C1)C(=O)NCC1CCCO1 c1(CC)cccc(C(N2CC3(CC3C(=O)NCCn3cc(CC)cn3)C2)=O)n1 N1(C(CN(CCOC)C)=O)CCCC(C2CCCCN2C(=O)C2CC2)C1 C1(CNC(Cn2c(C)nnn2)=O)CCN(C(c2cnn(CC(F)F)c2C)=O)CC1 C1(N(C(c2ccccn2)=O)CC)CCN(C(=O)C(C(C)C)c2cccnc2)CC1 N1(C(C2C3COCC23)=O)CCCC2(CCN(C(=O)C(C3CC3)C3CC3)C2)C1 c1(C(N2C(CNC(CC(C(C)C)O)=O)CCCC2)=O)ccc2c(c1)N(C)C(=O)C2 N1(CCCc2ccccc2)CC(N=c2cc(NCC3CC3)nc(C(F)(F)F)[nH]2)C1 CC(CN(C)C)CCC(=O)N1CCC(C(=O)N(C2CCC2)CCO)O1 CC1CC(NC(C2(NC(c3ccncc3F)=O)CC2(C)C)=O)CC(C)(C)C1 c1(CNC(=O)NC2C(c3ccc(C)cc3)C2)ccc2c(c1)nc(C)c(=O)n2C C1(CNC(C2C(C=C)C2)=O)(NC(=O)CN(C)C(=O)OC)CCOC1 CCC(C)(C)CCCC(=O)NC1(C)CCN(C(c2cccc(F)c2F)=O)CC1 c1(C(=O)NCCN(C(C)C)C(C2CCCCC2(C)C)=O)ccc(O)nc1Cl N1(C(C(C)(C)CO)=O)CCC2CCN(C(c3cc4sccc4n3C3CC3)=O)C2C1 N1(C(C=CC2N(C)CCC2)=O)CCCC(O)(CNC(c2ccc(Cl)cn2)=O)C1 c1(OC)cccc(C)c1.n12ccc(n1)C(=O)NCC2.N1(C)CCC(O)C1 C(=O)(C(CO)C(F)(F)F)NC(C(CC)C)C(=O)NCCC1NC(=O)NC1=O CN1CCOC(C(N2CCC(C(C)(C)NC(c3cnc4n3CCC4)=O)C2)=O)C1=O c1(C(=O)NCC(CCCC)NC(=O)CC(C)F)ccc2c(c1)CCCC2=O c1(NC(c2n(CCOC)nnn2)(C)CN2CCOC2=O)ccc2occc2c1 CN1CCN(C)C(CNC(C2(NC(=O)Cc3ccc(O)cc3)CCCC2)=O)C1 c12ccccc1NC2=O.CCC(C1CC1)(C1CC1)NC(C1CC1CF)=O CC1c2nncn2CCN1C(=O)C(O)CCNC(=O)C=CC(F)F C(=O)(CS(=O)(=O)CC(=O)NC(C)CCNC(c1c(C)cc(F)cc1C)=O)OC N1(C(CN(C(=O)CC2C=CCCC2)C)=O)CCCC1CN(C)C(c1ccco1)=O c1(C(=O)OCC(C(F)(F)F)n2cncn2)ccc(-c2nnco2)cc1 N1(C(CSC(C)(C)C)=O)CC(NC(C2(CC3CC3)CCCO2)=O)C(C)(C)C1 c1(CCCC(N2CCC3C(NC(C4CCC(C)O4)=O)C32)=O)ccc(O)c(F)c1 N1(CC(=O)N(CCCCCNC(Cc2nc(C)oc2)=O)C)CCCC(O)C1 c1(C(=O)NC)ncoc1CN.C(=O)(C(F)(Cl)C1CCC1)NCC1CC(N(C)C)C1 c1(C(=O)OCC)cc(-n2cc(C3CCC(C(=O)OC)CC3)nn2)nn1C C1(C(N2C(COC)(CNC(=O)CN3CSCC3=O)CCC2)=O)CCC(=O)CC1C c1(CC=C(C)OC)cn(CCC2CN(C(c3ccc(-c4cc[nH]n4)s3)=O)C2)nn1 C1(C(=O)NCCC)(NCc2cn(-c3ccccc3NC)nn2)CCCOC1 C(=O)(N=c1cc(C2CC2)n(C)[nH]1)C1(C(C)NC(c2cc(C)oc2)=O)CC1 C(C(C(=O)N1CC(C#N)(CCF)C1)C(C)C)NC(C=CCCC)=O c1(C(=O)NC(CN(C(=O)CN2CCC(C)C2)CC)C)nccc(OC)c1OC c1(C(=O)NNS(C)(=O)=O)sc2cccnc2c1Cl.C12CN(C1)CC(=O)NCC2 Cc1[nH]c(C(=O)NC23CC2CN(C(=O)CC2CCOC2=O)C3)c(C)c1[N+](=O)[O-] CC1CN(C(C2(S(C)(=O)=O)CC2)=O)CCC1NC(=O)COCC1(F)CC1 Cc1sccc1-c1cn(C(C)(C(=O)O)NC(c2ccc(C(=O)O)o2)=O)nn1 C1(NC(CCN(c2ccccc2)C)=O)CCN(Cc2ncc(C3CC3)o2)CC1O c1(CNC(C2CCC(NC(c3cn(C)nn3)=O)C2)=O)cnc2ccc(Cl)cn12 C=Cc1ccc(C(N2CCC(C(=O)NCC3OCCCC3(C)C)CC2)=O)cc1 c1(OC)ccnc(C(=O)NCC2CCC2NC(=O)CC(=O)N(C)C)c1 C1(CNC(c2c(C)nc[nH]2)=O)CN(C(C2(C3CCCCO3)CC2)=O)CCC1(F)F O=C1NCC2(CCN(C(C3CCN(C(=O)CC4CC(O)C(O)C4)O3)=O)C2)O1 c1(NC(=O)C(c2ccnc(F)c2)N2CCCC(O)C2)ccc2c(c1)OCCO2 C1(NC(c2c(CC)cno2)=O)CC=C(C(=O)NCC(CO)C(C)(C)C)C1 C1(C(F)(F)F)(C(=O)NCC(CNC(c2cnc(C(F)(F)F)s2)=O)O)CC=CCO1 N1(C(Cc2cn(CC)nc2)=O)CCC(C)C1C(=O)NC(c1cncnc1C)=O N1(C(C2C(C)(C)C2)=O)CC(NC(c2ccnc3c2CCO3)=O)C2(CCCC2)C1 C1(NC(C(CC)C(C)C)=O)CCCOC12CCN(C(=O)CC(O)C1CC1)CC2 C1(C(N(C)CCOCCCNC(C23CC(F)(C2)C3)=O)=O)CC12CCOCC2 Cc1cccc(C(O)C(N2CC=CC2CNC(c2nnn(C)c2C)=O)=O)c1 c1(CC)cc(C)c(C(=O)NCCCCN(C(=O)CSCc2cccs2)C)o1 C1(CNC(=O)CCn2cnnn2)CN(C(c2cccc(SC3CC3)c2)=O)CCO1 CN1CC(O)CCC1C(N1CCCN(C(=O)C(c2cccnc2)O)CC1)=O N1(C(CCC(C)=O)=O)CCC2(CC1)CC2NC(c1ccsc1)=O CC1(CNC(C2(C3CCCCO3)CC2)=O)CCN(C(c2n[nH]cc2Br)=O)C1 C1(C(=O)OCC)C2CC(O)C(C2)N1C(N1CC(C)(C)CC1CCO)=O Cc1ccc(Cl)c(NC(=O)CN2CC(CC(C)NC(=O)OC(C)(C)C)C2)n1 C(=O)(C1=C2CCCN=C2NN1)NC(C(C)C)CNC(=O)CCC=CBr c1(SC)cc(C(=O)NC(C2CCOC2)CNC(=O)C=Cc2ncc[nH]2)co1 N1(C(c2cc(OC)n[nH]2)=O)CCOCC(NC(=O)C(C)n2cnnn2)C1 CC1CC(NC(C2(c3cccnc3)CC2)=O)CCN1C(=O)Cc1ccccc1F c1(C(=O)NC(CCOC)CNC(=O)CC2CC(SC)C2)cnn(C(C)C)c1C C(CN=c1[nH]c(=NCCCC2CCCC2O)c2sccc2[nH]1)c1c(C)nc(C)s1 c1(C(N2C(CC)(CC)CC(NC(C3CCCSC3)=O)C2)=O)ccc(C#N)c(C)n1 C1(O)(CNC(c2onc(C)c2C)=O)CCCN(C(C2CN(C(N)=O)C2)=O)C1 N1(C(c2cc(CO)on2)=O)CCN(C(C2(C(=O)NC3CC3)CCC2)=O)CC1 c1(C(=O)NCCOCCNC(C2N(C)C(=O)CC2)=O)cc2c(cnn2C)nc1O C1(=O)CCCCN1C.n1(CC(=O)NC(=O)C=CC(C)(C)C)nccc1C CCCC(O)C(=O)NCCCC(C)NC(=O)C(C1CCC1)C1CCC1 S(=O)(=O)(c1ccc(I)cc1)NC1CCC(C(=O)Nc2cncc(O)c2)CC1 c1(C(=O)NCCC2CCN(C(c3c(CC)ocn3)=O)C2)ccnc(F)c1Cl c1(CNC(c2cc(I)c[nH]2)=O)ccc2c(n1)NCCC2 N1(C(c2c(C)cc(C)s2)C(=O)NCCOCC2CC2)CCC(C)(C)C1C CC1(C)COC(CCC(N2CCC(C(O)CNC(C3CNC(=O)C3)=O)CC2)=O)C1 C1(C(=O)NCC(N(OCC)C)=O)CCC(C)(C)N(C(C2CC3CCCC23)=O)C1 CC(C)CCC(C(=O)NC1CCC(C#N)CC1)NC(=O)CCc1nccn1C C(C)(C)(CCCCNC(C1CCOC(=O)CC1)=O)NC(COC(C)C)=O N1(C(C(C)N(C(c2cccc(O)c2)=O)CC)=O)CCCC2(CCCO2)C1 C1(N(C)C(C2CCSCC2)=O)CN(C(c2cccnc2C(F)F)=O)CC1F CCCC(CC)CC(=O)NCC(C)(C)CNC(C1CC1c1nccn1C)=O N1(C(C)=O)CCCC1C(=O)NC(C)(C)CCNC(=O)CCc1nc[nH]n1 c1(C(N2CCC(NC(C3(OC)CCCCC3)=O)C(C)C2)=O)cc(F)c(N)c(F)c1 N1(C(C(C)C)=O)CCSC(C(=O)Nc2ccc(-c3cccs3)cc2)C1 C1(CC)CN(C(c2cnc(O)n2C)=O)CCN1C(c1cc(C(C)(C)C)nn1C)=O C=CCCCCCC(=O)NC(C1CCCN1C(c1cc(C)ncn1)=O)(C)C C(C(=O)N1CC2C(C(=O)NCc3c(C)cccc3F)C2C1)(C(C)(C)C)OC c1(CC)nc(-c2ccnc(-n3cncn3)c2)n(CC(C)CO)n1 CN=c1ccc(C(N2CCC(C(=O)N(C)CC3CC3C)C2(C)C)=O)c[nH]1 N1(C(C2C(COC)C2)=O)CC(F)(CNC(=O)C(CN(C)C)N(C)C)C1.C(C)(C)S c1(C(CNC(c2ccn(CC)n2)=O)N(C)C)ccc(NC(C2CCS2(=O)=O)=O)cc1 O=C1CCC(NC(=O)CCC2CCCN2C(C2CCCC2)=O)C(=O)N1 c1(C(=O)NC(CN(C(=O)C(O)C(F)F)CC)C)ccc(N(C)C)cc1F C1(C(=O)N(C(CC=CC=C)=O)C2CC(C)C2)CCCN1CCCC c1(C(=O)NCCN(C(c2ccc(C#C)cn2)=O)CCC)ccc(S(N)(=O)=O)s1 C(C)(CNC(=O)CC1CC(OCCOC)C1)(CC)NC(CCC)=O N1(C(c2cnc(C)nc2)=O)CC2(CCN(C(=O)CCC3CCCC(O)C3)C2)C1 N1(C(c2cccc(SC)c2N)=O)CC(C2CCN(C(C)=O)C2)C1 C1(C(=O)NC(CC)C2CCC2)CC2(CCC2)CN1C(C1CCOC1(C)C)=O c1(CC)nc(C)c(C(=O)NCCCC2(NC(=O)CC3(O)CCCC3)CC2)s1 Cc1cc(=NCC2CC3(CC(N(C)C)C3)C2)[nH]cc1[N+](=O)[O-] C12(C(=O)NCC(C3CC3)NC(C(C3(O)CCCCC3)CC)=O)CCC(C)(C1)OC2 C1(C(=O)NC(COC(C)C)(C)C)CCCN(C(c2cccc(Cl)c2)=O)C1 C(=O)(CCCC(C)(F)F)NCC1(F)CCC(NC(C(=O)N(C)C)=O)C1 n1(CC(=O)N(C2CCN(C(=O)CN(S(C)(=O)=O)C)C2)C)nc(O)ccc1=O c1(CC)noc(CCNC(=O)C(C2CC2)NC(=O)C(C)c2ccco2)n1 C#CC(COC)NC(=O)C=CC(F)F.C1(=O)C=CC(C)N1 c1(OC)cc2c(C(N3CCOC(CN(C(=O)C(C)OC)C)C3)=O)c[nH]c2cc1Cl c1(OC)cnncc1C(=O)NC1(CC(=O)NC(C2CCCCC2)CO)CC1 C=CC(C)CC(=O)NCC1CCCN(C(c2ccc(C)n2C)=O)C1 CCN=C1NCC2CC(N1)C2(C)C.C1(C(=O)NC)CN(C(=O)OC(C)(C)C)C1 CC(CC(=O)N1Cc2occ(C(N3CC(F)CC(F)C3)=O)c2C1)C(C)(C)C N1(C(CCC2C(C)C2)=O)CCC2CN(S(=O)(=O)CC3CCC(C#N)CC3)CC2C1 C1(C(=O)NC23CC(NC(C4CCc5ncsc5C4)=O)(C2)C3)CCn2nncc2C1 C(CCC(=O)NCC1CC2(CCCO2)C1)(C(C)C)NC(C1(C#C)CC(=O)C1)=O NS(=O)(=O)c1ccc(-c2cc(CN3CC(O)C(F)C3)ccc2F)nc1 C12(C(N3C(NC(=O)NC4C(C)(C)C4CN=[N+]=[N-])CC3)=O)CCN(CC1)C2 C12(C(N3CC(OCCNC(c4n(C(C)C)ncc4)=O)C3)=O)CC1COC2(C)C C1(NC(=O)NCCCCCCCCCC)C2CCCNC2C1(C)C.C(C)(C)(C)O c1(OC2CC2)cccc(CC(=O)NCCC2(CC)CC2)c1.C1(=O)CCCN1 Cc1nccnc1C(N1CC(n2cc(CNC(C3CC4C=CC3C4)=O)nn2)C1)=O c1(C(N(C2(C(=O)OC)COC2(C)C)C)=O)ccc(Cl)c2ncccc12 CC(C(CC(=O)NC1CCN(C2CCCCC2)CC1)N(C)C)C(=O)O c1(CCC)cc(C(=O)NC2(CC)CN(C(=O)CC#N)C2)n(C)n1 Cc1cc(Cl)nc(Cl)c1CN1CC2CC2(C(=O)Nc2ccc(C#N)cn2)C1 C(=O)(C1=C(Cl)CCOC1)NCC(CNC(C1(CC#C)CCCOC1)=O)C C#Cc1ccnc(C(=O)NCC(C2CCCC2)NC(C2(C)CCNC(=O)C2)=O)c1 CCC(CC(F)(F)F)C(=O)NCC1=CCN(C(=O)CCSC(F)(F)F)CC1 c1(C(N2CC(CC)N(C(=O)CC(F)(F)F)CC2)=O)cc2cccnc2[nH]1 C(=O)(C1=NOC2(CCC2)C1)NCC1(F)CN(C(C2C(OC)CCCC2)=O)C1 C1(C(N(C(C)CN2CCCC2)CC)=O)(NC(c2cc(CO)on2)=O)CCN(C)C1 N1(C(CC(CC)OC)=O)CC(NC(=O)CCn2nc(C)cc2C)C2(CCC2)C1 CCC(C)C(C(=O)N1CCC(NC(=O)CN2CCOCC2=O)CC1)NS(C)(=O)=O N1(C(COCCC=C)=O)CCC(OCCNC(=O)CC(F)(F)Cl)CC1 CN1CC=C(CC(=O)N2CCN(C(c3c[nH]c(C#N)c3)=O)CC(CO)C2)CC1 c1(C(=O)NCCC(C)NC(C2(C)COC(=O)OC2)=O)cc2n(n1)CC(F)C2 c1(N(CCC(N2CCC(c3ccccc3Cl)CC2)=O)C)ccccc1[N+](=O)[O-] c1(CC)nc(NC(C2CC2C(C)NC(=O)Cc2cccnc2Br)=O)cc(C)n1 Cc1cccc(C(=O)NC2COCCC2C(N2CCC2(C)C(C)C)=O)n1 C(=O)(CC1=NNC(=O)C1)N1CCC(CC=C)(NC(=O)CC(=O)NC)C1 c1(NC(C2N(C(c3c(CC)nn(C)c3)=O)C(C)CC2)=O)cn(C)c(=O)nc1O N1(C(CN(CCC)C)=O)C2CCC1(CNC(c1c(C3CCC3)cnn1C)=O)CC2 c1(OC)ccc(C(N2CC=CC2(C)CNC(c2cc(C(N)=O)c[nH]2)=O)=O)cc1 c1(C(N2CCCN(C(C3CC(C)=C(C)CC3)=O)CC2)=O)cn(C)c2ccccc12 Cc1coc(C(N2CC(NC(=O)CCCSc3ccccc3)C(O)C2)=O)c1C c1(C(=O)NCC(C)NC(=O)CC2CCNC2=O)ccc2c(c1)CC2 c1(NC(C)C)ccc(C(C)C)cc1S(=O)(=O)NC(C)CNC1CC1 C1(n2cccn2)(SCC(=O)NCC(F)F)CCN(CC(=O)Nc2cnsn2)CC1 c1(N(CC(=O)NC2CCN(c3ccsn3)CC2)C)ccnc(NC2CC2)n1 C1(F)(CNC(C2(CCC)CCC2)=O)CN(C(C2CC2C(=O)NCCO)=O)C1 C1(C(=O)NC(C(=O)OCC)C(C)C)CCCC12CN(C(C)Cc1ccccc1)C2 C1(C)(OC)CN(C(=O)COc2cccc(C(F)(F)F)c2)CCC1(C)OCC C1(O)(C(=O)Nc2cn(CC)nc2)CCN(C(=O)Cc2cccc(Br)c2)C1 C(=O)(C1Cc2ccccc21)N(CCCCCCNC(C=CC(C)(C)SC)=O)C C1(SC)CC2(CCC2NC(N2CCN(C)CC2)=O)C1.C(C)(C)O N1(C(C(CCC)NC(=O)CC2CCC(=O)C2)=O)CCC2(CCOC2=O)C1 C12(C(=O)NC(C3CCCCC3)(CC)C)CCCCC1C2Br C1(CN(C(C(C)OCC)=O)C)CN(C(c2cnc(C)nc2OC)=O)CC12CC2 C(=O)(C(C)(C)CC(F)(F)F)NCC1(CNC(C(CC)(C)N(C)C)=O)CC1 CCC(O)C(C)C(=O)N(CCCCN(C)C(c1c(C)ncnc1O)=O)C c1(OC)nc(NS(=O)(=O)CCCCC2CC2)cc(O)n1 c1(C(N(C(CN(C(c2[nH]cc(CC)c2)=O)C)C)C)=O)ccc(F)c(OC)c1F c1(C(=O)NCC2(NC(CN(C3CCCC3O)C)=O)CC2)ncccc1N C1(C(N2C(COC)C=CC2)=O)CCN(C(c2ccc(C)o2)=O)CCO1 C(=O)(CC(F)(F)Br)NC(CCNC(CCCn1c(C)ncc1)=O)(C)C C(CNC(C1CCCN1CC(F)(F)F)=O)(CC(C)C)NC(CCCOC)=O C1(C(N2CC(O)(CN(C)C(c3ccn(CC(F)F)n3)=O)C2)=O)CC12CCOC2 C1(NC(C(n2cc(C)nc2)(C)C)=O)CCN(C(=O)C(C)OCC(C)C)C1(C)C C1(CNC(c2c(CC)cco2)=O)CCCN(C(=O)C(C(C)C)SC)C1.N(C)C C1(CC(N2CC(C#C)(N(C)C)C2)=O)CC(C)CN(C(=O)CCc2ccncc2)C1 N1(C(c2cccc(OC)n2)=O)CC2CC1CC2CNC(c1cn2ccsc2n1)=O S(=O)(=O)(c1ccccc1)NCCC(C(=O)NCc1c(OC)ccc(C)c1)N(C)C c1(NC(=O)C(F)C2CCOC2)nc(N2CC(OCCCCOC)C2)c(C)c(Cl)n1 Cn1cnc(C(=O)NCCC2(O)CCCN(C(C3CC(C)(C)CO3)=O)C2)cc1=O N1(C(C2CCN(C(CN(C(C)C)C)=O)C2)=O)CC(O)C(O)C12CCC2 N1(S(CC)(=O)=O)CCN(c2ncnc(Cl)c2F)C(C)C1.C1(CCC2CC2)C(=O)N1 c1(CC(=O)NCC(CCOC)NC(=O)C(C)(C)S(C)(=O)=O)ccc2occc2c1 N1(C(C=C(CCC)C)=O)CCN(C(C2(C)CCCOC2)=O)C2CCCC12 C(=O)(C(CC)C(C)(F)F)NCC1C(NC(c2cc(OC)c(F)cc2)=O)CC1 N1(C(c2c(CNC(C=C(C)C(C)C)=O)noc2)=O)CC2COCC2(C)C1 N1(C(CC(=O)OCC)=O)CCC2(CC1)CCN(C(=O)C(C)(C)c1sccc1Cl)C2 CCC(CC(=O)N1CC(C2CCCO2)C(O)C1)N(C(=O)CC#N)C CCC1CC(=O)N2CCCC(C2)C(=O)N1.c1(SC)ccnc(OC)n1 c1(C(=O)Nc2c(C)cc(OC3CCNC3)cc2)cnc2ccnn2c1 c1(C(=O)NCC(CO)NC(c2cn(CCc3ccccc3)nn2)=O)csc(Cl)n1 C1(C(N2CCN(C(C)=O)CC2C)=O)CCC2(CCCC2)O1 N#Cc1cc(C(=O)NCC2COCC2NC(=O)CCCc2cccs2)c[nH]1 C(=O)(C(O)CC(C)(C)C)N1CC(NC(c2ccnc(C)n2)=O)C(C)C1 Cc1snnc1C(=O)NCC1CCCN1C(C1(c2cccs2)CC1)=O C1(NC(=O)Cn2cccc2)CCC2CN(C(C3CCCCC3O)=O)CCC2C1 N1(C(c2c(OCC)scc2)=O)CCCN(C(c2cccc(OC)c2Cl)=O)CC1C c1(C(C(=O)NC)N(CC(C)(C)C2CC2)C)ccc(C(F)(F)F)cn1 c1(N2CC(C(F)(F)F)OCC2)nc(=NCc2ncoc2C2CC2)[nH]c2c1COCC2 C1(C(=O)NC2(CNC(CC(C)SC)=O)CCOC2)C2(CC2)C12CC2 CCCC(C)CC(=O)NC1C2CC3C1C3C2C(=O)NCC1CN2CCC1CC2 CC(C)CC(CN(C)C)N=c1[nH]c(=NCc2cc(Br)c[nH]2)[nH]c2c1CC(C)CC2 c1(CC)ccc(C(N2CCCC2C=CC(=O)NCC2(COC)CC=CC2)=O)cc1 C1(C(=O)N)CCCCC1O.N1(C(COCC(C)(C)C)=O)CCCC1C(=O)NC O=C(C1=Cc2ccccc2C1)OCC(F)(C(=O)NC1CCCCC1)C(F)(F)F C(=O)(C1SCc2cccnc21)N1CC2(N(C(CNC(=O)OC)=O)CCCC2)C1 Cc1cnc(C(N)=O)c(NC(=O)CC2(C)CCN2C(=O)Cc2cc(C)[nH]n2)c1 C1(NC(=O)C(c2cccc(Br)c2)O)COCCN(Cc2ccc(Br)s2)C1 c1(N(C)CC2C3CN(C(=O)C(C)(C)NS(C)(=O)=O)CC23)ccn2ccnc2n1 C1(C(C)C)N(C(=O)Cc2cncs2)CC12CCN(C(=O)C(O)CN(C)C)CC2 c1(OC)ccccc1OCCC(N1CCC(O)(CCNC(=O)C2=CCOC2)C1)=O CCC(CC)CC(=O)N1CCCCC(C(=O)NCCc2cncs2)C1 c1(C(=O)NC2(C)CCN(C(=O)C(F)n3cccn3)C2)cc(=N)[nH]c(Cl)n1 C(=O)(CC(C1CC1)NC(C12CSCC1C2)=O)NC1(CSC)CC1 C(=O)(C(C)(CC)CC)N1CCC(N(C(=O)Cc2cccc(C(N)=O)c2)CC)C1 c1(NC(C)=O)c(C(N2CC(NC(=O)CSCC(N)=O)CC2C)=O)cccc1C CC(C)C(C)C(=O)N1CCCC1CCCNC(=O)C=Cc1ccccc1 C1(C(C(=O)C(CC2(CC(=O)OC)CC2)=O)(C)C)CCCN(C(=O)CO)C1.N(C)CC c1(CN(C(C(C(C)=O)(C)O)=O)C)nc2ccccc2s1 N1(C(c2c(C)cn(C)c2)=O)CCC(NC(C2(NC(N)=O)CC2)=O)CC(C)(C)C1 CC1CC2CC2CC1C(=O)NC1CC(CNC(c2csc(C(F)F)c2)=O)C1 C1(C2CCOCC2)(C(N(CCN(C(c2cccc(C)c2Cl)=O)C(C)C)C)=O)CC1 c1(CC(N2CC=CC(NC(C=CC(N)=O)=O)C2)=O)ccc(F)c(Br)c1 C1(NC(c2ccc(COC)[nH]2)=O)CCC(C)N(C(c2ccc(C#N)cn2)=O)C1 N1(C(=O)NCc2ccc(CCCCCC)s2)CC2CC(C1)c1cccc(=O)n1C2 Cc1cccc2nc(C(C)NC(C(C3CC3)NC(N)=O)=O)cn12 C(=O)(CCCC(O)c1ccccc1)NCC1N(C(c2cc(CC)ncn2)=O)CCC1 c1(NCC(=O)Nc2nnc(C(C)C)o2)ccc2sc3ccccc3c2c1 C1(CC(=O)N(CCNC(c2c(C)sc(Br)n2)=O)C(C)C)CC(O)C12CCC2 C(=O)(CC1=CCOCC1)N1C(C)(C(N2CCCCC2CF)=O)CC(O)C1 c1(CCNCC(C)CCc2ccccc2F)nnc2n1CCC2 C=CCC(CC(C)C)C(=O)NC1(C(=O)NCC(C)O)CCN(C)C1 C1(Nc2c(Br)ncc(OC)c2)CN(Cc2c(F)ccc(Cl)c2Br)CC(F)(F)C1 CCC(C)CCC(=O)N1CC(C2CC2C(=O)N(C2(C(O)C(C)C)CC2)CC)C1 C1(C2CC2)(NC(C#CCCC)=O)CCN(C(C2CC(O)C(F)C2)=O)C1 C(CC(=O)NCc1ncsn1)(C(C)(C)C)NC(c1c(C)n(C)cc1)=O C1(NC(c2ccc(C)c(F)c2)=O)CCC2(CC1)CN(Cc1cc(Br)cc(I)c1)C2 c1(C(=O)NC2C3C(NC(C(C)SC)=O)CC(CC3)C2)ccc2ncc(C)n2c1 N12CCC(CC1)CC(=O)NCC2=O.C1(NC(=O)NC)(CN(C)C)CCCC1 Cc1cc(C(=O)CN(C[Si](C)(C)C)C(C)C(=O)N(C)C)cc2cccnc12 C(C)(CC(=O)N(CC(O)CN(C(=O)Cc1ncoc1C)C)C)OC CC(CN=c1nc2ncn(C)c2c(NCC2(C)CCC(F)(F)C2)[nH]1)n1cccn1 N1(C(c2c(SC)cccc2)=O)CC(NC(c2ccccc2Cl)=O)CC2(CC2)C1 C(=O)(CCCC(F)F)N1CCC2C(NC(COc3c(OC)cccc3)=O)C21 C1(C(=O)NC2CC(NC(=O)CN3CC4CC4C3)C2)CCC2(CCC2)C1 C(CC(C)C(=O)NC(CC1CCCC1)C(=O)NCc1coc(C)c1)OC C1(CNC(C2CC(NC(C(CO)N(C)C)=O)C2)=O)CCCCC1C(F)(F)F C1(CCC#C)(CNC(c2scc(CNC(=O)CNS(N)(=O)=O)n2)=O)CCCCC1 C1(C(N(C)Cc2cnn(C)c2)=O)CC2C=CC1N(C(=O)C=Cc1cnccn1)C2 c1(OC)cccc2c1CCCN2C(=O)CC(=O)Nc1ncccn1 C(=O)(CCCC(=O)OCC)NC1(C)CC(=C)C1.C1=CC(=O)N2C1CCC2 N1(C(C2N(C(CC3=NNC(=O)C3)=O)C3(CC2)CC3)=O)CCCC12CCCCC2 c1(C(N2C(C3(O)CN(C(CC(COC)C)=O)C3)CCC2)=O)cc(SC)cnc1O C(c1ccn(C)c1)=CC(=O)NCC=CCC(=O)NC(C1(OC)CCC1)C c1(C(=O)NC2(C(=O)OC)C(C)(C)C2)coc(S(N)(=O)=O)c1.C(=O)O C1(CN(C(=O)C(F)(F)C2CC2)C)CN(C(C2CCC23CCC3)=O)CCO1 C1(NC(C(CC)CC)=O)CC(O)CN(C(=O)CCOCC(F)F)C1 C(=O)(C(C)(C)CC(=O)NC1(C(=O)NCC(CSC)OC)CCN(C)C1)OC CCC(C)(C(=O)NC1CCC(CO)CC1)C(N)=O c1(C(N2CCC(C(=O)NCC3C(C)CCCC3)CC2)=O)ccc2[nH]ccc2n1 N1(C(CC2(C)CCCO2)=O)CCCC(C2CCN(C(c3cn[nH]c3)=O)CC2)CC1 N1(C(C(C)NS(C)(=O)=O)=O)CCC2(CCC(CNC(C3CC4CC4C3)=O)O2)CC1 C1(C(=O)NCC2(COC)CN(C(=O)C=C(C)C(C)(C)C)C2)CNC(=O)CC1C C(=O)(C1COc2ccc(Cl)cc21)NCC1N(C(COCC=C)=O)CCC(C)C1 c1(NC2(c3ccc(CCC(=O)OC)cc3)CCC2)ncc([N+](=O)[O-])cc1C C(=O)(CC(C(F)F)NC(c1cnn(C)c1N)=O)NCC(=O)OC O=C(C1=C(Cl)CCC1)NCC(CC(N1CC2C=CC1CC2)=O)C1CCC1 C12(C(N3CCC(CN(C(=O)CNC=O)C)C3)=O)CCN(CC1)C2 C1(C)CC1C1CCN(C(C=CCN(CC)CC)=O)CC1.C12CCC1C(=O)N2.OCC C1(C(=O)NCC2(NC(CCCC)=O)CC2)CC(F)(F)C1(F)F Cc1nc2ccccn2c1CC(=O)N(CCCNC(=O)CC(C)(C)O)CCO c1(C(=O)NCCC(=C)CNC(c2nccc(C(F)F)n2)=O)cc2c(s1)CCC2 c1(C(=O)OC)nccc2c1CCN(CC(=Cc1cccc(F)c1F)C)C2 c1(C(=O)NCCN(C(=O)C2OC(=O)c3ccccc32)C)cc2c(s1)C(C)(C)CCC2 C1(C(=O)NCCC(C)CCNC(C23CCC(CC2O)C3)=O)CCCCCCC1 C=CCC(C)C(=O)NC(c1cccc(Cl)c1)CNC(=O)C(C)(C)CC1CC1 N1(C(C(C(C)C)Cc2ccccc2)=O)CC2CC1CN(C(=O)CCOC(C)C)C2 c1(C(N2CCCC(C(C)C)C2)C(=O)NCCCOC)nccnc1Cl c1(C(=O)OC)ccc2c(c1)CCN2C(=O)C(C(C)O)NC(c1ccccc1F)=O C1(CC)CN(C(=O)Cc2ccon2)CCC1N=c1[nH]c(Cl)nc(C)c1Cl N1(C(C2N(C)CCC2)=O)CCOC(C)(CNC(c2cnn(CC3CCC3)c2)=O)C1 CCCC1CC(=O)NCc2c(cco2)C(=O)N1.c1(C)ccc(=O)n(C)c1.C(=O)NC N1(C(c2cncc(C)c2)=O)CCN(C)CC1C(=O)NCc1nnn(C)c1C Cc1nn(CC(=O)NCC2CN(C(=O)C(N3CCOCC3=O)C)CC2C)c(=O)o1 N(C(=NCCCCC1OCCO1)NCc1ccnn1C)CCOC C(=O)(C(CO)C(F)(F)F)N1CCCC(CCNC(C(C)(C)OC)=O)C1 C1(NC(C(CC)(C)O)=O)CN(C(=O)CNC=O)CCC1CO C12(OCC)CCC(C(N3CCOC(C)(CNC(=O)C(C(=O)OC)OC)C3)=O)(CC1)C2 c1(C(N2CC=CC(NC(=O)C(F)n3cccn3)C2)=O)csc2c1CCCC2 C(=O)(C1=CCCC1(C)C)NCCCCCC1CCN(C(CCN(C)CC)=O)CC1 Cc1cc(C2CC2)ncc1C(N1CCN(C(C2CSCCS2)=O)C2CC12)=O c1(C(N(CCCNC(c2ccc(O)c(Cl)c2)=O)CCO)=O)cc2cnccc2[nH]1 c1(C2(C(N3CCC4C(C(=O)N)C43)=O)CC2)ccc(F)cc1F.Cc1cnnn1CC1CC1 Cc1cccc2nc(CCC(=O)N(C(C)CCNC(=O)C=NOC)C)[nH]c12 CC1CCCC(C(=O)NC2CCC(NC(=O)C(F)(F)c3cscn3)CC2)C1 C#CC(C)(C)C(=O)N1CCCC(N(CCO)C(C2(C3CCCCO3)CCC2)=O)C1 c1(OC)ccc(-c2csc(NC(c3cnc(C(F)F)s3)=O)n2)cc1 C1(C(=O)NC2CCCN(CC(C)(C)O)C2)CCc2ccc(F)cc2N1 c1(N2CC(C(N)=O)OCC2)nc2ccc(S(=O)(=O)NCC(O)C3CC3)cc2s1 Cc1c(C(=O)NCC(F)CNC(c2ccc(OCCF)cc2)=O)noc1C1CC1 c1(CN2C(C(N3CCN(C(C)C)CC3)=O)CC(OC)C2)ccc(F)cc1Br C1(CC)CCC(C(=O)NCCCF)CN1C(c1ccc(F)cc1I)C(=O)OC C1(CCNC(C(CC)SC(F)(F)F)=O)CSCCN1C(=O)CC1COC(C)(C)C1 N1(C(C2N(C(c3c(C)cc(Cl)cc3)=O)CC(F)C2)=O)C2CCC1CC(N(C)C)C2 C1(C(N2C(CCCC)COCC2)=O)CCCN(C(C2(COC)COC2)=O)CC1 C1(CNC(C2(CC=C)CCCCC2)=O)CCC2(CN(c3ccc(CC)nn3)C2)O1 c1(C(N2CC=CC(NC(CCOCCCOC)=O)C2)=O)cnc2scc(C)n12 C12(CC(=O)NCC3CCCCC3NC(=O)COCCF)CCCN1CCC2 C12(CC)CN(C(=O)Cc3nc[nH]n3)C(CNC(C3(C)CCCC3O)=O)(C1)C2 C1(C2CCCN2C(=O)CN)N(C(=O)CCCCCC)CCC1(C)C.CN c1(CN(CC(=O)NCC(C)C(=O)O)C2CC2)ccc2c(c1)OCCO2 Cc1cc(F)ccc1C1(C(=O)NCC2CCCC2NC(=O)Cn2ccnn2)CC1 CCC(CC(=O)NC(CN(C(=O)Cc1csc(S)n1)C)CC)C(C)C CC1(C)CC(CNC(c2nscc2N)=O)N(C(=O)CCCCc2cnn[nH]2)C1 CC(C)CC(C)CNC(C1COCCC1NC(=O)CCn1ccnc1)=O c1(C(N2C3(CNC(C(C)(C)F)=O)CCC2CC3)=O)ccc2ncnc(O)c2c1 C1(C(N2C3C(CNC(C(CSC)C)=O)C(CCC3)C2)=O)CCn2c(O)nnc2C1 CC(C)CC(O)C(=O)N1CCOC(CC(=O)NC2(CN(C)C)CC2)C1 C1(O)(CNC(C(C)CSC(F)(F)F)=O)CCN(C(=O)CC2CCNC2=O)CC1 C#CC1(C)CCN(C(C2COCCC2NC(C2CCCN2CCC)=O)=O)CC1 C1(C2CCC2)(C(=O)NCC2CC(C)(C)N(C(=O)COCC3CCC3)C2)CC1(F)F N1(C(c2cc(Br)ncc2Br)C(=O)NCC)CCC2CCC(C1)N2C c1(-c2c(C)cccc2F)ccc2nccc(C(=O)NCC3COCCO3)c2c1 CC1(C)CC(CNC(=O)COC2CCCC2)N(C(c2cc([N+](=O)[O-])n[nH]2)=O)C1 C=C1CN2C(=O)CCC2(C(=O)NCC2CN(C(c3nccc(OC)c3N)=O)C2)C1 C1(C(=O)NCc2cccc(C#C)c2)CC12CCN(C(C1(F)CC=CCC1)=O)CC2 C1(CNC(CCNC(C)=O)=O)CCC2(CCC2)CN1C(=O)CC1CCCO1 Cc1nc2cc(C(N3CCC(NC(C45CC(C4)C5)=O)C(F)C3)=O)cnc2s1 CC1CC(C2CN(C(C34COC(C3)C(NC(=O)C(C)(F)OC(F)(F)F)C4)=O)C2)=NO1 c1(C(=O)NC(CNC(c2cc(OCC)n[nH]2)=O)CC)cccc(Cl)c1 CC1(C)CC1CCC(=O)NCCC1CN(C(C2CC2(F)Cl)=O)C1 c1(C(N(CCC(C)NC(C2CC2OC(C)(C)C)=O)C)=O)ccc([N+](=O)[O-])c(O)c1 c1(C(=O)NC(C(C)C)CNC(c2coc(Br)c2)=O)cc[nH]c(=N)c1N C1(C)(CNC(NC(C#C)C(C)(C)Nc2ccccc2)=NCCF)CCCC(F)(F)C1 C1(NC(C2CC(C)(C)O2)=O)CCN(C(=O)C=CC2CC2)CC1F c1(NC(C2C(CC(=O)NCCN3CCOCC3=O)C(O)C2)=O)ccc(CO)nc1 C1(C(=O)NCC(C)(CO)NC(c2cc(F)c[nH]2)=O)CCCCC12CCC2 c1(NC(C=C)C2CC2)nccc(=NCc2c(C3CC3)cccc2C)[nH]1 C1(C(=O)NCC2(F)COC2)C2CCCC1CN(S(=O)(=O)Cn1cccc1)C2 Cn1cnc(C=CC(=O)NC2CCCCC2NC(c2ccnn2C2CC2)=O)c1 C1(CCCC)CN(C(=O)OC(C)(C)C)CCN1C(c1cc(SCC)cnc1O)=O c1(NC(c2ccc(OC)cc2)=O)cnc(C2=CCCC2)cn1 C12(CNC(C(CC)COC)=O)CCC(CC1)CN2C(=O)CC1CC(=O)NC1=O c1(NC(N2CCC(CC#C)(C(=O)OC(C)C)C2)=O)ccc2c(c1SC)CCC2 C1(NC(C(C=CCCC)O)=O)CN(C(c2ccsc2Cl)=O)C2(CCCC2)C1 C1(CC)CCCCCCN1C(=O)CCCC(OC)OC.C1(=O)CC(OC)CN1 C1(C(=O)NCC2(N(C)C)CC2)CN(C(=O)C(C2CCCCC2)F)C2(CCC2)C1 Cc1ccc(C)c(C(=O)NCC2(O)CC(NC(=O)CSc3nnnn3C)C2)c1C c1(C(N2CC(C)C(CNC(=O)COC(F)F)C2)=O)ccc(O)c(OC(F)(F)F)c1 N1(C(C2(F)CCN(C)CC2)=O)CCCN(C(c2ccc(C(C)(C)C)s2)=O)CCC1 c1(CC(=O)NC2CCC(NC(c3cc(C(N)=O)no3)=O)C2)cc(F)ccc1F C1(C(=O)NOCC=C)(C(CNC(C2C(C(N(CC#C)C)=O)C2)=O)=O)CCCCC1 C1(NC(C2CC3(CCC3)C2)=O)CCCC12CCN(C(C1(CCF)CC1)=O)CC2 C1(C(=O)NC2(CCNC(c3cccnc3O)=O)CCC2)CCN(CCO)C(=O)C1 c1(CSC)nccc(C(C)C)n1.SCC C1(C(=O)NC2CN(C(c3c(CC#N)ccs3)=O)CC2O)CC12CCS(=O)(=O)CC2 CC1CCC(C(=O)NCC23CC2CN(C(c2ccncc2C(F)F)=O)C3)CC1 N1(C(c2c(C)nsc2)=O)CC(NC(=O)CC(C)n2ccnc2)C(N=[N+]=[N-])C1 C12CCC(C)(C)CN1N(CC)CC(=O)NC2.C1(C=O)CCN(C2CC2)CC1.CC CCCCC(C)C(=O)N1CC(O)(CN(C)C(c2scc(C)c2C)=O)C1 C(N=c1[nH]c(-c2cccc(CN3CCOCC3)c2)cs1)c1[nH]nc(CC)c1Cl c1(N2CCC(C)OC(C)C2)nc2ccccc2nc1N1CCSC(C)C1 C(C(=O)NC12CC(C(N3CC(O)(C(N)=O)C3)=O)(C1)C2)(C(C)(C)C)N(C)C N1(C(c2cnc(C(C)N(C)C)s2)=O)CC(NC(=O)C2=CCC2)CC1(C)C Cc1ccc(C(=O)O)cc1C(N1C(C(=O)Nc2ccc(F)nc2C)CC2CC12)=O C1(C(=O)OC(C)(C)C)CCCN(C(=O)NC2(OC(C)=O)CCCC2)CC1 C1(NC(CC(C)(C)NC(CN2CCC(C)CC2)=O)=O)CC2CCCCN2C1 Cc1cc(C)c(C(N2CCCC2CNC(=O)C(C)Oc2ccccc2F)=O)[nH]1 c1(NC(=O)NCCS(=O)(=O)NC(C)(C)C)nccc2ccc(F)cc12 C1(S(C)(=O)=O)(C(=O)NC2CC(C(=O)Nc3c(C(=O)OCC)nccn3)C2)CCC1 c1(C(N(C2CCCN(C(c3c(CC)csc3)=O)C2)CC)=O)ccnc(C)c1O C1(NC(C2(CCC=C)CCCC2)=O)CN(C(=O)CC(C)CC(=O)OC)CC1N=[N+]=[N-] N1(CC(C(CC)C)C)CC(C)c2cc(NC(=O)OC(C)(C)C)ccc21 c1(-c2c(C)n[nH]c2)nc(C(F)F)n(C(C)(C)C)n1 N1(C(c2c(CC)occ2)=O)CCC(C(=O)NCC2=NOC(C)C2)CC1(C)C N1(C(CC=C)=O)CC2(C1)C(NC(=O)C=Cc1nc(C)co1)CCS2(=O)=O CC1COCC(CC(=O)N(C)CC2(O)CN(C(c3coc(C(F)F)n3)=O)C2)O1 C1(OC)CN(C(=O)COc2cnccc2Br)CC1NC(C1CC1F)=O O=C(C1=Cc2cccc(Br)c2OC1)NC1CN(C(C2CC23CC(O)C3)=O)C1 C(=O)(C1=CC2(CCN(C(=O)C(C(C)C)NC(N)=O)C2)C1)NCc1ccc(C)s1 C1(C(=O)Nc2c(C)c(Cl)cnc2)N(c2ccnc(C#N)n2)CCCC1(C)C C1(C(=O)Cc2cn(CC3CCCOC3)nn2)CCOC(c2cccc(F)c2)C1 S(=O)(=O)(c1c[nH]c(C(=O)NCCC(C)N(C)C(C2(OC)CCSC2)=O)c1)NCC C1(NC(=O)NCC2CCCOC2)C2CC1N(c1ccncn1)C2 C1(OC)CC(CNC(c2snnc2C2CC2)=O)N(C(C2(c3cccs3)CC2)=O)C1 C(=O)(CC1=NNC(=O)C1)N1C(C)CC(NC(=O)C(c2ccc(O)cc2)=O)C1 C(=O)(C1CCCc2scnc21)NCC1(O)CCN(C(C2C(C#C)C2(C)C)=O)CC1 N1(C(C2C(C)C2C)=O)C2CCC(C2)C1C(=O)NCCC[Si](C)(C)C C1(C(N(CC(=O)Nc2ccc(NC)cc2)C(C)(C)C)=O)CCC(C)(C)CO1 O=C(NNc1ccc(F)c(F)c1)C1Cc2ccccc2C1=O CN1Cc2ccc(C(=O)NCC(CNC(=O)CC(F)(F)C(F)F)CO)cc2C1=O c1(OC)ccc(C(F)(F)F)cc1C(=O)NCC(CO)NC(=O)C(C)(C)C(=O)OC Cc1ccc(C(C)(F)F)cc1NC(=O)NCC1CCCC1c1nncn1C c1(CC2N(CC(=C)C)CCC2)ccc(CNC(=O)C(COC)OC)cc1 c1(N(C)C)ncc(C(N2CC(CC3CC3)(NC(=O)C=CC(C)(C)C)C2)=O)s1 c1(C(=O)NCC2(C)CCC(NC(C3(CCF)CC3)=O)C2)nccc2[nH]ccc12 CC1CN(C(c2cnn(C)c2)=O)CC1CNC(c1cc(CS(C)(=O)=O)on1)=O N1(OC(N2C(C)C(C(=O)NC(C)(C)C)CCC2)=O)CCc2scc(Br)c2C1 c1(C(N2CCCC(C(C)C(N3CCC(F)(CN(C)C)C3)=O)C2)=O)ccncc1Cl N12CCC3(CC1)CC(C3)N1CCCC1C2=O.n1(CC)cc(SC)cn1 c1(C(=O)OCC2(CC(=O)OCC)CNC2)ccc(C)cc1 N1(C(Cc2c(C)ccs2)=O)CC(CNC(C23CC(C(C)(C)C)(C2)C3)=O)CC1C C1(C(=O)NCC(O)C2CCC2)(COC)C=CCN1C(C1CCOCC1)=O CCCCCC(O)C(=O)N1CC2C(NC(=O)CN=S(C)(C)=O)C2C1 C#CCC(C)(C(=O)N(C(CCC)C(F)(F)F)CCO)NC(=O)COCCCCC c1(-c2onc(-c3cccc(C(=O)Nc4nn[nH]n4)c3)n2)nnc(O)nc1O c1(C(=O)NCC2CCCCC2NC(c2cncs2)=O)ccc2ncc(=O)[nH]c2c1 C12CC(OC)(C1)OCC(C)=CC(=O)NCCN2.C(=O)(C(C)(C)SC)CC c1(CNC(c2scc(C)n2)=O)c[nH]c2ccc([N+](=O)[O-])cc12.C12CCN(C1)C2=O C1(F)(CNC(c2c(C(=O)OC)occ2)=O)CCC(NC(C2CCCN2C)=O)C1 c1(C(n2nncc2NC(=O)C(=O)NC(CNC(N)=O)C2CC2)C)cccc(Cl)c1 C(=O)(C(=O)C(C)(C)C)NCC(C(=O)N(C(C)C(C)(C)O)C)OC C1(NC(=O)OC)CCN(C(=NC2CCS(=O)(=O)C2)NC2CCS(=O)(=O)C2)CC1 N1(C(=O)C=CC2CCC2)CC2CCN(C(=O)CCc3cccs3)C(C2)C1 CC(C)(CC(F)C(=O)N1CC(C#N)(CCF)C1)NC(c1cccc[n+]1[O-])=O CCCCC(C)C(=O)NC1(C)CCN(C(=O)CCc2nc(-c3ccoc3)no2)C1 C1(CC(=O)NCC2(C(N)=O)CN(C(CC=C=C)=O)C2)CC(O)C12CCC2 C1(NC(c2ccc(NC)cc2)=O)CN(C(=O)CCC(C)CN(C)CC)CCC1F N1(CC(=O)NC(C2CCC2)C)CCCNCC1 c1(C(N(CCCN(C)C(c2c[nH]nc2C2CCCO2)=O)C)=O)ccc(O)nn1 c1(C(=O)NCCC2(O)CN(C(C3(C)CC=CC3)=O)C2)ccc(CN(C)C)cc1 c1(C2(NCc3cc(C(C)(C)C)[nH]n3)CC2)ccc(C2=CCCCO2)c(C#N)c1 N1(C(C2(C)COC2)=O)CC(F)CC1CNC(C1COC(=O)N1)=O c1(CCC(=O)N2CC(C(F)Cl)C2)cccc(O)c1.n12ccc(n1)-c1cn(nn1)CC2 Cc1nc(NC2CCN(C(c3ccns3)=O)C2C)ncc1[N+](=O)[O-] Cc1ccc2c(c1)C(=O)OC(C)(C(N1CC3C4CCC(C3C1)NC4C)=O)C2 N1(CC)CCCCC1C(=O)NON1CCC(C)C1.C(=O)C=CC(C)C N1(C(Cc2cc(C)on2)=O)CC(C(=O)N(C)CC2CC(F)C2)CCC1C c1(C(N2C(C)(CNC(C(C(C)C)O)=O)CCC2)=O)cnc(Cl)c(C2CC2)c1 CC(CO)(C(=O)N(CCCO)CCO)NC(C1CCCOCC1)=O C1(C(=O)NC(C)(CNC(C2CC(n3ccnn3)C2)=O)C2CC2)OCCOC1(C)C c1(C(N(C(C(=O)OC)OC)C(C)=O)=O)ccc2ccoc2c1.C1(CN)CC(F)(C)C1 CC(C)(C#N)CC(C)(NCC1=CCCOC1)Nc1nnnn1-c1ccc(F)cc1 c1(C(=O)NCC(C)(C)NC(=O)CCOC2CCC2)ccnn1CC1CCC1 c1(C(=O)NCC(CC)NC(c2ccoc2)=O)ccc(N(C)C)c(F)c1 C1(C(=O)NCCC(C)c2cn[nH]c2)(NC(C=C(COC)C)=O)CCN(C)C1 N1(C(C2(CCC)CCC2)=O)CC2(CCN(C(C3(CO)CC3)=O)C2)C1 c1(-c2cn(CC3(COC)CN(C(C(CC)C4CC4)=O)C3)nn2)cccnc1Cl CCCC(C)C(C)NC(C12CC(C1)C(COC)O2)=O C1(CNC(c2ccc(C(=O)OC)cn2)=O)COCCN1S(=O)(=O)N(C)C CC1CCCCC1(CNC(C1(F)CCCCC1)=O)NC(=O)Cn1ccnn1 O=S1(=O)NCCN1c1cccc(Sc2nnc(-c3ncccc3F)o2)c1 N1(C(CCC(CC)C)=O)CCC(C)(C)C(CNC(c2ccc(C(N)=O)o2)=O)C1 CCN=C(NCC1C(C)(C)C1(C)C)N1CCN(C(C)(C)O)CC1 C1(c2cn(CC(=O)N(C(=O)C(C)(O)Cn3ccccc3=O)C)nn2)CCCNC1=O C1(CN(C(C(C2CCCC2)OC)=O)C)CC(F)CN1C(c1coc(C(C)C)n1)=O N1(C(C(C(=O)OCC)F)=O)CC(C)N(C(=O)C(C)CF)CC1C C=CC1CCCCN1C(C1C2CN(C(c3cc4occc4s3)=O)CC12)=O N#Cc1ccccc1-c1cnc(C(=O)Nc2cccc(CCO)c2)cn1 C1(C(=O)NCCCN(C)C)(COC)CCCN1C(C1CC1COC)=O.C1(C)CC1 N1(C(C(CC)CN(C)C)=O)CCN(C(c2csc(C3CCCN3C)n2)=O)CC1C c1(C(=O)NC(CC)CNC(C2CCCCC2)=O)ccnc(Nc2ncn(C)n2)c1 N1(C(=O)NCc2c(C)nc3ccccn32)CCC(O)(C2CCC2)CC1 c1(CC(=O)NCC(C)NC(C2C(C#C)C2)=O)ccccc1CC N1(C(c2c(C)noc2)=O)CCCC(C2CC2NC(c2cc3cscc3s2)=O)C1 Cc1cnc(C(N2CCCC(N(C(=O)C(C)Cn3ccnc3)CCO)C2)=O)nc1 C1(CCNC(C2CCC2(C)C)=O)(OC)CN(C(=O)CCN2CCOC2=O)C1 CCN=C(NCCc1ccccc1OC)N1CCN(CC)C(C)C1 C1(OC)CN(C(c2snc(O)c2Cl)=O)CC1NC(=O)CCc1ccnc(C)n1 c1(C(=O)NC(CC)CNC(c2c[nH]nc2C)=O)cc(Cl)c(O)cc1C N1(C(C(F)=CC)=O)CCC2(CCOC2)C(CNC(c2ccc(C3CC3)o2)=O)C1 C1(C(N(C2CN(C(C(CCCC#C)C)=O)C2)C)=O)CC2CCCC(C1)C2(F)F C1(C(=O)NCC2C(NC(C(C)NC(C=C)=O)=O)COC2)CC2(CC(=C)C2)C1 CC1(C)CC(O)CCN(C(c2ccsc2Cl)C(=O)NCC(F)F)C1 CC(C(=O)NC1CCN(C(c2cccn(C(C)(C)C)c2=O)=O)C1)C(C)(C)C N(C1CCNc2ccc(Cl)cc21)C(CC1CN(C)C(=O)C1)C1CC1 C1(CC=C)(NC(=O)CCCC)CCN(C(=O)C=Cc2ccncc2)CC1 c1(CC(N2CCCC(CCNC(C3N(CC)CC3)=O)C2)=O)ccc2c(c1)CCC2 n1(CCC(N2CCC(NC(C(C)C3CC3)=O)C2C(C)(C)C)=O)cnc2ccccc12 c1(OCC)cc(C)c(C(=O)NCCC(O)CNC(=O)C(O)C(F)F)cc1OC Cc1nn(C)c(C)c1C(=O)NCC1CCN(C(=O)CC23CCC(CC2)OC3)CC1 C1(CC(=O)N(C2CN(C(CCCOC)=O)CC2F)C)CCC(F)(F)CC1 C1(F)(CNC(Cc2cc(C)sc2)=O)CCN(CC2CC2c2ccccc2)C1 CCCC(C)CC(C(=O)NCSc1ccccc1)N1CCC(C(O)C(N)=O)CC1 C1(C(=O)NCC(CC=C)NC(c2cnns2)=O)CCCC2(CCC2)O1 N1(C(CSCCCC)=O)CCC(O)(CNC(C2CC2[N+](=O)[O-])=O)C1 C1(N(C(C=CC(=O)OCC)=O)C)CCN(Cc2cn(Cc3nccs3)nn2)C1 N(C(=NCc1ccc(Br)cc1Cl)N(C)CC1CCCO1)C(C=C)C c1(OCC)ccc(C(C(=O)NC(C)(C)C)N(CCc2cc[nH]n2)C)cc1CC N1(C(c2nc(COC)oc2)=O)CCC2CCN(C(c3cc(COC)cs3)=O)CC12 C1(C(=O)NC(c2nn[nH]n2)CC)CC12CCN(C(c1c(Cl)ccnc1Cl)=O)CC2 C1(CC)CC(C(N2CCCC(NC(=O)C=Cc3ccc(Cl)s3)C2C)=O)CC(=O)N1 c1(OC)ccc2c(c1)C(CC(=O)NCC1CN(C(=O)CCCCCF)C1)CCC2 C(=O)(CCCC(=O)NCCN1CCC(C(N)=O)C1)Nc1c(C)cccc1 C123CCCCC1(CC2)C(=O)NCCC1CCN(C1)C3=O.C(=O)(CC1CC1)N.CO Cc1cnc(C(=O)NC(c2ccccc2)CNC(c2cc(Cl)c(Cl)s2)=O)c(C)c1 N1(C(CN(C(=O)COCC(=C)C)C2CC2)=O)CCCC1CNC(C=C)=O c1(C(=O)NCC(COCC=C)(C)C)cccc(N)c1Br Cc1ccc(C(N2CC(O)CC2C(N2CCC3(CCC3)C2)=O)=O)cc1Br C(CC(O)C(=O)NC1CCCCC1NC(=O)CCc1cccc(C)c1)SC C12(C(N3CC(C#C)(O)C3)=O)COC(C1)C(NC(c1cn(C(C)C)nn1)=O)C2 C(=O)(C(C(C)CC)NC(c1csc(C)n1)=O)NC(COC)COC c1(NC(N)=O)cccc(C(=O)NCCC2CCCN2C(C2(CO)CCCC2)=O)n1 C(=O)(CC(C)(C(F)(F)F)N(C)C)NC1C(OC)C(C)(C)C1 C(N=c1cc(C)c(C#N)c[nH]1)C1(O)CN(C(c2ccn(C(CC)CC)n2)=O)C1 S(=O)(=O)(c1ccc(Br)c(C)c1)N1CC(C(N)=O)(OC)C1 N1(C(c2cc(C)[nH]n2)=O)CCC(C(=O)NC2CC(C3CC3)C2)C12CC2 c1(OC(C)(C)C)cccc(C(CF)NC2CCNCC2CO)c1 n1(CCOC)nnnc1C(c1nscc1Br)NCCCSC N#Cc1ccc(NC(c2csc(Nc3nccn4ccnc34)n2)=O)cc1F C1(CC=C)(NC(c2cncc(Cl)n2)=O)CC2CCC(C1)N2C(C1COC(C)C1)=O C(=O)(C(=O)CC(C)CC)N1C(C(N2CCC(CC#C)CC2)C2CC2)CC1C C1(NC(COCC=C)=O)CN(C(c2ccccc2CCC)=O)Cc2ccnn2C1 Cc1c(C(=O)NC2CCCN(C(C3CCS(=O)(=O)N3)=O)C2)nn2ccccc12 c1(C(=O)NC2CCC(NC(C3(COC)CCC3)=O)CC2)cc(C)cc(C)c1N Cc1ccc(C(C)C(=O)NCC=CCC(=O)NC(C)CC2CCOC2)o1 c1(CCCC)ccc(NC(=O)NCc2cnn(C(C)CC)c2CC)cc1 c1(C(CNC(c2cnc(-c3ccccn3)s2)=O)N(C)C)ccccc1Cl Cc1oc(C(=O)NCC(O)CC2CCC2)cc1Br N1(C(C2C=C(C)CS2)=O)CCCC(C(N2CCC(CCC(=O)N(C)C)CC2)=O)C1 C(=O)(C(F)CCC(C)C)NC(COC)CNC(c1nn(C)cc1Cl)=O c1(C(=O)NC(C)CCO)cc2n[nH]cc2cc1-c1ccc(N2CCCCC2)nc1 C1(CCC)(NC(c2ncc(C)cn2)=O)CCCN(C(c2nn(C)cc2SC)=O)C1 N1(c2ncn(C)c(=O)c2Br)CC2CCOCC2C1 C12CCCCN1C2=O.C(O)(C(F)(F)F)N1CC(OC(=O)OCCCC#C)C1 CC1(CO)CCN(C(=O)CCC2CC(NC(C3CCC(F)(F)CC3)=O)C2)CC1O N1(C(C(CCNC(C2(NC3CCC3)CC2)=O)OC)=O)CC2COCC2C1 Cc1ccc(C(=O)NCC2CC(NC(=O)CC(C)C3CCCC3)C2)cc1[N+](=O)[O-] C1(C(N2CCCCC2CO)=O)C2CCC(C2)N1Cc1ccc(F)c(Br)c1 Cc1ccsc1CC(=O)NOCC(=O)NCCOCC(F)F S(=O)(=O)(c1cc(C(=O)N(C(C)CSC)CC)co1)NC(=O)C1=CCCS1 C1(CC(=O)NCC(C)N(C)C)Cc2ccccc2CN1C(C1CC1F)=O N1(C(C2CC(=C)C2)=O)CCCC(F)(C(=O)N(CC(O)CO)CCO)C1 C(=O)(CCP(C)(C)=O)N(C1CCCCN(C(c2ncoc2C(C)(C)C)=O)C1)C CC1(C)CN(C(=O)COCCCN=[N+]=[N-])CC1C(N1CC(F)CCC1CO)=O C(=O)(CC(C)(C)C(F)(F)F)N1CC(OC)C(NC(=O)C(C)C(C)(F)F)C1 C1(CNC(c2c(C)cno2)=O)C(C)CCCN1C(c1cnc(O)cc1C)=O c1(C(N2CCC(CNC(C(COC)(F)F)=O)(OC)C2)=O)cccc2ccncc12 c1(C(=O)NC2(CC=C)CN(NC(C3CC4CC4C3)=O)C2)cc(C)c(CC)s1 C(=O)(C1=C(Cl)CCC1)N(c1c(C)[nH]cc1)CC1C2CN(Cc3ccccc3)CC21 C1(C(=O)NCCN(C(c2cc(C)cc(O)n2)=O)CC)Cc2nn(C)cc2C(=O)N1 C#CCC(C)(C(=O)N1CC(CO)(CO)C1)NC(c1cncc(C=C)c1)=O N1(C(CNC(=O)OC)=O)CC2CC2(CNC(c2cc(C)c(C)o2)=O)C1 c1(OC)cc(C(N2CCC(Oc3ccccc3F)C2)CSC)ccc1[N+](=O)[O-] C=Cc1cncc(C(N2CCC=CC2C(N2CC(C(C)OC)C2)=O)=O)c1 CC1(C)CN(C(C2CC3CC(O)CC(C2)C3)=O)CC2(CN(C(=O)COC(F)F)C2)O1 Cc1nc2cncc(C(=O)NC3CCCC3NC(=O)CNC(=O)OC(C)(C)C)c2[nH]1 CCC(CC(C)CO)NC1CCN(c2ccc(Br)cc2)C1=O C1(C(=O)NCC2N(C(c3cc(CCC)c(C)s3)=O)CC2)CCn2cncc2C1 CCCC(C)(C)C(=O)NCC(CCC1CCC1)OC.C(C)(CC(N)=O)C(=O)N C1(C(N(C)CC2COCCN2C(c2ccsn2)=O)=O)CCCC2C1C2(F)F C1(NC(=O)NC2(C)CCC2)CCC2(CCCCCC2)CC1 c1(C(=O)NC2(N)CCN(C(C)=O)C2)cccc2c1nc(O)n2C c1(C(=O)NC2CC(C)(NC(Cc3c(C)ccs3)=O)C2)ccc(C(F)(F)F)cc1O N1(c2nnc(C(C)C)s2)CCC(C(N)=O)c2ccccc21.C1(N)CCC(CO)CC1 C1(NC(C23CC(NC(CC(C)CN(C)C)=O)(C2)C3)=O)COCCC1(F)F C1(CC#C)(C(N2CC(NC(=O)CC#N)C(CCC)C2)=O)CCCCO1 N1(C(C(c2ccccc2)NC(C(C)C(F)F)=O)=O)CC(CO)C2(CC2)C1 N1(C(c2cnn(C=C)c2NC(=O)OC(C)(C)C)=O)CCn2ncnc2C1 C1(OCC(=O)N(C(C)C(=O)Nc2cnsc2)OCC)CCCC1 Cc1cccc2[nH]cc(CN3CCSC(C(N4CCCC(O)C4)=O)C3)c12 C=CC1(O)CN(C(=O)C(Cc2ccco2)NC(c2cccc(CC)n2)=O)C1 c1(OC)cc(C(=O)N(CCCCN(C)C(C2CCN(C)C2C)=O)C)cc(F)n1 C(=O)(C1=CC(O)CCC1)OC.C(C(C)C(C)C)N(C(=O)CCNC)CCCN C1(NC(C2C(C)C2)=O)CN(C(=O)CCn2ncc3c2CCCC3)CCC12CCC2 C1(C(C)NC(c2sccc2CO)=O)CCCN(c2cc(Cl)ncn2)C1 C(=O)(C1CCCn2cncc21)NC(C)CCNC(c1csc(O)n1)=O C1(CNC(C(C(C)(C)C)SC)=O)Cc2ccccc2CN1C(=O)CC(C)(C)O C1(CN(C(=O)C=C2CCC2)C)CCCC(NC(c2ccnc(C3CCC3)c2)=O)C1 c1(CNC2CC(CC(=O)OC)C2)cc(F)ccc1F N1(C(CC=C)=O)C2CCC1C(CNC(C1(C(=O)OC(C)(C)C)CCC1)=O)C2 c1(CC)cc(C(=O)NCc2nc(C(=O)NCCCOCCOC)co2)cs1 c1(CC)nc(C)c(C(C)N(c2nc(-c3cc[nH]n3)n(C3CC3)n2)C)s1 CC1(CC(=O)Nc2cnn(CC(N)=O)c2)CCN(C(=O)CO)C1 c1(OC)ccc(OC)c(CC(=O)NC2CC(C)N(C(=O)C=Cc3csc(C)n3)C2)c1 C(=O)(C(C)CCCOC)NCCC(C(=O)NCCN(CCC)C(C)=O)C C12(C(=O)NCC(CCNC(=O)Cc3cnccn3)O)C(=O)C3CCC1C2C3 N1(C(C2C(C=C)C2)=O)CCC2CCC(NC(c3cccnc3)=O)C1C2 CCCCCCC(C)(CC)C(=O)N(CCCCNC(=O)CC(CC)C(F)F)C CC1CN2CCN1C(C(=O)N(N1CCN(c3ccc([N+](=O)[O-])[nH]3)CC1)C)C2 C=Cc1ccc(C(=O)N(CCN(C(=O)C=Cc2cnc[nH]2)C)C(C)C)cc1 N1(C(CC2(C=C)CCCCC2)=O)CC2(C1)CN(C(c1ccc(F)c(C)c1)=O)CCO2 c1(OC)cccc(C(C)NC(=O)C(C2CCN(CCNC(C)(C)C)C2)F)c1F CC1C(C(=O)N(CCCNC(C2CC2c2cccs2)=O)C2CC2)C1C C1(NC(C2CCCC(O)C2)=O)CN(C(c2cccnc2O)=O)CC12CCC2 C(=O)(CCCC(F)F)NCCCCN(C)C(C1CC(C)(C)CCO1)=O C1(C(N2C(COC)CCCC2)=O)COC2CN(C(=O)CC(C)(C)C(=O)OC)CC12 C#CCCCN=C(NCCCN(C)C)N(C)Cc1ccc(F)cc1 Cc1csc(C(F)(F)C(=O)NC2CCC(CCNC(=O)CCC3(C)N=N3)C2)n1 Cc1cc(=NCC2(C)CCN(C(=O)CCc3ccccc3)CC2)nc(Cl)[nH]1 C1(NC(=O)CSCC(F)F)CC12CCN(C(C1CCC3(CC1)CC3)=O)CC2 C1(C(=O)OC(C(C)N(CC=C)CCC)=O)CCNC(C(F)(F)F)C1 C=CCCN=C(NCc1ccc(Cl)cc1)NCC(=O)NC1CCC(C)C(C)C1 CCCCC(CC)CCCN(C(=O)C(N1CCOC2C(O)CC12)=O)C CCC(C(N)=O)N1CC(NC(C2CCCC2C(c2cn(C(C)C(=O)O)nn2)=O)=O)C1 C#Cc1cc(OC)ccc1NCCC(CC)(CCCC=C)C1CC1 N1(C(C2CC(N(C)C)C2)=O)CC(C)(C(N2CCC(CO)C(O)C2)=O)CC1(C)C c1(C(=O)NCC2(CNC(C(C3CCOC3)OC)=O)CCC2)ncccc1Cl CCC(C)C(C(=O)N1CCOC(CNC(C2OCCC2(C)C)=O)C1)OC c1(C(=O)NCCN(CCC)CCC)ccc(C(C)(C)C)[nH]1 C(CC(F)F)(C(=O)NC1CC12CCC2)N(C(CCc1cc(C)no1)=O)C Cc1ccc(C=CC(=O)NCC(CC(C)C)NC(c2cnc3n2CCC3)=O)nc1 C1(NC(C2(OCC)CCC2)=O)CC2CCC1CN(C(C1(C(C)C)CC1)=O)C2 O=C(NNc1cc(Cl)nc(Cl)c1)C1CCC12CC2(F)F c1(C(N(CCOCCNC(C2CC(O)(CC)C2)=O)C)=O)ccc(CO)nc1 C1(NC(c2c(OCC)cc(Cl)cc2)=O)CCC2CC1CN2C(=O)C(F)=CCCF N1(C(c2[nH]c(C)c(C(=O)O)c2C)C=O)CCCC2(C1)OCC1CC21 C1(C(=O)OC)CN(C(=O)NCC(C2CCOCC2)(F)F)C2(CCCC2)C1 CC(=O)C(C)(C)CC(=O)N(C)CCc1cn(-c2cc(C)c(Br)c(C)c2)nn1 CCC(CC)=CC(=O)NCC=CCNC(=O)C(C)c1ccco1 N1(C(CCC(=O)N(C)C)=O)CC(C(=O)N(C2CC=CC2)C)C(F)(F)C1 C(=O)(C(C)CNC(=O)OCCCl)NCCN(C(C)=O)C Cc1cc(C(N2CC(NC(=O)CN3C(=O)CCC3=O)C(C(F)F)C2)=O)cc(O)n1 C1(CCC)CN(C(C2(CCNC(=O)CC3CCOCC3)CCC2)=O)CCO1 c1(C(N2CC(C)C(NCc3ccc(F)cc3)CC2)=O)ccc2ccccc2c1 c1(OC)ccc(C(O)C(=O)NCC(O)CN(C(=O)CSCC(C)C)C)cc1 N1(C(c2cnccc2Cl)=O)CC2OCCN(C(C3CC3C(F)F)=O)C2C1 C(=O)(C#CC1CCCOC1)NC1CCC(C)N(C(c2[nH]nnc2C2CC2)=O)C1 N1(C(=O)Cc2cn(C)cn2)CCCNC(=O)C1C.C(CC=O)NC(C)C CCC(CN=c1[nH]c2c(c(=NCCC3COCCO3)[nH]1)SCC2)N1CCOCC1 C#Cc1cccc(C(=O)NCCCCCC(=O)N(C)Cc2cnnn2C)c1 S(=O)(=O)(c1cc2sc(NC(C)CS(C)(=O)=O)nc2cc1Cl)N1CCCC(CCC)C1 C(=O)(CCCCCN(C)C(c1c[nH]ccc1=O)=O)NC(c1ccoc1)C C(c1ccc(Cl)nc1)=CCNC(N1CCCC(C(=O)NC23CCC(CC2)C3)C1)=O Cc1nc(NCC23CC(NC(c4ccc(C)s4)=O)(C2)C(C)O3)[nH]c(=N)n1 N1(C(C2C(=C)C2)=O)CCC(CC(=O)NCC(CC(C)C)OC)C1(C)C N1(C(C2CCCC(=O)N2)=O)CCc2ccc(NCc3ccnc(Cl)c3Cl)cc2C1 C1(C(C(=O)NCC2(OCC)CN(C(=O)Cc3ccccc3)C2)C)CCCN(C)C1 S(=O)(=O)(c1cccs1)NCCC(=O)N(C(C)CNC(C1CCCC12CC2)=O)C C1(C)(C(N(C2CCN(C(=O)C(C)SC)C2)CC)=O)CCCN1C(C)=O c1(C(=O)OC(C(c2ccc(OC)cc2Cl)=O)C)cnn2c1OCC(C)(C)C2 C12CC3CC(C3C1)NC(=O)C2N(CCC#N)C1CC1.CCOC Cc1nc(N)cnc1N(C(C(c1ccccc1)OC(C)=O)=O)C1CCCC1 Cc1c(C(=O)N(C(C)CNC(=O)C(C)N(C)C)C)cc(O)cc1N C1(C(N(C2CCN(C(=O)CCc3ccsc3)C2)CCC)=O)CS(=O)(=O)CC(=O)N1 C12(NC(c3cc(C)c(O)nn3)=O)CCN(C(c3cccc(CF)c3)=O)CCC1C2 C(=O)(CCNC(=O)Cn1cnnc1)OCC(=C)F C12(C(=O)NC3C(NC(C(c4ccn(C)n4)C)=O)COC3)CC(C)(CO1)C2 c1(SCCNC(C(N2CCC(C)C2)=O)=O)nc(C(F)(F)F)ncc1Br C(C(=O)NCC(C)CNC(C1CCCNC1=O)=O)(C(C)C)NC(=O)OC C1(OCC(=O)OCCCc2nn[nH]n2)CCCCCC1 C1(C)(C(=O)NCC(CNC(Cn2cc(C(C)=O)nc2)=O)(C)O)CC=CCC1 C1(C)(CNC(c2nc(CC)sc2)=O)CCCN1C(c1cc(F)n[nH]1)=O C1(C(=O)N(CC(C)(C)CNC(=O)CC2COCCO2)C)(OC)CCS(=O)(=O)C1 CCCCCCCCNC(=O)CC1CCN(C(=O)C(CC2CCCCC2)OC)C1 C#Cc1cc(C(=O)N(CC)CC2CCCN2C(=O)C(CCC)NC(N)=O)ccc1Cl C12(C(N3C(CNC(C4(OC)CCSC4)=O)CC(O)C3)=O)CCC(CC1)C2(C)C Cc1ccc(=O)n(CC(N2CCC3(NC(=O)Cc4csc(C)n4)CC3C2)=O)c1 C1(CCNC(C2CC2CC2CCC2)=O)CCCN(C(=O)CN2CCOCC2)C1 c1(C(=O)NCCCCCCNC(=O)CN2CSCC2=O)cc[nH]c2nccc1-2 c1(C(=O)NC(C(C)NC(C2CC(C#C)(O)C2)=O)C(C)C)cc(C)c(F)cc1Cl CC1CN(C(C2CCCCCC2)=O)CCC12CCN(C(=O)Cc1ccon1)CC2 c1(C(=O)NC2(COC)CCN(C(C3CCOC(C)C3)=O)C2)ccc2nn[nH]c2c1 c1(OC)cccc(CNC(C)C(N2CC(O)(CCNC(=O)CC3CCC3)C2)=O)c1 C=CCC(C(=O)NCCc1cnn(CC)c1)NC(=O)CC1CCCN(C)C1 c1(-c2ccnc(N(C3CN(C(C(C=C)O)=O)C3)C)n2)ccc(C(F)(F)F)cc1C C(=O)(C1=NOC2(CCC2)C1)N1C(C)CC(CNC(C2(C#C)CCCC2)=O)C1 c1(C(=O)NCCOCCCN(C(c2c(C)cns2)=O)C)nccc(C(F)F)n1 c1(C(=O)NCC2CCN(C(CC3(C)CCCO3)=O)C2)cccc2c1CCCCC2 Cc1cc(C(=O)NC(CNC(c2ccc(Br)cn2)=O)CC(C)C)sc1Cl n1(CC)nc(C)cc1C(N1CC(CNC(c2cc(C3(C)CC3)on2)=O)C(C)C1)=O c1(C(=O)NC(CN(C(C(C(C)C)N(CC)CC)=O)C)CC)cnn(C)c1C#N c1(CC(=O)NC2CCC(NC(C3CC(OCC)C3)=O)C2)c(C)nn(C)c1Cl N1(C(c2nc(C(C)OC)oc2)=O)CCCC(CNC(=O)CCc2cnoc2)C1 C(=O)(CCCCC(N)=O)N1C(CC(N2CCC(C)(O)C2)=O)CC1 CC1CCC(C(N2CC3CC3(CO)C2)=O)N(C(=O)CC2CCC(=O)C2C)C1 C#Cc1ccc(F)c(C(=O)NCCCN(C)C(C2CC3(C)CCC2(C)O3)=O)c1 CCC(F)(F)C(C)(C)C(=O)N1CC2CC(C1)N2C(=O)CC1(C)CCOC1 C(CCCO)(C(C)C)NC(C(C1CN(C(c2nonc2C)=O)C1)OC)=O c1(NC(C(=O)NCCC)C)ccc(C(=O)N(CC(O)CO)C(C)C)cc1 c1(C(=O)NCC2C(NC(c3c(C(C)C)onc3)=O)CCC2)ccc(C#N)cc1Cl c1(NC(=O)NCCCN(CC(C(C)C)C)C)cccc(Cl)c1 Cc1nn(CC(=O)NC2CN(C(=O)Cc3ncc(F)cc3F)CC2C)c(=O)n1C N1(C(C=Cc2n(CC)ncc2)=O)CCC2(CC1)CC2CNC(=O)C(C)C(=O)OC CCCC(C(O)C(=O)NCC1CC(F)C1)NC(=O)CSCC1CC1 CC(C)(CS(N)(=O)=O)C(=O)N1CCCC2(NC(=O)CS(C)(=O)=O)CC2C1 CCC(C)(C)C(O)C(=O)N1CCC(c2cn(-c3cc(Cl)c(F)cc3Cl)nn2)CC1 CC1=CC(O)CN(c2ncnc(NCCc3ccc(F)c(C(=O)O)c3)c2C)C1 C1(NC(c2cnc(C)[nH]2)=O)CC2CC1N(C(=O)CN1CCC(O)CC1)C2 N1(C(CC=CC)=O)CC2(CC(NC(=O)C(CCCC)N(C)C)c3nccn32)C1 CCCC(C)(O)CC(=O)NC(CNC(c1ccc(=O)n(CCO)c1)=O)C(C)(C)C c1(C(=O)NCCn2ncc(C(N3C(CCC)CCCC3)=O)c2)ncc(F)cc1C c1(C(N2CC(N(C)C(c3csc(S)n3)=O)C(F)C2)=O)ccn(C)c(=O)c1 C(=O)(C1=C(Cl)CCCC1)NC1(CF)CCN(C(Cc2cc(C)sc2)=O)C1 c1(C(N2CCC(CCNC(C(C)N(C)C)=O)CC2)=O)cc2c(C(F)F)nn(C)c2s1 C12(CCNC(=O)Cc3cnc(C4CC4)[nH]3)CCC1CN(C(=O)C(O)c1ccco1)C2 C1(NC(C2CCC(NC(C)=O)CC2)=O)CN(C(c2n[nH]cc2Cl)=O)CC(C)(C)C1 C(c1ccccc1C#N)=CC(=O)NCC12N(C(CCC=CC)=O)CCC1CC2 CC1(C)CN(C(=O)COc2cccnc2)CC1NC(=O)CCCn1cnc(C#N)n1 C1(COC)CCCN(CCN(c2ccccc2Cc2ccccn2)S(C)(=O)=O)C1 CC1CCC(C)(C(N2CCCC(CCCCNC(C3CC=CCO3)=O)C2)=O)CC1 c1(CN(CC(CC)O)C(=O)C(=O)NC2CC2)ccccc1-c1cc[nH]n1 C=C(C)CC(C)C(=O)NCCCCN(C(=O)CC1CCCC(C)(C)C1)C CC1(C)CC(CNC(C23CCCC2C3)=O)CN(C(c2cncnc2)=O)C1 c1(CN2C(C(F)(F)F)CCC2)ccc(-c2cccnc2O)cc1 C(=O)(C(C1=CCSC1)N1CCC(C(O)C(F)(F)F)CC1)NCC(C)(C)OC c1(C(N2CCC(CC=C)(NC(C3CC3(F)F)=O)C2)=O)c(C)nc2ncnn2c1C N1(C(C(C=C)(C)O)=O)CC(C2CCCN(C(c3ccc(C(N)=O)cc3)=O)C2)C1 Cc1cc(C(N2CCN(C(=O)CNC(=O)CC3CCC(C)(C)C3)CC2)=O)nn1C N1(C(C2CC(OCC)C2)=O)CCCC12CCN(C(c1cccc(CO)n1)=O)C2 C1(NC(C2(NC(C)C)CC2)=O)COC2(C1)CN(C(C1C3CCCC13)=O)C2 c1(N2C(C)CCC(NC(c3cc(=O)n(C)cn3)=O)C2)ncnc2c1COC2 C1(C(N(CCCCCCC)C)=O)CCCN(C(=O)Cc2cnnn2C)CC1 c1(C(=O)NC2(C)CC(NC(=O)CN3CCCCCC3)C2)cc(F)cc(N)c1N N1(C(C2C(C=C)OCC2)=O)CCOC2(C1)CN(C(C1CCCC1C(=O)OC)=O)C2 C#CCC(C(=O)NC(CO)CC=C)NC(C12CCC(C1)C2)=O C(=O)(N=c1ccn(CCc2cccc(Cl)c2)[nH]1)c1c(C)cc[nH]1 N1(C(C2(C#N)CCC2)=O)C(CC(N2CCC(O)C(F)C2)=O)C2CCCC12 C1(CC)CN(C(CC)C(=O)N2CC(C)(C(=O)N(CCC)CC)C2)CCO1 CC(C)CC(C(=O)NCC1CC=CC1)N(CCc1nccs1)C CC(C)C(O)(C(=O)NCC(C)CNC(=O)CCc1cnc(C2CC2)o1)C(F)(F)F C(=O)(C1=CCCCC1C)NCC1CC(NC(c2ccc(C)nc2O)=O)C1(C)C N1(C(c2c(COCC)noc2)=O)CCC2(C1)CN(c1ncnc3sccc13)C2 c1(C(N(CCCNC(C2C(C)CC2)=O)CCO)=O)ccc(CN(C)C)o1 c1(C(=O)OC)sc(NC(C)CCN2CCCC2)nc1Cl.C(C)(C)O CCCCC(CC(=O)NC1CC(O)(CO)C1)NC(C1OCCCC1(C)C)=O c1(C(N2C(CN(C(CC(C)SC)=O)C)COCC2)=O)cc(C)nc2c1CCCC2 C1(CCOC)CN(C(c2sccc2C)=O)CCN1C(=O)C(CCOC)OC C(=O)(C1=NOC2COCC12)NCC1N(C(C=C(C)C(C)C)=O)C2C(C1)CCC2 N1(C(COCCCC)=O)CCCC(C)C1CCNC(c1cccc(C(N)=O)n1)=O C(CC(C)(C)C)(C(=O)N(C(C(=O)NCC(C)CCO)C1CC1)C)OC N1(C(CCN(CCCCC)C)=O)CCN(C(c2cc(Cl)sc2Cl)=O)CC1CC C1(NC(C(C)SCC)=O)CCCN(C(c2ccc(C(N3CCCC3)=O)cn2)=O)C1 c1(CCC(C)O)cn(CC2C(CNC(C3CCN3C)=O)C2(F)F)nn1 C1(C(N2CC(OC)C(NC(=O)CC3(CSC)CC3)C2)=O)CCc2ncncc2C1 C12(C(=O)NCCc3n(C)c(Cl)nc3)CN(C(=O)OC(C)(C)C)CC1CCO2 C1(NC(c2nnc(CC)s2)=O)CC(C)N(C(=O)Cc2sc(C)nc2C)C1 C1(c2cn(CC(CC)O)nn2)CN(C(c2sccc2COC)=O)CCN1C N1(C(C2CCC(CCCC)CC2)=O)CCN(C(c2cccnc2)=O)CC1CF CC1CN(C(c2ccc([N+](=O)[O-])s2)=O)CCC1C(=O)NCCCNC(N)=O C(C(C(C)(C)C)NC(=O)CCSc1ccc(F)cn1)NC(C=CCCC)=O C1(C(=O)NC(CNC(c2c(C(C)C)onc2)=O)C(C)(C)C)CS(=O)(=O)CCO1 c1(N2CCCC(SC)C2)nc(NCc2cn(C)nc2C(C)C)c2cnn(C)c2n1 Cc1nc(NCc2cn(C)cn2)cc(=NC(C)c2cc(Cl)cc(Cl)c2F)[nH]1 c1(C(N2C(CNC(C3CCCC3)=O)CC(O)C2)=O)cc(C2CC2)nc(O)c1 C(C(CNC(=O)CCc1nncn1C)C(F)(F)F)NC(CC1CC(SC)C1)=O CN1CCN(C(=O)CC2CCNC2=O)C(CNC(c2ccc(CN(C)C)[nH]2)=O)C1 CC#CCC(C(=O)N1CCCCC1C1CC1)NC(c1ncc(F)cc1N)=O C1(CC(=O)N(CC=C(C)C)C2CC2)CCCN(C(C2(C#N)CC=CC2)=O)C1 C1(C(=O)NCC2(NC(c3cccc(C(F)F)n3)=O)CC2)CC2(CCC2O)C1 c1(OC)ccc(C=CC(=O)NC2(C3CCCN3C(c3cccc(Cl)c3)=O)CC2)s1 c1(C(C(=O)NCC(=C)C)N(CCC(=O)OC)C2CC2)cc(Br)c(C)o1 C1(NC(c2ccc(C)s2)=O)CC2CC1N(C(c1cscc1C(N)=O)=O)C2 N1(CC)CC(C(=O)NCCNC(c2cnn(C)c2C(F)F)=O)NC1=O c1(CNCC=C(C)CN2CCCCC2)ncnc(N2CCOC(C3CC3)C2)c1C CCCCCC(O)CC(=O)NC1CCN(C(c2ccc(N(C)C)nc2)=O)C(C)C1 C(CC(F)F)(C(=O)NCCc1ccncc1F)NC(=O)CC=Cc1ccccc1 N1(C(c2cccc(C(C)C)c2)=O)CC2(C1)CN(C(C1CC1F)=O)CC2CO C1(CNC(C2(SCC)CC2)=O)CCCN(C(=O)C(C)n2cccc2)C1 CC(C)C(C(=O)NCC(C)NC(=O)CSc1n[nH]c(O)n1)n1ccnc1 Cc1cc(C(=O)N(C2CCCCN(C(C34CCC(F)(F)C3C4)=O)C2)C)ccc1O C1(C(C)NC(C2N(CC)CC2)=O)CCN(C(c2ccc(C(=O)NC)cc2)=O)CC1 c1(C(=O)Nc2cn(CC=C)nc2)cc(S(N)(=O)=O)oc1C c1(CC(C(=O)NCC2(CNC(CC=C)=O)CCOC2)C)ccc(O)cc1 c1(C(=O)NCC2N(C(C=C(C)C(C)(C)C)=O)CC(O)C2)cc(O)cc(O)n1 C1(C(=O)NC2CN(CCNC(c3c(OC)n(C)nc3)=O)C2=O)CCC(C)(C)OC1 Cc1nc(C(N2CCC(Oc3cccc(F)c3)C2)C(=O)NC2CC(F)(F)C2)c(Br)[nH]1 c1(C(N2CCC(F)(C(N3C(C#C)CCCC3)=O)C2)=O)cc2ccccn2c1 N1(C(c2ncc(C)nc2)=O)CC2CN(C(=O)C(O)CC(N)=O)CC2C1 Cc1oc([N+](=O)[O-])cc1C(N1CC2CC(NC(c3cc(Cl)cnn3)=O)CC1C2)=O CCC(C(C)C)C(C(=O)NCC(F)F)N1CCc2sccc2C1 CCC(C)(C)C(=O)C(=O)N(CC(=O)NCCc1ccc(O)cn1)C(C)C CN1CCC(C(=O)NC(CCO)C2CCCC2)(NC(=O)Cc2cscn2)C1 n1(CC2CC(NC(C3C(C(=O)OC)C3)=O)C2)cc(C(C)C(C)(C)O)nn1 c1(C(=O)Nc2cccc(F)c2)cccc(S(=O)(=O)N2CC3CCC2CNC3)c1 C(=O)(C1CCc2ccccc21)NC1(CC(N2CC(N(C)C)C(CO)C2)=O)CC1 Cc1ccc(F)c(C(=O)NCC2CCCCN2C(=O)Cc2ccc(O)nc2)c1Cl c1(OC)ccccc1CNC(C1CC2CC2N1C(=O)CCc1ccncn1)=O c1(C(=O)NCC2(F)CN(C(C(C)OC)=O)C2)cccn2c(CC(C)C)nnc12 Cc1csc(CCCC(=O)NCC(C2CC2)N(C)C(c2coc(C3CC3)n2)=O)n1 C1(NC(=O)C(=O)NC2C(F)(F)C23CCC3)CCOC2(CCNCC2)C1 C(c1cnn(C)c1C)=CC(=O)NC1CN(C(C(NOC)=O)=O)CC1SC C1(C(=O)NC2C(NC(CN(C3CC3)CC)=O)C2)CCN(C2CCCCC2)C1 C(=O)(C#CC(C)(C)O)NCC(CNC(c1nn(C)c(O)c1)=O)(C)F C1(N(C(=O)Cn2nnc(-c3ccsc3)n2)C)CCN(C(c2cncs2)=O)CC1 N1(C(C2C(C#C)C2)=O)CC(CNC(c2cncnc2C(C)(C)C)=O)CC1(C)C c1(NC(C)=O)ccc(C(=O)NCC2C=CCN2C(c2[nH]c(O)nc2C)=O)nc1 C(=O)(CCCC(=O)N1CCCCC1CNC(c1sccc1F)=O)NC(C)C C1(C(=O)NC2CC(C)N(C(=O)COCCOCCO)C2)CCCCN1N=O C(=O)(C1=CCC(C)CC1)N(CC(N1CCN(C(CNC(CCC)=O)=O)CC1)=O)C c1(CC(=O)NCC(C2CCCN(C(CC(C)(F)F)=O)C2)(C)O)c[nH]ccc1=O CC1(C)CC(C(=O)NC2(c3cccnc3)CC2)(CNC(C2CC(CF)C2)=O)C1 C1(CC(=O)NC2C(C)(C)CC2)CCN(C(=O)CC2CCC3CC23)CC1 CCCC(C)C(C(=O)NC1CC1)N1CCCN(c2ccc(C#N)cc2C)CC1 C1(C(N(C(CCNC(C(CCC)OC)=O)C)C)=O)CCC(O)CN1C Cc1ccc2cc(C(=O)NC3(C)CCN(C(C4CCOC(C)(C)C4)=O)C3)cn2c1 N1(CCC(=O)NCC2(F)CC(NC3CCCCC3F)C2)CCCCCC1 N1(C(c2cc(CNC(C3C(CCOC)C3)=O)[nH]n2)=O)CCOC2CC12 c1(NC(C)=O)ccc(Br)cc1CC(=O)NC1CCCC1NC(c1cnc(C)[nH]1)=O c1(CCC(=O)NC(C)(C)CCNC(C2COCCO2)=O)ccccc1Br c1(C(N2CC(CNC(C(C)CSC(F)(F)F)=O)C2)=O)ccnnc1NC1CC1 C1(OC)(CNC(=O)CC2COCCN2C(c2cc(CC3CC3)c[nH]2)=O)CCCCC1 N1(C(CC2(C)CC2)=O)CC(O)(C2CCN(C(c3cnn4cnnc4c3)=O)CC2)C1 N1(C(c2cc(C)co2)C(=O)NCCCOC)CCC2(CC1)CC2 c1(C(N(C)C)=O)ccc(CNC(c2cc(Cl)c[nH]2)=O)cn1 C1(OC)CC(NC(=O)COCC2(F)CC2)CN(C(=O)CCN2CCOC2=O)C1 c1(C(=O)NCC(C(C)C)NC(C(CCC)O)=O)cc(C)n(-c2cccnc2)c1C CCCC(C)(C)CC(=O)NCC(C1CCCC1)NC(=O)C(CC(C)(C)C)OC c1(C(=O)NCC2CC(NC(C(CC(C)C)(C)O)=O)C2)nccc2ncccc12 C12(NC(c3c(C)nsc3)=O)CCCC(CN(C(=O)C(F)(F)c3ncccn3)C1)C2 C1(NC(CCNC(COC)=O)=O)CN(C(c2ccc(CO)s2)=O)CC1S(C)(=O)=O C1(C(N(C2CC(C)(C)C2)C)=O)CCCC(NC(=O)CCC(C)(C)F)CC1 C1(CNC(C(C)n2ccnc2)=O)CC(F)CN1C(=O)COCc1ccnc(O)c1 CC1CC=C(C(=O)NC2CCCCC2NC(=O)Cc2ccc3c(c2)CCC3)CC1 Brc1cccc(-c2cn(Cc3noc(C4CCOCC4)n3)nn2)c1 c1(OC)cnc(C(N2CCN(C(=O)CC3CC3(Cl)Cl)CC2)=O)c(F)c1 CCN=c1[nH]c(C(=O)NC2CCCC2NC(c2ccc(OC(F)F)cc2)=O)cs1 N1(C(c2ccc(N(C)C)cc2)=O)CCC(C2CC2)C1CNC(C1CC=CC1)=O CC(CN=c1nc2scnc2c(S)[nH]1)C(C)(C)C.C(F)F c1(C(=O)NC(CNC(C2(OCC)CCC2)=O)CO)coc(CO)c1 N1(C(c2nn(C)c3c2CCCC3)=O)Cc2ccccc2C2CC1C2 Cc1cc(C(N2CC3(CCN(c4ccc(C(F)(F)F)nn4)C3)C2)=O)c(C)cc1Cl C1(=CC(=O)NC2(CO)CCN(C(C3C=CCC3)=O)C2)CN2CCC1CC2 C(=O)(C(O)P(C)(C)=O)NCC(CN(C(=O)Cc1nc[nH]n1)C)O N1(C(C(F)=CCC)=O)CCC2CC1C(C)(C)C(=O)N2.C(c1ccccc1)=C.C1CC1 C1(O)(C(C(N2C3CC(NC(C4N(C)CCC4)=O)(C3)C2)=O)(F)F)CCCCCC1 S(=O)(=O)(c1ccccc1S(=O)(=O)NC1COC1)NCC(C1CCC1)OC N1(C(C2C(C)OCCO2)=O)CCC(O)(CNC(c2cc[nH]n2)=O)CC1 CC1CC(CNC(c2ccc(C(C)(C)C)o2)=O)CN(C(C2CCC(=O)O2)=O)C1 C(=O)(N1CC=CCO1)C1(COC)C=CCN1C(C1COCC(C)O1)=O N1(C(CCC=CC(C)C)=O)CCC(C)C1C(=O)NCCC1CCCCCC1 CC(C)CCCC(=O)NC1(C)CCN(Cc2cnc(N)c(Br)c2)C1 CCCC(CNC(=O)Cc1cccc(O)c1)C(=O)NCC1CC12CCC2 c1(C(=O)NC(C(C)C)CNC(=O)C(c2cccn2C)=O)ccc(C#N)o1 C1(C(N2CCC(C(C)C(N3CC4CCC3C4)=O)CC2)=O)CCC2(CCC2)O1 c1(C(C)NC(=O)C(N2CC(NC(=O)OC(C)(C)C)C(C)C2)=O)cccc(F)c1F c1(CCNC(=O)Nc2c(C)cc(C#N)cc2)cn(C)c2ccc(F)cc12 N1(CC2CN(C(C(F)=C(C)C)=O)C2)CCC2(CC1)CNC1(CC2)Oc2ccccc21 C(=O)(CCC(F)(F)F)NC(C)C(CO)NC(C1CC(=O)NC(=O)C1)=O CCCC(CC)CCC(=O)N1CCCC(C(C)(C)C(=O)NC(CC)C(F)(F)F)C1 CC(C)(O)C(F)C(=O)NCC1COCCN1C(c1ccnc(OCC(F)F)c1)=O C1(CNC(=O)OC(C)(C)C)CCN(N2CC(C(F)F)C3(CCC3)C2)CC1 c1(C(N2CCC(NC(C(CC)Nc3ccccc3)=O)CC2)=O)c(O)cccc1F C1(C)(NC(N)=O)CCOC1=O.N1(CC(=O)N(C2C(=O)N2)C)CC2CC2C1 Cc1cc(C(=O)N(C)CC2CCN(C(C3CC3c3ccccc3)=O)C2)ccc1O N1(C(c2c(C)ncnc2)=O)CC2CCN(C(c3cc(I)c(F)cc3Cl)=O)C2C1 C1(C(=O)NCC(C)CNC(c2nc(Cl)ccc2Cl)=O)CC2C=CCC(C1)C2 c1(CC)cc(C(=O)NCCCN(C(C2COC(=O)N2)=O)CC)cc2c[nH]nc12 N1(C(c2ccc(C#N)o2)=O)CC2CCCC2(C(N2CC3CCCC(C3)C2)=O)C1 c1(C(N(CC(O)CNC(=O)CC2CC=CCN2C)C)=O)cc2sccc2n1C N1(C(C2(C#N)CCC2)=O)Cc2ccc(C(=O)Nc3cc(Br)ccn3)cc2C1 C1(NC(C=CSC)=O)CCOC12CCN(C(=O)C(=Cc1cccnc1)C)CC2 N1(C(CSCC#C)=O)CCC(C(F)(F)F)C(NC(C2CCC(C(=O)OC)CC2)=O)C1 N1(C(CC=CC)=O)CC2(CCC2NC(c2cc(C3CCOCC3)[nH]n2)=O)C1 Cc1cnc(C(=O)N(C2CC(NC(C3CC4CCC3O4)=O)C2)C)cc1Br C(=O)(N=c1nc(C)nc2[nH][nH]cc1-2)C1CC(=C)CN1C(c1cc(Cl)cnc1F)=O n1(CCC)cc(C(=O)N(C)CC2C3CN(C(c4cccc(O)c4)=O)CC23)c(C)n1 Cc1cnc(C(=O)NC2CCN(C(=O)C=CC3CCC3)CC(C)(C)C2)cc1C#N c1(OC)ccc(S(=O)(=O)NC2CCCN(S(C)(=O)=O)C2)cc1CNC1CC1 c1(C(=O)NCC2(O)CCCN(C(C3(CC4CC4)CC3)=O)C2)cnc2c(Cl)cccn12 N1(C(C(=O)N(C)C)=O)CCN(C(=O)CCc2ccc[nH]2)CC2CCCCC12 C(c1ccccc1C)=CC(=O)NC1CCC(NC(C2C(SC)CCC2)=O)CC1 c1(C(=O)NC(C)C(C)NC(=O)CCc2ccc[nH]2)cccc(C2(O)COC2)c1 CC(C)CCC(F)C(=O)NC1CC(C)(C(=O)NCC2CC3CCC2C3)C1 C1(C(=O)NCC(C)OC)COC(NC(=O)CNc2ccccn2)C1 CC1C(NC(c2ncc[nH]2)=O)CC2CCC1N2C(c1cc2c([nH]1)CCC2)=O c1(-c2c(C)ccnc2C)ccc2c(C(F)(F)F)cccc2n1 N1(C(c2occ(C)c2C)=O)CCC(C2CN(C(=O)CN3CCP(C)(=O)CC3)C2)C1 C1(NC(CN(C(C)C)C)=O)CCOC(CNC(C23CC(C)(CO2)C3)=O)C1 N1(C(C(OCC)OC)=O)CCC(C(=O)N(CCCN2CCCC2=O)C)C1 c1(SCC(=O)OC(C(C)C)C(=O)Nc2cccs2)ccc(Cl)c(Cl)c1 c1(O)cn2c(C(F)F)cnc2s1.C1(C)CC1(F)F.N12CC(C1)CC2=O N1(C(CCCC(=O)OC)C(=O)NCC2CCOCC2)CCN2CCN(C)CC2C1 c1(C(N(C2CCN(C(=O)C(O)CC(N)=O)C2)C)=O)ccc(C(F)(F)F)c(O)c1 c1(C(=O)NCC23OCC(NC(CCCCC#C)=O)(C2)C3)cc(C)c(O)c(N)c1 N1(C(COC(C)=O)=O)CCN(C(=O)COc2cc(Cl)cc(Cl)c2)C(CF)C1 C1(OC)CC(C(N2CCC(n3cnnn3)C2)=O)N(C(=O)CSC(F)F)C1 N1(C(CCN(CCC)C)=O)CCC(C)(C)C1CC(=O)NC1CN(C(C)=O)C1 c1(N2CCC(CNC(C(CC)(C)C)=O)C2=O)cc(F)cc(F)c1 CCC(O)C(C)(C)C(=O)N(C1CCC(NC(=O)CCC(C)SC)CC1)C c1(CNC(C2CSCCN2C(c2cccc(O)c2F)=O)=O)ccnc(Cl)c1F N1(C(Cc2c(C)nc(Cl)cc2)=O)CC(C)CN(C(C2CC3CC3C2)=O)CC1C C(=O)(C1=CCCCO1)NC(c1ccc(F)cc1)CNC(c1c(C)ocn1)=O c1(OC)cc(C(=O)NC2(CCNC(=O)CCCC3CCC3)CC2)c(N)c(C)c1 C1(CC(N2CCC(CC(=O)NCC3CC(=O)NC3)CC2)=O)Cc2ccccc2O1 N1(C(c2cc(O)nc(O)c2)=O)CCC2(CCCN(Cc3cc(F)cnc3Br)C2)C1 c1(C(N2CCN(C(C(COC)N(C)C)=O)CC2C)=O)cc(C)cc(C)c1O C=C(C)C1OCCC1CNC(=O)CC(C(F)F)NC(=O)CC1COCC(C)O1 CC1(C)C(C(N2CCC(N(C(=O)CCc3ccc(N)cn3)CCO)C2)=O)C1(F)F N1(C(CCCSC)=O)CCCN(C(=O)C(C)n2cncn2)CC1C CP1(=O)CCN(CC(=O)NCC2CCC(F)(CNC(C3CCCO3)=O)C2)CC1 C(CCC(=O)NCC1(F)CN(C(=O)CNC(C)=O)C1)OC c1(CCCC(N2C(C(=O)NC3CC3(F)F)C=CC2)=O)ccc(F)cc1 N1(C(Cc2c(C)occ2)=O)CCC(C)N(C(=O)Cc2cc(C(C)C)no2)CC1 C(c1ccccc1Cl)=CC(=O)NCC1C(CNC(c2c(C)nc(C(C)C)o2)=O)C1 C(=O)(CC(C)C(C)(C)C)NC1CC2C(NC(CCCCOCC)=O)C2C1 CC1CCC(CCC(N2CC(C)(CCC(=O)N3CCC3CC3CC3)C2)=O)O1 CCC(CC)C(C)NC(=O)C(C)(CO)NC(=O)CC1(C#N)CC1 C1(C(=O)NCC2CC2CC(=O)Nc2ncc(CCO)s2)CCCC12CC2 C(CCCN=c1[nH]cnc(Cl)c1C#N)NC(C1N(C(CCC)=O)CCCC1)=O Cc1cccc(F)c1CC(=O)NCC(CNC(c1ccc(F)cc1Cl)=O)CO C1(CNC(CNC(c2c(C)occ2)=O)=O)CC(C)N(C(=O)C(F)C2CCC2)C1 CC1=C(C(=O)NC2CN(C(c3scnc3Cl)=O)CC2C)CCS1(=O)=O C(=O)(C(C)(CO)NC(=O)CC1C(N(C)C)CC1O)N(C(C=C)C1CC1)C C1(CNC(C2C(OC)CC2)=O)CCCC1NC(=O)Cn1cc(C2CC2)nn1 C(=O)(CCC(C)S(C)(=O)=O)N1CCC(CCNC(c2cncc(COC)c2)=O)C1 c1(C(C(c2ccccc2)N(C)C(c2cncs2)=O)=O)ccc(C(F)(F)F)cc1 n1(CCC)ccc(C(=O)NCCC2CC(NC(=O)C(C)(C)NC(=O)NC)C2)n1 C1(C(C)C)CC(NC(=O)CN(C)C(N)=O)C(O)C1.c12nnc(o1)CC(=O)NC2 C1(C2(NC(c3ncccc3F)=O)CC2)CCCCN1C(=O)C=Cc1ncc[nH]1 N1(C(c2ccc(C)cc2)=O)CCC(C(=O)NCCC2=CCC2)C1(C)C c1(C(=O)OCCCNC(C)=O)ccc(-c2nnn(C(C)(C)C)n2)cc1 C1(Oc2cccc(C)n2)CCN(C(=NCCC2CCC2)NC)CC1.C(C)(C(F)F)O N1(C(c2c(C)sc(Cl)n2)=O)CCC2CCN(C(c3ccc(F)c(O)c3)=O)CC12 C=C(C)CCCC(=O)NCC1CCN(C(C2CC(N(C)C)C2)=O)C(C)C1 C1(C(=O)NC(C)CCCCNC(C2CCC2)=O)CCCCC(=O)N1 C12(CNC(Cc3c(CC)con3)=O)CC(CN1C(=O)CCC=CC(C)C)C2 C1(c2n(CCC)nnn2)(NC2CC(F)(F)C2)CC(C)N(CC(=O)OC)C1 c1(C(=O)NC2(CNC(Cc3cnc(C)[nH]3)=O)CCOC2)cncc(N)n1 CC1(C)CCCCC1NC(=O)C(Cn1cccn1)NC(c1cnc(Cl)s1)=O c1(C(N2CCCC(C(C)NC(=O)C(F)F)C2)=O)ncc2c(F)cccn12 c1(C(N(CCCNC(CC2CN(C)C2)=O)C2CC2)=O)cc(F)cc(F)c1 C1(C=O)CC2CC2C1.N1(C(CC2(C(=O)NC)CC2)=O)CC(O)(CCN2CCCC2)C1 C12(CC(=O)NC3CN(C(c4ccc(C)s4)=O)C(C)C3)CCCN1CCC2 C(=O)(C1=C(Cl)CCC1)NC(COC)CC(=O)N(C1CC2CC2C1)C N1(C(c2cnn(C)n2)=O)CCCC(C2CCN(C(c3cnn(CCO)c3)=O)C2)C1 c1(OC)cc(C)cc(C(N2CCN(C)C(CNC(c3ccc(Br)o3)=O)C2)=O)c1N c1(C(=O)OC)cc(C(N2CCN(C(C3CCCSC3)=O)CC2)=O)ccc1Cl C1(C(N(C)CC2(NC(c3c(COC)scc3)=O)CC2)=O)CCCC(C)C1 Cc1c(NCCC2CC(C)(C)CO2)ncnc1NCCN1CCOCC1(C)C c1(C(=O)NC2C(NC(C(CC(C)C)OC)=O)CC2)ccc(N)c2ccncc12 N1(C(COCCCCC)=O)CCN(C(C2CCCC23CCC3)=O)CC1C C(N=c1ccn(CCC)[nH]1)(c1n(CC=C)nnn1)c1cnn(CCNC(N)=O)c1 C1(N(C(CNC(=O)NCC#C)=O)C)CCN(C(c2cnoc2COC)=O)CC1 N1(C(CCc2ccc(CC)cc2)=O)CC2OCCN(C(c3ncc[nH]3)=O)C2C1 C1(NC(C(C)SCCCC)=O)CCCC12CN(C(C1CCC(=O)O1)=O)C2 N1(c2nc(C)cc(OC)n2)CCC2C(CCCN2C(c2nc[nH]c3nccc2-3)=O)C1 c1(C(N2C(CNC(CSCC=C)=O)CC3(CC3)C2)=O)ccc2nnc(C)n2c1 c1(C(=O)NCC2(NC(C3OCC(C)(C)C3)=O)CC2)cnc2[nH]ncc2c1 c1(C(N(C2CCC(NC(CSC)=O)C2)C)=O)nccc2occc12 Cc1cccc(Br)c1C(=O)NC12CC(C(=O)NCCC3CCCN3C)(C1)C2 C1(NC(C(C(C)C)N(CC)CC)=O)CCN(C(C2CN(CC(C)C)C2)=O)CC1O C(N=c1cc(F)nc[nH]1)C1(NC(C(c2ccc(Cl)cc2)C)=O)CCCCC1 C(=O)(CCCCC(F)(F)F)NCC(CNC(CCCCNC(=O)OCC=C)=O)F c1(CC(C(=O)CCOC)=O)cnnn1C.N1(C(CNC)=O)CC(C(COC)N)C1 c1(C(C(N2CCN(c3ccc(F)cc3)CC2)(C)C)NC)c[nH]c2ccc(Br)cc12 CC(C(=O)NCCCC(C)(C)NC(C1CC2(C1)CC(O)C2)=O)C(C)(F)F c1(NC(c2c(C)nco2)=O)cccc(NC(=O)CN2CCCC2C)c1 C1(CC(=O)NC(C)CN(C(=O)CC2CC(=O)NC2=O)CC)(COC)CCOCC1 N1(C(Cc2c(C)noc2Cl)=O)CCCC(C2CN(C(=O)CSCC(F)(F)F)C2)C1 C1(C(N2C3C(C(=O)NC4C(OC)CC4O)C(C3)C2)=O)CC2CCC(C1)C2 c1(C(N(CC(C)NC(=O)C(c2cccc(C)n2)O)CC)=O)cc(F)c(Cl)cc1F C(=O)(C1=CCCC1C)N1CC(F)(CNC(CC(C)c2ccco2)=O)C1 c1(CN(Cc2cc(C)on2)Cc2ccc(Cl)cc2Cl)ccn2c1CCCC2 c1(NC(C2CC(NC(C3C(C(C)C)(COC)C3)=O)C2)=O)nnn(C)n1 N1(C(CC(C)OC)=O)CCCC12CCN(C(c1[nH]c(C)c(C(=O)OC)c1C)=O)C2 N1(C(c2c(C)cc(CC)o2)=O)CC(NC(=O)C(C)(C)CN(C)C)CC1(C)COC CCC(C)(C#N)C(=O)N1CCC(C)(C(=O)NCCCCCCC2CC2)CC1 S(=O)(=O)(c1ccc(Cl)s1)NCC(=O)NC(C)C1CC1.c1(C(=O)O)cc(I)cnc1Cl C1(C(=O)NC2CC(NC(C3CC=CC3)=O)C2)CCN2CCCC2C1 C1(O)(C(=O)NCC2C(NC(c3ncccc3C3CCCC3)=O)C2)CCCCC1 C1(C(N2CC(C(C(=O)N(C(C)C(N)=O)CC)OC)C2)=O)CC2(CCO1)CC2 C(=O)(C1=CCCCC1)NCC1(NC(C(C)NS(CCCC)(=O)=O)=O)CCOC1 c1(N(S(C)(=O)=O)C)nc(=NCCCOCC2CC(F)(F)CO2)[nH]c2ccsc12 c1(C(=O)NC2C(NC(Cc3cn(C)nc3)=O)CCOC2)ncc(Cl)cc1O c1(C(N2CCCC(C)(NC(c3cn(CC)nc3)=O)C2)=O)cc(Cl)cc(Cl)c1N C1(OC(C)C(F)(F)F)COCCC1NC(c1csc(Cl)n1)=O C(C(O)CC(=O)N(C1CCN(C(C2CC(OCCN(C)C)C2)=O)C1)CCO)SC C(=O)(CC(O)CCCC)NC(C1CC(NC(c2ccc(C=C)cc2)=O)C1)C C(=O)(C(F)C(C)(C)O)NCc1nccc(C(N(C2(C3CCCO3)CC2)C)=O)c1 C1(CC=C)(NC(=O)Cc2cncnc2)CCCN(C(=O)COC)C1 c1(OC)ccc(C(=O)NCC2CC2CNC(=O)C=Cc2ccoc2)cc1F c1(CCCC)cn(CC(C)NC(=O)CCN(S(C)(=O)=O)CCC)nn1 Cc1ccc(N)cc1C(=O)NCC1CC(NC(C2(C)C=CCC2)=O)C1 N1(C(c2cc(C)c(C)[nH]2)=O)CC2(COC(CNC(=O)C(F)C(F)(F)F)C2)C1 Cc1ncn(C)c(=O)c1C(=O)NCC1(O)CN(C(C2CCCN2C)=O)C1 c1(C(N(C)CCNC(C2CCC(=O)C2)=O)=O)ccc(S(N)(=O)=O)nc1 C1(NC(CSS(C)(=O)=O)=O)C2CC(O)C1N(C(=O)C1=CCCCC1)C2 N1(C(c2scc(CC)n2)=O)CCCN(C(=O)CCC(C)OC)CC1C c1(C(=O)NCC(C)N(C)C(c2cncn2C)=O)cc(F)c[nH]1 C1(NC(C2(CCCC)CC2)=O)CC(OCC)CN(C(=O)C#CC2CC2)C1 C(C(C)(CC(C)C)NC(=O)CCn1ccnc1)NC(C1(CC#C)CC=CCC1)=O C(C(C(=O)NCC(N1CCCC1)=O)NC(C1CNC(=O)C1)=O)OCC CCCC(C)(O)C(=O)NC1CCC1NC(=O)CCc1ccc(OC)cc1 CC(CN(C)C)CC(=O)NCC#CCNC(=O)C(C)Cc1cnc[nH]1 C1(C(=O)NCCCc2n(C)nnn2)CN(C(=O)C(C)(C)C2CCC2)CC12CCC2 C1(C(=O)NC2CCC(OC)C2)CC2(CC(NC(c3ccc(C)nc3C)=O)C2)C1 C(=O)(C(C)S(=O)(=O)C(C)C)N1CC(C2CN(C(Cc3ccc(OC)nc3)=O)C2)C1 c1(C(N2CCC(O)CC2)=O)cnc(Cl)cc1C(N1CCC(C(F)(F)F)CC1)=O C1(N(C(CN(CCCCCC)C)=O)C)CCN(C(=O)COCC(C)(C)C)C(C)C1 C(CC(C)C)(C(=O)NCC1CC(C)(C)CN1C(=O)CNC(C)=O)NC(=O)OC C1(C(=O)NCCCOC)CC2(CC(NC(C3CC3(C)C)=O)C2)C1 CCCCC(O)C(=O)N1CCCCC1C1(C(=O)NCc2ncc(Cl)cn2)CC1 C1(CNC(=NC)NCC2CCc3nccn32)CCC2(CC1)CC(C)(C)C2 Cc1nn(CC(=O)NCC2CC(NC(=O)C(=O)NC(C)C)C2(C)C)cc1Cl C1(C(N2CCC(NC(C3(OCC)CCCC3)=O)CC2)=O)CCCS(=O)(=O)N1 C(=O)C1CC(NCc2ncc(C(C)=O)cc2I)c2ccccc21.CC(C)(C)OC c1(OC)ncnc(C(=O)NC2CC(NC(C3CC(=O)N(CCN(C)C)C3)=O)C2)c1F Cn1ccc(C(C(=O)NC2CCCCC2)NC2CCCC2C2OCCO2)n1 C1(CC=C)CCN(C(c2cc(CNC(c3cnsc3)=O)[nH]n2)=O)C1 S(=O)(=O)(c1ccc(C(=O)OC(C2CCOC2c2nccn2C)C)cc1)NCC CCCCC(C)(F)C(=O)N1CC2CN(C(c3conc3C(F)(F)F)=O)CC2C1 C1(CNC(c2c(CNC(C(CCC)OC)=O)ocn2)=O)CC2CCC(C1)C2 C(=O)(C(CC=C)CC(F)F)NC(CCNC(CCCCC#C)=O)C c1(C(=O)NC(C(=O)NC2(C)CCOCC2)c2cccs2)ccn2ccnc2c1 N1(C(c2ccc(OC)nn2)C(=O)NCCC)CC(C)C(F)(F)C1 C1(C)(C(=O)NCCN(C(C2(C#N)CCCC2)=O)CC)CCC(F)(F)CC1 C1(CNC(C(CC)CC)=O)CCC2CN(C(c3ccnn3C(C)(C)C)=O)CC12 c1(C(=O)NC2CCCN(C(C(=O)NCC)=O)C2)coc2c1CSC2 c1(C(=O)NCC(CC(F)(F)F)NC(CC=C(C)C)=O)cnc2c(c1)NC(=O)CO2 c1(C(=O)NCC2CCCC(NC(=O)Cc3cncnc3)C2)cc2ccsc2s1 C(=O)(C1=NNC(=O)C1)N1CCC(CCOC)(NC(c2c(OCC)scn2)=O)C1 C(CC(N=c1ccnc(NC(c2cncn2C)N2CCCC2)[nH]1)c1ccco1)OC N=c1[nH]c2c(C(=O)NC3CC(CCNC(C4(F)CCOCC4)=O)C3)cccc2o1 C1(C(C)NC(CN(C(CN2CC(CC)C2)=O)CC2CC2)=O)CC(C)=NO1 C(=O)(C(O)C(C)(C)C)NCC(C)(C)CCNC(=O)C(F)CC1CCCC1 C(=O)(C(C)(CO)NC(=O)CC(C)CNC(=O)C=Cc1ccnn1C)OC C(C(CNC(C1CCC(N(C)C)CC1)=O)C(F)(F)F)NC(c1cn(CC)nc1)=O CCCCC(O)C(C)C(=O)N1CC(C(N2CCCC(F)(CO)C2)=O)C(CC)C1 Cc1c(C(N2CCC(F)(CNC(c3cccnn3)=O)C2)=O)cc(C2CC2)n1C C(N=C(NC1CC1C(F)(F)F)NC1CCS(=O)(=O)C1)c1n(C)ncc1 N1(C(c2ccc(C(=O)OC)o2)=O)CCC2CCN(C(C34CC(OC)(C3)C4)=O)CC2C1 Cc1cc(C(C)(C)C(=O)NCC2CC2NC(c2cncc(O)c2Cl)=O)ccc1F C(N=c1nc(N2CCN(C3CCCC3)CC2)c2c([nH]1)CCCCC2)C1C(C)C1 N1(C(CN(C(C(C)C)=O)C)=O)CC=CC1C(N1CCC(C(C)(C)O)C1)=O C1(CNC(c2c(C)nns2)=O)(NC(c2cnccc2N(C)C)=O)CCOCC1 c1(SC)c(C(N2CCCC(CNC(C3COCC3(C)C)=O)CC2)=O)cccc1F CC1(C(N2CCC(O)CC2C(=O)NCC2CC3(CC3)C2)=O)CCC(=O)NC1 c1(CC)nonc1C(=O)NC1(c2cn(Cc3ccnn3C)nn2)CCC1 c1(C(N2CCC3(CN(C(C(CC)COC)=O)C3)C2)=O)cccc(S(N)(=O)=O)c1C c1(CCC(=O)NCCCN(C(c2cnn(C)c2F)=O)CC)cccc(C#N)c1 N1(C(CC=C)=O)CCC(CCCN(C(=O)C(F)(F)CC2CC2=CC2CCCC2)C)CC1 N1(C(c2c(C)onc2-c2ccsc2)=O)CCCC(C)(Cc2ccccc2)C1 C1(C(=O)NC(C2CCN(C(c3[nH]ccc3-c3cccs3)=O)C2)C)CC(C)(O)C1 CC(F)(F)C(F)C(=O)NCCCC(=O)NC1CC(C)(C(N)=O)C1 N1(C(c2c(C)nc(CCC)s2)=O)CCC(C2CC2)(NC(=O)C=Cc2cc[nH]n2)C1 C(=O)(C(C)(O)CCN(C)C)N(C)CC1CCN(C(c2c(CCC)nco2)=O)CC1 N12CCC(C)C(C1)CC2=O.N1(C(C(C=C)OC)=O)CCC(C)C1OC C1(C(=O)NCc2ccc(C)s2)CCN(C(=O)CCCSC2CC2)CC1 CC1CCC=C1C(=O)NCc1cn(C2CN(C(=O)CC3CCCOCC3)C2)nn1 c1(OC)c(Br)ccc(CNC(C2N(Cc3c(O)cccc3F)CC(C)C2)=O)c1F N1(C(c2c(C)n[nH]c2)=O)CC2CC2(NC(=O)C(c2cscc2Br)=O)C1 C1(C(=O)NC(c2ccc(O)nc2)C)CN(C(=O)C(C)(C)CCF)CC1C1CC1 C1(C(N2CCN(C(C3CC(CC)C3)=O)C(CC(F)F)C2)=O)CN2CCN1CC2C c1(CCC(=O)NCC(C2(O)CCN(C(=O)C3CC3)C2)C)ncc(Br)cn1 Cc1cccc2ncc(C(N3CC(C)(CNC(C45CC(C4)C5)=O)C3)=O)n12 O=C(N=c1ccn(CCO)[nH]1)C1C=CCN(C(=O)Cc2cnns2)C1 CCC(CCOC)C(=O)N(C)CCN(C)C(C12CC1CCC2(F)F)=O c1(OC)ccc(C(N2CCC(NC(C3CC34CCC4)=O)CC2C)=O)cc1Cl C(=O)(C1CC=Cc2ccccc21)N1C2CN(C(CCC(C)(C)SC)=O)C(C2)C1 CN(C)NC(=O)CCC(=O)NCC1(F)CCC(NC(c2cn(C(F)F)cn2)=O)C1 C1(C(N2CC(NC(=O)CC3CCSC3)C2)=O)COc2c(cc(Cl)cc2[N+](=O)[O-])C1 CC(CCNC(=O)COc1cccnc1)C(=O)NCCc1cscn1 CC1(F)CCN(C(=O)C(C2CCC2)NC(c2cncc(O)c2)=O)CC1 c1(C(=O)NC2C(CNC(C=CC=CC)=O)C2)cccc(O)c1NCC Cc1c(Cl)ccnc1C(=O)NCCC(C)(C)NC(=O)CCC(C)N(C)C Cn1cc(NC(C2C(O)CCN2C(=O)CCc2ccnn2C)=O)c(O)nc1=O Cn1nnc2ccc(C(N3CCN(CC(=O)O)CC3)=O)cc12.C1CCS1 Cn1cnc2cc(C(N3CCC(NC(=O)CCc4ccon4)C(O)C3)=O)ccc12 C1(C(=O)NC(C(C)NC(c2onc(C)c2C)=O)C)CCc2nc[nH]c2C1 C(CC(=O)NC(C)CC(C)NC(c1ccnn1CC(F)(F)F)=O)(C(C)C)OCC N1(C(C2CC(SC)C2)=O)C2CCC1C(CNC(=O)C=C1CCC1)C2 N1(C(c2c(C)ocn2)=O)CCOC2(CCN(C(=O)CC(CN(C)C)C(F)F)C2)C1 C(=O)(CCC1=NNC(=O)CC1)NC1C(NC(c2c(OC)ccs2)=O)CS(=O)(=O)C1 c1(C(N2CCC3(C(C(=O)NCCC(C)C)C3)C2)=O)ccc2occc2c1 C1(CCC(=O)NCCCC(C)NC(c2cc[nH]c(=N)c2)=O)CC(C)(C)CO1 C1(NC(c2c(C)scn2)=O)CC1C1CCCN(C(c2ccn(C)c(=O)c2)=O)C1 C1(CNC(C2CC(O)(CC#C)C2)=O)CC(C)(C)CCC1NC(=O)C(F)F C=CCCCC(=O)NC(C)(COCC)C(=O)NCCc1cn[nH]c1 C(=O)(C#CC1(C)CC1)NC(CC)CNC(c1occc1C)=O.C1(C(=O)NC)CCC2CC12.N(C)N.C c1(C(N2CC(CCNC(c3cn4ccnc4s3)=O)C2)=O)cccc(F)c1F N1(C(=O)OC(C)(C)C)CC2CCC2(CCNC(=O)CCCNC2C=CCC2)C1 CCCC(C)(CCC)C(=O)NC1CCOC(C(=O)NC2COCC2F)C1 C1(CNC(C(CC=C)(F)F)=O)CC2(CO1)CN(C(c1ccc(Cl)cc1N)=O)C2 c1(C(=O)OCC(=O)NCC)ccc2cc(C)nc(OC)c2c1 C1(CC(=O)NCC2(OCC)CN(C(C3CCO3)=O)C2)CCC(=O)NC1 C1(C2CCN(C(C3CC34CCCC4)=O)C2)(NC(c2cnc3c[nH]nc3c2)=O)CC1 N1(C(c2c(C)n[nH]c2C)=O)CCC2CCCC12C(N1CCC(F)(F)C(F)C1)=O C1(CNC(c2scc(CNC(C(C)C3CC3)=O)c2)=O)CC(=O)NC1(C)C C1(CCOC)(NC(C2CCC(C)=C(C)C2)=O)CCN(C(=O)C(C)(C)N=[N+]=[N-])CC1 C1(NC(c2n(CC)nnc2C)=O)CC12CCN(C(c1cnoc1C(C)C)=O)CC2 C1(SC)CCC(N=c2[nH]c(N3CC(C(F)(F)F)C(F)C3)nc(=N)[nH]2)CC1 CC(C(=O)NCC(C)(C)NC(C1CC(C(F)(F)F)C1)=O)C1=CCCC1 Cc1cc(C#N)cc(C)c1CC(N1CC2CN(Cc3ccc(O)cc3O)C2C1)=O c1(C(=O)NC(CNC(C(CC=CC)CC)=O)C(C)C)cnc(O)c([N+](=O)[O-])c1 C1(NC(=O)C=CC2CCCC2)CN(C(c2cccc(-n3cccc3)c2)=O)CC1O O(NC(=O)C1=CCN(C(c2cc(C)nc(O)n2)=O)C1)C(C(=O)OC)C c1(C(=O)OC)nc(-c2cn(CCCC(=O)NCC3CCC(C)C3)nn2)c(C)s1 N1(C(c2c(C)nn(C)c2)=O)C2CCCC1CC(NC(c1cc(F)cs1)=O)C2 C(=O)(CC(C)C(C)(C)NC(=O)CCCCNC(N)=O)NCCc1cn(CC)nn1 Cc1c(C(=O)NC(c2cccnc2)CN(C(=O)C(C)(C)C)C2CC2)cnn1C1CC1 c1(C(N2C3(CNC(C(C(C)(C)C)O)=O)CC(C2)C3)=O)ccc(F)c2ccccc12 C1(C)(CNC(C(C(C)O)NC(=O)C=CC2CCCCC2)=O)CC2(CCC2)C1 c1(COC(C)C(=O)NCC2CCCN2C(C2CN(C)C(=O)N2)=O)ccc(O)cc1 C(=O)(CC(C(F)F)C(C)(C)C)N1CCCC(O)(CNC(CSCC=C)=O)C1 CCCN=C(NCCC(C)(F)F)N(C)CC(C)Oc1ccc(Br)cc1 N1(C(C(COC(C)=O)C)=O)CC(CNC(c2ccn(C(F)F)n2)=O)C(C)C1 c1(C(=O)NC(C(C)NC(=O)C(F)CC2CCCC2)C)cc2ccccc2nc1O N(C(=NCCCC(=O)OC(C)C)NC1CCS(=O)(=O)C1)CC1(COC)CCOC1 CCCC(F)C(=O)NCC(O)CN(C(=O)CCc1ncc(C)o1)C C1(CN(C(CC(=O)OCC)=O)C)CCCC(NC(c2ccc(N(C)C)cc2)=O)C1 C1(NC(CC(C)C2CCC2)=O)CCC2(CCN(C(C34CCC(C3)OC4C)=O)C2)C1 C=CC(CCC)CC(=O)N1CC2=C(C1)CN(C(C1CC3CCC1CC3)=O)C2 c1(CNC(C(COC)OC)=O)nnn(C)c1C(=O)NCC1CCOC1(C)C CCC(C)CC(=O)C(=O)N1CC(CCCCNC(c2ccoc2C2CC2)=O)C1 N1(C(c2sc(CC)c(C)c2)=O)CC(C)CN(C(=O)CCCN(C)N=O)CC1C C1(CSC)CCN(C(=O)Cn2cc(C34CCC(C3)C4)nn2)C1 C=CCC(F)(F)C(=O)N1CCC(F)(CNC(c2ccn(CCOC)c(=O)c2)=O)C1 C1(NC(C(CCCC)O)=O)COCCN(C(c2cc(Br)cn(O)c2=O)=O)C1 c1(C(=O)NC(C(C(C)C)NC(c2c(SC)snn2)=O)C)cc(C)c(C)c(C)c1 C(=O)(CS(=O)(=O)CC(F)(F)F)N1C2CC(NC(CCNC(=O)CO)=O)C1CC2 Cc1cnc(C(=O)NC2CCC2NC(C2(C)CC=CCC2)=O)cn1 C1(NC(c2c(C)nc(C)o2)=O)CN(C(=O)CCCN(C)N=O)C2(CCOC2)C1 C=CC1(C2(C(=O)NC3CCN(C(C4CC4F)=O)C3C)CCC2)CCC1 C1(NC(=O)CC2CC2)CCC2(CC1)CC(NC(C1CCn3nnnc3C1)=O)C2 C1(C(=O)NCC(c2ccccc2)CNC(=O)CC2CCSC2)CC2C=CC1O2 C12(NC(CN3C(C)CCCC3)=O)CC(CNC(c3ccco3)=O)(C1)OC2(C)C c1(NC(c2c(F)cc(Cl)cc2F)=O)cnc2c(c1)CN(C(c1cncs1)=O)CC2 N1(C(Cc2c(C(=O)OC)nco2)=O)CCCN(C(=O)C(C)(C)C(N)=O)CC1C c1(CCC(=O)NCC(CC)(C)NC(c2c[nH]nc2C(F)(F)F)=O)ccccc1Cl O=C(N=c1[nH]cc(Br)nc1Br)C1CN(Cc2ccc3ccccc3c2Br)C1 C(=O)(C1=NN(C2CC2)C2(CCOC2)C1)NC1CCCN(C(CCC)=O)C1 Cn1ccc2c(C(=O)N(c3ncnc4cc[nH]c34)C3CCNCC3)cccc12 c1(C(=O)NCC2CCCN(C(C(C=C)O)=O)C2)cccn2cc(C)nc12 C1(C(=O)NCCCN(C)C(c2ccc[nH]2)=O)CCCCC1O CCCCC(=O)C(=O)N1CCCC(CC(N2CCC(OCC(N)=O)C2)=O)CC1 C(=O)(CC1OCc2ncccc21)N1CC2C(N(C(CC=C=C)=O)C)C2C1 c1(OC(C)C(=O)NC2CC(NC(C3(CC(C)C)CCNC3)=O)C2)ccc(Cl)cc1 N1(C(CCC(C)SC)=O)CC2CC(NC(=O)CCn3cnnn3)C(C2)C1 N1(C(c2ccc(NC)cn2)=O)CC(C(=O)N(c2ccsc2)C(C)C)C2(CC2)C1 c1(NC(=O)NCc2ncc(C(NOC(C)(C)C)=O)s2)cncc2nc[nH]c12 N1(C(c2cn(CCC)c(=O)cc2)=O)CCN(C(=O)CS(=O)(=O)NCC)C(C)C1C c1(C2(C(=O)NCC3CCN3C(C3CCN3S(C)(=O)=O)=O)C(C)C2)ccccc1 Cc1[nH]cc(C(=O)NC2CC3CCC2N3C(c2ccnnc2)=O)c(=O)c1Cl C1(CNC(C(CCC)O)=O)CN(C(c2c(C)cccc2F)=O)C2(CCC2)C1 c1(CC(=O)NCCC(CNC(c2c(CCC)occ2)=O)O)ccc(O)c(F)c1 C(=O)(CCCCC(C)(C)C)NCC1(COC)CN(C(c2cccc(F)c2F)=O)C1 c12ccc(c(Cl)c1OC)[nH]c2=O.N1(CC(C(=O)OC)OC)CCSC(C)(C)C1 Cc1cccc(C)c1CNC(C1CCN1C(C1CC2CC1CC2=O)=O)=O C(=O)(C(C)(C)C(N)=O)NCC(CCOC)NC(=O)COC1CCCOC1 Cc1cc(CNC(=O)C(CCF)NC(=O)Cc2cn[nH]c2)cc(C)c1 c1(C(=O)NCC(C)(C)NC(C(c2c(OC)cccc2)C)=O)c[nH]cc(C)c1=O n1(CC(=O)OC)cc(O)c(=O)c2ccccc12.c12ccc(cc1)N1CCN(CC1)C2 CCCCCC(=O)N1CCC(N(C(=O)C(CC)OC2CCCC2)CC)C1 C(=O)(C1=CCc2ccccc21)N1CCC(CNC(COCCCC)=O)C(F)(F)C1 C(=O)(C1=NN(C)C(=O)CC1)N(C)CC1CCCN(C(c2ccc(C)cc2C)=O)C1 CCC(C)CCC(=O)NCC1CCN1C(=O)Cn1cc(-c2ccccc2)cn1 N1(C(C(c2ccc(C)cc2)=O)=O)CC(NC(C2CCCOC2)=O)C2CCCC12 c1(C(N(CCNC(CCCOCCOCCC)=O)C)=O)cnc2[nH]cncc1-2 Cn1nc(CC(N2CC=CC(NC(c3ccc[nH]3)=O)C2)=O)cc1C(F)(F)F N1(C(C2CN(C(CCN(CCC)C)=O)CC(C)O2)=O)CCn2c(C)nnc2C1 C1(N(C(c2snnc2C)C(=O)NCC2CCOC2)C)(COC)CCN(C)CC1 N1(C(CC2=NNC(=O)C2)=O)CC2(C1)CN(C(C1NC(=O)C3CCC13)=O)CCO2 N1(C(c2c(CC)nn[nH]2)=O)CCC(C)C(N(C)C(c2cc(C(F)(F)F)ns2)=O)C1 c1(C(N(C)CC2CCC(NC(=O)C(c3cccn3C)=O)CC2)=O)ncc(Cl)n1C C1(CNC(c2nccc3ccsc23)=O)C2CCCC1N(C(C1CCCSC1)=O)C2 CC1(C)CC(CNC(C2CCC(=O)O2)=O)CN1C(=O)CSC(F)(F)F C(CC1CC1)(C(=O)NCCCC(N)=O)NC(C1C(=C)C1)=O C1(N(C(CC(=O)NCC)=O)C)CN(C(=O)CCc2ccccc2)CCC1C c1(C(N2CC(O)(CNC(c3ocnc3C(F)F)=O)C2)=O)cccc2nccn12 CS(C)(=O)=Nc1nc(C(N2CCC(NC(C3CC34CC(F)(F)C4)=O)C2)=O)cs1 c1(C(N(C2CCCC(NC(CCCCN(C)C)=O)C2)C)=O)cnc2scnc2c1 N1(C(c2cnc(OC)s2)=O)CCC(NC(c2ccc(C(C)C)nc2C)=O)C(O)C1 c1(C(=O)NC2CN(C(CC3(N(C)C)COC3)=O)CC(O)C2)ccn2cncc2c1 N1(C(c2c(O)ccc(OC)c2)=O)C2CCC1CN(C(C1CCOC(C)(C)C1)=O)C2 c1(CCC)c(C(=O)NC(CNC(C2CCCC23CC3)=O)CO)cnn1CCO N1(C(=O)C(F)=CC2CC2)CCN(C(C2CC3C=CC2O3)=O)CC2(CC2)C1 C(=O)(CCS(=O)(=O)C(F)(F)F)N1C2C(CNC(C(C#C)(C)C)=O)(CCCC2)CC1 C1(NC(c2c(C)ncnc2)=O)CN(C(C2CCN2S(C)(=O)=O)=O)CC12CCC2 C1(OCCNC(CN(C(c2c(CC)c[nH]c2)=O)C)=O)(CO)CCC(C)(C)C1 CCC(CCOC)C(=O)NCc1ccc(C(N2CCC(OCC3CC3)C2)=O)o1 c1(C(=O)NC2C(NC(C3C(C(=O)OC)CCC3)=O)C2)ccc(C)cc1Br c1(NCC2(N(C(=O)C(C)(C)Oc3ccccc3)C)CC2)ccn(CC(F)(F)F)n1 Cc1ncc(CNC(C2(CNC(c3csc(Cl)n3)=O)CC2)=O)s1 N1(C(C(C)CBr)=O)CCOCC1CC(=O)Nc1cccc(OC(F)F)c1 N1(C(CCN(CC(C)C)C(=O)CNC=O)=O)CCC(F)(NC(=O)CC)C1 N1(C(Cn2ccc(C)c2)=O)CCC(C(N2CC(N=[N+]=[N-])C2)=O)C1C C1(C(=O)NCCC2(O)CN(C(c3nc(CC)oc3C)=O)C2)CCN(C)C(=O)C1 C(=O)(CC(C(C)(C)C)NC(=O)CC1CCC(=O)N1C)N(C(C)CS(C)=O)C N1(C(CSc2c(C)cccc2)=O)CCC2CCN(C(=O)C(C)CF)CC12 N1(C(Cc2ccc(C)s2)=O)CCCC2CN(C(=O)CCC3(C)CCC(=O)N3)CCC12 c1(C(N(C2(CN)CC2)C)=O)cc(Cl)cc(Cl)c1N C1(C#N)(NC(CC2CCN(C)CC2)=O)CCN(Cc2ccc(O)cc2Cl)C1 C1(C2(O)CCC2)(C(=O)NCCC2CC(NC(c3c[nH]nc3C3CC3)=O)C2)CC1 C(C(N)=O)(C(C)C)NC(c1c(CNC(C(C)=C2CCC2)=O)nnn1C)=O CC(CC(N)=O)C(=O)NCC1(C)CC(NC(=O)COC2CCOCC2)C1 C(CN=c1[nH]c(N2CCC(c3ccc(F)cc3)C2)nc(=N)[nH]1)c1c(C)cncc1 Cc1cccc2oc(OCCNC(=O)CC(F)F)nc12 c1(CCCN(C(C2CCC2CCC(=O)Nc2nnsc2C)=O)CC)ccccc1 C(N=c1[nH]cncc1I)C1CCC(NCc2cccc(C(OC)OC)n2)CC1 Cc1ccc(C(=O)NC2CN(C(=O)C(C)(C)C3CC3)CC2CO)cn1 S(=O)(=O)(c1cccc(NC2CCC(C(N)=O)C2)c1C)NC(=O)OC c1(C(N(CC(C)NC(C2(C)CC(C3CC3)=NO2)=O)C)=O)cc(Cl)c(F)cc1Cl N1(C(C2(CCOC)CCN(C(CCCCSC)=O)C2)=O)CCC(F)C(O)C1 N1(C(CS(CCCC)(=O)=O)=O)CC23CCCC2(C1)CN(C(C1C2CCCC12)=O)C3 N1(C(CC(C)CF)=O)CCN(C(=O)CC2CC=CC2)CC1CS(C)(=O)=O N1(C(C(C(=O)OC)C)=O)CCCC(O)(CNC(C2CC2c2ccc(C)s2)=O)CC1 c1(NC(C2C(C(=O)Nc3ncc(Br)cc3CO)CCC2)=O)ncc(F)cc1F Cc1nn(C2CCOC2)cc1C(=O)NCC1CN(C(=O)COCC(C)C)CCO1 C1(CC(=O)OCCOCC)CCCCN1C(c1nc(C)cn1C)=O C(=O)(C(CCF)NC(N(c1cccnc1C(F)(F)F)CC)=O)OC(C)(C)C c1(N(C)C)cc(C(=O)NCC=CCNC(=O)Cc2cc[nH]c2)nnc1C1CC1 c1(CCN(C(=O)C(C2CCC2)NC(=O)CN(C2CCCC2)C)C)cc[nH]n1 c1(OC)n[nH]c(NC(C2(F)CCN(Cc3ccc(I)c(F)c3)C2)=O)c1C#N CCC(F)C(=O)NCC1CCC1NC(c1ocnc1-c1ccccc1)=O C(C1C(=O)N(C)CCC2CCC(C2)O1)OCC.n1(CC)cc(C2(O)COC2)nn1 N1(C(C2(CC)CCC2)=O)CCN(C(C2CCC(C(F)(F)F)O2)=O)C(CC(F)F)C1 CC1=C(C)CC(C)(C(N2C3CCC2CC(N(C)C(C2CCC2)=O)C3)=O)CC1 c1(C(N2CCC(CN(C(C=CCC)=O)C)CC2)=O)cc2c(cc1N)CCCC2 c1(SC)cc(F)ccc1C(=O)NC(C(C)NC(=O)COC1CCOCC1)C(C)C c1(C(=O)NC2CC(C)(CNC(C3C(F)(C(=O)OC)C3)=O)C2)cc2cnccc2[nH]1 c1(C(N2CCN(C(c3c(C)n(C(C)C)nn3)=O)CC2)=O)nnn2c1CCCCC2 c1(C(=O)NCC(C2CCCC2)NC(C2CCCCS2)=O)cn2c(n1)CCCC2 c1(CC(=O)NCCC(CNC(C)=O)O)ccc(S(=O)(=O)CC(=O)N(C)C)cc1 N12CC(CC1=O)C(=O)N1CC2C1.c1(C(=O)NC2CC(SC)C2)cocc1C Cc1csc(C(=O)NCC(C)(CO)NC(=O)C(C)OCC2CC2)c1Br Cc1cnn(CC2CCN2Cc2cn(CCNC(c3sncc3C)=O)nn2)c1 C1(C(C)NC(COCCC#C)=O)CCCN(C(=O)Cc2cscn2)C1 [N-]=[N+]=NC1CN(C(=O)C(F)F)CC1NC(=O)Cc1cncnc1O C1(NC(C2CC=C(C(=O)N(CC=C)C)C2)=O)Cc2ccccc2C1 C(N=c1[nH]cnc(Cl)c1CO)c1ccc(CNC(c2c(C)con2)=O)cc1 C(c1cnn(C)c1)=C(C(=O)NCCC)C.C(=O)(CC1CC1C(F)(F)F)N(CC)CC.CCC CCCC(C(=O)NCCC1(OC)CCC1)NC(C1C(C)(C)C1(C)C)=O c1(C(=O)NC2(CC=C)CCN(C(=O)C(O)(C3CC3)C3CC3)C2)cc2cnn(C)c2s1 C1(C(N(C(CSC)C)C)=O)CN(C(=O)C=C(C2CC2)C2CC2)CCC1(C)C N1(C(c2cc(C(F)(F)F)ncn2)=O)CCC(C2CCN(C(=O)Cc3cncs3)C2)C1 CC(c1cnn(C)c1)=CC(=O)NC(C1CCCN1C(=O)CN(C)C(=O)C1CC1)C C(CCOCCO)(C(=O)NC1CCCC1(C)C)NC(CCC=C)=O Cc1cc(Br)cc(NC(=O)C(N2CCOCC(C(=O)O)C2)=O)c1N Cn1nccc(C(=O)NCC(N2CCNC(=O)C2)=O)c1=O.C12CCN(C1)C2=O Cc1cc(Br)c(C(=O)NCC2CCCN(C(c3c(O)cc(F)cc3F)=O)C2)cc1F C(=O)(C(F)(F)C(F)(F)C(F)F)N1CCN(C(c2c3c[nH]c(=N)n3ccc2)=O)CC1 N1(C(c2nc(CC)sc2)=O)C2CCC1CC(NC(=O)CC1CCCCC(=O)N1)C2 c1(N2CC3C(CO)C3C2)nc(=NCCOCC2CCOC2)[nH]c2c1CSC2 C(=O)(CC(C)(C)C(F)F)N(CCC(N1CC2(C)CC1(CO)C2)=O)CC=C c1(CNC(CNC=O)=O)ccc(CNC(C2C3(CC3)C23CC3)=O)c(F)c1 N1(C(C2(OC)CCCCCC2)=O)CCN(C(=O)C=Cc2nccs2)CC(CO)C1 Cc1cc(C(N2CC(NCc3cnccn3)C3(CC3)C2)=O)c(F)cc1F c1(CC(C(=O)NCC2(O)CN(C(CC3(C=C)CC3)=O)C2)C)c(C)noc1C N1(OC(c2cn(C)nn2)C(=O)NC2CC(CC(=O)OC)C2)CC2CC2C1 CC(C)(C)C(C)(O)CNC(c1coc(CNC(=O)CN2CC(=O)NC2=O)c1)=O C1(NC(=O)Cn2ncc(Br)n2)C2CN(c3ncc(Cl)cn3)CC12 C1(NC(C=CCC)=O)CCN(C(=O)CC2(CC)CCC2)CC1c1ccccc1 N1(C(C(=Cc2cnc[nH]2)C)=O)CCC(F)C(NC(=O)C=CCO)C1 N1(CC(=O)N(C2CCCCC2)NCc2sc(C)c(Br)c2)CCn2c(cnc2C)C1 CN1CC2(CCN2Cc2cn(CCCN3CCSCC3)nn2)C1 CON(C)C1CCN(C(=O)CC2CCC(NC(=O)C(C3CC3)SC)C2)C1 C(C(CO)N=c1ccc(C#N)n[nH]1)NC(C(CCCCC)CC)=O C1(CNC(C2(C)N(C)CCC2)=O)CC2(CC(NC(c3cnc4n3CCC4)=O)C2)C1 C(=O)(C(O)C1=CCCCC1)N1C(C(=O)NCC(C)(C)C(C)C)CC(OC)C1 C1(CNC(C2N(C)C(=O)NC2)=O)CN(C(c2cccc(=S)n2O)=O)C(C)(C)C1 N12CC3(CCC3)CC1CNC2=O.C#CC1CCCC(NC(C)=O)C1 CCCC#CC(C)(C)NC(C1N(C(=O)CCCCC2CC2)CCC1(C)C)=O C(=O)(CS(=O)(=O)C1CCCC1)NCC1N(C(C2N(C)CCC2)=O)CC2(CCC2)C1 N1(C(c2ccc(C)nc2)=O)CC(NC(=O)Cc2cc(C)[nH]n2)CCC1C C12(CNC(C(C)Cn3cccn3)=O)CC1CN(C(c1cccc(CC#N)c1)=O)C2 N1(C(COC(C)=O)=O)CCCC1(C)CNC(C1CCOC1c1ccc(Cl)cc1)=O Cc1nc2ccc(CNC(=O)NC3CCCCCC3CO)cc2s1 N1(C(C)=O)CSCC1C(=O)NC(C)(C)CN(C(=O)C(C)(O)C1CC1)C CC(CC(=O)N1CCN(C(c2cc(C(F)F)n(C)n2)=O)CC1C)C(F)F N1(CCCc2cn(C)nn2)CCOC(c2cccnc2)C1 c1(COCC)nnc(N2CCCC(CN(C)C)C2)n1C(C)COC C(=O)(CC(C)(C)CCC)NC(CC(=C)C)C(=O)NC(c1cnccc1C)C c1(CC(=O)N(C2CN(C(CC3(CCC=C)CC3)=O)C2)C)cc(=O)n(CC(C)C)[nH]1 C12(C(=O)NCc3c(C)ccnc3)CCN(C(=O)Nc3ccc(F)c(F)c3)CC1C2 N1(C(c2c[nH]c(=NC)o2)=O)CC2CC(NC(=O)Cc3cc(OC)no3)C1C2 c1(C(C)(C)C)nn2ccccc2c1NCC(=O)NC(C(=O)O)C(C)O c1(CC(=O)NC2CCC(CNC(C3(C)N(C)CCC3)=O)C2)cccc2nonc12 C(=O)(CCCC(C)(C)C)NCCN(CCCCC)CCC(=O)OC(=O)C1CC1 c1(C(N2C3CC(NC(c4c(CC)nn[nH]4)=O)C2CC3)=O)cnc2c(c1)ncn2C N1(C(C2CCC(=C)CC2)=O)CCC(NC(=O)CC(C)SC)C(F)C1 C1(NC(N2C(c3ccc(C)s3)CCC2)=O)(CO)CCN(C(c2ccccc2C)=O)C1 C1(COC)CCC(NC(c2csc(Cl)c2)C)C1 C(=O)(C(CC)CC(C)C)N(C1CCCC(NC(C23OCC(COC)(C2)C3)=O)C1)C C(=O)(C(O)C(C)(C)C)NCCC(CNC(c1c(CC)con1)=O)O c1(C(=O)NC2CCN(C(c3n[nH]cc3C3CC3)=O)C2)ccc(Cl)c2occc12 CC(C)CC(CNC(=O)CN1CCCNC1=O)C(=O)N1OC2C=CC1CC2 C1(C(=O)N2CC(C)(O)CO2)C2CCC1CN(C(C1CC(SC)C1)=O)C2 N1(C(c2cc(C)c(Cl)s2)C(=O)NCc2nnn(C)n2)CCC(N=[N+]=[N-])CC1 n1(CC#C)c(C)cc(C(=O)NCC(C)NC(c2ccc(=O)n(C)n2)=O)c1C c1(C(=O)NC2(COC)CN(C(C3CN(C4COC4)C3)=O)C2)cccc(OC)n1 N1(C(=O)CC=C(Cl)Cl)CC2OCCN(C(c3cnn4cc[nH]c(=O)c34)=O)C2C1 Cc1cc(C(=O)NNC(=O)NCCN2CCCCCC2)c(C)n1N Cc1ccc(N)cc1C(N1CC2CC(C1)C2NC(=O)C(c1ccccc1F)C)=O Cc1cc(C(N2CCN(C(c3cnn[nH]3)=O)CC2CO)=O)cc(C)c1Br N1(C(C2CCCN2c2ccccc2)=O)CC2OCC(NC(=O)C(F)(F)CO)C2C1 c1(OCCCNC(C2C(CC)N(C)CC2)=O)ccc(F)cc1F CC1CCN(C(=O)CC2CC(NC(=O)CCn3cnnn3)C2)CC1(C)C C1(O)(C(C(=O)NCCN(C(C2CCCC23CC3)=O)CC)(F)F)CCOCC1 C12(NC(c3ccc(C)o3)=O)CCC(CN(C(=O)C(C)n3ccnn3)C1)C2 c1(C(=O)NC(CN(C(C(CC)(C)OC)=O)CC)C)cccc(OC)c1F C12(C(N3CCC(N(C(c4c[nH]c(=NC)o4)=O)CC4CC4)C3)=O)CCC(C)(C1)OC2 Cc1nsc2cc(C(=O)NC3CN(C(=O)C(n4nccc4C)C)CC3C)cnc12 c1(C(=O)NCc2c(C(N(CC(COC)O)C)=O)n[nH]c2)ccccc1O N#Cc1ccsc1C(N1CCC2CC12C(=O)NCc1nccc(O)n1)=O C(CCCCCNC(C1CC(C(F)(F)F)CO1)=O)NC(C(=O)N(C)C)=O C(=O)(C1CCOc2ccccc21)N1CCC(C(=O)NC(C#CCC)(C)C)C1(C)C CN(CCCC(=O)N1CCC(=CCNC(=O)C=Cc2ccoc2)CC1)N=O CCCCCCC(F)C(=O)NC1(CNC(c2cc3n(n2)CCCC3=O)=O)CCC1 c1(C(=O)NC(Cn2cc(CCCOC)nn2)C)c[nH]ccc1=N C1(O)(CNC(CCCCOC)=O)CCCN(C(c2cn(CC(F)(F)F)cn2)=O)C1 C1(C(=O)NCC(CNC(C(C)OCCCC)=O)O)CN2CCCC2CO1 N1(CCC(C)N)CCCC(C)(C(=O)NC2(C#N)CCOCC2)C1 C1(C(=O)NCC23C(CN(C(c4c(C)con4)=O)C2)C3)Cc2ccccc2C1 c1(C(N2CC(OC)C(NC(=O)Cc3c(C)noc3C)C2)=O)ncc([N+](=O)[O-])n1C N1(C(CCc2scc(C)n2)=O)CC2CC(NC(=O)Cc3sc(S)nc3C)C2C1 C1(C(=O)NCC(=O)NCC(C)(C)C)CCS(=O)(=O)N1 CC1=C(C(=O)NCC(O)CNC(C2(CC(F)F)CC2)=O)Cn2ncnc2N1C C1(CNC(c2c(C)n(C3CCC3)nc2)=O)CN(C(=O)C(C)S(C)(=O)=O)CCN1C C1(NC(C2C(C)(Br)C2)=O)CC2(CCN(C(c3c[nH]c(=N)nc3O)=O)CC2)C1 N1(C(COCC)=O)CCOC(CCCNC(c2cc(C)sc2C)=O)C1 c1(NC(C)(C)CNC(=O)CC(O)CC(C)(C)C)ccc2c(c1)C(=O)NCCO2 c1(C(=O)NC(CNC(c2cc(C)c(C)s2)=O)CC(C)C)cnc2n[nH]c(C)c2c1 c1(C(=O)NC(CCC)CNC(=O)Cc2cncnc2O)cc2occc2s1 c1(C(N(CCN(C(=O)CC2CCCCO2)CC)CC)=O)[nH]c2ccc(C)cc2c1C N1(C(CCC2CCCN(C)C2)=O)CC(CO)C2(C1)CN(C(=O)COC1COC1)C2 CC1(C)CN(c2cccc(NC(C3CC(=O)N(C4CC4)C3)=O)c2)C(=O)O1 C1(CN(C(=O)C2=CCOC2)C)CCN(C(c2ccc(Br)cn2)=O)CC1 c1(C(=O)NCC(C(C)C)NC(=O)COC2(C)CCCC2)nc2ccccc2[nH]1 C1(NC(C)=O)CCC(C(N2CCC(N(C)C(c3cc(Cl)n(C)n3)=O)C2)=O)CC1 C1(n2cc(C(CC)(C)C)nn2)CCN(C(c2cc(Cl)ccc2Cl)=O)C12CC2 c1(N(CCS(C)(=O)=O)C)nc(N2CC3C4C=CC(C4)C3C2)nc2cc[nH]c12 c1(C(=O)NC(CN(C(c2ncncc2Cl)=O)CC)C)ccc(OC(C)C)c(F)c1 C1(CC(N2CC(C(=O)NCC3(CC)CC3)OCC2)=O)CCN(OC)CC1 C1(CC)(CNC(=O)CC(=O)N(C)C)CCCN1C(=O)CCCc1ccsc1 C1(Nc2c(C(C)C)c(C(F)(F)F)n[nH]2)CCC2CN(C(=O)OC(C)(C)C)CC2C1 C1(C(=O)NCCc2cc(C)on2)CC(F)(F)CN1C(=O)CC1CC(=O)C1 N1(C(CC2C(C)(C)COCC2)=O)CCC(NC(=O)C(Cl)=CCl)C(F)C1 N1(C(C2(OC)CC2)=O)CCCN(C(=O)C(C)N2CCC2)C(c2ccccc2)C1 C1(CC(NOCC(=O)OC)=O)C2CCCC2N1C(C1CC1C(F)(F)F)=O C1(CC=C)(C(=O)NCc2nn(C)c(=O)o2)CCCCO1 C#CCC(C)(C)C(=O)N1CCC(CO)(CNC(c2c(OC)ncnc2C)=O)CC1 CCCCC(O)C(C)C(=O)N1CCCC(NC(c2csc(CO)n2)=O)C1 CCC(CN(C)C)C(=O)NCC=CC(N1CCC=C(C)C1)=O C(CCC(=O)N1CCC(CF)C1)(C(C)C)NC(CCCC(C)C)=O C(=O)(CCCC(=O)N1CC(OC)C(NC(=O)Cc2c(C)nn(CC)c2C)C1)NC c1(C(=O)NCC23C(CN(C(CCc4cncc(C)c4)=O)C2)C3)cc(F)ccc1F C1(NC(CCc2cc(OC)no2)=O)CCN(C(=O)OC(C)(C)C)C(C)C1 N1(C(c2c(C)snn2)=O)CC(O)CC1CNC(c1cnn(C)c1N)=O C(=O)(NNC(=O)Cc1ccoc1)N(C(C)Cc1ccc(OC)cc1)CC CCCCC(C)(F)C(=O)NC1COCCN(C(c2cncc(OC3CNC3)c2)=O)C1 C1(C)(CC)C=C(C(=O)NCC(=C2CN(C(=O)CCC3CCC3)C2)F)C1 N1(C(c2ncn(C)c2)=O)CCC2C(CCCN2C(c2cccc(CO)n2)=O)C1 CC(C)C(O)C(=O)N1CCC(CNC(=O)CCNC(c2ncccc2O)=O)C1 N1(C(C2(CC=C)CC=CC2)=O)CCC(CCOC)(NC(c2ccsc2Cl)=O)C1 O=C(C1=CC2C=CC1C2)NC1(CNC(C2CC3(C2)CC2(CC2)C3)=O)CCCCC1 N1(C(c2c(C)coc2)=O)CCC(C2CC(NC(c3nc(C)c(C)nc3C)=O)C2)C1 C(=O)(C(C)C(O)C(C)C)N(CCNC(c1n(CCC)ccc1)=O)CCC C(C(=O)NNC(=O)c1ccccc1Cl)NC1(C)CCCCC1 N1(C(CCC(C(=O)NCC)C)=O)CCC(N)C(F)C1.c12ccc(O)c(c1)OC2=O.OC c1(C(N2CCN(C(C(C=C)(C)CC)=O)CC(C)C2)=O)cccc2cnccc12 N1(C(C=Cc2n(C)ccc2)=O)CCCC(NC(c2cscc2Cl)=O)C(F)C1 C1(NC(Cc2c(C)noc2)=O)CN(C(=O)CC2CCC3(CC3)CO2)CC1N=[N+]=[N-] c1(OC)ccc(C(=O)NCC(C)NC(=O)CC(F)(F)Br)c(OC)c1 C1(NC(COCCC=C)=O)CCCC(CC(=O)NCC(C2CC2)N(C)C)C1 n1(CCN(C)C)nccc1C(=O)NCC1CCC1NC(=O)CCC1OCCO1 c1(NC(=O)Nc2c(CNC(=O)OC(C)(C)C)nco2)ccc2c(c1)C(=O)CCN2 C(=O)(N=c1[nH]c(Cl)ncc1C)c1ccccc1NC(CC(C(C)C)OCC#C)=O Cc1c(-c2nc(C3CC3)nn2CCC2CC2)sc2ncc([N+](=O)[O-])cc12 c1(N2C(C(=O)Nc3cccc(OC)c3Cl)CC3CC32)ncnc2ncc(Br)cc12 N1(C(CC(C(=O)C(C(C)C)NS(C)(=O)=O)=O)=O)CCCN(C(=O)CCNCC)CC1.CCN Cc1nc(-c2ccc(C(C)NC(C3CC3c3cccc(F)c3)=O)cc2)sc1CO CCCCCC(O)Cc1nc(-c2cccc(OCCOC)c2)nn1CCS(N)(=O)=O c1(CC)ccc(C(=O)N(C)CC2CCCN(C(C3C4(CC4)C34CC4)=O)C2)cc1 C1(CNC(C2CN(C)C2)=O)CN(C(c2cccc(N3CCCC3)n2)=O)C(C)(C)C1 S(=O)(=O)(c1cnc2ccccn12)Nc1cccc(S(CC)=O)c1 C1(CNC(CCC(CC)=O)=O)CCC2(CN(C(c3cncc(OC)c3)=O)C2)O1 Cc1ccn(C)c(=O)c1NC(=O)C(O)C1CN(C(C2CCCC2C(C)C)=O)C1 C1(CC)(NC(=O)COC(C2CCCC2)C)CCCN(C(=O)CCc2ncccn2)C1 Cc1csc(C=CC(=O)NC(C)CNC(=O)COC2CCOC2)n1 Cc1ccn2c(C(N3CCC(C)(NC(=O)CC(=O)NC4CC4)C3)=O)cnc2c1 C#Cc1c[nH]nc1C(N1CCCC(NC(C2SCCS2)=O)C1)=O c1(CCN2CCCC(CC(=O)OCC)CC2)nc2cccnc2[nH]1 CCC(CNC(=O)CN(C(=O)C(C)CSC)CCOC)(CC)CC c1(C(N2CC(OCCNC(=O)C3=CCCOC3)C2)=O)cnc2ccncc2c1 N12CCCC(C1)c1ncc(s1)CNC(=O)C2C1CCC1.C(CC(=O)OC)OC c1(C(N2CC(NC(=O)C=Cc3nccs3)C3C2C3)=O)c(Br)nc2n1CCCC2 c1(C(=O)NCCC2(C(=O)NC3C(C)(O)CCC3)CC2)ccc2cccnn12 c1(N(C(c2ccccn2)C)C(=O)NC(C)CO)cccc(OC(C)C)c1 C(CNC(=O)CC1CC(F)(F)C1)(C(C)C(C)C)NC(Cc1cc(C(C)C)no1)=O c1(CC)cccc(C(=O)NC2CCCC(CO)C2)c1.C12(CCC1)CC(=O)N(C)C2 c1(CC)ccc(F)c(C(=O)NC(C)CCCNC(c2cncc(OC)c2C)=O)c1 c1(C(N2CCC(CCCCNC(C(C=C)O)=O)CC2)=O)cc(N)ccc1Cl c1(C(=O)NCC(CC=C)NC(c2cc(C)[nH]n2)=O)cc2ccsc2s1 C1(N(Cc2n(C)cnc2)CC2CCCCC2)CCCN(S(N)(=O)=O)C1 CCC(C)CCCC(=O)N1CC(C(O)C(=O)Nc2cnn(C)c2)C1 Cc1c(Cl)ccc2c1CN(c1nccc(=NCCCN3CCOCC3)[nH]1)CC2 N1(C(C2CCC(C(=O)OC)C2)=O)CCC2(CCN(Cc3cc(Br)ccc3F)C2)C1 CC(C)(C)CCC(F)C(=O)N1CCCOC(CNC(=O)CC2CC(=O)C2)C1 c1(C(C)=O)c[nH]c(CSCCCc2ncnn2C)c1C CC(C(C)(C)C(=O)N(C)CCC1CCCN1C)NC(c1ccsc1Cl)=O CCCC(C(O)C(=O)N1CC(n2cc(CO)nn2)CO1)NC(c1cccnc1)=O N1(C(C(C)(C)OCC)=O)C2CCC1CN(C(c1n[nH]c(C)c1F)=O)CC2 C1(CNC(C(COC)(C)C)=O)CC2CCC1N2C(c1cnsc1)=O Cc1nc(N2CC3CC2(CN2C(C(=O)NC(C)C)CCCC2)C3)c2c[nH]nc2n1 CC1CN(C(C2(Cl)CC23CCC3)=O)CCN1C(C1CC2(CC2)CO1)=O C1(C(=O)NC2C(NC(c3ccc(F)s3)=O)CCOC2)Cc2cccnc2C1 c1(C(N(C2CCCC2)CC(C)C)=O)cnc(CNC(=O)CC2CCC(C)O2)nc1 C1(C)(C(=O)NC(CN(C(=O)COCCOC)CC)C)CSC1 N1(C(C(F)=CC)=O)CC2CCCC1C2CNC(=O)CCc1cnn(C)c1 C(c1cc(Cl)cc(Cl)c1)=CC(=O)NC1(CNC(=O)NC2CCCCCC2)CCC1 C#Cc1ccc(C(=O)NC2CCCN(C(=O)C3=NOC(C)C3)CC2)cc1Cl Cc1nc2ncnn2cc1C(=O)NC1CC(C)(NC(=O)CN2CCCCC2C)C1 Cc1cccc(C(=O)NC(C)(C)C(=O)NCC2CCN(C3CC3)C2)c1C#N N1(C(CCCNC(=O)OC)=O)CC(CCNC(c2ccsc2Cl)=O)OC(C)C1 Cc1ccccc1C(=O)NCc1cccnc1CNC(=O)CC1CC2CCC1C2 CCCCCCCCCC(CN1CCC(C(F)(F)F)C1)C(C)NC(C)=O N1(C(=O)CC2CC23CC3(F)Cl)CCCNC(c2ccccc2)C1 c1(NC(=O)CNC(C2CC2CNC2CCCCC2)=O)cc(O)nc(O)n1 c1(OC)cc(CC(N2CCCCC2CNC(=O)CC23CCCC2C3)=O)ccc1O c1(CC)c(C(=O)NCC2N(C(c3csc(C4CC4)c3)=O)CC2)ccn1C C1(CCCC(=O)N(C)CC2(CNC(c3c(C)scc3)=O)CC2)CCCC(=O)N1 C(c1cnn(C)c1)=CC(=O)NCC(CC)(C)NC(=O)C(C)Sc1ccc(F)cc1 c1(C(N2CCC(N(C)C(c3cnn(C)c3)=O)C2)=O)nc2ccc(Cl)nn2n1 c1(N2CCC(C(=O)Sc3ccccc3)C2)cnc(CNC(c2c(C)ccs2)=O)cn1 Cc1cccn2c(=O)c(C(=O)NC3CC(CNC(C4C=CCCC4)=O)C3)cnc12 c1(C(N(CCN(C(C(CCC)C)=O)C)C)=O)sc(Cl)c(Cl)c1N c1(C(N(C2CCN(C(=O)CC3CCC(F)(F)C3)CC2)CC#C)=O)cc(=N)[nH]n1C Cn1cc(C(N2CCC(N(c3ccc([N+](=O)[O-])cc3)C3CC3)C2)=O)c(=O)c(Br)c1 C(=O)(CCCCSC)NCc1c(C(N2C(CC)CC2)=O)cco1 C1(C(=O)NC(CNC(=O)CCCC2CC2)C2CC2)CCS(=O)(=O)CC1 C1(NC(C(Cn2cncn2)NC(c2c(C)nc(C)s2)=O)=O)CC2(CCC2)C1O c1(CCC(N2CCC(NC(c3[nH]n(C)c(=O)n3)=O)(CF)C2)=O)nnc(S)nc1O N1(C(c2c(CC)nco2)=O)CC(NC(=O)CCn2ccnc2C)CC(O)C1 C1(c2nnnn2Cc2ccco2)(N(C)Cc2nnc(Br)s2)CCCC1OC(C)(C)C N1(C(C2CCC2)=O)CCCC1C(N1CC(c2ccc(Br)s2)C1)=O C(=O)(C(F)C(C)C(F)(F)F)NC(CC)CNC(=O)C=Cc1ccc(Cl)s1 C1(NC(CC=CC=C)=O)CCCCCC1C(N1CC(C(N)=O)C2(CC2)C1)=O c1(C(N2C(CC(=O)N(CCOC)CC)CCCC2)=O)c(-n2cccn2)cccc1F C1(NC(c2cccc(OC)c2)=O)CC1C1CCCN(c2nnc(CO)s2)C1 C(=O)(C1CCc2scnc21)N1C(C)CCC(C(=O)NCC2CCCSC2)C1 C12(C(=O)NCC(CNC(C3(n4ncc(C#N)c4)CC3)=O)F)CCC(F)(CC1)C2 c1(C(N2CCCC(N(C(C3CC3F)=O)CC)C2)=O)c(F)cncc1Br N1(C(c2ccc(C3(C)CC3)cc2)=O)CCN(C(C2CCCC(C#N)C2)=O)C2CC12 c1(CC(=O)NC2C(C)CCN(C(CSCCOC)=O)C2)cc(F)c(N)cc1F C(CCCC(=O)NCCCCc1cn(CC(N)=O)nn1)OC C12(C)CCCCC1N2.c1(OC(C)C)cccnc1N1CCCCC1 N1(C(C2(CC)CC2(F)F)=O)CC2(CCCCN2C(C2(OC)CCCC2)=O)C1 N1(C(c2occ(C)c2)=O)CC(NC(c2c(C)coc2C(C)(C)C)=O)CC(F)C1 c1(CN(C)C(=O)NC2CC3CCCC3C2)c(Br)nn(C)c1Br N1(C(c2ccc(-c3ccco3)s2)=O)CCC2(C1)CN(C(c1snc(O)c1Cl)=O)C2 CCCC(C)(C)CC(=O)NC1(CCNC(c2nccn3cnnc23)=O)CC1 N1(C(CC2CCCC(OC)C2)=O)CC2CCCC(C1)N2C(C1(C)CC=CC1)=O c1(OCC)cc(NCC2CCC(NC(=O)C(F)C(C)(C)O)C2)nc(OC)n1 c1(CC)cc(C)[nH]c(=NCC2(F)CC(NC(c3cccc4nc[nH]c34)=O)C2)n1 c1(C(C)=O)cc(=NCC2CCCN2C(=O)C(F)=C(C)C2CC2)[nH]cn1 C(=O)(CC1=CCOCC1)N(CCNC(c1cc2ncccn2n1)=O)C1CC1 C1(C(N2CCC(C(C)NC(c3cnc(C(F)(F)F)o3)=O)C2)=O)CC2(CCC2)CO1 CC(C)(C)C(CNC(=O)CC1(O)CCOC1)C(=O)NCC(C)(O)CO c1(C(=O)NC2CCC2NC(c2ccccn2)=O)cccc2ccnn12 C1(CC)CN(C(=O)CC2CCCCC2NC(=O)CC2(C)CCCC2)CCO1 C1(NC(c2c(CC)oc(C)c2)=O)CC2(CCN(C(C3(n4cnnn4)CC3)=O)C2)C1 Cc1cccc(C)c1OCCC(=O)NCC=CCNC(=O)CC(C)C1CCCO1 C1(C(=O)NC(CNC(c2cc(CC)sn2)=O)CC)CCCC(CC(F)(F)F)C1 c1(CC(N2CCCC(NC(C(CCOC)C)=O)C2C)=O)cccc2c1OCCO2 N1(C(C2CCCC23CCC3)=O)CC2(CCC(NC(C3(Cl)CC3(F)F)=O)CC2)C1 N1(C(CCOCCC)=O)CC(CO)C2(C1)CN(C(=O)CCn1nc(C)nc1C)C2 C1(CN(C(CCC=C)=O)CC)CCCC(NC(=O)CCOc2cncc(F)c2)C1 CC1CN(C(C2CSCCN2C(c2ccc(CO)nc2)=O)=O)CCCO1 C1(C)(C(N2CCC(OCC=C)C2)=O)CN(C(c2ncccn2)=O)C(C)(C)C1 C1(N)CCC2CC1CO2.c1(C(=O)NCC(CC2CN(C(C)=O)C2)(C)C)c[nH]n(Br)c1=O CC(C)(C)C(CNC(=O)C=Cc1ccoc1)NC(c1cnc(C2CCC2)s1)=O c1(C(C)NC(C2CCCC2)CNC(=O)OC(C)(C)C)ccccc1C N1(C(C(C(C)C)NC(c2cccs2)=O)=O)CC2CN(C(=O)CSC3CC3)CCC12 C1(NC(C(CC=CC)NC(=O)CCC(N)=O)=O)(CO)CC2CCCC12 C(=O)(CCCCCCCCCO)N(C)CC1(NC(c2oc(C)c(CO)c2)=O)CC1 Cc1[nH]c(C)c(C(=O)N(CCCCCNC(C2CC(=O)CCO2)=O)C)c1C c1(C(=O)NC2CCC(NC(=O)C3=CCC3)C2)c(OCF)cccc1F c1(-n2cc(C(C)N(C)C(C3CC3(Br)Br)=O)nn2)ccc(F)nc1 c1(C(N2CC(CO)C3CC23)=O)nc2n(c1Cl)CCCC2.C12(CCCCC1)C(=O)N2 c1(C(=O)NCC2CC(NC(c3ccc(N)cc3F)=O)C2)cc2c(nn1)CCCO2 C1(C(=O)NCC(C(C)C)(C)NC(c2cc(Cl)ccc2Cl)=O)CCC2(CCCC2)C1 N1(CC2CC(C)C2)C(=O)NC(c2cc3cccc(Cl)c3o2)C2=C1C(C(C)C)OC2=O c1(C(C)NC(=O)C(=O)NC(c2nccn2C)CO)ccc(C(F)(F)F)c(Cl)c1 C12(C(N3CC(c4c(C)n(C)nc4)C(CO)C3)=O)CC3CC(C1)CC(O)(C3)C2 C1(C(N(C)C)=O)CCCC(NC(N2CCC(CC(O)C(F)(F)F)CC2)=O)C1 C(C)(C)(C(=O)NC1CC(C(=O)NC2CCC(CC(=O)OC)C2)C1)OCCC C1(OCC)CC(N(C(=O)C(CCCCC=C[Si](C)(C)C)OCC)C)C12CCCC2 c1(OCCCC(=O)NCC(C2CC2)NC(C2CC2C2CCCO2)=O)cccc(F)c1 c1(C(=O)NC(CN(C(=O)CC(O)C2CCCC2)CC)C)ncc(C)cc1Br CC1(C)CN(C(c2cc(O)nc(O)n2)=O)CC1C(N1CC(F)(F)C1)=O c1(C(=O)NCC(C)(CNC(=O)C(O)C2CCCC2)OC)ccn2nccc2c1 c1(C(=O)NC(CC)CNC(C2CC(F)(CO)C2)=O)ncc(F)c2ccccc12 CCCC(C(=O)OC)C(=O)N(CC(C)(C)C(=O)N(C1CCCC(C)C1)C)C Cc1nnc2n1CC(C(=O)NC1CCSC13CN(C(=O)COCC(C)C)C3)CC2 C(C(F)(C(=O)N(C1CCNC1=O)C)C(C)C)NC(CSCCCC)=O N1(C(N2CCOCC2NS(=O)(=O)c2cccc(F)c2)=O)C2CCC1CCCCC2 C(=O)(C(F)(CNC(C1CSCCS1)=O)C(C)C)NCCc1c(C)n[nH]c1 c1(CN(C)C)ccccc1NC(=O)C(F)Cc1ccccc1 C1(NC(C2(CO)CCN(C(CC3N(C)CC=CC3)=O)C2)=O)CCC(=O)N(C)C1=O CCCC(CCCNC(=O)C(C)Cc1c(C)n[nH]c1C)NC(c1ccsc1C)=O c1(C(=O)NC2C(CNC(C3(C(N(C)C)=O)CC3)=O)CC2)cncc(C(N)=O)c1 CCC(COC)(CC)C(=O)NCC1CCCC1OCC(=O)Oc1ccccc1F c1(CC)cccnc1Cl.C1(N2C(=O)NC(C)c3nocc3C2)CCCSCC1 N1(C(C2C(OCC)C2)=O)CCOC(C(C)NC(=O)CCCc2cnccn2)C1 c1(CNC(C(CCCC)(C)F)=O)cccc2c1CCN(C(=O)CC1(C#N)CC1)C2 N(C(=NCC1CCC1)NCC1(C(F)(F)F)CC1)CC1CCCCC1 C(=O)(C1CCc2c(Br)cccc21)NC1CC(NC(C=CC(C)(C)SC)=O)C1 CCCCC(C)(F)C(=O)NCC=CCNC(=O)C(C1CCC1)OC N1(C(c2cc(-c3ccncc3)no2)=O)CC2CC1CN2C(C1(O)CC(F)(F)C1)=O C1(NC(C=C(C)C(C)(C)C)=O)CCC2(CCCN(C(=O)CCCF)C2)C1 Cc1cc(O)c(C(N2CC3C(CNC(=O)Cc4csc(C)n4)C3C2)=O)nn1 c1(CC(=O)NCCN(C(C2CCC(COC)C2)=O)C)ccc(F)c(Cl)c1F CC1CN(C(=O)CN2CCC2)CC(C)N(C(=O)CCc2cn(C)nn2)C1 C(=O)(C(C)CCCC(C)C)N1CCCC(F)(C(=O)NC(CC(=C)C)C(=O)OC)C1 C(=O)(C(CC)(CC)CC(=O)OC)NC1CCN(C(C(CC)OC)=O)C12CCC2 N1(C(C2C(C)=CCS2)=O)CCN(C(c2nn(C)cc2Cl)=O)CC1C C1(OC)(OC)CC(C)(C(=O)NCC(C(C)C)NC(=O)Cc2ccccc2O)C1 c1(C(=O)NC2(CC=C)CN(C(=O)C(C)(CC)C(N)=O)C2)ccc2c(ccn2C)c1 C12(C(=O)NCC3C(OC)CC3)COC(CC(=O)OC(C)(C)C)(C1)C2 C(C(CC(F)(F)F)NC(=O)CN(C)C(C)C)NC(C1C(=C)C1)=O C1(NC(C2CN(C(C)=O)C2)=O)CCC(C)N(C(C2CCOC2(C)C)=O)C1 C(C)(N=c1cc(C)nc(NCC2(C)CC2)[nH]1)C1CCN(C(COC)(C)C)CC1 C1(CNC(=O)C=CC(=O)NC2CC2)CC(F)(NC(=O)COC2CC2(F)F)C1 c1(C(=O)OCC)ccc(C(=O)NCc2ccc(N3CCOCC3)cc2)cc1 n1(CCC(=O)NC2CN(C(C3CC3CF)=O)C2)ccc2cc(Cl)ccc12 c1(C(=O)O)ccc(S(=O)(=O)N=c2sc3ccccc3cc2Cl)cc1 C1(C2CCCCC2)(C(=O)NCCCCC2CN(C(C=CC)=O)C2)CCCC1 c1(NC(C2CCCCC2c2cccc(F)c2)=O)ccc(F)cc1F N1(C(CNC(C(n2c(C)ccn2)C)=O)=O)CCN(C(=O)CC(C)(C)C)CC1 c1(C(N2CCCC(CNC(CC3CC(=C)C3)=O)C2)=O)n[nH]c2c(OC)cccc12 C(=O)(C1CCC(=O)c2ccccc21)NCC1N(c2ncc(C#N)o2)CCOC1 C1(SCC)=CC=C(NC(C2C(C)CCN2C(c2csc(COC)c2)=O)=O)C=CCC1 C1(CC(=O)NCCOCCNC(c2n(C(C)C)ccn2)=O)CCC=CCC1 C1(C2CCCN(C(c3noc4c3COCC4)=O)C2)(NC(C2CC3CC2C3)=O)CC1 c1(C(N2CCCC2CC#N)C(=O)NCCCC)cnc(Cl)c(C)c1 N1(C(C(C)n2cncn2)=O)CC2CCC1C(CNC(c1ccc(C3CC3)s1)=O)C2 C1(NC(C(C)=C(C)C)=O)C2CC3CN(C(=O)C(C)NC(=O)CC4C=CCC4)C1C3C2 C1(C(CC)(C)C)CCCN(CC(=O)N(C)Cc2ccccc2Cl)C1 C(=O)(CC(O)C(C)C)NC1(CCNC(c2nc(C(C)OC)oc2)=O)CCC1 C1(C(=O)NC2CC(C)(NC(=O)CC3CCC(F)(F)CC3)C2)COCC2(CCC2)O1 Cc1c(CCC(N2CC(C(C(=O)C(=O)C(C)(Cl)Cl)C(C)C)(O)C2)=O)cnn1C.C(C)N c1(CC)sc(C(=O)NC2CCCC2NC(C2CC(OC3CC3)C2)=O)cc1C C1(C(=O)NCC(O)CCNC(C2CCCS2)=O)CC2(CSC2)C1 C1(CC(=O)N(C2CCC(N)C2)C)CCCN(C(C2CCCO2)=O)C1 O(NS(=O)(=O)Cc1cn(CCN)nn1)C(C)C CCC(C(=O)N1CCOCC1)NC(N)=O.C1(c2ccoc2)C(=O)N1 C1(C(=O)NC2CC(NC(CS(=O)(=O)NC(C)(C)C)=O)C2)CC12CCCOC2 C1(C(=O)O)(C(N2CCCC(C(N3CCCCC3)=O)C2)=O)CC2CCC1CC2 N1(C(C(=O)NCC(CC)NC(=O)CS(=O)CC)C)CCc2ccccc21 c1(C(=O)NC(C)CNC(=O)Cc2cn(C)nn2)cc2ccc(C(C)(C)C)cc2[nH]1 N1(C(=O)NCc2c(OC)c(Cl)ccc2)CCC2CS(=O)(=O)CC2C1 c1(C(=O)NCC(C)NC(C2(CN(C)C)CCC2)=O)coc(C(C)(C)C)n1 c1(OC)cc(NC(c2ccccc2-c2nccs2)=O)c(F)c(Cl)c1 C1(C2CN(C(=O)Cc3cccc(F)c3Cl)C2)(NC(CSCC#C)=O)CC1 N1(C(C2=C(C)CCCC2)=O)CCC(C2(O)CN(C(=O)C(C3CCCC3)NC)C2)CC1 c1(CNCC2N(C(c3ncc(C)c(Br)c3)=O)CCOC2)cccc2c1CCC2 Cc1ccsc1-c1cn(CC2CCCN2C(c2c[nH]cc2C2CC2)=O)nn1 Cc1cc2c(C(=O)NCC34CC(CN3C(C3(C)CC3(Cl)Cl)=O)C4)nccn2n1 Cc1cc(C(=O)N(CCNC(C2(C3CC3)CCC2)=O)C2CC2)c(F)cc1Cl S1(=O)(=O)c2ccc(c(F)c2)NCC(C)CN1C.Cc1ccccc1C(C)N(C)C CC(C)CCC(C(=O)N(C)CCOC1CC1)NC(=O)C#CC1CC1 c1(C(N2CCCC(C(C)NC(C(F)=CC)=O)C2)=O)noc2cc(Cl)ccc12 N1(C(CCC(C)O)=O)CC2(CC2)CC1CNC(c1ccccc1F)=O C1(O)(C(C)C)CCN(C(C2(CNC(C3CCCO3)=O)CCCO2)=O)C1 N12CCC(CC1)NC(=O)NC(=O)C2C.c1(NC(c2sccc2Cl)=O)ccccc1 C(C(O)C(=O)N=c1ccn(C2(C(N)=O)CC2)[nH]1)NC(C(c1cnc(C)o1)C)=O c1(C(N2CCCCC2CO)C(=O)NCCN2CCCC2)csc2ccc(Br)cc12.CSC CC(C)P(=O)(CC(=O)NCC(C)CNC(=O)C(O)CCc1ccccc1)C(C)C Cc1nc(N(CC(F)(F)F)CCC#N)c2cc(-c3ccccc3)sc2n1.C C1(C(=O)NC(C(=O)NCCN2CCOC2=O)C2(O)CCC2)CC12CC2(F)F c1(OC)cc(-c2cnoc2)ccc1C(C1CC1)N.c12cccc(c1)C2 c1(CSC)ccc(C(=O)NCCN(C(=O)C(C2CCCO2)OC)C(C)C)cc1 n1(CC)nc(C(N2CCOC(C(=O)NC(C)C(C)(C)OC)C2)=O)cc1O CC(CC(=O)N1CCC(N(C)C(c2cccc3c2COC3)=O)C1)C(C)(C)C c1(C(=O)Nc2cccc(NC(C3CCC4CC34)=O)c2)cccc2c1CCCC2=O c1(C(=O)NCC(C)(C)NC(=O)CCc2nc(C(F)(F)F)n[nH]2)csc(F)c1 C1(C(N(CCCOCCC(=O)Nc2cnco2)C2CC2)=O)CCCC1O CCC(CC)C(C(=O)NCC1(F)CC(NC(=O)C(C)CCC)C1)OC C(C(=O)OC)(C1=CCCCC1)N(C(CCOC)C(=O)NCc1ccccc1Br)C N1(Cc2n(NC(C(c3nnn(C)n3)C)=O)nnn2)CCOC(C(F)(F)F)C1 C1(NC(c2ccn(CC)n2)=O)C=CCN(C(C2COC(=O)O2)=O)C1 C1(C(=O)NCC2CCCCC2CNC(=O)CN2CSCC2=O)(CC)CC(C)(C)C1 C1(N(C(C=C(CC)C)=O)C)CCCCN(C(c2ccc(C)cc2C)=O)C1 C1(NC(c2cc(CC)oc2C)=O)CN(C(=O)CCNC(=O)COC)CCC1CO C12(CNC(CC3(CC)CCC3)=O)CCC(CC1NC(c1ccc(C)s1)=O)C2 Cc1onc(CC(C(=O)CO)=O)c1C#N.C(=O)(C(F)OC(F)(F)F)NCCCN C1(C(=O)NCCCOCCC(N2CC(C)(CC)C2)=O)CCN(CCO)CC1 C1(CNC(C2(OC)CCC2)=O)CCC2(CN(C(=O)Cc3cnccc3C)C2)O1 N1(C(c2c(C)cco2)=O)CCC2CCCC12C(=O)NCc1nnn(C)n1 C(=O)(C(CC(=O)NCC1CC(C)CCN1C(=O)CCSCC)C(C)=O)OCC C12(C(N3CCC(C(C)(C)NC(C(COC)C)=O)CC3)=O)CCCCC1OCC2 C1(C)(N(C(=O)NC(C)Cc2ccnn2C)C)CCS(=O)(=O)C1 c1(C(N2CC3C(CNC(c4scc(COC)c4)=O)(C3)C2)=O)nc(C)ncc1Cl c1(C(C)C)cccc(OCC(=O)NC2COCCC2NC(=O)C(O)C2CC2)c1 C1(CC(=O)NCCC(C)N(C)C(c2sccc2CN(C)C)=O)C=NN(C)C1=O CCC(CCCC(=O)N1CC(C(F)(F)F)C1)N(C(=O)CCC(CC)OC)CC c1(OC)ccc([N+](=O)[O-])cc1.C1(=O)C(C2CCCC2)NCCN(C)CCC(=O)N1 C(C(O)CC(=O)NC(C12CCC(CC1)C2)CNC(C1CCCOC1)=O)N(C)C c1(C(N2CCCC(C)(NC(CC(CC)C(F)F)=O)C2)=O)cc2n(n1)CC1(CC1)C2 c1(C(N(C)CC2N(C(C3CCCCC3)C)CCC2)=O)cc2c(Cl)cc(F)cc2[nH]1 C1(C(=O)NCC2CC2CN)(C)CCCO1.C1(Cl)(C(=O)OC(C)(C)C)CC1(F)F c1(C(N2CC(C)N(CCO)C(C)C2)C(=O)NC)ccc2cncn2c1 C(=O)(C(F)(CNC(=O)CCC1CCOCC1)C(C)C)N1CCCC(CC)(CO)C1 c1(C(N2CCC(NC(C3CCC(OC)CC3)=O)(CO)C2)=O)cccc(S(C)=O)c1 C1(C(=O)NCC2CCN(C(C(CSC)C)=O)C2)CCN(C(N)=O)CC1 C(=O)(CCCC(=O)NCc1cc[nH]c1C(=O)NCC(N1CCCCC1)C1CC1)OCC c1(CC)cc(C(=O)N(CC(=O)N(C)CC2CCOC2)C(C)C)c(C)o1 c1(C(N2CCC(CN(C(C(CC#C)O)=O)C)C2)=O)cnc(O)c(F)c1 n1(CC(=O)OC(C)C)cc(NC(C(F)(F)F)C2CCOC2)cn1 N1(C(C(CC)=CC)=O)CC2=C(C1)CN(C(C1CCCN1N=O)=O)C2 N1(C(c2cc(C)sn2)=O)CCC(NC(c2cc(C(F)(F)F)cn2C)=O)CC(O)C1 N1(C(c2c(C(C)C)nns2)=O)CCC(NC(C2(C)CSC2)=O)CC(C)(C)C1 N1(c2n(CC)c(N3CC(C)(C)C34CC4)nn2)CCCC(O)(C(F)(F)F)C1 C1(NC(=O)CSc2cccc(Br)c2)CNC2(CCSCC2)C1 N1(C(c2c(CC)non2)=O)CCC(C(C)CNC(c2nnc(S)n2C)=O)CC1 C=CCC(C(=O)N1CCCC1CNC(=O)Cc1nocc1CC)C(C)(C)C N1(C(c2cc(C)[nH]c2C)=O)CC2(CCC2NC(=O)CN2CCOC2=O)C1 c1(C(C)CC=O)cc(F)cc(F)c1.C1(CC)CCN(C(=O)COc2ccon2)C1 Cc1ccncc1CC(=O)N(C(C)C(=O)NC=Cc1ccccc1)C1CCCC1 CCC(CC)(CC(=O)OC)C(=O)NCCC(C)NC(=O)CCCCc1cnn[nH]1 N1(C(C(CC=C)CNC(c2cccc(C#N)c2C)=O)=O)CC2(CCC(=O)O2)C1 c1(-n2cc(CCN(CC(C)C#N)CCC)nn2)cccc(Br)c1Cl c1(CCNC(N2C(C(=O)OC)CCC(O)C2)=O)cnc2n1CCCC2 Cc1nnnn1CC(=O)N(C(C1CCC1)=O)CC1(F)CC(NC(=O)CSC2CC2)C1 C1(CNC(C2CCCC2(C)C)c2n(CCCOC)nnn2)CCCC2(CCC2)O1 C1(CNC(c2ccc(C)c(F)c2)=O)CN(C(=O)CC2CC2C2CC2)CC(C)(C)O1 c1(CN2CC3C(NC(C4CC(=O)NC4)=O)(C3)C2)cc(Cl)cc(Cl)c1 CC1(C)OCc2c1n[nH]c2C(=O)NC12CC1CN(C(c1nnc(Cl)cc1N)=O)C2 CC(C)(C)C(O)CCC(=O)NC1CCCN(C(C2CCCC2(C)C)=O)CCC1 c1(N2CCOCC(C(=O)NCCCCO)C2)nn2cc(-c3ccco3)nc2s1 C1(C(N2CC(O)(CNC(=O)CCC3NC(=O)NC3=O)C2)=O)OC2CCC1CC2 C1(C(=O)Nc2c(CC)scc2)CC(F)(F)CN1C(=O)C(c1ccoc1)OC C#CCC(CC(=O)NCc1ccns1)NC(C12CCC(CC1)C2)=O C(CCC1CCC1)(C(=O)N(CC(O)CF)C)NC(C1C(C)=CCS1)=O C1(CC(=O)NCCC(CNC(C(C)=CC2CC2)=O)O)CCCC(=O)N1 N1(C(C=Cc2n(C)ccc2)=O)CC2CC(NC(c3ccc(C(F)F)cc3)=O)C1C2 C(=O)(C1=C(C)OCCS1)NC(C(=O)N(C(C(=O)OC)C)C)CCOCCO c1(NC(C23C(CN(C(CSC)=O)C2)C3)=O)c(Br)cc(Br)c(C)c1Br C1(CC)(NC(c2nc(-c3ccccn3)cs2)=O)CC(C)(C)C1 Cn1cnc(C=CC(N2CCC2CNC(C2(CC(F)F)CC2)=O)=O)c1 C12CCc3nc(ncc3C1)C(=O)N2.O=C(CCCn1cccn1)NC1CC1.C1CC1 C1(CNC(c2c(C)n(C)nc2)=O)CCC2(CO1)CC(NC(=O)C=CCF)C2 c1(C(=O)NC(C(N2C(C)CCC2)=O)CO)ccc(C#N)n1C Cc1ccnnc1C(=O)NCC#CC(=O)NCCCS(C)=O C1(CC(=O)NCC2CCC(F)(CNC(=O)CC3(CO)CC3)C2)CCCS1(=O)=O c1(CC)ccc2c(Cl)c(C(=O)NCCCNC(=O)C3=C(C)S(=O)(=O)CC3)sc2c1 C(=O)(C#CC1(C)CC1)NCC1(C)CCC(NC(Cc2cc(COC)on2)=O)C1 C=CC(CC)CC(=O)N(C1CCN(C(c2ccn(C(F)F)n2)=O)C1)CCC CCCCC(CNC(C1(C)CCC(=O)N1)=O)NC(c1cc(C)c(CC)s1)=O c1(OC)cc(Cl)cc(Cl)c1NC(C1C(O)CCN1C(c1cccc(Br)n1)=O)=O c1(C(=O)NCC(=O)OC(C)(C)C)ccc(C#N)c(Cl)c1F c1(C(=O)NCC2(CO)CCN(C(CCC(=C)C)=O)CC2)cnc2c(c1)ncn2C C(=O)(CC(C)(O)C=C)N(CCC(=O)NC(C1CCOCC1)C)CC#C C12(NC(c3cc(C)[nH]c3)=O)CCCC1CN(C(c1ccc(CO)nc1)=O)C2 Cc1nnc2cc(N3CCC(CNC(=O)C(c4ccc(F)c(F)c4)O)C3)ncn12 C(=O)(CCCCCF)NC1CC(C)(NC(c2ccc(C)nn2)=O)C1 Cc1cccnc1CCNC(CC(C)(C1CC1)NC(=O)CP(C)(C)=O)=O C12(COC)CC(C(N)=O)(CO1)C2.c12cn(nn1)C2.C12CC(C1)CC(=O)N2 C1(C(N(C(C(C)C)C)C)=O)CN(C)CCN1C(=O)C#CC1CC1 N1(C(C=C(C)CNC(C2(Br)CC2)=O)=O)CCOC(C(C)O)C1 c1(C(=O)NCCC(C)NC(c2cccnc2)=O)cccc(-c2cc[nH]n2)c1 C1(C(=O)OC(C)(C)C)CC(C(=O)OC)CN(C(=O)Cc2cnoc2)C1 C(=O)(CC(CC=C)NC(C1CCCC(=O)CC1)=O)NCCCC#C C(CCCCCC(=O)NCCc1ccccc1C)NC(C1(C(=O)OC)CC1)=O c1(C(=O)NC(C2CCCC2)CNC(CS(C)(=O)=O)=O)cc2scc(Cl)c2[nH]1 C1(COc2ccc(C(c3n(CC)nnn3)NC3(C)CC#CC3)cc2)CCCC1(C)C C1(C(=O)NC2(CN(C(=O)CC3CC4(CC4)CO3)C)CC2)CCc2nnnn2CC1 c1(C(N2CCC(O)(CNC(=O)C(F)(F)CC3CC3)C2)=O)cc(Cl)cc(Cl)c1 C1(C)(C(=O)NC2(CC=C)CN(C(=O)C3=CCCC3(C)C)C2)C2CC3CC(C2)CC1C3 C1(CC)(NC(=O)Cn2nnc(C)n2)CCN(C(c2ccc(C(F)F)cc2)=O)CC1 C=CCC(CC(F)F)C(=O)N1CCC1CNC(=O)C=CSC CC(C)CC(CS(C)(=O)=O)NC(=O)C(N1CCCC(CF)C1)=O C12(C(N3C(C4(NC(Cc5cn(C)nc5)=O)CC4)CCC3)=O)CCCC(C)(C1)OC2 c1(C(NOCC(C=C)C2CCCC2)=O)ccc([N+](=O)[O-])cc1[N+](=O)[O-] N1(C(COCCCOC)=O)CCC(NC(C2(C(=O)O)CC=CC2)=O)C(C(N)=O)C1 c1(CC)ncncc1NC(C1(CC)CN(C(C2CC(O)C2)=O)C1)=O N1(C(C(CCCNC(C(C(=O)NC)(C)C)=O)O)=O)CCC(C)(CO)CC1 C1(C(=O)NCC2CC(F)(CNC(C(C)OCCC#C)=O)C2)CC(=O)NC(=O)C1 Cc1ccc2oc(NC3(CNC(c4ccc(F)c(Cl)c4F)=O)CC3)nc2c1 C1(C(N2CC(C(C)NC(C3(CC4CCC4)CCC3)=O)C2)=O)(CC)CCNC1=O Cc1ccc(C(=O)NC2CCOC2C(=O)NOCC(C)(C)O)[nH]1 c1(NC2C(CCCC)C2)ncc(S(=O)(=O)N2CCCC(n3cccn3)C2)cc1Cl C1(C(=O)NC(c2ccc(C(C)C)cc2)C(=O)O)OCCN2CCOCC12 C1(NC(=O)NC(CC2(CCCC(=O)OC)CCC2)C2CC2)CCCCCC1C C12(NC(C(C=C=C)C)=O)CCOC(CNC(c3cncc(O)c3)=O)(C1)C2 Cn1cc(OCC(=O)NC2(CCNC(=O)C(O)Cn3cncn3)CCCC2)cn1 c1(NC)cnc(C(N2CC(C)C2C(=O)NCC(C)CCO)=O)cn1 C1(S(C)(=O)=O)(CNC(NCC(=O)N(CC)CC)=NCC(C)C)CCCC1 CCC(COC)C(=O)NCC(O)CNC(c1c(C)coc1C(C)(C)C)=O c1(C(=O)NC2(C)CCN(C(c3n(CC)ccn3)=O)C2)nc[nH]c2ncc(Br)c1-2 C(C(C)C(=O)N1CCC(C(F)C(=O)NC2CCOCC2)C1)OC c1(C(=O)NC2CN(C(C3CC3F)=O)CC2O)ccc(=O)n2c1CCCCC2 C1(C(N(c2c(NC)cc(C)s2)CC)=O)CC(F)CN1C(=O)Nc1ccccc1 c1(-c2nn(-c3nc(C)nn3C)c(C3CC(C)(F)C3)n2)ccc2c(c1)OCO2 c1(C(=O)NCC(n2cc(C(C)OC)nn2)C)ccc2c(c1)C(=O)OCC2 c12cccc(c1)CCC2F.C1(OC)C=CC(CO)C1.C(C)(C)(C)OC(=O)NC(=O)N CC1C(=O)N(CC(=O)NC(C)(CNC(=O)CCCC(F)(F)F)CO)C(=O)C1C c1(OC)cc(C)sc1C(=O)NC1C2CN(C(c3cnn(C)c3Br)=O)CC12 CC1CCCC1(C)NC(=O)C(C1CC1)NC(=O)C(C)N=[N+]=[N-] c1(SC)ccc(C=CC(N2CCCC(NC(c3ccc(=N)[nH]c3)=O)CC2)=O)cc1 C1(C2CCN(C(CCCOCC=C)=O)C2)CCCCN1C(=O)CCC1CC1 CC1C(C(=O)N(CCC2=CCCCC2)C)CCCN1C(C1CC(F)(F)C1)=O C#CCC(CC#C)C(=O)NCC(C)(C)NC(c1ccc(NC)cc1)=O C=CCC(C)C(=O)NCC(C)N(CC(O)COCCc1ccccc1)C N1(C(C2(CSC)CCC2)=O)CC=C(C(=O)N2CCC2)C1 C(=O)(CC(C)(C)C(F)F)N(C)CC1(CNC(=O)CSC2CC2)CC1 c1(OCC)cc(C(=O)NC2CC2CNC(=O)C2=NOCC2)ccc1[N+](=O)[O-] N1(C(C(C)C)=O)CCCC(C2CCN(C(=O)CC3CCC(C)(C)CO3)CC2)CC1 C1(C(NS(CCC)(=O)=O)=O)CCN(C)C(=O)C1.C1(=O)C(=O)NCC2(CCC2)CN1 N1(C(C(C2CCOCC2)OCC)=O)CC(CC)(NC(c2cnnn2C)=O)C1 N1(C(CN(C(C)=O)C)=O)CCC(CC(C)NC(=O)C(C)(C)OC2CCCC2)CC1 C12CCC(C1)CNC2=O.C1(N(C(C(=C)C)=O)CCC)(CNC(C)=O)CCCC1 C1(C(=O)NC(CC)CCOC)CCCCC1(C)NC(=O)CC1CCC(C)CC1 N1(C(C2(CC)CC2)=O)CC2CC1C2NC(c1sc(-c2ccccc2)nc1C)=O C=CCC(CC)C(=O)N1CCC(OCCNC(=O)C=C2CCC(C)C2)CC1 C(C(C)(C)CN=c1cc(NCC2CC(C)OC(C)C2)nc[nH]1)SC Cc1cc(F)cc(C)c1C(N1CC2CC1C2C(=O)NC1CCCCC1)=O c1(CC)ccc(NC(C2CC(OC)CN2C(=O)CSC(C)C)=O)c(Br)c1 Cc1c(C(N2CCCC3(NC(=O)CSC(=N)N)CC3C2)=O)sc2nccn12 c1(C(N2C(C(C)NC(=O)C(C)OCC(F)(F)F)CCC2)=O)nnn(C)c1N c1(C(N2CC(N(C(c3cc(C)cc(C)c3O)=O)C)C2)=O)cc(F)cc2nc[nH]c12 c1(NC(c2ccc(C(=O)OC(c3ccccc3)C)[nH]2)=O)cnc2ccsc2c1 CC1CC(C)N(C(=O)C(Cn2cccn2)NC(C)CCOc2cccnc2)C1 C(CN=c1ccn2ccnc2[nH]1)(c1cccs1)NC(c1c(CC)ocn1)=O N1(C(c2c(C)nns2)=O)CCCN(C(=O)C(C)CCCc2ccccc2)CC1CO n1(CCOC)cc(C(=O)NCC#CCN(C(=O)CNC=O)CCC)c(C)n1 CCCC(C(O)C(=O)N1CCC12CCCSC2)NC(c1cccnc1C)=O CC1CCC(F)(F)CN1C(=O)CCN(C(=O)CC1(C)CCC1)CCO C(C1=NOC2CN(C(=O)Cn3cc(Cl)c(O)nc3=O)CC12)NC(CCCC=C)=O Cc1ncc(C(=O)NCC2CCN2C(=O)CN2CCCCC2)c(C)n1 Cc1cnc(C(=O)NCC2CCC(NC(C3CCN(C)C3)=O)C2)nc1 N1(C(C(CSC)O)=O)CC=C(C(=O)NC(C)CCN(C)C)C1 C12(NC(C(CC3CC3)OC)=O)CCCC1N(c1nnc(-c3ccccc3)s1)CC2 Cc1nc(C)c(C(=O)N(C)CC=CC(=O)NCc2nc(N(C)C)n[nH]2)s1 N1(C(C2(C#N)CC2)=O)CC2CN(C(=O)CCc3ncc[nH]3)CC12 C(=O)(C1CCc2ccccc21)N1C(C)CC(CNC(c2ccc(N)c(N)c2)=O)C1 C1(C(=O)NCC(CCOC)NC(=O)C(SC)SC)CC2(C1)CC21CC1 C1(C(=O)NC(C(C)NC(C(CC=C)OC)=O)C)CC12CCCCC2 Cc1sc(O)nc1C(N1CC2C(NC(c3csc(C4CC4)n3)=O)C2C1)=O N1(C(c2cnc(C)s2)=O)CCC(CNC(C2CC(O)CN2C)=O)CC1 Cc1nc(CN(C(C2CCC(n3cc(-c4ccncc4)nn3)C2)=O)C2CC2)co1 C(C)(CNC(=O)C(C1CCCCC1)N(C)C)(C(C)C)NC(C=C(C)C(C)(C)C)=O C1(CC)CN(C(C(=O)NCCCSC)C2CN(C(C)=O)C2)CC(C)(C)O1 N1(C(C(COC)N(C)C)=O)CC(C(=O)NCC2(C)CC3CC3C2)CC(C)(C)C1 N1(C(c2ccc(C)o2)=O)CC(NC(c2c[nH]nc2[N+](=O)[O-])=O)C2(CCOCC2)C1 C1(CC(NOCC(CC)C)=O)CN(C(C2(CF)CC(=O)C2)=O)CC12CC2 N1(C(c2cccc(OC)c2)=O)CCCN(C(c2ccns2)=O)C(C)C1 n12cc(c(=O)cc1C)OC(C)C(=O)NCCC1(CC1)NC(=O)C2.C#CCOCF c1(C(=O)NCCCCCC)[nH]c2cc(C(N3CC(C)C3(C)C)=O)ccc2c1C c1(CN2CCC(CC(=O)NCC3CCC3)C2)cccc(Br)c1Br c1(C(=O)NCCN(C(c2cncc(OC)n2)=O)CC)cncc(C2CC2)c1 C1(C(N2CCN(C(Cc3c(C)occ3)=O)C(C(C)C)C2)=O)CC2(CCC2)CCO1 c1(C(C)C)ccc(C(C)(C)CN2CC3CC3(NS(=O)(=O)C(F)(F)F)C2)cc1 CC(CCC(C)(C)C)C(=O)NCC1CC(F)CN1C(=O)CC1=CCOCC1 c1(-c2cn(CCC3CCC(CCC)CC3)nn2)cnn2c1NCC2 C1(CC(N2CCC(O)(CNC(c3cnc(OC)nc3)=O)C2)=O)CCC(F)(F)CC1 CC1(C)CCC(C(=O)NCCC2CCOC2)(NC(=O)Cc2cnsc2)C1 C1(NC(c2cnc(C)c(Cl)c2)=O)CCCC12CN(C(c1cn(C)c(=O)n1C)=O)C2 c1(OC)cnc2[nH]c(C(=O)NC3CC(N(C(=O)Cc4nccn4C)C)C3)cc2c1 C1(CNC(CC2CCC(NC(C3(C=C)CCCC3)=O)C2)=O)CCC(F)(F)CC1 N1(C(=O)C2CC2)Cc2cnn(C3CCN(C(=O)C(O)Cc4cnc[nH]4)CC3)c2C1 c1(C(=O)NCC2N(C(C(=O)NCCOC)=O)CCC2(C)C)cc(F)c(F)cc1C c1(C(=O)NCC(C(C)C)NC(C2CCOC2(C)C)=O)cc[n+]([O-])cc1 C1(CCOC)CN(C(=O)CCCC(=O)OC)CCN1C(=O)C(F)=C(C)C C(=O)(C#CC1CCCOC1)NSCCCC(=O)OC(C)(C)C.N12C=CC(=NC(=O)C1)N2 N1(CC(=O)NC2CC(CNC(C3(COC(C)C)CC3)=O)C2)CCCCC1C C12(NC(c3n(C(CC)C)ncc3)=O)CC1CN(C(c1ccc(=N)[nH]n1)=O)C2 C1(=O)C(C)CC(=O)OCCN1CC(C)NC(=O)OC(C)(C)C.CNCC C12(NC(Cn3nnc(C)n3)=O)CCCN(C(C3CC(F)(F)C3)=O)CC1C2 c1(CC(=O)NC(C(C)C)CNC(=O)CN2CCCC2=O)cccc(NC(N)=O)c1 CCC(CC(C)C)C(=O)NCC1CCC1NC(c1cc(S(N)(=O)=O)cs1)=O C1(F)(C(=O)NC2CCN(C(=O)CC3COCCO3)CC2F)CCC(F)(F)CC1 Cc1ccnc(C(=O)NCCN(C(c2ccnc(Cl)c2O)=O)C2CC2)c1N CCCC(C(O)C(=O)NCC1(C)CSC(C)=N1)NC(=O)CC(C)C1CCCC1 N1(C(C#C)=O)CC(C)CN(C(=O)OC)C(C)C1.c12ccnc(n1)NC2(C)C C1(C(C)C)Cc2cnn(C)c2CN1Cc1ccn(C2CCNCC2)n1 c1(CC(N2CCC(C)(CNC(=O)C(c3ccccc3)F)C2)=O)ccc(F)cc1F CC1=C(C)CC(C(=O)NC2CC(C)(NC(=O)C(C)OCCC(C)C)C2)CC1 c1(-n2cc(CC(C(=O)OC)NC(=O)Cc3ccoc3)nn2)ccc(Cl)cc1 C1(O)(CNC(C(C)=O)=O)CCN(C(=O)C(C)SC(F)(F)F)C1 c1(C(=O)NCC(CCC)NC(C2(CC(C)C)CCC2)=O)cnc2[nH]cncc1-2 CC1(C(=O)NCc2c[nH]nc2-c2ccccn2)CCN(C(=O)C(=O)N(C)C)C1 c1(N2CCC(C(N3CCCC3c3ccsc3)=O)C2)ccc(Cl)c(Cl)c1 CCCCCCC(C)C(=O)N1CCCC(N(C(=O)COCP(C)(C)=O)C)CC1 C1(CCCc2nc(-c3csc(-c4ccccn4)n3)no2)CCC(F)(F)CC1.NC=O c1(C(=O)NCC2CC(NC(Cn3c(C)nc(C)n3)=O)C(O)C2)ccc(F)c(N)c1 c1(N2CCC(OC(C)C)C2)nc2c(c(=NCCCC(C)CC)[nH]1)CCCCCC2 C1(NC(c2nn(C)c(F)c2)=O)CC(CNC(c2ccccc2F)=O)C12CCC2 c1(CC(=O)NCC#CCNC(C2(C)CCNC2=O)=O)ccc(F)c(Cl)c1F CC(CNC(=O)C(Cc1ccc(=O)oc1)NC(=O)OC(C)(C)C)S(N)(=O)=O N1(C(Cc2cn(C)nc2)=O)CCC2(C(=O)NC3CC34CCC(=O)CC4)CCCC12 N1(C(=O)CC2CSCCS2)CCc2sccc2C1c1cccs1 C1(C(=O)NC(C(C(C)C)NC(CCN(C)CC)=O)C)CCc2ccccc2CC1 C1(NC(c2scc(C)c2Cl)=O)COC2(CNC(=O)C(C3CCOCC3)O)CC1C2 C1(C(=O)NCCOCCOC)CCC(NC(C2C=CCS2)=O)C1 C1(NC(C(C)SC(C)C)=O)CC2CCC1CN2C(=O)CCC(C)(C)F Cc1cc(C(=O)NC(C)C(C(C)C)NC(=O)Cc2c(F)cccc2F)nc(O)n1 N1(C(CCc2n(C)ccc2)=O)CCCC2(CC(NC(c3csnc3Cl)=O)CO2)C1 C(=O)(N=c1ccn(C2CC2)[nH]1)C1N(C(CNC(COC)=O)=O)CCC1CO c1(N(C(C(=O)NCCSC2(C)CC2)C2CC2(C)Br)CC)cccc([N+](=O)[O-])c1C N1(C(c2c(C)sc(-c3ccccc3)n2)=O)C2CCC1C(NC(=O)C=CC1CC1)C2 CC1(C)CC(NC(=O)C(c2ccccn2)O)CN(C(c2conc2C2CC2)=O)C1 C(C(C)(C)Cn1cc(CCCC=C)nn1)NC(CSCC=C)=O c1(C(N2CCCC(CCNC(C3=CCCC3C)=O)C2)=O)cn2cnnc2cn1 c1(C(=O)NC2CN(C(c3cccnc3Br)=O)CC2F)cc(Br)cc2cc[nH]c12 CC(=O)CCCC(=O)N1CCCC(CNC(=O)C(C)Oc2cccnc2)C1 C(=O)(CCN(C)N=O)NCC1CCN(C(c2c(C(C)C)[nH]cc2)=O)CC1 c1(C(N(OC)C)=O)cc(N2CCCC2C(=O)Nc2ccc(Br)cc2)ncn1 C=CC1CN(CC2CC2)CCO1.c12ccc(cc1)C(=O)NC2C(=O)NS(C)(=O)=O C1(C(=O)NC2CC(NC(C3(C=C)CCC3)=O)C2)CCCC2(C1)NC(=O)NC2=O c1(C(=O)NC2(C3N(C(C4OCCN(C)C4)=O)CCCC3)CC2)ccccc1C#N C(=O)(CC1=NN(C)C(=O)C1)NCC(=O)NC(CNC(CSC)=O)C1CCC1 CC1Cc2c[nH]nc2C(C(=O)N(C)CCC2CCN(C(=O)C=CC3CC3)CC2)C1 C1(C(=O)NC(C)CNC(=O)CCN2C(=O)CCC2=O)CCCCC1(F)F N1(C(c2cncc(Cl)c2)=O)CCC2CCN(C(C34CCC(C3)C4)=O)C2C1 C(CC1=CCN(C(c2ccc3nonc3c2)=O)CC1)NC(C(C(C)C)SCC)=O c1(C(=O)NC2CN(C(c3ccc(CF)cc3)=O)C2)cncc(OC(F)F)c1 C1(CC)CN(C(C2(C)CCCS2)=O)CC1C(=O)NC(C)C(=O)NC(C)C CC1(C)CC(NC(=O)C=C2CCCCC2(C)C)CN(C(C2(C)CC2(C)C)=O)C1 N1(C(C(C)C(F)(F)F)=O)CCC(C(=O)N(C)CC2(C#N)CC2)C(C)(C)C1 N1(C(C(C)=CC=C)=O)CC=C(CC(=O)N2CCC(O)C(F)C2)CC1 C(=O)(CCCN(C)N=O)NCC(CC)NC(=O)C(C)(C)C#N C1(CNC(C2C(F)(F)C23CCC3)=O)CCCCN(C(c2c(O)cccc2F)=O)C1 C1(COC)CN(C(=O)CCSC2CCCCC2)CCN1C(=O)C1=C(C)OCC1 c1(OC)cccc(Cl)c1C(=O)NC1CN(C(c2nocc2Cl)=O)CCC1O N1(CC(=O)NCCC(C)(C)NC(C2CCCCNC2)=O)CCS(=O)CC1 O=C(CC1=CCCC1)NCC(O)CNC(c1ccccc1Cl)=O c1(CCC)ccc(C(=O)NCC2CCC(NC(=O)CCCC3CCCO3)C2)cc1 Cc1cc2sc(C(=O)NC34CC(NC(C5CC(O)C5C(F)(F)F)=O)(C3)C4)cc2s1 c1(C(=O)NCC2CC(O)CN2C(C2CC2(F)F)=O)c[nH]c2cccc(Cl)c12 CC1CN(C(c2cnn[nH]2)=O)C(C)CN1C(c1ccc(OC(C)(C)C)cn1)=O N1(C(C2(COC)CCOC2)=O)CCCOC(CCNC(c2ncccc2N)=O)C1 C1(C(=O)NCC(=O)OC(C)C)CCCCN(C(=O)CCc2ccsc2)C1 C1(C2(NC(c3nnnn3C3CC3)(COC)C)CCC2)CCN(c2ccccn2)CC1 c1(C(=O)NCC(=O)NC(C)CN(C)C(C2CC2CF)=O)cccs1 C(=O)(C1CCCc2ccnn21)NC1CCN(C(CCP(C)(C)=O)=O)C12CC2 C(=O)(C(F)CC(C)(C)NC(C1CCC2CC1CO2)=O)N(CCC1CC1)CC c1(OC)ccc(I)c(C(N2CC3CN(C(=O)CC#N)CC23)=O)c1 Cc1cc(C(=O)NC2(C)CC(NC(C3CC3(C)C(F)F)=O)C2)c[nH]c1=N c1(C(=O)NC23CC(CNC(CN4CC(C(C)C)C4)=O)(C2)C3)noc2cc(F)ccc12 c1(C(=O)NCC2(C)N(C(C)=O)CC(F)(F)C2)cccc2c1c(Br)nn2C C1(CNC(c2cnc(C(=O)OC)s2)=O)CN(C(=O)CSC)C2CCN1C2 c1(COC)cncc(C(N2CC(N(C)C(C3C4CNC(=O)C34)=O)C2)=O)c1 C(=O)(CC(C(F)F)NC(c1ccsc1C#N)=O)N(C)C1CC1 c1(NC(CC2ON=C(C)C2)=O)cncc(C(=O)Nc2ccc(C(N)=O)nc2)c1 C1(NC(c2cc(CNC(C3(OC(C)C)CCC3)=O)no2)=O)CCCCC1F C1(C(C)NC(C(C)N(C(C)=O)C)=O)CCN(C(c2sccc2F)=O)C1 CC1(C)CCC(CNC(=O)CCC2NC(=O)NC2=O)(NC(=O)CC2CCOC2)CC1 C1(OCC(=O)N(CCCCNC(C(C)N(C(C)=O)C)=O)C)CCCOC1 N1(C(C2(CC=C)CCOC2)=O)CC=C(C(=O)NCC2(CO)CC2(C)C)CC1 N1(C(C2(N(C)C(C3SCCS3)=O)CC2)=O)CCCC2CCCCC12 C12(CNC(=O)Cc3csnn3)CCCC1N(C(c1sccc1F)=O)CCC2 c1(C2(C(=O)NCC3(NC(C(C)Cn4ccnc4)=O)CC3)CC2)c(F)cccc1F n1(CC)ncc(S(=O)(=O)NC(c2cccc(C(C)C)c2)C)c1C C1(O)(CC(N2CC(COC)(NC(=O)CCc3ccoc3)C2)=O)CCCCC1 C(C1=NOC2(CCC2)C1)NC(C(C)(CO)NC(C=CC(CC)C)=O)=O CCC(C)(CO)C(=O)N1CCCC1c1cn[nH]c1.c12nc(cs1)C(=O)O2 c1(CNC(=O)Nc2c(C)nn(C3CCCCO3)c2C)c(C)c2ccccc2n1C CC1(C(=O)NC2Cc3ccccc32)CCCc2ccccc21 C1(NC(C(C)NC(CC)=O)=O)CCN(C(c2nccc(C)c2N)=O)CC1O N1(C(C(C)(C)CC2CC2)=O)CC(C(=O)N(C)OC2CCCC2)C(C2CC2)C1 CON(C)C(=O)C(C)(C)CN(C)Cc1cccc(Br)c1 c1(C(=O)NC2(C)CCN(C(C(CC#C)O)=O)CC2)c[nH]c2ccc(C#N)cc12 N1(C(c2ccnc(OC)n2)=O)CCCOC(CCNC(C2(C)CCCO2)=O)C1 C#CCC(O)C(=O)NCC(c1ccc(F)cc1)NC(=O)COc1cnn(C)c1 c1(OCC)ccc(C(=O)N(C(C)CCNC(c2nccc(Cl)c2C)=O)C)cc1O c1(C(N2CC3(CC(NC(C45COCC4C5)=O)C3)C2)=O)cccc2cc[nH]c12 CC1CN(C(c2cnc(C3CC3)s2)=O)CCN1C(C1CC(C(=O)OC(C)(C)C)C1)=O c1(C(N2CC(C)C(CNC(c3ccccc3O)=O)C2)=O)cccc(C#N)c1Br c1(C(C)OCC(C)NC(=O)Nc2ccoc2)c(F)cccc1F C1(C)(NC(CCCC)=O)CCCCC1C(=O)NCC(=O)NOCCCC1CC1 C1(N(C(c2ncsc2Br)C(=O)NC)C)CCC2C3CCC(C3)C12 c1(C(=O)NCC=CCNC(C2(C#N)C(C)C2)=O)cc(F)cc2ccccc12 c1(C(=O)NC2(CCNC(c3cnsc3)=O)CCCC2)ccc(F)c(C(F)(F)F)n1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CCN(C(C2C(C(=C)C)OCCC2)=O)CC1O C(=O)(CCC(=O)N1CCCC(C(C)NC(=O)C(F)(F)CO)C1)N(C(C)C)C C1(CNC(CCc2onc(C)n2)=O)CC(C)N(C(=O)C(C)c2cc[nH]n2)C1 C(=O)(C(COC(C)(C)C)NC(=O)C(F)=CC1CC1)N(CC(O)CF)C C(=O)(CC(C(C)OC)NC(C1CC(=C2CC2)C1)=O)NCC=CC N1(C(CCC(C)C#N)=O)CCC(C2(NC(c3cc(Cl)no3)=O)CC2)CC1 Cc1ccc(Cl)cc1C(N1CC(NC(C2(O)CC(F)(F)C2)=O)C(C)C1)=O c1(C(=O)NC2(CO)CCN(C(C(C)OCC)=O)C2)cnc2[nH]cnc2c1 C1(NC(c2csc(-c3cnc[nH]3)n2)=O)COCCN(c2nccc(CC#N)n2)C1 c1(C(N2CCCC(N(C(c3c(C)cc(F)s3)=O)C)C2)=O)cccc2nc(O)oc12 c1(C(N2CCN(C(c3cnc(C)[nH]3)=O)CC2CCO)=O)cccc2c(C)coc12 c1(N2CC(O)C3(C2)CCCC3)nc(N2CCC=C(Cl)C2)nc2c1CCCCCC2 C1(N2C3CN2C3)CC(=O)N(OC)C1.C1(C=O)CC=CCN1C(=O)O.C(C)(C)(C)OC C(=O)(CCC(F)(F)F)NC(C(C)(C)NC(C1N(CCC)CCCC1)=O)C c1(OCC)ccc(C)cc1C(N1CC(OC)C(NC(=O)CCC2CCCO2)C1)=O S(=O)(=O)(c1cccnc1N1CC2CCCCC2C1)N1C(C)C(C)(C)CC1 N1(C(c2c(C)cc(C)c(Br)n2)=O)CCC2(CCC2c2nn[nH]n2)CC1 c1(CC)nc(=N)[nH]cc1C(=O)NCCC1(C)CCN(C(c2ncc(F)cn2)=O)C1 C(C1CNC(=O)c2cc(on2)CN(C(C)C)C1=O)OC.C1(CO)CC1 N1(C(c2cn(C(C)C)nc2-c2ccc(F)cc2)=O)CC2(CCC2)CCC1CO C(=O)(CC(O)C(C)CC)N1CCC(C=C)(C(=O)Nc2cnc(C)c(C)c2)C1 CCCC(C(=O)NCc1nc(C(=O)NCCc2cccn2C)co1)OC N1(C(CC2N(C(CC(C=C)(C)O)=O)C3C2CCC3)=O)CCC(C2CCC2)C1 N1(C(c2c(N)c(C)n(C)n2)=O)CCCC(C2CN(C(C3CCCC(O)C3)=O)C2)C1 c1(OC)cc(C)c(C(N2CCCC2CN(C(=O)Cc2ncoc2C)C)=O)cc1Cl C1(NC(C#CCNC(CC(=O)NCC#C)=O)=O)CCCN(C)C1C CCC1=C(C(=O)NC2CN(C(=O)CCCCSC)C3CCCCC23)CCCO1 N1(C(C2(c3c(C)cno3)CC2)=O)CCCC2CN(C(c3ccnc(C)n3)=O)CC12 CC1NC(=O)CCC1CNC(=O)C(O)C1CN(C(C2(C)CC(F)C2)=O)C1 c1(OC)ncc(C(N2CCCCC2CCNC(c2ccc(Cl)s2)=O)=O)cc1C CC1(C)CC(O)CCN(C(=O)C(CC(F)F)NC(c2ccc(F)cn2)=O)C1 c1(CC)cccc(C(N2CCCC(N(C(=O)C(C)(C)C3CC3)C)C2)=O)c1 c1(-c2cn(CC3CN(C(c4cn(CCC=C)nn4)=O)C3)nn2)c(F)cccc1F N1(C(CC2CCCC(C)C2)=O)CCCC12CCN(C(c1nonc1N)=O)CC2 N1(Cc2cc(C)c(Cl)cc2)CC2CN(C(c3ccccc3C#N)=O)CC2C1 Cc1cc(CNC(=O)CC=CCNC(=O)CCc2cc(C)no2)nc(C)c1 Cc1nc2c(F)cccc2cc1C(N1CCC(F)C(NC(C2C(C)C2C)=O)C1)=O Cc1cc(C(=O)NC(C(N2CC(F)(CO)C2)=O)C2CCC2)nc(C)c1 Cc1ccccc1CC(C)C(=O)NC1CC1NC(=O)Cc1nc(C)c(C)s1 CCC(CCC(=O)NCCOC1CCN(C(c2c(F)ccnc2Cl)=O)C1)OC Cc1ccccc1C(=O)NCC(CC(=O)NC1CC1(C)C(F)F)C1CCC1 C1(C(=O)NCCc2onc(C)n2)CN(C(=O)C(C)(C)F)CC1(F)F CCCCCCCC(C)CNC(=O)C(=O)NC1CCC(C)(C)CC1 C1(C(C)C)OCCCC1C(=O)N(C)CC1CCCN1C(=O)C=Cc1ccn(C)c1 C1(C(=O)NCCCCOCC)C2CCCC2CN1C(c1nnsc1N)=O CCC(C(=O)N1CC=C(C(=O)N2CCCC(C(C)C)CC2)C1)C(F)(F)F Cc1cc(OCC(=O)N(C)CC2CN(C(C3(O)CCC3)=O)CC23CC3)cc(C)c1 c1(N(CCOCCNC(C(c2cccc(Cl)c2)C)=O)C)nc2cc(F)cc(F)c2o1 c1(C(=O)NC2C(NC(C(CC)n3cncn3)=O)CCC2)cc(OC)cc(OC)c1 C1(NC(c2c(CC)[nH]c(=N)s2)=O)CCCCN(C(=O)CN2CCCC2C)CC1 CC1CCCCC1(CNC(c1cc[nH]n1)=O)NC(=O)CCn1cnnn1 c1ccccc1F.N(C(=NCC)NCC(CC)OC)C(C#C)CC C1(C(NOCCC#C)=O)CC2(CCN1C(=O)C=CC1(C)COC1)CC2 C1(O)(C(N(C(c2ccccc2)CNC(c2ncn(C)n2)=O)C)=O)CCCC(C)(C)C1 c1(C(N(C(C)C)CCN(C)C(C2CCSC2)=O)=O)cncc(F)c1Cl Cc1c(C(=O)NCc2cc[nH]c2C(=O)NC(C)C(=O)N2CCCC2)[nH]ccc1=O N1(C(C(C)=C2CCC2)=O)CCC2(C1)CN(C(=O)CCc1cn(C)nn1)C2 n1(CCCC(=O)NC(CNC(C=CC=CC)=O)(C)CO)nc(C)cc1C c1(C(N(C)CC2CCCC(NC(COCC)=O)C2)=O)c(C)[nH]c2ncccc12 c1(C(=O)NC(CNC(CCC(CC)C)=O)C2CC2)cccc2c(C)ccnc12 C1(C(=O)NCc2c(C(N(CCOC)C)=O)n[nH]c2)CC(C(C)C)=NO1 N1(C(c2c(C)nn(C)c2)=O)CCC(n2cccn2)(CNC(C2COC(=O)O2)=O)CC1 C1(NC(c2c(C)onc2)=O)COC2(CNC(=O)C(C)OCC(F)(F)F)CC1C2 Cc1cc(NC(c2nc(C)c(C)s2)=O)ccc1NC(c1cc(C2CCC2)[nH]n1)=O C=CCCC(F)(F)C(=O)NCC1CN(C(C2(CNC(=O)OC(C)(C)C)CC2)=O)C1 CCC(C)CCCC(=O)N1CCN(C(=O)C(N2C(=O)CCC2=O)C)CC1 c1(C(=O)NC2C(NC(C(C)NS(CC)(=O)=O)=O)C2)cc2c(C#N)cccc2[nH]1 C(=O)(C1CCCc2c1ncn2C)NCC(CC)NC(c1cc(CC)nc(O)c1)=O C1(C(C)C)CCC(C(N2CC(C)(NC(=O)C=CCO)C2)=O)C(=O)N1 c1(C(N2CC(c3ccncn3)C2)=O)nnn(C2CNC2)n1 C(CC(C)(C)C)(C(=O)NCC1CC1C)NC(Cc1c(C)non1)=O N1(C(CN(CCCCCC)C)=O)CCN(C(=O)C2=COCCO2)C(CF)C1 C(CC(C)(C)NC(=O)C(C1CC(C)(C)C1)F)NC(COCC(=C)C)=O C(=O)(C(C(C)(C)C)NC(N)=O)NCCCCN(C)C(c1coc(C(C)(C)C)n1)=O C(C)(C)(C#Cc1cn(CCC(F)(F)C(F)F)nn1)NC(C(C)NC(=O)NC)=O C(=O)(C(CNC(=O)C(CC)CC)C(C)C)N1CC=C(C)CC1 CCC(O)(CC(=O)N1CCC(CC)(NC(c2cnn(C)c2)=O)CC1)c1ccccc1 N1(C(C2CC(C)CN2C(C2CC(N3CCOCC3)C2)=O)=O)CCC(C)(N(C)C)CC1 N1(C(Cc2ccn(CC)n2)=O)CCN(C(=O)CCOc2cccc(Cl)c2)C(C)C1 C#Cc1ccc(C(N2CC(CCNC(=O)Cc3ccon3)OC(C)C2)=O)cc1Cl C(=O)(C1CCc2ccccc21)NCC(=O)NCCC(C)S(C)=O Cc1sccc1C(=O)NC(C1(O)CN(C(=O)C(C2CCCCC2)F)C1)C CN1CC=C(CC(=O)NCC2CCN2C(=O)COCC2(F)CC2)CC1 c1(NC(C(C2CCN(C(CC=C=C)=O)C2)F)=O)c(O)cccc1Cl N1(CCOC)C(=O)c2cccc(C(=O)OC(C)C=C3CCOCC3)c2C1=O C1(C2CCCN(C(c3sccc3COC)=O)C2)(NC(COCC#C)=O)CC1 Cc1ncc(C=CC(=O)NC2CCC(C)N(C(=O)C=Cc3cscn3)C2)c(O)n1 N1(C(CCOC(C)=O)=O)CC(NC(c2ccn(C)n2)=O)C(n2ccnn2)C1 c1(C(=O)NC(C(=O)NC)C)ccc2nc(-c3cc(C)cc(C)c3F)cn2c1 c1(C(N2CCOCC(CNC(C3OCC(C)C3)=O)C2)=O)ccn2c1CCCC2 CC1CC(NC(=O)C(O)C2CCC2)CCN1C(c1cn(C2CCC2)nn1)=O C=CCC(CC)C(=O)N1CCC(CCNC(C2(OC)CC2)=O)CC1 c1(C(N2C(C(N(CCC(=O)OC)CC#C)=O)C(CC)CC2)=O)occ2c1CCC2 C(=O)(CCC(C)(C)C)NCc1cn(C2CN(C(C3N(C)C(=O)NC3)=O)C2)nn1 N1(C(c2c(CC)onc2C)=O)CCC(F)(F)C(CNC(c2c(Br)nnn2C)=O)C1 C1(NC(CC(C)(F)F)=O)CC2CCC1N(C(c1c[nH]c(=O)cn1)=O)C2 C1(C(=O)N2CCCC2)CNCC(=O)N1.C1(OCC(=O)OC(C)(C)C)CCCC1 CC1C(C(N2CC(C)(C(N)=O)C2)=O)CCCN1C(=O)Oc1cc(N)cc(F)c1 C(CCCC(CO)NC(=O)Cn1ncccc1=O)NC(C1(OC(C)=O)CC1)=O c1(C(N2CCCC(C(C(=O)OC)N)C2)=O)nn(C)cc1S(C)(=O)=O CC1(C)NCCC1CSc1ccc(OC2CCOC2)cc1 N1(C(=O)N(C(c2ccccc2OC(F)F)=O)C2CC2)CCOC(c2nccs2)C1 Cc1ccc(NC(=O)CCCC#N)c(C(N2CCC(CNS(C)(=O)=O)C2)=O)c1 c1(NC)ccc(CCC(=O)NCC(C)N(C)C(c2cnccn2)=O)cc1 N1(C(C(CSC)C)=O)CCC(C)(CNC(c2cc(Cl)ns2)=O)C1 C1(C)(Cn2cc(C3N(C(N(C4CC5CC5C4)C)=O)CCC3)nn2)CCC(=O)N1 C1(C#N)(C(=O)NCC(C)CN(C(=O)C(c2ccccc2)C2CC2)C)CC1(C)C N1(C(C2(CCC=C)CC2)=O)CCCC(C)(CNC(c2ccc(O)nn2)=O)C1 C1(NC(c2cc(C)sn2)=O)CCS(=O)(=O)C12CN(C(=O)C(C)NC(N)=O)C2 c1(CC(=O)NC2CC(NC(C(C3CCOC3)OCC)=O)C2)csc(S)n1 CCCCC(O)C(=O)N1CCC(C)(CNC(=O)CN2CC3CCC2C3)CC1 C(C(=O)N1CCC(NC(=O)N(CCC(C)O)C)O1)OC(CC)(C)C c1(N2CCC(CNC(c3c(OC)ccnc3)=O)C2)nnccc1C#N c1(CNC(C2CC(NC(C(c3ccc(F)s3)C)=O)C2)=O)ncccn1 CC(C)C(C(=O)N1CC(CC2CC2)C1)NC(C1(O)CCOCC1)=O CCC(F)(F)C(C)(C)C(=O)NC1CCCC1NC(c1ccc(Cl)c(F)c1O)=O c1(CNC2C(C(N3CCCC(O)C3)=O)C2)ccc([Si](C)(C)C)cc1 C1(CNC(C(Cc2cnc[nH]2)NCCCC(C)(F)F)=O)CCCCC1(C)C C1(CC(=O)NC)CCCCC(C)(C)C1.Cc1ccno1.N12CC(C1)COCC2=O C1(NC(c2c(N)cn(C)n2)=O)CN(C(c2occ3c2CCC3)=O)C(C)(C)C1 C=CCCCC(=O)NCc1ccc(C(=O)NC(c2ncc(C)cn2)C)nc1 C1(C(=O)NCCN(C(C)C)CC)CCCN(C(C)=O)CC1.C(=O)(CCC)NCC C=CCC(CNC(C1(CC=C)CCCN1C(=O)C(C)C1(O)CCC1)=O)CC(C)C c1(C(=O)NC2(C)CCCN(C(=O)COC3CCCC3)C2)c(Cl)ccc2c[nH]nc12 N1(C(c2ccc(CCC=C)cc2)=O)CC2CC1CN2C(=O)CN1CCC(C)C1 Cc1n[nH]c(=NCCC2C(C)CCCN2C(C2CCCNS2(=O)=O)=O)o1 c1(C(=O)NCC2CC(C)N(C(=O)Cn3cnc(=N)[nH]3)C2)cc(F)ccc1C1CC1 c1(C(=O)NC2C3(CC(NC(C4CC(C)(O)C4)=O)C3)C2)onc2ccccc12 C12(O)CCN(C1)CCCNC2=O.CCC(C)N(C)CCC(C)(C)C N1(C(c2cccc(Cl)c2OC)C(=O)NCCCOC)CCC2(CNC(=O)C2)C1 N1(C(c2c(C(C)NC(C3CS(=O)(=O)C3)=O)noc2)=O)CCCC1(C)C(C)(C)C c1(C(=O)NCCC(CC)(C)NC(=O)CS(C)(=O)=O)cc(F)c(NC(C)=O)cc1F c1(NC(=O)NCc2cn(C)nc2OCCO)cnc2[nH]cnc2c1 c1(CCNC2C(CO)CCCC2)nnc2n1CCOC2 CC1CCC(CNC(c2cccc(O)c2F)=O)N(C(=O)Cc2ccc(O)nc2)C1 C(CCCN=C(NCc1ccccc1)NCc1cnns1)c1[nH]c(=O)sc1 CC(CCCCNC(=O)C=C(C1CC1)C1CC1)NC(C1CCCC12CC2)=O c1(CNC(N(C(C2CCCCC2)C)C)=O)sc(Cl)cc1Cl C1(CC)CN2CC1C2=O.c1(NC(=O)CCc2nccs2)cnc(OC)nc1 c1(C(=O)NCCC2C(C)CN(C(c3ccc(Cl)cc3)=O)C2)c2c(nn1C)CCC2 C1(C(=O)Nc2ccc(COC)nc2)CC2(CC(NC(C3COC(C)C3)=O)C2)C1 CN1CCN(C)C(C(=O)NCC2CCCC2NC(c2cnn(C)c2Cl)=O)C1 c1(CNC(C(C)N(C(=O)CC2CCC(C)C2)CC)=O)cccc(C)n1 c1(OCC)cnc(C(=O)NC2(C)CC(NC(c3cc(C4CC4)on3)=O)C2)nc1 N1(C(c2cnc(C)n2C)=O)CCC2(NC(c3ccc(C(N)=O)[nH]3)=O)CCCC12 c1(C(N2CC(OC)(CNC(C3CC(C)OC3C)=O)C2)=O)ccnc2nc(C)nn12 C1(OC)CN(C)C(C)(C(=O)NC(C)CCCCNC(c2ccc(Cl)c(F)c2)=O)C1 C1(C(N(CCN(C(=O)C(C)C2CCCC2)CC)CC)=O)CCNC1=O CC(C)C(C#N)C(=O)NCC1CCC(C(=O)NCCc2cnco2)C1 C1(CC(=O)NC)CN(C(c2ccsc2Cl)=O)CCN1C(=O)CSC.C1(O)CC=CC1 Cc1cc(CC(=O)Nc2ccnn2C)cc(F)c1 c1(C(N2CC(CNC(c3cnn[nH]3)=O)CC23CCC3)=O)cc2cccc(Cl)c2o1 CCC(CC1CCCC1)C(=O)NC1CCC(NC(C2CC(F)(F)CS2)=O)C1 C=C(C)C1OCCC1C(=O)NC(C)(CNC(=O)CC(C1CC1)C1CC1)CO c1(OC)ccc(Br)c(F)c1CNC(C1(F)CCCN(C(=O)C(O)CC(C)C)C1)=O N(C1CC(C)c2ccccc21)Cc1cc2ccc(C)cc2s1 N1(C(C(C(C)(C)C)NC(C)=O)=O)CCN(C(c2cc(Cl)ncc2N)=O)C2CCC12 C1(C)(C(N2C(C(=O)NC3CC(F)C3)(COC)C=CC2)=O)CC2CCC1C2 CC(C)CN=C(NCCSc1cccs1)NCCc1ncc(Cl)s1 c1(C(N2C(C)C(NC(c3cc(Cl)sc3Cl)=O)CC2)=O)c[nH]c2cccnc12 c1(C(=O)NC2CCN(C(C(=O)NCC)=O)CC2O)noc2c1COCC2 C#Cc1ccc(CC(N2CCC(C=C)(C(=O)NC3CCCC3(C)CO)C2)=O)cc1 c1(N(C(CC2(C#N)CC2)C(=O)NC2CCOC2)CC)ccc(C)cc1 c1(C2C(NCC(=O)OCC)C2)ccc(Cl)cc1Cl CCC(C)(C)C(=O)N1CCC(C(F)C(=O)NCC(C)(C)C)C1 c1(C(=O)NC(CC=C)CNC(=O)CN2CCSCC2)ccc(C2(OC)CC2)cc1 Cc1ccncc1C(C(=O)NCCC1CC1)N(C1CCCCC1)C(C)C C1(N(C)CCS(C)(=O)=O)CCC(c2nnnn2C)(NCC2CCOC2)CC1 CC1CC(NC(C2CC(C)(O)C2)=O)CN(C(=O)CCSc2ccccn2)C1 CCC(CC)C(F)C(=O)N(C)CC1(CNC(=O)CC2CCC(C(F)(F)F)O2)CC1 N1(CC(CCCC)CC)CCC(O)(CN2C(=O)CN(CC(C)(C)O)C2=O)CC1 N1(C(C2(SC(F)F)CC2)=O)CC2(CC(CNC(C3(O)CCOC3)=O)C2)C1 C(=O)(CCCCCCNC(C(O)CC=O)=O)NCCCCCCC S(=O)(=O)(c1ccc(NCC2CCC(OC)C2OC)c(Br)c1)N1CCC(CC)CC1 c1(C(N2CC(C)C(NCc3cn4ccc(Cl)cc4n3)C2)=O)ccc(Br)cc1[N+](=O)[O-] CC(C)CC(C)C(=O)NCc1ccc(C(=O)NCCCc2cc[nH]n2)o1 C1(NC(C2CC(C)CN2C(C2CC2(F)Cl)=O)=O)CCN(C)CC1C#N N1(C(CN(C(=O)OCC)C)=O)CCC(NC(=O)C=Cc2cnccn2)C12CC2 N1(C(C2CC3CCC2C3)=O)CCN(CC2CC2)C(c2ccc(OC(F)F)cc2)C1 CCCC(CC(C)C)C(=O)NC1COCCC1C(=O)N(C)Cc1nnc(O)o1 C1(CC(=O)NCC2(OC)CN(C(C3CC(=O)NC3=O)=O)C2)CCCCCC1 C1(c2n(C)nnn2)(Nc2cccnc2S)CCC(c2ccnn2CC(C)(C)C)CC1 N1(C(C=CSC)=O)CCN(C(c2cc3ccsc3s2)=O)CC1C1CCC1 N1(C(C2N(C(N)=O)CCC2)=O)CC(N=c2[nH]c3ccccc3n2C)CC(F)(F)C1 N1(C(C2CC3CCC(C2)C3)=O)CCC2CN(C(C3CCS3(=O)=O)=O)C2C1 CC1(C(N2CC=CC2C(=O)NCC(Cl)=CCl)=O)CCNC1=O CCCCCCC(C)C(=O)N1CCOCC(CNC(c2ccc(CO)nc2)=O)C1 c1(C(=O)NCC2N(C(CCC=C)=O)CC=C2)nc(CCC)c(C)s1 C#CCCCC(=O)NC1CC2(C1)CC2NC(C1CCCCO1)=O C(=O)(C(CCN(C)C)NC(C1CCCSC1)=O)NC(CC)CCO N1(C(CCn2c(C)ncc2)=O)CCCN(CCCNC(=O)CO)CC1 C1(C(N2CC(C)(C(=O)NOCC3(F)CCC3)C2)=O)CC2CCC1C2 C(=O)(C(C)(C)C(F)(F)F)NC1C2CN(C(CCc3nc(C)sc3)=O)C1C2 C1(C(=O)NCC(=O)NCC(N2CCC(CN(C)C)C2)=O)CC(=O)NC(=O)C1 C1(CC(N2C(C(CNC(Cc3nnc(C)s3)=O)(C)C)CCC2)=O)CCC(=O)NC1 C1(CN(C(C2CN(C(C)C)C2)=O)C)CCN(C(c2cnco2)=O)C1 N1(C(C2CN(C(C)=O)C2)=O)CCC2CN(C(c3ncc[nH]c3=O)=O)CC2CC1 c1(C(N2CC(O)CC(NC(C3CCC(CC)CC3)=O)C2)=O)cc[nH]c2nccc1-2 c1(-c2cc(OC)cc(C)n2)ccc2oc(C(N3CCN(C(C)C)CC3)=O)cc2c1 N1(C(c2c(C#C)c[nH]n2)=O)CC2CCCC(C1)N2C(C1CCCN(C(C)C)C1)=O C(CCCCCCC(=O)OC1CCCNC1)N1C(C)(C)C(c2ccccc2)CC1 c1(C(=O)NCc2cc(COC)c(Cl)cc2)cc([N+](=O)[O-])c(C)c([N+](=O)[O-])c1 c1(C(NOCC(=O)NC(C)(C)CCCF)=O)cnc(O)c(F)c1 C1(OCC)CC2CN(C(c3csc(C)n3)C(=O)Nc3cc(F)ccc3F)CC12 N1(C(C2CC(OC)C2)=O)CC(F)(F)CC1C(N1CC2C(C1)C2(C)C)=O c1(C(=O)NCC(=O)NCCN(C(CCS(C)(=O)=O)=O)C)ccc([N+](=O)[O-])cc1 N1(Cc2nc(C)sc2)CCN(C(c2cc(F)ccc2Br)=O)CC1C(C)C CC1CN(C(=O)CCc2ccccn2)CC1CNC(=O)C(F)C1CCC1 c1(C(=O)NCC(CC(C)C)(C)NC(C2CCCN2C)=O)cccc(P(C)(C)=O)c1 O=C(C1=NOCC1)NCCCN(C(c1cc(Cl)cnn1)=O)CC1CCCC1 C1(CN(C(C(C)NC(=O)CC2CCCO2)=O)C2CC2)CCCCO1 C(CC(C)C)(C(=O)N1CCOC(NCCNC(=O)C(C)NC(C)=O)C1)OC N1(C(C2ON=C(C)C2)=O)CCC(NC(C2OCCN(C)C2=O)=O)C2(CCC2)C1 C12CN(CC1C)C(=O)C(=O)N2.CCCCCCNC(=O)OC(C)(C)C.C1C(=O)N1 CCC(C)(CCC(C)C)C(=O)Nc1ncc(-c2cnn3c2NCC3)s1 CC1CCC(C)(C(=O)NCC2(CNC(c3nn(C)cc3Cl)=O)CC2)C1(C)C N1(C(c2cc(N)c(Cl)c(O)c2)=O)CCOc2ccccc2C1CO Cc1nc[nH]c1C(=O)NC(CNC(=O)CCc1nc(-c2cccs2)no1)CO CC1(C)C(CNC(=O)NCC(N2C(=O)CNC2=O)C(F)(F)F)C1(C)C c1(CC)c(C(=O)NC(C)(C)CCCNC(C2CC3(C2)CC3F)=O)nnn1C C1(NC(=O)Cc2cncc(F)c2)CCCN(C(c2ccccc2OC(F)F)=O)C1 c1(C2(C)CC2)nc(=NC2CN(c3nccnc3C#N)C3(CCC3)C2)[nH]o1 C1(C(C)NC(C(C2CN(C(c3nnc(O)o3)=O)C2)OC)=O)CCCN1C C12(CNC(C3C(C=C)OCCC3)=O)CC(NC(=O)COC(C)CC)(C1)C(C)(C)O2 c1(C(N(C2CC(NC(C3NC(=O)OC3(C)C)=O)C2)C)=O)cccc2c1COC2 O=C(CCC1CCc2ccccc21)NC1CC(NC(C2CC23CCC3)=O)C1 N1(CC(N2CCc3c(nc(C)n3C)C2)=O)C(=O)NC2(CCCC2(C)C)C1=O C(CCC(C)(C)C(=O)N(C)Cc1conc1CC)NC(COCCSC)=O C(=O)(C1CCOc2ccccc21)N(C1CCN(c2ncnc3n[nH]c(Br)c23)C1)C C(=O)(C1=NOC2(CCN(C(=O)C(C)OC3CCCCC3)C2)C1)N1CC2C(C)C2C1 c1(CONC(C2(F)CN(C(C3CCCCC3F)=O)C2)=O)ccc([N+](=O)[O-])cc1F N1(C(CCNC(=O)NC)=O)CC(NC(C2CCC(=O)N2C2CC2)=O)CC(C)(C)C1 N1(C(C2CCC(=C)CC2)=O)CCCCC(NC(c2ccc(-c3cccs3)o2)=O)C1 N1C(=NCCC(C)C)NCCC2CCC1O2.C(C1=CCCOC1)NC(C)=O C1(CNC(CC2N(C)CCCC2)=O)CC2(CC2)CN1C(c1cc(Cl)ns1)=O c1(N2CC(C)CS(=O)CC2)nc2c(c(=NCCc3ccc(Cl)s3)[nH]1)CCCC2 N1(C(CNC(CCC)=O)=O)CC(C)CN(C(=O)C=Cc2cncs2)CC1C CC(C)(C#N)CCC(C)(c1nnnn1Cc1ccccc1)NCC1C=CCCCC1 C12(NC(c3cc(-c4ccc(F)cc4)no3)=O)CCCC1CN(C(=O)C1CC1)C2 Cc1cnc(C)c(C(N2CC(N(C)Cc3c(O)cccc3Br)C2)=O)n1 CC1(C)OC(C(=O)NC2CCC2NC(c2c(Cl)ccc(F)c2F)=O)C(C)(C)O1 C(=O)(C1=CC2CCCCC12)NCC(C)NC(=O)COc1ccc(F)c(F)c1 C=CC(C)C(C)C(=O)NCCCCCC(=O)N(CCNC(C)=O)C Cc1ccccc1C(=O)NC(C)CCN(C(=O)C(c1ccc(C(F)F)cc1)C)C C(CS(=O)(=O)CC(=O)N1CC(NC(=O)C2=CCCSC2)C(C)C1)OC C1(NC(c2c(C)snn2)=O)CC2CN(C(=O)CNC(=O)CC(C)C)CCN2C1=O C1(CNC(C2CCN(C(=O)NCC)CC2)=O)CC2CCC(C1)N2C(C)=O C(=O)(CC(COC)NC(=O)CCC1CCCCC1)N(CC(=O)NC)C N1(C(Cc2n(C)ncc2)=O)Cc2ccccc2C(NC(=O)C(C)(C)C(C)(F)F)C1 c1(C(N2C(C)CC(NC(C3(O)COC3)=O)CC2)=O)n[nH]c2c1CC(F)(F)CC2 c1(-c2ccc(C(=O)NCc3ocnc3CO)s2)ccc(NC(=O)CC(F)(F)F)cc1 C#Cc1cn(C)nc1C(=O)N(C1CN(C(c2cccn2C2CC2)=O)CC1O)C c1(C(=O)NC(c2cnn(C)c2)C)cc(-c2cnc(C3CC3)nc2)cc2cc[nH]c12 c1(CCCC(=O)NCCN(C(=O)C(C)=CC(C)(C)C)CCC)ccc(F)c(F)c1 N1(C(C(C)(C)SC)=O)CCN(C(=O)Cc2cn(C)nn2)C(CF)C1 c1(C(=O)NCC(C#C)CC2CC2)nc(CNC(c2csnc2OC)=O)oc1C c1(C(N2CCC(N(C)C(c3cc(C4CC4)cs3)=O)C2)=O)cc(O)ncn1 C12(C(N(C)Cc3ccc(=O)oc3)=O)C(NC(=O)CC3CSCCO3)C3CC1C2C3 C1(NC(Cc2ccc(C)s2)=O)CCN(c2ncns2)CCC1CO C1(CC)(NC(=O)C(O)CC(F)F)CCN(C(=O)Cc2ccccc2COC)CC1 CCC(C)C(C(=O)Nc1ccc(F)nc1)N(C)C(c1n[nH]cc1Cl)=O N1(CCC#C)CCC(C(=O)NCC2CC2NC(C2COC(=O)C2)=O)CC1 N1(C(C2(OC)CC2)=O)CCCC(CNC(C2(Cl)CC23CCC3)=O)C1 c1(SCCC(=O)N(Cl)CCO)cc(Cl)cc(Cl)c1 O=C(NNC(=O)CSCc1ccccc1)c1cnc(-c2ccccn2)s1 C1(n2cc(C(N)=O)nn2)CC2CCC1(NC(=O)C(F)CC1CCOC1)C2 C(C(CC(=O)NCCCS(N)(=O)=O)NC(C1C2COCC12)=O)OC N1(C(CSSC)=O)CC(CO)C2(C1)CN(C(=O)C(C)SCC(C)C)C2 c1(C(N(CC(C)NC(=O)C(F)=C2CCC2)C)=O)ncncc1C#N N1(C(CCSCCC)=O)CCOC(C(C)NC(C2CC(O)CN2C)=O)C1 C(C1CCN(C(C2(F)C(C)(C)C2(C)C)=O)CC1)=CC(=O)N(C)Cc1cn[nH]c1 C(c1ccc(F)cc1Cl)=CC(N1CC2C(CNC(c3cncc(C)c3)=O)C2C1)=O CCCCC(C)CCC(=O)NC1CCN(Cc2ncc(C(C)(C)C)o2)CC1O CCC(CC(=O)NCC(=O)Nc1cc(Cl)cc(Cl)c1)C(C)(C)C Cn1nc2ccccc2c1C(=O)NC1CC2CCCC2C1 C1(C(N2CCC(=CCNC(c3c(C)cc(C)s3)=O)CC2)=O)CC(C2CCC2)C1 c1(CCC(=O)NCC(CC=C)NC(C2CC3C(C2)C3(C)C)=O)cccc(OC)c1F C(=O)(C#CC1(C)CCCO1)N1C(CN(C(C2C(C)=CCS2)=O)C)CC(F)C1 Cc1ccc(C(F)(F)C(=O)NCC(C2CCCC2)NC(=O)CSCCC#N)cc1 N1(C(C(CNC(c2c(CC)ccc(C)c2)=O)C)=O)CCC(F)(F)C(F)C1 C1(C(N2CC2C)=O)CCC(NC)CC1.C1(C(=O)NC)CCN(c2cnccn2)CC1 c1(C(=O)NCC(C)NC(C(C=C)O)=O)cccc(OCC=CC)c1 CC1(CNC(=O)CCN2CCCC2)CN(C(c2cc(Cl)nc(=N)[nH]2)=O)CCO1 c1(CC)cc(F)ccc1C(N1CCSCC1C(=O)NCC1C(C)(C)C1(C)C)=O c12cccn(c1=O)CC(=O)N2.N1(C(CCC2C(C)C2)=O)CC(C)(C)OC1=O N1(C(c2cnn(C(F)F)c2)=O)CCC2(CCCC(CO)O2)CC1 CC1CC(NC(c2ncsc2Br)=O)CCN1C(c1cc(Cl)no1)=O N(C1CCCn2nccc21)C(C(CCC)NC(C1CC2CC(=O)C1O2)=O)=O c1(CNC(c2n(CC)nnn2)Cc2ccc(C)n2C)cc(O)n2ncc(Br)c2n1 C(C(=O)NCC(C)C(=O)NC1CC2(C1)CC(O)C2)(C(C)(C)C)OC C(=O)(C1=NOCC1)NC(CC)CNC(=O)CCc1ccc(CCCCOC)o1.OC CC1(C(=O)NC(C)(C)CC2CCOC2)CN(C(C2CCCS2)=O)C1 c1(NC(C23C(CN(c4nccc(SC)n4)C2)C3)=O)ccc(C)cc1Br N1(CC)N=C(C(=O)N2CCC(CF)(NC(C34CCCC3OCC4)=O)C2)CCC1=O c1(CCNC(=O)NCC(c2ccc(F)c(Br)c2)(C)O)ccccc1[N+](=O)[O-] N1(C(c2ccccc2[N+](=O)[O-])=O)CCC2(CCCN(S(=O)(=O)C3CCOCC3)C2)C1 c1(C(COCC)(C)NC(c2nnnn2-c2ccccc2C)C)cc(Cl)cn1C N1(C(c2c(C)ocn2)=O)CCN(C(c2nn(C)cc2Br)=O)CC1CCO C1(C(=O)NCCCC(=C)Cl)CCN(C(C2CSC2)=O)C12CCC2 O=C(C#Cc1ccccc1)NC1CC(NC(c2c[nH]c3ncccc23)=O)C1 CC1CN(C(=O)COC(=O)C2CC2)c2cc(C(F)(F)F)ccc2O1 N1(C(CNC(=O)OC)=O)CC(C)(C(=O)NC(C2(C)CC2)C)C1 C1(NC(c2ccc(SC)o2)=O)C2CC3C(C2)C13C(=O)NCC1CC(C(N)=O)=NO1 C1(C(=O)NCCCC=C)C=CCCN1C(C1CC(F)(F)C1)=O Cc1c(C(N2CC3CCC(C2)N3C(c2ccc(O)c(Cl)c2)=O)=O)sc2nccn12 C1(C)(OC)CN(CC2C(C(=O)N(C(=O)CC3CC4(CC4)C3)C3CC3)C2)C1 Cc1ccn2ncc(C(N3CCN(C(=O)CCCCCF)CCC3C)=O)c2c1 c1(N(C(C)=O)CC)ccc(C(N2CCNC(=O)C2)=O)c(C)c1 C(=O)(C1=CCCCO1)NC(CC(C)NC(=O)CCSC1CCCC1)C c1(C(=O)NCC(C)OC)occc1CNC(c1cc[nH]c1)=O N1(C(C2C(C#N)C2)=O)CC2CCC(CNC(C3CCOC3)=O)(C2)C1 N1(C(C2C(COC)CC2)=O)CCC2(C1)CN(C(=O)CN(C)S(N)(=O)=O)CCO2 c1(C(N(CCC(=O)N(CC(C2CCC2)OC)C)C)=O)cc(O)ncc1F Cc1cc(C)c(C(N2CSCC2C(=O)Nc2cccc(C(F)F)c2)=O)o1 c1(OCC(=O)NCC(CNC(C(CC)N(C)C)=O)F)ccccc1[N+](=O)[O-] O=C1Cc2ccc(CC(=O)NC3CC(c4ncc[nH]4)C3)cc2N1 C1(C(N(C2CCCC2)CC=C)=O)CC2(CCN1C(=O)C(C)CC1CCCC1)CC2 N1(C(CC(=O)OC)=O)CCC(CNC(c2csc(C(F)(F)F)n2)=O)(OC)C1 c1(C(=O)NCCC2OCCN(C(c3cc(OC)no3)=O)C2)cc(C)c(Cl)cc1C n1(CC=C)ccnc1C(N1CC(O)(C2CCCN2C(=O)COCC)C1)=O C1(C(N2CC(OC)(CNC(=O)C(N3CCOCC3)C)C2)=O)COC(C)(C)C1 CC1CN(C(c2n[nH]c(O)n2)=O)CC1NC(=O)COC1CC(n2cnnc2)C1 c1(C(N(C2CCCN(C(c3cnc(O)o3)=O)CC2)C)=O)ccc(O)c(Cl)n1 Nc1c(C(N2CCCC(NC(=O)C3=CSCS3)CC2)=O)ccnc1Br c1(NC(C2CC(OC)CN2Cc2cnn(C)c2)=O)ccc(Br)c(C)c1F C(=O)(C1=CC2C=CC(C1)C2)N1C(C(N2CCC(C=C)(CO)C2)=O)CCC1 C(C(=O)N1CC(C)(O)C1)(C(C)O)NC(C=CC(CC)C)=O C1(C(=O)NCC(C(C)O)C)(NC(=O)C(=O)C2CCCC2)CCOCC1 C(=O)(C1=NOC(C)(C)C1)NCc1cn(CC(=O)Nc2cc(OC)ncc2C)nn1 c1(NC(=O)CCOCC(F)F)cnc(Br)nc1 c1(C(=O)NC2C=CCN(C(C=COCC)=O)C2)ccc(S2(=O)=NCCC2)cc1 CCCCCS(=O)(=O)CC(=O)N1CCN(C(c2c[nH]c(=N)s2)=O)C(CC)C1 N1(CC)N=C(C(=O)N2CC(F)(F)CC2CNC(c2cn(C)cc2C)=O)CCC1=O N1(C(CCNC(COC)=O)=O)C2CCC1C(CNC(c1cccc(N)c1C)=O)C2 c1(OCC)cc2ccccc2cc1CCNC(c1ccccc1F)CC(=O)O N1(C(C(C(C)C)N2CCCC2=O)=O)CC2(CCN(C(C3(C)CC=CC3)=O)CC2)C1 c1(C(N2CCN(C(=O)NCCCc3nc[nH]n3)CC2)=O)cc2ccccc2[nH]1 C12(C(N3CC(CNC(C(CCSC)N(C)C)=O)C3)=O)CCC(CC1)C(C)O2 C12(NC(COCc3onc(CC)n3)=O)COCCC1CN(C(C1CCC1)=O)C2 N1(C(CCC#CC)=O)CCC2CN(C(=O)CC(O)CCC)CC2C1 C(=O)(CC(C)(O)C(F)(F)F)N(C1C(C)CCN(C(c2sc(C)c(O)n2)=O)C1)C c1(NC(N2CC3(CC(O)C3)C2)=O)ccc(-c2nn[nH]n2)cc1F c1(CC)cc(C(=O)O)on1.n12cc(nn1)CNC(=O)NCC2 n1(CC(=O)NC2CCN(Cc3ncc(Cl)s3)C2)cnc(-c2ccccc2)n1 c1(OC)c(Br)cc(C(C(=O)O)NC(=O)C(N)CCNCCO)cc1Br CC1(C)C(NC(=O)CC2(N3CCCC3)CCC2)CC1CNC(C1CC(F)(F)C1)=O Cc1cccc(NC(C2CC(CNC(=O)COC3CCCC3)C23CCC3)=O)c1F c1(C(N(C(C)CN(C(=O)CN2CCC(O)CC2)C)C)=O)cc2ccnc(Cl)c2[nH]1 C1(C(=O)NCC(C)NC(c2scnc2C(F)(F)F)=O)CC2(CCO2)C1 C1(NC(C2N(C)C(=O)CC2)=O)CC2CN(C(=O)CCC3CCC(=O)NC3)CC2C1 C(C)(C(CC(=O)NCC1(C)CC(C)(C)C1)NC(=O)C=CC1CCCN1C)OC c1(C(=O)NCCC2CCCN(C(CCCOC(C)=O)=O)C2)nc(O)nc(O)c1F c1(C(=O)NCC2(F)CC(CNC(C34CCC(CF)(C3)OC4)=O)C2)csc2nccn12 C(=O)(C1=CCCCCC1)NCC#CC(=O)Nc1c(CC)noc1 Cc1ccc(I)cc1CCNC(=O)NCC1(c2ccccc2Cl)CC1 C(=O)(C(F)CCC(C)C)NC1C(NC(c2cncc(C(C)=O)c2)=O)COCC1 C1(NC(C2CCN(CC)C2)=O)C2CCCN(CC(=O)NCC3CC3)C2C1(C)C c1(OC)cc(C(N2CCN(CC(C)NC(C3CCC=CO3)=O)CC2)=O)cc(Cl)n1 c1(C(=O)NCC23C(CN(C(CCC(=C)Cl)=O)C2)CC3)c(CC)nc2ccccn12 Cc1cscc1C(=O)N(CCC1(NC(C2CCCC2C(F)F)=O)CCC1)C(C)C C(=O)(C1=CCCO1)NC(C(C)C)CNC(=O)C(C)(C)OCCS(C)(=O)=O N1(C(C2(C)CS(=O)(=O)C2)=O)CCC2(NC(c3ccc(C(N)=O)cc3)=O)CC2C1 C1(CC(=O)NCCCCN(C(=O)Cc2cscn2)C2CC2)C=CS(=O)(=O)C1 CC1(C)C(c2ccc(C(N3CC4C(NC(C5CC5F)=O)C4C3)=O)s2)C1(C)C C(C(=O)NC(c1c[nH]ccc1=O)C)(C(C)CC)NC(c1ccn(COC)n1)=O CC(CCCC(=O)NC1CCC(C)(CO)CC1)NC(C1CC1(F)Cl)=O c1(OC(=O)NCC(C(C)(C)C)CO)ccc(F)c(F)c1F.c12nc(cs1)NCC2 C1(C(=O)NCCCC(C(=O)NCC2(C#N)CCCC2)O)CC2(CCO1)CC2 c1(C(=O)NCC(CC)NC(c2cc(C(C)=O)c(C)o2)=O)ccn(CCO)c(=O)c1 c1(CN2CCC(NC(c3cc4ccccc4[nH]3)=O)C(O)C2)ccc(F)c(Br)c1F C1(C(C=C)C)CC(NC(=O)CN(C(=O)C(F)n2ccnc2)C)C1 c1(CC)cccc(C(=O)NC2CCCC2NC(C2CCCN2C(C)=O)=O)c1O N#Cc1ccc(CCC(N2CCC(F)C(NC(=O)COCC3CC3)C2)=O)c(F)c1 c1(C(N2CCC(F)(C(N3CCC(OCC(N)=O)C3)=O)C2)=O)ccn(O)c(=O)c1 C1(CNC(CCOCC#C)=O)COCCN(C(C2(CN(C)C)CCCCC2)=O)C1 C(C)(C(=O)N=c1ccn(-c2ccncc2)[nH]1)C1CCCN(C(c2c(C)ccs2)=O)C1 c1(CN2C(CNC(c3c(C)ccc(F)c3)=O)CCC2)ccc(Cl)cc1F C(C(C)C)(C(O)C(=O)NCC1CN(C(=O)CC2(C)CC2)CC12CCC2)OC C1(C(=O)NCC(C)NC(=O)C(C)(C)c2cnsc2)Cc2cccc(F)c2O1 CCC(CNC(=O)COCc1cccc(C)c1)(CC)NC(C1CC2CCCC12)=O C12(C(=O)NCCN(C(C3CC4CCCCC34)=O)CC)CC1COC2(C)C c1(-n2cc(C(C(C)C)O)nn2)ccccc1CNC(C1C2CCOCC12)=O c1(COC)nc(C)c(C(=O)NCC2CCN2C(=O)CCc2ccc(F)cc2)s1 C1(CCOC(C(Cc2ccccc2)OC)=O)=CCCCN=C1 Cc1cccc2c(=O)n(CC(=O)N(CCCNC(=O)CNC=O)C3CC3)cnc12 Cc1nc(N2CCC(C)C2CNC(C2CCCOCC2)=O)c(Cl)cc1[N+](=O)[O-] c1(C(=O)NC(C)CCNC(=O)C(C)(C)C2CCOC2)nc2c(s1)COCC2 C(CNC(c1ncsc1C1CC1)=O)(CC(F)(F)F)NC(c1n(CC)ncc1C)=O C1(CNC(C2C(C=C)CC2)=O)CC(F)(F)CN1C(=O)Cc1cc(C)no1 CC1CC(C)(C(N2CCC(CNC(c3cc(C4CC4)on3)=O)CC2)=O)CCO1 CC1(C)C(NC(C2CCN(CC(F)F)CC2)=O)CCN1C(C1CCS(=O)(=O)N1)=O C1(C(=O)NC(C2N(C(c3c(CC)ncs3)=O)CCC2)C)CN(S(N)(=O)=O)C1 C1(NC(CSCCOC)=O)CCC2(CC1)CC(NC(c1c[nH]nc1C1(C)CC1)=O)C2 CCCC(C(=O)NC1CCCN(CCNC(=O)C(=O)N(C)C)C1)NC(N)=O c1(C(=O)N(C2CCN(C(=O)Cc3nc(Cl)cs3)CC2)CC)ccc2cc(C)[nH]c2c1 C1(C2CCN(C(c3c[nH]c(C#N)c3)=O)C2)(NC(CN(C2CCSC2)C)=O)CC1 c1(OC(C)C)c(C(=O)NC(CNC(=O)C=CS(C)=O)C(C)(C)C)cccc1N C(=O)(C(C)CCC(C)(C)C)N(CCC(N1CC(C)C1(C)C)=O)CC#C S(=O)(=O)(c1c[nH]c(C(N2CC(NC(c3cc(CF)on3)=O)C3CC23)=O)c1)NC CN1CC(O)CCC1C(N1CCCC(CC(=O)NCC2(C3CC3)CCC2)C1)=O C(c1ccc2c(c1)OCO2)=CC(=O)NC(CNC(C#CC1(C)CC1)=O)C1CC1 N1(C(c2cnc(COC)nc2)=O)CC(C2CC2)(C(=O)N(CCO)OC)C1 c1(SCCC2CC(C)(C)OC2)cc(Br)cc(F)c1O C(CCCC(=O)N1CC(CNC(c2ccc(C(=O)N(C)C)nc2)=O)CC1C)SC c1(OC)cc(C)cc(C(=O)NCCCCNC(C2CCN(C)C2C)=O)c1C C(c1ccc(Cl)c(Cl)c1)=CC(N1CCN(c2ncccn2)C2(CC2)C1)=O CC(C)C(O)C(C)(C)C(=O)N1CCCC(CC(=O)NC2(C)CC(F)(F)C2)CC1 C1(CC(=O)NC2(CC=C)CCOC2)C2CCCC2N1C(=O)Cc1cc[nH]c1 C=Cc1cc(C(=O)NCC(C(C)C(C)C)NC(c2sc(C)cc2C)=O)cc(F)c1 C1(NC(C2=CC(C)(C)C2)=O)C2CCCN(C(=O)COCc3nc[nH]n3)C2C1(C)C C1(CC=C)CCCN(C(=O)CCN(C(=O)CC2CCC(C)(C)C2)C2CC2)C1.CCC c1(C(=O)NC2(CC=C)CN(c3cc(=O)n(C)c(O)n3)C2)cc2c(cn1)OCCO2 C1(NC(CCC(=C)Cl)=O)CCCC12CN(C(c1cn(C(C)C)nc1Br)=O)C2 N1(C(c2ccc(CSC)o2)=O)CCN(C(=O)Cc2c[nH]nc2O)CC1CF N1(C(C(CC=C)N(C)C)=O)CC2(C1)CN(C(C1CC(=O)NC1(C)C)=O)C2 c1(C(=O)NCc2c(-c3ccc(CCC)s3)cccc2)ccc2c(c1)C(=O)N(C)C2 C1(O)(CC(=O)NCC(C)(C2CCC2)NC(C2(C)CCNC2=O)=O)CCCCC1 Cc1cc(C(=O)N(C(C)CS(C)(=O)=O)C)cc(S(=O)(=O)Nc2ccccc2F)c1C N1(C(C(=O)NC(CC)(C)C)C(C)CC2CCCCC2)CCC2(C1)NC(=O)NC2=O C1(CC)C(NC(c2ccc(-c3cc[nH]n3)s2)=O)CCN1C(=O)Cc1csc(C)c1 C1(CC(=O)NCc2ncsn2)CC(F)CN1C(c1ccncc1F)=O c1(CC(N2CCN(C3CC3C(F)(F)F)CC2)=O)ccc2c(c1)OC(F)(F)O2 C(CCC(C)C)(C(=O)N1CC(C(=O)OC)C1)NC(COCCOCC#C)=O CCCC(C)CC(=O)NC1CN(C(C2CC2(C)C(C)C)=O)CC1F CC1CC(CNC(=O)Cc2csc(S)n2)CN1C(=O)Cc1cnco1 N1(C(COc2c(OC)cccc2)=O)CCC2CC1CN2C(=O)C#CC1CCC1 C1(N(C(CCOC)=O)C(C)CC#N)CNCC1(F)F C=CCC(C)(CNC(=O)CC(C(F)F)NC(=O)CN(C)C1CC1)CO CC(C(C)C(=O)NOCCF)NC(c1cc(F)c[nH]1)=O Cc1ccc(CCNC(CCCOc2ccc(F)cc2Cl)=O)cc1C C(=O)(CC1=CCOCC1)NC1CCCC(N(C(=O)CCc2nc[nH]n2)CC)C1 CC(C)C(C(=O)NC1C=CCCC1C(=O)NC1CC(O)C(F)C1)C1CCC1 C(C(=O)N1CCOCC1C(N)=O)(C(C)C)NC(c1cnc(C)o1)=O CC1=C(C(=O)NCC2CN(C(C3CCCC3)=O)CC2c2cncn2C)CCO1 C1(C2CC2)(C(=O)NCC(CC)(CC)NC(=O)CCc2nncn2C)CC=CC1 C(=O)(CCC(=O)NC)NCn1c(C(N(C(C)CO)CC)=O)cnc1 C1(C(N(C2(C(NOC(COC)COC)=O)CC2)C)=O)CC(C2CC2)=NO1 c1(NC(C2CC3CC3N2Cc2ccnnc2O)=O)cc(Cl)ccc1-c1nn[nH]n1 N(C1CCc2ccccc21)(C(C(=O)NCC=C)CC1CCC1)CC(C)C CC1CC(C)(C(=O)NC23COC(CNC(c4cc(C(N)=O)[nH]n4)=O)(C2)C3)CCO1 N1(C(c2cc[nH]n2)=O)CCC2(CCC(C(N3CC(F)(F)C(F)(F)C3)=O)CC2)CC1 Cn1ncc2cccc(C(N3CCC4CN(S(=O)(=O)CCCl)CC4C3)=O)c12 c1(C(N2CCC(C3N(C(Cc4n(C)ccc4)=O)CCC3)C2)=O)ccc(Cl)cc1Cl C12(CNC(C(CC)CO)=O)CCCCC1N(C(=O)C(O)C1CC1)CC2 C(CC(CN(CCCF)CCOCCSCCN)OC)NCCC.C(C)(C)(C)O O=C(C1=CCC(F)(F)CC1)NC1CCN(C(=O)NC(=O)C(Cl)(Cl)Cl)CC1 CC1C(NC(=O)COC(C)(C)COC)CCCN1C(c1cnncc1O)=O c1(C2CC2)nc2c(s1)CCCC2.C12(CC=O)CCCC1CC2 C1(NC(c2nnnn2CCSC)CCOCC=C)CC2CC(OC)C2C1 C(=O)(CCS(=O)(=O)c1cc(Cl)ccc1F)NC(CNC(C=CC(=O)OCC)=O)C N1(C(C(C2CC2)SC)=O)CCCC1CC(C)C.ONC C1(C(=O)NCCCC(C)NC(=O)C=Cc2cnc[nH]2)CC(=O)NC1(C)C Cn1nnc(C(=O)NC2COCC2CNC(C2CC2c2ccccc2)=O)c1N C12(C(C)C)CCC(C(=O)NCC(C)N(C)C3CC3)(CC1)CO2 c1(C(=O)NCC(CN(C(C2C=C(C)CS2)=O)C)O)ncc(N)nc1C N1(C(C(CCC)OCC)=O)CC(NC(C2OCCO2)=O)CC1(C)C C=CCC(CNC(=O)C(F)(F)C(C)O)C(=O)NC1CCC(=O)N(C)C1 c1(COC)nc(NCC2CN(C)C(C)(C)C2)cc(=NC2COC(C)(C)C2)[nH]1 C1(C#N)(NC(C(CC)C)=O)CCN(C(c2ccnnc2)=O)C1 N1(C(CN(C(=O)NCC)C)=O)CCC(C)C(NC(=O)CCC(=O)NC)C1 c1(C(N2C(C)(C)CC(NC(=O)CC3CCCCO3)C2)=O)coc2c1C(=O)CCC2 c1(C2(CN(C)CCNC(c3cn(C)nc3-c3nccs3)=O)CC2)ccc(F)cc1 c1(C(=O)NC(c2nocc2C(=O)NC2CC2C)C)cc2cccnc2[nH]1 c1(C(N2CCCC(NC(C(C)SCCCC)=O)C2C)=O)c(C)nn2ccccc12 c1(CCCN(C)C)cccc(-c2cccnc2-c2cn[nH]c2)c1 N1(C(CC(=O)OCC)=O)CCCCC12CC(NC(=O)CC1CC(C)(C)C1)C2 C(=O)(C(CC(C)C)C(N)=O)NC1C(NC(c2ccn(CCOC)n2)=O)C1.C(C)(=O)O C1(NC(C(C)CC2CCCN2C)=O)CCCN(c2ccc(Cl)cc2)C1=O Cc1cscc1C(=O)NC1CCC(CNC(c2ccc(C(F)F)o2)=O)C1 C1(NC(C(C)(C)c2ccncc2)=O)CC2CCC(C1)N2C(=O)C=CC(N)=O S(=O)(=O)(CCC(=O)N(C)CCOCCCNC(c1coc(C(F)F)n1)=O)NC N1(C(C2(CF)CC(=O)C2)=O)CCNC(=O)C1CCO.c1(SCC)ccoc1C(=O)N C(CCC(C)(C)C(=O)NC1CC2CCC(C1)O2)NC(C(C(C)C)=O)=O c1(NC2CN(C(C(=O)N(C(C)COC)C)=O)CC23CC3)cc(F)c(F)c(F)c1 N1(C(C(=O)NCC=C(C)C)=O)CC(CC2CCC3(C(=O)O)CC23)CC1C CC1CC(C(=O)NC2C3CC2N(C(=O)CCN(S(C)(=O)=O)C)C3)=NO1 C1(C(=O)NCC(CCCC)N(C(c2cccc(O)c2C)=O)CC)CC(=O)CC(=O)C1 c1(C(C(=O)OCC2CCOC2)(F)F)cccc(F)c1Br N1(C(C(COCC)C)=O)CCCC(CC(=O)NCCCOCCCO)C1 C1(NC(CCNC(=O)CO)=O)CCC2(CC1)CN(C(C1CCCCC1(F)F)=O)C2 c1(OC)cc(=NC(=O)C(C)N(C(=O)CC2CC3(CC3)CO2)C)[nH]n1C CN1CCC(OCCC(=O)NCC2(CNC(C3CCNC3=O)=O)CCCC2)CC1 C(=O)(C1=CCC(C)(C)CC1)N1C(C)CC(CNC(=O)CC2CCC(O)C2)C1 c1(C(=O)NC23C(CCN(C(CCC=C(C)C)=O)CC2)C3)cnc2ccncc2c1 c1(C(N2CC(CNC(C(C3(O)CCCCC3)OC)=O)C2)=O)cncc(C)n1 N(C(=NCCCCl)NCCC(O)CO)c1c(C2CN(C)C(=O)C2)nccc1 c1(C(=O)NCCN(C(c2nc(C(=O)NCC=C)sc2)=O)CC)ccc(C)cc1C C1(N(C)C)CCC(C(=O)NC2CCC2NC(C2(c3ccc(Cl)cc3)CC2)=O)CC1 CC(C)(C)C(CNC(=O)CC(O)C1CCCC1)NC(c1ccnc(OCF)c1)=O CC(CCN(C)C)C(=O)N(CCCNC(c1cnn(CC(F)F)n1)=O)C1CC1 c1(OC)c(F)cc(-n2cc(C(=O)Oc3ccnc(Br)c3)nn2)cc1F C(=O)(C(O)P(C)(C)=O)N(CC)CC1CCN(C(c2c[nH]c(Br)c2)=O)CC1 C1(C(=O)NCCN(C(c2c(CSC)noc2C)=O)CC)CCc2c(nnn2C)C1 Cc1cc(C(=O)NCC(CO)NC(C2C3CC4C(C3)C24)=O)nc(C)c1 Cc1cc(C(N2CC=C(CNC(c3ccc(CN(C)C)o3)=O)CC2)=O)nnc1C C1(O)(CC(=O)NCC2(C)CCCOC2)CCCN(C(C23CCC(CC2)C3)=O)C1 c1(C(=O)NCCCOCCN(C(=O)CN2CC3CC3C2)C)c[nH]c2cccnc12 C1(NC(C(c2n(CCC)cnn2)N(C)C)=O)(CC)CCC(O)C1 C1(CCC)(NC(C2CS(=O)(=O)C2)=O)CCCN(C(=O)CC2CCC(=O)NC2=O)C1 C1(C#N)(C(=O)NCC2COCCN(C(C(CC)(C)O)=O)C2)CC2CCC1C2 C1(CC(=O)NC(C2(O)CN(C(c3cccn3C)=O)C2)C)CN2CCN1CC2 C1(CNC(CC#C)=O)CN(C(=O)CCC2CCCN(C)C2)CCC1(F)F CC1CSCC1N=c1[nH]c(=NCCCOC2CCOCC2)[nH]c2c1CCCC2 N1(C(c2c(C)ncnc2)=O)CCC2CCC(NC(=O)C(C(C)C)N(C)C)C1C2 Cc1c(CC(=O)NCC(=O)Nc2ccccc2)cc(N)cc1O C1(C(=O)NCCCCNC(c2c(C3(C)COC3)noc2)=O)COCCC1C C(=O)(CC1COc2ccccc21)NC1(CO)CN(C(c2nn(C)c(O)c2)=O)C1 C(C(=O)N1OC2CCC1CC2)(c1cccnc1)NC(C1CC2CCC1O2)=O c1(C(=O)NC(CNC(C(CSC)(C)C)=O)C(C)C(C)C)cc(C)ccc1[N+](=O)[O-] Cn1nc(C(=O)Nc2c[nH]nc2Br)c2cc(-c3ccc4c(c3)CC(=O)N4)ccc12 c1(C(=O)NC2C(C(=O)Nc3cnc(C4CC4)cn3)C2)cc2cccnc2[nH]1 CC(CSc1ccccc1)C(=O)N1CC(F)(CNC(=O)CCCc2ccsc2)C1 c1(CCC(=O)NCC(CN(C(Cc2cc(C)sc2C)=O)C)O)ccc(Cl)c(F)c1 C12(NC(CC3CCN(C(=O)CCN4CCOC4=O)CC3O)=O)CCCC1C2(F)F c1(C(=O)NCC(CC)NC(c2nccnc2Cl)=O)coc2cc(O)ccc12 N1(C(C(CC)O)=O)CCC2(CC1)CC(NC(c1cnc3c(c1)CCOC3)=O)CO2 c1(C(N(CC(O)CNC(=O)C(=O)C(C)(C)C)C)=O)cccc2c1COC2 c1(OCC)nccc(=NC2CC3CN(C(=O)C(C)SC(C)C)CC23)[nH]1 c1(C(=O)NC(C2CCN(C(C3(P(C)(C)=O)CC3)=O)CC2)C)ccc(=O)n(C)n1 N(C1CCC(NC(=O)CCOCC(F)F)c2ccccc21)C(=O)CCC1CCC1 c1(OCC)cccc(-c2cnc(N3CCCC3)nc2)c1 N1(C(C(C2CCN(C(C(C)C(C)(C)C)=O)C2)(C)C)=O)CCc2c(O)noc2C1 Cc1cc(C(=O)NC2CN(C(c3c(C)cccc3I)=O)CC2C)c(O)c(C)c1 C1(C(=O)NCC2CCCC2Oc2cccnc2)CCCN1C(=O)Cc1cccs1 C(CCCC(=O)N1CCCC(CCC(=O)N(C)Cc2csc(C)n2)C1)OCC Cc1cc(=NCc2cncs2)[nH]c(N2CCN(c3cccc(F)n3)CC2)n1 Cc1cc(C(C)(C)C(=O)N(C2CCS(=O)(=O)C2)CCC(N)=O)n(-c2ccccc2)n1 CC(C)C(C(=O)N1CC(NC(C2C(C)(C)OC2C)=O)C(O)C1)n1cnnc1 c1(C(=O)NCC2C(C)CN(C(=O)C(F)C(C)(C)O)CC2)nccc2ncccc12 C(=O)(CCCC(F)(F)F)N1CCC(C(C)NC(c2coc(N(C)C)n2)=O)CC1 c1(NCCC2N(C(C3=NOC(C)C3)=O)CCCC2C)ncnc2c1ncn2C c1(SCC(N2CCCC(c3ccns3)C2)=O)ccccc1C1CCN1 Cn1ccc(C(N2CCCC(CNC(=O)CSCC#N)C2)=O)c1-c1ccccc1 N1(C(C(C)OC2CCCC2)=O)CCCCC1CCNC(=O)C=CC1CC1 N1(C(c2cc(CCC)on2)=O)CCCC1(CNC(=O)CC(=O)N(C)C)COC Cc1cc2ccc(C(N3CCC(NCc4cnc(F)c(C)c4)C(C)C3)=O)cn2c1 c1(C(=O)NC2CCC(NC(C(CCC=C)(F)F)=O)C2)coc2c1C(=O)NCCC2 c1(OC)ccc(C(C(=O)NCCC2CC2)N(C(C)C)Cc2ccco2)c(Cl)c1 C=CC(C)(C)CC(=O)NCc1ccc(NCC2C3CN(C(C)C)CC23)cn1 C1(C)(C(=O)NCCCCCN(C)C(C2CNC(=O)N2)=O)CS(=O)(=O)C1 N1(C(C(=O)NCC)=O)CCN(C(C2CC2(C)C(F)F)=O)C(CS(C)(=O)=O)C1 c1(CC2CCCN(C(CN(c3nn[nH]n3)C)=O)C2)c(F)cccc1Cl N1(C(C(C=CCCC)O)=O)CCN(C(=O)C2=C(C)CCC2)CC1c1ccccn1 C1(CC(=O)NC(C2CCCC2)CO)CN(C(=O)CC2CCSC2)CCO1 C(=O)(C(C(C)(C)C)N(C)C)N1CC(CNC(c2c(CC)cno2)=O)C(C(F)(F)F)C1 N1(CC(=O)NCC(CC)NC(C2(CC(F)F)CCC2)=O)CCC(C)(C)C1 N1(C(CCCO)=O)CC(C)N(C(=O)CCC(=O)OC(C)C)CC1C.CC=O N1(c2c(C)[nH]c(=NC)s2)Cc2ccc(C(C)C)cc2C1=O C1(NC(CC(C=C)C)=O)CCC(C)(NC(c2cc(-c3csc(C)n3)c[nH]2)=O)CC1 c1(C(N2CCN(C)C3C2C3)C(=O)NC(C)(C)C)cccc(C#N)c1F CC(C)(C(=O)NC(CNC(=O)CCCCCc1cccc(O)c1)CO)C(F)(F)F c1(C(=O)NC2CC(CNC(CCCC(N)=O)=O)C2)ccc2c(c1)NC(=O)CO2 CC(N=c1[nH]c(=NC(CCO)C2(C)CCCC2)[nH]c2ccccc12)c1nccs1 c1(NC(C(N2CCN(C)C(CO)C2)C)=O)cc(O)ccc1-c1ccc(C=O)s1 c1(CC)cc(Cl)ccc1C(N1CC(O)(CCNC(C2(C)CC2Br)=O)C1)=O C1(CC(=O)NC(CCCNC(c2n[nH]c(C)c2Cl)=O)C)CC2(CCC2)CO1 CC(N=c1[nH]c2c(c(=NC3CCC3)[nH]1)CSC2)c1css1 CCC(CC(=O)N1CC(C(=O)NC(C)(C)CC(C)(C)C)CCC1C)CC(C)C c1(C(N(C)CC2N(C(C(C)OCC)=O)CCCC2)=O)nnc(O)nc1O N1(C(C2ON=C(CC)C2)=O)CCOCC(F)(CNC(=O)CSCc2cccs2)C1 C1(NC(c2ccc(SCCC)cc2)=O)CN(C(c2csc(CO)n2)=O)CCC1C C1(CS(N2C(C(=O)OC)CN(C(C)=O)CC2)(=O)=O)Cc2ccc(OC)cc2O1 N1(C(c2cc(OC(C)C)ncc2)=O)CCCC(C)(NC(=O)C=Cc2cscn2)C1 N1(C(CNC(CCNC(=O)NC)=O)(C)C=O)CC2C3CCC(O3)C2C1.C1CO1 N(C1CCc2ccc([N+](=O)[O-])cc21)C(=O)Nc1nc2ncc(C)cn2n1 c1(SC)cccc(CNC(C)(C)C)n1.C12C3CC(CC13)C(=O)N(C)C2 Cc1cnc(C(N2CCC(N(C)C(C3(C)CC(O)CN3C)=O)CC2)=O)cc1C C(=O)(CC(C)(C)CC(=O)OC)Nc1cccc(CNC(C2(SC)CC2)=O)c1 c1(CCOC(c2c(C)scn2)=O)cn2ccsc2n1 CC1(C)OCC2CC12C(N1C2CCC1(CNC(=O)Cc1nc[nH]n1)CC2)=O N1(CC(Cc2c(C)ccs2)O)CC2(CCC(=O)O2)C1 C1(NC(c2cc(CF)on2)=O)COC2(C1)CN(C(c1c(Cl)csc1Cl)=O)C2 n1(CCC(=O)NCC2CN(C(CCc3c(C)ncs3)=O)C2)cnc2ccccc12 C(CC(C)(O)CC)NC(C1(CCC=C)CN(C(C2CCCC2F)=O)C1)=O Cc1cc(C(=O)NCC(=O)Nc2cn[nH]c2)cc(C#N)c1 C1(NC(C(C)c2ccco2)=O)CC(C(F)F)(NC(c2csnc2Cl)=O)C1 c1(C(=O)NC(C(NOCCC#C)=O)CSCC)cccc(C#N)c1C C(C(C(C)(C)C)NC(c1cc[nH]c(=N)n1)=O)NC(CC(C)OC)=O C(C1=NOC2CCCC12)Nc1n(-c2cccc(Cl)c2)nc(C)c1C CC(C)C(C(=O)NCCC(C)CCNC(=O)CCN1CCOC1=O)OC(F)(F)F c1(CNC(C2(CCNC(C(C)c3cc[nH]n3)=O)CCC2)=O)ncccc1F C1(NC(CC(CCC)O)=O)Cc2ccccc2C1NC(c1cc(C)nc(Cl)c1)=O c1(COCC(=O)N(CCc2cn(CC3C4COCC34)nn2)CC)cc(OC)ccc1F c1(C(=O)OC)[nH]c2cc(F)ccc2c1C(C)C.c12ccc(cc1)CN(C)C2 N1(CCC(=O)NC2CN(C(CNC(CC)=O)=O)C2)CCc2ccccc2C1=O N1(C(C2(C)CC2(F)F)=O)CC(F)CC1C(=O)NC(C(O)CO)C1CC1 C(C(=O)N1CC2CC2(NC(c2cc[nH]c2C(C)C)=O)C1)(C(C)C)NC(C)=O c1(C(=O)NCC2(COC)CN(C(=O)C=Cc3cnccn3)C2)cc2cscc2s1 c12ccc(C(F)(F)F)c(c1)NC2=O.C1(C(C)N(C)C)CN(C(=O)CCF)C1 Cn1cnc(C(=O)N(CCCNC(C2CC2(Cl)Cl)=O)C2CC2)n1 N1(C(C(CN(C)C)(F)F)=O)CC=C(C(=O)N2CC(C(C)(C)O)C2)C1 c1(C(N2C(CCCNC(C3(C=C)CC3)=O)CCC2)=O)cnc2c(c1)COC2 Cc1nn(C)c(N)c1C(=O)NC1(CC(=O)NC2COCC2C(N)=O)CCC1 c1(C(=O)NCC(CNC(C(CC)C#N)=O)C)cn2cccc(C)c2n1 C(=O)(CCCCC(C)(C)C)N1CCN(C(C(CCCOC)C)=O)CC1CCO c1(SCCNC(N=c2[nH]nc(CC(C)C)s2)=O)ccc2c(c1)OCCO2 C(=O)(CCCC(N)=O)N(C(C(N1CCC(N(C)CCO)C1)=O)(C)C)S(C)(=O)=O c1(OC)cc(CN(C)CCN(C(C2(F)COC2)=O)C2CC2)cc2c1OCO2 c12cccc(c1)NC(=O)CN(CC)C2=O.c1(C(C)(C)C)ccc(OC)cc1 CC1(O)CN(C(=O)C(c2cccs2)NC(c2cccs2)=O)C1 Cc1ccc(C(=O)NCCC2CCC(NC(c3cc(CCO)on3)=O)C2)c(F)c1 C1(NC(C=C(CCC)CCC)=O)CC(O)CN(C(=O)Cc2cc(C)ns2)C1 Cc1ccnc(C(=O)N(C)CCOCCNC(=O)Cc2cc(Cl)sc2Cl)c1N c1(C(=O)NCCC2(NC(Cc3nnc(C)s3)=O)CC2)cnn2cccc(Cl)c12 c1(C(=O)NCC(C)N(C(c2ccc(C)c(C#N)c2)=O)C)ccc2nnc(O)n2c1 C1(NC(C2CC3CCC2O3)=O)CC1C1CCN(C(C2(C(F)F)CC2)=O)CC1 C(=O)(CC(=O)NC(C)(CNC(=O)CCc1cnn[nH]1)CO)OCC c1(N(C(N2CC(C)=C(C)C2)=O)C)nc2ccccc2[nH]1 C1(CC(C)NC(C=CCC)=O)CC2CCC(C1)N2C(C1OCCC1C(C)C)=O C=CC(C)CC(=O)NCCC1CCCN(C(=O)CNC(=O)CC(F)(F)F)C1 Cc1cccc(C(=O)NC2CCN(C(C3(CC(C)C)COC3)=O)C2)c1F CC1C(C(=O)NCC2CCCCN2C(=O)CCCc2ccsc2)C1C1CC1 Cn1c(O)ncc(C(=O)NCCC2CCCN(C(=O)CCC#N)C2)c1=O CCCCC(C(=O)N1CC(C)(OCC(=O)NC2(C)CC2(F)F)C1)C(C)C CC(C)CC(O)C(=O)NC1CC(C)CN(C(c2cccc(F)c2C(F)(F)F)=O)C1 c1(C(N2C(C)C(C)(C)CC2)=O)coc2c1CN(C(=O)CC1CCC(O)C1)C2 c1(C(=O)NCCC2C(C)CN(C(=O)CNC=O)C2)ccnc(Br)c1N c1(C(=O)NC(CCCNC(C2=C(C)CC2)=O)C)nn(C)c2c1CCC2 C12(C(=O)NCC3CC(NC(C(c4ccc(CC)s4)=O)=O)C3)CCC(CC1)CO2 Cc1cc(O)ncc1CN(C1CC(C)(C(C)(C)C)C1)C CC(C)(CCCCNC(c1cncnc1)=O)NC(C1CC1Cl)=O C1(CNC(C2CSCCS2)=O)CCN(C(=O)Cc2ccc(Cl)nc2)CC1(F)F Cc1cc(N)c(Br)cc1C(=O)OCC1CC2(C(=O)OC(C)(C)C)CC1C2 C1(CNC(=O)Cc2cccs2)COCC1NC(=O)Cc1nc(C2CC2)cs1 C1CCCCCC(=O)N1.C1(N)CCCCN(C)C1=O.CC(O)C=O.C1C(=O)N1 C1(NC(c2cc(Cl)ncc2Cl)=O)CC2CCC(C1)N2c1ccnc(CO)n1 c1(OC)cc(-c2csc(CN3CCCC(CO)CC3)c2)cc(C)c1 Cn1ncc(C(=O)NC2CCCN(C(C3CCCCCC3)=O)C2)c1S(N)(=O)=O CCC(F)(F)C(C)(C)NC(=O)C(F)C1CC(NC(=O)C(=O)NOC)C1 C(=O)(CC(O)COC(C)C)NC1CC(C(F)F)(NC(c2cc(CC)on2)=O)C1 Cc1c(Cl)ccnc1C(=O)NC(C1CCCCN1C(c1cc(F)n[nH]1)=O)C C1(CC(C)(C)C)CN(C(=O)CS(C)(=O)=O)CC1NC(c1cc[n+]([O-])cc1)=O c1(N2CCC(C3C(NC(CC)=O)CS(=O)(=O)C3)CC2)nc(Cl)ncc1[N+](=O)[O-] C1(C(N(CCCOCCN(C(COCC=C)=O)C)C)=O)CCCC2(C1)CC2(F)F C12(NC(=O)CN3CCC(O)CC3)CCC(CC1NC(C1CC3(C1)CC3(F)F)=O)C2 c1(C(N2CCC(C(C)NC(c3cc(F)ccc3Br)=O)C2)=O)cc2cnccc2[nH]1 N1(C(c2cn(CCC=C)nn2)=O)CCC2(CC1)CN(C(=O)C1=CCC1)C2 C1(CNC(C(CN(CC)CC)F)=O)CC(O)CN1C(=O)C=Cc1ccc(CC)o1 c1(OC)ccc(-c2ccc(F)cc2C(N)=O)cc1C#N C1(CNC(COCCCCCC)=O)CCN(C(=O)C(n2nccc2C)C)CC1 N1(C(C2C(c3cn(CC(C)C)nc3)C2)=O)CCC(CCNC(=O)CCC#N)CC1 c1(C(=O)NC2CCCN(C(c3c(Cl)ncc(N)c3)=O)CC2)cccc2cnsc12 N1(C(c2c(N)nccc2)=O)CCC2(NC(c3ccnc(C(F)F)c3)=O)CCCC12 C1(CNC(CCCCC#C)=O)CCN(C(=O)C(c2ccc(C)cc2)C)C12CCC2 c1(CC(=O)NCC(CNC(c2c(OC)n(C)nc2C)=O)O)cccc2nsnc12 C(c1cc(Br)ccc1F)=CC(=O)NCC1C2CC1N(C(C1CC1F)=O)C2 c1(C(=O)NCCNC(N(C)Cc2ccno2)=O)cc(F)cc(F)c1Br C12(CNC(C3N(C(=O)CC4(O)CCC4)CC3)=O)CC(CCO1)C2 Cn1cnc2cc(-c3cn(C(C)(C)CC(=O)N(CC(F)F)C(C)(C)C)nn3)ccc12 c1(CC)cc(F)ccc1O.C1(CC=O)CCCCN1C(=O)NCCC1CC1 N1(C(C(CNC(=O)OC)C)=O)CCC(C2CC2)(CNC(C23CC(C2)C3)=O)C1 C1(C)(CN(C(C(C)OC)=O)C)CCCC1NC(=O)CCNC(N)=O C1(C(N(C2(C(=O)NCC34CCCC3C4)CC2)C)=O)CC(C)(O)C1 N1(C(C=Cc2occ(C)n2)=O)CCN(C(c2cc(CO)[nH]n2)=O)CC1C1CC1 c1(C(=O)NC(CC2CC(F)(F)C2)C(=O)O)cc2nc(Cl)ccc2o1 c1(C(N2CCCC(NC(C=CCCC(N)=O)=O)C2)=O)ccc2nc[nH]c2n1 C(=O)(C(Cn1cncn1)NC(C1CC=CC1)=O)NCC(C)Cc1ccco1 c1(CC(=O)N(CCC(=O)NC2CC(OC)C2)CC2CC2)cccnc1F c1(C(=O)NCCNC(C(CC)OC)=O)cc(-c2ccncc2)ccc1OC C1(CNC(CC2C(C)(C)OCC2)=O)C2CCCC1N(C(=O)C#CC1CC1)C2 c1(C(=O)NCCCN(C(=O)Cc2n[nH]c(C)n2)CC)cnc(C(C)(F)F)s1 CCCCCC(O)C(=O)N1CC2CC1CN2C(c1scnc1C(F)F)=O C(=O)(CC1=CCOCC1)NCC1(F)CCC(CNC(c2c(C(C)C)n[nH]c2)=O)C1 C#CCCCCCCC(=O)NC1CCC2CCC1N2C(c1cccc(CO)n1)=O C#Cc1cnc(C(=O)NC2C=CCN(C(c3ccc(CC)cc3F)=O)C2)c(C)c1 C1(C(N(CC(=O)OCC)C2CC2)=O)CCN(C(c2ccsc2C)=O)C1(C)C Cn1cc2c(n1)CCC(C(=O)NC1CC(NC(c3cnc4n3CCC4)=O)C1)C2 N(C1CCc2c(Br)cccc21)C(C(CCS(N)(=O)=O)N)=O c1(C(=O)NCC2N(C(c3c(C(=O)OC)ccs3)=O)CCC2)ccc(F)c2occc12 C1(C(N(CC(C(=O)OC)C)CC(N2CCOCC2)=O)=O)CC=CCC1C(=O)OC c1(C(=O)OC)ccc(C(=O)NCC(C)N(C)C(c2nnn(C)n2)=O)o1 C1(CC)CCC(C(=O)NCC(CO)NC(c2cnn(C(C)(C)C)c2)=O)O1 N1(C(c2nc(Cl)cs2)=O)CCC(c2ccccc2)(C(N2CC=CC2CO)=O)C1 Cc1cc(C(=O)NCC(C)(CC(C)C)NC(C2CCCO2)=O)nnc1O C1(C(=O)NCC2(C(F)F)CCOC2)CC(O)(CNC(C2N(C)CC2)=O)C1 Cc1nnc2n1CCCC2CNc1ccnc(N2CCC(NC(C)C)C(F)C2)n1 C1(C(=O)OC)C2=C(CCN(c3ccccc3N3CCC3)C2=O)N(C)C(=S)N1C(C)=O C1(NC(C(C)OCC)=O)CCOCC1NC(c1cn(C)nc1-c1cccnc1)=O C1(CNC(=O)CC2CC2)CCC(C(=O)NCCc2cccnc2)O1 C1(CN(C(Cc2nc(C(C)OC)sc2)=O)C)CCN(C(C2(C)C=CCC2)=O)CC1 CCCC(C(=O)NCC1CC2(CC2)CN1C(c1nccc(C(F)F)n1)=O)C(C)C C1(C(=O)OC)(NC(=O)CC2CN(Cc3c(Br)cncc3Br)C2)CCCCCC1 C(=O)(CN=C(NC1CCCC1)N1CCCC(n2ccnn2)C1)NC(CC)C c1(N2CC(C(C)NC(C(C)Cc3ccccn3)=O)C2)ncc2c(n1)NC(=O)C2 c1(C(=O)Nc2c(O)ccc(OC)c2OC)cnn2c1C(C)CCC2 C(CCNC(C1C=CCS1)=O)(C(=O)NC(c1nc(C)cs1)CO)OC CC1(C)CC(NC(c2ncccc2CO)=O)CN(C(c2csc(=N)[nH]2)=O)C1 CC(C)(CC(C(=O)NCCOCCOCCCNSC(F)F)c1ccccc1)C(=O)O C(C1CCOCC1)=CC(=O)N(C1CCN(C(=O)Cc2cn[nH]c2)C1)CC#C C12(C(N3CC(N(C(c4cc(C)ns4)=O)C)C(O)C3)=O)CCC(CF)(C1)OC2 C1(C(=O)NCCCNC(CCC=CC)=O)(Cc2ccccc2)CCCCC1 N1(CC(=O)NC2CCN(C(c3cc(C(C)=O)oc3)=O)C2C2CC2)CCCCCC1=O C1(CN(C(C(=O)NCCCC)c2cc[nH]n2)CCC#N)CCCCC1 C(=O)(C1=CS(=O)CCC1)NCC1C(CCC)C1 Cc1nc(C)c(C(N2CC=CC2C(=O)NCc2ncsn2)=O)o1 C1(NC(=O)OC)CC2CCCC(C1)N2C(=O)NCC1C(C(F)(F)F)C1[N+](=O)[O-] C1(C(=O)NC2CC(C(C(N3C(C(=O)NC)C=CC3)=O)F)C2)CC2COCC2C1 C1(CC(CO)NC(=O)NCCn2ccc(Br)n2)CCC(F)(F)CC1 c1(CNC(CCOCC#C)=O)cn(CC(C)NC(=O)COC)nn1 N12CCC3(CCN(CC3)C1=O)C2.O=C(C=NOC1CCCCC1)NC1CCOC1 C(CNC(c1cc(F)cs1)=O)(CC(C)C)NC(c1cc(C)oc1)=O C1(C(N(C)CCOCCCNC(C2CC2Cl)=O)=O)CCCCC1n1ccnc1 N1(C(CN2CC(C)(C)C2)=O)CCCCC(C2CN(C(=O)C(=O)C(F)(F)F)C2)C1 C1(NC(=O)Cc2cc(F)cc(Cl)c2)CCC(O)CN(C(=O)C(F)=CCCF)C1 C1(C(=O)NC2C(SC)COC2)CN(C(c2cnn(C)c2Cl)=O)CCC1(C)C C(C)(C(CC(=O)N(C)Cc1ccn(C)n1)NC(=O)C=Cc1ccn(C)c1)OC N1(C(c2c(C)n(C3CC3)cc2)=O)CC2C3CCC(C2C1)N(C(=O)C(C)N(C)C)C3 c1(C(c2ccc(F)cc2)NC2(CC)CC2)ccnc(Br)c1C C(=O)(C(CNC(c1ncccc1O)=O)CC(C)C)NC(CC#C)CC#C C(=O)(CC(CC(C)C)NC(C1CCC(N(C)C)C1)=O)NCc1cc(C)on1 c1(C(=O)NCCCOCCCNC(C2N(C)CCOC2)=O)ccc2occc2c1 C1(C(=O)NCCC2ON=C(C)C2)(CNC(=O)C(C)C2CCOC2)CC2(CC2)C1 Cc1ncoc1C(=O)N(CCCNC(=O)CCSCC(N)=O)C(=O)N.C1CC1 C1(NC(C(C=C)(C)C)=O)CCN(C(c2ccc(CC(=O)OC)cc2)=O)C(C)C1 c1(CC)oc(C)cc1C(=O)NC(CN(C)C(C1(CC2CC2)CCC1)=O)C c1(C(=O)NCCCN(C)C(c2cc3ccncc3[nH]2)=O)cccc2cncn12 c1(C(=O)NCCC2CN(C(C=CSC)=O)C2)ccc(C)c(CO)c1 C1(C)(CC)CCC(C(=O)NCCC2(C(=O)N(C3CCOC3)CC3CC3)CC2)O1 N1(C(C(CC=C)OC)=O)CCCC(CC(=O)N(C2CCN(C)C2)CC)CC1 C(=O)(C1CCCc2nc[nH]c21)NC1CC2(CN(C(C3(CC)CCC3)=O)C2)C1 Cc1c(NC(N2CC(NC3CC(=O)N(C4CCCCC4C)C3)C2)=O)cccc1Cl C1(C(C)C)(C(C)C)CN(C(=O)C(F)(F)C(C)O)CC1N(C(=O)C(F)(F)F)CCO c1(C(=O)NCCC(C)NC(C(C)SC(C)C)=O)cnnn1C(C)C CC1C(CC(=O)NC2(c3ccccc3)CC(NC(C3CSC3)=O)C2)C1(F)F C(=O)(C1CCc2cccnc21)NC(CC=C)CNC(=O)Cc1cc[nH]n1 C1(O)(C(C)NC(C(C)=C2CC2)=O)CCCN(C(C2(C#N)CC23CCC3)=O)C1 c1(CC)cc(C(=O)NC2CC(N(C(=O)CN3CCC(C)C3)CC)C2)nn1C CCC(C)(C(=O)OC)NC(=O)CC1CC(F)CN1C(=O)C(CN(C)C)N(C)C Cc1cc2cc(C(=O)NCC3CC(NC(C4(N(C)C)CCC4)=O)C3)ccc2[nH]1 c1(C(=O)NC(C)CC(C)NC(=O)CO)c(S(C)(=O)=O)cnn1C CC1CCC(C(=O)NC23CCCC(NC(=O)CC4=CCCC4)(C2)C3)CC1C C1(C(=O)NCCC2COC(C)(C)O2)CCC2(CC2)N1C(c1ccc(CO)s1)=O Cn1nc(SCC(N2CCCC2C(=O)Nc2cnc(C#N)cn2)=O)cc1CO c1(OCC)cnc(NC2CCC(C(=O)NCC(O)CO)CC2)nc1 C1(C(=O)NCCC(C)N(C(c2c(C)ccnc2O)=O)C)CCc2ccccc2O1 c1(Cn2cc(-c3cnc(C4CC4)o3)nn2)ccc(C(F)(F)F)cc1.O=C(CF)N C(c1ccccc1OC(F)(F)F)=CC(=O)NCCNC(C1CC(C2CCC2)C1)=O N1(CCC(N2CCC(OCCNC(Cc3c(C)cco3)=O)C2)=O)CCCCC1=O c1(C(N(CCCN(C)C(c2cnnn2C)=O)C)=O)sc2sccc2c1Cl NC(=O)CC(O)C(=O)NCC1CC(C(=O)NCc2nn[nH]n2)=NO1 C1(C(=O)Nc2n(C)nc(O)c2)CCCN(Cc2cccc(Cl)c2F)CC1 CC(C)C(F)(F)CC(=O)NC1CC(C)(NC(=O)CC2CC3CCC(C2)C3)C1 C(=O)(C#CC(C)(C)C)NCC(c1ccc(OC)cc1)NC(=O)C(O)C1CC1 c1(C(=O)NC2(CO)CCN(C(c3ncc(C)c(C)c3)=O)C2)cccc2[nH]ccc12 C1(C(=O)NC2CC(NC(=O)COCc3nc[nH]n3)C2)CCCCC1C1CC1 N1(C(C2CN(C(C)=O)C2)=O)CC2CCC(C1)C2CNC(C1CCCC2(CC2)C1)=O N1(C(C(C)NC(=O)C2CC2)=O)CCCC(CO)(CNC(C2COCC2(C)C)=O)C1 Cc1noc(C)c1NS(=O)(=O)CC1CNCCC1C.C12=CC=C(C=C1)C2 C1(NC(CCC(=O)N(C(C)C)C)=O)CC2CCC(C1)N2C(=O)C(C)C(C)O CCCCC(C)(F)C(=O)NCC1C=CCN1C(c1nc(C)c(C)nc1C)=O CC1CCN(C(=O)CCC2CCOCC2)CCN1C(=O)CCc1cc[nH]n1 N1(C(CCC(=O)N(CCC)CCC)=O)CCCCCC1CNC(=O)C(O)C1CC1 N1(C(c2[nH]c(=NCC)sc2)=O)CCn2ncc(CN(C(=O)C3=CCCS3)C)c2C1 c1(OC)cc(C(=O)NC2CCC2NC(=O)C(C(C)C)CNC(C)=O)cc(Cl)c1 N1(CC(=O)NCC(C)(C2CC2)NC(C=CCN(C)C(=O)C2CC2)=O)CC(=O)NC1=O N1CC2(C)CC1CO2.C(c1ccncn1)=CCn1cc(CCn2ncc(C)c2)nn1 C(F)(C(=O)NNc1ccc(Br)c(O)c1)=CCCC N1(C(C(C=CCCC)O)=O)CCC(C)C(N(C(=O)CCCC)C2CC2)C1 C(C)(CC(C)(C)C)Nc1cn(C2(CCNC(C3C(OCC)C3)=O)CC2)nn1 C(C)(C)(CCC(=O)NC1CCCN(C(c2cncn2-c2ccccc2)=O)C1)OC CCCCC(C(=O)NC(C)(CC)CC)NC(=O)C(N1CCOCC1=O)C CN1CCC(NC(C2CC3CCC2N3C(C2CN(C3CCC3)C2)=O)=O)CC1=O CN1Cc2ccccc2CC1C(N1CC2C(C1)N2C(c1c(O)cccc1O)=O)=O N1(CC(=O)NC(C)C)CCCC(C2CCCN(C(=O)C3=CCCCC3C)C2)C1 C(CCc1ccccc1)(C(C)NC(=O)C=CSC)NC(C=C(CC)CC)=O c1(SC)cc(C)ccc1NC(=O)N(C)C(=O)NCC1C2COCC12 N1(C(C(c2ccccc2)C)=O)CCOC(C)(CNC(=O)Cc2ccc(Cl)cc2F)C1 C1(C(=O)NC2CC(C(C)C)OC2)CCN(C(c2cnsc2)=O)CC1(C)C C1(C)(C(=O)NCC(C)(C)CCO)CCCN(C(c2cc3n(n2)CCC3)=O)C1 Cc1nc[nH]c(=NCCC2CCCC2)c1Br.c12c[nH]c(c1)N(CCO)CC2=O N1(CCONC(CC2N(C(CN(C)C3CC3)=O)CCC2)=O)CCOCCC1C1CC1 c1(C(=O)NCC(C)CN(C)C(c2coc(C3CCOCC3)n2)=O)cncc(F)c1 C(=O)(CCS(=O)(=O)NCC(N1CCCC1)=O)NC(C)CC(=O)NCC#CCl N1(Cc2cccc(OCC)c2C)CC2CCN(C(c3cnnn3C)=O)C2C1 C1(C(=O)OC)CC(n2cc(C3(C)CSC3)nn2)CN1C(=O)CC1OCCC1(C)C c1(C(N2CCC(NC(CC=C)=O)C(C)(C)C2)=O)c[nH]c2cccc(F)c12 c1(C(=O)NC2CC(C)(NC(c3c(C)c(C4CC4)on3)=O)C2)ccc2nc[nH]c2c1 Cc1ccc(NC(=O)CCC2(C)CCCN2C(c2ccnc(C)n2)=O)c(C)n1 C1(CC)CCC(O)(C(=O)NC2CCC(N(C(=O)Cc3cnn(CC)c3)C)CC2)C1 n1(C(C)C)cnnc1CNC(C1(N2CC(O)C2)CCC1)=O C(=O)(C(C)(F)CCCC)NCC(CC(C)C)NC(c1nnc(C#C)s1)=O CC(C)CC(C)CC(=O)NC1CCN(C(c2c[nH]nc2OCC(F)F)=O)C(C)C1 C12(C(=O)NCC3CC(NC(C4(OC)CCOCC4)=O)C3)CCC(CC1)C(C)O2 N1(C(C(=O)Nc2c(-c3cccc(C)c3)cccc2)=O)CCC2(CCCCC2)CC1 C1(C(C)NC(C2CC2CF)=O)CN(C(c2csc(-c3nc[nH]n3)n2)=O)CCO1 c1(C2(C)CN2)nnnn1CC1(c2ccoc2)CC1.N1(C(=O)OC)CCCCC1 C12(CNC(C=CC(C)(C)C)=O)CC(NC(=O)CC3COCCO3)(C1)C(C)(C)O2 N1(C(c2ccc(C)nc2)=O)CCC2(CC1)CC(NC(c1cnc(S)[nH]1)=O)CO2 N1(CC(=O)NCCC(C)NC(c2ocnc2C2CC2)=O)CCCNC1=O N1(C(c2cn(C(C)(C)C)nc2)=O)CCCC(O)(CNC(=O)CC(F)(F)F)CC1 N1(Cc2[nH]c(C)nc2C)CC=C(CCNC(c2ccc(C(=O)OCC)[nH]2)=O)CC1 C1(CNC(CCN(C(C)=O)C)=O)C(C)CCN1C(=O)C(C(C)C)n1cnnn1 c1(CC(=O)NCC(C)CNC(=O)C(N2CCOCC2=O)C)ccccc1C(N)=O N1(C(c2ccnc3[nH]ncc23)=O)CCN(C(c2sccc2Cl)=O)C2(CCC2)C1 c1(C(=O)NC(CC=C)CNC(=O)CC(c2cccc(F)c2)O)ccc(C)nc1O CC1(C)CCC(NC(=O)C(CC2CCC2)NC(=O)CCN2CCCC2=O)C1 N1(c2cc(C(=O)NC3(CC)CCC3)[nH]c2)CCC(C(C)NC(C(C)OCC)=O)C1 N1(C(C2C(NC(C)=O)CCC2)=O)CC2OCC(NC(c3cnn(C)c3)=O)C2C1 c1(CC)cc([N+](=O)[O-])ccc1C(=O)NCC(C)(C)NC(=O)CC1CC(C)OC1C c1(C(=O)NCC2(O)CC(Nc3ncnc(Cl)c3CO)C2)cccc2nccn12 C12(c3nc(-c4ccc(C)cc4Cl)nn3Cc3cnoc3CO)OCCCC1C2(F)F CCC(C)(C)CC(=O)NCC(CCNC(C1CC(C)(C)CCO1)=O)OC C1(CC)CN(C)C(=O)CN1C(=O)CC(O)CNC(C1C(C)C1C)=O C1(C(C)C)CN(C(C2CCC(C(N)=O)O2)=O)CCN1C(c1ccn(C)n1)=O c1cc([N+](=O)[O-])c(N)cc1F.C(=O)(CC(C)C)NCC.C1(=O)CCO1 C12(NC(c3ccc(Cn4ccnc4)cc3)C)CC3CC1C2C3N N1(C(C2c3nnc(C)n3CC2)=O)CCC2OCCCC2(c2nn[nH]n2)C1 C1(CNC(C23N(C(c4c(C(C)C)noc4)=O)CC(C2)C3)=O)CC2CCC1CC2 C#Cc1cccc(C(N2CC(CC(C)NC(C3(Br)C(C)C3C)=O)C2)=O)c1F C1(C(N(CCN(C(c2c(O)ccc(C(C)C)c2)=O)C)C)=O)CN2CCCN1CC2 CC1(C)CC=CCN(C(=O)CC(C(F)F)NC(=O)C=Cc2ccc[nH]2)C1 c1(NC(CCOC)CNC(=O)C(C)SC(F)(F)F)nc(OC)cc(OC)n1 CN1CCC(NC(C2(NC(=O)CC3CC4(CC4)CO3)CCC2)=O)CC1=O c1(C(=O)OC)ccc2c(c1)C(C)CN2C(c1ccnc(NCC(F)(F)F)c1)=O C1(n2cc(C3(N(C)C)CC3)nn2)CC2CCC1(NC(c1ccc(=O)n(C)n1)=O)C2 c1(C(C)NCCN2CCCCC(O)C2)cccc(S(N)(=O)=O)c1 Cc1nc(C(=O)NCCC2CN(C(C34CC(F)(C3)C4)=O)CCO2)cn1C Cc1sccc1CC(=O)N(CCCC(=O)NCC(c1ccco1)O)CCO c1(C(=O)NC(c2ncccn2)(CC)C)ccc(Br)nc1[N+](=O)[O-] C(CCC(C)(C)C)(C(=O)NC(C)(C)CC)N1CCN(CC#C)CC1 c1(C(N2CC(COC)(NC(C3CC(C)OC(C)C3)=O)C2)=O)ccc2c(n1)CCO2 C=CC(C(=O)N(CC(C)(C)NS(C)(=O)=O)C)c1ccccc1 N1(Cc2cccc(C)c2)CCCC(C)(C(=O)NCc2ccnc(OC(F)F)c2)C1 C(=O)(C1=CC2(CN(C(=O)CCc3nc(O)n[nH]3)C2)OC1)N(C)Cc1cscn1 c1(C(C)NC(=O)CC2CCCN2CC=CC(C)(C)C)c(F)cccc1F C1(C(=O)NCC2CN(C(C=Cc3cn(C)nn3)=O)C2)CCc2cncn2C1 N1(C(C2CCN(Cc3cn(CC)nc3)CC2)=O)CCCCC1C(=O)OC CC(C)CC(C)(O)C(=O)NC1CC2(C1)CC(CNC(=O)CCOCC1CCC1)C2 N1(C(CC(CNC(C(=O)NC(C)C)=O)C2CCC2)=O)CC(O)C(C)(C)C1 c1(C(=O)NCCCNC(COc2c(C)cccc2)=O)cccc(F)c1I n1(CC)nccc1CC(=O)NC(C(=O)Nc1ccsc1)c1ccoc1 C(c1cc[nH]n1)=CC(=O)NCC1CC1NC(=O)CCc1ccsc1Br N=c1nc(N2CCCC(C(N)=O)CC2)[nH]c(=NCCc2nc3ccccc3[nH]2)[nH]1 c1(C(C(=O)NCCNC(C2(C)CC2(F)F)=O)O)cccc(Oc2ccncc2)c1 C(=O)(CC(CC)SC)NC(C1(CNC(c2c(CC)noc2)=O)CC1)C Cc1nn(CC(N2CC(CN(c3nnc(O)s3)C)C2)=O)c(C)c1C(F)(F)F N1(C(c2n(CCC)nc(C)c2)=O)CCC(C2(NC(C34CC5CC3C4C5)=O)CC2)C1 c1(C(N2C(COC)C(C(=O)OC)C(OC)C2)=O)cc(Cl)cc(Cl)c1F C(=O)(C1=NN(CCO)C(=O)CC1)NCCNC(=O)CCC1CCCC1 N1(C(C(C)=C2CCC2)=O)CCCC(C)(NC(c2cnc(C)n2C)=O)C1 CC1CC(NC(C2(CF)CC3(CCC3)C2)=O)CCN1C(=O)CCC1CCCCC1 C(=O)(C1CCc2c[nH]nc21)N1CCC(OC)(CNC(=O)C=CSC)C1 c1(C(N(C2CN(C(C3CCC(C)O3)=O)C2)C)=O)coc2c1NC(=O)CCC2 C(=O)(C1CCCn2cncc21)N(CCNC(C(CC)OCC)=O)CCOC c1(-c2cc(OCC)cc(C)c2)cc(C(=O)NCc2nccn2C)c2[nH]ccc2c1 CCCC(CC)CCC(=O)NC(CC)CCCC(=O)N(c1ccc(CSC)cc1)C Cc1cc(-n2nc(C3CCOC3)nc2C2CCCS2)ccc1O C(=O)(CCC(C)(C)NC(=O)CC1CCCC12CC2)NC(COC(C)C)C Cc1cc(C(N2CCC(CF)(NC(C3CC=CCC3C)=O)C2)=O)cc(O)c1 N1(CCNC(CCN(C)CC)=O)CCC(NC(C2CCOC2C)=O)CC1 C1(C(=O)NC)CC2(C1)CC21CC1.C(C1C(=O)N(C2CC(C#N)C2)CC(=O)N1)OC c1(CCNC(=O)NCCc2cncs2)cc(Br)cs1 Cc1sc(CC(C)C)nc1C(=O)NC1CCN(C(C2CC2(c2ccccc2)F)=O)C1 CCC(CNC(C1(c2ccccc2)CCN(C)C1)=O)(CC)NC(=O)CCCC C1(C(=O)NC(C(=O)N(C)CC2CCCCO2)CC2CC2)CCCCC(=O)C1 N1(C(C(n2c(C)ncc2)C)=O)CCn2ncc(CNC(c3sccc3F)=O)c2C1 C1(CC(=O)NC2C(NC(c3ccn(C)c3)=O)C2)SC2=NCCN2C1=O N1(C(C2C(C(C)(C)C)CC2)=O)CCCC(CCNC(=O)C=Cc2cccs2)CC1 CC(C)C(CCC(=O)NCCC1CC(=O)N(C)C1)NC(c1ccc(O)cn1)=O CCC(O)CC(=O)NC(CCOCCO)C(=O)Nc1ccsc1 C(=O)(CCCC(F)(F)C(F)(F)F)NCC(CCNC(CC(C)C)=O)O c1(OC)ccc(-c2ccc(C)c(Cl)c2)cc1S(=O)(=O)N1CC2CN(S(C)(=O)=O)CC12 c1(OC)ccc(C(F)(F)F)cc1CO.N12CCC(CC1)OCC2 c1(C(=O)NCC(N(C(C(CCC)C)=O)C)C2CC2)c(C)nn(C)c1Br n1(C(CC)CC)nc(-c2cccc(N(C)C)c2)nc1-c1ccc[nH]1 C1(C(N2CCC(C(C)NC(c3n(C(C)C)ncc3)=O)C2)=O)CC2(CCO1)CC2 C1(N(C(Cc2c(C)occ2)=O)C)C2CN(C(=O)CC(C)C3CCCC3)CC12 N1(C(c2[nH]cc(CC)c2)=O)CCC2CN(C(C3CC3c3ccccc3F)=O)C2C1 CCC(CCC(=O)N(C(C)CC(C)CC)C)NC(c1ccn(C(C)C)n1)=O N(C1CN(C(C2Cc3ccc(F)cc3C2)=O)Cc2ccccc21)C(C=CCC)=O Cc1ccc(Br)c(C(=O)NC2CC(C)CN(C(c3cc(N)ccn3)=O)C2)n1 C1(COCCOC)COCCN1C(C1C2CCC1(C(F)(F)F)C2)=O.C(C)(C(=O)OC)O n1(C(CC)CC)ncc(C(N2C(CNC(=O)CC3CC34CC4)CC3CC23)=O)c1C N1(C(CN2CC(C)C2)=O)CCOC2CCN(C(=O)C(F)C3CC3)CC12 CCC(N=c1nc2ncn(C)c2c(NCC=CCOC)[nH]1)c1cccc([N+](=O)[O-])c1 C1(C(N2CCCN(C(c3c(C)scc3)=O)CC2C)=O)Cc2c[nH]cc2S1(=O)=O CCCCC(CC)CC(=O)N(C)CC1(NC(c2c(F)cc(C)cc2F)=O)CC1 C1(C(C)C)CN(C(c2cc(F)cc(Cl)c2)=O)CCN1C(c1cc(Cl)c(Cl)s1)=O CCC(CC(=O)N1CCOC(C(C)NC(=O)CCS(=O)(=O)NC)C1)C(F)F N1(C(CC(n2c(C)cc(C)n2)C)=O)C2CCC1C(F)C(NC(=O)CC1(C)CCC1)C2 Cc1ncc([N+](=O)[O-])n1CC(N1CC(C)N(C(C23CC(F)(C2)C3)=O)CC1C)=O c1(C(N2CCC(CNC(C(c3ccn(C)n3)(C)C)=O)C2)=O)nc2ncccn2n1 C1(C(=O)NCC(C)NC(=O)CN=S(C)(C)=O)CC12CCC(C)(C)CC2 CCC(C)(C(=O)N(C)CC=CC(=O)NCCCC1(C)CC1)C(N)=O C1(C#N)(C(=O)NCC(C)(C)CNC(=O)CC2C=CCC2)CC2CCC1CC2 C1(O)(C(=O)NCC2N(C(c3c(C)nsc3Cl)=O)CCCC2)CCOC1(C)C N1(C(CC(CC)OC)=O)CC(NC(c2ccccc2)=O)CC2(CC2)C1 CCCC(C)(O)C(=O)NC1CCN(C2CCN(C(C3(C)CCCC3)=O)CC2)CC1 C1(NC(=O)C(CC2CCOCC2)NC(c2ccncc2Cl)=O)CCCCCC1F C(C(=O)NCC1(F)CCC(CNC(c2nc(Cl)cs2)=O)C1)(C(C)C)NC(COC)=O N1(C(C=CC(=O)NCC(C)N(C(c2c[nH]nc2CC)=O)CC)=O)CCCC(C)C1 c1(C(=O)OC(C)C)cc(=NC(C)Cc2cn[nH]c2)[nH]c2ccccc12 CCCC(C)(C)CC(=O)NC(C)C(C)NC(=O)CSC(F)F c1(C(=O)NC2CCC(CNC(CN(C3CC3)CC)=O)CC2)cnn2cc(C)cnc12 c1(OC)ccc(CCC(=O)NC(C)CC(C)NC(=O)C2=NNC(=O)C2)cc1C Cc1nc(S)sc1CC(=O)N(C1CN(C(C2CC(O)CN2C)=O)C1)C N1(C(CC2CC(=O)NC2=O)=O)CC(=O)NCC1C(=O)N(C12CC(C1)C2)C1CC1 N1(C(C2C(C=C)C2)=O)CCC(NC(=O)C=CC2(C)CCOCC2)C(C)(C)C1 N1(C(C2C(OC)C2C)=O)CCCC(C)(CNC(c2cccc(N)n2)=O)C1 n1(CCSC)nnnc1C(C)(CCCl)NCc1nscc1Br c1(C(=O)NCCC(=C)CNC(=O)C(F)C2CCOC2)ccc(Br)c(OC)c1 CC1CC(NC(c2cn3ccsc3n2)=O)CCN1C(=O)CN1CCCOC1=O C(=O)(CCC(=O)NCC1C=CC(NC(=O)C(C(C)O)NC(C)=O)C1)OC Cc1nn(C)cc1CCNC(=O)C(C1(C)CC1)NC(c1ccccc1)=O c1(C(N2CCC(C(N(c3ccnc(Cl)n3)CCC)=O)C2)=O)cccc(OC)c1Br c1(COC)ccc(C(=O)NC(CO)C(C)NC(=O)C=Cc2cocn2)o1 Cc1cccc(C(=O)NCC2CCCCN2C(c2n[nH]cc2I)=O)c1OC(F)F c1(C(=O)NCC(C2CCC2)NC(c2occ(C)c2)=O)[nH]c2ccc(Cl)cc2c1Cl c1(NC2CCC(CNC(C3CS(=O)(=O)C3)=O)C2)cnc2ccccc2n1 N1(C(C2(SC)CC2)=O)C2CCCC1CC(CNC(=O)CCC1CC1(C)C)C2 c1(CC)cnc(C(N2CC(C(=O)N(CCCOC(C)=O)CCO)C(F)C2)=O)nc1 C(C(C)CC(=O)NCC(C)(C)C(N)=O)NC(C1(CC)CCOC1)=O C=CCC(C(=O)NCCN(CC(C)O)C(c1cnc(C)s1)=O)C(C)C c1(C(C2(C(C)C)COC2)C2(C)COC2)nnnn1C1CCC1 O=C(C1=CCC(F)(F)CC1)NCC1CCN(C(=O)CC2=CCCCC2)C1 C(=O)(C1Cc2c(Cl)cccc21)N1CC2CC3C(NC(CS(C)(=O)=O)=O)C1C2C3 CC1=CCC(C(=O)O)CC1.c1cncnc1N(C)C C(=O)(C(F)(F)CC(C)C)NC1C(NC(CCCOCC)=O)CCOC1 C(=O)(C#CC(C)(C)CNC(=O)CSCCN1CCCCC1)NC1CC(C)OC1=O N1(C(c2c[nH]c(=NC)s2)=O)CCCC(CC(=O)NCc2cc(O)ccc2F)CC1 N1(C(C2C(=C)CC2)=O)Cc2ccccc2OC2(C1)CN(C(=O)COCCF)C2 n1(CC(=O)NC2(c3ccc(OC)cn3)CCCCCC2)cnc2ccccc2c1=O C1(O)(CNC(c2ccc(F)c(Cl)c2)=O)CCCN(C(C2COC3(CCC3)C2)=O)C1 C1(C(N2CC3CCN(C(C4CC=CCO4)=O)C3C2)=O)CCn2nnnc2C1 c1(C(C)(C2CC2)NCc2n(CCC)nnn2)c(F)ccc(F)c1Br N1(C(=O)OC)CC2C=CC1C(C(=O)NC1CC(CO)N(C(=O)CNOC(F)F)C1)C2.OC c1(C(N)=O)ccc(Br)cc1NC(C1CCN(Cc2cnn(-c3ccccn3)c2)C1)=O C1(O)(C(C(=O)NC(c2cnn(C)c2)C)NC(c2cc(CO)[nH]n2)=O)CCCCC1 CC(C)C(C)C(CNC(c1ccnnc1)=O)NC(=O)CSc1cccc(C#N)c1 c1(C(N2CCC(N(C(=O)CC3COCC(C)O3)CC)CC2)=O)cnc(C)cc1Cl C(C)(C(CC(=O)OC)NC(c1nc(F)ccc1Br)=O)OC C1(CC(N2C(C(=O)NCCC(COC)O)CCC2)=O)CC2(CCC2)C1 CC(=O)CCN=C(NCC(F)(F)CO)NC(c1ccccc1F)C c1(C(=O)NC2CN(C(C(CCC)(C)C)=O)C3C2C3)ccc2c(n1)COCC2 C(=O)(CS(=O)(=O)NC(C)C)N1CC(O)(C(C)NC(c2nc(CC)sc2)=O)C1 C(=O)(CC(C)(C)C(C)(F)F)N1CCC(N(C)C(C2CC3(CCCC3)CO2)=O)C1 N1(C(c2c(N)cc(Br)cc2)=O)CC2CCC1C(NC(=O)CC1CCCC1)C2 N1(C(Cc2c(C)non2)=O)CCC(C(F)(F)F)C(NC(=O)Cc2cn(C)nn2)C1 C#CC(CC(C)(C)C)NC(C1CCN1C(=O)C(O)C=C)=O c1(C(=O)NCCC2(OC)CN(C(C(CC)=CC)=O)C2)ccc(F)c(F)c1 C1(C(=O)NC)C(C)CCN1C(=O)Cc1ccccc1NC(C=NOC)=O.C(C)(C)O C1(Cl)(C(=O)OC)CC1C(=O)N(C)CC1(NC(=O)COCC(F)(F)F)CC1 C(=O)(CC1C(=O)Nc2ccc(F)cc21)NCC(CO)NC(c1cc(C)ncc1)=O CC1(C#N)CCN(C(C2(F)CCCN(C(C3CCC(CO)CC3)=O)C2)=O)C1 CC(C)C(F)(CNC(=O)CC1COC(=O)C1)C(=O)N(C)CC1CCSC1 C1(CNC(N2CCC(OC)CC2C)=O)CN(C(=O)OC(C)(C)C)CCC1(C)C CCCCCC(=O)N(C1CCCCC1)CCNC(c1csc(CCC)n1)=O C1(OC)(CNC(C2CN(C(N)=O)C2)=O)CN(C(c2c[nH]nc2C)=O)C1 Cc1c(CNc2nc(CC(=O)Nc3conc3CN)cs2)cncc1Br n1(CC(=O)NC2C(NC(=O)CC3CC3(Cl)Cl)CCCC2)ccc(=O)c([N+](=O)[O-])c1 C1(CC=O)CCC2(CC1)CC2.c12nsc(n1)N(C)CC1CCN(C1)C2=O.CO Cc1oc(C)c(C(N2CCOC(C(=O)NCc3cc(O)ncn3)C2)=O)c1C C(=O)(C(CNC(=O)CCc1ncccn1)CC1CCCC1)NC(C)(C)CO N1(C(=O)NC2CC(OCC)C2)CCC2C(C(=O)NCC(c3cccnc3)O)C2C1 N1(C(CC#N)=O)CCN(C(=O)CC2CC(n3cnnc3)C2)C2COCC12 Cc1noc(C2C(CNC(=O)N(C)C3CC3)C2c2ccccc2)n1 C1(CCCl)CC(O)CN1c1nnc(-c2ccco2)n1CC1CCOC1 c1(C(=O)NCC(C)CN(C(=O)C(C)CNS(C)(=O)=O)C)cccc(Cl)c1 C1(NC(CCCSC(C)(C)C)=O)(CO)CCN(C(=O)CCC2CC(C)C2)CC1 N1(C(CSCC(C)C)=O)CC(C)CN(C(C2C3C4CCC(C4)C23)=O)CC1C c1(OC)cc(CC(N2CC(NC(=O)CC(C)C)CC(F)C2)=O)cc(OC)c1OC CCC(CC(=O)N(C(C)CCC(C)C)C)NC(c1occc1C1CC1)=O Nc1cc(C(=O)NCC2(CCNC(C3CCCC34CC4)=O)CC2)c(F)c(F)c1F c1(NC(CCCN(C)C(C2CCCCNC2=O)=O)=O)cccc2c1OCO2 c1(N2CCC(C#CC)C2)ccc(S(=O)(=O)N2CCCC2C(C)C)cc1Cl c1(OC)c(NC2CCCC(CC(N)=O)C2)cc(Br)cc1Br C(C(CCC(=O)O)S(C)(=O)=O)NC(=O)NCCc1ncc(C)cn1 N#Cc1cc(C(N2CCCC2C2CCN(C(c3n[nH]cc3Cl)=O)CC2)=O)c[nH]1 c1(C(N2C(CN(C(=O)C(F)F)C)CCC2)=O)ccc(Cl)c(Cl)c1 C(c1ccc(C)o1)=CC(N1C(CN(C(=O)Cc2ccccc2C)CC)CCC1)=O c1(OCC)cnc(CN2CCC(CCNC(=O)CC3CCCC(=O)N3)C2)nc1 C1(C)(CNC(c2ncn(CC)n2)=O)CCCN(C(=O)C=C2CCCCC2(C)C)C1 Oc1ncc(Br)cc1C(CCc1ccccc1)NCc1ccc(-c2cc[nH]n2)o1 CCCC(CCC)CC(=O)NC1CN(C(c2ccc(CC)c(Cl)c2)=O)CCC1C C1(NC(COC)=O)CC12CC(NC(=O)C(O)Cc1cc(C)sc1C)C2 C1(C(=O)NCC2CC23CC3(F)F)(CC)CCN(C(=O)C(C)(C)N(C)C)C1 C1(NC(C2C(F)(F)C23CCC3)=O)COC2CN(C(c3csnn3)=O)CC12 c1(C(=O)NC2C(NC(C(CC)(C)CC)=O)CCCC2)cccc2nc(O)ccc12 CCC(CC(=O)N(C1CCCN1N1CC(F)(C#N)C1)C=O)c1ccccc1 O=C(C1=Cc2cc(Br)ccc2OC1)Nc1c(CO)cncc1O c1(C(=O)Nc2ccc(C(C)NC(=O)NCCC)o2)ccc(C(=O)OC)c(F)c1 CC1CCCC(C)N(C(=O)CCCCCNC(C2(C)CC(F)C2)=O)C1 Cc1cnc(C=CC(=O)NCC2C3CN(C(c4scnc4Cl)=O)CC23)[nH]1 N1(C(C(CC#C)C)=O)CC2CC(NC(c3ccc(Br)c(Cl)c3)=O)C(C2)C1 Cc1ccc(OCCC(=O)N2CC(CNC(C3(C)CC=CCC3)=O)C2)c(C)c1 c1(C(N2CCC(F)(CNC(C3(CCCC)CCC3)=O)C2)=O)cnc(OC)c(Cl)c1 N1(C(CC2(N(C)C)CC2)=O)CCC2CCCC(C1)N2C(c1ccncc1Cl)=O Cc1cc(NC2CC3CN(CCN(c4ccncc4)C)CC23)ccc1[N+](=O)[O-] C1(C(=O)NCC2(O)CN(C)C2)CN(C(=O)CC2CC2)CC1N(C)CC C(=O)(C1CCOc2ccccc21)NC(C(C)C)C(c1cc(Cl)cc(Cl)c1)=O c1(C(C)Nc2cccc(-c3cccc(N(C)C)n3)c2C)cccc(F)c1F Cc1ccc2c(c1)CN(C(C1CC(F)CN(C(=O)CCN(C)C)C1)=O)C2 c1(C(=O)NC(C)(CNC(C2CC(F)(CO)C2)=O)CO)nnn2c1C(=O)NCC2 N1(C(C(C)(C)CF)=O)CCCCCC(NC(c2ccc(C(F)F)s2)=O)C1 N1(C(=O)COCc2nc[nH]n2)CCC2(CCCCN(C(c3ccsn3)=O)C2)C1 c1(C(N(CCOCCN(C(CC(C=C)C)=O)C)C)=O)ccc2ccoc2c1 O(NC(=O)C(O)C(C)CC)C(C(=O)NC1C(C)(COC)C1)CC(C)C N1(C(C2C(C)=C2)=O)CCC(NC(c2nc(Br)sc2C)=O)C(O)C1 C1(n2cc(COC3CCN(C(C4CCS(=O)(=O)N4)=O)C3)nn2)CCC(CO)CC1 C1(N(C)C(n2ccc(C3CC3)n2)=O)CCCC(NC(=O)COc2ccccc2)C1 c1(C(=O)NCC(COC)NC(=O)CCn2cccc2)ccc(OC(C)=O)nc1 C(=O)(C(C)C(C)C(C)(C)C)N1CCN(C(c2cccc(OC)c2F)=O)CC1 C1(NC(c2c(C)cncc2)=O)Cc2ccccc2N(C(=O)Cc2ccc(Cl)s2)C1 CC1CSc2ccccc2CN1C(c1cc(F)c(Br)cc1F)=O c1(C(N2CC(C(=O)NCC3CC4C=CC3O4)(SCC)C2)=O)cc(O)nn1C c1(OC)cc(C(=O)NCC#CCNC(=O)CNc2ccccn2)c2c(c1)CCC2 CC(C)(C)C(=O)C(=O)NC1CCN(C(c2cncc(C(F)(F)F)c2)=O)CC1CO C1(NC(CC2(CC)CCC2)=O)CC2(C1)CN(C(C1(C)CCCC1C)=O)C2 C1(C(=O)NC(C)CO)N(C(c2cc(C#N)c[nH]2)=O)CCCC1(C)C c1(C(N(C2CCN(C(=O)CCCC(C)(C)C)C2)CC)=O)cnn2ccccc12 C12(NC(CNC(=O)OC)=O)CCCC1CN(C(=O)CCN1CCOCC1=O)C2 c1(C(=O)NC(C)C)ccc(-c2cn(C(C3CCOC3=O)C)nn2)cc1Br CC(N=[N+]=[N-])C(=O)N1CCCCC1C(=O)NCCCc1cnccn1 c1(CN2CC(CNC(=O)Cn3cc(Cl)cn3)C2)ccc(F)c2ccoc12 c1(C(=O)NCC(c2ccccc2)NC(CCOC(C)C)=O)cc(N)c(Cl)c(O)n1 C(C(C)C)(C(O)C(=O)NCC1CC(O)CN1C(C1CCC1)=O)OC Cc1cc(C(=O)NC(c2ccnn2C)C(=O)NCC(c2ccco2)O)c(C)s1 c1(C(=O)NCCN(CCC)C(c2csnc2OC)=O)cc(Cl)cc(C)c1N C1(C)(CC)CC(OC)CN1C(c1cnc(CNC(=O)C=Cc2nccs2)nc1)=O C1(CC(=O)NCc2ncon2)CN(C(=O)Cn2ccccc2=O)CCO1 C1(SC)CC(CC(=O)NC(C(=O)NC(C)C(=O)NC(C)C)C2CCC2)C1 CN1C(=O)CCCC1C(=O)N(C)Cc1cccc(CNC(C2CNC(=O)C2)=O)c1 N1(C(C(CCC)NC(C)=O)=O)CCC(NC(c2sccc2Cl)=O)C12CCC2 Cc1cnc(NC(c2csc(NC(C3CCC(=O)NC3)=O)n2)=O)c(Br)n1 C(CC1CCOC1)(C(=O)NC1CCCO1)N(CC#N)CC1CC1 c1(C(=O)NCC2C(NC(c3csc([N+](=O)[O-])c3)=O)C2)cccn2ccnc12 c1(CCC)cc(C(=O)Nc2cccc(N(C)Cc3cnn(C)c3C)c2)ccc1F c1(C(=O)NCC(CC)NC(=O)C(N2CCCC2)SC)cc(NC(C)=O)cc(F)c1 c1(C(=O)NCC(CN(C(CCCc2onc(C)n2)=O)C)(C)C)scc(C)c1Cl C1(CNC(C2C(C)CCO2)=O)CCC(NC(=O)COCCN(C)C)CC1 c1(C(N2CCC(C(=O)Nc3ccc(O)c(F)c3)C(O)C2)=O)ccnc2cc[nH]c12 N12CC3CC1CN(C3)C(=O)c1c(F)ccc(OC)c1C2=O.c1(CC)cnn(CC)c1 C12(C(=O)NC3COCC3CN)C3C4C1C1C2C3C41C#N.C(CCC=O)OCC=C c1(C(=O)NCC2C(NC(Cc3ccn(C)n3)=O)C2)ccc2c(c1)CCCS2 N1(C(c2cc(OC)ncc2)=O)Cc2nccn2CC(NC(C2(O)CCOC2)=O)C1 C1(COC)CN(C)C(=O)CN1.C12CCN(C1C(C)C)C2=O c1(C(C)=O)ccc(C(C#N)N(C2CC3CCC2C3)S(C)(=O)=O)cc1 N1(C(C(CCSC)NC(Cc2cn(CC)nc2)=O)=O)CCC(F)(F)C(F)C1 c1(C(C)C)cc(C(=O)NCC(C)N(C(=O)C(C)Cc2ccnn2C)C)ccc1F C(=O)(CCCCOC)C(CN(C(=O)C(F)C1CCCC1)CC)=O.NCC c1(C(=O)NC23CCC(CNC(CC(CC)C)=O)(C2)C3)ccnn(C)c1=O c1(OC)ccc(O)c(C(N2CCN(C(=O)CC3(C)CCCO3)CC2C)=O)c1 N1(C(c2c(C(C)=O)ccs2)=O)CCC2CC2(NC(c2snnc2C)=O)CC1 C1(C(=O)NCC(CC)(CC)NC(C2C3CCOCC23)=O)CCCC(C)(C)C1 C1(C)(C(=O)OC)CC(C(N2CCCC2CN(C(=O)C(COC)OC)C)=O)C1 c12cc(OC)c(SC)cc1NC(=O)NCC1CCN(CC1)C2=O.C(CO)OC.CO c1(CNC(c2cc(C)n(-c3nccs3)c2C)=O)ccc2n[nH]cc2c1 C1(O)(CC)CCCN(C(C2(C)CCCN(C(=O)CC(C)(C)OC)C2)=O)C1 C1(C)(C(=O)NC(CNC(=O)OC)C)C=CCN1C(c1cc(CO)[nH]n1)=O N1(C(C(CC=CC)C)=O)CCC2CN(C(=O)CC3CCS(=O)(=O)CC3)C2C1 N1(C(C2C=CC(=O)N=N2)=O)CC(NC(c2nccnc2Cl)=O)CC12CCC2 C12(CNC(C(C)OCCC=C)=O)CC(NC(=O)C(C)NC(C)(C)CC)(C1)C2 c1(CNC(C2CCN(C(c3n(C)cnc3)=O)C2)=O)cccc(Br)c1F c1(OC(C)C)cc(C(=O)N(CC(C)CNC(=O)CN(C)C(C)C)C)ncc1Br C(CC(=O)NOCC(N)=O)N(CC(C)C)C(=O)CC1CCC(C)(C)C1 N1(C(c2cccc(N(C)C)c2)=O)CCC(O)(CNC(C2(Cl)C(C(C)=O)C2)=O)C1 c1(CC2(C(=O)O)CCC(C)(OC)CC2)cn(C)c2c(C)cccc12 N1(C(C(C)OCCOC)=O)CCOC(CN(C(=O)CCC2CCCCN2C)C)C1 Cc1c(C(=O)NCc2ccc(C(=O)NCC3(C(F)(F)F)CC3)o2)cccc1O Cc1ccc(S(=O)(=O)N(CC(N2CCCCC2C(C)C)=O)C)cc1 N1(C(c2c(N)cccn2)=O)CCN(C(C2C3CCC4C(C3)CC24)=O)C2COCC12 C1(NC(=O)CN2CC=CC2)COC2(CCN(C(C3CCS3(=O)=O)=O)CC2)C1 N1(C(C2CCCN(C(c3cncs3)=O)C2)=O)CCn2ncc(-n3ccnc3)c2C1 N1(C(CCCCC=C)=O)CCN(C(c2ccc(C(C)=O)[nH]2)=O)C2CCCCC2C1 c1(-c2nc(-c3ccc(C)cc3)nn2CCOC2CCOCC2)nccc2occc12 C1(O)(CC)CCCN(C(C2(NC(c3cc(C(N)=O)[nH]n3)=O)CC2C)=O)C1 c1(C(N2C(CNC(CC)=O)(CNC(C(C)OC)=O)CCC2)=O)c(C)nc(C)n1O N1(C(CCOC(C)C)=O)CC2CCN(C(=O)Cn3nc(Cl)ccc3=O)CC2C1 N1(C(c2nn(C)c(F)c2)=O)CCC(NC(c2cc(C#N)c[nH]2)=O)C(F)C1 C1(C)(CC(=O)NC2C(NC(C3(CN(C)C)CC3)=O)COC2)CCCCC1 C1(N(C(C(C)OCC)=O)CC)CCCN(C(=O)CCSc2ccc(C)cc2)C1 C1(NC(C2CCC(CC)CC2)=O)CC(C)CN(C(c2csc(C)n2)=O)C1 C1(NC(CC(C)C)=O)CCN(C(=O)C(C)CSc2ccccc2)C1(C)C Cc1cc(N)c(C(=O)NCC2CCN2C(C2CC(C)OC2=O)=O)cc1C Cc1c(OC(C2COC3(CN)CC2C3)=O)cccc1CNC c1(C(C)C)ccccc1C(N1CCC(C)(NC(=O)CCC(C)N(C)C)C1)=O C1(NC(c2nc(CC)oc2)=O)CCN(C(c2cn(C3CC3)cn2)=O)C(C2CC2)C1 CC1CN(C(C2CCCC(F)C2)=O)CC(C)CN1C(c1ccc(C(N)=O)cn1)=O c1(C(C2N(C(C3C(CCC)C3)=O)CC2)=O)ccccc1Br N1(C(CCc2onc(C)n2)=O)CC(F)CC1CNC(=O)C(C)NC=O N1(c2nc(C(C)C)nc(N(C)C)c2)CCCCN(C(C2CC2(C)C)=O)CC1 c1(C(N2CCC(NC(CCOCC#C)=O)(CF)C2)=O)ccc(OC)c(Cl)n1 c1(CCNC(=O)NC23CC(C)(C2)OC3(C)C)ccc(S(C)(=O)=O)cc1 c1(N(C(=O)CCCCCCc2ccccc2)C)cc(Br)cc2c1OCC2 Cc1cnccc1C(C)C(=O)NCC=CCNC(=O)CNC(c1ccsc1)=O C(C(C)CC(=O)N1CCCCC1C1CCC1)NC(c1c(C)occ1)=O NS(=O)(=O)CC(=O)NC1(CO)CCN(C(=O)CCC2CNC(=O)N2)C1 N1(CCNC(c2c(C)c(F)ccc2)C)CCC(C(F)(F)F)C2(CCC2)C1 C(=O)(C(CC)C(=O)N1CCN(CCN(C)C(C2NC(=O)OC2C)=O)CC1)OCC S(=O)(=O)(CC(=O)NC1CCN(c2nc(C)ns2)CC1)N(CCCOCC)C c1(Oc2cn(CCOC)nc2)ccc(C(n2[nH]nnc2=N)(C)C)cc1 N1(C(C(C=C)(C)C)=O)CCC=C(C(=O)NCC2CS(=O)(=O)CC2c2ccccc2)C1 C1(N(C(CCC2CCN(C(COCC(C)C)=O)C2)=O)C)CN(C)C(=O)N1 C1(NC(CSCC=C)=O)CCCCC12CCN(C(=O)C(C)(C)c1cncnc1)C2 C1(C)(C(=O)NC(C)C(CO)NC(c2ccc(CO)s2)=O)CCOC1C C(=O)(C(=O)Cc1cccs1)NCCCN(C(C=C(C)C1CC1)=O)CCO C1(NC(c2ccc(-n3ccc(C)n3)cc2)=O)CCN(Cc2ccco2)CC(O)C1 C1(CC)CCCN(C(c2cnn(CCO)c2)=O)C1C(N1CC2(CC2)C1)=O N1(C(CC2CC(=O)NC(=O)C2)=O)CC2CCN(C(=O)C(O)C3CCCC3)CC12 C1(C(=O)NC2C(NC(c3cc(C)sn3)=O)C2)CCCCC12CC2 C1(C(N2CCC(NC(C)=O)CC2)=O)CC(F)(F)CN1C(=O)Cn1[nH]cnc1=N N1(CC)CCN(C(c2cc3c(Br)cncc3s2)=O)CC12CCOC2 C1(NC(CC(=O)OCC)=O)(CC)CCCN(C(C2CCCCC2C(F)(F)F)=O)C1 C(C(C)N=c1nc(N(CC(C)C(C)(C)C)C)c2c([nH]1)CCOC2)NC(=O)OC CC1(C=CC(=O)NCCCN(C(=O)C=CSc2ccccc2)CCO)COC1 n1(CC)nc(C(N2C3CCC(C3)C2CNC(C)=O)=O)ccc1=O CCCC(C(=O)N1CC(NC(=O)C(F)CC2CCOC2)C(CC(C)(C)C)C1)OCC C1(NC(c2c(C)cc(CC)o2)=O)C2CC1CN(C(c1ccsc1C(F)F)=O)C2 CC1(CNC(c2nccnc2N)=O)CN(C(C2CCOCC2)=O)CCO1 C1(C(=O)Sc2cccc(OC(F)F)n2)CCCN(CC2C(c3n(C)ncc3)C2)C1 C1(C(=O)NC23CC(C(=O)OC)(C2)C3)CC2CCC1O2.C12CCN(C1)C2C CCC(O)(C(=O)NC1CCCCC1NC(=O)CCF)c1ccccc1 C(CN=c1[nH]c(N2CCC(C(N)=O)CC2)nc2c1COC2)N(C)CC CCC(C)C(O)C(C)C(=O)NCCC(C(=O)NCC1(C(N)=O)CCCCC1)OC CC1CC=C(C(=O)NC2COCCN(C(C34CCOC3CCOC4)=O)C2)CC1 N1(C(CCc2ccc(C)cn2)=O)CCC2C(CCN2Cc2c(F)cccc2I)C1 c1(C(N2CCC(CCC)C2)C(=O)NC(C)C)ccc(C)c2c1CCC2 c1(CNC(CNC(C2COCC(C)O2)=O)=O)cc(C(=O)O)ccc1Br C1(NC(CCCCCC)=O)CN(C(c2n[nH]c(CC)n2)=O)C2(CCCOC2)C1 C(=O)(CC(O)C(Cl)(Cl)Cl)NC1CCN(CC(=O)N(C2CCCCC2(C)O)CC)C1 c1(C(=O)OC)cc(C(F)(F)F)cc(C)c1.c1(N2CC2)cc(C)ns1 c1(N2CC(C)C(CNC(C3CC4OC3C3CC43)=O)C2)ncnc2ccc(F)cc12 N1(C(C(C=C)(C)O)=O)CCCC(CO)(NC(c2cncc(F)c2)=O)C1 c1(C(N(CC(CC)NC(c2cc(=O)n(C)o2)=O)C)=O)ccc2cc(Cl)ccc2c1 N1(C(COCC(=O)NC)=O)CCC(F)(F)C(CNC(C2COCCN2C)=O)C1 C1(N(C)C)CC2CC1CN2C(=O)NC1CCN(C(c2ccsc2)=O)C1 C(=O)(C1=CCc2ccccc21)N1CC(C)(C)C(CNC(=O)CC2CCC(=O)N2)C1 c1(OCCC(=O)NC2CC2NC(c2ccnc(C3CC3)c2)=O)ccccc1F C1(N(C(=O)CC2CC=CCC2)CC)CCN(C(=O)C(C)Cc2ccccc2)CC1 c1(C(=O)NC2C(C)CN(C(=O)COCC(F)F)C2)cn2cccc(Br)c2n1 N1(C(c2c(C)nco2)=O)CCC(C(=O)N(CC(N)=O)C)C12CCC2 CCCCCC(C)(CC)C(=O)NC1CC2(C1)CC2NC(C1CCCC(=O)C1)=O S(=O)(=O)(c1cc(C(=O)NC2CC(NC(C3CCCC3F)=O)C2)ccc1C)NCC C(CCC(=O)N(C(C)CN(C(=O)CNc1ccccn1)C)C)OC C(C(F)C(=O)N1CC(C(=O)N)C1)OCC.C1(C)(CNC(=O)CC2CC2)COC1 N1(C(CCN(C(c2cc[nH]c(=NC)c2)=O)CC)=O)CC(C)CCC1C C(C1CCCO1)=CC(=O)NCC(F)CNC(=O)CNC(=O)Cc1ccccc1 N1(C(CC2CCC(NC(c3c(C)nn(C)c3N)=O)CC2)=O)CCC2CCC(C1)S2 N1(C(c2c(CC)[nH]cc2)=O)CCC2(NC(C3CC4(CSC4)C3)=O)CCCC12 C1(C(=O)NCCCCCNC(c2csc(-c3cnc[nH]3)n2)=O)CCCC12CCC2 C12(NC(C=C(C)Cl)=O)CCCC1N(C(c1ncc(C(N)=O)cc1Cl)=O)CCC2 CCC(C)CC(=O)NC(Cn1cccn1)C(=O)N1CC(COC)C1 CC(C)C(C(=O)NCC1CCCC1NC(=O)CS(N)(=O)=O)N1CCCCC1 C1(CC(=O)NC(CC)C(=O)OC)C2CN(C(C3CC(n4cnnc4)C3)=O)CC12 C1(C(c2n(CCCC)nnn2)NC(C)C(C)n2cncn2)(CCl)CCOCC1 Cc1[nH]c2ccnc(NC(c3nnnn3CC(F)(F)F)CC3(C)CC3)c2c1C C(=O)(CC(C)C(=O)N(CCC(=O)NCC1=CCCC1)CCO)OC N1(C(C=C(C)C(F)F)=O)CCOCCC1C(=O)NCC1CC1c1ccncc1 C(CC(=O)OC)(C(F)(F)F)OC(c1cc(C)cc(NC)c1C)=O N1(C(c2c(CC)[nH]nc2Cl)=O)CC(C)C(Nc2cnc3ccccc3n2)C(C)C1 c1(C(N2C(CN(C)CCC3CCCO3)CCCC2)=O)cc2cc(Cl)ccc2[nH]1 C(=O)(C(O)C1=CCCCC1)N(C)CCNC(=O)CNC(c1ccc(NC)cc1)=O N1(C(C2C(CNC(c3cc(C(C)=O)on3)=O)C2(C)C)=O)CCC2(CCC2)C1 CC1CC(CC(N=c2nc3sccc3c(-c3ccncc3)[nH]2)=N)N1CC1CC1.CC1CC1 n1(CC(=O)NC(C)C(C)(C)NC(C2CC(=O)N(O)C2)=O)nnc2ccccc12 CC1(C)CN(C(=O)CNC(C2CCCS2)=O)CC1CNC(c1ccc(Cl)cc1)=O c1(-c2cn(CC)nn2)ccc2nsnc2c1.C1(=O)C(CCO)OCCN1CC(=O)O C(=O)(CC(C(F)F)c1cccc(F)c1)N1CCCC(NC(c2cn[nH]c2)=O)C1 c1(CN(C2CCCCC2)C(C(N2C(CC)CCC2)=O)=O)ccc(CC(F)(F)F)cc1 C1(CNC(c2cnsn2)=O)CC(F)CN1C(=O)CCN1CCC(F)C1 C(=O)(C#CC1CCCCC1)NCC(CCCC)NC(c1ccc(F)c(O)c1)=O c1(SC)cc(C(=O)NC2CCC(CNC(=O)CSCCC#N)C2)ccc1N c1(CC(=O)NC2CC2CNC(C2(O)CCCCCC2)=O)ccc2c(c1)OCCO2 N1(C(C2(C#C)CC(=O)C2)=O)CCC2(CC1)CC2C(=O)NC(C)CCC(C)C C1(NC(C(c2ccoc2)NC(c2ccc(CO)cc2)=O)=O)CC12CCCCCC2 C1(O)(CN(C(C2C(CC)C2)=O)C)CN(C(c2cc(C)co2)=O)C1 c1(CN(C(=O)NC(C)C(c2ccccc2Cl)O)C2CC2)cccc2nc(O)oc12 c1(C(=O)NC2(CNC(C3CCC(C)CC3)=O)CCOC2)cc(F)c(F)c(F)c1N C(C)(CCCC(=O)NCC1CC1(F)F)NC(C1CN(C(C)C)C1)=O C#CC1(C(=O)Nc2cnccc2N(C)C)CCN(C(C2CCCCNC2=O)=O)C1 C1(N(C(C)(C)C)C(C2CCNC2=O)=O)CCN(C(C2(C)CC=CCC2)=O)CC1 N1(C(C2C3(CC(NC(C(NOC)=O)=O)C3)C2)=O)CCS(=O)CC1C N1(C(C2CCCN(CC)C2)=O)CCN(C(=O)CCCN2CCCC2)C2COCC12 C(=O)(N=c1[nH]nc(C2CC2)s1)NCCC(C)OC c1(CCCO)nc(-c2ccc(C(C3CC3)=O)cc2)n(C2CCCC2)n1 C1(=CC(=O)NC2(CF)CCN(C(c3cccnc3S)=O)C2)CN2CCC1CC2 C1(CNC(=O)CCN2C(=O)CCC2=O)CC(NC(c2sccc2F)=O)C12CCC2 C1(CC)CCCN(CC(=O)NCC(C)(C)NC(c2ccc(C3CC3)o2)=O)C1 C(CCCS(C)(=O)=O)(C(=O)O)NCc1nc2cccc(OC)c2[nH]1 N(C(=NCCN1CCCC1)NCC1(C)CC1(C)C)CC1(CC)CC1 CC1(C)CC(C(=O)NC2CCC(NC(=O)CC3(C(F)(F)F)CCC3)CC2)=NO1 N1(C(C(C)P(C)(C)=O)=O)CCCC(NC(=O)C=Cc2cc[nH]n2)CC1 N1(C(c2c(C)cno2)=O)CCCC2C(NC(=O)Cc3sccc3Cl)C(C)(C)C12 C(=O)(CCCC)N(C)CC.C12(C(=O)OC(C)=O)CC(c3ccccc3)C1C2 c1(C(N2CC(C)(NC(C(C)NC(=O)NC)=O)C2)=O)ccc(Cl)c(C(=O)NC)c1 c1(NC(=O)NCCC2C(C)(C)C2(C)C)ccc(F)cc1NS(C)(=O)=O C1(C(N2CCC(C(F)(F)F)C2)=O)CCCN(CCn2ccnc2)C1 CC1CN2CCN1CC2C(=O)NC1COCC1NC(c1cnc(O)o1)=O N1(C(C(C)C)=O)CCCC(C)(C(=O)N(C2CCC2)C2CCC2)C1.N1CCC1 CCC(C)(C)C(=O)N1CCCC1CN(C)C(C1CCN1C1CCCC1)=O Cc1ccccc1C=CC(N1CCN(C(=O)C(O)CC(N)=O)C(CC2CC2)C1)=O CCC(C)CC(=O)NCCCNC(C1(C(C)(F)F)CC1)=O c1(C(c2coc(-c3ccccn3)n2)N(C)C(=O)NCC2(C)COC2)cccc(Br)c1 c1(C(N(CCCNC(=O)COC(F)F)C)=O)c(O)ccc2ccccc12 C(=O)(CC(CN(C)C)C(F)F)NCCC(C)NC(c1cccnc1C(F)(F)F)=O CCCC(CC)C(C(=O)Nc1c(C)cccc1C)N1CC2C(C1)C2(C)C C1(C(N2CCC(C(C)NC(c3nccc(C)n3)=O)C2)=O)(CC)CCNC1=O CCC(C)CCCCC(=O)N1CC(NC(c2ccnnc2)=O)CC1(CC)CC c1(C(C)C)c(C(=O)NCC2(C(C)NC(c3cccnc3O)=O)CC2)cccc1F N(C(=NCC(F)F)N1CCOC(C(C)C)C1)C(CC)CC(=O)OC C1(NC(C=CC(=O)N(C)C)=O)C2CC1N(C(=O)Cn1cnccc1=O)C2 C(=O)(N1CC(C)(O)CO1)C1(CNC(C2(CC)CCCO2)=O)CCCCC1 c1(CN(c2cc(OC)ncn2)C2CCCNCC2)c[nH]c2cc(F)cc(F)c12 c12ncnc(OC)c1CN(C)C1CN2C1.c1(C)cccc(C(C)(C)C)c1.CO C1(CN)CCCC(NC(c2cccc(F)c2)=O)(CC2CC2)C1 c1(-c2cc(CNC(c3csc(-c4nn[nH]n4)c3)=O)on2)c(F)cccc1F c1(CC(=O)NCC2C(NC(C(CCCC)O)=O)C2)cn(C)c2c(cnn2C)c1=O CC1CCCN(C(=O)CCOc2cccnc2)C1CNC(=O)C1=COCC1 Cc1cc(C(N2CCCC(CN(C(=O)CCNC(=O)CO)C)C2)=O)c(O)c(C)c1 Cc1ccc(NC(=O)CC2(C)CCN2C(c2cnco2)=O)cn1 CN(C1CC(F)(F)C1)N1CCOC(COC(C)(C)C)C1 N1(C(C2C(C)(C)CC2)=O)CC2CC(C1)CN(C(c1ccnn3ccnc13)=O)C2 Cc1csc2ccc(C(=O)N(C(C)CNC(C3(C)CCC(=O)NC3)=O)C)cc12 C12CCC(CC1)C(=O)N2.c1(CCCNCC2CCCO2)cc(C2CC2)[nH]n1 c1(NC(C(C)NC(=O)CN(C2CCC2)CCO)=O)cnn(C(C)(C)C)c1 CC1CN2CCCN1N1CC3C(C3C1)C2=O.C(=O)C1=CCSC1 c1(C(N2C(C)CCC(NC(C(CC)F)=O)C2)=O)ccc2c(c1)NC(=O)CO2 C1(C(=O)NC2C3CN(C(CSSC)=O)C2C3)CCc2ccccc2C1 c1(CNC(C2CCC(NC(C3C4CCCC34)=O)C2)=O)ccccc1Br c1(CC)ncc(CNC(c2conc2CNc2cn(CC3CCC3)nn2)=O)s1 C12(NC(C=C(C)C3CC3)=O)CCCN(C(C3CCC(C)CC3)=O)CC1C2 c1(C(N(CCC)CCNC(=O)Cn2cnc(C)c2CC)=O)coc(S(C)(=O)=O)c1 C1(C(CNC(C)=O)C)COCCN(C(c2sc(C)c(C)c2Br)C)C1 C1(C(N(CCC2N(C(CCC=C)=O)CCCC2)C)=O)C(F)(F)C12CCC2 C(c1cncnc1O)=CC(=O)NCC1CN(C(Cc2cc(C)sc2)=O)C(C)C1 Cc1cc(=NC(=O)C(=O)N(C2CC3CC2N(C(=O)C=Cc2cc[nH]n2)C3)C)[nH]o1 c1(C(=O)NC(C)C(C(=O)N)NC2CC3CCC(C2)C3)cc(C)cc(C#N)c1.CC=CC c1(C(=O)NC(CC=C)CNC(c2cc(Br)ccn2)=O)cc(=N)[nH]c(Cl)n1 C1(NC(CCCC)=O)CCN(C(=O)CCc2cc(C)[nH]n2)C(C)C1 C1(NC(CC2C(C)CCCC2)=O)CCCOC12CCN(C(C1CNC(=O)N1)=O)CC2 c1(C(C(=O)NCC=C)N(C(C)C(C)(C)C(=O)OC)C)ccc(OC)c(OC)n1 Cc1oc(S(N)(=O)=O)cc1C(N1CC(CNC(=O)C=CCO)CC(C)C1)=O CCC(C)CCC(=O)N(C1C2CN(C(=O)CC3OCCCO3)CC12)C C=CCC(CNC(=O)CC1CCCO1)C(=O)Nc1c(C)noc1C(C)C c1(C(N2CC3CCC2C(O)C3)C(=O)NC)cc(C)nc2ccccc12 c1(C(=O)NCCC(C)(C)N(C2CCCC(C)C2)CC(=O)OCC)cnn(C)c1C#N [N-]=[N+]=NCC(C(=O)N1C2CCC1COC2)NC(=O)CC1CCOCC1 C1(CNC(N2CC3CCC(C2)N3CC(F)(F)F)=O)CC2CCCCN2C1=O C(=O)(C(C(=O)N1CC(C(C)NC(c2ccc[nH]2)=O)C1)C(C)C)OCC N1(C(CC2N(C)C(=O)CC2)=O)CCN(C(C2COCCOC2)=O)C2COCC12 c1(C(N2CC(CCNC(C(CC)=CC)=O)C2)=O)ccc(C)c(OC(C)=O)c1 N1(C(c2cccc(SCCC)c2)=O)CCC(C)CC1CNC(=O)C(C)(C)C#N n1(CC)nc(C(N2CC(OCC(=O)NCc3nc(N(C)C)no3)C2)=O)cc1O CC(CC#N)C(=O)NC1(CNC(=O)CCc2cccc(O)n2)CC1 N1(C(C2C(C)OCCC2)=O)CCC2(NC(=O)Cc3cnn(C)c3)CCCC12 N1(C(C2CC(C#C)(O)C2)=O)CCC(C2CCN(C(=O)C=Cc3cnc(C)s3)C2)C1 C(=O)(C(C)(C)S(C)(=O)=O)O.C1(OC)(CNC(=O)Cn2cc(F)ccc2=O)CCOCC1 Cc1ccccc1CCNC(=O)CCC1CCCCN1C(c1ccns1)=O c1(-n2ncc(C(=O)NCC(C)N(C(=O)CC3CCCC3)CC)c2)cccc(O)c1 C1(NC(CCCN(C)C)=O)CCCC12CCN(C(=O)CCC1CC(F)(F)C1)CC2 N1(C(CC(OCC)OCC)=O)CC2CCCC2(NC(=O)CC2(C)CCCCC2)C1 c1(C(N2CCC(N(C(C3C(C)CCC3)=O)C)C2)=O)cccn2c(CO)nnc12 C(c1ccc(C#N)cc1)=CC(=O)N(C(C)C)CCNC(=O)C(C)C(C)(C)C C1(C(=O)NCCC2(CNC(c3scnc3C(F)F)=O)CC2)CCCCS1(=O)=O c1(CCCC)ncc(C(=O)NCC(c2cccnc2)(C)NC(=O)COCCF)s1 C1(S(N)(=O)=O)(C(=O)NC2CCC(c3c(OC)ccc(Br)c3)C2)CCCC1 c1(C(N2CC(NC(C3N(C)CCOC3)=O)C(O)CC2)=O)coc2ccc(F)cc12 C(=O)(C(C(C)C)NC(=O)CCN(C(c1cnc(N)cn1)=O)C(C)C)NC N1(C(C(C)CN(C)C(C2CCNC2=O)=O)=O)CC2(CCCO2)C1 C1(C2(NC(C3CC(C(C)C)C3)=O)CC2)CCCCN1C(=O)C=C1CC1 c1(C(C)C)ccc(C#N)c(N(C)CC2CCCN(C(C3CCC(C)C3)=O)C2)n1 Cc1cc(C(=O)NC2CC3CN(C(=O)OC(C)(C)C)CC23)c(C)n1CC1CC1 C(=O)(C(N)CCc1cn[nH]c1)NCC(C)(F)CN1CCCC1 c1(C(N2CC(NC(c3cnn4ncccc34)=O)C2)=O)cccc2c(O)nncc12 n1(CC)nc(C)c(C(=O)N(CC(c2ccc(C)nc2)O)C(C)C)c1Cl C1(C(N2CCC(C)C2C(=O)NCC=CC(=O)OC)=O)C2C3CC4C1C1C2CC3C41 C(C(=O)N=c1ccn(C2CCCN(C(c3c[nH]c(=NC)o3)=O)C2)[nH]1)C1C(=C)C1 c1(C(N(C(CNC(C(C)=CC)=O)Cc2ccccc2)C)=O)cnc2ccsc2c1 Cc1cc(F)ccc1C(=O)N(C1CN(C(=O)C(C)C2CC2)C1)C c1(C(=O)NCC2CC(OC)CN2C(C2CCC(C)O2)=O)c[nH]cc(Br)c1=N N1(C(CC(CC)O)=O)CCC2(CC1)OCCCC2NC(=O)CC1CCOCC1OC c1(C(=O)NC2C(C)(C)CN(C(C3CS(=O)(=O)C3)=O)CC2)cc2c(F)cccc2[nH]1 C=C(Cn1cc(C2(NC(=O)CCC=CC(=O)N(C)C)CC2)nn1)C1CCOCC1 N1(C(c2cc3cccc(C)c3s2)=O)CC2(CCCN(C(=O)CC3(C)CCC3)C2)C1 N1(C(=O)CCOC2CC2)CCN(C(c2ncsc2-c2cccnc2)=O)CC1 c1(CN(C(COC)=O)CCF)ccc(Cl)cc1 N1(C(CN(C)C(N)=O)=O)CCCC1C1CCN(C(C2CC3CC2C3)=O)C1 C1(C(N(C2(CNC(=O)C=CBr)CC2)C)=O)CCOC1C(F)(F)F C(=O)(C(C)CCOC(C)=O)N1CCC(CCCC)C1.C12(CCCC1)C(=O)N2 CC1OC(=O)NC1C(=O)NC1CN(C(=O)C(=CC2CCCCC2)F)CC1O Cc1cc(C)c(C(=O)NC(C(F)F)C2CCCO2)c(C)c1 c1(C(=O)NC(c2cc(C(F)F)oc2CCC2C(CCF)C2)=O)cccc(C(F)F)n1 Cc1ccc(F)c(C(N2CCC(C(C)(C)N)C2)=O)c1.C1(=O)CCOCCN1 c1(CC(=O)NCCN(C(C(CO)N(C)C)=O)C2CC2)ccccc1N1CCOCC1 N1(C(c2ccc(OC)nc2F)=O)CC2CCN(C(=O)CCCCN(C)C)CC12 c1(C2(CNC(C3CC4CC4N3C(=O)CC3COCCO3)=O)CC2)ccccc1F CCC(C)C(C(=O)NCc1nc(C)c(C)[nH]1)N(C)C(c1cnns1)=O Cc1cc(C(=O)N(C)CC=CC(N2CCC(C(F)(F)F)C2)=O)nc(C)c1 Cn1ncc(C(=O)NCC2CN(C(=O)CC3CCO3)CC2C(F)(F)F)c1C(F)F C12CCN(C1)C(=O)N2.c1(N2CC(CN(C)C)C2)ccncn1 N1(C(C(C(C)C)OCC(C)C)=O)CCCCCC1CNC(=O)C1=CCCCO1 CC1CN(c2nnnn2Cc2cccc3c2CCCC3)CC(C)S1(=O)=O c1(NCC(C)CNC(c2cccc(N)c2OCC2CC2)=O)nnn2ccccc12 N1(C(c2cc(C)ccc2Cl)C(=O)NCCOCC)CCC2(CC1)NC(=O)CO2 c1(C(N2C(CNC(=O)CS(=O)(=O)NCC3CC3)C=CC2)=O)cc2scnc2[nH]1 C(=O)(C1CCc2scnc21)N(C1CCN(C(C2(C(=O)OCC)CC2)=O)CC1)C Cc1ccnc(O)c1C(N1CC=C(CNC(C2(F)CCS(=O)(=O)C2)=O)CC1)=O C1(N(C(c2c(F)ccc(C)c2)=O)C)CCN(C(C2(C#N)CC2(C)C)=O)CC12CC2 C(=O)(CC(C)(C)C)NC(C)C(N1CCC(CF)(NC(=O)CSc2nc[nH]n2)C1)=O CCC(C)CC(C)C(=O)N1CCOC(C)(C)C1C(=O)OCC N1(C(C(C)SC(C)C)=O)CCCC(C)C1CN=c1[nH]nc(O)s1 c1(C(=O)NCC2(C(F)F)CCN(C(CCCCOC)=O)C2)cnc2sccn12 Cc1c2ncnc1CN1CCC(C1)SCCN2.c1(CSC)ncn(CC(C)C)n1 c1(C(C)C)nc2c([nH]1)CC(C(=O)NCC(C)(C)CNC(=O)Cc1cnc[nH]1)CC2 c1(C(=O)NC2C(C)CCN(C(c3c(C)cc[nH]c3=N)=O)C2)c(C)ccc(C)c1O C1(C(=O)NCC2COC(=O)O2)C(O)CCN1C(c1csnn1)=O N1(C(C(N2CCCCCC2)C)=O)CCC(F)C(NC(=O)CCc2cnco2)C1 c1(OCC(=O)N(CCCNC(=O)COCCF)CC)ccsn1 c1(CC(=O)NC(CNC(c2c(CC)noc2)=O)C2CCC2)sc(O)nc1O c1(C(C)C)cc(C(=O)N(C(=O)OCC2CC2)C)[nH]n1 CCC(C)(CC)C(=O)N1CC(C)(C(=O)NC2CCC2OC)C1 c1(C(=O)NC2C(NC(c3csc(Cl)c3)=O)CC2)ccc(F)cc1Br c1(C(=O)NC(C2CN(C(=O)C=CCF)CCO2)C)cc2c(cc1F)OCC(=O)N2 C=CCC(C(=O)NCCCN(C(=O)CCCn1ccnn1)CCOC)N(C)C C1(OS(Cc2c(C)nc(Cl)s2)(=O)=O)CC2CCC1C(N)C2 n1(CCC(N2CCC(F)(CNC(C3CCN(C)C3)=O)C2)=O)cc([N+](=O)[O-])cn1 N1(C(=O)CN2CC3CC3C2)CC2(C1)SCCC2NC(C1CCN(C2CC2)C1=O)=O c1(C(=O)NC(C)CNC(=O)Cc2cc(C3CC3)on2)cc2c(cc1Cl)OCCO2 C1(C(=O)NCCN(CCOC)C(c2cc(C)c(C)nc2O)=O)CCc2nnnn2C1 N1(CC=CC(N2C3N(COC)C(=O)C(C3)C2)=O)C(=O)Cc2ccccc2C1=O N1(C(c2ccc(CC)cc2)=O)CC2CCC1C(CNC(=O)CC1CC(C)=NO1)C2 C#CCC(C(=O)NC)NC(C1CN(C(=O)C(C)NC=O)CC1CCC)=O C(=O)(CCC(=O)N1CCCCC1C1CCN(Cc2c[nH]c(Br)c2)C1)N(C(C)C)C c1(OC)cnccc1C(N1CC(CCOC)(NC(C2CC3CCCC23)=O)C1)=O CC(N=c1nc2sccc2c(NCCO)[nH]1)c1nnc(CC(CC2CCC2)CO)s1 N1(C(C(CC)(C)C#N)=O)CC2(CCCN(C(c3ccc(N(C)C)cc3F)=O)C2)C1 c1(C(N(CCNC(C(C(CC)O)C)=O)C2CC2)=O)ccc(Cl)c(C#N)c1 C12(C(N3C(CN(C(C(C(C)C)OCC)=O)C)CCCC3)=O)CCC(C1)C(C)(C)O2 c1(OC)ncc(Br)c(=NCC2CCCC(NC(C3C(C)(C)C3(C)C)=O)C2)[nH]1 c1(C(N2C(C)C(NC(=O)CCC(F)(F)F)CC2)=O)ncn2c1CCCC2 c1(N(CC(=O)NCC(C)(C2CC2)NC=O)C)cc2cc(Cl)ccc2o1 CCCCCC(C)CC(=O)NC1CCC1NC(=O)C(c1ccc(F)c(Cl)c1)O c1(OC)ccc(OC)c(CCNCC(c2ccc(Cl)cc2Cl)N2CCCCC2)c1 C1(OCC(C)NC(C2(C3CCCCO3)CCC2)=O)CCOCC1 C1(NC(C(N2CCOC2=O)C)=O)CCC(CNC(=O)Cc2ccnc(F)c2)CC1 N1(C(C(C(C)C)N2CCCCC2)=O)CCC2C(C1)NC(=O)CN2C(=O)CO c1(C(=O)OC)ccc(NC(C2CCN(Cc3cc(Cl)ccn3)CC2O)=O)c(Cl)c1 c1(OC)ccc(CC2CN(C(=O)C=CC(N)=O)CCO2)cc1Br.C12(CC1)NC(=O)N2 c1(C(N2C(CC)C(NC(C3C(F)(F)C34CC4)=O)CC2)=O)cc2cc(F)ccc2o1 C#CCC(C)(C)C(=O)NC(C1CCCN(C(=O)Cn2nnnc2C)C1)C N1(C(C2C(C(=O)OC)C2)=O)CC(NC(c2csc(-c3ccoc3)n2)=O)C(C)C1 C1(C(N(C)Cc2ccc(CNC(C3C=CCS3)=O)cc2)=O)C2CCC(F)(F)C12 C1(CNC(N2C3C=CC(C3)C2c2ccccc2)=O)CC2COCC(C1)C2 c1(OCC)ncccc1NC(C1CC2CC2N1C(C12CC(C1)C2)=O)=O C#CC1(CNC(=O)CCC2CCCN(C(c3nc(Cl)cs3)=O)C2)CCCC1 CC(C(=O)NC1CCC(CCC(=O)N(C2(C3CC3)CC2)C)C1)C(F)(F)F N1(C(C=CC(C)C)=O)CCC(CC(C)NC(=O)CCC2CCCN2C)CC1 C1(F)(C(=O)NC(C)C(C)(C)O)CCN(C(=O)Cc2cccc(O)c2)C1 C1(C(N2C(CN(C(C3=C(C)CCC3)=O)C)COCC2)=O)CC2(CO1)CC(F)(F)C2 c1(OC)c(C(=O)OCc2cc(O)c(F)c(F)c2)cc(I)cc1F C1(C(=O)NCC(C(C)(C)C)NC(C2C(C)CCO2)=O)CC(C)(C)OC(C)(C)C1 C1(NC(CC2CC(OC)C2(C)C)=O)CC2(C1)CC(NC(c1nocc1C1CC1)=O)C2 c1(C(N(c2ccnn2C2CCC2)CC(COC)O)=O)cnn(C(C)(C)C)c1 N1(c2nnc(CC)o2)CCC2C(CCCN2C(c2ncoc2COC)=O)C1 Cc1cc(C(=O)NC2CN(C(c3nc(-c4ccccc4)[nH]c3Cl)=O)CC2C)cnn1 C(CCCCC(=O)NC1(CO)CC2CCCC12)N(C(c1cn(CC)nn1)=O)C c1(C(N2CCC(NC(c3cnc(Br)o3)=O)C2)=O)ccc(Br)cc1F C#CCCCCCC(=O)N1CCC(OCCNC(c2cn(C)nc2-c2ccoc2)=O)C1 c1(C(=O)NCC2N(C(C(C)CC(N)=O)=O)CCCC2)ccc(S(=O)(=O)CF)cc1 CCC(F)(F)CC(=O)NCc1cn(CC(C)NC(C2CCC(C(N)=O)O2)=O)nn1 C1(NC(CNC(=O)OC)=O)CC2CCC(C1)N2C(=O)CC(C)CN(C)C c1(C(=O)NC2C(NC(CCCSC)=O)CCC2)cccc(NC2CC2)c1.S(C)(=O)(=O)N N1(CC2(CO)CCN(c3nc(C4(C#C)CCCC4)on3)C2)CCCN(C)CC1C N1(C(C(F)=CC)=O)CCN(C(c2cccc(CCC)c2)=O)CC1C(C)(C)C n1(CC(N2CC(NC(C(CCC)O)=O)C2)=O)nc2n(c1=O)CCCCC2 C(C1CCN(C(=O)CCc2ccsc2)CC1)=CC(=O)NCCCCCSC N1(C(c2c(C)occ2)=O)CCC(C2CN(C(C3(CC(C)C)CCC3)=O)C2)CC1 Cn1cc(NC(=O)CC2CC3(CC3)CN2C(c2cncc(F)c2)=O)c(C#N)n1 C(C(=O)Nn1ccccc1=O)C1(NC(C(C(C)(C)O)F)=O)CCC1 S(=O)(=O)(c1cccc(=NC2CCC(F)(F)CC2)[nH]1)NC1C(C)(CC)C1 c1(CNCC(c2ccc(OC)cc2)C)cc(Br)c(O)c(Br)c1 N1(CC(=O)N(C)C)CCC(N(C(N)=O)Cc2ccccc2)C1=O.C1C(=O)O1 C1(NC(COCCCCCC)=O)C2CN(C(=O)CSCCC#N)CC12 C(c1ncccc1C)=CC(=O)N(C1C(NC(c2cc(C)c(C)s2)=O)CCCC1)C c1(OC)cc(C#N)ccc1C(=O)NCC1CCCN1C(=O)CCC1CCOC1 c1(C(=O)OCC)cnc(N(CCOC)CC)nc1C.c1(C(=O)O)nccc(Cl)c1F C1(CNC(C2CN(C)C2)=O)CN(C(=O)CCCn2cccc2)CCO1 c1(C(=O)NCCCN(C(=O)C(O)Cc2cnc[nH]2)C)cc2c(cc1Cl)CCCC2 N1(C(c2c(C)ncnc2)=O)CC2(CCCC2)C1C(=O)NC(c1cc[nH]n1)C C1(C(C(=O)NC2C(NC(=O)CC3(O)CCCC3)CCC2)O)CCS(=O)(=O)CC1 C1(NC(C(CSC)OC)=O)CN(C(=O)CCc2ccc(F)cc2)CC1C(F)(F)F Cc1nn(C)c([N+](=O)[O-])c1C(=O)NC(C1(O)CN(C(=O)CCCS(C)(=O)=O)C1)C N1(C(C(C#C)(C)C)=O)CCC2(C1)CN(C(c1occ(C)c1C)=O)CC(C)O2 c1(CC)noc(C(=O)N(C)CCOCCNC(C2CCCN(C(N)=O)C2)=O)c1C c1(CNC(c2n(CC=C)nnn2)c2cncnc2)cc(Cl)nc(Cl)c1 CCC(C)C(C(=O)NCc1cncnc1)N(C)C(c1cnc(Cl)s1)=O C1(CCNC(=O)CSC(F)(F)F)CSCCN1C(C1CCSCC1)=O c1(C(N(CC(C)NC(=O)CNC(=O)CC(F)(F)F)C)=O)cnnc(C2CC2)c1 c1(C(=O)NC(C)CC2CN(C(C3CC3OCC(F)(F)F)=O)C2)nn(C)cc1CO C1(CNC(c2cnc(C(C)OCC)s2)=O)CCN(C(=O)CCCCCF)CC1C c1(OCc2noc(CO)n2)ccc(Cl)cc1Cl.N1(C(C(COC)OC)=O)CCCC12CN2 C(C)(C)(CC(=O)N1CCCCC1C1(NC(=O)CCCC2CCCO2)CC1)OC O(NC(=O)C(CNC(=O)CC1CC(=O)NC1=O)CC=C)CC(=C)Cl c1(NC(C2CCCCN2C(c2cnc(C3CC3)nc2)=O)=O)ccc(Cl)cc1F c1(CCCC)ncc(C(=O)N(CCC(Cc2ccccc2)NC(=O)CC=C)C)s1 c1(C(N(CC(C)NC(=O)C(F)(F)c2ccccc2)C)=O)cc2nc(=O)ccn2[nH]1 N1(C(c2ncn(CCOC)c2)=O)CCCN(C(=O)Cn2nc(C)oc2=O)CC1 c1(NCCC(C)(c2nnnn2C)NCCNC(=O)OCC)ccc(F)c(Cl)c1Cl C1(C(N2CCC(C)(CC)C2)=O)CC(F)CCN1C(=O)Cc1cncnc1O C1(CCN)CCCCN1C(=O)C(C)C.c1(OC)csc(C(N2CCC2)=O)c1 c1(OCC(=O)NCCN(C(CCC)=O)CC2CCCCC2F)ccc(Cl)c(Cl)c1 N1(C(C(C)c2cc[nH]n2)=O)CCN(C(c2cnn(C)c2C(F)(F)F)=O)CC1C1CC1 c1(CNC(C(CSC)O)=O)cc(Cl)ccc1F c1(C(=O)NCC2CCC(NC(C(C)C3CCOC3)=O)C2)n[nH]c2c1COC2 C1(O)(CCNC(CN(CCCCCC)C)=O)CCN(C(=O)Cc2nncs2)C1 C(CC)(CC)(CCNC(=O)CC1COC(C)(C)CO1)NC(C=CCCC)=O N1(C(C(COC)O)=O)CCC2(CCOCC2)C(CNC(C23CC(CCO2)C3)=O)C1 C1(CC(=O)NCC(C)C(=O)NCCc2ncccn2)CC(=O)NC1=O C#Cc1cc(C(N2CCN(C(c3ccnc4[nH]ncc34)=O)C3CC23)=O)cc(F)c1 O=C1CCC(C(=O)NC2CCCC(NC(C3(O)COC3)=O)CC2)=NN1 C1(C(N(C2CC(CCO)C2)C)=O)CC12CCN(C(=O)CC1(C#N)CCC1)CC2 N1(C(CCOC)=O)CC(C2CN(C(c3cc(C(C)=O)oc3C)=O)C2)C1.CC(F)(F)F c1(C(=O)NCC23N(C(CCC#C)=O)CCC2CC3)c([N+](=O)[O-])cnn1CC(F)F c1(C(N2CC(O)(CNC(c3cnc(SC)s3)=O)C2)=O)cnn2c1OCCC2 c1(NCC)cc(S(=O)(=O)NCCC(C)(C)C)ccc1C=CCC(=O)NC1CC1 CC(CC(=O)NCC1CCC1NC(=O)C=C1CCOCC1)n1cccn1 C1(CNC(C(C=C=C)C)=O)CC2(CCN(c3nnc(COC)s3)CC2)CO1 CC1=CC(NC(C2(CO)CCN(C(=O)CN3CC(C)(C)C3)C2)=O)CCC1 CCC(CC(C)O)N=c1cc(C)[nH]c(=NCCCNC(=O)Nc2ccsc2)[nH]1 N1(C(c2c(C)ocn2)=O)CCC2CN(C(=O)C(C)NC=O)CCC2C1 C1(NC(C(C=C=C)C)=O)CCN(C(=O)C2=C(Cl)CC2)CC12CCC2 C1(NC(CC=CC=C)=O)CC(CNC(c2cccc(C)n2)=O)CC1O C1(C(=O)NC2CC3(CC(NC(C4CC(C)(O)C4)=O)C3)C2)COCC2(CCC2)O1 C1(C(N(CCCNC(=O)CCCCCNC(C)=O)CC)=O)CCN2CCOCC12 C1(COC)(NC(C2CCCN2C)=O)CCN(C(=O)C(C)CC2CCCC2)CC1 Cc1cc(C(N2CCCC2(C)CNC(=O)Cc2cc(C)ccc2O)=O)cc(C)c1 c1(C(=O)NCC=CCC)cc(SC)oc1C.N12CCCC1C1(CC1)C2=O c1(C2(O)CN(C(C(=O)Nc3cnn(-c4cccnc4)c3)=O)C2)cccc(F)c1 c1(C(=O)OCC)sc(NC(=O)CC2CN(C(c3cncc(C)n3)=O)C2)cc1C C1(C(N2C(CN(C)C(c3nnc(O)cc3O)=O)COCC2)=O)CCCC2(CC2)C1 Nc1cc2ccccc2c(NC(N2CCC(OC(F)F)C2)=O)n1 N1(C(c2cc(C)c(O)cc2)=O)CC(NC(=O)CC2(O)CCCC2)C2CCCCC12 N1(C(C(CCN(C)C)NC(CC2C(C)CCO2)=O)=O)Cc2ccc([N+](=O)[O-])cc2C1 Nc1ccc(C2CCCC(NCCC3CC3c3ccccc3)C2)cc1 c1(C(N2C(C)CCC(NC(Cc3c(C)noc3)=O)C2)=O)ncnc2c1cnn2C Cn1c(C(F)(F)F)ccc1-c1cn(C2CN(C(c3cccnn3)=O)C2)nn1 C1(C(N(C(C)CNC(c2csc(-c3ccco3)n2)=O)CC)=O)CC2C=CC1O2 CN1CCCCC1C(=O)NC12CC1CN(C(c1sc(NC3CC3)nc1Cl)=O)C2 c1(C(N(CCN(C(c2ncccc2CO)=O)CC)CC)=O)c(OC)ccnc1O C=CCCCC(C(=O)NC1CC(CC)C1)NC(c1cc(C)[nH]c1C)=O N1(C(C=C(C)C(C)C)=O)CC(NC(C23CCCC2(C(N)=O)C3)=O)CC(C)C1 N1(C(c2c(C(C)C)ncs2)=O)CCC(CNC(C2(C(N)=O)CC2)=O)(OC)C1 Cc1noc(C(C)C)c1C(=O)NCC1CC(C)N(C(c2ncc(Cl)s2)=O)C1 N(C(=NCC(F)F)N1CCC(S(=O)(=O)N2CCCCCC2)C1)C(COC)C c1(C(=O)NCCC(C)NC(c2nc(C)sc2)=O)ccc(C2CC2(F)F)cc1 CCC(C)(C#N)C(=O)N1CCC(C)(CCNC(c2cc(C)cc(C)n2)=O)C1 C(C(C)(C)C(=O)NCC1CCC1NC(c1cccc(C)n1)=O)NC(C)=O Cc1nc(C(=O)N(C(C)(C(=O)N2CC(c3ccon3)C2)C2CC2)C)co1 C1(C(=O)NCCSCC(=O)NCC(n2cccn2)C)CC2CCC2C1 N1(C(C(COC)NC(C)=O)=O)CCN2CCCC2C1.N12CCCC1C2=O c1(C(N2C(C(=O)NC(c3cnccn3)C)C=CC2)=O)ccc(CC#N)cc1 c1(OCC(=O)OC(C)C)ccccc1CN=C(NCC(F)F)NC1C=CCCC1 CCC1=NOC(C(=O)NCC=O)C1.C(CNC(N)=O)O C1(NC(CCOCC(C)C)=O)CC2CCC1(C(=O)N(CC(F)(F)Cl)C)C2 C1(=CC(=O)N(CCNC(c2cc(C(N)=O)n(C)n2)=O)CC)CCC(C)(C)CC1 Cc1nc(O)nc(C)c1CC(=O)NC1CN(C(c2cccn2C)=O)CCC1(C)C N1(C(=O)OC)CCC2(CC1)OCCC2.c1(C(=O)NC(C)(Cl)C2CC2)cc[nH]n1 C(=O)(CC(C)CCC=C(C)C)NCC(C)N(C(=O)CN1CCS(=O)CC1)CC C#CC1CC2(CC(C(N3CC4C(NC(=O)CN5CCC(C)C5)C4C3)=O)C2)C1 C(=O)(CC(F)(F)C(C)C)N1CCC(CNC(C2(C=C)CCC2)=O)CC1C N1(C(CC2(NC(C(C)=C3CCCC3)=O)CC2)=O)C2CCC1CN(C(=O)CO)C2 CC12CC(NC(c3cccc(F)n3)=O)(C1)C1(CN(C(=O)CC3CCC(O)C3)C1)O2 n1(CC)ncc2c1CCCC2NC(=O)CCNC(=O)C(F)OC(F)(F)F n1(CC)cnc2c(N(CCCF)C)[nH]c(=NCCCc3cc(C)[nH]n3)nc12 c1(C(=O)NCC(C)NC(C(C)(CO)OC)=O)cccc2nc(O)n(C)c12 N1(C(c2c(C)nsc2)=O)CCC(NC(c2ccn(CCO)c(=O)c2)=O)C(F)(F)CC1 c1(C(=O)NC2(CNC(c3nc4ncccn4n3)=O)CC2)ccc(=O)n2c1CCC2 C1(NC(C)=O)CC12CCN(C(=O)CC1CC(OC)C1)C2.C1C(=O)N1CC C1(NC(C2(COC(C)C)CC2)=O)CCN(C(=O)CCC2CC2(F)F)C12CC2 c1(C(=O)NC(C(=O)OC)CC2CCCCC2)cc2cc(C)ccc2nc1C C#Cc1cncc(C(N2CCC(CCNC(=O)C(C)C#N)C2)=O)c1 CC(C(C)(C)C(=O)NCCc1ccncc1F)NC(C1CC(=O)NC1(C)C)=O Cc1ccc(C=CC(=O)NC(C(C)NC(=O)CN2C(=O)CCCC2=O)C(C)C)cc1 c1(CC(=O)NCC(C)(C)NC(=O)C(F)CC2CCC2)ccccc1C(F)(F)F Cc1cc(C(=O)NCC2(C(F)F)CCN(C(c3ccno3)=O)C2)ccc1Cl n1(CC)cnc2c(NCc3cc(C)co3)nc(N(C)Cc3ccc(Cl)o3)nc12 c1(CN(C(=O)C(c2ccc(Cl)cc2)CO)C(C2CC(=C)CN2)=O)ccc(Br)c(C)n1 c1(C(N2CCC3CN(C(CCCC4C(C)C4)=O)CC32)=O)cnc2ncnn2c1O O(NC(=O)C#CCNC(=O)CC1(COC)CC1)CCC=C C1(CCOC)CN(C(c2cccc(N(C)C)c2)=O)CCN1C(=O)CC(CC)OC c1(C(=O)NCC23OCC(NC(CCC(=C)C)=O)(C2)C3)ccc(C#N)cc1 c1(C(=O)NCC(C)NC(=O)CC2(CO)CCOCC2)cc2c(nc1N)CCC2 N1(Cc2nc(NC(=O)NCCCCCCCC)sc2)CCc2cc(Cl)nnc2C1 C12CCC(c3nnnn3C)(C1)NC2=O.c1(CC)cccc(CSC(C)(C)C)c1 N1(C(c2cc(CNC(c3nc(CC)oc3C)=O)oc2)=O)CCC12CC(C)C2 c1(C(N(CC(C)(C)CNC(=O)C=CC2CCC2)CC)=O)cc2nc(C)ccc2o1 C1(NC(c2cc3n(n2)CCCN3)=O)CCC2CCN(C(=O)C=CCF)C1C2 C1(S(C)(=O)=O)(C(=O)NCC(CN(C(C2(CCC=C)CC2)=O)C)C)CC1 CC(C)C(CCC(=O)NCC1CCCC1O)NC(C1C2COCC12)=O c1(C(N(C2CC(C)(C)C2)C)=O)cc(S(=O)(=O)NCC2CC2)ccc1F CCC(CC(=O)NC1(CNC(C2CCN(C)CC2)=O)CCCCC1)C(C)(C)C c1(-c2ccc(CN(C)Cc3ccc(OC)cn3)nc2)ccc(O)cc1Cl c1(OC)c(C(=O)NC2CCN(C(c3ccn(C)c3)=O)C(C)C2)oc2ccccc12 C(=O)(CCCC(F)(F)F)NCC1(C)CCN(C(c2cc(OC)nc(C)c2)=O)CC1 C1(CC)CCC(C(=O)NCCCCCNC(C2COCCN2CC(F)F)=O)CC1 Cc1cccc(C2CC2C(=O)NCC2CC(NC(c3cc(C)sn3)=O)C2)c1 N1(C(C(C=C)OC)=O)CC(NC(=O)Cc2csnc2C)C2(CC2)C1 C(C(C)(C(=O)N(C)C(C1CCCC1)C)NC(c1cc(=N)[nH][nH]1)=O)SC c1(NC2(CNC(C(CC)(CC)CC)=O)CCOCC2)ncnc2c1c(Br)nn2C C=C(C)C(C)(O)C(=O)NCC(C)(O)CNC(c1cccc(F)c1C1CC1)=O C1(OCC)CCCN(C(=O)CCCN(C)C(c2nc(=N)cc[nH]2)=O)C1 c1(C(=O)NCC2OCCN(CCC=C)C2)cnc2nc(Cl)ccc2c1 C(CC)(CC)(C(C)C)N(n1ccnc1Cc1ccsc1-c1ccccc1C)CC N1(C(=O)Cn2nnc(=O)[nH]2)CCC2CN(C(c3cc(C(F)F)on3)=O)CC2C1 C1(CN(C(CN(C(=O)CCOCCOC)CC#C)=O)C)CN2CCC1CC2 C(c1ccccc1)=CCn1cc(C2CCN(C(CC3(C#N)CC3)=O)C2)nn1 c1(C(=O)NC2(c3cccc(Cl)c3)CC2)ccc2c(c1)NC(=O)CCN2C c1(CN(C=O)CC2CN(S(CC=C)(=O)=O)C2)cc(C)cc(F)c1 N1(C(c2c(C)cc(=N)[nH]c2)=O)C2CCCC1CN(C(C1CCC(F)(F)CC1)=O)C2 C1(N(C(c2ccc(CCNC(C(C)=C3CCC3)=O)[nH]2)=O)C)CCCCC1C C(=O)(CC(CC)NC(c1cc[n+]([O-])cc1)=O)N(CC(CC)OC)C c1(C(=O)NCC(CC(=O)OCC)C)cc[nH]c(=N)c1N CCC(CC)C(C)C(=O)NCC1CCN(C(=O)CN2CCCC2CO)CC1(F)F C1(C(=O)OC)CN(C(=O)NCC(C)(C)CC(C)O)CC1(C)CCC C(c1ccc2occc2c1)=CC(N1CCN(C(CC(CC)SC)=O)C(CC)C1)=O c1(C(=O)NCCN(C(=O)CC2CCCN(C)C2)CC)c(F)cc(F)cc1Br Cc1cc(C(N2CCCC(C)(C)C2CNC(C2CCCO2)=O)=O)c2c(c1)CCC2 N1(C(C(C)CC(N)=O)=O)CC2CCC(N(C)C(c3cc(F)ccc3N)=O)C2C1 c1(C(N2CC(N3CCCCC3=O)C2c2ccccc2)=O)sc2c(c1CO)CCC2 C1(C(N)=O)C2CC3C(C2NC(C2(CNC(C4CCC4)=O)CC2)=O)C13 C1(n2ccnc2)(C(N(C(CNC(=O)Cc2csnn2)C2CC2)C)=O)CCCC1 c1(C(N(CCN(C(C(C)SC(C)C)=O)C)C(C)C)=O)cc(C(C)C)on1 C(=O)(CCS(=O)(=O)C(F)(F)F)N1CC(NC(C2(C=C)CC2)=O)C(CO)CC1 n1(CC(=O)NCCC(N2CCC(CN(C(=O)C=C3CCC3)C)C2)=O)ccccc1=O C1(CC)CC2CCC(C1)N2C(=O)C(Cc1ccco1)NC(=O)CCC(C)C N1(C(C2CCC(=O)O2)=O)CC2(CCC2)CC1C(N1CCC2CCCC2C1)=O N1(C(C23OCC(C)(C2)C3)=O)CC2(COC(CNC(C3CCC(O)CC3)=O)C2)C1 C12C(C)CCCN1C2=O.c1(NC(c2cccc(OC)c2)=O)nccc(OC)c1C C1(N2CC(C3CN(C(C(=O)C=Cc4ccsc4)=O)C3)C2)CC2CCCCC2NC1=O c1(C(=O)NCC(CN(C(=O)CCCn2ccnn2)C)O)nc(C(F)(F)F)cn1C c1(C(=O)NCC2CCC(NC(c3c(CC)scc3)=O)C2)cc(OC)cnc1F Cc1cc(C(=O)NC2CCC2CNC(c2cn(C3CC3)nn2)=O)cc(C)c1Cl CN1CCC(N(C)C(c2ccc(CO)cc2)=O)(Cc2nc(C3CC3)nn2C)CC1 c1(C(N2CC(NC(C(C)=CC3CC3)=O)C3(C2)CCC3)=O)n[nH]c2ccc(F)cc12 CC1(C)C(NC(=O)Cn2ccccc2=O)CCN1C(=O)C1=CCCCC1 c1(C(N2CC(CNC(C(C3CC3)OCC)=O)C(O)C2)=O)nccc2occc12 Cn1c(C(=O)NCC(C)(C)CC2CN(Cc3cc[nH]n3)C2)cc(Cl)c1Cl C1(NC(C2CC=CCC2)=O)CCSC12CN(C(c1scnc1C(F)F)=O)C2 C1(CNC(C(CC)SC)=O)CCCCN(C(=O)CC2CCC2)C1 C1(CC)CCC(NC(N2CC(c3ncnn3C)(CC#N)C2)=O)CC1 C1(N(C(=O)C=CC=C(Cl)Cl)CCC)CCN(C(=O)C(F)F)C1 C1(C(c2nnnn2C2CC2)NC(C(CC)OC)=O)CN(C(=O)C2CC2)CC1(F)F CC12COC(C(=O)NCC=C3CN(C(=O)CN(C4CCCC4)C)C3)(C1)C2 C1(NC(CNC(c2cnc(OC)s2)=O)=O)CC12CCN(CC(=O)NC1CC1)CC2 C(=O)(C(C(C)C)N1CCCS1(=O)=O)NCCCC1N(C(CC=C)=O)CCC1 C(C(C)C(F)C(=O)NC(c1nc(=O)o[nH]1)(C)C)N(C(COC(C)C)=O)C1CC1 N#CC1(CC(N2CCN(C(C3CCC(O)CC3)=O)CC2)=O)CCCCC1 C1(C(N2CCC(NC(CCCN(C(C)C)C)=O)C2(C)C)=O)CCCCCC1(F)F C(C1=CCN(C(=O)OC(C)(C)C)CC1)NC(C(=O)NCCC)=O Cc1ccnc(C(=O)N(C2CCN(c3nccc(CC#N)n3)CC2)C)n1 N1(C(C(c2c(C)noc2C)(C)C)=O)C2CCC1C(CNC(=O)C(C)NC(N)=O)C2 C1(C(=O)OC)CCN(C(=O)c2cccc(Cl)c2C)O1 N1(C(C(CC)C2CC2)=O)CCN(C(c2cc(C3(C)CC3)on2)=O)C(CN(C)C)C1 C1(C(=O)NCCCCNC(=O)CCc2cn[nH]c2)C2CCC3C(C2)CC13 C12(NC(c3c(-c4cn(C)nc4)ocn3)=O)CC1CN(C(C1C3CC4C(C3)C14)=O)C2 C1(C(N2C(C)CN(C(C3CCC3)=O)CC2)=O)CCn2c(O)nnc2C1 N1(C(C(C=C)C)=O)CCC(CNC(=O)CSc2ccc(C)cc2)C12CCC2 C1(CNC(C(C)OCC)=O)CC2CCC1N(C(C1C3CCOCC13)=O)C2 c1(OC)ccc(Cl)c(CN2CCSC(C(=O)Nc3ccc(Cl)c(C)c3)C2)c1F N1(CC2CC(=O)N2)CCOCC(NC(c2ccn(-c3ccccc3)n2)=O)C1 C#CCC(CC#C)C(=O)N1CC(C)C(C)(CNC(=O)C=Cc2cncnc2O)C1 N1(C(C2(OC)CCOC2)=O)CCN(C(=O)CCN2CCCC2)C(C2CCC2)C1 c1(C(N2C(C)(C(=O)NC)CC(O)C2)=O)ccc2ncccc2c1 CC(=NO)C1CC(C(N2CCC(C)(CNC(C3(C)CC3)=O)C2)=O)C1(C)C C1(C(=O)NCC2N(C(c3c(OC)ccs3)=O)CC(O)C2)CN2CCN1C(C)C2 n1(CC)nnc(C(N2CCC(CCCNC(C3(C)C=CCCC3)=O)CC2)=O)c1C Cc1cc(C(=O)NC)nc(O)n1.N12C3CCC1C(C3)C(=O)C1CN2C1.C(C(F)F)O C1(NC(c2ccc(CC)o2)=O)COCCC1NC(C1CCC(N(C)C)CC1)=O N1(C(c2cnn(-c3cccnc3)c2)C(=O)NCC(C)C)CCS(=N)(=O)C(C)C1 Cc1ccc(C(N2CC3C(CNC(C4C5CC6C(C5)C46)=O)(C3)C2)=O)c(F)c1 c12ccn(c1)CCNC(=O)C1(C(OCC)CNC2=O)CC1.C1(CC)CCCO1 N1(C(C(n2c(C)nnn2)Cc2ccccc2)=O)CC2CC(NC(=O)CO)C(C2)C1 c1ccc2oc(OCCOc3ccc(I)s3)nc2c1 C(=O)(N=c1cc(Cl)nc(SC)[nH]1)C1N(C(c2cc(OC)cc(C)c2)=O)CCSC1 Cc1c(C=CC(=O)NCC2CC(NC(c3cc(N)c(Cl)cn3)=O)C2)cnn1C N1(C(C(C)C(F)(F)F)=O)CCOC2CN(C(C3(F)CCS(=O)(=O)C3)=O)CC12 c1(CC(=O)NC2C3CCN(C(c4ncc(C)nc4)=O)C32)cccc2c1OCCO2 Cc1cccc(F)c1C(=O)NCCN(C(C12COCC1C2)=O)C1CC1 C1(C(N(c2nccc(N)c2Cl)C)=O)CCC(=O)N(CC(=O)O)CC1 C(=O)(C1=CC2CCCCCC12)NCC1C2CN(C(CC(CCCCC)O)=O)CC21 N1(C(COCCC=C)=O)CCC(F)(CNC(C2CCC2C)=O)C1 c1(NC2CCN(C(c3c(C)cc(C)nc3)=O)CC2C)[nH]c(=O)n(C)c(=O)c1C#N O=C(C1SCCc2ccccc21)NCC1CCCN1C(=O)Cc1cccc(F)c1 CON(C)S(=O)(=O)c1ccc(Cl)c(C(=O)N(C)CCNC(C2(C)CC2(F)Cl)=O)c1 Cc1oc(Br)c(C)c1C(N1CC(NC(c2cnc(O)o2)=O)C(C)C1)=O c1(N2CCC3(C(C(=O)NCC(C)(F)F)C3)C2)ncc2ccc(F)cc2n1 C12(NC(CCCCC)=O)CCCC(NC(=O)Cc3ccc(F)cc3Br)(C1)C2 CC1(C)CC(CC(=O)NC2CCN(C(=O)CCCc3nccs3)CC2F)C(=O)O1 N1(C(C(C)c2cccs2)=O)CCCC1(C)NC(=O)CSc1n[nH]c(O)n1 C(=O)(CCC1CC1)NCC(N(C(C1C(CN(C)C)C1)=O)C)C1CC1 CC1CCC(F)(F)CN1C(=O)CCNC(=O)CN(C(=O)C(O)CN(C)C)C c1(CS(C)=O)cccc(C(=O)NCC(O)CNC(C2CC23CC3)=O)c1 C1(CNC(C(CCOC)(C)C)=O)CC2CCC(C1)N2C(=O)C=C(C)I c12cc(ccc1F)C1C=C2CC1.CC(F)(F)C1(CC(=O)NCCCNC(N)=O)CC1 C=CCCCCCC(=O)NCc1nc(Cl)oc1C.C12CC(C)(C)CN1C2=O c1(N2CCC(C)C(C)(C)C2)nccc(=NC(C)c2ccc(Br)s2)[nH]1 c1(C(=O)NC2(CC(N3CC(C)C(CN(C)C)C3)=O)CC2)c[nH]c2cccnc12 C1(N(C(CCN(C(=O)CC2CCCO2)C)=O)C2CC2)CCC(=O)NC1 C(C(=O)NOCCN(C)C)N(C(CC1CC(=C)C1)=O)CC c1(C(N2CCN(CCCO)CC2C)CC(=O)NC)c2c(nn1C)CCOC2 NC(=O)CCCCC(=O)NCCC1(C(=O)NCC(O)CN(C)C)CCC1 CC(c1cccc(Cl)c1)=CC(=O)NCC12CC1CN(C(c1cnc(C)nc1C)=O)C2 C1(C(N(C)CC2CCOC2)=O)CCN(C(c2ccc(O)cn2)=O)C12CC2 CN1CCN(C)C(CNC(C2(C)CCCN(C(=O)CN3CCC(F)CC3)C2)=O)C1 CCCC(N=c1[nH]c(=NCC(Cl)Cl)[nH]c2c1CSC2)c1ccc(Cl)s1 CC1(C)OC2(C(=O)NCC3(NC(C4CCCCC(=O)N4)=O)CCOC3)CC1C2 C(=O)(CCCCC(C)(C)OC)NCC(CCCC)NC(=O)Cc1ccno1 N1(C(c2cccc(OC)c2F)=O)CCC(NC(C2(F)CCC2)=O)C(CO)CC1 C1(NC(C(C)N(CC(C(=O)OCC)C)CC)=O)CCCOC1c1cc[nH]n1 CC(C)C(CNC(=O)C(C)C1CC1)NC(=O)C(F)CC1CCCC1 c1(C(=O)NCCN(CCC)C(c2cc(C)[nH]n2)=O)cnc(Br)s1 N1(CC)CC2CCCOC2C1.c12ccc(cc1)C(C(C)C)C(=O)N2 C(C)(C(O)C(=O)NCc1ccc(C(=O)N(CCc2cccc(O)c2)CC)o1)SC C1(CC)CC(CC(=O)NC(c2ccc(F)cn2)C)CCO1 O=C(C1=C(Cl)CCCC1)N1CCN(C(=O)CN2CC(F)(F)C2)C(C2CCCC2)C1 c1(C(=O)NC2C(C)N(C(C3CCN3C3CCCC3)=O)CC2)cccc2c[nH]nc12 c1(C2C(C(=O)NC3CCC(C(C)(C)C)C3)C2)cccc(O)c1Br c1(NCC2N(C(C34CC(C)(OCC3)C4)=O)CC2)cc2c(cn1)C(=O)CCC2 c1(C(=O)NCC(C)NC(C(C=C)O)=O)cnn2c(C)ccnc12 N1(C(c2cn(CCCCF)nn2)=O)CCCCCC1CNC(C12CCC1C2)=O Cc1ccc(C)c(SCC(N2CC(NC(=O)CC3CCCOC3)C(C)(C)C2)=O)c1 N1(CC(F)(F)F)CC(=O)N(CCC(N)=O)C1=O.CC1CSC1 c1(NCCNC(C23CC(C(=O)OC)(C2)C3)=O)c(Cl)cnn1C1CCC1 c1(CNC(=O)NCc2ccc(C(=O)OC)cn2)cnc(C2CCCC2)[nH]c1=NC C#CCCCC(C)C(=O)NC(C)(C)CCNC(=O)COCC(=O)N(C)C Cc1nc2c(C(N3CC4(CCC4N)C3)=O)cccc2o1.N1(C(=O)CC2CC2)CCCC1 N1(CC(=O)NC(C)CCNC(c2cnn(C(C)(C)C)c2N)=O)CCCCCC1=O c1(C(N2C(CNC(CCC)=O)CC2)=O)nc2ncccn2n1 c1(CNC(C(=O)N(C2C(C)=C(C)CCC2)CCO)=O)cccc2nccnc12 c1(CC)onc(C(N2CCCC(CCNC(=O)CN3CC(C)C3)C2)=O)c1C N1(C(C2(OCC)CCOCC2)=O)CCC2CCN(C)C2C1.n12cc(nn1)c(=O)[nH]2 C1(C(=O)NC(C(C)NC(c2cc(C(C)=O)on2)=O)C)CCc2nc(O)[nH]c2C1 c1(C(N2CC3CN(C(C4CC(OCC)C4)=O)C3CC2)=O)cccc2nccnc12 C1(NC(=O)CSC(F)F)CCC(C(=O)NCC(CNC(N(C)C)=O)(C)C)CC1 c1(C(=O)NCC(C)NC(=O)CS(=O)(=O)CC2CCCO2)cncc(Cl)c1Cl c1(C(=O)OC)cc(CNC2C3CC4C(C3)C24)ccc1OC c1(C(=O)NCC(CO)NC(C23CSCC2C3)=O)coc(C2CCC2)n1 C(CN=c1ccc(C#N)n[nH]1)(CC(C)C)NC(c1c(C)ccc(C)c1C)=O c1(C(=O)NC2C(F)CCN(C(c3nc(CCC)oc3)=O)C2)ccsc1S(N)(=O)=O CC1c2sccc2CCN1C(=O)Nc1cc(Br)ccc1O N1(CC(=O)NCCCN(C)C(c2occc2Cl)=O)CCOC1=O C(=O)(C(COC)CC(C)C)N1CC(N(C(CC(CC)(F)F)=O)C)C(C)(C)C1 C(=O)(C(C)C(C)C(C)(C)C)N1CC(N(C(Cc2cc(C)on2)=O)C)C1 N1(C(C2(CC)CCCC2)=O)CCCC(O)(CNC(c2cc(C(F)(F)F)n[nH]2)=O)C1 c1(C(N(C)CC2CCCC(NS(=O)(=O)C3CC3)C2)=O)ccc(NS(C)(=O)=O)nc1 c1(CN(c2cc(N3CCC(C)(O)CC3)ncn2)CC)cnn2cccc2c1 C(=O)(CCCC(C)(C)NC(c1cc(C)ns1)=O)NCc1cccc(CC)c1 C1(CC(=O)N(CC(CCOC)NC(C=C(CC)CC)=O)CC)(OC)CCOCC1 c1(OC)cnccc1CNC(=O)C(=O)NCCCc1cn(CC(F)(F)F)nn1 c1(C(=O)NC(CN(C(C2CCCC(OC)C2)=O)C)C)ncnc2ccsc12 c1(NC(C2N(C(c3ccc(CC#N)cc3)=O)CCSC2)=O)csc2nccnc12 CC1CC(CS)CN1c1cccnc1Oc1ccncc1.c1(S)ccccc1 c1(CC)cc(C(N2CCCC2C(C)NC(c2ccc(Cl)o2)=O)=O)sc1C C(=O)(CCC(C)CN(C)C)NCc1c(CNC(C2CCC(C)O2)=O)occ1 C(=O)(C#CC1(CC)COC1)N1CC(CC)N(C(C2C=C(C)CS2)=O)CC1 N1(CC)CCN(C(C2CN(C(=O)C(F)CC3CCOC3)CCO2)=O)CC1 C(C)(CCOC)(c1nnnn1C1CCC1)NC1(CC)CCC1 C1(CCc2cn(C(C)C(=O)O)nn2)CCCCC(=O)C1.C1C(=O)N(CC#N)CCS1 C(C(=O)NCC1CC(O)CN1C(=O)CC(C)(C)O)(C(C)C)SCC CC1(CNC(=O)CCc2ccc(Cl)s2)CCC(NC(=O)CCCOC(C)(C)C)C1 C1(NC(CC(CC)CC)=O)CN(C(=O)Cc2c(C)cccc2C)C2(CCC2)C1 C1(C(=O)NCC(CCCC)NC(c2cc(C)c(=O)n(C)c2)=O)CCCC1P(C)(C)=O C12(OCC)CCC(C(=O)NCCn3cc(CN(C)CCO)nn3)(CC1)C2 N12CCCC(C)(C1)C2=O.N1(C(CCC(C)SC)=O)CCCC(C)(F)C1 N1(C(CC(C)O)=O)CCC(C)N(C(=O)Cc2c[nH]ccc2=O)CC1 N1(CC(=O)NC(CCN(C(Cc2scc(C)n2)=O)C)C)C(C)CCC1C C1(OC)CCCN(Cc2ccc(N3CCCOC3=O)cc2)C1C(=O)O N1(C(CC2C(C)C2(F)F)=O)CCN(C(=O)CC2OCCO2)C(C2CCC2)C1 N1(C(c2n(C)ncn2)=O)CCC(C2CCCN(C(c3cnc(O)n3C)=O)C2)CC1 N1(CCCC)CCC2(CCCC2C(=O)N=c2cc[nH][nH]2)C1.C(=O)N CCC(CC(=O)NCC(c1ccccc1F)NC(C1(F)CCOCC1)=O)SC C(CN(C)C)(CO)(CO)NC(N1CC(Oc2cn(C)nc2)C1)=O.C(C)(C)(C)C(=O)O C(CO)(CCC(C)C)NC(C(C1CCC1)NC(CC1ON=C(CC)C1)=O)=O C1(CNC(C(C)SC)=O)CC2(CCOCC2)CN1C(C1(C)CC(C#N)C1)=O C1(C(=O)NC2(C=C)CCCCC2)CC2(CCN(C(c3cnsn3)=O)C2)C1 C=CCCCCCN(C(=O)C(CCC1CCC1)NC(=O)C(C)N1CC(C)C1)C C1(C(N2CCC(N(C(c3cc[nH]n3)=O)CC3CC3)CC2)=O)CCC2CC2CC1 C(=O)(CC(C)(C(F)F)N(C)C)N1CC(C)C(c2ccc(C(F)(F)F)cc2)C1 N1(C(CCCN(CCC)CCC)=O)CCC(NC(C2CN(C)C(=O)N2)=O)C(O)C1 N1(CCC)CCCN(C(CCc2ccc(C)c(C)c2)C(=O)NC2CC2)CC1 N1(C(C(C)CN(C)C)=O)CCCC(C2CCN(C(=O)C(C)C)CC2)CC1 C1(=O)C(C)(CC)C(=O)NCCCC2CN1CCO2.C(C(=O)OCC)=CCOC O=C(C1=CCC(F)(F)CC1)NCC1CCN1C(=O)CCS(=O)(=O)c1ccccc1 C(=O)(C(CNC(=O)C(c1ccc(C)cn1)(F)F)Cc1ccc(I)cc1)NC Cc1ccc2c(c1)SC(C(=O)N(C)CCNC(C1CCn3nncc3C1)=O)C2 c1(C(N(C)CC2CCN(C(=O)CCC3CC3)C2)=O)cnn2cccc2c1 C1(C)(CC(N2CC(NC(c3n(CC)ccn3)=O)C(C)C2)=O)CCS(=O)(=O)N1 C1(O)(c2cn(C3CCC(C)CC3)nn2)CCN(C(C2(Br)CC2)=O)CC1 C(C)(C(=O)NCC1CCC1NC(=O)Cc1cn[nH]c1)OCCC#C N1(C(c2ccc3nc(N4CCCC4)oc3c2)=O)CCC(O)C2(CCCNC2=O)C1 C1(O)(CCNC(c2scnc2Cl)=O)CCN(C(C2(c3ccccc3Cl)CC2)=O)C1 C12(NC(c3cnc(NC(C)=O)o3)=O)CCCN(C(=O)CC(C)(C)C)C1C2 CCCCC(O)C(C)C(=O)N(CCC(C(C)C)NC(=O)CC(C)(C)CCOC)C C1(CNC(C=Cc2ccc(C)o2)=O)CC2CN(C(c3ccc(C#N)cn3)=O)CC12 N1(C(C(CCC)C)=O)CCN(C(=O)Cc2nocc2CC)C(C2CC2)C1 CC(=O)C(C)(C)CC(=O)N1CC2=C(C1)CN(C(C1CCC(N(C)C)C1)=O)C2 C1(NC(c2ccc(C)nc2)=O)CCCN(C(C23CC(C(F)(F)F)(CO2)C3)=O)CC1 N1(C(C)C)CCC(NC(C2CCC2(F)F)=O)C(C)C1 N1(C(CNC(=O)OC)=O)CCN(C(c2sc(OC)nc2C)=O)C(C2CC2)C1 c1(C2(C(=O)NC3C(NC(C=CCC)=O)C3)CC2)ccc(OC)c(F)c1 c1(CCOC)n[nH]c(=NC2CCCCN(C(c3nc(=O)n(C)[nH]3)=O)C2)s1 c1(OC)ccc(C(=O)NC2CC(NC(c3ncccc3C(F)F)=O)C2)nn1 c1(CCC(=O)NC2CCCC(C(=O)O)C2)cccc(C(=O)O)c1 O=S(=O)(c1ccc(C(F)F)c(Br)c1)Nc1ccncc1N1CCOCC1 Cn1ccnc1C(F)(F)C(=O)N1CC(CNC(=O)C=CCN2CCCC2)C1 N1(CC(N2C(C(C)C)C(NC(=O)C(O)CN(C)C)CC2)=O)OC(C)(C)CC1=O C#CC1CN(C(c2cc(CC3CC3)on2)=O)CCN1C(c1ccc(=N)[nH]n1)=O c1(CCC(=O)NC2(C)CN(C(c3cnn(CC(F)F)c3)=O)C2)cccc(F)c1 C1(NC(CCC=CC)=O)COC2(CCCN(C(c3ccccc3C3CC3)=O)C2)C1 c1(CNC(=O)CSc2cn(CC(O)C(F)(F)F)nn2)ccc(F)cc1F C1(C(N(CC(C)NC(=O)CNC(c2ccncc2)=O)CC)=O)CCC(C)(C)CO1 c1(CC)ccc(CC(N2CCC(C(=O)NOCc3scnc3C)C2)=O)cc1 C1(CC)CN(C(C2(n3cncn3)CC2)=O)CC1C(=O)NCC=Cc1ncco1 CCC(CC)(C(=O)NC1CC2C=CC1N(C(=O)CNC(=O)CC(C)C)C2)C(C)C Fc1cccc(Br)c1-c1noc(OCC2CCOC2)n1 C1(C(=O)NCCN(C(C=C(CCC)CCC)=O)CC(C)O)CCC(C(C)C)NC1=O c1(C(=O)OCCC#N)ccc(NCC2CC(=O)N(CCc3ccccc3)C2)cc1 C(=O)(CCCC1CCCO1)N.C1(C(C2(C)CC2)=O)(NC(=O)OC(=O)CCN)CC1C n1(CC=C)c(C(=O)NCCC(c2nnnn2C)NC(N)=O)cc2ccccc12 C1(C(N2CCC(CNC(c3cccc(C)n3)=O)CC2)=O)Cc2cc(F)ccc2O1 c1(CNC(C(C)OCC(C)C)=O)cc(C(N2CCC2CO)=O)n(C)n1 C1(NC(CCSC)=O)CCN(C(=O)C(c2nc(F)ccc2Cl)C)CC1O c1(NC(C(Cc2ncccn2)NC(=O)OC(C)(C)C)=O)cc2nc(Br)sc2[nH]1 C12CCCCN1C2=O.Cc1ccc(CNC(C2CC2c2ccoc2)=O)o1 Cc1cc(CN(C)C(c2conc2CNC(=O)CCCC2CC2C)=O)nn1C CCCCC(CC)C(=O)N1CCCC1c1nc(CC(C)(C)C)nn1C(C)C N1(C(Cc2c(C)n(C)nc2)=O)CCC(C2CC2)C1C(N1CC(C(C)(C)O)C1)=O c1(N2CCC(C)(CSC)C2)nc2cc[nH]c2c(=NCC2(S(C)=O)CC2)[nH]1 c1(C(N(Cc2cn(C3C(OC)COCC3)nn2)O)=O)ccc(C)cc1F C(=O)(C(C)(C)C(C)C)NCC12CC(NC(c3ccc(OCCOC)cc3)=O)(C1)C2 c1(C(N(C)CCOCCNC(=O)CC2CS(=O)(=O)C2)=O)cc([N+](=O)[O-])c[nH]1 CCC(C)(C)CC(=O)NC(C)(C(=O)N(C)Cc1ccccc1F)C1CCC1 CC1(c2ccc(Br)cc2)CCN(CC(=O)NCc2csc(-c3ccccc3)n2)CC1 C(=O)(C1=CCCC1P(C)(C)=O)NC(CN(C)C(C1C=CCC1)=O)(C)C c1(N2CCCC(C)(CC)CC2)[nH]c(=NCC2(C)CC(C)=NO2)nc2scnc12 N1(C(C(=O)NCCOC)=O)CCCC(C(=O)NC(c2ccccn2)(C)C)C1 C1(C(N(CC(CC)(C)OC)C)=O)CN(C(C2(F)CCCCCC2)=O)CC12CCC2 C1(N(C(CC(C)F)=O)C2CC2)CN(C(C2(n3cncn3)CC2)=O)CCC1F C(C1c2ccsc2CCN1C(C1CCC(=O)N1C)=O)NC(CCC(=C)C)=O C1(C(CNC(CCNC(c2coc(C(N3CCCC3)=O)c2)=O)=O)O)CCCC1O C1(C)(CC)CC(C(N2CCN(C(c3c(C)coc3C3CC3)=O)CC2C)=O)CCO1 c1(C(N2CCN(C(CSCC=C)=O)CC2C(C)C)=O)cc(N)cc2c1OCCO2 C1(C(=O)NCC(=C)CCNC(=O)CC(C)OC)CCc2ccccc2C1 c1(C(c2n(CCCC)nnn2)NC(C)Cc2cccs2)ccc(N(C)C)cc1 C1(F)(CNC(C=C(C)C2CC2)=O)CCN(C(C2CC3CCC2O3)=O)CC1 c1(C(=O)NCCNC(c2ccc(C#C)cn2)=O)cc(C)nc(Cl)c1N C1(C(=O)NC(c2c(C)noc2C)C)CCN(C(c2cncn(C)c2=O)=O)CCO1 c1(CC)c(C(=O)N(C2CCN(C(=O)C(C)C#N)CC2)CC(C)C)csc1C C1(CNC(C(C)C2CCCO2)=O)CC2COCC2N1C(=O)C(C)(C)CC(C)C C=C1CCN(C(=O)CCCCOCC)C(C(=O)NC2COC(C(F)F)C2)C1 c1(C(=O)NCCC2(CNC(C(C)OCC)=O)CC2)ccc2c(c1)OC(C)(C)OC2 N1(C(C=Cc2n(C)ncc2)=O)CCN(C(c2cc3n(n2)CCC3)=O)C2CC12 c1(CCOC)ccccc1-c1nc(CCOC)nn1-c1ccccc1C c1(NC(=O)NC(C2CC2C2CC2)C)ccc(C#N)c(Cl)c1 N1(C(C(c2ccc(C(C)(C)C)s2)C)=O)CC(CNC(=O)CCCC2CC2)C(C)(C)C1 N1(C(C(CCC)C)=O)CCCC(C)(CNC(=O)CCc2cccn2C)C1 C1(C(=O)NC2CC(O)C2)(CC)CCN(C(=O)CCCC2CCCO2)CC1 Cc1cc(C(N2CCC3CN(C(C4CC4C(F)F)=O)C3C2)=O)cc(F)c1C n1(CC(=O)N(CCN(C(C)C)C(C2CC2C(F)(F)F)=O)C)nnc2ccccc12 C1(C(N(CC(=O)NCC2C3COCC23)C(C)C)=O)C2(CC2)C12CC2 C(CCC(=O)C(=O)COCC1(C(=O)NCCNCC2CCCC2)CC1)N(C(C)=O)C N#CC1=C(C(=O)NCCC2CCN(C(c3ccncc3F)=O)C2)CCC1 C1(NC(CC)=O)CC12CCC(NC(c1cc(-c3cccc(Br)c3)no1)=O)CC2 N1(C(=O)C2=CCSC2)CC2(C1)CN(C(=O)CCOCC1CCCO1)C2 N1(C(c2c(C)ccc(OC)c2)=O)CC(NC(=O)C(C)CC(C)(C)O)CC12CCC2 c1(C(=O)NC(CN(C(=O)CCc2cnc[nH]2)CC)C)cc(C)c(N)c(C)c1 C(=O)(CN1C(=O)CCCc2ccccc21)N(CC(CNC(CC=CC)=O)C)C c1(CC(=O)NCC2(COC)CN(C(=O)C(CO)N(C)C)C2)cncnc1O C1(CC)CN(C(=O)C(C2CC2)C2CC2)CC1C(N1CCC(CF)C1)=O C12(C(N3CCN(C(c4cncc(C)n4)=O)CC3)=O)CCC(CC1)C2(C)C c1(C(=O)NC(C2CCCC2NC(c2cnnn2C)=O)C)n[nH]cc1C(F)(F)F C1(CC(=O)NC(c2ccccc2)CC)CCC(NC(=O)Cn2ccc(C)c2)CC1 CC(C)C(O)(C(=O)N1CC(C)(NC(=O)C(C)NS(C)(=O)=O)C1)C(F)(F)F c1(CNC(=O)Nc2c(Br)nc(C)n2C)cn2cc(Cl)cc(C)c2n1 C1(COC)(NC(c2ccc(-c3ccco3)s2)=O)CCN(C(c2csc(S)n2)=O)C1 c1(CCC)cc(C(=O)NCCN(C(=O)C=Cc2ccco2)C(C)C)ccn1 C(c1ccc(=N)[nH]c1)=CC(=O)NCCCCC(C)NC(C1CN(CC)C(=O)N1)=O C1(C(=O)NCCOCC(=O)NCC(C(=O)OCC)(C)O)CCCCC1(C)C c1(C(=O)NCC2(C)CC(NC(=O)CN3CCSCC3)C2)cnc2[nH]nnc2c1 C1(C(=O)NC(CC)CO)(SC)CN(C(=O)C(C)CN2CCCC2)C1 N1(C(c2cccc(SCCC)c2)=O)CCC(NC(=O)C(O)C(C)(C)C)CC1C C1(NC(=O)NC2CCN(C(C3(OC)CCOC3)=O)C2)CC(C2CCCC2)C1 S(=O)(=O)(c1cccs1)N1C(Cc2ncn(CCNC(=O)OC(C)(C)C)n2)CCC1 CC1(C)CC(CNC(c2cc3occc3[nH]2)=O)N(C(=O)CCc2cncnc2)C1 n1(CC(=O)Nc2ccc(C)c(CN)c2)ccc(=O)c(O)c1C C1(C2C(NC(CCC3C(C)C3)=O)CCO2)CCN(C(=O)CCn2cccn2)CC1 C1(OC)CCC2(C(N3CCCCC3C3CCCN(C(C4CCCS4)=O)C3)=O)CCC12 C(=O)(CCCCC(F)F)N1C(CN(C(COCCC=C)=O)C)CCC1 CC1CCN(C(c2nocc2Cl)=O)C1CNC(c1csc(C2CC2)c1)=O N1(C(COC(CC)(C)C)=O)CCC(C(=O)NC(COC)CO)(OC)C1 CCCCCCC(C)(CCC)C(=O)N1CCN(Cc2nc(O)n[nH]2)CC1C C1(N(C(COCCSC)=O)C)CCC2CN(C(=O)C(=O)CC(C)C)CC12 O=C(C1CCCc2cncn21)NCCCN(CCCN)S(C)(=O)=O C1(NC(C(CC)n2cccn2)=O)CN(C(=O)CCN(C)CCO)CCC1C c1(NC2CC(F)(CNC(c3c(CC)cno3)=O)C2)ncc2c(n1)CCCC2 c1(C(=O)NC2(CO)CCN(C(C3(CC)CC3(F)F)=O)C2)cnc2c(c1)CCOC2 C1(CNC(=O)Cn2cc(CO)nn2)CCC2CN(C(=O)C3=COCCC3)CCC2C1 C1(C#N)(C(=O)NC(C(C)NC(c2cc(CCC)on2)=O)CO)CC=CC1 CP1(=O)CCN(CC(N2CC(O)CC2C2(NC(=O)Cn3nnc(=O)[nH]3)CC2)=O)CC1 C(c1cncnc1O)=CC(=O)OC.N1CC2CC1C2CN(CCCCC)C Nc1sc2c(c1C(=O)NCC1CCCCC1NC(c1csnn1)=O)CCSC2 Cc1cc(Cl)cc(N)c1C(=O)NCC1(CNC(=O)C(C)CC(C)(C)C)CC1 CC(C)(CCCNC(=O)NCC(=O)OCc1ccco1)NC(C1CCC(=O)N1)=O C(C1=NOC2OCCCC12)N1CCC(=O)C(c2ccc([N+](=O)[O-])cc2)C1 C=Cn1nccc1C(N1CCC(CO)(CNC(C2CCN2CC)=O)C1)=O C1(CNC(CCOC)=O)CCCCC1NC(=O)CC1(O)CCOC1 c1(NC(C(CC=C)NC(=O)C=C(C)C(C)C)=O)cnccc1C#N Cc1coc(C2CC2)c1C(N1CC(NC(C2CC2F)=O)C(c2nccn2C)C1)=O Cc1cc(N)c(C(N2CCC=C(CNC(=O)C3=C(Cl)CCC3)C2)=O)c(F)c1 C1(C(=O)NCC(C)O)CN(Cc2ccc(OC(F)(F)F)nc2)CC(F)(F)C1 N1(C(CC2CCC(OC)CC2)=O)CCN(C(C2CC2(F)F)=O)CC1C c1(C(N2C(C)CC(NC(c3n[nH]c(C)c3C(F)(F)F)=O)C2)=O)ccc(O)c(F)c1 CN1CC(O)CC1C(=O)NCc1ccc(C(=O)NCC2CC2CO)nc1 CCCCCC(=O)NC1COCCC1NC(c1n[nH]cc1-c1ccncc1)=O N1(C(=O)C=Cc2ccccc2Br)CCC2CN(c3ncc4[nH]ncc4n3)CCC12 C1(CCCC)CN(C(c2n[nH]cc2OC)=O)CCN1C(C1C2COCC12)=O C1(NC(C(C=CC)O)=O)CCOC12CCN(C(=O)C(C)=CC1CC1)CC2 C1(C(=O)NCCCNC(c2cc(CS(C)(=O)=O)on2)=O)CCCC1(F)F CCC(CC)CCC(=O)N1CC(CC(=O)N(C)CC2CCOC2C)C(C)C1 c1(CC)c(C(=O)N(CC(C)NC(c2cnc(NC(C)=O)o2)=O)C)[nH]c2ccccc12 N1(C(C2C(CC)CCCC2)=O)CCC2(C1)CN(C(C1(C)CCCO1)=O)C2 N1(C(C(C(C)C)(F)CNC(C2(C(C)C)CC2)=O)=O)CC(C2CCCCC2)C1 CC(C)CC(C)(O)CNC(=O)CN(C1CCC1)C(C1CC1[N+](=O)[O-])=O c1(C(=O)OC)cc(=NC(=O)C2(NS(C)(=O)=O)CC(C[Si](C)(C)C)C2)[nH][nH]1 c1(OC)cncc(CC(=O)NCC(C(C)(C)C)NC(C2CN(C)C(=O)N2)=O)c1 C(=O)(CC(C)C(C)(C)NC(c1cnn(CCF)c1)=O)NC(C)C(C)(C)C CC(C)(C)CC(O)C(=O)NC1CN(C(=O)CCc2ccccc2F)CC1O C1(N(C(CN(C(c2cc(C)nn2C)=O)C2CC2)=O)C)CCCC(C)(C)C1 CC(C)C(CCNC(C1CCCN1c1nccs1)=O)NC(=O)C(C)c1cccs1 N1(C(Cc2c(C)ocn2)=O)CCN(C(=O)C(F)=CCCN2CCOCC2)CC1C Cc1cccc([N+](=O)[O-])c1C(=O)NC(C)CNC(C1CC2CCCCCCC12)=O C1(CNC(C2(C#C)CC2)=O)CN(C(C2CC2(C)CC)=O)CC12CC2 CP(C)(=O)C(O)C(=O)N1C(CNC(C2(N(C)C)CCCC2)=O)CC2CC12 N1(C(C=C(COC)C)=O)CCC(C(C)CNC(c2cc(O)ncn2)=O)CC1 C(CC(C(=O)NC(C1CC2(CCC2)C1)C)NC(=O)C(c1ccn(C)c1)C)=CC C1(C(=O)NC(c2c(CN)occ2)=O)(NC(N)=O)CCOC1.C1(CCF)(C)CC1 C1(C)(C(N2C(CO)CC(NC(CCC(=O)NCCC)=O)C2)=O)CCC(C)=C(C)C1 C1(NC(c2n(CC)nnn2)CCc2ccc(F)cc2)CC2C=CCC(C1)C2 C1(OC)CN(C(c2cn(C)c(=O)n2C)=O)C(C)(CNC(=O)CCC2CC(C)C2)C1 c1(OCC)ncccc1-c1noc(C2CCOC2c2ccccc2C)n1 Cc1ccc(Cl)c(O)c1C(=O)NCCN(C(C12CCCCC1C2(F)F)=O)C(C)C c1(C(=O)NC2CCC(C(=O)NC3CC(=C4CC4)C3)C2)cncc2nc[nH]c12 N1(C(C2CN(C(C)=O)C2)=O)CC(C2CCN(C(=O)CC3COC(C)(C)C3)CC2)C1 C=CC(C)(CC)C(=O)N1CCC(NC(=O)CC2OCCO2)C(OC)C1 Cc1cccc2[nH]cc(C(=O)NC(CNC(=O)CC(C)O)C3CC3)c12 N1(C(CS(=O)(=O)N(C)C)=O)CCCC12CCN(C(c1ccc(C#N)c(Cl)c1)=O)C2 CC(C(=O)NC(c1ncc[nH]1)CO)NC(=O)C=CCF c1(C(=O)NC2CC(NC(c3cnn(CC)n3)=O)C2)noc2c1CCCCC2 C1(N(C)C)CCN(C(=O)CN(C(=O)CCNC(C2CCCO2)=O)C2CC2)C1 NS(=O)(=O)c1ccc(CC(=O)NCCC2(CNC(C3CCCO3)=O)CC2)s1 C(=O)(C(CC)CCNC(=O)C(C)(C)C)N1CC(NC(C(CCC)O)=O)C1 N1(C(C#CC)=O)CC2CN(S(=O)(=O)C3CC3)CC12 N1(C(C(=O)NCCNC(C)=O)=O)CC(NC(=O)CC2CCCC(=O)CC2)CC(C)C1 C1(C(=O)NCCCCCNC(CS(=O)(=O)NC)=O)C2CC3C(C2=O)C13 C(=O)(C(F)(F)CC=C)NCC1C(C(=O)NCC(=O)OC)C1(C)C CON(CCC(=O)NCc1ccncc1Cl)C(=O)CC1CCC(CO)O1 C1(N2C(=O)CC3(CCC3)C2)(CC)CC(C)CC(C)C1.CCON Cc1c[nH]cc(C(=O)NCc2ccc(CNC(=O)CCOCC3CC3)cc2)c1=O N1(C(C(=O)NCC2CC2)=O)CCC2CCN(C(C34CCCC(CO3)C4)=O)CC2C1 c1(C(=O)NC2CCCC(CN(C(CC3(OC)CC3)=O)C)C2)ccc2c[nH]nc2n1 C1(CNC(c2c(C(C)C)nns2)=O)CN(C(C2COC2)=O)CC1C(F)(F)F N1(C(c2c(CC)cno2)=O)CCN(C(=O)CCc2cccc(OC)n2)C(C)C1C C(=O)(C(C)C(C)(C)C)N(C1CCN(C(c2cn(CC3CC3)nn2)=O)C1)CC C(CNC(c1c[nH]nc1Cl)=O)(CCNC(C1CC1(C)C(C)C)=O)OC c1(OC(=O)NCCCOCc2c(C(=O)OC)c(C)[nH]n2)cc(C)cc(C)c1 S(=O)(=O)(c1c(F)cccc1F)NCC(=O)NC1CC(NC(c2ccc(N)cn2)=O)C1 c1(C2C(CC)N(C(=O)C(O)C(C)C)CC2)cc(C)c([N+](=O)[O-])cc1Br C1(CNC(c2c(C)scc2)=O)CCC(C)N(C(c2ccnc(Cl)c2F)=O)C1 C1(NC(CCOC)=O)CN(C(c2cnsn2)=O)CC1F C(C)(C(C(C)C)NC(c1ccoc1C)=O)NC(CCOC)=O c1(C(N(C(CC)CNC(C2CNC(=O)C2)=O)C)=O)cnc(COC)n1C c1(C(N2C(CN(C(c3n(CC)c(O)nc3)=O)C)CCC2)=O)cn2c(n1)CCC2 c1(C(=O)NC2C(NC(C(C)(F)F)=O)C2)ccc(-c2cccnc2)nc1O Cc1nc2cc(C(N3CCC4(C3)CN(Cc3cc(I)cc(I)c3)C4)=O)ccc2s1 N1(C(CC2(COC)CC2)=O)Cc2[nH]nc(C(N3CC4(CCOC4)C3)=O)c2C1 c1(CC)cc(C(N2CC3CC2C3NC(C2CC2[N+](=O)[O-])=O)=O)ccc1Cl c1(C(=O)NCCN(C(=O)CN(C)C2CC2)CCOC)cc(C)nc2[nH]nc(C)c12 C(=O)(C(C)(F)C(C)(C)F)NCC(C)CNC(=O)CCS(=O)(=O)N(C)C C(=O)(CC(C)(F)F)N1CCC(C(N2CCC(N(C)C)C2)=O)C1 CC(CC(N)=O)C(=O)NCC1CN(C(=O)C=CC(C)(C)C)C2CC12 C1(CCC)CCCC1C(=O)NC(C1CCCC1)CNC(=O)C=CSC C1(CNC(c2c(C(F)(F)F)nc(C)o2)=O)CC2CCC(C1)N2C(=O)Cc1ccoc1 C1(C(N2CCN(C3CCN(C(c4cccc(Cl)c4)=O)C3)CC2)=O)CC(=O)N(O)C1 c1(C(N2C(C(=O)NCC(F)(F)C(F)F)CC(O)C2)=O)ccc2c(c1)OCCO2 c1(OC)cccc(C(N)=O)c1F.c12ccc(c(Cl)c1)CN1C(CC3CC13)C(=O)N2 N1(C(CSCC#C)=O)CC2(CCN(C(=O)C(C)Cc3ccccc3Cl)C2)C1 n1(CC(=O)NCC(CNC(CC2CC(CC)C2)=O)C)nnnc1C n1(CCC)nccc1C(C)NC(=O)CCN(C(=O)CCCOCC)C CC(C)(CS(C)(=O)=O)C(=O)NCC1(F)CCCN(C(c2ccc(Cl)cc2)=O)C1 c1(C(N2CCC(N(C(c3cc(C(C)C)no3)=O)CC3CC3)C2)=O)cncc(F)c1 c1(C2(NC(C3CCCCC3)=O)C(C)C2)cccc(C2(C)CC2)c1 Cc1nc(C(N2CCCC2C(C)(C)CNC(=O)CC2(C#N)CC2)=O)c(Br)s1 CC1CC(C(=O)NCCOC2CCN(C(=O)CC(C)C3CCCC3)C2)=NO1 c1(C(=O)NC2(CNC(c3c(C)noc3C)=O)CC2)ccnc(OCC2CC2)c1F N1(C(C2CC(SC)C2)=O)C2CCC1CC(CC(C)NC(c1cncc(C)c1)=O)C2 C1(CN(C(c2nc(CC)oc2)=O)C)C2CN(C(=O)Cc3csc(COC)n3)CC12 c1(C(=O)OC)c(C(=O)NC(=O)C(C2CCCN(C(C)(C)C)C2)(C)C)cnn1C Cc1ccc2c(c1)C(N(C(N1CC=CCC1)=O)C1CC1)CCCO2 N1(C(C(C(C)C)NC(c2cccs2)=O)=O)CC(C2CN(C(=O)C(N)=O)C2)C1 c1(N2CCC(NC(CCc3ccnc(C)n3)=O)CC2)ncnn2cccc12 C1(OC)CC(CNC(=O)C(C)NC(N)=O)N(C(c2ccc(-n3ccnc3)cc2)=O)C1 C1(CNC(c2cn(C3CCC3)nn2)=O)CCCCN1C(=O)C1=NOCC1 CCCCC(=O)N1CSCC1C(=O)NC1CC1c1cnn(CCOC)c1 C1(COC)CN(C(=O)C=CCF)CCN1C(=O)Cc1c(O)ncnc1O NC(=O)CCCC(=O)NCC(N1CCN(C(C2CC2CF)=O)CC1)C(F)F C1(NC(CC(C)(C)OC)=O)CC(NC(=O)CCC(CF)CF)C12CCOCC2 C1(NC(CC=C)=O)CC2C(NC(c3sc(F)cc3C)=O)C2C1 N1(C(c2c(C)occ2)=O)CCN(C(c2cc(F)c(F)cc2N)=O)C2CCCCC12 CC(CC(=O)NCCOCCOCCNC(c1cccc(O)n1)=O)P(C)(C)=O N1(C(C(C)OCOC)=O)CCC(C)(C(=O)N(C)C(c2nccs2)C)CC1 C=CC1CC(NC(=O)CCCNC(=O)C(C)NC(=O)NC)C1 c1(C(N2CCC(N(C(C3CC4CC3C4)=O)CC)C2)=O)cccc2ccoc12 C1(C(=O)NC2CC(C(=O)NCC(F)(F)Br)C2)CC1C1CC1 N1(C(C=C(C)Cl)=O)CCC2CCC(NC(c3cc(Cl)nc(Cl)c3)=O)C1C2 C(C)(C)(CCCN=c1cc(C(=O)OC)cn[nH]1)OC C1(N(C(=O)NC(c2cc(F)c(F)c(F)c2)C)C)COc2ccccc2C1 N1(C(CCN2CCN(C)CC2)=O)CCC2(C1)CN(C(C1(C)CCC(=O)NC1)=O)C2 c1(C(N2CC3C(CCNC(CCCC#C)=O)(CC3)C2)=O)coc(S(N)(=O)=O)c1 C(=O)(CCCC(C)(C)NC(=O)Cc1cn(C)cn1)N(C)Cc1ncn(C)n1 C(=O)(C1=C(CC)OCCC1)NC(CC#C)C(=O)NCCOC1CCCCC1 Cc1cn2c(n1)CCC(C(=O)NCCOCCNC(c1cnn3c1NCC3)=O)C2 Cc1ccncc1C=CC(=O)NCC1(C)CCCN1C(c1cccc(Cl)n1)=O c1(C(=O)NCC2CCN(C(C(CCC)C)=O)CC2)ccc2nc(N(C)C)oc2c1 N1(C(C(CCC)C#N)=O)CCCC(C)(CNC(C2C3CC4C(C3)C24)=O)C1 N1(C(C=Cc2n(CC)ncc2)=O)CCC(NC(=O)C2=CCCSC2)C(O)C1 C(=O)(CC(CC)C(C)C)NC(CCNC(c1cc(CC)cc(C(F)(F)F)c1)=O)C CC1(C)OC2C3CC(CNC(=NCCCF)NC4CC45CCCC5)C(C3)C2O1 c1(C2(C(N3CC4CC4(CNCc4ccc(Cl)nn4)C3)=O)CC2)cc(Cl)ccc1Cl c1(NC(C(C)C)CNC(c2nccs2)=O)ncc(C#N)cc1Cl C12(F)CCC(C1)NC(=O)C(=O)NC2.C1(C(=O)Nc2ccoc2)CCOCC1 c1(OC)ccccc1C(C)=CC(N1CCC(NC(=O)Cc2cnoc2)C(O)C1)=O C12(C(N(C(CNC(C3(C)CCCOC3)=O)C3CC3)C)=O)CC(C)(C1)OC2C C1(CNC(=O)C=Cc2ccsc2)CCN(C(=O)CCC(=O)N2CCOCC2)CC1 CC(C)S(=O)(=O)C(C)C(=O)NC1CC(C)(NC(=O)CC2(C#N)CCCCC2)C1 N1(C(C2N(C)CCOC2)=O)CCC(NC(=O)CC#N)C(c2ccccc2)C1 C(CC(C(=O)NC1(CN(C)C)CCC1)NC(=O)CC(C)COC)=CC CC(C)C(O)CC(=O)NC1COCC1CC1(C(=O)N)CCCC1.C(=O)(C1CC1)NC c1(C(=O)NC(C2CC2C(=O)NC(C)Cc2nn[nH]n2)C)nccc2[nH]ccc12 C1(N(C)C(C2(F)CCCC2)=O)CN(C(=O)C(c2ccc(Cl)cc2Cl)O)CC12CC2 C1(NC(Cc2cc(OC)c(C)cc2)=O)CN(C(C2CCCC2)=O)C2(CCCC2)C1 CCCCCCCCCC(C(=O)OC)N1CCc2ccccc21 C12(NC(=O)COCc3ccc(OC)cc3)CCN(C(=O)Cc3cccs3)CC1C2 C1(CNC(CCN(C(C2(CC)CCOC2)=O)CCO)=O)CC12CCOCC2 CC1(C)CC(O)(CC(=O)NC2CC(CNC(=O)C3=C(Cl)CCC3)C(O)C2)CO1 C12(CNC(C3CN(C)C3)=O)CCC(CN(C(=O)COc3c(Cl)cccc3Cl)C1)C2 C1(CC(c2nnnn2-c2ccccc2)NCC(CCC)OC)(OC)CCCCC1 c1(N(CCC(C)O)C)nc(=NCC2C(F)(F)C23CCC3)[nH]c2c1CCCCC2 c1(OC)sccc1C(=O)NCC(O)CNC(=O)CSCc1cscn1 c1(NC(=O)C=Cc2ccc(C(F)F)o2)cc(S(=O)(=O)N2CCOCC2)ccc1O CCC(C)C(C(=O)N1CCC1CC1CCCC1)N(C)C(c1nnc(S)n1C)=O C1(CCNC(C2CC(C)N(C)C2)=O)CCCN(C(=O)Cc2ccnc(CO)c2)CC1 N1(C(C2N(C(c3ccc(C)o3)=O)CC(O)CC2)=O)CC(C)(C)C12CCC2 CC1=C(c2ccc3c(c2)SC=C(CC)C=C3)CCCC1.N1(CCOC)CCC1 C(=O)(CC(CNC(=O)NC(c1ccc(Br)s1)C)C(C)C)OC CC(C)(CS(C)(=O)=O)C(=O)NC1CC1CNC(=O)C(F)(F)C(C)(C)O CC1(C)CN(C(c2cc[nH]c(=N)c2N)=O)CC(CNC(C2(C(F)F)CC2)=O)O1 C(CNC(=O)C1=CCCOC1)(C(C)C(C)C)NC(c1ccc(SC(C)C)cc1)=O C1(C(N(C(CCNC(Cc2cc(C)on2)=O)C)C)=O)CCCCN(C)C1=O CCCCC(C(=O)N1CC(c2ccccc2)(NC(=O)Cc2ccsn2)C1)N(C)C CCC(C)(C(=O)NCC(C(C)C)NC(c1sccc1SC)=O)OC N1(C(c2c(C)nn(C(C)(C)C)c2)=O)CCN(C(C2(N(C)C)CCCC2)=O)CC1CO N1(C(c2ccc(C#C)cc2)=O)CC(NC(=O)C(c2ccccc2)C)CC2(CC2)C1 N1(C(c2n(CC(=O)OCC)ncc2)=O)CC(O)C(O)C1CO.C12CC(C1)SC2=O CC1(C)CN(C(c2cnc(N)c(N)c2)=O)CC1CNC(=O)CCC1CCCO1 C(=O)(C(CC#CC)NC(=O)CCCC(=O)OCC)NCC(C=C)(C)C O(NC(=O)CCC1CCCN(C(=O)CNC=O)C1)CC#C c1(C(N2CC(O)(CCNC(c3ccc(OC)s3)=O)C2)=O)ccc(C)c(F)c1F CC1CN(c2cc(C(=O)NCC3CCN(C(S(C)(=O)=O)=O)C3)ccn2)CC(C)O1 c1(SC(C)CNC(N2CC=CC2(C)C)=O)ccnc(C(F)(F)F)c1 C(=O)(C(C)(COC)COC)N1CC(CNC(C(C=C)(F)F)=O)C(C)C1 S(=O)(=O)(c1ccc(C)c(C)c1)NCCc1nccc(=NCC2(OC)CCOC2)[nH]1 CC1CN(C(c2cccc(N(C)C)c2)=O)CC1NC(C1CC(=O)CO1)=O c1(C(=O)NC(C2(O)CN(C(C3(C4CC4)CC3)=O)C2)C)cnn(CC(F)(F)F)c1 C1(C)(CC)C=C(C(=O)NC(C(=O)NCCOCCC(C)C)c2ccoc2)C1 C1(CC(=O)NC2CC3(C2)CN(C(C2CCC24CCCO4)=O)C3)CN2CCN1CC2 c1(C(N2CCCC(CN(S(C)(=O)=O)C)C2)=O)cccc2c1NC(=O)C2=O N1(C(C(CC(F)F)NC(C(CC)OC)=O)=O)CCCCC(C)(F)C1 C(=O)(CC(C(C)(C)C)NC(=O)C(C)N1CCCC1)NC(C#C)CC1CCCC1 c1(C(N(CCNC(C2CC(C)(C)O2)=O)CCOCCO)=O)ccnnc1O Cc1cc(=O)n(CCC(=O)N2CC(=C(F)CNC(=O)C(CC)CC)C2)cn1 c1(CC)ncnc(Nc2ccc(OCC(C)C)cc2Cl)c1F c1(OCC(=O)NC(CC)(C)CNC(=O)C(C#N)C2CC2)cc(Br)ccc1Cl c1(NC(CNC(c2n(CC)nnn2)(C)CSC)(C)C)ccc2c(c1)OCO2 N1(C(CCn2ccc(C)n2)=O)CC2CC(C(=O)NC3(C)CS(=O)(=O)C3)C(C2)C1 C=CCCCC(C)(C)C(=O)NCC(C)CNC(=O)Cc1cnn(C)c1 C(=O)(C(C)CCCOC)NC1(C(C)(F)F)CCC1.C=C1CC2(C1)C(=O)NC2 C1(NC(C=CC(N)=O)=O)CCN(C(c2ccc(=O)n(O)c2)=O)C12CCCC2 C1(C)(C(=O)NCCN(C(=O)CSCC(F)F)C)CCCC1 CC1(C)CCCC(CC(N2CC3CC2CN3C(c2ccc(F)c(C#N)c2)=O)=O)O1 C1(NC(COCC(=C)C)=O)CCOC(C(=O)NCCN2CCOC2=O)C1 c1(C(=O)NCCCC(CCC)NC(C2CC=C(C)CC2)=O)cccc2sccc12 c12ccc(o1)S(=O)(=O)N2.O=C1CC(CC2CN(c3ccncn3)C2)CN1 c1(CC#N)cccc(C(=O)NC(CNC(C2CC23CCCC3)=O)CO)c1 N1(C(c2scc(C)c2)=O)CCOC2(C1)CN(c1ncc(F)cn1)C2 Cc1cc(C(N2CCCC(N(C)C(c3ccsc3Cl)=O)CC2)=O)cc(C)c1O CCC(CN(C(=O)CNC(=O)OCC)C)N(C(=O)C(O)C1CCCC1)C CC1CC(N=c2cc(C#N)nc(CNC(=O)CC3CCC=CCC3)[nH]2)CCO1 CC1CC2(CCN(C(=O)C(C(N)=O)C(C)(C)C)CC2)CN1C N1(C(c2nccc3cc(OC)ncc32)=O)CCC2(CC=CCO2)C1 c1(C(N2CCCC(CNC(C(C)C(C)(C)C)=O)CC2)=O)cccc2[nH]ncc12 N1(C(C(CC=C)C)=O)CC2CCCCC2(NC(=O)CCC2CC(F)(F)C2)C1 N1(C(c2cnn(C(C)C)c2N)=O)CCC(NC(c2cc3sccc3[nH]2)=O)C(C)C1 N1(C(C2(COC)CCCC2)=O)CC2CCC1CN2C(=O)C(C1CCCCN1)=O C(CCCC=C)(C(=O)NCCCc1ncnn1C)NC(c1ccc(C#C)cc1)=O C1(C)(C(=O)NCC(CC=C)NC(=O)CN2CC3CC3C2)CCC(O)CC1 C1(OC)CCCC1C(=O)NC1(C)CC(NC(=O)C=C(Cl)Cl)C1 C12(NC(C(CC)OC)=O)CCC(C1)N(C(=O)C=CC1CCCCC1)C2 CC1(C)CCC(=CC(N2CC(CNC(=O)CCC(F)F)C3(CC3)C2)=O)CC1 c1(OC)cc(C(=O)NC2CC3(NC(=O)CCCc4cccs4)COC2C3)cnc1O N1(CC)CCC(OCC(CC(N)=O)c2cn(C3CCOCC3)nn2)CC1C Cc1nn(C)cc1CC(=O)NC1(C(=O)NCC(O)Cn2cccn2)CCN(C)C1 N1(C(N2CC(OCCOC)C2)=O)CCCC(C)(CNC(=O)OC)C1 N1(C(C=CCN(CC)CC)=O)CCCN(C(c2c(Cl)n[nH]c2C2CC2)=O)CC1 C1(NC(C(C)OCCOC)=O)CCC2CC1CN2C(C1(C)CC(C)=NO1)=O N1(C(C(c2c(C)cccc2)C)=O)CCC(C)(C)C(Nc2ncc(F)cn2)C1 C1(CNC(c2c(Cl)cccc2Cl)c2n(CC(=C)C)nnn2)CC2CC1C1CC21 C1(CC(=O)NCC(CC)NC(C2CN(CC(F)(F)F)C2)=O)(CN(C)C)CCCC1 c1(C(=O)NCC(CNC(C2(CCC)CCC2)=O)C)nc[nH]c2ncnc1-2 C(c1cc(Cl)cc(Cl)c1)=CC(N1C2C(NC(C3(C)ON=C(C)C3)=O)CC(C2)C1)=O C12(NC(Cc3c(C)ccc(F)c3)=O)CCCN(C(C3CC(=O)CO3)=O)CC1C2 c1(C(=O)NCCCN2CCCC2)c(NCc2cc(O)cc(Br)c2)cccc1F C(=O)(CCC(CC)CC)NC(CC#C)C(=O)NCc1cnn(CC)c1C N1(C(c2ncn(C)c(=O)c2)=O)CCC2(CC(NC(=O)C(N)=O)CO2)C1 n1(CCSC)nnnc1C(c1ncsc1C)NCc1ncnn1C(C)C C(C)(c1ccc(OC(C)C)cc1)=CC(=O)NC1CCC(N(C(COC)=O)C)C1 C(CC(=O)NCCC1(O)CCCCC1)(C(F)F)NC(C1N(C)CCOC1)=O CCCC(C(=O)Nc1cc(F)c(C(=O)OC)cc1NC(C)=O)S(N)(=O)=O Cc1cnc(NCc2ncoc2C(C)(C)C)c(S(=O)(=O)N2CCCN(C)CC2)c1 c1(NC(C(COCC)OC)=O)nnc(C#N)s1 n12cc(nn1)COC(=O)CNC(=O)C2.c1(C(N(CC(C)C)C2CC2)=O)ccc(Cl)s1 C=CCC(CC=C)C(=O)NCC1CN(C(=O)C(C)SCc2ccccc2)CCO1 N1(C(c2c(Br)cn(CC)n2)=O)CCCC12CN(C(=O)CCc1ccc[nH]1)C2 c1(C(N2CCC(NC(C#CC(C)C)=O)C23CC3)=O)cc(Cl)c(N)cc1F c1(C(C)=O)ccc(NC2(CNC(=O)C)CCC2)nc1.C(=O)(C(C)c1ccsc1)N N1(C(c2ncc(OCC)cn2)C(=O)NCC=C)CC=C(C(C)(C)C=C)C1 Cc1ccc(C(=O)NCC2COCCN(C(C3(O)CCCCCC3)=O)C2)nc1C C1(NC(c2n(C)ccc2)=O)CC12CC(NC(=O)CSc1nnc(-c3ccco3)o1)C2 C(=O)(CC1=CCCCC1)NCCCCC1CCN(C(c2ncc(C)nc2)=O)CC1 c1(CNC(=O)NCc2cc(C)cc(O)n2)cnc2n1CCCC2 CC(CC(=O)NC1CC(C(=O)Nc2ccsc2C(N)=O)C1)C(C)(C)C CC1CCC(CNC(c2ccc(F)o2)=O)CN1C(=O)CCc1cnco1 N1(C(C2CC(C(=O)OC)C2)=O)CC=CC1(C)C.C12OCCC1C(=O)N2 C1(CC)CN(C(C2CC(C)N(C(c3ccnn3C(F)F)=O)C2)=O)CCN1C C(C(CNC(=O)C(C)n1cccn1)CO)CC(=O)OC.CC(C)C(=O)N C1(C(C)C)CCCC1NC(=O)COCCCNC(=O)CSCC(F)F N1(CC2CN(C(CC3CCC(=O)C3)=O)C2)CCN(C(=O)Cc2c[nH]nc2O)CC1 C#CCC(CC(F)F)NC(C1CC(C)CCN1C(c1cc(Cl)no1)=O)=O CC(C)CC(CNC(=O)C(C)OCCN(C)C)C(=O)NC1CCC12CCCC2 N1(C(CCc2scc(C)n2)=O)CC2CC(NC(c3cc[nH]c3)=O)C(C2)C1 c1(NC(C(=O)N(C(C)CNC(c2cc(C3CC3)[nH]n2)=O)CC)C)ccccc1 C1(NC(C2CCc3c[nH]nc3C2)=O)CN(C(C2CSCCS2)=O)CCC12CCC2 C1(C(=O)NCc2n(CC)ncc2)COCCC1NC(=O)CC1(NC)CCCC1 C1(c2cn(CCCOCC)nn2)CCCCN1C(=O)C(=O)NCC1CCC(=O)NC1 C1(CCC)CN(C(=O)CC2COCCO2)CC1C(=O)NC(CC1CC1)C(=O)OC C(CC(N)=O)(C(=O)OC)OC(CCCOC)=O C1(O)(CNC(C(C)C)=O)CCN(C(=O)C(C(C)(C)C)N(C)C2CC2)CC1 Cc1nccnc1C(=O)N(CCCNC(=O)C(C)(C)C1CCC1)C(C)C C1(C(=O)NC(C)Cc2cn[nH]c2)CN(C(=O)C(C)(C)CCCF)CCC1(C)C CC(=O)CCCC(C)C(=O)NCCC(C)(C)C(=O)NCCC1CCC1 C1(CN(C(C(C)OCCOCCCOC)=O)C)CCN(C(c2ccco2)=O)C1 N1(C(COC2(C)CCC2)=O)CC2CCC(C1)N2C(C1CC1C1CCCC1)=O c1(C(=O)NCC2C(C)CCN(C(=O)COCC(F)F)C2)[nH]nc2c1COC2(C)C C=C(Cl)CC(C(=O)Nc1cncc(C)c1)NC(=O)C(C)CC c1(C(=O)NCCCC(C)NC(c2cccc(CN=[N+]=[N-])c2)=O)cnc(O)cc1O c1(C(=O)NCC(C)N(C(=O)CCC(C)(C)C)C)nc(Br)n2c1COCC2 Cc1c(CS(=O)(=O)C)cc(F)cc1[N+](=O)[O-].c1ccc(S(C)(=O)=O)c(F)c1 N1(C(CCC#C)=O)CC2(C1)CN(C(c1ccn3ncccc13)=O)CCO2 c1(CCC(N2CCCC(CO)C2)=O)ccc(COC(F)F)cc1 c1(C(=O)NC(CNC(c2cc(C)on2)=O)C)nnc2ccccc2c1O c1(CC)ccc(C(C)NC(c2nnnn2CCC2CC2)C(C)C2CC2)s1 C(c1ccc2occc2c1)=CC(=O)N(C1CN(C(=O)CC2(C)CCCCO2)C1)C C1(CNC(C2(CC)CC2)=O)CN(C(C2CC(=O)C2C)=O)CCC1C C=CCC(C(=O)N1CCCC(C(F)F)C1)NC(c1ccccc1F)=O c1(C(N(C(CC)COCc2nccc(CO)n2)C)C)ccc(S(N)(=O)=O)cc1 C(=O)(CC(O)CCCCCC)N(C1CCN(C(=O)C=CC(C)C)C1)CC#C C(=O)(CC(C)N(C(=O)CC(C)SC)C)N(CC#C)C c1(CC(N2CCC(COC)(NC(c3cc[nH]c3)=O)C2)=O)c[nH]c2ccc(Cl)cc12 C1(NC(C2C(C=C)OCC2)=O)CN(C(c2cc(OC)ccc2F)=O)CCC1C c1(C(=O)NCC2C(Cl)(C(=O)NCC3(SC(=O)OCC)CC3)C2)cc(C)cs1 Cc1cccc(O)c1C(=O)NCC1C(C)CCN1C(=O)Cc1nc(C2CC2)cs1 N1(C(c2c(CC)nn[nH]2)=O)CC(CC(=O)NCC(O)C(F)(F)F)C(C)C1 C1(COC)(NC(C2CC2C(=O)OC)=O)CCCN(C(c2coc(C)n2)=O)C1 c1(C(=O)NCC=CCNC(CCc2ccc(N(C)C)cc2)=O)cccn2nnnc12 N1(C(C(C=CCCC)O)=O)CCC(O)(C(C)NC(c2cc(C)nn2CCC)=O)C1 CCCCC(CC)C(=O)NC1CN(C(C2CC2C2CCC2)=O)C1 C1(C(N2C(C)CC(CNC(=O)Cn3cc(CO)nn3)C2)=O)CCc2nccn2C1 C1(NS(CCC=C)(=O)=O)COCCN(Cc2cc(=O)c(OC)co2)C1 c1(C(N(CC(CC)NC(C2CCC(=O)N2)=O)C)=O)cc(=O)c(OC)co1 N(C(=NCCc1ccc(OC)cc1)NCCC)C(C#C)C.C(c1ccccc1)=CC Cn1cc(I)c2c(NC(C3(O)CCN(Cc4ccc(O)c(I)c4)C3)=O)ncnc12 Cc1ccc(NC(=O)C(Cc2cc[nH]n2)NC(c2ccc[nH]2)=O)cc1Cl C1(CC(=O)N(C2CCN(C(c3ccoc3CC(N)=O)=O)C2)CC)COCCOC1 CCC(C)C(C(=O)NC1CC1)N1CCC(CN2CCOCC2)CC1 C(=O)(C(CNC(=O)CC1(OC)CCC1)CC1CC1)N1CC(NC(=O)OC)C1 c1(CN2CCC(NC(C3=CC=NC(=O)C3)=O)C(O)C2)cc([N+](=O)[O-])ccc1Br C1(NC(c2cccc(C(N)=O)n2)=O)CC=C(C(=O)NCC2CC2Cl)C1 c1(C(=O)NCC2C(C)CCN2C(=O)CC(C)c2ccco2)noc2ccccc12 C1(C(C)(C)N)CCN(C(=O)CCC(F)F)CC1.N1(C(=O)OC)CCCC1C(=O)O N1(C(C2(CC)CCN(C(=O)OC)C2)=O)CCN(C(c2ncnn2C)=O)CC1C C1(NC(C2CC(C#C)(O)C2)=O)C2CCC1N(C(C1CCCN1C(=O)NC)=O)C2 CC1=NNC(=O)C1CC(=O)N(C(C)(C)CC(=O)NCCSC(F)F)C N1(C(CC(C(C)C)C)=O)CCCC2(C1)C(NC(C1CCCN1C)=O)CCN2C CC1=NN(C)C(=O)C1CC(=O)NC1(C)CC(NC(c2nnn(C)n2)=O)C1 c1(C(=O)NCC(c2ccc(Br)cc2)C)cccn(C2CCC2)c1=O C1(C2CCN(C(=O)Cc3cnoc3)C2)(NC(C2CC3CCC2O3)=O)CC1 N1(C(c2cc(C(C)C)sn2)=O)CCCC(C2CCN(C(=O)C3=NOCC3)C2)C1 C(=O)(N1CC(O)CO1)C1(F)CCN(C(C2(CO)C(C)CC2)=O)C1 c1(OC)cc(N)c(C(N2CCN(C(=O)C3=CCCS3)CC(O)C2)=O)cc1O c1(C(N2CCCN(C(c3c(C)nc[nH]3)=O)C(C)C2)=O)cc(Cl)c(N)c([N+](=O)[O-])c1 CCCCN(CCCN(C(=O)COC)CCNC(=O)NC1CC1)C N1(C(c2cn(CC)nn2)=O)CC(NC(=O)C(N)=O)C(S(C)(=O)=O)C1 C1(CCOC)CCCN(c2nnc(-c3cnn(C)c3)n2CCn2cccn2)C1 N1(C(c2nc(CC)sc2)=O)CC2CCCC1C2CNC(=O)CC12CCC(CC1)C2 O=C(C#CC1CCOC1)NCC1CCN(C(c2cn3c(n2)SCC3)=O)C1 c1(SC)ccc(C(=O)NC2CC(F)(CNC(=O)Cc3nnc(C)s3)C2)o1 CC1(C)CC(=O)NC1CNC(=O)CCC1CCN(C(c2cc(O)cc(F)c2)=O)C1 c1(C(=O)NC2CN(C(CCC(=C)C)=O)CC23CC3)ccc2nc(O)[nH]c2c1F C1(C(=O)NCC(CC=C)NC(C2(CC)CCCC2O)=O)CCC(CO)CC1 n1(C(C)C)cc(C2CC2C(=O)NCCCN(C(=O)CC2CCCCO2)C2CC2)cn1 c1cccc(S(C)=O)c1.C1C(O)CNC(=O)C2(CC2)CC(=O)N1C.CS C(=O)(CCCC(=O)NCC(C1CCCC1)NC(=O)Cc1nnc(C)s1)OC Cc1cn2c(CC(N3CC(NC(=O)CC(=O)OC(C)(C)C)CC3C)=O)csc2n1 c1(C(=O)NC(C2CC(NC(c3onc(CC)n3)=O)C2)C)cccc(F)c1F C1(NC(C=CC(C)NC(=O)CN2CSCC2=O)=O)C(O)C2CCOC12 O=C(CCc1ccc(O)cc1)NOCc1cccnc1-c1ccccc1 C(C(=O)N(CC(C)(C)NC(=O)Cc1cnccc1C)C)(C(C)C)SC N1(C(=O)CSC(F)F)CCN(C2CCN(C(C3CC34CC4)=O)C2)CC1 C(=O)(C(C)(C)C(C)(F)F)NCC(c1ccc(F)cc1)NC(C(CSC)O)=O CC(C)CCC(O)C(=O)N(CCCCC(=O)NC(CO)C(=O)N(C)C)C C1(C(=O)NC(CNC(c2c(C)nsc2)=O)C)CCOCC1(C)C CS(=O)(=O)c1sccc1C(=O)NCCOCCNC(c1cc2c([nH]1)CCC2)=O C(=O)(C1=CS(=O)(=O)CCC1)N(C1CC2CN(C(CC(C)C)=O)C1C2)C C(CS(=O)(=O)c1ccc(F)cc1)OC.c12ccc3c(c1)CCC3OCC(=O)NC2 C1CCCCC(=O)N1.C1(CC(=O)NC2CCSC2)(OC)CCCCC1 C(CN=C(NCC1(NS(C)(=O)=O)CCOC1)NC1CC1)C1C(C)(C)C1 N1(C(c2ccc(C(=O)OC)c(Br)c2)C(=O)NC(CC)C)CCc2nocc2C1 CC1(C)CCCN(C(=O)Cc2ccc(Cl)s2)C1CNC(=O)C#CC1CC1 C1(C(N2C(CNC(c3c(OC)nsc3)=O)CC2)=O)OC2CCC1C2 C(=O)(C(C)(C)CCNC(=O)CC1CC(=O)C1)N(C1(c2ccoc2)CC1)CC c1(CNC(C2(CC=C)CN(C(=O)CCN3CCC(F)C3)C2)=O)ncncc1OC c1(OC)cccc(OC)c1NC(C1CCCCN1C(c1ccsc1S(N)(=O)=O)=O)=O c1(CC)nn(C)c(CNC(=O)CNC(=O)C(c2ccsc2C)N)c1Br C(CS(=O)(=O)c1cc(Br)ccc1Cl)N(C(c1ccccn1)C)C c1(C(=O)NCC2C(NC(C(COCC)C)=O)CCC2)cc2n(n1)CC1(CC1)C2 N#CC1(C(N2CCC(Cc3cn(C4CCCC4O)nn3)C2)=O)CCC(=O)CC1 N1(C(C(C2CC(F)(F)C2)OC)=O)CC(C)C(C)(CNC(C2(CF)CCOCC2)=O)C1 C(=O)(C(CCC)CC(C)C)NC1(C(=O)NC2CCC(CCC)CC2)CC1C c1(C(=O)NCC=CCNC(C2OC(C)(C)OC2(C)C)=O)coc2c(Cl)cccc12 C1(NC(c2cc(CCCC)oc2C)=O)CC(NC(=O)CC2=CCCC2)C12CCC2 c1(C(=O)NC(C(C)NC(=O)CC2COCC(C)(C)O2)(C)C)ccc(Cl)c(F)c1N c1(C(N2CCC(NC(C3(C4CC4)CC3)=O)C(F)C2)=O)ccc2nnn(O)c2c1 N1(C(COCCCOC)=O)CCC(C)(C)C(CNC(=O)Cc2c[nH]nc2O)C1 CC(C)C(C(C)C)NC(=O)CC1CCCC1NC(c1cc(Cl)n[nH]1)=O C1(N(C(C2(CC)CC(C(=O)OC)C2)=O)C)CCN(CCC(C)CC)CC1 N1(C(C(C(CC)O)(F)F)=O)CCCC(C2CCN(C(=O)CN3CCC(C)(O)C3)C2)C1 C1(N(C(C(C)=C2CC2)=O)C)CCCC2CN(C(c3cc(CC4CC4)on3)=O)CC12 Cc1nc(CNC(=O)CC2CN(C(=O)C(c3ccc(Cl)cc3)C)C2)sc1I c1(C(N2CC(C(C(=O)NCc3cncn3C)OC)C2)=O)cnn(C)c(=O)c1 N1(C(C(C)(C)C2CCC2)=O)CCC2(CCCN(C(c3cccn3C3CC3)=O)C2)C1 c1(C(=O)NC2CC(NC(C3C(C)CC3C)=O)C2)cnc2nc(O)ccc2c1 c1(CC)nn(C)c(CC)c1C(=O)N(CC(O)CNC(C1(CO)CCOC1)=O)C C1(NC(c2cc(C)n(C)n2)=O)COC2(CCN(S(=O)(=O)c3ccc(F)cc3)CC2)C1 C=CC(C)(CC)C(=O)N1CCC(CN2CCN(C(=O)CC3CCCC3)CC2)CC1 C(=O)(C(CN(C(C1CCOC1C(C)C)=O)CC)(CC)CC)NCC1N(CC)CC1 c1(C(=O)NC2C(NC(c3c(C)n(C)nc3Cl)=O)CC2)ccc2nnc(S)n2c1 c1(C(N)=O)ccc(CC(=O)NCC2CCCN2C(=O)CCC2CC2C2CC2)cc1 n1(CC(C)C)cc(C(=O)NC2CCC(NC(=O)C(C)N(C)C)C2)c(C(F)F)n1 c1(CC)ccccc1OCC(=O)NCCCCN(C(=O)C(C1(O)CCCC1)F)C n1(C(CC)C)nnnc1C(C1CC1)NCCNC.c1(C)snnc1C1CC1 C1(CCNC(c2nc(CCCC)sc2)=O)C(C)CCCN1C(c1cccn1C)=O C(=O)(C#Cc1ccc2c(c1)OCO2)N1CCCC(Cc2ccc(OC)c(C)n2)C1 N1(C(c2c(C)ccc(C)n2)=O)CC(C)N(C(c2cnn(C3CC3)c2C)=O)CC1C c1(C(=O)NCC2CCCN(C(C3CCN(C(N)=O)CC3)=O)C2)cccc(F)c1Cl c1(C(N(C2CCCN(C(=O)CCc3cccc(O)n3)C2)CC)=O)[nH]ncc1C#N C1(CNC(c2ccc(SC)o2)=O)COCCN(C(c2cc[n+]([O-])cc2)=O)C1 Cc1nnsc1C(=O)NCC(C)(C)CN(C)C(C1(CO)CCCO1)=O CC1CN(C(=O)CC2CCC=CCC2)CCCN1C(C1CC12CCOCC2)=O c1(C(N(C2CCCN(C(=O)C(C)(C)c3ccccc3)C2)CC)=O)ccc(C#N)s1 c1(CNC(N(C)CCOc2c(O)cccc2Cl)=O)cccc(S(C)(=O)=O)c1F C#Cc1ccnc(C(=O)NC(C(=O)N(C)CC2(O)CCC2)C2CC2)c1 C1(c2noc(C3CCCN3C3CC3)n2)(NC(C2CCCO2)=O)CCCCC1 c1(C(=O)NC2(CC=C)CCN(C(=O)C(C)C(=O)OC)C2)nc(C)n2ccccc12 CC(C)(CC(F)F)C(=O)OC1CCCCCC1F c1(C(=O)NC)ccc(C(=O)NCCCCCCNC2CCCC(OC)C2)cc1F c1(C(=O)NC(C(=O)NCc2c(CCC)nns2)C2CCOC2)ccccc1CO N#CC1(CN2CCOC(C(F)F)C2)CCNCC1 N1(C(CSCC=C)=O)CCC(CC(=O)NCc2cccnc2Cl)C1(C)C CCC(CC(F)(F)F)C(=O)N1C2COCC1CC(NC(c1ccns1)=O)C2 CCC(C)CC(=O)NCC1CCN(C(c2cnc(N)cn2)=O)C1 c1(C(N2CCCC(NC(c3csc(Cl)c3)=O)C2)=O)ccc2nsnc2c1 CCC(CC(=O)N1CCC(C(F)C(=O)NCc2cc(Cl)no2)C1)C1CCC1 c1(C2N(CCCc3nnn(CCOC)n3)CCC2)ccc(OC)c(C#N)c1 N1(C(CNS(CCCC)(=O)=O)=O)CC2CCN(C(c3nnsc3C)=O)C2C1 CCC(O)(C(=O)NCCC1CCN(C(=O)CC(C)CF)CC1)c1ccccc1 c1(C(C)NC(c2ccc(-c3cnco3)cc2)=O)ccc(N2CCCS2(=O)=O)cc1 n1(CCN2C(CC(=O)Nc3c(C#N)scc3)CCC2)ccc2ccc([N+](=O)[O-])cc12 N1(C(=O)CCN2CCCCCC2)CCC2C(CCN2C(c2ncccn2)=O)C1 C1(NC(=O)CCc2cnco2)CCCC12CN(C(C1(O)CCCCC1)=O)C2 N1(Cc2nc(-c3cc(OC)c(C)cc3OC)sc2)CC2CC(CO)CC(C2)C1 CC(=O)CCCC(=O)NCC1CCN(C(=O)CC2(O)CCCOC2)C12CC2 CC1CCCC1(O)CNC(C1CCC(NC(c2cc(CO)[nH]n2)=O)C1)=O c1(C(N2C(C)CC(CC(=O)NCCCn3cnnc3)C2)=O)ccc(F)c(O)c1 C12(CNC(C(C)Cc3ccc(F)cn3)=O)CC(NC(C3CC3F)=O)(C1)C(C)(C)O2 N1(C(c2scc(C)c2C)=O)CCC2(C(=O)NCC(O)C3(Cl)CC3)CCCC12 C1(N(C2(c3nnnn3CCC3CC3)CCCSC2)CCNS(N)(=O)=O)CC(F)(F)C1 c1(C(N2CC(O)(CCNC(c3nn(C)c(=O)cc3)=O)C2)=O)cccc2c1COC2 c1(C(CC(=O)N(CC(C)NC(C(C)=CC)=O)C)NC(=O)OC)ccc(F)cc1 C1(NC(c2n[nH]c(CC)c2Cl)=O)CCC2(CCCN(C(=O)CC(F)F)C2)C1 c1(C(N2CC(CNC(CN(C)CCO)=O)OCC2)=O)cnc2c(c1)C(=O)CCC2 N1(C(c2nc(OC)oc2)=O)CC2(C1)CN(C(C1(NC(C)=O)CC1)=O)C2 N1(C(C(c2cccc(F)c2)(C)C)=O)CC(NC(C2(CO)CCC2)=O)C(O)C1 CC1(C)C(C)(C(N2CCC(O)(CNC(C3CCNC3=O)=O)C2)=O)C1(C)C c1(C(=O)NC2(C)CC(NC(CCC3(C)CC3)=O)C2)cc2nc(Cl)ccc2o1 C(CC(C)C)(C(=O)Nc1cc(O)cc(F)c1)NC(c1c(C)csc1)=O c1(NC(CC2CC(NC(CCC=CC(C)C)=O)C2)=O)cc(C#N)ccc1F C(=O)(CS(=O)(=O)CC(C)C)Nc1cccc(NC(C(C)OCCC=C)=O)c1 N1(C(c2c(C)onc2)=O)CC2CN(C(=O)CCN3CCC(F)C3)CC2C1 C1(=CCNC(CC=C=C)=O)CCN(C(C2CC(C)OC2=O)=O)CC1 c1(C(=O)NCC2(CNc3ncc(I)cn3)CC2)ccc2cc(O)ccc2n1 c1(C(N2CCC(CC(C)NC(C3OCCCO3)=O)C2)=O)ccc(N2CCC2)cc1 C#Cc1ccc(C(N2CC3OCCN(C(c4cnc(S)[nH]4)=O)C3C2)=O)c(F)c1Cl C(=O)(C(C)(C)CC(C)(C)C)NC1C2CN(C(CCc3c(C)noc3)=O)CC1CC2 c1(OC(=O)NCC(c2c(C)occ2)=O)cc(Br)cc(Cl)c1F C1(NC(c2cccc(SC)c2)=O)CN(C(=O)C(CO)C(F)(F)F)CCC12CCC2 C1(C)(CC(=O)N(C2CCCN(C(c3cn(C)c(O)n3)=O)C2)CC)CCS(=O)(=O)N1 c1(CC)cc(N)c(C(=O)N(CCCCNC(=O)CC(O)C(C)C)C)c(F)c1 CCCC(C(=O)N1CC(=O)N2CCC(CC2)C1)OC.C(N)(=O)NCC C1(C(=O)NC2C3(CN(C(CC4CC(=C)C4)=O)C3)CCC2)CCc2cnc(C)n2C1 N1(C(CCc2cccc(C)n2)=O)CCC(C(=O)NC2CCCSC2)C(C)C1 c1(C(N2CC(OCC)(CNC(C3CCCO3)=O)C2)=O)nnn(C(C)C)c1C N1(C(C2(CC=C)CCOCC2)=O)CC2COCCC2(NC(=O)CC#N)C1 CC1CCc2c(sc3ncnc(NC(C4CCC(Nc5cnnn5C)C4)=O)c23)C1 Cc1ncnc(O)c1C(=O)NC(C)CCN(C)C(c1ncnc(O)c1F)=O Cc1c(NCCC(N)=O)nc[nH]c1=NCc1c(-c2ccccc2)cnn1C C1(CC(=O)N(CCN(C)C)CCO)CCCCN1C(c1ccc(=N)[nH]c1)=O C1(C2C(=O)N2)CC2CC2C1.CC(C)(C)OC(CCCF)=O.C1CN1 C1(NC(c2cccc(C)c2C)=O)CN(C(=O)C(F)C(C)C)CC(C)(C)C1 N1(C(C2C(C(C)NC(c3cnn(C(C)(C)C)c3)=O)C2)=O)CCCCC1CF C1(F)(CNC(Cc2c(C)ocn2)=O)CCN(C(=O)C(O)Cc2ccccn2)CC1 c1(C(=O)NCC(CC=C)NC(C2CC(N(C)C)C2)=O)ccc2sccc2c1 C1(NC(c2c(CC)cno2)=O)CN(C(=O)C(c2cc(C)ccn2)(F)F)CC12CC2 Cc1nonc1CC(=O)NCC1(NC(c2conc2C2CC2)=O)CC1 N1(C(C2(C(=O)OC)CC2)=O)C2CCCC1CC(NC(c1ncc[nH]1)=O)C2 C1(CNC(C(CC#C)C)=O)CCC2(CCN(C(C3COC3)=O)CC2)O1 c1(C(=O)NC(Cc2cc(C)n(C)n2)C)cc(S(=O)(=O)N2CCCCC2)ccc1Cl C1(C(=O)NCc2c(C(=O)NCC(C)(C)CC3CC3)[nH]cc2)CC12CCOC2 CC1=C(C(=O)NCCCC2CCCN2C(C2CCC(O)CN2C)=O)CCC1 C(=O)(C(C)CCC(C)(C)C)NC1(CCOC)CCN(C(CCOCC#C)=O)CC1 CC(C)(CNC(C1CC2(CC2)CO1)=O)CC(=O)Nc1cnc(Cl)nc1 c1(C(=O)NCCN(C(=O)CCC2CCCO2)CC(C)O)occ2c1CCOC2 c12nnc(n1CC1CC1(C)C)N(C)C2C.C(C(F)F)OCCOC c1(C(C(=O)NC2CC(F)(F)C2)N(C2CCCC2)CC(C)C)cc2ccccc2[nH]1 N1(C(c2ccc3ncnn3n2)=O)CCc2sccc2C1c1ccccc1 c1(C(=O)NC2(C3CN(C(C(C)N(C)C)=O)C3)CC2)cnc2ncnn2c1O c1(C(N(CCCNC(=O)CCSCCC(N)=O)CC)=O)ccc(C#N)[nH]1 c1(CC)cccc(NC(C2CC(C)CN2Cc2ncc(Br)cc2Cl)=O)c1OC C1(CC(N2CC3C(NC(c4nn(C(F)F)cc4Cl)=O)C3C2)=O)CN2CCN1CC2 C1(NC(c2c(COC)cc[nH]2)=O)CN(C(c2cnc(N)c(Cl)c2)=O)CCC1CO N1(C(C(C2CCOCC2)C)=O)CCCC12CCN(C(c1cccc3[nH]ncc13)=O)C2 c1(C(N(C)CC2N(C(CC(=O)N(C)C)=O)CCC2)=O)cc(F)c(F)cc1N C1(NC(c2c(CC)cns2)=O)CCN(c2nnc(CO)s2)CCC1CO CN1CCCN(C(=O)CC2N(C(C3CC(=O)NC(=O)N3)=O)CCC2(C)C)CC1=O c1(-c2cn(NC3(CF)CCN(C(COC(CC)(C)C)=O)C3)nn2)c(C)cccc1C CC1(C)CC(C(=O)Nc2cnc(C(N)=O)cn2)CN1C(=O)C(F)C1CCC1 c1(CNC(C(N2C(c3cccc(OC)c3)C(O)CC2)=O)=O)cccc(Br)c1C#N C=CCC(CNC(=O)C(C)(C)CN(C)C)C(=O)N1CC(CO)C2(CC2)C1 c1(CNC)cc(C(=O)OCC(CC(=O)OC)(F)F)c(F)cc1C C(CN(C(=O)CN1C(=O)CN(C)C1=O)C)(CO)(CO)NC(CC1(COC)CC1)=O C(=O)(CC(C(=O)NCc1nc(CNC2CC2)cs1)NC(=O)OC)OC(C)(C)C C1(C2(O)CN(C(C3CC(C4CC4)=NO3)=O)C2)(CNC(C(C2CCC2)OC)=O)CC1 CC(C(=O)NCC1CCCN(C(c2cnoc2C2CC2)=O)CC1)C(C)(F)F Cc1ccc(C(=O)NC2(CNC(c3ccsc3C)=O)CC2)cc1S(C)(=O)=O CCCC(C)(O)CC(=O)NCC(C)(C)C#CC(=O)N1CC(O)CC1(C)CO C(C(O)CC(=O)N1CCN(C(C)(C)C)CC1)NC(C(n1ccc(C)n1)C)=O C1(CC=C)(NC(=O)CCC2CCC2)CCCN(C(=O)C(C)(C)C(C)O)C1 C1(C(N2CCC(C(C#C)C)CC2)=O)CCCN(C(=O)C(C)(C)C)CC1 c1(OC)ccc(CC(=O)NC2CCC(NCc3cc(O)cc(F)c3)C2)cc1O Cc1ccc2cc(NCC3CN(Cc4ccccc4)CC(C)S3(=O)=O)cnc2c1 n1(CC(=O)NC(C(=O)NC(CC=C)CC)CN(C)C)c(C)ccc1C C=C(Cl)CC(C(=O)Nc1cc(F)ccc1C)NC(=O)CC1CC=CCC1 N1(C(CC2CCCN(C)C2)=O)CC(CNC(c2n[nH]cc2Cl)=O)OC(C)(C)C1 CC1(C)CCC(CC(N2CCC(NC(=O)CSc3ccc(F)cc3)CC2)=O)OC1 c1(C(=O)NC2C(C=C)CN(C(=O)CS(C)(=O)=O)C2)cccc2ccn(C)c12 c1(C(=O)NC(CN(C(CCOC(CC(C)C)C)=O)C)C)ccc(C2CC2)cn1 C12(NC(C=COCC)=O)CCCC1N(C(=O)COc1ccc(Cl)c(CC)c1)CC2 c1(C(N2C3CC(CNC(C(CSC)(C)C)=O)C2CC3)=O)c(O)cc(F)cc1F c1(C(=O)NC2CCC(N(C)C(C3(C)CCCC3)=O)C2)cc2cnc(Cl)cc2s1 c1(N2CC(C)CN(C)CC2)nc(N(CCCF)C)nc2c1CCC2 c1(SC2CC(CC)N(C(=O)OC(C)(C)C)CC2)cc(F)ccc1[N+](=O)[O-] N1(C(CC=C(C)C)=O)CCC(NC(C2(c3ccn(C)n3)CC2)=O)C1(C)C N1(C(C2(Cc3cnn[nH]3)CC2(F)F)=O)CCCN(C(c2ccccn2)=O)CCC1 C1(O)(CNC(C2CCC(NC(C(C)(F)c3ccon3)=O)C2)=O)CC2CCC1O2 c1(C(N2C(CNC(=O)C(C)NC(C)=O)CC(OC)C2)=O)ccc(Cl)c(Cl)c1 C=CC(O)(C(=O)NCC=CCNC(=O)CC1SC(=N)NC1=O)C(F)(F)F N1(C(CC=C(C)C)=O)CCC(OCCNC(=O)C(C)Cn2ccc(C)n2)CC1 Cc1nn(C)c(N)c1C(=O)NC1CC1CNC(c1cccc(Cl)c1Cl)=O N1(C(C(CC=C)(F)F)=O)CCC2CN(C(=O)Cc3cccc(F)c3O)CC2CC1 c1(C(N2C(COC)CN(C(c3sccc3C#N)=O)CC2)=O)cc(F)c(F)c(F)c1 c1(C(=O)NC)cccc2ccncc12.C1(C(=O)NCCOC2CC2)(C)CCCN1OC C1(COC)(NC(C2CCC(O)C2)=O)CCN(C(c2ccc(-c3nc[nH]n3)cc2)=O)C1 c1(C(N(CCNC(C=C(COC)C)=O)CC2CC2)=O)sc(C2CCCC2)nc1C Cc1nc(O)c(C(=O)NCC(C)NC(=O)CC2NC(=O)CNC2=O)nc1C c1(OC)cc(CN2CCC3(CC3C(N3CC(F)(F)C(F)(F)C3)=O)C2)c(Br)cc1O CCCCC(=O)C(=O)NC1(CO)CCN(C(=O)C(CO)N(C)C)C1 CC(C)C(CC(=O)NCC1(NC(C2CCCCS2)=O)CCC(F)(F)CC1)C(C)C C1(N(C(c2c(C)nc(C)o2)=O)C)CCN(C(=O)C(C)c2cccs2)CC12CC2 c1(C(N2C(Cc3cn(C4C=NN(C)C4=O)nn3)CCC2)=O)ccc(F)c(CO)c1 C(=O)(C(F)C(C)(C)O)NC1(C(=O)NCC(C)OCC#C)CCCC1C c1(OC)cc(C(N2CC3CC3(CNC(=O)C(=O)NC(C)C)C2)=O)ccc1Cl CC1CN(C(=O)Cc2c[nH]nc2O)CCC1NC(=O)CCc1nnc(S)nc1O N1(C(C)=O)CCC(CNC(=O)CCN(C(C)C)Cc2[nH]nnc2C)CC1 CC(C)(O)CC(=O)N1CCN(CCCNC(=O)CC2CCSC2)CC1 C1(NC(c2ncn(CC)n2)=O)CC(C)CN(C(c2ccc(C3CC3)c(F)c2)=O)C1 CC(C)C(C)C(CNC(c1ncsc1Br)=O)NC(c1ccn(C)c1)=O CC(C)C(CCNC(=O)C1=CCC1)NC(=O)CSc1nncn1C1CCCC1 N1(C(C(C#N)=CC(C)C)=O)CCN(C(=O)CN(C)C(C2CCCC(O)C2)=O)CC1 N1(C(C(C)NC(=O)C=Cc2cc[nH]c2)=O)CC2CC2C2CC12 C1(C(C)C)COC(CNC(C)CCN2CCCC2=O)C1 C=CCCCCCNC(=O)C(C1CC1)NC(=O)C(C)Cn1cccn1 c1(C(N(C2CN(C(=O)CN3CC=CC3)C2)C)=O)cnccc1Br Cc1ncoc1C(=O)NCCOCC(=O)NC(CO)C1CC1 N1(C(CC(CC)(F)F)=O)CC2CCCC(NC(C3(COC)C=CCC3)=O)C2C1 C=CCC(CNC(=O)C(=O)Nc1cc(C(=O)O)ccc1C)CC(C)C(C)C c1(C(N(C(C)CNC(C2CC3CCC2O3)=O)C)=O)cccc2scnc12 N1(C(c2c(NC(C)=O)cncc2)=O)CCC(NC(=O)CSC2CC2)C(C)C1 c1(CC)nc(N(C2CCN(C(=O)CC3CCC4CC4C3)CC2)C)[nH]c(=N)n1 c1(C(N2CCC(CN(C)C(c3nnc(S)n3C)=O)C2)=O)n[nH]c2c1CC1CC21 C=CC1(C(=O)NCC(=O)OCCO)CCN(C(C2CCC(O)CN2C)=O)C1 c1(CN(C(CC)C)Cc2cccc(Cl)c2)c(C)[nH]c2ncccc12 CCC(C)CC(C(=O)N1CCC1C)NC(=O)C1=CC(C)(C)C1 N1(C(C(C(C)C)SCC)=O)CCC(C2CC2)C1C(=O)NCC1(CN(C)C)CC1 C(=O)(C(C)C(=O)N1CCC(N(C)C(C23CC(C(=O)OC(C)(C)C)(C2)C3)=O)C1)OC C(=O)(n1ccccc1=NC(=O)c1csc(C2CC3CCC2C3)n1)OC(COC)=O C(C)(CC(C)CC)NCC1(CCC(=O)NC(c2c(CCCC)onc2)=O)CCCC1 CC1(C)C2CN(C(c3csc(Br)c3)=O)C(C(=O)NCc3ccno3)C12 C12(C(N3CCC(C(C)C)(C(=O)NCCCC4CC4C)C3)=O)CC(C)(CCO1)C2 C1(CC)(NC(c2cnc(Br)s2)=O)CCN(C(=O)Cc2cnc(C)s2)CC1 CC1CC(NC(c2cnn(C(C)(C)C)c2N)=O)CN(C(=O)COCCF)C1 Cc1cc(C(N2CC(NC(c3nn[nH]c3Cl)=O)CC(C)C2)=O)c2ncccc2c1 C(=O)(C1=C(Cl)CCOC1)NC12CC(NC(CC(C)(O)c3ccccc3)=O)(C1)C2 C(=O)(CCC(C)(C)NC(=O)C(C#N)C(C)C)NC1C(C)(CC)C1 CC1CCC(NC(c2coc(-c3cccnc3)n2)=O)CN1CC1CCCC1 N1(C(C2C(C)C2)=O)CCC(C2(O)CCN(C(=O)CC(F)(F)C(F)F)C2)CC1 CC(CCC(=O)NC(C(F)(F)F)C1CC1)NC(=O)Cc1cc[nH]c1 C1(CCC)CN(C(=O)C(C)SC(F)(F)F)CC1NC(=O)C(c1cnn(C)c1)O N1(C(C2CC3OC2C2CC32)=O)CCN(C(C2C3CC4C(C3)C24)=O)C(CO)C1 c1(C(=O)NC(c2cccc(OC)c2)CNC(C2(O)CCC2)=O)cc(F)cnc1O C(C)(CCC(=O)N1CCCC1C=CC(=O)NC(C1(OC)CCC1)C)OC C(=O)(C1COc2ccccc21)N1CCC(C2(NC(c3coc(Br)c3)=O)CC2)C1 C12(C(=O)NCCCN(C(C(CC)C(C)C)=O)CC)CCCC(=O)N1CCC2 CCCC(C)(C)CC(=O)N1CC(CC(=O)NC(c2cscn2)C)CC1(C)C c1(N2CCCC(NC(=O)C(c3ccccc3)O)C2)ccc([N+](=O)[O-])cc1 N1(C(CCOC)=O)CCOC(CN(C)C(C2(N3CCOCC3)CC2)=O)C1 C12(NC(c3cc(-c4c(OC)cccc4)[nH]n3)=O)CCN(C(=O)CNC=O)CC1C2 C1(CC(=O)N(C2CCN(C(c3ocnc3CC)=O)C2)CCC)CC2(CCC2)CO1 C#CCC(C)C(=O)NC1CCCC1CNC(c1oc(Br)cc1C)=O S(=O)(=O)(c1ccc2c(c1)C(=O)NCCC2)N(C)CC1C(C(F)F)C1(C)C c1(N(C)CCSc2ccccc2F)ccnc(N)c1 C1(NC(C2CC23CCCC3)=O)(CO)CCCN(Cc2cc(Cl)sc2Cl)C1 CN1CCCC(C)(COCC2CCN(C(C(=O)NC3CCOC3)=O)CC2)C1 n1(CC2C(C)C2)nc(-c2cccc(F)c2)nc1Cc1cnc(C2CC2)o1 C1(OCC)CC(O)C12CCN(C(C(=O)NCCCc1ccccc1)C(C)C)CC2 C1(OCC)CN(C(=O)C(C(C)C)SCC)CC1NC(=O)CS.C(C)(C)(C)S(C)(=O)=O c1(OC)cccc(O)c1CN1CC(NC(c2nc(C)cnc2C)=O)C1 Cc1cc(C(=O)N(CC(C)NC(=O)CC2(C(F)F)CC2)C)ccc1S(N)(=O)=O N1(C(CC(=O)NCC#C)=O)CCN(C(=O)Cn2cc(C(F)(F)F)cn2)CC1C c1(NC(C(Cc2ccc(OCC)cc2)=O)=O)c(F)ccc(OC)c1Cl C1(OCC)(CNC(=O)C(n2ccc(C)n2)C)CN(C(=O)C(F)F)C1 C(CCCC(C)NC(C1CC1(C)C)=O)NC(c1nc(C(C)C)oc1)=O c1(CC(=O)NC2CC(C)(C)N(C(C3CC4(CCC4)C3)=O)C2)ccc2c(c1)CCC2 CCCC(C(=O)N1CCN(CC(C)NC(=O)C(C)(C)CC)CC1)NC(C)=O C(C(=O)NCC(C)(C)C(C)O)(C(C)O)NC(CCc1cc(C)on1)=O c1(C(=O)NC(C(C)NC(C2(CC)CC2)=O)C(C)C)cc2c(nc1O)CCC(F)(F)C2 N1(C(C=C(CC)CC)=O)C2CC=C(C(=O)N3CCN(C)C(CO)C3)C1CC2 CCCC(C)(C)CC(=O)NC1(CNC(c2ccc(Br)c(N)c2)=O)CCOC1 N1(C(c2cccc(OCC)n2)=O)CCCC(C2CN(C(=O)C(C)NC(C)=O)C2)C1 N1(C(c2c(OCC)nccc2)=O)CC2CC(NC(=O)C(O)CC(N)=O)CC1C2 c1(OCC)ccc(C)cc1C(=O)NCC(C)CNC(=O)CC1CC2(CCC2)CO1 C1(C)(C(=O)C(=O)NC(=O)C(C(C)C)n2ccc(C3CC3)n2)CCC(=O)N1.CCC(C1CC1)N CP(C)(=O)c1ccccc1C(=O)NC1CN(C(c2ccc(F)cc2)=O)CC1CO C1(NC(C=CC(C)(C)C)=O)CCN(C(=O)Cc2cncnc2)CC1O c1(C(=O)NCC(CN(C)C(c2ccon2)=O)(C)C)ncccc1Br n1(CC(=O)NCC2(NC(C(C3CCOC3)OC)=O)CCCC2)ncccc1=O c1(C(CC(=O)NC2CCCC2NC(=O)COc2ccccc2O)O)ccc(F)cc1 C1(NC(C2N(CC)CC2)=O)CCN(C(C2CCC2(OC)OC)=O)C12CCC2 c1(CC(C2(C)CCCO2)NC(CCC(C)C)C)ccc(C(F)(F)F)c(Cl)c1 Cc1cc(C(N2CCC(O)(CNC(C3CC34CCCCC4)=O)C2)=O)cc(C)n1 c1(OC)cc(CCNC(=O)C(N2CCC(C(C)(C)O)C2)=O)c(NC(C)=O)cc1Br Brc1ccc2c(c1)C1(CC2)CCN(CC2(C3CC3)CCCCC2)CC1 c1(OC)c(CNC(c2ccncc2C)c2ccccc2C)cccc1C Cc1cc(C(=O)NC(C2CCN(C(=O)Cn3ncc(O)nc3=O)C2)C)cnc1O N1(C(CC2C(CNC(C3C(OC)CCC3)=O)C2)=O)CCc2ccc(O)cc21 CC1CC(C)(C)CCC1NC(C12CC(CN1C(c1cccc(=O)o1)=O)C2)=O C1(CCC(=O)N(C(C(C)SC)C)C)CCCN(C(c2cc(C#N)c[nH]2)=O)C1 C(CC(C)CCNC(C1C2CN(CC(C)C)CC12)=O)NC(CC)=O c1(C(=O)NCC(C)OC2CCCC(C)C2)[nH]nc2ncccc12 C1(NC(C(=O)NC(C)C)=O)CC2CCC1N(c1ccc(C#N)cn1)C2 CCC(C(=O)N1CC(C(C(=O)NOCCOC)NC(C)=O)C1)C(C)(C)CC C(=O)(C1=C(Cl)CCC1)N(CCC1CCN(C(c2c(CCC)onc2C)=O)CC1)C c1(C(=O)NCC23C(CN(C(C=CCCC)=O)C2)C3)cc(Br)ncc1N(C)C C1(NC(COCC)=O)C(CNC(=O)CN2CC3CC3C2)CCC12CCC2 N1(C(c2c(CC)nn(C)c2)=O)CCN(C(c2ccccc2Cl)=O)CC1CO c1(C(=O)NCC=CCNC(C2(CC=C)COC2)=O)ccc(O)nn1 C(C)(CCCCNC(=O)COc1nn(C)cc1Br)NC(C1C(C=C)C1)=O N1(C(C(C)NC(COC)=O)=O)CC2(CO)CC1(C(=O)N(CC(F)Cl)C)C2 C(=O)(C(C)C(C)S(C)(=O)=O)NC(CC1CN(C(c2c(OC)scc2)=O)C1)C C1(O)(COC)CCOCC1NC(=O)CCCSc1ccc(Cl)cc1F c1(CC)c(C(N2CCCCC2CNC(=O)C(c2cncnc2)C)=O)cccc1F C12(CNC(C3OCC(C)(C)C3)=O)CC(C1)C(NC(=O)C(C)(F)F)CO2 C12(OC)CCC(C(=O)NC3CC3CNC(=O)CC3CCC4CC34)(CC1)CC2 c1(C(=O)NC(C)CN(C)C(C2(c3ccc(F)cn3)CC2)=O)ccc2c(c1)NCCC2 CC1(C(=O)NCCn2cnc(NC(N3CCC(O)CC3)=O)c2)CC2(CC(=O)C2)C1 C1(NC(C2(CC=C)CCC2)=O)CS(=O)(=O)CC1NC(c1ccncc1Cl)=O C(=O)(C(CC(F)F)NC(C1CN(C(=O)OC(C)(C)C)CCN1C)=O)OC C1(NC(C(CC=C)OC)=O)CC2CC(NC(c3cnc(OCC)s3)=O)C1C2 C1(C(N(CCCN(C(=O)C(O)c2ccsc2)C)C)=O)CCN(C2CCOC2)CC1 N1(C(c2ccc(OC)nc2)=O)CC(C)(C)CC1C(N1CC2(CCCC2)C1)=O c1(C(C)NC(C)CCc2ccccc2)ccccc1I.CC#N c1(C(=O)NC(CN(C(=O)C(C)CN2CCCC2=O)CC)C)cc2occc2n1C C(=O)(CC(C)(C)C(C)(F)F)NC1C(N(C(=O)C(C)(C)CC(F)F)C)CCCC1 c1(C(N2CCC(NC(CSC(C)(C)C)=O)C2)=O)ccc(F)c(C(C)(F)F)c1 N1(C(C(C(C)C)n2cnnn2)=O)CCC2(CC1)CN(C(C1CCCOCC1)=O)C2 c1(C(=O)NCC(C)NC(COCC(=O)OC)=O)c[nH]c(=N)s1 CCC(F)(C(=O)OC)C(=O)NC1CC(c2ccc(Cl)cc2C(C)=O)C(O)C1 C(=O)(CC(F)(F)C(C)C)N1C(CNC(c2cncc(O)c2)=O)CC(COC)C1 C(N=c1[nH]c(=NCc2csc(Br)c2)[nH]c2c1SCC2)c1nc(=N)s[nH]1 c1(C(=O)NC(C(C)NC(c2ccon2)=O)CO)cc2ncccn2n1 c1(C(=O)NCC2CC(F)(CNC(Cn3ncc(C)c3)=O)C2)cc2n(n1)CC(F)C2 N1(C(c2ccc(C)s2)=O)CC2CCC1C(CNC(C1(C)CC1(F)Cl)=O)C2 c1(OC(C)(C)C)ccc(C(=O)NC2CCC2NC(c2ncoc2C2CC2)=O)nc1 CC1(C)CC(O)CCN(C(C2CC(F)(F)CN2C(C2C3CCCCC23)=O)=O)C1 N1(CCc2nc(C)[nH]n2)CCCC(C(=O)NC(C)C(C)C)C1 c1(C(=O)NCC2(F)CCC(CNC(C3CC(=C)C3)=O)C2)c(S(N)(=O)=O)cnn1C Cc1cc(C(=O)NC2CCC(CNC(C3CCC(=O)C3)=O)C2)ccc1S(C)(=O)=O CC(C)(C)C(C(=O)NC1CCCC1NC(c1cnc(O)o1)=O)NC(N)=O C(=O)(CCC(N)=O)N(C1CCN(C(C2(C#N)CCC2)=O)CC1)CC c1(COC)nc(C(=O)N(C)CCNC(c2cn(CC3CC3)nn2)=O)co1 C(=O)(C(Cc1ccccc1)C(C)C)N(CCCNC(C1(OC)CCC1)=O)C C1(NC(c2nc(C3(C)CC3)oc2)=O)CC2CCCC(C1)N2C(C12CSCC1C2)=O c1(C(=O)NCC2(F)CC(NC(C3(COC)CCC3)=O)C2)cccn(CCO)c1=O c1(C(=O)NCCNCCOC)cnn2ccncc12.C(C=O)(C(C)C)OCC Cc1cccc(C)c1NC(=O)C(C(C)(C)C)NC(=O)NCC(c1ccc(O)cc1)O CCC(C)(F)C(=O)NCC1CC(NC(c2nncn2CC)=O)C1 N1(C(c2cnc(C)s2)=O)CCCCC(CNC(c2occc2Cl)=O)C1 CC(Cc1nc(C(C)(F)F)no1)S(C)=O C#CCC(C)(C)C(=O)NCC1CCCN(C(=O)CC2CCCC(F)(F)C2)C1 N1(C(CC(=O)OC)=O)C2CCC(C2)C1C(=O)Nc1cccnc1C c1(C(c2cc(F)ccc2Cl)NCc2n(CCCOC)nnn2)nccc(Cl)c1C N1(C(Cn2ncc(C)c2)=O)CCC2(COC(CNC(C3CCCN(C)C3)=O)C2)C1 c1(CC(=O)NCc2c(C)nc(CNC(C(COC)OC)=O)o2)ccc(C)c(C)c1 Cc1cc(C)n2cc(C(=O)NC3CCC(C)N(C(C45CC(CO4)C5)=O)C3)nc2n1 c1(C(=O)NC(CC)CNC(c2cn(CC(N)=O)nn2)=O)c(C)ccnc1NC N1(C(C2CCN3CCOCC23)=O)CCC2(CCC(O)CC2)CC1 CCC(C(=O)N1CCN(C(=O)COC(C)C)C(c2nccn2C)C1)C(C)C C(=O)(C(CNC(c1nnn(C)c1N)=O)CC1CC1)NCc1c(C)nco1 C12(CNC(c3c(C)[nH]c(C(F)(F)F)c3)=O)CCCCC1N(C(=O)C=CI)CC2 C1(NC(C(C)N(C)C)=O)CC2CC1N(C(=O)CCc1cc(Br)ccc1F)C2 C1(CC(C)NC(=O)CSC(F)F)CCN(C(C2(C)COCCO2)=O)CC1 C(=O)(C(C(F)(F)F)NC(=O)OCC)OCC1(CC(=O)NC(C)(C)C)CC1 c1(C(=O)NCCCN(C(c2c(CC)c[nH]n2)=O)CCO)cncc(NC(C)C)c1 N1(C(C(C)Oc2ncccn2)=O)CC2CCN(C(C3(CF)CC3)=O)CCC2C1 C12C(O)CCN1NC2=O.c1(C(=O)NC)ccc(C(F)(F)F)nc1.c1(C)cc(Br)ccn1 c1(OC(C)C)cccc(C(N2CCCCC2CNC(=O)C(C)C2CCC2)=O)n1 c1(C(=O)NC2C(NC(=O)CCc3cc[nH]n3)CCCC2)ccc(F)cc1[N+](=O)[O-] c1(C(=O)NCC2COCCN2C(=O)COCC2CCOC2)cc(F)c(F)cc1F Cc1cc(C(=O)NC2CCCC(NC(=O)C(F)(F)C(F)F)CC2)cc(C)c1O c1(OC)ccc(OC)c2c1CN(CCCCCC(C)C)CC2O C1(C(=O)NC(C)(C)CNC(=O)CC2SC(=N)NC2=O)CC2(CCC2)CCO1 C1(C(N2CC(OCCNC(C3C(C=C)C3)=O)C2)=O)C2CN(CC(F)(F)F)CC12 N1(C(CC2CCN(C)C2)=O)CC2(NC(c3cn(C(F)(F)CO)nn3)=O)CC1C2 N1(C(c2c(CC)c[nH]c2)=O)CCC(C)(CCNC(C2(CCCF)CC2)=O)C1 C1(CC)CN(C(C2CC(C3CC3)=NO2)=O)CCN1C(c1sc(C)cc1Cl)=O CC1(C)C(C(=O)NCCC(O)CNC(=O)Cc2csc(S)n2)C1(F)F C1(NC(C=CC=C)=O)C2CC1(C)CN2C(=O)C(C)(C)NC(=O)OCC=C.C(C)(C)C C1(N(C(=O)CNC(c2cccs2)=O)C)CCCCN(C(C2CCCN2N=O)=O)C1 c1(C(=O)NCC2C(NC(C3(C)CC3(Cl)Cl)=O)CCC2)cnc(O)nc1O C1(NCC2(c3[nH]c4ccncc4c3)CCCCC2)CCCC12CCCCO2 c1(-c2c(CN3C(C)(c4ccccc4)CCC3)cccn2)cc(C(F)(F)F)ccc1N c1(C(=O)NC2(C)CCN(C(C(CCSC)O)=O)C2)ccc(C)c(F)c1N C(=O)(C(F)(F)CC)N(CC(C)NC(=O)CCC1CCC1)CC C12CC3CCC(C1)N3C(=O)C1(c3cn2nn3)CC1.C(CC(F)=C(F)F)OCCOC c12cn(C)nc1C(=O)N2.C(=O)(C(C)NC(=O)CCC1CC1CO)NCCOC C1(C(N(CCNC(C2(S(N)(=O)=O)CC2)=O)CC)=O)OCC2CCCCC12 C1(NC(CC2(CC=C)CCCC2)=O)CC2(CCC(CNC(C3CC3C)=O)OC2)C1 C1(F)(C(N(C(C)C)CCN(C(=O)C=C2CCN(C)C2)C)=O)C2CCCCC12 N1(C(c2c(OCC)ccc(C)c2)=O)CCN(C)c2ncccc21 N1(C(C2(C)CC2)=O)CC(NC(c2cc3ncccc3s2)=O)CC2(CCOCC2)C1 C1(CC)CN(C(c2cc(Cl)cc(Cl)c2)C(=O)NC(C)C(=O)OC)C(C)CO1 c1(CC2CC(C)(N(C(=O)CC=CCN(C(C)(C)C)C(=O)C3CC3)C)C2)ncn(C)n1 C(CCCCCNC(c1ccncc1C(F)(F)F)=O)NC(=O)CC1CCC1(F)F C1(NC(C(c2ccn(C)n2)(C)C)=O)C2CN(c3ncccc3Cl)CC12 N1(C(c2ccc(NC)cc2)=O)CCC(CO)CC1C(N1CCOC(CCF)C1)=O c1(CC(C(=O)NCC(C(C)C)NC(C2(COC)CC2)=O)C)ccccc1Cl c1(C(N2C(C)(CNC(CNC(C(C)(C)C)=O)=O)CCC2)=O)ccc2cc[nH]c2n1 c1(OC(C(=O)N(CC)CC2(O)CN(C(=O)C(F)F)C2)C)ccc(Cl)cc1 CC(C)C(C)C(CNC(=O)C(C)(C)C)NC(c1c(C(F)(F)F)cnn1C)=O C#Cc1c[nH]nc1C(=O)NC(c1nocc1C(=O)NCC1(Cl)CCC1)C C1(C(C(C)NC(=O)CNC(c2cccc(Cl)c2)=O)C(=O)O)CN2CCCC1C2 C1(C(N2CCN(C(C)C)CC2)=O)CCOCCN1C(=O)CCC1(C)N=N1 C1(NC(C(C)NC(CC)=O)=O)CN(C(c2cc(C)nn2C)=O)CC12CCCC2 C1(OCC)CC(C(C(=O)NC2(C)CC2)N(C)Cc2ccnn2C)CC1OC C(=O)(C(C)(C)C(F)F)NCCCC(C)NC(=O)CSc1ccccc1F C1(NC(C2CC(C3CC3)=NO2)=O)CCC2CCN(C(c3csc(O)n3)=O)C1C2 CC(C)C(N=[N+]=[N-])C(=O)NC12CCC(C(=O)NCCOCC3CCCC3)(CC1)C2 CCCC(CCC)CC(=O)N1CCOC(CC(N2CCCC2(C)CC)=O)C1 CN1CCCC(C)(C(=O)Nc2c(CN3CCCC(N)C3)cccc2)C1 CCCCCCCCS(=O)(=O)NC1CN(C(c2nc(Cl)ccc2F)=O)CC1C#N C(=O)(C(CO)N(C)C)NCC(CC)NC(=O)C(C1CC1)OC(C)=O C1(C(=O)NC2CC2C(=O)OC)COCCC1NC(C1(C(=O)NC)CC1)=O c1(NC(c2n[nH]c(C)c2C)=O)ccc2c(c1)CCCN2CCN(S(C)(=O)=O)C C1(C)(C(=O)NC2CN(C(=O)NC)C2)CCCN(CC(C)CC(C)C)C1 c1(COCCOC)nc(-c2cccc(OC(C)(C)C)c2)n(CC2CCCOC2)n1 c1(COC)cc(C(=O)NCCC(C)N(C(=O)C(C)SC(F)(F)F)C)n[nH]1 C=Cn1nccc1C(N1CC=CCC1C(=O)NC1(c2[nH]c(C)nc2C)CC1)=O C1(N(C(Cc2cc(CC)no2)=O)CC)CCCN(C(c2cc(C(C)C)[nH]n2)=O)C1 c1(C(=O)NCC(C)CNC(=O)CC(c2cccc(F)c2)N(C)C)cccc[n+]1[O-] c1(C(=O)NCCOC2CCN(C(CCC)=O)C2)cccc2c1ccn2C c1(C(=O)NCCN(C(C2(C)CCC(C)C2)=O)CC)cc2n(n1)CCO2 c1(CN2C(C(=O)NCC3CCN(C)CC3)CC(=C)C2)cc(Br)ccc1O N1(C(c2cc(C)c(F)c(C)c2)=O)Cc2ccccc2OCC1C N1(C(c2c(C)nc[nH]2)=O)CCC2(NC(=O)Cc3ccsc3)CC2C1 C1(NC(C2CC(SC)C2)=O)CCC(=O)NC1C1CCN(C(=O)OC(C)(C)C)CC1 CCC(CC)CC(=O)N1CCC(C(C)NC(=O)CC(O)C2CCCC2)C1 N1(C(CC(CCC)C)=O)CCC2(CC1)CC(NC(=O)C=Cc1nc(C)cs1)C2 C1(CNC(=O)NC23CC(C#N)C(C2)C3)CCC2(CC1)OCCO2 CC1CCCCC1(CNC(c1cn(CC(N)=O)nn1)=O)NC(c1cccnc1)=O c1(C(N2C(C)CCC(CNC(C=CC)=O)C2)=O)ccnc2[nH]c(O)nc12 C(C1CC1)(C1CC1)=CC(=O)NC(C1CCN(C(=O)COC(=O)CO)C1)(C)C c1(C(N2CC(F)CC(NC(C3(CC)CC3)=O)C2)=O)cnc2c[nH]nc2c1 N1(C(CC(C)SC)=O)CCC(C2(NC(=O)Cc3n[nH]c(=NC)s3)CCC2)CC1 N1(C(C2CCCN2CC(F)(F)F)=O)CCC2(CCN(c3ncncc3I)CC2)C1 C1(NC(C=C(CC)C)=O)CCCN(C(=O)C(CC(C)C)C2CCC2)C1C C(CCCCCN=[N+]=[N-])NC(C(C(CC)C)N(C)C(c1nccnc1C)=O)=O N1(C(C(C=C)(F)F)=O)CCN(C)C(CNC(C2CC2c2ccccc2C)=O)C1 N1(C(C=Cc2ccn(C)c2)=O)CC2(CCN2c2ccncn2)C1 N1(C(C2OCCN(C(=O)CN3CCCC3)CC2)=O)CCC2CCC(C1)S2 N1(C(CC2N(C(CN3C(C)CCC3)=O)C3C2CCC3)=O)CC(CO)CC(C)(C)C1 CC(C#CC(=O)NCCN1CCC(NC(=O)OC(C)(C)C)CC1)NC1CC1 C(=O)(C(CC(F)F)C1CCC1)NC1CN(C(COC(C)C)=O)CC1CC1CC1 c1(C(=O)NC2CCC(CNC(c3cccc(C)c3C)=O)C2)nc(C)c(C)nc1O N=c1ncc(C(=O)NC2CCN(C(C3C4CC5C(C4)C35)=O)CC2)c[nH]1 N1(C(C=CCCC)=O)CC(NC(c2cccc(COC3COC3)c2)=O)CC1C Cc1cc(C(=O)NCC2(CNC(=O)CCc3ccc[nH]3)CC2(F)F)cc(C)c1O c1(C(=O)NC(CNC(C(CC)OC)=O)CO)cc2cccnn2c1 C(=O)(CC1=CCN(C)CC1)NCCC1CC(NC(CCC(CC)C)=O)C1 N1(C(CC(C)NC(C(COC)(C)C)=O)=O)CC2(CCC(=O)N2)C1 C#CCCCCCC(=O)NC(CNC(=O)C(C)C(C)CC)(CC)CC C(=O)(C(C)(C)C(=O)NC1CCN(C(c2ccc(F)c(C(F)F)c2)=O)CC1O)NC c1(CC)nc2cccc(C(N3CCC4(C3)CN(C(C3CNC(=O)C3)=O)C4)=O)c2[nH]1 c1(NC(=O)Cc2csc(=NCc3c(F)cccc3Cl)[nH]2)ncnn2cccc12 CC1=C(C(=O)N(C2CCCN(C(=O)CCc3cn(C)nn3)CC2)C)SCCO1 C1(NC(c2c(C(C)(C)C)n[nH]c2)=O)CC(NCCC2CC3CCC2O3)C12CCC2 CC(CC(=O)NCC1(CNC(=O)CCc2cnoc2)CCCC1)c1ccco1 CC(CCCCCO)NC(=O)CC1CC2(C1)CN(C(c1c[nH]ccc1=O)=O)C2 C1(NC(=O)Cc2csc(Cl)c2)CCOCC1NC(c1coc(Cl)c1)=O N1(C(c2ccc(OC)cn2)=O)CC2CC1CCC2NC(=O)C(C)(C)n1cnnn1 CCC(CCOC)C(=O)NC1CC(C(=O)NC(c2cn(C)nn2)(C)C)C12CCC2 C1(NCCN(C(CCC)=O)CCC2CCCCC2)(CF)CC(F)(F)C1 c1(C(N(C2CCN(C(c3cc(N)cnc3Cl)=O)C2)C)=O)cccn2c(O)nnc12 N1(C(C(CC)(C)O)=O)CC2(C(=O)NCC(O)C3CC3)CCC1CC2 c1(CCNC(c2cc(Cl)nc(Br)c2)=O)nc2ncc(Br)cn2n1 c1(C(=O)NCC(C)CNC(C2(Br)C(C)C2C)=O)n[nH]c2c1CCOC2 N1(C(C(c2c(C)cccc2)C)=O)CCC2(C1)CN(C(c1c(C)nccc1C)=O)C2 c1(OC)cccc(CC(c2nc(-c3ccc(F)cc3)nn2C2CCCOC2)C)c1 C1(C(C(=O)NCC(C)NC(COCCC)=O)O)CCOCC1 c1(CC)c(C(=O)NCCC(C)NC(c2cc[nH]c(=NC)c2)=O)[nH]c2ccccc12 CC1(C)CCC(CC(N2CC(O)(CNC(c3n[nH]cc3Cl)=O)C2)=O)OC1 N1(C(c2cnc(OCC)nc2)=O)CCC(C)C(NC(C2CN3CCN2CC3)=O)C1 C(N=c1[nH]cnc(Cl)c1OC)C1(NC(C(CCC)(C)C)=O)CCOCC1 N1(C(C(CCC)OCC)=O)CCC(C)(C)C(CNC(=O)C(O)Cc2cnc[nH]2)C1 N1(C(c2cnc(C)c(N)c2)=O)CCC2C(C1)CN2C(=O)CC1COCCN1C c1(NC2CCN(C(COCC)=O)CC2)cc(OC)c(S(N)(=O)=O)c(Cl)c1 C=CCCCCCN(C(=O)C(CC1CCOCC1)NC(=O)CC(C)SC)C c12ccc(o1)C(=O)NCc1nc(sc1)CNC2=O.c12nncn1C2.C(C)(C)N.COC C(=O)(C(C)(C)CC(C)=O)N(CCC(=O)NCc1onc(CC)n1)C N1(C(Cc2c(C)ocn2)=O)CC(C)CN(C(=O)C#CC(C)(C)C)C(C)C1 C1(C(N(C(CSCC)C)C)=O)CCCC(NC(c2cc(CO)on2)=O)CC1 N1(C(CC(C)C2CCCO2)=O)Cc2ccccc2CC1CO C1(C(CO)N)CCCCC1.C(C(F)(F)CO)N(CC(O)CN(C)C=O)C N1(C(c2nc(CC)[nH]n2)=O)CCC(O)(CNC(=O)C=CCn2cncn2)C1 CC(C)C(=O)C(=O)NCC1CCCC1NC(=O)CCc1cncc(O)c1 C1(C(N(C(C)C)CCNC(=O)CCc2ccon2)=O)CCCS1(=O)=O c1(NC)ccc(O)c(C(=O)NCC2CC(C(N3CCN3)=O)C2)c1 C1(NC(CC2(C)CCN2C(=O)C2CC2)=O)CCC2CCCC1O2 N#CC1CC(C(=O)NCC2(CNC(c3csc(O)n3)=O)CC2)C1 C1(C(=O)NCC(CNC(c2cc(OC)no2)=O)OC)CCC(C2CCC2)CC1 C1(C(=O)NOC(C)(C)CO)(CC=C)CCN(C(c2cnc(N)cn2)=O)C1 C1(O)(C(C)NC(c2cc(CCCO)on2)=O)CCN(C(C2CC2(C)C)=O)C1 CN1CCN(C(=O)CC2CCCN(Cc3ccn(C4CCCOC4)n3)C2)CC1 c1(C(=O)NCCCCC(C)NC(=O)CN(C)C)c(F)ccc(Cl)c1N c1(NC(N2C(C3CCN(C(CCC#C)=O)CC3)CCC2)=O)cc(Br)ccc1C N1(C(C=CC)=O)CCC(CNC(c2ccc(-n3cc(Br)cn3)cc2)=O)C(C)C1 C1(NC(C(CCSC)O)=O)CN(C(=O)C(=Cc2cnn(C)c2)C)CC1N=[N+]=[N-] N1(C(C2N(C(c3c(C)cccc3C)=O)CCOC2)=O)CCC2(CCN(C)C2)C1 c1(C(c2noc(CC3CCCCC3F)n2)(C)C)ccc(F)c(F)c1 c1(C(N(C2CCCC2)CCOC)=O)cccc(CNc2cnccn2)c1 C1(CNC(c2ccnnc2)=O)CCC(C(=O)NOCC2(F)CCC2)O1 CC(C(=O)N1CCC2CN(C(=O)C3=CCSC3)CCC12)S(=O)(=O)C1CCOCC1 C1(C(N2CC(C#C)(C(=O)NCC=Cc3ccco3)C2)=O)CCC(C)(C)OC1 N1(C(c2c(C)nc[nH]2)=O)CCCC(C2CCCN(c3nnc(C(C)(C)C)o3)C2)C1 C=CCC(C)(C)CCNC(C1CNC(=O)CN1C(=O)C(CC)SC)=O C(C)(C)(CCC(=O)NCCCN1CCC(O)C1)N(C(C=CCCC)=O)C(C)C CCCCCC(CC)C(=O)N1CCC2CCN(C(C3CCC3OCC)=O)C2C1 C(CC(C(C)(C)C)NC(=O)CC1(C#N)CC1)N(C(C(C)Oc1ccc(Cl)cc1)=O)C CCCC(O)CC(=O)NC(C(=O)N1CC(NC(C)=O)C1)C(C)C C(=O)(C1=NNC(=O)CC1)N1CC(C)C(N(C)C(c2ccn(C)c2)=O)CC1 c1(NCCC(=O)NC(CNC(c2nccc(C)n2)=O)(C)C)ccc(Cl)cc1Cl c1(CN(CCC)CCNC(C2(O)CC2(C)C)=O)ccc(Cl)cc1F C(=O)(C1=Cc2ccccc2C1C)N1CC(CC=C)(NC(C2CCC=CCC2)=O)C1 Cc1c(C(N2CCN(C(C3CCCS3(=O)=O)=O)CC2CO)=O)sc2ccccc12 C(=O)(C(C)(C)C(=O)N1CC(C(=O)NC(C)Cc2ccccn2)C2(CC2)C1)NC CCC(C)(C(=O)NC1CC(OC2CCN(C(=O)CC(C)C3CC3)CC2)C1)OC C1(CC(=O)NC2CCCN(C(C3(C)CC(=O)C3)=O)CC2)Cc2ccccc2C1 c1(CCC(=O)NC(C)C(C)NC(=O)CSCC2CC2)nnc(-c2ccccc2)o1 c1(C(=O)NC(Cn2cc(-c3cc(C)c(C)s3)nn2)C)cnc2cccc(C)n12 C1(C)(C(=O)NCC2(F)CC(CNC(CC(C)(C)C#N)=O)C2)CCCCCCC1 c1(C(=O)NCC(CC)NC(=O)C(C)NC(C)=O)cc2cc(Cl)sc2[nH]1 Cc1c(N(C(CCc2ccsc2)C(=O)NC2CC2)C)cnn1-c1ccc(Cl)cc1 N1(C(C(C2CN(C(=O)CN3CSCC3=O)C2)O)=O)CCC12CCOCC2 C1(CNC(C(OC)OC)=O)CN(C(c2sc(C3CC3)nc2C)=O)CC1C C12(NC(CCC)=O)CC3CC(C1)CC(NC(=O)CC1CCCC(C#N)C1)(C3)C2 C(CC(C)C)(C(=O)NC1CCN(C(c2cnn(C)c2N)=O)C1C(C)(C)C)OC C(=O)(CC(O)C(C)C)NCCCN(C(c1cc(CSCC)on1)=O)CC c1(OC)cnccc1C(=O)NC(CNC(=O)C(C1CCCOC1)OC)CCOC c1(NC(C=C)COC)ccc(S(=O)(=O)NCC2CCCC(C)O2)cc1Br C1(CC=C)(C(=O)N(C)C(C)C2CC2)CCCN(C(C2CC23CCCCC3)=O)C1 N1(C(c2cc(C)nnc2)=O)CCC(CNC(=O)Cn2ccnc2C)C(C)C1 C1(COCCC)CC(NC(CCCOC)=O)CN1C(c1cnc(OC)cn1)=O Cc1nc(N2CCOC(C(C)NC(c3cc4ccccc4[nH]3)=O)C2)ncc1C#N c1(C(=O)NC2CC(NC(c3cnc(C)c(C#N)c3)=O)C2)ccc2ncccc2c1F CC(CN=c1nc(C2(N(C)C)CC2)[nH]s1)NC(c1cnc(C(F)(F)F)s1)=O N1(CCC)CCN(C(C2CC2(F)F)=O)CC1.c12ccc(nc1)N1CC(C1)NC2=O CC12CCCC(C(N3CCCC(CNC(c4cc(C#N)no4)=O)C3)=O)(CO1)C2 c1(C(=O)NCCNC(C2(OCC)CC(CF)C2)=O)c(C)c[nH]c1CC(N)=O c1(C(N2CCC(N(C(c3cc(C)c(C)[nH]3)=O)CCO)C2)=O)nc2cccnc2s1 c1(C(=O)NCCC2CC(NC(c3c(C)n(C)nc3)=O)C2)cc2c(s1)CCC2=O N12CCCC1CN(C)C(C)C2=O.C1(NC(c2cncnc2)=O)(CO)CCCC1 CC(CCN1CCOCC1)N=c1nc2scnc2c(N(C)Cc2nc[nH]n2)[nH]1 c1(CN2CC(COC)N(C(=O)CCn3cncn3)CC2)cc(F)cc([N+](=O)[O-])c1 n1(CC)cc(C(=O)NC2CCN(C(C34CSC(C3)C4)=O)CC2F)c2ccccc12 c1(CCCC(=O)N(C2C3CN(C(C4CCCCC4O)=O)CC23)C)ccc(Cl)nc1 C(C(C)(C)C(=O)N1CCC(NC(N)=O)C1)NC(C=C(C)C(C)(C)C)=O N1(C(CN(C(=O)CC2CCOC2=O)CCOC)=O)CC(N(C)C)CC1(C)C C(C(C)(C)CCCO)NC(C1C2CN(C(C(C)CC3CC3)=O)C1C2)=O c1(OC(CC2(NC(=O)OC(C)(C)C)CCC2)=O)cccc(N)c1Br CCCCN=C(NCCSc1cncn1C)NCc1ccco1 n1(C(C)C)ncc(CCN(c2cc(Br)cn2C)C2CC2c2cccc(Cl)c2)c1F C(C(C)C(=O)N(CCCNC(=O)CC1(O)CCC1)C)OCC CC(C)CC(=O)C(=O)NCCC1(C)CCN(C(=O)C2=COCCC2)C1 CC(C)C(CC(=O)Nc1cnc(O)c(F)c1)NC(C1CN(C)C(=O)N1)=O CCC1=NOC(CC(=O)NCC2(O)CN(C(=O)C(CC#C)C3CC3)C2)C1 CCCCC(O)C(C)C(=O)N1CC(O)CCC1C(N1CC(CC)C(F)C1)=O CC(=O)CCCC(=O)N(CCCC(N1CCOC(C)CC1)=O)C CC12CC(CC(N3CCCC(CNC(c4coc(Br)c4)=O)C3)=O)(CO1)C2 c1(C(=O)NC2(CN(C(=O)CC3(O)CC3)C)CC2)cscc1Br N(C1CSc2ccccc21)CCC(c1cccc(Cl)c1)N C1(NC(C(C(C)C)C)=O)C2CCC1CN(C(=O)C(C)(O)C(F)(F)F)C2 C#CC1(F)CCN(C(=O)C(C2CCCC2)NC(c2cnncc2C)=O)CC1 C=CCC(CC(C)C)C(=O)NC1CC2CN(C(c3ncsc3C(F)(F)F)=O)CC12 Brc1ccc2c(c1)CCN(c1nccc(=NCC3C4COCC34CO)[nH]1)C2 c1(NC(=O)Cc2c(F)cc(Br)cc2Br)ccc2c(c1)S(=O)(=O)C=C2 c1(C(=O)NCC(C)NC(C2CC(O)CN2C)=O)c[nH]c2ccc(O)cc12 C1(C(=O)NC2CCC(CNC(=O)Cc3ccsc3Cl)CC2)CC2CCC(C1)S2 C(CN=C(NCC1CN(S(C)(=O)=O)C1)N1CCCC(C)C1)OCC C1CCC(=O)NCCO1.C(C(C)=CC(=O)N(CCF)C(C)C)OC Cc1nc(C(C)NC(=O)CC(c2ccc(Cl)cc2)NC(N)=O)c(C)o1 C1(CC)CN(C(=O)Cc2nocc2C)CCN1C(c1cnccc1C1CC1)=O c1(OCC(C)NC(c2cnn(CC3CCCC3)c2)=O)ccc(Cl)cc1Cl C1(CC(=O)N(CCCO)CCOC)C2CCCC2N1C(=O)CC1CCSCC1 c1(CC)cc(C(N2CCCC2CNC(=O)C(c2c(C)noc2C)C)=O)ncn1 C(CCC(=O)NCCCN(C(=O)COc1cc(C)on1)C)=CC Cc1cc(C#N)nc(N2CCC2C(=O)Nc2cc(C(F)(F)F)ccn2)n1 c1(C(N2CCCC(N3CCNCC3=O)C2)=O)ccnc(Br)c1 C1(NC(c2cc([N+](=O)[O-])c[nH]2)=O)CN(C(=O)COCCO)CC12CCOCC2 N1(C(C(C(C)C)C2(C)CC2)=O)CCCC(NC(c2cc(C)c[nH]2)=O)CC1 c1(C(N(CC(C)N(C(C(CC)COC)=O)C)C)=O)cccc2c1NCC2 C1(C)(C(N(C2CCCN(C(C3(CO)CCOCC3)=O)C2)C)=O)CC=CCO1 N1(C(CCCOCC)=O)CC2CCC(C1)N(C(c1[nH]cnc1C#N)=O)C2 N1(C(c2nc[nH]n2)=O)CCC=C(c2ccccc2-c2ccc(F)cc2)C1 N1(C(c2n(CC)ncc2C)=O)CC=C(C(=O)NCc2nccn2C)C1 n1(CC)cc(C(=O)NCC(C)NC(C2CCCNC2=O)=O)c(C(C)C)n1 c1(C(N2CCN(CC(C)(C)NC(C3CC(Cl)(Cl)C3)=O)CC2)=O)cc(Cl)ccc1N c1(NC(=O)CN(C(=O)COCCCF)C2CCC2)ccc(F)c(O)c1 Cc1cc(-c2ccc(NCc3c(F)cc(F)cc3F)c(F)c2)c2ccccc2n1 N1(C(C=CCN(CC#C)C)=O)CC(CCNC(C2(C(C)(F)F)CC2)=O)OC(C)C1 n1(CCN(C(C)CN(CC(=O)N(CC(C)(C)C)C)C)C)cnc2c(N)ncnc12 C1(NC(C2C(CC)C2)=O)CC2CCC(C1F)N2C(C1(S(C)(=O)=O)CC1)=O c1(CN2C(C(=O)Nc3cccnc3I)CC(=C)C2)c[nH]c2ccc([N+](=O)[O-])cc12 C(=O)(CCCOC(C)=O)NC(C(=O)NC(c1ccnn1C)C(=O)OC)C C(c1cn(C)nn1)=CC(=O)NC(CC)C(=O)NCC1CCN(C(C)C)C1 c1(OC)c(CN2CCN(C(=O)CC3CCC(F)(F)C3)CC2)cccc1F C(=O)(C1=C(C)OCCC1)NC1(C)CCC(NC(C2CCC(C(C)C)C2)=O)CC1 C1(NC(c2ccccc2CO)=O)CCSC12CN(C(=O)Cc1ccco1)C2 c1(C(=O)NC(CNC(c2c(OC(C)C)nccc2)=O)(C)C)c(N)cc(Cl)nc1Cl O=S(=O)(c1cccc2c1OC(F)(F)O2)N1CCC(c2ccccc2)C1 N1(C(c2cn(CC)nc2)=O)CCC(COC)C(NC(=O)C(C)(C)N2CCCC2)C1 c1(CC(C)C)c(C(=O)NC2CCN(C(C3CC4(CC4)C3)=O)CC2)cnn1C N1(CC)CC2CCC1CN2C(c1cc(C)[nH]n1)C(=O)NC1CCC1 C1(C(=O)NC2C(C)CCC2C)COCCN(C(c2cccc(C#N)c2)=O)C1 N1(C(CCC2C(=O)NC(=O)N2)=O)CC2CC(C1)CN(C(c1ccnc(Br)c1)=O)C2 N1(c2nnc(CC(C)C)s2)CC=C(CNC(=O)CN2C(=O)CNC2=O)CC1 C1(C(C)NC(C(C)=C2CC2)=O)CCCN(C(=O)CCc2cncc(F)c2)C1 N1(S(c2cccc(C(C)C)c2)(=O)=O)CCC2(CCCN2C)CC1 N1(C(c2cn(CCC=C)nn2)=O)CCC(CNC(=O)C(O)C(C)C)(OC)CC1 N1(C(C(C)CNC(=O)C(C2CCCCC2)C)=O)CC(O)(C2CCC2)C1 n1(CCOC)ccc(C(=O)NCCCCn2cc(C3CCCOC3)nn2)n1 C1(NC(c2c(CC)nns2)=O)CCCC1(C)CNC(=O)C(O)CCc1ccccc1 c1(N2CC(NCc3cccc(C)c3F)C(C)C2)ncnn2cc(Br)cc12 c1(C(N)=O)ccoc1C(N1CCC1CC(=O)NC1CCCOC1)=O c1(OC)cccc(NC(=O)CCC2CC(NC(C3(CC4CC4)CCC3)=O)C2)c1 N1(C(=O)CCOC2CCC2)CC2CC1CN2C(=O)C(CC(F)F)c1ccccc1 c1(SCC(=O)NCC(C)N(C(CC(=O)OCC)=O)C)cc(=O)n2nc(C)sc2n1 c1(C(=O)NC2(COC)CCCN(C(=O)C(C)=C3CC3)C2)nc(C)n2ccccc12 c1(OC)cc(C)nc(NCc2ccc(=O)n(CCN3CCOCC3)c2)n1 N1(CC)CCN(CCNC(C)CNC(=NC)NCC(Cl)Cl)CC1 N12CCN(CC1)c1ccc(o1)NC2=O.N1(CCn2nnc(C)n2)CCOCC1C C1(NC(c2c(C)n[nH]c2C)=O)CC2CCC(C1)N2C(c1c(C)nc(C)nc1C)=O C1(NC(COC2CCN(C(C3CCC(=C)CC3)=O)CC2)=O)C2CCCCCC12 C(=O)(C1=CCC(C)(C)CC1)NCCN1C(=S)NC(CCCC)C(C(=O)OC)=C1C C1(CNC(Cc2n(C)cnc2)=O)CC(NC(=O)CN2CSCC2=O)CCO1 C(=O)(CC1=CCN(C)CC1)N1C(C(N(C(C)CC(N)=O)C)=O)C=CC1 C12(C(=O)NCC(CCCC)NC(c3ccc(COC)[nH]3)=O)CCC(O)(CC1)CC2 Cc1ncc(CC(=O)NCC2COC(CNC(=O)Cc3cc(C)[nH]n3)C2)s1 C#CCC(CC#C)C(=O)NCCN(C(c1ccc(C(C)C)nc1)=O)CC1CC1 c1(C(C)(C)NC(=O)NCc2n[nH]cc2I)cccc(Cl)c1 S(=O)(=O)(c1c[nH]ccc1=NCC1(OC(C)=O)CCOC(C)C1)NCCCCCCC=C C1(CNC(C(CO)N(C)C)=O)CCN(C(c2csc(CO)n2)=O)C12CC2 c1(C(N(C2CCN(C(c3c(C)nn(C)c3C)=O)C2)C)=O)cccc2c1CC(=O)N2 S(=O)(=O)(c1ccc(OC)c(C)c1)Nc1cc2[nH]cc(C(=O)NC)c2cc1 N1(C(c2c[nH]c(=NC)s2)=O)CC2(NC(C3CCC(F)C3)=O)CCC1CC2 c1(C(C(=O)NC2C(C)CN(C(C3CC(C)(C)CO3)=O)C2)O)ccc(F)c(Cl)c1 CC(CS(C)=O)C(=O)NCC1(CNC(C2(F)CC=CC2)=O)CCCCC1 c1(N2CCCC(N(C(c3cccc4ccoc34)=O)CCF)C2)ncc([N+](=O)[O-])cn1 C(=O)(C(Cc1ccccc1)C(F)(F)F)NC1(C)CCN(C(=O)CCCF)C1 c1(C(=O)NCC(C)(CO)NC(C2C(C)CC2)=O)cccn2ccnc12 N1(C(c2ccc(OC)cn2)=O)C(CNC(=O)Cc2cncs2)CC2CCCC12 C12(C(N(CC(C)(C)CNC(=O)CCCC3CCCCC3)C)=O)CCCC1CC2 Cc1cc2cc(C(=O)NCCCN(C(=O)CC3CCC(=O)NC3)C)oc2cc1C C(c1cccc(Cl)c1)=C(C)C(=O)NCC1(CNC(C2OCCOC2C)=O)CCC1 Cc1c(Cl)cc(C(=O)NC2CN(c3ncnc4c3CCC4)CC2F)cc1Cl Cc1ncccc1CCCNC(c1cc(CCOC(C)C)[nH]n1)c1nnnn1C c1(N2CCN(C(c3ccc(C(C(C)O)=O)cc3)=O)CC2)c(F)cc(F)c(F)c1F C12(CNC(CC(=O)NCC(CC)C(=O)NCC3CC3)=O)CC3CC(CC1C3)C2 Cc1ccc(C)c(C(N2CC=CC(NC(=O)C(C)OCC3CC3)C2)=O)c1 C1(CC(=O)NC2CS(=O)(=O)CC2N2CCOCC2)CCCC2(CC2)C1 C1(C(N(CCCCNC(=O)CC2(C)OCCO2)C)=O)CC=CCC1C(N)=O CCC(C)(C)C(O)C(=O)NCC(C(C)C)NC(c1cccc(O)n1)=O C1(=O)CCC(=O)N(C2CCCO2)C2(CC2)CN1C.c1(C(C)C)nnc(OC(C)C)s1 C1(NC(COCCOC)=O)CC2CN(C(c3ncccn3)=O)CC2C1 C(=O)(CC(C)CN(C)C)N1C(C(C(=O)NC2(c3c(C)ncs3)CC2)(C)C)CCC1 c1(CSCC(=O)N(CCN(C(C)C)C(C2CCCO2)=O)C)noc2c1COCC2 c1(C(N2CCC(NC(C(C)OCC)=O)C(O)C2)=O)cn(C)c(=O)c(C)n1 C1(CC)CCC(C(N2CCC(O)(CNC(=O)COCCOCCO)C2)=O)CC1 Cn1c([N+](=O)[O-])cnc1C(N1CCC(N(CCO)CC2CCC2)CC1)=O n1(CC)c(C)nn(CC(N2CCCCC(CNC(=O)CCN3CCCC3)C2)=O)c1=O c1(C(=O)OC)ccc(C(C)Nc2ccccc2SS(C)(=O)=O)c(Cl)c1 C1(CCC)(CO)CCCN1C(=O)CN(C(c1ccco1)=O)CC1CCCC1 C1(F)(C(=O)NC2(CCCNC(CCSCC(C)C)=O)CC2)CCN(C)CC1 C1(C(N2C(CC(C)C)CC2)=O)CC=CCC1NC(C1CC(F)C1)=O C(c1cnccn1)=CC(=O)NC1CC(NC(=O)C(F)C2CC2)CC1O c1(C(=O)NC(CC#C)C(=O)NCc2cc(COC)no2)cc(C)c(F)cn1 N1(C(CCc2cnc(C)o2)=O)CCC(CNC(c2nnc(C)s2)=O)C12CC2 C1(C(=O)NCCC(O)C2CCCC2)(NC(C(C=C)O)=O)CCOCC1 n1(CCOc2cccc(C(NC=O)C3CC3)n2)c(O)nc2cc(Cl)ccc12.C(C(F)F)O C1(C(=O)NCC(c2ccccc2SC)(OC)OC)CCS(=O)(=O)CC1 Cc1cccc(F)c1C(=O)NC1COCCN(C(c2cnn(C)c2C2CC2)=O)C1 CC1(C#CC(=O)NC2C3CN(C(C4(C)CCCNC4=O)=O)CC23)CC1 C(C(CC(=O)N1CCC1C(=O)OC)C1CCC1)NC(Cc1n(C)ccc1)=O c1(C(=O)NCC2CN(C(CC(CC)CC)=O)C(C)(C)C2)cc(Cl)cc([N+](=O)[O-])c1 c1(C(=O)NC(CNC(c2cnn(CC)n2)=O)CO)ccc([N+](=O)[O-])c(C)n1 N1(C(c2cc(C)n[nH]2)=O)CCC2(CC1)CCN(C(C1CC3CCC1O3)=O)CC2 Cc1cc(=NC2CCC(C)(N3CCC3)CC2)[nH]c(=NCc2cncn2C(C)C)[nH]1 c1(OC)ccc(C(N2CCC(CN(C)C(C3C4CCCC34)=O)C2)=O)c(OC)c1 C(=O)(CCC(F)(F)F)NC(CN(C(C1(SC)CC(=O)C1)=O)C)C N1(C(c2cnn3ccn(C)c32)=O)C2CCC1CN(C(=O)CC1CCC(C)(C)C1)CC2 C(=O)(CCC(CF)CF)N1CCC(CNC(CCSC)=O)CC1 c1(C(N2CCC(OCCNC(C(COCC)(C)C)=O)C2)=O)cc(Cl)ncc1O C1(O)(CN(C(C2C(CC)C2)=O)C)CN(C(c2cnc(CN)[nH]2)=O)C1 C(N=c1[nH]c2ncc(Cl)cc2s1)C12CCC(NC(c3cncn(C)c3=O)=O)(C1)CO2 N1(C(Cc2c(C)nn(C)c2)=O)CCC(C(=O)NCCC#CCO)C(O)C1 C1(CN(C(=O)CCOc2ccc(Cl)cc2)CC)CCCCN1C(=O)CC1(O)CC1 C1(CC)CC(O)(CNC(C2CC2)=O)C1.C(=O)(COCC1CCC1)NC C1(CCC(=O)N(CCN(CC=C)C)CC)CCN(C(C2CCN(CC)C2)=O)C1 C1(C2C(NC(CC=CC)=O)C2)CCCN1C(=O)CN(C1CCC1)CC C12(NC(C=Cc3scc(C)n3)=O)CCCN(C(c3cc(=N)[nH]n3C)=O)CC1C2 C12(C(=O)OC)CN(C(c3ccc(F)s3)=O)C(CO)(C1)C2 CCS(=O)CC(=O)NCCCN(C(c1cccc(-n2ccnc2O)c1)=O)C(C)C c1(C(=O)NCC2(C(=O)NC3CC(C#C)C3)CC(C)(C)C2)cccc(C#N)c1C N1(C(CN(C(C(C)CC(F)(F)F)=O)C2CCC2)=O)CC2(CCC(O)CC2)C1 N1(C(CC(COC)C)=O)CCN(C(C2CC(=C3CC3)C2)=O)C(c2nccn2C)C1 N1(C(c2[nH]c(=N)sc2)=O)CCN(C(c2cc(C3CCCC3)[nH]n2)=O)C2CC12 N1(CCC(=O)NC(C)CN(C(=O)C(C)(C)O)C)CCN(C)CC1 O=C(NNC(=S)Nc1ccc(I)cc1)C(F)CC(Cl)C(F)(F)F C1(C)(NC(C2(CC(=O)OC)CC2)=O)CC(NC(=O)CCC=CC(C)CC)C1 c1(NC(CCC(C)NC(C2N(C(C)=O)CCC2)=O)=O)c(C)cc(C)nc1C c1(NC2CCN(C)C2=O)cc(Br)ccc1S(=O)(=O)NC1CCCCC12CCCC2 O=S(=O)(c1ccc(Cl)s1)N1CCN(S(=O)(=O)Cc2ccc(C(=O)O)cc2)CC1C c1(CNC(C(c2ccc(C)cc2)N2CCCC2)=O)ccc2c(n1)NCCC2 C(=O)(CCCCCC(C)C)N(CC(C)(C)CNC(c1cc(SC)oc1C)=O)CC N1(C(C(C(=O)OCC)F)=O)CCC(NC(C2(c3ccno3)CCC2)=O)C(O)C1 N1(C(c2c(C)nc(C3CC3)o2)=O)CC(NC(C2CC(=C3CCC3)C2)=O)CC1(C)C c1(-c2cncc(C)c2)ccc2cnc(NC(C3CCN(CC4CC4)C3)=O)nc2c1 C1(NC(C2(CCC)CC2)=O)CN(C(c2cnn(C)c2Br)=O)CC1C(F)(F)F c1(C(N2CCC(NC(C(=O)NCCOC)=O)C(F)C2)=O)cc(OC)cc(Cl)c1O C(CS(=O)c1ccccc1F)NC(=O)NC1(CC=C)CCNC1 c1(C(N2CCC(O)(C(C)NC(c3cccs3)=O)CC2)=O)cccc2nsnc12 CC1CCCN1CC(=O)NC1CCC(NC(=O)C(C2CCOCC2)O)C1 c1(C(=O)NC2(CCNC(C(CC)F)=O)CC2)ccc2c(c1)NC(=O)CNC2=O C1(C(=O)Nc2cnc(Cl)cn2)CN(C(c2c(I)ccnc2O)=O)CCC1O Cn1cc(S(C)(=N)=O)c(NC2CC3(CCC3)CN2C(=O)OC(C)(C)C)n1 c1(CNC(=O)COc2cccc([N+](=O)[O-])c2)cc2c(=O)[nH]ccn2n1 C1(NC(C2C(NC(C3CC(F)(CF)C3)=O)CCC2)=O)CCC2(CC2)C1 C=C1CCN(C(C2CCCN(CCCC)C2)C(=O)NC2CCCC2)CC1 c1(C(=O)OCC(c2c(C)nn[nH]2)=O)cc(Cl)c(Cl)n1C N1(C(C(C)N(CC)CC)=O)CC(C#N)(N(C)C(C)C)C1 C=CC1CN(C(=O)CC2CN(C(c3cccc(C#N)c3)=O)CC2C)CC1O c1(C(=O)NCC(CNC(C2(COC)C=CCC2)=O)(C)C)cnc2ccsc2c1 Cc1cc(O)ncc1C(=O)N(CC(C)O)CCNC(c1cscc1C#N)=O Cc1ccc(C)c(C2(C(=O)NNC(=O)C3CC(OC(F)(F)F)C3)CC2)c1 Cc1[nH]nc(Cl)c1C(=O)NCC(C1CCCC1)NC(=O)CNC(N)=O c1(C(=O)NCCCCN(C)C(C2CCOC2)=O)cc2cccnn2n1 CC1CCCC=C1C(=O)NC(CC(C)(C)C)C(=O)N(CCCn1ccnc1)C CC(C(=O)N(CCCNC(c1nc[nH]n1)=O)CCO)=CC(C)(C)C c1(C(c2n(CCC)nnn2)NCc2cc(C3CCC3)on2)ccc(C)cc1Br C(C#CC1CCCCO1)N1C(C(N2CCC(N)CC2)=O)CCC1 c1(OC)nc(C)ncc1NC(C1CCCN1C(c1cc(Br)cnc1O)=O)=O C1(CNC(Cc2cn(CC)nc2)=O)(CO)CC12CCN(C(=O)C1CC1)CC2 C(=O)(C(C(=O)N(C1(CC(=O)NCCC2CCCOC2)CC1)C)OC)OC C(=O)(C(F)(F)C(F)F)NC1C(C(=O)NCC(C)CC(F)F)CCC1 Cc1cc(C(=O)NCC2CC(F)(CNC(=O)C(F)=CCCF)C2)cnc1C c1(C(=O)NC2C(CC)CN(C(=O)CCCC(N)=O)CC2)cnc2n(c1=O)CCS2 CCCCC(C(=O)Nc1cccc(C(=O)OC)c1)NC(c1conc1C1CC1)=O c1(OCCC)ccc(C(=O)N(CC(C2CC(F)(F)C2)OC)C)cc1[N+](=O)[O-] N1(C(CC2OCC(C)(C)C2)=O)CCC2CC2(C(=O)Nc2ccc(N=[N+]=[N-])cc2)CC1 C(=O)(C(C)(C)C(=O)N1CC2CC1CN2C(C1CCC=CCCC1)=O)OC(C)(C)C c1(C(=O)NC2(C3N(C(C(C)N4CCCC4)=O)CCC3)CC2)ccc2occc2c1 C(=O)(C1=CCCN(C(=O)C(C(=O)OCC)OC)C1)N1CC2C(CCC)(C2)C1 c1(OC)ccc(C(=O)NC2CCCC(NC(=O)CC(F)(F)Cl)C2)cc1O C1(NC(C2CC3(C2)CS(=O)(=O)C3)=O)CCN(C(c2cccc[n+]2[O-])=O)C12CCC2 N1(C(c2n(CC)cc(Cl)c2)=O)CCCC(C)C1CNC(c1cc(Cl)ns1)=O n1(CC)cc(C(=O)NC(C)(C)C(C)NC(=O)CCc2ccc(Cl)cc2)c(C)n1 C(=O)(C(C)(C)C1=CCSCC1)NC(CC(C)C)(C)CNC(=O)CN1CSCC1=O c1(C(N(C2CCCCN(C(c3ccnc(F)c3)=O)C2)C)=O)ccc(C#N)c(O)c1 N(C(=NCCCCN1CCN(C(C)C)CC1)NCC(C)(O)CC1CC1)C(CC)C Cc1nsc(C)c1C(N1CCCC1C(C)NC(c1cnn(C(C)(C)C)c1)=O)=O C(C1CCCN1C(=O)CC1CCSC1)=CC(=O)NCCCC(=C)Cl CC1(C)CN(C(c2cscc2Cl)=O)CCC1NC(=O)C1=CS(=O)CCC1 c1(C2N(C(C3CC(C)(NC(C4CC(Cl)(Cl)C4)=O)C3)=O)CCC2)cccc(F)c1F c1(N2C(C)(CNC(Cc3cncc(C)c3)=O)CCC2)cc(C)nc2ncnn12 CC1(C(N2CC(O)(CNC(=O)CC3CC(=O)NC3=O)C2)=O)CCC(=O)C1 Cc1nc(C(C(C)(C)NC(N2CCCC2CC(C)(C)C)=O)C)no1 C1(S(N)(=O)=O)(C(N2CCC(C(C)NC(c3cccc(CF)c3)=O)C2)=O)CCCC1 C1(NC(c2cn(CCOC)nc2C)=O)CCCCN(C(=O)C(O)COC)CC1 c1(OC)cc(C)c2cc(C(=O)NC(CNC(=O)CC(F)(F)Cl)C(C)(C)C)[nH]c2c1 c1(OC)ccc(-c2ccccc2)cc1C.n1(CO)nc(CO)nc1-c1ccn(C2CC2)n1 c1(NCCOC2CN(C(C=C(CC)C)=O)C2)cc(C)c2n[nH]cc2c1 N1(CCCNC(c2[nH]nc(N(C)C)c2Br)=O)CCN(C(=O)CO)CC1.C1(CC2CC2)CC1 C1(NC(Cc2c(C)ocn2)=O)CC(C)CN(C(=O)CS(C)(=O)=O)C1 Cc1cc(C(=O)NC2CCCCC2NS(=O)(=O)c2cccs2)cc(C)c1F C(=O)(C(C)C(=O)OC(C)(C)C)NC1C(NC(c2c(CC)[nH]cc2)=O)CCC1 n1(CC(C)O)cc(C(=O)NCC2CCN(c3cccc(F)c3)C2=O)ccc1=O CC(=O)CCCC(C)C(=O)NCC(C)C(=O)NC1CCC(N(C)C)C1 N1(C(COCCCC#C)=O)CCC(NC(c2cc(C(N)=O)cn2C)=O)C(F)(F)CC1 c1(OCC(=O)N(C(CNC(c2scc(C)c2C)=O)C)C2CC2)nc(O)nc(O)n1 CCCCC(C(=O)N(C)CCC)C(C)C.C(C)(C(=O)NCC(C)C)N1CC1=O Cc1cc(Cl)c(C(=O)NCC2CCN2C(=O)C=Cc2cccs2)cc1Br N1(C(CCc2c(C)ncs2)=O)CCC(C)(NC(=O)CCSCc2ccccc2)C1 c1(C(=O)NCC(CN(C)C(C2(C#N)CC3CC3C2)=O)O)cccc(F)c1F CC(C)C(C)(CNC(c1cc(-c2ccco2)on1)=O)NC(C1CCCO1)=O c1(CC2C(NC(CCc3ccc(OC)nc3)=O)C2)nc2ccccc2[nH]1 N1(C(C2CCCCC2F)=O)CCN(C(=O)C(=O)Nc2ncc(Br)s2)CC1 N1(C(CC(C(=C)C)OCC)=O)CCC(C(=O)NC2CN(C)NC2=O)=C(F)C1 N1(C(CNC(CC)=O)=O)CC2CC(NC(=O)CCS(=O)(=O)NC)CC2C1 Cc1cncc(CC(=O)NC2(CN(C(=O)CCN(CCC(C)(C)C)C)C)CC2)c1 c1(CC(=O)NC2CC(C)(NC(c3nc(C)oc3)=O)C2)c[nH]c2cnccc12 CCCS(=O)(=O)C(C)C(=O)NCC(CCOC)NC(c1cc(C#N)cc(C)n1)=O c1(-n2cc(C=CC(C)N(C(C)(C)C(=O)O)C)nn2)ccc2cnn(C)c2c1 c1(CC)cnc(CC(N2CCC(C(C)NC(c3cc(Br)n[nH]3)=O)C2)=O)[nH]1 CC(CC(N)=O)C(=O)N1CC(C(=O)NCCNC(=O)CC2CCCCC(=O)N2)C1 c1(CC(=O)N(CC(C)N(C(CCCOCCOC)=O)C)C)cc(C)ccc1C CC1CN(C(c2cc(O)nc(O)n2)=O)CCC1N(C)C(c1cc(C#N)no1)=O C=C=CCCC(=O)NC(CNC(c1c[nH]nc1C)=O)(CC)CC c1(C(N(CCCNC(C(CC)OC)=O)CC)=O)cc2c(F)ccc(F)c2s1 S(=O)(=O)(c1ccc2nc(Cl)sc2c1)N1CCCC(COC)CC1 c1(C(=O)NC2(C(=O)OC)CSC(C(C)C)C2)ccc(Br)cn1 N1(C(C2(N(C)C)CCCC2)=O)CCC2(CC1)CC2CNC(C1CC(F)C1)=O C12(NC(CCCC#C)=O)CCOC(CNC(=O)CNC(N3CCCC3)=O)(C1)C2 C(=O)(CC(C(C)C)OCC)N(C(CCNC(C1(C#C)CC1)=O)C)C c1(N2C(C(=O)N(CCCN3CCOCC3)CCO)CC3CC32)nc(Cl)c2c(n1)COC2 N12CCCC(C1)C2=O.n1(C(=O)NC2CC(C)(NC(C)=O)C2)nc(N(C)C)cc1C C(=O)(C1=CCCOCC1)N1CCC(CNC(c2c[nH]cc(C)c2=O)=O)C(C)C1 c1(C(N2CC=C(CCNC(C(F)=C(C)C)=O)CC2)=O)ccc2n[nH]c(C)c2c1Cl C1(NC(C2C(=C)CC2)=O)COCCN(C(=O)C=C2CCC2)C1 N1(C(c2n(CC)ccc2)=O)CCC2CCCN(C(C3CC(CC4CC4)C3)=O)C2C1 C1(C(=O)NCCCC2N(C(C(N)=O)=O)CCC2)COc2cc(Cl)ccc2C1 C(=O)(CC(C)(C)C1CC1)NC1(C)CN(C(=O)COCC2CCCOC2)C1 C1(NC(=O)COc2cccc(CO)c2)CC2(NC(=O)Cc3cc[nH]n3)COC1C2 N1(C(=O)C(O)c2ccsc2)CC2ON=C(CNC(=O)CC34CCC(CC3)C4)C2C1 CCC(CC(=O)NCCN1CCN(C(c2cccn2C(C)C)=O)CC1)C(C)C Cc1cccc(C(=O)NC2CCC(C)N(C(C)C(=O)NC(C)(C)C)C2)c1C C1(CC(=O)OC)CN(C(=O)C(C)SC)CCN1C(C1(Br)CC1)=O C1(CNC(c2ccc(-c3ccccn3)s2)=O)CN(C(C2CC(Cl)(Cl)C2)=O)CCO1 C(C(C)C(F)C(=O)NC1CCC(O)C1)NC(C=CCCC(C)C)=O C1(C(C)(O)CNC(=O)CC2CC2)CCN(C(=O)CNC(C2CCCC2)=O)CC1 N1(C(c2cc(C(C)=O)on2)=O)CCOCC1CN(C)C(C1CC1CF)=O CCCCCC(C)CC(=O)NCC(C(C)C)NC(=O)C(C)(C)C N1(C(c2c(C(C)=O)cccc2)=O)CC(C2CN(C(c3c[nH]cc(F)c3=O)=O)C2)C1 C1(NC(C2C(CC)OCC2)=O)CN(C(=O)CCC(C)(C)O)CC2(CC2)C1 c1(C(N2CCC(CC)(NC(C3CCC(=O)N3C)=O)CC2)=O)cccc2nsnc12 c1(C(=O)NC2CC(CNC(=O)COCc3cccnc3)C2)c(Cl)cccc1Cl O=C(C1=NNC(C(F)(F)F)C1)N1CCC(O)(CCNC(C2CC(O)C2)=O)C1 Nc1c(C(=O)NC2CC2CNC(c2csc3cncn23)=O)cc(F)cc1Cl c1(C(=O)NCC2CN(C)C(C)(C)C2)cccc2cccnc12 c1(CC(C)NC(=O)CCNC(c2cscc2Br)=O)ccccc1F C(CC(N)=O)(C(=O)NC1(c2ccccc2)CC1)NC(C=Cc1ccc(C)o1)=O c1(CN=C(NCC(C(=O)OCC)(F)F)NCC(C)C)nccc2ccc(OC)cc12 C1(OC(C)C)CCCN(C(C2CC3(C2)CC3NC(=O)CCCN(C)C)=O)C1 C1(CC=C)(NC(C2CC2(F)F)=O)CCCN(C(=O)CC(C)C2CCCC2)C1 C1(C(N2CC(C(C)NC(c3cnsc3)=O)OCC2)=O)CCc2nnc(O)n2C1 CN1CCC2C(CCN2C(C2CC(NC(=O)CC3CCOC3)C2)=O)C1 c1(C(=O)NCCOCCCNC(C2C(N(C)C)CCC2)=O)cncc(O)c1 c1(OCC(=O)N(C)CC2CCCC2NC(=O)COCCCC)ccc(Cl)c(F)c1 C12(NC(=O)CC3CC4(CCC4)CCO3)CCCCC1N(C(c1csnn1)=O)CC2 C1(NC(=O)C2=CCCS2)CCC2CN(C(C3C4(CC4)C34CC4)=O)CC2C1 C#Cc1ccc(C)c(NC(=O)C(CC(C)C)N(C(=O)CC(O)C(C)C)C)c1 C1(C(=O)NCc2ccc(C)nn2)(COC)C=CCN1C(=O)CC1C(C)(C)C1(F)F c1(C(=O)NCC(C)NC(c2cc(OC)ncc2)=O)coc2c(F)cccc12 C(=O)(CCCCCc1ccsc1)OC(C)C(=O)N1CC(N(C)C)C1 CC(CNC(=O)C(F)(F)c1ccc(Br)s1)(Cn1cccn1)NC(=O)C1CC1 CCCC(CNC(C1(C)CC(=O)N(C)C1)=O)C(=O)NCCc1ccnc(O)c1 c1(NC(C2(O)CCN(C(COCCSCC)=O)C2)=O)ccc(OC)c(Br)n1 C1(C)(C(=O)NCCN(C(c2c(C)n(CC(C)(C)O)nc2)=O)C)CCCCC1C c1(C(N2CCCN(C(=O)C=CC(F)(F)F)CC2)=O)csc(=NC2CCCCC2)[nH]1 c1(CC(=O)NC2(C(=O)NC(C3CC3)C3CC3)CC(F)C2)cncnc1O c12ccc(cn1)C(=O)N1CCC(O)(C1)CN2.c1(C2C(C(=O)OC)C2)cccc(Br)c1 Cc1nnc2n1CCC(C(=O)NCC1C3CCCC1N(C(c1cc[nH]c1)=O)C3)C2 C=CC(CCC)CC(=O)N(C)CC1(O)CCCN(C(=O)CC2CC(=C)C2)C1 N1(C(CCC2C(C)(C)C2)=O)CCC(NC(c2cnc3[nH]ccnc2-3)=O)CC(O)C1 N#Cc1ccccc1CNC(=O)CC1C(NC(C2OC3CCC2C3)=O)CC1O C1(CNC(C(C)NC(C)=O)=O)CCCCN(C(C2COC(C)C2)=O)C1 Cc1nnc(CCC(=O)NCC(C)(C)NC(=O)C(C)CC2CC2)n1C CON(CCC(=O)N(CCCC(=O)NO)C)C(=O)c1sccc1C c1(C(N2C3C(NC(C(CC)O)=O)C(CC3)C2)=O)coc(=O)c2ccccc12 N1(C(CC(CC=C)NC(=O)C(C)N2CC(C)C2)=O)CCC(F)(F)C(F)C1 S(=O)(=O)(c1cccs1)N1C(NC(N(C2C(C)COCC2)C)=O)CC(O)C1 C1(NC(CCOCC#C)=O)CCC12CN(C(c1ccc(C)nc1C1CC1)=O)C2 C(CCCCC(=O)N(CC(C)COC)C)N(C)CC.C12CC1COC2=O C12CCCN(CC1)C2=O.CCC(CC1CCCC1)C(=O)NCC(=O)NCC(F)(F)F C12(C(=O)NC(CCNC(CCCCOC)=O)C)CCCN1S(=O)(=O)CC2 C1(NC(Cn2ccc(C(C)C)n2)=O)CCN(C(C2CCCOCC2)=O)C1C1CC1 C1(C(=O)NCC#CCNC(C2(CC)CC2)=O)CCc2nn[nH]c2C1 C(=O)(C1=CC2(CCN(C(c3sccc3C#N)=O)C2)C1)NC(C)Cc1ncn(C)n1 c1(CNC(c2csc(C(=O)NCC3CCCCO3)n2)=O)ccc2nccnc2c1 c1(CC(=O)NCC(C(=O)N(C)CCc2ncon2)N(C)CC)c(C)cnn1C CC(CCNC(c1ccoc1CNC(=O)CN1CCC(F)CC1)=O)CCO C(C(C)(C)N=c1ccc(Cl)c(Cl)[nH]1)OC(C)(C)C C1(CNC(C=C2CCC(C)C2)=O)CC12CCN(C(=O)C(C)(C)C(C)(C)C)CC2 CCCCCC(CC)C(=O)NCc1ccsc1C(=O)N(c1ccccc1)C C(C(C(=O)NCC(C)(C)C1CCOC1)NC(=O)Cc1ncccn1)SCC c1(C(=O)NC2CN(C(COC)=O)C(C)C2)ccc(=NCCOC)[nH]c1 c1(C(N(C(C)CN(C)C(C2(n3cccn3)CC2)=O)C)=O)cnn(C)c1Cl N1(C(CC2(OC)CN(C(C(COC)N(C)C)=O)C2)=O)CCSC2(CCC2)C1 c1(C(=O)NCC2N(C(C(CSC)O)=O)CCCCC2)cc2c(ncn2C)[nH]1 c1(C(C(C)NC(=O)Cn2cnnc2)NC(=O)CCOC2CC2)ccccc1 c1(C(N(CCCCNC(=O)CC2COCCN2C)C)=O)noc2c1CCCC2 c1(NC(C#C)(C)C2CC2)ccc(C(F)(F)F)cc1Cl Cc1ncc(Cl)c(C(=O)NCC2CC(NC(=O)C(c3ccccc3C)=O)C2)n1 N1(C(C(CCC)NC(C)=O)=O)CCC(F)(CNC(c2cc(COC)no2)=O)CC1 CCC(CC(=O)N1CCC(O)(CNC(=O)CC2(CS(C)(=O)=O)CC2)C1)OC C(=O)(C(C(C)(C)C)C1CCCC1)N1CC2C(CNC(c3c(C)ncn3C)=O)(C2)C1 N1(C(C(C)(C)SC)=O)CCCCC(CNC(=O)CC(C)C)CC1 N1(C(CC2(C)CC2)=O)CCOCC(NC(C2CCCCC2)=O)C1 C1(CNC(C2CC(N(C)C)C2)=O)CN(C(c2csnn2)=O)C2CC12 CN1CCC(C(=O)NCCC2CCC3CC23)(NC(=O)CCC2OCCO2)C1 C(CC(C)C)(C(=O)N1CCCC(OCC2CC2)C1)NC(COC)=O.C1C(=O)N1 Cc1cc(C)c(CNC(CN2CCCC2)C(C)(C)C)cc1C c1(C(=O)NCC(CN(C(C=C(C)C(F)F)=O)C)C)cccc2c1C(C#N)C2 C1(C(=O)NC2CN(C(CCOCCN(C)C)=O)CC2F)CN(C)CC12CC2 C(N=c1nc2sccc2c(NCCc2cc[nH]n2)[nH]1)C1(SC)CC1 C1(CNC(C(CC)(C)CC)=O)CC2CCC(C1)N2C(c1sc(C(C)C)nc1C)=O C1(CNC(c2c(CC)oc(C)c2)=O)CCN(C(=O)CCc2cccs2)C(C)C1 C1(CC(=O)NCC(C(=O)NCCc2cn(CC)nc2)N(C)C)CCNC(=O)C1 CC(c1ccco1)=CC(=O)NC(CC(=O)NCC1CC1CO)C1CC1 c1(C(=O)NC(CC)(C)CNC(=O)Cc2ccns2)cnc2ncnn2c1O c1(-c2ccc(SC)cc2)ccc2c(C(=O)N(C)CCSC)nsc2c1 C1(CNC(CC=CCC)=O)CN(C(C2CC(F)(F)C2)=O)C2CCCC2O1 c1(C(=O)NC2CC(NCc3cnc(F)c(F)c3)C2)cc(F)c(F)cc1Br CC1(C)CCN(C(C2(F)CCCCC2)=O)CCO1.C1(=O)C2=NOC(C2)CN1 c1(OC)cc(C)ccc1C(=O)NC1CN(C(c2[nH]c(C)cc2C)=O)CCC1CO c1(NCCC(C(C)C)NC(c2cn(CC)nc2)=O)ncnc2ccsc12 N1(C(CC=C=C)=O)CCN(CC(=O)NCC2CC23CC3(F)F)CC1 Cc1ccc(C(N2CC(NC(=O)Cc3cc(Br)cs3)C(O)C2)=O)nc1C N1(C(c2c(OC)ccs2)C(=O)NCc2nnn(C)n2)CCC12CCCOCC2 Cc1c(Br)sc(Br)c1C(=O)NC1C=CCN(C(=O)C=CC(C)(C)C)C1 C1(CNC(C(F)=CC)=O)CN(C(c2[nH]nnc2C2CC2)=O)CC1C C1(CC)CN(C(c2ccc(C)o2)=O)CCC1OCC(=O)N1CC1 C(=O)(C(F)(F)C(F)F)N(C(C)(C)CC(=O)N1CCC(N2CCC2)CC1)C CC1CC(C(N2CC3(CCN3C(=O)CC3SCCO3)C2)=O)CC(=O)N1 N1(C(CC(=C=C)C)=O)CCC2CCN(C(c3cc(SC)oc3C)=O)CC12 c1(CC)[nH]c(C(N2CCC(N(C(=O)C(C)C(F)F)CC(C)C)CC2)=O)nc1Cl c1(CNC(CSC)C2CCC2)coc(-c2cnn(C)c2)n1 c1(C(N(C(CCNC(C2(CC#C)CCCO2)=O)C)C)=O)ncnc(C)c1OC N1(CC(=O)N(C2CCC(NC(=O)CO)C2)C)CSCCSC1 C1(CC2(O)CC(OC)C2)CC(C)CN1C(=O)CN(CC(C)(C)C)C c1(C(=O)NCCN(CC(C)O)C(C2CC3CCC(C2)O3)=O)nc(O)nc(O)c1F C(=O)(C1CCCc2ccnn21)N1C(CNC(c2nc(Cl)c(Cl)s2)=O)CC(F)(F)C1 N1(C(=O)NC(CC)Cc2ccccc2Cl)CC(c2ccccc2)OC(C)(C)C1 c1(C(=O)NC(C)CN(C)C(C2(Oc3ccccc3)CC2)=O)coc2c1CSC2 C(=O)(n1cncc1CN1CCCC(C(=O)NCCCCCO)CC1)NC(C)C C(=O)(CCCC(F)(F)F)N(CC(C)NC(=O)C(C(C)C)OC)CC N1(C(C)C)CCCN(C(=O)C(CC2(C)N=N2)N(C)C)CC1 N1(C(CC=C=C)=O)CCN(C(C2CCCN(C(C)C)C2)=O)CC1CC(C)(C)C c1(C(C)C)c[nH]nc1CNC(=O)CCOCCN(C(=O)C(C)n1cccc1)C N1(C(Cc2n(C)cnn2)=O)CCCC(NC(c2cnn(CC(F)F)c2C2CC2)=O)C1 c1(N2CCC(NC(c3nccnc3N)=O)C(O)C2)ncnc2c1nnn2C=O.C1CC1 Cc1nnc(O)c(C(=O)NCC2(C)CN(C(=O)C(C)C3=CCCC3)CCO2)c1C c1(NCC(CC)C(C)C)[nH]c(=NCCN2CCOCC2)nc2c1ncn2C CC(C)(C)CC(C)(C)C(=O)NC1CCC1NC(=O)CNS(C)(=O)=O c1(NC2(C3CCN(C(c4cc(Cl)c(Cl)[nH]4)=O)CC3)CC2)ncc2cccnc2n1 N1(C(c2[nH]cc(C)c2)=O)CCCC(O)(CN(C(=O)C=CCF)C)C1 CCCCCNCCC(=O)NCCCCNC(CCN(C)C(c1cccs1)=O)=O C1(C(N2CC(COC)(NC(c3ccsc3OC)=O)C2)=O)CC(C(C)=NO)C1(C)C C1(NC(C(c2cccc(OC)c2)O)=O)CC2CCC(C1)N2CCCCF C=CCC(CC(=O)N(C)Cc1ccncc1)NC(=O)Cc1sccc1C C1(NC(c2n(C)ncc2)=O)CC2CC(C1)N(C(c1cc3ccsc3[nH]1)=O)C2 N1(C(=O)OCC)CCC(C)N(C(=O)Cc2ccco2)CC1.C1CCC(=O)O1 Cc1cccc(C)c1C(N1CCCC(C(=O)NCC2(O)CCC2)C1)=O c1(CC(N2CC(NC(CN(C(C)=O)CCO)=O)C3C2C3)=O)cc(C)ccc1O c1(C(=O)NCCN(C(C2N(C(C)C)CCCC2)=O)C)nsc2ccccc12 C1(C(N(OC)C)=O)C=CCCN1C(C1CCC1)=O N1(C(C=CCCC)=O)CCCC2(C1)CN(C(=O)CCc1nnc(S)n1C)CCO2 Cc1[nH]nc2ccc(C(=O)NCC3(C)CCN(C(=O)C(=O)N=S(C)(C)=O)C3)cc12 N1(C(C(C)NC(c2ccc(F)cc2)=O)=O)CCC(O)(CNC(c2cncn2C)=O)C1 C(=O)(CC(CC(C)C)ONC(C1(OC)CCCC1)=O)NC(=O)CC#N c1(CCN2CCC(N3CCN(C(C(C)CC4CC4)=O)CC3)C2)ccc(Cl)cc1Cl C(=O)(CCCCC(=O)NC1CCOC1CC1CCC1)OC.C12(CC1)C(=O)NC2 c1(OC)ccc(N)c(C(=O)NCC2(C)CCN(C(C3C(C)(C)C3(F)F)=O)C2)c1 c1(C(=O)NCCC(C)N(C(COCCCC)=O)C)cccc(C2CCOC2)c1 CCC(C)(O)C(=O)NCCCCCNC(=O)CC1CCOC(C(C)C)C1 c1(CNC(COCCNC(C(C)c2cc[nH]n2)=O)=O)ccccn1 CCC(C)(C(c1nnnn1C(c1ccccc1)c1ccco1)NCCCF)OC c1(NC)ccc(C(N2CC3C(CNC(=O)CCc4cn(C)cn4)C3C2)=O)cc1F Cc1cc(C(=O)NCC(c2ccccc2)NC(=O)C(C)N(C)C)c(C)nc1C C(=O)(CCC(C)(C)[N+](=O)[O-])NCC1CN(C(C2ON=C(C)C2)=O)C(C)(C)C1 c1(OC)ccc2c(c1)C(C(C)C)N(C(C1(c3ccccc3C#N)CC1)=O)CC2 N1(C(C(C)Cc2ccco2)=O)CCOCC(F)(CNC(c2nnn(C)n2)=O)C1 c1(C(N2CCC(N(C(CC=C=C)=O)CC)C2)=O)c[nH]cc(Br)c1=N c1(C(=O)NC2C3CN(C(C4(C)N(C)CCC4)=O)CC2C3)cscc1S(C)(=O)=O C1(n2cc(CN(C(C(CC(C)(C)C)c3ccccc3)=O)CC)nn2)CCCNC1=O N1(C(c2c(OCCC)nccc2)=O)CC2CCC(C1)N2c1nc(C)nc(=N)[nH]1 C(=O)(CC(C)(C)C(F)F)N(CC(=O)NCC(=O)NCCC)C Cc1nc2ccccn2c1C(=O)NC(C)C(CO)NC(=O)C(CN(C)C)C1CC1 c1(OC)ccc2oc(C(=O)NC3CCCC3NC(=O)CCNC(C)C)c(C)c2c1 Cc1cc2ncc(C(N3CCN(C(c4cc(C)c(Br)cn4)=O)CC3)=O)cc2[nH]1 C=CC(F)(F)C(=O)OC1CC(c2ccccc2F)(C(=O)OC)C1 C(=O)(CC(C)C(C)(C)NC(c1cnc(C)nc1C)=O)NC(C=C)C CC(C(=O)N1CC(C(C(N2CCC2(CO)CO)=O)N(C)C)C1)C(F)F C1(NC(=O)CC(O)Cc2ccccc2)COCCN(CCn2ccccc2=O)C1 N1(c2cc(NCCc3cccc(Cl)c3)nc(COC)n2)CCN2CC(C)CC2C1 N1(C(C2N(C(CN3CCN(C)CC3)=O)C3C(C2)C3)=O)CC2CCCCC12 c1(C(=O)NCC(CN(C)C(C2(C)CCOC2)=O)O)cnc(N)cn1 N1(c2nc(C)c(F)cn2)CCC2(CCN(C(=O)C3=CCCC(C)(C)C3)CC2)CC1 N1(C(CNC(CCC)=O)=O)CCCC(F)(CNC(c2csc(C3CC3)n2)=O)C1 C(=O)(C(CCCOC)NC(=O)Cc1nocc1C)NCc1ccn(CC)n1 N1(C(C(C)C)=O)CCC(CO)C(NC(=O)Cn2cc(F)ccc2=O)C1 C1(N=[N+]=[N-])(C(N2C(CSC)CCC2)=O)CCN(C(=O)Cc2cnc(C)s2)C1 c1(OC)cnc(F)c(C(=O)NC2CC(NC(c3[nH]ccc3C3CC3)=O)C(O)C2)c1 C(=O)(C(F)C(F)(F)F)N(C1CCN(C(=O)C(CCSC)NC=O)CC1)CC#C CON=C(C(=O)NC1COCCN(C(=O)Cc2cccc(F)c2O)C1)c1ccco1 c1(CN2C3CN(C(=O)Cc4cccnc4Br)CC2CC3)cc(O)ccc1[N+](=O)[O-] c1(CC)cc(C(=O)NCCCOCCNC(=O)CC2CCC2(C)C)c(C)o1 c1(C(=O)NC(CC(C)NC(c2cc(C)[nH]n2)=O)C)cnc(C(F)(F)F)c(C)c1 C1(C(=O)NCCN(C(CNS(CCOCC)(=O)=O)=O)CC)CCC2CCC12 c1(C(N2CC(CN(C(C(C(C)O)(F)F)=O)C)C2)=O)nc2ccccc2nc1O c1(NC(=O)NC(c2nnc(C3CCCOC3)o2)C)cccc(-c2nc(C)no2)c1 N1(C(C2(CC#C)CC2)=O)CC(CNC(=O)C(c2ccc(OC)cc2)CF)CC1C c1(NC(N(CC(c2ccc(Br)cc2)O)C)=O)cc(Cl)c(F)cc1C#N C(C)(C)(CC(=O)N(CC(C)(C)CNC(C1CC1(C)C(F)F)=O)C)OC C1(CC)(NC(c2c[nH]ccc2=O)c2nnnn2-c2cccc(Cl)c2)CC(C)(C)C1 c1(OC)ccc(NC(c2ccn(CCNC(C3CCCSC3C)=O)c2)=O)c(F)c1 C(=O)(C(CC)C(=O)NC1CCC1NC(c1ccc(Br)cc1C)=O)OCC N#Cc1ccccc1OCCNCc1c[nH]ccc1=O.C12CC(C1)NC(=O)N2 c1(CC)nc(=N)[nH]cc1C(=O)NCCC(C)NC(C1CC1Br)=O CCC(CNC(=O)C(C(C)CC)NC(C)=O)N=c1[nH]c(Cl)ncc1C(C)C CC1OC2(C(=O)NC3CC(CNC(C4(C)CC(F)(F)C4)=O)C3)CCC1C2 Cc1c(C(=O)NC(C)CC(C)NC(=O)C(O)C2CCCC2)sc2cccc(F)c12 CC1CC(C(=O)O)CC(C)N1C(C1COCC(=O)N1Cc1ccccc1)=O CCC(C)(C(=O)OCc1cn(C)nc1-n1cncn1)OC CCC(CO)CN=c1[nH]c(=NCCCCCCSC)[nH]c2c1CCC2 c1(CC)ocnc1C(=O)NCC1CC1CNC(c1cnn(CC)n1)=O N1(C(c2cc(C)c(C)[nH]2)=O)CCC(F)(CNC(c2cccc(C)c2O)=O)CC1 c1(NCC(=O)NCC(CNC(C2C(C=C)C2)=O)O)ccccc1[N+](=O)[O-] N1(C(C(C)NC(c2ccsc2Cl)=O)=O)CCCN(C(=O)COC2CCCC2)CC1 C(C1CCCn2ccnc21)NCC1C(C(C)(C)C)OCC1 NC(C(=O)NNC(=O)C1CC=CC1)C1(O)CN(C(=O)OC(C)(C)C)C1 C1(c2c(C)n(C)nc2)C(NC(c2csc(OCCF)n2)=O)CC(=O)N1C c1(CN2CCC(O)(C(=O)NC(C)CN3CCCCC3)CC2)cccc([N+](=O)[O-])c1 C1(CC(=O)NCC2C(NC(CC=C)=O)C2)COC2CC1C2 C(CC(=O)N1CCN(C2CC2)C(=O)C1)(C(F)F)NC(C1(C(C)=O)CC(=O)C1)=O c1(C(=O)NC2COCCN(C(C3(O)CCOCC3)=O)C2)ccn2c1CSCC2 c1(C(C)C)ncc(C(=O)N(C2CCCC2)CCNC(=O)C(C)(O)C2CCC2)cn1 c1(OC)cc([N+](=O)[O-])ccc1C(N1CCCC(CN(C)C(c2cnns2)=O)C1)=O N1(C(C(C)(C)SC)=O)CCN(C(c2nc3c(s2)COCC3)=O)CC(C)(F)C1 c1(C(N(C)Cc2ccncc2)=O)coc2c1CN(C(=O)COC1CCCCC1)C2 C(=O)(C1=CNC2=NCCCN12)NCC1(C)CCN(C(C(C)OCC)=O)C1 c1(C(=O)NC(C(C)C)CNC(=O)C(F)CC2CCC2)cn2c(n1)SCC2 N1(C(CCC2OCC(C)(C)C2)=O)CC(CNC(=O)C(F)C2CCC2)C2(CC2)C1 N1(C(c2nc(CCC)oc2)=O)CC(O)CC1CNC(C1(C(F)(F)F)CCC1)=O N(C(=NCCC1CC1)N1CCC(S(C)(=O)=O)CC1)Cc1c(OC)cncc1OC CCCC(C(=O)NC1(C(=O)NCC=Cc2cccnc2)CCCCC1)NC(C)=O C1(C2CC2)(CC(N2CC(CCNC(C3(C(F)F)CC3c3ccccc3)=O)C2)=O)CC1 Cc1cc(=O)oc(C)c1C(=O)NCC(CNC(=O)CSCC(F)(F)F)S(C)(=O)=O CC(C)CC(C(N)=O)NC(=O)CC1(CN)CCC1.C(S(C)(=O)=O)C1CC1 C1(C(=O)N)CCCCC(=O)N1.CC(C(=O)N)N(CC=CCCCOCC(F)(F)F)C O=C(C1=NOC(C(F)F)C1)N1CC2(CO)CC1(CNC(C1(C3CCC3)CC1)=O)C2 c1(C(N2CCC(O)(CNC(c3c(CC)cco3)=O)CC2)=O)ccc(C)c(C#N)c1 CCC(O)C(=O)NCCCN(C(=O)C(C)C1CC1)CC c1(C(=O)NC(C)(CNC(C2CC=CCO2)=O)C2CC2)cc(C(F)(F)F)ncc1Cl c1(NC(c2c(CNC(C(C(CC)C)C)=O)occ2)=O)ccn2nccc2c1 N=c1[nH]c(C2CC2)ncc1C(=O)NC1CC(CNC(c2csc(C3CC3)n2)=O)C1 CCC(CC)C(C)C(=O)NC(CNC(=O)Cc1cc(C)on1)C(C)C C(C(=O)NNC(=O)C(=O)NCc1ccc(F)cc1)(C1CC1)NC(C(C)(C)CC(F)F)=O Cc1nc(C(=O)NCCCOCCNC(C2CC2c2ccncc2)=O)c(C)n1C O=C(C(O)CCNC(C12COCC1C2)=O)NC12CC(C1)C2 c1(C(=O)NC2C(OC)CN(C(c3cnc(C)s3)=O)C2)ccc(Cl)c2occc12 Cc1cc(Cl)ccc1OCC(=O)NCCCC(C)NC(c1csc2nnsc12)=O N1(C(C(C(CC)O)C)=O)CC2CCCC(C1)N2C(c1cc(C)ccc1SCC)=O C=CCC(C)(C)CC(=O)N(CCCNC(c1cc(C(F)F)ncn1)=O)C C1(CCNC(CCc2ccn(C)c2)=O)CCCN(C(=O)Cn2[nH]cnc2=N)CC1 C1(NC(C(C)C2CCC2)=O)CC2(CCN(C(c3c(C#N)cnn3C)=O)C2)C1 c1(C(=O)NCCCNC(COCCCC)=O)ccc(C(C)=O)n1C N1(C(CCCOC(C)=O)=O)CC(CNC(=O)C(C)Cc2cccc(Cl)c2)C2(CC2)C1 O=C(C1Cc2ccc(F)cc21)NCC1CCCCC1NC(C1CC1F)=O c1(C(N2CCC(CCNC(=O)COC3CCOC3)C2)=O)cc2ccnc(Cl)c2[nH]1 CC(C)C(O)C(=O)N1CCC(O)(CNC(c2cnn(C(C)C)c2Cl)=O)C1 C1(OC)(CNC(=O)CCSCC2CCCC2)CCN(C(C2CC2C#N)=O)C1 N1(C(COC)C)CCC2(CC1)CN(C(=O)CC1CCN(C)C1=O)C2 c1(COC)ccc(C(N2CC(=C(F)CNC(c3cc(CF)on3)=O)C2)=O)o1 c1(C(=O)NCC2(OC)CCN(C(C(COC)(C)O)=O)C2)c(N(C)C)cccc1F N#Cc1cncc(NCCc2c(F)cccc2Cl)n1 C(C)(c1ccc(F)cc1F)=CC(=O)NC1C2CCN(C(COC(CC)(C)C)=O)C21 C(=O)(N=c1cc(C)n(C(C)C)[nH]1)C1(C)N(C(c2c(CC)cns2)=O)CCC=C1 c1(C(N(C2CN(C(=O)Cc3ccc(O)cc3)C2)C)=O)ccc(NS(N)(=O)=O)cn1 C(C(=O)NCC=CCC(=O)NC1(CCOC)CC1)(C(C)C)SC N1(C(c2cc(C(C)C)[nH]n2)=O)CC2CN(C(=O)CC(O)C3CCCC3)CC2C1 CCCCCCCC(=O)NC1C2CC3C(C2)C13C(=O)NC(CC1CC1)C1CC1 N1(C(CCCC(=O)N2C(C)CC(Nc3ccsc3)C2)=O)CCCN(C)C(=O)C1 C1(NC(C(C)(O)C2CCC2)=O)CCN(C(C2CN(C3CCCCC3)C2)=O)CC1F c1(NC(C(C2CN(C(=O)Cc3cnn(C)c3O)C2)OC)=O)cccc(F)c1O c1(C(N2CCC(C)(CNC(c3c[nH]c(Br)c3)=O)C2)=O)cn2ccccc2n1 c1(OC)cc2c(cc1OC)CN(c1nc(C)cc(=NCc3n[nH]c(=N)s3)[nH]1)CC2 C1(N=c2cc(Cl)c(O)n[nH]2)(CCNC(CC2(OC)CCC2)=O)CCC1 c1(C(=O)NCC(CO)NC(c2nc(C(F)F)cs2)=O)cncc(OCCF)c1 c12cc(nc(C)n1)N2.c1(C(=O)OC)nc(CN2CCC2(C)N(C)C2CC2)cs1 C(CC(C)C(=O)N(C1(CNC(=O)COc2ccc(Cl)cc2)CC1)C)=CC C1(C#N)(NC(Cc2ccc(SC)cc2)=O)CCN(C(=O)C(O)Cc2ccccc2)C1 c1(CNC(C2CC3CCC(C2)N3Cc2nc[nH]n2)=O)ccc(Cl)c(C#N)c1 N1(C(Cc2cc(C)on2)=O)CCC2(CNC(=O)C(C)C)CCCCC12 c1(CC)onc(C(=O)NCC2(NC(C3CC3C)=O)CCCC2)c1C c1(CCCNC(C2CC2c2cccs2)C)ccccc1F Cc1cc(C)n(C(C)C(=O)NCC2CCN2C(=O)CCn2ccccc2=O)n1 C(=O)(C1CCCc2sc(NC(=O)CCSc3ccccc3Br)nc21)OC C(CC(O)(CC)CC)NC(CNC(CNC(C1C(C(C)C)OCC1)=O)=O)=O C(=O)(CCCC(=O)NCC(CO)NC(c1ccnc(SC(C)(C)C)c1)=O)N(C)C c1(OC)ccc(C(N2CC(NC(c3c(C)csc3Cl)=O)C(F)C2)=O)cc1OC N1(c2nccc(OC)n2)CCCC(N(C)C(c2n[nH]c(C)c2Br)=O)CC1 C1(C(=O)NCC2N(C(=O)C(F)CC3CCCCC3)CC2)CCC2CC2CC1 C1(C(N(CCCNC(=O)C(c2ccnn2C)C)CC)=O)COCCN1C=O c1(CN2CC(C(N=c3cc(OCC)o[nH]3)=O)OCC2)cc(O)c(O)c([N+](=O)[O-])c1 C(C(C(=O)NC(C)(C)CNC(C1(F)CCC(C)CC1)=O)C(C)(C)C)OCC=C c1(NC(=O)OC(C)(C)C)cc2ccncc2[nH]1.C(CCC1C(=O)N1)OC N1(CC(=O)N(C)C(c2cnsn2)=O)OC(C)(C)CC1=O.C12C3CN(CC13)C2 CC1CC(CNC(=O)Cc2cnsc2)CN1C(C1CC12CC2)=O S(=O)(=O)(CCCCS(=O)(=O)N1CCOCC1)NC(CCC(C)=O)=O c1(C(N(C(Cc2cn(CCCF)nn2)CC(=O)O)C)=O)cc2ccc(O)nc2s1 c1(COC)ccccc1CNC(=O)CC1CN(C(c2cc(F)n(C)n2)=O)CCO1 N1(C(C(C2CC(CC)C2)NC(=O)Cc2scnc2C)=O)CCN(C2CC2)CC1 c1(-n2c(N(C3CC3)OC(C3(C)CC(=C)C3)=O)nnn2)ccc(C(F)(F)F)c(F)c1 N1(C(CCOC)=O)CCCC1(C)CCNC(=O)C=Cc1cc[nH]n1 C1(C(N(C2(C)CC2(C)C)C)=O)CCC(C)(C)N(C(=O)CCC2CC(N(C)C)C2)C1 Cc1nn(C)cc1CC(=O)NCC12CC1CN(C(c1cc(Cl)ccn1)=O)C2 C1(C(=O)NC(c2ccccc2F)CNC(C(C#C)(C)C)=O)CN2CCN1CC2 c1(CC)ccc(C(=O)NCCN(CCOC)C(C2CCCC2C)=O)cc1Cl N1(C(c2c(C)nsc2)=O)CCC2(CCCCN(C(=O)CCC3CCCO3)C2)C1 C1(NC(C2CC(C)(C)C2)=O)CCSC12CN(C(=O)CCSC(F)(F)F)C2 c1(OC)c(C(=O)NC2CN(C(c3ncc(Cl)nc3Cl)=O)CC2C)nc(O)nc1O N1(C(CCOCC#C)=O)CCC(CCOC)(CO)C1.c12conc1NC2=O c1(OC)cc(F)c(CN2CCC(N3CCC(F)(F)CC3)C2)cc1Cl C1(C2CC2)(NC(C(C(C)(C)O)F)=O)CCN(C(=O)CCCS(N)(=O)=O)C1 C12(CNC(C3CC(C)OCC3)=O)CCCC1N(CCC(C)F)CCC2 N1(C(c2cccc(C(N)=O)c2)C(=O)Nc2ccc(Cl)cc2)CC2CS(=O)(=O)CC2(C#N)C1 C1(CC)CC(C(=O)NC(C)CCN(C)C(C2CN(c3nncs3)C2)=O)C1 c1(C(N(C(C(=O)NC(CC=C)(C)CC=C)C)CC2CC2)=O)cccc2[nH]ccc12 c1(C(N(CCC)CCNC(=O)Cc2csc(C(F)(F)F)n2)=O)cccc(O)n1 N1(C(c2c(C)n(C)cn2)=O)CCC2(CC2NC(C2CC3CCC2CC3)=O)C1 N#Cc1nccc(NCCC2CCCN(C(=O)Cn3ccccc3=O)C2)n1 Cc1cc(O)ccc1NC(=O)C(C1CCCN(C(c2ccnn2C(F)F)=O)C1)C C12(NC(c3cc(C)sc3C)=O)CCC(C1)N(C(c1ccc(C3CC3)cc1)=O)C2 c1(C(N2C(COC)CN(C(=O)COC3CCC3)CC2)=O)cnn2cccnc12 Cc1cc(C(N2CCC(NC(=O)C(=O)N(C)C)C2)=O)c2c(C)nn(C)c2n1 C1(NC(c2cc(C(=O)NCCOCC#N)no2)=O)CC(=O)N(CC2CC2)C1 C(C)(C)(C(C)CC(=O)NCc1ncccn1)NC(C(CC=CCC)C)=O c1(OC)ccc2c(c1)OCC(C(=O)NC1CC(NC(=O)CC3CC34CC4)C1)=C2 N1(CC(C)C(=O)NCc2nc(C3CC3)n(C)n2)CCC(C(N)=O)(C(=O)O)CC1 Nc1cc(F)cnc1C(N1CC(C(O)C(=O)NC(CO)C(F)F)C1)=O c1(C(=O)NC(C)C(=O)NCCc2cc[nH]n2)cc(O)cc(=O)o1 N1(C(CNS(CC)(=O)=O)=O)CCN(C(C2(C#N)CCCCC2)=O)CC1CF CCC(CNC(c1nnnn1CCOCC)C(C)C1CC1)(CC)CC n1(CC)nc(C)c(Cl)c1CN1CC2C(C(N3CCCC3C3COCCO3)=O)C2C1 O=C(C1=CCOCC1)N1CCC(NC2CN(C(C3(CO)CC3(F)F)=O)C2)CC1 c1(OC)cncc(CCC(=O)NC2CC(O)(CNC(=O)Cc3nccn3C)C2)c1 C(=O)(CC(=O)OC(C(=O)N(C(CCC)C)C)C)NCCNC(C)=O CCC(O)(C(=O)N1CCOC(CNC(=O)COc2cnn(C)c2)C1)c1ccccc1 C1(CCNC(C(C)NC(=O)NC)=O)COCCN1C(c1ccccc1N(C)C)=O N(C(=NCc1c(Br)cnn1C)NC1CCN(C2CC2)CC1)C(CC)C C1(C(=O)Nc2ccc(CC)nc2)CN(C(=O)CCc2ccn(C)c2)CC12CC2 Cc1cccc(C)c1CC(=O)N(C1CCCCC12CC2)CCNC(=O)C(C)C(F)F CCCCCC(O)C(=O)NCC1(NC(C2OCCC2C)=O)CCC(F)(F)CC1 Cc1ccc(C)c(OCC(N2CCC2CNC(c2cc(F)cs2)=O)=O)c1 C#CC1(C(N2CC3(CCC3O)C2)=O)CCN(C(=O)C(C2CC2)SC)C1 C1(NC(CS(CC)=O)=O)CN(C(c2cc3c(nn2)CCOC3)=O)CC2CCCC12 c1(SC)nc(=NCC2CCCCN2C(=O)CCC(C)N(C)C)s[nH]1 CCC(COC)C(=O)NC12CC1CN(C(c1cnc(C)s1)=O)C2 CC1CN(C(c2occc2F)=O)CCC1NC(=O)CCCCN(C)C C(C(=O)ON1CCOCC1)(C(C)C)NC(CCCOCC)c1nnnn1C(C)C c1(OC)c(C(=O)NCC(C)NC(=O)C(C)OC2CCCC2)cccc1F c1(NC(=O)NC2CCCC2C(F)(F)F)nccc(SC2CCCO2)n1 c1(NC(C)=O)ccc(C(=O)NCC(CC(F)(F)F)NC(=O)C(C)O)c(F)c1 C(CCC(C(=O)N(CCCCO)C)NC(=O)COC1CCC1)OC C1(N(CCC)C(c2cc(C)co2)=O)CCN(C(C2CCC=CCC2)=O)CC1 Cc1ccc2cc(C(=O)NC(C)CNC(C3(C#N)CCCCC3)=O)cn2c1 C1(C(N2CCOCC(NC(CCP(C)(C)=O)=O)C2)=O)CCC2(CC1)CC(O)C2 N1(C(C23CCC(C)(CC2)OC3)=O)CCC2(CCCN2C(=O)CNS(C)(=O)=O)CC1 C1(NC(c2c(COC)cco2)=O)COC2(C1)CN(C(c1cnns1)=O)C2 C(CN(C)C(C1(Cl)CC1)=O)(CO)(CO)NC(c1c(CCC)nco1)=O C12(CNC(c3c(CC)nccn3)=O)CCC(CC1)N2C(=O)C=CC(C)(C)SC Cc1cc([N+](=O)[O-])cnc1C(N1CC2C(N(C(=O)C=CC3CCCO3)C)C2C1)=O N1(CCCCN(S(C)(=O)=O)C)C(=O)CN(Cc2ccnc(F)c2)C1=O O=C(N=c1[nH][nH]c2cccnc12)C1CC(F)CN1Cc1ncccc1O C12(NC(C=C(C)C)=O)CCCC1N(C(=O)CCc1csc(C)n1)CCC2 C12(C(=O)NC(Cn3cc(-c4c(C)cccn4)nn3)C)CC3CC1C2C3O Cc1cccc(C(=O)O)c1S(=O)(=O)N(C1Cc2ccccc2CN1)C c1(COC)ccc(C(=O)NC2CCCC2CNC(=O)C(F)(F)c2cnn(C)c2)s1 C=CCC(CNC(=O)C=CCN1CCC1)C(=O)N1CCC2C(O)CC12 c1(C(=O)NCC(c2cccc(C)c2)NC(C2CCCS2)=O)cc2n(c1)CCCC2 c1(C(=O)OC)cc(C)c(C(N2CC(O)CC2CNC(=O)CC2CC3CC3C2)=O)o1 CCC(C)CCCC(=O)N(C)CC1(O)CCN(C(c2cncc(C3CC3)c2)=O)C1 N1(C(CCCOC)=O)CCC2(CC1)CC2CNC(=O)CCc1cc(Cl)no1 Cn1ccc2[nH]c(C(N3CCCC3(C)CNC(C3(C)CCCCO3)=O)=O)cc12 C(=O)(C(F)(F)C(F)(F)F)N(CCOCCCN(C(c1ccc(C)nc1)=O)C)C C1(NC(c2c(CC)nc(C)s2)=O)CCOC12CCN(C(=O)CC(C)(C)C#N)CC2 C1(C(=O)NCc2snc(CC)n2)CCCN1NC(=O)CC1CC(C)=NO1 [SH](=O)(=O)C1(C(=O)NCC2CN(C(C3(CO)COC3)=O)CC2C)CCCCC1 C1(C(N(CCC(=O)NCCc2cnc(C)o2)CC=C)=O)CCCCC1C C(=O)(C(C)CC(F)F)N1CCC(N2CCN(C(CCCC#C)=O)CC2)C1 C1(CCCNC(C(=C(C)C2CC2)F)=O)CCCCN1C(=O)C(C)C1CCCC1 CC(C)CC(CC(C)C)C(=O)NCC1(C(C)NC(C2CC(O)C2)=O)CC1 C1(C(=O)NCCC2(NC(CN3CCN(C)CC3)=O)CC2)COC2(CO)CC1C2 N1(C(c2ccc(CNC(CCCN(C)C)=O)o2)=O)CC2(C)CCC2(C)C1 Cc1nn2cc(C(N3CC(C(=O)N(C)CCc4ncon4)CC(F)C3)=O)nc2s1 c1(CNC2C3CN(C(c4nc(C)oc4)=O)CC32)ccc(O)c(I)c1 N1(C(c2cc(CC(C)C)[nH]n2)=O)CCC(C2CN(C(C3CCC3F)=O)C2)CC1 C1(N(C(C2N(C)CCCC2)=O)C)CC2CC1N(C(=O)CC1(C)OCCO1)C2 Cc1ccc(C(=O)NC(C(=O)NCC2CC23CCC3)C2CCOC2)o1 c1(CC)cn2c(n1)CC(C(=O)N(C)CCN(C(=O)COCCOC)CC)CC2 CCCCCCCCCCC(=O)N1CCCC1CNC(=O)Cn1cccnc1=O C1(CC)CN(C(=O)C(C2CCCCC2)NC(=O)CC(C)SC)CCN1C c1(CCOCC)nc(C(N2CCCC2C(=O)NCCNC(=O)NC)=O)cs1 C(=O)(CCCCC(C)(C)C)NC1CC(C)(NC(COCCCOC)=O)C1 CN(C1CCc2ccc(Br)cc21)C(=O)CCCCCC1CC1 N1(C(C2(F)CC(C(=O)OCC)C2)=O)CCCN(C(=O)C(C2CCCCC2)O)CC1 C12CCCC13CN(C3)C(F)(F)CN2.N1(C(CC)C(=O)OC)C(=O)CCC1=O CCC(C(=O)N1CC(CNC(=O)CCNC(=O)C=CCl)(OC)C1)C1CCOCC1 C1(CN(C(C(C)NC(CC)=O)=O)C)COCCN1C(C1CCCN1C(C)C)=O N1(C(=O)OC(C)(C)C)CC(C(=O)Nc2ccoc2)C2(CC2)C1 C1(CC=C)(NC(=O)COCC(=C)C)CCN(C(=O)C=Cc2ccncc2)C1 c1(C(N(C(C)C(=O)N(CCCC(C)O)C)CC)=O)ccc(O)c(C)c1 N1(C(C2(CN(C)C=O)CC(C)(C)C2)=O)CCOC(C)(C#N)C1 C1(C(=O)NC(CCOC)C)CC(=O)CN1C(=O)Cc1cnnn1C c1(C(N2CC(C(C)NC(c3cnc(C)o3)=O)OCC2)=O)nccc2ccsc12 C1(CNC(C=C(C)C(C)C)=O)C2CCCC1N(C(=O)C=Cc1nccs1)C2 C(C)(CCC(=O)N1CCCC(NC(c2ccccc2SCCO)=O)C1)OCC CC(C)C(C)(C)C(=O)NC1CCN(C(c2csc(-c3ccsc3)n2)=O)CC1O C(=O)(C1=NOC2COCC12)N1CC=CC(C(=O)NCC(C)N(C)C2CC2)C1 Cc1ccc(COC2CCN(C(=O)CCOC(C)C(=O)N(C)C3CC3)CC2)cc1 C(c1cscn1)=CC(=O)NCC(C)(C1CCC1)NC(c1csc(CO)n1)=O c1(CC(C(=O)NC2CCCN(C(=O)C=CCF)CC2)N(C)C)c(F)cccc1F Cc1c(N)ccc(C(=O)NCC2CC(NC(=O)CC3CCOCC3)C2)c1C C1(C(=O)NC(C2CCOC2)C)CCC2(CN(C(=O)Cc3ccc(Cl)c(F)c3)C2)O1 C(=O)(C(CCC)OCC)N1C(C(N(CC#CC)CC#C)=O)CCC1 C(CCCC(C)C)(c1nnnn1Cc1nnn(C)n1)NC(C)CC1CC1 C(=O)(C1=CC(O)C(NC(C2COCC2C(N)=O)=O)C1)NCc1nc(C)sc1C C12(NC(=O)CCc3cnoc3)CCCC1N(C(=O)Cn1cnnc1O)CC2 c1(C(N2CCC(CC=C)(NC(=O)C(C)C)C2)=O)cn(C)cc(Br)c1=O C(=O)(C1=COCCO1)NCCC1CCN(C(c2cc(CNC(C)=O)on2)=O)CC1 n1(CCC(=O)NC2CCCC(NC(Cc3c(C)scc3)=O)C2)c(C)c(C)sc1=O c1(NC(C(=O)NC2(C(=O)OC)CCOCC2)=O)ccc(CS(C)(=O)=O)cc1OC C(CC(C)(C)C(=O)NCC12CC(NC(=O)CC3CN(C(C)C)C3)(C1)C2)OC C(=O)(C1=C(Cl)CCC1)NC1C(NC(Cc2c(C)cco2)=O)CCC1 C1(C(N2C3CN(C(C(C(C)(C)C)CO)=O)CC2CC3)=O)CSc2ccccc2O1 n1(Cc2nc(C(CC)O)nn2-c2cnnn2C)c(=O)sc2ccccc12 CC1CC(NC(=O)COc2cncc(Br)c2)CN1C(C1CCCCCC1)=O n1(CC(N2CC(CC=C)(C(=O)NCC3(OC)CCCC3)C2)=O)nc(C)oc1=O c1(COC)cccc(CC(=O)NCC(F)CNC(=O)C2=NOCC2)c1 N1(CC)CCCC(C(=O)NC2(CO)CCN(C(=O)CNc3ccccn3)C2)C1 C1(C(=O)NCC2CC(NC(c3cnc4n3CCC4)=O)C2)CC2CCCCN2C1 C(=O)(CCCC(=O)N1CCN(C(=O)CNC(=O)C(C)CC)C(CO)C1)OC C(=O)(CC1=CCCC1)N(C1CCCN(C(=O)Cn2ccccc2=O)C1)CC Cc1ccc(CC(=O)NC2COCC2NC(=O)C(c2ccccc2)N(C)C)cn1 Cc1cc(C(N2CCCC2CC(=O)Nc2cnn(CCO)c2)=O)cc(Cl)n1 Cn1nnc2c1CCN(C(C1(NC(C3CC(C4CC4)=NO3)=O)CC1)=O)C2 c1(CC)noc(C(=O)NC(C)(C)CCN(C(=O)C=Cc2ncc[nH]2)C)c1C C1(C(N2C(CCNC(c3c(SC)csc3)=O)COCC2)=O)CC2CCCC(C1)C2 CC1OCC2(CCNCC2)C1N(CC(F)(F)F)C(c1cnn2ccccc12)=O O=C(C1CCc2ccccc21)NCc1csc(Cl)n1 C1(CC)COCCN(C(=O)CC2CCN(C(=O)C(C)CCOC)CC2)C1 Cc1cc(O)nnc1C(N1CCN(CCCNC(=O)C(O)C2CCC2)CC1)=O C(C(C)CC(=O)N1CC2CC1C2CNC(c1ncccc1COC)=O)OC Cc1cccc2c1OC(C(N1CC(C(C)NC(C3CC3(F)F)=O)C1)=O)C2 CC1CC(Cn2cccn2)(CO)C1.C12(CC(=O)NC(c3c[nH]nn3)=O)CCCC1C2 C(C(=O)O)(N=c1cnc2cc(F)c(F)cc2[nH]1)c1ccc(C)s1 C(=O)(CCN=C(NCC1CCCSCC1)NCC1CC1(F)F)N(C)C N1(C(CCSc2nc(C)[nH]n2)=O)CCN(C(=O)CSC2CC2)C(C(F)F)C1 C12(CNC(C3CC(C)(O)C3)=O)CC1CN(C(c1ccc(C(F)(F)F)nc1)=O)C2 c1(C(=O)NC2C(C)CCN(CCc3cn(C4CC4)nn3)C2)c[nH]c2ccccc12 C1(C(=O)NCCC(C)(C)N(C)C)(NC(C(C)=C(CC)C)=O)CC(CO)C1 C12(C(N3CCC(CNC(C4(CC=C)CC=CC4)=O)C3)=O)CCCC(=O)N1CCC2 N1(C(CCOC)=O)CC(O)CC1CNC(c1ncoc1-c1cnn(C)c1)=O c1(C(=O)OC)ccccc1CN1C(C(=O)Nc2cnccc2Br)CC2CC12 C1(C)(C(=O)NC(C)CC2CN(C(C3(NCc4ccccc4)CC3)=O)C2)CNC(=O)C1 N1(C(C2(NC(CC3(NC(C)=O)CC3)=O)CC2(C)C)=O)CCN(C)C2(CCC2)C1 S(=O)(=O)(c1cccc(N)c1)C(N(C)CC1CC(C)C1CCNCC)C C12(CNC(c3c(OC)nccc3)=O)CCC1CCN2C(c1csc(Cl)n1)=O Cc1cc(C(=O)NC2COCC2NC(c2cc(C)sn2)=O)c2nccc(C)c2c1 CC1=C(C(=O)NC2COCCC2C(=O)NCC2CCCOC2)CCO1 C(=O)(C(C)(O)CC(F)F)N1CC(CC)N(C(c2nn(CC)nc2C)=O)CC1 O=C(C1=CCCCCC1)NC1CN(c2ccnc(C(F)(F)F)n2)CC1F C1(NC(C=C(C)CNC(C2CCC2(F)F)=O)=O)CCCC(O)C1 c1(C(=O)NC(CN(C(C(COC)N(C)C)=O)C)(C)C)cnc2ccccc2c1C CC(C)C(C(=O)NC1CCCC1NC(c1nnsc1N)=O)c1cccnc1 c1(CCC(=O)N(C(C)CNC(C2CN(C)C(=O)N2)=O)CC)ccc(Br)cn1 N1(CC(=O)Nc2ccc(Cl)c(Br)c2)CCC2CCCCC12 C(c1nccs1)=CC(=O)NCC(CO)NC(c1c[nH]nc1Cc1ccccc1)=O Cc1ccc(C(C)C(=O)NC2CCC(CNC(C3(c4cc[nH]n4)CC3)=O)C2)cc1 c1(N(C2C(CC)CCCC2)C)nc(=N)nc(N2CCC(CF)CC2)[nH]1 c1(C(N2CC(NC(C3(CCC)CC3)=O)C(O)C2)=O)ccc2nc[nH]c2c1 c1(NC(=O)C2CC2)ccc(-n2cc(C(=O)OCC)nn2)cc1 c1(C(=O)NC2CCN(CC(=O)Nc3cccc(O)c3)CC2)c(O)cccc1O C1(C)(NC(c2nncc(OC)c2)=O)CCCN(C(c2ccc[n+]([O-])c2)=O)C1 C(=O)(C(C)(C)OCC(C)NC(COCCC(C)C)=O)NC.C(C)(C)(C)O c1(C(=O)OC(C)(C)C)csc(=NCC2CC3(CC3)C(=O)O2)[nH]1.CC(C)C1C(=O)O1 C1(COC)CN(C(C2COCCN2C(=O)CC23CCC(CC2)C3)=O)CCO1 Cc1nc(NCC2(C)CCN(C(C3CCCCC3)=O)CC2)cc(C(C)C)n1 c1(C(=O)NC2CCN(CC3(N(C)C)CC3)C2)c(N(C)C)ccc(F)c1F c1(OC)cc(C)c(C(=O)NC(C)CCCCNC(c2nccn2C)=O)cc1Cl c1(C(=O)NCCC(C)NC(=O)C(c2ccccc2)=O)cncc(-n2cnnn2)c1 C1(C(C)C)CN(C(=O)C(CO)NC(N)=O)CCN1C(C1CCC(F)(F)C1)=O C(=O)(C1=NOC2(CCOC2)C1)N(CCNC(=O)C(CC(C)C)NC(C)=O)CC C1(CN(C)C)CCC(C(=O)NC2CC(C)(NC(=O)C(=O)NC3CC3)C2)O1 N1(C(C=CCOC)=O)C(C(N2CC(C(C)OC)C2)=O)CC2CCCC12 c1(OC)ccc(CCCCC(=O)NCCNC(C2CCC(C)CC2)=O)cc1OC N1(C(C2CCN(C)C(=O)C2)=O)CCC(C2CN(C(C34C=CC(CC3)C4)=O)C2)CC1 C1(CC(=O)N(C2CCN(C(=O)COCC3CCCC3)C2)CC#C)CC(CC)=NO1.C CCCC(C(=O)NCCc1cnccn1)NC(C1(C)CC(F)(F)C1)=O Nc1cc(C(N2CC3C(CNC(C4(CO)CC(F)(F)C4)=O)C3C2)=O)ncc1Cl N1(C(COCCCC)=O)CC2(CC(NC(C3(C)CCOC(C)C3)=O)CO2)C1 O=C1NCC2(CCCN(C(C3CCC4(CCC4)CO3)=O)CC2)O1 c1(C(N2CC(C3CN(C(c4ccncc4)=O)CCO3)C2)=O)cccc2occc12 C(=O)(C1=CS(=O)(=O)c2ccccc21)NCC1CCN(C(CNC(N)=O)=O)C12CC2 N1(C(c2c(OC)ccc(Cl)c2)=O)C2CCC1CN(C(c1ccc(C)nn1)=O)C2 Cc1ccc(NC(C2CC23CC(NC(c2ccc(C)c(C)n2)=O)C3)=O)c(C)n1 S(=O)(=O)(c1c[nH]c(=NCc2csc3c(Cl)cccc23)cc1C)NC1C(COC)C1 CC(C)CCC(C)NC(=O)CC1CCN(C(=O)CCCn2cccn2)C1 N1(C(c2c(CC)noc2)=O)CC(NC(c2ccc(-c3cnco3)cc2)=O)CC1C c1(C(=O)NC(c2ccc(F)cc2)CNC(COCCCC#C)=O)n[nH]c(C)c1O c1(OC)ccc(NC(C2CC(CNC(=O)CC(C)c3cccnc3)C2)=O)cc1 c1(OC)cccc(CC(=O)NCC2CN(C(c3cocn3)=O)C2)c1 Cn1cc(C(=O)NCC2(CN3CCCCCC3)CC2)c(=O)c2cnn(C)c12 C1(C(=O)NC(C2CCCC2)CNC(C2CCC(CC)O2)=O)CCC(C)(C)CC1 N1(C(C2(CC=C)CCCN2C(c2c[nH]c(=N)c(C)c2)=O)=O)CC(C)=CC(C)C1 C1(C(N2C(CNC(c3n(C)cc(C(N)=O)c3)=O)CC2)=O)CCC([N+](=O)[O-])CC1 c1(C(N2CC(C(=O)NCCC(C)c3cn[nH]c3)OCC2)=O)cn2ccccc2n1 C=CC1(O)CCN(C(=O)CC2CCCCN2C(C23CC(CO)(C2)C3)=O)C1 N1(C(CC=C)=O)CCC(C2(CNC(C3(C#N)CCCC3)=O)CCOCC2)CC1 S(=O)(=O)(c1ccc2c(c1)CCCC2)NC(CC1CCCC(C)C1=O)=O CCCCCCCC(=O)NC1(C2CCN(C(=O)Cc3ccc(C)cc3F)C2)CC1 N1(N2C3CNC(C3)C2)CCc2cccnc2C1.Cc1c(C)cncc1Br c1(C(N2C(CCC)C(C)CC2)C(=O)NCCSC)cccc2ccccc12 C(C1CN(C(C2OCCC2(C)C)=O)CC1C(=O)N(C(C)(C)C)CCOC)=CC C(=O)(CC(C)(C)C(F)F)N1CC(C)C(CNC(=O)CCP(C)(C)=O)C1 C1(F)(CNC(CC=CC=C)=O)CC(NC(=O)CC2(COC)CCC2)C1 C(N=c1[nH]c2cc(Cl)ccc2s1)C1(O)CC2N(C(COCC)=O)C(CC2)C1 C(=O)(C(C)N(C(=O)COC)C)N(C1C(CCC)C1)C C(CC(C(=O)NC(C)Cc1cnn(C)c1)NC(=O)CC1CC1CC)OCC C1(C)(C(=O)NCC(CCNC(c2c(OC)n[nH]c2)=O)O)CC2(CC2)C1 C=CCC(C(=O)NC1CC(CNC(=O)Cc2c[nH]c(=N)nc2O)C1)C(C)C N1(c2cc(NCC(CCCC)CC)nc(C)n2)CCC(NC2CC2)C2(CC2)C1 Cc1c(C(N2CCC(C)C2CNC(=O)CS(=O)(=O)N(C)C)=O)cnn1CC(F)F C1(NC(CCC=C)=O)CC2CC1N(C(C1C3CC4C(C3)C14)=O)C2 C(=O)(CCCCC(N)=O)NC(C(C)C)(C)CNC(C1(C2CCCO2)CC1)=O c1(CNC(c2c(C)nsc2N)=O)cnn2c1CN(CC1CCN(C(C)=O)C1)CC2 C1(C)(NC(CN(C(C(CC)n2cncn2)=O)Cc2cn[nH]c2)=O)CCCCC1O c1(C(N2CCC(N(C)C(C3CCNC(=O)C3)=O)C2)=O)cnc2n1CCCC2 Cc1nn(C)c(Cl)c1C=CC(=O)NC1CN(C(=O)C(C)O)CC1n1ccnn1 C1(F)(CNC(c2c(C)csc2)=O)CCN(C(c2ccc(C)cc2O)=O)CC1 N1(C(C(CC2CN(C(c3cc(C)[nH]c3C)=O)C2)F)=O)CCC2(CCSC2)C1 c1(NC(C2C3CC2N(Cc2ccc4nccn4c2)C3)=O)ccc2nnsc2c1 C(=O)(CCCCCc1ccc(O)cc1)N1CC(O)(CNC(C2CC3CC3C2)=O)C1 CN(C1CCc2ccccc21)C1CC2CCC(C1)N2CCC1CCS(=O)(=O)CC1 C(CCC(=O)N1C(C(=O)N(C)CCn2cccn2)CC1C)OCC=C C1(C(=O)NC2CC(C)(CC)C2)CC2(CCN1C(c1cc(Cl)ns1)=O)CC2 c1(C(=O)NCCC(=C)CNC(c2nc(=N)cc[nH]2)=O)cc2cccc(Cl)c2s1 c1(OCC)nc(C)ncc1Br.C12CN(CC1n1ccnn1)C(=O)C1CC1C(=O)N2 N1(C(CCOCCC)=O)CCC2CCCN(C(c3c(N)sc(C)c3C)=O)C2C1 C1(CNC(CC(=O)OC)=O)CN(C(c2occc2-c2ccccc2)=O)CCCO1 C(=O)(CS(=O)(=O)C(C)C)NC1CCCCN(C(c2c(C)sc(Cl)n2)=O)C1 CCCCCCCC(=O)NCC1CC(NC(=O)C(F)=CC2CC2)C12CCC2 CN=c1[nH]cc(C(N2CCC(O)(C(C)NC(c3ccoc3C(C)C)=O)C2)=O)s1 CC1C(NC(C23CC(NC(=O)CC4(O)CCOCC4)(C2)C3)=O)C2CCN1CC2 c1(NC(=O)Nc2cccc(NC(CCSCC(=O)OC)=O)c2)ccc(F)c(F)c1 c1(NC(C(N2CCC(C(C)NC(C)=O)C2)C)=O)ccc(F)c(C)c1 C1(CNCC)CCC(NC(=O)C(C2(O)CCCC2)F)CC1.C(C)(C)=CC CCCC(CC)C(=O)NCC(O)CN(C(=O)Cn1cnc(Br)c1)C Nc1cc(Cl)ccc1C(=O)NC12CCC(CC1NC(c1ccc(N(C)C)nn1)=O)C2 C1(CC(=O)NC2CC2)C2CN(CC(F)(F)F)CC12.C12CC3(C1)CC3CNC2=O N1(C(C2CCC3CC(C)CN3C2)=O)CCN(C(=O)Cn2cnnn2)CC12CCC2 N1(C(CC2(NC(c3c(C)nn(C)c3)=O)CCCCC2)=O)CCN(C)C2CC12 c1(CC(N2CCCC(CNC(Cc3c(C)cc(C)s3)=O)C2)=O)ccc(Cl)c(O)c1 C1(C(=O)NC2CN(C(c3cc(O)nc(O)n3)=O)C3CC23)CCn2nncc2C1 C(C(=O)N1CC(CNC(=O)CN2CCOC2=O)(OC)C1)(C(C)C)SCC Cc1ccc(CC(=O)NCCC2(NC(=O)C(C)S(C)(=O)=O)CCC2)cc1Cl Cc1cncc2cc(C(=O)NC(C3CCCCC3)CNC(=O)CC3(C)CC3)sc12 c1(CNC(C(C)N2CCC2)=O)cn(CCNC(c2cnc(O)o2)=O)nn1 C12CN(C(=O)C(C)=CC(C)(C)C)CC1O2.C(CCCCOCCc1ccccc1)OCC Cc1cc(C(=O)NCCN(C)C(c2ncnc3sccc23)=O)c2cnn(C)c2n1 CC1CCCC(OCC(=O)N(C(C)CCNC(=O)C(C)(O)C2CCC2)C)C1 CN1C(=O)CCCC1C(=O)NC1CCCC1NC(c1cncc(F)c1Cl)=O C1(NC(c2c(C)con2)=O)COC2(CCN(C(C3(n4nccn4)CC3)=O)C2)C1 c1(NCC2OCCN(C)C2)[nH]c(=NCC2CCC(=O)NC2)nc2scnc12 N1(C(CC(C)SC)=O)CC(NC(c2c(F)cc(F)cc2F)=O)C2CCCC2C1 N1(C(C2(CC(C)C)CCC2)=O)CC(NC(C2C(OC)CCC2)=O)C2(CC2)C1 N1(C(COC2CN(C(c3cnc(C)o3)=O)C2)=O)CCOC(C(N)=O)C1 Cc1cccc(CC(=O)NC2CC3(C2)CC3C(=O)NCCC(O)CC(C)(C)C)c1 N1(C(C2(C)CCN(C(CCCCOC)=O)C2)=O)CC(C(N)=O)OC(C)C1 N1(C(CCOC(C)=O)=O)CCc2nc(C(N3CC(=CCN(C)C)C3)=O)cn2CC1 C1(C(=O)NC(C(CC)C)C(=O)OC)CC2(CCN1C(=O)C(C1CC1)SC)CC2 c1(C(=O)NCC(C)CNC(=O)Cc2cc[nH]c2)cnc2[nH]nc(O)c2c1C(F)F C1(NC(=O)C=Cc2cnc[nH]2)CN(C(c2ccnc(-n3cncn3)c2)=O)C2CC12 C(=O)(C(C)(C)CC(=O)NC1CCC1NC(=O)C(c1cccc(Cl)c1)O)OC C1(CNC(C(CCC)(C)CC)=O)CCC12CCN(C(=O)Cc1ccoc1)CC2 C1(CNC(CC(C)C)=O)CCCC(CNC(c2cc[n+]([O-])cc2)=O)C1 C1(CNC(=O)CNC(c2cccc(Cl)c2)=O)CC2CCC1N(C(C1CCC1)=O)C2 c1(C(N2C(C(N3CCCC(C)(F)C3)=O)CC3CC32)=O)ccc(Br)c(Cl)c1F Cc1cc(C(F)(F)F)ccc1NC(=O)CONC(=O)C(C)c1cccnc1 C=CCC(CC(C)C)C(=O)NCC(C)(CO)NC(=O)CCn1c(C)c(C)sc1=O N1(C(C(=O)NCC2CCOC2)CCc2ccccc2)CC(C2=NOCC2)C1 c1(C(=O)NCC(C(F)(F)F)NC(c2nc(CCC)sc2)=O)cc(CC)ccc1C N1(C(CCN(CC)CC)=O)CC(NC(C2CC(C)(C)OC2(C)C)=O)C2(CCC2)C1 c1(OC)ccc(C(N2CC3CC3(C(=O)Nc3cnncc3Cl)C2)=O)cc1C Fc1cc(Cl)cc(Cl)c1CCN1CCCC(C(F)F)C1 N1(C(C(C(=O)NC)(C)C)=O)CCC(C2CN(C(C3CC3C3CC3)=O)C2)CC1 c1(C(=O)NCC(C)(C)NC(=O)CC23CCCC2C3)csc2c(F)cc(Cl)cc12 C1(C(=O)NCC(C)(C)NC(C2CN3CCCN2C3)=O)(OC)CCS(=O)(=O)C1 C(=O)(C1CCCc2ncccc21)NCCC(C(N)=O)NC(c1n(C)c(S)nc1)=O c1(C(=O)NCCOCCNC(C2(C)CCC(=O)N2)=O)cc2c(Cl)cccn2n1 O=C(C(=O)N=c1cc(CCO)o[nH]1)NCC1(CCNC(=O)CC23CC(C2)C3)CC1 c1(CC)ccc(C)cc1C(=O)NC1CCC(C)N(C(=O)CCC=C(C)C)C1 c1(C(=O)NC2(CO)CCN(C(COCC)=O)CC2)c(F)ccc2c1OCO2 CCC(CC(=O)N1CC(C)(CNC(=O)CC(CC)CC)C1)C(C)C C1(OC)CC(NC(c2scnc2C2CC2)=O)CN(C(=O)C(C)C(F)(F)F)C1 C1(NC(c2ccc(C)o2)=O)C2CC3C(C2)C13C(=O)N(C1CCC1)C1CCC1 C=C=C(C)CC(=O)NCc1ncccc1C(=O)NCC1CCC1CO C(C1CCN(C(C2C=CCCC2)=O)CC1)=CC(=O)NCCCOCC1CC1 c1(CNC(C2CC(N(C)C)C2)=O)nc(CNC(c2ccc(C#N)cc2)=O)cc(O)n1 N1(C(c2ccc(CC)cn2)=O)CCN(C(=O)CC2CC=CC2)C2CC12 C(C)(CCC(=O)NCC1C2CN(C(C3CCC3(C)C)=O)CC12)OC C1(CNC(c2cc(C)ncn2)=O)CCC(C)(C)CN1C(c1cnc2sccn12)=O C(C(C(=O)N1CCCC1C(=O)N(C)C)C(C)(C)C)NC(CCS(=O)(=O)N(C)C)=O c1(C(C#C)SCC#CCO)c(F)cccc1Cl c1(C(C(=O)NC2CN(C(C3(C)CCCS3)=O)CC3C2C3)=O)cc(F)c(F)cc1F c1(C(=O)NC2CCCC(OCC(F)(F)F)C2)cc2c(cc1[N+](=O)[O-])OCO2 C1(C(=O)NC(C)CCCNC(=O)C(C)n2cncn2)CC2(C1)CC1(CCC1)C2 c1(C(=O)NCC2(O)CN(C(c3cc(F)c[nH]3)=O)C2)cccc2ccoc12 c1(C(=O)NCC(C)N(C)C(C2(C(F)(F)F)CC2)=O)cc(S(=O)(=O)N(C)C)cn1C C1(NC(C(C)N(C(c2cnn(C3CC3)c2)=O)CC)=O)CCC(=O)N(C)C1=O Cc1cc(C(N2CCCC(C)C2CNC(=O)CCc2cc(O)no2)=O)cnc1C CC1=C(C(=O)N2CC(CC(C)NC(C3CCC(F)CC3)=O)C2)CCCC1 c1(C(C(=O)NC(C(C)NC(c2nn[nH]c2Cl)=O)C)O)ccccc1F Cc1ccc(C)c(C(N2CCC=CC2(C)C(=O)O)=O)c1C C1(CC(=O)N(C)Cc2nncs2)CC(C)(C)CN1C(=O)CC1CCOC1(C)C c1(C(=O)NC2(C(N(CC#CC)C)=O)CC(O)C2)cc(C)cc(F)c1 N1(C(CCCC(=O)N(C)C)=O)CC2CC(Nc3nnc(C(C)(C)C)s3)C(C2)C1 C1(C(N2CCC(C(=O)NCCOCCO)CC2)=O)CS(=O)(=O)c2ccccc2O1 C1(O)(CNC(c2cccc(I)c2)=O)CCCN(c2nccc(N3CCCC3)n2)C1 c1(C(C)C)cc(C(=O)NCCC2CCN(C(=O)COCCC(F)(F)F)C2)n(C)n1 C(=O)(C(C)CC(F)F)NCCc1c(CNC(Cc2cccc(C)c2)=O)nco1 N1(C(C(CC2CC2)NC(C)=O)=O)CCCC1(C)c1cncn1C CCC(C)(CC(=O)O)C(=O)N1CC(C)(c2cn(-c3ccc(N)cc3)nn2)C1 c1(C(N(C2CCCN(C(=O)CSCC(N)=O)C2)CCC)=O)cnncc1O C(C1(C)CCC(C)C1(C)C)=CC(=O)NC(C1CCN(C(=O)CC(C)C(C)C)C1)C c1(C(=O)NC2CC3CC(NC(=O)C4=COCCC4)C3C2)c(Cl)sc2nnsc12 CCC(CC)C(C(=O)N1CC(NC(c2ccc(OC)s2)=O)CC1C)OC c1(C(N2CCC(C#N)C2)=O)n[nH]c2c1CN(C(C1CC3CCC(C1)O3)=O)C2 c1(CC(=O)NCCNC(=O)C(c2ccccc2)=O)cn2ccsc2n1 c1(C(N2CCC(C(N)=O)(CC3CC3)CC2)=O)ccc(C#C)cc1F.C1(=O)CN1CC C1(C(=O)NC2CCN(C(CCC(C)(C)OC)=O)CC2)CCCC2(C1)CC2(F)F Cc1coc(C=CC(=O)NC2CCC(CNC(c3n[nH]c(C)c3N)=O)C2)n1 N1(C(COCCCC)=O)CCC2(NC(c3snnc3C)=O)CCCC12 N1(C(c2ccc(OC)cn2)=O)CCCC12CCN(C(=O)CCP(C)(C)=O)C2 c1(C(=O)NC2CC(NC(C3(COC)CCCO3)=O)C2)cc2ccccn2n1 CN1CCC(C(=O)N(CCC2(NC=O)CCC2)CCSC(F)(F)F)C1=O N1(C(CCC)=O)CCCC(C(N2CCCCC2CNC(=O)CCCOCC)=O)C1 Cc1coc(C(=O)NC(C(N2CCC(N3CCCC3)C2)=O)C2CCCC2)c1 C1(CC(c2onc(CC)n2)=O)CCCC(=O)C1 Cc1ccc(COCC(N2CCCC2CNC(c2ccc(Cl)s2)=O)=O)s1 N1(C2CCN(C(=O)Cc3nc(C4CC4)n[nH]3)C2)CCN(C(C2CCC2)=O)CC1 C(=O)(CC(C)CNC(C1(CC(=O)OC)CC1)=O)N(C(COC)C)C C1(CC(=O)NCC2(OC)CC2)CC2(CC2)CN1C(c1nnc(O)nc1O)=O Cn1ccc2ccc(C(=O)NC3CC(CNC(c4cc(F)ccc4Cl)=O)C3)cc12 c1(C(=O)NCCCC2CCCN2C(c2cc(Cl)c[nH]2)=O)coc2c1C(=O)NCC2 c1(C(=O)NCC(C)CNC(=O)CCN(S(C)(=O)=O)C)cnc(N)cn1 N1(C(c2cnc(CC)o2)=O)CC(C(N2CCCCCC2C)=O)C(C)(C)C1 c1(OC)coc(C(=O)N(C2CCN(C(=O)CC3CC3(C)C)C2)C)cc1=O C(CC(=O)NNC(=O)C1CC(C)OC(C)C1)Sc1onc(C)n1 c1(CC)cscc1NC(=O)CCN(C(c1ccns1)=O)C(C)C c1(C(N2C(C)CCN(C(c3ccc(C)cc3C)=O)CC2)=O)cnc2c(c1)COC2 CC(CCCCNC(=O)CCc1nncs1)NC(c1cc(C#N)c[nH]1)=O C1(NC(c2occc2CNC(=O)NC2C(OCC)CCC2)=O)CC2(C1)CC(C)C2 CC1CCCC1(C(=O)NCCn1cccnc1=O)NC(=O)C=CCO C1(NC(CC=C)=O)CN(C(=O)CCC(=O)c2ccccn2)CC1(C)C C1(NC(CC(CC)O)=O)CCN(C(c2ccccc2O)=O)CC1C C#CCCCC(C)C(=O)NC(C1CCCCC1)C(=O)NCCCP(C)(C)=O C1(NC(CN(C(C2(CCOC)CC2)=O)C)=O)CC(C(N)=O)C12CCC2 C=CC1COCC1NC(C12CC(NC(C3CCCN3C(C)=O)=O)(C1)C2)=O N1(C(CN(C)CC)=O)CC(CCNC(c2sccc2C(C)C)=O)OC(C)C1 c1(C(=O)NCCC(C)NC(c2ccc(CN(C)C)nc2)=O)cc(C#N)c(F)cc1F C(CCC(=O)OCC)(S(C)(=O)=O)NC(CC=C)CC.C(C)(C)C C1(F)(C(=O)NCC2C(C)C2(F)F)CCN(C(=O)CCCC#N)CC1 C1(C(N2CCN(C(C3(OC)CCOC3)=O)CC2)=O)OCC2COCCC12 N1(C(CC(C)F)=O)CCN(C(=O)CCNC(N)=O)CC12CCC2 C1(CCNC(C2CC(OC)C2)=O)CCCN1C(=O)CNC(=O)CC1CC(F)C1 C=CC(CCC)CC(=O)NCC1(F)CCCN(C(C2CCC(CC)O2)=O)CC1 C(CC(C(=O)NCC1CCCC(O)C1)NC(C1CN(C(N)=O)C1)=O)N(C)C CC(C)CC(C(N)=O)NC(C1C=CC(NC(C2CC(=O)N(C(C)C)C2)=O)C1)=O CON(CCC(=O)N1CC(CNC(=O)CC2CC2)C1)C(=O)OC(C)(C)C Cc1cc(C(=O)NCC(O)CNC(c2nc(Cl)cs2)=O)cc(C(F)F)c1 O=C1NC(C(=O)NCC2CCN(C(=O)C(c3ccc(Cl)cc3)(F)F)CC2)CCO1 C1(CNC(c2n(CC#C)ccc2)=O)CCCCCN1C(c1ccc(CO)cc1)=O CC1=NNC(=O)C1CC(=O)N(C)CC1CCCCN1C(c1ccsc1C(F)F)=O c1(OC)nc(C(=O)N(C)CC2CCCN2C(=O)CCC2OCCO2)cc(O)n1 CC(C)(F)C(C)(F)C(=O)N1CC2CC(Nc3cc(CC4CCCC4)ncn3)CC1C2 CC(CCCNC(=O)C=CCc1ccccc1)NC(C1CCC1COC)=O N1(C(C2CC(OC)C2)=O)CC(CNC(=O)CCc2cn[nH]c2)CCC1C N1(C(C2(COC)CC(=C)C2)=O)CCC(C)(C(=O)NC(C)CN(C)CC)CC1 Cc1nc2nccc(C(=O)NC3CCC(NC(c4n[nH]cc4Cl)=O)CC3)n2n1 c1(CC(N2CC(C(=O)OCC=C)C2)=O)c(F)cccc1F.C1(=O)CO1 C(=O)(C#CC1CCCCC1)NCc1cnc(NC(=O)CCCCCF)s1 CS(=O)c1cccc(C(=O)NCC2CN(C(c3cncc(F)c3Cl)=O)CC2O)c1 N=C1NC(=O)C(CC(N2CCCC2CNC(C2CCCN2C(=O)C2CC2)=O)=O)S1 C=C1CCC(CNC(C2(N(C3CCN(C)C3)CC)CCC2)=O)CC1 c1(C(=O)NCC2N(C(c3ccc(C(CC)C)cc3)=O)CC2)cc(O)cc(Cl)c1 c1(C(N2CCCC(CCCCNC(COC)=O)C2)=O)cc2c(Cl)cncc2s1 C1(NC(CN(CCOC)C)=O)CC2CCC(C1)N2C(C1SCC=C1C)=O c1(C(=O)NCCC2(O)CCN(C(=O)C#CC3CCOC3)C2)ccn2c1CSCC2 N(C1CN(C(C23CC(C)C2C3)=O)Cc2ccccc21)C(c1c(C)oc(CO)c1)=O c1(CC)ccc(NC(=O)N(CCC(=O)NC(c2ccccc2OC)C)C)cc1 C1(C#N)(C(N2CC(C(=O)NC3CC(C)CCC3O)(OCC)C2)=O)CCCCC1 c1(CC)ccc(C=CC(=O)NCC2CC(NC(=O)C=CCF)CCO2)o1 C(C(O)CN(C(=O)CC1CCC1)C)NCCOCC#C C1(NC(CC(C)C)=O)CCCN(C(C2CCCC(C)CC2)=O)C1C c1(C(N(CC(C)(C)CNC(=O)CC2CCC2)CC)=O)c(N)sc2c1CCC2 Fc1cc(CN=C(NCC(N2CCCC2)=O)NCc2ccccn2)cc(F)c1 Cc1cc(C(=O)NC(C(=O)NCC(C2CC2)C2CC2)C2CCOC2)ncc1F CC(C)CC(O)CC(=O)NC(C)C(C(C)C)NC(c1ccnn1C(C)C)=O c1(OC)cc(C(C)=O)cc(OC(=O)C(C(C)C)c2ccc(N)cc2)c1OC c1(C(C)C)noc2ncc(C(=O)NCCN(C)C(C3CCS(=O)(=O)C3)=O)cc12 c1(C(N(C)CC)=O)ccccc1Cn1cc(C(c2ccccn2)O)nn1 N1(CC(C)C)N=C(C(=O)NC(=O)Cc2ccc3ccccc3c2)CCC1=O n1(C(C)(C)C)nccc1C(=O)N(C1CC1)CC1CC(NC(c2ccn(C)c2)=O)C1 C1(C(=O)NCCc2ncon2)NCCC1C1CC1.c12ccc(cc1)CO2 C1(NC(C(C)OCCC=C)=O)CCCN(C(=O)C2=CCCC2)C1C C1(C(=O)NC2(CNC(CC)=O)CC2)CC(CC(F)(F)F)C1 c1(NC(C2(OC)CCN(C(=O)C(O)CN(C)C)C2)=O)cnn2cccnc12 c1(-c2cn(C3(NC(=O)CCn4cccn4)CC3)nn2)cc(F)cc(F)c1 c1(OC)ccccc1C1(C)CC1.C12(OC)CC(C1)C(=O)NC1CC(C1)NC2=O C1(NC(C(CCC)C)=O)CC2CCC1CN(C(c1cn(C)c(C)n1)=O)C2 C(=O)(C(O)CC(C)C)N1CC2C(CNC(c3c(OCC)scc3)=O)C2C1 c12cn(C)nc1C(=O)OC2.N1(C(C(OC)OC)=O)CCC(C)(C(N)=O)C1 C1(C(N2CC(N3CCOCC3)C2)=O)(COC)C=CCN1C(C1CCSC1)=O CC1CN(C(C2(C#N)CC2)=O)CCC1NC(c1cc(C(F)(F)F)cs1)=O C1(NC(c2nc(C)[nH]c2Br)=O)CCCN(C(=O)Cc2csnn2)CC1 N1(CC(=O)N(C(C(=O)NC(C#C)CC2CC2)C2CCOC2)C)CCOCC1 c1(C(CO)NC(Cn2cc(C3CCC(=O)C3)nn2)=O)ccc(F)c(Br)c1 c1(C(=O)NC(C2CCCN(C(C3(CCOC)CC3)=O)C2)C)c(N)cc(Cl)cc1F N(C(=NCC)NC1CCCN(CCSc2ccccn2)C1)C(C=C)C C1(C(N(C2CN(C(C(C)OC3CCCC3)=O)C2)C)=O)CCSCC1.C1(=O)CCCN1 C(c1ccc(-c2cccnc2)cc1)=CC(=O)OC.C12CCN(C1=O)CC(=O)N2 C1(NC(C=CC(CC)C)=O)CC(NC(c2cc(CCOC)on2)=O)CC1O C1(CC(N2CCCCC2CF)=O)CC(F)CN1C(=O)C#CC1CC1 C1(CNC(C2(C(C)C)CN(C(C3(C)CCN(C)C3)=O)C2)=O)CC2CCCC2C1 c1(CC(=O)NC(CCNC(CCC)=O)(C)C)nc(C)sc1Cl N1(C(CC(=C)C)=O)CCN(C(=O)C(C(C)C)n2cccc2)CC(C)(F)C1 c1(C(N2CCC3(NC(c4n(CC)ccn4)=O)C(C2)C3)=O)ccc2nc(C)ccc2c1 Cn1ccnc1CCC(=O)NCC1C=CCN1C(c1c[nH]nc1Cl)=O c1(C(N2CC(C)N(C(C3CC3CF)=O)CCC2)=O)cncc2c(O)nccc12 N1(C(CCN(C)CC)=O)CCCC(NC(=O)C(N2CCSCC2)C)C1 C(=O)(CCCC(C)(C)C)N1CCC(NC(Cn2c(C)ncc2)=O)C(F)C1 c1(CNC(c2ccc(-c3ccc(CN(C)C)s3)cn2)=O)ccc(Br)cc1[N+](=O)[O-] c1(CCCCNC(=O)NCC2CCCCNC2)cccc([N+](=O)[O-])c1 c1(C(C(=O)OC)N(C(=O)CCc2ccc(Br)cc2)C)cccc(Br)c1 c1(OCC)cnccc1C(N1CC(=CC(C)NC(=O)Cc2ccnn2C2CC2)C1)=O N1(C(c2c(C)nn(C(C)C)c2)=O)CC=C(CNC(c2ccnnc2)=O)CC1 N1(C(CSCC)=O)C2CCCC1CN(C(C1CCC(=O)NC1)=O)C2 S(=O)(=O)(c1[nH]c(=NC2CC3C=CC2C3)ccc1Br)NCCOC1(C)CCCC1 S(=O)(=O)(c1ccc(C(N2CCN(C(C3CCC4CC34)=O)CC2C2CC2)=O)o1)NC N1(CC2CC(OC)C2(C)C)C(=O)C2Cc3ccc(O)cc3CN2C1=O C1(C(=O)OC)CCN(C(=O)Nc2cnn(C3CCOC3)c2C)CC1(F)F Cc1ncccc1CCC(=O)N(C1CCC(NC(C2CCCSC2)=O)CC1)C C1(O)(CN(C)C(C2(CF)CC(F)(F)C2)=O)CCN(C(=O)C2=CCCC2)CC1 CCC(C)C(=O)NCCC1(C(=O)N(C(CC)C(=O)OC)C)CCC1 C1(NC(c2n(CCC)ccc2)=O)CN(C(c2ccc(CSC)o2)=O)C2CC12 N1(C(C(C)Cc2cnn(C)c2)=O)CCCC(N(C(=O)CCn2cncn2)C)CC1 c1(C2CCCN(C(=O)Nc3c(CN(C)C)cccc3)C2)ccc2nc(O)oc2c1 C(=O)(C(C(C)(C)C)NC(=O)CC1(O)CCC1)N(C)Cc1cnccn1 C(=O)(C(C)(C)CC(=O)OC)NC1CCN(C(CSCCC)=O)CC1C C=CC1(CC(=O)NC2CCCC(F)C2)CN(C(=O)C=CC2CCCCC2)C1 C(c1cccc(F)c1)=CC(=O)NC(C)(C)CCNC(=O)CCC1CCC(=O)NC1 CC(=O)CCN=C(NCc1ccsc1)NC1C(C)(C)C1(C)C C1(NC(C(=C)C(F)(F)F)=O)CN(C(c2ccc(C)nc2F)=O)Cc2nccn2C1 Cn1ncc2c(O)cc(C(=O)NCC(CNC(C3(C)CC(C)(C)C3)=O)CO)cc12 N1(C(C(C2CCC2)NC(c2cc(C)on2)=O)=O)CC2CCCCC2C1C c1(C(N(C2CN(C(CSCC#C)=O)CC2F)C)=O)cc2cn[nH]c2cn1 C1(CNC(CCCSC)=O)CN(C(C2CCCCC2(C)C)=O)CC1(C)C N1(C(=O)Cn2cnnc2O)CC(C(=O)NCc2ccc(F)c(F)c2)C2(CC2)C1 O(NC(=O)C(C)(c1ccccc1Cl)N1CCOCC1)C(C)(C)C c1(CCC)cc(C(=O)NC(C)CC(C)NC(=O)COC2CCC2)n(C)n1 CC1CN(C(C2OCCO2)=O)CCC1NC(c1ncn(-c2ccccc2)n1)=O C(CC(O)(C(F)(F)F)c1ccc(F)cc1)NC(N1C(c2cn(C)nc2)CCC1)=O N1(C(C(CCCCC)O)=O)CC2CCCN(C(=O)CCc3ccon3)C2C1 C(=O)(CC(C)C(C)(C)C)NCCC(=C)CNC(=O)CSc1ccncc1 N1(C(CNC(=O)CC(F)(F)F)=O)CCN(C(c2cc(Br)n[nH]2)=O)CC(O)C1 c1(OC)ncc(F)cc1CN1CCC(O)(CNC(c2ccncc2)=O)C1 N1(C(c2cccc(-c3ccc[nH]3)c2)=O)CCOc2cc(Cl)ccc2C1 c1(OC)ccc(CC(N2CCCC(CN(C(=O)CC3C=CCC3)C)C2)=O)nc1 c1(NC(N2C(C)CC(C3CC3)C2)=O)ccc(F)cc1NC(=O)CN1CSCC1=O c1(OCC)ccccc1C=CC(=O)NC1(CCSC)CCCC1 N1(C(C(c2cccc(F)c2)(C)C)=O)CCOC(CNC(C2CCC2CF)=O)C1 c1(C(CC)=O)ccc(C(=O)NC2(C)CN(C(c3ncccc3F)=O)C2)cc1 c1(C(c2c(C)cccc2)NC2CCC(C#N)CC2)cccc2ccsc12 C(=O)(C(C)CCCC(C)C)N1CCN(C(C(COC)OC)=O)C(c2ncc[nH]2)C1 N1(CC(c2ccccc2F)CC)CCOc2cc(Cl)ccc2C1 c1(C(C)C)cccc(C(N2CCOCC(NC(=O)CC(C)N(C)C)C2)=O)c1N N1(C(C(C)=C2CC2)=O)CCC2(CCCN(C(c3sc(=N)[nH]c3C)=O)C2)C1 CC#CC1CCN(C(C2CCC=CC2NC(=O)CC(CC)OC)=O)C1 CS(=O)(=O)c1cccc(C(=O)NCCC#N)c1.C1CC(=O)N1CCCO N1(C(CC(CC)CN(C)C)=O)CC2CCC(C1)N2CC(N1CCC(C(N)=O)CC1)=O C1(C(=O)NCC(=O)NC2C(C)CC2)(CNC(c2cnccn2)=O)CC(C)(C)C1 C(=O)(C(CCC)C(C)C)NC(CCC=C)C(=O)NCCn1ccc(=O)cc1 C1(C(=O)NCC(c2ccccn2)C)(CF)CCN(C(c2ccc(C(F)F)o2)=O)C1 CC1C(NC(=O)Cc2cccc(Cl)c2)CC2CCC1N2C(C12CC1C2)=O c1(C(N2CCC(N(C(CC=C)=O)C)CC2)=O)ccc2c(c1)C(C)CN2 C(=O)(CCS(N)(=O)=O)NCC1CCCC(NC(C2CC(OC)C2)=O)C1 c1(C(N(CCOC)CCNC(=O)C(C2CCOCC2)F)=O)ccc(C(C)O)cc1 Cc1nn(C)cc1NC(=O)CC(CC1CC1)NC(c1ccc(Cl)cc1)=O c1(C(N2CC(NC(c3ccc(COC)[nH]3)=O)(CO)C2)=O)cccn2c(C)nnc12 Cc1cc(C(=O)NCC(C(C)C(C)C)NC(c2ccn(C)c2)=O)cnc1C(F)(F)F C(=O)(C(C)C(O)CC(C)C)NCC(C(C)C)C(=O)NCC1(O)CCOC1 Cc1cnc(C(N2CC(Oc3cc(F)cc(F)c3)C2)=O)c(F)c1 N1(C(CC(C=C)(C)C)=O)C2CC=C(C(=O)N3CCn4nncc4C3)C1CC2 CC(C)C(C(C)NC(C1CSC1)=O)NC(=O)C(C)(C)CC1CC1 CCCCCCC(CC)C(=O)NC(C)CCNC(=O)COc1ccc(F)cc1 CCCCCCCCC(=O)NCCCN(C(C1CC1CC)=O)C1CC1 c1(CN2CCN(C(Cc3c(C)cc(F)cc3)=O)CC2C)cc(F)c(O)c(F)c1 C1(C(N(C)CC2(CNC(C3CCCN3C)=O)CC2)=O)CCCCN1S(C)(=O)=O Cc1ccc(C(N2CC(CNC(=O)C(C)(O)c3ccccc3)C2)=O)o1 c1(CC)ccc(F)cc1C(=O)N(CC(C)CNC(C1(CF)CCC1)=O)C C(=O)(C(C)(CO)NC(c1nc(Cl)oc1C)=O)N(CC=C)CCOC C(c1ccc(OC(=O)OC)cc1OC)=CC(N1CCC(CCCCC)CC1)=O N1(C(c2nc(C(C)OC)oc2)=O)CCN(C(=O)CC2(C)CC(F)(F)C2)CC(O)C1 c1(C(N2CCCCCC(NC(C(C(C)C)C)=O)C2)=O)ccc2c(c1)CN(C)C2 c1(C(N2C(C)CCC(NC(c3ccc(C)c(F)c3)=O)C2)=O)cc(Cl)c(F)cc1N c1(C(=O)NCC(CC)NC(c2ccc(CO)cc2)=O)nc2n(c1Cl)CCCC2 c1(CCn2c(C)ncc2)ncc(C(F)(F)F)cc1C1=CCC(C(C)C)CC1.C(CO)N C1(NC2CCC(c3cc(Br)ncc3)OC2)CC2(CCCNC2)C1 N1(C(C(CCCC)NC(=O)COc2cccnc2)=O)C2CCC1CN(C)C2 C(C1Cc2ccccc21)NC(C(C(C)C)CNC(=O)CC(C)n1cccn1)=O C(=O)(CCN(C)C(C)=O)OCCC.C12CN(C1)C(=O)C(C)S2 Cc1coc(Cl)c1C(=O)NC(C)CNC(=O)CC1CCC1NC(=O)OC(C)(C)C c1(CN(c2cc(Nc3ccn4ccnc4c3)ncn2)C)ccc(O)cc1[N+](=O)[O-] CC1CCC(NC(C2CCC3CC23)=O)CN1C(C1C2CCCOC12)=O C1(C(=O)N(C)CCN(C(=O)Cc2cc(C(C)C)on2)C(C)C)(OC)CC(C)C1 N1(CC(=O)NCCNC(=O)CCc2ccsc2)CCS(=O)CC1 c1(N2CCC(OC)C(C)(C)C2)nc(=NCC(C)C(C)(C)C)[nH]c2cccnc12 c1(C(=O)NC2C(NC(c3c(OC)nn(C)c3)=O)CCC2)ncc(N)cc1Cl C1(NC(c2ncc(C)nc2)=O)CN(C(=O)COC2CCCC2)CC2(CC2)C1 N1(C(Cn2cnc(C#N)n2)=O)CC2CCCC(CNC(=O)COC3CCC3)C2C1 C(C)(C)(C(=O)N1CC(OCCNC(=O)C(F)(F)C2CC2)C1)OC Cc1cc(C=CC(=O)NCC(C)NC(=O)CC2OCCC2C)c[nH]c1=N C12(NC(COCCC=C)=O)CC(CN1C(=O)CCC(C)O)C2 Cc1ccc(CCC(=O)NCC=CCNC(=O)CCC=CBr)cc1C N1(C(C2(CCOC)CC2)=O)CC(NC(=O)CC2CCCO2)C1.COC c1(CCNC(c2nnnn2C)(C2CCCCC2)CC)c(F)ccc(Cl)c1F C1(O)(CCNC(C2CCC3(CCC3)C2)=O)CCCN(C(C2(F)CC2)=O)C1 N1(C(C2(C)CC(C)C2)=O)CCN(CC2CN(C(=O)CCc3cncn3C)C2)CC1 C1(NC(C=CC=CC)=O)CCN(C(c2ccc(C(C)=O)o2)=O)CC1F c12ccc(cc1)c1ccc(nc1)[nH]c2=O.CC1(C(=O)Nc2ccccn2)CCCC1 C1(C(N(CC(=O)NCC2C=CCOC2)C)=O)CCCC1(F)F C1(C(N(C2CCCCC2)C)=O)CNC(=O)CN1C(C1C2CC(=O)CC12)=O c1(C(N(C)CC2N(C(C(CC)OCC)=O)CCC2)=O)cccc(C2(O)COC2)c1 c1(C(=O)NC2C=CCN(C(c3c(=N)[nH][nH]c3)=O)C2)cc(Cl)c(F)c(Cl)c1 C=CCC(CNC(=O)C(C)(C)C1(O)CCC1)C(=O)NC(c1ccsc1)C c1(C(=O)NCCNC(c2cnc(-c3ccoc3)s2)=O)cnc2c(Cl)cccn12 CCCCCCOC(C)C(=O)NCC1CCN1C(c1ccnn1CC)=O c1(OC)cc(=NC(=O)c2n[nH]c3cc(-c4cnn(CCO)c4)ccc23)[nH]c(Cl)n1 c1(C(C)=O)ccc(=NCc2nc(C)c(COC)o2)[nH]c1Br C1(NC(c2c(CC)c[nH]n2)=O)CC2(C1)CC(CNC(C1CCC(C)O1)=O)C2 C1(NC(=O)NCCN(CCN(C(C)=O)CC)C)(CO)CC2CCC1CC2 c1(C(N2CCC(C(C)NC(C3(CCC)CCC3)=O)C2)=O)ccc2nc(O)sc2c1 CC1CCC(CNC(c2cc(Cl)cn2C)=O)CN1C(c1cc2ccsc2s1)=O C1(CC(=O)NC(C)CC2CN(C(=O)CN(C)C3CC3)C2)CC=CCC1 C(=O)(C1=CC2CCC1C2)NCCNC(C1(C)CC1)=O.N12CSCC1C2=O CC1CN(C(c2cc(C3CC3)ccn2)=O)CCC1NC(c1cc(C(N)=O)cs1)=O N1(C(c2cccc(C)n2)=O)CCC2(CNC(=O)CC(F)(F)C(F)F)CCCCC12 C(=O)(C(O)C(F)F)NC(CCNC(COCc1c(C)ncs1)=O)(C)C c1(CC)[nH]nc(Cl)c1C(=O)NCC(C(C)(C)C)NC(=O)CC(C)(C)C1CC1(Cl)Cl c1(C(N2CC(C)C(NC(=O)COCC3CC3)CC2)=O)cc2scc(Br)c2[nH]1 N1(C(C=CCCC)=O)CC(NC(=O)COc2ccc(Cl)cn2)C(CC)C1 CN=c1cc(C(=O)NC2(CNC(=O)C(C)C3CCOC3)CCCCC2)cc[nH]1 C1(C(=O)NCC(C)(C2CC2)NC(c2coc(Cl)n2)=O)Cc2ccccc2S1 Cc1c(CC(=O)N(CCCC(=O)N(C2CCOC(C)C2)C)C)ncn1C C(N=c1[nH]cncc1I)C1C(NC(=O)CCc2cccc(O)n2)CCC1 c1(OCC(N2CC(O)(C)C2)=O)cncc(C)n1.c12c[nH]nc1NC2=O.CC O=C(C1=CCN(C(c2ccc(F)c(O)c2)=O)C1)NCC1CCOC1 c1(C(N2CC3C(CNC(C4CC5(CC5)CO4)=O)C3C2)=O)cnc2[nH]c(O)nc2c1 CCC(CCC(=O)N(C)Cc1cncn1C)NC(=O)C(O)CC1CCCC1 C(CCCCCC(=O)NCCCCC1CCN(C(=O)C2=CCCS2)CC1)SC c1(C(=O)NC(c2cccc(C)c2)CNC(CN(C)CC)=O)nc(Cl)c(Cl)s1 CCC(CC(=O)N1CCN(C(CNC(=O)C=Cc2cncs2)C)CC1)C(C)(C)C c1(SCC)c(C)c[nH]c1C(=O)NCC(C)(C1CC1)NC(C(C)NC(=O)OC)=O c1(C(N2CCCC2CCO)C(=O)NC(C(=O)OC)CC)ccc(F)cc1 c1(C(N2CCC(C(=O)N(CCO)CC)CC2)=O)cc2c(s1)-c1ccccc1OC2 C1(C(N2CCCCC(N(C)C(C34CC5CC3C4C5O)=O)C2)=O)CC2(CCOC2)C1 N1(C(=O)C=CCF)CCCC2(C1)CN(C(c1nscc1Br)=O)CCO2 C1(C(N2CC(F)(CC(=O)NC3(C4CCC4)CC3)C2)=O)CC1C1CCCC1 c1(CN2CC(CC(F)(F)F)(NC(c3csc(C4CC4)n3)=O)C2)cc(F)ccc1F Cn1nc(C(=O)OCc2ccn(-c3ccc(Cl)cc3)n2)cc1Cc1ccccc1 N1(C(C(CC#C)C2CC2)=O)CCC2CCCC12C(=O)NCCc1csnn1 N1(C(c2cc(CC)sn2)=O)CC(CNC(c2ncccc2C)=O)C(F)(F)C1 c1(C(=O)NCCCCN(C)C(C2CN(c3nncs3)C2)=O)cnn(CC2CC2)c1 C(=O)(CN(C)NC(=O)c1nccs1)N1CCCC(c2onc(CC)n2)C1 O=[N+]([O-])c1ccncc1NC1CCC1 C1(O)(CCNC(C2CCC(OC)C2)=O)CCN(C(c2coc(C(N)=O)c2)=O)CC1 N1(C(C2(CC#C)CC2)=O)CCCC1CN(C(=O)CSc1ccncc1)C C1(N(C(=O)Cn2cnnc2O)C)CCN(C(=O)Cc2cnc[nH]2)CC1CO c1(C(=O)NC(C2CCCN(C(COC)=O)C2)C)cc(O)nc2c(F)cc(C)cc12 c1(CC)cc(C)ccc1C(=O)NCCC(C)(C)NC(c1csc(CO)n1)=O C(=O)(CCCCC(=O)NCC1(F)CCC(CNC(=O)Cc2ccoc2)CC1)NC C12(NC(CC(CCC)C)=O)CC(C)(C1)OC21CN(C(=O)Cc2ccnnc2O)C1 CC1(C)C(CNC(C2(C(F)F)CCCC2)=O)CCN1C(=O)Cc1cccs1 N1(C(CNC(C2CC(C)C2)=O)C)CCN(C(=O)Cn2cnc(=N)[nH]2)CC1 N1(C(c2c(C)oc(Cl)n2)=O)CCN(C(c2ccccc2F)=O)CC1CC(C)(C)C CCCCC(C)C(=O)N(CC(C)NC(=O)CC1CCOC(C)(C)C1)C C(=O)(CC(C)(C)CNC(c1ccccc1F)=O)NC1(CC=C)CC1 C1(C(N2CCCC(c3nc(C4CC4)no3)C2)C(=O)NCCOC)CCCC(C)(C)C1 C1(NC(CSc2n(C)nnn2)=O)CC(F)CN(C(=O)CCc2cnco2)C1 C1(CC(=O)NC2CCN(C(CCOCC(C)C)=O)CC2)CC(C)(C)CCO1 S(=O)(=O)(c1cccs1)NCC(N1CCC(CC=C)(NC(=O)C=CS(C)=O)C1)=O c1(OC)cc(C(N2CCN(C(=O)Cn3nc(C)ccc3=O)C3CC23)=O)cc(Cl)n1 C1(C(=O)NCCC2C(C)C2)C2CC(O)C(C2)N1C(c1cnc(Cl)s1)=O CC(CC(=O)N1CCC(C(=O)NCC2CCCO2)CC1)C(F)F C1(C(=O)NCCC=C)CCCN(C(=O)CN(C)C(=O)OC)C1 c1(C(=O)NCCC2CCN(C(c3c(C)noc3)=O)CC2)cc2n(n1)CCCC2O C1(NC(C(C2CC2)NC(c2cccc(CO)c2)=O)=O)CC12CCCCC2 C1(C(c2nnnn2CCCF)NC(CCSC)C)CC2(C1)OCCO2 N1(C(C2(F)CN(C(c3cc(OCC)no3)=O)C2)=O)CCSCC1C1CC1 c1(N2C(NC(N3CC(C)C(O)CC3)=O)CC3(CC3)C2)ncc2c(n1)CCC2 N1(C(CC=C)=O)CC(CCNC(C2CCCN(C)C2)=O)C(C)C1 C(C)(CCCCC)NC(COCC=C)=O.N12CC(C1)OCC2=O C1(C(N2CCC(CN(C(C3(CSC)CCC3)=O)C)C2)=O)CCN(C)C1=O c1(CNC(C(C(C)NC(c2c(CC)ocn2)=O)C)=O)ncc(C)cc1C C1(CNC(C(C)Cc2ccco2)=O)CCN(C(c2cn3ccnc3s2)=O)C12CC2 c1(C(N2CC(Cn3cc(CCCOC)nn3)C2)=O)ccc(C)cc1F C1(C(C)C)CN(C(=O)C(N2CCOCC2)C)CC1C(=O)NCC1(C#N)CCC1 C=CC1(O)CN(C(=O)C(O)CNC(C2(C)CCCS2)=O)C1 C1(NC(c2cc(C)oc2C)=O)CC2CN(C(=O)CC3CCC(=O)C3)CC2C1 c1(C(=O)NC2CC(F)(F)CC2NC(C2CC=CC2)=O)cc(Cl)cc(Cl)c1O CCC(CC(F)(F)F)C(=O)NC1CC(F)CN(C(c2ccc(C)cc2)=O)C1 CC1CC(CNC(=O)C(O)C2CCCC2)CCN1C(=O)Cc1cnnn1C C1(C(=O)NCC(C)(C)OCC(=O)NCC#C)CCCN1CC1CCC1 C(=O)(CCP(C)(C)=O)N(CCCNC(=O)C(C)CC1CCCC1)CC CS(=O)(=O)CCCC(=O)NNC(=O)NC1CCC(O)CC1 N1(C(CC(CC)C)=O)CC(C2CN(C(c3nc(Cl)sc3C)=O)C2)C1 C(CS(=O)(=O)CC(=O)N1CCN(C(c2cccnc2OC)=O)C(C2CC2)C1)OC C1(NC(=O)CCn2cc(C(N(C3CCC3)C)=O)nn2)CCCCC1 C1(NC(C=CCN(C)C)=O)CCN(C(c2c[nH]cc2C(C)(C)C)=O)CC(C)(C)C1 N1(C(C(C)(C)c2cccnc2)=O)CC2(CC(NC(=O)CC3CS(=O)(=O)C3)CO2)C1 c1(C(=O)NC(CCCC)c2nnnn2C2CCCCC2)cnc(C)c(C#N)c1 c1(CC(N2CC(C=C)C(NC(=O)C(C)(O)C(C)C)C2)=O)cccc([N+](=O)[O-])c1C C1(C(=O)NC2CN(C)C2)CCCN1C(C1CC1F)=O C(=O)(C(O)CCC(C)C)NCC(C(=O)NC(c1ccco1)COC)N(C)C C(=O)(CCP(C)(C)=O)N1C(CNC(CC2(C(=O)OC)CCOCC2)=O)CCC1 CCC(C)C(C(=O)N1C2CCC1C(CNC(C1(N3CCOCC3)CC1)=O)C2)OC C12(NC(C3CC(NC(CNC(=O)CC4CC5(CC5)C4)=O)C3)=O)CC1COC21CCC1 c1(N(C)Cc2cccc(Br)c2C)cc(NCCSC)nc(C(F)(F)F)n1 N1(C(CSCC(=O)OC)=O)CCCC1C1CCCN1C(=O)C(C)n1cccn1 N1(C(C2(C)C(C)CCC2)=O)CC2CCC(N(C(=O)C(F)=CC3CC3)C)C2C1 N1(C(C(CO)OC)=O)C(C(=O)N(C)C(c2ccccc2)C)CC2CC12 c1(CNC(C2(CNC(c3cn(C)nc3)=O)CCC2)=O)cccnc1Br c1(C(C2(NC(c3cnc(C4CCC(=O)N4)s3)=O)CC2)=O)ccc(Br)cc1 C(CC(=O)NCC1C2CCCCCC12)(C(F)(F)F)NC(c1cnn[nH]1)=O Cc1ccccc1C1(N2CC(n3cc(C4(C)CCCO4)nn3)C2)CCCCC1 C1(C(=O)NCc2[nH]nc(COC)n2)CC(C)(C)CCN1C(c1ccnnc1C)=O C(C(=O)NCC12CC(NC(C3CCCC(C)CC3)=O)(CCO1)C2)(C(C)(C)C)SC N1(C(=O)Cc2cnns2)CC2OCCN(C(c3cn(C4COC4)nn3)=O)C2C1 c1(C(=O)OC)ccnnc1N(C)C(C12CC(NC(=O)C(c3ccccc3)F)(C1)C2)=O C1(CC=C)(C(=O)NCc2ncoc2C)CCCN1C(=O)CC(=O)NC1CC1 C1(CNC(c2c(CC)csc2)=O)CCCC2(CC2)C1.c12cc(c(C)s1)CNC2=O N1(C(c2ccc(Cl)nn2)=O)CC2CC(C1)CN(C(C1(Br)CCC1)=O)C2 c1(CNCC2CCC(O)C2)noc(CCc2ccccc2)c1Cl Cc1cccc(CC(=O)NC2CC2CNC(=O)CC2(O)CCOCC2)c1F c1(C(=O)NC(C(C)NC(C=CCCC)=O)CO)cc2ncc(C(C)C)cc2[nH]1 c1(CN(S(=O)(=O)CC2C3CCCCC23)C)ccc2oc(O)nc2c1 N1(c2cc(SC)ncn2)CCC2(CC1)CC(NC(=O)Cn1nnc(=N)[nH]1)CCO2 C1(NC(c2cnn(CC)n2)=O)CC2(C1)CC2NC(c1cnc(SC)[nH]1)=O N#CC1(C(=O)NC(C=C2CN3CCC2CC3)C(=O)O)CC2(CC2)C1 N1(C(C(C)OCCOC)=O)CC(n2ccnn2)C(C)(C)C1.C12CCCC1C(=O)N2 C1(C(=O)Nc2c(C(=O)OC)scc2)C=CCN(C(C2CC23CC(O)C3)=O)C1 C1(C)(C(=O)OC(C)(C)C)CCCN1OC(c1nc(C(CCCC2CC2)C)on1)=O c1(C(N2CC(CNC(=O)Cc3ccnc(F)c3)C2)=O)cn2c(n1)CCCC2 c1(NCC2CC(C)C2)ccc(S(=O)(=O)NCC2(C)CCCCO2)cc1Br C1(C(=O)NCC2C3CN(C(CCCCOC)=O)C2C3)C2Cc3ccccc3C12 C1(CC)CN(C(c2cc(C#N)cn2C)=O)CCC1CNC(=O)C=Cc1cncs1 C(CN=c1cc(NC(c2ccc3c(c2)NC(=O)C3)C)nc(C)[nH]1)C1(OC)CCC1 C=C(Cl)CC(C(=O)NCC1CCCN1C(C)=O)NC(=O)C1=CCCC1 C=CCC(C(=O)N1CCC(CNC(c2ccn(-c3ccncc3)n2)=O)C1)C(C)C C12(C(=O)NCCN(CCC)C(c3cc(COC)on3)=O)CCOCC1C2 c1(C(=O)NC(c2ccc(C)cc2)C(O)C2CC2)ccc(C)c([N+](=O)[O-])c1 C(=O)(C#CC1(C)CCCO1)N(CCCN(C(c1ccc(C)c(C)c1)=O)CCO)CC Cc1cccc(F)c1CC(N1CC(NC(C2(O)CC2)=O)CC(O)C1)=O Cc1ccnc2ccc(C(=O)NC3CN(C(C4CCCNS4(=O)=O)=O)C3)cc12 c1(C(=O)NC(C(=O)NC(CCCC)CO)CCC2CCC2)cc(C)c(F)cn1 C1(OC)CCC(C(N2CCC(CCC(=O)NCC3(C)CC(O)C3)C2)=O)C1 C12(C(N3CCN(CCN(C)C(c4cnn(C)c4N)=O)CC3)=O)CCCC(C1)OC2 CC1(NC(C2CCCS2)=O)CCC(NC(=O)CCc2cccnc2)CC1 C(=O)(CCCCC(C)(C)C)NC(CCNC(c1cc(C)c(F)cn1)=O)C C1(CC(=O)NCC(C)NC(C2C=CCS2)=O)CCC(C)(C)C1 C(C#Cc1cn(-c2ccc(F)cc2)nn1)NC(C(C)CCc1ccc(F)cc1)=O N1(C(C2N(CC)CC2)=O)CCN(C(c2coc(CSC)c2)=O)C(CO)C1 O=C(Cc1ccc(F)cc1)NNC(=O)c1ncoc1Br C=CC(C)(CC)C(=O)N(C1CCC(CNC(=O)C(C)(C)CCC)CC1)C C1(C(C(=O)N2CCC2)F)CCN(C(=O)Cc2cncnc2)CC1.C1(N)CC1 CCCC(CCCNC(C1SCC=C1C)=O)NC(c1coc(C(N)=O)c1)=O N1(C(c2n(CC)ccc2)=O)CC(CC(=O)N(CC(F)F)CCO)C(C)C1 Cc1cccc(C2CC2C(=O)NCCCCN(C)C(c2cnc(N(C)C)s2)=O)c1 c1(NCc2cnn(Cc3ccccc3)c2)ccc(Br)nc1I.C12CCN1C2=O c1(CCNC(=O)Cn2cncn2)ocnc1CNC(=O)CC1CCC2CC12 C1(NC(C2(OC)CCC2)=O)CCCCN(C(c2snnc2C)=O)C1 N1(C(CC2(NC(C3CC34CCC4)=O)CC2)=O)CCC2(CC2)C1 C12(C(=O)NC3(CF)CC(F)(F)C3)OC3C4C5CC(C6C5C3C16)C24.C1(CO)C(=O)N1C.CO C=CCC(C)(C)CC(=O)N1CC(NC(=O)C(C(C)(C)C)NC(=O)OC)C2(CC2)C1 c1(C(=O)NCC2CC3CC2CN3C(C2CC2F)=O)cc2cnc(Cl)cc2s1 Cc1cccc2c1c(CC(N1CCC3(CC3C(=O)NC3CC(C)C3)C1)=O)cn2C C1(C(N2CCCC(CC=C)C2)=O)CCC2(CCNC2=O)CC1 C1(C(=O)NCC(C)CN(C)C(c2ccccc2SC(F)F)=O)CCCCN1C CC(C)(CC(=O)NCC1C2CN(C(=O)Cc3cnns3)CC12)C(F)(F)F c1(C(N2CC(CC)C(C(=O)NC3CNC(=O)C3(C)C)C2)=O)ccc(C)cc1O Cc1nnc2n1C(C(=O)NC(CNC(=O)Cc1cncn1C1CC1)C1CC1)CC2 N1(c2nnc(C)s2)CC2C(CN(C(=O)CC3CC34CC4)C(c3ccccc3)=O)C2C1 C1(C(N2CCN(CCCNC(CC(C)(C)OC)=O)CC2)=O)CC12CC(C)(C)C2 C1(CC)CN(C(=O)C(C)(C)c2ccccn2)CCC1NC(=O)CCC(C)OC C(=O)(CC(C)(C)C)N.C1(CNC(=O)CC2CC2)CC(CNC(C2CC(CC)C2)=O)CO1 N1(C(c2c(C)n[nH]c2C)=O)CC(NC(=O)CC2OCCC2(C)C)CC2(CCC2)C1 c1(OC)nccc(C)c1NC(=O)CC1CCCN(C(c2cc(Cl)c(Cl)s2)=O)C1 N1(C(C2(F)CCCCC2)=O)CC2(CCCCN2C(=O)C(C2CCOCC2)O)C1 c12nc(nc(=N)[nH]1)C(CCCC)SCCCC(C1C(C)C1)NC(=O)N2 C=Cc1cc(C(N2CCN(C(=O)CC3CCS(=O)(=O)C3)C(CO)C2)=O)cc(F)c1 CC(C)CC(O)C(=O)NC1CC(O)(CNC(c2cc(C3CC3)[nH]c2C2CC2)=O)C1 c1(CCC(=O)N(C2CCCC2)CCNC(c2ncccn2)=O)ccncn1 c1(C(=O)NCC(C)CN(C)C(C2(CCF)CC2)=O)cccc(Br)c1Cl c1(C(=O)NC(C2CN(C(c3sccc3C#N)=O)CCO2)C)cnc2n1CCS2 C1(C(=O)NCCCCCNC(C2CC(C)OC2)=O)CN2CCN1C(C)C2 C(=O)(C(C)C(C)NC(=O)CCCF)OC.c12cccc(c1)NC(=O)C2 CC(C)C(C(=O)N1CCCC1CN(C)C(C1(C)CC1Br)=O)n1cnnn1 N1(C(c2ccns2)=O)CCC2(CC1)CN(c1ccnc(Br)n1)C2 c1(C(N(CCN(C(CN(CC)CC)=O)C)C)=O)nn(C)c2c1CCCC2.C1CO1 C=CC(C)(C)CC(=O)NC1CC(C(F)C(=O)NC(CCO)C(C)C)C1 n1(CC(N2CC(C)(NC(c3c(OCC#C)nccc3)=O)C2)=O)cc([N+](=O)[O-])cn1 N1(C(C2(C(N(C)C)=O)CC2)=O)CCC(N(c2ncc(I)cn2)C)CC1 N1(C(N(CCC)OC)=O)CCC2CCN(C(=O)CCC3CCC(=O)C3)CC12 O=C(C1=CC2(CCOCC2)C1)NC1CC2(C1)CC2NC(=O)Cc1ccnnc1O C1(OC)CC2(CCC(C(=O)NC3CC(NC(c4ccccn4)=O)C3)CC2)C1 N12CCCCC1C(=O)OCCC2=O.n12cc(nn1)C(=O)N1CC2C1.CCC(=O)O N1(C(C(C)C)=O)CCC(C)C1CNC(C12CCC(CC1)C2)=O N1(C(CS(C)(=O)=O)=O)CCC2(C1)CN(C(C1COCC(O)C1)=O)C2 CCC1=NOC(c2nc(C34CC(CN3C(=O)CC(C)CO)C4)no2)C1 c1(C(=O)NC2CCN(CC(CCC)OC)CC2)cnc2[nH]c(C)nc2c1 c1(C(=O)NC(C(C)OC(C)CN(C)C(C2CCC2)=O)=O)ccc2nc(=N)[nH]n2c1 C1(NC(C(C)C2CCC2)=O)CN(C(=O)CCCCCc2ccccc2)CC1(C)C c1(CC)nscc1NC(=O)CC1CCCN1C(=O)CCc1cn[nH]c1 N1(C(C(CC)OC)=O)CC(N(C)C(C2CN3CCC2CC3)=O)C2(CC2)C1 CC1COc2c(C(=O)NC3CC(NC(c4cc5ccncc5[nH]4)=O)C3)cnn2C1 CC1=NS(=O)(=O)N(C)C=C1C(=O)NC1CC1CNC(C1CC2(C1)CC(O)C2)=O C1(C(=O)NC(c2ccccc2)C(=O)NC(CCN(CC)CC)C)CCCSC1C N1(C(c2ccc(CC)[nH]2)=O)CC2CC(C1)N(C(C1COC3COCC3O1)=O)C2 C(C(C(C)C(C)C)NC(=O)CCc1cnc(O)[nH]1)NC(COCCC)=O C(=O)(C1=NN(C)C(=O)CC1)N1CC2C(NC(c3ccc(C)c(C)c3)=O)CC(C2)C1 C1(CC)CN(C=Cc2ccccc2OC)CCN1C(c1cccc(C)c1O)=O c1(C(N(C2CCCN(C(C(C)N(C(C)=O)C)=O)C2)CCO)=O)cc(C#N)ccc1C C12(C(N3CC(C)N(C(=O)C=Cc4cncn4C)CC3)=O)CCC(CC1)C(C)O2 c1(C(N(C2CCC(NC(=O)Cc3ccco3)C2)C)=O)c(N)cc(F)cc1F c1(C(C)(C)C)ccc(CNC(=O)NOCCCCC(C)(C)C)cc1 C1(C#N)(C(N2CCC(CNC(c3ccc(SC)cc3)=O)CC2)=O)CC2(CC2)C1 CCC(C(=O)N1CCN(C(=O)Cc2cnn(C3CC3)c2)C(C)C1)C(C)(C)CC N1(CC)CCC(N(C(=O)C(N2CCC(c3nc[nH]n3)CC2)=O)C)CC1C C12(NC(CC(C)F)=O)CCCC1N(C(C1(c3ccc(Br)cc3)CCCC1)=O)CC2 C(c1c(C)coc1C)=CC(=O)NCC1(F)CCC(NC(C=CC=CC=CC)=O)C1 N1(C(c2ccn(CC)c2C)=O)CCOC2(C1)CN(C(=O)CC(C)F)C2 O=C1Nc2ccc(F)cc2CC1C(N1CCN(Cc2ccccc2O)CC1)=O c1(SC)cc(C(N2CCC(NC(C3CC(OC(F)F)C3)=O)C(F)C2)=O)ccc1F Cc1[nH]c2ncccc2c1C(=O)NC1CC(NC(=O)C#CC2CC2)C1 c1(CNC(N2C(c3ccc(C)c(N(C)C)c3)CCC2)=O)cccc2c[nH]nc12 c1(C(=O)NCC(CNC(c2c(C)cnnc2)=O)O)cc2c(F)cc(Cl)cc2[nH]1 C1(C(=O)NCC(C)NC(C(C(C)C)F)=O)CC(=O)OC1(C)C C12(C(=O)NC(C)(CNC(=O)C(C3CCCCC3)=O)C3CCC3)CCCC1CCC2 C(CC(=O)OC)N(C1CN(C(=O)C(C)=C(C)C)C1)CCC c1(C(=O)NCC2(CO)CC2)cn(C2CCC(CO)C2)nn1.C1(C)CC1 c1(OC)cc(N)c(C(N2CCC(NC(c3cncs3)=O)C(CO)CC2)=O)c(F)c1 CS(=O)(=O)C1CN(C(c2ccc(C(F)(F)F)o2)=O)C2(CCC2)C1 C12(CN3CCN(CN4CC(O)C(c5ccc(Br)cc5)C4)CC3)CCC(CC1)OC2 c1(OC)cc(C(=O)NCCC(C(C)C)NC(C2(OC(C)=O)CC2)=O)ccc1O C1(C)(CC)CN(C(C2CC2C(C)NC(=O)C(C)N=[N+]=[N-])=O)CC1C CC1C(C(=O)NCC(C(C)(C)C)NC(c2nccc(Cl)c2F)=O)=NOC1C N1(C(C(CCC)F)=O)CCC2(CC(NC(=O)CC3CC3c3ccccc3)C2)C1 C1(NC(CN(CCC#C)C)=O)CCN(C(c2ccc(COC)nc2)=O)C(C)C1 C(=O)(CCCCCC(C)(C)C)NCC1CC(NC(c2c(OC)nsc2)=O)C1(C)C C(=O)(C(C(=O)N(CCCCCCNC(C)(C)C)C)SC)OC.C(C)(=O)O C1(NC(c2cc(CC)c(F)cc2)=O)CCN(C(=O)C2=CCCCC2C)CC1(C)C C1(CNC(C=CC(C)C)=O)CC2CN(C(c3ccc(-c4ccccn4)s3)=O)CC12 C1(C(=O)NCC(CC)O)C(CC)CCCN1C(c1ccc(=N)[nH]c1)=O C1(C(N2CCC(N(C(=O)C=CC(C)(C)SC)CC)C2)=O)CCC2CCCCC2C1 Cc1ccc(Br)c(N)c1C(=O)NC(C)CNC(c1cnc[nH]1)=O C1(C(=O)NC2CC3C(NC(C(C)=C4CCC4)=O)C3C2)CC(=O)C12CCCC2 Cc1cn(CC(N2CCCC(C(=O)N)(CO)C2)=O)c2ccccc12.c1(CO)ccoc1 c1(CCC)cc(O)nc(CC(=O)NCC2SCCS2)n1 N1(C(=O)C=CSc2ccccc2)CCN(C(C2CCCC2c2nc[nH]n2)=O)CC1 c1(C(=O)NCCC(C)(C)NC(=O)CC2CCCC(F)(F)C2)cncc2c[nH]nc12 c1(NC(c2c(C)nc(NC(=O)CCCN(C)C)s2)=O)cc(O)ncc1Br c1(C(N2CC(N(C(C(C)N(C)C)=O)C)C2)=O)cc(C2CC2)cc(F)c1 N1(C(C=CC(C)C)=O)CCCC1CCNC(c1cc(Cl)cs1)=O C1(CS(C)=O)CC2CCC(C1)N2C(c1cn(CC2(c3ccncc3)CC2)nn1)=O C#CCCCCCC(=O)NC(CC(=O)Nc1ccc(N(C)C)cc1)C(F)(F)F C(=O)(CCC(C)(C)F)N1CCC(N(C(=O)CSc2nnc(N)s2)CC)C1 N1(C(C(CCC=C)NC(C)=O)=O)CCN(C(=O)C(O)COC)C2(CCC2)C1 c1(N2CCC(NC(c3c(SC)nn(C)c3)=O)C(F)C2)cc2ncnn2cn1 c1(C(=O)NCCCC2N(C(COCC=C(C)C)=O)CCC2)cc(C)n(C2CC2)n1 C(=O)(C1=CC(O)C(NC(=O)CC2=CCOCC2)C1)NC1(C(=O)OC)CC1 C1(CC(=O)NC(C)CNC(=O)COCCn2cncn2)COCC1O Cc1cc(CC(N2CCC(OCCNC(=O)CSC(F)F)C2)=O)cc(C)c1 C1(CNC(=O)COCCn2nccc2C(=O)NC)COCCN1C(c1ccco1)=O C1(C(=O)NCc2nnc(C)s2)CC(C)(C)CCN1C(=O)CC1=CCOCC1 c1(SC(C)CC(=O)NCCC(C)(C)NC(=O)CC2CCNC2=O)ccc(Cl)cc1 C(CNC(C1(NC(C2CC(F)C2)=O)CC1(C)C)=O)(C(C)C)OC c1(C(N2CCCC3(NC(=O)CC4CC=CC4)C(C2)C3)=O)nnc2n1CCCCC2 c1(C(=O)NCCCNC(=O)CCOCC2CCCO2)cccc(C(F)F)c1F c1(C(N2CCCC(O)(CNC(CNC(C)=O)=O)CC2)=O)cnc2n1CCC(C)C2 C1(NC(C2C(OCC)C2C)=O)CCN(C(=O)COc2cccc(Cl)c2)CCC1CO C1(C(=O)NCC2C(NC(c3c(C(C)C)nns3)=O)C2)OCCOC1(C)C N1(C(CCN(C)C)=O)CC2COCC(C1)N2C(c1cc(O)ccc1I)=O c1(N(CC(=O)NCCCC)C)nc2ccccc2c(C)c1C(=O)OCCOC N1(C(C2C(C)=CCS2)=O)CC2CCC1CC2NC(=O)CCC(N)=O Cc1ccc(CCC(=O)N(C)CC2CCN(C(C3SCCS3)=O)C2)cc1C C1(C(CO)NC(CSCCOC)=O)CCN(C(c2ccc(=O)oc2)=O)CC1 C(CCCCCCCF)NC1OCCN(C(=O)OCC(C)C)C1 CCC(C)C(O)C(=O)NCC(CC(=O)N(C1CC(C)(C)C1)C)OC C1(C(N)=O)(NC)CCN(N2CCCC(CCc3ccccc3)C2)CC1 c1(NC(C)=O)cnc(O)c(C(N2CC(CO)(NC(C3CCC(=O)N3)=O)C2)=O)c1 Cn1nc(C(N2CCC(CO)C(NC(=O)Cc3ccc(O)nc3)C2)=O)c(Cl)c1Cl C(=O)(C1=CC2CCCC12)NC12CC(CNC(C(C)CN(C)C)=O)(C1)C2 C(=O)(CN1C(=O)CCCc2sccc21)N1CC(NC(=O)C#CC2CCC2)C(O)C1 c1(C(=O)NC2(CF)CN(C(C(C)OCC)=O)C2)cn2c(n1)CCC(C)C2 C=CC(CCC)CC(=O)N(NC(C1CCC(C)CC1)=O)CC.c1(N)cc(F)ccc1F N1(c2ncc(C)cn2)CC(NC(=O)C=Cc2cncn2C)CCC1C c1(C(N(C(C)C(N2CCC(C#N)C2)=O)CC)=O)[nH]ccc(=O)c1C c1(CC(=O)N(CC(C)NC(C2(C#N)CC(=O)C2)=O)C)c[nH]c2cc(Cl)ccc12 C1(NC(=O)C=Cc2ccco2)CC(O)CN(C(c2cnn3c2CCC3)=O)C1 Cc1cc(N)c(C(=O)N(C)CCNC(=O)CCc2nnc(S)nc2O)c(F)c1 Cc1c(C(=O)NC23CCCN(C(=O)Cn4ccsc4=N)CC2C3)sc2nccn12 C1(CNC(=O)Nc2n(C)nc(C)c2Br)CCC2(CCOC2)O1 N1(C(C2(OCC)CCOC2)=O)CCC(CO)(CNC(C2CC(C)=NO2)=O)CC1 Cc1nc2ncnn2c(C)c1CC(=O)NC1(CNC(C2CC2C(F)F)=O)CCC1 c1(CN2C(C(=O)Nc3cnc(Br)c(F)c3)CCC2)ccc(O)c2ncccc12 C1(C(N2C(C(N(CCCCC=C)C)=O)COCC2)C2CCC2)CC2(C1)CC(O)C2 c1(C(=O)NC(C2(O)CN(C(C3CC(C(=O)OC)C3)=O)C2)C)c[nH]c(=N)nc1C c1(C(=O)NC2CN(c3ncc(OC)cn3)CC2C#N)cc([N+](=O)[O-])c(C)cc1C CC1CN(C(=O)Cc2ccn(C)n2)CCC1CNC(=O)C(C)(C)CC#N N1(C(c2c(C(C)=CC)noc2)=O)CCCC12CCN(C(c1cc(C)cc(F)c1)=O)C2 c1(C(N2CCC(C3N(C(C(C)C4CCC4)=O)CCC3)C2)=O)ccn2nccc2n1 c12cc3cc(ccc3[nH]1)S2.c12sccc1C(=O)NC2.C1(C(=O)OC)CC1C(=O)OC C(CC(C)(C)C(=O)NC(C1CCN(C(=O)C(C(C)C)NC(C)=O)CC1)C)OC c1(NC(=O)CC2CCN(C(c3ccc(F)nc3)=O)C2)ncnc(Cl)c1Cl n1(CC)nc(C)c(C(=O)NC2CC2NC(C2(CC3CC3)CCCO2)=O)c1C CS(=O)(=O)CCCCCNC(=O)C(O)Cn1cncn1 N1(C(=O)CC=Cc2ccsc2)CCC(c2ccccc2)C(O)C1 c12nccc(Cl)c1CN1CCC1(C)C(=O)N2.N1(CC)CC2CC1CN2C C1(NC(C(N)=O)=O)CCC(O)CN(C(=O)CNC(=O)NC2CCOCC2)C1 c1(C(N2CC3C(CCNC(CC(CC)(F)F)=O)(CC3)C2)=O)ccn2ccccc12 C1(CCNC(CCC(=O)NC)=O)CCN(C(=O)C(C)(C)C2CC2)CC1C C#CC1CCC(C(N2CCC(CNC(=O)C=Cc3cnccn3)C(C)C2)=O)CC1 CC1(C)C(C(=O)NCCCC2(NC(=O)CC3CSCCO3)CC2)CC1O c1(CCCC(N2CCOCC2CC(n2ccnn2)=O)=O)cc(F)c(F)cc1F n1(CC)ccc(C(N2CCC(O)(Cn3cc(-c4cc[nH]n4)nn3)C2)=O)c1C N1(C(CSCC(=O)Nc2ccc(=O)oc2)=O)CCN(C(=O)CN2CCCC2)CC1 C1(CNC(C(C)NC(=O)NC)=O)CN(CC=Cc2cccs2)CCC1(F)F C(=O)(C(=O)C(C)(C)C)Nc1cccc(-n2cc(CC(=O)OCC)nn2)c1 c1(C(=O)NC(CCNC(CC(C=C)(C)O)=O)C(C)C)cc(F)cc2c1CCC2 C(=O)(C(=O)NC(C(=O)NCCc1ncon1)C1CC1)N(C)C Cc1oc(C)c(C(=O)NCC2OCCC2C(=O)NCC(C)C(=O)N(C)C)c1C C1(NC(c2ccc(C#C)cc2)=O)CC1C1CCN(C(=O)C(O)c2ccsc2)CC1 c1(NC(C(C)C)CN2CCCC2)nc(CO)c(Br)s1 N1(C(c2nnc(-c3ccncc3)o2)=O)CCC(O)C2(CCC2)C1 C(c1nnn(C)n1)=CC(N1C(CN(C(=O)CN2C(=O)CNC2=O)C)CCC1)=O C(=O)(C(=O)C(C)(C)C)N1CCN(C(=O)Cc2c(C(=O)OC(C)C)nco2)CC1 N1(C(CC(C)C2CC2)=O)CCC(N=c2nc(C(F)(F)F)[nH]s2)C2(CCC2)C1 c1(C(N2C(C)CCC(CO)C2)=O)cnc2ccccc2c1 CC1C=C(C(=O)NC(c2ccccc2)CNC(C2C3C4CCC(C4)C23)=O)CC1 Cc1ccc(OCCCC(=O)NC2CN(C(c3ccsc3)=O)CC2(C)C)cc1C C1(NC(Cc2ccn(CC)n2)=O)CCN(C(C2CCC=CCCC2)=O)C(C)C1 c1(C(N2C(C)(C)C(CNC(=O)C3=CCCO3)CC2)=O)cc2ccc(F)cc2o1 N1(C(C(C)(CO)OC)=O)CC(C2CCCN(C(c3scc(C)c3C)=O)C2)C1 O=C(NNc1ccc(Br)c2ccncc12)c1ccc(Br)cc1Cl Cc1cc(C)c(C(=O)NCC(C2CCCC2)NC(=O)C(N2CCCCCC2)C)s1 C12(C(CNC(C3CC3Cl)=O)NC(C=C(C(=O)OC)C)=O)CCC(CC1)C2 c1(OC)ccsc1C(=O)N(CCNC(c1coc(-c2cccnc2)n1)=O)C(C)C N1(C(c2c(NC(C)=O)sc(Cl)c2)=O)CCCC(NC(=O)CN2CC(C)(OC)C2)C1C C1(C(N2CCCC(CO)C2)=O)CCCN(Cc2ccncn2)C1 c1(OC)nc(N2C3CC2CN(Cc2c(C)cccc2C)C3)ncc1Br c1(C(=O)NCC(CNC(C(=Cc2cccs2)C)=O)(C)C)cncc(S(C)(=O)=O)c1 C(=O)(C1CCCc2n[nH]cc21)NC(CNC(c1cc(OC)ncc1Cl)=O)C(C)C N1(C(CNC(C2C(C)C2)=O)=O)CC2CN(C(=O)CC34CCC(CC3)C4)CC2C1 Cc1cn2c(n1)CC(C(=O)NC(C)CNC(=O)COC(F)F)CC2 C(C(=O)N1CCC(C(N2CCC(C)(CCO)C2)=O)O1)(C(C)C)OC c1(CC)cc(C(=O)NC(C)(CO)C(=O)NCC2(C)CC(F)C2)n(C)n1 C1(C(=O)NC2C(CNC(C3(CC)CCCC3)=O)CCC2)CCC2(CCC2)CO1 C1(CNC(c2ccc(COC)o2)=O)CC(C)(C)CN1C(c1csc(Cl)c1OC)=O C1(CNC(CC(COC)C)=O)CC2CCC1N2C(=O)CC(=O)NCC1CC1 C(C)(CC(OC)OC)(c1n(CC(=C)C)nnn1)NC(C)(COC)C1CC1 CC1CCN(C(=O)C(C)(C)N(c2ncn(C(C)C)n2)S(C)(=O)=O)CC1 n1(CCC)cc(C(=O)N(C)CC2CCN(C(=O)CC3CCCCCC3)C2)c(C)n1 C1(C(=O)NCCCC)CCCN(C(=O)CC(C)(C)c2cccs2)CC1 C1(C(=O)NC(C)CN(C(=O)CCc2cnoc2)C)C2(CC2)C12CC2 C(c1nc(C)cs1)=CC(=O)NC1CCC(CNC(C(CC)F)=O)C1 c1(C(N(CC(CNC(C2(SC)CCC2)=O)C)C)=O)ccc(C(C)(F)F)cn1 CCC(F)(F)C(=O)NCCC1CCC(NC(c2csc(C)c2)=O)C1 N1(CC)CCC(CNC(c2n[nH]cc2CNC(c2ccc(C(C)=O)[nH]2)=O)=O)C1 CCC1=NOC(CC(=O)NCC2(CCNC(=O)CC(C)n3ccnc3)CC2)C1 C1(N(C(c2c(C)cno2)=O)C)CCN(C(C2CC(CC(C)(C)C)C2)=O)CC12CC2 N1(CC(=O)NCCOC)CCC(NC(C2(Br)CC2)=O)C(C)(C)C1 CC1=NS(=O)(=O)NC=C1C(=O)N1CCCC1(C)CNC(=O)CCc1ccc(C)o1 C1(NC(c2c(-c3cc(C)no3)n[nH]c2)=O)CN(C(=O)CCCC#N)CC12CCC2 N1(C(CN(C(=O)CC2CCCO2)C(C)C)=O)CCC2(CCOC2)CC1 C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)NC1(CCNC(C(C)O)=O)CCC1 C(CC(=O)NC(c1ncccc1F)C)(C(F)(F)F)NC(CCc1cc(C)on1)=O C1(C(=O)Nc2cccc(C(=O)NC(C)CN(C)C)n2)CCC(=O)N2CCCCC12 C12(NC(C(C)=CC)=O)CCN(C(c3nn(CCC)cc3Cl)=O)CC1C2 C1(CNC(CCCC#CC)=O)C(C2CC2)CCN1C(C1CCCC(F)C1)=O N1(C(C2C(C)OCCC2)=O)CCN(C(=O)CCn2cncn2)CC12CC2 c1(CNC(C=C(CC)CC)=O)cc[nH]c1C(=O)N(CC)Cc1ccccn1 c1(C(=O)NC2CCC(C)(CNC(=O)CC#N)CC2)cc(C#N)ccc1F N1(C(C(C)=C2CCC2)=O)CC2(CC(NC(c3cnc(-c4ccccc4)s3)=O)C2)C1 C1(C(=O)NCC2N(C(c3c(C)scc3)=O)CCOC2)CC(O)C12CCC2 c1(COC)ccc(C(=O)Nc2ccnn2-c2ccc(C)cc2)c(C(=O)OC)c1 CC1C(C(N2CC(F)C2)=O)CCN1C(C1CC2CC2C1)=O Cn1cc(C(=O)NCC(O)COCc2ccc(F)cc2)c(=O)c2cnn(C)c12 Cc1cncc(-c2cn(CCCNC(C3CCC(N(C)C)C3)=O)nn2)c1 c1(CN(CC(C)O)C)cc(Oc2ccccc2C)cc(C(F)(F)F)c1 CC(C)C(CO)NC(=O)C(c1ccccc1)NC(C1CC12CCC2)=O c1(C(=O)NC(c2ccccc2)CNC(C2CCSC2)=O)ccc(F)cc1F C(N=c1[nH]c(=NCCCN2CCc3ccccc3C2)c2ncccc2[nH]1)C1C(Br)C1 C1(NC(c2nc(Cl)cs2)=O)CC2C(NC(c3cc(F)c[nH]3)=O)C2C1 N1(C(c2n[nH]c(C)c2Cl)=O)CCC2CCN(C(=O)CN3C(=O)CN(C)C3=O)C2C1 N1(C(C(C(CC)(C)C)=O)=O)CCCC2(C1)CN(C(c1cnccc1Cl)=O)CCO2 Cc1cc2n(n1)CCN(C(c1cc(CNC(C3CC4CCC3CC4)=O)on1)=O)C2 c1(C(=O)NCc2cccc(CN3CCCC3)c2)cc2cc(F)cc(F)c2[nH]1 C(=O)(CC(C)(C)C(F)F)N1CC(CC(=O)NCCc2cc(C)no2)OCC1 N12CCN(CC1C)CCn1nccc1C(=O)N1CCCC1(C)C2=O.CO C1(COC)(NC(c2occ(C)c2C)=O)CCCN(C(c2ccc(CO)nc2)=O)C1 CC(CC(F)F)C(=O)N1CCC(N2CCN(C(C3(C4(C)CC4)CC3)=O)CC2)C1 N1(c2nc(COCC)nc(C)c2)CC(C)CN(C(C2(SC)CC2)=O)CC1C CC(C)P(=O)(CC(=O)NCC(F)CNC(c1cc2n(c1)CCC2)=O)C(C)C c1(C(=O)NC2CC(CNC(C34CCC(CC)(OC3)C4)=O)C2)coc2c1CCCC2 C(=O)(C1CCCc2sccc21)N(C(C)CNC(c1cc2c(Cl)nccc2o1)=O)C N#Cc1c[nH]c(C(=O)NC(C(=O)NCc2ncsn2)C2CCCO2)c1 c1(C(=O)NCC(C)(F)CNC(=O)CCc2ncco2)ccc(F)cn1 C1(C(N(C2CCN(C(=O)CCOCC(F)F)C2)CC#C)=O)CC12CCOCC2 C(=O)(CC(C(F)F)N1CCOCC1)NCC(CCCC)NC(C1CS(=O)(=O)C1)=O C1(CNC(C2(C)C=CCC2)=O)CCC2CN(C(=O)C=CCO)CCC2C1 c1(-c2n(CCC)nc(-c3ccc(Cl)s3)n2)cn2c(n1)SCC2 N1(C(C2C(C)C2C)=O)CCC2(CCN(C(c3ccc4sc(=N)[nH]c4c3)=O)C2)C1 c1(C(N2CCCC(n3cc(C4CCCC(C)C4)nn3)C2)=O)ccc([N+](=O)[O-])n1C N1(C(C(c2cnn(C)c2)OC)=O)CCC2(CCC(NC(=O)C(C)(C)F)CC2)CC1 CCC(CCC(=O)N1CCCC(N(C(c2cnc(OC(C)=O)s2)=O)CC)C1)OC CC1(C)CC(=O)NC1CN1CCCCC1.c12cc(cc(Br)c1)C(=O)N2 C1(NC(=O)CCc2ccon2)CN(C(c2ccc(F)c(CO)c2)=O)C2(CCC2)C1 c1(N(CCCNC(Cc2ncc(CC)[nH]2)=O)C2CC2)ncc(C#N)cc1C(N)=O C(CC(=O)N1CCC(CC(C)C)C1)(C(F)(F)F)NC(c1c(COC)cco1)=O c1(C(=O)NC2CC(CNC(C=CS(C)=O)=O)C2)scc2c1CCCC2 n1(CC(N2CCN(C)CC2)C)cnc(S(=O)(=O)N2CCCc3sccc3C2)c1 C1(N(C(C(C)n2ccnc2)=O)C)CCC2CN(C(C34CCC(C)(C3)OC4)=O)CC12 Cn1cccc(C(=O)NCc2cccnc2-c2ccc(-c3ccccc3)s2)c1=O c1(C(=O)OCc2cccc(C#N)c2Cl)ccc(Br)c(S(N)(=O)=O)c1 C1(C)(CCNC(CC2C(CC)C2)=O)CCN(C(=O)Cc2cc(C3CC3)no2)C1 c1(C(C)C)ccc(C(=O)COC(C2CCC=CO2)=O)c(C(F)(F)F)c1 N#Cc1c(F)cc(-c2cnc3[nH]c(-c4noc(C(C#N)C(N)=O)n4)cc3c2)cc1F C1(OC)(CNC(c2[nH]ccc2SC)=O)CCN(C(c2c(C)ncn2O)=O)CC1 C1(OCC(=O)NCC(C)N(C(=O)CC2CCCC2)C)CCCCC1C C(C(CC(C)C)NC(C1CCC=CO1)=O)NC(CCSC)=O c1(C(=O)NCCCCCF)ccccc1-n1cc(C2CC2C(=O)O)nn1 c1(CC)c(N(C)CCN(C)C(C2(C)CCC(F)(F)C2)=O)ncnc1Cl CCC(CCCC(=O)NCC1CC2CCC2C1)NC(C1CC(N(C)C)C1)=O CC(=O)CCCC(=O)N1CCCOC(NC(=O)COCP(C)(C)=O)C1 N1(C(C(CCC)CC)=O)CCC2(C1)CN(C(C1CCCC(=O)CC1)=O)CCO2 c1(C(N2CCC(C(C)C(=O)N(C)Cc3cnnn3C)C2)=O)cnn2c1CCC2 Cc1cc(OCC(=O)NCC(CNC(C2CC(CC3CC3)C2)=O)CO)no1 Cc1nc2sc1C(=O)NC2.c1(NC(=O)C(O)c2ccsc2)cnn(CC(C)C)c1 CC1CCCCN1CC(=O)NC1CC(NC(=O)C(O)Cc2cnc[nH]2)C(O)C1 c1(C(N(CC(CC)NC(C(CC=CC)CC)=O)C)=O)cc(OC)cc([N+](=O)[O-])c1 c1(C(=O)NCC(C)NC(CCCC(=C)C)=O)ccnn2ccnc12 CCC(C(=O)N1CCC(F)(CNC(c2cnn(C)c2)=O)C1)C(C)(C)CC C1(F)(C(=O)NC2(C(=O)OC)CC2)CCC(NC(=O)CSCC(F)(F)F)C1 c1(OC)cc(CNC2CCN(c3ncnc(Cl)c3C)CC2C)ccc1Cl C1(C(N(CC(CNC(C2(CC)COC2)=O)(C)C)C)=O)CCc2cnn(C)c2C1 C(CCCCCNC(C1(n2cc(Cl)cn2)CC1)=O)N(C(c1cc(C)no1)=O)C CC12CN(C(C3(c4cccnc4)CC3)=O)C(C(N3CC(C(N)=O)C(O)C3)=O)(C1)C2 c1(C(N(CCCNC(c2ccc(SC)cc2)=O)C2CC2)=O)cnc2[nH]cnc2c1 C(=O)(CCC(F)(F)C(F)F)N1CCCC(N(C(CC2ON=C(C)C2)=O)CCF)C1 C(=O)(C1=CC(O)C(NC(=O)CSc2nc[nH]n2)C1)N1CC(C#N)(F)C1 C1(NC(C)=O)CCCN(C(C2(c3ccccc3C#N)CCC2)=O)C1C N1(C(c2cccc(C)n2)=O)CC(O)CC1(C)C(=O)NCCCOCC(C)C c1(OC)c(C(=O)NC2(C3CN(C(=O)C(O)CCSC)C3)CC2)cccc1F C(=O)(CCC(C)CC)N1C(COC)(CNC(=O)C(C)CSC)CCC1 C1(C(C)OCc2occ(C(=O)OC)n2)CN(C(=O)C(C)N(C)C(C)=O)CCO1 N1(C(C2CC3(CC3)CN2C(c2coc(CO)c2)=O)=O)CCc2nnnn2CC1 Cc1cccc(N)c1C(=O)NC1CN(C(c2cccc(C3CC3)n2)=O)CC12CC2 C1(CN(C(C(CSC)OC)=O)C)CCN(C(=O)CC2C=CCCC2)CC1 C1(CC=CC)CCN(C(=O)C(=CC2CCCC2)C)C1.c1(C2C(=O)N2)cnn(C)c1 Cc1nc(C(=O)NCC(C2CCCCN2C(=O)CCOC(C)C)(C)C)ccc1C#N C(C1CCCC1)=CC(=O)NC1CC(N(C(C(C)NC(=O)NC)=O)C)C1 N1(C(CN(C(C2CC(C)OCC2)=O)CC2CC2)=O)CC2CC2C2CC12 C1(O)(C(C)NC(C2(CC(C)C)CCC2)=O)CCN(C(c2cc(C3CC3)[nH]n2)=O)C1 C(C(CC(F)(F)F)NC(=O)C(F)=C(C)C)NC(c1nncc(CCC)c1)=O N1(C(C2CCCCCN2C(=O)CN2CCCCC2)=O)CC2CCC(CC2)C1 N1(C(C(C(C)C)(C)C)=O)CC2(CCN(C(=O)CCC(=O)c3ccccc3N)C2)C1 C(=O)(C1=CCCCO1)NCC(C)(C)CNC(=O)C(Cc1ccccc1)SC(C)(C)C Cc1cc(C(N2CCC(C)(C(=O)NC(c3cccnc3)C)C2)=O)n(C)n1 N1(C(c2cccc(C)c2)=O)CC2CCN(C(=O)Cc3ccsc3C)CCC2C1 N1(C(C(C=C)(C)C)=O)CCC(C)C(CNC(=O)Cn2cccnc2=O)C1 Cc1cnc2ccccc2c1CCN1C(=O)CN(C)CC(C)C1=O c1(OC)nc(CNC(C2CNCCN2Cc2cnn(C)c2OC)=O)nc2[nH]cnc12 c1(C(=O)NC2CN(C(C=C(C)C)=O)CC2F)cnc2c(c1)c(C(C)(C)C)nn2C N1(C(c2n(CCC)ccc2)=O)CCCC(C)(C)C1CNC(=O)CC(C)(C)OC c1(CC(=O)N(CCNC(C(CC)n2cccn2)=O)CC)c[nH]c2cnc(Cl)cc12 C12(CNC(CC(=O)NCC)=O)CCC(CN(C(c3cncc(C#N)c3)=O)C1)C2 N1(C(CCSC)=O)CCN(CCNC(=O)CC2C=CCC2)CC1 C12(NC(c3c(C)cncc3)=O)CCN(C(c3ccc(Cl)cc3C(F)F)=O)CC1C2 c1(C(=O)NCC(c2ccnn2C)NC(C(F)OC)=O)c[nH]nc1C1CC1 C1(C(=O)NCCC(=C)CNC(=O)CCC(C)(C)C)CC2CCC1CC2OC CC(C(C)(C)C)=CC(=O)NCC(C(C)C)NC(=O)C=CC(C)C c1(C(=O)NC2(C)CCN(C(=O)C(F)(F)C3CC3)CC2)cccc2oncc12 N1(C(C(C2CCN(C(c3cccc(F)c3)=O)C2)C)=O)CCC2(CCCO2)C1 C1(NC2CC(c3cccc(O)c3)(C)C2)C2CC1N(C(=O)C(F)(F)c1ncccn1)C2 C(C(CC1CCCC1)C(=O)N(C)CCc1ccncc1)NC(CC=C(C)C)=O N1(C(C=CSC)=O)CCC2(NC(c3cc4ccnc(Cl)c4[nH]3)=O)CCCCC12 c1(C(C)C)cc(C(=O)N(C)CCN(C(=O)CN(C)C(C)C)C)c(C(C)C)[nH]1 c1(CNc2n[nH]cc2NC(=O)CCc2ccc(Br)s2)ccc(C(=O)NO)o1 c1(C(c2nnnn2C2(C)CC2)CNCC2(COC)CC2)cncc(C)c1 N1(C(C(CC)N(C)C)=O)CC2(C(=O)NC3CC3C(F)(F)F)CCC1CC2 C1(OC)CCCC1(c1nnnn1CCCNC(=O)OC(C)(C)C)NC1CC1C Cc1ccncc1C=CC(=O)NCC1CCN(C(=O)C=CCN(C)C)CC1 Cc1nn(C)c(Cl)c1CN1CC(C)OC(C)C1.N12CCC(CC1)C(C)C2=O c1(NC(C(C)NC(=O)NC)=O)scnc1C(=O)NCCCOCCCN(C)C N1(C(CC=CC=C)=O)CCCC2(N(C(=O)Cc3ccc(Cl)nc3)CC)CC12 C1(N(C(=O)C(=O)NC2CC2)CC#C)CCN(C(=O)CCn2ncn(C)c2=O)CC1 Cc1ccc(S(=O)(=O)NC2CCC(C=Cc3cccc(N)c3)CC2)c(F)c1 C1(C(N(CC#C)CC)=O)CCN(C(=O)C(C)N(C2CCCC2)CC)C1 CC(CC(=O)NC1(CCO)CN(C(C2CNC(=O)C2)=O)C1)CC(C)(C)C C(CCNC(=O)C=Cc1cscn1)(C(=O)N1CCCC1CN=[N+]=[N-])OC C1(CNC(C#CC(=O)N(C)C)=O)CCCCN(C(c2csc([N+](=O)[O-])c2)=O)C1 NCC1OCCc2sc(C(=O)NOCc3ccccc3F)cc21 c1(C(C)C)ccc(C(=O)NCC(O)CN(C(=O)CC2(C)CCCO2)C)c(O)n1 C(=O)(C(C)(C)C(C)O)N(CC(CC)NC(c1ccc(CO)c(F)c1)=O)C N1(C(CCC(=O)NC)=O)CC2CN(C(=O)CCC(C)SC)CCC12 C1(C(=O)NC(C)(C)CC=CC(=O)NCCN2CCCNC2=O)CCCCC12CCC2 C1(NC(C)=O)CCN(C(=O)CC2(NC(C3SCCS3)=O)CCCC2)C1 C(=O)(C(C)(C)CCCNC(=O)CCOCCNC(=O)Cc1cccnc1F)OC Cc1cc(C#N)c(F)cc1NC(C1C2CC1N(C(C1(C(F)(F)F)CC1)=O)C2)=O c1(NCC2N(C(C(CC)CC(C)C)=O)CCN(C)C2)cc(C)ccc1[N+](=O)[O-] C12(C(=O)NC3(C)CCN(C(CS(CC)(=O)=O)=O)C3)CCC(OC)(CC1)CC2 N1(C(COCCCOC)=O)CCC2(COCC(CNC(=O)CC(C)(F)F)O2)C1 c1(CCC23CC2CN(NC(CC2(N(C)C)CCC2)=O)C3)nc2ccc(F)cc2[nH]1 c1(C(C)NC(C2CC(NC(C(COC)OC)=O)C2)=O)ccc(C)nc1 N1(C(COCCOC)=O)CCN(C(c2ccnc3[nH]cnc23)=O)C(C)C1C N1(C(CN(C)CC)=O)CC(NC(=O)Cc2ccc(C)cc2)C2CCCC12 c1(C(=O)NC2CN(C(C(C)=C(CC)C)=O)CC2C)cnn2c(O)cc(C)nc12 N1(C(C2CC(OC)C(OC)C2)=O)CCC(C)(C)C(NC(c2ccnc(C)c2)=O)C1 CC(O)C(C)(C)C(=O)N1CC2CC(C(=O)N(CC(F)F)CCO)(C2)C1 Cc1ccc(CC(CO)NC(=O)Nc2ccc(C#N)cc2)cc1C c1(CCC)nc(C(=O)NCC2CCN2C(c2csc(-c3nc[nH]n3)n2)=O)co1 Cc1nn(CC(=O)NC2(CNC(C3CC4CCCC4C3)=O)CCCC2)c(C)c1Cl NC(=O)CCC(C(=O)N1CC(Oc2cc(F)cc(F)c2)C1)Nc1cnns1 C12(C(=O)NCC(=C3CN(C(c4cncc(SC)c4)=O)C3)F)CC3CC1C2C3O CCC(CC(=O)NC(C)(C)CN(C)C(c1ccn(CC)n1)=O)C1CC1 c1(OC)cccc(SCC(=O)N(C2CCN(C(=O)Cc3c[nH]nc3O)CC2)C)c1 C12(CNC(CC3(C)CC3)=O)CC1CN(C(=O)CNC(=O)NC1CC1)C2 Cc1cc(N2CCCC(CNC(c3cnsc3C)=O)CC2)cc(C#N)c1[N+](=O)[O-] N1(C(C(F)=CC)=O)CCN(C(C2COC(=O)C2)=O)C(c2cn[nH]c2)C1 N1(CC(=O)NC(C(C)C)CNC(=O)C(=O)N(C)C)CCC(=O)NC1=O c1(C(N2CC(N(C(CC(=O)OCC)=O)C)C2)=O)cnc(C(=O)O)nc1 Cc1cc(C(=O)NCCNC(C2NC(=O)OCC2C)=O)c(C)s1 N1(C(c2c(C)nc(C)[nH]2)=O)CCC(NC(=O)C=CC2CCCC2)CC(C)(C)C1 C1(C(N2C(C(N3CCCC(O)(CO)C3)=O)CC2)=O)CCC([N+](=O)[O-])CC1 Cc1ccc(C)c(C(=O)N(C(C)CCNC(C2(CF)CCC2)=O)C)c1 c1(N2CC(C)SCC2)ccc(S(=O)(=O)NCC2CC(N(C)C)C2)cc1Cl C12(CNC(c3n[nH]c(C)c3C)=O)CCC(CN(C(C3OCCC3C)=O)C1)C2 n1(CC(=O)NC2C(CNC(C(C)n3cncn3)=O)CC2)cc(CO)nn1 C1(C(=O)NCC2C(NC(C3C=C(C)CS3)=O)CCCC2)CCN(C)C(=O)C1 c1(NCC2(F)CC(NC(C(C(CC)C)C)=O)C2)ncnc2c(Cl)cc(Cl)cc12 C(=O)(C#CC1CCCCC1)N1C(CN(C)C(C2CCC3(CCOCC3)C2)=O)CCC1 C(=O)(C(=O)NOC)NCCCC(=O)NC(CC)C C1(CC(=O)NCC2CC(C)CO2)(NC(C=C(C)C(C)C)=O)CCCC1 O=C(CSC1CC(C(=O)NOCC(F)(F)F)C1)NOCc1cn(C2CCC2)nn1 Cc1ccc(C(=O)N(CC(C)(C)CNC(C2C3CC3C3CC23)=O)C)c(C)n1 C1(CNC(C2(COC)CC2)=O)(CO)CCN(C(C2CCCCC2(C)C)=O)CC1 N1(C(C(CC)OCC)=O)CCOCC1CCNC(c1nc(C)sc1C)=O Cc1ncnc(C(=O)NC2CN(C(=O)Cc3csc4nccn34)CC2F)c1C N1(C(C2(CC)CC2)=O)CC(NC(=O)C(C)(C)OCCOC)CC1(C)C CC1(C)CN(C(=O)C(=O)C=Cc2ccccc2)CC1NC(C1CC(N(C)C)C1)=O CC(C)C(C(=O)NC1CC(NC(=O)CCc2cc(Cl)no2)C1)c1ccncc1 c1(CC(=O)N(C(C)(C(=O)NCCN2C(=O)CCC2=O)C2CC2)C)cccnc1O C(CC(C)C(=O)NCCOC1CCN(C(c2cc(COC)on2)=O)CC1)=CC N1(C(C2OCCN(C)C2)=O)CC2(CCCC2NC(=O)CCCc2cnccn2)C1 C(=O)(C(C(C1CCCC1)OC(C)(C)C)N(c1nnn(C(C)(C)C)n1)C)NCCCC C1(NC(C(C)(C)C2CCOC2)=O)CCOCC1NC(=O)C1=CCSC1 CC(C)(F)C(=O)NC1COCC1NC(=O)CC1CNC(=O)C1 c1(C(=O)OCCOc2c(CC)cccc2)cc(OC)c2c(c1)OC(F)(F)O2 C1(C(=O)NC(C(=O)NCC2COCC(C)O2)CN(C)C)CCC2(CCC2)O1 C1(NC(CCN(C)CC)=O)CC2(NC(=O)CC3CCCC3)COC1C2 c1(OC)n[nH]c(C(=O)NC2CCC(NC(=O)Cc3csnc3C)C2)c1Cl CCC(C)C(CC(=O)N(C1CCC(CO)CC1)C)NC(C1CC1(F)Cl)=O C12(CC)CCC1CN(C(c1cccnc1CNC(c1ccccc1NC)=O)=O)C2 c1(CNC(C(=O)NCCSC)=O)ccnc(F)c1Cl C1(C(N2CC(CSC)C2)=O)CN(C(=O)Cn2cc(C#N)cn2)CCC1(C)C CC(C)CC(CNC(=O)CC1(N2CCCC2)CC1)NC(=O)Cc1cccc(F)c1 C1(OC)CN(C(C2CC2C2CC2)=O)CCC1NC(=O)CC1CC(OC(C)(C)C)C1 C1(C)(C(=O)NCC(C)(C2CC2)OC)C=CCN1C(=O)COCCC(C)C C1(C)(C(=O)NC2CCN(C(C(CC(C)C)(F)F)=O)CC2C)CC(C2CC2)=NO1 CC1CC(CO)N1C(=O)CSCCNC(C12CC(CO)(C1)C2)=O C12(CCOCC1)C(=O)NC2.c1(CNC(CCSC)=O)ncc(C)cn1 C1(C(C)C)N(C(=O)CCC2(C)N=N2)CC12CCN(C(=O)COCC1CC1)CC2 C1(C(=O)NC2C(CCC)C2)(NC(c2ccnn2C(F)F)=O)CCSC1 c1(C(COCC)CNCC(c2ccc(F)cc2)(C)C)ccc(F)cc1F c1(C(C)=O)cc2ccccc2[nH]1.C1(NC(C2(C)CNC2)=O)CCCCCC1CO c1(C(=O)NC(C2CCN(C(Cn3ccc(C)n3)=O)CC2)C)nccc2nn[nH]c12 c1(NCCC2CC(=O)NCC2)ccc(Oc2cccc(Cl)c2)c(I)c1 C1(C(=O)NC2(CC=C)CCC2)CCCN(C(c2c[nH]c(=NC)s2)=O)C1C C1(NC(=O)C=Cc2cncs2)CN(C(=O)CC=C(Cl)Cl)CC12CCOCC2 C1(NC(CC2(C)CCCC2)=O)CN(C(=O)CCCC(F)F)CCC1CO C(=O)(CC1=CCCCC1)NCC1C(NC(COc2ccc(C#C)cc2)=O)CCC1 N1(C(C2C(CCC)CCC2)=O)CCC(C(C)(C)C)(CNC(c2c[nH]c(=N)s2)=O)C1 c1(C(N2CCC(F)(C(N3CCC(CO)C3)=O)C2)=O)cc(O)cc(F)c1 CN1CC=C(CC(=O)N2CC(O)(CCNC(C3(F)CCOCC3)=O)C2)CC1 c1(OCC(=O)NC2C3CN(C(C=CC)=O)CC32)ccc(F)c(F)c1 C1(C(=O)NCC(C=C)O)(CNC(c2ncn(C(C)C)n2)=O)CC2(CC2)C1 C=CCCCCCC(=O)NCC(C)(C1CCC1)NC(C1CC12CCOCC2)=O CN1CCN(C(=O)C=CC(C)(C)C)CC1CNC(C1CC(=O)C12CCC2)=O C(=O)(C1=CC(O)CCC1)N1CC(NC(c2ncc[nH]c2=O)=O)CC(C)C1 C=C(F)C1(CC(=O)NCC2CN(C(c3cc(C)c(C)[nH]3)=O)C2)CCC1 C12(C(=O)NC(C(CC=C)C)=O)CCC(NCC3CC4(CCC4)C3)(CC1)C2 C1(CCC)CN(C(=O)C(S(C)(=O)=O)C2CC2)CCN1CC(=O)NC1CCCCC1 CN=c1[nH]cc(C(=O)NC(CCC2CC2)C(=O)N(CCCO)C(C)C)s1 C1(NC(CC2CCN(C(CCC#C)=O)CC2)=O)CCc2nn[nH]c2C1 C1(C(N(CC(N2CC(CCOC)C2)=O)C(C)C)=O)CCCC1OC N1(C(c2c(CC)scc2)=O)CCC(OCCCNC(=O)CC2CCCC2)CC1 C1(NC(CC2C(C)(C)CCC2)=O)CC(C(N)=O)=NO1 C1(NC(CCOCCC)=O)CCCCC12CCN(C(=O)Cn1cc[n+](C)c1)C2 C1(NC(c2cc(OCC)ncc2)=O)CN(C(=O)C(O)C(C)C)CCC12CCC2 CCC(CNC(=O)C(c1ccccc1Cl)N(C)C)CC(=O)OC(C)(C)C C1(C(=O)NC2(CN(C)C(c3ccc(C(N)=O)cc3)=O)CC2)CC2(CCC2)CO1 Cc1cccc(O)c1C(N1CC(C(N)=O)(CNC(C23CCC(C)(C2)OC3)=O)C1)=O C1(C#N)(C(=O)NCc2ccc(CN(C(C(C(C)C)F)=O)C)cc2)CC2(CCC2)C1 C#Cc1ccc(CC(N2CCC(C)(CNC(=O)C(C)P(C)(C)=O)C2)=O)c(F)c1 CCC(C(=O)N(C1CCCC(NC(=O)Cc2nc[nH]n2)C1)C)C(F)(F)F c1(C(N2CC(C(=O)Nc3ccc(C)cc3C)C3C2C3)=O)cc(C)c(=O)n(C)c1 C1(CCC)CN(C(c2nn[nH]c2Cl)=O)CCN1C(=O)C=Cc1ccc(C(N)=O)o1 C12(CCNC(C=C(C)C(C)(C)C)=O)CCC(C1)N(C(=O)CN1C(=O)CNC1=O)C2 c1(C(=O)NC2CN(C(C(CN(C)C)O)=O)CC23CCC3)ccc2cnccc2n1 N1(C(C(C=C)(C)C)=O)CCC2(NC(c3cnn(C)c3Br)=O)CC2C1 CC(CC(=O)N(CCOCCO)C1CC1)C(C)(C)NC(=O)CCCF C(C1c2ccsc2CCN1C(=O)CCSC(F)(F)F)NC(=O)C(C1CCOCC1)F Cc1ccc(CC(N2CC(NC(=O)C=Cc3ccco3)CC2C)=O)cn1 n1(CC(N2CCC(CNC(C3(CF)CC3)=O)C2)=O)cccc(C(F)(F)F)c1=O C#Cc1ccc(Cl)c(C(=O)NC(CNC(c2cc(C#C)ccc2Cl)=O)CC)c1 c1(NC(C2N(C(c3sc(C)c(Br)c3)=O)C3C(C2)C3)=O)cc(C(F)(F)F)cc(F)c1 N1(C(C(Cc2ccc(OC)cc2)N)=O)CCC2(CC=CCO2)C1 C(C(=O)N(C(C)C(F)F)C)(C(C)(C)C)NC(c1nnn(CC)c1C)=O C1(C(=O)NC(CN2CCN(C(COCCSC)=O)CC2)C)CCC(C)(C)CC1 N1(C(Cc2ccc(C)o2)=O)CCCOC(CNC(c2nncs2)=O)C1 C1(C(N(C)C2CC2)=O)C2CC1N(Cc1cccc(F)c1)C2.c12ccc(cc1)NC2 c1(C(=O)NC(C(C)NC(C2CN(C(C)C)C2)=O)CO)ccc(CO)c([N+](=O)[O-])c1 N12CCCC(CC)(C1)C(=O)N1CC(C=C)(C1)CC2=O.C1(C)(CO)CCC(=O)N1C C1(C(=O)N(C(C)C(=O)NCC2CC23CCC3)C2CC2)(OC)CCSC1 C(C)(C)(CCN(C(=O)CC1CCCN1C)C)NC(CSCC#C)=O C1(C(=O)NC2CCCN(C(C3C(C)CC=CC3)=O)C2)CC(=O)CC12CCC2 c1(C(=O)NC2CC(NC(C3CC3CC3CC3)=O)C2)ccc(CCCO)cc1Cl Cc1nn(C)cc1CN(C)C(C1(CNC(=O)C(F)OC(F)(F)F)CCCC1)=O C12(NC(=O)CCC(F)F)CC3CCC(C1C2)N3C(c1ccccc1CCCCl)=O N1(C(c2c(C)nc(-c3ncc[nH]3)s2)=O)CCC(NC(c2csc(O)n2)=O)C1(C)C C1(CC)CN(C(=O)C2=NOCC2)CCC1NC(=O)C(C)(C)c1cnsn1 Cc1[nH]nc(C(C)C)c1C(=O)NC(C1CCN(C(C2CNC(=O)N2C)=O)CC1)C C1(OC)CCCC1C(=O)NCC1CCC1NC(=O)Cc1n[nH]c(=N)s1 CN(C(=NCc1ccco1)NCC1CCOC1)CCc1ccoc1 C1(NC(C(CNC(CCC2CC(C)C2)=O)C)=O)CN(C)CCN(C)C1 c1(S)ccc(Br)cc1OCCC#C.C1(=O)C(=O)NCCOC(C)(C)CN1.C(C)(C)O c1(C(=O)NC(C(C)C)CNC(c2cc(N)cnc2Cl)=O)cnc2[nH]cncc1-2 Cc1c(Br)ccc(CN(C)CC2CCCNCCC2)c1O N1(C(CCC(=C)Cl)=O)CC2CCCCC2(CNC(c2cc(C#N)ccc2C)=O)C1 C1(NC(c2cn(CC)nn2)=O)CCC2CCN(C(=O)C(c3ccccc3Cl)C)C12 C(=O)(C1=NOC2(CCC2)C1)NC(C)CCCC(=O)N(C)Cc1ccncn1 C#Cc1ccccc1CC(N1CCC(CO)C(NC(=O)C=Cc2cnc[nH]2)C1)=O N1(C(CCCC)=O)CC(CNC(C23CCC(OC)(CC2)C3)=O)OC(C)(C)C1 C1(CC(=O)OCC)CN(C(=O)CS(=O)(=O)CC)CCN1C(c1ccc(O)nc1)=O C12(NC(c3cc(CC)ncn3)=O)CCN(C(c3sc(C)cc3C)=O)CC1C2 N1(C(C2N(Cc3c(C)cc(Br)cc3)CCC2)=O)CCc2c(O)n[nH]c2C1 C1(C(N2CCC(C)(CC(=O)NC)C2)=O)CCCCCCN1C(=O)CCn1cccn1 C=CCC(C)(CNC(=O)CC(C)N(C(=O)C=Cc1cocn1)C)CO C1(NC(=O)CCCC2OCCO2)(CO)CCN(C(=O)C(F)=C2CCC2)C1 c1(C(=O)NC(CC)CNC(=O)CCn2cc(C)cn2)nn(C)c(Cl)c1Cl c1(CN2C(C(N3CCCC(O)C3)=O)CC(C)C2)ccc2ncnn2c1 N1(C(C2CCC(NC(C3CCC4(CCC4)C3)=O)C2)=O)CC=C(CO)CC1 C(=O)(C(C)(O)Cn1ccccc1=O)NC1C(CNC(C(C)=CC)=O)COC1 c1(OCC)c(C(=O)NC2CC2NC(=O)C(c2cncn2C)O)cccc1Cl C1(C(=O)NC(C)CCC(=O)NC(CC2CCC2)CO)CCC2(CCC2)C1 c1(OC)ccc(C(=O)NCC2CCCCN2C(=O)C(=O)NC2CC2)c(C)c1 C(c1nc2cccc(Cl)c2s1)=C1CCC(C#N)C1 Cc1cn2nc(N3CCC(CF)(NC(c4cc(CC(C)C)[nH]n4)=O)C3)sc2n1 C1(C(N(C)N(C(C2(CO)CC2)=O)C2CC2)=O)(C(N2CC(C#N)(CO)C2)=O)CC12CCC2 N1(C(C2(SC)CNC2)=O)CCCCC(NC(=O)CCCN(C)C(C)=O)CC1 C1(O)(CN(C(CCCC#C)=O)C)CCCN(C(c2occc2C(=O)OC)=O)C1 C(=O)(C(C)(C)CCCc1ccccc1)NCC1CC1C(=O)NC(COC)C(C)C C(C(C)C(C)(F)F)NC(CCOCCNC(C(C)C)=O)=O C(=O)(C1=NOC(C)C1C)NCCC(=C)CNC(=O)CN(S(C)(=O)=O)C CN1CC(C(=O)NCC(O)C(=O)NCCCP(C)(C)=O)CCC1=O c12ccc(cc1)s2.C(=O)(C(O)CC1CC1)NCCC(C)N(C(=O)CNC=O)C c1(NC)cnncc1C(N1CCN(C2CCCN(C(=O)C=C(C)C)C2)CC1)=O C1(CN(C)CC2CCN(C(=O)C(=O)NCCC(N)=O)CC2)CCCCCS1(=O)=O Cn1cc(C#N)cc1NC(C1CCCCN(C(C2CCCOCC2)=O)C1)=O N1(C(CC(c2c(C)n[nH]c2C)C)=O)CC(O)(C2(CNC(=O)C(C)(C)CF)CC2)C1 C1(NC(c2cc(Cl)ncc2O)=O)CC2(CCN(C(=O)CCOCC(F)F)CC2)C1 N(S(C)(=O)=NC1CC1)C(CC1(C)CCN(C(=O)Nc2ccccc2)C1)=O FC1(F)CN(c2cnc3n2CCOC3)CCN(c2ccc(OC(F)F)cc2)C1 Cc1c(C(=O)NCCC2CCN(C(C3CN(C)CCO3)=O)C2)nnn1C(C)C C1(NC(C2(CCCC)CC2)=O)CCN(C(=O)CC2(C3CC3)CC2)CC1C C1(C(=O)OC(C)(C)CCN(C)C(=O)OC(C)(C)C)CCN(CC)C2(CCCC2)C1 N1(C(C(C)Oc2cccc(Cl)c2)=O)CCC2C(C1)CN2C(=O)C1=CCCCC1 C=C1CCN(C(C2CC2OC(C)(C)C)=O)C(C(=O)NCC(O)C(F)(F)F)C1 c1(CC(=O)NCCNC(c2nn(C)c(C3CCCO3)c2)=O)ccc(O)c(F)c1 C(=O)(C(F)(F)CC1CC1)NCC(C1CC1)NC(c1cn(CCC)nc1)=O c1(CC(=O)N)cc(CNC(=O)NCC)nc(OCCn2cccn2)n1.C1CC1 c1(CNC(C(C)N(C(=O)C(C)(C)OC(C)C)CCC)=O)ccc2n[nH]cc2c1 c1(C(=O)NCCC2(O)CN(C(C3CCC(C)S3)=O)C2)cc2n(n1)CCNS2(=O)=O c1(NC(C(N2CCCC(c3nc(C(=O)OCC)[nH]n3)C2)=O)=O)ccc(Cl)c(F)c1 C(C)(C)(CCCNC(C1CCCN1CCC(C)C)=O)NC(C(CC)NC(C)=O)=O Cc1nc(C)c(C(N2CCC(NC(C3CC3c3ccnn3C)=O)C2)=O)[nH]1 Cc1nn2cc[nH]c(=O)c2c1C(=O)NCCC1CCCCN1C(=O)CC(C)F C(=O)(C(O)CCC(F)(F)F)N1CCC(NC(CSCCCC)=O)(CO)C1 c1(C(N2CC(CC(C(N3CC(O)(CC(C)C)C3)=O)F)C2)=O)nn(C)cc1Cl c1(C(N2CC(CCC)C(NC(c3cc(C)n(C)c3C)=O)C2)=O)ccc([N+](=O)[O-])s1 n1(CC)cc(NC(=O)C(C2CCC2)NC(=O)CC(C)c2ccco2)cn1 c1(CC(N2CC(NC(C3(COC)CCCC3O)=O)C2)=O)ccc(OC)cc1Br c1(C(N2CC(O)(C(C)NC(C(C)SC)=O)C2)=O)cc(C)c(C(C)C)nc1O c1(C(=O)NCC2N(C(c3cccc(NC)n3)=O)CCCC2)ccc(F)c(F)c1F N1(C(C2C=C(C)CS2)=O)CCC(C(=O)NCc2ccc(C(N)=O)o2)CC1(C)C C1(C(=O)NC2CC(SC)C2)CC12CCN(C(c1ccc(N3CCC3)nc1)=O)C2 CS(=O)(=O)C1(C(=O)NC2CCC(CNC(C3C=CCC3)=O)CC2)CCCCC1 c1(C(N2CCCC(NC(c3cnc(O)s3)=O)CC2)=O)ccc2[nH]c(=O)cnc2c1 C(C)(C)(CCC(=O)NCC(C)(C)CNC(c1cc(Cl)on1)=O)OC c1(-c2c(C)nn(C)c2C2COCCN2C(C)C)ccc2c(c1)NC(=O)C2(C)C N1(C(CC(C)(F)F)=O)CCC2(CCOC2)C(CNC(c2cc(C(N)=O)[nH]n2)=O)C1 N1(C(CNC(CNC(C)=O)=O)=O)CCC2(CNC(c3ccno3)=O)CCCCC12 c1(CNC(c2sccc2Cl)COC)ccn(-c2ccccc2)n1 c1(CC(=O)NC(C(C)NC(C2N(CC)CC2)=O)C)ccc(F)cn1 C1(CC(=O)NC)CN(C(=O)CN(C)C(C)C)CCN1C(C1CCCN1C=O)=O C(=O)(C(C)(C)C(=O)NC)NCC(c1ccc(F)cc1F)NC(CSCCC)=O CC(C)(C)S(=O)(=O)CC(=O)NCC1C(C2CC2)CCN1C(c1n[nH]c(=N)[nH]1)=O N1(C(CCNC(=O)NC)=O)CCC(C(=O)NC2C=CC(COC)C2)C12CC2 c1(C(=O)NCC2C(NC(CC3CCC(=O)NC3=O)=O)C2)snc2ccccc12 c1(OC(C)C)ncccc1S(=O)(=O)c1cc2ncccn2n1 C1(NC(CCOCCCNC(c2c(C)ocn2)=O)=O)C(C#N)C1(C)C Cc1c(C(=O)NCC2(CNC(C3CCC3C)=O)CCC2)nnn1C c1(C(=O)NC(CC)CNC(C2CCC2C)=O)cc2sc(S(N)(=O)=O)cc2s1 Cc1ccc(C(=O)NC2(CN(C)C)CN(C(=O)Cc3c(C)noc3Cl)C2)cc1C C=CC(C)(C)C(=O)N1CC(NC(=O)C=Cc2cocn2)C(n2ccnn2)C1 c1(NC(=O)CNC(C2COC2)=O)ccc(C(F)C(F)(F)F)cc1 c1(CC(=O)NCC(CNC(C2C(C(N)=O)C2)=O)CO)ccnc(Br)c1 C1(NC(CCC(=O)NC)=O)CCN(C(=O)Cc2n[nH]c(=NC)s2)CC1F CC(CC(N)=O)C(=O)NC1(C2CN(C(=O)CCn3cnc(=N)[nH]3)C2)CC1 c1(C(=O)NC2(C)CCN(C(=O)Cc3csnn3)C2)cccc2oncc12 C1(C)(C(=O)NC(C(=O)NCc2n(CC)nnn2)C)CC2CCC1O2 c1(CC)ccc(Cl)c(C(N2CCCC(C)(NC(c3cc(SC)nn3C)=O)C2)=O)c1 N1(C(C(CC)ONC(=O)OC)=O)CCC(CO)CC1 c1(C(=O)NCCCN(C)C(C2CCN2C2CCCC2)=O)csnc1Cl CN1CCC(C)(CNC(=O)C(C)(CO)NC(c2ccon2)=O)C1 c1(N2CC3(CCN(C(C(C)(C)SC)=O)C3)C2)cnc(C#N)c(C#N)n1 C(=O)(C1CCc2cc(F)ccc21)NC(CC(C)NC(c1c(C(C)C)scn1)=O)C N1(C(C2(CCOC)CCC2)=O)CCCCCC(NC(=O)CSCC(N)=O)C1 CC1CN(C(C2CC(C)(O)C2)=O)CC(C)N(C(C2CCC(=O)N2)=O)C1 Cc1c(C(=O)NCC(C)CC(=O)NC2(CC(N)=O)CC2)nnn1C C1(F)(CNC(C2(CCC)CCC2)=O)CN(C(=O)CCc2nc[nH]n2)C1 c1(C(N2CCC(C)(CNC(CN(C3CC3)CC)=O)C2)=O)ncn2c1CCC2 N1(C(C(C)CC2CCCC2)=O)CCOCC(C(=O)N(C)Cc2ccsc2)C1 C1(C(=O)NCC(C)(CNC(=O)Cc2ccoc2C)OC)CCCCC1O N1(C(C2CN(C)C(=O)N2)=O)CC2(CCC(CNC(=O)CC3CCN(C)C3=O)O2)C1 c1(C(=O)NC(CNC(C(CC)COC)=O)C(C)(C)C)nn(C)c(C)c1Cl c1(C(=O)NCCCO)ccnc(CNC(c2sc(C(F)(F)F)nc2Cl)=O)c1 C1(CC#C)(C(=O)NCCN2C(=O)CC=CCSCCOCCC2)C=CCC1.CC c1(C(N(C)CC2(C)CCOC2)=O)ccc(N)c(N(C)C)c1 N1(C(C(C)CC2CCC2)=O)CC2(CCN2C(=O)CCCC2CCCC(=O)N2)C1 Cc1c(C(=O)NCC2(NC(c3cccs3)=O)CCC2)cccc1[N+](=O)[O-] C1(C(=O)NCC2(CNC(C(C)=CC)=O)CCC2)CCCC1c1cnn(C)c1 N1(C(Cc2cc(OC)c(Cl)cc2)=O)CCC2CCN(C(=O)C(O)CC(C)C)C2C1 C1(CCNC(c2ncc(C)cn2)=O)C(C)CCCN1C(=O)CCCn1ccnn1 c1(C(N(CC(C)N(C(CCC(=C)C)=O)C)C)=O)cnc2ncnn2c1O C(=O)(CC1COc2ccccc21)N(CC(C)N(C(=O)C#CC1(C)COC1)C)C N1(C(Cc2c(C)nc(S)s2)=O)CCC(NC(=O)CNC(=O)C(F)(F)F)C(F)C1 C1(CC(N2C(CNC(C=CC)=O)CC(OC)C2)=O)CCn2cncc2C1 N(C(=NCCc1ccccn1)NCCc1cccc(C)c1)C(C(COC)C)C N1(CC(=O)N(CC(C(C)C)C)C2CC2)CCN(C(=O)CC2NC(=O)NC2=O)CC1 N1(C(C(CC)O)=O)CCCC2(CCCN2C(c2ncc(C)cc2C)=O)C1 c1(C(CC)CC)nc(-c2cnn(CC)c2)n(C(c2ncnn2C)C)n1 N1(C(C2C(C)C2c2ccccc2)=O)CC2CCN(C(=O)CCC3CC3)C2C1 c1(C(=O)NC2C(CNC(CCCCNC(C)=O)=O)CC2)cnn2c1OCC(F)C2 C1(OCCCOC)CN(C(=O)CC2CCCC2OC)CC1c1cnn(CC)c1 CCCCC(O)C(C)C(=O)NNC(=O)c1cc(OCC(F)(F)F)ccc1C C1(C(=O)NC(CC#C)(C)C)CCN(C(c2cnn3c2OCC3)=O)C(CC)C1 c1(CC(=O)N(CC(CC)NC(c2occc2C)=O)C)cccc(C)c1Br N1(C(C2C(=C)CC2)=O)CC(F)(F)CC1CNC(=O)C1=C(C)CCC1 Cc1nc2ccc(C(=O)NC(CO)C(C)NC(C3(C#N)CCOCC3)=O)cc2o1 c1(C2(C(=O)NCCCN(C(=O)C(C)CF)C(C)C)CC2)ccc(Br)cn1 C1(NC(CCc2nnc(C(C)C)o2)=O)CC2CCC(C1)N2C(=O)COCCCF C1(C(=O)NCCC(C(=O)NC)O)CCCCCN1C(=O)C(C1CC1)C1CC1 c1(C(N2C3CC(CNC(C4CN(C(C)=O)C4)=O)C2CC3)=O)cc2ccncc2[nH]1 Cc1csc(NC(c2sccc2NC(c2ccc(N3CCCCC3)o2)=O)=O)c1C C1(NC(C2CCS(=O)(=O)CC2)=O)CC2CC1CN2C(=O)CCc1cnoc1 C1(C(=O)NCC(CNC(c2[nH]cc(CC(C)C)c2)=O)C)CCC2(CC1)CC2(F)F C1(C(N(C)CCOCCNC(c2sccc2C#N)=O)=O)CCCC2(CCC2)O1 N1(C(C2(OC)CCCC2)=O)CCCC(C(N2CCCC2CO)=O)C1 C1(c2nnnn2C2CC2)(Nc2c(C)ncnc2C)CCC2(CC1)COC(C)(C)C2 N1(C(C2CCC(C)O2)=O)CC(NC(c2csc(-c3ncc[nH]3)n2)=O)CC1C C1(CC(=O)N(C2CCCN(C(C3CC3C)=O)C2)CC)C2CC3CC(C2)CC1C3 C(=O)(CC1=CCN(C)CC1)NCC(C)N(C(=O)C=Cc1cocn1)C C1(OC)CC(CNC(=O)Cc2nn(C)cc2Br)N(C(c2conc2C)=O)C1 C1(O)(CNC(C2CN(C(C3CN(C4CCC4)C3)=O)CCO2)=O)CC2CCC1O2 c1(SCC(=O)NCC(=O)NCC(=O)Nc2coc(CO)n2)n[nH]c(O)n1 C1(CNC(=O)NC(C(=O)OCC)CCSC)CC2(CCC2)CO1 C1(CNC(CC2(C)CCOC2)=O)CN(C(=O)C(O)CC2CCCCC2)CC1(C)C CC1(C)CCCCC1C(=O)NCC1(CNC(c2cncc(C(F)F)c2)=O)CC1 C1(CNC(c2c(C)occ2)=O)CCN(C(=O)Cc2ncoc2C)CC1C Cc1ccc(C(=O)N(CCCNC(C2CCS(=O)CC2)=O)C)nn1 C(=O)(C(O)C(C)(C)CC)NC(C(N1CCCN(CC=C)CC1)=O)COC C1(C)(CNC(C2(C=C)CCC2)=O)CCC(NC(c2nnsc2C)=O)CC1 CC1=NOC(C(=O)NC2CN(C(C)C)CC2N2CCCC2)C1C N1(c2c(Cl)cnc(OC)n2)CC(NC(c2ccc(F)cc2F)=O)C2CCCCC12 C(=O)(CC(C)(C)CNC(=O)CC(O)C(C)C)N(C1CCN(C)C1)CC N1(C(c2cccc(CNC(C)=O)c2)=O)CC(NC(=O)CCC2CCOC2)CC(F)C1 c1(NCC(=O)NC)ncccc1S(=O)(=O)NC1CCC(C2CC2)C1 N1(C(C(CO)NC(C(C=C)O)=O)=O)CCC(F)(C#C)CC1 C1(C2(O)CCOCC2)(NC(C2C(c3cccc(F)c3)(C)C2)=O)CC1 N1(C(c2n(CC#C)ccn2)C(=O)NCCOC)CC(C)=CC(C)C1 C(=O)(C(C)(CNC(=O)Cc1cncnc1)CC)NCCCCCCSC c1(N(C)CCn2cc(-c3ccn(C4CC4)n3)nn2)cccnc1OC(F)F.C(CO)O C(=O)(C(C)(C)C(F)F)NCC(CCOC)NC(=O)C(c1ccncc1)C C(=O)(C(O)CC[S+](C)C)NC1CCC(N(C)C(c2ccnn2C)=O)C1 C1(CNC(=O)CCCCC2CC2)CCC2(CCC2)N1C(C1CC2CCC(C1)C2)=O CC1(CNC(=O)CC2CC=CCC2)CCN(C(C2CNC(=O)C2)=O)CC1 c1(N2Cc3c(CNOC)n[nH]c3C2)ncnc2[nH]cc(C#N)c12.C12CC(O)CN1C2=O C(=O)(C(CNC(c1c[nH]nc1CC)=O)CC(C)C)NC(CCC)C(=O)N(C)C Cc1nc(CO)ncc1C(=O)NCC1(F)CCC(CNC(C2CCC2C)=O)CC1 C1(NC(C2(C)C(C)(C)C2)=O)CC=C(C(=O)N2CCN(CCF)CC2)C1 C1(C(N(CCNC(c2n(C)ncc2)=O)C2CC2)=O)CC2CCC(C1)N2C1CC1 C1(C(=O)NC(C#C)C2CCC2)(OC)CCN(C(C2CC=CCC2CC)=O)C1 C1(CN(C(C)(C)C)C(=O)NC(CC)C(=O)NO)CCCOC1c1cn[nH]c1 C1(CC(=O)NCC(C(C)C)NC(=O)CCc2cnn(C)c2)CN2CCN1CC2 c1(OC)cc(C)c(CN(CCC(=O)NO)C=O)cc1Br.C(CO)S c1(NCC2(OC)CCCSC2)nccc(=NC(C)c2cn(C)nn2)[nH]1 c1(C(N2CCCCC(NC(C3C(C)(C)CCC3)=O)C2)=O)ccnc2cc[nH]c12 C[Si](C)(C)C1(CNC(c2cn3ccsc3n2)=O)CC1 c1(CC(=O)NCC2CC(NC(c3cnc(OCC)s3)=O)C2)nnc2n1CCCC2 C1(C(N(C(C(C)C)C)C)=O)C=CCN(C(c2cc[nH]n2)=O)C1 C(CN=c1[nH]c2c(cc1C#N)c(C)nn2C)(C1CCC1)NC(c1c(C)coc1)=O C(c1c(F)cccc1F)=CC(=O)NC1C(NC(C2C(=C)C2)=O)COCC1 c1(C(=O)NC(C)CCNC(C2NC(=O)C3CC23)=O)cc2c(Cl)cccc2s1 CS(=O)(=O)c1ccc(CN(C)C(c2ccc(N3CCNC3=O)cc2)=O)cc1Cl C1(C(=O)NCC2(F)CC(NC(c3ccon3)=O)C2)CCS(=O)(=O)C1 c1(C(=O)NCCN(CCC)C(C2CN(C)CC2C)=O)cc2ncc(C)cn2n1 CCC(CC(=O)N1CCCC(C)(CNC(c2cccc[n+]2[O-])=O)C1)C(F)F C1(NC(CCC(C)OC)=O)(CNC(=O)CN2CC(C)C2)CCC(F)(F)CC1 CCC(CCCC(=O)NC1(c2cccnc2)CC1)NC(c1cnns1)=O CCC(CO)C(=O)N1CCN(C2CN(C(C3CCCN3C(C)C)=O)C2)CC1 C1(CCC(=O)N(C2CCCN(C(C3CC(F)(CO)C3)=O)C2)CC)NC(=O)NC1=O C#CCCCCCC(=O)NCCCN(C(C1CC1c1nc(C2CC2)no1)=O)CC C(CCCCCC(=O)NC1(C)CCCS1)NC(c1n(C)nc(C2CC2)c1)=O c1(N(CCN(C)CCO)C)ncc(S(=O)(=O)NC2(C)CC3(CCC3)C2)cc1Cl N1(C(CCCC=C)=O)CCC2CN(C(c3ccccc3Br)=O)CC12 c1(CCC(=O)NCC(C)(C)NC(=O)CCc2cnoc2)nnc(C(F)F)o1 CC(C(=O)N1CCC(CCC(=O)Nc2cnc(C3CC3)nc2)C1)C(F)F Cn1c(C(=O)NCC2(F)CCC(NC(=O)CSc3ccc(F)cc3)C2)cnc1O C=CCC(F)(F)C(=O)N1CCN(C(C2CNC(=O)C2)=O)CC1CS(C)(=O)=O c1(C(=O)NC2C(C(=O)NCC(C)N(CC)CC)CCC2)ccc2nncn2c1 C1(CC)C(NC(=O)Cn2cc(Cl)cn2)CCCN1C(c1ccccc1Cl)=O CC(C)C(C)(O)C(=O)N(C1CCN(C(=O)CCOC2CCCCC2)C1)C c1(CNC(C2CCCN(c3nc(C4CC4)ns3)CC2)=O)cccn2nncc12 c1(OCC(=O)N(CC(C)NC(C2CC23CCCC3)=O)C)c(F)cccc1F C12(CNC(C(C)=C(C)C)=O)COCCN1CCN(C(=O)CC1CC3CCC1O3)C2 c1(OC)cc(C(C)C)n[nH]c1=NCC(C)N(S(C)(=O)=O)C C1(C)(NC(C2CCC(NC(CC(=O)NCC)=O)C2)=O)CS(=O)(=O)C1 c1(C(N)=O)ccc(S(=O)(=O)NC2CC3(C2)CC(NCC2CCC(O)CC2)C3)cc1 Cc1c(C=CC(=O)NCC23CCC(CC2)N3C(C2CCSC2)=O)cnn1C N1(C(C23CC(OC)C2C3)=O)CC2(CCCN(C(c3cc(N)ccc3F)=O)C2)C1 C(=O)(C1=C2CCCN=C2NN1)NC1CC(CNC(CCC(=O)NC)=O)C1(C)C N1(C(Cn2nnc(C)n2)=O)CCC2(CC1)CN(C(c1cnn(C)c1N)=O)C2C(C)C CCC(C(=O)NC1CC=C(C(=O)N2CC3(C2)CN(C(C)C)C3)C1)C(C)(C)CC N1(S(c2c(C)nn(CC(F)F)c2C)(=O)=O)CCOC2CCN(C)CC12 N1(CCOC)CCC(N=c2[nH]c(=NCCc3nnc(C)o3)c3sccc3[nH]2)CC1 C(=O)(C(CC(F)(F)F)c1cccc(F)c1)NCC(C)C(=O)OC(C)(C)C O=C1CCCC(C(=O)NC(CC2CCCC2)C(=O)NC2CCNC(=O)CC2)CC1 C1(NC(C2CCCC(=O)C2)=O)C2CC3C1C3C2C(=O)NCC12CCC(CC1)C2 c1(NCCC(C(F)(F)F)OC(C)(C)C)ccc2oc(O)nc2c1 Cn1nnc2c(C(N3CC4CCN(C(C5CCO5)=O)CC34)=O)cc(Br)cc12 c1(OC)ncc(C(=O)NCC2(N(C(=O)Cc3cn(C)nc3C)CC)CCC2)c(C)n1 c1(C(=O)NC(C2(O)CN(C(c3cc(C)ns3)=O)C2)C)cnc2n1CCCC2C C(=O)(C1=C(c2ccccc2)SCCO1)NCC1N(C(CC(C)CF)=O)CCCC1 Cc1ccnc2c(C(N3CCCC3CN(C)CCSc3ccccc3Br)=O)cnn12 c12ccc(cc1C(F)(F)F)[nH]2.C(=O)(C(C(C)O)NC(=O)CSC(C)C)OC CCCC(C)(O)C(=O)N1CCCC(O)(CCNC(c2nn(C(F)F)cc2Cl)=O)C1 C12(NC(C(Br)=C(C)C)=O)COC(C1)C(NC(c1scnc1C1CC1)=O)C2 c1(CC2OCC(C(=O)NCCOC(C)(C)CNC(C3(O)CCC3)=O)C2)ccccc1 C1(O)(CNC(CC2C(C)(C)CC2)=O)CCCN(C(c2ccc(C3CC3)cn2)=O)C1 C1(C)(NC(c2oc(C)c(Br)c2)=O)CCCN(C(C2Cc3nccn3C2)=O)C1 N1(C(C(C(CC)c2cccc(Br)c2)N)=O)CC2(CCC2)OCC1CO N1(C(c2c(OC)c(F)ccc2F)=O)C2CCCC1CN(C(=O)C(O)C1CC1)CC2 C(CN=C(NCC(F)F)N1CCCCC1)c1ccc(N(C2CCCCC2)C)nc1 N1(C(c2nc(CCOCC)oc2)=O)CC(C(=O)NCCCC(C)O)CC(C)(C)C1 c1(C(N(C2CC(NC(CSCc3nc(C)sc3)=O)C2)C)=O)cc(F)cnc1O Cc1oc2ncn(C)c(=O)c2c1C(=O)NCC1CC(F)(CNC(=O)CC(C)O)C1 c1(CC(=O)NCC23CC(NC(=O)Cn4nc(Cl)ccc4=O)(C2)C3)ccc(Cl)c(Cl)c1 n1(CCCF)nnnc1C1(C(C2CC(n3cncn3)C2)N)CC1.C1(C)CC1 N1(C(c2cc(OCC)n[nH]2)=O)CC2CC1(C(=O)NC(c1c(C)n[nH]c1C)C)C2 C(=O)(CC(C)CC(F)(F)F)NC(CNC(c1c(C#C)cnn1C)=O)(C)CO Cn1cnnc1CCCC(=O)NC(C1CCCN1C(=O)C=Cc1ccsc1)(C)C N1(C(CCCC)=O)CCC(N(C(=O)Cc2cc(CC)no2)CCO)CC1 c1(C(=O)NCCC(C)CCNC(=O)CC(C)(C)C#N)ccc2ncccc2n1 c1(C(N(CCCNC(C=CC)=O)Cc2ccccc2)=O)c(C)ccc(Cl)c1F c1(C(=O)NC23CC2CN(C(=O)CCCN2CCCC2)C3)cc(Cl)ccc1Cl c1(NC(C)CC(N)=O)[nH]c(=NCC2CCCC(F)C2)nc2c1ccn2C CC(C)CC(C(=O)N1CC(C)C(C(=O)NCC2CC(OCCO)N2)C(C)C1)C(C)C C1(NC(Cc2nn(C)c(Cl)c2)=O)CCN(C(=O)CCc2ccoc2)CC12CCC2 c1(OC)cc(CC(N2CC=CC2CNC(C23COCC2C3)=O)=O)ccc1O C(=O)(C1=NNC(C(F)(F)F)C1)NC1CCC(N(C)C(c2nc(Cl)cs2)=O)C1 C1(NC(C(CC)n2nccc2C)=O)CCOCC1NC(c1ccccn1)=O Cc1cc(C(C(=O)NC2CC2)N(CCCc2cccnc2)C)cc(C)c1F N1(C(C2(C)N(C(C=CCCCCC)=O)CCC2)=O)CCc2ccc(Br)cc2C1 c1(CN(CC(C)NC(=O)CC)C(C2(CCC)CCC2)=O)ccnn1CC N1(CC(=O)N(C2CCN(C(c3ncn(CC)c3)=O)C2)C)CCN(C)C(=O)C1 C1(C(=O)NCC(C)NC(c2ccc(F)nc2)=O)CC1C1CCCCC1 C1(C(=O)NCC(C)(C2CCC2)OC)CCN(C(=O)C=CC(C)C)CC1(C)C c1(OC)cc(NC(C2CCCC2CNC(=O)CC2CC=CC2)=O)ccc1[N+](=O)[O-] N1(C(C(CCC)OC)=O)CC2(CC(N(C(=O)CCOC3CC3)C)C2)C1 C1(C(=O)NCC2CN(S(C)(=O)=O)C2)CN(C(=O)CSC(F)F)CC1(C)C C(CCC(C(=O)N(C)C(C=C)C)NC(=O)C#CC1CC1)CC=C C1(OC(=O)Cn2ncc(Br)n2)Cc2ccc(Br)cc2C1 C1(O)(CNC(c2cnc(C)[nH]2)=O)CCN(C(=O)C=Cc2sccc2C)CC1 N1(C(c2nc(C)nc(O)c2)=O)CCN(C(C2COC(=O)N2C)=O)C2COCC12 N1(C(C(CC)Cc2ccccc2C)=O)CCC2C(C1)CN2C(c1cn[nH]c1)=O c1(CC)ccccc1C(=O)N(CC(O)CN(C(=O)COC(C)(C)C)C)C C(=O)(CC(C)(C)C(F)F)NCCC1N(C(C2N(C)CC(O)CC2)=O)CCCC1 C1(NC(c2cccc(CC)n2)=O)CN(C(=O)CC2CC(C)(C)CO2)CC12CCC2 N1(C(c2ccc(OC)o2)=O)CC(CCNC(=O)Cn2cnc(=N)[nH]2)OC(C)C1 N1(C(c2csc(Br)c2)=O)CC2OCC(C(N3CC4CC4C3)=O)C2C1 c1(CNCC)ccnc(C(N2CCN(C(=O)NC(CC=C)C)CC2)=O)c1 Nc1cc(C(N2CC(F)CC2CNC(C2(N3CCCC3)CCC2)=O)=O)cc(Cl)n1 c1(N(CC(C)C)C)ccc(C(=O)NC2COCCC2NC(C2(F)CC2C)=O)cn1 C1(CCNC(CCC)=O)CCCCN1C(=O)CCCC1CCCCC1 N1(C(c2c(C)nc(C)o2)=O)CC(CO)C2(CCN(C(C3CCCC3)=O)CC2)C1 O=C1CCN(Cc2ccc3occc3c2)C(=O)N1CCc1nccc(C2CC2)n1 C1(OC)CC(CNC(=O)C=Cc2cnc(C)s2)N(C(=O)C(c2nc(C)cs2)C)C1 c1(CNC(C2(C#C)CC2)=O)ocnc1C(=O)N(C1CCCC1)C1CC1 c1(SCCOCC2C(C#N)CN(c3ncccn3)C2)ccc([N+](=O)[O-])c([N+](=O)[O-])c1 C(C(F)(F)C(F)(F)F)OCCC(=O)NC1(C)CCN(C(c2cc(CC)no2)=O)C1 CC(C)CC(C)C(=O)NC1CN(C(c2ccc(C(F)(F)F)nc2N)=O)CC1F N1(C(c2cnn(C)c2C(F)F)C(=O)NCCCCCC)CCCCCC1C C(C1=CCN(C(c2conc2C(C)NC(=O)C(=Cc2ccco2)C)=O)CC1)OC N1(C(c2ccc(CC)cc2C)=O)CCC2CCN(C(=O)C(CC(C)C)OC)C2C1 CC(C)CC(C(=O)N1CCC(C(=O)NCC2CCC(=O)C2)C1)c1ccc(Cl)cc1 C(CC(C)(C)CC(=O)NC1CC(C)CN(C(c2cnn(C)c2C)=O)C1)OC c1(CC)noc(CCCNC(C2(CC)CN(C(=O)CC3(O)CCC3)C2)=O)n1 N1(C(C2CN(C)C2)=O)CCC2(CCCCC2NC(=O)CCc2cncn2C)C1 CC(C)C(CC(=O)NCC(CNC(=O)CN(C)C1CC1)CO)C(=O)OC(C)(C)C CN=c1nc(N2CCCC2)[nH]c(=NCc2ccc(Br)o2)[nH]1.C(CC#N)NC C1(NC(c2cccn2Cc2ccccn2)=O)CCCC12CN(C(=O)C1CC1)C2 c1(OC)cc(C(=O)OCCNC(C2(C3CCCO3)CC2)=O)cc2cn(C)nc12 Cc1ncoc1C(=O)NCCCCCNC(=O)C=CC(=O)NC(C)C c1(C(=O)NC2CC(C)N(C(=O)COc3ccccc3OC)C2)cc2ccsc2s1 c1(NC(N(CCC=C)Cc2ccccc2)=O)cc(F)cc(F)c1O c1(C(N(CCCNC(=O)C(C)c2ccsc2)CC)=O)cc2c(cc1Cl)N(C)CC2 c1(CC)oc(C(N2CCC(C(=O)NCC3CNC(=O)O3)C2C(C)C)=O)cc1C CCCC(O)CCNC(c1cc(C(=O)OCC)[nH]n1)=O.C(=O)C(C)(C)C N1(C(C2CC(C)OC2)=O)CC=C(CCNC(=O)Cn2cc(C3CC3)nn2)CC1 C(=O)(CCC(C)CC)NC(CCNC(c1nc(CCC)oc1)=O)COC n1(CC(OCC)OC)c(N2CCN(CC)CC2)nnc1CC1CC12CCOC2 C#CCCCCCCC(=O)NCC12CCCC(CN1C(c1cc(=O)cc[nH]1)=O)C2 C1(O)(C(C)NC(C2(CC#C)CCC2)=O)CCN(C(C2(C(F)F)CCC2)=O)C1 C1(C(=O)NCC23CC(CNC(C4ON=C(C)C4)=O)(OC2)C3)CCN(C(C)C)C(=O)C1 C=CC(C)(CC)C(=O)NCCCCCNC(=O)C(F)(F)CCn1ccnn1 C1(CNC(C(C2CC2)OC)=O)CN(C(C2(CC(C)C)COC2)=O)CCC1(C)C c1(CC(=O)N(CCCCCCNC(C2CC2(F)F)=O)C)ccc(Cl)cc1F c1(SCC)cncc(C(=O)NC(CNC(=O)Cc2cccc(Cl)c2)C2CCC2)n1 c1(CCC(=O)NCC2(O)CN(C(C3CCC(=O)N3)=O)C2)cncnc1 c1(C(=O)NCC(C)(O)CO)ccc(CNC(c2cccc(O)n2)=O)cn1 c1(C(N2CC(N(C(CCCc3onc(C(C)C)n3)=O)C)C2)=O)ncc(N)cc1Cl N1(C(CSCCOC)=O)CCN(C(=O)CCOCCOC)CC1.C1CCCO1 N1(C(CCOCCCOC)=O)CC2(CC2)CC1CNC(=O)CCC1CCOC1 C1(C(N2C(C#C)CC2)=O)CSCCN1C(=O)CC1CCCCN1C c1(N(C(c2csc(Br)c2)=O)CC2CNCC2O)cc(Cl)ncc1[N+](=O)[O-] c1(CCC(=O)Nc2c(C(=O)NCC(C)(C)C)n[nH]c2)ccc(Br)cc1 Cc1ccc(O)c(CC(N2CCC(C)(NC(c3cnnc(C4CC4)c3)=O)C2)=O)c1 N1(C(C2(C(C)C)CCCO2)=O)CC2(CC(NC(=O)CC(O)CN(C)C)CO2)C1 c1(C(N2CC(NC(=O)CSc3ccc(F)cc3)(CO)C2)=O)cc2cc[nH]c2cn1 C(=O)(C1=CC2(CCOCC2)C1)N1CCC(NC(C(CCCC)O)=O)(CO)C1 N1(C(C2C(CCC)C2)=O)CCC(F)(CNC(c2cnn(C(C)C)c2)=O)C1 c1(C(=O)NCC2(O)CC(C(=O)NCC(=C)Cl)C2)cccn(C)c1=O C(C)(C)(CCCC(=O)NCCCC1(O)CCC1)NC(c1n(C)nc(O)c1)=O c1(C(N2CC(C)C(CNC(c3ccc(C(N)=O)[nH]3)=O)C2)=O)ccc2c(n1)CCO2 CC1CC(CC(=O)N(CC(=O)N(c2ccccc2)C)C2CCC2)C(C)O1 N1(C(C2C(OC)(OC)CC2)=O)CC(NC(C2CC(C)(C)CN2C)=O)C(C)(C)C1 c1(C(=O)NC2CN(C(C3C(CCOC)C3)=O)CC2C)ccc2ncc(=O)[nH]c2c1 C1(C(N(CCNC(CCC=C)=O)CC2CC2)=O)CN(C(=O)CC(C)(C)C)CCO1 n1(CC(=O)NC2CC(C)(C)N(C(C3CC=CC3)=O)C2)ncn2nccc2c1=O c1(C(=O)NCC2(F)CCC(NC(COCC#C)=O)C2)c(C)ccc(C)c1C CCC(CC(=O)OCOC)NC(=O)C(CO)c1ccccc1.C1(CCF)C(=O)N1 N1(C(COC(CC)C)=O)CCC2(CCCC2NC(c2nncs2)=O)CC1 C(CC(C)(C)C(=O)NC1CC(CCNC(c2onc(C)c2C)=O)C1)OC C(=O)(C(C)CNC(=O)C(C)NC(c1cc(C)cs1)=O)OC CC(CN(C(C1CCOCC1)=O)C)C(=O)N(C(CC(=O)NCC(F)(F)F)C1CC1)C S(=O)(=O)(c1cnc(NCC2(F)CC2)c(Cl)c1)N1C(C)C(N(C)C)CC1 C1(CC)C(=O)NCCCN1C(=O)C(CN(C)C)NC(=O)Cc1cscn1 C(c1ccnc2ccccc12)=CC(=O)NCC1CC(NC(C2C3COCC23)=O)C1 C12(CNC(CC(C(C)C)O)=O)CC(NC(=O)C(C)CS(C)(=O)=O)(C1)C(C)(C)O2 c1(C(N2C(C)C(C)NC(=O)C2)=O)cn2cc(Cl)cc(Cl)c2n1.c12cccc(c1)CO2 CC(C)(C)C#CC(=O)NCC1CCC(NC(c2ccnn2C2CCCC2)=O)CC1 N(C(=NCCCNC(=O)OC(C)(C)C)NC1CCCC1)CC#CC c1(CC)ccccc1C(CNC(=O)CCC1CC1(C)C)NC(c1sccc1C)=O CC(C)(C)CC(O)CNC(c1coc(CNC(c2coc(CO)c2)=O)n1)=O CC1CCCC1(C)C(=O)NCC1(CC(=O)N(C)Cc2ccsc2)CC1 C1(CC(N)=O)CCN(C(C2CCCCN2C(=O)C(C2CCCCC2)=O)=O)CC1 C1(NC(c2cnc(C(C)(C)C)[nH]2)=O)CCSC12CN(C(c1c(Cl)csc1Cl)=O)C2 CCC(CC(=O)N(CC(CC)NC(c1ccc(Cl)nc1N)=O)C)CC(C)C c1(SC(c2ccc(Br)nc2)C)nc2ccccc2n1C c1(C(c2n(CCC)nnn2)NCCC2CCC(=O)N2)cc(C(F)(F)F)cc(C)c1 c1(N)cc(C)nn1CCCN1CCCC1.N1(C(=O)NCC=CC)CC(C(=O)OC)C1 CCCCCC(O)C(=O)NC1CC2(C1)CN(C(C1CCCC13CCC3)=O)C2 C(CCN=c1[nH]c(=NCCn2cnc3ccccc23)[nH]c2c1CSC2)N(C)C N1(C(CC2CN(C(C)=O)C2)=O)CCC2CN(C(=O)C3=CCC(F)(F)CC3)CCC2C1 CCC(C)CN=c1[nH]c2c(c(=NC3CC(C(C)(C)C)C3)[nH]1)COC2 C(N=c1[nH]ccc(C#N)c1[N+](=O)[O-])C1OCC(CNC(COc2cccc(C)c2)=O)C1 N1(C(C2(C)N(C(CC=C(C)C)=O)CC=C2)=O)CCC2C(C(N)=O)C2C1 c1(C(N2CC(CNC(CC=CC=C)=O)C(C)C2)=O)c(F)ccc(F)c1OC C=CC(C)(C)C(=O)N1CCC(CN(C(=O)C(C)(C)COc2ccccc2)C)C1 C1(CN(C)C(C2CC(c3ccc(Cl)cc3)(O)C2)=O)CCCN(C(C2(Cl)CC2)=O)C1 Cn1cncc1C(=O)Nc1c[nH]nc1C(=O)NCCc1cc[nH]n1 C1(OC)CN(C(=O)Cc2cncc(O)c2)CC1NC(=O)CC(C)C Cc1c(C(N2CC(NC(=O)CCCN=[N+]=[N-])C(C3CC3)C2)=O)ccc(F)c1F C1(CC)CN(C(c2cnc(N(C)C)cn2)=O)CCN1C(c1ncccc1F)=O CCCC(C(=O)NCC(CCOC)NC(c1c[nH]nc1OC)=O)S(N)(=O)=O C1(C(N2CC(C)(OCC(N3CC(CO)(CO)C3)=O)C2)=O)CC2CCC1CC2 Cc1ccc(C(=O)NC2CCCCC2NC(=O)CN(C)S(=O)(=O)N(C)C)nc1O N1(C(C2CCC(C)CC2)=O)CCCC2CN(C(c3csc(Cl)n3)=O)CCC12 C1(O)(CNC(C(C)Cc2ccccc2)=O)CCN(C(=O)Cn2cc(CO)nn2)C1 N1(C(CCOCCC)=O)CC(C(N2CCC3(C=CCO3)C2)=O)CC12CCC2 C=CCC(C(=O)N1CC(C(O)C(=O)NC2(COC)CC=CC2)C1)C(C)C O=C1Cc2c(N3CCc4[nH]nc(C(=O)Nc5ncnc6ccsc56)c4C3)ncnc2N1 n1(C(CC)C)nnnc1C(C)(CCCl)N(CC(F)(F)F)CCCOCC C(CNC(=O)CC(C)N1CCCC1=O)(C(C)(C)C)NC(C(CC)c1ccccc1)=O C(=O)(CCCC(=O)OC)NCC1CC(OC)CN1C(c1ccc(CF)cc1)=O C1(C)(CNC(CC(C)(C)OC)=O)CN(C(=O)C(C)C2=CCCC2)C(C)(C)C1 N1(C(c2csc(Cl)c2)C(=O)NCCOCC)CC2OCC(COC)C2C1 CC1CN(C(=O)CCCOc2ccc(F)cc2)CC1CNC(=O)COC(F)F Cc1cc(C(=O)NCC2CN(C(=O)CCC3CCOC3)CC2(C)C)nc(C)n1 N1(C(C(C)c2ccsc2)=O)CC2CC2(CNC(=O)CSCCN2CCOCC2)C1 c1(C2(C(N3C(CN(C(CC=C)=O)CC)CCC3)=O)CC2)cccc(Br)c1C c1(C(N2CC=C(CNC(C3=C(C)CC3)=O)CC2)=O)ccsc1S(N)(=O)=O N1(C(C2CC(O)(CC#C)C2)=O)CCN(C2CCN(C(=O)COCC(F)(F)F)C2)CC1 C1(NC(C=C(C)C(C)C)=O)CCCC(C(=O)NCCc2ncnn2C)CC1 CC1(C)CC(CNC(C2COCCN2C(=O)CC2(CO)CC2)=O)CCO1 C1(OC)CCC2(C(=O)NCCCCC3CCCN(C(=O)CCCF)C3)CCC12 Cn1ccc2nc(N3CCC(F)C(NS(=O)(=O)C(Cl)(Cl)Cl)C3)ncc12 CCCCCC(O)C(=O)NC12COC(C1)C(NC(=O)CN1CC3CC3C1)C2 N1(C(CC(CC)(F)F)=O)C2CCC1C(C)C(NC(c1c(OC)ncnc1C)=O)C2 C1(CN(CCC)CCNC(C2(O)CCSC2)=O)CC(c2ccccc2)=NO1 C1(CNC(CC(C)O)=O)CC(C)N(C(=O)CNC(c2ccccn2)=O)C1 C1(OCC)CC2(C1)CC2NC(C1(CNC(C2CC23CC3)=O)CC12CCC2)=O CC(C(=O)N1CCC(C)(CNC(c2cnn[nH]2)=O)C1)C(C)(C)O Cn1cc([N+](=O)[O-])cc1C(N1CCN(C(=O)C(C)(C)NS(C)(=O)=O)CC1CO)=O N1(C(C2C(COC)C2)=O)CC(NC(c2ccc(Cl)c(Br)c2)=O)CC1(C)C c1(C(C2CC2)NCC(C)CCO)cnc(Cl)c(F)c1.c1nnnn1C1CCCC1 C1(CC(=O)NCCOC2CCN(C(C3CC(O)C3)=O)C2)(CC=C)CCCC1 N1(C(c2c(C)nn[nH]2)=O)CCCCC2(C1)CN(C(=O)C1CCc3c[nH]nc31)C2 C(=O)(CCCC(F)(F)F)N1C(C)CC(CNC(c2ccc(CC)[nH]2)=O)C1 N1(C(CC2N(CC)C(=O)CC2)=O)CCCN(C(=O)CCOC(C)C)C(C(C)C)C1 c1(CC(=O)N(CC(C)N(C(=O)Cc2ccccc2Cl)C)C)cc(F)cc(Cl)c1 N1(CCC(C)(C)C#N)CCC2(CC1)CC(n1cc(NC(=O)C3CC3)nn1)CCO2 c1(C(N(CCC(=O)NCC(C(CC)(C)C)O)C)=O)c(C)cccc1C Cc1oc(C)c(C(=O)N(CC(C)Oc2ccc(Cl)cc2)C)c1C C(=O)(C(F)(F)CNC(=O)OC(C)(C)C)NC(CN(C(=O)Cc1csc(Cl)n1)C)C c1(C(N(CC(C)NC(c2c(SC)cccn2)=O)C)=O)cc(F)cc2nc[nH]c12 C1(C(=O)NC(C(=O)NCC2=CNC(=NC)C[SH]2OC)CCF)CC2CCCC2C1 c1(NC)ccc(C(=O)NC(C2CCN(C(=O)CC34CCC(CC3)C4)CC2)CO)cn1 C1(NC(CCC(=O)N(C(C)C)C)=O)COC2(C1)CN(C(C1(S(C)(=O)=O)CC1)=O)C2 N1(C(C(C)SCC)=O)CC(NC(=O)C(C)(C)COC(C)C)CC(O)C1 C(=O)(N=c1ccn(C(C)(C)C)[nH]1)C1N(C(C2CCCN2C=O)=O)CCC(CC)C1 c1(C(=O)OC)cc(S(=O)(=O)N(C)Cc2cccc(OC)c2O)c(C)cc1F N1(C(c2c(C)nc(CC3CC3)s2)=O)CCOCC(NC(=O)Cc2cc[nH]n2)C1 C1(C(N2CCC(NC(CCCC(=C)C)=O)C2(C)C)=O)CCc2cnnn2C1 c1(NC(C2C(NCc3cc(C#N)cc(Cl)c3)C2)=O)cc([N+](=O)[O-])ccc1Cl CCCC(CC1CCCCC1)C(=O)NCC1(C)CCCC1NC(=O)CSC(F)(F)F C1(CNC(C(C)=CC)=O)CC2(CCN(C(C3C4CCC(C4)C3(C)C)=O)C2)CO1 c1(C(N2CC(C)C(CNC(=O)C(O)C(F)(F)F)C2)=O)cn(CCO)c(=O)nc1O N1(C(C=Cc2cc(C)no2)=O)CCC(O)C(CNC(=O)C(Cl)=CCl)C1 c1(C(=O)NCC2N(C(CCN(CCC)C)=O)CC=C2)c(C)oc2ncnc(O)c12 S(=O)(=O)(c1ccc(Br)c(F)c1)NC1CCN(Cc2cccc(C#N)c2)C1 c1(C(=O)NCC(CO)NC(c2ccc(OC)nc2)=O)ccc2[nH]c(C)c(C)c2c1 c1(SC)cccc(F)c1C(N1CCCC(CN(C)Cc2cn(C3CC3)nn2)C1)=O N1(C(c2cc(C)cc(F)c2)=O)CC2CCC(C1)C(NC(=O)Cc1ccccc1)C2 C(=O)(C(O)CC(C)C)NCCCC(=O)NC(CC=C)C(=O)NC N1(C(C2C3CCC(=O)C32)=O)CCC2C(NC(=O)CCOCC3CC3)CC12 C1(CNCC(c2ccccc2)C)CCCN1NC(=O)C1CCOCC1 C(=O)(CS(=O)(=O)C1CCCC1)N1C2CCC(NC(c3c(C(N)=O)csc3)=O)(C2)C1 C(=O)(C(F)CCC(C)(C)C)NC(CCCC)C(=O)N(C)Cc1cn(C)nn1 c1(CC(C)=CC(=O)NCCC(C)NC(=O)Cc2ccc(C)o2)nncn1C CC1CN(C(C2CCC(C)N2C(=O)C2=CCCSC2)=O)CC(C)(C)O1 c1(COC)cn2ccccc2n1.C1(N2C(=O)C(C3CC3)NCC2)CCCCCC1 C(=O)(C(CNC(c1cnc2cc[nH]c2c1)=O)C(C)(C)C)NC1C(OC)COC1 Cc1ncsc1C=CC(=O)NC1(CNC(c2c(C)n[nH]c2C)=O)CCCCC1 N#CCCCCCC(=O)N1CCC(C(C(=O)NOC2CC3CCC2C3)OC)C1 C1(C(=O)NC23CN(C(c4n(C)ccn4)=O)C(CC2)C3)CCCC2(CCC2)O1 C1(C(=O)NCCCCCN(C)C(c2cccc(F)c2Cl)=O)C2CS(=O)(=O)CC12 Cc1ccccc1C=CC(=O)NCCC(C)N(C(=O)C=Cc1cscn1)C Cc1ccc(Cl)c2[nH]c(C(N3CC(NC(=O)CC(C)CN(C)C)C(F)C3)=O)cc12 N#Cc1cncc2[nH]c(C(=O)OCC(N3CCSCC3)=O)cc12 N1(C(C(C=CCCC)O)=O)CC2(CCCN(C(=O)COCCCOCC)C2)C1 c1(C(N(C2CC(NC(=O)C(F)CC3CCCCC3)C2)C)=O)cnc2sccc2c1 CC(C)(CCCNC(=O)C(c1cccc(Cl)c1)O)NC(=O)CC1CC1 c1(C2C(NC(N3CCn4c(CC)nnc4C3)=O)C2)ccnc2ccccc12 C(C(=O)NOCCC(C)C)OCCCC.C1(CC=O)C=CCCC1 C1(CC(N2C(CC(=O)NCC(C)CC3CC3)CCC2)=O)CC(=O)NC1=O CC(CC(=O)N1CC2CCC(C1)N2C(c1cscn1)=O)CC(C)(C)C CCCCC(C)CCC(=O)N1CC=CC(NC(C2(C)CC2(F)F)=O)C1 C(CC(C)(C)CC(=O)N(CC(O)CNC(=O)C1=NNC(=O)CC1)C)OC C(CC(N)=O)(C(=O)NCCc1ccncc1C)NC(CCCCC)=O CCC(C)CCCCC(=O)NCC1CC(F)CN1C(c1ccnc(C2CC2)n1)=O CC(C)C(C)(CNC(C1CC2C=CC1C2)=O)NC(c1cn(CC2CC2)nn1)=O CC1(C)CC(CC(N2CC(Cc3ccco3)C2)=O)N(C(c2cnc(O)o2)=O)C1 C1(NC(C2(CC)CCCN2C(=O)CN2CSCC2=O)=O)COC(C)(C)C1 Cc1cccc2c(CC(=O)NCCNC(C3CN(C)CC3C)=O)c[nH]c12 C1(CN(C(COCCOCCOC)=O)C)CC(C)CN(C(C2CC2C)=O)C1 N1(C(c2n[nH]c(C)c2C)=O)CC(NC(C2CC=CCO2)=O)C2(CCC2)C1 C(C(=O)NCCc1ncc(C)s1)(C(C)CC)N(C(CCC=C=C)=O)C C(=O)(C(C)S(C)(=O)=O)N(CC(CC)NC(=O)COc1ccc(F)cc1)C c1(C(=O)NCC(CC)NC(c2ccccc2)=O)ccc(Cl)cc1 C1(C(N2C(C(C)C)CN(C(C3CN(C)C(=O)N3)=O)CC2)=O)CCn2cncc2C1 C(C(C)(C)CNC(=O)CC1CCCO1)N(C(=O)CCn1cc(Cl)cn1)C c1(NC(C2(C)N(C(C3C(C)C3)=O)CC2)=O)cnnc2cc(Br)ccc12 N1(C(C(C)Oc2c(OC)cccc2)=O)CCC(NC(c2csnn2)=O)C1(C)C N1(C(c2cccc(C#C)c2C)=O)CCN(C(=O)C(F)CC(C)(C)C)C2(CCC2)C1 N1(C(C2CCC(CC)O2)=O)CC(C(=O)NCC(O)COC)CCC1(C)C Cc1cc(Cl)cc2cc(C(=O)NCC(C)CN(C(=O)CCN(C)C)C)[nH]c12 C1(NC(CCCN=[N+]=[N-])=O)CC2CC(NC(=O)Cn3cnc4c3CCCC4)CC2C1 N1(C(C(CC(=C)C)NC(C)=O)=O)CCC(C2CC2)C1CNC(C1CCCC2CC12)=O c1(C(=O)NC2(C)CC(NC(C3N(C)CCOC3)=O)C2)cc(O)cc(O)n1 c1(C(=O)NC2(CCOC)CCN(C(C3CCCS3)=O)C2)occc(=O)c1OC c1(C(=O)NCCNC(=O)Cn2cccnc2=O)nn2c(c1Br)CCC2 CCC(CC)CC(=O)NC(C(C)NC(=O)C(=Cc1cnc[nH]1)C)C(C)C c1(C(=O)NCCCCC2CCCN(C(COC)=O)C2)nsc2ccccc12 O=C1CN(CC(=O)NCC2(F)CCC(NC(=O)CCCn3ccnn3)C2)C(=O)N1 c1(C(N2CCC(NC(CC3C(C)C3(F)F)=O)(CF)C2)=O)ccc(S(N)(=O)=O)s1 CCN=c1cc(C(=O)NCC(CC(C)C)NC(c2cnn(CC)c2Cl)=O)cc[nH]1 N1(C(CC(=C=C)C)=O)CCN(C(C2CCCCO2)=O)CC1c1c(C)cccc1C C(=O)(CC1=CCN(C)CC1)N1CCCC(C(=O)NC(c2nc(C)on2)(C)C)CC1 Cc1ccc(O)c(C(N2CCC(CNC(c3ccc(Cl)c(F)c3)=O)C(C)C2)=O)c1 C(=O)(C(F)(F)C(F)F)N1CCCC(C(C(=O)NCC#CC)C)C1 Cc1ncc(C#N)c(N2CC(F)(C(=O)Nc3cnc(O)c(Br)c3)C2)n1 C(=O)(C#CC1CCOCC1)N1CC(CC)C(NC(=O)Cc2n[nH]c(=NC)s2)CC1 C1(C(N2CC(NC(CSCCCC)=O)C2)=O)CCc2n[nH]c(C)c2C1.C1C(=O)O1 c1(C(N2CC(NC(C(C=C)OC)=O)CC(F)(F)C2)=O)cc2cc(C)ccc2[nH]1 N1(C(C(C)OCC=C)=O)CCN(C(=O)C(F)(F)c2nccs2)CC1C1CC1 n1(CC(N2CC(C(C)NC(C3COC(C)(C)C3)=O)OCC2)=O)ncc(O)nc1=O C1(c2n(CCC)nnn2)(NCCc2cc(Cl)ccc2Br)CCOCCC1C C1(O)(CCNC(C2(C)C(C)C2)=O)CN(C(C2CC(c3ccccc3)C2)=O)C1 C1(NC(CCCCNC(C2C=C(C)CS2)=O)=O)CCCCC12CC2 C1(NC(c2ccc(OCC)nn2)=O)CCN(c2nc(C)cc(C)n2)CC1O N1(C(C(CC)OC)=O)CCC(C2(NC(=O)CN3CCN(C)C(=O)C3)CCC2)CC1 c1(C(=O)NCC(C2CC2)NC(Cc2c(C)nc[nH]2)=O)oc2ccccc2c1C C1(CC)CCOCCN1C(=O)CNC(=O)CNC(=O)NC1CCCCC1CC CC1CN2CCN1C(C(N1CC3CN(C(C45CC(C)C4C5)=O)CC3C1)=O)C2 C(=O)(CC1=NNC(=O)C1)NCC1(C)CCN(C(CSCC(=O)OC)=O)C1 c1(NC(C(N2CC(CNC(CNC(CC)(C)C)=O)(OC)C2)=O)C)c(C)noc1C c1(CC)ccc(C(N2CCC2CNC(C2CCCN(C3CCC3)C2)=O)=O)cn1 C(=O)(CCCC(N)=O)NC(C1(O)CCN(C(c2nc(OC)c(C)s2)=O)C1)C c1(C(=O)NCC2C(C)(C)CN(C(c3cc(C#N)c[nH]3)=O)C2)cc(Cl)c(O)c(Cl)c1 N#Cc1cc(CN2CCCC(C(=O)Nc3cc(Cl)cnc3F)C2)cc(Cl)c1 C#CCC(CC(=O)N(C)CC1OCCC1(C)C)NC(c1cncc(O)c1)=O c1(C(N2C(C)CC(NC(=O)Cn3ccc(=N)[nH]3)CC2)=O)ccc(O)c([N+](=O)[O-])c1 Cc1cc(O)n2ncc(C(=O)NC(C3(CO)CCC3)=O)c2n1.C12CC(C1)NC2 c1(OC)cc(NC(C)C)ccc1NC1CCOC(c2cccc(C(F)(F)F)c2)C1 C(=O)(C1CCc2scnc21)N1C(C)(C)C(CNC(=O)COC2CCOCC2)CC1 c1(-c2c(C)occ2)nc(C(C)CCN(C)C)n(-c2ccc(C(C)C)cc2)n1 C1(NC(C(C#C)(C)C)=O)CCCCN(C(c2cc(C)c(Br)o2)=O)C1 C1(CC(N2CCC2C2CC2)=O)CCN(C(c2cn(-c3cccnc3)nn2)=O)C1 C(=O)(C1CCCc2sc(C)nc21)N1CC(CCNC(C2N(CC)CC2)=O)(OC)C1 c1(C(=O)NCCCN(C(=O)C=Cc2sccc2C)CC)cc(C)c2[nH]nnc2c1 S(=O)(=O)(CC(=O)NC(C)C(C(C)C)NC(=O)CSc1ccccc1C)NC c1(-c2cn(-c3nn[nH]n3)nn2)ccc2c(c1)CCC2=O.c1(CC)ccc(Cl)c(S)c1 Cc1nn(CC(=O)NCC=CCNC(c2c(C)nsc2N)=O)c(C)c1[N+](=O)[O-] C1(C(=O)NCC2CN(C(c3ccc(Cl)cc3F)=O)C2)C2C3CC4C1C1C2CC3C41 N12CCC3CCC(C13)C2=O.N1(CCC)CCCCC1C(=O)OCC C(=O)(C1=CCCCO1)N1CCN(C2CN(C(c3cn(C)cc3C(F)(F)F)=O)C2)CC1 N1(C(C2(c3cc(C)no3)CCOCC2)=O)CCCC(C(=O)NC2CC2)CC1 N1(C(C2N(C)C(=O)OC2)=O)CCC(NC(=O)CC2CCC3(CC2)CC3)C1(C)C C1(CNC(=O)CCc2nc[nH]n2)CN(Cc2ccc(O)nc2)CCO1 C1(CC)CN(C(C2(NC(=O)NC3CC(OC)C3)CSC2)=O)CC(CC)O1 CC1=NS(=O)(=O)NC=C1C(=O)NC1Cc2ccccc2CN1c1ccnc2ccccc12 N1(C(C(c2ccccc2F)(C)OC)=O)CCC2(CCN(C(C3CCCO3)=O)C2)C1 N1(C(CCc2cc(C)oc2C)=O)CC(c2ccccc2)Cn2nc(C)cc21 Cc1nn(C)c(C)c1CC(N1CC(NC(c2cnc(O)nc2O)=O)CC(F)C1)=O C=Cc1cncc(C(=O)NC2CC(CO)N(C(C3CC(SC)C3)=O)C2)c1 c1(C(=O)NC2C(NC(Cc3c(C)cccn3)=O)C2)c[nH]nc1S(N)(=O)=O C1(C(C)C)CCC(C(=O)NCC2CC(F)(CNC(=O)CCN3CCCC3)C2)CC1 N12CCCC(C1)C2=O.C1(n2ncc(SCC)c2)CN(c2cncc(Cl)n2)CCO1 C1(CNC(C2(C=C)CC2)=O)CN(C(c2cc(OC(C)=O)n[nH]2)=O)C2CCN1C2 N1(C(C(C=C)(C)O)=O)CCC(C2(Nc3ncc4ncnc-4[nH]3)CC2)CC1 Cc1cc(Br)ccc1S(=O)(=O)N1CCCC12CN(C(c1cc(Cl)ccc1Cl)=O)C2 N#Cc1nnc(N2CC=CC(NC(=O)COc3ccc(F)cc3)C2)s1 C=C=CCC(=O)N(CC(C)N(C)C(c1n[nH]cc1C)=O)C C1(C)(CC(=O)NCC(C)(CNC(C2CN3CCC2C3)=O)OC)CCOCC1 N1(C(CC(C)N(C)C)=O)CC(NC(C2CC2C(C)(F)F)=O)CC(F)(F)C1 c1(-c2cccc(COC(C)C)c2)cccc(S(C)(=O)=O)c1 c1(CCC(=O)N(CCOCCNC(C=CC(CC)=CC)=O)C)ccc(C)s1 N1(C(C2COCCN(C(C(CCCC)F)=O)C2)=O)CCc2sccc2C1 C(=O)(CS(=O)(=O)C1CCCC1)N(CCNC(Cc1n(C)nc(CC)c1Cl)=O)CC C1(C(=O)NCCC(C)N(C)C(c2ncn(C)n2)=O)CCCC2(CCC2)O1 c1(C(N2Cc3cccc(-c4nccs4)c3C2)=O)cc2ccc(O)cc2o1 Cc1cc(F)c([N+](=O)[O-])cc1NC(c1ccnc(Cl)c1O)=O c1(C(N2C3C(NC(CCC#CC)=O)C(C3)C2)=O)cnc(Br)c(OC)c1 Cc1cc(C(=O)N(C(c2ccccc2)CNC(=O)Cn2cnnn2)C)nnc1O C1(NC(C(c2cnn(C)c2)C)=O)CC(F)(CNC(C2CC2c2cccnc2)=O)C1 C12(C(=O)NCC3(CC)CCCCO3)CCC(CC1)N(C(=O)CN(C(C)CC)C)C2 c1(OCC)cc(Br)cc2c(CNCC3CCCCN3CC(F)F)c[nH]c12 CCCC(C(=O)N1CCOC(CNC(=O)C(F)=C(C)C)C1)NC(=O)OC(C)(C)C c1(NC(C2CCC(C(C(Cn3cccn3)NC(N)=O)=O)C2)=O)nc2ccccc2[nH]1 CC1(C(N2CCC(C)(C(N3CC(O)(C(N)=O)C3)=O)C2)=O)CC2CCC1O2 c1(OC)cc(CNCC23CC2CN(C(=O)CNC(=O)C2CC2)C3)ccc1F N1(C(c2cnc(Cl)cn2)=O)CCC=C(C(=O)NCC2N(C)CCC2)C1 CCC(CN(C)C)C(=O)NC1CC(NC(=O)C(O)Cn2cncn2)CC1O C1(CNC(c2cc(OC)nn2C)=O)CC2(CO1)CN(C(=O)CC1CC(OC)C1)C2 C1(C)(CNC(C(C=C)NC(=O)OC(C)(C)C)=O)CCCN(C(=O)CSC(C)C)C1 C(=O)(NNc1cccc(C(F)(F)F)c1)c1[nH]cc(C)c1C c1(C(N2CC(CC)N(C(c3c[nH]c(=NC)s3)=O)CC2)=O)ccc2nc(C)[nH]c2c1 N1(C(C=C(CC)C)=O)CC2CC(OCC)C2C1.C1(C)C(=O)N2CC(C2)C(=O)N1 C(=O)(C1=C(C)OCCC1)NC(CC(=C)Cl)C(=O)N(C(CO)C1CC1)C CC(C)(CCNC(=O)C=CCO)NC(=O)CC1CC1(C)C C1(N(C(=O)COCC2CCCO2)CC)CCN(C(C2(CN(C)C)COC2)=O)C1 N1(C(c2cc(C)sc2N)=O)CC(O)CC1(C)C(=O)NC1CCC(C)(C)CC1 c1(C(c2ccc(OC)cc2OC)NC(C2CC2C)=O)cc(OC)c(OC)c(I)c1 C1(CC(N2CCC(C(CNC(C3(CCC)CCC3)=O)(C)C)C2)=O)CCCCC1O CCC(C)CCCC(=O)N(CC(C)CNC(C1(Cl)CCC1)=O)C C=C1CCC(C(N2CCCC2CN(C(=O)C(O)C2CCCC2)C)=O)CC1 C1(N(C(c2cc(C)ns2)=O)NC)CCN(C(=O)CC2CCCCO2)CC1.C1COC1 N1(C(C(c2ccc(F)cc2)C)=O)CCC(O)C(NC(C2CC23CCCCC3)=O)C1 C#CCC(C(=O)OC)NC=O.C1(C(=O)NC2(CCCN)CC2)CCCN1C(C)=O C1(NC(C(CC)(C)COC)=O)CN(C(c2cn(C)c(O)n2)=O)C2(CCC2)C1 C=CC1(C(N2CCC(O)(CN(C)C(C34CCCC3C4)=O)CC2)=O)CCOCC1 c1(CF)cnc(NC(c2nnnn2CCCSC2CC2)c2ccco2)c(Cl)c1 C1(NC(C(c2ccccc2)N(C)CC)=O)CN(C(C23CCC(C2)C3)=O)CCC1F N1(C(c2ccnc(C(C)C)n2)=O)CCC2CCC(C1)N2C(=O)C1=CCCOCC1 C1(C(=O)NCC(F)CNC(C2(C)CC(C(F)(F)F)C2)=O)(NC(C)=O)CCCC1 c1(C(=O)NC(CC)CN(C(C2CCCC2SC)=O)CC)nc2ccccn2c1F CC(C)(CC(=O)N1CCCC(NC(=O)CCCn2cncn2)CC1)CC(F)(F)F C1(C(=O)NC2(CC)CCN(C(=O)CCC(C)(C)OC)CC2)CCCC2CCCN12 c1(CC)ncccc1C(=O)NC(C1CN(C(C2C(C)C2C)=O)C1)C CS(C)(=O)=NCC(=O)N1C2CCC1C(CNC(=O)C=CC1CCCCCC1)C2 c1(CC)oc(C)cc1C(=O)NC(CCSC)C(=O)NCC1CC12CCC2 C(=O)(CCS(=O)(=O)Cc1ccccc1)N1CCC(C)(NC(CCOCC)=O)C1 N1(c2nc(C#N)cc(C)n2)CCC2(CCCN2C(c2cc[nH]n2)=O)CC1 N1(C(C(C(CC)(C)C)O)=O)CC2CC(N=c3[nH]nc(C(C)C)o3)C2C1 N1(C(c2ccc(CC)c(OC)c2)=O)CC(C)N(C(=O)COC2CCCCC2)CC1C c1(C(N2CCC(C3CC3)(Nc3ncccn3)C2)=O)cc2ccccc2cc1F C(c1ccccc1Cl)=CC(=O)NCC1CC(OC)CN1C(c1c(C)cnn1C)=O C1(C2C(C3CCCN3C(=O)NCC(C3CCCOC3)(C)C)C2)CC2CC1C1CC21 Cc1cc(C(=O)NC2CCCCC2CNC(=O)Cc2csc(=N)[nH]2)cnc1O C1(C(N2CCC(C(C)(C)O)C2(C)C)=O)Cc2ccccc2C1N Cc1cc(C(=O)NCC2CCC(C(=O)NCCC3CC3C)CC2)cc(O)n1 c1(OC)nccc(C(=O)NCC(C)(C)CN(C)C(c2ccc[nH]2)=O)c1F c1(C(=O)NCCN(C(COC)=O)CC(C)O)cc(C(C)C)ccc1F O=C(CCC1CC1(F)F)NCC1CC(NC(=O)CCc2cnoc2)C1 C1(C(=O)NCC(C2CCC2)NC(c2occ3c2CCC3)=O)C2CCC(F)(F)C12 CC1(C)CCC=C1C(=O)N1CCC(C2OCCC2NC(=O)C(N)=O)CC1 N1(C(c2ncn(C)n2)=O)CCC2(CC1)CC2NC(c1ccc(S(C)=O)cc1)=O Cc1nc(C(C)C)cc(CNCC2(NC(c3cnco3)=O)CCCCC2)n1 CCCCCC(F)C(=O)NCC1(OC)CN(C(C2CC2(F)Cl)=O)C1 N1(C(c2c(OC)ccc(F)c2)=O)CC2CN(C(=O)C(C)NC(C)(C)C)CC2(C)C1 c1(C(N2CCC(O)(CN(C)C(C3(C)CC(C)(C)C3)=O)C2)=O)ccc2ccsc2c1 C(=O)(C(C(C)(C)C)NC(=O)CN1CCC(=O)CC1)N(C(C)CC(N)=O)C c1(C(N2CCC(CCNC(CCC(C)SC)=O)C2)=O)ccc2nn[nH]c2c1 C1(CC)CCCC1CNC(=O)N(c1sccc1SC)C C12(C(=O)NCCC(C)NC(c3cc(N)ccc3O)=O)CCCN(CCC1)C2 C1(C(C(=O)OC)(C)C)CCN(N2CCCCC2C2CCCCC2)CC1 C(=O)(C1=CCOCC1)C1C(C2CCCCN2C(=O)Cc2cccnc2O)(C)C1 c1(C(C)NC(c2cccc(-c3ccc(CCC)s3)c2)=O)ccc(Cl)c(Cl)c1 C1(O)(CNC(CN2CC(CC)C2)=O)CCN(C(c2ncccc2C)=O)CC1 Cc1nc(C(=O)NC(C)CC(C)NC(=O)CCOCCN(C)C)c2ccccn12 C=CC(F)(F)C(=O)NCCCCCN1CCN(C(=O)CC2OCCC2C)CC1 C1(C)(CNC(C(=O)Nc2c(C)cccc2C)=O)CN(C(C2CC2F)=O)C(C)(C)C1 C1(OC)(CNC(C2COCC2C(N)=O)=O)CCN(C(=O)Cn2cc(C)cn2)C1 C1(CC(NOCCCN(C)C)=O)CN(C(=O)Cc2cn(C)cn2)CCC1C c1(C(=O)NCC(C2CCOC2)NC(c2n(CC)ccc2)=O)ccc(Cl)nc1C C1(C(N2C(C)CC(CC(=O)Nc3ccccc3CCO)C2)=O)OCCCC1(C)C N1(C(c2ccc(CC)[nH]2)=O)CCCC2C1CCN2C(=O)CCC1CCCN(C)C1 C(=O)(C1CC(=O)c2ccccc21)NC1Cn2c(cc(C(=O)O)n2)OC1 N1(C(CCOCCCOC)=O)CCN(C(c2cc(F)n(C)n2)=O)CC1CCOC C1(NC(C2(Br)CC2)=O)COC2CN(C(C3CCC4(CCC4)CO3)=O)CC12 CCCCCC(C)(CC)C(=O)N1CCC1CNC(c1c(Cl)n[nH]c1C)=O c1(SCC(=O)NC(CN(C(=O)CC2C=CCC2)C)(C)C)nncn1C C1(F)(CNC(C(C)OCC=C)=O)CCN(C(c2cc(CN)on2)=O)C1.C(C)(C)(C)O c1(C(=O)NC(CC)(CNC(C2CC2C2CCCO2)=O)CC)ccc(C)c(C)c1Cl C1(C(N(CC(CN(C)C)O)C)=O)CCC=CCC1NC(c1ccnnc1O)=O c1(N2CCC(CCC#N)CC2)nc(CC(=O)N2CCC2)c2ccccc2n1 C1(C(N2CCC(CNC(CC(C)CN(C)C)=O)CC2)=O)CS(=O)(=O)CC(=O)N1 c1(C(N2CC(CCNC(C(C)n3ccnn3)=O)C2)=O)ccc(OCCOC)cc1 Cc1c(C(N2CCCCC2C(=O)NCCc2ncccc2F)=O)nnn1C N1(C(C=CC(=O)OCC)=O)CCC(C)C(NC(c2ncccc2OCC)=O)C1 c1(C(N2CC(C)CC(NC(C3(CC)CC3)=O)C2)=O)cc(F)cc2nc(C)c(C)nc12 c1(NC(C)=O)ccc(C(N2CCN(C(c3ccc(F)nc3C)=O)CC2)=O)cc1C C1(NC(C2C(C(=O)NC(CC(=O)OC)C)C2)=O)CC(=O)N(C(c2ccccc2)C)C1 O=C(C1CCc2cc(F)ccc21)N1CC2CC(C1)N2C(=O)Cc1ccc(O)nc1 C1(NC2CCC(CC)CC2)CCC12CCOCC2 c1(N2C(=O)CC(C(N(CC#N)CC3CC3)=O)C2)ccc2c(c1)CCC2 C(CCCCCNC(C1(C(C)(C)O)CCC1)=O)NC(C(c1ccccc1)C)=O C(CCC(C)CC(=O)NCCCCC(C)NC(c1c(C)ccn1C)=O)=C(C)C C1(CC(=O)NC(CO)CO)CC2(C1)CN(CC1CCCS1)C2 N1(C(c2ccc(OC)o2)=O)CCN(C(C)CNC(C2CCCN(C)C2)=O)CC1 N1(C(C2C(C(C)(F)F)C2)=O)C(C(=O)NCC2(C)CC3(CCC3)C2)CCC12CC2 C1(CCCC(=O)NC)CCCN(C(=O)NC2CC(c3cc(CCOC)on3)C2)C1 C1(N(CCOC)C(c2ccn(C)n2)=O)CCN(C(=O)C(O)CN2CCCC2)CC1 N1(C(C(CC)(F)F)=O)CCc2nnc(N3CCSc4ccccc4C3)cc2C1 N1(C(CCC=C)=O)CCN(C(c2csc(Br)n2)=O)C(CO)C1 CC(C)(C)C#CC(=O)NCC1CCCC1NC(=O)C=CC(c1ccc(N)cc1)=O CCC(CC(=O)NCc1nccc(O)n1)NC(=O)CCc1nc(C)no1 C=CC(O)C(=O)NCCN(C(=O)CCc1nc(C(C)(C)C)no1)CC N1(C(c2c(C)ccnn2)=O)CC2CN(C(C3(CO)CCCC3)=O)CCC2(CO)C1 C=CCCCC(C(=O)N1CC=CC1CF)NC(c1ncccc1CC)=O Cc1[nH]c2ncnc(N3CCCC(CO)(NC(=O)Cc4cccs4)C3)c2c1C N#CC1(C(c2nnnn2C2CCCC2)NCC2CCCC(F)C2)CCCCC1 C(CC(C)(C)CC(=O)NCC1CC(C)(C)CN1C(=O)C(C)C(C)O)OC C1(CCN(C)C)OCCC12CN(C(=O)Cc1ccc(OC(F)(F)F)cc1)C2 c1(C(N(CCCNC(C(F)OC)=O)C2CC2)=O)ccc(-c2cscn2)cc1 C=CC1(CC(=O)NCC2CCCN(C)C2)CN(C(c2c[nH][nH]c2=N)=O)C1 CC(C)(CCSc1ccccc1)N=c1nn[nH]n1CC(F)(F)F c1(OC)cncnc1N1CCC(CC(=O)NCC2(CCO)CCC2)C1 N1(C(c2c(C)cc[nH]2)=O)CCC2C(NC(c3cccc4sccc34)=O)C2CC1 Cc1nc(N2CCCC3(NC(C4CC45CC(C)(C)C5)=O)CC3C2)cc2nncn12 CC1OC2(C)CC1(C(=O)NC1CC3CC1N(C(=O)CCn1cnnn1)C3)C2 n1(CC=CC)c(CN2CCC(N(C)C)CC2)nnc1-c1ncc(C)o1 c1(CC(=O)NCC(C2CCC2)NC(C2C(C(=O)OC)C2)=O)cn(C)nc1C C1(CNC(C2C(C(C)O)C2)=O)C(C)CCN1C(=O)Cc1cncnc1 N1(C(CCC=C)=O)CCCC(C)(NC(c2ocnc2-c2ccccc2)=O)C1 C(CC(C)(C)C(=O)NCC(C)C(=O)OC)NC(C(C=C)CC)=O C1(NC(=O)Nc2c(OC)c(C#N)c(F)cc2)CCC2C3C=CC(C3)C12.C(C)(=O)N c1(C(N2CCC(OCCNC(C3(C)CCCO3)=O)C2)=O)cn2c(n1)CCCC2 C1(CC)CCCN(C(C2CC(O)CN2C(=O)CC2CCOC2(C)C)=O)C1 CCCCC(C(=O)NCC1CN(C(C2(CN(C)C)CC2)=O)CCC1(F)F)C(C)C Cc1cc(C(=O)Nc2ccc(NC(C3CC4CCC3C4)=O)nc2)cnc1F C(=O)(C(Cc1cn[nH]c1)NC(c1nccn1C)=O)NC(C)C(C)n1cncn1 N1(C(C2(CNC(CN(C)C)=O)CC23CCC3)=O)CCC2CCC(C1)N2C.C1C(=O)N1 c1(C(=O)NC2CCN(C(C(C3CCCC3)OC)=O)C2)ccnc(Br)c1 CC(c1ccccc1F)=CC(N1CCOC(CNC(c2cc(O)nn2C)=O)C1)=O N1(C(C(C(F)(F)F)OC(C)=O)=O)CCN(C(c2nc(C)oc2C)=O)CC(O)C1 N1(C(CON)=O)CC2CCC2(NC(=O)C(c2ccc(NC(N)=O)cc2)=O)C1 C=CCCCC(C(=O)O)NC(=O)CCC1CCCOC1 c1(CC)cnccc1Cl.n12nnnc1C2.C1CO1.C1CO1.C(C)C N1(C(C(=O)NCCCSC)CCc2ccccn2)CCCSCC1C1CC1.C1CN1 C12CCN(C(=O)C1)C2=O.c1(CC(N2CC(O)C2)=O)csc(-c2ccsc2)n1 CC(C)(CC(=O)NC1CCN(C(C2CC(F)C2)=O)C12CC2)CC(F)F C(=O)(C(C)(F)C(C)(C)F)NC1(CNC(CCN2CCN(CC)CC2)=O)CC1 CC12CCC(C(=O)NCCOc3cccc(F)c3C(N)=O)(CC1)OC2 C(=O)(C1CCc2c(Cl)cccc21)NCC(C)CNC(=O)COC1CC=CC1 C1(OC)(CNC(C2CC2C)=O)CN(C(c2cnn(CC3CCCCC3)c2)=O)C1 c1(CNC(=O)NCCNCCNC(c2cccc(C)c2)=O)n[nH]c2c1CC1CC21 CC1CCCC(CC(N2CCC(NC(C3CCCCC3)=O)CC2)=O)C1 N1(C(Cc2ccc(OC)cc2)=O)CCCC1C1CCCN1C(c1cncs1)=O N1(C(=O)Nc2c(OC)cc(OC)c(Br)c2)CCN2CCCCC2C1 C(CCN=c1cccc(S(=O)(=O)N(C)CC2CC3(CC3)C2)[nH]1)OC=C C1(C(=O)NC(CC)CC)CCCN(C(C2CCCN(C)C2)=O)C1 c1(C(=O)OCC)coc(C(C(=O)Nc2cn(CCO)nn2)N(C2CSC2)C)n1 c1(C(=O)NCC2CC(NC(CC3CCCC(OC)C3)=O)C2)cc(O)cc(F)c1 C(=O)(C1OCCc2ccccc21)NCC1CN(C(C2(CCOC)CCCC2)=O)C1 c1(C(C)C(=O)NCC2CCCCN2C(=O)Cc2nc(=N)[nH][nH]2)ccc(Cl)cc1F C1(C(=O)O)CCCC2(CCN(C(C3Cc4ccccc4OC3O)=O)C2)O1 C1(C(CC)NC2(C(=O)OC)CCNC2)(OC)CCCOC1 c1(C(N2C(C)CC(NC(C3CCC(C(N)=O)O3)=O)C2)=O)cc2c(Cl)cccc2s1 c1(CC)ccc(C(=O)NCC2CCC2NC(c2cc(O)nc(C)n2)=O)cc1OC CC1(C)COC(C(N2CCC(CO)(NC(c3cnns3)=O)C2)=O)C1 Cc1ccc(C)c(SCC(=O)NC2CCN(C(=O)C=CC3(C)CCOCC3)C2)c1 C(C)(C)(CC(=O)NC1CC(C#N)C1)N(C(CC1C(C)CCC1)=O)C N(C(=NCCCC(=O)OC)NCCCOC)C1CC(n2cc(C(=O)N(C)C)nn2)C1 C(=O)(C(CC(C)C)OC)NCC(CC=C)NC(=O)CC1(O)CCCCCC1 C(=O)(CCCCCCN=[N+]=[N-])N1CC(CNC(C(CCC)(C)C)=O)OCC1 c1(N(CC(=O)NC23CC(C2)C3)C(=O)NCCCc2csc(CO)n2)ccc(Cl)cc1 C1(O)(CCNC(COCCCCC)=O)CCN(C(=O)C2=CCCSC2)CC1 c1(C(N2CCC(Nc3cccc(C)n3)C2)=O)cc(C#N)ccc1Cl N1(C(CCCCC)=O)CCC2(CC1)CC2NC(c1cc(Cl)cc(Cl)c1)=O N1C2c3ccccc3CC2C1=O.CC1(C#CC(=O)NC2(C(N)=O)CCC2)CCCO1 C1(C2CCCN(C(=O)Cc3nc[nH]n3)C2)(NC(CN(C(COC)=O)C)=O)CC1 Cc1cc(CCNC(c2occc2CNC(=O)C(C)NC(N)=O)=O)ccn1 c1(-n2c(C(n3ccnn3)C)nc(CCC(C)(C)C)n2)ccc(F)c(F)c1 CC(C)(C)C(O)C(=O)NCCN(C(=O)C=Cc1sc(Cl)nc1Cl)C1CC1 C1(C)(C(=O)Nc2c(C)nccc2)CC(F)(F)CN1C(=O)COCC1CCOC1 N1(C(c2n(C)cnc2)=O)CCCC(C2CC2NC(=O)C(c2cccc(Cl)c2)O)C1 Cc1nc(CC(C)C)oc1C(=O)N(CC(C)CNC(=O)CC1CCC1)C C1(NC(CCn2ncc(C)c2)=O)CC2CC1N(C(=O)CCC(C)N(C)C)C2 CC1CCc2n[nH]cc2C1C(=O)N1CCC(F)(CNC(C2(O)CC2)=O)CC1 N1(C(CC=CCCCCC)=O)CCC2(CC2NC(c2nn(C)cc2Cl)=O)C1 N1(C(c2c(C)ocn2)=O)CCOC(CC2(C(N(C)C(C3CCCC3)=O)=O)CCC2)C1 CN1C(=O)CSC1=CC(=O)NCC1CCC(NC(c2cc3ccccn3c2)=O)C1 c1(CC)c[nH]nc1C(N1CCCC1CNC(c1ccc(C(=O)OC)[nH]1)=O)=O CC(O)CC(C)(C)CNC(C1(CNC(c2ccoc2)=O)CCCCC1)=O c1(C(=O)NC2(CNC(c3cccnn3)=O)CC2)ccc2c(c1)CC2 C(=O)(C1CCCn2nccc21)NCCCCN(C)C(C1CCc2nn[nH]c2C1)=O N1(C(CC2CCN(C(C(C)OCCC=C)=O)C2)=O)CCOC2(CCC2)C1 C1(CC(=O)NC(CC)CNC(=O)CNC(=O)OC)CCn2c(C)cnc2C1 Cc1nnc2n1CC(C(N1CC(C)C(C)(CNC(=O)C(Cl)=CCl)C1)=O)CC2 N12CCCC(C1)OCc1cn(nn1)C(C)(C)C2=O.c1(C(=O)NC2CC2)cnn[nH]1 c1(CC(=O)NCC(C)CN(C)C(c2sccc2Br)=O)csc2nccn12 C12(C(=O)NC3C(C)CN(C(=O)CCc4cnoc4)CC3)CC(CO)(C1)OC2(C)C N1(C(=O)NC)CC2CC1CN2C(=O)C(C1CCN(C(C2CCN(C)C2=O)=O)C1)F C1(C(=O)NCCC2(CNC(=O)CCNS(C)(=O)=O)CC2)(CC)CCC(O)CC1 C(=O)(C1=C(C)OCCC1)N(CC(CNC(c1cncc(C=C)c1)=O)(C)C)C C(C1c2ccccc2CN1C(c1cnc(C(F)F)nc1)=O)OC Cc1cncc2cc(C(=O)NCC(C3CCCN3C(C3CCNC3=O)=O)(C)C)sc12 C1(C)(CN(C)Cc2scnc2-c2ccc(Br)cc2)CC(=O)C12CCC2 c1(C(N2CC3OCC(C(=O)NC4CCN(C)CC4)C3C2)=O)[nH]nc2ccncc12 N1(C(C2(C(F)F)C(C(=O)O)C2)=O)CC2(CCN2C(c2ccc(F)cc2)=O)C1 C(=O)(C1=COCCC1)N(CCNC(c1c(C(C)C)ncnc1)=O)C CC(C)(C)CCCCC(=O)NC1CC12CC(NC(=O)C(F)n1cccn1)C2 N1(C(CC=CC=C)=O)CCC2(CC2NC(c2ccc(C(F)F)nc2)=O)C1 c1(NC)cnccc1C(=O)N(C)CCN(C(c1cc(C)sc1N)=O)C(C)C N1(C(CN(CCC)C(C2CC2(C)CC)=O)=O)CCC(C)(C)C(=CC2CCC2)C1 N1(C(C2(NC(c3cc(C)oc3C)=O)CCC2)=O)CCC2(CCOC2)C1 c1(C(=O)NC(C)CNC(=O)CC2(O)CCC2)csc(C(C)OC)n1 C1(C(=O)NCCSCC=C)CC=CCN1C(C1CCC1COC)=O C12(C(=O)NCCCN(C(Cc3ccc(C#N)cc3)=O)CCO)CCCCC1OCC2 c1(C(N2CC(NC(Cc3c(C)nccc3)=O)C(F)C2)=O)ccc2nccn2c1 C1(CNC(c2c(C)nc[nH]2)=O)CN(C(=O)CCC=Cc2ccccc2)CCN1C C1(C(C)(C)CNC(c2cncs2)=O)CCN(C(C2(C)COC(=O)C2)=O)CC1 c1(C(=O)NCCCN(C(=O)CN(C)C(N)=O)CCC)cn(-c2ncccn2)cn1 C(=O)(CS(=O)(=O)CC1CCCO1)NC(C1CN(C(C(=O)NCCOC)=O)C1)C C(=O)(C(C)(C)NC(=O)CC1CC1C1CC1)NCC(C1CCC1)OC c1(CCNC(C(C=C)(C)CC)=O)cc2cccnc2nc1C.C1(=O)C2=CCN1C2 C1(C(=O)NCC2(O)CN(C(=O)Cc3csc(C)n3)C2)(OC)CCCCCC1 C1(NC(CC=C)=O)CCC(C)N(C(=O)C=Cc2ccccc2OC)C1 C1(C(=O)NC2C(NC(C(C)OCCOC)=O)C2)CCOC1c1ccncc1 S(=O)(=O)(CCCCS(=O)(=O)N1CCc2c(F)cccc2C1)NC(C(=O)OCC)C C1(OC)CCCC(C(=O)NCCCCC(C)NC(C2CCCCN2C)=O)C1 N1(C(c2n[nH]c(C)c2O)=O)CC(O)CCC1C(=O)NCCCC(C)CO C(CO)(C(C)(C)CO)NC(C(COC(C)=O)NC(C(CCC)C)=O)=O C1(C(N(C(CNC(CC2CC(C)C2)=O)C)C)=O)C(C)C1(F)F c1(CC(=O)NCC2(F)CCN(C(C(C)(C)SC)=O)C2)cccc(C)c1Cl c1(C(=O)NCC(C)(C)SC)cnn2ccc(-c3ccc(O)c(C)c3)cc12 CCN=C(NC)NC1CC1c1ccco1.c1(C=O)cc(C(C)C)no1 C(=O)(C1=COCC1)NCCC(=C)CNC(=O)C(O)Cc1ccccc1Cl c1(C(=O)NCC(CNC(C2(C)CC=CCC2)=O)O)ccc2nc(N(C)C)sc2c1 N1(NCCOC(=O)CC2CCC(C(F)(F)F)O2)CCNC(C2CC2)C1=O n1(CCOC)nccc1C(N1CCC(CN(C)C(C23CC(C)C2C3)=O)C1)=O N1(C(C(COC)C)=O)CCn2c(CNC(=O)CC3COCCN3C)nnc2C1 c1(C(=O)NC(c2cc[nH]n2)C)ccn2c(Br)cnc2c1 CC1CCCC(OCC(=O)NC2CC(C)(NC(=O)COC3CCOCC3)C2)C1 Cc1ccc(C)c(CNC(C2(F)CCCN(C(=O)C=CC3CC3)C2)=O)n1 CCC(CNC(=O)CCC(C)NC(=O)C(C)NC=O)C(C)(F)F CC1(C)CCCN(C(c2cc(CCO)on2)=O)C1CNC(c1csc(O)n1)=O C1(C(=O)NC(CNC(Cc2ccn(CC)n2)=O)(C)C2CC2)CN2CCN1CC2 CC1CCCN2C1CNCC2=O.c1(NC(=O)C=C2CC2)ccc(O)cc1 Cc1onc(CC(N2CCCC2CN(C(=O)C=CC2CCCO2)C)=O)c1C#N C(=O)(C(C)CC(N)=O)N(C1CCN(C(CC=CCC)=O)C1)C c1(C(N2C(C(=O)NC3(C(=O)OC)CC3)CCC3CC32)=O)ccccc1C#CC1CC1 C(CC(C(=O)N1CCCC(C)C1)NC(=O)CNC(c1ccco1)=O)=CC C1(C(=O)NCCOCCN(C)C(C23CCC(CC2O)C3)=O)CC2CCC(C1)C2O C1(SC)CN(C(c2cnccc2Cl)=O)CC1NC(=O)CC1NC(=O)NC1=O N1(Cc2n(C)ncn2)CCC(C)(NC(=O)NC2CCC(O)CC2)CC1 S(=O)(=O)(CC(=O)NCC1CC(F)(CNC(C2CCS(=O)CC2)=O)C1)NC N1(C(c2ncc(OC)nc2)=O)CCC2CN(C(=O)C(=Cc3cccs3)C)C2C1 CCCC(CC)C(=O)NCc1nc(CNC(C2CC(CF)C2)=O)cc(O)n1 N1(C(C2CC(C#N)C2)=O)CC(CNC(C2CNC(=O)C2)=O)OC2(CCC2)C1 C1(C(=O)NCc2ccsc2)(NC(CN(S(C)(=O)=O)C)=O)CCN(C)C1 C1(CC)CCN(C(=O)C(C(C)C)OC)C1CC(=O)N(C)CC1(OC)CCC1 C1(C(=O)NCC(=O)OC(C)(C)C)CC12CN(C(=O)C(c1ccc(Br)cc1)(C)O)C2 N1(C(C2C(C(CCC)=O)C2)=O)CC2C3COCC3C2C1.c12ccc(cc1)o2 N1(CC)CCCC(C(N2CC(OCCC(N3CC(C)(CC)C3)=O)C2)=O)C1 c1(CC)cccc(C(=O)NC2CCN(C(=O)C(O)Cc3ccccc3)C2C)c1N O=Cc1ccsc1-c1ccc(-c2ccc(N3CCN(C(=O)CBr)CC3)nc2)cc1 C(=O)(C(C)(C)N(C(N)=O)C1CC1)N(CC(F)(F)Br)C N1(C(CCn2cc(COCC=C)nn2)=O)CC(c2ccccc2)C(C#N)C1 CCCC(C(O)C(=O)N(C1CC1)CCc1ccccn1)NC(C1CCOC1)=O C1(CC(=O)NCCOCCC#C)CC(NC(c2cn[nH]c2)=O)C1(C)C c1(C(C)C)cnn(CC(N2CC(NC(c3coc(CN(C)C(C)C)c3)=O)C2)=O)c1 C1(C(N2CCC(N(C)C(c3nccnc3C(N)=O)=O)C2)=O)CC(C)(C)CN1C c1(C(=O)NC(C)CN(C)C(c2cc(C(F)(F)F)on2)=O)cncc(Cl)c1 C1(C(N(C2CCCC2)CCC#C)=O)C=CCN(C(=O)CP(C)(C)=O)C1 c1(C(=O)NCCCC2(NC(CC3(C#N)CC3)=O)CC2)c(Cl)cccc1Cl Cc1cnsc1C(=O)NC(C(=O)N(C1CC(C)(C)C1)C)c1cccs1 CC(C)CC(O)C(=O)NC1CCN(C(c2cccnc2NS(C)(=O)=O)=O)CC1O N1(C(c2c(C)ccnc2)=O)CC2CCN(C(c3cc(Cl)c(Cl)cc3Cl)=O)C2C1 C1(CNC(c2cc(C)nc(O)n2)=O)CC2CCC1N(C(C1CC13CC3)=O)C2 C1(NC(=O)NCC2(CC(NOCC)=O)CC2)CC2CCCC2C1 C1(CCNC(C2CC23CCSCC3)=O)CCCN(C(=O)Cc2csc(S)n2)CC1 C1(C(=O)NC2CCN(C(C(C)(C)n3cnnn3)=O)C2)CNC(=O)CC12CCC2 Cc1nc2c(o1)CCCC2OC(C1CCCC(OC(F)(F)F)C1)=O C1(CN(C(=O)C(=O)NC2CC2)C)CCCN1C(=O)COC1CCCC1 c1(-n2c(C(COCC)(C)Nc3nnc(C)o3)nnn2)ccc2c(c1)OCO2 C1(NC(c2ncccc2Br)=O)CC(CO)N(C(=O)CSc2n[nH]c(O)n2)C1 C(=O)(CCP(C)(C)=O)NC(CC=C)CNC(C1CC(=O)N(CCN(C)C)C1)=O C(CC1=CCCCC1)NC(CCC1(NC(CC(C)n2cccc2)=O)CCCC1)=O N1(C(C2CCCN(C)C2)=O)CCC(C#N)(C(N2C3CCC2COC3)=O)C1 C#Cc1ccc(C(=O)NCC2COCCN2C(=O)C(n2ccc(C)n2)C)cc1C C1(C(=O)NCC2CCCN(C(c3cncc(O)n3)=O)C2)CCn2ncnc2C1 N1(C(=O)OC)CCCC(C(=O)NCCC(C)(C)NC(C2CC(=O)N(O)C2)=O)C1 c1(C(N2C3CN(C(c4cccc(OC)c4OC)=O)CC32)=O)cc(O)ccc1[N+](=O)[O-] CCC(C)C(O)C(C)C(=O)N(CC(=O)NCC(CC)C1CCC1)C c1(OCCCCOC(C)=O)cccc(NC(=O)CC(c2ccc(F)cc2)C)c1 c1(C(N(C2CCC(C)(C)C2)C)=O)cccc(NS(=O)(=O)Cc2ccccc2Br)c1 C1(C)(NC(C2CC(OC)CN2C(=O)C=Cc2ccncn2)=O)CCC(=O)NC1=O N1(C(C2(C(C)C)CNC(=O)C2)=O)CC2OCCN(C(c3cnc(=N)[nH]c3)=O)C2C1 c1(OC)cc(CN(C2CCNCC23CC3)C(=O)CNC(=O)C(C)(C)C)cc(Cl)c1 c1(C(N(CC(CNC(CCOC)=O)C)C)=O)ccc([N+](=O)[O-])cc1[N+](=O)[O-] C1(NC(CCOC(C)C)=O)CC2(CCN(C(=O)C(C(C)C)c3cccs3)CC2)C1 c1(C(CC)NC(=O)C(C)=CCNC(c2coc(C(C)C)n2)=O)ccncc1 c1(C(N2CC=CC(C(=O)NC3(C)CC(=C)C3)C2)=O)ncc(N)cc1C N1(C(Cc2cnc(C)[nH]2)=O)CCC2(NC(C3CC4CCC3CC4)=O)CCCC12 CC1CC(CNC(c2snc(O)c2Cl)=O)CCN1C(=O)C1=CCCSC1 C1(CNC(c2sccc2Cl)=O)CN(C(=O)C=Cc2ccsc2)CCCO1 c1(CC(N2CCN(C(c3cnccn3)=O)C3CC23)=O)cc(Cl)c(F)c(Cl)c1 c1(CC(=O)NCC2CCC(NC(c3c(C)noc3)=O)C2)cccc2c1CCC2 Cn1nccc1CCC(=O)NC1CCC1.C12(CCCC1)C(=O)N1CCC(C1)OC2 CCC(C(=O)Nc1cc(C(=O)CC2(C)COCC(C)(C)O2)cnc1OC)C(C)O C1(CNC(C(C2CC2)OC)=O)CCC(C)(C)CN1C(c1sccc1C#N)=O C1(CNC(C2N(C)S(=O)(=O)CC2)=O)CN(C(C2CC(O)C2)=O)C2(CCOCC2)C1 CCC(C(=O)NC1CC2CC(C1)N(Cc1nc(C(C)(C)C)no1)C2)C(C)(C)CC N1(C(c2n(C(C)C)cnc2)=O)CC2CC2(CNC(c2nccnc2C(N)=O)=O)C1 N1(C(c2ccc(=O)oc2)=O)CC2ON=C(CC(=O)NC34CC(C3)C4)C2C1 C12(C(N3CC(CNC(CCCOC(C)=O)=O)OCC3)=O)CCC(=O)N1CCS2 c1(OC)cc(CNC(=O)C=CCN(C)C(C2CCC(F)CC2)=O)n(C)n1 C12(NC(C(=O)NCC)=O)CC(CNC(c3ccc(SC)s3)=O)(C1)OC2C c1(OC)cc(C)nc(N2CCC(CN)(CO)C2)n1 CC(C)(C(=O)NC(CNC(C1CCO1)=O)C1CCC1)N1CCCC1 c1(OC)ccc(Cl)c(C(=O)N(CC(O)CN(C)C(C2COC(C)C2)=O)C)n1 c1(C(=O)NC2CCC(=O)N(CC(=O)O)C2=O)cccc2c1C(=O)NC2 C1(C2CCOCC2)(C(N2CCCCC(CNC(c3ccco3)=O)C2)=O)CC1 c1(CC(=O)NCC(C(=O)NCC(N2CCCCC2)C2CCC2)O)ccccc1Cl C1(NC(=O)COCCCF)CCN(C(=O)C(c2cccnc2)O)CC1O c1(NC2CN(CC(N)=O)C2)nccc(N2CCCC(C(=O)N(C)C)C2)n1 CC1CCCn2cc(C(=O)NCC3CC4CCC3N4C(c3sccc3Cl)=O)nc21 c1(C(=O)NCCN(C(c2cc(C(C)C)no2)=O)CC)cncn1C Cc1ccc(Cl)cc1CN(C)CCN(C(=O)Cn1cc(CC(C)(C)C)nn1)C c1(C(=O)NCCN(C(C2(OC)CS(=O)(=O)C2)=O)C)ccc2[nH]c(=O)c(=O)[nH]c2c1 c1(C(=O)OCC)cncnc1C(=O)OC1CCCN(C(=O)CC)C1 N1(C(C(CCC)C#N)=O)CC2(C(=O)NC(C)(C)CF)CC1CCO2 c1(CC)nc(C)n(C)c1C(=O)N(C(C)CNC(C1CCCO1)=O)CC C12(NC(CC(C)SC)=O)CC(CNC(c3ccc4occc4n3)=O)(C1)OC2(C)C Cn1ccc(-n2cnc(C(=O)NCC(C)(C)NC(=O)CC3CNC(=O)C3)c2)n1 CCCCC(Cc1nc(-c2ccc(N)cc2)nn1C1CCCC1C1CC1)CO N1(C(Cc2c(C)n[nH]c2C)=O)CC2OCCN(C(c3cccc(Br)c3O)=O)C2C1 C(CC1CC1)(C(=O)NCC(F)Br)NC(C(C)OC(C)(C)C)=O N1(C(c2c[nH]nc2C(F)F)=O)CCC(C(=O)N(C2(C3CCCCO3)CC2)CO)CC1 c1(C(=O)NC23CC(NC(C=CCC)=O)C(OC2)C3)cnc2nc(C)[nH]n2c1=O C1(NC(CCC(C)C)=O)CC2CN(C(=O)C(=O)Cc3ccc(Cl)cc3)CC12 CCCC(C)(O)CC(=O)NC(C1(C)CCN(C(=O)CCOC(C)C)C1)(C)C C1(CNC(c2ccc(CC)s2)=O)CC(OC)CN1C(=O)Cn1cnc(C(F)(F)F)c1 C(C(C)(C)C(=O)NCCN(C(c1ccc(Cn2ccnn2)cc1)=O)C1CC1)SC c1(CC)ncc(NC(=O)CNC(C2CCN(C(=O)NC(C)(C)C)C2)=O)c(C)n1 c1(C(=O)NC(C(C(C)C)C)CNC(c2n[nH]cc2Br)=O)c(F)ccc2c1OCC2 N1(C(CC2(N(C)C)COC2)=O)CC2(C1)SCCC2NC(C1CC2CCC2C1)=O CC12CN(C(=O)NCC3C4CC5COC3C5C4)CC1C1C=CC2C1 C1(NC(C2CCC3(CCC3)C2)=O)CCCC12CN(C(c1cnn[nH]1)=O)C2 Cc1cc(=NCc2cc(C)[nH]n2)[nH]c(NC2CCc3cc(Br)ccc32)n1 C1(CC(=O)NC(CCC)C)CCCCN1C(c1cnccc1Cl)=O C(=O)(C(O)C(C)CC)NC1(C2N(C(COCCCC)=O)CCC2)CC1 Cn1ccn2cc(C(=O)NC3CCC3NC(=O)CC3(C)CC3(Cl)Cl)nc2c1=O c1(C(=O)NCCCN(C(C(C)CC(N)=O)=O)C2CC2)cccc2oc(=N)[nH]c12 CC(C)(F)CCC(=O)NC(C)(CNC(=O)CN1CCC(O)CC1)CO Cn1cccc(C(=O)NC2CCC2CNC(=O)Cn2nccn2)c1=O C1(NC(C2C(OCC)C2)=O)(CF)CN(C(=O)CC2CCC2)C1 N1(C(C(c2cc(C)oc2C)C)=O)CC2(CC(NC(=O)Cc3cc(C)n(C)n3)C2)C1 c1(-c2cn(CC=C)nn2)ccc(N(C)C(c2coc(-c3ccccn3)n2)=O)cc1 C(CCCl)(CCCl)(c1n(C(C)(C)C)nnn1)NCC1(CC2CC2)CCOC1 c1(OC)cccc(C(=O)NCC2CCC(NC(c3c[nH]c(Br)c3)=O)C2)c1 N1(C(C=NOC)=O)CC2(CC(NC(=O)CCSc3cc(C)cc(C)c3)CO2)C1 c1(OC)ccc(C(N2CCOC(C(=O)Nc3ncc(F)cc3C)C2)=O)c(O)c1 CC(C)(C)C(C(=O)NC1CCCC1CNc1cccc(CO)c1)N1CCNC1=O C(=O)(CC(C(F)(F)F)NC(=O)CNC(c1c[nH][nH]c1=N)=O)NC(CC)(C)C c1(C(=O)NCC2OCCN(C(C(=C(C)C3CC3)F)=O)C2)ccc2ncccn12 C1(=CC(=O)NC(C2CCN(C(=O)CCN3CCCC3)C2)C)CCCCC1 C1(C(=O)NCC2CCN(C(c3c(CC)nn[nH]3)=O)C2)CCCOC1c1cc[nH]n1 c1(SCC(N2CC(C)(NC(C3CCN(CC)CC3)=O)C2)=O)nc2ccccc2s1 C1(CC)CN(C(c2ccc(C3CC3(F)F)cc2)=O)CCN1C(c1cnsn1)=O C(=O)(CC(C)COC)NCCCN(C(=O)C(C)C(F)F)CCC c1(COCCC(N2CCCC2C(N2CCC23CC3)=O)=O)cn2c(n1)CCC2 C1(C(=O)NCC2C(NC(C3(C)CC(=C)C3)=O)C2)CCCCN1C(=O)OC(C)(C)C c1(C(N2C(CNC(C(c3ccc(F)cc3)C)=O)C=CC2)=O)ccc(C#N)s1 C1(C(=O)OC)Cc2ccccc2N1C(=O)CNC(C1CC1c1ccccc1)C N1(C(C#CC2(CC)COC2)=O)CC2(C)CN(C(=O)CC(F)(F)C(F)F)CC2(C)C1 N1(N(C)C(C2CNCC2(C)C)=O)CCN(CC(N2CCOCC2)(C)C)CC1 N1(C(C)=O)CCOCC1C(=O)NCC(O)CN(C(=O)Cc1nnc(O)s1)C C1(C(N2C(CNC(c3nc(C)[nH]n3)=O)CC3CC32)=O)Cc2cncn2C(=O)N1 C12(CC(=O)NCC(C)N(C(=O)Cc3ccon3)C)CCCN1CCC2 c1(C(C(=O)NC)N(CC(C)(C)C#N)CC)sc(=O)n(C)c1Cl C(=O)(CC(C)(C)CCOC)N1C(C)CC(CNC(CNC(CC)=O)=O)C1 Cc1cccc(CC(=O)NCCN(C(c2cscc2C(F)F)=O)C(C)C)c1F C1(c2n(C)ncc2)CCCN(C(=O)NCC2(Cc3ccccc3)CC=CCC2)C1 CC12CCC1CN(CCC#N)C2.N12CC3(CCN3C(=O)c3cccc1n3)C2 C1(C)(C(N2CC(OC)(CNC(c3ccnnc3)=O)C2)=O)CC(C)OC(C)C1 Cc1cn2[nH]c(=NC3C4CN(C(C5CC(C)CC(C)(C)C5)=O)CC34)sc2n1 C1(NC(Cc2ncc(CC)[nH]2)=O)CCC2CN(C(=O)C(C)(C)CC)CC2C1 c1(CC(=O)N(CC(C)NC(Cn2c(C)ncc2)=O)C)cccc2c1OC(C)(C)C2 c1(OC)ccnc(C(=O)NCCN(C(c2ncccc2Br)=O)C2CC2)c1 c1(NC(C=Cc2occ(C)n2)=O)ccc(OCc2cccc(Cl)c2C)c(C)c1 CCCS(=O)(=O)C(C)C(=O)NC(C1CCCN1C(=O)Cc1ccoc1)C c1(C(=O)NC2CC2CNC(C2OCC3CCCC23)=O)cnc2nccnc2c1 N1(C(CC(C=C)CCC)=O)CCC2(CCCN2C(=O)COCC(=O)NC)C1 C(=O)(CC(C(F)(F)F)n1cccn1)Nc1c(OCCN(C(C)C)C)cccc1 Cc1ccc(CCNC(=O)CN2CCCN(CC(C)O)CC2)c(C)c1 C=CCCC(F)(F)C(=O)N1CC(C(F)(F)F)C(CNC(C2(C)CCC(=O)N2)=O)C1 C1(OC(C2(CF)CCOCC2)=O)CCC(OC(F)F)CC1 c1(N(C(=O)C(O)Cn2cncn2)CC2CC2)cccc2cccnc12 C12(C(N(CC(C)NC(CC3(C=C)CC3)=O)C)=O)CCC(=O)N1c1ccccc1S2 N1(C(CCC=C=C)=O)CC(C)C(C)(CNC(=O)COC(F)F)C1 C#Cc1ccc(C(=O)NC2CCC(NC(=O)C(F)C3CCCC3)C2)c(F)c1 N1(C(c2c(F)cc(Br)cc2F)=O)CCCC12CCN(C(C1CC1(F)F)=O)C2 c1(C(N2CCC(O)(C(C)NC(c3cnsn3)=O)CC2)=O)cnc2ccccc2c1 CC1(c2nn[nH]n2)CCN(C(=O)CCCn2cncn2)C1 n1(CC)ccc(C(=O)NC2CN(C(=O)C3=CCCC3C)CC2(C)C)cc1=O c1(CC2C(C(=O)NC(CNC(=O)C(C)n3cccn3)C3CCC3)C2)ccccc1 C(=O)(C(F)(F)C(F)(F)C(F)F)N1CC(O)(C(C)NC(c2cc(Cl)ncc2O)=O)C1 C=C1CC2(C1)CN(C(=O)C(c1ccoc1)NC(=O)CC1CNC(=O)O1)C2 CC(O)CC(C(=O)O)NC(c1ncoc1C(=O)OC(C)(C)C)=O c1(C(=O)NC(C)CN(C)C(C2CN(S(C)(=O)=O)C2)=O)cccc(C(=O)N(C)C)c1 c1(C(N2CC(C)(C(N3C(CC)CCC3)=O)C2)=O)cnnc(C)c1C c1(OC)c(C(c2nnnn2C2CCC2)NCC2(C)CCOC2C2CC2)c(C)nn1C n1(CC)cc(Cl)cc1C(=O)N(CCCNC(=O)Cc1nnc(C)o1)C(C)C C(=O)(CCCCCc1cccs1)NC(C1(O)CN(C(Cc2c(C)ocn2)=O)C1)C N1(C(Cc2c(C)cnn2C)=O)CCN(C(=O)C(N2CCOCC2)C)CC(C)(C)C1 N1(C(C(C(C)C)SC)=O)CC2OCCN(C(c3ccc(CC(C)C)s3)=O)C2C1 C1(CNC(C(=O)NCc2nc(C)c(C)n2C)=O)Cc2ccccc2C1(C)C Cc1cnc(C(=O)NCC2CCN(C(=O)Cc3ncccc3C)CC2C)c(C)c1 C(=O)(CC(C)C(=O)N1CC(=O)NCC1C(=O)NCC1CCCO1)OC c1(NC(CC2CCCN(CC3CCC(C)(C)O3)C2)=O)cc(Br)cnc1O c1(CNC2C(CC(C)(C)C)C2)ccc(CNC(=O)C(C)(C)C)cc1 Cc1cccc(C(=O)NC2CCC(NC(=O)COCC3CCOC3)CC2)n1 Cc1ccc(C2=CCN(C)CC2)c(NC(c2ccc(Cl)cc2)C)c1 C1(F)(C(=O)NCC2CC(NC(c3c(CC)scn3)=O)C2)CS(=O)(=O)CC12CCC2 c1(OC)ccc2cc(C=CC(N3CC(NC(=O)C(C)C(F)(F)F)C3)=O)ccc2c1 N1(C(CN2CCC(C)(C)C2)=O)CC2(CC(C(=O)CC3CCOCC3)C2)C1 C1(C(=O)NC2CC(CC(=O)N(c3ncccc3CO)C)C2)CC2(CCCCO2)C1 N1(C(C(C)N(C(C2(OC)CCOC2)=O)C2CC2)=O)CC2CC(C)(C)C2C1 Cc1ncncc1C(=O)N(CCCNC(c1cn(Cc2cccs2)nn1)=O)C c1(OC)ccc(Cl)cc1C=CC(=O)NCCC(C)N(C(=O)C(C)C1CCCC1)C N1(C(c2cc(C)oc2)=O)CC(F)(F)CC1CCNC(=O)Cc1ccnn1C c1(CC)c[nH]c(C(=O)NC(CNC(C2CC(N(C)C)C2)=O)CO)n1 Cc1cc(C(=O)NCCN2CCN(C(=O)C=C3CC3)CC2)cn2c(C)cnc12 C1(CC(N2CCN(C(C(CC(=C)C)C)=O)CC2CC)=O)SC2=NCCN2C1=O N1(C(C2COCCN(C)C2)=O)CC(NC(=O)CC2COC(=O)C2)CC2(CCC2)C1 c1(C(=O)N(CC2C(NC(CC3CC(=C)C3)=O)CCC2)CC)cccn(C2CC2)c1=O c1(N(C(COC)=O)C(C2CS(=O)C2)=O)cc(C)cc(C)c1O.C12CC(C1)O2 c1(OCC(=O)NC)ccc(C(N2CC=CC2CNC(=O)CC2(C)OCCO2)=O)cc1 N1(C(c2[nH]cc(C(C(C)C)=O)c2)=O)CCCC(NC(=O)Cc2csc(C3CC3)n2)C1 C(CC(C)C(=O)NC(C(=O)N1CC(CCO)C1)C(C)C)OC C(C(C)C(=O)N1CCC(CN(C(=O)Cc2cnn(C)c2)C)C1)OC N1(C(c2cnc(C(C)(C)CF)o2)=O)CC2CC2(NC(C2COC(=O)C2)=O)C1 N1(C(CSC)=O)CCN(C(=O)Cc2cc(-c3ccccc3)ccn2)C(CF)C1 Cc1ccc2nc(CN3CCN(CC(c4nc[nH]n4)=O)CC3)[nH]c2c1C N1(C(C(C)NC(C)(C)C)=O)CCCCCC1CNC(c1cc(CCCO)on1)=O C1(CCNC(c2cnc(O)s2)=O)CN(C(=O)C(c2ccccn2)O)CCCO1 c1(CC)cc(C(N2CCC(CNC(=O)Cc3cccc(C)c3)CC2)=O)cc(O)n1 C1(NCc2cc(C)no2)CCC(C)N(C(C)C(=O)Nc2ccccc2C)C1 c1(CC2(C(=O)NCC3C(NC(=O)CN4CCNC4=O)C3)CC2)ccc(F)cc1 C1(CC#C)(C(=O)NCC(C)(C)NC(=O)CC2CC2(C)C)CCOCC1 c1(C(C)=O)cc2c3ccccc3n(C)c2s1.c12ccccc1OCC(O)CN2 N1(C(COCCC(C)C)=O)CC2CC2(CNC(=O)CC2CCNC2=O)C1 C(=O)(C1=CC2CCCCC12)N1CC(CNC(CC(C)(C)NC(C)=O)=O)N(C)CC1 c1(C(N(C2CCCN(C(c3n(CC#C)ccc3)=O)C2)CC)=O)c(C)cccc1N C1(C)(NC(C2CCC(C)O2)=O)CCN(C(c2cn(CCCF)nn2)=O)C1 C1(F)(CN)CCCN(C(c2cnc(C(C)C)s2)=O)C1.C=C1CC(CN)C1 CC(CCC(=O)NCC1(CO)CC=CC1)NC(c1cnccn1)=O CCCCCCOCC(=O)NCC(CC)N(C(=O)CC1CC1C(F)(F)F)CC N1(C(C(CCC)S(N)(=O)=O)=O)Cc2ccccc2C1CNC(C1CC(C)CO1)=O N1(C(c2nc(C)n(C)c2)=O)CCCC2(NC(C3CCOC3C)=O)CCCC12 C1(N(C(C(c2cccnc2)NC(C=CC=CC)=O)=O)C)CCC2CC12 Cc1nc(C)n(-c2ccc(C(N3CCCC3CNC3CCC(=O)NC3)=O)cc2)n1 C#CCC(O)C(=O)NC(CC)C(=O)NCC(=O)N(C)OC CCCC(CCCNC(C12CCCCC1C2)=O)NC(c1cncc(N)c1C)=O C(=O)(CCNC(C1(CCNC(=O)Cn2nccn2)CCC1)=O)OC C1(CC(=O)NCC2(NC(c3c(C)c[nH]c3)=O)CCC2)CC(O)C1(C)C c12nc(ccc1Br)NC2=O.C(=O)(C(F)(F)F)N1CCC1 N1(C(CNC(NCCOC(C)C)=S)=O)Cc2[nH]nc(Cc3ncon3)c2C1 N1(C(CSc2ccc(C)cc2)=O)CC23CCCC2(C1)CN(C(=O)CSC(=N)N)C3 N1(C(C(CSC)(C)C)=O)CC(CNC(c2cc(F)ncc2C)=O)C2(CCC2)C1 N1(C(COCC)=O)CC2CCN(C(c3ccc(OC)c(C)c3C)=O)C(C2)C1 Cc1ccccc1CC(N1CCC(CF)(NC(c2csc(F)c2)=O)C1)=O C(CC(=O)NCC1(F)CCN(C(c2cc(C)cc(Cl)c2)=O)C1)(C(C)C)OCC N1(C(C2CC(C(=O)OC)C2)=O)CCCC(C)(C(N2CCOC(C)(C3CC3)C2)=O)C1 CC1=C(C(=O)N(CCCNC(=O)C#CC(=O)N(C)C)CCO)SCCO1 CCC1=NOC(CC(=O)NCC2(CNC(=O)C(C)(C)CO)CCC2)C1 c1(C(C)(C)N(C(c2cn(CC3CCCN3)nn2)=O)C2CC2)cnc2[nH]ccc2c1 C1(F)(CNC(=O)CCc2cncs2)CN(C(c2cnn(-c3nccs3)c2)=O)C1 c1(N2C(C)CC(CNC(c3cnn(C)c3C3CC3)=O)C2)nc(Cl)nc2ccccc12 C1(NC(c2cc(F)cc3cc[nH]c23)=O)C2CC3CN(C(C4CCCO4)=O)C1C3C2 C(CC(=O)NCC1CCCCN1C(c1ccsc1Cl)=O)(C(N)=O)NC(C)=O Cn1ncc2c(NCCC3(O)CCN(C(C4CC5CCC5C4)=O)CC3)ncnc12 C1(C(=O)NC(C)CCCCNC(=O)CCP(C)(C)=O)COc2ccc(F)cc2C1 Cn1cc(I)c2c(N3CC4CC4(C(=O)NCCN4CCNC4=O)C3)ncnc12 c1(CCNC(=O)C(N2CCCC2CCO)=O)ccc2ccccc2c1 C1(C(=O)NCCCC(C)(C)NC(CCCOCCC)=O)CCCC(F)(F)C1 c1(N2CC(CNC(c3ccc(CCC)[nH]3)=O)C(C)(C)C2)c[n+]([O-])ccc1[N+](=O)[O-] c1(C(=O)NC(C2CCN(C(C3CCCCS3)=O)CC2)COC)cnc(OC)c(F)c1 O=c1cc(-c2ccccc2)ncn1C1CCN(CCc2ccccc2)C1 C(=O)(C1=Cc2ccccc2C1O)NCCCNC(c1c(N)cncc1)=O CC1CN(C(c2cccnc2Cl)=O)CCC2(CCOC2)O1 c1(C(=O)NC2C=CC(CNC(C(C)(C)c3cnco3)=O)C2)ncccc1F CC1CN(C(=O)CCF)CCC1N(C)C(c1cn(CC2(C)COC2)nn1)=O N1(C(CC2(OCC)CC2)=O)CC(C)CN(C(c2cc(C)sc2C)=O)C(C)C1 c1(CC(=O)N(CCC)CCNC(=O)C=CSc2ccccc2)cccc(Cl)c1F C=C1CC(C(=O)NCCC(C)N(C)C)(CNC(=O)C(C)N2CCCC2)C1 c1(CC(=O)NNC(=O)c2cccc(Cl)c2Cl)ccc2c(c1)C=CC2 N1(C(CCCC2C(C)C2)=O)CC2CC1C2CNC(=O)C(O)C1CC1 C1(NC(C(C2CN(C(c3cocc3C)=O)C2)OC)=O)CCC(F)CC1 C=CC(CCC)CC(=O)N1CC2C(NC(c3c[nH]c4nccc-4c3)=O)C2C1 Cc1c(Br)cnn1CC(=O)NCCCN(C(C1CCCSS1)=O)C(C)C CN1CCCC(C(N2CSCC2C(=O)NCc2cn[nH]c2)=O)C1 C(=O)(C#CC(C)(C)C)N1CC(CC)C(C(N2CCCC2CC(C)C)=O)C1 c1(CC)[nH]nc(C(=O)NC2CCC(C)N(C(=O)CCc3nncs3)C2)c1[N+](=O)[O-] S(=O)(=O)(c1ccc2cc(Br)ccc2c1)NC(C1(CC=C)CCNCC1)=O C12(C(=O)NC(C3CCN(C(C(c4cncnc4)C)=O)C3)(C)C)CCCCC1C2 N1(C(CC2CN(C)C2)=O)CC2CCN(C(C3(N4CCOCC4)CC3)=O)CC2C1 N1(C(c2c(C)ncs2)=O)CC2CCCC(NC(=O)CC(C)n3ccnc3)C2C1 Cc1cccc2c(N3CC4C(CO)C4C3)ncnc12.N12C3CCC1CN(C3)C2=O C1(COC)CN(C(c2nc(=O)n(C)[nH]2)=O)CCN1C(=O)C(O)Cc1cnc[nH]1 N1(C(c2n(C)nc(CC)c2Cl)=O)CC(C)N(C(c2oc(Br)cc2C)=O)CC1C C1(CNC(CCOCCN(C)C)=O)CN(C(c2cn(C3CC3)cn2)=O)CC1C Cc1cc([N+](=O)[O-])ccc1C(=O)Nc1cccc(N2C(=O)CCC2=O)c1 C(CC(C(C)(C)C)NC(=O)CC1(O)CCCCCC1)N(C(C1(CC#C)CC1)=O)C C(C(CC(C)C)C(=O)NC1CC(C)(CC(=O)NCCSC)C1)OC C(=O)(C(F)(F)C(C)(C)O)N1CCC(C(CNC(c2ncc(C)c(Cl)c2)=O)O)CC1 c1(CCC(=O)NC2CCC(CNC(C3(CCCC)CC3)=O)C2)ccncc1Br N#CC1CCN(C(=O)CCC2CCCN2Cc2cnc(O)c(Cl)c2)CC1 N1(c2cc(C)ncn2)CCN(C(C2(c3cnccn3)CC2)=O)CC1CC#N C(=O)(C#CC1CCCO1)NCc1ccc(C(N2CCC2Cn2ccccc2=O)=O)o1 c12ccc(cc1)C(NC(C1CC13CCCC3)=O)C(=O)N2.N1(CC)CCOCC1 C12(C(=O)NCC3CCN(C(CC=C(C)C)=O)C3(C)C)CC3CC(C1)CC(F)(C3)C2 C1(CC#C)(C(=O)N(C)CC2CCCN2C(c2cc(Cl)cs2)=O)CCCOC1 c1(C(C)C)nccc(=NC2CC(CNC(c3ccc(OCCO)cc3)=O)C2)[nH]1 C1(C(=O)NC2(COCC)CC2)CN(C(=O)Cn2nccn2)C(C2CCC2)(CC)C1 Cc1ccc(NC(C2C=CCN(C(=O)CC3CC4C=CC3C4)C2)=O)c(C)c1O N1(C(CCCC#C)=O)CCC2(CC1)CC2NC(=O)CC12COC(C)(C1)C2 CC(CC(N)=O)C(=O)N1CCC(C)(C(=O)NC2(CO)CC2)C1 N#Cc1cccc(CC(=O)NCC=CC(=O)NCc2ccc(O)nn2)c1 N1(C(COCCOC)=O)CCCC2(C1)C(NC(c1cccc(C)n1)=O)CCN2C N1(C(C2CC(=C)C2)=O)CCC2(CC1)CC(C)N(C(=O)COCC1CCC1)C2 c1(C(=O)OC(C)(C)C)nnc(O)cc1O.C12COCCN1C2 CC1(C)CC(CC(=O)NCC2(C(N)=O)CCCC2)CN1C(=O)C(F)C(F)(F)F N1(C(C2(C#C)CN(C(=O)CCc3ccc[nH]3)C2)=O)CC2(CCC2)OCC1C c1(NC(c2c(OC)cccc2)c2nnnn2CC2CCCO2)ccc(O)cc1OC c12cc(nc(C)c1)S2.c1(C(CC)=O)cccc(Nc2ccc(C(N)=O)cn2)c1 CC(CC(F)F)C(=O)N1CC2CC(NC(=O)CCN3CCCC3=O)C1C2 c1(CN2CCC(C(=O)NC(C(C)C)CCO)C(O)C2)ccc([N+](=O)[O-])c(O)c1 C1(CNC(C2(OC)CCC2)=O)CN(C(c2nc(C)ncc2Cl)=O)CCC1C c1(CCC(C)C)nc(-c2cccc(N3CC=CC3)c2)n(CC(F)(F)F)n1 N1(C(CCn2ncc(C)c2)=O)CCC(C)(C)C(NC(=O)C=CC(F)(F)F)C1 C1(NC(c2cc(C)c(C)nn2)=O)CCN(C(C2COCCN2C(C)C)=O)CC(O)C1 C(CCCCC(=O)NC(CO)C(N)=O)N(C(c1cc(CC)[nH]n1)=O)C C(=O)(CC1=CCN(C)CC1)NC1CCC(NC(c2c(C)cc(Br)cc2)=O)CC1 c1(NC(c2cncc(OC)c2)C2CC2)ccc(O)c(Br)c1 N1(C(c2cccc(Cn3cc(C(C)(C)OC)nn3)c2)=O)CCCN(C=O)CC1 N1(C(C2CCCC(C(=O)OC)C2)=O)CCOC2(C1)CN(C(=O)C(O)C(F)(F)F)C2 CCCCCCC(C)(C)C(=O)N1CC(NC(=O)CSCCOC)C(C(F)(F)F)C1 c1(C(=O)OC)sccc1S(=O)(=O)N1CCC(Nc2ncc(C)s2)C(O)C1 Cc1ccc(C(C)C(=O)NCCCN(C(=O)Cc2[nH]cnc2C)C(C)C)cc1 N1(C(C=CCC)=O)CC2CC1CC2CNC(=O)C(F)(F)c1csc(C)c1 C1(NC(C(C2CC2)SC)=O)CCCCC1NC(C1CCC(C)CC1)=O C(C(=O)NOCCCC(=CC(C)(C)C)C)N(CC#C)C(=O)CC1CCOC1 Cn1cc(C(=O)NCC(C2CC2)NC(C2CCCCC2)=O)cc1Br N1(C(c2c(Br)cc(C)s2)=O)CCCC2(C1)CN(C(C1C=CCCC1)=O)C2 c1(C(=O)NC(C#C)(C)C)c[nH]nc1CCNC(C1CC(=C2CCC2)C1)=O N1(C(c2cnc(C)nc2)=O)CC2CCN(C(C34CC(CO)(C3)C4)=O)CC2C1 CCCCCCC(F)C(=O)NC1CC(O)(CNC(=O)Cc2c(C)n[nH]c2C)C1 c1(NC(CSCC)=O)cc(C)c2c(c1)CCCN2.N12CCN(CC1)C(C)(C)C2 CS(=O)CCCCNC1CCC(NS(C)(=O)=O)CC1 c1(C(=O)NCC(CC)NC(=O)CCOc2cccc(C)c2)ccnc(OC)n1 C1(C(=O)NCCN(c2csc(C3CC3)n2)C(c2ccc(O)nc2)=O)CCCCCC1 C1(C(=O)NC(c2cccc(O)c2)C)CC2CCC1N2C(=O)C1CC1CCCO c1(OC)ccccc1C(C)N(C)C(C1(c2ccc(Br)s2)CC1)=O Cc1ccc(Cl)c(N)c1C(N1CCCC(NC(=O)COCCC(C)C)CC1)=O C1(C(=O)NCC(C#C)C(C)C)CCC(O)CN1C(c1cnc(NC)cn1)=O CC1=C(C(=O)N2CCC(CO)(NC(C3C4(CC4)C34CC4)=O)C2)CCS1(=O)=O N(C(=NCCN1C(=O)NCCC1=O)NC(C1CC1)C1CC1)C(c1ccsc1)C.C1(C(C2CC2)CC)CC1.CC1CC1.N C(=O)(C(C)(C)CCOC)N(CCN(C(c1c(CC)nns1)=O)C)C C1(NC(CSCCC)=O)CN(C(=O)CC2(n3cccn3)CCOCC2)CCC1C N1(C(C(CC)NC(C2(CO)CCCO2)=O)=O)CCC(CC(C)C)CC1 c1(OC)cc(C(N2CCC(C(=O)NC(c3ccccn3)C)C2)=O)ccc1Br N(C)(C(=NCC(O)C(C)(F)F)NCC)C(C)C.C(C(F)F)NC C1(C(=O)NCC2(OC)CCOC2)CN(C(c2csc(C)c2)=O)CC1C1CC1 N1(C(c2cncc(C)c2)=O)CCC(C)(NC(=O)CCC2CCC(=O)N2)CC1 C1(C(N2CC(CC(C)NC(=O)Cc3ccnc(O)c3)C2)=O)CCCS1(=O)=O N1(C(c2cc(OC)nn2C)=O)CCC2C(C1)CN2C(c1ccoc1Br)=O C1(CC#C)(OC(C2CCCCN2Cc2cccc(C)c2)=O)CCN(C(C)=O)C1 N1(C(C(CC)C)=O)CCC(F)(CNC(C2CCCNCC2)=O)CC1 C1(NC(c2c(COC)noc2)=O)CC(C)CN(C(c2sccc2SC)=O)C1 C(=O)(CCCCCN(C(=O)COC(C)(C)CNC1CC(C)OC1=O)C)OC N1(C(C(Cc2cn(C)nc2)O)=O)CC=C(C(=O)NCCn2ccnn2)C1 N1(C(c2c(C)noc2C(F)(F)F)=O)CC(NC(=O)C=CC2CC2)CC(C)(C)C1 c1(C(=O)NCC2CN(C(c3nn(C)c(O)c3)=O)CC2O)cc2c(s1)CCC2 N1(C(c2cc(C)c(C)[nH]2)=O)CC2CC1CN(C(C1CCC(C)NC1=O)=O)C2 c1ccc(C(=O)NC(C)C(=O)N2CCCC2)o1.N1(NC(C(C)C)=O)CCC(CS)C1 c1(C(=O)NC2CCC(NC(C3CCS(=O)(=O)C3)=O)CC2)nccc2occc12 C(=O)(C(C#N)C(C)C)N(CC(=O)NCC=C(C)C)CC(C)C CC1CC(CNC(=O)Cn2ccccc2=O)CN1C(=O)C[SH](CCC#N)CCF c1(CNS(CC2CCC(COC)O2)(=O)=O)ccc2cc(OC)c(F)cc2n1 Cc1ccc(Br)c(CS(=O)CC(=O)NCC2CCCSC2)c1 c1(C(C(=O)O)NC(C(=O)NCC2CC2c2ccco2)=O)ccc(F)c(Br)c1 C(c1ccccc1C)=CC(=O)NCC(C)N(C(c1c(CC)nns1)=O)CC Cc1cccc2cc(C(=O)NCCCCN(C(=O)CCC(C)(C)F)C)[nH]c12 c1(C(C(=O)NCC=C(CC)C)(C)C)ccc(CNC(=O)C(C)SC)cc1 N1(C(C(C)SCCCC)=O)CCSCC1CCNC(C1(CO)CC(F)(F)C1)=O C(=O)(C(C)NN(C)C(C1CCC1C(=O)OC)=O)NC c1(C(N2CCN(C(C=C(C)C)=O)C(C)C2)=O)ccc2c(c1)CCO2 C1(C(N(CCCN2CCCC2)C)=O)COC2(C1)CN(C(c1cnnn1C1CC1)=O)C2 N1(C(CCC(C)NC(c2c(C)cc(CC)o2)=O)=O)CCC(C)CC1C c1(C(=O)NCC(CNC(C2=CCCC2C)=O)O)ccc(N)c([N+](=O)[O-])c1 N1(C(C2CCCCC2(C)C)C(=O)NCC(C)C)CCNC(=O)CC1(C)C C(=O)(C(CC(F)(F)F)C1CC1)NC(C1(F)CCN(C)CC1)=O.c12ccc(cc1)CC2 O=C(CCC(=O)N1CC(CC(F)C(=O)N2CC(c3nocc3Cl)C2)C1)C1CC1 C=CCC(C)(C(=O)N1CCC(CNC(=O)C(O)C(C)(C)C)CC1)N(C)C c1(CCN(C(C(=O)NC)C2CC2(Br)Br)C2CC2)c(C)[nH]c2c(C)cccc12 C1(F)(C(=O)OCCCSCC)CCCN(C(=O)CCCN(C)C(C)=O)C1 c1(C(=O)NC(C(=O)NCC(CCC)O)c2ccoc2)nccc2[nH]ccc12 N1(C(C(C)S(C)(=O)=O)=O)CCC2CN(C(C3CC3C3(C)COC3)=O)C2C1 C1(CNC(COCCCCOCC#C)=O)CN(C(C2COC(C)C2)=O)C(C)(C)C1 N1(C(CC2CC(NC(C3N(C)CCC3)=O)C2)=O)Cc2ncccc2C1 CC(C(C)(C)NC(=O)CNC(c1cnc(O)o1)=O)NC(=O)CNc1ccccc1 Cc1c(C(NC2COc3ccc(F)cc32)=O)oc(=O)c2ccccc12 c1(C(N(C2CCN(C(c3c(C(C)C)occ3)=O)C2)C)=O)cc2ccc(Cl)cc2o1 Cn1nc([N+](=O)[O-])cc1C(N1CCN(C(C2C=CCCC2)=O)CC1C(C)(C)C)=O n1(CC(=O)NC(CNC(C2(OC)CCSCC2)=O)CC(C)C)ccc([N+](=O)[O-])n1 N1(CC)CCN(C(=O)CC2C3CCC(C3)N2C(=O)Cn2cc(C)cn2)CC1=O CN1CCCCC1CCC(=O)NCCOC1CCN(C(=O)CCN2CCC2)CC1 N1(C(c2c(C)onc2)=O)CC(C)CN(C(C23CC4CC2C3C4(F)F)=O)C(C)C1 CCCCCC(C)(C)C(=O)NC1CCCC1CNC(c1ccc(N(C)C)cc1)=O N1(C(c2ccc(C3CC3)cc2)=O)CC2CCCC2(C(=O)NCC2(CO)COC2)C1 N1(C(CC)=O)CCCC(C(C)(C)CNC(C(C)CCC=C(C)C=C)=O)C1 N1(C(c2nc(OC)oc2)=O)CCC(CNC(c2cnn(C3CC3)c2C)=O)C1(C)C Cc1cc(C(N2CCCC2(C)CNC(=O)C2=CCCCO2)=O)cc2ccoc12 N1(C(c2nn(C)c(C(F)F)c2)=O)CC2(CCCCN2C(C2CCC(O)C2)=O)C1 C1(C(=O)NCCC2N(C(COCCN(C)C)=O)CCC2)CS(=O)(=O)CC(=O)N1 C=CCCCC(=O)N1CC2CC1(CNC(=O)CN1CCC(C)(C)C1)C2 c1(C(N2C(C(C)C)C(C(=O)NCC3CCCC3)CC2)=O)cc(F)cnc1O c1(C(N(C(CCNC(C2C(C(N(CC#C)C)=O)C2)=O)C)C)=O)ccc(N)c(N)n1 CC1CN(C(=O)CNC(c2ccoc2)=O)CC1NC(=O)C(CO)N(C)C C(=O)(C1=NNC(C(F)(F)F)C1)N1CC(C)C(Nc2nccc(CC#N)n2)C1 C1(COC)(CNC(C23COCC2C3)=O)CCCN1C(C1CC12CCC2)=O c1(C(=O)NCC2(NC(c3snc(O)c3Cl)=O)CC2)csc2ncnc(O)c12 C(CC1=CCN(C(C2CC3(C2)CC(O)C3)=O)CC1)NC(c1ccc(C#C)cn1)=O c1(C(=O)NCc2ccnc(Cl)c2F)ccc2c(c1)CN(Cc1cc(I)c[nH]1)CC2 C(CC(C(=O)NCCc1cocn1)NC(=O)CCc1nc[nH]n1)OCC CC1CC2CCN2C(=O)C1=O.c1(CC(=O)OC(C)(C)C)cnn(C)n1.C(C)(C)(C)O C1(O)(C(C)NC(CC2(OC)CCC2)=O)CN(C(C2(C3CCCO3)CC2)=O)C1 N1(C(c2c(OCC)ccs2)=O)CCC(Nc2ccc(I)cc2C(F)(F)F)C(F)C1 c1(C(=O)OC)cccc(C(N2CCOC(CNC(C3CN(C)CCO3)=O)C2)=O)n1 C1(C(C)(C)C)C(=O)N2CCC(OCCC=C)(C2)C(=O)N1.C(C)(C)(C)OC(C)=O c1(Cn2cc(CN(C(=O)COCCc3cccc(F)c3)C)nn2)cccc(Cl)c1 N1(c2nnc(-c3cn(C)nn3)n2C)CCC2CNC(=O)C2C1 c1(C(C(=O)NCC(C)CNC(c2cccc(F)c2)=O)SC)cccc(Cl)c1 C1(C(=O)NCC(C2CCC2)OC)CCOCCN1C(=O)CSC(F)F N1(C(C(CC(=C)C)NC(c2cnncc2OC)=O)=O)CCN(CC)C(C)(C)C1 N1(C(CC(CCC)NC(=O)C(O)CC2CCCC2)=O)CCC2(CCCO2)CC1 C(CC(CC)C(=O)N(C)CC1(O)CCN(C(c2nc(=O)cc(C)[nH]2)=O)C1)=CC n1(-c2cc(C)on2)c(C)cc(C(=O)N(c2cccc(Cl)c2)CCS(C)(=O)=O)c1C Cc1c(C(=O)NC(CNC(c2ncc(Cl)cc2F)=O)C(C)C(C)C)cncc1Cl N1(C(C(C(C)(C)C)SC)=O)CC(C)(CNC(=O)Cc2cccc(F)c2)CC1(C)C c1(CN(C(c2ccccn2)=O)CCO)cc2cnn(CO)c2nc1Cl.C1(CO)CC1 CN=c1nc(N(C)Cc2ncn(C)n2)[nH]c(=NCC2CCC(F)(F)C2)[nH]1 C1(C(N2CCC(NC(CCOCCOCC)=O)C2)=O)CCC(CCCCC)CC1 N1(C(c2nc(C)[nH]n2)=O)CC(C)N(C(=O)Cn2cccc(O)c2=O)CC1C N1(C(C(C=C)O)=O)CCCC(C(=O)NCC2(SCC)CC2)C1C C1(CNC(Cc2c(C)cccc2)=O)CN(C(=O)C2CC2)CC1(F)F.C12CN(C1)C2=O C1(NC(C(CC)SC)=O)C2CC3C(C2)C13C(=O)NC(CC1CCCC1)CO C1(C(=O)NCCN(C(c2n[nH]cc2C)=O)CC)CC2CCCC(C1)C2=O Cn1ccc(C(N2CCSCC2C(=O)NCCN2CC3CC3C2)=O)cc1=O c1(CNC(c2ccc(Oc3ccc(F)cc3)cc2)CC)cc(I)cc(I)c1Br c1(N2CCC(CC(N)=O)C2)nc(=NC)nc(N2CCC(OCCO)C2)[nH]1.CCC C1(C(=O)NC(C2CCCC2)C#C)CCN(C(=O)CC2CCCC3CC23)O1 C(=O)(CCN(CC(C)C)N1CCCC1C(=O)OC)Nc1ccc(C)cc1 c1(C(N2C(CNC(C3CCC(C(=O)OC)C3)=O)CC2)=O)cc(C(N)=O)cc(F)c1 CC1CN(C(c2sccc2CO)=O)CC1(C)CNC(c1cnccn1)=O CCN=C(NCc1cccc(CCN(C)C)c1)N1CC2CCCCC12 N1(C(CCC(=O)NC)=O)CCC2(CCN(C(=O)CSc3nncs3)C2)C1 CC1OC2(C(C(=O)OCCC3CCOC3)(C)C)CC1(C(=O)OC)C2 C1(NC(C(C)=C(CC)C)=O)CN(C(c2ccc(CC)cc2)=O)CC1OC C12(C(=O)NCC3(CCNC(C4CCCCO4)=O)CCCO3)CCC(CO)(CC1)C2 C1(OC)CC(NC(c2cnc(O)n2C)=O)CN(C(=O)CC2(N(C)C)CCCC2)C1 Cc1cccc(C)c1C1(C(N2CCN(C)C(CNC(=O)COC(F)F)C2)=O)CC1 c1(CNc2ccc(NC(CC)=O)cc2)cnn2cccc(Cl)c12 CCC(CC)C(C)C(=O)N1CCN(C(=O)C(C)Cc2ccccc2Cl)C(C)C1 CCC(CNC(c1nnsc1C)=O)(CC)NC(C1CC1c1ccc(F)nc1)=O C(c1ccc(C)c(C)c1)=CC(N1CCC(CC)(NC(=O)C(F)=C2CCC2)CC1)=O c1(COc2ccc(C)c(Cl)c2)ccc(O)c(F)c1F c1(OCCC(=O)NC2CCCN(C(C3CCCCS3)=O)CC2)ccc(Cl)c(F)c1 C=C(C)CC(C(=O)N1CCN(C(c2ccc(C(=O)OC)cn2)=O)C(C2CC2)C1)OC c1(OC)cc(Cl)c(NC(=O)C(n2ccc(C)n2)C)c(Br)c1 CN1CC(C(=O)NC2COCC2NC(C2(C(C)(F)F)CC2)=O)CC1=O C=CC(CC)CC(=O)N(C)CC1CCCN(C(=O)COCC(=O)OC(C)(C)C)C1 N1(C(CN(C(=O)COCCOC)CC#C)=O)CCC(C(C)(C)O)C1 N1(C(CCC2CCC(NC(c3cc(C)nc(O)c3)=O)C2)=O)CC(O)C2(CCCC2)C1 S(=O)(=O)(c1ccc(Cl)cc1)NCC(N1CCCC(NC(=O)C(F)CC2CC2)C1)=O Cc1cc(C(N2CC(N3CCN(C(c4cc(C#N)cs4)=O)CC3)C2)=O)cnc1O C1(CC)CC(C(=O)OC)CN1C(C(=O)OC)C1CC(CNC2CC2)C1 C1(OC)CC(CO)(NC(=O)C)C1.c1(C(C(=O)NCCC(C)SC)C)ccn(C)c1 C1(C(N2CC(O)(C(N)=O)C2)=O)C(C2CC2)CCN1C(=O)Cc1cn[nH]c1 c1(OC)cc(NC(C23CC(CN2C(=O)C(C#N)C(C)C)C3)=O)ccc1F C(=O)(C(O)C(O)C(=O)NNC(=O)OC(C)(C)C)NCC(=O)Nc1c(F)ccc(C)c1 c1(N2CCN(C(c3cc(-c4ccccc4)no3)C3CC3)CC2)ccc2nncn2n1 c1(C(=O)NC(CNC(C(CC)Cc2cccc(C)c2)=O)C)cnn2c1NCCC2 Cc1cc2cccc(-c3ccc(NC(c4cccc5[nH]ncc45)=O)cc3F)c2[nH]1 C1(NC(C2N(CC)CCC2)=O)CCN(C(c2cnn3ccn(C)c23)=O)C12CCC2 N1(C(C2(OCC)CCC2)=O)CC(NC(c2cc(C)n(C)c2C)=O)C2(CCC2)C1 C1(N(C(C(CC#C)O)=O)C)CCCN(C(c2nc(C)sc2C)=O)CC1 C1(CNC(c2cnc(S)[nH]2)=O)CC2(CCN(C(=O)CC=C(Cl)Cl)C2)CO1 C(=O)(C1=NOC2COCC12)N1CCC(NC(C2C(CC)OCC2)=O)C(C)C1 Cc1cc(F)cnc1C(=O)NC(C(N1CC(CO)C(O)C1)=O)c1ccco1 CC(C)(O)CC(=O)NCc1c[nH]nc1C1CCN(C(=O)C=CC2CC2)C1 N1(CC)CC(COC)Oc2ccccc21.c12cccc(c1C)C(=O)N2C C1(NC(c2cc3nc[nH]c3cc2F)=O)CCC2(CCCN(C(=O)C=CCF)C2)C1 c1(C(N2CC(N(C(c3cccc(OC(F)(F)F)c3)C)C)C2)=O)ccnc(C2CC2)c1 c1(OC)cnccc1CNC1CCCC1c1ccccc1 CCC(C)C(O)C(=O)NC1COCCN(C(=O)Cc2csc(-c3ccoc3)n2)C1 C12(NC(C=C(COC)C)=O)CCC(C1)N(C(c1cc(C(C)(C)C)oc1C)=O)C2 C1(C2CC2)CC(=O)N1.C(c1ccsc1)=CC(=O)NC1CC(NC(C)=O)C1 CC1(C)CC(CNC(C2CC(C)(C)C2)=O)N(C(c2cccn2C2CC2)=O)C1 c1(C(=O)NC2(CNC(C(CC=C)C)=O)CCCC2)ccc(OC)cc1C C1(C(C)NC(=O)C(n2cc(Cl)cn2)C)CCN(C(C2CC2(C)C(F)(F)F)=O)CC1 n1(CCC)ccc(C(=O)NCCn2cc(C(=O)N(CCS(C)(=O)=O)C)nn2)n1 C(CC1CCCN1)(N=c1nc(COC)[nH]s1)c1c(CC)cccc1 C=CCCCCCC(=O)NCC1OCCC1C(=O)N(C)CCC1CCCC1 Cc1ncnc(C)c1CC(=O)N(C(CNC(C1CCCC1C1CC1)=O)C1CC1)C c1(C(N2CCC(CNC(C(C(C)C)n3cc(C)nc3)=O)C2)=O)occ2c1CCC2 c1(C(=O)NC(CC=C)CNC(=O)C(C2CCCC2)SC)cn(C)nc1OC c1(C(N2CCC(C(C)NC(c3cnn(C)c3C(F)F)=O)C2)=O)ccc(N)c(F)n1 C1(C)(CN(C)C)CCN(C(C2COCCC2NC(=O)C(O)C2CCCC2)=O)C1 C1(NC(=O)Cn2nnc(=O)[nH]2)COC2CN(C(=O)C=C3CCOCC3)CC12 N1(C(c2scc(C)c2C)=O)CC2CCN(C(C3C(C)(C)C3(F)F)=O)C2C1C CN(Cc1cccc(Cl)c1Cl)N1CC(F)(F)C(F)(F)C1 C1(OC)COCCC1(c1nnnn1CC1CCC1)Nc1ccc(OC(F)F)cc1 C(C(C)(C)C(=O)N1CCC(C(C)(C)CNC(c2cc(Cl)ns2)=O)CC1)OCC CCC(C)(C)CCCC(=O)N1CC(O)CC1(C)C(N1CC(F)(C2CC2)C1)=O c1(CCN2CC(C)C(C(=O)OC(C)(C)C)CC2)cc(Br)cc([N+](=O)[O-])c1 C(=O)(C1=CCCCO1)NC(CNC(c1nc(C(C)OCC)sc1)=O)CC N1(C(C(C)(C)c2ccccn2)=O)CC2CCCC(C1)N2C(=O)CCF CCCCC(CNC1CC2C=CC1C2)NC(=O)C(C)(C)NC(=O)C(F)(F)F C(=O)(CCCCCn1cc(CCSC)nn1)N(C(CC)C)Cc1ccn(C)n1 c1(C(=O)OC2CCCC=C2Br)cccc2c1CCO2 c1(OC)ccnc(OC)c1C(=O)N(C)CC1CN(C(c2cc(C)c(N)cn2)=O)C1 CON1CCC(C(=O)N(CC(O)CN(C)C(C2(F)CCOC2)=O)C)CC1 N1(C(C2(CCC=C)CCCC2)=O)CCCC(C)(CNC(C2(C)CS(=O)(=O)C2)=O)C1 c1(OC)c(CN2CCCC(N3CCC3)C2)ccc2ccccc12 C(C(O)C(CC)CC)NC(CC1N(C(C(CC=C)NC(C)=O)=O)CC1)=O C(C)(CCCCNC(=O)C(c1cccnc1)O)NC(C1(CC)CC1(F)F)=O C(C(C)(CC(C)C)NC(c1cc(C)c(N)cn1)=O)NC(c1cc(OC)no1)=O N1(C(c2cc(F)cnc2Cl)=O)CCC2(C(=O)N(C3CCCC3)CCO)CCCC12 C12(CCN(C(=O)CCC3CCCOC3)C1)C(=O)N2.C1(COC)CC(O)C1 NS(=O)(=O)N1CCC(C(=O)NCCn2cc(CC3CCCOC3)nn2)CC1 N1(C(c2c(C)n[nH]c2C)=O)CC2(CCN(C(c3cnnc(Cl)c3)=O)CC2)CC1C N1(C(C(Cn2ccnn2)NC(=O)COC2CCCCC2)=O)CCc2ncsc2C1 N1(C(C)=O)CCC(C(=O)N(CCC(C)NC(c2c(C)noc2C2CC2)=O)C)CC1 C1(C(=O)NCCCOC2CCN(C(C(C(C)C)O)=O)CC2)CC2OC(=O)OC2C1 c1(OC(C)C)cccc(-n2c(-n3cccc3)cnc2C(=O)NC(CO)C(C)O)c1 C(C(C)C(C)C(=O)N1CCC(c2nc(OC)cc(O)n2)CC1)OC C1(C(=O)NCC(C)C)(CC2CC2)CCN(C(=O)CCCC2CCCC2)C1 C1(C(=O)NC(C2CCC2)C)CN(C(=O)C(C)(C)n2cccn2)CC1F c1(C(N2CC(CNC(Cc3c(CC)cccc3)=O)C(O)C2)=O)ccnc(F)c1N O(NC(=O)CN(C(=O)CC(C)C1CCCCC1)CCOC)CCOCC C(=O)(C(O)C(F)(F)F)NCC1CCN(C(C2(CC)CCOC2)=O)CC1 c1(C(C)=O)cc(C(=O)NC2CCCC2NC(C2CCC3(CCC3)C2)=O)ccc1C c1(C(N2CC(CNC(C(C(CC)C)O)=O)C(O)C2)=O)cccc2c1OC(F)(F)O2 Cc1nn(C2CC2)c(Cl)c1C(=O)NCCCCCCN(C(=O)C(C)C(C)C)C1CC1 C1(NC(c2cn(CCNC(c3c(OCC)cnnc3)=O)nc2)=O)CCCCNC1=O c1(C(N2C(C)COCC2)=O)n[nH]c2c1CN(C)CC2 n1(CC)c(C(=O)NC2CN(C(c3onc(C)c3C(F)(F)F)=O)CC2O)cnc1O c1(C(=O)NCCC(CCNC(CCN(C(C)=O)C)=O)C)ccc2ncnn2n1 C1(OC(F)F)CC(C(=O)NC2(CNC(=O)CCNC3CCCO3)CC2)CC1OOC.O C1(CC(=O)NC(CN(C(c2cncc(COC)c2)=O)CC)C)COC(C)(C)CO1 c1(CNC(C2CCCN(C(=O)CCc3cccnc3)C2)=O)cc(Br)cnc1O C1(C(=O)NC2(C)CN(C(c3ccc(OC)nn3)=O)C2)C2CCC3C(C2)CC13 C1(CNC(CCC2CCCN(C)C2)=O)CC2CCC1N2C(=O)C(C)(C)C#N C1(COC)CCCCN1C(=O)CC(CC1CC1)NC(c1ccc(C2CC2)cc1)=O c1(SCC(=O)NC(CC)CNC(=O)C(CC2CC2)OC)cc(Cl)ccc1Cl N1(C(CN(CCOC)C)=O)CCC(NC(=O)Cc2cccc(Cl)c2F)CC1C Nc1cc(F)ccc1C(=O)NC1CCOC(CNC(c2nnsc2C(F)F)=O)C1 C(=O)(CCC(=O)NC(C)(C)COCCCNC(C1CC(C)C1(C)C)=O)NC C1(CNCc2cn(C)nc2C(F)F)C2CCCC1C(=O)N2 N1(C(CCC(CC#C)NC)=O)CCn2ncc(-c3nn[nH]n3)c2C1 C1(NC(c2n(CCC)ncc2)=O)COC2(CCN(C(=O)CC3CCOC3)C2)C1 Cn1nc(C(N2CCC(C)(CNC(C3CCCSC3)=O)C2)=O)cc1Br C#CC1(NC(c2cc(CNC(c3csnn3)=O)nn2C)=O)CCCCC1 n1(CCC)cc(C(=O)NC(CN(C)C)C(=O)NC(C)C(C)n2cccn2)nn1 CC1CCc2ccc(C(=O)NC3CC4(C3)CC4NC(=O)CCC3CC3)nc2C1 c1(NC(=O)NC(c2ccc3nc(O)[nH]c3c2)C)c[nH]c2c(Cl)cc(Cl)cc12 N1(C(COCCC=C)=O)CCN(C(=O)CC(C)OCCCC)CC1C(C)C N1(C(C2CCC3(CCC3)C2)=O)CC(NC(c2cn(C)nc2)(C)C)CC(O)C1 c1(C(N2CCC(C(C)NC(C3(OC)CC3)=O)C2)=O)cc(Cl)nc(Cl)c1 N1(C(C)C)CC2CCC2(C(F)(F)F)C1.C1(O)CCCC1.C1(=O)CO1 c1(C(N2CCC(CC#C)(NC(=O)C(C)OC)C2)=O)coc(S(=O)(=O)NC)c1 C1(C)(CNC(c2n(CCC)ccc2)=O)COCCN(C(=O)C2=CCCSC2)C1 N1(SC)CCCC(CN2CCCC2)C1.C1CCC(=O)N2CC(C)(C2)c2cn1nn2 Cc1ccc(-c2ccc(C(=O)NCc3cc(Cl)ccc3I)nc2)c(CO)c1 c1(CNC(CSCC)C)cc(NC(=O)C(N2CC3CCC3(C)C2)=O)c(OC)c(F)c1 c1(C(c2nnnn2CCCc2ccccc2)NCC(CO)OC)cnc(Cl)s1 Cn1cnc2cncc(C(=O)NCCC3CCCN(C(C4(C)CCCS4)=O)C3)c12 C(=O)(CS(=O)C(F)(F)F)N(CC(C)NC(=O)CCn1cnccc1=O)C N1(C(CCNC(C2C(C)C2)=O)=O)CC2(CC(NC(=O)CC3COCCO3)C2)C1 c1(OC)ccc(C(=O)NCC(CNC(C2(C)COC(=O)C2)=O)CO)c(F)c1F N1(C(c2nn(C)c(O)c2)=O)CCC2(CCC2)C(NC(=O)C2=COCCO2)C1 Cc1ncnc(C(=O)NCC2CCN(C(C3(C)CC3(Cl)Cl)=O)CC2)c1C n1(CCCC=O)c(O)nnc1O.C1(SCC(=O)N2CCC(O)C2)CCS(=O)(=O)C1 CC(CC(F)(F)F)C(=O)NCCNC(=O)C(C)(O)C(F)(F)F CC1(C)CN(C(=O)C2=COCCO2)CCC1NC(c1cc(Cl)cc(F)c1N)=O C(=O)(C(O)(C(F)(F)F)c1ccccc1)NCC(C)CNC(=O)C(N)=O c1(OC)c(C(=O)NC2CCCN(C(=O)CO)C2C)ccnc1F C=Cc1ccc(C(C)NC(c2sncc2C)c2nnnn2CCC2(C)CC2)cc1 c1(C(=O)NC(C(C)NC(CC2(NC(C)=O)CC2)=O)CO)cccc(C)c1F C1(NC(c2cc(C(N)=O)ncc2)=O)CC(CNC(C2CC3(CC3)C2)=O)C12CCC2 c1(OC)ccc(CNCC2(NC(=O)OC(C)(C)C)CC3CCC2C3)c(OC)n1 C(C(=O)NCCC(C)N(C)C(c1ccc(N2CCCC2)cc1)=O)(C(C)C)SC C=C(Cl)CC(C(=O)N1CC(CCO)(CC)C1)NC(C1CC(C(=O)OCC)C1)=O C1(C)(NC(C(CC)(O)c2cccc(Cl)c2)=O)CCN(C(=O)C(O)C(F)(F)F)CC1 C1(CCC)(NC(=O)C(C(C)C)NC(N)=O)CCN(C(=O)CCOC2CCC2)C1 Cc1noc2ncnc(N3CC(C)(C)CC3CNC(c3ccc4n[nH]cc4c3)=O)c12 c1(CC)ccc(OC)c(Br)c1OC.C1(O)(C)CCN(C(C2CCC(=O)N2C)=O)C1 N1(C(C(n2cc(-c3ccncc3)nn2)C)=O)CCOC(c2ccccc2Cl)C1 C(=O)(CC(C)P(C)(C)=O)N1CC2(N(C(C(CC)(F)F)=O)CC2)C1 N1(Cc2ccc(CC)cc2)CCN(CC(=O)NC(c2ccccc2)C#N)C(=O)C1 c1(C(=O)NC2C(NC(C(CC)(C)OC)=O)CCCC2)cc(C2CC2)cc(F)c1 c1(NCc2nnc(C(C)C)s2)nccc(=NCc2nc(C(F)(F)F)n[nH]2)[nH]1 CCCC(CNC(c1cscn1)=O)C(=O)NCC1CC(O)C12CCC2 C1(NC(c2coc(C3CCC3)n2)=O)CCCC(NC(c2cc(C(F)F)[nH]n2)=O)C1 C1(NC(C(CCO)N(C)C)=O)CC2CCC(C1)N2C(=O)C(c1cccc(Cl)c1)O c1(SCC(N2CC(O)(C3CCCN3C(c3ccncn3)=O)C2)=O)nnc(S)s1 c1(C(=O)NC(CCOC)CNC(c2cn(C)c(C)n2)=O)cnc2c(c1)CCC2 c1(C(N(CCCCN(C)C(C2C3CC3C3CC23)=O)C)=O)cc2ncccn2n1 CC(F)(F)CCCCN(C(c1ncccc1Cl)C(=O)NC(c1ccccc1)C)C c1(NCc2c(C)ccs2)ccc(S(=O)(=O)NCC(C)(C)n2ccnc2)cc1Br C(=O)(CC(F)(F)CNC(c1nnnn1Cc1ccco1)C1CCCOC1)OCC C1(C(=O)NCC2(F)CN(C(c3ccc(C)nc3C)=O)C2)CCCCC12CCC2 C(=O)(C1=CC2(CCN(C(C3CCC(OC(C)=O)CC3)=O)C2)C1)N(CCCC)C1CC1 C1(OC)CC(NC(=NC)NCCC2CC2)C12CCC2.C1(C=O)CCCC1 CC1(C)OC2(CO)CC1(C(N1CC(O)CC1CNC(=O)CN1CCCCC1)=O)C2 C=C1CCC(C(=O)N(CC(O)CN(C)C(c2cscc2SC)=O)C)CC1 N1(C(=O)CCC2CCCC2)CC2CCCC2(C(N2CC3(C=CCO3)C2)=O)C1 C1(CNC(CNS(CC)(=O)=O)=O)CCCC1C(F)(F)F C(=O)(CC(C=C)CC)N(CC#C)CCF.c1(C2C(=O)N2)ccc(C2CCC2)cc1 CCC(N=c1[nH]c(N2CCC(C)(NC)CC2)nc2cccc(F)c12)c1nccs1 c1(OCC(=O)NCC2C(NC(c3nc(C)nn3C)=O)CCC2)cc(Cl)ccc1C C(=O)(C(O)C(F)(F)F)OC.C1=CCOc2nccc1c2 Cc1cc(C(N2CC(C)(C)CC2CNC(C2CC23CC3)=O)=O)c(C)cn1 CN1CCNC(CNC(C2CC23CN(Cc2cnc(-c4ccccc4)s2)C3)=O)C1 C(=O)(CC(C)(C)CN(C)C)NC(C(C(=O)NC1(c2onc(C)n2)CC1)C)C C#CC1CN(C(=O)C(C)CC=C)CCN1C(=O)COCCC(C)C Cn1cc2cc1C(=O)N2.N1(C(C2CC2c2cccnc2)=O)CCC(F)C1 C(=O)(C(CCC(N)=O)N(C)C)NC1C(C)CN(C(=O)COCCOC2CCC2)C1 c1(C(N(C(C)CCNC(C2(C)CCC(=O)N2)=O)C)=O)coc2c1CSC2 Cc1noc2ncc(C(=O)NCC(CC(C)C)NC(=O)C3=COCCO3)cc12 c1(C(=O)NC2(CNC(c3occc3C3CC3)=O)CCC2)cc2c(=O)[nH]ccn2c1 CCCCCCC(C)C(=O)NC1C2CCC1CN(C(=O)C1=COCCC1)C2 N1(c2ccccc2)CCCC(NC(C2(NC(=O)NC)CC2(C)C)=O)C1=O.C(C)OC C=CC1OCCCC1C(=O)NCC1(NC(c2cc(CC)no2)=O)CCCC1 C(C)(C(C)(C)C)N(C(CCN(C(=O)CCc1ccccn1)CC=C)=O)C c1(C(N(CC(C)NC(C2(CF)CCC2)=O)C)=O)ccc(Cl)c(F)c1F N1(CCN2CC(c3nncn3C)(C(=O)OC)C2)CCCS1(=O)=O N1(C(C)C2CC2)CCCC(C)(NC(N2CCC(CS(N)(=O)=O)C2)=O)C1 C(=O)(CC(C)C(F)(F)F)N1CC(CC(N2CCC(N(CC)CC)C2)=O)C2(C1)CC2 C1(C(=O)OCC)OCCC1CNC(c1cc(Cl)ns1)=O C1(CC)CCC(C)N(C(=O)C(c2ccccc2Cl)C)C1.c1(C)cn(CCCS)nn1 C12(C(=O)NC(CCC(C)C)C)C(NC(C3CCCC(O)C3)=O)C3CC1C2C3 C1(C(N(CCCCNC(C2CC3(CC3)C2)=O)C)=O)CCOC(C)(C)C1 c1(NC(C)=O)ccc(C(=O)NC(C2CCN(C(c3coc(Cl)c3)=O)C2)C)nc1 C1(C(=O)NCC)(NC(=O)C(=O)NCCSCCCO)CC1(C)C N1(C(c2nnc(C)s2)=O)CCCN(C(c2[nH]nnc2-c2ccccc2)=O)CC1C C(=O)(C(CC(C)C)NC(C1C=CCN(C(=O)CC2CCCN2C)C1)=O)NC N1(C(c2c(F)ccc(C)n2)=O)CCCC12CCCN(C(C1CC3CCC1C3)=O)C2 N1(CCC2CCN(C(CN(C(CN(C(=O)OCC)C)=O)C)=O)C2)CCN(C)CC1 c1(NCCCOCC)nccc(=NC2CCCSC2)[nH]1 c1(C(C)CC(N2CC(NC(=O)CP(C)(C)=O)C(C(F)F)C2)=O)ccc(F)c(F)c1 c1(C(=O)NCC(CC=C)NC(COCC#C)=O)ccnnc1S CC(C)(O)C(F)CNC(=O)COCCC1CC1.C1(=O)C(O)CN1 C1(NC(C2CCCCC2C(F)(F)F)=O)CC2CCC(C1)N2CC1CCOC1 c1(C(N(C(CNC(C(n2cc(Cl)cn2)C)=O)C)C)=O)c[nH]c2ccccc2c1=N C1(C(N(CCCCNC(C2(CC#C)CCCO2)=O)C)=O)CCc2ncnn2C1 C1(NC(=O)CC2CCCC2)CCCN(C(c2occc2Cn2cccn2)=O)C1 c1(CC)nc(C)n(C)c1C(=O)NCC(C)(C)CN(C(=O)CC1CN(C(C)=O)C1)C c1(C(N2CCN(C(c3ccnnc3)=O)C3CC23)=O)cc(Br)cc(C(F)(F)F)c1F N1(C(C(C)C)=O)CCC(C(F)C(N2CC=CC2C(=O)N(C)C)=O)C1 C(CC(C(=O)N1CCN(Cc2cccnc2)CC1)NC=O)SC.C12CN(C1)C2=O N1(CCCNC(C=CC(C)(C)C)=O)CCN(C(c2cnc(Cl)[nH]2)=O)CC1=O Cc1ccc(Cl)c(C(N2CCC2CNC(C2CCC(=O)NC2=O)(C)C(=O)O)=O)c1 c1(C(N2CCN(C(C3(OC)CCSC3)=O)CC2C)=O)ccc(C#N)cc1C C1(CNC(C=C(C)C)=O)CC(F)CN1C(=O)C(F)CC1CCC1 C(=O)(C(CNC(=O)CCCCC1CC1)CC1CC1)NCC1CN(C(N)=O)C1 C1(N(C(CCOCCCOC)=O)C)CCCCN(C(C2CNC(=O)N2)=O)C1 c1(CNC(C2CC3(CC(NC(=O)Cn4cc(Br)cn4)C3)C2)=O)nc2ccccc2[nH]1 c1(CNC(c2ccccc2)COC)ccc(C2=CCOCC2)nc1 O=C1NC2(CO1)CC(C(N1CCCC1CN(C(C1COCCO1)=O)C1CC1)=O)C2 C(=O)(CC(F)(F)CC)NC(CC)CNC(=O)CC1CCN(C)C1=O S(=O)(=O)(C=Cc1ccccc1)NC(C(=O)OCCC)Cc1cc(Br)ccc1C c1(C(=O)NCCNC(c2cccc(OCCC)c2)=O)cccc(F)c1Br c1(CC(=O)NC(C(C)C)C(C)NC(c2ncn(C)n2)=O)c[nH]c2cccnc12 C=C=C(C)CC(=O)NCc1cc(C(=O)NCC(CSC)OC)co1 c1(C(N2C3CN(C(CC(=O)NC4CC4)=O)C(C3)C2)=O)cnn2c1OCC2 CCC(C#N)C(=O)N1CCC(C(=O)NCc2ncoc2C(C)C)CC1 N1(C(c2n(CC)ncc2)=O)CCC2(CC(NC(=O)C(C)(C)C3CC3)CO2)C1 CC1(C)CCC(CNC(C2CCS2(=O)=O)=O)N(C(c2sccc2OC(F)F)=O)C1 c1(C(=O)NC2(CNC(=O)COC3CCC3)CC2)cccc(-c2ccsc2)c1 c1(C(=O)NCC(CNC(=O)C(N2CCOC2=O)C)OC)cccc2c1C(=O)NC2 c1(CC(=O)NCCN(CCC)C(c2cc(C(N)=O)n(C)n2)=O)ccc(C)c(F)c1 c1(NC)ccc(C(=O)NC2CC2CNC(c2cc(C(F)(F)F)ns2)=O)cc1[N+](=O)[O-] Fc1ccc2[nH]cc(CNc3ccc(I)cc3)c2c1 C(CNC(=O)C(O)CCc1ccccc1)(CC(F)(F)F)NC(c1ccsc1)=O C1(NC(c2n(-c3c(C)cccc3)nnn2)(C)C)CC2(C1)CC(O)C2 C=CCC(CC)C(=O)NCCCOCCOCCC(=O)NC1CCC1 c1(OC)ccc(C(CO)NC(=O)NCc2ccc(-c3scnc3C)cc2)c(Br)c1 c1(C(C(=O)N(CCCN)C2CC2)O)cccnc1.C(=O)(CC)C=O c1(Cc2nc(CC(N3CCC(N(CCC)C)C3)=O)sc2)ccc(F)cc1 C(=O)(CC(C(C)(C)C)NC(=O)CCCc1cnn[nH]1)NC1CCN(CC)C1 N1(c2ccc(CSCCCC(=O)N(C)C)cc2)C(=O)C(CCCCO)N(C)C1=O CCCCCC(O)C(C)C(=O)N(CC(O)CNC(=O)CN(C)C1CC1)C c1(OC)cccc2c(C(=O)N(C3CC(NC(C4(C)CCOC4)=O)C3)C)csc12 CCC1=C(C(=O)N2CC(CCNC(c3cc(C)nc4ncnn34)=O)C2)CCCO1 c1(C(=O)OCC)ccnc(C(N2CC(CO)(NC(=O)CN3CCCC3=O)C2)=O)c1 N1(c2ccc(NCc3n(CC)c(C)nc3)cn2)CCS(=O)CC1C C(=O)(C1=CC2CCC1C2)N1C2C(NC(c3c(C)nn(C(C)(C)C)c3)=O)CC(C2)C1 C(C(C)C(C)C(=O)NCCC(C(=O)NC(C)(C)CN(C)C)OC)OC C1(C(C)C)(C(=O)N(CCN=[N+]=[N-])C)CCN(C(c2nccs2)=O)C1 Cc1cc(C)c(C(=O)NCCN2CCCN(C(=O)CCCN(C)C)CC2)cc1C C(=O)(C(CNC(C1(C(F)(F)F)CCC1CO)=O)(CC)CC)OC CC1=CCC(C)(C(N2CC(CNC(c3cccc(F)c3)=O)C(C)C2)=O)CC1 c1(NC(CC)=O)c(C(c2nnnn2C2CCCC2)NCCF)cccc1C CC1Cc2c[nH]nc2C(C(=O)N2CCCC(N(C(=O)C(Cl)=CCl)C)C2)C1 c1(NC(C23C(CN(C(c4cncc(COC)c4)=O)C2)C3)=O)nc(C)c(N)cc1C N1(C(CN(C(=O)C(O)C(C)(C)CC)CC#C)=O)Cc2cncnc2C1 N1(C(CSCCOC)=O)CC2(CCN(C(C3(C)CCC(C)(C)CC3)=O)CC2)C1 N1(C(C=CC(=O)OCC)=O)CC(C(N2CCC23CC(C(N)=O)C3)=O)CCC1C Cc1cc(C(N2CCN(C(=O)CSC(C)(C)C)CC2C)=O)c([N+](=O)[O-])cc1F CC#CCCC(=O)NC1(C2CCCCN2C(C2CCCSC2)=O)CC1 Cc1cccc(CN(C)CC2CCCN2C(=O)C(=O)Nc2sc(C)cc2C)c1 CC1(C)CN(C(C2CCN(C(c3ccc(Cl)cc3)=O)CCO2)=O)CCO1 c1(NC(C(C)N(C(=O)CCN2CCCCC2=O)CC)=O)ccc2ccccc2c1 C1(C(=O)NC(CC=C)CNC(=O)Cc2cc(C(C)C)no2)CCC(N(C)C)CC1 C(C(C)(C)CNC(C1CC1(C)Br)=O)N(C)C(C1(O)CCC1)=O CC1CCCN(C(=O)CN(C(=O)C=Cc2cn[nH]c2)CC2CC2)C1CO c1(C(=O)NC2CC(NC(C3(COC)CCCCO3)=O)C2)ccnc2c1cnn2C c1(OC)cc([N+](=O)[O-])ccc1NCc1csc(CNC(=O)OC)n1 c1(CC(C)C)ccc(CC(N2CCC(C)(CNC(C3(C)CC=CC3)=O)C2)=O)cc1 C(N=c1[nH]c(N2CCC(F)C(F)C2)nc2c1CCC2)C1(OC)CCS(=O)(=O)C1 C(CCCCC(=O)N1CC(N(C(=O)Cc2ccn(C)n2)C)C1)SC N1(C(C(C)C2(O)CCC2)=O)CCCC(C(=O)NC(C2CC2)C2CC2)C1 C1(C(=O)NCC(CC)n2cccn2)C2CC3C(C2NC(c2ccc(=N)[nH]c2)=O)C13 c1(C(=O)NC(CCNC(C2(COC)CC=CC2)=O)(C)C)cc(C#N)cc(C)n1 N1(C(C(CC)NC(C)=O)=O)CCC(C(=O)N)=C(F)C1.c1(CC)ccnn1C c1(CN2C(C(N3CCCN(CCC)CC3)=O)CC(C)(C)C2)c[nH]c2cnccc12 N1(CC2C(C(=O)NCCNC(c3cocn3)=O)C2)CCCCC1 C(C)(N=c1[nH]c(=N)[nH]c(=NCC(C)C)[nH]1)c1cc(C)sc1C C1(NC(C(C)CC2CCC2)=O)CCN(C(=O)C=Cc2cnccn2)C1C Cn1cc(C(=O)NC2COCC2NC(=O)Cn2cnnc2O)nc1C(F)F CC1(C)CCCC(C(=O)NCC(C2CCCN2C(=O)C2=C(Cl)CC2)(C)C)CC1 N1(CCNC(C2CCN(C(C3(Oc4ccccc4)CC3)=O)C2)=O)CCC(O)CC1 c1(C(C(=O)NCCCN(C(c2cccnc2N)=O)CC)C)ccccc1C CCC(C)CCCC(=O)N1CC2C(CNC(C3(c4ncccc4F)CC3)=O)C2C1 C1(NC(=O)CNC(c2ccc(Cl)s2)=O)C=CC(CNc2cnns2)C1 N1(C(c2ccc(-c3cc(=N)[nH]cc3)o2)=O)CC2(CCC2)c2ncccc21 C1(CNC(C2C(OCC)C2)=O)CN(C(=O)Cn2nnnc2C(C)C)CC1O C(C(C)(O)CC(=O)N1CCCC(CCNC(=O)CCNC(C)=O)C1)OC N1(C(=O)COc2cccc(Cl)c2)CCN(C(c2c(Cl)cncc2Cl)=O)C2CC12 C1(C2CCOCC2)(C(N2CC(CCNC(CCOC(C)C)=O)C(C)C2)=O)CC1 N1(c2sc(C(=O)OC)c(C)n2)CCC(F)(CNC(=O)C(=O)NC2CC2)CC1 N1(C(CNC(CC(C)(C)C)=O)=O)CC2CCC(NC(c3cnc(O)o3)=O)CC2C1 C(=O)(C(F)C(C)CNC(c1ncccc1F)=O)N(C(C(=O)OC)C)C C1(C(=O)OCC(=O)Nc2cccc(C)c2)C(O)C(=O)N(C)C1C N1(CC(C)NC(C2(C)CC2)=O)CCN(C(C2(C(F)F)CC2)=O)CC1 c1(OC)ccc(Cl)c(C(N2CCC(NC(c3cncc(Br)c3)=O)C2)=O)c1 C1(CNC(C(C)N(C)C)=O)CN(C)CCN1C(c1ccc(C(C)(C)C)cc1)=O c1(CN(c2cc(NCC3CCCC34CC4)ncn2)C)ccc(F)cc1F CC1(C)COCC1C(N1CCCCC1CC(=O)Nc1ccsc1)=O Cc1nn(C)c(Cl)c1CN1CCN(C(c2cc(Cl)c(Cl)s2)=O)C2CC12 c1(C(C(=O)NCC)N(C2CCSCC2)CCCC)ccc(C)cc1OC C(c1ccc2c(c1)CCO2)=CC(=O)NC1CN(C(C2CC3(CC(C)(C)C3)C2)=O)C1 C1(CC=C)(C(=O)NCC(C)S(C)(=O)=O)CCCN1C(c1cnc(C)s1)=O C(=O)(C(C#N)CCC)NCCN(CCC#C)C(C1CC12CCCCC2)=O Cc1ccn(CC(C)C(=O)C(=O)C(C)OCC(C)C)n1.C1(CCN)(N)CCC1 c1(CCC(=O)NCC2CCN(C(c3ccc(F)cc3)=O)C2)n[nH]c2c1CCCC2 C(=O)(C1Cc2ccccc21)N1CC(CCNC(c2c(CC)nccn2)=O)(OC)C1 C12(NC(C=C(C)C(C)(C)C)=O)CC1CN(C(=O)CSCc1cscn1)C2 C1(CNC(=O)CC2CSC2)Cc2ccccc2CN1C(=O)CC1CCC12CCC2 N1(C(c2ccc(CC)[nH]2)=O)CCCC(CC(=O)NCCc2cc(C)on2)CC1 C1(C(=O)NC2CCCCN(C(C(C(C)C)(C)O)=O)C2)CCc2nncn2C1 C1(N(C(Cc2cc(C)[nH]n2)=O)C)CN(C(C2CCCC2(F)F)=O)CC1(C)C c1(C(=O)OC)cccc2c1CN(C(=O)CC1CCCN1C(C1C=CCC1)=O)C2 C1(CN)(NC(c2cnns2)=O)CCCCCC1.n1(CC(=O)C(=O)CC2CC2)ccnn1 C(CCCCNC(c1c[nH]nc1-c1ccc(Cl)s1)=O)NC(c1sccc1Cl)=O C1(NC(Cc2c(C)noc2C)=O)CCC2(CCN(C(C3(O)CC3)=O)CC2)C1 c1(CC(=O)NC(C2CCN(C(CCCCC)=O)C2)C)cccc(OCC)c1Cl N1(C(C2CCN(C(C(CCC(C)C)F)=O)C2C)=O)CCc2nc(O)[nH]c2C1 CCCCC(CNC(c1c[nH]cc1COC)=O)NC(=O)CC1(C)CCOCC1 C1(CNC(c2ccccc2Cl)=O)CC(NC(=O)CC2(C(F)F)CC2)C12CCC2 c1(C(=O)NCCCCCC)cccc(CN2CCCC2c2ncc[nH]2)c1 N1(C(C(c2cccnc2)NC(CCC(=O)N(C)C)=O)=O)CCC(F)(CF)CC1 C(CC(C(=O)NCCF)NC(C1COC(=O)N1)=O)OCC c1(C(C(=O)NC2CCC(CNC(c3c(CC)ccs3)=O)C2)=O)ccc(F)cc1C c1(C(=O)NC2C(NC(COC(CC)C)=O)CCOC2)sc2nccn2c1C C1(NC(c2c[nH]ccc2=O)=O)CCN(CCN)C1=O C(=O)(C1=CS(=O)CCC1)N1C(C(C)NC(c2cc(C)c(C)nn2)=O)CCC1 C1(CCNC(=O)CC(C)CF)(OC)CCN(C(=O)C(C)OCCC2CCCO2)C1 N1(C(CSc2c(C)cccn2)=O)CCCC(C)(NC(=O)CCCF)C1 CC1CN(C(=O)NCC(F)SC2CCC2)CCC1(O)C(F)(F)F N1(C(c2nc(C(C)(F)F)sc2)=O)CCCCC(NC(c2ccc(CF)cc2)=O)C1 N1(C(C(C)OC)=O)CC(C)(C)OCC1CNC(=O)C(C)(C)c1cnc[nH]1 N1(C(COCCC)=O)CCOCC(CNC(=O)CC2COCC(C)(C)O2)C1 C(N=c1[nH]cnc(Cl)c1C#N)C1CC(NC(C(=O)NC(C)C)=O)C1 N1(C(c2cncn2C)C(=O)NCCSC)CCOCC(C(C)C)C1 N1(C(C(COC)O)=O)CCC(C)C1C(=O)N(C1CCCCC1)C N1(C(CC(C)(C)C)=O)CCN(CC2CCCCO2)CC(O)C1.C1(=O)CN1 C(C1CCC(C)CC1)=C(C)C(=O)NCC1CCN(C(=O)Nc2cccnc2)CC1 C=Cc1cncc(C(=O)NCC2CN(C)CCN2C(c2ccc(C)c(C)n2)=O)c1 C(=O)(C(O)C1=CCCCC1)N.C(CCC(=O)NCCCOCCOCCOC)SC C1(CC(=O)OCC)CCCN(C(c2ccc(Br)nc2)C(=O)NCCCSC)CC1 C=C(C)C(C)(C)C(=O)N1CCN(C(=O)C=Cc2sccc2C)C(C2CC(CC)C2)C1 CC1C(C(N2CCN(C3CN(C(C45CSCC4C5)=O)C3)CC2)=O)CCN1C c1(C(=O)NCC2N(C(C3CCN(CC)C3)=O)CC(F)C2)cc2sccc2s1 Cn1cncc1C(O)C(=O)NCCCOCCNC(c1conc1C1CC1)=O O=C1NC(=O)C2CN(C(C3CCCCN3C(C3CCCO3)=O)=O)CC12 CCC(C)(C#N)C(=O)NCc1cc(C(=O)NCC(O)COC)cs1 C(=O)(CC(C)(C)C1CC1)NC(C(=O)N(C)CC1(OCC)CCC1)c1cccs1 N1CC2CN(C(c3ccc(O)nc3)=O)CCC12.CN(CCc1ccccc1)N=O c1(CCC)cc(C(=O)NC(C)CN(C(=O)COCc2cncc(F)c2)C)n(C)n1 Cc1ccc(C(=O)NC23CCN(C(c4nccc(Cl)c4C)=O)CC2C3)cc1O CC1CCCCC1C(=O)NC1CCC(NC(=O)OC2CCC2)CC1 N1(Cc2ccc(OC)c(F)c2)CCC2(CCCC2C(N2CC(C)(O)C2)=O)C1 c1(OC)ccc(F)c(NC(C23CCN(C(C4CC5CCC(C4)C5)=O)CC2C3)=O)c1 c1(C(=O)NCCNC(C2(CC=C)CC2)=O)nn(-c2ccc(Cl)cc2)c2c1CCC2 Cc1nccn1CCNC(C1CCCC1NC(=O)Cc1ccn(C)c1)=O N1(C(C(=O)NC2CCN(CC(=O)N(CC)CC)CC2C)=O)CCC(P(C)(C)=O)C1 n1(CCOC)ccc(C(=O)N(C2CCN(C(C3(N(C)C)CC3)=O)C2)C)n1 c1(OC)ccccc1NC(C1CCN(C(=O)C=CI)C1)=O N1(CCN2CCC(OC)C2)C(=O)CCN(CC2CC2)C1=O N1(C(=O)CC2CC2c2cccc(O)c2)CCC(N=c2[nH]nc(C(F)(F)F)s2)C1 C1(OC)CC2(C1)CC(C(=O)NCCC1CSCCN1C(c1ccc(CO)cn1)=O)C2 C1(OC)CC(C(=O)N(CC(CO)C2CCC2)Cc2ccco2)N(C2CCCC2)C1 C(CC(C)C(=O)NCC1CCCN1c1cc(OC)ncn1)OC c1(C(N2CCC(O)(CN(C)C(C3CCCC3)=O)C2)=O)cc(Cl)ccc1[N+](=O)[O-] CC1OC2CCC1(C(=O)NCCCCCCN(C(=O)CC1(N(C)C)CC1)C)C2 n1(CCCC)cc(C(=O)NCC(O)CN(C(=O)C=CC(C)(C)C)C)nn1 C(=O)(C1=CCC(NC(c2cn(CCO)nn2)=O)C1)NC1(c2cc(C)on2)CC1 C(C)(CNC(C1CC=CCO1)=O)(C(C)C)NC(C1CC(CC(=O)OC)C1)=O C1(NC(CSCCC)=O)CCC2(CC1)CC(NC(c1ccc3ccnn3c1)=O)C2 c1(CC)oc(C)cc1C(N1CCOCC1CNC(=O)CCc1c(C)noc1C)=O n1(COC)nccc1C(=O)NC(C)(C(=O)NCC(C)CC1CCC1)C1CCC1 CCC(C)(COC)C(=O)NCCCCCN(C)C(c1cc(C)cc(Br)c1)=O C1(NC(c2cccc(C3CC3)c2)=O)CC(CO)N(C(=O)C(F)OC(F)(F)F)C1 C(=O)(C(C)(C)CCCF)N(C(c1cn(-c2ccc(Br)cc2C)nn1)CCC)CC N1(C(CC(C)C)=O)CC2COCC2(C(=O)N(C)Cc2ncn(C)n2)C1 N1(C(C(C)C2CCCC2)=O)CCC2(CCCC2NC(c2ccn(O)c(=O)c2)=O)C1 N1(C(C(=O)NCCc2ccccc2Cl)=O)CCCC2CC3(CCC3)C12 N1(C(c2[nH]cc(C#N)c2)=O)CCCCC1C1CCCN1C(c1cc2n(n1)CCO2)=O C1(CNC(c2n(C(CC)CC)ncc2)=O)CCCN(c2ncc(Cl)cn2)C1 Cc1cc(C)n(C(C)C(=O)NC2CN(C(C3(C(F)F)CCC3)=O)CC2C)n1 Cn1cc(C(=O)NCC(CNC(=O)CC2(n3ccnc3)CC2)CO)ccc1=O N1(C(C2N(C(Cc3c(C)n(C)nc3)=O)CCCC2)=O)CC(C)N(C)C(C)C1 C(=O)(C(CCCC)C(C)C)N1CCC(C#C)(C(=O)NC2CN(C)C2)C1 c1(CCC(=O)NC(C(=O)NCCCCC)c2ccco2)conc1C c1(N2CC(N(C(C(=CC3CCCC3)C)=O)C)C2)ncnc2ccccc12 CCCC(C)(O)CC(=O)NC(CC1CC1)CC(N1CCCN(C=O)CC1)=O Cc1c(CNCC2NCCC2C2CC2)cccc1Cl CC(CCO)N=c1[nH]c(=N)[nH]c(=NCC2Cc3cc(Cl)ccc3O2)[nH]1 N1(C(c2n(CC)ccc2)=O)CCC2(NC(C3CCN(C(C)C)CC3)=O)CC2C1 n1(CCN(C(=O)CC2CCCC2NC(=O)OC(C)(C)C)C)ccc(=O)n(C)c1=O O=C1CCN(Cc2ccc(Cl)cn2)C(=O)N1CC(F)F.c12ccc(cc1)SC2 S(=O)(=O)(c1cccc(C(N2CCC(C(=O)NCCc3ncc[nH]3)CC2)=O)c1)NC N1(C(c2cc(C)on2)=O)CCC2(CC1)COC(C(N1CCCC3CCCCC13)=O)C2 Cc1cc(C#N)nc(=NCC2CN(C(=O)Cc3ccccc3C)CCCO2)[nH]1 CC(C)(C(=O)NCC(O)CCNC(C1CC(=O)N(CCN(C)C)C1)=O)C(F)F c1(NCC(C)CCCO)nccc(=NCC(CO)c2ccc(F)cc2)[nH]1 c1(CC)cc(CC)[nH]c(=NCCCNC(C2(C)CCCC2(F)F)=O)n1 c1(C(=O)NCC(C)NC(c2csc(C(F)(F)C(F)(F)F)c2)=O)ccnn(C)c1=O c1(C(N2CC3C(CNC(C4(C#N)CCC4)=O)C3C2)=O)ccc2c(c1)CCOC2 C1(NC(C2CC(=O)NC2)=O)CCCCC1C(=O)NC1(c2ncc[nH]2)CC1 CCC(C#N)(CC)C(=O)NCC(C)(F)CNC(C1CCCNC1=O)=O c1(NC(C2CCN(C(C3CCC3(C)C)=O)C2)C)c(F)cc([N+](=O)[O-])cc1F C1(NC(CC(C)SC)=O)CC2(CCN(C(=O)CSc3ccc(F)cc3F)CC2)C1 N1(C(C(C)=C(C)C)=O)CCCC(O)(CNC(=O)C(C2(O)CCCC2)F)C1 N1(C(CC(CNC(C2(CC)CCOC2)=O)OC)=O)CCC2(CCCC2)C1 C(N=c1[nH]c(C#N)c(Cl)s1)C1C(NC(C2(C(C)(C)C)CCCC2)=O)CCC1 N1(C(CSCCC#N)=O)C(CNC(c2cccc3nonc23)=O)CC2COCC12 c1(OC)nccc(C(=O)NC(CNC(=O)Cc2cc(Cl)n(C)n2)C(C)C)c1F C1(CNC(C2CCC(C(F)(F)F)C2)=O)C2CN(C(=O)COc3ccsc3)CC12 Cc1cc2n(n1)CCN(C(C1CCN(C(c3cc(F)cc4cc[nH]c34)=O)C1)=O)C2 CC1C(C)N(C(c2cn(C)nc2Cl)=O)CCN1C(=O)C=Cc1c(F)cccc1F C1(NC(CCCOCC)=O)CCCN(C(=O)CC2CC(C(C)(C)C)C2)CC1 N1(C(c2cc(OC)ns2)=O)CCCCC(CNC(=O)CCC2CCC(=O)N2)C1 N1(C(CN(C2CC2CC(C)(C)C)C)=O)CCC(C)(CC(=O)N)C1.N1(CC)CC=CC1 Cc1cc(CNC(C2CC=CC(NC(=O)C(F)=C(C)C)C2)=O)ncn1 N(C1c2ccccc2CC1O)C(=O)NC1CC(NCc2c(C)ccc(C)c2)C1 c1(C(=O)NCC2(NC(CN3CCC(N(C)C)CC3)=O)CC2)cc(Cl)c(Cl)[nH]c1=N N1(C(=O)CC2CC3CCC2C3)CC2CCN(C(=O)Cc3cncc(F)c3)C2C1 C1(CNC(C2CCCC2(F)F)=O)CCN(C(c2cccc(F)c2F)=O)C12CCC2 N1(C(C(CC=CC)CC)=O)CCCN(C(=O)Cc2cnc(Cl)cc2C)C(C)C1 c1(N(CCCC)C)nc2ccsc2c(=NCC2(NC(C)CC)CCC2)[nH]1 S(=O)(=O)(CCC(=O)NCC(CNC(=O)CC1CCCC1C)OC)NC C1(C2CC2)(NC(c2c(C)oc(CO)c2)=O)CCN(C(C2C3CCCOC23)=O)C1 C#CC1COCCN1C(C1(CC)CCN(C(=O)CC2CC3(CC3)CO2)C1)=O CC(C)C(O)C(F)(F)C(=O)N(C1CCCC1)CCNC(=O)CC(C)C(F)(F)F c1(OC(c2csc(N3CCCCC3)n2)=O)nc(Br)ccc1Br c1(CN(C(=O)C(n2cc(C(N)=O)nn2)C)CCOCC)cncc(OC(C)C)c1 c1(CN2CCN(C(c3cccc(C(F)(F)F)n3)=O)CC2)cn2ccccc2n1 N1(C(C(CCCC)N(C)C)=O)CCn2ncc(N(C)C)c2C1 c1(C(=O)NC(CCOC)CNC(C2(OC)CC2)=O)cc(=O)n(C)c2ccccc12 C(C)(CNC(=O)CCCSc1cccnc1)(Cn1cccn1)NC(CC)=O Cc1cc(C(=O)NCC(C2CC2)NC(=O)C(C)C(F)(F)F)cc([N+](=O)[O-])c1O CCCC(CNC(=O)CC(=O)NC)C(=O)N1CCCN(CCO)CC1 C1(NC(CCOC2(C)CC2)=O)CC2CC1N(C(C1(C)CC1(C)C)=O)C2 c1(OC)cc(C(=O)NCC(C)NC(=O)CSCc2ccncc2)ccc1C#N c1(NC(CC(N)=O)C2CC2)[nH]c(=NCc2cn(C3CCC3)nn2)nc2scnc12 N1(C(CCCC(C)(F)F)=O)CCCC(C2CC2NC(C2CCC=CCCC2)=O)C1 N1(C(c2c(C)n3c(s2)cnc3)=O)CCOc2nccnc21 c1(OCC(=O)NC(CCNC(Cc2ccc(C)cc2)=O)C)ccc(Cl)c(Cl)c1 c1(C(=O)NCC23CC(C(N4CCC(CC)CC4)=O)(C2)C3)nc(Cl)ccc1Cl C(=O)(C(CC(F)F)N(C(=O)C=Cc1cncn1C)C)NCC(C(C)C)(C)C c1(C(c2nnnn2C2CCCC2)NCC=CC)ccnc(N2CCN(C)CC2)c1 S(=O)(=O)(c1c(Cl)cc(Cl)cc1[N+](=O)[O-])N1CC(COC)C(c2ccccc2)C1 c1(OC)ccc(F)c(C(=O)NC(C2CN(C(=O)C(C)CC(F)(F)F)C2)C)c1N c1(C(N2CCC(CNC(C(c3ccccc3)N(C)C)=O)C2)=O)sc(C#N)cc1Cl C1(OC(C)=O)CCCCC1(C)C.C12(CCN(C(=O)C(F)(F)F)C1)C(=O)NOC2 N1(C(CN(C(C)=O)C)=O)CC(CO)C2(C1)CN(C(c1c[nH]c3cccnc13)=O)C2 C#CC1CCCN1C(=O)CC1CCCN(C(c2cnsn2)=O)C1 Cc1ncc(Cl)cc1CC(=O)NC1CCCC1CNC(=O)C(C)Cn1cccn1 C(=O)(CCCCCF)NC1CCCC(CNC(CN(CC(C)(C)C)C)=O)C1 C1(NC(CC(=O)OCC)=O)CCN(C(=O)CC2CC=CC2)CC1C c1(-c2cn(CCCCNC(C3CCn4ccnc4C3)=O)nn2)cccc(Cl)c1Cl c1(C(N(C(C)CNC(=O)Cc2cnc(C)[nH]2)CC)=O)cc(C)cc(Cl)c1 c1(C(N2CC3C(N(C(CC(COC)OC)=O)C)C3C2)=O)nccc2[nH]ccc12 c1(OC)ccc(C(C)NC(=O)C(=O)N(C(C)(C)CCO)C)c(F)c1 N1(C(CC=CCC)=O)CCN(C(c2ccc(=O)n(C)n2)=O)C2CCCC12 C1(C(N2CCC(CCNC(CCCC#C)=O)CC2)=O)CCc2c[nH]nc2C1 c1(N(CC(=O)NCC(C)(CO)NC(C2CC23CCC3)=O)C)ccc(Cl)cc1 c1(OC)ccc(C2=NOC(C(C)NCc3cc(F)c(F)c(F)c3)C2)cc1 CCC1=NOC(NC(c2sc(-c3ccc(-c4ccc(C(C)=O)o4)cc3)nc2C)=O)C1 O=C(N=c1cc(CC2CCC2)[nH][nH]1)c1cc(F)ccc1OC(F)(F)F C1(OC)CN(C(=O)COC(c2c(Oc3ccsc3Cl)noc2C)=O)CCC1CO c1(-c2nncc(C(=O)NCC=C)c2)ccc2c(c1)OCO2 C#Cc1ccc(C(N2CC(F)CC2CC(=O)NCCCCc2ncc[nH]2)=O)o1 c1(C(N(C)C2CC2)=O)n[nH]c(C)c1[N+](=O)[O-].C(C(=O)NC1(C)CC1)NC(=O)OCC=C N1(C(C(CC)(C)C)=O)CCCC(C2CN(C(c3cc(S(N)(=O)=O)ccn3)=O)C2)C1 C(c1ccc(F)cc1)=CC(N1CCCC(CNC(c2n(C)cc(C)c2)=O)C1)=O N12CC(C(O)C1)NC(C)C2=O.N1(CC(=O)Nc2ccccn2)CCC(CO)CC1 c1(CC)ccc(C(N)=O)cn1.c12cscc1C(c1nnnn1C)N2 c1(C(N2CC(C(=O)C3CC3)(CNC(C3(C)CC3)=O)C2)=O)cccc(-n2cccc2)n1 C1(NC(CNS(CCOCC)(=O)=O)=O)CN(C(=O)CCSC(C)C)CC2(CCC2)C1 CCC(C)CCCCC(=O)NC(CC(=O)N1CCC(C)C1)C(C)C c1(C(N2CC(O)(CN(C(C(COC(C)=O)C)=O)C)C2)=O)ncc2ccccn12 Cc1cc(C(C)C(=O)NCC2CN(C(C3CSC3)=O)CCO2)cc(C)c1 c1(-c2c(C(N3C(CC(C)C)COCC3)=O)n[nH]c2)cn(C)c2cc(CO)ccc12 N1(C(C(C)=CC2CC2)=O)CC2(CCC2)CC1C(=O)N(C)CC1CCCC2CC12 C1(O)(C(N)=O)CCN(C(c2c[nH]nc2CCC(=O)C=Cc2cnccn2)=O)C1 CC1CN(C(=O)C(Cl)=CCl)CCCN1C(=O)CNC(=O)NC1CCCCC1 c1(OC)cccc(Cl)c1CN(CC(C)O)CCOC(=O)CCCc1ccccc1 c1(SCCS(=O)(=O)N(C)C)cccnc1CN1CCC1C1CCC1 N1(C(c2cc(Br)ccc2F)=O)CC2CC(C1)N(C(C1COC3(CCC3)C1)=O)C2 N1(CCCOC)CCN(CCN(C)CCc2c(C)noc2C)CC1 c1(C(=O)NCCCC(C)NC(=O)C(C)CO)cc(Cl)cnc1O C1(C(N2C(CNC(C(C=C=C)C)=O)CCCC2)=O)COC2(CCC2)CO1 C(=O)(C(C)CC(F)(F)F)NC(CNC(C(C(CC)O)C)=O)C c1(OC)ccc(F)c(C(=O)NC2CN(C(=O)CN3CCC(F)CC3)CC2O)c1 C(C)(C)(CCCC(=O)NCc1nnc(O)n1C)NC(C(CCCC)O)=O Cc1nn(CC(=O)NCC2(C)CCN2C(=O)CC2NC(=O)NC2=O)c(=O)n1C C(c1ccc(F)c(F)c1)=CC(=O)NC1CCC1NC(c1cnn(C(F)(F)F)c1)=O c1(CNC(CC2C(C)(C)COC2)=O)cc2n(n1)CCN(C(=O)CC1CC1(C)C)C2 CC(F)(F)CCCC(=O)NCC1CCCC1NC(C1(C2CCCCO2)CCC1)=O c12ccc3c(n1)N2CC3.c1(C(CN(CC(=O)OC)C)O)ccccc1 Cc1cnc2cc(C(N3CCC(NC(=O)CC(C)(C)C)C3C3CCC3)=O)nn2c1 C12(CNC(C=CCC)=O)CC(CNC(=O)C=CC(F)(F)F)(CN1C(C)=O)C2 CC1CC(C)N(Cc2c(F)cccc2Br)CCN1 C(N=c1[nH]c(=NCN2CCC(C(C)O)CC2)c2ccccc2[nH]1)C1(OC)CCC1 Cc1ncc(C(N2CC(NC(C3OCCCO3)=O)C2)=O)c(=N)[nH]1 N1(C(C2NC(=O)C(F)C2)=O)CCC2(CCN(C(=O)CS(N)(=O)=O)C2)C1 N1(C(C2CC(C)C2)=O)CCN(C(C2CN(S(N)(=O)=O)C2)=O)CC12CCC2 C1(NC(C(C)Cn2cccn2)=O)COCCC1CC(=O)Nc1cn(C2CC2)cn1 N1(C(C(=O)NC2CC2F)=O)CCS(=O)(=O)CCC1c1ccccc1 c1(CC(C(=O)NCCCN(C(C2CC2(C)C)=O)CC)O)ccccc1C(=O)O N1(C(COCC)=O)CC2COCC2(C(N2CC(CC)C(F)C2)=O)C1 C1(CNC(CC(C)OC)=O)CCC(C)(C)CN1C(c1ccc(=O)n(C2CC2)c1)=O C1(CNC(C(n2cnc(C#N)n2)CC)=O)CN(C(c2ns[nH]c2=O)=O)CC1O c1(CCC(=O)N(CCNC(C(C)OCC#C)=O)C2CC2)ccncc1 C1(C(N2CCC(NC(C=CC(=O)OCCCC)=O)C(C)C2)=O)CC12CCCCCC2 c1(C(=O)NC2(CNC(CCOCCOCC)=O)CCC2)ccn(C(C)C)c1C c1(C(N2CC(CNC(c3n(CC)ccn3)=O)(OC)C2)=O)ccc(N)c(O)c1 CCC1=NOC(CC(=O)NC2CCCC(NC(c3nc(O)sc3C)=O)C2)C1 c1(CC)ccccc1C1(NC(=O)CNC(=O)NCc2ccc(O)nc2)CC1 C1(C(=O)NC(C(O)CO)C2CC2)CCCN1C(C12CC(CO)(C1)C2)=O N1(C(C2C(CC)CCC2)=O)CC2CCC(C1)N2C(=O)CC(C)c1cccnc1 N1(C(c2sc(CC)c(C)c2)=O)CCCC2CN(C(=O)CC(C)(C)OC)CCC12 C=Cc1cncc(C(=O)NCC(CC(=O)NCC2(C#N)CCOCC2)OC)c1 C(c1ccccc1C#N)=CC(=O)NC(CN(C(CCC=C=C)=O)C)C C1(C2CCN(C(c3cnc(O)c4ccsc34)=O)CC2)(NC(=O)COCCF)CC1 C1(CNC(=O)Cc2ccc(O)nc2)CC2CCC(C1)N2C(=O)C(F)CC1CC1 CC1CCCC(C(=O)SCCNCC2CCNC2)C1.C1CN(C)CCOCCO1 c1(C(=O)NC(CNC(c2nn(C)c(Cl)c2Cl)=O)C2CC2)ccc2ncncc2c1 C1(C(=O)NC(C)C)CNC(=O)CN1C(c1ccon1)=O CC1C(C)N(C(C23CC(C)(C2)OC3(C)C)=O)CCN1C(c1cnc(C2CC2)nc1)=O C1(CN(C(c2[nH]cc(C)c2)=O)C)CCCN(C(c2csc(=N)[nH]2)=O)C1 C(=O)(C1OCCn2ccnc21)N1C(CCNC(Cc2ccn(C)n2)=O)CCC1 C1(CC(=O)N(C)CC2(C)CC2)(OC)CN(C(=O)C(C)N2CC(C)C2)C1 N1(C(C(C)(C)O)=O)CCC2CCN(C(C3(CCF)CC3)=O)CC2C1 C1(CSC)CN(C=O)CC12CC2.c1(OC)ccc(CNC(c2[nH]ccc2)=O)cc1 c1(OC)ccccc1SCC(=O)NC(C)(CNC(C1(C)CCOC1C)=O)C(C)C C(CCCCC(=O)NC1CCC(CNC(C23CCC(C2)OC3)=O)CC1)SC C(C(=O)N(CCCN(C(=O)C(C)N1CCCC1)C)C)(C(C)(C)C)OC C(=O)(CCCC(C)(F)F)NCC1CCCN(C(CCOCCCC)=O)C1 N1(C(COC)=O)CCC2(CCCCN(C(c3cc(Br)n[nH]3)=O)C2)C1 N1(C(=O)N(C(C)CCO)CCCCC2CCCC2)CCC(O)(C(=O)N(C)C)C1 Cn1cnc2c(C(=O)NCCC3CCC(NC(=O)CCC4CC4)C3)ccnc12 CC(CNC(=O)C(=O)NCc1ccc(C(C)C)c(C)n1)CC(F)(F)F C(=O)(CCC(C)S(C)(=O)=O)N1CCC(OC)(CNC(=O)C(C)(C)OC)C1 Cn1c(=O)n(C)c2cc(CCCNC3CC4CC4CC3C)ccc12 c1(C(N2CCC(NC(c3c(C)noc3Cl)=O)C2)=O)cccn(C(C)(C)C)c1=O c1(C(=O)NCC2N(C(CCC#C)=O)CCC2C)cc2ccncc2s1 c1(C(=O)NC2CC(NC(C3(C)CC(F)C3)=O)C2)cc2ncccc2o1 c1(CNC(C2C3CCCOC23)=O)cccc2cn[nH]c12 C1(CC(=O)NC2(C(=O)NCCOCC(=O)NC)CC2C)CCCCC1 c1(C(=O)NC(CNC(C2C(C)C2)=O)(C)C2CCC2)nnn2c1CCCCC2 c1(CC(=O)NC2(CNC(CCC=CC)=O)CCOC2)c(CC)noc1CC C=CCCCCCCCCC(=O)NC(C)CN(C(=O)CN(S(C)(=O)=O)C)C C(C(F)(F)Cn1cc(C)nn1)NC(C(C1CCC1)SC)=O.C(C(C)O)OC C(=O)(CC(O)C(C)C)N1CC(NC(C(c2ccccn2)C)=O)(CO)C1 C1(O)(CNC(C2C(C)N(C)CC2)=O)CCCN(C(c2cnn3ccsc23)=O)C1 N1(C(C(C2CCOCC2)OCC)=O)CCCC(NC(=O)CCCC#N)C1 C12(NC(C(CCC=C)NC(c3ccn(CCF)n3)=O)=O)CCC(C1)C(O)C2O c1(C(=O)NCCCN2CCN(C(CN(C)C)=O)CC2)cc(=N)[nH]cc1Br CC(C#N)C(=O)N(CC(c1cnn(C)c1)O)CCO C(C)(C)(CC(C)NC(=O)C(C)(c1cccs1)NC(=O)CCC1(C)CC1)OC O=C(Cc1nnc(-c2sc(Br)nc2Cl)o1)N=c1ccn2ncc(I)c2[nH]1 CCC(CC)C(C(=O)N(C1(CC(=O)NC2CCCCC2(C)C)CC1)C)OC C1(C(=O)NCCCN(C(=O)C(C)(C)c2cnco2)C)CCS1(=O)=O C12(CC)CCC(C(=O)NCC3CC(NC(c4cnc(N)cn4)=O)C3)(CO1)C2 c1(C(=O)NC2CCC(C)(CNC(C3(C=C)CCC3)=O)C2)cnc(N(C)C)c(Cl)c1 Cc1ncc(N)cc1C(=O)NCCNC(c1ncnc(C)c1C)=O N1(C(C=C(C)C2CC2)=O)CC(NC(=O)Cc2cc(C)on2)C(C(F)F)C1 c1(C(=O)NC2C(NC(C3(CCOC)CCC3)=O)CCC2)c(C)cccc1O C1(NC(C(COC(C)=O)C)=O)CCCC12CCN(C(C1CCC(NC)CC1)=O)CC2 N1(C(=O)OC(CC(C)C)C)CCCCC1CNC(=O)CCC(C)O C(CCCCC(=O)NC1(C(=O)NCC2CCCS2)CC1(C)C)=CC C12(C(=O)NCCC(C)(C)NC(c3cc[nH]c3)=O)CC(N=[N+]=[N-])C1C2 c12ccc(cc1)CCS2.C1(C)(C(=O)OCC)CN(C(c2[nH]cnc2C)=O)C1 C12(CNC(C(C=C)O)=O)COCCN1CCN(C(=O)COCCCC(C)C)C2 C1(NC(c2c(CC)ocn2)=O)CCCN(C(c2nc(OC)cc(OC)n2)=O)CC1 C1(CC(=O)NCCCc2nnc(C)o2)CC2(C1)CN(C(=O)OC(C)(C)C)C2.C(C)S C1(C(=O)NC(C(O)CO)C2CC2)(CC)CCCN(C(C2CCN(C)C(=O)C2)=O)C1 c1(C(=O)NCC(CCC(C)C)NC(=O)C2=C(Cl)CCCC2)coc(S(N)(=O)=O)c1 c1(C(=O)NCCN(C(c2cc(NC)ccc2F)=O)CC)nn(C)c2c1C(=O)CCC2 N1(CCSC2CC2)Cc2ccccc2C1.c12cncc(c1)NC(=O)C(=O)N2C c1(C(N(CCCOC(N(C)C)=O)C)=O)cccc(F)c1OC(F)F c1(C(N(CCNC(C2C(C(=O)OCC)CCO2)=O)C)=O)cccc2c1OCC2C C=CC1CN(C(=O)C(C2CCCCC2)O)CC1NC(c1cc(C)sc1C)=O C=CCCCCCCCC(=O)N1CCC(NC(c2n[nH]c(C)n2)=O)C(F)C1 c1(C(C(=O)NCC2(Cc3cn(CC(=O)O)nn3)CC2)O)ccc(F)c(Cl)c1 C(=O)(CC(CC1CC1)NC(=O)CC12CCCC1C2)NCC1CC(=C)C1 c1(C(=O)NC2CCC2CNC(C2CC(F)C2)=O)cc(F)c(C(F)F)c(F)c1 C1(CNC(C2CCCCCN2C(=O)C(O)C2CC2)=O)CC2(CCC2O)C1 c1(N(CC(C)(C)C(C)(C)C)C)cccc2c(CN(C)C)cccc12 C(CN=c1[nH]c(Cl)ncc1Br)Oc1c(OC)cc(Cl)cc1 N1(C(C(C)c2ccsc2)=O)CC(CO)(NC(=O)C(O)CC2CCOCC2)C1 C1(NC(=O)CC(F)(F)F)CN(c2ncc(F)cn2)CC2(CCOCC2)C1 c1(C(N2CC3CN(C(C(C)(C4CC4)OC)=O)CC3C2)=O)[nH]nc2c1COC2(C)C C1(C#C)(C(N(CCCC#C)C)=O)CN(C(C2CC2(F)Cl)=O)C1 CCCCC(=O)NC1CC(C(F)C(=O)NC2COCC2OCC)C1 Cc1cccc(NC(=O)C=CS(C)=O)c1CN=c1nc(CC2CCCC2)[nH]s1 CONC(=O)C(=O)NC1CN(C(=O)C(C)n2cccn2)CC1C(C)C c1(-c2n(C(C)C3CC3)nc(C(F)F)n2)cc(F)c2[nH]nnc2c1 C1(CNC(C2N(CC)CC2)=O)CC(C)(C)CN1C(=O)CSC(F)(F)F C12(c3nc(CNC(N4CC5CCC4C(O)C5)=O)sc3)CC3CC(CC(C3)C1)C2 c1(C(=O)NC(C2CC(NC(C3(CS(C)(=O)=O)CCC3)=O)C2)C)cncc(Cl)c1 Cc1cc(NC(=O)CCC2CC(NC(=O)C(C3CCOCC3)F)C2)cs1 c1(C(N2C(C)CC(NC(=O)CCC(C)(C)C)C2)=O)cc2sc(N(C)C)nc2s1 Cc1cc(-n2nc(-c3nccs3)nc2C2CC2(F)F)ccc1-n1cccn1 c1(CC(=O)NCC2(NC(C=CCCC)=O)CCC2)cc(F)cc(F)c1 N1(C(CNC(C2(C(F)F)CCC2)=O)=O)CCN(C(=O)CC2(O)CCC2)CC1 c1(C2C(C(=O)NC3(n4cc(C(CC)O)nn4)CC3)C2)ccc(Cl)c(F)c1F c1(C(=O)NC(C)CNC(c2ccc(OC(F)F)c(F)c2)=O)cnc2c(c1)CCC2 C12(NC(CS(=O)(=O)NC)=O)CCOCC1CN(C(c1cn3ccnc3s1)=O)C2 C1(NC(CNC(C2C(C)C2)=O)=O)CC2(C1)CN(C(c1c[nH]c(C(F)(F)F)c1)=O)C2 C1(NC(C=CC(CC)=CC)=O)CN(C(C2CN3CCCN2CC3)=O)CC2(CC2)C1 c1(C(=O)NC2CN(C(CCN(CCC)C)=O)CC(C)(C)C2)ccc2nn[nH]c2n1 C1(NC(C(C)(O)C2CC2)=O)CC2(CCCN(c3snc(Cl)c3C#N)C2)C1 c1(N2CCCC(CN(C)C)C2)nc2c(c(=NCC3CC(CO)CO3)[nH]1)COCC2 c1(C(=O)NC(C2CCOC2)CNC(c2c(C)nc(C)o2)=O)nccc(Cl)c1Cl c1(C(=O)NC2C3(CC(NC(c4cccs4)=O)C3)C2)cnn2c1S(=O)(=O)NCC2 c1(CC)nc(C)c(C(=O)NCC2(F)CC(NC(=O)CSC(C)(C)C)C2)c(C)n1 c1(C(N2C(CNC(c3ccc(F)cn3)=O)CC2)=O)n[nH]c2c1COC2 c1(OC)cc2cnc(C3CC3)nc2cc1CN1CCN2CCCCC2C1 c1(C(N2CCC(OCC(=O)NCC3CCN(C)CC3)C2)=O)cc(O)ccc1F CCC(=O)CCC(=O)NC1CC(CC(=O)N(CC(C)C)C(C)C)C1(C)C CC1CC(NC(=O)C(C)(C)N(C)C)CN1C(C1CCCN1S(C)(=O)=O)=O N1(C(C(CC)COC)=O)CCCCC(N(C)C(c2cc(Cl)c(Br)[nH]2)=O)C1 c1(CCNC(C(c2cn(C)nc2)NC(=O)CC2CC2(Cl)Cl)=O)ccc(O)cc1 C=CCC(F)(F)C(=O)NCCC1CC(CNC(c2cc(O)nc(O)c2)=O)C1 CC(F)(F)C(F)C(=O)NC(CC(N1CC2(CC(OC)C2)C1)=O)C1CCCC1 C(=O)(N=c1[nH]nc2[nH]ccnc1-2)c1ccc(-c2ccc(C)cc2C)cn1 C#Cc1ccccc1CC(N1CCC(C)(CNC(c2cccc(OC)n2)=O)C1)=O c1(NCCC2CCCN(C(c3c(CC)c(C)sc3)=O)C2)nnc(C)c(C)n1 c1(C(N2CCC(CCNC(C(C)C3CC3)=O)C2)=O)cccc(-c2nncn2C)c1 c1(C(=O)NCC23N(C(C(C)P(C)(C)=O)=O)C(CC2)CC3)cc2c[nH]cnc-2n1 c1(NC(C)=O)cncc(CC2CCCN2C(=O)Cc2nc(C3CC3)cs2)c1 C1(O)(C(=O)NC)CCN(C(C2CC23CCOC3)=O)CC1 c1(C(N2C3CCC2CN(Cc2cc(I)ccc2Br)C3)=O)cnc2ccccc2n1 N(C(=NCCC(C)N(C)C)N1CC(c2ccccc2)C2(CCC2)C1)C(CC)C C(C(=O)NCc1cn(C(C)C(=O)NC2(C(C)C)CCCC2)nn1)(C(C)(C)C)NC C1(NC(=O)CSc2ccc(Cl)cc2)CN(C(=O)C=CI)CCC1CO C1(C(=O)NOC2CCOC2)C(C2CC2)CCN1C(=O)CCCC(F)(F)F.O=C C(C1=CCN(C(c2c(C)[nH][nH]c2=N)=O)CC1)NC(C(COC)NC(C)=O)=O c1(C(=O)OC)cnc(N2CC3C(NC(C4CCCCC45CC5)=O)C3C2)cc1C Cc1cc(C)c(C(=O)NCC2CC(=O)N(CC3CC3)C2)c(C)c1 C(=O)(C1Cc2ccccc21)NC(CC=C)CNC(=O)Cn1cnc2c1CCCC2 C1(N(C(CCOCCC)=O)C)CN(C(c2cc(C3CC3)no2)=O)CC12CC2 C1(CN(C(C(C)CN(C)C)=O)C)CCCCN1C(c1cnn(C2CC2)c1)=O N1(C(C2N(C(C(CCC)F)=O)CCCC2)=O)CCn2nc(C)cc2C1 C1(C(N2CC(CNC(c3ccc(C(=O)OC)s3)=O)C2)=O)Cc2ccccc2CO1 Cc1ccc(C)c(C(=O)N(C(CNC(C2CC3CCC3C2)=O)C2CC2)C)c1C Cc1ncc2cc(C(N3CCN(C(C4CC4F)=O)C(C(C)C)C3)=O)c(O)nc2n1 N1(C(CC2(NC(c3c(C)nsc3)=O)CC2)=O)CCC(CC(C)O)CC1 c1(OC)cnc(C(N2CC(NC(=O)C(C)c3cncs3)C2)=O)cn1 c1(C(C)NC(C2(CNC(C(COC)N(C)C)=O)CCCC2)=O)ccccc1C C1(c2cn(CCCCCC#N)nn2)(NC(=O)NCCCCCC2CC2)CC12CCC2 N1(C(C(C)CC2CC2)=O)CC2(CCC2)CC1CN(C(=O)C=CC=C(Cl)Cl)C1CC1 c1(CNC(=O)NCC(c2cccnc2)C)ccc(-n2cncn2)cc1 N1(C(C2C(NC(C(N(C)C)NC(C)=O)=O)CC2)=O)CC(C)CCCC1C C1(C(N(CCCCN(C(=O)CC2CSCCS2)C)C)=O)CCC(C)(C)OC1 c1(OC)ccc(CNC(C2CCCCC2Nc2ncc(F)cn2)=O)cc1CCO Cn1cnc(CC(=O)N(CCCNC(C2CC23CCC3)=O)Cc2cccnc2)c1 C=C(C)C(CC(=O)NCCCSCC1(F)CCN(C(=O)CCC(=O)NC)C1)OCC Cc1noc(C)c1S(=O)(=O)N1CC2CC(C1)N(c1ncc3ccsc3n1)C2 C=CC1(C(N2CC(N3CCN(C(C4CC4C#N)=O)CC3)C2)=O)CCOCC1 c1(C(=O)NCC23CCC(CC2)N3C(=O)Cc2cccnc2)ccn2nnnc2c1 c1(CNC(=O)C(N2CCC(O)(c3ccc(Br)cc3)C2)=O)c[nH]c2cc(Cl)ccc12 C(=O)(CCC(=O)N(CC(C)NC(c1coc(N(C)C)n1)=O)CC)NCC C(CC(C(=O)NCCc1ccon1)NC(C1C=CCS1)=O)OC Cc1ccc(C(c2nnnn2C)NCC(O)CC(C)(C)C)nc1C C1CCN=C2C=C(C(F)=CN2)O1.C(=O)(NN1CCCC1)OC(C)(C)C CC(CC(=O)N1CCCCC(C)(F)C1)C(C)(C)NC(=O)C1=C(C#N)CCC1 c1(C(=O)NCC2C(NC(c3ncccc3Br)=O)C2)cc2c(nn1)CCCO2 c1(C(=O)NCC(CNC(c2n(CC=C)ccn2)=O)O)ccc(N(C)C)cc1 C1(C)(CNC(C(C)C2CCOC2)=O)CCN(C(C2CCN2C2CCCC2)=O)C1 C1(C(N2C(=O)CN(S(CCC)(=O)=O)C2=O)C)CCC2(CCOCC2)CO1 c1(NCC2(CO)C(C)CCC2)nccc(=NCc2cnn(-c3ccccc3)c2)[nH]1 c1(C(=O)NCCN(C(=O)Cn2cnc(=N)[nH]2)CCC)ncnc(C)c1C C(CCC(C)NC(=O)CCc1cnn(C)c1)NC(C1CC(CN(C)C)C1)=O C(C)(CCC(=O)N(C1CCN(C)CC1)C)NC(COC(CC)CC)=O C1(NC(c2cccc(C)n2)=O)CN(C(c2cc(O)ccc2C)=O)C2(CCOC2)C1 c1(CNCC(CN(C(=O)CC(C)C)C(C(=O)OC)C)(C)C)cc(Cl)cc(Cl)c1 C(C1Cc2ccccc21)NC(CC1C(NC(c2ccn(C)n2)=O)CCCC1)=O C1(C(=O)NC(CC(C)NC(c2c(C)nsc2)=O)C)CCCN(C(C)(C)C)C1=O c1(CC(=O)NCC2CCCC2NC(C2C3CCCOC23)=O)ccncc1Cl N1(C(=O)Nc2ccc(C)cc2)CCC2CN(C(c3cc[nH]c3)=O)CC12 Cc1ncn2ccc(C(=O)NC3CCN(C(c4ccc5cnnn5c4)=O)C3)cc12 n1(C2CC(N)C2)cc(-c2nccs2)nn1.C1C(=O)NCC1 C1(NC(=O)CSC(F)F)CC2CCC(C1)N2C(c1ccsc1C(F)F)=O c1(C(=O)NCC2C(NC(C(C)C3(O)CCC3)=O)CC2)ccc2n[nH]cc2n1 N1(C(c2cc(C)ns2)=O)CCCN(C(=O)COC2CCC(F)(F)CC2)C(CO)C1 CCCC(CCC)=CC(=O)NCCOCC(N1CCCC1c1cn[nH]c1)=O n1(CC)cccc1C(=O)NCC1CCCN1C(c1csc(C(C)=O)c1)=O n1(CC(=O)N(CC(CC)NC(c2cc(C)ccc2Cl)=O)C)c([N+](=O)[O-])cnc1C c1(C(CC)NC(=O)NCc2conc2C2CCCO2)csc(Cl)c1OC N1(C(C(C)C)=O)CCCC1CCNC(=O)Cc1n[nH]cc1Br Cn1c(C(=O)NCCCNC(=O)CC2CCC(=O)NC2=O)ccc1C#N N1(C(C(C=C)(C)O)=O)CCC2(CCCN(C(C3CC3C(=O)OC)=O)C2)CC1 N1(C(C(CN(CC)CC)F)=O)CCC(C)(CNC(=O)C(F)F)C1 N1(C(C(CNC(C(C=C)C)=O)C)=O)CCn2c(C)nnc2C1 C1(N2CCCC(C)(C(N(C(c3cscn3)C)C3CC3)=O)C2)CC2(CCNCC2)C1 c1(C(N2C(C)CN(C(=O)C3=CCCS3)CC2)=O)cc2ccc(F)cc2[nH]1 C=CC(CCC)CC(=O)NCCc1ocnc1CNC(c1cc(Cl)c([N+](=O)[O-])[nH]1)=O c1(-c2cn(C(CC)C)nn2)c(CCNC(c2oc(C)cc2C)=O)cccc1F n1(C2C(C)CC2)c(C2CC2c2ccccc2)csc1=Nc1ccnc(Cl)c1 C1(C(=O)NC2(CC=C)CN(C(c3ccncc3C)=O)C2)CC(=O)NC2CCCCC12 n1(CC)c(C(=O)NCC2(C)CC(OC)CN2C(C)=O)nc2ccccc12 CC1CCOCC1C(=O)NC1CC(CCNC(c2ccc(C#N)[nH]2)=O)C1 N1(C(C2(C(CC)(F)F)CC2)=O)CCCC(C)(NC(c2onc(Br)c2C)=O)C1 N1(C(C(c2cnn(C)c2)C)=O)CCCC(F)(CNC(C2(O)CCOC2)=O)CC1 N1(C(CCCOC)=O)CCCCCC1C1CCCN1C(=O)CC1CC(C)(C)CO1 N1(C(c2c(C)cn(C)c2)=O)CC2=C(C1)CN(C(=O)CCC(C)(C)NS(C)(=O)=O)C2 c1(C(=O)NCC2CCN(C(c3ccc(C(C)C)o3)=O)C2)ccc(Br)cc1N c1(CC)ncccc1C(=O)NC(CCSC)C(=O)NCC1(C)CC=CCC1 CCC(C)(C)C(=O)NC1CCCCC1CC(N1CCC(Cc2ccccc2)C1)=O Cc1c(CO)cccc1CNC(C1CCN(C(c2ccnn2C)=O)CC1)=O C=C1CCN(C(c2cn(C)c(C)n2)=O)C(C(N2CC(OC)CC(C)C2)=O)C1 C1(C(=O)NC(C(C)C)CCN(C)C(c2cccc(F)c2)=O)CCc2cncn2C1 c1(C(=O)NCC(C)(F)CNC(=O)C=C(Cl)Cl)ccc(=N)[nH]c1 CC1CCN(C(=O)NCCn2cc(Cl)cn2)CC1.N1(CC)CCOCC1=O Cc1cc(C#N)ccc1C(N1CC(C)(C)CC1C(=O)N(CC(C)C#N)C1CC1)=O c1(C(=O)NCCCN(CCCNC(=O)CC2C=CCC2)C)sccc1Br Cc1cc(C(=O)NC(C2(O)CN(C(=O)C(C)OCCC(C)C)C2)C)nnc1C Cc1ccc(C(=O)NCC2CC(NC(=O)C(C(C)C)N(C)C)C2)c(O)c1C c1(C(N(CCNC(=O)CCc2nnc(C)n2C)CC)=O)ccc2ncncc2c1 N1(C(c2ncc(C)c(Cl)c2)=O)CCCN(C(=O)C=CC2CCCO2)C(C)C1 c1(NC(=O)NCC#C)ccc(Cl)c(C(N2CC(c3ccsc3)C2)=O)c1.C1CN1 CN1C(=O)CCCC1C(N1CCC(NC(=O)CC2CCCSC2)CC1)=O c1(C(N2C(CN(C(=O)C3=CCCC3)C)CCC2)=O)ccnc(F)c1N N1(C(c2cccc(C)c2C)=O)CCC2CCCC12C(N1CCC12CCSCC2)=O CC1CN(C(c2ccccc2-n2cc(C3CC(=O)C3)nn2)=O)CCCO1 c1(C2C(C(N(CC(CN(C(=O)CSCC(N)=O)C)O)C)=O)C2)ccn(C)n1 C1(C(NOCCOCC#C)=O)CC(NC(=O)Cn2cnnc2O)C1(C)C C123COC(C1)(C2)CNC(=O)C3.C(N=c1nc[nH]s1)C1(F)CC(OC)C1 C1(Nc2cnc(Br)c(C)n2)CC2(C1)CN(C(c1ccc(COC)cc1)=O)C2 C1(NC(C(C)N(CC)CC)=O)CCCC(NC(=O)CSCc2cccnc2)C1 c1(N(C2CCNCC2)Cc2c3ccc(C)cc3[nH]c2)ncnc2[nH]cc(C#N)c12 N(C(=NCCCF)N1CCC(O)CC1)CC1CCCN(C(=O)NCC)C1 C(C)(C(=O)C(CNNC(C(=O)N(CC(F)Cl)C)c1ccco1)=O)N(CCC)C C1(NC(=O)C2=CCCC2)CCCC2CN(C(C3CCc4ccccc4C3)=O)CC12 n1(CC(=O)N(CCNC(c2scc(C)c2)=O)C)cc(C#N)cn1 c1(C(N2CCC(N(C(=O)CC3(C(F)(F)F)CC3)C)C2)=O)cccc(C(F)F)c1F N1(C(=O)C#CC2CC2)CC2C3CCC(C2C1)N(C(c1ccsc1C(F)F)=O)C3 c1(NC(CN2C(C)CCC2)=O)ccccc1CNCC(C)(C)CCO c1(OC(C(C)CNC(=S)Nc2ccccc2)=O)ccc(Br)cc1 C(C)(C)(CC#Cc1ccccc1)N(C1CC1)Cc1cn(CCC)nn1 c1(CSC)ccc(C(=O)NCC(C2CCC2)NC(C2(N(C)C)CCCCC2)=O)cc1 CC(CCCC(=O)NCC1([Si](C)(C)C)CC1)NC(C1CC(F)(F)C1)=O C(C(=O)NCC1CCN1C(=O)OC(C)(C)C)(C(C)O)N(c1ccnn1C1CC1)C Cc1ccnc(NC(=O)NC(C)CC(C)N)c1F CC1CCN(C(=O)CNC2CCCC2)C(CNC(c2cnn3c2SCC3)=O)C1 C1(C(=O)NC(CCOC)CO)CC(C)CN1C(c1cc(C)c(C)o1)=O C(CCC(C(=O)N1CCC(C(F)(F)F)C1)NC(C1CN(C(C)C)C1)=O)OC c1(C(CC)C)cc(C(=O)NC2C=CCN(Cc3cn(CC)nn3)C2)cc(C)c1 Cc1c(C(=O)NCCCNC(c2ncc(Br)cc2O)=O)cccc1F c1(OC)c(C)csc1C(N1CCCC1C(C)NCc1ncccc1C(F)(F)F)=O c1(CN(C)CC2CCN(C(=O)Cc3ccc(F)cn3)CC2)cc(F)c(F)cc1F C(=O)(CCCCCC(C)(C)C)NC(C1CCCN(C(c2cn(C3CC3)cn2)=O)C1)C C(C)(c1ccco1)=CC(=O)N(C)CC1CCN(C(C2(COC)CC=CC2)=O)C1 C12(C(N(C3CCC(O)C3O)C)=O)CC(CO)(CN1C(C1CC1(F)F)=O)C2 c1(OC)ccc2c(CNC(=O)COCc3ccnc(OC)c3)csc2c1 C1(C(=O)NCCCC(CC)C)CN(C(=O)CCC2CCC(=O)C2)CC1(C)C CC(C)(C)C(O)C(=O)N1CCC(CCNC(c2ccc(Cl)nc2F)=O)C1 n1(CC)c(C)nn(CC(=O)NC2CCC(NC(=O)C(C)CC(C)(F)F)C2)c1=O CC(C)CCC(C)N(C(=O)C(O)C1CN(C(=O)Cn2cc(CN(C)C)nn2)C1)C CN1CC(CC(=O)NCC(O)CNC(C2CC2C(F)(F)F)=O)c2ccccc21 c1(N2CCC(C(C)NC(=O)CC3CC3)CC2)nc2ccccc2s1 N1(C(c2nc(OCC)oc2)=O)CCCN(C(C2CN(CP(C)(C)=O)C2)=O)C(C)C1 Cc1c(C(=O)Nc2ccc(C(=O)Nc3cnc(Br)c(Br)n3)nc2)cncc1Br Cc1cc(Cl)cc2cc(C(=O)NC(CNC(C3CCN3C(C)(C)C)=O)CO)[nH]c12 N1(C(=O)NCCc2ccc3c[nH]nc3c2)CCOCCC12CCC2 N1(C(CCOC)=O)CCC2(CC1)CCN(C(C1CC1C(=O)NC1(C)CC1)=O)CC2 c1(COC)ccc(C(=O)NCC2CC2NC(C2(C)COCCO2)=O)cc1 C#CCCCCC(=O)NC(C)CNC(=O)C(c1ccc(F)c(Cl)c1)C c1(C(C(=O)NC2CC(C)(NC(CCc3cc(C)no3)=O)C2)OC)ccccc1C CC1CC(C(=O)NCCSC(F)F)N(C(c2ccc(Cl)o2)=O)C1 c1(C(=O)NC2CN(C(c3cc(C)c(C)nn3)=O)CC(F)C2)cccc2nccn12 c1(OC(C(C(=O)OC(C)(C)C)NC(=O)OCC)=O)cc(Cl)c(F)cc1C C1(CNC(C(C2CCOC2)OC)=O)CCCCN(C2CC3CC2CN3C(C)=O)C1 CC(CC(F)F)C(=O)NC1CCC(CC(=O)Nc2cncc(C3CC3)c2)C1 c1(OC)ccc(CC(=O)NC2CCN(C(=O)CSc3nc[nH]n3)C2C)nc1 N1(C(CCCCNC(C)=O)=O)CC2CN(C(c3cccs3)=O)CCC12 C(CC)(CC)(CCNC(C(C)OCCC=C)=O)NC(=O)C(C1CC(F)(F)C1)OC N1(CC(=O)NCCOC(CC)C)CCN(C(c2nc(C)sc2C)=O)CC1 C(=O)(C(C)C(C)S(C)(=O)=O)NC(C)CCNC(c1ccc(C(F)(F)F)s1)=O n1(CC(=O)NCC(CNC(C(CC)(C)CC)=O)(C)F)ccc2ccccc12 CC(C)(CC(F)(F)F)C(=O)NC1CCCCC1NC(c1c(Cl)ccc(O)c1N)=O c1(C(=O)OC)ccc2c(c1)nc(O)n2Cc1cn(C)nn1 C12(n3cccn3)CCN(CC1)C2.c1(CN(C)C)cccc(O)n1 N1(C(c2c(C)nc(C)o2)=O)CCN(C(=O)C(C)C2CCC2)C(C)C1 C=C(Cl)CC(C(=O)NC1CN(C)CC1(C)C)NC(C1COC(=O)N1)=O C(C(=O)NC(C)(C)CCNC(C1(N2CCCCC2)CCCCC1)=O)(C(C)C)SC N1(C(C(C)OCC(C)C)=O)CCCC1C(=O)NC1CC2CC2C1 Cc1c(Cl)ccc(C(=O)NCC2C3CN(C(=O)Cn4ncnn4)CC23)c1Cl c1(N(CC2=CCSC2)C)nc(N2CCN(C(C)(C)C)CC2)nc2c1CC(C)CC2 C1(Nc2c(Cl)nc(OC)c(Br)c2)COc2ccc(C)cc2C1 N1(C(C(N2CCC(O)CC2)C)=O)CCN(C(=O)Cc2cn[nH]c2)CC(C)(C)C1 C1(CN(C(=O)C=Cc2nnn(C)n2)C)CCCN(C(=O)CCn2cnnn2)C1 C1(C(=O)NCC(C2(O)CN(C(C3CS(=O)(=O)C3)=O)C2)(C)C)CC2CC2C1 Cc1ccn(C(C)(C)C(=O)NC(CO)C(C)NC(c2cncn2C)=O)n1 c1(CCC(=O)N(C(C(=O)N(C(C)C(=O)NC)CC#C)C)C)cnc(O)[nH]1 N1(C(c2n[nH]c(C)c2O)=O)CC(O)C(O)C1CNC(=O)CCCN1CCOC1=O c1(C(=O)OC)cc(CN2CC(C(=O)OC)(CN3CCOCC3CO)C2)ccc1O CC1=NOC(C)(C(=O)NC(c2nocc2C(=O)NCC2CCCC2CF)C)C1 c1(C(=O)NCCN(C(C2CC(SC)C2)=O)C)cnc(C2CCC2)o1 C1(C(=O)NCCOc2ccccn2)CC2CCC1N2C(c1cccc(=O)n1O)=O Cn1ncc2c1CCCN(Cc1nc(-c3ccncc3)no1)C2 c1(C(=O)NCC=CC(=O)NCC2(CO)CCN(C)C2)cc(O)ncc1F N1(C(CC2CCC(=O)NC2)=O)CCC2(CC1)CN(C(C1CCCCS1(=O)=O)=O)C2 c1(C(=O)OC)cc(=NCC(C2CC2)NC(=O)Cc2c(C)cccc2C)[nH]c(C)n1 N1(C(C(C)CS(C)(=O)=O)=O)CCC2CCN(C(C34CCOC(C)(C3)C4)=O)CC12 Cc1cccc2c1OC(C(N1CC3CC3(CNC(=O)C(C(C)C)N(C)C)C1)=O)C2 N1(C(C(COC)O)=O)CC2CC(C1)CN(C(C1CCN1C(=O)OC(C)(C)C)=O)C2 c1(OC)cccc(O)c1C(=O)NCC(C)(C(C)C)NC(C1CCCC(C)(C)C1)=O C1(NC(CCCC#C)=O)CC2CC(C1)N(C(=O)Cc1c(C)ncnc1C)C2 c1(C(N2CC(CNC(CSCCN(C)C)=O)OCC2)=O)cncc2cnccc12 c1(CNC2CC(C(=O)Nc3ccc(C)c(O)c3)C2)c(F)ccc(O)c1F C1(C(C)C)CCCN1C(=O)CC1CCCN1C(c1cncs1)=O C1(N(C(=O)Cc2ccsn2)C)COC2CN(C(=O)Cn3ccnn3)CC12 C1(CC(N2C(CNC(Cc3scc(C)c3)=O)CC(F)C2)=O)CCCC(C)(C)C1 C1(C(C)NC(=O)Nc2ccc(-c3cccc(O)c3F)cn2)Cc2ccccc2O1 C1(C)(COC)CC(NC(c2cnc[nH]2)=O)CN1C(c1nc(C)ccc1OC)=O c1(SC)ncc(C#N)c(N2CC3CN(Cc4cc(Cl)sc4Cl)CC23)n1 C1(C(=O)NCCOCCCNC(c2cnsn2)=O)CC(n2cnnc2)C1 N1(C(C2CC(=O)OC2)=O)CC2CN(C(c3ccc(OC(F)F)nc3)=O)CC12 C1(CC(N2C(C(=O)NC)CC2)=O)CCCC(NC(=O)CC(C)(C)C)C1 N1(C(C2C(OCC)C2C)=O)CCOC2(CCN(C(=O)C=CC(C)(C)SC)C2)C1 c1(NC(CC(C)OC)=O)sc2c(c1C(N1CCC3(CC3)C1)=O)CCCC2 c1(C(=O)NCc2c(NC(C3(CCO)CC3)=O)nns2)n[nH]c2c1COC2 Cn1nnc2cc(C(N3CC4CC(NC(C5(CN(C)C)CC5)=O)C3C4)=O)cnc12 C(c1cccc(F)c1Cl)=CC(=O)NC1CCN(C(C=C(C)Cl)=O)CC1O c1(C(=O)NC(C(C)(C)NC(C2(SCC)CC2)=O)C)cc(F)cc2ccncc12 c1(OCC)cccc(O)c1C(N1CCC(N(C)C(c2n[nH]c(C)c2C)=O)C1)=O N1(CC(N2CC(N(C(c3ccc(CNC(C)=O)o3)=O)CC)C2)=O)CCOCC1=O N1(C(c2c(CC)con2)=O)CCC(C)(C)C(CNC(=O)C(CC)CC(F)F)C1 C1(N(C(c2c(C)nns2)=O)C)CCCN(C(=O)C(CO)NC(N)=O)CC1 C#CC1CC2(CC(C(N3CCN(C(c4occc4Br)=O)C(CC)C3)=O)C2)C1 C1(F)(C(N(CCCOCCNC(=O)CC2(C)CC2F)C)=O)CCCC1 Cc1cc(C(N2CCC(NC(=O)CSc3c(C)n[nH]c3C)C(O)C2)=O)cc(C)c1 C(C(CC1CCCC1)CO)N(C(C(C)O)c1ccco1)Cc1cccs1 C1(C(N(C2CCC(NC(=O)C(=O)NCC(F)F)C2)C)=O)CSC(c2ccccc2)=N1 c1(NC(c2cccc(Br)c2)CC)ccncc1S(=O)(=O)NC(C1CCCO1)CO CCC(C)CCCC(=O)N1CC2CCN(C(=O)CN3CCS(=O)(=O)CC3)C2C1 Cc1cc2nccnc2cc1C(N1CCN(C(=O)CC2=CCCC2)CC1CO)=O C1(C(=O)NCC2CC(C)N(C(C3CC3(Cl)Cl)=O)C2)CCC2(CC1)N=N2 Cc1ccc(OCC(=O)NCC(F)CNC(C2CC(C)CCC2C(C)C)=O)cc1C C(=O)(C1=C(Cl)CCOC1)N1C(C)CCC(CNC(=O)C=CCN2CCOCC2)C1 N1(C(C(C)SC)=O)CCC(NC(=O)C2CC2)CC1C.C12CCCN1CCNC(=O)C2 N1(C(CC(C)(C)OC)=O)CC2CCCC2(CNC(c2cncc(N)c2)=O)C1 N1(C(CC(CN(C)C)O)=O)CCCC(CNC(=O)Cn2nnc(=O)[nH]2)CC1 C12(C(=O)NCC=CC(N3CC(C)N(CC#N)CC3)=O)CC3CC(C1)CC(CO)(C3)C2 C(c1ccc(F)cc1)=CC(=O)NCCC(C)N(C)C(C1CCC(O)CC1)=O CCC(F)(F)CC(=O)NC(CC(=O)N(C)CCc1cccs1)C(F)F N#Cc1cncnc1C(=O)NCC1CC(F)(F)CN1C(=O)CCCC1CCOCC1 C1(CCNC(C2(OC)CCC2)=O)CN(C(=O)CCOC2CC2)CC1C Cc1csc(C=CC(N2CC(NC(=O)CCS(C)=O)CC2C(N)=O)=O)n1 C1(NC(CC2(NC(CC3CC(=C)C3)=O)CC2)=O)CCCCC1N=[N+]=[N-] C1(C)(CNC(C(CC)F)=O)CCN(C(=O)Cc2ncc(Cl)s2)CC1 CC1(C)CN(C(c2ccc(CO)nc2)=O)CCC1NC(c1cnn[nH]1)=O C12(NC(=O)C3=CCCCC3)CCCC1N(C(=O)CC1C=CCC1)CC2 N12CCC(C1)C(F)C(=O)N(C(c1cn[nH]c1)C)CC2=O.CC(C)COC c1(Cc2nc(C3CCS(=O)(=O)C3)on2)ccc(O)c(F)c1F c1(C(=O)NCC2CN(C(c3cnns3)=O)CC2O)ccc(=O)n2c1CCCC2 c1(C(=O)NCCC(C)NC(c2ccc(C3CCC3)nc2)=O)cc(F)c(N)cc1F Cc1[nH]c(=NC2CC(CNC(=O)C(F)(F)c3ccccc3)C2)ccc1C#N c1(C(C)NC(=O)Nc2ccc3cnn(C(F)F)c3c2)cccc2cccnc12 c1(OCC(N2CCC(CNC(=O)CCCF)C2)=O)ccc(F)cc1O C1(CNC(C2C(OC)C2)=O)(CO)CC12CCN(C(=O)CN1CC3CC3C1)CC2 O=C1CCc2cc(S(=O)(=O)N3CCc4c(O)nc(O)nc4C3)ccc2N1 C=C(Cl)CCC(=O)NC(C(=O)N(C1CCNC1=O)C)C(C)C CN1CCC(C(N2CCCCC2CNC(c2ccnn2CC(F)(F)F)=O)=O)CC1 c1(CC#N)ccc(C(=O)NCC(CNC(c2ccnc(C3CC3)n2)=O)CO)cc1 c1(N2CC(n3ncc(N(c4ncc(C)c(C)n4)C(C)=O)c3)C2)ncnc2sccc12 c1(SC)ccc(C(=O)N(CC(C)O)CCNC(c2cnnc(C)c2)=O)cc1 C1(NC(C(CCC)N(C)C)=O)CC2CN(C(c3ccc(C(N)=O)o3)=O)CC2C1 C(c1ccc(F)cc1F)=CC(=O)NC(C)CCNC(=O)Cc1cc(C2CC2)no1 C1(C(C)C)CN(C(=O)C=CC2CCOC2)CCN1C(c1ccc(Cl)s1)=O CCC(CC)C(=O)NC1(C)CC(NC(C2CCN(c3ccncn3)CC2)=O)C1 Cc1cc(-c2cn(CCN(C)C(CC(C)O)=O)nn2)oc1Br c1(CC)csc(CN2CC(O)C2)n1.C1(Cc2nccn2C(C)C)CCNC1=O c1(CC(=O)NCC2CCN(C(C3SCCS3)=O)C2)coc2cc3c(cc12)CCC3 Cc1coc2ccc(C(=O)NCC3COCCN3C(C3C(C)C3(F)F)=O)cc12 O=C1CCCC(C(N2CCC(NC(C3(F)CC=CCC3)=O)CC2)=O)N1 c1(C(N2CCN(C(C(CCC)C)=O)C(CC(F)F)C2)=O)ccc(C)c([N+](=O)[O-])c1 c1(CC)ccc(C(=O)NCCC2(O)CN(C(c3nnn(C)c3CC)=O)C2)c(C)n1 c1(C(=O)NC2(CN(C(C(C)OCC)=O)C)CC2)cc(O)cc(Cl)c1Br c1(C(=O)NCCC2(OC)CN(C(=O)C(O)C3CCC3)C2)nnc2ccccc2n1 C1(C#N)(C(=O)NC2(C)CCN(C(c3n(CC)ncc3)=O)C2)CCN(C)C1 C1(CC)CCC(C)(C)OC1.C12OCCC1C(=O)NC1CN(C1)C2=O Cc1nc[nH]c(=NCC2C3CN(C(c4nc(Cl)c(Cl)s4)=O)CC23)c1C(N)=O N12CCC(CO)(CC1)CC2=O.C(C(O)C(C)C)OC.C1(CCOC)CC(NC=O)C1 N1(C(C)C)CCCC1C(=O)NC1CC(NC(c2cnc(C(C)(C)C)s2)=O)C1 C1(CCC(=O)NC2CC(CNC(C(C)OCCC=C)=O)C2)CCC(=O)NC1 C(=O)(CC(C)C(C)(C)C)N1CC(NC(c2c(Cl)cnc(C)n2)=O)C(F)CC1 C1(C(=O)NCc2ccnc(Br)c2F)CN(Cc2cccc(O)c2Br)CCC1(F)F N1(C(C2(CCN(C)C)CC2)=O)CC(NC(=O)C=CC2CC2)CC2(CCC2)C1 N1(C(Cc2ccn(CC(C)C)n2)=O)CC2C(CNC(=O)Cc3scnc3C)C2C1 Cc1cc(C(=O)NCC=CCNC(=O)CCCCN(C)C)cc(C)c1OC(F)F n1(CCC(N2CC3C(CNC(C(C)SCC)=O)C3C2)=O)cc[nH]c(=O)c1=O C1(CCNC(=O)CO)CSCCN1C(=O)CCN1C(=O)CCC1=O Cc1nc2c(o1)CCN(C(=O)C(C)(C)C1CCN(C(C3CC3(F)Cl)=O)C1)C2 c1(CC)nccnc1C(=O)NCCC(C(C)C)NC(c1nn(C)cc1COC)=O C1(NC(CN2C(C)CC2)=O)CCC(C)(C)CC1CNC(=O)CCc1csc(=N)[nH]1 C1(NC(C2OCCN(C)C2)=O)CCCN(C(=O)CCc2cnn(C)c2)CC1 c1(C(N(CCN(C(=O)CCC2CC2C)CC)CC)=O)cc2ccccc2s1 c1(SC(C)C(=O)NCCC2(NC(=O)CCCCCF)CCC2)nc2ccccc2s1 c1(OC(C)C)cc(C(N2CC(NC(=O)C#CC(C)(C)C)C(F)C2)=O)cc(Br)c1 c1(C(=O)NCC(C)(C(C)C)NC(c2ccc(OC)o2)=O)cc(F)c(F)cc1F CC1(NC(=O)CCCCCNC(c2cncn2C2CC2)=O)CCCCCC1 c1(C(N2CCN(C(C)C)C(C)C2)C(=O)NCC)cc2cccc(Cl)c2o1 C1(NC(CSc2ccc(C)cc2)=O)C2CCN(C(C3CC4CCC3CC4)=O)CC12 N1(C(C(C)CN(C)C(C2CC(Cl)(Cl)C2)=O)=O)CCC(CC2CC2)CC1 CP(C)(=O)c1cnn(CC(=O)NC2CCN(C(=O)OCCCCl)CC2)c1 c1(C(=O)NC(CC)CN(C)C(c2ncc(C(F)F)s2)=O)cncn(C)c1=O N1(C(CC2CC(=C)C2)=O)CC2CC1CC2CNC(c1cccnc1S)=O C12(CNC(=NCCC)NCC(C)C(=O)OC)CC(CO)(C1)OC21CCC1 c1(C(N(CCOCCN(C(C2C(OC)C2)=O)C)C)=O)c[nH]nc1-c1cnn(C)c1 C1(NC(C2(C(C)NC(C3CCCCO3)=O)CC2)=O)CC=CC(O)C1 C#CC1(C)CCCN(C(C2CC(CNC(=O)C=C(C)COC)C2)=O)C1 C12(NC(=O)COCC(F)(F)F)CC1CN(C(=O)Cn1ccc(C3CC3)n1)C2 C1(NC(C(C)SCC)=O)CN(C(c2ccc(C(C)(C)C)o2)=O)CC1C(F)F C1(C(=O)NC(CCOC)CNC(c2ccsc2C(F)(F)F)=O)CC2(CCC2)C1 N1(C(c2ccc(OC)[nH]2)=O)CCCC(C2CCCN(C(=O)C3=C(C)OCC3)C2)C1 C(=O)(C(C)(C)CCNC(=O)CC1CC1(C)C)N1CCC(NC(CC)=O)C1 c1(CN(CCC)CCN(c2ncn(C)n2)CC)ccc(-c2ccccc2CC)cc1 c1(C2(CC(=O)NC3CC3COCC)CC2)c(C)cccc1C.C12CC(C1)NC2=O CC(C)(C(=O)N1CCN(c2ccc(C(=O)NCC(C)(C)CCO)cn2)CC1)C(F)F C(=O)(C(CC(C)(C)C)OC)Nc1ccc(NC(C(C)NC(CC)=O)=O)cc1C C(=O)(C(C)(CO)OC)NC1CC(C)(C(=O)NCCOC(CC)CC)C1 C1(CNC(CC(C)OC)=O)CN(C(c2cnn(C)c2F)=O)CC2(CCC2)O1 Cc1ccc(NC(=O)COC(F)F)c(C)c1.C1(C)CCNC(=O)CCN1C C1(C)(C(=O)NCCCC(C)NC(C23COCC(C2)C3)=O)CCN(C)C1=O C(=O)(C(CN(C)C)C(C)C)Nc1c(C(N2CCN(C(C#C)C)CC2)=O)nco1 C=C(C)CC(C(=O)N(C1CCCC(C)(C)C1)C)NC(=O)CCc1csnn1 CCCC(CCCNC(c1nc(C)sc1C)=O)NC(c1ccc(C)cc1Cl)=O C(=O)(CC(C(F)(F)F)NC(c1ccc2cccnn12)=O)NC(CC(C)O)C(N)=O C(=O)(C(O)C(F)(F)F)NCC(C1CCN(C(=O)C=Cc2ccoc2)CC1)(C)O C1(OCC)COCCC1N=c1[nH]c(N2C3C=CCC2CCC3)nc2c1SCC2 c1(CCNC(N2CCC(CC3CC3)C2)=O)cn(CC2CCCO2)nn1 C1(C(=O)NCC(CNC(C2NC(=O)C(F)C2)=O)CO)CC2(C1)CC(O)C2 N1(C(c2c(NC3(C)CCCC3)cccc2)C#N)CCCN(c2ccccc2)CC1 c1(CC)cc(CNC(C2(C(=O)N(CCC(=O)N(C)C)C)CCCO2)=O)n[nH]1 N1(C(CC2(CC)CC2)=O)CC(OC)CC1CCNC(=O)C(F)(F)c1csc(=N)[nH]1 C(=O)(CC(C)C(=O)NC1(C)CC(C(N2CC(OC(F)F)C2)=O)C1)OC C1(NC(=O)CCC2CCCC2)CCN(CCCc2cc(CN)c[nH]2)C1.C(=O)C1CC1 CCCCC(CC)CCC(CNC(=O)NCc1cccc(-n2nncc2C)c1)CC S(=O)(=O)(c1cccc(F)c1)NC12CCC(NC(c3cccc(CO)c3)=O)(CC1)C2 Cc1ccc(OCCC(=O)NCC(C)NC(c2cnn(C(C)(C)C)c2Cl)=O)cc1 CCC(C)C(C(=O)NCCc1ocnc1CNC(=O)CN1CC2CC2C1)OC N1(C(c2ccn(C(C)(C)C)n2)=O)CCC(C2CCN(C(C3CC3Cl)=O)CC2)C1 c1(OCC)ccc(C(=O)N(C)CCN(C(=O)C(C)Cn2ccnc2)C)c(F)c1F CC1(C)CC(NC(c2coc(CNC(C3CCC3C(C)(C)C)=O)n2)=O)CO1 Cc1cnc(C(=O)Nc2ccc(C(=O)NCc3ccc(O)c(Cl)c3)cn2)c(Br)c1 N1(C(C(OC)OC)=O)CCCC2(NC(c3cccc(C)n3)=O)CC2C1 c1(C(=O)NCC(CNC(C(c2ccccc2)C)=O)(C)O)ccc2ccoc2c1 N1(C(C(c2n(C)cnc2)O)=O)CC(NC(c2coc(Cl)n2)=O)C(O)C1 c1(C(N(CC(CC)NC(C2COCCN2CC(F)F)=O)C)=O)cncc(CO)c1 C1(C(=O)NCCC(=O)NCCC)CCN(C(=O)Cn2cncn2)CC1(C)C c1(C(=O)NC2CC3CC(NC(C4CS(=O)(=O)C4)=O)C3C2)cc2c(cn1)OCCO2 c1(C(=O)NC2(CN(C(C(CCC)COCC)=O)C)CC2)cnc2cc[nH]c2c1 c1(CC)c(C(N2CC(NC(=O)C3CC3)C(NC(=O)COC)C2)=O)cnn1CC O(C=CC(=O)NC(C)CC(C)NC(=O)CN1CCC(C)C1)CC C12(NC(c3csc(C(F)(F)F)n3)=O)CCC(CNC(C3CCSC3)=O)(CC1)OC2 c1(C(N2CCC(NC(c3c(SC)scc3)=O)C(C)C2)=O)cc2c(s1)CN(C)CC2 CC1CC(F)(F)CCN1C(=O)CC(C)(C1CC1)NC(c1ncnc(O)c1F)=O c1(C(N(CCCC(=O)NC2(CC=C)CCOC2)C)=O)ccc(F)cn1 C(C(C(=O)N(CCC(=O)N1CCC(OC)C12CCC2)OC)OC)OC c1(CN2CCC(CC(=O)NC)CC2)ccc2c(c1)CNC2.n12cc(nn1)C2 C1(CN(C(C2CNC(=O)C2)=O)CC)CCN(C(C2CCC2C)=O)CC1 c1(NC(C2(COC)CC2)=O)ncc(CN(C(=O)C2CC2)C)cn1.C1(=O)CN1 S(=O)(=O)(c1cccs1)NC(C)C(N1CC(NC(=O)CC2C=CCC2)C(O)C1)=O c1(CNC(C2N(C(C(=O)N(C)C)=O)CC(F)C2)=O)ccc(=O)n(C)c1 C(C(C)(C)CC(=O)NCc1cccc(F)c1F)NC(c1cn(C)nn1)=O c1(CC)cccc(C(=O)NC(C)CNC(c2cn(C(C)(C)C)nn2)=O)c1 c1(C(N2C(C(=O)NC(c3cccc(O)c3)C3CC3)CCC2)=O)ccc(F)cc1 C1(CC(N2C(CN(C(CCC(C)C)=O)C)COCC2)=O)CCCCC12CC2 N1(C(C(C)O)=O)C2CCCC1CN(C(C1(C#N)CC13CCCC3)=O)C2 C1(CNC(C2(C=C)CC2)=O)CC12CCN(C(c1ccc(C(C)(F)F)cc1)=O)CC2 CN=C(NCCc1cnn(-c2ccccc2)c1)NCC(C)(C)C1CC1 c1(OCCNC(NC(CC)C(N)=O)=S)c(Br)cc(F)cc1Br C1(C(=O)OCC)CC2CN(N3CCOC(CC)(CC)C3)CC(C1)C2 N1(C(C(=O)NC(C(CC)(C)O)NC(=O)OC(C)(C)C)=O)CC2NC(=O)C(=O)NC2C1 N1(C(C2OCCC(NC(C(CCC)=CCC)=O)C2)=O)CCc2cccc(C)c21 Cc1ncc2cc(C(N3CC(NC(C4CC=CCO4)=O)C(O)C3)=O)c(O)nc2n1 c1(C(c2n(CC=C)nnn2)NC2CCC(SC)CC2)cc2cccc(Br)c2o1 CCC(C(C)NC(=NCC1(c2ccccc2)CC1)NC(C1CC1)C1CC1)C(C)C C1(C(=O)NCC2(CC(C)C)CC2)CC(C)(C)CCN1C(=O)C(F)n1ccnc1 C1(C(N2C(CNC(Cc3c(C)scc3)=O)CC2)=O)CC2C=CC1C2 Cc1ccc(NC(=O)CC(C)N(C)C(C2CCC(=O)C2)=O)c(C)c1O CCC(CN=c1[nH]c2c(c(=NCc3cc(Br)c[nH]3)[nH]1)CCCCCC2)CCOC C1(NC(c2c(CC)cccc2)=O)CCN(C(C2(C#N)CCC2)=O)CC1CO c1(C(=O)NCC2CN(C(CCCC#C)=O)C(C)C2)cc(C)ncc1C c1(OC)cc(C)c(NC(=O)CC(C)CNC(=O)CC2(OC)CC2)cn1 C(C(=O)N1CCCC1CNC(=O)CC1(C)CC1(F)Cl)(C(C)C)OC c1(C(=O)NCC(CC=C)NC(c2c[nH]nc2C(C)C)=O)cc(C)ccc1OC N1(C(C(CC#C)C)=O)CCC2C(CCN2C(c2cc(Cl)c([N+](=O)[O-])[nH]2)=O)C1 c1(OC)cc(C(N2CC(CC(F)C(=O)NCC(C3CC3)N(C)C)C2)=O)ncn1 CS(=O)CC(c1ccccc1)CNC(=O)CCn1cc(C(C)(C)C)nn1 Cc1ccc(-c2cnc(N3CCN(C(C4CC4(F)Cl)=O)CC3)nc2)cc1C c1(C(C(N2C(C)C(NC(=O)COC3CCCCC3)CC2)=O)O)ccc(C#N)cc1 N1(CC)C(=O)CCC1C(=O)NCC1CN(C(=O)C(C)NC(=O)CC2C=CCC2)C1 c1(N2CCC(NC(c3n(CC)ncc3)=O)C(C)C2)cc2nnc(C(C)C)n2cn1 C(=O)C1CCN(C(C2CC2CNC(C2COCCC2C)=O)=O)C1.CO CC(C)CC(C(=O)NC1CCCN(C(C)C)C1)ONC(C1CC=CC1)=O C=CC(C)(O)CC(=O)N(CC(=O)NC1C(O)C2CCOC12)CCC c1(C(=O)NC2CCN(C(CCSC)=O)CC2F)cc(Br)ccc1[N+](=O)[O-] CC(CN)CC(=O)N1C(CC(F)(F)F)CCC1C1CC1 C1(C(=O)NCC(C(=O)N2C(CCCC)CCC2)C(C)C)CCC2CC1C2(C)C C1(C(N2CCC3C(C2)CN3C(=O)COc2ccsn2)=O)CC1C1CCCCC1 c1(CCC(=O)N(CCN(C(C2CC2C)=O)CC)CC)nc2cccc(Cl)c2[nH]1 CN(C(=NCC1(S(C)(=O)=O)CC1)NCn1ccnn1)CC1CCCO1 C(C)(N=c1ccc2ncc[nH]c-2n1)C1N(C(C2OCC(C)(C)C2)=O)CCCC1 C1(C(=O)NCc2cc(CC)[nH]n2)COCCC1NC(c1c(C)nsc1C)=O S(=O)(=O)(c1[nH]c(=NCCNC(CCC)C2CCC2)ccc1Br)NCC(CC)C(C)C C1(C(=O)OC)CCC(C(=O)O)CN1C(c1cc(C(F)(F)F)ccc1Cl)=O CC(C)(C)CC(CO)NC(C1CCN(C(c2ccc(Cl)s2)=O)CCO1)=O C1(NC(CCNC(=O)NC)=O)CN(C(c2c(C(F)(F)F)ncn2O)=O)CCC1C N1(CC=C)CCN(C(=O)NC2CC3CC2C2CC32)C(C)(C)C1=O C(C1CN(C(=O)C(O)C2CCCC2)CC1C(=O)NCCCc1cncnc1)=CC c1(OC)ccc(-c2noc(-c3csc(N4CCCCC4=O)n3)n2)cc1OC Cc1ccc2[nH]cc(CC(=O)NC34CCCC3C4)c2c1 c1(C(N2CCC(C(CNC(CC(C)(C)F)=O)(C)C)CC2)=O)cccc(Cl)c1F CCCCCCCCCC(=O)N1CC(C)(C)CC1CNC(c1cocc1C(N)=O)=O C1(C(N2CC(CO)C(C)C2)=O)(CNC(C2(C)CC(=C)C2)=O)CC12CCC2 C1(CNC(C(c2ccccc2)SCC)=O)C(O)C(O)CN1C(c1sccc1C)=O N1(C(c2c(CC)nccn2)=O)CCCC(CO)(CNC(c2onc(C)c2C)=O)C1 C1(CC)CN(C(=O)C(CNC(c2ccnc(C)c2)=O)N(C)C)CC1F Cc1cc(C)c(C(=O)NCC2C3CN(Cc4ncccc4O)CC23)c(C)c1 C1(C(N(C(CCNC(C2(CC#C)CCOC2)=O)C)C)=O)CCC(C)(O)CC1 c1(NC(C2CCCC2O)=O)cc(O)nc(=O)n1C.CC1CC2CN1C(=O)CN2 C1(CNC(C2N(C)CC(F)C2)=O)CC(C)(C)CN1C(=O)C1=C(C#N)CC1 CCCC(CNC(=O)C(CC)n1cncn1)C(=O)N1CC(c2nncs2)C1 CCCC(C(=O)N1CCC2C(OC)C12)NC(=O)COCC1CCCC1 c1(C(C)C)ncncc1C(=O)NCC(O)CNC(=O)CC=CC(C)(C)C N1(C(C2CCC(C(N)=O)C2)=O)CC2(CC(NC(c3cc4sccc4s3)=O)C2)C1 N1(CC(C)(C)NC(c2nc(Cl)c(Cl)s2)=O)CCN(C(=O)CC2C=CCCC2)CC1 N1(C(c2ccc(=NC)[nH]c2)=O)C2CCC1CN(C(=O)Cc1ccno1)C2 c1(CC(=O)OC)nsc(N2CC(OCCNC(=O)C(C)n3cncn3)C2)n1 c1(N(c2ccccc2)C(=O)NCCOC)cc(N2CCCC2)ccn1 C1(CC(=O)N(CC(N)=O)CC)CN(C(C2(C(=O)NC)CCC2)=O)CCC1C c1(OC)nccc(N(C)C)c1C(=O)NNC(=O)C1CCN1C(C)=O c1(C(=O)NCCNC(C2CC(OC)C(OC)C2)=O)cncc2ccsc12 c1(CNC(C23CCC(CC2)O3)=O)cnn2c1CN(C(=O)CN1CCOCC1)CC2 C1(NC(c2nccc(C)c2)=O)CC2CC1N(C(c1cc3c(s1)CCC3)=O)C2 c1(C(=O)NCC2(F)CCCN(C(CCCSC)=O)C2)cn(C(C)C)c(=O)nc1O C(C#Cc1cccnc1)NC(CC(C(F)F)NC(C1(OCC)CCOC1)=O)=O C1(C(=O)NC23C(CN(C(c4n(C=C)ncc4)=O)C2)C3)CCCCCCCC1 c1(C(N(C2CN(C(C3CC4(C3)CC4F)=O)C2)C)=O)ccc(N)c(F)c1F c1(C(=O)NCC(C)NC(c2conc2C2CC2)=O)csc(C(F)F)n1 C1(c2c(C3CC=C(C)CC3)cccc2)CC(=O)N(COC(F)(F)F)C1=O Cc1nsc(C)c1C(=O)NCCOCCN(C(=O)C(C)C(C)C)C N1(NC(=O)OC)CCN(CCCCC2(N(C)CN3CC4CC4C3)CC2)CC1 c1(C(c2nnnn2C2COC2)NC(c2ccc(C)o2)C)cc(C)c(Cl)c(C)c1 c1(C(=O)NC2CC(NC(CSC)=O)C2)cc(S(=O)(=O)N(C)CC)c[nH]1.C1CCC1 C1(NC(c2c(CC)cccc2)=O)CCCN(Cc2ccncc2C(=O)NC)CC1 N1(C(CCc2c(C)ncs2)=O)CC(CNC(C2CC2F)=O)C(C)(C)C1 Cc1c(C(N2CCN(C)CC2C(C2CC2)NC(=O)COCCF)=O)cccc1Cl C1(CNC(C(=O)N(C)C)=O)COCCN(c2ccnc(-c3nccs3)n2)C1 N1(C(COCCCC(C)C)=O)CCC(C)C(NC(=O)C(C)Sc2ccncc2)C1 CCC(CC(=O)NCCC(CNC(=O)CCCNC(N)=O)OC)CC(C)C N1(C(C2C(C(C)=O)C2)=O)CCCC(CC(=O)NC2(C)CCSC2)C1 CC(=O)CCCC(=O)N1CCC(O)(C(C)NC(=O)Cc2cnn(C)c2)C1 Cc1coc(C(C)C)c1C(=O)NC12CC(CNC(=O)CNC(=O)N(C)C)(C1)C2 C1(C(=O)N(C2CCN(C(c3ccc(C#N)[nH]3)=O)C2)CC)(CC)CCC(F)(F)CC1 C1(CNC(c2cc(CC)nc(O)c2)=O)CN(C(=O)C(C)COC)CCC1C(F)(F)F c1(CC(=O)NC23CCCC2CN(C(C24CCCC2C4)=O)C3)noc2ccccc12 C1(=O)C(C(C)C)N1.C1(OC)(CN(C(=O)CN(C2CCC2)C)C)CC1 C(CC(=O)NCC(C1CC(C)(C)C1)O)(C(F)(F)F)NC(C=C(C)C(F)F)=O CN1CC(O)CC1C(=O)NC1CCC(C(=O)NCC2COCC2N(C)C)C1 CC1CCCCC1(CNC(C1CCCCC1(F)F)=O)NC(C1CC=CCO1)=O N1(CC(=O)NC(CC(C)C)c2ccccc2)CCCCC1Cc1ccc(F)cc1 Cc1ccc(C(N2CCC(C(C)(C)NC(c3csc(Cl)n3)=O)C2)=O)nc1O Cc1ccc2c(c1)C(N(C(c1cc(-c3ccc(C)cc3)c(C)s1)=O)C1CC1)CC2 N1(C(COCC)=O)C(C(=O)NCc2cc(NC)nc(Cl)c2)CC2CCCC12 C(c1ccccc1C#N)=CC(=O)NCCC1CC(NC(C(C)c2ccco2)=O)C1 CC1=NOC(C)(C(=O)NCCCCCNC(C2(c3ncccc3F)CCC2)=O)C1 N1(C(CCC(CC)C)=O)CCC(C(=O)N(C2CCOC(C)C2)C)=C(F)C1 N1(C(C(=O)NCCCOC)Cc2ccn(CCF)n2)CCN2CCCCC2C1 N1(C(C(CCN(C)C)NC(c2cc(F)n(C)n2)=O)=O)CC2(CCC(=O)N2)C1 c1(C(N2CCC3CN(C(C=NOC)=O)CC3C2)=O)cc2c(F)cc(Cl)cc2[nH]1 C1(CC(=O)NCC(CN(C(C23CC(OC)C2C3)=O)CC)(C)C)CCCCC1(C)C C12(C(=O)NCC(CNC(C=C(COC)C)=O)OC)C3CCC(CC13)C2(F)F N1(C(C(=O)NCCOC)C(C)(C)C)CCCC2(C)COCCC12 CC(C)C(O)C(F)(F)C(=O)NC1CC(CNC(c2ncn3cc(Cl)ccc23)=O)C1 C=C1C(NC(N2CCC(Nc3cccc(Cl)c3)C2)=O)CC2CC1C2(C)C N1(C(c2c(C)cco2)=O)CCCC2(NC(=O)C(C)C3CCCC3)CCCC12 c1(C(=O)NC2(C(=O)NCC(F)C(C)(C)O)C(C)(C)C2)ccc(N=[N+]=[N-])cc1 Cc1cc(-c2ccccc2)oc1C(N1CC(F)CC1C(N)=O)=O c1(C(=O)NC(CCOC)CNC(=O)C(C2CC2)C2CC2)cnn2c1C(=O)NCC2 N1(C(C(CC)(C)CC)=O)CC2CN(C(=O)CCc3cn[nH]c3)CC2C1 c1(C(N2C3CN(c4nccc(C#N)n4)CC2C3)=O)cnc2[nH]ccc2c1 C1(Cc2ccccn2)CCC(c2nc(-c3nnc(C(F)(F)F)o3)no2)CC1 C1(C(N(CCCN(C)C)CC)=O)CN(C(=O)C=CC(C)(C)C)CCO1 C1(C(N(C2CN(C(Cc3c(CC)cccc3)=O)C2)C)=O)CN2CCCC2CO1 CCN=C(NCC(C)Oc1cccc(C)c1)NC1CC1(F)F C(=O)(CC(C)(C)c1cccs1)N(CC(C)NC(c1cc(COC)on1)=O)C C(=O)(C1CCc2nccn21)N1CCC(N(C(CC2(C=C)CCC2)=O)CCC)CC1 C1(CNC(c2cccc(CC)n2)=O)CC2(CCN(C(=O)CC(C)(C)SC)C2)CO1 C1(NC(c2cc(CC)no2)=O)CCCCC1N=c1cc(C)nc(C2CCC2)[nH]1 N1(C(c2c(CC)non2)=O)CC2CN(C(=O)C(F)C3CCCC3)CCC12 C1(NC(COC)=O)CC2CCC(C1)C2NC(=O)CC(C)c1cnn(C)c1 c1(NC(CC(=O)OCCSCC(C)C)=O)ccccc1OCCF c1(CC(C(=O)OC)NC(C2CCCC(=O)N2C)=O)ccc2ccccc2c1 Cc1cc(C(N2CCC(F)(c3cc(F)cc(F)c3)CC2)C(=O)NC(C)C)ccc1Br n1(CC)cc(C(=O)NC2CC(C)N(C(=O)CN3CC(C)(C)C3)C2)c(C(C)C)n1 C(=O)(C1=CCC(C)CC1)NCc1c(CNC(C=C(CC)C)=O)n[nH]c1 c1(OCCC(=O)NC2C(NC(=O)CCc3ccncn3)CC2)ccc(Cl)c(F)c1 N1(C(=O)Cc2ccc(F)cn2)CC2CCC(Nc3ncncc3Br)CC2C1 C1(F)(C(=O)NC2CN(C(C(C)(C)O)=O)CC2O)CS(=O)(=O)CC12CCC2 C=CCCCC(=O)N1CC(C(=O)NC)(CNC(C2CCCN(C)C2)=O)C1 CC1(C)OCc2c1n[nH]c2C(=O)NCCCNC(=O)CC1CCCOCC1 c1(C(=O)OC)c(C)ccc(C)c1C(=O)NC(C)CCNC(C1(C)CC=CCO1)=O C(=O)(C1CCCc2nc[nH]c21)N1CC(C)(C)C(NC(=O)C2=COCCO2)CC1 C1(CNC(c2c(CC)nccc2)=O)CCCN(C(=O)CC2CCC(=O)N2C)CC1 c1(CCC(=O)N(CCOCCCN(C(=O)Cc2nccn2C)C)C)cccnc1 C1(NC(CSC)=O)CCC2CN(C(c3nnc(O)nc3O)=O)CC2C1 c1(OCC)cc(CC(=O)NC2CC(CNC(C3CC3(F)F)=O)C2)on1 N1(C(c2nc(CC)sc2N)=O)CCC(NC(=O)C(C)N(C)C(C)=O)CC(C)(C)C1 N1(C(CCc2ccc(CC)cc2)=O)CC(NC(C2CCC(=O)N2)=O)C2(CCC2)C1 C1(O)(CCNC(c2c(C)noc2)=O)CCCN(C(c2ccnn2CC2CC2)=O)C1 Cc1cc(Br)ccc1C(=O)NCCCNC(C1(NC(N)=O)CCCCC1)=O Cc1cc(F)c(C(=O)N(C)CC2CCCN2C(=O)Cn2nccc2C)c(Cl)c1 CC1CCN(C(=O)CN(C(=O)C(N)CN)CC(=O)N(C)C)C1(C)C C1(C)(CNC(C(CC)OC(F)(F)F)=O)CN(C(=O)CSC(F)F)C(C)(C)C1 C(CC(C)C)(C(=O)NCCC(C)(C)CNC(c1cnnn1C1CC1)=O)NC(C)=O c1(C(=O)NCC(CNC(c2cc(OCC)no2)=O)F)cccc(=O)o1 C(C(C)NC(=O)C1=CCCC1)(C(C)C)NC(C=CC=CC)=O c1(CC)ccccc1C1CCN(C(c2c[nH]nc2-c2cnccc2Cl)=O)C1 C(=O)(C(F)C(F)(F)F)N1C(CNC(CC(C)(C)C2CC2)=O)C=CC1.C1CCS(=O)(=O)C1 c1(C(=O)NC(C2(CNC(c3ncc(F)cn3)=O)CC2)C)ccc(C(F)F)cc1F c1(C(N2CC3C(CNC(C4C(C(=O)OC)CC4)=O)C3C2)=O)cc2cccnc2o1 C1(OC(N2CC(=O)N(CC(=O)O)C2)=O)CC(C(N(C(C)(C)C)C2CC2)=O)C1(C)C c1(C(C(=O)OC)N(CCCOC)CC2CC(OCC)C2)ccc2cncn2c1 CCC(CCCC(=O)NCCCc1nc(C)no1)NC(c1cnsc1)=O Cc1cc(Cl)c(Br)cc1C(N1CCCC(NC(=O)Cn2nccc2C)CC1)=O C(=O)(C=C1SCC(=O)N1C)NC1COCC(CNC(C(CC)(CC)CC)=O)C1 N1(C(c2ccccc2C(N)=O)=O)CCN(C(c2ccccc2Cl)=O)C2CC12 Cn1nc(Br)cc1CCNC(=O)C(=O)NC1CCC(C#N)C1 C1(C(CC)C)CCCN1C(=O)CCC1CCCC1.C12CC(C)(C1)NC(=O)C2 C1C(O)C(=O)N1CCOC.C(C)(C(=O)NC1CC1)OCC=C N1(CC)CC(C(=O)NCC2CCC2CNC(=O)C(F)F)CC1=O c1(C(=O)OCC)cc(C)cnc1N1CCC(NC(=O)Cc2cc(C)ccc2O)C1 c1(CC(C(=O)NCCC2CCC(NC(c3c(C)con3)=O)C2)C)ccccc1Cl N1(C(CC2CC(CC)C2)=O)CCCOC(CN)C1 S(=O)(=O)(c1c(Cl)cccc1Cl)NC.CC(N(C)N=O)C1CC1 c1(C(N(CC(C)NC(C(C)SCC)=O)C)=O)cc(Br)cn1C1CC1 C1(C(=O)NC2(C3N(C(c4cccc(C)n4)=O)CCC3)CC2)CCn2nncc2C1 CC1CCC(NC(c2c[nH]nc2-c2cccnc2)=O)CN1C(=O)CC1(O)CCCC1 C(C)(CC(F)(F)F)NC(C(CNC(C(CC)N(C)C)=O)C)=O n1(CCCC(=O)NCC2N(C)CCN(C(=O)CO)C2)cnc2ccccc2c1=O C1(=O)C2=CCC(C2)N1.C#CC1CCCCC1.C1(=O)C(CCC)N1 N1(C(c2nccc(C)n2)=O)CCC(NC(=O)COc2c(C)occc2=O)CC1C S(=O)(=O)(c1ccc(F)c(C(=O)NC(C2CCCO2)CC)c1)N(CC(=O)NC(C)C)C N1(C(=O)C2CC2)CCc2c(C(C)=O)csc2C1 C(=O)(C(F)C(=O)N1CCC(CCCC=O)C1)OCC.N(CCC1CC1)CC c1(C(C(=O)NCCCOC)N(CC=C)Cc2ccc(C)o2)cc(Br)ccn1 c1(C(=O)NCC(CN(C(CCC(CCSC)O)=O)C)C)ccc2c(c1)NC(=O)C2 c1(NC(N2CCC(C#C)(C(=O)OC(C)(C)C)C2)=O)cc(Cl)cc(Cl)c1CC1CCC1 CC1CCN(C(C2CC(NC(c3cccc(O)c3)=O)C2)=O)CC1(C)C C(=O)(C(C)(O)CCC1CCCC1)N(CCC(=O)O)C C1(C(=O)NCC(CCOC)O)CN(C(c2oc(C)nc2C)=O)CC12CCC2 c1(N(CCCNC(C(C2CCCOC2)OC)=O)C2CC2)ncnc(C)c1OC C1(NC(CCNC(=O)NC)=O)CCN(C(=O)C(C)CCC2CCOCC2)CC1 c1(C(N2CC(=C(CNC(c3cccc(Cl)c3)=O)F)C2)=O)cc(O)ncc1F N1(CC)C2CCC1CN(C(=O)C(N1CCOC(C(C)(C)C)C1)=O)C2.C1CS1 C1(NC(C2CC(C3CC3)C2)=O)CCCC(NC(C23COC(CF)(C2)C3)=O)CC1 C(C[Si](C)(C)C)(C(=O)O)C1C(NC(C=Cc2ccc(C)cc2)=O)CCCC1 c1(CC=C)ccccc1C(=O)NC(CC(N1CCOC(O)C1)=O)C1CC1 Cc1cc(C(=O)NC23CC(CNC(=O)CNC(=O)CN(C)C)(C2)C3)c(C)cn1 C(=O)(CCCCCCN(C)C)NC1CCC(C)N(C(=O)CCCCN(C)C)C1 S(=O)(=O)(c1cccc(C(C)C)c1)N1CCN(C(=O)NCC2ON=C(C)C2)CC1 c1(CN(C2CCCN(C(c3n(C)cnc3)=O)C2)CCO)ccc(O)c(O)c1 C(=O)(C1=CCN(OCC)C1)N1CC2N(C(C3(CCOC)CCCCCC3)=O)C2C1 n1(CC)c(=O)nc(O)c2c1nc(C(C)NC(=O)CC1COC(C)(C)C1)n2C C(=O)(CC(C)(C)C)NCC(=O)NCc1cc(C(=O)NCC(c2cnc[nH]2)C)on1 N1(C(c2c(C)scc2)=O)CCC(F)(F)C(NC(c2occc2Br)=O)C1 C=CCCCC(C)(C)C(=O)NCCN(C(=O)Cn1cc(C)ccc1=O)CC1CC1 O=C(C1=CCCSC1)NC1(CO)CCCN(C(=O)CCCc2nccs2)C1 c1(NCC)cncc(C(=O)NC(C)C(C)(C)NC(=O)C=C2CCC2)c1 C(=O)(C(CC)C(C)(F)F)NC1(CNC(c2nc(COC)oc2)=O)CCCCC1C c12nccc(n1)N1CCC(C1)C(C)NC2=O.C1(C(=O)OC)(CCF)CC1 c1(NC(N2CCC(n3cc(C(C4CCCO4)O)nn3)C2)=O)ncccn1 c1(C(N2CCC(C)(O)C2)C(=O)Nc2cccc(OC)c2)cc(C)cc2c1OCC2 C1(NC(c2cnco2)=O)C2CCC1CN(C(=O)CCCCc1cccc(O)c1)C2 N1(C(CC(C)(C)O)=O)CC2CCC1C(CNC(C1CCc3ncsc3C1)=O)C2 CC1C(C)N(C)CCN1C(C1(C)CCN(C(=O)CCc2cnn(C)c2)C1)=O c1(CC)oc(C(=O)NC(C)CC(C)NC(c2cccnc2)=O)cc1C Cc1cc(Cl)ccc1NNC(=O)c1ccnc(-c2cccnc2)n1 C(=O)(C(C)(C)CC1CCN(C(=O)NC(C2CC3CCC2C3)C)CC1)OC CON(CCC(=O)N1CC(C)OC(C)(C)C1)C(=O)Cc1cc2cccnc2[nH]1 C(=O)(CCC(C)CCCC)NCCOC1CN(C(c2cc(C#C)c(C)cc2)=O)C1 c1(N(CCN(C(C(=O)OC)=O)C)C(C2CCC(N(C)C)CC2)=O)ncccc1F C1(CNC(c2c(OCC)scc2)=O)CCCCCN1C(=O)C(O)C1CC1 S(=O)(=O)(CCC(=O)N1CCC(C)C(NC(=O)C=Cc2ccc(Cl)s2)C1)NC C1(C(=O)NC(C)CN2CCN(C(C3CCC(C)O3)=O)CC2)CC(=O)NC1(C)C c1(OC)cc(N)c(C(=O)NC2CC(NC(c3ccc(F)c(F)c3C)=O)C2)cc1F c1(CC)nn(C)c(CC(N2CCC(O)(CNC(=O)C(C#N)C3CC3)C2)=O)c1Cl Cc1ccc(C(N2CCC(NC(=O)CSCC3CCCO3)C2)=O)c(N)c1F c1(C(=O)NC(CC=C)CNC(C2CC3(CC3)C2)=O)cccc2[nH]ccc12 C1(C(=O)NCC(C#C)OC)CN(C(c2cccc(O)c2F)=O)CC(C)(C)C1 C12(NC(c3ccc(OC)o3)=O)CCCC(CN(C(c3ccc(C)c(Cl)c3)=O)C1)C2 c1(C(N2C3CC(CN(C(C(P(C)(C)=O)O)=O)C3)C2)=O)ccc2c(c1)OCCCO2 Cc1cc(=O)c(C(=O)NC2CCCCC2CNC(=O)COc2ccon2)cn1C N1(C(C(C2CN(C(c3cc(O)n(C)n3)=O)C2)OC)=O)CCOCC2(CC2)C1 C(C)(CNC(=O)CC=C(Cl)Cl)(C(C)C)NC(c1nc(C(C)OC)oc1)=O C1(CC(=O)NCC(C2CC2)OC)CCN(C(=O)C=CC2CC2)C1 C1(C(N(C2CC(NC(c3c[nH]nc3Br)=O)C2)C)=O)CCC1(F)F C1(C(=O)NCC(CNC(C2SCCCS2)=O)C(F)(F)F)(OC)CCS(=O)(=O)C1 C=CC1(C(=O)N(CCCF)C)CCN(C(=O)CC2=CCCC2)C1 c1(C(N(C2CCC(NC(=O)CCN3CCCC3=O)C2)C)=O)cncc2[nH]ccc12 C(=O)(CCCCN(C)C(c1c[nH]nc1CNC(c1sccc1C)=O)=O)NC C1(CC(=O)N(CCCNC(=O)C(C)NC(c2ccoc2)=O)CC)CC2CCC1O2 O=C(C1=NOC2(CCC2)C1)NC1(C2CCCN(C(c3coc(O)n3)=O)C2)CC1 C#Cc1cccc(N(C(=O)CCCC2CCCC2)C2CCOCC2)c1 c1(SC)ncc(C(N2CCCC2CNC(c2ccnc(Cl)c2N)=O)=O)c(O)n1 N1(C(CSCc2cccc(C)c2)=O)CCC(NC(C2CC3(CC3)C2)=O)C(O)C1 C#CC1CN(C(c2ccsc2OCC)=O)CCN1C(c1cnncc1OC)=O C(CC(=O)NCC1CC(CCC(=O)NC(=O)CN(C)C)C1)(C(F)F)NC(=O)OC c1(OC)ccc(C(O)CNC(c2cccc(Cl)c2F)C)cc1F c1(CNC(C2CC(O)CCN2C(c2ccc(Br)s2)=O)=O)cccn2nccc12 N1(C(CSc2n(C)cnn2)=O)CCCC(O)(CCNC(C23CCC2CC3)=O)C1 c1(C(N(C(C)CNC(C2CC3(CC3)C2)=O)CC)=O)ccc2c(c1)CCCO2 CN1CCC(Cc2nc(-c3cccc(SC(C)(C)C)n3)nn2CCC(C)(C)C)CC1 C(C1CN(C(c2ccsc2)=O)CC1C(=O)NC(CCO)C1CC1)=CC N1(C(C2C(CCC)CN(C(C3CCC=CCC3)=O)C2)=O)CC=C(CO)CC1 c1(C(C(=O)NC(CNC(C=C)=O)C2CC2)C)ccc(Cl)c(Cl)c1 c1(-c2cc(NC(c3nc(Cl)ccc3Cl)=O)ncc2)cc2cc(F)ccc2[nH]1 C#CC1CCCCN1C(=O)CCC(CC)NC(=O)C=Cc1ccsc1 C1(N(C(=O)CO)CC)CCCN(C(c2cc(-c3ccccn3)ns2)=O)C1 C1(C(=O)NC2CC3CCC(C2)O3)(CC)CCN(C(=O)Cn2nccn2)CC1 c1(C(C(=O)NC)C)c(C(N2CCN(C(=O)CC3C(C=C)C3)CC2)=O)cccc1F c1(NC(C(C2CCN(C(CC(=C=C)C)=O)C2)F)=O)cc(C)c(O)cc1C c1(CC)c[nH]cc1C(N1CCC1CC(=O)NCC(=O)NC1CC1)=O N1(C(c2c(OC)cc(N)cc2)=O)CCC2(CCCN2C(c2cc(F)n[nH]2)=O)C1 CCCCCOCCNC(=O)CN(C(C1(C(=O)N(C)C)CC1)=O)C1CC1 CC1=C(C)CC(C)(NC(=O)C(Cc2cc[nH]n2)NC(=O)C=Cc2ccn(C)c2)CC1 C1(N(C(c2c[nH]nc2C2CC2)C(=O)NCCCSCC)C)CCCC(C)C1 C(=O)(CCC(=O)N1CCCC(N(C(=O)COC2CCOC2)C)C1)c1ccc(C)s1 N1(C(c2cc(N(C)C)ncc2)=O)CCN(C(C2CC3(C2)CC3F)=O)C(C2CC2)C1 c1(CC(=O)NC2C(CNC(c3c(C)n[nH]c3)=O)C2)ccc(Cl)c([N+](=O)[O-])c1 C1(C(N(CCC(=O)NCC2(CCC=C)CC2)CCO)=O)C2CCCC12 C(=O)(CCC(C)NC(=O)CC1CCC2CC12)NCc1c(OC)nsc1 C1(F)(CNC(C(C)NC(N)=O)=O)CCN(C(=O)Cc2cnoc2)CC1 N#Cc1cc(Br)ccc1C(=O)NCCCNC(=O)NCCOCCOCCO c1(C(=O)NC2C3(CCN(C(C4CC(C)=C(C)CC4)=O)C3)C2)ccc([N+](=O)[O-])cc1 c12ccnc(c1)C(=O)N(C1CC1)CCNC(=O)C2.C=C1CCC1CC1CC1 C1(C(=O)NC2(C)CC2)CCC(CNC(=O)C=CCF)CC1 Cc1ncc([N+](=O)[O-])cc1C(N1CC(CNC(c2cc(Cl)cs2)=O)C(C)(C)C1)=O CC1=C(C)CN(C(c2occc2CNC(C2COCCN2C)=O)=O)CC1 c1(CC(CC)N(CCCc2cnc(N)c(CO)n2)C)c(F)cccc1F c1(NC(C)=O)cnccc1C(N1CC(NC(C2(C)COC2)=O)C(C)C1)=O c1(OC)ccsc1C(=O)N(CC(C)C(=O)NCC(c1ccco1)O)C c1(CN2CC3C(C(=O)Nc4c(Cl)ccc(C(=O)OC)c4)(C3)C2)c(F)cccc1F C(C(C(C)C(C)C)NC(=O)C(=O)N(C)C)NC(C(C=CC)SCC(F)F)=O c1(C(=O)NC(c2cccc(C(=O)OC)c2)C)cnc2[nH]nnc2c1 N(C(=NCCc1cccs1)NCC(c1ccc(F)cc1)O)CC(N1CCCC1)C C1(C(=O)NC(C2CCN(C(C3C4CCCC34)=O)C2)C)(CO)CCOCC1 C(=O)(C(Cn1ccnn1)NC(=O)COCCF)N(C)Cc1ccoc1 c1(N(CC(=O)NCCCC)C)ccc(NC(c2nnnn2C)C(C)OCC)cc1 N1(C(CCCCN(C(C2(OC)CCOCC2)=O)C)=O)CC2C(C1)C2(C)C C1(NC(c2c(OC)n(C)nc2)=O)CCN(C(C2CCC2C#N)=O)CC1O C1(NC(c2cnc(C(C)C)n2C)=O)CCC12CN(C(c1ncn(C)n1)=O)C2 c1(C(=O)NCC(=O)NC(CNC(C2C(C=C)C2)=O)CC)c(F)cccc1Cl N1(C(C(C)SCCCC)=O)CCCC(NC(CCC(=O)N(C)CCOC)=O)C1 C(CC(C(=O)NC1CCCCC1NC(c1cc(C)co1)=O)NC(N)=O)SC N1(C(CCC(C)(C)C)=O)CCC2(CC1)CN(C(=O)C(C)(C)CC#N)CCO2 c1(C(=O)NC(CNC(C2C(=C)C2)=O)CO)[nH]nnc1C1CC1 C1(CCC)CCN(N2CCC2c2ncccn2)CC1 C(CCC(C)(C)C)(c1nnnn1CCCSC)Nc1ccc(OC)nc1 S(=O)(=O)(c1ccc(N2CCN(C3COCC3O)CC2)cc1Br)NC(CCSC)C c1(NC(Cc2ccc(=N)[nH]c2)=O)cc(F)cc2nc[nH]c12 C12(CNC(=O)CC3C=CCC3)CN(C(=O)Cc3cc(F)ccc3F)CC1CCO2 N1(C(Cn2c(C)ccc2C)=O)CCN(C(C2CCCC(C)(C)O2)=O)CC1C c1(C(=O)NCc2ccc(Cl)cc2-c2nn[nH]n2)cc(Br)c2cccnn12 C(=O)(C(CC1CCOCC1)NC(=O)C(C)CC1CC1)NC(c1ccn(C)n1)CC c1(C(=O)NC2(C(N(CCC(C)C)C3CC3)=O)CCC2)ncoc1C(C)C CC(C#N)C(=O)N(CC(=O)NC(c1ncc[nH]1)CO)C c1(C(C)NC(C2CN(C(c3cscc3Br)=O)CCO2)=O)cc(Br)cc(Br)c1 C1(NC(CC(C=C)C)=O)CCCC12CCN(C(c1cc(F)c(C)cc1Cl)=O)CC2 Cc1cc(C(=O)NCC(C)(C)C(N2CC(O)C(C)(C)C2)=O)ncc1F n1(CC(=O)NCC2CN(C(=O)CSCc3cccs3)C2)cnnn1 C1(CC(=O)N(C2CCN(C(=O)C(=O)N(C)C)C2)CC)CC2(CC2)C1 C1(NC(C2CC3CCC2CC3)=O)COC2(C1)CN(C(=O)C(C1CCOCC1)F)C2 c1(C(N(C2CCN(C(C=CC(C)(C)SC)=O)C2)C)=O)c(C)ncnc1O C=CCCCCCC(=O)N1CC(CO)OCC1C.C123CCC(CC1)(C2)NC3=O c1(CC)nc(-c2cccc(C)n2)nn1C(C)C1CC1.n12nccc1C2 CC1=NC(C)(CNC(=O)C(CCC2CCC2)NC(=O)CN2CCOC2=O)CS1 C(CC)(CC(C)CO)NC(CN(C(C1CC(=C)C1)=O)C)=O C1(NC(C(CC#C)C)=O)CC2CCCC(C1)N2C(c1nc(Cl)sc1C)=O CCCC(C)(O)CC(=O)N1CCN(CCCCCCNC(=O)C(C)S(N)(=O)=O)CC1 C1(C(=O)NC2CC2)C(O)CCN1C(=O)C1CC1 C=Cn1nccc1C(=O)N(CC)CC1CC(F)CN1C(=O)CCSC1CCCC1 C(C)(C)(C(=O)N1CC(O)(CCC(N2CC(C)(C(F)(F)F)C2)=O)C1)OC(C)=O Cc1c(C(N2CC(NC(c3ccccc3Br)=O)C3CC23)=O)ccn1C C1(CC=C)(N(C(=O)COC)Cc2ccc(Br)s2)CCCN(CC2CCCCO2)C1 Cc1ccc(Oc2cccc(C(N3CCC(SC(F)F)C3)=O)c2)c(C)c1 c1(OCC)c(Cl)cc(C)nc1C(N1CCC(=CCNC(C2OCCO2)=O)CC1)=O N1(C(c2nc(C3CC3)cs2)C(=O)Nc2c(C)cc(F)cc2)CCC(=C(F)F)CC1 N1(C(CNC(CCC)=O)=O)CC(C(=O)NC(C)CCO)C(=O)C1 N1(C(COC(C)=O)=O)CC2CC1CC2NC(=O)CCCc1ccc(Cl)cc1 C#CCCCCC(=O)NC(C1CCCC1)CNC(c1nn[nH]c1C(F)(F)F)=O C(CC1CC1)(C(=O)NCc1ccc(C(=O)NCC(C)(Cl)CC)o1)OC n1(CCC)nc(C)cc1C(=O)NCC12CC1CN(C(C1(SC)CC1)=O)C2 N1(C(CC2C(C)CCO2)=O)CCC(O)(C(C)NC(C2CCSCC2)=O)CC1 c1(NC(c2c(Cl)cnn2C)c2n(C(CC)C)nnn2)ccc(Br)c(C#N)c1 n1(CC)cc(C(=O)N(C)CC2(CNC(C3(SC)CC3)=O)CC2)cn1 c1(CNC(C2CCN(C3CCCN(C(C(C)(C)F)=O)C3)C2)=O)ccc2cc[nH]c2n1 C(=O)(CC1=CCOCC1)NC1CCC(CCNC(C2C3CCC2CC3)=O)C1 c1(N(C)Cc2cc(C)nn2C)[nH]c(=NC(C)C(C)F)nc2c1ncn2C(C)C c1(C(=O)NCC2C(NC(c3cn(CCOC)nc3)=O)C2)cncc2[nH]ccc12 N1(C(C(C(C)C)C)=O)CCCC2(NC(=O)CC3CSC3)CC2C1 C(=O)(CCC(CC)NC(c1c(C)ccn1C)=O)NC(CC#CC)CO c1(OC)ccc(NC(C2CC(O)CN2Cc2ncc(Cl)s2)=O)c(OC)c1 CC1OC(C)CC1C(=O)NC1CCN(C(c2coc(C(F)F)n2)=O)C1 C#CCC(C)(CC)C(=O)NCCOCCCN(C)C(c1ccc(OC)nc1F)=O Cc1cc(C(O)CNC(CCC2=CCOCC2)=O)ccc1F C(c1ccccc1)=CCCC(=O)NC1CC(C)(NC(c2coc(C(=O)O)c2)=O)C1 C1(C(=O)NCc2ccc(CC(C)NC(CC(C)OC)=O)cc2)CC(F)(F)C1(C)C c1(C(=O)NC(CC)CNC(C2CC=CCC2C)=O)cc2cc(Cl)cc(Cl)c2[nH]1 N1(C(C(C)S(C)(=O)=O)=O)CC2OCCN(C(=O)CN(C)C)C2C1 Cc1c(Br)cnn1CC(N1CCCC1(C)CNC12CC(C1)C2)=O c1(CNCC2C(C)CCN(C(c3cc(C(C)=O)on3)=O)C2)cnn2ccncc12 N12CCc3nc(cn3CC1)CC(=O)C(C)(CO)C2=O.C1(C)CCOC1.CO C1(CNC(c2cn(C)nc2C2CC2)=O)COCCN(c2ncc(Cl)c(O)n2)C1 c12ccc(cc1)C(C#C)NC2=O.c1(CCc2nn[nH]n2)nc(C(C)(C)C)n[nH]1 N1(C(c2cncc(C)n2)=O)CC(NC(=O)Cc2cccc(F)c2)CC12CCOC2 c1(C(N(C(CNC(C(CC)NC(C)=O)=O)C)CC)=O)cc(Br)c(C)cc1F N1(C(c2c(OCC)cccn2)=O)CCN(C(=O)OC(C)(C)C)CC1CC(F)(F)F C1(NC(CC=C(C)C)=O)CCC(NC(=O)CC=CCc2ccccc2)C1 C1(NC(c2c(C)cns2)=O)CC2CC(NC(=O)CN(C)C3CC3)C2C1 c1(OCC)ccc(C=CC(N2CC(C)(NC(C3CCCOC3)=O)C2)=O)cc1Br c1(N)ccc(N=[N+]=[N-])cc1.C12CCN(CC1)C(=O)CN2CC1CC1.C(CCF)O c1(C(=O)NC2CCCN(C(c3cncnc3)=O)CCC2)cc(Cl)cc2c1OCC2 C12(CC(N3C(CN(C(=O)CN(S(C)(=O)=O)C)C)COCC3)=O)CCC(CC1)CC2 Cc1cc(C(=O)NCC(C2CC2)NC(=O)CCC(C)(C)N(C)C)cc(C)c1F N1(CC)CC(C(=O)NCCCC(C)(C)NC(C2C(C)OC(C)C2C)=O)CCC1=O C=CC(C)(O)C(=O)NCC(C)(F)CNC(=O)Cc1cc(C)cs1 C1(C(=O)NCCCCNC(C(CCOC)C)=O)CSC(c2ccccc2O)=N1 C(CC(C)(C)C(=O)N(C1CCCOC1)C)NC(c1cc(C)on1)=O C(=O)(C#CC1CCCCO1)NCC(C)CNC(c1cn[nH]c1)=O c1(CNC(C(C2CN(C(COC(C)=O)=O)C2)O)=O)nn(C)c(=O)n1C C(=O)(C1=CCC2CCC1N2C(=O)C(O)C(F)(F)F)NC(C=C)COCC c1(C(=O)NCCC(C)N(C(=O)CSC2CC2)C)ccc2[nH]c3c(c2c1)CCCC3 c1(CN(C(C(C)NC=O)=O)C)cccc(CNC(C2(C)CCNC2=O)=O)c1 CN=c1[nH]nc(CC(N2CCC(C)C2CNC(=O)CC2CC=CC2)=O)s1 C=CC1CN(C(=O)CCC(C)(C)OC)CC1NC(=O)COc1cccc(F)c1F C(CCCCCNC(c1nocc1Br)=O)NC(CN(C)C1CC1)=O c1(CC(=O)N(CC(CO)(CO)NC(CSCC#C)=O)C)cc(F)ccc1Br C(=O)(CS(=O)(=O)CC(C)C)N1C2CC(NC(CC=C)=O)CC1CC2 C1(NC(N(C)Cc2c(C(F)(F)F)n[nH]c2C(F)(F)F)=O)CCCC1P(C)(C)=O C(=O)(C(C)CC(F)(F)F)NCC(C(C)(C)C)NC(c1c(CC)nns1)=O c1(C=O)cc(I)c(O)c(I)c1.N12CCC(C(O)C1)C2.N12CC3C(C1)N23 c1(C(N(C2CCN(C(CC(=C)Br)=O)C2)CCO)=O)cccc(OC)c1C C(=O)(C(C)(C)CCCO)NCC1(NC(C)=O)CCCC1.N12CCC(C)C(C1)C2=O c1(C(=O)NCC(C)NC(CCN(CC)CC)=O)cccc(Cl)c1[N+](=O)[O-] C1(N(C(C2C(NC(c3cc(C)oc3)=O)CC2)=O)CC2CC2)CCS(=O)CC1 c1(C(C(C)NC(=O)Cn2nnnc2C)NC(COCCOC)=O)cccc(Br)c1 Cc1c(C(N2CCC(F)(CNC(=O)C(C)(C)N(C)C)C2)=O)cccc1O c1(CC)cnsc1C(c1nnnn1C1CCC1)NCCC(Cl)Cl C(=O)(C1=CC2CCCCCC12)NC1(COC)CN(C(c2c(C)noc2N)=O)C1 N1(C(c2c(C)cccc2N)=O)C2CCC1CN(C(c1cccc(C(F)F)c1)=O)C2 c1(OC)cc(CN2CC(OC(=O)Nc3cccc(F)c3C)C2)cc(O)c1O N1(C(C(C)CF)=O)CCC2(CCCN2C(c2nc(Cl)cc(N)c2Cl)=O)C1 c1(OCCOC)ccc(CNCCc2ccc(NC(=O)CCC)cc2)cc1 C(CC(=O)NC1CC=CCC1C)(CC(C)C)NC(c1nc(CCC)oc1)=O CON(C(=O)C(F)C1CN(C(c2cnnn2C(C)C)=O)C1)C(C)C c1(C(=O)OC)ncnc(N2CCC(OC)C2)c1OC.c12cccc(c1)C(=O)N2 C1(NC(=O)Cc2ccsn2)CCCC(NC(=O)Cn2ccc(Br)n2)C1 Cc1cc(NC(=O)CC23CCC2CN(C(=O)C2=CCCCCC2)C3)c(C)c(C)c1 c1(C(N2C(CNC(C#CC3(C)CC3)=O)COCC2)=O)c(O)ccc(Cl)c1F CC(C)CCCCCC(=O)NC1CN(C(=O)Cn2cnc(C#N)n2)C2CCCC12 c1(C(=O)NC(CN(C(=O)CC(C)n2cccn2)CC)C)nc(Cl)c(=O)[nH]c1N C(=O)(C(C)CC(N)=O)NCC(c1ccccc1)N(C(c1ccc(C#C)o1)=O)C c1(CNC2CN(C(c3n(C(C)C)ncc3)=O)CC2C)ccc2c(O)nccc2c1 CC(CNC(=O)CCCN1CCCC1)C(F)C(=O)N1CCC(C)(CCO)CC1 CC1(C)CC(NC(c2ncccc2C(c2ccccc2)=O)=O)CO1 C12CCN(C(=O)C3(OCC)CCN(C3)C1=O)O2.C1(OC)(CO)CCC1 C1(CNC(CCOCCOC)=O)CC2COCC2N1C(c1cnc(N)cn1)=O N1(C(CC2(C(=O)OC)CC2)=O)C2CCC1CC(N(C)C(C1CN(C)CCO1)=O)C2 C1(C(=O)OC)C2CC(NC(c3ccc(C4(N)CCC4)o3)=O)CC12 C1(NC(c2cc(C)c(=N)[nH]c2)=O)CC2CC1CN(C(=O)CC(C)(C)F)C2 C1(NC(C=C(CCC)C)=O)CCC(O)CN(C(C2CCCC2(F)F)=O)C1 CCC(CC)(CO)C(=O)N1CC=C(C(=O)NCC2CCC(C)C2)C1 C12(C(=O)OCC)CC(CC3COC4CC3C4)(C1)OC21CN(C(C)=O)C1 c1(C(=O)NCC(CNC(C(CC=CC)C)=O)F)ccc(S(=O)(=O)NC)o1 c1(C(N2C(C)(C(=O)Nc3nccs3)CCC2)=O)cccn2ccnc12 C(=O)(C1=C(Cl)CCC1)NC1(CCNC(c2c(C(C)C)n[nH]c2)=O)CCOCC1 C(=O)(C1Cc2ccc(Cl)cc21)N1CCC(CCNC(C(C)(C)C2CC2)=O)C1 C1(NC(C(C(F)(F)F)OC(C)=O)=O)CC2CC(C1)N(C(c1cc(Cl)no1)=O)C2 c1(C(=O)NCC(CNC(C2(C)COCCO2)=O)O)cccc2c[nH]nc12 Cc1nc(=NC(C)CC(C)NC(=O)CCCCN2CCCCC2)s[nH]1 c1(C(=O)NC2C(C)CN(C(c3ccsn3)=O)CC2)ccc(C#N)cc1Br CCCC(C(=O)NCCCO)NC(C)=O.C1(C(N(C)C)=O)COCCN1CC N1(C(c2cccc(S(=O)(=O)N3CCCC3)c2)=O)CCC(S(=O)(=O)c2ccccc2)C1 c1(CSCC(=O)NC(CNC(CNC(CCCC)=O)=O)C2CC2)ccc(F)cc1 N1(C(C(C(CC)C)O)=O)CC2CC(C)N(C(c3ccc(C(F)F)cc3F)=O)C2C1 C1(=CC(=O)N(C(CNC(c2ccccc2)=O)Cc2ccccc2)C)CCN(C)C1 C(=O)(C1=NOC2(CCOC2)C1)N(C1CCCCN(C(=O)CC=CC(C)(C)C)C1)C c1(C(=O)NC(C2CCCN(C(=O)CCCCN=[N+]=[N-])C2)C)ccc2cc[nH]c2n1 C1(CC)(CC)CCN(C(=O)C(c2cccs2)NC(C2CC=CCC2)=O)C1 C1(NC(c2c(CC)[nH]nc2Cl)=O)CCC2CCN(C(c3ccc(SC)s3)=O)C1C2 Cc1ccc2oc(C(=O)NC(CNC(c3ccc(Br)cc3)=O)CO)cc2c1 N1(C(C(n2ccc(C)n2)C)=O)CC2C(CNC(=O)CSC(C)C)C2C1 c1(C(N2CC3C(CNC(c4ccc(C(C)N)cc4)=O)(C3)C2)=O)cc(I)cnc1Cl CC(C)CN=c1[nH]c(=NCC(F)(F)C(F)F)c2cc(OC)ccc2[nH]1 Cc1ccc2c(c1C)C(NC(=O)CCc1c(C)nc(O)nc1O)CC2 C(=O)(C(CCCC1CC1)N1CCOC(CS(N)(=O)=O)C1)NCCOC c1(C(N(CCCNC(COC(CC)C)=O)C)=O)c(C)nn(C)c1OC C1(CC(C)C)(C(N2CCC(N(C(=O)C(C)NC(N)=O)C)CC2)=O)CCOCC1 N12CCC(C)(CC1)CCC2=O.C1(C(=O)NC)CCCOC1.C(C(=O)C(N(C)C)=O)N C1(NC(c2ccco2)=O)CC12CCC(NC(c1ccnn1C(F)F)=O)CC2 N1(C(COc2cn(C)nc2)=O)CC(CNC(C2CNC(=O)C2(C)C)=O)CC1(C)C CCCCC(C(=O)NC1CN(C)CCC1O)NC(=O)C=Cc1cn(C)cn1 c1(C(N2CCC(O)(CN(C(c3onc(C)c3C)=O)C)C2)=O)ccn2ccnc2c1 C1(C(=O)NC2CC(NC(C=Cc3c(C)cncc3)=O)C2)Cc2c(F)cccc2O1 C(=O)(C1=NN(C)C(=O)CC1)N1CCC(C(C)NC(c2c(C)cccn2)=O)CC1 CC1CN(C(C2CCOC(=O)N2)=O)CCN1C(C1C2CCCCCC12)=O c1(C(=O)NC2CC(C)(NC(C=C(CCC)C)=O)C2)cnn(-c2ccccc2)c1C Cc1ncnc(C)c1C(N1CCN(CCNC(=O)CNC(=O)NC2CC2)CCC1)=O C1(CNC(C2ON=C(C)C2)=O)CN(C(=O)CN(C(=O)CCC)C)CC1O c1(C(N2CCC(NC(C(COC)(C)OC)=O)C23CC3)=O)cc(C#N)ccc1F N1(C(C(C)(C)CC2CC2)=O)CCC2(CC1)CC2NC(=O)Cc1ccno1 N1(C(CCCOCC)=O)CCC(CF)(NC(c2ncnn2C)=O)C1 C1(C(=O)NC2(C(=O)NCc3cnc(C)s3)CCCC2)CC(=O)CC12CCC2 Cc1cccc(Cl)c1OCC(N1CC(NC(C2(C)CCOC2)=O)C(O)C1)=O CCCC(C(=O)NCC1C(O)C(O)CN1C(=O)Cc1cnc[nH]1)S(N)(=O)=O CC1CCC(CNC(=O)CCOC2CC2)CN1C(c1cc[n+]([O-])cc1)=O C1(NC(C2(C)CC2(F)Cl)=O)CCCCN(C(=O)CC2CC3(CC3)C2)C1 CC1(C(=O)NCCC2CCCN(C(=O)CCCC#N)C2)CC2(CCC2)C1 N1(C(C=C(C)C)=O)CC2CC(C1)N(C(c1ccc(F)c(C3CC3)c1)=O)C2 C(c1ccc(O)cc1)=CC(N1CCCC(CN(C(=O)CCCCCBr)C)C1)=O Cc1cc(C(=O)NC2CCCC(CC(N3CCC(CO)C(O)C3)=O)C2)ncc1Cl C12(CNC(c3cc(C)[nH]n3)=O)CCC(C1)N(C(=O)CCC1CCC(=O)NC1)C2 C(=O)(C(C)C(O)C(C)CC)NC(C(N1C(C=C)COCC1)=O)CO CP(C)(=O)c1cnc(O)c(C(=O)NCC(O)CNC(=O)Cc2cnsc2)c1 c1(C(=O)NCCN(C(C(=O)N(C)C)=O)C)cc([N+](=O)[O-])nn1C C1(NC(c2cc(OC)ncc2)=O)(CO)CCCN(C(C2CCCSC2)=O)C1 c1(NC(c2ccc(CNC(C)=O)s2)=O)ccc(C)cc1 c1(OCC(=O)NC2C(CNC(C(C)C(C)(F)F)=O)C2)ccc(Cl)c([N+](=O)[O-])c1 C(N=c1ncc(F)c[nH]1)C1CCCC(N)C1.c12cnccc1C1CC(C1)C2=O C1(C(=O)NC2C(NC(c3c(OCCOC)cccc3)=O)C2)CC(F)(F)C1(F)F c1(C(=O)NCCN(C(C2CC(C)OCC2)=O)C)sccc1S(=O)(=O)C(F)F N1(C(C=CCCC)=O)CC2CCC(C(=O)NC3C4CCCC3CC4)(C2)C1 C1(NC(C2C(C)(C)C(NC(=O)C=C3CCOCC3)C2)=O)CC2(C1)CC(O)C2 C1(CNC(C2C(C(=O)OC)CC2)=O)CN(C(=O)CCN2CCNC(=O)C2)CC1O C(C)(C)(CC(=O)N1CCC(C(C)CO)CC1)OC1CCN(C(COC)=O)C1 C1(CNC(C(C)OCCOC)=O)CC2(CCN(c3ncnc(Cl)c3C#N)C2)CO1 C(CC1=CCN(C(=O)C(C)(C)F)CC1)NC(C1N(C)CC(O)C1)=O C1(C(=O)NCC2CC3CN(C(c4ncccn4)=O)CC23)CCCCC12CCC2 C(=O)(C#CC(C)(C)C)N1CC(CCNC(CCc2oc(C)c(Br)c2)=O)OCC1 N1(C(C(CO)N(C)C)=O)CCCC2(CCN(C(=O)CCc3csc(=N)[nH]3)C2)C1 c1(SCC(=O)NC2(C)CCN(C(C(CCOC)(C)C)=O)C2)ccc2n[nH]cc2c1F CC1CCC(NC(c2csc(-c3ccoc3)n2)=O)CN1C(c1ccccc1F)=O C(=O)(C(C)(F)C(=O)NCC(C)(CO)NC(c1sc(CC(C)C)nc1C)=O)OCC c1(C(N2CC(CNC(C(C)NC(C)=O)=O)OCCC2)=O)ccc(C(C)(C)C)cc1N C=CCC(C(=O)NC1CCCC1NC(c1nnc(S)n1C)=O)C(C)C S(=O)(=O)(c1cc(OC(F)F)nc(Cl)c1)N(C)Cc1c(C(C)C)nccc1.C(C)N N1(C(C(C=C)(F)F)=O)CCCCC(NC(=O)C(N2CCOCC2)C2CC2)C1 C(C(C)(O)C(C)C)NC(C(C)(N(C(c1ccc(CC)o1)=O)C)C1CC1)=O N1(C(CC(C)CF)=O)CC2(CCC2)CC1CNC(=O)CC1CN2CCC1CC2 CC1(C)CCCN(C(c2ccc(O)c(O)c2)=O)C1CNC(=O)COC1CCOC1 C1(CC=C)(NC(C2(COC)CCC2)=O)CC2CCC(C1)N2C(C1CCNC(=O)C1)=O CCC(C(=O)Nc1nc(C(=O)C(C)(C)C)cs1)c1ccccc1 C1(CNC(c2c(CC)noc2)=O)CC2(CC2)CN1C(=O)C(C)OCCN(C)C C1(C)(C(=O)NCC2(COC)CC2)CC(O)CN1C(=O)CCOC1CCCC1 C1(C2N(C(C=CC(CC)=CC)=O)CCC2)CCN(C(=O)C(N)=O)CC1 C(CN=C(NCC(=O)NCCc1ccc(Br)cc1)N1CCCC(C)(C#N)C1)OC N1(C(CCCn2nc(C)c(C)c2C)=O)CC2CCN(C(C3CC(F)C3)=O)CC2C1 c1(C(=O)NCC(C)NC(C(C(C)(C)C)OC)=O)nn(C)c2c1C(=O)CCC2 C1(C(=O)NC2CCC(C)N(C(C34CCC(C3)C4)=O)C2)COc2ccccc2C1 CC1CCn2c(C(=O)NC(C)(C)CCNC(=O)CC3NC(=O)NC3=O)cnc2C1 CC(C)CC(C)(C)C(=O)N1CCCC(CCNC(=O)CCCCCC#N)C1 c1(CC)cc(C(=O)NCCNC(=O)CCCCCNC(N)=O)ccc1C N1(C(C2(OC)CCN(C(C)CO)CC2)=O)CC2(CCC2)C1C1CCCO1 C1(NC(c2cnc(COC)s2)=O)CCC(F)(CNC(=O)CC2CCCO2)C1 C(=O)(C(CCF)NC(c1ccc(CO)o1)=O)NCCC(C)N1CCCC1 C(=O)(C1CCc2ccccc21)NC12CCCC(NC(COC(C)=O)=O)(C1)C2 C1(C(N2CC(CC)(NC(=O)CN3CCCC3=O)C2)=O)COCCC1(F)F C(C(=O)NC(CNC(C1(C(F)F)CCC1)=O)C(C)C)(C(C)C)NC(CC(C)C)=O N1(C(C(CC)CC)=O)CC2CC1CN2C(=O)Cc1ncc(C)s1 CCC(CC)C(=O)NCC(=O)NC1CC(CNC(=O)CCNC2CCCC2)CO1 N1(C(CCCCC)=O)CCC(C2(O)CCN(C(=O)CCCCC(=O)OC)C2)CC1 O=C(CC(C(F)F)c1ccccc1F)NC1CC(NC(N2CC3C=CC2C3)=O)C1 Cc1cc(N2CCC(NC(C3CCCO3)=O)C2)ncn1 C(CC(O)CC(=O)N1CC(C)(C)CC1CNC(c1ccnc(O)c1)=O)SC Cc1nc(O)nc(C)c1C(=O)NC1(C2CCN(c3ncnc4[nH]ccc34)C2)CC1 N1(C(CN2CCN(C)CC2)=O)CC2(CC2)CC1C(=O)Nc1cnc(Cl)cc1C(N)=O c1(C(C(C)NCc2cc(-c3c(F)cccc3F)on2)O)c(F)cccc1F c1(C2C(C(=O)NCCCC3(NC(CC4CC(=C)C4)=O)CC3)C2)c(C)cccc1C C12(C(c3ccc(Cl)cn3)=O)CCCC1N(C(=O)C(C(C)(C)C)=O)CCC2.CO C(CCN=c1[nH]c(Cl)ncc1Br)NC(C)COC(F)(F)F N1(C(C2(C#N)CCOC2)=O)CCN(C(=O)CC2CCSCC2)C(CC(F)(F)F)C1 CC1(C)C(CC(=O)NC(CNC(=O)CCc2ccccc2Br)CO)C1(C)C C12(CNC(c3cc(C(=O)OC)ncc3)=O)CCCC1CN(C(=O)C=CCO)C2 C1(CNC(C2CN(CCC)C(=O)C2)=O)CN(C(C2CCCN2C)=O)CCC1(F)F N1(C(C2(C)SCCS2)=O)CCC(=CCNC(C2CC3(CC3)CO2)=O)CC1 Cc1c(CC(=O)NCCC2(C)CCN(C(C3CC(CC4CC4)C3)=O)C2)cnn1C C12(CNC(CC=CC)=O)CN(C(=O)Cn3ncccc3=O)CC1CS(=O)(=O)C2 c1(OC)cc(C)c(C(=O)NCC2(CNC(=O)C3=CCCS3)CCC2)cc1OC Cc1nc(C2C(=O)N2c2ccccc2)sc1Br.c1(C(CSc2cnn(C)c2)=O)ccccc1 C(N=c1[nH]c(=NCCN(S(C)(=O)=O)CCO)c2ccccc2[nH]1)c1n(C)cnc1 C1(C(=O)NC(CC)C(C)(F)F)CN(C(c2ccc(CO)s2)=O)CCC1(C)C C1(C(N2CC(CNC(c3occc3Br)=O)OCCC2)=O)CCCC2CCCN12 C12(NC(CC(CC3CC3)NC(C=CCN(C)CC)=O)=O)CCC(CC1O)C2 C1(C)(CNC(C(CC#C)CC#C)=O)CN(C(=O)C(C)CC2CCCC2)C(C)(C)C1 C1(CNC(c2n(CC)ccn2)=O)CN(C(c2ccc(F)c(N)c2)=O)C(C)(C)C1 c1(CC(N2CC=CC(NC(C(CC(C)=O)(C)C)=O)C2)=O)c[nH]c2cc(Cl)ccc12 C12(C(N3C(CNC(CC(c4c(C)noc4C)C)=O)CC3)=O)CC(C)(C1)OC2=O CC1c2c(F)cccc2CCN1C1CC2CC1CN2Cc1ccc(NCCl)cc1 N1(C(CNC(C(CC)C)=O)=O)CC(C(=O)NC2(n3cncn3)CC2)C2(CCC2)C1 Cc1cncc(OCC(N2CC(F)(NC(=O)CCN3CCN(C)CC3)C2)=O)n1 Cc1n[nH]c(C)c1CC(C)C(=O)N(CCNC(=O)CC1CCS(=O)(=O)C1)C(C)C C1(NC(C(C)OCC)=O)CN(C(=O)CN(C)S(=O)(=O)N(C)C)CC1(C)C C#CCCCC(=O)NC(C)CC1CN(C(c2snc(Cl)c2Cl)=O)C1 C1(OC)CCN(C(C2(C3CC3)CN(C(=O)C=CCN3CCC3)C2)=O)CC1(C)C c12cc(on1)CCNC2=O.C(=O)(CN(C)CCOC)N(C)CC Cc1cccc(C)c1C(O)C(=O)NC1C2CN(C(c3ccsn3)=O)CC12 N1(C(CCC#C)=O)CC2CCC2(CNC(C2CC3C(C2)C3(C)C)=O)C1 C1(N(C(C(C(C)C)F)=O)C)CN(C(=O)COc2ccsn2)CC12CC2 c1(CN2CCC3(C(C(=O)NC(CCC)CCO)C3)C2)c(C)ccc(F)c1O C1(NC(CC(C)c2ccncc2)=O)C(C)(C)C(NC(c2ccc(Cl)s2)=O)C1(C)C C=CCC(C)(C)CC(=O)NCC1CN(C(=O)C(F)CN(CC)CC)CCC1(C)C C(C(C)(C)CC(=O)NCCC(C)NC(C1(Cc2ccc(F)cc2)CC1)=O)N(C)C CC1(C)OCC2CC12C(N1CCC(OCCNC(=O)Cc2cccnc2)C1)=O N1(C(c2c(CC)noc2)C(=O)NCC2CCOCC2)CC(C)C(C)C1 CCCCCC(C)(C)C(=O)OC(C)(C)C.C12CCC(=O)NC1C(=O)NC2 C1(NC(C(C2(O)CN(C(c3n(C)nc(O)c3)=O)C2)F)=O)CCCC(C)(C)C1 C#CCCCCCC(c1nnnn1C1CC1)NCC1(C)COCCO1 N1(C(CN(C(C(C(C)(C)C)O)=O)c2cccc(C(F)F)n2)=O)CCC(O)C(F)CC1 C(CCC(C)C(=O)NC(C)C(C)(C)NC(c1cn(CCOC)nn1)=O)OC C1(CC(=O)NCC=C)CCCCN1C(c1ccnc(O)c1)=O Cc1ccn2nc(C(N3CCC(NC(C4CCC5(CC5)C4)=O)C3(C)C)=O)nc2n1 CC#CCC(C(=O)NC1CC(CC)C1)NC(=O)CC1CCC(=O)NC1 C1(CNC(c2c(C)cc(F)cc2)=O)CCCCC1N=c1[nH]nc(C2CC2)o1 Cc1nn(CC(=O)NCCC2COCCN2C(=O)C(C)C#N)c(=O)n1C Cc1cnc2c(c1)N(S(=O)(=O)CCCCCC1CCC1)CCN2 c1(N2C(C)C(NC(=O)C=CC3CCOC3)CCC2)ncc2c(n1)CCCCC2 c1(C(N2CC(CC=C)(NC(=O)CC3CCN(C)C3)C2)=O)ccc[n+]([O-])c1 C1(C2CCCN(C(=O)C#CC3CCC3)C2)(NC(C2CCCC2CF)=O)CC1 c1(NC(CCC=C)C2CC2)nccc(=NCc2ccc(F)cc2C)[nH]1 N1(C(c2n(C)ncc2CNC(C2SCCS2)=O)=O)CCCCCC1CO CCCC(C)C(=O)NC(Cn1cncn1)C(=O)N(CCC(C)C)C N1(C(C(C(CC)C)NC)=O)CCCNC(=O)C12CCC2 CC(C)C(O)CNC(=O)C(CO)NC(c1cocc1C(N)=O)=O N1(C(CSCCCC)=O)CC(NC(c2cncc(C)c2C)=O)C2(CCC2)C1 c1(C(N(CC=C)CC)=O)snnc1C C1(C(N2CC(C3C(C)C3)C2)=O)(CO)CC2CCC1C2.C1C(C2CCC2)CC(=O)N1 c1(-c2cc(OC)c(C#N)cc2)cncc2sc(C(=O)NCCC(C)CO)cc12 N1(C(C(c2cc(C)sc2)(F)F)=O)CC2(CCCC2CNC(=O)C=CC=C(Cl)Cl)C1 C(C(=O)NCCCC(=O)Nc1ccnn1C1CC1)(C(C)C)N(CC)CC C(C(CC1CC1)C(=O)NCCCCCNS(C)(=O)=O)NC(=O)CCN1CCCC1 C(=O)(C1=NOC2(CCC2)C1)NC1CN(C(Cc2cccc(OC)c2)=O)C(C)(C)C1 C1(CCO)(NC(CC)=O)CN(C(=O)CC2CC(C(F)F)C2)C1 N1(C(c2cnc(CC(C)C)s2)=O)CCC(NC(C2C=CCCC2)=O)CC(C)(C)C1 C1(CC(=O)NC(CCNC(C(c2cccnc2)C)=O)(C)C)(N(C)C)CCCCC1 c1(CN2C(C(=O)Nc3n(C)ncc3Br)C3CCC2C3)c[nH]c2cccnc12 C=C1CC(C(=O)N(C)CCN2CCCCC2)(CNC(=O)C=C(CC)CC)C1 N1(C(C(c2c(C)cncc2)C)=O)CCN(C(C2(C)CC2)=O)CCC1C c1(C(N)=O)cc([N+](=O)[O-])ccc1NCC1CN(C(=O)C2=C(Cl)CCOC2)CCO1 c1(C(N2CC=CC(NC(C3(C)CC3(F)F)=O)C2)=O)cc2c(cc1Cl)OCO2 c1(CCOC(c2nnn(C)c2C2CCC2)=O)cc2ccccc2s1 c1(C(N(C)CCNC(=O)CC2CCC(=O)C2)=O)cccc(OCc2ccco2)c1 C12(CNC(=O)CCF)CC1CN(C(C1CCC(CN3CCCCC3)O1)=O)C2 N1(C(c2nc(-c3c(OC)cccc3)sc2)=O)CC(=O)NCC1C(=O)O C1(CCC)CCCN(C(=O)C(=O)NC2CN(CC3CC3)CC2C)CC1 Cc1nc(C=CC(=O)NCCNC(=O)C(F)(F)Cl)[nH]c1C N1(C(Cc2c(OC)cccc2)=O)CCCC(O)(C(=O)Nc2ccccn2)C1 C(=O)(C(C)C1=CCCC1)N(CC(CNC(c1c(OC)c(Cl)ccc1)=O)C)C CCC(CC(F)(F)F)C(=O)N(CCCN(C)C(C1CCC2CC2C1)=O)C C=CC(CCC)CC(=O)NC(C)(C)CC=CC(=O)N(C)CC1CN(C)C1 n1(CCCC)nc(C(C)Sc2nnc(SC)n2C2CNC2)c2ccccc2c1=O Cc1cn2ccccc2c1C(=O)NCC1(F)CCC(NC(C2(F)CC=CC2)=O)C1 C1(C(=O)NC2CC3(CC(NC(CCCC(=C)C)=O)C3)C2)CCCC(F)(F)CC1 c1(C(N(CCNC(CCCSCCCC)=O)CCOC)=O)cc(CO)oc1C N1(C(C=CCC)=O)CCOC2CN(C(=O)C(c3ccc(Cl)cc3Cl)C)CC12 c1(CC)cc(C(=O)NC2(C)CCCN(C(C34CC(C3)C4)=O)C2)ccc1F CON(CCC(=O)N(CC(O)C(C)(C)C)C)C(=O)c1cnn(CC2CC2)c1 C1(C)(C(N(C2CCN(C(=O)COCCCN=[N+]=[N-])C2C)C)=O)CCCCC1C N1(C(C2(CN(C)C)CC2)=O)CCC2C(CCN2C(=O)CCCc2ccccn2)C1 N1(C(C2C(C=C)OCC2)=O)CC2(CC(NC(=O)C(C)(C)COC3CCCC3)C2)C1 c1(C(=O)OCC2(C)CCC(C)CC2)ccc2c(c1)C(=O)NCCO2 N1(C(C(CCCC)O)=O)CC2CC(NC(=O)CCCC3CCCC3)CC2C1 Cc1c(C(c2ccccc2)NCc2cccc(SC(F)(F)F)c2)cc(Br)cc1F Cc1cc(C(=O)NC2CCC(NC(=O)CCCCn3ccnn3)CC2)nc(O)c1 C1(C(=O)NC(C)CN(C(=O)CCN2CCCCCC2)C)CCc2ccccc2N1 c1(C(N2CC(NC(C3(C#C)CC3)=O)C(F)CC2)=O)ccc(C#C)cc1F c1(C(N2CCC(N(C(=O)Cc3cccc(F)c3)C)C2)=O)cnc2n(c1=O)CCS2 N1(C(=O)Nc2n(CC)ncc2)CCCC(O)(CO)C1.c12cccc(c1)NC2C C(c1cccc(Cl)c1)=CC(=O)NC1CCN(C(c2ccncn2)=O)CC1F C12(NC(c3cc(C(CC)C)no3)=O)CCN(C(=O)Cn3ncc(O)nc3=O)CC1C2 c1(C(=O)NC(C#C)(C)C2CCCC2)coc(CNC(C2CC23CCC3)=O)n1 C(C(C(=O)NCc1ncccn1)NC(=O)C(Cl)Cl)N(C)C c1(C(N2CC(C(C)NC(C3(C)C(CC)CCC3)=O)C2)=O)ccc2c[nH]nc2c1 CC1CC(NC(c2sccc2Cl)=O)CN1C(c1cccc(O)n1)=O c1(CNC(C(C2CCCO2)NC(C2C=C(C)CS2)=O)=O)cccc(C)c1O Cc1cc2[nH]c(C(N3CC(O)(C(F)CNC(=O)CC4(C)CC4(F)F)C3)=O)cc2o1 N1(C(c2nc(C)sc2)=O)CC2CCC(NC(=O)C(C)C3CCCC3)CC2C1 C1(CNC(C2(C)CC2F)=O)(CNC(=O)C=CCF)CCOCC1 C12(C(=O)NCC(C)CNC(=O)CC(F)(F)C(F)(F)F)CC3CC(CC(C3)C1)C2 c1(C(N2CC(C(N(c3ccccc3C)CC)=O)OCC2)=O)ccccc1Cl.C(C)(=O)O Cc1cc(Cl)ccc1C(=O)NCCN1CCN(C(=O)C(F)(F)C2CCCC2)CC1 c1(C(CC)C)cc(C(=O)NCC2(NC(c3ccccc3)=O)CCCC2)on1 c1(C(=O)NCC2N(C(C(C)(CO)OC)=O)CCCC2)nc(C)ncc1Cl c1(C(N2CCOCC2CCC2CCCCC2)C(=O)NC(C)C)nc(F)ccc1Br c1(C(=O)NCCCNC(=O)CC(=O)NCC(F)(F)F)ccc(C2CC2)nc1 C1(NC(=O)C(C2CCC2)C2CC2)CC2CC1N(C(c1cn(C3CCC3)nn1)=O)C2 C1(NC(Cc2n(C)ncc2)=O)(CO)CCN(C(C2CC(C)(C)CO2)=O)CC1 c1(C(=O)NC2CC(NC(CN(S(CC)(=O)=O)C)=O)C2)cn2nc(C)sc2n1 CCCC(O)CC(=O)NC1CCN(C(=O)Cc2ccc(C)s2)C(C)C1 CC1(C#N)CCCN(C(=O)CC2CCN2C(C2CC2(F)Cl)=O)C1 C1(C)(C(N2CCN(C(C(C)OCCC=C)=O)C(C)CC2)=O)Cc2ccccc2C1 c1(CNC2C(C(=O)Nc3cnc(Br)c(Cl)c3)CCC2)cccc2c[nH]nc12 c1(N2CCC(COC)C2)nc(N(C)Cc2cc(C)ccn2)c2ccc(C)cc2n1 c1(C(N2C(C(=O)NC(c3ccc(Cl)cc3)C)CC(O)C2)=O)cc2cc(F)ccc2[nH]1 C1(C#N)(CC(=O)NC2(CCOC)CCN(C(=O)CSC(F)F)C2)CCCCC1 C1(C(=O)OC)CC(C)CN(C(CCc2cc(NC(=O)COC(C)=O)[nH]c2)=O)C1 C1(C(=O)NC2CN(C(C3CCCO3)=O)C2)CCCN1C(=O)CCc1ccccn1 N1(C(c2sc(Cl)nc2C)C(=O)NCC(=C)C)Cc2ccc(O)cc2CC1C N1(C(C)C)C(=O)COCC1C(=O)Nc1ccccc1.c12cc(c[nH]1)COC2=O c1(C(C(=O)NCCC(=O)OCC)N(C23CC(C2)C3)CC)ccc2nc[nH]c2c1 C1(NCc2cn(-c3cccc(S(=O)(=O)N(C)C)c3)nn2)CCc2c(nnn2C)C1 CCCCC(C)C(=O)N(CC(C)N(C)C(c1nc(C)ccc1F)=O)C C1(N(C)C(c2ccc(C(F)F)o2)=O)CC2CCC(C1)N2C(=O)CC1CCOC1 N1(C(c2c(C)cc(C)s2)=O)CCN(C)C(C(N2CC3(CC3)C2)=O)C1 CC1CCC(CNC(=O)CC2(O)CCOC2)CN1C(=O)Cn1cncn1 c1(OC)ccc2cc1-2.N1(CC)CC(C(C)CNC(C23CC2C3)=O)C1 C(=O)(C1=CC(O)CCC1)NC1CC(CCNC(=O)Cc2csc(S)n2)C1 C1(CC)CN(C(=O)C=Cc2ccc(OC)cc2)CCC1NC(=O)CC(C)CF C=CC1(C2(C(=O)NC3C=CCN(C(=O)C(CO)C(C)(C)C)C3)CCC2)CCC1 N1(C(Cc2cnn(C)n2)=O)CCC2(CNC(=O)Cc3cn(C)nn3)CCCCC12 C(=O)(C(CC(C)C)N(C)CC)NC(CC1CN(C(c2oc(CC)c(C)c2)=O)C1)C C1(C#N)(NC(c2cc(C)no2)=O)CCN(C(c2cccn(C)c2=O)=O)C1 CCCCCC(O)CNC(C1CC12CC(NC(c1coc(CCC)n1)=O)C2)=O N1(C(CC(CC)C)=O)CCCC12CCN(C(C1CCCCC13CCC3)=O)C2 Cc1cc(O)ncc1C(=O)NCC1C2CN(CC(=O)NCC3CC3)CC12 c1(-c2c(C)nccc2)cc2c(s1)CCN(c1nc(C(F)(F)F)nc3sccc13)C2 C(CCF)(C(=O)NCCOCc1nc[nH]n1)NC(=O)CC1CC1C1CC1 C1(C(N(C2CC(OCC)C2)C)=O)CC(OC)CN(C(C2CCC(O)C2)=O)C1 N1(C(c2c(F)cc(C)c(F)c2)=O)CCCCC2(C1)CN(C(=O)C(F)C(F)(F)F)C2 N1(C(COCCC#C)=O)CCCC(NC(c2cccc(O)c2F)=O)CC1 N1(CC(N2C(CNC(C(C)n3cncn3)=O)C=CC2)=O)CCC(F)CC1 N1(C(c2c(C(C)C)n(C)nc2)=O)CCC2CCC(C1)N2C(C1(C)CCC(=O)C1)=O Cc1ncc(Cl)c(C(N2CC(NC(c3ccc(F)cc3Cl)=O)C3CC23)=O)n1 C1(NC(C2CC(CCNC(C3CC(=O)OC3)=O)C2)=O)CCC([N+](=O)[O-])CC1 C12(C(N(CC(CCC)C)C)=O)CC1CN(C(=O)COc1ccn(C)n1)C2 C1(CNC(c2cnc(Cl)s2)=O)CCN(C(=O)CCn2cc[nH]c(=O)c2=O)C12CC2 c1(CNC2CC(CC(=O)NC3(c4cc(C)[nH]n4)CC3)C2(C)C)c(C)cccc1F CCC(C)C(C(C(=O)Nc1ccc2ccc(Cl)cc2n1)N1CCN(C)CC1)OC C1(C(=O)NC(c2nc(C)sc2)C)CC(F)(F)CN1C(c1cnsc1)=O C1(C(=O)NC(COC)C)CCN(C(=O)CCc2ccccn2)O1 c1(C(N(CC(O)CNC(c2cncs2)=O)C)=O)ncc(C(C)(C)O)cn1 Cc1nc2cccc(C(=O)NCC34CCCC3CN(C(=O)C(N)=O)C4)c2[nH]1 N1(Cc2[nH]nc(COC)n2)CCC2(CCN(C(C3(F)CCOC3C)=O)CC2)C1 N12CCC(C)CC1CNC(=O)C2.C1(C(F)(F)F)(C(=O)OCC)CCCC1 C1(NC(C(F)=CC)=O)CC(C)N(C(c2ccc(-c3csc(C)n3)cc2)=O)C1 C(CN=c1[nH]nc(C2CC2)o1)N(C(c1c(CC)oc(C)c1)=O)C C1(CNC(c2[nH]nc(OC)c2Cl)=O)COCCN(C(=O)CC(F)F)C1 c1(CC2C(CC(C)NC(C)CCCO)C2)ccc(Cl)cc1 C1(C)(c2cc(OC)cc(OC)c2)NC(=O)N(NC(=O)C2CCC(F)(F)C2)C1=O N1(C(CSC)=O)CCCC1CNC(c1cncc(NC)c1)=O N1(C(COCCSC)=O)CCC(C)C(N(C)C(c2cc3n(n2)CCC3)=O)C1 CC(C)(C(=O)NC1CC(CCNC(C2CCC(=O)O2)=O)C1)c1sccc1Cl N1(C(c2nc(C(C)OCC)sc2)=O)CCC(C)(CNC(=O)C2=CCOCC2)CC1 c1(OC(C2CC(C)CC(C)(C)C2)=O)cccc2nc(O)ccc12 CC1CCN(CC(N2CCC(C(=O)NC(N3CCOCC3)C)CC2)c2ccncc2)CC1 c1(C(=O)NCC2CC(C)N(C(c3cnc(C(F)F)s3)=O)C2)cc(Cl)c(N)c(Cl)c1 CC(Cc1ccco1)C(=O)NCCCCNC(c1c[nH]nc1-c1ccccn1)=O C(=O)(CCCCO)NCC(=O)NC1(CNC(C(C)OCC(C)C)=O)CCOC1 C12(CC(=O)NCC(C)(F)CNC(=O)C(c3ccc(F)cc3)F)CCCN1CCC2 C1(C(=O)NCCN(CC(=O)NC)CC)CCCN1CCC(C)C CC(C(O)C(=O)N1CC(N(C(=O)C(F)C2CCCC2)C)C1)c1ccccc1 C#CCC(N)=O.c1(CC(=O)NC2C(CNC(C)=O)C2)scnc1C Cc1cc(C)c(CC(=O)NC2CN(Cc3ccc(O)c(F)c3Br)CC2F)c(C)c1 C1(NC(COc2ccn(C)n2)=O)CCN(c2ccnc(C#N)n2)CC1O N1(C(C=C(C)C)=O)CC2CCCC1C2CNC(c1ncc(Cl)cc1F)=O CC1c2c(Br)cccc2CCN1C(c1sc2nccc(C)c2c1N)=O C1(NC(CC(=O)OCC)=O)CCCC(CNC(=O)CC2CCCOCC2)C1 C1(C(=O)NCCC2N(C(C3(CC)CCOCC3)=O)CCSC2)CC(S(C)(=O)=O)C1 N1(C(C(C)(O)C2CCOCC2)=O)CCC(NC(=O)CCNC(N)=O)C2(CCC2)C1 C1(NC(=O)C=Cc2ccc[nH]2)CCCCC12CCN(C(=O)C=CC1CC1)C2 c1(C(=O)NC2C(F)CCN(C(CNC(C)=O)=O)C2)ccc2cc(O)ccc2n1 c1(OC)cc(C(C(=O)NCCC2CC2)N(C2CC3C=CC2CC3)C)ccc1SC N1(C(C2C3CN(C(=O)Cc4cccc(Br)c4)CC32)=O)CCC2(CCOC2)C1 C1(CNC(CC2(NC(c3cc(C)oc3)=O)CC2)=O)CC2(C1)CC(O)C2 C1(NC(c2c[nH]nc2C2CCCO2)=O)CCCN(C(=O)C(=O)C(F)(F)F)CC1 c1(OCC)cnc(C(=O)NCC(C)CNC(c2nccc(SC)n2)=O)c(Cl)c1 c1(C(CC)NC(c2nc(C)ns2)=O)cccc(F)c1 c1(NC(C2N(C(CCCn3c(C)ncc3)=O)CC=C2)=O)ccc(Cl)nc1Cl CCC(CCC(=O)N1CCCC(OC)C1)NC(c1nscc1C)=O N1(C(C(CC)n2cccn2)=O)CCC2C(NC(=O)CCc3ccco3)CC12 Cc1ccc(CCCN)c(NC(c2sc(-c3ccsc3C#N)nc2C)=O)c1 C1(C(N2CCC(CNC(C(CCC)C)=O)CC2)=O)Cc2cc(O)ccc2CN1C Cc1cc(C(=O)NCC2(NC(c3cccc(OC(F)(F)F)c3)=O)CC2)cnn1 c1(CC)onc(C(=O)NCC2CCCCC2NC(=O)CCCOCCOC)c1C C1(NC(=O)COC(F)F)CN(C(c2ccno2)=O)C1 C1(NC(C2(OC)CC(C)C2)=O)CC2CN(C(C3CC(F)(F)C3)=O)CC2C1 C1(CC)CCN(C(C2CCC(O)C2)=O)C(C(N2CCC2CN=[N+]=[N-])=O)C1 c1(OC)ccc(F)c(C(N2CC3(NC(=O)Cc4cccc(F)c4)CC2C3)=O)c1F C1(COCC)CCC(CNC(C2CCCC2COC)=O)CC1.C1(=O)C(C)(C)N1.OC c1(CC)ncccc1C(N1CC(CCNC(c2ccc(CSC)o2)=O)C(C)C1)=O C1(CNC(C(COCC)C)=O)C(C)CCN1C(c1ccnn1COC)=O N1(C(c2cccc(OC)n2)=O)CCC(C)C(NC(=O)Cc2cc(C3CC3)on2)C1 N1(C(C2ON=C(C)C2)=O)CC(C2CC2C(N2CCCN(C)CC2)=O)C1 C1(NCc2c(N(C)C)cccc2Cl)C2CCOC2C1(C)C C#Cc1ccc(C(N2CCCC(C)(C)C2C(=O)NCc2csnc2C)=O)cc1C c1(C(=O)NC(CC)CN(C(=O)C=Cc2ccc[nH]2)C)cc(C)cc2ccoc12 C1(CNC(CNS(CC)(=O)=O)=O)(OC)CCN(C(C2(F)CCOC2C)=O)C1 c1(C(=O)NC(C)CCN(C(=O)Cc2cc(Cl)c[nH]2)C)ccc(-c2ccon2)cc1 Cc1cccnc1C(=O)NCC1CCCN(C(=O)CN2CCC(C)(O)C2)C1 c1(CN(C(=O)NCC23CCC(COC2)O3)C2CC2)c(Br)ccc2c1OCO2 C(C)(CCC(=O)NC1CCCSC1)NC(c1n(COC)ncc1)=O Cc1cccc2c1CCC2NC(c1ccc(F)c(OCF)c1)C(=O)NC1CCOC1 n1(C(C)C)ncc(C(=O)NCC(C2CCOC2)NC(c2coc(Cl)n2)=O)c1N C=CCCCC(C)(C)C(=O)NC1CC2CC(C1)N(C(c1cc(Cl)n[nH]c1=N)=O)C2 C(=O)(CCC(CC)NC(c1cscn1)=O)N1C(CC(=O)OC)CCC1 C1(NC(CNC(CNC(CCCOC(C)=O)=O)=O)=O)C(C)(C)C(O)C1(C)C N1(C(CC(C)Cc2ccco2)=O)C2CCC1(CNC(=O)C=CC(C)(C)C)CC2 c1(C(=O)NCC(C)N(C)C(C2(C)CCOC2)=O)cc([N+](=O)[O-])n[nH]1 CC(O)C(C)(C)C(=O)NCCC1CCCN(C(=O)CN2CCC(F)CC2)CC1 C1(C(=O)OC(COC(C)=O)CO)CCCN(C(c2nc(C)no2)=O)C1 c1(CC)cccc(C(=O)NC(C)(C)CCCNC(=O)CCF)n1 c1(NC(C(C)OCCOCC)=O)ccccc1CNC(=O)C=Cc1cn[nH]c1 C1(C(=O)NC(C)CNC(=O)C=C2CCCCC2(C)C)CC2(CCCCC2)C1 c1(C(N(C)CCNC(C2CC2C2(C)COC2)=O)=O)ccc2cc(Br)ccc2n1 N1(C(c2cc(C)n(C(C)C)c2C)=O)CCCCc2ccncc21 C(C(C)(O)CNC(=O)C(CC1CCOCC1)NC(=O)CCc1ccc[nH]1)OC C1(CNC(c2ncoc2C2CC2)=O)CC(F)(F)CN1C(c1ccc(O)nc1Cl)=O n1(C(C)C)cccc(C(=O)NCC2CN(C(c3n[nH]cc3Cl)=O)CCC2C)c1=O c1(C(N2CC3CC3(N(CCF)CC)C2)=O)c(F)ccc(OCc2ccccn2)c1F C=C1CCN(C(CC2CCC3CC23)C(=O)NC2CCC(C(=O)OC)C2)CC1 C1(NC(C2(COC)COC2)=O)CCN(C(c2cnn(C3CC3)c2Cl)=O)C(C)C1 CC(C)(C)CCCC(=O)NC1CC2(CCN(C(=O)Cn3ccc(=N)[nH]3)C2)C1 C1(c2cn(CC(C)(C)C(F)F)nn2)CCCC(=O)CC1 C1(C(=O)NC2CCC3CC23)(COC)CN(C(c2cn(C)cn2)=O)C1 C(=O)(CC(C)(C(F)F)N(C)C)NC1CC(NC(C(C)Cc2cccc(Br)c2)=O)C1 c1(C(N2CCC(N(C(=O)C(C)c3cc[nH]n3)CC#C)C2)=O)sc(C)cc1C c1(OC)ccc2nc(C(=O)NC3CCN(C(=O)CSCCC(C)C)CC3)cn2n1 c1(C(=O)NCC2(O)CCN(C(=O)C=Cc3cnc[nH]3)C2)cc(F)cc2cc[nH]c12 C1(NC(C(C)C(F)(F)F)=O)CN(C(c2nc(Cl)ccc2N)=O)CC2(CCC2)C1 C12(C(N3CCCC3)=O)CCC(ONC(C(c3ccc(OC)cc3)N(C)C)=O)(CC1)C2 C1(CCN(C(=O)Cc2ccccc2O)C)CCCC(NC(=O)COCC(N)=O)C1 c1(OCC(=O)NCC(C)CNC(=O)CCC(=O)NN(C)C)ccc2c(c1)CCCC2 C1(C(=O)NC2(CCCCC)CC2)CCCCC1CNC(=O)COC1CCCOC1 CCCCCC(C)(C)C(=O)NC1CCN(C(=O)CCF)C(c2ccccc2)C1 C(=O)(CC1NC(=O)c2ccccc21)N1CCC(N(C)C(C2CCOCC2)=O)C1 c1(C(N(CC(CN(C(C(CC)=CC)=O)C)O)C)=O)cccc(COC)c1 C1(OC)CC2N(C1)C(=O)C1CC1C(=O)N2.c1(N(CCC(C)C)C)ccncc1 C(=O)(CC(C)O)N(CCC(=O)NC(COC)C)CCCO c1(C(=O)NC(CC=C)CNC(C2CC2F)=O)cc2cccn2cn1 N1(CCCC(=O)Nc2nnc(-c3n(C)ncn3)o2)CCc2ccccc2C1 C1(NC(c2c(CNC(CC3CCC(C)(C)C3)=O)ccs2)=O)(CO)CC2(CCC2)C1 c1(C(NOCCCCC=C)=O)nn(-c2ccccc2Cl)c(C)cc1=O C1(S(N)(=O)=O)(C(=O)NC2CC3(C(NC(c4c(C)n(C)nc4)=O)C3)C2)CCCC1 c1(C(N2CCC(N(C(=O)CCC(F)(F)F)CC)C2)=O)sc2cc(F)ccc2c1C C1(NC(c2cc(N(C)C)ncc2)=O)CN(C(c2cnns2)=O)C2(CCOC2)C1 CC(c1cnn(C)c1)=CC(=O)NC1CN(C(C2(C#N)CC(=O)C2)=O)C1 c1(NC(C(C)(C)OC)=O)cccc(N2CCN(Cc3ccnc(Cl)c3)CC2)c1 C1(C(=O)NCCC(C(=O)NCc2nc(COC)sc2)OC)CC2(C1)CC(C)C2 N1(CC(N2CCCC(C(=O)NC3CC4COC(=O)C34)C2)=O)CCS(=O)(=O)CC1 C1(C(=O)NC2CCCC2CN(C)C)(NC(C(C=CC)O)=O)CCOCC1 Cc1c(Br)cnc(O)c1C(=O)OCC12CC(CO1)N(C(=O)OC(C)(C)C)C2 n1(CC(=O)NC2CN(C(c3cc(CCC)on3)=O)CC2F)ccc(=O)c(O)c1C N1(C(C(c2n(C)ncc2)O)=O)CC2(CC(C(=O)NCCCCn3ccnc3)CO2)C1 c1(C(N2CCC(CN(C(Cc3cnc(C)s3)=O)C)C2)=O)ccc(Cl)cc1 CC1(C)CCC(C(N2CC3CC2(CNC(=O)CC2CC2)C3)=O)CO1 C(=O)(C1=CCSC1)NC1CN(C(=O)C(Cc2ccoc2)Oc2cccnc2)C1 c1(C(=O)NC2COCCN(C(c3cccc[n+]3[O-])=O)C2)cn2cc(Cl)cnc2n1 C1(C(=O)Nc2cnccn2)C2CC1N(C(c1cncc(O)c1)=O)C2 C1(C(N2CCC(O)CC2CC)=O)(CC)CCCN(C(C2CCOC2C)=O)C1 C1(n2c(C(N(C(CNC(C(C)(C)OC)=O)C)C)=O)cnn2)CCS(=O)(=O)C1 c1(C(=O)NC(C)CCNC(=O)CCC2CC(C)CO2)cccc2c1ncn2C c1(C(N(CC(CCC)O)C)=O)ccnc(CNC(=O)CCOCC2CCC2)c1 Cc1coc(C(C)C)c1C(N1CCCCC1CN(C)C(C12CCC(C1)OC2)=O)=O C(CC(O)CNC(C1CCC2CC12)=O)NC(c1cncs1)=O O=C(CCC(F)(F)C(F)F)NC1CC2CC(C1)N(C(=O)C=CC1CCCO1)C2 N1(C(C(COC)NC(C)=O)=O)CC2CCC(C1)C2CNC(c1nnc(S)n1C)=O N1(C(C(C2CC2)SC)=O)CCC(OCC(=O)Nc2cn(CC(F)(F)F)nn2)C1 CC(CC1CC1)C(=O)Nc1cc(Cl)on1.n1(CCNC)cccn1 N1(C(C2C(C)CCCC2)=O)CCC(CO)C(NC(=O)CC23CNC(=O)C(C2)C3)C1 c1(NC)ccc(F)cc1C(=O)N(CCCN(C)C(C1(CC2CC2C)CC1)=O)C c1(OCCCC2(NC(C(C)C)=O)CCC2)ccc(C(N2CC(O)C(F)C2)=O)cn1 N1(C(CSC(C)(C)C)=O)CCN(C(c2ccn(CC(F)F)n2)=O)C(CC2CC2)C1 c1(OC)ccc2nc(Nc3ccc(CN4CCCCC4)c(Cl)c3)[nH]c2c1 CCCC(O)CC(=O)NCC1CC(NC(=O)COc2cc(C)on2)CCO1 CC(CNC(=O)NC(c1ccccc1)CN(C)C)N=[N+]=[N-] C1(N(C(C)=O)C)CN(C(C2CC23CCSCC3)=O)CC1(C)C C1(NC(C2CN(CCC)C(=O)C2)=O)(CO)CCN(C(=O)CC2(C#N)CC2)CC1 c1(C(=O)NCC2C=CC(NC(C=CCN(CC#C)C)=O)C2)nccc(Cl)c1Cl CC1(C)CCC(CCNC(=O)C(C2CC2)NC(=O)COCC2CC2)C1 c1(C(=O)NCC2CCC(NC(C3(CC4CC4)CC3)=O)C2)ccc(Br)c(O)c1 N1(C(C(=O)CC2CCC23CCC3)=O)CCCN(C(=O)N)CC1.C1(O)(N)CCCC1 C1(C2(O)CN(C(c3cnc(C4CC4)s3)=O)C2)(CNC(Cc2c(C)nc[nH]2)=O)CC1 c1(C(=O)NCC(N(C(C2(C#C)CC2)=O)C)C2CC2)sccc1CC C1(NC(CC2(C)CCCC2)=O)(CO)CCCN(C(C2CC3(CCC3O)C2)=O)C1 CC(C)S(=O)(=NC(=O)c1cnn(CCn2ccnc2)c1)C(C)C C1(CCNC(c2cc(CF)on2)=O)CCCCN1C(c1cc(C(F)F)ccn1)=O Nc1cc(C(=O)NC2CC(NC(C3CCCCNC3=O)=O)C2)cc(Cl)n1 c1(CC)cc(C(N2CC(CCNC(C34CCCC3C4)=O)C(C)C2)=O)ccc1C CC(C)(C(=O)N1CCC1C1CCC1)C1=CCN(C2CC2)C1.c12cc(ccn1)NC2=O c1(OC)cc(C(N2CC(C)(NC(c3cnc(C)nc3)=O)C2)=O)c2ncccc2c1 C1(C2CC2)(C(=O)OCC)CCN(C(=O)Nc2cnc(N3CCCCC3)cn2)C1 CC1CC2CCCCC2N(C(c2noc3ccc(F)cc23)C(=O)NC2CCC2)C1 c1(C(N2CCN(CC(C)NC(CCCCCC)=O)CC2)=O)cc(C#N)ccc1O C1(NC(COC)=O)CC(C)CN(C(C2CCC2CC(=O)OC)=O)C1 Cc1coc(C(N2CCC(Oc3ccccc3F)C2C)=O)c1C C(N=c1[nH]c(C(N2CCCC2)=O)nc(=N)[nH]1)c1c(CC)n[nH]c1 CC(C)S(=O)(=O)CC(=O)NC1CCOC1C1CCN(C(C2(CCO)CC2)=O)CC1 N1(C(c2c(OC)n(C)nc2)=O)CC(NC(=O)CCC(=O)c2cccs2)CC(C)C1 CC(C)C(C(=O)N(C)CC1CCCOC1)NC(c1coc(C(F)F)c1)=O N1(C(C(C)S(C)(=O)=O)=O)CCC2(CC1)CC2CNC(c1cc(F)cc(F)c1F)=O C=CCC(CC=C)C(=O)N(C1CCCN(c2ncnc(O)c2Br)CC1)C c1(CNC(C2(CCNC(CSCCOC)=O)CC2)=O)cc(C)nc(C)c1 C(=O)(C1=NOC2(CCCN(C(=O)C=C3CCC3)C2)C1)Nc1ccc(OC)cc1C c1(C(C(=O)NC(C)C(=O)OC)N(CC)CC2CCCCC2)cnc(OC)c(Cl)c1 C(=O)(C1=CCCCO1)NC1(CCNC(C2N(CC)CC2)=O)CCC1 CC(C)C(CNC(=O)COC(C)C)C(=O)NC(C)C(F)(F)F C1(O)(CC#C)CCN(C(=O)C(CN(C)C)NC(C2CN(C)C(=O)N2)=O)CC1 C=CC1CCN(C(c2ccnc(CNC(=O)Cc3ccccc3O)c2)=O)C1 Cc1cccc(C)c1C(=O)NC1CC(CC(N2CCNC(=O)C2C)=O)C1 Cc1cnc(C(=O)NCCCCN(C)C(C2(C)CCC(=O)NC2)=O)c(F)c1 C1(C(C)NC(C(C)OCC)=O)CN(C(=O)CCNC(C2CCC2)=O)CCO1 CC1CN(C(=O)COc2ccsn2)CCC1NC(=O)CCCC1CCCC(=O)N1 CCCCC(C)CCC(=O)NC12CCC(C1)N(C(c1cn(C)nc1C(C)C)=O)C2 C(CC(C(C)(C)C)NC(=O)CC1COC(=O)C1)N(C(=O)CP(C)(C)=O)C Fc1cc(F)c(Cc2nc(-c3ccc(Cl)cn3)nn2C23CC(C2)C3)cc1F CC1(C)CN(C(=O)CCCn2cccc2)CC1CNC(=O)CN1CC=CC1 CCC1=C(C(=O)NCC2CC3CCC2N(C(c2cocc2C)=O)C3)SCCO1 C1(C(=O)NC)COCCN1C(C1CCN1C(=O)Cc1cc(C)no1)=O c1(COC)cc(C(=O)N(CCCNC(c2c[nH]c(Br)c2)=O)C(C)C)no1 C1(C(=O)NC2C(OC)CN(C(=O)CCS(C)(=O)=O)C2)CC(C)CC(C)(C)C1 C1(C)(C(N(CC(CC)O)C)=O)C=CCN1C(c1cccc(O)c1)=O CC(C)C(CC(=O)N1CC(NC(c2cc(Br)cnc2N)=O)CCC1C)C(C)C c1(CC)ccc(Br)c2nc(NC(C3CC(C)C3)=O)sc12 CCCCCCCCC(C)CC(=O)Nc1ccc(NC(=O)C(O)CSC)cc1C c1(C(N2CC(C)(CNC(C3CC34CCC4)=O)OCC2)=O)n[nH]c2nccc(Cl)c12 c1(CC=C)cccc(C(=O)NC(CNCCOCCN=[N+]=[N-])C(=O)NC)c1 C1(CC(=O)NC2C(NC(c3[nH]cc(CC(C)C)c3)=O)CC2)CCCCCCC1 Cc1ncnc2c1CC(C(=O)NCC1(O)CN(C(C3CCNC(=O)C3)=O)C1)CC2 C1(CC(=O)NCC)C=CCCC1.C12(CCC1)CC(=O)N(CCC#C)CC2 Cc1cnc(C(=O)N(C)CCn2cc(CCC(=O)CCN3CC4CC4C3)nn2)cc1Br C=Cc1cc(C(=O)NC2CCN(C(C3CC(OC)C3)=O)CC2O)cc(F)c1 c1(C(=O)NC2(CC=C)CN(OC(=O)CCS(C)=O)C2)n[nH]c2cc(C)ccc12 c1(CC2(C)COC2)cn(Cc2csc(C(F)(F)F)c2)nn1 Cc1ccc([N+](=O)[O-])cc1NC(C1CCC1CC(=O)O)=O c1(OCCCCNCC(CNC(=O)OC(C)(C)C)(C)O)cccc(F)c1 c1(C(=O)NC2CC3(C2)CN(C(=O)CC2OCCO2)C3)ccc(=O)n2c1CCCC2 C1(CN(C(=O)CC2OCCCC2(C)C)C)CCC2(CCC(C)(C)CC2)O1 C12(C(N3CC(CC(C(=O)NC4(C#C)CCOC4)F)C3)=O)CCC(CO)(CC1)C2 N1(C2CN(C(N3C(SC4CC4)CCC3)=O)C2)CC(C(=O)Oc2cnn[nH]2)CC1=O Cc1cccc(CN2CCC3(CC3C(=O)NCc3cnnn3C)C2)c1F N1(C(CCCC(C)C)=O)CC2(CCC2)CC1C(=O)NC(C)CN1CCCC1 CS(=O)(=O)c1sccc1C(=O)NC1C2CCC1CN(C(=O)C1=NOCC1)C2 N1(C(c2cc(C3CC3)ccn2)=O)CCCC1C1CCCN1C(=O)C=Cc1cscn1 CC1C(=O)N1.C(C(O)CNC(=O)C(C)C1CC1)N(C(C)(C)C)C(=O)O.CCC#N Cn1c(O)nc2c(C(=O)NCC3(NC(c4cc(Cl)c[nH]4)=O)CC3)cccc12 c1(CN2CCC(NC(c3cc(C)oc3C(F)(F)F)=O)C2)c[nH]cc(Cl)c1=O C(=O)(CC(CCCC)NC(=O)C(C)(C1(C)CC1)OC)N1C(CC#C)CCC1 C(C(N=[N+]=[N-])C(=O)[N+](CC(C)CC(=O)N(C)CCOC(F)F)(C1CCC1)[O-])OC c1(C(=O)OC)ncc(Br)cc1-c1cn(C(C)COC)nn1 c1(CC)cc(C)c(C(=O)NCc2ncc(C(N3CC(n4ccnn4)C3)=O)cn2)o1 S(=O)(=O)(C1CC2C=CC1C21CC1)C(C(C)CC1CCCC1)=O C1(CNC(COCCCC)=O)C2CCCC1N(C(C1(O)CCSC1)=O)C2 CC(C(=O)NCC(c1ccccc1)Nc1cc(OCC#N)ncn1)S(N)(=O)=O c1(C(=O)NCCN(C(=O)C(C)(C)N(S(C)(=O)=O)C)C)cc2c(s1)CCC2=O CCC(C)C(C)C(=O)NCCCN(C(=O)CCc1ccccc1O)C1CCCC1 C(C)(C(CC(=O)N=c1cc(C(N)=O)n(C)[nH]1)NC(c1sccc1F)=O)OC c1(CC(N2CCOC(CNS(=O)(=O)CCCCl)C2)=O)ccc2ccccc2c1Cl c1(C(=O)NCC23CC2CN(C(C2CC2C2CCC2)=O)C3)cc2cn[nH]c2cn1 C1(NC(c2c(C)nsc2Cl)=O)CCCC2CN(C(C3CSC3)=O)CC12 C1(C(C)C)(C(=O)NCCN2CCOCC2)CCCN1C(c1ncn(C(C)C)n1)=O N1(c2n3c(nn2)C3)CCn2ncc(Br)c2C1.C1(C)CCCCO1.C(COC)OC N12CC3CN(C3C1)Cc1cccc(c1)C2=O.N1(Cc2cnco2)CCCCC1 c1(C(N2CCC(C(C)NC(=O)CC(C)(C)O)CC2)=O)n[nH]c2ccc(O)cc12 N1(C(=O)C(N2CC=CC(O)C2)=O)CC2CCCC1C2 C1(NC(=O)NCCn2ncc(C(=O)OC)c2)CCCN(CC(F)(F)F)CC1 C1(C(N2C(CNC(C(C)CO)=O)CC2)=O)COC2CCCCC12 CCC(C)(C)C(C)NC(=O)C(CCSC)NC(c1sc(C)nc1C)=O CC1CCC(C)(C(N2CCC(CN(C)C(c3cn[nH]c3)=O)C2)=O)C1 c1(C(=O)NC2CN(C(C3(C)ON=C(C)C3)=O)C3C2C3)c[nH]c2cccc(F)c12 CC1CN(C(=O)Cc2ccc(-c3ccc(C#N)cc3)cc2)Cc2c(Br)cccc21 c1(CC(=O)NC(CNC(C(C)C2CCOC2)=O)(C)C)cncnc1 c1(C(N2C(CNC(C3N(CC)CC3)=O)CC3CC32)=O)cc(C)cc(C)c1C N1(C2CCN(C(=O)C=CC3CCCO3)C2)CCS(=O)(=O)CC1 CCC(CC)C(C)C(=O)NCC1(OC)CCN(C(c2ccc(C#N)c(C)c2)=O)C1 N1(C(C(C)(C)C2CCOCC2)=O)CCOC(CNC(=O)Cc2cncc(F)c2)C1 c1(C2(C)CC2SCCCCCl)ccccc1F N1(C(C(c2scc(C)n2)C)=O)CCCOC(CNC(c2cccc(Cl)c2C)=O)C1 c1(C(N2CCC(NC(CSCCC)=O)C(O)C2)=O)nn2c(c1C)CCCC2 C1(CNC(CCOCC)=O)CC2CCCCC2N1C(C1CNC(=O)N1)=O N1(C(COCCCC(C)C)=O)CCCCC1CCNC(c1sccc1CC#N)=O N1(C(c2nn(C)cc2Cl)C(=O)NCCOCC)Cc2c(F)ccc(Br)c2C1 N1(C(c2c(C)scc2)=O)CCN(C(=O)Cn2cc(C3CCOC3)cn2)CC1CO N1(C(C(CCC)OC)=O)CCC2(CCCCN(C(=O)CCC(C)(C)F)C2)C1 N12CCC3CN(CC13)NC(=O)C2=O.c1(C(C2CC2(Cl)Cl)C)ccc(F)cc1 CCCC(CCC)CC(=O)N1CC2CC2(NC(c2cnc3cc(C)ccn23)=O)C1 n1(CCC(N2CC(C)N(C(=O)CN(C)C(C)C)CC2)=O)ccc2cccnc12 C1(C(=O)NC(C)CNC(c2ncccn2)=O)C2CCCCCC12 CC#CCCC(=O)NCCn1cc(C(=O)N(CC(C)CNC(=O)OC)C)cn1 N1(C(c2ccc(COC(C)C)cc2)=O)CCCC(NC(C2C3CCC23)=O)CC1 N1(C(C2CC(OC(C)(C)C)C2)=O)CCCC2(CC(NC(=O)CCP(C)(C)=O)C2)C1 C(c1cccc(CO)c1)=CC(=O)NC1CCCN(C(=O)C2=CCC2)CC1 C1(NC(c2c(CC)cccc2)=O)CC(NC(c2scc(C)c2Cl)=O)C12CCC2 Cn1cnc(C(=O)NCC2(NC(C3COCCO3)=O)CC(F)(F)C2)cc1=O Cc1cc(C)c(C(=O)N(C(C)CCNC(C2CC2c2nc[nH]n2)=O)C)cc1N C1(NC(c2cc(C(C)=O)sc2)=O)CC2CC(NC(=O)CCC(=O)NN(C)C)CC2C1 C(=O)(CCC(C)(C)F)NCC(C(=O)NC1CCC(c2n(C)ccn2)C1)(C)C C(=O)(CCCCC(=O)NC1COCCC1C(=O)NCc1nccc(OC)n1)OC c1(C(N(CC(CN(C(c2c(C)cccc2F)=O)C)O)C)=O)cnc([N+](=O)[O-])n1C c1(OC)ccc(C(=O)NC(C)CCNC(=O)CC2(C(F)F)CC2)c(C(F)(F)F)c1 C1(CNC(C2CC=CCC2)=O)CC2CCC(C1)N2C(=O)Cc1cn[nH]c1 c1(-c2n(CCN(C)C)nc(-c3nc(C(F)(F)F)cs3)n2)cc(Cl)c([N+](=O)[O-])[nH]1 c1(C(N2CCC(C)(CNC(C3C(C)CCO3)=O)C2)=O)nn2c(c1Br)CCC2 N1(C(c2cc(OC)ns2)=O)CC=C(C(=O)NCC2CC2c2ccoc2)C1 C(C1=NOC2CCCC12)NC(=O)C1=CCN(C(C2CC23CC3)=O)C1 C(c1cc(C)ccc1OC)=CCN(C(C(=O)N(CC(CC)OC)C)=O)C N1(c2cc(NC3CC(CC)C3)nc(C)n2)Cc2cc(Cl)ccc2C(C)(C)C1 c1(CC(=O)NCC2CN(C(C(C)(Cl)Cl)=O)C2)ccc2c(c1)OCO2 N1(C(c2ccc(N)cc2F)=O)CCC2(CCCN(C(C3(O)CCC3)=O)C2)C1 Cc1ccnc2c(C(N3CCC(N(C)C(C4CCC4)=O)C(C)C3)=O)cccc12 C1(N(C(=O)CC2CCOC2)CCC)CCN(C(c2cc(CO)on2)=O)CC1 Cc1c(Br)c(C(=O)NCC(C)(CC(C)C)NC(C2CC23CC3)=O)nn1C C1(C(=O)NCC2C(NC(c3cc(C)no3)=O)C2)CCC(C)(C)CO1 Cc1ccc(C(N2CCC(C(C)NC(C3(C(F)(F)F)CC3)=O)CC2)=O)cn1 CN1CCCN(C(=O)C(C)(C)CCNC(=O)Cc2cnsc2)CC1 c1(CC)ccccc1NC(=O)C(c1cccc(F)c1)N(C)C(C1CCCC1)C c1(C(CC)NC(c2ncc(C)o2)C)ccc(OC)c(Cl)c1 c1(N(C)C)cccc(NC(=O)NCCc2cc(C(F)F)ccn2)n1 C(=O)(C#CC1CCCOC1)NCCOC1CCN(C(C(CCC)OC)=O)C1 c1(CC(N2CCCC(NC(Cc3n(C)cnn3)=O)C2)=O)c(F)cccc1Br C1(=O)C(O)(C(F)(F)F)CN1.N1(C(CN(C)C(=O)C2CC2)=O)CCOC(C2CC2)C1 c1(OC)cc(C(=O)NC2CN(C(=O)CCCC(C)=O)CC2F)ccc1OC(F)F C=CC1CN(C(c2cc(Cl)cn2C)=O)CCC1CC(=O)O Cc1cc(Cl)cc(C)c1CN1C(C)CC(NC(=O)CNC(C2CCOCC2)=O)C1 CC1CN(C(c2ccc(C(F)F)nc2)=O)CC1CNC(C1(F)CC=CCC1)=O c1(C(N2CCCC(CCC(=O)N3CCC3C(=O)O)C2)=O)ccc2c(c1)CCC2 N(C(=NCCSC)NC1CCOc2c1ccc(Cl)c2Cl)CCC(=O)NC C1(C)(CNC(c2nc(CC(C)C)sc2)=O)CCN(C(c2coc(N(C)C)n2)=O)C1 c1(C(N2CCC=C(CNC(C3CCCOC3)=O)C2)=O)cnn2ccc(Cl)c(F)c12 C1(NC(c2cc(CCC)[nH]n2)=O)CCC(O)CN(C(c2nccc(Cl)c2F)=O)C1 CC1CC(=O)NC(C(N2CC(CNC(=O)CC3CCOC3=O)C(F)(CO)C2)=O)C1 c1(C(N2CCC3CN(C(C4C(=C)CC4)=O)CC3C2)=O)c[nH]c2cc(C#N)ccc12 N1(C(c2c(N)cccc2Cl)=O)CC2(C1)CN(C(C1CC13CCOC3)=O)CC2CO C1(C(N(C2CCC(NC(c3ccc(O)nc3)=O)C2)C)=O)Cc2ccc(F)cc2O1 N1(c2ccc([N+](=O)[O-])cn2)CCC2C(CCCN2CCC2CCCCO2)C1 c1(OC)ccccc1C(C)NC(C1CCN(C(=O)Cc2nc(O)n[nH]2)CC1)=O c1(C(=O)NCC2(CNC(c3c(CC)cccc3)=O)CC2)ccc(N)c(C)c1Cl c1(C(=O)NC(C(C)NC(c2cc(OC)n[nH]2)=O)C)cc(O)ccc1Cl Cc1ccc2c(C(=O)NC3(CO)CN(C(=O)CCCCC#N)C3)csc2c1 CC(=O)CCC(=O)NC12CC(NC(c3sccc3C)=O)(C1)C2 C=CCCC(C)C(c1nnnn1-c1c(C)cccc1C)Nc1ccc(Cl)nc1C C1(O)(CC(=O)NC(C(=O)NC2C(CCC)C2)C2CCC2)CCCC1 c1(C2C(C(N(c3cnn(C(C)C)c3)CCC)=O)C2)cc(F)cc(Br)c1 N1(CCC(=O)NC2(C(=O)NCCC3CC=CCC3)CCC2)CCOCC1 c1(C(C(N2CC=CC(NC(CCCC=C)=O)C2)=O)O)cc(Cl)cc(Cl)c1 c1(C(C)(C)SC)cn(CCC(=O)Nc2cc(-c3ccccn3)on2)nn1 n1(C(C)C(=O)NCCCCNC(c2ccc(-c3cc[nH]n3)s2)=O)cnc(C#N)n1 N1(C(C(=O)NC2COC2)=O)CCOC(CCc2cn(Cc3ccccc3)nn2)C1 c1(C(=O)NCCN(C(c2ccc(CC)cc2)=O)CCOC)nn(C)c(Cl)c1Cl N1(C(c2ccc(Br)cn2)=O)CC2(CCC2)CC1Cc1nn[nH]n1 CC(O)(C(=O)NC1CCCC(NC(=O)CC2CC3(CC3)C2)C1)C(F)(F)F CC1CC(NC(C2CC2(C)C(F)F)=O)CCN1C(=O)Cn1nc(Cl)ccc1=O C1(C(=O)NCCc2nc(CC)on2)CCC2CCC1N2C(c1cocn1)=O C(CCN=c1[nH]c(Cl)nc2c1CCC2)N(C(=O)CCC1(C)CCCO1)C Cc1ccc(C(C)NC(c2nccs2)C)c2[nH]ncc12 c1(OC)ccc2c(c1Br)OC(F)(F)O2.C=Cc1cccc2c1CO2 C(N=c1[nH]c2cc(F)ccc2o1)C1(NC(C(C)=C2CCCC2)=O)CCCCC1C Nc1cc(Cl)ncc1C(N1CC(F)(F)CC1CCNC(C12COCC1C2)=O)=O c1(CNC(C2C=CCCC2)=O)ccc(C(=O)NC(CC2CC2)C2CC2)cc1 C1(C2CC2)(NCC(C)CS(C)(=O)=O)CCN(C(=O)OC(C)(C)C)C1 C1(CCOC)(NC(C2CCC(=O)NC2)=O)CCN(C(=O)CN2CC=CC2)C1 Cc1csc(C(C)NC(=O)CC(C)NC(c2ccoc2Cl)=O)n1 C1(CNC(C(c2cnn(C)c2)OC)=O)CC(C)N(C(C2CCCN(C)C2)=O)C1 N1(C(C(CC2CCCC2)NC(c2c(C)oc(Cl)n2)=O)=O)CCn2c(cnc2C)C1 c1(C(N2CC(CC(C)NC(C3=NOC(C)C3C)=O)C2)=O)cc(S(N)(=O)=O)n(C)c1 N1(Cc2cccc(C)c2F)CC2(C)CN(C(=O)C(C3CCCCC3)=O)CC2(C)C1 Cc1cc(=O)oc(C)c1C(N1CC(OCCNC(=O)CC2CN(C)CC2O)C1)=O N1(C(CC(C)C2CC2)=O)CCCC(C(=O)NCCC(=O)OCCN(C)C)C1C c1(C(=O)NCC(C)(C2CC2)NC(CCCC#C)=O)ccc(C)cc1Cl Cc1cc(CC(=O)NCC2CC(CC(=O)NCCC3CC4C=CC3C4)C2)nn1C C1(C(N(C)CC2CCN(C(c3c(COC)cco3)=O)C2)=O)CCc2c[nH]nc2C1 C1(NC(c2n(CC)nnc2)=O)CCN(C(=O)C(O)COC)C1c1ccccc1 C1(C(=O)NCCOCCC=C)CCCCCN1C(c1ccc(F)cc1C)=O Cc1noc2nc(C(=O)NC(C3CN(C(=O)Cc4cnns4)CCO3)C)ccc12 O=C(C1CCCc2ncnn21)NCC1C2CC1N(C(c1coc(Cl)c1)=O)C2 N1(CC(=O)NCNC(C)C)CCN(S(C)(=O)=O)CC1.C12CC(C1)OO2 c1(C(=O)NCC2CC(CNC(c3cc(C(C)=O)sc3)=O)C2)n[nH]c2c1CC1CC21 C1(C(=O)NCC(CC)N(C(=O)COCC2CCCC2)C)CCOC1C(C)C c1(C(=O)NC2CC3(C(NC(c4ccc(CC)s4)=O)C3)C2)cc2cccc(Cl)c2o1 C1(NC(c2nc(N(C)C)sn2)=O)CC(NC(=O)CNC(c2ccco2)=O)C(O)C1 N1(C(Cc2ccc(C#C)cc2)=O)C2CCC1CN(C(=O)CN(C1CCSC1)C)C2 C=CCC(CC(C)C)C(=O)NCC1CC1NC(c1cc(C)c(C)nc1O)=O N1(CC)CCCC(O)(N2C(=O)C3(OCCO3)C2)C1.C(N)=O C(N=c1cc(Cl)nc(C(C)(C)C)[nH]1)C1CCC(CNC(C(C=C)O)=O)C1 C(CC(C)(C)NC(=O)CCc1ccsc1)N(C(=O)CC1CSC1)C n1(CC(=O)NCCOC(C)=O)cc(NCC2CCCOC2)cn1 CC1CC(C(=O)NC2CCCN(C)C2=O)CCN1C(C1CCCC(C#N)C1)=O N1(C(C2CCCN(C(C=C)=O)C2)=O)Cc2occ(NC(=O)CC(C)(O)C=C)c2C1 c1(C(N(CCCN(C)C)CCNC(C2(O)CCC2)=O)=O)cn(C)nc1C1CCCO1 CCC(CC)CC(F)C(=O)NC(C(=O)NC1CCCC(O)C1)C1CC1 Cc1c(Cl)ccnc1C(=O)NC(C1CCCN(C(=O)CCc2nncs2)C1)C CC1=C(C(=O)N2CCCC(C(=O)NCCCCc3ncc[nH]3)CC2)CCC1 Cc1cc(C(=O)N(CCCCN(C)C(c2occc2C2CC2)=O)C)ccc1F c1(C(=O)NC(C(C)NC(c2cscc2Cl)=O)(C)C)ccc2cc[nH]c2n1 CCCCC(CC)CC(=O)NC(CCC(C)C)C(=O)NCC(C)(O)CCO N1(C(C(C(C)O)C)=O)CCCCC(NC(C2CCCCO2)=O)C1 c1(C(=O)NCC2CCN(C(CCOc3ccc(C)cc3)=O)C2)cc2n(n1)CCO2 c1(SC)cc(C(=O)CN(C)Cc2ccccc2Cl)cc(O)n1 c1(C(=O)NCC2(NC(C(CC(CC)C)C)=O)CC2)ccc2c(c1)OCCNC2=O c1(-c2scc(NC(N3CCC(F)(CC(=O)O)C3)=O)n2)ccc2c(c1)CCC2 C(=O)(CCC(=O)c1cccc(C(=O)NC2C(CNC(N)=O)C2)c1)NCCOC1CC1 C1(S(C)(=O)=O)(C(=O)NC(CC)CNC(c2cc(C(F)(F)F)c[nH]2)=O)CCCCC1 C1(CN(C(Cc2cc(C)sc2)=O)C)CN(C(C2CCCC(=O)N2)=O)CCO1 C1(NC(CC(CNC(CCCCCN(C)C)=O)O)=O)CCn2cnnc2C1 C#Cc1cccc(CC(=O)NC2CCCC2C(=O)OC(C2CC(N(C)CC)C2)=O)c1 CC1OC2(CNC(=O)CC3CCCSC3)CC1(NC(C1CCCCC1)=O)C2 N1(C(C2C(CC)N(C(c3ccn(C)c3)=O)CCC2)=O)CCCOC(C)(C)C1 C1(NC(COCCN(C)C)=O)CCC(CCNC(c2cc(C3CC3)no2)=O)C1 N1(C(C=CC2N(C(C)=O)CCC2)=O)CC2CCC1CN2Cc1ccc(C)c(F)c1F C(C(CC(C)C)NC(=O)Cc1ccc(C(C)=O)s1)NC(c1ccc(CC)s1)=O C1(C(=O)OCC)CCN(C(=O)CCOC(c2oc(C(=O)O)cc2C)=O)C1C N#CC1(F)CCN(C(=O)CC2(N3CCC(F)(F)CC3)CC2)C1.n12cc(nn1)C2 C1(NC(=O)C(F)CC2CC2)CN(C(=O)CN2CCS(=O)CC2)CC12CCC2 c1(-c2scc(C(=O)NCCCN(C(=O)C(C)O)C(C)C)n2)cc(F)ccc1F C12(CNC(C(C=C)(F)F)=O)CCC(CC1)CN2C(=O)C(CC)NC(C)=O N1(C(C2CCC(CC)CC2)=O)CCCC2CN(C(=O)C(C)(C)C)CCC12 C1(O)(C(C)NC(C2CCC(=O)O2)=O)CCN(C(C2(CO)CCCCC2)=O)CC1 CC1COCCN1N(CC(c1ccccc1)c1ccccc1)CC1CC2CCC1C2 C1(C(=O)NCCN(C(c2c(CC)onc2C)=O)C)C2CCCC(=O)C12 Cc1cc(C)c(CC(=O)NC2CCC2NC(=O)Cc2cn[nH]c2)c(C)c1 C(CC(=O)Nc1cccc(F)c1)(C(F)F)NC(C1CC(=O)NCC1)=O C1(CC(=O)NC2(CO)CC(=C)C2)CC2(C1)CN(C(c1ccsc1C)=O)C2 C1(C(=O)NC(C)CCN(C)C)(CC)CCCN(C(C2OCCC2(C)C)=O)C1 N(C1CCS(=O)(=O)c2ccc(Cl)cc21)C(=O)NC1CC(C)(O)C1 C1(NC(c2c(C)n(C3CCC3)nc2)=O)CN(C(C2CCC2(C)C)=O)CCC1(C)C CCCC(CCC)C(=O)N1CCC(C(C)NC(=O)C(C)c2ccsn2)CC1 CC1(CNC(C2CC3CC3C2)=O)CN(C(c2ccc(C(F)(F)F)nc2)=O)CCO1 c1(OC)cc[n+]([O-])c(C(N2CCCOC(CNC(=O)CC3CCN(C)C3)C2)=O)c1 c1(C(=O)NC2CC(NC(c3cc(C(N)=O)co3)=O)C2)cc2c(=O)[nH]ccn2n1 c1(C(=O)NCCN(C(c2ccc(C)o2)=O)C)cn(-c2cccc(F)c2)nc1C c1(C(=O)NC2(CC(=O)N(CC(c3ccco3)O)C)CCC2)cccc2cncn12 c1(CCC)cc(C(N2CCCCC2CCNC(=O)CC(C)C2CC2)=O)sc1C c1(C(=O)NCC2N(C(CCC3C(C)=NNC3=O)=O)CC2)ccc(OCF)cc1F C(CN=c1nc[nH]s1)C1CCC(N(C2CCCCC2)C(c2cc3ccsc3s2)=O)C1 C(N=c1[nH]c(=N)[nH]c(Cl)c1[N+](=O)[O-])C1C(C)CN(C(=O)CN2CCCNS2(=O)=O)C1 N1(C(Cc2nn(C)c(Cl)c2)=O)CC2CS(=O)(=O)CC2(N(C(=O)C=CCF)C2CC2)C1 c1(C(N(C)CC2(OC)CCCC2)=O)cc2c(F)c(F)c(F)cc2[nH]1 CCCCCCCCNC(=O)C(CC(C)C)ONC(=O)CN1CCOC1=O CCC(CCC(=O)N1CCC(C(=O)N(C(CC)C(=O)N(C)C)C)O1)OC CCC(C)(C)C(O)C(=O)N(C)CC1CN(C(c2ccc(O)c(F)c2)=O)CCO1 N1(C(c2cc(C)c(N)cc2)=O)CCCC(NC(=O)CC2CC2(C)C)CCC1 CC(C)(CC=CC(=O)NC1CCCO1)NC(C1CC(NC(=O)OC(C)(C)C)C1)=O c1(OC)ccc(NC(=O)CC2CN(C(C3(c4ccccc4)CC3)=O)CCO2)cn1 N1(C(Cc2cnn(C)n2)=O)CCC(NC(c2coc(C(F)F)c2)=O)C(CO)CC1 N1(C(c2cc(CC)on2)=O)CCOC(C)(CNC(c2ncccc2C(N)=O)=O)C1 c1(C(=O)NC(CC2CN(C(C3CC(CC)C3)=O)C2)C)cc(C)cc(C)n1 c1(C(=O)NC2C(CNC(C(C)NC(N)=O)=O)CC2)ccc2nnn(O)c2c1 C1(NC(Cc2n(C)cnc2)=O)CCC(NC(=O)CCc2cscn2)CC1 C1(NC(=O)CCc2cccnc2)CC2CN(C(c3cc([N+](=O)[O-])n[nH]3)=O)CC2C1 c1(C(N2C(C(=O)NCC(C(=O)OC)(C)O)CC2C)=O)ccc(C)nc1O C1(NC(CN(CCOC)C)=O)C2CCN(C(=O)Cc3cccc(O)c3)CCC12 N1(C(Cn2nc(C)oc2=O)=O)CC(NC(=O)C(C)C2CC2)CC2(CC2)C1 c1(CC)ccccc1C(CNC(=O)Cc1cnc[nH]1)NC(c1cc(Cl)n(C)n1)=O CC1(C)CC(C(N2CCC(=CCNC(C3CC3C(F)(F)F)=O)CC2)=O)CCO1 C1(CC)CN(Cc2cc(C)cc(Cl)c2)CCN1C(c1cccnc1OC(F)F)=O N1(C(C23CC(C(=O)OC)(C2)C3)=O)Cc2ccccc2C(CNC(C2CC2Cl)=O)C1 N1(C(c2n(CC)ncc2Cl)=O)CCCC(CCNC(C2(C)CCOC2)=O)CC1 C(=O)(C(CC(C)C)C(N)=O)N(C1CCCN(C(c2cc(C)[nH]c2C)=O)C1)CC C(=O)(CC(C)C(F)(F)F)NC1(C(C)NC(c2coc(CN(C)C)c2)=O)CC1 N1(C(CNC(C)=O)=O)C2CCCC1CN(C(C1COC3CCCCC13)=O)CC2 C1(NC(C(CCCOC)C)=O)Cc2ccccc2C1NC(C1COC(=O)O1)=O Cc1c(Cl)ccnc1C(=O)N(C1CCCN(C(=O)C(C#N)C(C)C)C1)CCF c1(CN(C(C(C)COC2CCCCC2)=O)C)cccc(Cl)n1 C(=O)(C(CCC(N)=O)N(C)C)N1CC(NC(CCCC)=O)C(C)(C)C1 C1(NC(C(c2nc(C(F)(F)F)cs2)N(C)C)=O)CCC2(CC2)C1 Cn1cnc2ncc(NC(C34CCC3C4)=O)nc12.c12cccc(c1)NC(=O)CC2 Cn1ncc2c(N3CCC(OC(F)(F)CF)CC3)ccnc12 c1(C(=O)NC(CCC)C)ccc(-c2cnn(CC(C)O)c2)cn1 N1(C(c2cocc2Br)C(=O)NCCCC)CCOC(CNS(C)(=O)=O)C1 C1(C(N(C)Cc2c(C)nco2)=O)C2CC2CN1C(c1cn[nH]c1)=O N1(C(C(c2ccn(C)n2)C)=O)CCC2(NC(c3c[nH]cc3C(C)(C)C)=O)CC2C1 c1(OC)ccccc1NCC(N1CCCC1CCNC(c1nnc(S)n1C)=O)=O Cc1c[nH]c2ccccc2c1=NCCNCC(C1CCOCC1)C C1(N(C)C)CCC(C(=O)Nc2cc(CNC(=O)OC(C)(C)C)cs2)S1 C1(NC(CCN(CC)CC)=O)CCN(C(C2C3CCN2CC3)=O)CC1CC C1(C(N(CCN(C(C=CC(C)C)=O)C)C(C)C)=O)CCc2[nH]nc(O)c2C1 c1(CN2CCC(C3N(C(c4c(C)cccn4)=O)CCC3)C2)ccc2cc[nH]c2c1 N1(c2c(C(C)=O)cnc(C)n2)C2CCC1C(C)C(NC(C1CCOC(C)C1)=O)C2 CC1(CNC(=O)CC2CCC2)CCC(NC(=O)CC2CS(=O)(=O)C2)C1 N1(C(COCC)=O)CCC2(CC1)CN(C(c1csc(SC)n1)=O)CC2C(=O)O c1(C(=O)NCC(C)OCC#C)cnc(CNC(C2OCCOC2C)=O)nc1 N1(C(c2ncn(C(C)C)n2)=O)CC(NC(C2(CC3CC3)CCC2)=O)CC(C)C1 C(=O)(C(C#N)C(C)(C)C)N1CC(C)(C(=O)NCC2N(C(C)=O)CCCC2)C1 c1(C(N2C(C(=O)Nc3cn(CC)nc3C)CC(F)(F)C2)=O)ccc2c[nH]nc2c1 CC(F)(F)CCC(=O)NCC(C)(C)NC(=O)CC1CNC(=O)C1 c1(C(=O)NCc2c(Cl)ncc(C(=O)OC)c2)ccc(F)c2cccnc12 C1(NC(=O)OC(C)(C)C)C2CCC(C(=O)Nc3cccc(C#N)c3)C2C1(C)C C1(NC(=O)C2=C(Cl)CCOCC2)CCC2(CCN(C(=O)C3CC3)C2)C1 C1(C=O)Cc2ccccc2O1.C1(CC(N2CC(O)C2)=O)CCN(C(=O)C2CC2)CC1 C(=O)(C1=Cc2ccccc2C1)NCCN(C(=O)C(C)NC=O)CC(C)O C1(Cc2n(C)ccn2)CCN(N2CCC2Cc2ccccc2Cl)C1 CCC(C(=O)N(C)C)N(c1nnnn1C1CC1)CCCSC(F)F N1(C(Cn2c(C)ccn2)=O)C(C)CN(C(=O)CC2CCCC2(F)F)CC1C C1(O)(CN(C(C(C2CC2)OCC)=O)C)CCN(C(=O)CCN2C(=O)CCC2=O)C1 n1(CC(=O)OC)nc(C)c(Cl)c1NC(CN(C1CCOCC1)C)=O Cc1cc(C(N2CC(NC(C3(n4cccn4)CC3)=O)CC2C)=O)cc(F)c1 N1(C(CCCC(OC)OC)=O)CCC(NC(c2cc(OC)cs2)=O)C(C)C1 c1(C(c2nnc(-c3cccc(OC)c3)o2)N(CCNC)CC)ccc(F)c(Cl)c1 C1(C(=O)NCCOCCC(=O)NCC2CC23CCOCC3)OCC2CCCC12 Cc1cccc(N)c1C(=O)NCC1CCN(C(c2cc3sccc3[nH]2)=O)C1 N1(C(C(CCC)=CCC)=O)CCC(NC(c2cc(C(C)C)cc(F)c2)=O)C(O)C1 N(C1CCCc2c[nH]nc21)C(C1(NC(=O)Cc2ccco2)CC1)=O N1(C(CC2(NC(CCC(C)SC)=O)CCC2)=O)CCC(C)(C)C(CO)C1 c1(OC)cccc2c1C(C(=O)NCC1CN(C(=O)Cc3cc[nH]n3)CCO1)CC2 CC1(CO)CC2(CCN2C(C2(CNC(=O)OC(C)(C)C)CCNC2=O)=O)C1 N1(C(C=CCC(C)(C)NC(C2CN(CC)C(=O)C2)=O)=O)CCN2C(=O)NCC2C1 C1(NC(CC(=O)NC)=O)CCC2CN(CC(O)COc3ccc(Cl)cc3)CC2C1 Cc1c(C(N2CCCC(NC(=O)COC3CC=CC3)C2)=O)cnc2ccnn12 C=CCCCC(C)(C)C(=O)NOC(CC(C)C)C(=O)NC1(C)CC1 c1(C(=O)NCCC(C)O)ccnc(CNC(C2CC2c2ccncc2)=O)c1 C1(C(=O)NCC(CC)NC(=O)CC2CCOCC2)CC(S(C)(=O)=O)C1 C1(CC(N2CCC(OC3CN(C(C(C)OC)=O)C3)CC2)=O)CCN(OC)CC1 c1(C(=O)NCC(CNC(CC2CC(OC)C2)=O)O)cccc2ncn(C)c12 C1(C(=O)NC(C2CCOC2)CC)COCCN(CCNCc2ccccc2)C1 CCCCC(C)CCC(=O)NCc1cc(C(=O)N(CCCC)CCC)n[nH]1 C1(C(=O)NC(C2CCN(C(=O)CNC(N)=O)C2)C)Cc2ccc(C)cc2S1 c1(-c2c(C(=O)O)con2)cccc(OCc2cn(CC(O)C3CC3)nn2)c1 C1(C(=O)NC2CC3CCC2N3C(=O)C(F)F)CCCC(F)(F)CC1 C=C(C)CCC(=O)N1CCCC1C(C)NC(=O)COCCCN(C)C C1(NC(C(C)=CC2CC2)=O)CC(C)N(C(=O)Cn2nnc(-c3ccccc3)n2)C1 Cc1cccc(C)c1C(O)CNC(=O)C(F)Cc1ccc(Cl)c(F)c1 C12(CC(=O)NC(C)CN(C)C(C3OCCO3)=O)CCC(CC1)C2(C)C C1(OC)CN(C)C(C)(C(=O)NC2CN(C(C3(S(C)(=O)=O)CC3)=O)CC2C)C1 N1(C(C23CC(C)C2C3)=O)CCCN(C(c2cn[nH]c2)=O)C(CO)C1 Cc1cnc(N(CC(C)C#N)C(c2ccc(NC3(O)CCCC3)cc2)=O)nc1 C(=O)(CC(O)c1ccccc1)N(CCNC(c1cc(C(F)F)[nH]n1)=O)CC C1(COC)(CNC(c2cocc2C)=O)CCCN1C(C1CCCCS1)=O c1(C(N(C2CCN(C(c3coc(C(C)C)n3)=O)C2)CCC)=O)cc(CCO)on1 Cc1cscc1C(=O)NCC1CCCN1C(C1CC(OC(C)(C)C)C1)=O C(=O)(C1=CCCCCC1)NC1C(NC(c2nc(OC)oc2)=O)CC1 C12(CNC(c3cc(C)[nH]n3)=O)CC(NC(C3CC3C)=O)(C1)C(C)O2 CC1(C)CN(C(=O)CN2C(=O)CNC2=O)CCC1C(=O)NC1CC(=O)N(O)C1 c1(C(=O)NC2CCC(F)(C(=O)OC)C2)cc2c(Br)coc2cn1 Cc1ncc(NC(=O)CC2(C)CCN2C(=O)C(C)(C)C2CCC2)c(C)n1 C(=O)(C(F)(F)C(F)(F)F)N1CCC(N(CC(C)C)C(c2ccnn2C)=O)C1 C(=O)(C(C)(C)C1=CCN(C(c2cccnc2O)=O)C1)NCC1CCN(OC)CC1 CC1(CNC(C2CNCC2NC(N)=O)=O)CCCOC1 C(=O)(CCCCC(F)(F)F)NCC1N(C(CCCCCN(C)C)=O)CC2(CC2)C1 Nc1ccc(O)c(C(=O)NC2CCCCC2CNC(c2ccc(NC)cn2)=O)c1 C(CS(=O)(=O)CC(=O)Nc1ocnc1C(=O)NOCCOC(C)C)NC N1(C(C2C3CN(C(CC(=O)OC)=O)CC32)=O)CCC2(CCCOC2)C1 c1(CCC)nc(C)c(C(=O)NCC2CCCCN2CCn2cc(Cl)cn2)s1 c1(C(=O)NCCCN(C(=O)Cc2nnc(O)s2)C)nccc(-c2cnccn2)n1 c1(C(N2C(CNC(=O)CCC3CCOC3)CC(OC)C2)=O)cnc2[nH]ncc2c1 c1(C(C)C)c(C(N2CCC(O)(C(C)NC(=O)CCF)CC2)=O)cccc1F C(c1ccc2c(c1)CCO2)=CC(=O)NC(CNC(C1(OC)CCC(C)C1)=O)(C)C C1(C(=O)NCc2cc(Br)cs2)CN(C(c2ccccc2)=O)CCC1F c1(CN(C(C2CCN(CCc3nn[nH]n3)C(C)C2)=O)CC)cc(Cl)c(Cl)cc1O N1(C(CC2ON=C(CC)C2)=O)CC(NC(c2cc(COC)on2)=O)C2(CC2)C1 c1(C(=O)NC2(CNC(=O)CCC3CCC3)CCCCCC2)nccn2cnnc12 c1(C(=O)NCC(CC)NC(c2sc3ccccc3c2Cl)=O)cc2c(C)cccn2c1 C(=O)(C(C)(O)COC)N(CC(CC)NC(=O)Cc1n[nH]c(C)n1)C CCN(CCCCC)N1CCOC(c2ccccc2Br)C1 C(=O)(C(F)(F)CNC(=O)CNC(c1n[nH]cc1C1CC1)=O)OCC c1(OC)ccccc1-n1ncc(NC(=O)C(C)C2CC2)c1C1CC1 C1(NC(c2ccc(CSC)o2)=O)CC(C)CN(C(=O)C(C)=C2CCCC2)C1 c1(OC)cccc(NC(C2(Nc3nccc(C)n3)CC(CO)C2)=O)c1 c1(C(=O)NCCCNC(C(c2ccccc2)SC)=O)c(O)cnc2ccc(Cl)cc12 N1(C(c2c(C)nn(C)c2N(C)C)=O)CCOC2(CCN(C(=O)CCF)C2)C1 c1(C(=O)NC2CCN(C(C(CC)(C)CC)=O)CC2C)scc2c1OCCO2 S(=O)(=O)(c1[nH]c(=NC2CN(Cc3cccs3)C2)ccc1Br)NCC(CC)CCO C1(NC(C23CC(C(=O)OC)(C2)C3)=O)CCCCN(C(C2CCC(=O)N2)=O)C1 N1(NC(=O)CC2(Nc3nc(CC(F)(F)F)cs3)CC2)CCN(C2CCOCC2)CC1 c1(C(=O)NCCOCCCNC(c2c(CC)ocn2)=O)ncccc1C(=O)OC c1(NC(=O)NC2N(Cc3ccc(C)c(C)c3)CC=C2)cccc2c(Br)cccc12 C1(CCC(=O)NCCN2CCNC2=O)CCN(C(c2ccncc2Cl)=O)CC1 C1(O)(CNC(C(CC2CCC2)NC(=O)CCc2ccoc2)=O)CCOCC1 c1(C(=O)NCCC(COC)O)ccnc(CNC(c2[nH]nnc2C)=O)c1 C1(C(N2CCC(COC(C)=O)C2)=O)C(C)OCCN1C(=O)Cc1ccsc1C CN1CCCC(O)(CC(=O)NC(C)(C)CCCNC(c2ccnn2C2CC2)=O)C1 C(=O)(CS(=O)(=O)CC)NCC1(C)N(C(c2c(CCC)[nH]cc2)=O)CCC1 c1(C(=O)NC2C(NC(c3cncnc3)=O)CC2)cc2c(nn1)CCCC2 c1(CCC)cccc(CC(=O)NC2CCC(N(C(=O)CC3CCC3)C)C2)c1 C(C)(C(=O)NCC(CO)NC(c1csnn1)=O)N(C(C)=O)C N1(C(C(C=C)(C)O)=O)CCC2(CC1)CC(NC(=O)CCc1cncc(OC)c1)C2 C1(NC(COC(CNC(c2c(CC)cncc2)=O)(C)C)=O)CCC2CCCC1O2 Cc1ccc(C(=O)NCC2CCN2C(c2sc(C)c(C)c2C)=O)cc1F c1(CN=C(NC(CC)C2CC2)NCC2CC(C(=O)OC)C2)c(OC)ccc(Cl)c1Cl N1(C(c2c(C)nc(C3CC3)[nH]2)=O)CCC2CN(C(c3ncoc3C)=O)CCC2C1 c12nc(co1)N(C)C2=O.C1(NC(COCCOCC)=O)CC(C(=O)OC)C1 N1(C(C(COCC)C)=O)CCC(C)N(C(c2cn(C)nn2)=O)CC1 n1(CC(=O)NCCNC(C2CN(C(C(C)(C)OC)=O)C2)=O)ncc2cc(C)cnc12 c1(C(=O)NC2CCC2NC(c2csc(CO)n2)=O)cnc(O)c([N+](=O)[O-])c1 CCCC(C)(O)C(=O)NCC1C(C)CCCN1C(c1sc(C)cc1OC(F)F)=O C1(CC=C)(NC(=O)Cc2csc(C)n2)CCN(C(C2(Cl)CC2(C)C)=O)C1 c1(NC(C2CCCN2C(c2nc(Cl)ccc2Cl)=O)=O)c(Br)cc(Cl)cc1[N+](=O)[O-] Cc1nc2ccccn2c1C(=O)Nc1nc(C(F)(F)F)ccc1Cl C1(C(C(=O)NC(C#C)CCC)C)CCN(C(c2cc(C)co2)=O)CC1 C(=O)(C1=COCC1)NCCCNC(C1CN1C=O)=O.C(C)(C)(C)OC(=O)C1CC1.CS c1(C(=O)NCC(O)CCNC(=O)C(C2CCCC2)C2CCC2)cc(F)cnc1O Cc1cnc(C(=O)NC2CC(CNC(=O)CNC(N)=O)CC2O)cc1Cl CC(C)CCC(=O)NOCC(=O)N(C)Cc1ccn(C)n1 c1(C(=O)NC2C(NC(C(C(C)(C)C)CO)=O)C2)cc(N)cc(S(C)(=O)=O)c1 C(C1CCCN1C)=CC(=O)NC1CC(CCC(=O)NCc2n(CC)nnn2)C1 c1(C(=O)NC2CCC(NC(c3cc(C)c(C)o3)=O)CC2)cncc2c1CCC2 N1(C(C(C2CC2)OCC)=O)CCCC(C2CCN(C(c3cnsn3)=O)CC2)C1 c1(CC(=O)NC23CC2CN(C(C2(CF)CCOCC2)=O)C3)cnc2cccnn12 C12(NC(C3CC4(CC(=O)N4)C3)=O)CCCC1N(C(C1CC(=O)N1)=O)CC2 C1(C(=O)NC2CC(C(=O)NC)C2)CN(C(=O)COCC2CCOCC2)CCO1 C1(NC(CSc2nc(C)[nH]n2)=O)C2CC1N(C(=O)CN(C1CCCC1)C)C2 N1(C(Cn2c(C)ccn2)=O)CC2CCC(C1)N2C(=O)CCOCC1CCC1 Cn1cnc2cccc(C(=O)NC3C=CCN(C(c4cc(Cl)ccn4)=O)C3)c12 c1(C(C)(C)C)cc(Br)ncc1F.n12c(nnc1-c1ccc(Br)cc1)CC(Cl)NC(=O)C2 N1(c2ccnc(COC)n2)CCCC(CCNC(c2snnc2C)=O)CC1 C(=O)(C(CC(C)C)NC(C)=O)NC1CCC(CCNC(C2(CC)C=CCC2)=O)C1 C(CC(C)(C)C(=O)NCC(C)(CO)NC(=O)C(c1ccc(F)c(C)c1)=O)OC Cc1ccc2sc(C)c(C(N3CCCC(N(C)CC4COCC45CC5)C3)=O)c2c1 C=C(C)CCC(=O)N1CCC(CC(C)NC(c2ccc(Cl)o2)=O)CC1 N1(C(CCC2CCN(C(C(C(CC)C)O)=O)CC2)=O)CC(C)(C)C12CCCC2 c1(NC(C2CC(NC(C3C(C)(C)C3)=O)C2)=O)ccc(C(F)(F)F)nn1 C1(CNC(=O)CCNC(c2ccoc2)=O)CC(C)N(C(c2nc(C)sc2)=O)C1 C1(NC(C2CN(C)C(=O)CC2)=O)CN(C(=O)CC2CC(F)(F)C2)C2(CCCC2)C1 c1(C(N(C(CC)CNC(=O)CC2(O)CCOCC2)C)=O)ccc(C)c(C#N)c1 c1(C(=O)NC)ccc(-n2nc(-c3cccc(Cl)c3)nc2CC2CC2C)cc1 c1(OC)cc(N)cc(NC(N2CC(=O)N(C)C(C)C2)=O)c1OC CC1(C)CCCN(c2nc(Cl)ncc2Br)C1CNC(=O)CC1CCC(O)C1 N1(C(C2(CNC(C3C(C4(C)CCC4)C3)=O)CCC2)=O)CCN(C2CCC2)CC1 c1(C(N2CCC(NS(=O)(=O)C(F)(F)F)C(F)C2)=O)c(I)ccnc1F C=CCCCC(=O)N(C(C)(C(=O)NCC1COC(=O)N1)C1CC1)C C12(C(=O)OC)CCCCC(CC1)N2S(=O)(=O)C1=C(C)CCC1 N1(C(COC(C)C)=O)CC2CC(NC(=O)C(C)NC(=O)OC(C)(C)C)C2C1 CC1CCCCC1(C)n1cc(C2CCCN2C(=O)CCCF)nn1 N1(C(CCN(C)CC)=O)CCCC(C)(C(=O)NC2CCCC(O)C2)C1 C(=O)(NNc1ccc(-n2cccn2)cc1Cl)c1c(N)cncc1 N1(C(C(C)C)=O)CCC(NC(=O)C=Cc2ccccc2Cl)C(C)C1 c1(C2C(C(N(C(C)CCNC(C3(C(C)C)CCC3)=O)C)=O)C2)c(Cl)cccc1Cl CC#CCCC(=O)N1CCC(CNC(c2oc(C)nc2CC)=O)C1 c1(C(=O)NC(C(=O)NCC2C(C(=O)OCC)C2)C2CCOC2)ccccc1Cl N1(C(C2(C)CC(=O)C2)=O)CCC2(CC1)CC2C(=O)NCCF N1(C(C2(C)CC3(CC3)C2)=O)CCCCC(NC(=O)Cc2nc[nH]n2)C1 CC1(C)CC(O)CCN(C(=O)C(C2CC=CCC2)NC(=O)Cc2ccccn2)C1 N1(C(C(C)N(C(CCC)=O)C)=O)CC(C(=O)OC)C(F)C1 N1(C(C(CC)C(C)(C)CC)=O)C2CC=C(C(=O)NCc3ccc(C)nc3)C1CC2 CCC(CC)(CCNC(c1ccc(-n2cncn2)cn1)=O)NC(C1C=CCC1)=O S(=O)(=O)(c1cc(NC(=O)CSC)ccc1C)NC1(C(=O)OC)CCC1 CC1CN(C(=O)CC2(C)CC2)CC1CNC(c1cc(O)n(CCF)n1)=O c1(C(N(C2C3CN(C(=O)C=Cc4cscn4)CC23)C)=O)cccc2c1CCOC2 c1(C(=O)NCC(CC)NC(=O)C(C)C2CCC2)ccc(C(F)F)nc1 N1(C(C=CC(C)(C)NC(c2c(CC)occ2)=O)=O)CC(C)C12CCOCC2 C1(NC(CSCC(N)=O)=O)CCCC(COCCC(=O)N(CCCO)C(C)C)C1 CC1CCCC(CNC(c2cc(CNC(=O)CCN3CCCC3=O)cs2)=O)CC1 c1(C(=O)NCC(C)CNC(C2(C)CC(=O)N(C)C2)=O)ccsc1S(C)(=O)=O c1(C(C2(C)CC(NC(c3ccc(CC)o3)=O)C2)=O)ccc(-n2cncn2)nc1.N C(=O)(CCC(C)(C)C#N)NC(C(=O)N(CCC(C)(C)O)C)Cc1cc[nH]n1 C1(NC(C=Cc2n(C)ncc2)=O)CN(C(=O)Cc2ccsc2Cl)CCC1CO C1(CCNC(c2c(CC)ccs2)=O)C(C)CCCN1C(=O)COC1CC1 c1(C(=O)NC2(C)CCN(C(C(n3ncc(C)c3)C)=O)C2)ccc(Br)c(Br)c1 c1(C(C(=O)NCCN(C(C2(C)CC2C(F)(F)F)=O)CC)=O)cc(Br)co1 C(=O)(C#CC1(C)COC1)N(C)CC1CCN(C(CC(C)CN(C)C)=O)C1 C12(CCOCC1)C(=O)N2.C1(CC)CCCC1N(C(c1ccns1)=O)C1CC1 Cc1nc(C=CC(=O)NCC2(NC(=O)CC3CCCOC3)CCOCC2)[nH]c1C C(=O)(CC(C)N1CCCC1=O)N1CC(C(C)NC(CC2CC(SC)C2)=O)C1 N1(C(C(C2CCC(=O)N2)C)=O)CCCC1CN(C)C(c1cc(Br)n[nH]1)=O N1(CN(C)C)CCCC(C(N2CCC(C)(CCNC(=O)CO)C2)=O)C1 N1(C(N2CCC3C(CCN3c3nncs3)C2)=O)CCC(C2CCOCC2)C1 CC1CC(CNC(=O)CCCC2CC2)CN(C(=O)CC2(C)CCOCC2)C1 N1(CC(C2CCC2)OC)CCC(CNC(c2[nH]ncc2Cl)=O)CC1 C1(O)(CNC(c2c(C)nco2)=O)CCCN(C(=O)C2=CCCCC2)C1 C1(CC(=O)NC(C(N2C(C)(C)CC2)=O)C2CCCC2)CCC(C)(C)O1 c1(C(C)(C)CC2CCCN2C(C2CCCN2CC(F)(F)F)=O)ccc(Br)cc1 N1(C(C2CN(CC)C(=O)CC2)=O)CCC(O)(C(=O)NC2CN(CC(F)F)C2)CC1 c1(OC)c(Cl)cc(NC(N2CC(O)CC2CNc2ccc(C#N)nc2)=O)cc1Cl C(C1=CCN(C(=O)C(C(C)C)N2CCCCC2)CC1)NC(C(COC)O)=O c1(OC)cc(C(=O)NCC2(F)CCC(CNC(=O)COC(C)C)CC2)cc(C)n1 CC12CCCC1N(C(=O)C#CC1CCCC1)CCN(C(C1CN3CCC1C3)=O)C2 c1(C(CNC(c2nccn2C)=O)NC(c2nc(CC)sc2)=O)cccc(Cl)c1 c1(C(=O)NCCNC(C2CCCCC2(F)F)=O)c[nH]c2cc([N+](=O)[O-])ccc12 Cc1cc(F)ccc1C(=O)NCC1CN(C(=O)C(C)(C)C(=O)N(C)C)CCC1C N1(C(c2noc(CC)c2C)=O)CC2(CCN(C(=O)Cc3ccccc3O)C2)C1 N1(CC2(Cc3ccccn3)CCN(C)C2)CCC(=O)N(CCCCN(C)C)C1=O C1(C(N(C)CC2CCCN2C(=O)C(F)=C2CCCC2)=O)C(C2CC2)C1(F)F N1(C(c2cncc(COC)c2)=O)CC(NC(=O)C(C)(O)C(C)C)CC12CCC2 c1(N(CC(=O)NCC)C)nc(N2CCC(C)C(C)C2)nc2ncn(C)c12 C(=O)(C(C)(C)S(C)(=O)=O)N(C1CCN(C(c2cccc(F)c2C)=O)C1)CC CN1C(C(N2CC(F)CC2CNC(=O)COc2ccccc2O)=O)CCS1(=O)=O C1(CC#C)CCCCN1C(=O)C(=O)NC(c1ccccc1)COC(C)(C)C c1(C(=O)NC2(C3CN(C(=O)CCc4cc[nH]n4)C3)CC2)ccc2nccnc2c1 c1(C(=O)NC2CC(NC(CC3(C=C)CC3)=O)C2)cc2c(F)ccc(Cl)c2[nH]1 CC(C(F)(F)C(F)(F)F)=CC(N1CC2CCCC2(NC(c2ccn(C)c2)=O)C1)=O c1(C(N2C(CNc3ncc(C(=O)OCC)s3)CC2)=O)cn2cc(Cl)ccc2n1 N1(C(C(=O)N(c2cnn(C)c2)CCOC)=O)CCC2CC1C(=O)N2C C1(NC(C(C)SCCCC)=O)(CO)CCCN(C(c2cn(C)nc2COC)=O)C1 C1(O)(C(C)NC(C(C(C)C)C)=O)CCN(C(C2CNC(=O)O2)=O)CC1 c1(C(=O)NC2CCCN(C(C3C(C)(C)C3(F)F)=O)C2)nccc(C#N)c1F CCC(CNC(c1ccc(C#N)s1)=O)(CC)NC(=O)C(F)CC1CCC1 C1(NC(N2CCC(OCC(OC)OC)C2)=O)CCC(=O)CC1 N1(C(C(C(C)(C)O)F)=O)CCC2(CCOCC2)C(NC(c2ncccc2O)=O)C1 C1(COC)(CNC(=O)CCC2(NC(=O)CC3CCC3)CCCC2)CCCO1 C(CCCOC)(C(=O)NC(C)CC(C)C)NC(C=C(CCC)CCC)=O C1(N(CCc2ccc(C(N3CCN(C)CC3)=O)cc2)CC)CCCC12CCNCC2 CON(CCC(=O)NC1C2CCC(F)(F)C12)C(=O)C(C(C)C)N(C)C N1(C(c2cc(C)nn2Cc2ccccc2)=O)CCN(C(=O)CCC(F)F)CC1CF c1(C(N(C)CC2CCN(C(C(CCCC)C)=O)CC2)=O)cnc2sc(C)c(C)n12 c1(CC2C(C(C)(C)C)C2)cc(=NCC2COC(C)(C)CO2)[nH]c(N2CCCC2)n1 CC(CC(=O)NC1CCC1NC(C1C2COCC12)=O)Oc1ccccc1 C1(CNC(c2cc(C(C)=O)on2)=O)CN(C(C2(C)CC(C)C2)=O)CCC1(C)C C#Cc1cc(Br)ccc1NC(=O)CCCSC1CCCC1(F)F C1(NC(=O)C=CC(C)(C)SC)CC12CCN(C(c1nccs1)CC)C2 C(=O)(NNc1c(Cl)cccc1Cl)O.C(CCCCC)C(C)(C)C S(=O)(=O)(c1cc(Cl)cnc1N)NC(c1cccc(C(=O)OC)c1)C Cc1ccc(CC(=O)NC2CC2CNC(=O)CC(F)(F)F)cc1Br C(=O)(C1Cc2ccccc21)CC(O)CF.c1(NC)ccc(Br)c(S(=O)(=O)N(C)C2CC2)n1 C(=O)(C1CCCc2scnc21)NC1CN(C(c2ccc(C#N)[nH]2)=O)C2(C1)CCC2 N1(C(C2(C#N)CC2)=O)CC(NS(=O)(=O)CCCCCl)C(F)(F)C1 CCC(C)CC(C(=O)NCCOCCOC)NC(=O)CSC.C(C)(C)S c1(NC(=O)NC(C)C(C)Oc2ccc(C(F)(F)F)cc2)cccc2ccoc12 C1(CC)C(NC(=O)Cn2ccnc2)CCCN1C(C1CCC(=O)N(C2CC2)C1)=O c1(CCC)ccc(C(=O)CCC(=O)N(C)CCNC(C2C=CCC2)=O)cc1 c1(-n2c(-c3cc(C#C)cc(OC)c3)nc(C3CC3)n2)nc2cc(C)cc(C)c2[nH]1 CC1(C(N2CCCC(Cn3cc(-c4cncnc4O)nn3)C2)=O)COCCO1 c1(C(=O)NCC(C)NC(C2CCC3CC3CC2)=O)cc(Br)cnc1N N1(C(C2(C)CN(C(C(CC3CC3)OC)=O)C2)=O)CCc2ccccc21 CC1(CNC(C2(C(C3CC3)C)CCCO2)=O)CC(NC(=O)Cc2cncs2)C1 N1(C(C2(CNC(C(CC=C)C)=O)CC23CCC3)=O)CCC2CCCC12 c1(NCc2n(CCC)nnn2)ccc(OCc2ccccc2)c([N+](=O)[O-])c1 C(=O)(CC(O)CC(C)(C)C)N(CCC(=O)NCc1cccnc1O)C(C)C c1(OC)cc(C(=O)NCC(C)CNC(C2CCN(C)C2)=O)c(C)c(Br)c1 C(CCC(C)(C)C(=O)N1CC(C)(C)C1c1cn(C2CN(C)CCO2)nn1)OC Cc1ccccc1C(c1nc(-c2cccc(F)c2)n(-c2cnc(C)s2)n1)C C1(COC)CN(C(=O)CCCCNC(=O)CC2C=NN(C)C2=O)CCO1 c1(NCCO)cccc2c1CCC2.N12CC3CC1CN3C(=O)C2=O N1(C(CC(=C)Br)=O)CCC(N(C(=O)C(C(C)C)NC=O)C(C)C)CC1 CC(CS(N)(=O)=O)NC(=O)N(C1CCCN(Cc2ccco2)C1)CCO C1(CC2CCC(NC(CN(C(CN(C(C)=O)C)=O)C)=O)C2)(CO)CC(C)(C)C1 Cc1cc(C(N2C(C(=O)NCc3ccc(Cl)cc3F)CC3CC23)=O)cc(C)c1F C1(NC(CCCNC(C(CC)O)=O)=O)CCCC12CC2 Cc1ccc(CSCC(=O)NCCC(C)NC(=O)C=Cc2ccccn2)cc1 c1(C(=O)NC2C(CNC(c3cc(C(C)C)on3)=O)CC2)cnc2sccc2c1 N1(C(C(C(C)C)C)=O)CC2(C1)CN(C(=O)COCC=CC1CCCC1)CC2CO C(=O)(C(O)(C(F)(F)F)c1ncc[nH]1)NC(CC)CN(C(=O)COCC(=O)NC)C N1(C(CCCSC)=O)CCC(C(N2CC(O)(CC(C)C)C2)=O)C1C(C)C C1(CCC(N2CCC(CN(C(=O)Cc3cncn3C)C)C2)=O)OCCCC1(C)C c1(CC)ccoc1C(=O)NC(C)CC(C)NC(=O)CCc1cc(C)on1 C1(OC)CCCN(C(=O)CCOC(C)(C)C)C1OC1CC1.C12(CC1)C(=O)NCC2 N1(C(c2cc(CC)[nH]n2)=O)C2CCC1CN(C(c1cscc1F)=O)CC2 N1(C(CCC(C)C)C(N)=O)CCCOCC1(C)C C=CC1(CC(=O)NC2CC3CC2N(C(c2csc(C(F)F)c2)=O)C3)CCCCC1 N1(C(=O)COC2COC(C(F)(F)F)C2)CC2CC2(C(=O)NCC(N2CCCC2)=O)C1 C1(C)(CNC(CCn2ncc(C)c2)=O)CCCN(C(=O)CC2(C(F)(F)F)CCC2)C1 C1(C(C)C)(C(=O)N(C2CCC(O)CC2)C)CCN(C(c2cc(Cl)no2)=O)C1 C12(NC(CC(CC)NC(=O)CN3CCOCC3=O)=O)CC1COC21CCC1 C1(CN(CCC(=O)NS(C)(=O)=O)C)CCCCO1 C1(CC=C)(NC(C2CCOC(CC)C2)=O)CCN(C(=O)Cc2cccnc2OC)C1 c1(OC)ccc2c(C(=O)Nc3[nH]nc([N+](=O)[O-])c3Cl)csc2c1 N1(Cc2cc(C(C)C)no2)CC(n2cc(C3CC4(C3)CC4F)nn2)C(C)C1 C1(CNC(c2cncn(C)c2=O)=O)N(C(=O)CC2(CO)CC2)CCCC1(C)C CC1(C)C(C)(CNC(C2COCCC2NC(C2CCC(=O)O2)=O)=O)C1(C)C C1(CC)CN(C(C2(CC(C)C)CC2)=O)CCC1NC(=O)Cn1cnc(C#N)n1 C(=O)(C(CN(C)C)N1CCC1)NC(CN(C(COCC)=O)C)C.C12CC(C1)C2 c1(OC)ccc(CC(=O)NC2COCC(C)C2)cc1NC(=O)C(C)(C)C C=CCCC(C)(C)C(=O)N1C2CCC1C(CNC(C1CCCCCCC1)=O)C2 c1(C(=O)NC2CC(NC(C3(C)CCOC3)=O)CC2O)cccc2c1OC(F)(F)O2 C1(n2c(SCC(=O)N(C)C)nc(-c3cscn3)n2)CCOC2(CCCC2)C1 C(CNC(C1C(C)C1C)=O)(CC)(CC)NC(C=C(CC)C)=O N1(C(c2nc(SC)sc2)=O)CCC2CN(C(=O)C(O)Cc3cnc[nH]3)CC2C1 c1(C(N2CC(CC(=O)NCCc3c(C)cccn3)C(C)C2)=O)cccc(C#N)c1 c1(OCC)nc(C)ccc1C(N1C(CNC(=O)CC(C)(C)F)CC2CC12)=O C(=O)(CC(C)(C(F)(F)F)N(C)C)N1CCC(CN(C(c2ccc(CC)s2)=O)C)C1 C#CCC(C(=O)NCc1ccc(C(N2CC(OC(=O)NC)C2)=O)o1)C1CC1 c1(NCC2OCCN(C)C2)ccc(S(=O)(=O)NC2CCC3(CCC3)C2)cc1Br N(C1CCCc2occc21)C(CCCNC(C(C)(C)OC(C)=O)=O)=O C12(CNC(c3n[nH]cc3C3CCC3)=O)CC1CN(C(=O)CNc1ncccn1)C2 c1(CCCO)ccc(-c2cnn(C(=O)NCCn3c(C)ncc3)c2)c(F)c1 C(C(C)C(=O)NC(C)CC1CN(C(c2c[nH]nc2C(F)F)=O)C1)OC C1(COC)(NC(=O)C(C)n2cccc2)CN(C(c2ccccc2)=O)C1 C(c1ccc(F)c(F)c1)=CC(=O)NCC1CN(C(=O)Cn2cnnc2)CCO1 Cc1ccc(CO)cc1NC(=O)CNC(=O)NCC=Cc1cc(Br)cn1C N1(C(CCC(CC)OC)=O)CC2(CCC2)CC1CNC(=O)C(CC)SC C1(C2(O)CN(C(C3CCOC3)=O)C2)(CNC(c2nn[nH]c2Cl)=O)CC1 C(C)(C)(CCCNC(c1c(C)noc1C(F)F)=O)NC(CCc1ncc(C)[nH]1)=O N(C1CCCn2ncnc21)C(C(CC1CC1)NC(C(CC)C(C)C)=O)=O C=C(C)CC(C(=O)N1CC(CC(F)C(=O)NCC2(OC)CCC2)C1)OC C1(C(N2CCC(N(C(c3scc(C)c3)=O)CC3CC3)C2)=O)C(C)(C)OC1(C)C CCC(C)(C(=O)NC(CNC(c1cnc(CC(C)(C)C)s1)=O)C(C)C)C(N)=O C1(C)(NC(C(CCOCCO)NC(C2(F)C(C)(C)C2(C)C)=O)=O)CN2CCC1CC2 c1(C(CC)C(=O)NCC(O)CCNC(c2cncn2C)=O)c(C)noc1C C(C)(CN=c1[nH]cnc2cccnc12)(CC(C)C)NC(Cn1ncc(C)c1)=O N1(C(c2cc(CC)ncn2)=O)CC2CCN(C(=O)C=C=C(C)C)CC12 CC1=C(C)CC(C(N2CC3(C)CC2(C(=O)NCCCN(C)C(C)C)C3)=O)CC1 c1(C(N2C(c3cnc(C)s3)CCC2)=O)ccc(C(=O)N(C)C)cc1 CN1CC(C(N2CCN(C(=O)Cn3cc(CO)nn3)CC2CF)=O)OCCC1=O c12ccccc1NC2=O.c1(C(CC)(C)O)cn(CC2(C(C)C(C)C)CC2)nn1 S(=O)(=O)(c1ccc(C#N)cc1)NC(C(=O)NCCN(CCOC)C)C c1(C(=O)NCC2N(C(C(C)N(C(C)=O)C)=O)CCCC2)ccc2ncccc2n1 c1(CCC(C2CCOCC2)NCC(=O)NC2(CO)CCC2)ccccc1 CC(C)C(C)(O)C(=O)NCC1(CNC(c2ccc(Cl)c(F)c2)=O)CC(F)(F)C1 C1(NC(C2CCN2C(c2cccnn2)=O)=O)CC12CCCCCC2 Cc1c(C(=O)NC2CC3CN(C(c4[nH]cnc4Cl)=O)CC3C2)nn2c1OCCC2 c1(CC(N2CCC(C)(CNC(c3ccnn3CCF)=O)C2)=O)cc(O)nnc1O C(=O)(C1=CS(=O)(=O)CCC1)NC(CCNC(C(C)Sc1nncn1C)=O)(C)C C1(C(=O)NCC(C(=O)NC2C(CC=C)CCC2)O)CCS(=O)CC1 Cc1ncc([N+](=O)[O-])n1CC(=O)NC1CC(NC(=O)C(C)P(C)(C)=O)C1 c1(C(=O)NCC2(NC(c3ccn(C(F)F)n3)=O)CCCC2)c(Cl)ccc(Cl)c1O C(C(F)(F)F)=CC(=O)N(CC(=O)N(CC(O)CN(C)C)C)CC=C c1(C(C)C)ocnc1C(N1CCCC1Cc1cn(CC(C)(C)O)nn1)=O C1(F)(C(N(C)Cc2c(C)ccnc2)=O)CCN(C(=O)CC2CCC(C)(C)C2)CC1 N1(CCNC(c2ccsc2)=O)CCC2(CCCCN(C(c3csc(O)n3)=O)C2)C1 N1(C(CN(c2ccccc2)C(C)=O)=O)C(CNC(=O)CCSC)CC2COCC12 CC1CCc2sc(C(=O)O)cc2C1.N12CCC(C)(CC1)CNC(=O)C2=O C1(NC(C2(COC)CC(=C)C2)=O)CN(C(c2cccn2C)=O)CC1F C1(C(N2C(CN(C(COCC#C)=O)C)COCC2)=O)CCc2nnc(O)cc2C1 C1(C(=O)NCc2cnc(C)s2)CC(O)CCN1Cc1cccc(F)c1Br C1(CC)CCCC1C(=O)NOCC(=O)NCC(=O)N(CC)Cc1ccncc1 C(CC(C)C)(C(=O)NCc1cn(-c2nn(C)cc2C#N)nn1)SC C(=O)(C1=CCCCO1)NC(C1CCCN1C(c1ncoc1-c1ccccc1)=O)C N1(C(c2snc(C)c2N)=O)CCC(C(=O)NC(c2ccccn2)CO)C(C)C1 C1(NC(c2nc(C)oc2)=O)CC2CC1N(C(C1(CO)CCC1)=O)C2 c1(OC)ccc(Cl)c(C(=O)NCCC2(O)CCCN(C(=O)C=C(C)C)C2)c1 N1(C(c2ccc(COC)s2)=O)CCC2(CC1)CCN(C(C1(CSC)CC1)=O)CC2 c1(C(N(CCCNC(CC(C)(C)SC)=O)CCO)=O)cnc2cc(C)nn2c1 N1(C(CSC)=O)CCC2CN(C(=O)C(C(C)C)n3ccc(C4CC4)n3)C2C1 c1(C(N(CC(C(=O)N(C(CC)CC)CC)C)C)=O)nc(C)ccc1C c1(C(=O)NCC(CC)(C)NC(C2CCC=CCC2)=O)ccc(C(C)C)nc1 c1(-c2cn(C3(CCN(C)C(=O)OC(C)(C)C)CC3)nn2)cccc(C#N)n1 c1(OC)ncc(C(=O)N(C2CN(C(=O)CC3COCC3O)CC2(F)F)C)cc1C C1(O)(c2c(C(=O)NCCC)scn2)CCN(C(=O)C(C(C)C)c2cnc(C)s2)CC1 Cn1cc(NC(C2CC(c3ccccc3)C2)=O)cc1C(=O)NC1CCC(=O)NC1 c1(C(C)(CO)NC(N(CCC)CC2CCCO2)=O)ccc(C)cc1 c1(C(C)C)ccc(C(=O)NCCC(C)CCNC(C2CCCSC2)=O)c(F)c1 N1(C(c2c(C)cccc2Cl)=O)CCC(O)(C2(NC(c3csc(Cl)n3)=O)CC2)CC1 C1(C(=O)NC(C2CN(C(Cc3c(C)ncc(Cl)c3)=O)C2)C)CCCC2CCCN12 C1(CC)CCN(C(=O)Cc2ccc(C)nc2)C1C(=O)NCc1nccc(OC)n1 C1(NC(C2N(C(C3(Cl)C(C(C)=O)C3)=O)CC(O)C2)=O)CC2C=CCC(C1)C2 c1(C(N(CCOCCCN(C(Cc2cnc(C)s2)=O)C)C)=O)csc2cncn12 C(C(C)(C)CNC(=O)CCc1nnc(C2CCCC2)o1)NC(C=CC(CC)C)=O C1(CNC(c2n(CCC)ccc2)=O)CCCC(NC(c2nc(=N)cc[nH]2)=O)C1 c1(C(=O)OCC(c2c(N(C)C)cccc2)=O)cc(Br)cnc1O c1(CC(=O)N(C2CCN(C(c3csc(C(F)(F)F)c3)=O)C2)CC)ncc(C)s1 C(=O)(C(CCC(N)=O)n1cc(-c2ccc(N)c(N)c2)nn1)N1C(C(C)C)CC1 c1(NC(=O)CC2CN(S(=O)(=O)CCBr)CCO2)cc(F)c(F)c(F)c1F C1(C(C)C)(NC(C2CCCN2C(=O)C(C)(C)C)=O)CC(O)C1 C(C(C)(C)C(=O)NCc1cc(C(N2CCC(CN(C)C)CC2)=O)co1)N(C)C N1(C(c2cnc(CC(C)C)s2)=O)CCC2(CC1)CCN(C(=O)Cc1ccoc1)C2 CC1CC(C(=O)NN2CC(C(N(C(C)(C)C)CC3CCC(=O)N3)=O)C2)=NO1 c1(OC)cc(C#N)cc(Br)c1NC(C1CCN(Cc2cccc3ccnn23)C1)=O N1(C(C(COC)C)=O)CC=CC(C(=O)Nc2cccc(OCC(C)C)c2)C1 CC(C)CCCCCCC(NC(=NCCCF)NCC(c1nc(C2CCC2)no1)=O)=O C(=O)(C(CCCC)C(C)C)N1CCC(F)(CNC(CC=CC)=O)C1 C=CCCC(C(=O)NCc1cccc(C)c1C)NC(=O)Cc1ccsc1C c1(CC)cc(Cl)ccc1C(=O)NC1CCCC1NC(=O)C(C)(F)F C12(NC(C(C)SC(C)C)=O)CCC(C1)N(C(c1cc(O)cc(F)c1)=O)C2 c1(NC(c2cc(-c3cc(F)cc(F)c3O)cnc2Cl)=O)nnc2ccc(Cl)nn12 c1(OC)cc(F)c(Cl)cc1C(=O)NCC12CC1CN(C(c1cc(Cl)ncn1)=O)C2 CC(C(=O)NCCC1CCN(C(C2CC3(CCO3)C2)=O)CC1)S(N)(=O)=O C1(C(=O)OC)CC12CCN(c1nnnn1C1C3COCC13)CC2 CC1(O)CON(C(=O)C(F)C2CCN(C(=O)CC3OCCCO3)C2)C1 C=CCC(CC)C(=O)NC1CCC(N(C(=O)Cc2cnnn2C)C)CC1 CC(C)C(C#N)C(=O)N1CCN(C(=O)CCC(C)(F)F)C(c2cccc(Cl)c2)C1 C1(NC2C(C)(C)CC(=O)NC2)C2CCC(O2)C1(F)F [nH]1ccc(OC(C)(C)C)n1.CC1C=CC(=O)NCCC2(CC2)C(=O)N1.C1(=C2CC2)CC1 C(=O)(C(F)CCC(C)(C)C)N1CCCC(F)(CNC(C(C)C(F)(F)F)=O)C1 N1(C(CN(C)CC)=O)C(C(=O)N(C2CCCN(C)C2)C)C2CC(O)C1C2 C1(CNC(CCOCCOC)=O)CCCC1NC(=O)CCC1CC1(C)C Cc1cc(NC2(CNC(=O)C=CCOCCC(C)C)CCC2)nc(C(F)(F)F)n1 Cc1cc(C(=O)NC(C2(O)CCN(C(=O)C(C)O)CC2)C)cc(Br)c1C c1(CCC)cccc(C(=O)NC(C)CCCNC(C2CCCC(=O)N2)=O)c1 N1(c2snc(C(C)C)n2)CCC(NC(C2Cc3nccn3C2)=O)C12CC2 O=C(N=c1nc2ccccn2[nH]1)C1(C(F)(F)F)CCNC1 c1(C(N(C2(CC(N3C(C#C)CC3)=O)CC2)C)=O)n[nH]cc1C#C c1(C(C(=O)NCC(C)N(C(CC=CC)=O)C)C)ccc(-c2ccccc2)cc1 C#Cc1ccc(C(=O)NC2CC(C(=O)NC(C=C)C(F)(F)F)C2(C)C)cc1C c1(C(=O)NCC2CC(NC(c3ccc[n+]([O-])c3)=O)C2)ccn2nccc2n1 C=CC(C)(C)CC(=O)N1CC(NC(c2ccc(OC)nc2C)=O)C(C)C1 N1(C(c2cnc(C(C)C)[nH]2)=O)CCOC2(C1)CN(C(=O)CCCc1cccs1)C2 C1(CNC(COCC(=O)NC)=O)(OC)CCCN(C(C2CCNC2=O)=O)C1 c1(NC(C2CCC(NC(c3cnc(Cl)nc3)=O)C2)=O)c(O)cccc1O C(=O)(C(C)C(O)CC)N1CC(C=C)(CC(=O)N(CCCCC(C)C)C)C1 O=C(CC(O)CN(C(=O)CCc1csnn1)C1CC1)Nc1ccc(O)nc1 C(=O)(CCC(C)CCCC)N1C(C#C)CN(C(=O)C(C(C)CC)OC)CC1 C1(C(N2CCCC(n3cc(C(=O)NC45CC(C)(C4)C5)nn3)C2)=O)CC(CC)CCO1 CN(C)S(=O)(=O)N1CC(CNC(=O)NC2CCCC2O)C1 C1(C#CC(=O)NC(C)C(C)C(=O)N(C)CCOC(C)=O)(CC)COC1 N1(C(CCC=CCC=C)=O)CCCN(CCNC(=O)C(C)CC(N)=O)CC1 C(C(O)CN=c1nc2scnc2c(NCCn2ccccc2=O)[nH]1)OC(C)C CC(C(=O)N1CCC(C(=O)N(C)Cc2cccnc2)(CF)C1)S(N)(=O)=O c1(C(=O)NCCCN(C(=O)CCC2(C)CC2)C(C)C)cn2c(n1)CCC(C)C2 CCCC(C(=O)N1CC=CC(NC(=O)Cc2csc(CC)n2)C1)C(C)C CC(C)C(C)(C)C(=O)NCC1CN(C(=O)CC2CCCCCO2)CCCO1 N1(C(c2cnc(C)nc2O)=O)CCCC2CN(C(=O)C3=NOC(C)C3)CC12 Cc1ccc(C(=O)N(CC(C)O)CCNC(=O)C(CC(C)C)N=CCl)c(F)c1C c1(CN(Cc2c(OC)ccs2)Cc2ccccc2)ccc(Cl)c(Cl)c1 C1(C(=O)OCC2CC(C)(c3ccccc3)C2)CC(=O)NC(=O)N1 c1(C(N2C(CNC(C(F)=CCC)=O)C(C)(C)CCC2)=O)[nH]cc2c1CCS2(=O)=O Cc1c(C(=O)NC(C)(C)CN(C(=O)CCn2ccnc2)C)cncc1Cl N1(C(Cn2ncc(CC)c2)=O)CCC2(CC2)CC1C(N1CC(C(N)=O)C1)=O c1(C(N2CCN(C(C3CCN3S(C)(=O)=O)=O)C(CO)C2)=O)cnn2cccnc12 O=C(CCC(F)(F)Cn1cc(-c2cccnc2)nn1)NC1CC2CCCC2(O)C1 CC1CCC(CNC(c2ccc(OCF)c(F)c2)=O)N(C(c2ccsc2Cl)=O)C1 c1(CNC(CCC(=O)OCC)C)ccc2cc(OC)ccc2c1 C=CC1(C(=O)NCCCc2scnc2C)CCN(C(=O)CCCOC(C)(C)C)C1 C(=O)(C(CCC)CC(C)C)N(CC(CC)NC(=O)C=C(Cl)Cl)C.C=O C1(OC)(CNC(=O)C=CC2CCC2)CCN(C(=O)C(C2CCN(C)CC2)O)C1 C#CCC(C)(CC)C(=O)NC(CNC(=O)CCN(C)CCC(C)C(C)C)CO C(C(=O)NCc1cnc(Cl)s1)(C(C)C)N(C(C=CC(=O)OCC)=O)CC C1(NC(c2c(SCC)nccn2)=O)CC2CCC1N2C(c1cccc(Cl)c1)=O C(=O)(C#CC(C)(C)CNC(C1COC(=O)N1)=O)N1CC(C)SCC1 C(=O)(C(O)CCS(C)=O)Nc1c(OC)ccc(CSCCCO)c1 C1(CNC(c2nc(CC)oc2)=O)CN(C)CCN1C(=O)CC(=O)NC1CC1 c1(OC)cc(OC)cc(C(=O)NC2CCC(NC(n3nc(C)n(C)c3=O)=O)C2)c1 C(C(O)CC(c1ccc(Cn2cccn2)cc1)NC1CC(OC)C1(C)C)OC S(=O)(=O)(CCCC(=O)O)NCCc1nc(CSCC(=O)NC(C)C)on1 C1(C(=O)NCc2c(C(=O)NCC(c3scc(C)n3)C)nco2)CC12CCCCC2 N1(C(C(=O)NC(C)C)=O)CC2CCC1C1CN(C(C3COCCN3C)=O)CC21 c1(C(=O)NCC(CNC(=O)Cc2cnns2)OC)ccc(F)c(C(F)F)n1 c1(C(=O)NCC2(NC(=O)CN3CCCC3CO)CCCC2)ccc(Br)cn1 C1(C(=O)NCC2CCCN(C(c3c(CN(C)C)cco3)=O)C2)CC(C)(C)CN1C C1(OC)CN(C(=O)CCC(C)NC(C2(C)CCOCC2)=O)CC12CC2 Cc1c(CC(=O)NC(C)CN(C(=O)CSCC(N)=O)C)cnn1C CC1=CCC(C(=O)NCC(C2CC2)N(C)C(C2(C)CCOCC2)=O)CC1 CN(C1CCOCC1)N1CCC(OC(C)(C)C)C1 C(=O)(C1=Cc2ccccc2C1O)NC(C)(C)CNC(c1cc2n(n1)CC1(CC1)C2)=O C(=O)(C(CC(C)C)NC(c1csc(=N)[nH]1)=O)N(C1C(NC(C)=O)CCCC1)C C1(CNC(c2ccc(Cl)o2)=O)CC(CNC(=O)CCc2ccco2)CO1 Cc1nccc(C(=O)NCCC2(C)CCN(C(=O)C(C3CCOCC3)C)C2)n1 C1(C(=O)NCCN(C(=O)C(F)C(F)(F)F)C)CC2OC(=O)OC2C1 Cc1cccc(C(=O)NC2CC2CNC(C2CCCN2C)=O)c1C#N C1(C)(CN(C(Cc2c(C)noc2)=O)C)CCCC1NC(C1CCCC1O)=O C12(NC(CCc3ccn(C)n3)=O)CCCC1CN(C(C1CCCCC1(F)F)=O)C2 N1(C(COC2CCN(C(c3ccn(CCC)n3)=O)C2)=O)CCC(F)(F)C1 C1(C(C)(C)S(C)(=O)=O)c2nnnn2C2CCC1C2.CC(CCS(C)(=O)=O)NCC C1(C(N2CC(O)(C(C)NC(c3cn(CCCC)nn3)=O)C2)=O)CCC=CCC1 c1(OC)ccc(C(N2CC(CC(C)NC(=O)C(C)(C)C(F)(F)F)C2)=O)c(N)c1F C(=O)(CC(F)(F)C(F)(F)F)N1CC2CC(NC(c3c(C)ccc(OC)c3N)=O)C2C1 C1(C2CC2)(CNC(c2nc(OC)c(C)s2)=O)CCN(C(C2(C)CC(C)(C)C2)=O)C1 CCCCCS(=O)(=O)CC(=O)N1CCCCC(NC(=O)C(C)(CC)OC)C1 c1(C(N2CC(NC(c3c(COC)scc3)=O)C3(C2)CC3)=O)ccc(F)c(C)c1N Cc1cc([N+](=O)[O-])ncc1C(N1CCCC(O)(CNC(=O)CSC(C)C)C1)=O CC1CN(C(C(=O)NC2(C)CC2)c2ccsc2)C2(CCC2)C1 C(=O)(C(C)(C)C(C)NC(=O)C#CC1CC1)NC(C)CCn1cncn1 c1(C(=O)NCC(C)(C)NC(C2C3CCC(F)(F)C23)=O)ccc(C(F)(F)F)c(O)c1 C(=O)(C(C(C)(C)C)NC(C)=O)N(CCC)CCOC(=O)C=CCNC.C(C)(C)(C)O Cc1cc(=O)n(C)nc1C(=O)NC1CCC1CNC(=O)C1=NNC(=O)CC1 N1(CCC)CCCCC1C(=O)NCCCNC(c1ccnn1CCF)=O C(=O)(C#CC1(CC)COC1)NCC(CCCC)NC(=O)CC(C(C)C)OCC N1(C(CCCCSC)=O)CCC2(CC1)CCN(C(=O)CC1CCOCC1)CC2C Cn1cc2ccc(C(=O)NCC3COCCN(C(c4ccsn4)=O)C3)cc2n1 c1(OC)cc(C(N2CC(NC(=O)C(F)(F)C(C)O)CC2(C)C)=O)cc(F)c1C#N c1(C(N2CC3C(CNC(=O)C(F)(F)CO)C3C2)=O)cc(Br)c2c(c1)CCO2 C12(NC(C3CCN(C(C(C)n4ccnn4)=O)C3)=O)CCC(C(N)=O)(CC1)C2 c1(CC(N2CCC(NC(CCC=C)=O)CC2C2CC2)=O)cccc([N+](=O)[O-])c1 C=C(C)C(C)(O)C(=O)NCC1CCN1C(=O)Cc1cccc(OC(F)F)n1 Cc1ccc2cc(C(N3CCC(NC(c4ccn(C)n4)=O)C3)=O)cnc2c1 C1(NC(c2c(C)cco2)=O)C2CC3CN(C(c4ccn(C)c(=O)c4)=O)C1C3C2 n1(CC)ccnc1C=CC(=O)NC1CN(C(=O)Cc2cccc(Cl)c2)CC1C C(=O)(C(C)(O)C(F)(F)F)N(CCC(=O)NC(CO)C(C)(C)CO)CC C1(C(N(CCOCCCNC(c2c(C)cco2)=O)C)=O)CC2CCCCN2C1 N1(C(=O)CSc2ccon2)CCCCCC(N=c2nc(C3CCCC3)[nH]s2)C1 N1(C(C=CC=CCC)=O)CCC(C(N2CCCC(C(C)C)CC2)=O)C(C)(C)C1 n1(C(C)C2CC2)nnnc1C1(NCCCn2ccnc2)CC(C(F)(F)F)C1 CCN=C(NCC(=O)NOC)NCC1CCCCCC1 c1(CC)cc(=NCC=CCNC(=O)CCSC(F)(F)F)[nH]cn1 C1(C(N2CC(CC(C(=O)N(C)Cc3ncco3)F)C2)=O)CCOC1(C)C N1(C(C2CS(=O)(=O)C2)=O)CCOC2(CCN(c3ncnc(Cl)c3[N+](=O)[O-])C2)C1 C(=O)(C#CC1(C)CC1)NCC1CN(C(C(C(C)C)OC)=O)CC1O C(=O)(CC(C)CC(C)(C)C)N1CC2C(C(N3C(C#C)CC3)=O)(C2)C1 c1(OC)cc(NC(=O)COc2cccc(C(=O)OC(C)=O)n2)ccc1N=[N+]=[N-] c1(C(=O)NC2CC(NC(c3n(C)cc(Br)c3)=O)C2)c[nH]c2cc(F)c(F)cc12 c1(C(=O)NCCN(C(C(n2cnc(C#N)n2)CC)=O)CC(C)O)ccc(Cl)cc1Cl c1(C(NNC(=O)Nc2cc(C)c(N(C)C)cc2)=O)cccc2c(C(=O)O)cccc12 c1(C(=O)NCC(C)N(C(=O)Cc2nc(C(=O)OC)no2)C)cnc(C(C)(C)C)o1 C1(OC)CN(C(=O)C(C#N)C2CC2)CC1CNC(=O)Cc1csc(C2CC2)n1 C1(CNC2C(C(NOC(C(=O)OCC)C)=O)CC=CC2)CC2CC1CC2O n1(CCOC)cc(C(=O)NCC2CCC(NC(=O)CCN(S(C)(=O)=O)C)C2)cn1 c1(C(N(CCC)CCNC(c2cnns2)=O)=O)cnccc1OC c1(OC)cc(C(=O)NC2CC2NC(=O)C(F)n2ccnc2)cnc1Br C(=O)(C(CNC(=O)CCCC1CCC1)c1cn(-c2cccnc2)nn1)OC N1(C(C2(OC)CCOCC2)=O)CC(C)(C)CCC1CNC(=O)Cn1ccnn1 C(=O)(C(C)CC(=O)N1CCCC(CNC(c2ccc(C)cc2SC)=O)CC1)OC C1(NC(C(COC)SC)=O)C=CCN(C(=O)COCCc2ccccc2)C1.C(C)O C(=O)(C#CC1CCCCO1)N1CCC(CNC(c2c(C)cccc2Cl)=O)C1 C1(N(C(c2c(NC)cncc2)=O)C)CCCN(C(C2(C3CC3)CCCO2)=O)CC1 C1(C)(CC(=O)N(C)CC2CCCO2)CCN(C(c2ccnnc2)=O)C1 C12(C(N(CCCC=C)C)=O)CC(CO)(CN1C(=O)CCC1CCCOC1)C2 c1(CC)ccc(C(=O)NCC2(F)CCC(NC(C3CCCC3CC)=O)C2)c(C)c1 c1(NC(C(CN(c2ncc(I)cn2)C)(C)C)=O)ccc(Cl)c(C(F)(F)F)c1 C1(C(N2CCC(CN=c3nc(CC)[nH]s3)CC2)=O)CCc2cncn2C1 N1(C(c2cc(C)n(C(C)C)c2)=O)CCC(C)C(NC(C2CCCCC2(C)C)=O)C1 CC(C)C(C(=O)N1CC(CNC(c2ccc(C)n2C)=O)C2CC12)NC(N)=O n1(CCNC(C23CSC(C2)C3)=O)cc(C2CC2)c(-c2ccccc2)n1 Cc1cc(C(=O)NC2C3CN(C(=O)CC4CN(C)C4)CC23)c2c(c1)C(C)CCN2 c1(C(C)NC(=O)CNC(C2(C)CCOC2)=O)c(F)cncc1F Cc1nc(C)c(C(=O)OCC(C)C)s1.N12CCCC1C(=O)CC2=O c1(C(N2CCC3C(NC(C(CC#C)O)=O)C32)=O)ccc([N+](=O)[O-])nc1 c1(C(=O)NC(CCNC(C(CC(C)C)O)=O)C(C)C)ccc2c(ccn2C)c1 c1(C(CNC(C)=O)NC(c2nnc(C(F)F)o2)=O)cccc(N(C)C)c1 c1(C(C)(C)C)cc(NC(c2ccc(Cl)nc2)c2nnnn2C2(C)CC2)ncn1 Cc1cc(C(=O)NCc2cccc(N3CCC3=O)c2)cc(C)c1Br c1(C(=O)NC(CNC(c2cccc(OC)c2)=O)C2CC2)cc(C(N)=O)ccc1C C#Cc1cnn(C)c1C(=O)NC(CNC(C1CC(C)OC1C)=O)CC(C)C C(C(N=c1cc[nH]c(=NCCc2nccn2C)[nH]1)c1ccc(Cl)cc1Cl)N(C)C N1(C(C2CC(=C)C2)=O)CC(OC)CC1CNC(c1cccc(C(F)F)c1)=O C1(C(=O)NC2CC2)CCN(Cc2ccc(-c3ccccc3F)nc2)CC1(F)F c1(C(=O)NCC(C)C(=O)NC(C)CN2CCCC2=O)ccc(Cl)cc1 c1(C(N2CCC(CNC(c3cc(Cl)c(Cl)s3)=O)C2)=O)ccc(=O)[nH]c1 N1(C(C(C)C)=O)CCC(C(C(=O)NC2CCOC2)N(C(C)C(F)F)C)CC1 C1(C(N2CC(C)C(CNC(C3(C)COC3)=O)C2)=O)CCC2C(C1)C2(F)F c1(OCC)cc(C(=O)NCC2(O)CCCN(C(c3ncccn3)=O)C2)cc(F)c1 C(=O)(C1=CCCC1C)NC(C(=O)NCC(c1cnn(C)c1)C)c1ccoc1 C1(C(=O)NCCC(C)NC(c2cn(C)ccc2=O)=O)C2C3CCC(C3)C12 N1(C(C(CC)OC)=O)CCCCC(N(C(=O)C(C)SC(C)C)C)C1 N1(C(C=Cc2ccc(C)s2)=O)CC2CCCC(N(C)C(C3CCC=CO3)=O)C2C1 N1(C(c2c(C)ocn2)=O)CCC2(CCCN2C(c2cn(C(C)C)cn2)=O)C1 CCC(O)C(F)(F)C(=O)N1CCC1CNC(c1occc1Br)=O c1(C(=O)NC2CCCCN(C(C(CCC#C)O)=O)C2)cc(F)cc(C#C)c1 N1C2CCCC1CC(NC(C(C1CCOC1)OC)=O)C2.C(=O)(CO)NCCN(C)C CC1(CNC(CCO)c2cncs2)CC2CC2C1 C(=O)(C(C(C)CC)N(C)C(C1CCC(C(N)=O)CC1)=O)NC(CCC)C1CCCC1 c1(C(=O)NCC2(O)CCN(C(c3cc(CC)ncn3)=O)C2)c(C)cc(C)nc1C c1(C(N2CCC(F)(C(N)=O)C2)=O)cccc(C(=O)Nc2ccsc2CO)c1.CC N1(C(CSCCCC)=O)CCC(CNC(=O)CC2(NC)CCCC2)C1(C)C c1(C(N2C(CCNC(C=NOC)=O)CCC2)=O)cc(F)cc(F)c1O C1(CN(C(COCC(=O)NC)=O)C)CC(F)CN1C(c1cnsc1C)=O CC1CC1C1CC1C(=O)N(C)CC1CCCN(c2cc(-c3cccs3)ncn2)C1 Cc1cn2cc(C(N3CC4(C3)CN(C(=O)Cc3c[nH]nc3C)C4)=O)cc(C)c2n1 c1(OCC#C)ccc(C(N2CCCC2CNc2ccc(C(=O)NC)cn2)=O)cc1 N1(C(C2CN(OC)C(=O)C2)=O)CCC2(CC1)CC2C(=O)NCC1COC(=O)N1 N1(C(c2scc(C#N)c2)=O)CCC2(CCN(C(c3c(F)ccnc3F)=O)CC2)C1 Cc1cc(C(N2CC=C(C(=O)NCC3CC4OC3C3CC43)C2)=O)cc(C)n1 C1(NC(C(CNC(C2N(CC)CCCC2)=O)O)=O)CCCC(C)(C)C1 S(=O)(=O)(c1cccc(Cl)c1Cl)N1C2CN(C(=O)Nc3cc(Cl)c(Cl)c(Cl)c3)CC21 Cc1ccc2c(c1)CN(C(c1csc(Cl)n1)C(=O)NC1(C)CC1)C2 CN1CCCC(CC(=O)NC2CC(CC(=O)NC3CCN(C(N)=O)CC3)C2)C1 C1(CNC(c2[nH]cc(C)c2)=O)CC(C(C)C)CCN1C(c1cc(=O)n(C)cn1)=O c1(C(N(CCNC(C2C(C=C)OCC2)=O)C2CC2)=O)cccc(=S)n1O c1(CC(=O)NC(CN(C(C2C(C#C)C2)=O)C)C)ccc(C)nc1 c1(C(=O)NC2C(C)CN(C(CNC(C)=O)=O)CC2C)cc(Cl)c2c(c1)OCCO2 CCC(C)(CCNC(C1CCCC1SC)=O)NC(c1ocnc1C(C)C)=O C1(N(C)C)CCC(C(=O)Nc2ccoc2CNC(=O)CC(F)F)CC1 Cc1cccc(C(N2CC=CC2C(=O)N(C(C)CO)C)=O)c1C Cc1c(Cl)cnn1CC(=O)N(C1CCC(NC(=O)CS(=O)(=O)N(C)C)CC1)C N1(C(COCCOCC)=O)CCC(N(C(=O)C=Cc2cncs2)C)CC1 Cc1nc(C(N2CCC(C(=O)NC3(C)CC(O)C3)(CF)C2)=O)c(C)o1 c1(C(C)C)ccc(C(=O)NC2CCCN(C(=O)C(C)NC(C)(C)C)C2)c(CO)c1 c1(C(=O)NCC2C(C(=O)Nc3nc(C)c(C)s3)CCCC2)cnn2c1CCC2 C(=O)(C1CCCc2nncn21)N(CC(C)NC(c1sccc1C(C)(C)C)=O)CC C1(C(N2CC3CC(C)C3C2)=O)CC2(CCN(C(=O)C(C)(F)F)C2)C1 C1(O)(CN(C(=O)Cc2n[nH]c(=N)s2)C)CCN(C(C2C3(CC3)C23CC3)=O)C1 S(=O)(=O)(c1cc2ccccc2cc1C(C)=O)Nc1c(C(=O)OCC)cccc1 C1(C#N)(C(=O)NCCN(CC(C)O)C(=O)C=Cc2nccs2)CC1(C)C C12CN(CCO1)CCOC2=O.C(=O)(C(C)Cn1cccn1)C(N1CC(OC)C1)=O C1(NC(C2(C(N)=O)CC2)=O)CN(C(=O)CC2C=CCC2)CC1C(F)F c1(C(N2CCCC2)=O)cnc2ccccn12.CCC(CSC)N CCCCC(CNC(C1(NC(C)=O)CC1)=O)NC(c1cnnn1CCOC)=O C1(C(C)C)COCCN(C(C2CCC2NC(=O)CC(C)(C)C#N)=O)C1 Cc1cnnc(O)c1C(=O)NCCC(O)CNC(=O)CCc1cccn1C c1(C(N(CCCNC(c2coc3c2CSC3)=O)C)=O)cc(F)c(F)c(F)c1N C1(CC(=O)NC(C)CCNC(c2cc(C#N)c[nH]2)=O)CCC(C)C(C)C1 c1(C(=O)NCC23CC(NC(C4CC5CC4CO5)=O)(C2)C3)cc2cc(Cl)ncc2[nH]1 C1(NC(c2scc(C(=O)OCC)c2)=O)CCCC(NC(c2cnc(O)nc2)=O)C1 CC(C)(C)CC(=O)NCC(C1CCCN(C(=O)CCOC2CC2)C1)F c1(C(=O)NCC2CC(OC)CN2C(c2ccc(Cl)cc2)=O)ccc2cc[nH]c2n1 C1(C(=O)OC)CCN(C(=O)c2ncoc2-c2cn(-c3ccccc3)nn2)O1 CCCCCCCCCc1cn[nH]c1.C12(C#N)CCN(C1)C2c1cccnc1F Cn1nc(C(=O)N(CCNC(c2cn(CCCC#N)nn2)=O)C2CC2)cc1F N1(C(c2csc(C)c2C)=O)CCCC1C1CCCN1C(c1cnc(NC(N)=O)o1)=O c1(C(=O)NC(CCOC)CNC(C2CCCN2N=O)=O)cc2c(cc1Cl)OCO2 c1(CC(=O)NCC(CC(C)C)NC(c2cccc(N)c2)=O)ccc2occc2c1 C1(CC=C)(NC(=O)C=CBr)CCN(C(C2CCCOC2)=O)C1 N1(C(CC(=C=C)C)=O)CCN(C(=O)Cc2ccsn2)CC1CS(C)(=O)=O Cc1cc(NC(=O)CC23CCCC2C3)ncc1[N+](=O)[O-] C1(NC(=O)CC2CC=CC2)CN(C(=O)C(O)C2CC2)C2(CCOCC2)C1 C(=O)(CC(CNC(C1CC12CCC2)=O)C1CCC1)N(C1CCSCC1)C Cc1cnc(C(N2CCOC(CNC(=O)C(=O)N(C)C)C2)=O)cc1C#N c1(OCC)nccc(C)c1C(=O)NCC1CC1NC(=O)C(N1CCOCC1)C C1(NC(C(CSC)(C)C)=O)CC2CN(C(=O)COC3CCOCC3)CC2C1 C1(N(C(c2ccn(C)c2)=O)CC)CCCN(C(=O)CCC2C(=O)ON=C2C)C1 c1(C(N(CCC)CCNC(C2CC2CC)=O)=O)ccc(OC)c(N)c1 N1(C(C(Cc2c(C)nc[nH]2)O)=O)CCN(C)CC1CNC(c1cnc(Cl)s1)=O c1(C(=O)NC(CNC(CC2CCCC(C)O2)=O)(C)C)cccc2[nH]ncc12 c1(C(c2nnnn2CCSC2CCC2)SCC)cc(F)ccc1CNC1CCC1 c1(C(=O)NCCCC(C)NC(COC(C)C)=O)ccc([N+](=O)[O-])o1 C1(C(=O)NCC2N(C(C=C(C)C(F)F)=O)CCC2)CC2(C1)CC21CCC1 c1(C(N2CC(C(C)NC(C3C(C=C)CC3)=O)OCC2)=O)cc(N)cnc1Cl c1(CNC(=O)NC2CCN(C(C)=O)CC2)nc2cc(Cl)cnc2[nH]1 N1(C(c2c(OC)c[nH]n2)=O)CC2(NC(c3cn(C)nc3Br)=O)CCC1C2 N1(CC)CC(C(N2CC(C(N3CCC4CCCC34)=O)C3(CC3)C2)=O)CCC1=O C1(N(C(c2cn(CC)nc2C(C)C)=O)C)CCCN(C(c2cc[nH]c2C)=O)CC1 CC(C)CC(CNC(=O)Cc1cn[nH]c1)C(=O)N1CCC(O)(C(F)(F)F)C1 C1(CC)CCCN(C(=O)CCCc2cnn[nH]2)C1C(=O)NC1(CO)CCC1 CCCC(C(=O)NCC1(C(=O)NCC(C)(C)n2ccnc2)CC1)OC CC1C(=O)N2CC(C2)CS(=O)(=O)O1.C1(NC(=O)COCC(F)F)CCCC1 C(F)(c1ccccc1)=CCCOC(c1ncoc1C1CCCCC1)=O C(=O)(C(C(=O)OC(C)(C)C)C1CC1)NCC(C)Cn1cc(C2(C)CCCO2)nn1 c1(C(CC)NC(c2ccc(Sc3ccsc3)cc2)=O)ccccc1OCCO Cc1c(C(=O)NCC23CC(C2)C(NC(=O)C(C)N(C)C)CO3)sc2ccccc12 CC1(C)CCN(C(=O)Cc2ccc(CO)cc2)CC1CNC(=O)CC(F)(F)F Cc1noc(Cl)c1CCC(=O)N(C1CCN(C(=O)C(C)(C)C2CCCO2)C1)C c1(CC(=O)N)sc2ccccc2c1Cl.N12CC3CN(CC13)c1ncc(Br)c2n1.[nH]1cc(I)cc1 c1(C(N2CC(N(C(CCCOC)=O)C)C(C)(C)C2)=O)cc2cccnn2n1 c1(OC)cc(OC)c(F)c(C(N2CCC2CNC(=O)C(C)n2cccn2)=O)c1 c1(NC(CN(C(C)=O)C)=O)ccc(NC(C2CC2C(N)=O)=O)c(C)c1 N1(C(C(C2CCOCC2)OC)=O)CC2(CC(NC(C3CC(F)C(=O)N3C)=O)C2)C1 C(C)(C(=O)O)(C(CCN)CCNC(=O)COCC(F)F)OC C1(NC(=O)CCc2ccsc2Br)CCCC12CN(C(=O)CO)C2 C(C(C)C)(C(O)C(=O)NC1(C(=O)O)CC(O)CCC1)OC c1(C(=O)NC(C(C)NC(C2CCCO2)=O)C)nn(C)c2c1CCC2 C1(=O)C(C)CCN1.C1(C)(OCC)CN(C(=O)C(CN(C)C)N(C)C)C1 C1(CNC(c2c(C)noc2C)=O)CCN(C(=O)CCCC(=O)C2CC2)C12CC2 CCC(CC)(CCC(=O)NC(=O)C1=NOC2COCC12)[N+](=O)[O-].C1CCCN1C Cc1cc(C(=O)N(CC(C)NC(C2(C3CCCCO3)CC2)=O)C)nn1C(F)F C(CCCCNC(=O)CSc1nncn1C)N(C(C1C(OCC)C1)=O)C C#Cc1ccc(C(=O)NC2CCC(C(=O)N(CC)CC3CCOC3)CC2)cc1C C1(NS(=O)(=O)c2cccs2)CCCC(N=c2ccn3nccc3[nH]2)C1 C1(C)(CNC(C2C(C)OC(=O)N2)=O)CCCN(C(C2(CC(F)F)CCC2)=O)C1 C1(C(N(C2CCN(C(c3ccccc3Cl)=O)C2)CCC)=O)CC(=O)N(CC)C1 c1(-n2cc(CC(CC(=O)O)ONC(c3csc(Br)n3)=O)nn2)cc(F)ccc1F CC1C(NC(=O)CCCN=[N+]=[N-])CCCN1C(c1cnc(C(F)F)nc1)=O C1(NC(C(CCSC)NC(N)=O)=O)CC2CC1CN(C(=O)CCN(C)C1CC1)C2 Cc1sc(C(=O)NC2CCN(C3CN(C(=O)COC4(C)CCC4)C3)CC2)c(C)c1C N1(C(C(C)CN(C(=O)Cc2cccc(C)c2)CCC)=O)CCC2(CC=CCO2)C1 C1(O)(CCNC(C2CCCN2C(=O)C(=O)Nc2cnns2)=O)CCCCC1 C1(C(=O)NCCCNC(C=C(CCC)C)=O)(CCF)CCOCC1 Cc1nc(C)c(C(=O)NC2CCCC2(C)C(N2CCC(C(F)C(=O)O)C2)=O)o1 C1(CNC(C2(CSC)CC2)=O)CCN(C(C2OCCC2C(C)C)=O)C1 C1(NC(c2nccc(C)n2)=O)CCOC12CCN(C(c1ccc(Cl)cn1)=O)CC2 N1(C(c2c(N)cccc2)=O)CC2(CCCC(CCO)O2)C1 c1(N2CCC(CC=C)(NC(=O)C(=O)N=S(C)(C)=O)CC2)nc2c(C)cccc2o1 C1(N(C)C(C2CC2C#N)=O)CCN(C(C2CCCN2C(C2CCOC2)=O)=O)CC1 c1(C(N2CCC(NC(C(C)SC)=O)C(O)C2)=O)cnc2ccnn2c1N C1(NC(CC(CC)NC(c2cnc(OC)s2)=O)=O)CCCCC1C#N C1(NC(CC2(CC)CCC2)=O)CN(C(=O)CSCCOC)CC(C)(C)C1 Cc1ccc(-c2ccc(NCCCNC(=O)C(N3CCSCC3)C)o2)cc1 c1(NC2C(F)CCN(S(=O)(=O)c3cn[nH]c3)C2)c(C(F)(F)F)ccc2[nH]ccc12 c1(C(C(=O)NCc2c(CNC(C=CC)=O)ocn2)(C)C)ccc(F)c(F)c1 C1(NC(=O)NC(C)(C)C)CC2CC(O)C(C1)C2.C1(=O)C(C(C)(C)C)O1 N1(C(CC(=O)NCC)=O)CCN(C2CN(CCn3ccc(COC)n3)C2)C(=O)C1 Cc1nc2ncc(C(N3CCC(NC(C4CC4CC(C)(C)C)=O)C3)=O)c(=O)n2[nH]1 c1(C(N2CCCC(N(C(CCOCC)=O)C)C2)=O)ccc(F)c(N)c1Br C1(C)(CC(=O)N(CC(C)(CO)NC(CSc2n(C)nnn2)=O)CC)CCCCCC1 C1(NC(C(C(C)C)CO)=O)CCC2(CC1)CCN(C(=O)Cc1cn(C)cn1)C2 c1(CC)cnccc1C(=O)NC1CCCCC1NC(c1c(C2CC2)cnn1C)=O N1(C(c2c(Cl)cc(OC)s2)=O)CC2(CC(NC(=O)C=CCOC(C)(C)C)CO2)C1 C1(CC)CCCN(C(=O)C=CCNC(C)=O)C1C(N1CCCC(NC)C1C)=O C(CN=c1nc(N2CCCC(C3CCCCO3)C2)c2c([nH]1)CCOC2)SC CCCC(C)(C)C(=O)N1CC(C(=O)Nc2cccc(C(C)O)c2)C(O)C1 Cc1cn2nnc(C(=O)NC3CN(C(=O)C=Cc4ccco4)CC3C)c2c(O)n1 c1(C(=O)NC2CC(Nc3cc(OC)nc(C)n3)C2)cc2cccc(C)c2[nH]1 C1(O)(C(C(=O)OCC)F)CN(C(N2CCC(C)C2)=O)C1 N1(C(C2(C)CC(F)C2)=O)CCCCC(NC(=O)CNC(C2CCC2)=O)C1 N1(C(C(F)=CC)=O)CC(N(C)C(c2cn(C)nc2C2CCOC2)=O)C(F)C1 C1(CNC(c2c(C)ccc(Cl)c2)=O)CN(C(c2cc(Cl)sc2Cl)=O)CCC1(C)C N1(C(C(C)OCC)=O)CC2C(NC(=O)CC)C2C1 N1(Cc2cc(OC)no2)CCCC(O)(OCC(=O)Nc2ccc(F)c(F)c2)CC1 C(=O)(CCNC(=O)NC1C(CN)C1)N(C(C)C)CC.C(=O)(N(C)C)OC Cc1cc(C(=O)N(CCC(C)NC(c2cnc(N(C)C)nc2)=O)C)ccc1Cl CC1=C(C(=O)N2CC(NC(=O)C3=CCCCC3C)C(O)C2)Cn2ncnc2N1C N1(C(C(c2ccncc2)C)=O)CC2CCC1(CNC(=O)CC(C)(C)O)CC2 C12CCCC13CCN(C3)C2=O.c1(NC(Cc2cncc(C)n2)=O)ncc(Br)cc1O N1(C(CCc2n[nH]c(=N)s2)=O)CCCCCC1CNC(=O)C=CC1CCC1 c1(C(N2CC(NC(C3C(C(C)C)OCC3)=O)C2)=O)ccc(-c2nnc(S)o2)cc1 Cc1ccc(C#N)cc1C(=O)NCCN(C(=O)C(C)(C)C(F)F)CC1CC1 N#CC1CCCC(C(N2CCC(NC(=O)Cc3ccon3)C2)=O)C1 c1(C(=O)NCC(CNC(COCCOC)=O)(C)C)c(N)ccc(Br)c1F Cc1c(Br)noc1C(=O)N(C(C)CNC(C1(CS(N)(=O)=O)COC1)=O)C Cc1cc(C(=O)NCC(C2(O)CN(C(C3CCCCS3)=O)C2)(C)C)cc(C)n1 CC(CNC(c1c(C#N)ncn1C)=O)C(F)C(=O)NC1CC(CO)(CO)C1 N1(C(CC)=O)CCN(Cc2cccc(C(F)(F)F)c2)C(CC)C1 c1(CC(=O)NC2C(NC(=O)C=Cc3cscn3)C2)c[nH]c2ccccc12 N1(C(COCC(=O)NC)=O)CC2CC1CN(C(=O)C(C)=C1CCC1)C2 C1(C(=O)NCCC2(NC(C3C(CC)C3)=O)CCC2)CC12CC(O)C2 CCC(CCC(=O)N1CCCC(C(=O)N(CC(C)(C)C#N)C(C)C)C1)OC N1(C(c2cc(C)on2)=O)CCN(C(c2cnn(CCO)c2C)=O)CC(O)C1 Cc1oc(Cl)nc1C(=O)NCC(CC1CC1)C(=O)NC(CO)CCOC C1(C2CC2)(NC(C23N(C(C4CC45CCCCC5)=O)CCC2C3)=O)CCCCC1 c1(C(=O)NCC2OCCC(NC(C3CC(O)(CC#C)C3)=O)C2)cc(Cl)c(C)cn1 c1(C(=O)NCCC(C)N(C(=O)CC#N)C)cccc2ccccc12 C(=O)(C1=NOC(C)(C)C1)NCCC1(C)CCN(C(c2cn(CCOC)nn2)=O)C1 C#Cc1ccc(C(=O)NCC2CN(C(=O)CCC=C)CCCO2)nc1 c1(CNC(c2cnc(CC)s2)=O)cnn(C)c1C(=O)N(CC(COC)OC)C C12(CNC(=O)Cc3cc(Br)cs3)CC1CN(C(=O)CN1CCOCC1)C2 CCCC(C(=O)N1CC(N2CC(NC(C3(CC)COC3)=O)CC2=O)C1)OCC c1(CNCCN(C(Cc2c(C)nc(CC)nc2C)=O)C)ccc2nc(C)[nH]c2c1 Cc1cc(Cl)ccc1OCC(N1CCC(O)C1C(=O)NCc1ccc(Cl)nc1)=O C1(C2(NC(c3cnc(C4CC4)[nH]3)=O)CC2)CCCN1C(C1CC1CF)=O CC(C)CCC(C(=O)NC1CC1)NC(c1cccc(Cl)c1)=O c1(C(N2CCC(C(C)NC(C(C=CC)O)=O)CC2)=O)cc2n(n1)CC1(CC1)C2 N1(C(c2c(CCC)nns2)=O)CCOC(C(C)NC(c2cnco2)=O)C1 N1(C(C=CC(C)C)=O)CCC2CN(C(=O)CSn3cncn3)CC2C1 n1(CC=C)cc(C(=O)N(C(CC)C(=O)NC2CCN(CC(N)=O)C2)C)nn1 N1(C(CC2CC(=O)OC2)=O)CC2C(CNC(c3ccc(CO)nc3)=O)C2C1 N1(C(c2cccc(N(C)C)c2)=O)CCCCC(CNC(=O)C=Cc2cncs2)C1 c1(C(C)C)nc2c([nH]1)CC(C(=O)N(C(C)CNC(C1C=CC=CC=C1)=O)C)CC2 C1(NC(COc2ccc(OC)cc2)=O)CN(C(c2ccsn2)=O)CCC1F C(=O)(CCC(CC)SC)NC1(CC=C)CN(C(c2cc(COC)cs2)=O)C1 Cc1cc(C(=O)NC2CC(CNC(=O)C(F)CC3CCC3)CC2O)c(C)nc1C Cn1nc(C(F)(F)F)c(I)c1CNC(c1cc(-n2cnnn2)cc(Br)c1)=O C1(O)(CC(C)C)CCN(C(=O)C(c2cccs2)NC(c2ccnn2C)=O)C1 N1(C(C2(CO)CC(C)(C)C2)=O)CCCC(CC(=O)NCC(=O)NCC2CC2)CC1 C(=O)(CC(F)(F)C(F)F)NCC1CC(OC)CN1C(c1cnn(C(F)F)c1)=O CCCC(C)(O)CC(=O)NCCC1COCCN1C(=O)C=Cc1cocn1 CC1CC(C)(C(=O)Cn2cc(-c3ccc(OC(F)(F)F)cc3)nn2)CCO1 c1(CNC(C(CNC(c2scc(C)c2C)=O)C)=O)ccc(C#N)cc1 c1(CNC(COCC=C)=O)ccccc1CNC(C1CC(C)C1(C)C)=O C1(CC(=O)N(CCN(C(c2nc(Br)c[nH]2)=O)CC)CC)CCC(C)CC1 N1(C(C)C)CC2CC(NCCNC(=NCC3(F)CCCC3)NC3CCC3)CC2C1 c1(OCC(N2CCC(NC(C(C)c3cc[nH]n3)=O)C2)=O)cccc(F)c1 C#Cc1ccc(C(N2CC3CC2CN(C(=O)CC2COCC2O)C3)=O)cc1Cl c1(NC(C(CC)NC(c2cn(C)cn2)=O)=O)cncc(OC)c1 C1(OC)CC2(C1)NC(=O)N(Cc1cc3ccc(Br)cc3o1)C2=O c1(C(N2CCCN(C(C(CCSC)O)=O)CC2)=O)csc2ccc(F)cc12 N1(C(Cn2nc(C)c(Cl)c2)=O)CC(NC(C2CCNC(=O)C2)=O)C2CC2C1 CCCCCC(F)C(=O)N1CC(CNC(=O)CNC(=O)CCC)(OC)C1 CCCC(CNC(c1ccc(F)c(O)c1)=O)C(=O)NCCC1(C)CCOC1 C1(CNC(C(CC)F)=O)CN(CCc2cn(Cc3ccc(F)cc3)nn2)CCO1 C1(N(C)CC)CCN(C(C2CCN(C(=O)C#CC3CC3)C2C)=O)CC1 N1(CCC(=O)NC2COCCN2)CC2C3CC(C2)CC1C3.c1(CO)ccccc1 CC(C)(C)C(CNC(=O)CCNC(C1CCC1)=O)NC(C1OCCO1)=O c1(C(C(=O)NCc2ccccc2)N(C2CCC(=O)NC2)C)cnn2c1CCC2 CCC(C)(O)C(=O)NC1CCCCC1CC(=O)N(C1CCOC(C)C1)C N1(C(CN(C)C)=O)CCN(C(c2cnc(N)c(Br)c2)=O)C(CC(F)F)C1 c1(C(C)OCC)nc(C(N2CC(CC3CC3)C2)=O)c(C)o1.C(CC(F)(F)F)N(C)C1CC1 c1(C(=O)NC2CN(CC3CCN(C)C3)C2)cc2c(nc1O)CCC(C(C)(C)C)C2 Nc1c(Cl)c(NC(c2ccc(Cn3cccc3)cc2)=O)nc(F)c1Cl C1(C(=O)Nc2nnc(C3N(CC#C)CCC3)s2)CCC(C(=O)OC)CC1 CCC(C)(CCC(C)C)C(=O)N1CC(N(C(=O)COCC(C)(C)C)C)C1 c1(C(N2CCC(CCOC)(NC(=O)C(C)=C(C)C)C2)=O)cccc2scnc12 C1(C(=O)NC(C2CC2C(=O)NC2CCCC2)C)CCc2n[nH]cc2C1 N1(C(C(CC)O)=O)CCOC(c2cn(CC(c3ccccn3)(F)F)nn2)C1 C(=O)(C1=CC2C=CC(C1)C2)N1C2(C(=O)NC3(CC)CCC3)CC2CC1 C1(S(=O)(=O)c2ccccc2)(C(=O)NC(CNC(=O)CC2CC=CC2)C2CC2)CC1 C(=O)(C1=CN(Cc2cc(OC(F)(F)F)cc(F)c2)CCC1)N1CC(C)OCC1 N1(C(C(C2CCCN(C(c3c(C(C)C)occ3)=O)C2)C)=O)CCC(F)(F)C(F)C1 c1(C(=O)NCCC(C)N(C)C(C2CCN(C3CC3)C2=O)=O)ccc(N)c(Cl)c1 O=S(=O)(c1ccccc1)CN1CCN(S(=O)(=O)c2ccccn2)C(C(F)(F)F)C1 c1(CC(=O)NC(C)CC(C)NC(=O)CCNC(N)=O)ccc(N(C)C)nc1 CC(C)C1=NOC(C)(C(N2CCC(F)(CNC(c3cn(C)cn3)=O)C2)=O)C1 c1(C(N2C(COC)CC(OC)C2)C(=O)NC2CCC2)ccc(Br)cc1F c1(C(=O)NC2(C)CN(C(CCc3cc(C)on3)=O)C2)ccc2c(c1)N(C)CCO2 N1(C(C=CSC)=O)CCC=CC1C(N1CCC(c2cnco2)C1)=O C1(C)(NC(c2c(CC)nccn2)=O)CC12CCN(c1ncccc1OCC)CC2 N1(C(C(CCCC)O)=O)CC(NC(C23CC(C(F)F)(CO2)C3)=O)C2CCCC2C1 c1(C(N(CC(=O)NCC(=O)N(C)C)CC#C)=O)cccc(C)c1C c1(C(N(CCCNC(C2C(C)OCC2)=O)C)=O)cc(C(F)F)ccn1 c1(CC(N2CC(CN(C(C3CCC(C)C3)=O)C)C2)=O)noc2ccc(F)cc12 CC1=NOC2(C1)CC(C(=O)NCC(C)N(C)C(C1CC(C)(C)C1)=O)C2 C12(NC(C3(CNC(CC(COC)(C)C)=O)CC3)=O)CC3CC(CC1C3)C2 c1(C(N2CCC(C)(C(N3CC4CSCC4C3)=O)C2)=O)cccc2cnnc(O)c12 c1(C(=O)NCC(CNC(=O)C=C(C)C(F)F)OC)ccc(Br)c(N)n1 Cc1nc(C(N2CCN(C(c3ccnnc3C)=O)CC(O)C2)=O)c2n1CCCC2 c1(OC)c(-c2nc(CCSC)nn2-c2cccc(F)c2)cccc1Br Cc1cc(F)ccc1C(N1CCCC(N(C(=O)C=Cc2ccc(Cl)s2)C)C1)=O C(=O)(C(O)C(F)F)NCCCN(C(CC1(OC)CCC1)=O)CC1CCCC1 Cc1cc(C=CC(N2CCCC2CN(C(=O)CCCC(N)=O)C)=O)c[nH]c1=N CC(C)C(C(=O)N1CC(Cn2cc(CNC(C3CCNC3=O)=O)nn2)C1)N(C)C C1(C(N(C2(C(N3CC(NC(C)=O)C3)=O)CCCC2)C(C)C)=O)CCCC(C2CC2)O1 C(=O)(C(C)(C)C(F)(F)F)NCC1N(C)CCN(c2ncnc(CC(=O)OC)c2F)C1 n1(C(C)C)ncc(C(=O)NC(CO)C(C)NC(C2(O)CCOC2)=O)c1C(F)(F)F N1(C(COC(C(CC)(C)C(F)(F)F)=O)=O)Cc2ccccc2CC1CO CC1CCC(NC(c2ccc(C3CC3)cn2)=O)CN1C(C1CCC(C)CC1)=O C1(C(N(CCN(CC=C)C)CC)=O)CC(CO)N(C(=O)Cc2cc[nH]n2)C1 n1(CC#C)cccc1C(=O)NCCC(C)N(C(=O)CC1(COC)CC1)C Cc1oc(C)c(C(=O)N(CCCC(=O)NCc2cccc(Cl)n2)C)c1C c1(C(=O)NC(CN(C(=O)COCc2cccs2)CC)C)cc2c(s1)CN(C)CC2 C1(C(=O)NCC2CC(O)C23CCC3)CCCCCCN1C(=O)CC1CCOC1=O Cc1ccc(O)c(C(N2CC3CC3(NC(=O)C=CSCc3ccco3)C2)=O)c1 c1(C(N2CC3C(NC(C(C(C)C)OCC)=O)(C3)C2)=O)cccc2c1NCCC2 C(=O)(C(C)(C)CCCNC(c1ccnc(O)c1)=O)NC(C)Cc1ccncc1 N1(C(C2C(C)C2)=O)CCC(N(C(=O)CSCc2cccs2)CC2CC2)CC1 C1(NC(c2n(C)ncc2)=O)CN(C(c2cc(-c3cccc(Br)c3)no2)=O)CC1F N1(C(C(CCCC)CC)=O)CC(NC(c2ccnnc2)=O)CC12CCCCCC2 Cc1cc(O)ccc1CC(=O)NCCC1CC(NC(=O)CC2CSCCS2)C1 N1(CC(c2noc3c2COCC3)=O)CCOc2cc(Cl)c(Cl)cc21 c1(C(C(C)NCCc2ccnc(N3CCOC(C)(C)C3)n2)O)c(F)cccc1F C12(NC(C=C(CCC)C)=O)CCOCC1CN(C(=O)CC(CC)CC)C2 c1(NC(CC(C)NC(c2ccc(F)c(O)c2)=O)=O)cccc2c1OCO2 N1(C(C)=O)CCCCC1C(=O)N(C)CC1(CNC(=O)C(C)(C)n2cc(Cl)cn2)CC1 C1(NC(c2c(C)nn(C)n2)=O)CN(C(=O)C(N2CCSCC2)C)CC1(C)C c1(C(=O)NCCCCNC(=O)COCc2cccnc2)ccc2scnc2c1 c1(NC(N2CC(C(C)C)N(C)CC2)=O)cc(S(=O)(=O)C(C)C)ccc1N(C)C C(=O)(CCC(=O)NCC1(C)CC(NC(C2CC(CC(C)(C)C)C2)=O)C1)NC N1(C(c2c(C)con2)=O)CCC(C(=O)NC2(CCO)CCC2)CC1(C)C N1(C(c2c(C)ncnc2)=O)CC2CCC(CNC(=O)CC3CCC3(F)F)(C2)C1 c1(NC(C(CNC(=O)C#CC(C)(C)C)N(C)C)=O)ccc2nc[nH]c2c1 N1(C(=O)NC2Cc3c(nc(C)s3)CC2)CCN2C(=O)NCCC2C1 C1(CC(=O)NC2C=CCN(C(C3C(Cl)(Cl)C34CC4)=O)C2)CCCCCC1 c1(-n2c(N(C)CC3CC3)nnc2-c2ccoc2)ccc2c(c1)OCCO2 C1(CNC(C(c2ccoc2)NC(C2C(CC(C)C)C2)=O)=O)CCC(CO)O1 CCC(CC)C(=O)NCC(C1CCOC1)NC(=O)C=Cc1ccsc1 N1(C(C2C(CC)OCC2)=O)CC2C(C1)C2N=c1[nH]nc(-c2cccnc2)s1 C=C=CCCC(=O)N1CCC(C2OCCCC2NC(=O)CC2(O)CCC2)CC1 N1(C(C2C(C)=CCS2)=O)C(C(N2CCCN(C)CC2)=O)C2CC(O)C1C2 C(CCCCC(=O)NC1CCCN(C(=O)CC2CN3CCC2CC3)C1)N(C)C1CC1 c12cc(ccc1C)C1CC(n3cc(nn3)C3OCCN(C3)C2=O)C1.C(C)(C)C.CO N1(C(C(COC)(C)C)=O)CC2CN(C(c3cccc([N+](=O)[O-])c3C)=O)CC2(C)C1 N1(C(C2ON=C(C)C2)=O)CCCC(C)(NC(C2(C)CCC(C)C2)=O)C1 c1(C(=O)Nc2cncc(NC(=O)OC(C)(C)C)c2)ccc(S(N)(=O)=O)cc1Cl C1(c2ccccc2)(C(=O)NCC2CN(C(CCOCCC)=O)C2)CC1(Cl)Cl C1(NC(C=CC=CCC)=O)CCCC12CCN(C(c1cn(C)nc1C(C)C)=O)C2 Cc1ncnc(N(C2CN(C(=O)C(C)n3ccnc3)C2)C)c1F C(C(=O)NC(c1ncc(F)cn1)C)(C(C)(C)C)NC(c1c(COC)nco1)=O CC1(C)CC1(O)C(N1CCC(OCCNC(c2ccc[nH]2)=O)C1)=O C(C(C)C(C)C(=O)NCC1(C(=O)NCC=CCSC)CCCC1)OC C1(C(=O)NCCN(CCC)C(C23CC(N(C)C)(C2)C3)=O)CC(=O)N(C2CCCC2)C1 CC(CC(=O)NCc1ccc(C(N2CCN3CCC2CC3)=O)cc1)CC(C)(C)C N1(C(CN(C)C(C2CCCOC2)=O)=O)CCNC(=O)C1CCO N1(C(=O)NC(c2ccc(OC)cc2)CF)CC(O)CC2(CCOCC2)C1 C1(C2CCN(C(=O)Cn3cc(N)cn3)CC2)(NC(Cc2ccc(C)o2)=O)CC1 N1(C(c2c(C)oc(Cl)c2)=O)CCC2(CCN(c3ncc(Br)c(C)n3)C2)C1 C1(C(=O)NCC(CC)(CC)NC(C2(C)CCC(=O)NC2)=O)CCCC(C)=C(C)C1 c1(CC(=O)NCCC(C)NC(C2CCOCC2)=O)ccnc(Cl)c1F Cc1noc(Cl)c1CCC(=O)NC1CC(=O)N(C2CN(C(=O)CC(C)N(C)C)C2)C1 c1(C(=O)OC)cnc(OC)nc1C(=O)NNC(=O)c1cc(C)[nH]n1 C1(OC)CC(NC(c2cnn[nH]2)=O)C12CCN(C(c1ccc(Cl)c(F)c1)=O)CC2 CN1CC2(CCN2C(=O)C(C2CCN(C(=O)Cn3cccc3)C2)F)C1 C(=O)(C1=CCCCO1)NC12CC(CNC(c3n(C)cc(Br)c3)=O)(OC1)C2 C=CCC(C)(C)CC(=O)NC(C(=O)NC1(CC=C)CCC1)C1CCOC1 N1(C(c2ccc(CCC)cc2)=O)CCC2CCC(NC(=O)C(C)(C)F)C1C2 CCCCN=C(NCC=Cc1cccs1)NCc1ccnc(NC)c1 c1(Nc2c(C)cn(C)n2)cc(Br)ccc1S(=O)(=O)N1CCCC(C(C)C)CC1 N1(C(C2(F)C(C)C2)=O)CC(C2(NC(c3coc(Br)n3)=O)CC2)C1 C(CCC1CC1)(C(=O)NC(C)C(C)(C)O)NC(C(C)SC(C)C)=O N1(C(=O)Cn2cccc2)CC(C(N2CC(C)C(C(=O)OC(C)(C)C)C2)=O)CCC1C N1(C(c2c(CC)noc2)=O)C2CCC1C1CC1(NC(C1CN(C(N)=O)C1)=O)C2 C1(CC(=O)Nc2c(C)csn2)C=CS(=O)(=O)C1.C(C)(C)(C)N(CC=CC)CC C1(C(=O)NC(CCC(=O)OC)C)CCC(O)CN1C(=O)C=CC1(C)COC1 C1(NC(C(C)SC)=O)C=CCN(C(=O)CCNC(=O)C=CCl)C1 c1(C(N2C(C(=O)Nc3cccc(CF)c3)CCC2)=O)cc(Cl)c(Cl)cn1 c1(C(N(C(C)CNC(C2(CC)CCC2)=O)CC)=O)cc(Cl)c(F)c(Cl)c1 C(=O)(C#CC1(CC)CC1)N(CC12C(CN(C(C3(SCC)CC3)=O)C1)C2)C1CC1 C1(C(=O)OC)C(C)CCN1C(=O)CC1CN(C(C2OCCC2C)=O)C1 c1(CN(C(C)=O)C)ccc(NC(N2CCCC2c2ccn(C)n2)=O)cc1 N1(C(c2csc(-c3csc(C(F)(F)F)c3)n2)=O)CC2CCCCC1C2 O=C(C1=CCCCO1)NCC(O)CCNC(=O)Cn1cnc(C(N)=O)n1 c1(C(N2C(C(C)NC(C3CCCC3O)=O)CCC2)=O)ccc(C2CC2)nc1O N1(C(C)=O)CCOC(CC(=O)NC(C2CCN(Cc3cccc(C)n3)CC2)=O)C1 C(C(CC1CC1)C(=O)NCc1cccnc1)NC(CC1CC(=C)C1)=O Cc1c(N)ccc(C(=O)N(C)CC2CN(C(=O)C(C)CO)CCO2)c1Cl C(=O)(C(CCC(C)C)NC(=O)C(C)C)NC(CC)C1CC1 C=C(C)CC(C(=O)NC(C(O)CO)C1CC1)NC(=O)CC1CCC=CCC1 C1(C)(C(=O)NC23CC(C)(C2)C3)CN(C(=O)Cc2ccc(F)nc2)C(C)(C)C1 C(=O)(C1CCCc2ncnn21)N(CCCCN(C(=O)C1=CS(=O)(=O)CCC1)C)C N1(C(C2(F)CCN(C(c3cc(COC)no3)=O)CC2)=O)CCCC(F)(F)CC1 CC1(C)CCC1(C(=O)O)NC(c1c[nH]nc1C1CCCO1)=O C1(C(=O)NC2CC(C)C2)CCc2nc(-c3cccc4ccncc34)sc2C1 c1(C(=O)NC2CCN(C(CNC(=O)OCC=C)=O)C2)cc2cc(F)c(Cl)cc2[nH]1 C(=O)(CCCS(N)(=O)=O)N(C1CCC(NC(C=Cc2nc(C)sc2)=O)C1)C C12(CNC(C(=O)N(C)Cc3ccsc3)=O)CC(C(F)F)(C1)C2 CC(C)C(C)C(CNC(c1ccc(N)c(O)c1)=O)NC(=O)C(C)CN(C)C c1(Sc2c(NCC)cccc2)c(C)ncnc1C Cc1cc(C)n(C(C)C(=O)NCCCC2CCCN2C(c2nc(C)n(C)n2)=O)n1 c1(COCC)nc(-c2cnn(CC)c2)n(C(C)Cc2ccccc2)n1 c1(C2C(CN3C4CC(NC(C(C)Cc5cnc[nH]5)=O)(C4)C3)C2)ccc(F)cc1Cl C1(CCNC(C2(COCC)CCCCC2)=O)CC(F)(F)C1(F)F N1(C(C(C=C)O)=O)CCC(CNC(=O)CC2CCC(C(F)(F)F)O2)CC1 C(=O)(CS(=O)(=O)CCC(F)(F)F)N1C(COC)(CN(C(=O)CCC(N)=O)CC)CCC1 C(CC(C(=O)NC1(C)CCOC1=O)NC(C1CCN1C(C)(C)C)=O)OC c1(CNCC(O)Cc2ncccn2)nc(Cl)ccc1Br c1(Cc2cc(OC3CCN(C(C4C(C)CN(C)C4)=O)CC3)no2)ccc(C#N)cc1 C1(C(C)(C)NC(C2CCC(C)O2)=O)CCN(C(=O)Cc2cnc[nH]2)CC1 n1(CC(=O)Nc2cnn(C3CC3)c2)ccc2nc(O)nc(O)c12 c1(SCCC(=O)NC2(COC)CN(C(CSSC)=O)C2)ccc(C)c(C)c1 CC1N(C(=O)CC2C3CCCC3N2C(c2ncccc2F)=O)CCCC1(C)C C1(C)(CCC)CN(N2CCOC(c3ccc(Br)cc3)C2)C1 C1(CC(=O)N(CCOCCCNC(COC(C)=O)=O)C)OCCCO1 N1(C(C2=CCC(NC(CSCCOC)=O)C2)=O)CCC2(CC1)CC2CO C1(C2CCCO2)(C(=O)NCCC2CCN(C(CC)=O)C2)CCOCC1 CC(C)(C)C(O)C(=O)NC1CCC1NC(c1c[nH]nc1-c1cccc(Cl)c1F)=O C1(N(C=O)CC)CCN(C(=O)COCCOC)CC1.c1(C(C)(C)C)cc(CSC)no1 C(=O)(C(CC(C)C)NC(N)=O)N1CC(OC)(CNC(=O)CCNC(C)=O)C1 C12(NC(Cc3ccc(SCC)cc3)=O)CCC1CN(C(=O)CCC(F)F)C2 CONC(=O)C(=O)NCC1(C(N)=O)CN(C(=O)CC=Cc2ccccc2)C1 S(=O)(=O)(c1ccc(NC(=O)N(C)C)c(F)c1)N1C(C(C)(C)C)CCC1 c1(C(=O)NC(c2cn(Cc3nscc3Br)nn2)CCC)nc(CC)sc1I C1(C)(CNC(C=NOC)=O)CCCN(C(c2c[nH]c(=N)o2)=O)C1 O=C1Nc2ccccc2CC1SCC(N1CCC(C(F)(F)F)C1)=O C1(C(N2CC(F)(CO)C2)=O)(COC)C=CCN1C(=O)Cc1cccnc1O n1(C(C)C)cnc(C(=O)NCCC(=O)NCCN(C)C2CC2)c1 c1(CC(=O)N(C2CCCN(C(C3CC(C#N)C3)=O)CC2)C)cccc(C#N)c1 c1(OCC(C)C)ccc(OCCC(=O)NC2CN(C(N3CCCC3)=O)C2)cc1 CCCCCC(C)(CC)C(=O)NC1CCN(CCNC(=O)C(C(C)C)OC)C1 c1(C(=O)NCC2CN(C(CCOCC#C)=O)C3C2C3)occ2c1CCC2 C#CC1CN(C(C2CC3CC2CC3NC(=O)CCc2csnn2)=O)CCO1 C(=O)(C(CCC)C(=O)OC)N1CC(C(C(=O)NC(CC#C)CC)OC)C1 N1(C(C(C)(c2ccccc2)N(C)C)=O)CC(C2CN(C(=O)Cc3nc[nH]n3)C2)C1 n1(Cc2nc(C)sc2)nnc(NC(=O)N(C)CCOc2ccccc2)c1C c1(CCC(N2C3CC3C3CC23)=O)cc(F)c(Cl)cc1F C(CC(C)CC)(C(=O)N1CCCN1CCO)NC(CC=CC)=O N1(C(C23C(CN(c4nc(C)c(F)cc4)C2)COC3)=O)CCCc2ccccc2C1 C(=O)(CCCC1CCCO1)NCCN(C(=O)C(C)C1CC1)C(C)C C1(CNC(C2ON=C(C)C2)=O)CN(C(c2ccnn2C(F)F)=O)CC1(C)C C(=O)(CC(C)(C)C(C)(F)F)N1CCN(C(C(C=C=C)C)=O)C(CCOC)C1 C1(S(C)(=O)=O)(C(N(CC(C)O)CCNC(=O)C2=CCSC2)=O)CCCC1 C(=O)(C1=CCS(=O)(=O)C1)N1CCN(C(COC)=O)C(C(C)C)C1 O=C(C1CCc2c(Cl)cccc21)NCCC1CN(C(=O)C=Cc2ccsc2)C1 C12(C(=O)O)C(NS(=O)(=O)CC3C4CCCCC34)CCC(CC1)C2 C(=O)(C(S(C)(=O)=O)C1CC1)NCCN(C(c1[nH]c(C)cc1C)=O)CC C(=O)(CC1OCCc2sccc21)NC1C2(CCN(C(c3c(CC)ncs3)=O)CC2)C1 C(=O)(CCC(C)(C)N(C)C)N(CC(CC)NC(=O)COc1ccccc1OC)C c1(C(N2CCC(F)(CF)C2)C(=O)NCCOCC)csc([N+](=O)[O-])c1 N1(C(=O)NCc2csc(C(F)(F)F)c2)CCC(C2CCCNC2)CC1 C(=O)(C1SCc2cccnc21)NC1CCN(C(CSCCC(C)C)=O)CC1O C1(CC)CN(C(c2ncncc2Cl)=O)CCC1CNC(=O)C(C)C(C)(C)C C(CC(O)CC(=O)NCCCN(C(=O)CCc1cncn1C)C1CC1)SC c1(CNC(=O)NC(CCN(C)CCC2(C3CCCO3)CCC2)=O)ccncc1 c1(C(C)(C)C)ncc(CCNC(=O)C(=O)NCCC(Cl)(Cl)Cl)cn1 C1(C(=O)NC2(CCC(=O)NCC(C3CC3)OC)CCC2)(CO)CCCCO1 C=C(C)CC(Cc1ccccc1)NCC12CC1CCN2C(C)=O c1(CC)noc(C(=O)NCC(C)CN(CCCSC)C(c2ccccn2)C)n1 CCCCCCC(C)C(=O)N(CC(C)O)C1(CNC(=O)COc2cc(C)on2)CC1 C(=O)(C1=C(C)CCCC1(C)C)N1CC2CN(C(C(CCC)OCC)=O)C2CC1 N1(C(c2ccc(Cl)o2)=O)CC2CCN(C(=O)CCOc3ccc(Br)cc3)C2C1 c1(OC)cc(C(=O)NC2CCCC2CNC(=O)CCCC2CCCO2)n(C)n1 c1(CCC(=O)NCCN(CCC)C(C2(Cl)CC2(F)F)=O)ccccc1 c1(CC)ccc(OC2CCCC(NC(=O)Nn3cnnn3)C2)cc1 c1(C(C(=O)NC(CC)C)N(CC(=O)NC)CC)cc(C(F)(F)F)ccc1F c1(C(N2C3C(NC(C(C)C)=O)C(C3)C2)=O)oc2ccccc2c1-c1cccs1 N1(C(c2cc(CC)c(C)s2)=O)C2CCC1C(C)C(NC(=O)CCc1nncs1)C2 CC1=C(C(=O)N(C2CCC(NC(=O)CCCOc3ccc(F)cc3)C2)C)CCC1 c1(OC)cc(C(=O)NC2(C(F)(F)F)CC(F)C2)cc(OC)c1Cl CC1(C)CCC(CO)N(C(c2c[nH]nc2CNC(=O)CCCC2CCCO2)=O)C1 c1(C(=O)NC(C2N(C(CSCc3onc(CC)n3)=O)CCC2)C)ccc(=O)oc1 Cc1cccc2c(C(=O)NC(C34CC(CO3)C4)C)cnn12 C1(C(N(CCCNC(c2onc(CC)n2)=O)C(C)C)=O)CCc2nc[nH]c2C1 CC1(C(N2CC(NC(c3cc(O)cc(O)n3)=O)C(O)C2)=O)CCC(=O)NC1 C1(CC)(NC(c2ccc(NS(C)(=O)=O)o2)=O)CCCN(C(=O)C2=CC(C)(C)C2)C1 N1(C(CCCCCC)=O)C(CNC(c2ccc3nn[nH]c3n2)=O)CC2COCC12 N(C1CCc2cc(CNC(c3nn(C)nc3C)=O)ccc21)C(C=C(CCC)C)=O N1(C(c2ncc(C)cn2)=O)CCCC(F)(CNC(c2cnn(CC(F)F)c2)=O)C1 N1(C(C(C)NC(CC)=O)=O)CCC(CNC(=O)C(F)(F)C(C)O)(COC)CC1 Cc1cc(C(=O)NCCCCCCNC(c2cnc(Br)s2)=O)c(C)o1 C1(CC(=O)N(C(=O)CC(C)Sc2csc(C)n2)CC)CCN(CC(C)C)CC1 C1(NC(C(COC)OC)=O)CCCCN(C(c2ccncc2C)=O)C1 N1(C(C(CC(C)C)=O)=O)CC2CCC(C1)N2C(=O)CCc1c[nH]c2ccccc12 Cc1cc(CC(=O)NCC2OCCC2C(N2CC(N3CCOC3=O)C2)=O)no1 c1(C(N(C)Cc2ccc(OCc3ccccc3)cc2)=O)cnn2c1NCCC2 N1(C(CCC(=O)NCCC)=O)C2CCC1C(NC(=O)C(C)(C)C1CC1)C2 c1(CC)cccc(C(N2CCC(C(=O)N(CC(N3CC=CC3)=O)C)CC2)=O)n1 C=CC(CC)CC(=O)NC1(C2CCCN2C(c2nn(C)c(Cl)c2Cl)=O)CC1 C12(C(N3CCCC(C(C)NC(c4cc(C(C)C)no4)=O)C3)=O)CCOC(C)(C1)C2 c1(C(=O)NCC2CN(C(C(C)NC(C)=O)=O)CC2O)ccc(F)c(C(F)(F)F)c1 C(CC(O)CC(=O)NC12CC1CN(C(=O)C=CC1CCCCC1)C2)SC CCC(F)(F)CC(=O)N1CCC(CNC(=O)CCOCC2CCC2)(CF)C1 N1(C(c2cnn(CC3CC3)c2)=O)CC2CN(C(c3ccn(C4CC4)n3)=O)CC2C1 N1(C(C2N(C(C3N(C)C(=O)CC3)=O)CC(F)(F)C2)=O)CCC2(CCOC2)C1 N#CC1CC(c2ccc(Br)cc2)(N2CCCC2CC2CCC2)C1.c1ccc(F)cc1 c1(CC(=O)NCC#CCNC(C23CCCC2C3(F)F)=O)ccc(Cl)cc1F C(=O)(C1=COCC1)N.c1(C(C)(C)C)ccc(C(F)(F)F)nc1.C12(O)CC(C1)N(C)C2=O C1(O)(CCNC(COC(CNC(C(C(C)C)N(C)C)=O)(C)C)=O)CCCCCC1 C1(C(N(C)C)=O)CCC2(CCN(NC(C3CCCOC3)=O)CC2)O1 N1(C(C(Cc2cc[nH]n2)NC(c2ccn(C)n2)=O)=O)Cc2ncsc2C1 C(C)(C(CC(=O)N(C1CC(O)C1(C)C)C)NC(=O)C(C)(C)O)OC c1(-c2nc(CCCCC)nn2C2CCCC(SC)C2)cc2c(s1)CCOC2=NO N1(C(C(C2(O)CN(C(Cn3cnc(=N)[nH]3)=O)C2)F)=O)CC(=O)N2CCCC2C1 c1(CC)cnc(C(=O)NC2CCCC2NC(=O)CSS(C)(=O)=O)cn1 c1(NC(=O)NCC(c2ccc(Br)cc2)(F)F)ccc(I)c(Br)n1 N1(C(C(C)(C)OCc2ccc(F)cc2)=O)CCN(C(C2CCC(F)(F)C2)=O)CC1 C(=O)(C(C)(C#N)CC)N1CCCC(CCCCNC(c2c(CC)oc(C)c2)=O)C1 c1(COC(C)C)ccc(-c2cccc(CN(C3(CN)CC(F)(F)C3)C)c2)cc1 Cc1ncc([N+](=O)[O-])n1CC(=O)NCC(C)NC(=O)C(C)C(=O)OC(C)(C)C C1(CNC(C(Cc2ccc(OCC)cc2)C)=O)CN(C(=O)CO)CCN1C C1(C)(NC(COC)=O)CCCN(C(c2n[nH]c(C)c2Br)=O)C1 C1(CCC)CN(C(=O)CN2CCNC(=O)C2)CCN1C(=O)C(CO)OCC(C)C C1(NC(C=CCC(C)(C)NC(C2CCC(C)(F)CC2)=O)=O)CCCCC1N=[N+]=[N-] CC1(C)CC(O)CCN(C(=O)CC2(c3cn(C(C)(C)C(=O)O)nn3)CCCCC2)C1 N1(C(c2ccc(-c3nc(C)sc3)s2)=O)CCC2CN(C(c3oncc3C)=O)CC12 C1(N=[N+]=[N-])(NCCc2cccc(C(=O)OC)c2)CCNCC1 Cc1nn(C)cc1C(=O)N(C1CN(C(=O)C(C2CCCO2)OC(C)C)C1)C N1(C(CCC)=O)CCCC(C(N2CCN(C(=O)CCn3cncn3)CC2)=O)C1 C1(OC)CCC2(CCN(C(=O)CC(C(F)F)NC(=O)OC(C)(C)C)C2)C1 c1(C(N(CC(=O)NCCC2CCC3CC23)C(C)C)=O)ccc2c(c1)CCC2 c1(C(=O)NCC(C(=O)NC2C(OC)C(O)C2)C(C)C)cc(C)cc(C#N)c1 C1(C(=O)NCC(CNC(C(OCC)OCC)=O)O)SCCCS1 N1(C(CNC(=O)Cn2cccn2)=O)CCN(C(C2CCC(=O)O2)=O)CC1 c1(NC2C=CC(C(=O)NCCCCN(C)C)C2)cc([N+](=O)[O-])ccc1Cl Cc1ccccc1OCC1N(C(=O)OCC(N(C)C)Nc2c(C)cnn2C)CCC1 C=CCN=C(NCCCC1CCCO1)NCc1cc(C)c(O)nn1 N1(C(CN(CCC#C)C)=O)CCC(NC(=O)CCCN2CCCC2)CC1C C1(NC(c2cc(C)ncc2C)=O)CN(C(c2ccoc2C)=O)CC1C1CC1 N1(C(CN(C2CC2)CC)=O)CCCC(C)(C)C1C(=O)N(CCC(N)=O)C C1(CC)OCCCC1N=c1[nH]c(=NC2CCSc3ccccc32)[nH]c2c1CCC2 C1(C2CC2)(NC(C(COC)C)=O)CCN(C(c2cc(-c3ccccc3F)no2)=O)C1 CC1(C)C(C(=O)NCC(O)CC2CCCC2)CCN1C(=O)C1=COCC1 c1(C(N2CCC(CNC(c3ncc(Br)cc3Cl)=O)C2)=O)nccc(Cl)c1Cl CS(=O)(=O)CCCCC(=O)NC1CC2CC(C1)N(c1ncns1)C2 C(C(C)(C)C(=O)N1CCC(OCC(N)=O)C1)N(C)C(C1CCCC(O)C1)=O N#Cc1cc(F)cc(NC(N2CCCC(CCCO)C2)=O)c1Cl Cc1cc(N2CCCC(N3CCOCC3)C2)n(C)n1 CC1(C)CN(C(=O)C2=CCCSC2)CC(CNC(c2ccns2)=O)O1 C1(C(=O)NC(CCCCNC(c2cc(OC)no2)=O)C)CCc2nnnn2C1 C1(NC(C2N(C(c3cc(C)sc3C)=O)CC(O)C2)=O)CCC(=O)CC1(C)C CC1C(NC(=O)CCc2cccs2)CCCN1C(c1cc([N+](=O)[O-])n[nH]1)=O N1(C(CC(=O)NCC#C)=O)CCC(C(=O)N(C)CCN(C)CCC)CC1CC C1(CC)CC(O)CCN1C(=O)CN1CCN(C(C2CCCC(=O)N2)=O)CC1 C1(CN(C(C2(CC=C)CN(C(C3CCCC3OC)=O)C2)=O)C)CCCN(C)C1 CC1CC(NC(c2ccccc2)=O)CCN1C(c1ccccc1C(C)O)=O C#Cc1cccc(C(N2CCC(C)(NC(=O)CC3CCC(C)(C)CC3)C2)=O)c1 c1(C(N2CC(F)(CNC(C(C)SC)=O)C2)=O)cc(F)cc(N)c1F n1(CC)nc(C(C)C)cc1C(=O)NC1CC1CNC(C12CCC1CC2)=O c1(C(N2CCCC(C(=O)NCCOC3CCCOC3)C2)=O)ccc(F)c(O)c1 C12(NC(Cc3nc(C)sc3)=O)CCC(CC1C(=O)OCc1ccc(C#N)cn1)C2 Cc1ccc(SC2(CNC(C3CCN(C(C4C=CCCC4)=O)CC3)=O)CC2)cc1 c1(C(N2CCN(C(COC(CC)(C)C)=O)CC2)=O)ccc(F)c(C2CCC2)n1 c1(C(N2CCCC(N(C(=O)C(C)C#N)CC)C2)=O)cccc2c1OCCCO2 Cc1c(CN2CCC(c3ccccc3)C2)sc2ccc(F)cc12 c1(C(=O)NCC2CC(NC(C(F)OC)=O)C2)cnn(C(C)(C)C)c1N Cc1cnccc1C(C)C(=O)NC1(CCCNC(=O)C=Cc2sccc2C)CC1 c1(C(N2C(CN(C(CCC(C)(C)OC)=O)C)CCCC2)=O)ccc([N+](=O)[O-])nc1 N1(C(C(C=C)(C)CC)=O)CCc2ccccc2C(N(C)C(=O)CCC2CCC2)C1 NC(=O)CCN=c1[nH]c(=NCc2n[nH]cc2C2CC2)[nH]c2c1CCCCCC2 C1(C(=O)NC2CC(CNC(C(C)NS(CC)(=O)=O)=O)C2)CC2(CC2)CO1 CCCCCCC(=O)N1CCN(C(c2cc(C(F)(F)C(F)(F)F)on2)=O)CC1 C(=O)(CCCC(F)F)N(C)Cc1c(CNC(C(COC)OC)=O)cccc1.SC Cc1nn(C)c(N)c1C(=O)N(C)CC1(NC(C2CCCN2CC(F)(F)F)=O)CC1 Cc1cc(C(=O)NC2CC(CCNC(c3ccc(C)c(Cl)c3)=O)C2)c(N)cc1F N1(C(N=C2c3ccc(OC)cc3CC2)=O)CC(C)(C)C(CN(C)C)Cn2ncnc21 C1(C(=O)NCC2CCCN(C(c3c(OC)noc3C)=O)C2)CCCNS1(=O)=O Cc1ccc2c(c1)C=C(C(=O)NCCc1cc(Br)ccc1C)CO2 CCCC(C)CC(=O)N1CCC(NC(c2cccc(-n3cnnn3)c2C)=O)CC1 N1(C(c2nc(Cl)cc(N)c2Cl)=O)CCCC12CCN(C(=O)CC1CCCS1(=O)=O)C2 C(CN=c1[nH]c2cc(F)cc(F)c2o1)C1CCN(C(c2cc3c([nH]2)CCCC3)=O)C1 C1(C(=O)NCCOCCN(C(=O)C=Cc2cc[nH]n2)C)CCCC1C(F)F CC1(C)CN(C(c2cocc2C(N)=O)=O)CC1NC(c1csc(C2CC2)n1)=O c1(CN2C3CN(c4c(F)cnc(C)n4)C(C3)C2)ccc2sc3ccccc3c2c1 C(C(=O)N1CCCCC1CNC(c1csnc1C)=O)(C(C)C)NC(COC)=O c1(OC)cc(C=CC(=O)NCC2CC2CNC(c2ocnc2C)=O)sn1 CCC(O)C(C)(C)C(=O)N1CC(NC(c2cc(C)ccn2)=O)C(F)C1 C1(C(=O)NC(C2(O)CN(C(=O)CCn3cc(Cl)cn3)C2)C)CCC2C(C1)C2(F)F c1(CC(=O)NCC2CC(NC(C(C(=O)OCC)(C)C)=O)C2)cccc2ccoc12 C=C(Cl)CC(C(=O)NCc1cccc(COC)n1)NC(C1OCCC1(C)C)=O c1(NCC2(CNC(c3cnc[nH]3)=O)CC2)nc(Cl)[nH]c2nccc1-2 c1(CNC2(c3nnnn3C)CCN(CCOC)CC2)c[nH]c(=O)c2ccnn12 c1(C(=O)NCC(CC)NC(C2CCCC2(C)C)=O)cnc2ccnn2c1O C=CC(C)(CC)C(=O)NCC(C(=O)NCCc1cnn(CC)c1)N(C)C N1(C(C(CC)NC(C)=O)=O)CC(F)CC1CC(N1CCC(CC(=O)NC)C1)=O CC(C)C(C)CC(=O)N(C1CCCN(C(C2CCC3(CC3)C2)=O)C1)C c1(CC(=O)NC2(CCNC(C(C)SCC)=O)CCC2)ccccc1C(N)=O C1(NC(C2(OC)CCOC2)=O)(CO)CCCN(C(=O)COC2(C)CCOCC2)C1 C1(NC(CCCCCC)=O)CC2CCC1CN(C(=O)CN1CCCNC1=O)C2 C(=O)(CC(C)CC(C)C)NCC1CCCC(NC(CNC(=O)OCC=C)=O)C1 CCC(C)C(C(=O)N(CCNC(c1cc(C(F)F)n(C)n1)=O)CC)NC(N)=O CC1CCC(C(=O)Nc2cccc(OC(C)(C)C)n2)CN1C(=O)C1=CC(C)(C)C1 c1(CCC(=O)NCC(C(C)C)NC(c2ncn(C)n2)=O)cncnc1O c1(C(N(C(CNC(c2c(CCC)[nH]cc2)=O)CC)C)=O)ccccc1C(C)(F)F n1(C(C=C)C)ncn(CC(=O)OC(C)(C)C)c1=S C(=O)(CC(F)(F)C(C)(F)F)N1CCN(C(c2ccc(C)cn2)C)CC1 C1(NC(c2cc(C)[nH]c2C)=O)CC(NC(C2CC(=O)NC(=O)C2)=O)C12CCC2 N1(C(CCc2nc(C)c(C)o2)=O)CC2COCCC2(NC(=O)CC(C)C)C1 N1(CC)CC2CCC1C1CN(C(=O)CC3CCN(CCNC(N)=O)CC3)CC21 Cc1cc(C(=O)NC(C)CC(N2CC3C(CN(C)C)C3C2)=O)c(C)o1 c1(CS(C)=O)cccc(C(=O)NCC2CC2NC(C2(C)C=CCC2)=O)c1 C#Cc1ccc(C(N2CCOCC(NC(=O)C=CS(C)=O)C2)=O)cc1 c1(C(C2(C3CN(C(C(CC(C)C)F)=O)C3)CC2)=O)ccc2[nH]c(=N)oc2c1 C(=O)(C1=C(C)OCCS1)NC1C2(C(=O)NC(CC=C)CC)C3CC1CC23 c1(C(N(CC(CNC(CN(C(=O)OC)C)=O)O)C)=O)cc2c(F)cc(C)cc2[nH]1 C#Cc1cccc(C(=O)NCC2C(C)CCN2C(c2nn(C)cc2Cl)=O)c1Cl N1(C(CCC2C(C)=NOC2=O)=O)CCC2CN(C(=O)CCOCC(F)F)CC2CC1 c1(C(=O)OC)cc(C(=O)NCC2CCC(NC(=O)CCC3(C)N=N3)C2)ccc1F C(=O)(CCC(=O)NC1CC1)N(CCC(=O)NC1(CO)CC1C)CC=C C1(NC(c2ccc(OC)s2)=O)CC2CC(C1)CN(C(=O)Cc1ccn(C)n1)C2 C(=O)(C(C(C)C)n1cnnc1)N1C(C2(NC(c3cc(C)on3)=O)CC2)CCC1 c1(C(=O)NC(=O)CC2CCN(C(C3(CC)CCCCC3)=O)C2)cc2cccnn2c1 CCCC(C(=O)NC1CN(C(c2ncccc2SCC)=O)CC1F)S(N)(=O)=O Cc1cc(C(=O)NC2CCN(C(C3CNC(=O)C3)=O)C2)cnc1Cl CC1CN(C)CC1NC(=O)C=CC(C)(C)N.C(=O)(CCC1CCCC1)C(=O)C C1(CCOC)(NC(C(C)=CC)=O)CCN(C(c2ccnc(C3CCC3)c2)=O)C1 c1(C(N=c2ccc(CC)n[nH]2)=O)cccc(S(=O)(=O)N2CCCC3(CNC3)C2)c1 N1(C(c2c(C)scc2)=O)CCOCC(C)(CNC(=O)CS(N)(=O)=O)C1 C(=O)(C(C)(C)C1=CCN(C(C2(C#N)CCC2)=O)C1)N(CC(C(=O)NC)C)C c1(C(=O)NC(C)CCCCNC(=O)Cc2cccn2C)cc2c(nn1)CCOC2 N1(C(=O)NCC=CC(C)(C)C)CCC2(CCCC2Nc2ncnc(Cl)c2F)C1 C1(C(N2CCOC(CNC(=O)CNc3nccs3)C2)=O)(OC)CCCC(C)C1 N1(C(CC2N(C(c3ccn(CCC)n3)=O)C3C2CCC3)=O)CC(C)(C)OCC1C CCC(C)CCCC(=O)N1CCC(C(=O)Nc2csc(Cl)c2)O1 c1(C(C(=O)NC2CCOC2)N(C2(CCC)CCOC2)C)cc(S(N)(=O)=O)cs1 C(=O)(C1=CCc2ccccc21)N1CCCC(C2(NC(c3c(C)nco3)=O)CC2)C1 CC(C)C(F)(CNC(C1CCOC1CO)=O)C(=O)N1CCCC(O)(C(N)=O)C1 Cc1ccc(Cl)cc1-n1cc(CCC2CN(C(C3(C)CC3(F)F)=O)C2)nn1 C1(CC)CN(C(=O)CCC(C)NC(c2cc(F)cc(F)c2)=O)CCCO1 c1(C(N(C2CCC(NC(c3cnc(O)s3)=O)C2)C)=O)cccc2nonc12 C1(NC(C2CC(C(=O)OC)C2)=O)CCN(C(c2cccc3[nH]ncc23)=O)C(C)C1 N1(C(CC2CC(=C)C2)=O)CCN(C(c2nocc2C(C)C)=O)CC1CC Cc1cc(C(=O)NCC2CCN(C(=O)CCc3cn(C)cn3)C2)sc1Br C12(NC(CC=CC=C)=O)CCCC1CN(C(=O)Cn1cncn1)C2 C1(NCCC(NC(=NC)NCCCOC)(C)C)CCCN(C)C1 O=C(CS(=O)(=O)N1CCCCC1)N1CC(O)(C2CCCN2C(=O)CO)C1 c1(CC(N2CCC(CNC(c3c(OC)cncn3)=O)CC2)=O)cc(C)ccc1C S(=O)(=O)(c1ccc(NC(N2CCCCC2)=O)c(F)c1)N1C(C(C)C)C(O)CCC1 c1(C(=O)NC(CC)(C)CNC(C2NC(=O)OC2C)=O)ccc(N)c(Cl)c1 N1(C(CC=CCC)=O)CC=C(CNC(c2ccc(F)cc2C2CC2)=O)CC1 c1(NCC(OCC)OC)ncc(C)cc1S(=O)(=O)N1CCCC(CC)C1 c1(CN(C)C(c2ccc(NCc3cccc(F)n3)nc2)=O)cccc(Br)c1O Cc1cc(NC(C2CCCC(n3cc(C4CCS(=O)(=O)CC4)nn3)C2)=O)c(C)cn1 C1(C(=O)NC2(c3nc(C)[nH]n3)CC2)CC2CC2N1C(=O)CC1CCCC(=O)C1 C(N=C(NCc1ccnn1C)N1CC=C(F)C1)c1c(CC)n(C)nc1 CC1CN(C(C2(c3ccn(C)n3)CC2)=O)CCN1C(C1CCNC1=O)=O N1(C(c2ccc(CC)c(N)c2)=O)CC(NC(=O)C(CC)SC)C(C2CC2)C1 CC1(C)CCCCC1C(=O)NCCC1(NC(C2CC(C#N)C2)=O)CCOCC1 Cc1cc(=NCc2sc3ccccc3c2C)[nH]c(N2CC3CCCC3C2)n1 c1(C(=O)NCC2(CNC(=O)C(O)C3CCCC3)CCC2)ccc2c(c1)COC2 C=CCC(CC)C(=O)NCC12CC(CN1C(=O)C(C)CCCc1ccccc1)C2 c1(C(=O)NC(CC)(C)CNC(C2CCN(C)CC2)=O)ccc(F)c(OC)c1 C(N=c1[nH]cc(Br)c2nnnn12)c1[nH]c(=N)sc1 c1(C(=O)NCC(C(=O)NCCC(C)O)C)cccc(CO)n1 C(=O)(C1=C(C)OCCS1)N(CCCN(C(CCC1C(C)=NOC1=O)=O)C)C CC1CCC(NC(=O)C(=O)NC2CC2)CN1C(c1cncc(Cl)n1)=O c1(C(=O)NCC2(CNC(C3(C)CCNC3=O)=O)CC2)cc2c(nn1)CCOC2 C1(NC(CCC(C)C)=O)CCN(C(c2cnn(CC(F)(F)F)n2)=O)C(C)C1 c1(C(=O)NC2C(c3cccc(Cl)c3)(C)C2)cc(Br)cnc1Cl C1(NC(CCC(=O)NC)=O)CCCC(C(=O)NCCCCc2ncc[nH]2)CC1 N1(C(C2CCOCC2)=O)CC2CN(C(C3CC=CCC3)=O)CCC12 C1(NC(c2cccc(NS(CC)(=O)=O)c2)=O)CC(O)CN(C(=O)CN2CC(C)C2)C1 C1(C(N2CC(OC(F)F)C2)=O)CC(=O)NC1=O.CC1(C)C2C1CNC2=O S(=O)(=O)(c1ccc(O)c(Br)c1)CNC(COCC)CO c1(C(=O)NC(CN(C(=O)Cn2ccc(C)n2)CC)C)nc(COC)sc1N N1(C(CN(C(CC(C(C)=O)(C)C)=O)C)=O)CCC(F)(F)C(F)C1 C(N=c1cc(C)c(C#N)c[nH]1)C1CCCN(C(Cc2cc(OC)no2)=O)C1 C1(C(N2CCN(C(=O)Cn3cnc4ccccc34)CC2)=O)CC1C1CCCCC1 C1(CNC(c2c(Cl)cnc(C)n2)=O)CN(C(=O)C(F)CC2CC2)C2CCCC2O1 c1(C(N2C3CCC(CCNC(CCC4C(C)C4)=O)(C3)C2)=O)ccn2nccc2n1 c1(CCC)nc(C(=O)NCCCNC(c2cc(Cc3ccco3)c[nH]2)=O)cs1 C(=O)(C1=NN2CCCN=C2N1)NC1C2CC3CN(C(COCCC#C)=O)C1C3C2 CN1CC(C)(C)CC1C(=O)NC(C(=O)NCC1(Cl)CC1(F)F)C1CCCC1 N1(C(c2cc(C(C)=O)n(C)c2)=O)CCC(C2CC2)(CNC(C2CC3CC3C2)=O)C1 c1(N(C)C)cnc(C(=O)NCC2CCN2C(=O)CC2CCNC2=O)cn1 N1(C(C2C(C)(C)C2)=O)CCC(CCC(=O)NCC=CC(F)(F)F)C1 C(=O)(CC(C)Cc1cccc(F)c1)NCCN(C(c1c(C)noc1)=O)C(C)C C12(CNC(C(C(C)C)N(C)C)=O)CCC1CN(C(=O)Cn1cnnc1)C2 c1(C(N(C)CC2CCN(C(c3nonc3N)=O)C2)=O)cc(S(C)(=O)=O)cs1 C(=O)(CCCCC(=O)N1CCC(C(C)NC(c2csc3nnsc23)=O)C1)NC N1(C(C2(C=C)CCOCC2)=O)CCc2c(CNC(=O)C(O)C(=C)C)cccc2C1 CCC(C)(C(=O)N1CCCC1CCNC(=O)CCC1CCCN1C)C(N)=O C1(CCC(=O)NCC(C(=O)NC)C)CCN(C(c2cc(OC)no2)=O)C1 N1(C(COC(C)=O)=O)CCCC(C)(C)C1C(N1CCOCC1)=O N1(C(C2CC(C)(C(C)(C)C)C2)=O)CCCC(NC(=O)CC2(c3ccon3)CC2)C1 Cn1nccc(C(N2CCC(CF)(NC(=O)C(c3ccccn3)O)C2)=O)c1=O C1(C(F)(F)F)(C(=O)NC(CNC(C(C)NC(C)=O)=O)(C)C)CC=CCO1 CC(C)C(C(=O)NCC(C)(CO)NC(c1cc(CO)[nH]n1)=O)c1cccnc1 C(=O)(C(COC)(CC)CC)N(CCCNC(C1(COC)CCCOC1)=O)C c1(C(N2CCC(NC(C3CCC(C)CC3)=O)(CF)C2)=O)cn(C)c2ncccc12 c1(CC(=O)NCC2CC2CNC(c2ccncc2F)=O)ccc(F)cc1F Cc1cc(C)c(C(=O)NCC2CC(NC(CO)CC(C)(C)C)C2)c(=O)o1 N1(C(CCCC(OC)OC)C(=O)NCCSC)CCOCC(C)(C)C1 c1(C(=O)NCCC(C)NC(C(C)OC(F)(F)F)=O)ccc(C(=O)NC2CC2)cc1 c1(COC)ncc(C(=O)NCC2(O)CCCN(C(c3ccsc3C)=O)C2)c(=N)[nH]1 c1(CCSCCn2cc(C(c3n(CC)nnn3)N)nn2)c(C)cc(Br)cc1C c1(Nc2ccc(OCCCC)c(SC)c2)ccc(OC)c([N+](=O)[O-])c1 Cc1cccc(O)c1C(=O)N(CCCOCCNC(C1CC2CC2C1)=O)C Cc1cc(C#N)cnc1C(=O)NC1CCN(C(C2(F)CCCOC2)=O)C1 N1(C(CC2CCCN(C)C2)=O)CCC(O)C(NC(=O)C(C)(C)c2ccccc2)C1 C(=O)(C(CCC(C)C)NC(c1ccn(C(F)F)n1)=O)N1CCCCC(CC)C1 c1(C(=O)OC)ccc(CNC(=O)Nc2nc(Cc3ccccc3)[nH]c(=N)n2)nc1 C(c1ccccc1Br)=CC(=O)NCCCN(C)C(C1(C)C=CCC1)=O C1(C(=O)NCC2CC2)(COC)C=CCN1C(=O)CC1CCC(=O)C1C N12CCN(C(C)CC1C)C(=O)COc1ccc(cc1F)C2=O.C(CC(C)C)OC C1(O)(CNC(C(=Cc2ccncc2)C)=O)CCCN(C(c2nc(C)oc2C)=O)C1 c1(OCC)ccc(F)cc1C(=O)NC1(CNC(=O)C(F)=C2CCCC2)CCOC1 C1(C(=O)OC)CN(S(=O)(=O)N2CCCCC2CC2CC2)CC1C1CCC1 c1(C(=O)NC(CNC(c2cc(C)on2)=O)(C)CO)ccc(C(F)(F)F)cn1 c1(C(=O)NCCCN(C(C2CCN(C(C)=O)C2)=O)C)ccc(C)c(N)c1 C12(CNC(CCc3nc(C)sc3)=O)CC1CN(C(c1cnoc1CC(C)C)=O)C2 N1(C(N2CC(OCCNC(C3N(C(C)=O)CCC3)=O)C2)=O)CC2CCC1C2 c1(CC(=O)N(CCNC(C(C)=C(C)C)=O)C(C)C)csc(Cl)n1 CC1CC2CN(C(=O)CCCC(=O)NCC(F)F)CC2N1C(C1CNC(=O)C1)=O C12CCOCC1NC(=O)C2.CNS(=O)(=O)NCC(=O)NCCN(C1CC1)C(C)C C1(c2n(CC)nnn2)(NCC2(CF)CC(F)(F)C2)CCCC(C(F)(F)F)C1 c1(CC(=O)NC(C(=O)N(CC)CC2CC2)SC)ccnn1C c1(OC)ccc(C(=O)NC2CC(CNC(c3csc(C)c3OC)=O)C2)c(N)c1F CCCS(=O)(=O)C(C)C(=O)NCCCN(C(=O)COc1cccc(C)c1)C Cc1ccc(CN2CCC(CNC(c3ocnc3C3CC3)=O)C2)o1 C#Cc1ccc(C(=O)NCCN(C(=O)CCC(C)(C)C)C2CC2)c(C)c1 C=CC1CN(C(=O)CCCN(C)C2CC2)CC1NC(C1CCOC1C)=O C1(CNC(=O)COC(F)F)CCCCN1CC1(c2ccccc2Br)CCCC1 c1(OCC)ncc(NC(C2CCOCC2)=O)s1.c12nc(cs1)CN2 CP(C)(=O)C1(C(=O)NCC2(NC(=O)C(F)C3CCC3)CC2)CC1 C(=O)(C(F)C(F)(F)F)N1CC(C(N)=O)(CNC(C(C)(C)OC(C)C)=O)C1 C1(NC(CCNC(=O)C=CCl)=O)CCCCN(C(=O)C=Cc2ccccn2)CC1 c1(CC)[nH]nc(C(N2C3CCC2CC(NC(=O)CCCCC2CC2)C3)=O)c1[N+](=O)[O-] N1(C(c2cnn(C(C)C)c2F)C(=O)NCC(=C)C)CCC2(CC1)CNC(=O)N2 c1(NC(c2c(F)ccc(Br)c2C)c2n(CC)nnn2)ccc(C#N)cc1COC C1(CCc2c(C(=O)NC3CN(C)C3)snn2)COc2c(F)cc(F)cc2C1 C#CC1(NC(=O)NCc2cccc(SC)c2C)CCCCC1 c1(C(C(=O)OC)F)ccc(C(=O)OCc2nc(C(F)(F)F)n[nH]2)cc1 Cc1ccc(C(N2CCCC(CNC(C3(C)CC(C)C3)=O)C2)=O)c2c1CCCN2 CCCC(C)(O)C(=O)NCC1(OC)CCN(C(=O)C(C(C)C)OCC)C1 C12(Nc3c(C(=O)OC)sc(Br)c3)CCCCC1OCC2 Cc1sccc1CNC(c1nnnn1CCCSC1CC1)C(C)C1CCC1 c1(C(N2CCCN(C(CC(C)(C)OC)=O)CC2CO)=O)cnc2c(c1)CCOC2 C1(C(=O)NC2C(CC(=O)NOCC3CCCC3)CCC2)CC2CC1CC2O Cc1ccc(F)c(-c2cn(C3COCC3NC(=O)CCCN(C)C)nn2)c1Br C(F)(F)(C(=O)NNc1ccc(F)c(NC(=O)C2CC2)c1)C12CCC(C)(CC1)CO2 Cc1c(O)ccnc1-c1ccc(N2CCN(c3nnc(C4CC4)s3)CC2)cn1 C1(C(=O)NC(C2CN(C(=O)C(C)(Cl)Cl)CCO2)C)CCCCCCC1 c1(C(=O)NCCCOC2CCN(C(C(C)=C3CCC3)=O)C2)ncc(F)cn1 C(N=c1[nH]c(N2CCCC3(CCC3)C2)nc2c1COCC2)C1CCCC(F)C1CO C#CC1(O)CCCN(C(=O)C2=CCN(C(C3(Cl)CC3)=O)C2)C1 c1(N(C(C)CCNC(=O)CSCCN(C)C)C)ncnc2sccc12 C1(CNC(c2n(CC(=C)C)nnn2)c2cnn(C(C)C)c2)(OC)CCOCC1 N1(C(c2cc(CC)ccc2OC)C(=O)NCCCC)CC(C2CC2)CC1C1CC1 c1(C(N2CCC(O)(CNC(c3c(OC)cncc3)=O)C2)=O)ccc(Cl)c(F)c1O C1(NC(c2cn(CC(CC)O)nn2)=O)CCCN(C(=O)CCSCC(N)=O)C1 N1(C(C2N(C(CC3C(=O)NCC3)=O)CCC=C2)=O)CCC(F)CC1 Cc1ccc(N2CC(CN=C(NC(C)C)NC3CCC3C3CC3)CC2=O)cc1 C(=O)(C(O)C(C)(C)C)NCC(CC(=O)NCC1(C)CC2(CCC2)C1)OC c1(COC)cccc(CC(N2CCCC(NC(C3CC=CCO3)=O)C2)=O)c1 c1(C(c2ccccc2)NC(=O)Nc2ccc(N(C)C)cn2)ccc2c(c1)CCC2 C(=O)(CCCC(=O)NOC(C)(C)C)NC1CC2CN(C(C#CC(C)(C)O)=O)CC21 C1(O)(CNC(CCC(C)OC)=O)CCCN(C(=O)CC(=O)OCCC(C)C)C1 c1(C(=O)NCCCN(C(=O)CCC2(C#N)CCC2)CCC)cnc2[nH]cncc1-2 C1(C(N2CCN(CC=C)CC2)=O)CCCN(C(C2(OC)CCCCC2)=O)CC1 C(=O)(C(O)CCC(F)(F)F)N1CC=C(CNC(CCc2cc(C)no2)=O)CC1 c1(C(=O)NC2CN(C(C=CC)=O)CC2C)cc(C)ccc1NC1CC1COC N1(C(CC(C)OC)=O)CCC(=CCNC(=O)C(C)(C)Sc2ccccc2)CC1 CC(C)CN=C(NCS(C)(=O)=O)N(C)C(C1(OC)CCOC1)C1CCCO1 C1(CC(=O)NCCN(C(=O)CSc2n[nH]c(O)n2)C2CC2)CC2CC2C1 C1(=O)C(F)(F)CCCCN1.c1(-n2cc(C3(C)CCCC3)nn2)ccc(F)cc1Br C1(CC(N2CCC(CNC(C3CSCCS3)=O)C2)=O)(COC)CCOCC1 N1(C(C(C)NC(COC)=O)=O)CCN(C(c2ccnc(OC)c2Cl)=O)CCC1C C1(C)(CNC(Cc2cc(C)ns2)=O)CCCN(C(c2n[nH]c(C3CC3)n2)=O)C1 c1(CCNC(CC(CC)C)C)nc(C(C)C)c(Cl)cc1Br c1(C(=O)NCCC2CCCN(C(C(F)OC)=O)C2)c(C)ncnc1C N1(C(=O)CCc2cnoc2)CCOC(C(=O)NC2CC(n3cncn3)C2)C1 c1(OC)ccc(C)c(C(N2C3CCC2C(CNC(C2CC4CC4C2)=O)C3)=O)n1 c1(N(C(C(C)(C)C2CCCO2)=O)CC2C(CNC3CC3)COC2)ccc(Cl)nc1 C1(C)(CNC(C(F)OC)=O)CC(F)(F)CN1C(c1ccc(C(C)(C)C#N)cc1)=O C1(CCNC(C(CC)OC)=O)CC2CCC(C1)N2C(c1nn[nH]c1C(F)(F)F)=O Cc1nc2cc(CNC(=O)CC(C)CC(C)C)ccc2s1.C123CC(C1)(C2)C(=O)N3 Cc1c(F)ccc(Cl)c1C(N1CCN(C(=O)C(=O)NC(C2CCCO2)C)CC1)=O CN(C)N=Nc1ccccc1C(N1CCC(NC(C2CC(=O)NC(=O)N2)=O)C1)=O c1(OCCCC)ccc(C(=O)N(C2CCCC2)CCO)cc1.C1(=O)C(CO)N1 N1(C(CCOCCCOC)=O)CCCOC(CNC(c2cccc[n+]2[O-])=O)C1 C1(CNC(Cc2cc(OC)no2)=O)C2CN(C(c3cc(CCCO)on3)=O)CC12 C1(CNC(C2(C)CC2F)=O)(CNC(=O)Cc2ccccc2Cl)CCCCC1 N1(C(C(CCOC)OC)=O)CCCN(C(=O)COc2ccc(Cl)nc2)CC1C Cc1cc(Cl)cc(C)c1C(N1CC(O)(C2CCCN2C(=O)C(=O)N(C)C)C1)=O N1(C(C(=O)NC(c2ccccc2Cl)C)C)CCC2(CCCC2)CC1 c1(N(C(=O)CCCC(=O)C(C)(C)C)C)nc(=NCC2C3CCCC23)[nH]c2cc[nH]c12 N1(C(=O)C(c2ccc(OC(F)(F)F)c(Cl)c2)=O)CC2CC(C1)CN(C(=O)CO)C2 C1(C(N2CC3CCN(C(c4c(C)nco4)=O)C3C2)=O)CCc2ccccc2C1 c1(CCO)ccc([N+](=O)[O-])cc1.N1(C(C2(C3(C)CCCO3)CC2)=O)C2CSC1C2=O N1(C(C=CCCCCC)=O)CC2CC1CN(C(=O)C(O)(CC)c1ccccc1)C2 c1(C(=O)NC2CCN(C(C(CCCC)=O)=O)CC2F)ccc2c(c1)C(C)(C)CO2 N1(C(CCNC(=O)OCC)=O)CC(C)N(C(=O)CCNc2ncccn2)CC1C CC(C)(C#N)CCCC(=O)N1CC(NC(C2CC2c2cccs2)=O)C(F)C1 Cc1ccc(C(=O)OCCOC2CC(C)C2)cc1I C1(C(N(C(c2ccc(N3CCCCC3=O)cc2)C)C)=O)CCCS(=O)(=O)C1 C1(NC(C2C(=C)C2C(=O)OC)=O)CCOCC1C(=O)NCCn1ccc(=O)cc1 c1(CSCC(=O)NCCC(C)N(C(C(C)C)=O)C)nc(-c2ccncc2)no1 C1(C(=O)NCC(CCNC(c2cccc(OCCF)c2)=O)O)CCCC12CCC2 N1(C(c2c(C#C)cc(F)c(OC)c2)=O)CCC(C2=NOC(CN)C2)CC1 C1(c2c(C(=O)OC)c[nH]n2)CCCCN1C(=O)Nc1ccc(Cl)cc1 C1(CCOC)CN(C(=O)C=Cc2ncc[nH]2)CCN1C(C12COC(CF)(C1)C2)=O CC1=C(C(=O)N2CC(C)C(C)(CNC(=O)Cc3cc(C)cc(F)c3)C2)CCCC1 CCC1=C(C(=O)NC2CCC2CNC(c2cnc(O)c(F)c2)=O)SCCO1 c1(C(=O)NC2(C)CCCN(C(Cc3c(C)ccnc3)=O)C2)cc2ccccn2n1 c1(-c2nc(SC)sc2)ccc(C(N2CC3C(c4ccc(SC)o4)(C3)C2)=O)cc1F N1(C(C2C(C)C2)=O)CCC(C)(NC(c2coc(OC(C)C)n2)=O)CC1 C=CC1(CO)CCN(C(C2(NC(=O)C(O)C(F)(F)F)CCN(C)C2)=O)CC1 CC(C)(CCCNC(=O)C(C1CCCCCC1)F)NC(=O)C=CC1CCCCC1 C(C)(C(=O)NC1CCC(NC(c2coc(C3CCC3)n2)=O)C1)(C1CC1)OC C1(NC(=O)C=Cc2cc[nH]c2)CC2CC1N(C(c1ccccc1Cl)=O)C2 C1(C(N2CC(C(C)NC(C3C(OC)C3)=O)OCC2)=O)CC12CCSCC2 c1(SCC)nccnc1C(=O)NC1CCC(C)(CNC(=O)CC2OCCO2)C1 N1(C(CNC(c2ncc(C)o2)=O)=O)CC=CC1(C)C CCCCC(C(=O)N1CCC1)NC(=O)CNC1CCN(C(C)(C)C)C1 C1(C(=O)NCC2(CNC(c3nc(OC)oc3)=O)CC2)CC2(C1)CC(F)C2 C1(NC(C(C(C)C)N(C)C)=O)CC2CCC(C1)N2C(c1ccc(=O)n(O)c1)=O C#CC(CNC(=O)C(F)CC(C)(C)NC(=O)Cc1cnn(C)c1)CC(C)(C)C N1(C(=O)Nc2c(COc3c(C)ccc(C)c3)cccc2)CC2(COC(=O)C2)C1 N1(C(=O)C2=COCC2)CC2CCN(C(c3cc(F)c(F)cc3O)=O)CCC2C1 Cc1cc(=NCC(F)(F)C(C)C)[nH]c(N(C)Cc2cccc(S(C)(=O)=O)c2)n1 CC(C)CC(C(=O)N1CCOCC1CNC(=O)C(F)CC1CC1)N(C)C c1(CC)cc(=NCC2OCCC2NCCn2cccn2)[nH]cn1 C(=O)(C1CCCc2c[nH]nc21)N1CC2CC(NC(CC(C(C)C)OCC)=O)C2C1 N1(C(C(CSC)O)=O)CCCC(CCNC(=O)CC2(O)CCCCC2)CC1 c1(C(=O)NCC(C)NC(=O)CC(C)c2ccco2)cnc(CC2CCCC2)[nH]1 c1(C(=O)NCC(C(C)C)NC(=O)CC2CCCN2C)cc(O)nc2c1CCC2 C(C(C)CNC(=O)COC(C)(C)CNC(=O)C(C)n1ccnn1)OCC C(=O)(C1=C(Cl)CCOC1)NCC1(C)CCCC1.N12CCC1C2=O C=C(C)CCC(=O)NC1CCC(CNC(C2OCCC2C)=O)C1 c1(SC(C)C)ccc(C(=O)NCC2(F)CCN(C(=O)C(C)c3ccsn3)C2)cc1 c1(C(N)=O)cncc(NC(C2(C)CCCN2C(c2cccc(O)n2)=O)=O)c1 Cc1cccc(CC(=O)NC2C=CCN(C(=O)CC(C)n3ccnc3)C2)c1 c1(C(C)C)ccc(C(=O)NC(C)(CNC(=O)C(=O)NCC(F)F)C(C)C)cn1 c1(C(=O)NCC2(CNC(c3ncc[nH]c3=O)=O)CC2(F)F)cc2ccccc2s1 CC(CC(C)NC(C1CCCN1C1CC1)=O)NC(=O)C(C)NC(=O)C1CC1 Cc1cc(C)c(C(N2CCC3C(NC(C4CCCC(=O)N4)=O)C3C2)=O)cn1 C(C(C)(C)C(=O)NCC1C(C(=O)NOCC2CCCO2)C1(C)C)NC(C)=O Cc1oc(C)c(S(N)(=O)=O)c1C(=O)NCC1CC1CNC(=O)CC1(C(F)F)CC1 c1(CC)nnsc1CCCNC(=O)C(O)CC1CCCC1.C12CC(C1)NC2=O C(=O)(C(CCC(C)C)NC(C1CN(C)CCO1)=O)N(C)Cc1c(CC)noc1 Cc1ncnc(C)c1C(N1CCN(C(=O)C(=O)NC(C)C)CC1C1CCC1)=O Cc1cc(C(=O)NCC2CC3CN(C(c4cnsc4)=O)CC23)c(Br)cn1 CC(C)C(C)(CNC(=O)C(C)n1ccnc1)NC(=O)Cn1nnnc1C1CC1 N1(C(CCN(C(C(c2cccnc2)C)=O)C)=O)CCC(O)C(N(C)C)C1 Nc1ccc(Cl)nc1C(=O)NC1CCCCC1NC(=O)CNC(=O)CC(F)(F)F c1(C(N2C(C(C)(C)NC(c3onc(COC)n3)=O)CCC2)=O)cc(O)cnc1N c1(C(N2CC3C(CNC(C(CCOC)(C)C)=O)(CC3)C2)=O)cnn2cccnc12 N1(C(c2cc(OC)ns2)=O)CC(C)N(C(=O)Cc2ccsc2)CC1C C(C1CN(C(=O)CCC(N)=O)Cc2ccccc21)NC(C1CC(C)=C(C)CC1)=O C(=O)(C1=C(C)CCCC1)N(CC(CC)NC(C1CC12CCC2)=O)C Cc1c(O)c(=O)ccn1CC(N1CCC(OCCNC(=O)C#CC2CC2)C1)=O c1(C(N2CC(C)C(NC(C3CCCN3C)=O)C2)=O)c(F)cccc1[N+](=O)[O-] CCCCCC(O)C(=O)NCCOCCCN(C)C(c1c(C)cccc1N)=O C1(NC(=O)OCC)CCC(CCNc2ccnn2CC(F)F)CC1 C1(N(C(C(=Cc2cccnc2)C)=O)C)CCCN(C(=O)C(C)(C)CC2CC2)CC1 CC(CNC(=O)CNC(=O)Cn1ccnn1)CC1CCCC1 N1(C(C(C)(C)O)=O)CCC(CO)(NC(=O)CCN2CCOC2=O)C1 Cc1oc(C(N2CCC(C)(CNC(=O)C(F)(F)CO)C2)=O)cc1-c1ccccc1 CC#CCC(C(=O)Nc1cccc(CCF)c1)NC(c1ccc(C)n1C)=O c1(C(=O)NC2CCN(C(Cc3nc(C)sc3)=O)C(C)C2)coc2c1C(=O)NCC2 C1(OC)CC(CNC(=O)Cc2ccn(CC(C)C)n2)N(C(=O)CN2CCCC2)C1 c1(C(=O)NCC2C3CN(C(C(C)OCOC)=O)CC32)cccc(=S)n1O C12(C(=O)NCC(CNC(C3(C(=O)OCC)CCC3)=O)O)CCCN(CCC1)C2 C(=O)(C(C)(C)COC(C)C)NCC1(CNC(C(C=C)O)=O)CCC1 c1(CSc2nc(C(C)NC(N)=O)sc2)nc2cc(Cl)cnc2[nH]1 C1(C(N(C2CCCN(C(=O)CNS(N)(=O)=O)CC2)C)=O)CCC(C2CCC2)CC1 CC1C(C)N(C(C2(CO)CC2)=O)CCN1C(c1cnnc(C2CC2)c1)=O N1(C(CCC=CC)=O)CCOC(CN(C(=O)C(C(C)C)NS(N)(=O)=O)C)C1 C(N=c1[nH]c(=NCCCC2CCCCO2)c2sccc2[nH]1)C1C(O)CCC1 C1(NC(C2C(C)(C)CCCN2C(C2CC23CC3)=O)=O)CCn2nccc2C1 N1(C(c2ccc(CC)s2)=O)CC(NC(=O)C2=CC3C=CC2C3)CCC(O)C1 C(=O)(C1=CC2C=CC(C1)C2)N1CCC(C(=O)NCC(C)OC(F)F)C12CCC2 C1(CNC(CCc2nnc(C)o2)=O)CC2COCC2N1C(=O)CC1(O)CCCC1 C1(F)(C(=O)NC(C2CCCC2)CNC(CC2CC(=C)C2)=O)CS(=O)(=O)CC12COC2 C(CCCCC(=O)N1CC(NC(=O)C(C2(O)CCCC2)F)C2(CC2)C1)OC c1(CC)oc(C)cc1C(=O)NCCCC(C)(C)NC(C1CC1c1ccccc1)=O C1(NC(C(F)OC)=O)CCN(C(c2ccc(Cl)nc2N)=O)C12CCC2 C(CCSC)(C(=O)N1CC(CC(C)NC(c2ccc(OC(C)C)cc2)=O)C1)OC CC#CCC(C(=O)NC1CN(C)CCC1O)NC(c1occc1C)=O Cc1cc(C(=O)NCC(C)(C)NC(=O)CC2CCC(C)O2)ccn1 c1(C(N2CC3C(CNC(c4c(C)nsc4)=O)(C3)C2)=O)nc(Br)cnc1N C1(CNC(c2ccc(C(C)C)s2)=O)(OC)CCCN(C(=O)C2CC2)C1 C(=O)(CCCC(C)=O)NC1CCC(NC(c2cn(CCOCC)nc2)=O)CC1 C12(NC(C3CC=CC3)=O)COC(CNC(c3ccc(-c4ncc[nH]4)cc3)=O)(C1)C2 N12CCC(C3(CCC3)NC(CC)C1=O)CC2.C1(=O)CC(C)(C)N1.O(C)OC CC1(C)C2CCC(C2)C1C(=O)NCC1(COC)CC1.[nH]1cc(-c2nc[nH]n2)nn1 C(CC(C)C(=O)N1CCC=CC1C(=O)N(C)Cc1cscn1)=CCC C1(NC(C(N2CCCC(N3C(=O)CCC3)C2)=O)=O)C2CC3CC(C2)CC1C3 c1(CC)nc(C)[nH]c1C(=O)NC(C)(C)CN(C(=O)CSCCOC)C Cc1cc(C#N)c(NC(C2NCCCCC2(F)F)=O)cc1F Cc1cc(C(N2CCOC(C(C)NC(c3ccc(CF)cc3)=O)C2)=O)nn1C Cc1ccc(Br)c(C(=O)NC2C3CCN(C(C4CC(N(C)C)C4)=O)CC23)n1 C1(CCC)CN(C(C2CC(=O)N(C(C)C)C2)=O)CC1NC(C1CN(C)CCO1)=O C(C)(CCCNC(C1CN(CC(C)C)C1)=O)NC(C(C)NC(C)=O)=O N1(C(c2cnc(C)[nH]2)=O)CC2CCN(C(=O)C(C)S(N)(=O)=O)CC(C2)C1 c1(CN(C(=O)CC=CCNC(=O)C(CO)N(C)C)C)ccc(C#N)o1 n1(-c2cccc(C(=O)OC)c2)ncc(=NC(=O)C2CCCC2C2CC2)[nH]1 N1(C(C2(C)C=CCC2)=O)CC2(COC(CNC(c3cc(C4CCC4)no3)=O)C2)C1 CC(CCN(C)C)C(=O)NC(Cc1ccco1)C(=O)NCCc1ccon1 C1(C(C)(C)C)CCC(=CC(=O)NCC2CC(C)N(C(c3cncc(C)n3)=O)C2)CC1 C1(CC(C)C)CCCN(c2nnc(C(C)(C)C3CC3)n2CCC(C)C)C1 C(=O)(C1=CCOC1)NC1(C)CC(NC(c2cnc(S)[nH]2)=O)C1 C(=O)(CCCN=[N+]=[N-])NC(CNC(C(c1cccs1)SC)=O)(C)Cn1cccn1 c1(C(=O)NCCOC2CCN(C(c3ccco3)=O)C2)cc(F)cs1 CCC(CC)C(C(=O)NCC1CCN(C(=O)C(F)(F)c2ccncc2)C1)OC N1(C(CS(=O)(=O)NCC)=O)CCC(NC(C2(CO)CC2(F)F)=O)C(CC)C1 c1(C(=O)NC2C(C)N(CC3CC34CCOC4)CCC2)ccc2ncsc2c1 C(CCO)(C(F)(F)F)NC(CC1C2CN(C(Cc3n(C)ccc3)=O)CC21)=O C1(C(=O)NC2CC(C)(NC(=O)OC(C)(C)C)C2)(OC)CN(C)C1 N1(C(C(c2cnccn2)C)=O)CCCN(C(c2ccnc3c2CCC3)=O)CCC1 Cc1nc2ncccc2cc1CC(=O)N(CC(O)CN(C)C1CC1)C N1(C(CCCOC(C)=O)=O)CC2(CC(C(N3CCC(C)(CO)C3)=O)CO2)C1 CCC(CC(F)F)C(=O)N1CCC(C(N2CC3(C2)CN(C(C)C)C3)=O)CC1 c1(OC)ccnc2c1CCN(C(=O)Nc1cc(C)ncc1C#N)C2 c1(NCCC2CC(NC(C(Cc3ccccc3)OC)=O)C2)ncnc(C)c1Br C1(C(=O)NCC(=C2CN(C(c3ccc(F)cc3F)=O)C2)F)CC2C(C1)C2(F)F c1(OC)cc(C(=O)NCC2CN(Cc3cc(F)c(F)cc3C)C2)ccc1C#N Cc1nc2ccc(C#N)cc2cc1C(N1CCC(c2ncccn2)CC1)=O C1(C(=O)NCC(CN(C)C(c2ccc(O)c(N)n2)=O)O)CCC2(CC1)CC2 N1(C(=O)CCOC2COC2)CCCC(F)(CNC(=O)CCOC2CC2)CC1 c1(C(=O)NCC2C(CNC(Cc3cc(C)nn3C)=O)C2)cccc(Br)c1N c1(OC)ccc(Cl)cc1CC(=O)NC(CNC(C1CCCCC1(C)C)=O)C1CC1 C=C(C)CCC(=O)NC1CC1NC(=O)CSCc1cnn(C)c1 C(C1CCOC1)=CC(=O)NCCN(CCC)C(C1CCOCC1)=O CC1(C)OCCC1NC(c1sc(Br)cc1I)=O N#CCCCCC(=O)NC1CCCCC1CNC(c1cn(C2CCCC2)nn1)=O Cc1ncc(C(N2CC(F)(CNC(=O)C(F)=C3CCC3)C2)=O)cc1CC(C)C C1(NC(c2cc(C(C)(C)C)n[nH]2)=O)CC2CC1N(C(C1(c3ccsc3)CC1)=O)C2 c1(C(=O)NC2CC(C)CN(C(=O)CCSC3CCCC3)C2)cc(S(N)(=O)=O)c[nH]1 C1(C(=O)NC(c2cnn[nH]2)C)CC(NC(C2CCC3(CC3)C2)=O)C(O)C1 c1(CC)nc(C)c(C(=O)NCCCCN(C(=O)CN2CCNC(=O)C2)C)c(C)n1 CC1CN(C(=O)Cc2cn[nH]c2)CCC1CNC(C1(C)CCC1)=O CCCC(O)CC(=O)NC1CCC1NC(c1ccc(Cl)cc1F)=O N1(C(C(C)OC)=O)CC(CO)C2(CCN(C(c3ccn4nccc4c3)=O)CC2)C1 c1(N2CC(CCO)(NC(CC3(CC)CCC3)=O)C2)cc(CC)ncn1 c1(OC)ccc(C(N)=O)c(NC(=O)C(N2CCC(O)C2)c2ncco2)c1 C1(C(N2C(CN(C)C)CCC2)=O)CCC(O)CN1C(=O)CN1CCC(F)CC1 c1(C(N2CC(C)(C)C(NC(C3(F)CC=CC3)=O)C2)=O)ccc(S(N)(=O)=O)cc1 C1(C(=O)NC2CC(C(C)NC(c3c(CC)cno3)=O)C2)CCC(N=[N+]=[N-])C1 C(=O)(C(C)CC(C)(C)C)NCCc1nc(C)c(-c2cccc(Cl)c2)o1 C(=O)(C1CCCc2ncnn21)N1CCCC(NC(=O)COCCF)C1 c1(C(N2CCC(O)(C(C)NC(c3csc(Cl)c3Cl)=O)CC2)=O)nc2ncccn2n1 CC(C)C(C(=O)NCC(C)(C)CNC(=O)CCOCC)NC(=O)OC(C)(C)C c1(CC(=O)NC(C2CCN(c3nnc(C)o3)C2)C)cnccc1C C12(C(N(CC=C)Cc3cn(CC4CNC(=O)O4)nn3)=O)CCCCC1OCC2 C12(COC)CCC(NC(c3ccc(C)c(I)c3)c3nnnn3C)(CC1)CO2 c1(CC(=O)NCCN(C(=O)CCC2CCC(=O)N2)CCC)nc(C)sc1C N1(C(c2c(CC)nc(C)o2)=O)CC(NC(=O)CCc2nc[nH]n2)C2(CC2)C1 C1(C(=O)NCCSCC)(C(C)C)CCN(C(=O)C(C)CC2CC2)C1 N1(C(C(CC)O)=O)CC2CC(C1)N2C(=O)CCc1c(C)noc1C C1(C(=O)NCCCNC(=O)C(F)(F)CC2CCCO2)CC2CC(O)C(C1)C2 Nc1ccc(C(F)(F)F)cc1C(N1CCOCC1CNC(C1(Cl)CC1(F)F)=O)=O c1(C(=O)NCCC(C(=O)NCc2nnc(O)n2C)OC)cccc(C)c1O C1(CNC(CSCCCC)=O)C(C)CCCN1C(c1cc(Cl)cn1C)=O C(CCC(C)(C)C(=O)N1CCC(c2nc[nH]n2)C1)NC(c1ccn(CC)n1)=O C1(CNC(c2ccc(C)cn2)=O)CCN(C(c2cc(C)on2)=O)C12CC2 CS(=O)(=O)c1ccc(N2CC3CCCC2C3CNC(C2(C(=O)NC)CC2)=O)nc1 c1(C(=O)OCC)ccc2c(c1)N(C(=O)C(=O)NC(C1CN(C(C)C)C1)C)CCC2 C(c1ccc(F)cc1F)=CC(N1C(C)(C)CC(CNC(C2CCCS2)=O)C1)=O N1(C(C(C)OC2COC2)=O)CC2(CC(NC(=O)CC3CCOC(C)(C)C3)C2)C1 C(C(=O)NNC(=O)C(=O)Nc1nc(-c2cccc(C)c2)cs1)(C(C)C)SCC N1(C(C(C2CCC2)NC(c2ccc(C)nn2)=O)=O)Cc2ccc([N+](=O)[O-])cc2C1 c1(OCC)cnc(C(=O)NCC2CC(NC(C3(OC)CC3)=O)C(O)C2)cn1 C(CC(C)C(F)(F)F)CCC=O.C(CC1CCC1)(C(=O)N1CCC1CC1CC1)OC CCC(O)C(C)C(=O)NC(CNC(c1ccc(Cl)cc1N)=O)(CC)CC N1(C(C2CC(OCC)C2)=O)CCC2(CC1)CCN(C(=O)CC(C)O)C2 C12(C(N3CC(CC=C)(NC(C4CC(CC)=NO4)=O)C3)=O)CC3CC(CC1C3)C2 Cc1ccc(S(=O)(=O)CCN2CCC(C(=O)NCCc3ncc[nH]3)CC2)cc1 c1(C(=O)NCCCN(C)C(C2(Cl)CC23CCC3)=O)ccnnc1O N1(C(C2CN(C(C)C)C2)=O)CCCC(CO)(NC(c2cc3occc3s2)=O)C1 c1(C(=O)NC(C(=O)N2CC(C(C3CC3)CC3CC3)C2)c2cccs2)cnccn1 c1(C(=O)NC2CC(NC(CC#CCC)=O)C(O)C2)c(F)ccc(F)c1F c1(C(N2CC(F)(C(C)(C)CNC(=O)CSC3CC3)C2)=O)cc(Cl)cc(F)c1N N1(C(c2c(C)csc2C)=O)CCC(C)(C)CC1C(=O)N(C)Cc1cc(C)on1 C(=O)(C#Cc1cccs1)N(c1cccc(C)n1)C1CC1 C(=O)(CC(C)(C)CN(C)C)N1CC(CCNC(c2c(CC)cccc2)=O)C(O)C1 N1(C(CCNC(CC(C)C)=O)=O)CCCC(NC(=O)CN(c2ccoc2)C)C1C c1(OC)cc(C(=O)NC(C)(C)CNC(=O)CC2(n3ccnc3)CC2)sn1 N1(CCCCC=C)CCn2cc(-c3cn[nH]c3)nc2C1.c1(N)[nH]nc2cnccc12 Cc1ccc([N+](=O)[O-])c(OCCSCc2cc(F)c(F)c(F)c2)c1 C(=O)(CCC(=O)C(C)(C)C)CC(=O)N(CC)CC.c1(C(N2CC(O)C2)=O)cc(C)co1 CCC(C)(CNC(=O)CCN(C(c1cc(C#N)n(C)n1)=O)C(C)C)C(C)O C1(C(=O)NC2C(C)(C)C2C(=O)NC2CC(O)(CO)C2)CC2(CSC2)C1 C1(C(N2CCN(C(c3cc(CC)no3)=O)CC2C(C)C)=O)CCc2c[nH]nc2C1 c1(N2CCCC(C)(C(N3CCCC(C)(O)CC3)=O)C2)nccc(S(C)(=O)=O)n1 C12(CNC(C=NOC)=O)CC(NC(=O)COc3cc(C)on3)(C1)C(C)(C)O2 C1(CNC(c2nc(CC)[nH]n2)=O)CCN(C(c2nc3c(s2)CCC3)=O)CC1C CCC(CC)C(F)C(=O)NC12CCC(C(=O)NC3CCNC(=O)C3)(CC1)C2 c1(C(N2CC(N(C(c3c(COCC)noc3)=O)C)C2)=O)c[nH]c2ccc(Cl)cc12 C(=O)(C(F)(F)C(F)F)NC1CCN(CCNC(C2N(C(C)=O)CC(O)C2)=O)CC1 C1(C(N(CCCCCCNC(C(CC)(C)O)=O)C)=O)CCCCCC1(F)F c1(NC(N(C(c2ccc(I)cc2)C(=O)OC)C)=O)ccc(O)nc1 C=CC(C)(O)CC(=O)NC(CNC(c1sccc1F)=O)C1CCC1 CCC(C)C(O)C(=O)N(CC)CC1CCCN1C(=O)CCc1nnc(C2CC2)o1 c1(N(C(=O)NC(CC2CC2)C2CC2)C2CC2)cccc(C(F)(F)F)c1 C(=O)(CN=c1cc[nH]cc1)NC(CC(C)NC(C1CC2(CCOC2)C1)=O)C C1(CNC(CC=CC=C)=O)CC2CC1CN2C(=O)Cc1nnn(C(C)(C)C)n1 Cc1ccccc1C(CN(CC(CO)NC(C1CCCCC1)=O)C)N(C)C N1(C(Cc2cc(C)cc(F)c2)=O)CCC2CN(Cc3cc(C#N)ccc3Cl)CC12 N1(C(c2n(CCC)ccc2)=O)CCN(C2CC(NC(c3ncsc3C)=O)C2)CC1 C1(=O)C(CC(C2CCCCC2)OC)N1.c1(CCCN(CC=C)CCO)ccccn1 c1(N(CCNC(C(C)N(C(C)=O)C)=O)C(C)C)cccc(F)c1[N+](=O)[O-] C1(NC(CSC)=O)CCC(C)N(C(=O)CC2CCOC2(C)C)C1 N1(C(COC(CC)C)=O)CC(C)C(C)(CNC(=O)CCC(=O)c2ccncc2)C1 C1(OC)CCN(C(C2CCC(NC(c3cc(C)nc(O)c3)=O)C2)=O)C(C)C1 c1(OC)ccc(F)c(C(=O)NC2CCN(C(=O)Nc3ccc(F)cc3)CC2)c1F N1(C(C(F)=C(C)C)=O)CCC(C(=O)NC2CCN3CCC2C3)C1(C)C C1(F)(CNC(CCCN(C)C)=O)COCCN(C(=O)COc2ccccc2F)C1 C1(C(N(C)CC2(CNC(C3C(C)CCO3)=O)CC2)=O)CCn2c(O)nnc2C1 C=CC1(CC(=O)N(CC(F)F)CC)CN(C(=O)C2COC2)C1.OCC S(=O)(=O)(c1ccc(NCCOCCF)c(Cl)c1)N1C(CC)CC(O)C1 n1(CC)cc(C(=O)NCC2CN(C(C3(F)CCOC3)=O)C2)c(C(F)(F)F)n1 Cc1cnccc1C(=O)N(CCNC(=O)Cc1ccnc(O)c1)C1CC1 C1(CNC(C2(CC#C)CCC2)=O)CC(C)(C)CN1C(c1ccc(F)c(C)c1)=O c1(NC(c2ccccc2)CNC(c2cnc(CC)s2)=O)cncc(Cl)n1 c1(C(=O)NC2(CN(C)C)CC2)cc(CNC(C2CC2(F)Cl)=O)cs1 c1(C2C(NC(C(C)OCC)=O)C2)ccccc1Br CC(C)(C)C(O)C(=O)NCC1CCN(C(=O)COCC(=O)Nc2ccccc2)C1 C1(C(=O)NCCCC(=C)Cl)CCC(NC(=O)Cn2nnc(C)n2)CC1 C1(NC(=O)CSc2ccccc2)CC2CN(C(C3SC4C=CC3CC4)=O)CC12 N1(C(C#CC)=O)CCCCC(NC(C2SCCCS2)=O)C1 c1(C(=O)NCC2CC(NC(C(C)=CC(C)C)=O)C2(C)C)ccc2c(c1)CCC2=O CC1(NC(C2CCC23CCC3)=O)CCCN(C(C2CCCCC2(C)C)=O)C1 N1(C(C(C2CCCCC2)OC)C(=O)NCC(C)C)CCCC2CN(C)CCC12 C1(C2N(C(Cc3nc(C)sc3)=O)CCC2)CCCN(C(c2cccnc2Cl)=O)C1 C(=O)(CCC(=O)NC(C)(C)CNC(=O)C1CC1)Nc1c(-c2cn(C)nc2)cco1 C1(C)(CCN(C(c2ccn(C)c2)C)CC)CCOC1C C1(C(=O)OC)CCCCN1C(=O)CC1CCCN(C(=O)CN2C(=O)CNC2=O)C1 C1(CN=[N+]=[N-])CN(C(C2CCOC(C(F)(F)F)C2)=O)CCO1 N1(C(C2C(C)C2c2ccccc2)=O)CCC(CNC(=O)C(=O)Nc2ncc[nH]2)C1 Cc1ncccc1CCC(=O)NCC1CCN(C(c2ccc(CO)o2)=O)C1 C(=O)(C1=CC2C=CC(C1)C2)NCC(C1CC1)NC(CCOCc1nnc(C)s1)=O c1(N(CCC2(C(N(CC)OC)=O)CC2)C(=O)NN2CCOCC2)cncc(C#N)c1 C1(C#N)(C(N2CC(CNC(CC(C)c3ccccc3)=O)C2)=O)CC1(C)C c1(CC)oc(C)cc1C(=O)NC1(CCC(=O)NCC(O)C(C)C)CCC1 N1(C(c2scc(C)c2)=O)CC2CC1CN2C(C1CCC(C(C)C)CC1)=O C1(NC(C(C)CO)=O)CCCCCCC1NC(=O)CCCS(C)(=O)=O CC1CC2(CC(NC(=O)C(F)C3CC(NC(C4OCCC4(C)C)=O)C3)C2)C1 CC(C)CCCCCC(=O)NC1CC(C)(NC(=O)CN2CCCC2C)C1 C1(NC(CC(CCC)(C)O)=O)CC1C1CCCN(C(c2ccc(F)nc2F)=O)C1 C(=O)(C(C)(O)CC(C)C)NC(C1(O)CCN(C(CCCC#C)=O)C1)C c1(C(=O)NCC(CNC(C2CCCC(C(=O)OC)C2)=O)O)cc2sccc2n1C n1(CC(=O)N(C(CC(C)C)c2ncccn2)C2CC2)cc(I)c(=O)c(I)c1 c1(OC)cc(C(=O)NC2CCCC2CN=c2nc[nH]s2)ccc1F c1(OC)cc(CC(=O)NCC2CC(NC(C3CCC(=O)N3)=O)CCO2)ccn1 N1(C(c2c(C)sc(O)n2)=O)CCCC(NC(=O)C(CC#N)c2ccccc2)CC1 N1(C(C(C(C)C)C)=O)CCCN(C(c2occ3c2CCOC3)=O)CCC1 C1(C2CCN(C(c3nc(=N)[nH][nH]3)=O)C2)(NC(C2ON=C(C)C2)=O)CC1 c1(N2CC(C)(CNC(C(CCC)OC)=O)OCC2)cc2c(cn1)C(=O)CCC2 C1(CC(=O)NCC2(NC(c3c(F)cccc3F)=O)CC2)Cc2ccccc2O1 C1(CCOC)CN(C(c2ccc(CCO)cc2)=O)CCN1C(c1ocnc1C)=O C1(C2CC2)(NC(C(C)OCC)=O)CCN(C(c2csc(Cl)n2)=O)C1 c1(N(C)Cc2ccc(C3CC3)cc2)ccc(Br)c(C#N)c1 c1(C(=O)NC2N(C(C(=O)NCCC(=O)OC)=O)CCC2)cnc(CCOC)n1C Cc1cc(C(N2CCN(C(=O)CCCC#N)CC2)=O)c(C)n1-c1ccncc1 C1(NC(C(C2CC2)OC)=O)CCN(C(c2ccc(O)nc2Cl)=O)C1(C)C N1(C(C=Cc2ccc(C)cc2Cl)=O)CCOC2CCN(C(c3cnn[nH]3)=O)CC12 c1(N2CC(F)CC(OC)C2)[nH]c(=NC2C=CCC2)nc2c1cnn2C(C)C c1(SC)cc(C)ccc1C(N1CC(NC(C2CC2C(F)F)=O)C(O)C1)=O C(=O)(C1=C(C)CCCC1)NC(CCC)C(=O)NC(CC)CCOC c1(C(=O)NCC(C2CC2)NC(CC2(N(C)C)CCCCC2)=O)ccc(Cl)c(Cl)c1 N1(C(C(C2CCOCC2)C)=O)CCC(C(=O)NCC2(C)CCCS2)=C(F)C1 c1(OC)c[nH]c(C(N2CCCCC2C2CCOCC2)=O)cc1=O C1(CNC(COCCCC)=O)CCC2CN(C(=O)Cc3csnn3)CCC2C1 C(C)(CO)(C(F)(F)F)NC(c1c(CNC(c2c(C)scc2)=O)n[nH]c1)=O Cn1cc(Br)c(C2CCCN2C(=O)NCCC2CN(C(=O)OC(C)(C)C)CCO2)n1 S(=O)(=O)(c1ccc(NCC(c2cccs2)O)cc1Cl)NCC1(CC#N)CC1 C(=O)(C1=NNC(=O)CC1)N(C1CCCN(C(c2ccc(CC)c(N)c2)=O)C1)CC C(=O)(CCN=c1nc2cc(C(F)(F)F)ccc2c(N2CCCC(C)C2)[nH]1)NC N1(C(COCC(=O)OC)=O)CC(F)(CNC(=O)COCCF)C1 N1(C(CCc2n(CC)ccn2)=O)CCCC(NC(=O)CCCNC(=O)OC)C1C CCCS(=O)(=O)CC(=O)N1CCCN(C(=O)CC2CCC(C)O2)CC1 c1(C(N2CC3C(NC(C(CC)C)=O)C3C2)=O)cc(Br)c2ncccc2c1 N1(C(CC)C(=O)NC2(NC(=O)COC(C)C)CCOC2)CCN(CCO)CC1 c1(C(=O)NC2CC(NC(CCCOCCC)=O)C2)cnc(S)nc1 N1(C(=O)NC(=O)C(CC)NCC2CCCO2)CCN(CC2CCN(C(C)=O)CC2)CC1 c1(-n2ccc(SCc3onc(-c4[nH]cc(Br)n4)n3)n2)ccc(F)cc1 CC1(C)CN(C(C2CCC(O)CC2)=O)CC1NC(c1cccnc1)=O C1(C)(NC(CCCn2cc(-c3c(C)noc3C)nn2)=O)CCCN(S(C)(=O)=O)C1 C(=O)(N(CCO)OC)c1cc(CCC)[nH]n1.C1(=O)C(C)C(C)O1 c1(C(=O)OCCSC(CC)C)cccc(-n2cccc2)c1 C1(CCOCC)(NC(c2cnc(C)[nH]2)=O)CCN(c2ncc(C)cn2)C1 C(C(C)(O)CNC(=O)CN(C(c1ccn(C(C)C)n1)=O)CC1CC1)OC N=c1nc(C(=O)NCc2cc(C(=O)NCC#CC3CC3)co2)cc[nH]1 CCCCN=C(NCC1(CO)CCCO1)N1CCC2(CCC(O)CC2)CC1 c1(C(=O)NC(C)CN(C)C(c2ccc(CS(N)(=O)=O)cc2)=O)cn2ccsc2n1 c1(C(N(CC(=O)NCc2nc(C)[nH]n2)C)=O)ccc(C)c(C#N)c1 c1(C(N2C(CNC(C3N(C(C)=O)CCC3)=O)CC3(CC3)C2)=O)cccc2nncn12 c1(C(C)NC(=O)N(C)Cc2ccc(SC(F)F)cc2)cccc([N+](=O)[O-])c1 S(=O)(=O)(c1ccccc1F)N1C(CC(=O)Nc2c(C(=O)OC)nccn2)CCC1 C=CCCCCC(=O)NC(CNC(C1CCCC(N(C)C)C1)=O)C(C)(C)C C(=O)(C#CC1CCCC1)NC1CCCC(CN(C(=O)CC2(O)CCCCC2)C)C1 c1(C(=O)NCC(C)N(C(=O)C=CS(C)(=O)=O)C)nc2cc(F)ccc2o1 N1(C(CC(C(C)C)C)=O)CCC2CCN(C(c3cc4cc(O)ccc4[nH]3)=O)CC12 CC1(C)CC(C(=O)NC2CC3(CCCO3)C2)CN1C(C1CN2CCC1C2)=O N1(C(C2N(C(=O)NC)CCC2)=O)CCN(C(c2cc(F)n[nH]2)=O)C(C2CCC2)C1 C(=O)(C1=NN2CCCN=C2N1)NC(C)CC(C)NC(C1COCCO1)=O Cc1ccc2c(c1)C(NC(=O)C(=O)N=S(C)(C)=O)CN2C(=O)C(F)(F)Cl c1(OC)ccc(C(=O)NC2CCCN(C(=O)CC3C=CCC3)CC2)c(Cl)c1OC CCCC(C)CCN(C(=O)Nc1ccc(OCCC)cc1)C1CC1.C1(O)CC1 N1(C(C2(C)CCOCC2)=O)CCC2(CC2C(=O)NCC2CCCC2)C1 N1(C(CC(C)n2cccc2)=O)CC(C2(NC(=O)CCCc3cc[nH]n3)CC2)C1 C1(NC(C(c2cccc(OC)c2)O)=O)CC2CCC1N(C(=O)C(C)C(C)O)C2 c1(NC(C2CC2C(N2C(C)C(O)CCC2)=O)=O)cccc2c1OC(F)(F)O2 C(CC(C(C)(C)C)NC(=O)C(C)C)NC(C(CCSC)OC)=O.N12CCCC1C2 c1(OC(CC)C(=O)NCCNC(=O)CCCN2CCCC2)ccccc1F c1(C(=O)NC(CCC)C2CC2)cccnc1CNC(C1(N(C)C)CC1)=O C#CCC(C(=O)N1C=CCCC1C(=O)N(CCF)C(C)C)C1CC1 c1(C(N2C(CC)CN(C(=O)C(CO)OC)CC2)=O)cccc2cnnc(O)c12 N1(C(C(COCC)NC(c2n[nH]c(C)c2O)=O)=O)CC2CCC(C1)C2O C(=O)(C(C)(C)CCCF)NC(CCN(C)C(C1CCCCC1O)=O)C(C)(C)C CCCC(C#N)C(=O)N1CC(OC)C(C(=O)NCC(C)(C)CC)C1 c1(CC)ccc(OC)c(C(=O)N(C2CCNCC23CC3)C)c1.C1(=O)CCO1 C1(NC(C23OC(C)C(C2)C3)=O)COCCN(C(C2(C#N)CC2)=O)C1 c1(SC)cccc(F)c1C(=O)NCC(O)CNC(C1CC12CCOC2)=O Cc1cnc2cc(C(=O)NC3CN(C(c4cncnc4)=O)CCC3(C)C)nn2c1 c1(NC(=O)Nc2ccc(F)nc2F)ccc(Br)nc1I.C12CN(CCO1)C2=O Cc1c[nH]nc1CNC(=O)CC1CCCN1C(=O)CCCc1nccs1 CCC(C)CCC(=O)N1CCC(C(=O)NCCCCC2CC2)O1 C1(C(N(C2CCCC2)CCNC(C(C)(C)C2CCC2)=O)=O)CC(F)(F)C1(F)F C=CC(C)(C)CC(=O)NC12CC(NC(=O)Cn3ccc(Br)n3)(C1)C2 C(c1cncc(C)c1)=CC(N1CCC(CNC(CCSCC)=O)(CO)C1)=O N1(C(CC(C)(C)C#N)=O)CCC(C2CN(C(c3cc(Br)cnc3N)=O)C2)CC1 N1(C(C(C)N(C(C2(CC#C)CC2)=O)C)=O)CCC2(COC(C)C2)C1 c1(C(=O)NCC(C)CNC(c2ccc(C(C)(F)F)cc2)=O)cc(O)c(F)cc1N c1(C(=O)NC(CCNC(C(C)=C2CC2)=O)C)cc2cccc([N+](=O)[O-])c2[nH]1 C(=O)(C(C)(C)C(=O)NC)NC(c1cn(Cc2ccc(C(=O)OCC)cc2)nn1)C N1(C(c2ccc(C(C)C)nc2)=O)C2CCCC1CN(C(c1cnc(S)nc1)=O)C2 c1(CC(=O)NCCCCC(=O)NCc2ccc(C#C)cn2)cc2ccccc2[nH]1 C1(C(N2CCCC(OCCC)C2)=O)CC(C)(C)CN1C(C1OCCC1CC)=O C1(C)(NC(c2[nH]cc(CC)c2)=O)CCN(C(=O)C(O)CN2CCOCC2)C1 O=C(C(c1ccoc1)NC(C1CC12CCC2)=O)NOCc1nc[nH]n1 C=CCCCCCC(=O)NCC1(F)CCCN(C(c2cnc(=N)[nH]c2)=O)C1 C12(C(N(CCNC(CC3C(C)(C)CCO3)=O)C3CC3)=O)CC1COC2(C)C Cc1ccc(F)c(OCC(=O)NC(CO)CCCCNC(C23CCCC2C3)=O)c1 C1(C(N(C(C)CC2CC2)C)=O)C(C)CCN1C(=O)CCc1ncnn1C C1(C(c2nc(CC3CCCC3(F)F)n(-c3ccccc3)n2)=O)COC2(CCC2)CN1 c1(C(=O)NC(CC(C)NC(=O)C(C)(C)C2CCC2)C)cc2c(F)c(Cl)ccc2[nH]1 C1(C2N(CCCC(C)N3CCCC3)CCC2)CCN(C(=O)OC(C)(C)C)CC1 n1(CC)nnc2c1CCC(C(=O)NCC(C)NC(C1CCC(C)CC1)=O)C2 C1(C(=O)NC(CNC(C2(OC(C)C)CCC2)=O)C2CC2)CCCNS1(=O)=O c1(OC)ccc(C(=O)CCC(=O)NCCCC(C)(C)NC(=O)C#CC2CC2)cc1 C12(CNC(Cc3[nH]c(=N)sc3)=O)CCC1CN(C(C1CC(O)C1)=O)C2 c1(C(=O)NCC2(F)CCCN(C(CN(C)CCO)=O)C2)nccn2nccc12 CC(C)CC(CN(C)C)CC(=O)N(C1CC(C)CC(C)C1)CCCOC1CCOC1 CC1CCc2sc(C(=O)N(CC(C)NC(c3c[nH]c(Br)c3)=O)C)cc2C1 c1(C(=O)NCC(C2(C(=O)NCCSCC(C)C)CC2)OC)cnc(Cl)s1 N1(C(C2(CC)CCNC2=O)=O)CC2CCC1CN2C(C1CC2C(C1)C2(F)F)=O C(CCCCC(=O)N1CCC1CC(=O)NC(c1nnnn1C)C)OCC C1(C(=O)NC2CC(NC(=O)CSC3CCOC3)C2)(CO)CC1(F)F C1(NC(C2(OC(C)C)CCC2)=O)CC2CCC(C1)N2C(=O)C(C)(C)c1cscn1 c1(N2C(CNC(c3ccc(C)[nH]3)=O)CC(F)(F)C2)ccc([N+](=O)[O-])cc1 CC1CC1C1CC1C(=O)NCC1COCC1NC(=O)C(N)=O c1(C(N2CC(Cc3cn(CCOCCO)nn3)C2)=O)cnn2ccccc12 CCCCC(C(=O)NCC1CC(COC)C1)NC(=O)C(CO)N(C)C(=O)OC N1(C(c2ccc(C)c(O)n2)=O)CCC2CC2(NC(c2cnc(C(C)C)s2)=O)CC1 c1(C(C)(C)C)nnc(CC(=O)NCC2(NC(=O)CNC(N)=O)CC2)o1 N1(C(C(C)=C(C)C)=O)CCC(C(=O)NOCC(O)CO)C1C c1(C(=O)OC)cnc(N2CC(CC(C)NC(c3cnc(C)[nH]3)=O)C2)c(C)c1 C=CCCC(C)C(C)NCCN1CCN(CCNS(C)(=O)=O)CC1 n1(C(CC)C)nc(C(=O)NCC2CCCN(C(C3(C)CCC3)=O)C2)cc1C C1(NC(c2nc(C(C)NC(=O)CCN3CCCC3=O)oc2)=O)C=CC(C)(C)CC1 c1(C(=O)NC2CCC(C(=O)Nc3ncc(I)nc3Cl)C2)ccc([N+](=O)[O-])c(F)c1 C=C1CC(CC(=O)NC2(CNC(C3CC(CCO)C3)=O)CCC2)C1 c1(C(=O)NCCN(CC(C)O)C(C2CC(N=[N+]=[N-])C2)=O)cccc2c1OCCO2 c1(CNc2cc(NC(c3scc(C)n3)C)ncn2)cccc2nsnc12 C12(C(N3C(C)C(NC(C4CC4F)=O)CCC3)=O)CCC(N=[N+]=[N-])C1C2 c1(C(N2CC3C(NC(CCOCCOC)=O)(C3)C2)=O)ccc2cnnn2c1.C1CC1 c1(C(=O)NC(CNC(C(CSC)O)=O)C(C)C)cc(S(C)(=O)=O)ccc1Cl c1(C(=O)Nc2nc(C)cnc2NCC2CCCN2CC)cccc2cnccc12 N1(C2CN(C(c3coc(Cl)c3)=O)C2)CC(NC(C2CCC(=O)N2)=O)CC1=O C#CC1(NC(=O)C(CC)NC(C2CC2C(=O)OCC)=O)CC2CCCC12 C12(CNC(=O)CCNc3ccccn3)CCC1CN(C(c1cc(F)c[nH]1)=O)C2 c1(OCCC(=O)NC2C(NC(=O)CSCC(F)(F)F)C2)ccc2ccccc2c1 C12CCC(CC1)NC2=O.CC1(OCC(=O)NC2CCC2C(C)(C)C)CCCC1 c1(NC(CCC2N(C(c3cc(C)oc3C)=O)CCCC2)=O)ccc(C#N)c(O)c1 c1(COC)cncc(C(=O)N(CCCC(=O)NCCCOCC(F)F)C)c1 N1(C(C2(F)CN(C(C3CNC(=O)N3)=O)C2)=O)CCC(C2CC2)CC1 c12c(cc(Cl)cc1Cl)N(C=O)C2.C(C(COC)C(C)C)OC c12ccc(C(C)C)cc1C(=O)N2.C1(OC)COCC1NCc1ccc(C(C)(C)C)s1 c1(CCCNCc2ccc(OCCOCC)cc2)cc(OC)c(O)c(N)c1 C12(NC(c3nc(C)sc3)=O)CCN(C(c3cn(C(F)F)c(C)n3)=O)CC1C2 N1(C(C(C)N(C(C)=O)C)=O)CC(CNC(c2ncoc2C)=O)CC1(C)C n1(C(C)C)cc([N+](=O)[O-])c(=NCc2ccc(-c3ccc(C=O)o3)cc2C)[nH]1 C1(C(=O)Nc2cn(CC(=O)NCC(c3ccncc3)C)nc2)CCCC(CF)C1 CC1(F)CN(C(c2ccncc2Br)=O)CCN(C(C2CCC23CCC3)=O)C1 C1(C(=O)NC(CC=C)C(=O)OC)CC2(CCC2)CN1C(C1CCCCO1)=O C1(NC(C(C=C=C)C)=O)CC2CCC1(C(=O)NOCc1ccnc(OC)n1)C2 CC(C)C(O)C(=O)NCC(C1CCCC1)NC(c1cccc(C2CCCC2)n1)=O C12(NC(c3nn(C(CC)C)c(C)c3)=O)CCCN(C(=O)CCOC(C)C)CC1C2 C1(NC(C(C)SC(F)(F)F)=O)CCC2CN(C(C3(C)CC3(F)F)=O)CC2C1 N1(C(CS(C(C)C)(=O)=O)=O)CCC2C(CCN2C(c2cc(Cl)cn2C)=O)C1 N1(C(C=NOC)=O)CCCC(C2CCN(C(c3coc(C#N)c3)=O)CC2)C1 C(=O)(C1=CCCCC1C)N.Cc1cc(C)n(CC(=O)NCCC2COCCN2C)n1 Cn1nc(C(=O)NC2COCCC2NC(C2CCC3(CCC3)O2)=O)c2c1CCC2 S(=O)(=O)(c1ccc(C(N2CCN(C)CC2C)=O)cc1)NCCC#C N1(C(C=NOC)=O)CC(CNC(C2(C)C=CCCC2)=O)OC2COCC12 c1(C(=O)NC2(CC=C)CCN(C(CCCC#CC)=O)C2)coc2ccc(F)cc12 C1(NC(C2CCS2(=O)=O)=O)CCN(C(=O)COc2cccc(F)c2)C12CC2 C1(C(=O)NC(C(=O)NCCC)C)(NC(c2nnn(C)c2N)=O)CCOCC1 N1(C(c2cc(-c3ccc(C)s3)[nH]n2)=O)CC(CNC(=O)C(C)CF)C(C)(C)C1 c1(C(=O)NCC(CO)NC(=O)CCC2CCCCO2)ccc(-n2cncn2)cn1 CCCCCC(CC)NC(=O)NCCCC1(CS(C)(=O)=O)CC1 C(=O)(C(F)(F)C1(OC)CCCC1)NCCC(C)NC(C1(COCC)CCC1)=O c1(CN2C(C(=O)Nc3cc(F)cnc3Cl)C=CC2)c(Cl)c[nH]c2nccc1-2 C1(C2CC2)(CNC(c2c(CCC)onc2C)=O)CCN(C(=O)CCC(C)OC)C1 c1(NC(=O)NCCN2CCOC(C3CC3(F)F)C2)ncnc2sccc12 N1(C(C(CC=C)OC)=O)CC(CNC(c2ccncc2N(C)C)=O)CC1(C)C C1(CC2(C(=O)Oc3ccc(C=C)cc3)CC3(CC3)C2)CCCCC(F)(F)C1 N1(C(C(C)C2CC2)=O)CCCN(C(=O)CS(=O)(=O)Cc2cccs2)CC1CO Cc1ccnc(C(=O)NC(C)C=CC(=O)NC2(CO)CCC(C)C2)c1 Cc1cc(C(N2CCCCC2CNCCCN(S(C)(=O)=O)C)=O)nc(C)c1C#N CCC(CCC(=O)Nc1ccc(F)cc1CO)NC(=O)CCCn1cccc1 C1(CC=C)(NC(=O)CNC(=O)C(C)(C)C)CCN(C(c2ncoc2C(C)C)=O)C1 c1(N(C2CCCN(C(C(C)Cn3ccnc3)=O)C2)CCO)nc(C#N)c(Cl)s1 C(=O)(CC(C)n1ccc(C)n1)N1CC(C(=O)NC(CCNC(C)=O)=O)C1 C1(F)(NC(CNC23CC(C)C2C3)=O)CCCN(C(=O)CCn2ccccc2=O)C1 N1(C(C2(C=C)CCOCC2)=O)Cc2cc(O)ccc2C(C(=O)O)C1 C1(CCNC(CCOC)=O)CCN(C)C(=O)O1.c12cn(nn1)C1(CC1)C(=O)N2 c1(CC23CC(C(N4CCC(N(C(CC(C)O)=O)CC)C4)=O)(C2)C3)cccc(Cl)c1 CC1CN(C(=O)COc2cccc(Cl)c2)CC1NC(c1n[nH]cc1Br)=O C1(C)(CC(=O)NC(CCNC(c2c(CC)nn(C)c2)=O)C)CCCCCC1 N1(C(CC2CCC(C)C2)=O)C2CCC1CN(C(c1cnc3n1CCCC3)=O)C2 N12C(=O)CCN(C1=O)Cc1c(nccc1)C2.N1(C(N)=O)CC(COC(C)(C)C)C1 C(=O)(CCCCC(=O)NCC(C1CC1)N(C)C(C1CC(F)C(=O)N1C)=O)NC c1(C(N2CC(OC)C(NC(c3ccc(C)s3)=O)C2)=O)ccc(F)c(O)c1 CC(CNC(=O)CNC(=O)CNC(=O)CCc1cnn(C)c1)C(C)(F)F Cn1cc2c(n1)CCCC2C(=O)NCC(O)CCNC(=O)C(C)(C)C(N)=O c1(C(C(c2cccc(Br)c2)(C)OC)=O)ncnc2nc(N3CCOCC3)sc12 CC1(C(N2CCCC(CNC(c3cc(C(F)(F)F)no3)=O)C2)=O)CS(=O)(=O)C1 C(=O)(CC1=CCCCC1)N(CC(C)C(=O)NCCC(=O)NCCF)C N1(C(c2cc(C(=O)OC)on2)=O)CC2CCCC1CN(C(=O)CCCC(F)(F)F)C2 N1(C(c2c(Br)c(C(F)(F)F)nn2C)=O)CCC(OC2CC2)C(F)(F)C1 O=C(CCCC(F)F)NC1CCN(C(=O)C(c2cc(Cl)ccc2Cl)(F)F)C1 N1(C(C)C)CCCC(N=c2[nH]c(N3CCC(F)(F)C(F)C3)nc3cc[nH]c23)CC1 O=C(CC1OCCc2ccccc21)N1CC(NC(C23CCC(CC2)CO3)=O)C1 n1(CC(=O)N(CC(C(=O)NCCC(C)OC)C)C)cccnc1=O c1(C(=O)NC2CN(C(C(CC=C)(F)F)=O)CC2F)cc2n(n1)CC(F)C2 c1(CC)cc(C(=O)NC2CCCCC2NC(C2(CO)CCOCC2)=O)n(C)n1 c1(C(N2CCN(C(CCCCC)=O)C(CC3CC3)C2)=O)cn2c(n1)CC(C)CC2 Cc1nn2c(C(N3CC4(C3)CN(C(=O)C3=CCC3)CC4CO)=O)c(C)nc2s1 c1(CNC(c2c(C)cno2)=O)ccc2c(c1)CCC2NC(c1ccccc1Cl)=O N1(C(CNC(c2cc(C)c(C)nn2)=O)=O)CC(C)(C)OC(C)(C)C1 c1(C(=O)NC2CC(NC(C(C)(C)OC(C)C)=O)C2)ccc(F)c2ncccc12 C1(OC)CN(C(=O)C(C(C)C)SC)CC1NC(c1nocc1C(C)(C)C)=O c1(C(N2C(C(=O)NC(C(C)C)C)CC(=O)C2)=O)cccc(O)c1F C(N=c1[nH]c2cc(F)ccc2o1)C1C(NC(c2cscn2)=O)C2(CC1)CCC2 N1(N(C2CC23CC(NC(=O)C(F)(F)C2CC2)C3)C)C2CCCC1CN(C)C2.C=O Cc1cc(Cl)nc(N)c1C(=O)NC1CC1NC(c1cccc(CS(C)(=O)=O)c1)=O C(C(CNC(c1coc(-c2ccccc2)c1)=O)CO)NC(C(C)NC=O)=O C1(CNC(c2cn(CC)nc2C(C)C)=O)CCC(C)CN1C(=O)Cc1ccsc1 C(C(F)(F)F)CCN(CCN(C)C)C(C1CN(C2CCC2)C1)=O c1(OC)cc(C(N2CCC(CN=[N+]=[N-])CC2)C(=O)NC2CC2)c(F)cc1Br C1(C(N2CCC(N3CC(O)C3)C2)=O)CCCOCC1.C12(CCC1)C(=O)NC2 CN1CCC(NC(c2cc(CNC(c3cc(Cl)no3)=O)no2)=O)CC1 C=CC(C)(CCOC)C(=O)NCc1ncoc1C1CN(C(C2CC2CF)=O)C1 c1(-n2cc(CC3CCN(C(C4COCOC4)=O)C3)nn2)ccc(Br)cc1 c1(SC)ccc(Cl)c(C(N2CC(CC(C)NC(=O)CNC(=O)C3CC3)C2)=O)c1 Cn1cc2c(n1)CC(C(=O)N(CCNC(C1(C3CCCO3)CC1)=O)C1CC1)CC2 Cc1cccc(C(O)C(=O)NCC2CC(NC(c3cccc[n+]3[O-])=O)C2)c1F Cc1ccccc1C(=O)NC(Cc1ccco1)C(N1CCC(CC(C)O)CC1)=O CN1CCC(NC(=O)C2=CCC(NC(C3CN(C(N)=O)C3)=O)C2)C(C)(C)C1 c1(NC(C(=O)NCC2CC3CCC2CC3)=O)cc2c(cc1Cl)OCCO2 c1(C(=O)NC2CC(NC(c3n(CCC)ccn3)=O)C2)ccnc(C)c1O c1(C(N(C)CC2N(C(C(C3CCOC3)OCC)=O)CCC2)=O)cc(C2CC2)n(C)n1 C1(C(=O)NCC2=NOC(C)C2)CCN(C(c2cccc3occc23)=O)C12CCC2 N1(C(CCCS(C)(=O)=O)=O)CC2CC(NC(=O)C=Cc3cscn3)CC(C2)C1 c1(C(=O)NCC(C(C)C)NC(c2ccc(C3CCC3)nc2)=O)cc(Cl)cnc1O C12(C(=O)NCCCC3CC(NC(=O)C(O)CC4CCCC4)C3)CCC(CC1)CO2 c1(CCC)nnsc1C(N1CCCC1C1CCOC1)C(=O)NCCCSC C1(C(=O)NC2CCC(F)(F)C2)CCCN(C(=O)CCn2cccn2)CC1 c1(C(=O)NCC(CCC)NC(=O)CCC(C)(C)C)cc([N+](=O)[O-])c(C)s1 C1(C(=O)NCC(CNC(C(C2CCCCCC2)C)=O)O)C(C)(C)C1(C)C c1(C(N2CC(C)C(CNC(C3CCCOC3)=O)C2)=O)cc(F)ccc1S(C)(=O)=O c1(C(=O)NCCN(CCOC)C(C2C3CCN2CC3)=O)scc(C)c1C c1(CC)nnc(NC(=O)CCC2OCCO2)s1 Cc1nn(C)c(Cl)c1C=CC(=O)NCC1CN(C(c2ccncc2F)=O)CCO1 Cc1c(C(=O)NCC(C)CNC(=O)C(F)CC2CCOC2)[nH]c2cc(F)ccc12 c1(NCC=C(C)C)nc(=NCc2ccnc(C)c2)[nH]c2c(C)nn(C)c12 c1(C(N2C3CC(NC(C4N(CC)CCCC4)=O)C(C3)C2)=O)cccc([N+](=O)[O-])c1 c1(C(c2c(C(=O)OC)nc[nH]2)NC(C)CC)ccccc1F.C12CC1C(=O)N2 c1(C(=O)NCC2C(NC(c3c(CC)oc(C)c3)=O)C2)cc2c(F)ccc(F)c2s1 c1(C(=O)NC(CC(C)C)CNC(C2CCCC2CF)=O)cc2cccnc2cn1 N1(C(Cc2nnc(C)s2)=O)CCC(NC(C2CC23CCC3)=O)C1C N1(C(c2c(C)[nH]nc2Cl)=O)CCCC2(C1)C(NC(c1cn(C)nn1)=O)CCN2C N1(c2cc(S(=O)(=O)NCCC(C)F)cc(Cl)n2)CCOc2ccccc2C1C Cc1cc2c(cc1C(N1CCC3CN(C(=O)CC#N)CC3C1)=O)OCCCO2 C1(C#CC(=O)N2CC(CNC(=O)CN3CCOCC3)(OC)C2)(CC)CC1 C1(NC(c2cnoc2)=O)CN(C(C2CCCC23CC3)=O)CC2(CCC2)C1 C(CC)(CCC(=O)NCCC(C)C(F)F)NC(CC=C=C)=O C(C1CCC(C)CC1)=CC(=O)N(CC(CNC(C=C(C)C)=O)O)C C(=O)(CCC(C)S(C)(=O)=O)N1CC2CN(C(c3cc(C)n(C(F)F)n3)=O)CC2C1 CC(C)C1=NOC(C(=O)N(CCC(=O)N(C)C)CCO)C1.C1(C)C(=O)N1.OCC c1(OC)cccc(F)c1N(C)C(c1csc(C2OCCO2)c1)=O N1(CC(=O)NCC(C)(C2CCC2)NC(C(C)NC(C)=O)=O)CC(=O)NC1=O CC(C)(CNC(=O)CCC1CCCC1)CC(=O)NCCC(O)C(F)(F)F N1(C(CCOCC(C)C)=O)CCN(C(c2nnc(Cl)cc2N)=O)CC(C)(C)C1 C1(c2ccccc2)(C(N(C(C)CNC(c2[nH]nnc2C)=O)CC)=O)CCCC1 N1(C(Cc2c(CC)con2)=O)CCC2(CC1)CC2NC(=O)CC1CSCCS1 C(=O)(CCCCCN=[N+]=[N-])N1C2(CNC(C(CN(C)C)(C)C)=O)CCCC2CC1 Cc1cccn2c(C(N3CCCC3C3CCC3)=O)ccc12 c1(C(N2CC(C(C)NC(COC(CC)C)=O)C2)=O)c[nH]c2cc([N+](=O)[O-])ccc12 N(C(=NCCOC(C)C)NC1CCCOC1)C(COC)C1CC1 CC(C)C(C#N)CS(=O)Cc1ccc(F)cc1Br c1(NCCc2ccc(OC)cc2Cl)ccc(S(=O)(=O)NCc2cncnc2)cn1 Cc1nc(C(=O)NCCC2(NC(=O)C(C3CCOCC3)C)CCCC2)cc(O)n1 c1(C(=O)NC2C=CCN(C(c3ccc(C#C)cc3)=O)C2)ccc2nc(O)[nH]c2n1 Cc1cc(=O)oc(C)c1C(=O)NC(C)C(C(C)C)NC(=O)CC1(O)CCCC1 C(=O)(CC(C(F)F)NC(=O)CCCCCn1cc(C(C)(C)SC)nn1)OC n1(CC(=O)NCC2(CN(C(C(CC)COC)=O)C)CC2)ccc(C)cc1=O c1(CCNC(C2C(=C)C2)=O)ocnc1CNC(c1cnn(CCC)c1)=O N1(C(CC(C)N(C)C)=O)CCC(OC2CN(C(C3CC4C=CC3C4)=O)C2)CC1 Cc1nn(C(F)F)c(C)c1C(=O)NC(=O)N(CC(C)(C)C)CCO N1(C(C(C)=O)=O)CC(NC(C2CC3(C2)CC3(F)F)=O)CC(C)(C)C1 Cc1nc(O)sc1C(=O)NCC(C)(C)OCCC(=O)NCC(F)C1CCC1 C1(CNC(c2ccc(SC)cc2)=O)CC2CCC1N(C(=O)C=CC(C)=O)C2 Cc1cc(CCC(=O)NCC(C)CNC(c2cc(CN(C)C)on2)=O)on1 C(=O)(CC1=NNC(=O)C1)NCC(C)(CO)NC(C(=CC1CCCC1)C)=O C(=O)(C(F)C(C)CNC(C1OCCCC1(C)C)=O)NC(CCN(CC)CC)C C(CC(C(=O)NC1(CNC(c2nn(C)cc2Cl)=O)CCCC1)NC(N)=O)SCC Cn1cc(C(N2CC3(CC3)CC2CNC(C2CNC(=O)C2)=O)=O)c(O)nc1=O N1(C(=O)COC2CCCN2C(=O)CC2CCC=CCC2)CCC12CCCCC2 C1(NC(CCCC=C)=O)CN(C(c2c[nH]cc(C)c2=O)=O)C(C)(CC)C1 c1(C(=O)NCC(CN(C)C(C2CCCCC2O)=O)(C)C)cc(N)c(Cl)c(O)c1 N1(C(c2ccc(C)[nH]2)=O)CC(C(=O)N(C2CCN(C)C2=O)C)CC1(C)C c1(C(N(C2(CNC(c3nccs3)=O)CC2)C)=O)c(F)ccc(F)c1Cl CCCCC(C)CCC(=O)NC1CCC(CC(=O)NC2CC(C)CC(C)(C)C2)C1 CC1CCN(C(=O)C=CC(=O)NCCC(C)NC(c2nccn2C)=O)CC1 C1(C)(C(=O)NCCN(C(C2CC3(CO)CC2C3)=O)CC)CCCC1O c1(C(=O)NC(CN(C(=O)CC2CCCOCC2)CC)C)ncccc1Br C123CN(C1COC2)C3=O.C1(CN(CCO)CC)CC(F)CN1C C#Cc1ccc(CNC(=O)CC2C=CC(NC(C3CCC4CC34)=O)C2)cc1 CC1CC(C(=O)NC2COCCN(Cc3cccnc3)C2)CCN1C n1(C(C(=O)N(C2CN(C(=O)Cc3ccc(Cl)s3)CC2F)C)(C)C)cc([N+](=O)[O-])cn1 Nc1ccc(F)c(C(=O)NC2CCC(NC(c3ccc(F)cn3)=O)CC2)c1F C1(CNC(c2c(CC)nco2)=O)CCCN(Cc2[nH]c(C)nc2-c2nn[nH]n2)C1 C(=O)(C1=CC2CCC=CCCC12)NCCCC(C)NC(C1(CC)CCCC1)=O C12(NC(C(C(C)C)C)=O)CCCC1CN(C(c1ccn(CCF)n1)=O)C2 CC1(O)CCN(C(C2CC(N)C23CCC3)=O)CC1O n1(CC(=O)NCCC(C)NC(C(CC)F)=O)nc2n(c1=O)CCCC2 N1(C(C=CC(C)(C)C)=O)CC2(CC1CNC(c1ccn3ccnc3n1)=O)CC2(F)F c1(NCCCNC2CCN(CCOC)C2)cc(=NCCOC)[nH]c(C(F)(F)F)n1 c1(CC(=O)NC(C)CCNC(C2CC2c2ccncc2)=O)cccnc1O CCCC(C(=O)N1CC(n2cc(CC(=O)Nc3ccccn3)nn2)C1)NC(C)=O CC1CC(NC(c2sccc2F)=O)CN1C(c1ccc(SC(F)(F)F)o1)=O c1(COC)cncc(C(=O)N(CCC(=O)Nc2ccncc2SC)C(C)C)c1 CC(CNC(c1n[nH]cc1CNC(=O)C(C)(Cl)Cl)=O)CC(F)(F)F c1(CCC(=O)NC2CC(NC(CN3C(C)CC3)=O)C2)ccc(S(N)(=O)=O)cc1 S(=O)(=O)(c1[nH]c(=NCCC2(CO)CCC2)ccc1Br)N(C)CC1C(C)CCCC1 CN1CCN(C(=O)CC2CCCNC2=O)C(C(N2CCCN(C3CC3)CC2)=O)C1 C1(C)(NC(C(COCC)C)=O)CCCN(c2nccc(SC)n2)C1 c1(C(=O)NC(CC(C)NC(c2ccc(C#N)c(F)c2)=O)C)cc2c(o1)CCCC2 C=CC1CN(C(=O)CC2CCCOCC2)CC1NC(c1cnc(C)cc1C)=O C=CC(C)(CC)C(=O)NCCNC(c1ccccc1SCc1nnn(C)n1)=O Cc1ccncc1CC(=O)NC(C1CCCC1)CNC(=O)Cn1ccnc1C C#Cc1c[nH]nc1C(=O)NC1COCC1C(=O)NC(CC=C)CC=C N1(CCOC)CCC(NC(=O)CCN2CCCCC2C)C(O)C1 c1(NC)ccc(C(=O)NCC2CC(O)CN2C(=O)CC2CCCSC2)cc1 c1(CC)nnc(N(CCCCNC(C2CNC(=O)CC2C)=O)C)c(C#N)c1CC C1(C(=O)NCC2CN(C(C(C)(C)C)=O)CC2C(F)(F)F)CSc2ccccc2O1 N1(C(=O)OC(C)(C)C)CC2CCC(C1)C2C(=O)NC(C1CCCO1)CO C#CC1CC2CCC1N(C(=O)C(C1CC1)N(C)C(C1CC3(CCC3O)C1)=O)C2 Cc1ccnc(C)c1CNC(=NCC1CC12CC2)NCc1ccc(Br)cc1F C(=O)(CCN=C(NCC(CO)C(F)(F)F)NCC(c1nc(C)cc(O)n1)(C)C)NC N1(C(C2(CC)CC2)=O)CCCC(CC(=O)NCC2CCCCC2)CC1 C1(C(N(C2CCCCCC2)C)=O)CC2(C1)CC1(CNC1)C2 C=CCC(CNC(c1nonc1N)=O)C(=O)NC1CC2C=CC1C2 C#CCC(CC(F)F)N=c1[nH]c2c(c(=NCCN(C)CC)[nH]1)COCC2 C1(CC)C(CC(=O)NCCCN(C(=O)C(C)NC(=O)CC)CC)C1(F)F Cc1[nH]c(C#N)cc1C(N1CCOCC1CCNC(c1cnc(Br)s1)=O)=O C(=O)(C(O)C(C)CC)N(C1CCN(C(c2n[nH]cc2C)=O)CC1)CC#C c1(C(=O)NC2C(CNC(C(C)(C)OC(C)C)=O)C2)ccc(O)cc1Cl C1(CC=C)(NC(=O)C(C(C)O)N(C)C)CCCN(C(C2CCCOC2C)=O)C1 N1(C(COCCCCC)=O)CCCC(NC(C2(CSC)CC2)=O)C(F)C1 N1(C(CC2(N(C)C)CCCC2)=O)CC(O)(C2(CNC(=O)Cc3cc[nH]n3)CC2)C1 N1(C(c2nc(C)n(C)c2)=O)CC(CNC(C2(C)CCCCO2)=O)OC(C)(C)C1 N1(C(CCCC=C)=O)CCOC(C)C1C(=O)NC1C(C)(C)C1(C)C C1(NC(c2ccc(CC)o2)=O)CCN(C(=O)Cc2ccn(C(C)C)n2)CC1(C)C c1(C(=O)NC2C(NC(c3scc(COC)c3)=O)CCC2)cc2cc(Cl)ccn2n1 Cc1cc(C(N2CCC(O)(CCNC(=O)CCc3nc(=N)[nH][nH]3)C2)=O)sc1C C1(C(N2CCC(CC#N)(CC)C2)=O)C2CCCC2CN1C(=O)CCNC(=O)OC C1(NC(C2C(NC(c3ccc(O)nc3)=O)CCO2)=O)C2C=CC(C2)C1CO c1(C(=O)NCC(C)(C2CC2)NC(c2cc(SC)nn2C)=O)cn2ccsc2n1 C(=O)(C1=CCc2ccccc21)N1CC(NC(c2c(C)[nH]nc2Cl)=O)CC12CCC2 c1(C(=O)NCC2(F)CN(C(C3(C)CC3F)=O)C2)cc2n(n1)CCNS2(=O)=O N1(C(CCc2cccc(C)n2)=O)CCC2(CC2NC(c2cccc(F)c2C)=O)C1 C(=O)(CS(=O)(=O)CCO)N1CC(CCNC(C2C(CC)C2)=O)C(C)C1 c1(C(=O)NC(CNC(=O)CC2COC(=O)C2)CO)ccc2nc(O)oc2c1 C1(CNC(C(CC#C)O)=O)CCN(C(c2ccc(F)cc2SC)=O)C12CC2 CCC(C(=O)N1CCC(C)C(NC(=O)CNS(C)(=O)=O)C1)C(C)O C(=O)(C(CC(C)C)C(C)C)N1CC(C(=O)NC(CC#C)C)(Sc2ccccc2)C1 C#CC1(C(=O)NOC2CCCN(C(=O)CC(=O)OC(C)(C)C)C2)CCCCC1 O=C(CCC(=O)c1ccncc1)NCCCC1CCCCN1C(=O)C(F)C1CC1 C(=O)(C(C(C)(C)C)NC(=O)C(C)CCOC)NCC(CC)(C)CO Cc1cccc(C(N2CC(C(=O)NCCN3CCCC3=O)C3(CC3)C2)=O)c1C#N N1(C(C(CC#C)C)=O)CCC2CN(C(=O)C=CCN(CC(F)(F)F)C)CC2C1 C1(CC(=O)NCC2(F)CC(CNC(C(=O)NCC3CC3)=O)C2)CCC2(CC2)CO1 C1(CC(=O)N(CCC(C(C)C)NC(=O)C(C)(F)F)C)CC(O)C12CCC2 C1(N(C(c2ccnn2C)C(=O)NCCC2CC2)CC(C)C)CCCC(C)C1 c1(C(N2CCN(C(CNC(CCSC)=O)C)CC2)=O)cnc2ccnn2c1 N1(C(C=Cc2cnc(C)s2)=O)CC(C)CN(C(C2CCSCC2)=O)CC1C C1(C2CCCN(C(c3cc(C(N)=O)co3)=O)C2)(NC(C(CC(C)C)(C)O)=O)CC1 C1(C)(CCC(=O)NCCOCC)CCCN1C(c1oc(CO)cc1C)=O C1(CC(=O)NCCCN2C(C)CCC2)C2CCC(C2)N1C(C1CCOC1)=O c1(OC)cnc(C(=O)NCCN(C(=O)CC2CCCCC2C)CCOC)nc1 C=CC(C)(CC)C(=O)N1CC(F)(CNC(c2ccc(CNC(C)=O)c(F)c2)=O)C1 C12(NC(C3C4CC4C4CC34)=O)CCC(CC1)N(C(=O)CS(=O)(=O)CC1CCCO1)C2 c1(C(=O)NC(C)CN(C)C(C2CCCCN2C)=O)cccc2c1NCCNC2=O Cc1cc2ncc(C(N3CCCCC3Cc3cn(CCCF)nn3)=O)c(C)n2n1 CC(O)(CC(=O)NC1(CNC(C2(C3CCCO3)CCC2)=O)CCCC1)C(F)(F)F Cc1cc(CNC(=O)C(CC(C)C)N(C(=O)CCCCNC(N)=O)C)cc(C)c1 N1(C(c2c(C)nc(CCC)s2)=O)CCCN(C(=O)CC(F)(F)C(F)F)C(C)C1 N1(C(CC2CC(=C)C2)=O)CC2CC(NC(=O)C(C)(C)COCCC)CC(C2)C1 c1(C(N(C2CCN(C(=O)CN3CCOCC3)C2)C)=O)sc2cccc(F)c2c1Cl C(=O)(CCCCN1CCOCC1)NCC1N(C(CCOCC(C)C)=O)CC1 c1(C(CNC(c2snnc2C)=O)NC(CNS(NC)(=O)=O)=O)ccccc1F C1(NC(c2cnn(C)n2)=O)CN(c2nc(C(N)=O)ns2)CC2(CCOCC2)C1 C(CC1=CCN(C(=O)CSc2ccccn2)CC1)NC(c1c(CC)oc(C)c1)=O N1(C(CSC)=O)CCOC(CCNC(c2csc(-c3cnccc3C)n2)=O)C1 CCCC(=O)NCCNC(=O)C(C)C1(N(C(=O)OC(C)(C)C)C2CC2)CC1 CCCC(C(=O)OCc1ccc(OC)c(OC)c1)C(=O)OC C1(C)(C(=O)NCCCCCOC)CC(O)CN1C(c1cc(O)ncn1)=O c1(C(=O)NC2CN(Cc3c(C)cc(O)cc3)CC2C#N)cc(Cl)c(Cl)c(Cl)c1 C1(C(N2CC(F)(CNC(C3(O)CCCC3)=O)C2)=O)CC(C2CC2)=NO1 c1(CN2CCN(C(=O)NC(C(=O)OCC)C)CC2)cc(Cl)cc(I)c1 C1(CNC(CN(CCC#C)C)=O)CC(C)CN(C(C2CC3CCC2O3)=O)C1 C(=O)(C(C)C(O)C(C)C)N1C2C(N(C(c3[nH]cc(OC)c(=O)c3)=O)C)CC(C2)C1 C1(NC(c2c(C)nc(O)[nH]2)=O)CCN(C(C2CC(C(=O)O)C2(C)C)=O)CC1F Cn1ncc(C#N)c1C(=O)NCCOC1CCN(C(c2ccc(Cl)o2)=O)C1 N1(C(c2cnc(CC)o2)=O)CCCC(C2CCN(C(=O)CC3=CCOCC3)C2)C1 N1(C(C2CN(CC(F)F)C2)=O)CC2(C(=O)NCC#CC#CCO)CC1CO2 c1(N(CC)CC)ccccc1C.N12CCN(CC1)CC2=O.C(C)C C(=O)(C(C)(F)C(F)(F)F)NC1CN(C(=O)CC=C(Cl)Cl)CC1C(c1ccccc1)C N(C(=NCCCN1CCC(O)CC1)NCCF)Cc1cn(CC#C)nc1 c1(C(N2CCN(C(C3(C(=O)OC)C4CCC34)=O)C(C)C2)=O)cc2ncccc2o1 c1(CC(=O)NCCC2CN(C(C3SCCCS3)=O)C2)cccc(C(F)(F)F)n1 C(c1ccc([N+](=O)[O-])s1)=CC(=O)N(C1CN(C(c2ccn(C3CC3)n2)=O)C1)C Cc1cncc(C(=O)NCC(CC2CCCC2)C(=O)NCc2cnn(C)c2C)c1 C1(CCNC(C(C)OCCC=C)=O)CCCCN1C(c1nc(Cl)sc1C)=O Cc1nc(C(=O)C(=O)N(CC(O)CNC(C2(CC(C)C)CCC2)=O)C)cs1 C1(C(N(CCCNC(c2ccc(-c3cccs3)o2)=O)CC)=O)CCC2CCC12 c1(CNC(c2cn(CCN(C)C)nc2)=O)ccc(COc2ccccc2N)cc1 C1(C(=O)NC(C2CCN(C(C3CC3F)=O)CC2)(C)C)C(C)(C)C1(F)F C(CCCCC(=O)N1CC(NC(=O)CC2OCCCC2(C)C)C(C)(C)C1)SC N1(C(c2c(C)noc2C(F)F)=O)CCN(C(C2CCC(=O)N2C)=O)CC(O)C1 c1(OC)cc(F)ccc1C(=O)NCCN(C)C1CC1 N1(C(c2c(C)con2)=O)CCN(C(=O)CC(C)c2ccco2)C(C(C)C)C1 CCCCCC(C)CC(=O)NCC1(C)CCCN(Cc2[nH]c(C)c(C(N)=O)c2C)C1 C1(C(N2C(C(CC)O)CCC2)=O)C2CCC(C2)N1C(c1cncc(F)c1)=O C1(C(N)=O)CN(C(c2ccc(C(N)=O)s2)=O)CCC1N=c1nc[nH]c2[nH]c(Cl)cc12 n1(CCNC(C2CC(CCN)C2)=O)cc(Br)c(C)n1.C(C)(C(=O)N)CCCC Cc1nc(-c2nc(C3CCOCC3)nn2Cc2ccsc2)sc1C N1(C(C2(C)CC3CC3C2)=O)CCCC(O)(CNC(=O)C2=CCOCC2)CC1 C(=O)(CCCc1cc[nH]n1)N1C2(CC2)CC1.C=CCCOC(COC)=O N1(CC(C)C)Cc2ccc(NC(c3cccn(CC(C)C)c3=O)=O)cc2C1 c1(C(N2CC(C)(CNC(=O)CCc3ccon3)OCC2)=O)cc(Cl)c(N)cc1F C1(C(=O)NC(C)C=CC(N2CC(CO)(CO)C2)=O)CN2CCN1CC2 Cc1ccc(NC(=O)COC2CC(NC(=O)COC(C(O)CO)C3CC3)C2)n1C C1(CC)CN(C(=O)Cc2cnc(C)o2)CCC1NC(c1cc2n(n1)CCC2)=O CC1(C)C2CCC13CCN1C(C2)N(C=C(Cl)C(C(=O)O)=NN3CCSC)CC1=O N#Cc1cc(CC(=O)NCC2CC3CC3N2C(C2CCC(=O)O2)=O)ccc1F Cc1cc(F)ccc1C(C)NC(c1cc(=N)[nH][nH]1)=O c1(OC)cc(C(N2CCC(CC(N3CCC(C)(O)C3)=O)C2)=O)cc(Br)c1Cl CC1CC2(CCN(C(c3ccc[n+]([O-])c3)=O)CC2)CN1C(C1CC1C(F)F)=O N1(C(C2CC23CCOC3)C(=O)N(C2CCCCC2)C)Cc2cccc(F)c2C1 C(=O)(C1=CCCOC1)NCc1c(C(N(CC(C)(F)F)C)=O)c[nH]n1 C1(CNC(c2c(C)snc2)=O)N(C(=O)C(N2CCNC2=O)C)CCC1(C)C c1(CN(C(C)C)Cc2cc3ccccc3o2)cccc2c1NC(=O)CO2 NS(=O)(=O)CCCC(=O)N1CC(NC(=O)CC2CC2C(F)(F)F)CC(F)C1 C1(CNC(CNC(CCC(C)C)=O)=O)CCCCN(C(C2CCCS2(=O)=O)=O)C1 c1(C(N(C(C)CNC(C2CC2CC(C)C)=O)C)=O)cc(OCC(F)F)cc(F)c1 CC1CCC(CCC(=O)NCC(C)(C)CNC(C2CC(N3CCOCC3)C2)=O)O1 c1(CNC2(C(=O)OC)CC(CO)C2)cc[n+]([O-])cc1 c1(Nc2c(C(=O)NC3C(C(=O)OCC)CCC3)ccs2)ccc(OC)cc1F N1(C(C2CC(SC)C2)=O)CCCC(NC(c2ncn(C)n2)=O)C1C Cc1ccc(C(=O)NC2(CF)CCN(C(c3c(C)coc3CO)=O)C2)c(N)c1C c1(C(=O)NCCC(C)(C)NC(c2n(CC#C)ccc2)=O)cn(C)c(=O)cc1C C12(C(=O)NC(C)CCC(=O)OC(C)(C)C)CCCCC(=O)N1CCC2 CC1(C)CCN(C(=O)Cc2cc(C(F)(F)F)n[nH]2)C(C(=O)NCC2(O)CCCC2)C1 Cc1ncc(CNC(C2CC(C)N(C(c3ncc(F)cn3)=O)C2)=O)n1C C1(C(=O)NCCC=CCCC)(C(=O)Nc2cc(C)[nH]n2)CCCC1C S(=O)(=O)(c1ccc(C#N)cc1NC1CCOCC1)N1CCC(F)(C(=O)OC)C1 n1(CC)nc(C(=O)NC2(C)CN(C(C3(N4CCOCC4)CCC3)=O)C2)c(C)n1 C1(NC(C2ON=C(C)C2)=O)CCOC12CCN(C(c1ccc(C)c(O)c1)=O)CC2 C1(NC(CCC)=O)C2CCN(C(=O)CC3CC3)CCC12 c1(-c2n(CCC)nc(C)c2)ccc(C)n2cc(C(=O)NC3CC3C)nc12 C12(C(=O)NCC(C(C)C)NC(=O)Cc3ccc(Cl)cc3)COC(CC3CC3)(C1)C2 c1(C(=O)NCC(C)CNN)ccc(N)cc1.C(=O)(C(C)OC(=O)SOC)O.C(C)(C1CC1)OC N1(C(CN(C)CCO)=O)CC2CCC(C1)N2C(C1(Sc2ccccc2F)CC1)=O c1(OC)cc(Br)cc2cncc(N3CCCC(C)(F)C3)c12 N1(C(=O)NCC(C)(O)C2CCC2)CCC(C(=O)CONC(=O)NC(C)(C)C)C1 C1(C(=O)NCC2(C)CCC2)CC2CCC(C1)N2C(c1ccc(Br)c(C(F)(F)F)c1)=O Cc1nc(N2CCCC(CCNC(=O)CC(C)(C)O)C2)cc2nncn12 C(CC(C(=O)N1CC(O)(OC(=O)N(C)C)C1)NC(c1cnc(OC)s1)=O)OC CCC(CC(=O)N1CC=CCO1)NC(=O)C(O)CC(C)C N1(C(C(N)=O)=O)CCCC2(CCCN2C(=O)CCCOc2ccccc2)C1 C12(C(N(CCCc3nn[nH]n3)C)=O)CCC1CN(C(=O)CNC(N)=O)C2 CCC1=C(C(=O)NC2(C(=O)NCC3(N(C)C)CCCC3)CC2)SCCO1 S(=O)(=O)(c1cnn2ccc(=NCc3cc(C4CC4)nn3C)[nH]c12)NC(CCC)CC CCCCC(CNC(c1ccc(C2CC2)s1)=O)NC(=O)CNc1cccnc1 N1(C(=O)Cn2ncc(O)nc2=O)CCC2C(C1)CN2C(=O)C(O)C(F)F N1(C(C(C(C)NC(C=CCCC)=O)C)=O)CC2(C1)NC(=O)NC2=O N1(CCN(C)C(C2C3CCCCC23)=O)CCN(C(c2ccncn2)=O)CC1 N1(C(C(=O)NCCCC(C)(C)O)=O)CCC12CCCSC2 c1(NC(c2n(C)ccn2)=O)ccc(=O)n(CCCC(F)(F)F)c1 C1(C(=O)NCC2C(CNC(c3cc[nH]n3)=O)C2(F)F)(OCC)CCOC1 C12(NC(c3c(C)cc(SC)o3)=O)CCCC1N(C(c1[nH]c(O)nc1C)=O)CCC2 C1(CCNC(C2CC3(C2)CS(=O)(=O)C3)=O)CN(C(=O)C(O)C2(Cl)CC2)CCS1(=O)=O C1(C(=O)NCC2CCCSC2)CC(NC(C2(C(=O)OCC)CCCC2)=O)C(O)C1 C1(C(=O)NCc2ccc[nH]2)C=CCN1C(c1cnc(C(F)(F)F)s1)=O c1(C(C)NC(C(CC2CC2)NC(C(COC)(C)OC)=O)=O)ccc(C)c(F)c1 C1(NC(C2CC3CCC3C2)=O)CC2CC(NC(c3cc4c(s3)CCC4)=O)C2C1 C1(NC(CCC(C)C)=O)CC2CCC(C1)N2c1nnn(C)n1 C#Cc1cncc(NC(C2CN(C(=O)CN3CCOCC3)C2)=O)c1 n1(CCNC(C2(CF)CCC2)=O)cc(-c2ccncc2)nn1 c1(C(=O)NC(CCOC)CNC(=O)CCCN(C)C(C)C)cccc(C(C)C)c1 N1(C(c2cnc(C(C)C)s2)=O)CC(C2(NC(=O)CN3CCCC3C)CC2)C1 N1(C(CCc2n(C)cnc2)=O)CCC(N=[N+]=[N-])(C(=O)N(CC(F)F)C2CCC2)C1 C(=O)(C1=COCCC1)NC1CC(C(N2CCC(CC#C)C2)=O)C1 c1(CC)ccc(Cl)c(S(=O)(=O)N(C)Cc2ccccc2CCCc2ccccc2)c1 CN=C(NCC1CC12CCOCC2)N1CCC(CCC)C1 C(=O)(CN=c1cc[nH]cc1)NC(C(=O)NCCC)C1CCCC1 C1(C)(C(N2CC(CC=C)(CNC(C3(COC)CCCC3)=O)C2)=O)CCNC1=O c1(OCC(=O)NCC2CN(C(CC(C)(C)SC)=O)CC2O)cc(C)ccc1F c1(C(=O)NC2C(NC(=O)C=CCO)CC2)cnc2ccccc2c1C(F)(F)F C(=O)(C#CC1CCC1)N1C(C(=O)NCCNc2ccccc2)CC1 c1(SC)nccnc1C(=O)NCC(C1CCN(C(=O)Cc2csnn2)CC1)O CCCCCC(C)C(=O)NC1CCC(CC(=O)NCc2cnn(C)c2C)CC1 c1(OC)cc(C=CC(=O)NC(CC2CC=CCC2)CO)ccc1OCC(N)=O N1(C(C2C(C)(C)C2)=O)CCC(CNC(c2cc3ccccn3n2)=O)C(F)(F)CC1 N1(C(C2(C)CC2(F)F)=O)CC(NC(c2ccc(C(N)=O)cn2)=O)C2(CCC2)C1 Cc1cc(-c2csc(=N)[nH]2)ccc1OCc1cnncn1 c1(SCC(N2CC(O)(CNC(C34CC(OC)C3C4)=O)C2)=O)ccc(C#N)cc1 C1(NC(c2cncc(C)n2)=O)CN(C(=O)CCN2CCCCC2)C2CCCC12 C1(C(=O)NC(CCCNC(c2cc(C)ns2)=O)C)CN2CCC1C2 C1(C(N(c2cncc(C(N)=O)c2)C)=O)(CO)CCCN(C(=O)OC(C)(C)C)C1 N1(C(C2(CCOC)CC2)=O)CCC(CC(C)NC(C2CC2(Cl)Cl)=O)CC1 N1(C(c2ccc(OC)cn2)=O)CCCC(C)C1CCNC(=O)CN1CC=CC1 C=C1CCC(C(=O)NCc2cc(C(=O)Nc3ccccc3F)ccn2)CC1 CC1(C(=O)NC2CCN(CCCO)C2)C=CCN1C(c1cc(Cl)ns1)=O C1(CC#C)(C(=O)NC2CCCC2F)CCN(C(c2ccc(O)cn2)=O)C1 c1(N(C2CC3CNC2C3)C(C(C)OC)=O)cc(Cl)cc(Cl)c1 c1(CNC(C2(NC(Cc3ccn(C)c3)=O)CCC2)=O)cncc(Cl)n1 c1(N(C(C(N2CCC(=C)CC2C(=O)O)=O)CCC)C(N)=O)cccc2c1CCO2 N1(C(C(F)OC)=O)CCCC(CCC2CCCN2C(=O)CCC2CC2)C1 N1(C(C2C(C(C)C)C2)=O)CC(C)OC2(CCN(C(=O)CSc3ccccn3)C2)C1 c1(OC(NOCCCC(=O)NC2CC(C)C2)=O)cccc2c1CCC2 CC1CC(C(=O)C(N2CCCCC2=O)F)CN1C(=O)CCCc1ccc(F)cc1 CCCCCCC(CC)NC(=O)C(CCC1CC1)NC(=O)CCC1CCCCC1 c1(NC(C)C(F)(F)F)ccc(C(F)(F)F)cc1S(=O)(=O)Nc1cccc(Cl)c1Cl C1(F)(CNC(C(CCCC)C)=O)COCCN(C(c2nocc2Cl)=O)C1 c1(C(N2CCC(CCC(=O)NC3(CC#C)CCOC3)C2)=O)ccccc1CC#N C1(C)(CC(=O)N(CC=C)CC2CC2)CCN1C(=O)C(C)(C)O C1(NC(=O)C2=CSCS2)CCOCC1NCC1CC1.C12CCN(C1)CC(=O)N2 C1(C)(C(=O)NC23CC(CNC(COCP(C)(C)=O)=O)(C2)C3)CNC(=O)C1 n1(CC)nc(C)cc1C(N1CCC(C(=O)NCC2CC23CCC3)(CO)C1)=O N1(C(C(C2CCC2)NC(C)=O)=O)CC2CC(NC(c3cnn[nH]3)=O)C1C2 N1(CCC(N2C(C)C(NC(=O)C(=O)NCC3CC3)CCC2)=O)Cc2ccccc2C1 C1(CNC(c2c(C(C)C)nns2)=O)CC2CCC(C1)N2C(C1(C#N)CC1(C)C)=O CCC1=NOC(C(=O)N(CC(C)NC(c2ccc(C3CC3)o2)=O)CC)C1 c1(C(=O)OC)cccc(C(N2CCC(C)(CNC(=O)CC3CC=CCC3)C2)=O)n1 CC(C)CC(C)C(=O)NCCC(C)N(C)C(c1c[nH]cc1-c1ccccc1)=O Cn1nc(C(N2CCCCC2C(=O)Nc2cn[nH]c2)=O)cc1O C(=O)(C(CN)CC(=O)Nc1ccnc(OC)n1)OC N1(C(c2c(OC)cncc2)=O)C2CCC1CN(C(c1scc(OC)c1Cl)=O)C2 N1(C(c2cc(OC)n[nH]2)=O)CCC2(CC1)CN(C(c1ccno1)=O)CC2CO N1(c2nnc(CC)s2)C2CCC1CN(C(C1CC(=O)NC1(C)C)=O)C2 CCC(CCC(=O)N1CCC(O)(N(C)C)CC1)OCCOC N1(CC(C)=CC(C)C)CCC(N(S(C)(=O)=O)C)CC1 Cn1cc(N)c(C(N2CCCC(OCCNC(c3nc(C4CC4)cs3)=O)C2)=O)n1 C1(C(N(C2CCN(C(=O)C=NOC)C2)CC#C)=O)CCSCC1 C1(C(=O)NCC2CCN(C(=O)COC3CCCC3)C23CC3)CCn2nncc2C1 N1(C(c2[nH]cc(C#N)c2)=O)CCCC(C2CC2NC(C2CC(=O)N(O)C2)=O)C1 c1(CSC)noc(CC(=O)NCCN(C(=O)C(F)C2CCOC2)C(C)C)n1 c1(OC)ccc(C(C)NC(=O)C(N2CC(C)CCC2CO)=O)c(Cl)c1 C=CC(O)(C(=O)NC(c1ccccc1)CNC(c1cc(=O)cc[nH]1)=O)C(F)(F)F C(CCC(=O)NC1(CCNC(C2CN(C3CCOC3)C2)=O)CCC1)=CC C=C(Br)CCC(=O)NC(C1(CNC(c2cn(-c3cccnc3)nn2)=O)CC1)C c1(CC(=O)NCC(C)(CO)NC(C2CCCC(=O)N2)=O)ccc(Br)c(O)c1 C1(NC(c2cn(CC(F)F)cn2)=O)CCN(C(=O)CCc2cocn2)C1 N=c1cc(C(C2CCCC2)NC(N2CCC(C(F)(F)CO)C2)=O)cc[nH]1 C(C)(C)(CC(F)C(=O)NCC1(C)CC=CCC1)NC(CC(C=C)C)=O CCC(O)(CNC(=O)CC(C)CNC(=O)COc1cnn(C)c1)CC N1(C(c2cc(OC)n[nH]2)=O)CC(C)CCC1CNC(=O)C=Cc1ccoc1 C1(NC(CCc2cc(C)on2)=O)CN(C(=O)COC2CCC2)C2(CCOC2)C1 c1(C(=O)NCCNC(C2(CC#C)CCOC2)=O)ccccc1SC1CCCCC1 Cc1c(C(=O)NCC2(C(C)NC(C3(CC4CC4)CCC3)=O)CC2)cncc1F C1(CO)(CO)CCC2CCC1N2Cc1cc2ccc(Br)cc2[nH]1 C1(C(=O)NC2(C)CC(NC(COCCN(C)C)=O)C2)Cc2ccccc2S1 C1(C(=O)NCc2csc(O)n2)(CNC(=O)CC2CSC2)CC12CCC2 c1(CNC2CC(NC(c3ccc(OC(F)F)cc3)=O)C2)ccc(Cl)cc1 C1(CNC(c2c(C)cc(C)o2)=O)CN(C(=O)CCC(F)F)CCCO1 c1(C(=O)NCC23N(C(C(C)=C(C)C)=O)CCC2CC3)cnc2c(c1)NC(=O)CO2 c1(C(=O)NC2CC(C)(COC)N(C(=O)Cc3ccon3)C2)cc(N)c(F)cc1C C(N=c1[nH]c2c(C)cc(C)cc2s1)c1nnc(CC(CC)C)n1C C(=O)(C1=CS(=O)CCC1)N1CC(CNC(c2ccnn2CC(F)F)=O)C(O)C1 CCC(CC(=O)N1CCCC2CN(C(C34CC3C4)=O)CCC12)CC(F)(F)F C(=O)(CC(C)(C)C=C)NC1(C)CC2(CC(OC)C(C#C)NC2=O)C1 N1(C(c2cc(CNC(c3nsnc3O)=O)[nH]n2)=O)CCC2(CCCC2)CC1 c1(C(=O)NC2C(C)CN(C(=O)CCn3ccnc3)CC2)nn(C)c2c1CSCC2 CC12CCC(C(=O)NCCC3CCN(C(C4CC4F)=O)C3)(CC1)C(C)(C)O2 c1(CCC(=O)N(CC(O)CCNC(=O)CCC(C)(C)F)CC)ccc(C)cc1O c1(C(=O)NCCCCCN(C(COCC=C)=O)C)cc(C(C)=O)oc1C c1(CNC(C2(CC#C)CCCO2)=O)cccc2c1OC(C)(C)O2 n1(CC)nc(C(N2CC(NC(c3cnn(C)c3Cl)=O)CC2C)=O)c(Br)n1 N1(C(CCC(=O)NCC)=O)CC2CN(C(c3ccc(OC)cc3OC)=O)CC2C1 C(=O)(CC1CCc2ccccc21)NC(CC)CN(C)C(c1ccc(Cl)nc1O)=O CCN=c1ccc(C(=O)NC2CCCCN(C(C3Cc4nnsc4S3)=O)C2)c[nH]1 CCCC(C)(O)C(=O)N(C)CC1(O)CN(C(=O)C(CN(C)C)c2ccccc2)C1 c1(NC2(CO)CCCN(C(C3CC(CC)OCC3)=O)C2)cc2nnc(C)n2cn1 C1(NC(c2sccc2Cl)=O)CC2CC(NC(=O)CC3CC4(CCC4)CO3)C1C2 C(C(C)(O)C(=O)NC(C)CCNC(C1(c2ccc(C)cc2)CC1)=O)OC C1(NC(C(CC)n2ccnc2)=O)CN(C(=O)C=Cc2nccs2)CC2(CC2)C1 c1(OC)cnc(C(N2CCC(C)(CNC(=O)CN3CC(C)C3)CC2)=O)c(F)c1 Cc1ccsc1C=CC(=O)NCCCN(CCCNC(=O)CC1COC(C)C1)C N1(C(c2ccn(CC(F)(F)F)n2)=O)CC2(C1)CN(C(c1cc(O)ncn1)=O)C2 C(=O)(C(F)C(F)(F)F)N1C(C)C(NC(=O)C(C)O)CC1 c1(C(N(C(C)C(=O)NC2CCN(CC)C2)CC)=O)cccc(CO)n1 Cc1cc(C#N)ccc1C(N1CC(CNC(=O)C(c2cccnc2)O)CC1C)=O C1(C(=O)NCC2N(C(CC(=O)OC)=O)CCOC2)COc2ccccc2O1 N1(C(C(C=CCCC)O)=O)CCC(CNC(c2nc(C)sc2C)=O)C(F)(F)C1 N1(C(COCCCC)=O)C2CCC1CN(C(c1n[nH]c(C3CC3)c1Br)=O)C2 C1(C(N2CC3(CN(C(CC4CC(=O)NC4=O)=O)C3)C2)=O)CC1C1CCOCC1 CC1(CO)CCN(C(=O)CCCCNC(=O)CCC2CCOC2)C1 C(CCCOC)(C(=O)NC1CC(F)C(=O)N1)NC(C(C)SCCCC)=O C1(C(N(CC(C(=O)NC(CCCC=C)C)(C)C)C)=O)CC(C)CC(=O)N1 C(=O)(C1CCCc2ccccc21)NCCC1(NC(C(CC)NC(C)=O)=O)CCC1 C1(C)(CC(=O)N(C2CCN(C(C34CC3CCC4(F)F)=O)C2)CC)CCCCCC1 C1(C(C)NC(c2n(CC)ncc2)=O)CN(C(=O)CCN2CCC(F)C2)CCO1 C(C(=O)NC1CCCC(NC(=O)CCn2cc(C)nn2)C1)(C(C)C)SCC C1(CC(C)(C)C)CCN(C(=NCc2ccncc2)NCCOc2ccccc2)C1 C(=O)(C(C)CS(C)(=O)=O)NCC(C1N(C(c2c(F)ccc(C)n2)=O)CCC1)(C)C c1(CC(=O)NCCN(C(=O)CCc2cc(OC)no2)CC)ccc(Cl)c(F)c1 CCC(F)(F)CC(=O)N1CC(CNC(c2ncc(OC)cc2F)=O)C2CC12 Cn1ncc2ncc(C(N3CC(NC(=O)C(F)n4ccnc4)CC(O)C3)=O)cc12 C1(=CCNC(CN(C(COC)=O)C)=O)CN(C(C2(c3ncco3)CC2)=O)C1 C1(C(=O)NC(CC)CO)CN(C(=O)C(C)(C)C2CCCN2)CCNC1=O N1(C(CC2(NC(CCCCC(C)C)=O)CCCCC2)=O)CC(=O)N2CCCC2C1 N1(CCC)CCC(C(=O)N(C)CCN(C(c2cc(C)cs2)=O)C(C)C)C1 C(c1cccc(F)c1)=C(C(=O)N(CCN(C(C(COC)C)=O)C)C(C)C)F N1(C(C(C(=O)NC)(C)C)=O)CC=C(C(=O)N(CC(C)(O)C2CC2)C)CC1 C1(C(C)CNC(=O)CCc2cnc[nH]2)CCN(C(=O)Cc2cc[nH]c2)CC1 N1(C(C(C=C)OC)=O)CC(NC(=O)CCc2cc(F)ccc2F)CCC(O)C1 C(=O)(CCC1=CCCCC1)NCCC1(C(=O)NC2(C(COC)O)CC2)CCC1 C1(NC(CC(=C=C)C)=O)CC(NC(c2ccc(C(F)(F)F)o2)=O)C12CCOCC2 N1(C(c2nc(C)oc2)=O)CCN(C(c2ccc(C(F)(F)F)cc2)=O)C2CCC12 Cc1ccc(Cl)c(CN2CCOCC2C(=O)Nc2cccc([N+](=O)[O-])n2)c1F CC1=C(C(=O)N2CCCC(CO)C(NC(C3(CO)CC3(F)F)=O)C2)CCC1 C1(C)(NC(=O)NS(CC(CCC)(C)C)(=O)=O)Cc2ccccc2C1 C(CC(=O)NC(C)(C)CCCNC(c1ccn(C)n1)=O)(C(F)(F)F)OC c1(CNC(C(C2(C)CC2)NC(C(SC)SC)=O)=O)ccnc(C)n1 CCC(F)(F)C(C)(C)C(=O)N1CC(C)CN(C(=O)CCC(C)C)C(C)C1 Cc1ccc(C(C)NC(=O)C(C2CC3(CC3)C2)C2CCCC2)cc1F c1(NC(C=CC(C)(C)NC2CCN(C(=O)C(O)C(F)(F)F)C2)=O)ccc(Cl)c(F)c1 c1(OC)cc(C#N)ccc1C(N1CCN(C)C(CNC(=O)C(O)CSC)C1)=O CN1CCC2(CC1)CC2NC(=O)NCC1CN2CCCN1CC2 c1(C(N2CCN(C(C(C)OC)=O)CC2C2CCC2)=O)ccc2ccccc2c1C N1(C(C(CC)OCCC)=O)CSCC1C(N1CC(CC(=O)OC)C1)=O c1(NC(C)=O)ccc(O)c(-c2cn(CCCC(=O)NC3COCC3O)nn2)c1 C(=O)(CCCCC(=O)c1ccccc1)NC1C(NC(c2nccc(C)n2)=O)C1 c1(C(=O)NCC2N(C(c3c(CC)c(C)sc3)=O)CC2)cnc2c(c1)NC(=O)CN2 c1(C(C)C)c(NC(=O)COC(=O)Cn2ncnn2)cnn1-c1ccccc1 C12CC3CCC(C1)N3C(=O)CCNC2=O.C=CC1CC1C(=O)NCC1CCC1 C1(C(CO)NC(C2(C#N)CCC2)=O)CCN(C(=O)Cn2ccnn2)CC1 c1(C(N(C2CCCC(NC(C3CC(C4CC4)C3)=O)C2)C)=O)n[nH]c2c1CCC2 c1(CC(=O)NCCOCCn2cc(-c3cccc(C)n3)nn2)ncc(Cl)cc1Cl CC1(C(N2CCCC2CNC(=O)CC2(O)CCCCC2)=O)CCCCCCC1 c1(C(=O)NC(CC)CN(C(=O)C=Cc2ccsc2)C)cc(C)c(F)cc1N c1(C(=O)NC2CC(C)(NC(c3cc(CC(C)C)nn3C)=O)C2)ccc(=O)n(C)c1 CCC(C)(C(=O)NC1CN(C(C2(Br)CC2)=O)CC1OC)OC C(=O)(CCC(C)(C)C(=O)OC)NC(CC)(CNC(C1CCOC1)=O)CC CC1(C)CCCCCC1NC(=O)C(CCF)NC(c1nsnc1O)=O c1(SCC)cncc(C(=O)NC(C2CN(C(=O)Cn3nnc(=N)[nH]3)CCO2)C)n1 N1(CC(=O)NCC(C)(C)OCC(=O)N(CC2CC2)CC2CC2)CCOCC1 N1(C(=O)COC(C2CCCC2)=O)CCCCC1C1CCCN1c1nnc(C(F)F)s1 C(CC(=O)OC)(C1=CCCC1)OCC.C12CCCC1N2 c1(C(=O)NCC2CC(NC(C3C(C)(C)NC(=O)C3)=O)C2)cc2c(Cl)ccnc2s1 CN1CCOCC1CC(=O)NC1COCC1C(=O)NCc1ncc[nH]1 c1(OC)ccc(C=CC(=O)NCCN(C)C(c2ccnc(C)n2)=O)cc1OC C#CC1CN(C(c2cccnc2N)=O)CCN1C(=O)CC1OCCCC1(C)C C1(NC(CN2C(C)CCC2C)=O)CCCCCCC1NC(=O)CCc1ccsc1 C(=O)(C1=CC12CC(N(C)C(=O)OC(C)(C)C)C2)N1CCC(C(=O)OC)C1 C1(CCCOC)(C(N2CC(n3cc(CNS(N)(=O)=O)nn3)C2)=O)CCCC1 C1(CNC(C)=O)CN(C(=O)Cn2nc(O)ccc2=O)C2(CCOCC2)C1 n1(CCN(C)C)ccc(=NC(=O)C2C(C(=O)Nc3ccc(C#N)cc3)CCC2)[nH]1 C(CCN=C(NCC1CCOC1)N(C)Cc1ccncc1Br)SC c1(C=O)cc(Cl)c(O)cc1O.c1(CS(N2CCN(CCO)CC2)(=O)=O)cccc(Cl)c1 c1(C(=O)NC(CCCC)CNC(c2ccc(CC)cn2)=O)cn2cc(C)sc2n1 c1(NC2C(CCC)CCCC2)ncnc2cc(F)c(OC)cc12 C1(C(=O)NC2(CCOC)CCN(C(=O)CCC(C)(F)F)C2)CCCCC1C1CC1 c1(C(=O)NCC(CNC(c2c(OC)cccc2Cl)=O)C)cccc(P(C)(C)=O)c1 CC(C)CCCC(=O)N1CCN(C2COCC2NC(=O)CCc2cn[nH]c2)CC1 C(C(=O)NC(CCSC)C(=O)NCCC1(OC)CC1)(C(C)C)OC C=CC1(C(=O)NCc2c(C)ccnc2C)CCN(C(=O)C=CC(C)CC)C1 c1(NCc2n(C)ccn2)nc(=NC2CC(c3cccnc3)C2)[nH]c2c1CCC2 C(CN=C(NCc1cc(C)ccc1Br)NC1CC1Cc1ccccc1)OCC C1(C(=O)NCCC2(C(=O)NC(C)CN(C)C)CCCC2)CC2C=CC1C2 c1(C(N2CC(NC(c3c(F)cc(Cl)cc3Cl)=O)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 C1(C(=O)NCC2C(C(N3CC(CF)C3)=O)C2)CCN(C2CCSC2)CC1 c1(SC)ccc(-c2cccc(C(O)CN3CCCC3)c2)cc1 C1(NC(C2CC(CF)C2)=O)CN(C(c2ccc3c[nH]nc3c2)=O)CC12CCC2 c1(C(=O)NC(C(C)NC(CC(CCC)C)=O)CO)nccc2ccsc12 C1(C)(C)CC(=O)N2CC(CC2C)NC1=O.C1(N(C)C)(CO)CCCCC1.CS C(CC(C(=O)NCC(c1ccccc1)C)NC(c1ccnn1CCF)=O)=CC C1(OC)C(C)(C)CN(C(c2c[nH]c3ncc(F)cc23)=O)C1(C)C C(N=c1[nH]nc(CO)s1)C1CCN(C(=O)CC2CCCSC2)C1 N1(C(c2ccc(O)nn2)=O)CC2CCN(Cc3cn4ccccc4n3)C2C1 c1(-c2c(CC)cccc2)cccc(C(N2CC3CC(C2)N3C(=O)CCBr)=O)c1N c1(C(=O)NC(CN(C(=O)CC2CC2)CC)C)cc(OC(F)(F)F)c2ncccc2c1 c1(OC)c(C(=O)NC2CC(F)CN(C(=O)CCN3CCCC3)C2)cccc1Cl c1(CC(=O)NC(C2CCCCC2)C(=O)N(C(C(=O)NC)C)C)ccc(C#N)cc1 c1(CCC(=O)NCC(CC=C)NC(C2CC2C2CC2)=O)ccc(F)c(F)c1 N1(C(C2CON(CC)C2=O)=O)CCCCC(N(C(=O)Cn2nc(C)cc2C)C)C1 C1(CNC(c2cnn(C3CCCCO3)c2)=O)CN(C(c2cc(F)cs2)=O)CCO1 N1(C(C=C(COC)C)=O)CC2C(CNC(c3cnc(C(=O)OC)s3)=O)C2C1 c1(OC)cscc1C(=O)NC1(C)CC(NC(=O)CCC=CC(C)C)C1 c1(-c2cccc(C(=O)NCC3CNCC(C)C3)c2)cccc(C#N)c1 c1(C(=O)NC2(CNC(C3C(C)OC(=O)N3)=O)CCOC2)ccc(Cl)c(F)c1F C1(CC(=O)N(CCCN(CCO)C(C2CSCCS2)=O)C)CCCCC1(C)C c1(C(C)C(=O)NC2CC(N(C)C(C3CC4CC3C4)=O)C2)ccc(C#N)cc1 C(=O)(C(F)(F)C(O)C1CC1)NCC(C1(O)CCN(C(C2CC(O)C2)=O)C1)C C(CC(C)(C)C(=O)N1CCC1CNC(c1csc(-c2csc(C)n2)c1)=O)OC c1(C(N(CC(C)NC(=O)CNC(N)=O)C)=O)ccc2c(Br)cncc2c1 c1(CC)ncccc1N(C)C.c1(C2CNC(=O)N2)nc(C(=O)N(C)C)co1 N1(C(c2n(C)cnc2)=O)CC2(CNC(=O)CCOc3cccc(F)c3)CCC1C2 N1(C(C2C(CNC(C3N(C)CCOC3)=O)C2)=O)CC(O)(C2CCC2)C1 CC1(C)CC(NC(=O)NC(c2cc(F)cc(F)c2)CO)C12CCC2 c1(C(=O)NCCC2(NC(C=CS(C)=O)=O)CC2)cc2c(s1)CCCCCC2 C1(CC(=O)NCC=C2CCN(C(CC(C)(C)C3C(C)C3)=O)CC2)CCCC(C)(C)O1 c1(C(=O)NC2CN(C(CC3(OCC)CC3)=O)CC(O)C2)ccc(C)c(C)c1Cl C1(C(N(CCCNC(CC(=O)NCC#C)=O)C2CC2)=O)CC(=O)N(CC=C)C1 c1(S)ccc(F)c(F)c1.C(=O)(CCC1CCCC1)N.CC(C)N1CC1 C(C)(C(C(=O)N1CC2(CCCCC2)C1)C(C)C)NC(C(C)SC)=O CN=c1[nH]cc(C(N2C(C(=O)NC(C)C(C)(C)CO)CCC2C)=O)o1 O=C1CC2(CCN(C(c3ccnc(Oc4ccccc4Br)c3)=O)CC2)CN1 c1(C(N(C(C)CNC(c2cn[nH]c2)=O)CC)=O)ccc(Cl)c(Cl)c1C CN1CCCCC1C(N1CCCCC1CNC(=O)Cc1ccccc1CC#N)=O c1(C(N2C(CNC(C3C(CC(C)C)C3)=O)CC(F)C2)=O)nnn2c1C(=O)NCC2 c1(CNC(C2C(O)CCN(S(CCC)(=O)=O)C2)=O)n[nH]c2ccccc12 C1(NC(C(C)=C(C)C)=O)CCCN(C(c2cc(Cl)ccc2Cl)=O)CC1F C(=O)(C(C(C)O)N(C)C)NCC(CC)N(C)C(C1CCCN1N=O)=O CC1(C#N)CCN(C(C2CN(C(c3ccon3)=O)CC23CC3)=O)C1 c1(NC(=O)Nc2cccc(NC(N3CCCCC3)C)c2)cccc(S(C)(=O)=O)c1 C1(C)(C(N(CCCNC(=O)C(c2ccc(F)cn2)(F)F)C)=O)CC(O)CN1C C(=O)(CC(C)O)NC(C)CC.C(=O)CCNC(=O)CCN(C)CCO C=CCC(CC)C(=O)NCC(C)(C)NC(c1cnc2n1CCS2)=O c1(C(N2CC(C)C(NC(c3cocn3)=O)C2)=O)cc(O)nc2ncn(C)c12 c1(C(N2CC3C(CNC(CC(C)F)=O)(C3)C2)=O)c(F)cc(Br)cc1F C(CCC(C(=O)NCC(=O)N(C)C)NC(=O)CC1CC=CCN1C)OC C1(C(=O)NC(C)CN(C)C(c2ccnn2CCF)=O)CC2(CCOC2)C1 C1(NC(c2cnn(CC(CC)C)c2C)=O)CC2CN(C(c3cccn3C)=O)CC12 C12(C(=O)OC)CCCC1(C(=O)NC(CCN(C)C(c1cncs1)=O)C(C)C)C2 C1(C(=O)N(CC(C)CNC(c2cnn(C(F)F)c2)=O)C)(OC)CCCOC1 c1(NC(C)=O)ccc(S(=O)(=O)N2CCN(Cc3ccncc3F)CC2)cc1 c1(OC)c(F)cc(S(=O)(=O)Oc2ccc(SCC(F)(F)F)cc2)cc1Cl C(CCC(C)C(=O)N1CCN(C(=O)CC2(O)CCCCC2)CC1COC)OC c1(C(=O)OCCc2cc(OC)cc(Cl)c2)ccc([N+](=O)[O-])cc1O N1(c2ncn(-c3nc(C)c(C)s3)n2)CCOC2(CCC2)C1.N12C(CC3CC13)C2=O N(C(=NCCN1CCCC1)NCc1ccco1)CC1CC(C(F)(F)F)C1 c1(C(N(C2CC(NC(c3c(OC)ccnc3)=O)C2)C)=O)ccc2c(c1)COC2=O C1(NC(c2ccc(CNC(c3ccc(CCC)[nH]3)=O)nc2)=O)CC1C1CCCC1 c1(C(=O)NCC(CC(C)C)NC(c2c[nH]c(=N)o2)=O)cccc2c1COCC2 c1(C(N2CCN(C(C3CCC(=O)N3)=O)C3C2C3)=O)cnc2c(n1)CCCC2 C1(C(=O)NC(CC)CNC(c2ccncc2Cl)=O)Cc2cccnc2C1 CC(C)(C(=O)N1CC(O)(CCNC(=O)C(F)(F)C2CC2)C1)c1ccncc1 Cc1csc2ncnc(NC3(c4cccc(C(F)(F)F)c4F)CC3)c12 c1(C(N2CCC(CCNC(C(C=C)c3ccccc3)=O)C2)=O)cc(O)nn1C c1(N2CCC(N(C(C)C)C(c3cnccc3C(F)F)=O)CC2)nc(Cl)ncc1F C(=O)(CS(=O)(=O)C1CC1)N1C(C(C)NC(C2(c3ccno3)CC2)=O)CCCC1 c1(N2C(C)COC(c3ccccc3)C2)ccc2oc3ccccc3c2c1 C1(c2nn[nH]n2)(Nc2c(C(=O)OC)sc(Br)c2)CC2CCC1C2 Cc1ccc(C#N)cc1C(=O)Oc1ccc(N2CCCC2)c(F)c1 C12(C(=O)NCCCCSCC)CC(C)(CN1C(C1C3CCCOC13)=O)C2 S(=O)(=O)(c1cncc(C(=O)O)c1)N1CCC(=O)N(c2ccccc2F)CC1 CCC(CC(=O)N(CC(O)CNC(=O)C(C)CCOC)C)SC c1(CC)nnsc1C(N1CC(C(C)NC(=O)C(C)N(C)C(C)=O)C1)=O CCP(=O)(CC)c1ccccc1-c1cc(C(=O)OC)ccc1OCCN(C)C N1(C(c2cc(CSCC)on2)=O)CC2(NC(=O)C(O)CC(C)(C)C)CCC1CC2 CC(CC(=O)N1CCCC1CCNC(=O)COc1ccn(C)n1)n1cccn1 c12ccccc1NCCc1cn-2nn1.c1(N(C(C)=O)C)cccc(Cl)c1 C1(C(=O)NCCC(CCNC(c2c(C)cno2)=O)C)CC2CC(F)(F)C2C1 C1(C(C)(F)F)(C(=O)NCC(CN(C(c2cncnc2)=O)CC)O)CCOCC1 C=CCCCCCCCC(=O)Nc1c(C(=O)Oc2cccc(Cl)c2F)c[nH]c1C Cc1ccc(C(C)C(=O)NC(CNC(=O)COCCN(C)C)CO)cc1 CC(O)(CC(=O)NCC(C1CCC1)NC(c1cncc(F)c1)=O)c1ccccc1 C(=O)(CCC(C)S(C)(=O)=O)NCCN(CCC)C(c1cc(Cl)ccc1F)=O C(=O)(CCNC(=O)CN(C(c1cc[nH]n1)=O)CC1CC1)NC(C)C c1(OC)cc(C(=O)NC23CC(NC(=O)C(O)CCSC)(C2)C3)cc(OC)c1O CCCCC(CC)C(=O)N1CCCCC(NC(=O)Cn2ccc(C(F)(F)F)n2)C1 CN1CCN(C)C1=NCC1CCN(c2ncccn2)CC1 C=C(C)CCCN1CC(n2cc(C(=O)NC3CC(CN4CCCC4)C3)nn2)C1 CCCN=C(NCC1(N2CCOCC2)CCSC1)NC(C)COCC(C)C C1(CNC(CC(C)(C)OC)=O)CCC2(CCN(C(=O)C(C)(C)C3CCC3)CC2)O1 C(=O)(CC1=NNC(=O)C1)N1CCC(N(C(c2n(C)c(S)nc2)=O)CC)CC1.OC CC(C)CC(=O)OC1C(c2ccccc2)OCC(C(=O)N(C)Cc2ccco2)N1 C(=O)(C(C)(C)C(=O)NCC12CCCC1N(C(c1cc(C)cc(F)c1)=O)CC2)NC c1(C(N2CCCCC(NC(c3cc(C)nn3C)=O)C2)=O)cc(F)c(C#N)c(F)c1 c1(-c2cn(CC(=O)OC)nn2)ccccc1C(C)NC(=O)CCOCC1CCCO1 c1(C(=O)NCCCC(C)NC(CCCC=C)=O)cnc2ccccc2c1OC CN1CCC(NC(=O)CCOCCNC(c2cc(O)ncc2F)=O)CC1C c1(C(N2C(CCOC)CN(C(=O)CSC(C)C)CC2)=O)cc2c(o1)CCCC2 Cc1cc(C(N2CCCC2C(C)NC(=O)CCC2CCC(=O)N2)=O)cc(C)c1F C(=O)(CC(C)CC(F)(F)F)NC1CCC(NC(C(C)Oc2cccc(C)c2)=O)C1 C1(C2CCCO2)(C(N2CC3CN(C(c4ncc(C)nc4)=O)CC3C2)=O)CCCO1 C#Cc1ccccc1CC(N1CC(C)CC1C(=O)NCc1occc1C)=O C1(C(=O)NC(c2cn[nH]c2)C)CCCC12CCN(C(=O)C1=CCCC1(C)C)CC2 N1(C(c2nc(COC)oc2)=O)CCCC2(CC(NC(=O)C(C)(COC)OC)C2)C1 C1(C(=O)N(C2CC(C(=O)NC(C(=O)OC(C)C)C)C2)CC)CCCCC1 c1(CNC(C(C)CNC(=O)CN2CCOC2=O)=O)c[nH]c2cnccc12 C1(C(=O)NCC(C)CN(C(=O)C(C)(C)CC(F)(F)F)C)CCc2nc(O)[nH]c2C1 N1(CCn2ncc(C)c2)CC2CC2(C(=O)NCc2cc[nH]n2)C1 C1(NC(=O)CC2CC=CC2)CC(O)CN(C(c2cncs2)=O)C1 Cn1ccc2nc(N3CC(F)CC3C(=O)NCCC3CCOC3)nc(Cl)c12 c1(NC(C2C3(CN(C(c4cc(C)ncc4)=O)C3)C2)=O)csc2nccnc12 S(=O)(=O)(c1ccc(NC2CCC2)c(Cl)c1)NC1CCCC(C(C)C)C1 C1(C(N2CC(O)(C(C)NC(=O)Cn3cc(C(F)(F)F)cn3)C2)=O)CCCCC1C c12cccc(c1)CNC(=O)C1(CC1)C2=O.c1(C(=O)NC)ccc(Cl)cn1.C1CC1 C(c1cccc(NC2CC2)c1)=CC(=O)NCC(C)NC(CNS(CCC)(=O)=O)=O CC1(C)OCC2CC12C(=O)NCC(C1CCCCC1)NC(c1cc(Br)c[nH]1)=O c1(C(=O)NCc2c(C)cc(Cl)nc2)c(C)cc(O)cc1C.C1(CN)CN(C=O)CCO1 C1(COc2cn(C)nc2)CCCC(NCC2CC3C=CC2C3)C1 c1(C(N2CC(NC(c3c(C)ocn3)=O)C(O)C2)=O)cc2cc(Br)ccc2o1 C12(C(=O)NC3CN(C(c4c(CC)cno4)=O)C(C)C3)CCC(C(F)F)(CC1)CC2 C1(NC(C(C2CN(C(C(CC)(C)COC)=O)C2)OC)=O)CCN(C)CC1C#N C(=O)(CCC(C)(F)F)N1CC(C=C)(CC(=O)NCC2CN(C)CCO2)C1 c1(CC(=O)NC2CC(CNC(C(CC)N(C)C)=O)C2)nc2c([nH]1)CCCC2 N1(C(C(CC#C)C2CC2)=O)CCC2(C1)CN(C(=O)C1=C(C#N)CCC1)C2 c1(C(=O)NCCCCCCN(C)C(C2COC(=O)C2)=O)cc2n(c1)CCCC2 C(C(=O)N=c1cc(C)[nH][nH]1)NC(c1ccc(F)cc1)C(=O)NC(COC)C C1(CC(=O)NC(C)CCNC(=O)Cc2cnsc2)OCCOC1(C)C c1(C(N2C3CN(C(c4ccc(C)c(C)c4)=O)CC32)=O)cccn2nccc12 c1(C(N(C(C)CNC(=O)C(C)Cc2cnn(C)c2)C)=O)ccc(C2COC2)cc1 c1(N(CC(CC)C)C)ccnc(NCCSc2cccc(F)c2)n1 CCCC(CNC(=O)C(CC)NC(C)=O)C(=O)NC1CCC1O S(=O)(=O)(CCC(=O)N1C2CCC1C(CNC(=O)CC1CCC(=O)O1)C2)NC c1(C(=O)NCCCN(C(C2CCC(=C)CC2)=O)C2CC2)nccc2occc12 c1(C(=O)NC2CN(C(CN(C)CCO)=O)C(C)(C)C2)cc(F)c(N)c(F)c1 N1(C(C2CN(C)C(=O)C2)=O)C(NC(C23CCCN(CCC2)C3)=O)C2CC(O)C1C2 CC1(C(=O)NCCCOCCNCC2CCC2)CCCN1C(c1ccon1)=O N1(C(=O)C=C2CCOCC2)CC2(CCN2C(=O)C(F)C2CCOC2)C1 N#Cc1ccc(CC(N2CCOC(CNC(c3nccnc3Br)=O)C2)=O)cn1 Cc1cc(Cl)c(C(N2CCCC(C(C)NC(=O)CCC3CCC3)C2)=O)cn1 N1(C(C23CCC(CNc4c(C)cnc(C)n4)(CC2)C3)=O)CC2CCC(CO)(C2)C1 N1(C(CSCCOC)=O)CCCC(C)C1CNC(=O)CS(N)(=O)=O C1(c2cn(CC3CCCC4CC34)nn2)CCCCN(C(=O)C(C)(C)N2CCOCC2)C1 c1(C(=O)NCC2N(C(c3n(C)cc(C(N)=O)c3)=O)CCCC2)cc2sccc2s1 N1(c2ccc(C(=O)Oc3cn(C)nc3C(F)F)o2)C(=O)C2C3C=CC(C3)C2C1=O N1(C(=O)NCc2c(C)con2)CCOC(c2ccccc2)(C(F)(F)F)C1 c1(NC)ncccc1C(=O)NCCOCCCNC(c1cc(CO)c(C)o1)=O c1(C(=O)NC2CC(NC(C(C)(C)c3ccns3)=O)C2)ccncc1O c1(C(=O)Oc2ncccc2C)cc(SC)ccc1NC(=O)NC(C)(C)C C12(CNC(C(C)Nc3cccs3)=O)CC1CN(C(=O)CC=Cc1ccccc1)C2 n1(CC(=O)N(CCN(C(C(CC=CC)C)=O)C)C(C)C)nc(C)n(CC)c1=O c1(C(N2C(CN(C(c3n(CC#C)ccc3)=O)C)CCC2)=O)ccnc(C(C)C)n1 C=CCC(CC)C(=O)NC(CNC(c1ccnc(O)c1Br)=O)C1CC1 C1(NC(C2CN(CC)C(=O)C2)=O)Cc2cccc(C)c2C1 C1(C(=O)NC2CN(C(CSC)=O)CC2(C)C)CN(C)C(=O)CCO1 N1(C(c2c(C)cc(OC)c(Br)c2)=O)CCc2c(Br)cccc2C1C C12(CNC(C3(COC)C=CCC3)=O)CN(C(=O)C(C)CSC)CC(F)(C1)C2 N1(C(CCN(C(CNC(C2C(C)C2)=O)=O)C)=O)CC(CO)C1(C)C C1(NC(C=Cc2cnc(C)s2)=O)CC(NC(=O)C(C)(C)c2ccns2)C12CCC2 Cc1cc(C(N2CCCC(C(C)NC(=O)CC=C(Cl)Cl)C2)=O)c(F)cc1N c1(C(N2CCC(N3CCC(C(=O)OC)CC3)C2)=O)cccc(O)c1OC(F)(F)F C12CC(C1(C)C)CC(=O)N2.CCCCNCCCOCC.C1(=O)CN1.C(=O)N.CC C1(NC(c2c(OCC)scc2)=O)CCN(C(=O)Cc2ccc(C)c(O)c2)CC1C c1(C(=O)Cc2cccc(Br)c2)ccc(CS(=O)(=O)CF)c(C(F)F)c1Cl CC(CC(F)(F)F)C(=O)N1CCC(CCCNC(=O)CN2CC3CC3C2)CC1 C1(CNC(=O)NC(COc2c(C)cccc2C)C)CC(C)(C)OC1(C)C N1(C(CCCCC)=O)CCC2(C1)CN(C(=O)C(c1ccnn1C)O)CCO2 C1(CN(C(=O)C2=NOCC2)CC)CCN(C(C2CC2C(F)F)=O)CC1 C1(C)(C(N(CC(=O)NC2CC(C(C)C)OCC2)C2CCC2)=O)CCCN(C)C1 CC(CC(=O)NC1CCCC(NC(=O)CCc2cccc(F)c2F)C1)P(C)(C)=O N1(C(C(CC)NC(c2ccc(C)s2)=O)=O)CCCCCC1C(=O)OC N1(C(c2cnc(O)c(Cl)c2)=O)CCc2cnccc2C1 N1(C(C(C)n2cccn2)=O)CC2CN(C(=O)COCC3CCCCO3)C2C1 C(=O)(C(CC(CC)CC)N(C1(C)CC1)Cc1ccc(I)cc1)NC CC1CN(C(=O)Cc2ccc(F)c(C)c2)CC(C)C1NC(c1cc(CO)on1)=O C(c1ccccn1)=C(C)C(=O)N(C)CC1CCN(C(=O)C=Cc2cc[nH]n2)CC1 N1(C(C(C)NC(=O)C2CC2)=O)CCC(C(=O)NCC2=NOC(C)C2)C1(C)C c1(C(=O)NC2CN(C(CC(C)(C)O)=O)CC2F)cc(O)ccc1Cl c1(C(=O)NC(C2(O)CCN(C(=O)CCC3CCCC3)C2)C)ccc(C(N)=O)nc1 c1(C(=O)NCC=CCNC(=O)C2=CCCOC2)c(F)ccc2c1OCO2 N(C(=NCC(F)(F)c1ccccc1)NCC(F)F)CC1C(c2ccccc2)(C)C1 c1(NCC2(C(C(N3CCCCC3)=O)Nc3ccccc3)CC2)cc(F)cc(F)c1O N1(C(CCOCC)=O)CCCC2CN(CC(O)COC3CCC(C)CC3)CC12 N1(C(Cc2c(C)nc[nH]2)=O)CCCC2(CC(NC(C3CCCC(CF)C3)=O)C2)C1 C1(NC(=O)C=CC=C(Cl)Cl)CN(C(c2ccc3c(c2)CC3)=O)CCC1C(F)(F)F CN1CCN(C(=O)CSCC(N2CCCC2CNC(=O)COCCF)=O)CC1 C1(C(N(CC(CN(C(CCOCCN(C)C)=O)C)O)C)=O)CC(=O)C12CCC2 CCC(CNC(=O)C=Cc1cc(C)no1)(CC)C(=O)NCC1(C#N)CCC1 c1(C(N2CC(CNC(C(C)(C)N(C)C)=O)OCC2)=O)ccc2[nH]cc(C#N)c2c1 N1(C(C(C(=O)OCC)C2CC2)=O)CCOCC(NC(=O)C(C)OC)C1 c1(C(=O)NCCCNC(c2cn(C)nc2)=O)ccc2cc(F)ccc2n1 N(C1CCc2c1ccc(Cl)c2Br)CC(=O)NC(c1ccc(F)cc1)=O C12(C(N3CC(O)(CN(C(CC(=O)N(C)C)=O)C)C3)=O)CC(C#N)(C1)C2 C1(CN(C(=O)CC2CSCCO2)C)CCN(C(C2CCC(F)C2)=O)CC1 n1(CC)nc(C(=O)N(CCC(C)NC(c2ncnn2C(C)C)=O)C)c(C)n1 C1(C(=O)OCC(CC#C)(C)C)OCc2ncnc(O)c21 N1(C(C(c2ccccc2)OCC)=O)CCN(C(c2cncc(N)n2)=O)C2COCC12 N1(C(=O)CSc2ccc(Cl)cc2)CC2(CCN(C(=O)CCSC3CC3)CC2)C1 N#Cc1ccnc(C(=O)NCCC2(O)CCN(C(c3n[nH]cc3Cl)=O)C2)c1F C1(NC(C(C(C)C)S)=O)CC2CCC(C1)N2C(=O)CS(C)(=O)=O Cc1ccc(C(=O)NC2COCC2NC(=O)C(N2CCCC2)C2CC2)cc1 N1(C(CCC(=C)C)=O)CC2CCC1C(CNC(=O)CNS(C)(=O)=O)C2 c1(C(N2C3C(NC(C4(C)CC4Br)=O)CC(C3)C2)=O)ccc2n[nH]cc2c1 Cc1ccc(C)n1CC(=O)NC1(CO)CC(C)(CO)C1 C(CC(=O)NCC1C(C)(C)C1(C)C)(C(F)(F)F)NC(Cn1nnc(C)n1)=O C1(C(=O)NCCn2nnc(=N)[nH]2)CCCCC1NC(=O)CCN1CCOCC1 c1(C(=O)NCCCN(C(c2ccc(Cl)s2)=O)CC)ccc2sc(C)nc2c1 C12(NC(C(C)NC(N)=O)=O)CCC(CNC(c3cnc(C(F)F)s3)=O)(C1)OC2 N12CCN(CC1)c1ccc(cc1)NC(=O)C2=O.N1(CC#C)CCCCC1C C(=O)(C(C)(C)CCSC)N(CCC)CCNC(=O)CC1CCC(=O)N1 CC1=C(C(=O)N2CCC(C)(CNC(=O)Cc3nncs3)C2)Cc2ccccc2O1 C1(C(=O)NCc2c(C(=O)NCC3(F)CCCCC3)[nH]cc2)CC2CCC(C1)O2 C1(NC(c2ccc(C(C)C)cc2)=O)CCCC2CN(C(C3CCC(=O)O3)=O)CC12 N1(C(C(CC)(C)OC)=O)CCCC2(CCCCC2NC(c2cc(Br)n[nH]2)=O)C1 c1(N2CCC=C(C)C2)ccncc1S(=O)(=O)NCc1cccc(-n2cccn2)c1 c1(C(=O)NC(C2CCCCC2)C(=O)NC(c2ncc[nH]2)C)cccc(O)n1 C1(c2cn(CCCSC)nn2)COC(C)(C)OC1.N12CC(O)C(O)C1C2 c1(CNC(C2C3(CCN(c4cc(C)ncn4)CC3)C2)=O)c(Cl)ccc2c[nH]nc12 C1(CNC(C(c2ccc(F)cc2)OC)=O)CC(F)CN1C(c1cccnc1S)=O n1(CCC(=O)NCCc2ccc(CNC(CC)=O)cc2)cnc2ccccc12 N1(C(C(C)Sc2ccccn2)=O)CCN(C2CCN(C(=O)C(C)C(C)O)CC2)CC1 C1(C2CCN(C(=O)CC(F)(F)F)C2)(NC(C(C)N(c2ccccc2)CCO)=O)CC1 c1(N2C3C(O)CC(CC3)C2)nc(=NCc2cnns2)[nH]c2c1CCC2 c1(C(N2CC(CC(=O)NCc3snc(CC)n3)C(C)C2)=O)ncc(C)cc1F CC1C(NC(c2cc(=O)cc[nH]2)=O)CCN1C(c1cnc(C(C)(C)CF)o1)=O CC1CC=C(C(=O)N2CC(CCNC(C3(CCN(C)C)SCCCS3)=O)C2)CC1 Cc1cnnc(O)c1C(=O)NC1CC(C)N(C(c2ccc(Br)cc2O)=O)C1 c1(C(=O)NCC2CN(CCCC#C)C2)c(O)nc2ccccc2c1Cl N1(C(c2c(C)cncc2)=O)CCN(C(=O)CCc2cnccn2)C(CC(F)F)C1 C1(C2CC2)(CNC(c2c(C)noc2C)=O)CCN(C(C2Cc3nncn3C2)=O)C1 c1(CNC(C2CC(O)(CC)C2)=O)ccnc(C(N)=O)c1.c12ccccc1C(=O)N2 N1(C(CNC(N)=O)=O)CC2(CCN(C(C3CC3c3cccc(O)c3)=O)C2)C1 CC1(C)OCCC1CCNC(=O)C(c1ccco1)NC(=O)CCn1cncn1 C1(NC(C2CCC(C(=O)OC)C2)=O)CCC(C)N(C(=O)Cn2cccnc2=O)C1 c1(NC(=O)CCC2CCCN2C(c2cc(O)ncn2)=O)ncc(C(F)(F)F)cc1Br C(=O)(C(O)CCNC(c1cc[nH]c1C)=O)NCC1CC(OC)C1 C(CCCC(=O)NCCC(C)(C)NC(c1[nH]nnc1C1CC1)=O)N(C(C)=O)C CC1CCCCC1(CNC(C1CN(C(N)=O)C1)=O)NC(=O)CC1(O)CCC1 C12(CNC(C3C(C(=O)OC(C)C)CCO3)=O)CC1CN(C(=O)CCCC1CC1)C2 C1(C)(CC)CC(NC(=O)CC2CC(F)CN2C(C2COCCN2C)=O)CCO1 Cc1cc(CCC(=O)NCC2CCOC2)on1.c12cn(nn1)CCN(C)C(=O)C2 C(=O)(C1=CCCC1P(C)(C)=O)N1C(COC)CN(C(c2coc(O)n2)=O)CC1 c1(C(=O)NCC(CNC(C(CC)OCC)=O)O)cccc(-c2nc(O)n[nH]2)c1 C1(NC(c2c(C)occ2)=O)CN(C(=O)COC2COC2)CC(C)(C)C1 C1(CC)CN(C(=O)CCOc2cccc(C#N)c2)CCN1C(=O)CC1CC1(Cl)Cl C12(C(=O)OC)CC(CO)(CN1CC(=O)C(C)CC)C2 C1(CC(=O)NC(C2CN(C(=O)Cn3cnc(Br)n3)C2)C)CCCOCC1 c1(C(=O)NC(C(=O)NCCC=CCCC)Cc2ccoc2)cncc(C#N)c1 c1(C(c2n(CCCSC)nnn2)NCc2cn(C3CC3)nn2)cnn(C)c1C CCCCC(O)CC(=O)NCCC(C(C)C)NC(=O)Cn1cc([N+](=O)[O-])nc1C S(=O)(=O)(CCC(=O)N1CCC(NC(=O)CSCC2CCCO2)C(F)C1)NC CC1CC(NC(c2ccc(-c3ccccc3)s2)=O)CN(C(c2sccc2Cl)=O)C1 N1(C(C2CCCN(S(CCC)(=O)=O)C2)=O)CCn2nc(-c3cnc[nH]3)cc2C1 C1(C(N(CC(CC)O)C)=O)(C(C)C)CCN(C(=O)Cn2cncn2)C1 c1(C(N2CCC(NC(c3c(CC)cco3)=O)C23CC3)=O)cc(F)cc(Cl)c1O c1(C(N2CCC(NC(CCCOC)=O)C(F)C2)=O)cc(Br)c(OC)cc1O N1(c2snc(CCC)n2)CCC(NC(=O)C(C)(C)COC)C(O)C1 C1(CCNC(c2nc(C)sc2)=O)CCCN(C(c2ncsc2C2CC2)=O)C1 c1(N(C)CC2CNCC2(C)C)ncnc2c1ncn2C1(CO)CCCC1 N1(C(c2ccc(SCC)cc2)=O)CCC(NC(c2c[nH]c(=N)nc2O)=O)C(C)C1 C(C(N=c1cc(C(C)C)nc(Cl)[nH]1)C(C)C(C)C)NC(CCSC)C(=O)OC(C)C C(CC1=CCN(C(C2CCCCC2O)=O)CC1)NC(c1c(C)noc1)=O N1(C(CCSc2n(C)nnn2)=O)C2CCC1(CNC(C1CC(C)(C)C1)=O)CC2 N1(C(C=CCOC)=O)CC(NC(c2cc(-n3cccn3)ccn2)=O)C(C2CC2)C1 C12(C(=O)OC)CC1CN(C(C1CCCN(C(=O)CC3COC(C)(C)C3)C1)=O)C2 C1(N(C(C(C2CCC2)OCC)=O)C)CCCN1C(=O)C(C)(C1CCOCC1)OC C1(N(C)C(c2cc(C#N)no2)=O)CCC2CN(C(C3CCCC(C#N)C3)=O)CC12 c1(OC)nccnc1C=O.C1(CNC(c2cn(C3CC3)nn2)=O)COC(C)(C)C1 C1(C(=O)N2c3ccc(cc3)C(=O)N3CCC2C3)CC12CC(F)(F)C2.N#Cc1nc[nH]n1 N1(C(=O)NC(C(C)(C)C)C)CCN2CCN(C(=O)CCC3CCCN(C)C3)CC2C1 C12(C(=O)NCCC3CCC(NC(c4c(C)noc4)=O)C3)CCC(CO)(CC1)CC2 C1(C(N2CCC(NC(CCSCCC)=O)C(C)C2)=O)CC2(C1)CC1(CC1)C2 C(=O)(C(C)(C)C(C)O)N1CC2C(C(=O)N(CC(C)(C)CO)C)C2C1 CCC(C)(CO)C(=O)N1CCCC(CNC(c2ccc(C(=O)NC)nc2)=O)C1 c1(C(C(=O)NCCC2CC(NC(C(C)(C)C3CCCC3)=O)C2)=O)cccc(O)c1 CCC(CC)CC(F)C(=O)NCC1CN(C(=O)C(C2CCOCC2)C)CC1C C(=O)(NNc1cc(C)ccc1[N+](=O)[O-])Nc1ccc(OCC)cc1C C=CC(C)(O)CC(=O)NCc1occc1C(=O)NC1CN(C)NC1=O c1(C2N(C(C(CSC)C3CC3)=O)CCC2)ccc(O)nc1 c1(C(N2C(C)CN(C(CCC(CC)C)=O)C(C)C2)=O)ccc(SC)c([N+](=O)[O-])c1 c1(C(N2C(CN(C)C(C3CC(C4CC4)=NO3)=O)CCC2)=O)c(F)ccc(O)c1F c1(CCC(N2CC(SC)C(NC(C3CC3C)=O)C2)=O)cccc(Cl)c1Cl N1(C(c2c(Cl)cn(C)n2)=O)CCN2CC3(CC3)CC2C1 c1(C(=O)NC(CN(C(c2coc(CO)c2)=O)CC)C)ccc2c(c1)NC(=O)CN2 c1(-c2cn(CCC(=O)NCCOC)nn2)cccc(C)n1.C1C(=O)O1 n1(CC)ccc(=NC(=O)c2ccnc3[nH]ncc23)[nH]1 C(C)(CCC(=O)NCCCCCCNC(=O)CCNC(C1CCCCC1)=O)SC C1(c2nc(CCC3C(C)CCO3)on2)CC2CCC1C2 C1(NC(c2cnc(N(C)C)o2)=O)C2CCC(C2)C1C(N1CCS(=O)(=O)CC1)=O N1(C(CC=CC(C)(C)C)=O)CC2CCC2(CC(=O)NC2(C3CCCC3)CC2)C1 C1(C(=O)NC2CCCC(NC(CN(C)C(=O)C3CC3)=O)C2)CCCC1P(C)(C)=O CC12CN(C(=O)CC3(C)CCOC3)C(C(=O)NCCOCCCO)(C1)C2 C=CC1CN(C(=O)C(C)(CC)CC)CC1NC(c1ccn2ccsc12)=O C1(C2CN(C(C3CCCCC3)=O)C2)(NC(c2cc(C)sc2C)=O)CC1 N1(C(CSCCCC)=O)CC(C2CCCN(C(c3cn4cc(C)sc4n3)=O)C2)C1 c1(NC(=O)CC23CC(C2)C3)ccc(-c2cn(-c3cncc(O)c3)nn2)cc1 c1(OC)nccc(C(=O)NCC(CCNC(C2CC3(CC3)CO2)=O)OC)n1 c1(COCC(=O)N(CC)Cc2cn(CC(=O)O)nn2)cc(OC)cc(C)c1 C=CCC(C(=O)N1C(C(=O)NCCc2cncc(C)n2)CC1C)OC N1(C(COCC(=O)OC)=O)CC(C)(CCC(=O)NCC(c2cccnc2)O)C1 N1(C(C2(OC)CCSCC2)=O)CC(CNC(c2cnco2)=O)C2(CCC2)C1 c1(C(=O)NC(CC)CNC(C2CCCC2C)=O)cccc(OC)c1OC Cc1ccc(Cl)cc1C(=O)NCCC1CCN(C(C2CC3(CCC3)C2)=O)C(=O)C1 C1(CC(=O)NCC23CCC(C(=O)OC)(C2)CO3)SC2=NCCN2C1=O N1(C(c2c(CC)ccs2)=O)CCOC(CNCc2ccnc(SC)c2)C1 C12(CNC(c3cn(C(C)C)nc3)=O)CCC(C1)N(C(C1CCCCNC1=O)=O)C2 c1(OC)ccc(Cl)cc1CC(N1CC(O)(CNC(=O)C(C2CCOCC2)F)C1)=O C1(C(=O)N(C2CCN(C(C3CC(C(F)F)C3)=O)C2)CCO)COC2(CCC2)CO1 Cc1cccnc1CN1CCNCC1C(=O)NC(c1cccnc1)C1CC1 c1(C(=O)OC)ccc(C(=O)N(CCCN(C)C(c2cccc(C)c2)=O)C)c(C)c1 C1(COC)(CNC(=O)C=C(C)c2ccco2)CCCN1C(=O)CC1(C)CCC1 C12(COC)CC(C(=O)N(CC(C)N(C(=O)C(c3ccc(F)cc3)F)C)C)(CO1)C2 N1(C(c2c(C)non2)=O)CCC(C(=O)NCC(C)(C)C2CC2)C(C)(C)C1 C1(C(=O)NCc2ncc[nH]2)(NC(c2nc(CCC)oc2)=O)CCC(C)(C)C1 c1(C(=O)NCCC(C)(C)NC(C2C(CC(C)C)C2)=O)ccc2c(c1)CCCC2 c1(CSCC)cccc(C(=O)N(CC(CC)NC(c2[nH]cnc2C#N)=O)C)c1 C1(CNC(CC2CC(NC(=O)CCOCC(F)F)C2)=O)CC2CCC(C1)C2 C1(NC(C2CCCC2)=O)CCCN(C(=O)Cc2ccc3occc3c2)CC1F c1(C(N(C(CNC(CCSC)=O)C)C)=O)coc2c(C)cccc12 N1(C(C(CC)=CC)=O)CCC2C(CCCN2C(c2nc3ccccn3n2)=O)C1 C1(C)(COC)CC(NC(=O)CC2(C)CC2)CN1C(c1ccccc1F)=O C(CC(CNC(C1CCCN1C(C)=O)=O)NC(=O)C(c1ccccc1)C)OC C1(C)(CNC(C2(CC=C)CCC2)=O)CN(C(=O)C(COC)N(C)C)C(C)(C)C1 c1(CSC)noc(C(=O)OC)n1.C12(CC1)C(=O)N2.C12(CC1)NC2 C12(CN(c3c(C)noc3C)C)CCCCC1C2(F)F n1(C2CN(C(CN(C)C(=O)C3CC3)=O)C2)cc(C2CCCC2)nn1.C1(SS)CCCC1 N1(C(C(CC)C#N)=O)CC2CC(NC(=O)Cc3c(OC)cccc3F)C2C1 C1(C(CNC(C(c2ccc(Cl)s2)C)=O)(C)O)CCN(C(c2cccn2C)=O)CC1 C1(NC(CC2C(C)CCC2)=O)CC2(CCN(C(c3cnn(C)c3N)=O)C2)C1 C1(NC(C(CCC)(C)O)=O)CC2(CCN(C(=O)C(C)CF)CC2)C1 Cc1c(C(=O)NCC2CCC2NC(C2CCCOC2C(C)(C)C)=O)ccn1C C1(NC(C2CC3CCC2O3)=O)CN(C(=O)C(c2ncccc2F)(F)F)CCC1F c1(C(=O)Nc2cc(Cn3cc(CCO)nn3)sc2Br)cc2[nH]ccc2nn1 CC1CCC(=CC(=O)N(C2CCN(C(C3CN(S(=O)(=O)C(F)F)C3)=O)C2)C)CC1 N1(C(C2(F)CC2)=O)CCCC(C(=O)NC2C(NC(=O)OC(C)(C)C)CCC2)C1 O=C(CCC1CC(NC(=O)C(CO)c2ccccc2)C1)N=c1c(Cl)c[nH]cc1I N1(C(CCCC)=O)CCC2CCCN(C(C34CCC(CC3)C(C)O4)=O)C2C1 CC1(C)CN(C(=O)C(F)(F)CC2CC2)CCC1NC(c1ccnc(S)c1)=O c1(C(N(C)C)=O)cccc(C2COC2)c1.C12CCCC1C(=O)N2.c1(=O)c(=O)n1C1CC1 CC1CCN(c2ncccc2S(=O)(=O)NCc2nc(=N)[nH][nH]2)CC(C)O1 N1(Cc2c(N(C(=O)OC)C)cccc2)C(=O)CCN(CC2CCC(F)C2)C1=O c1(C(N2CCN(C(COC(CC)(C)C)=O)CC2CC)=O)coc2c(F)cccc12 N1(C(CCCC)=O)CC2CC1CN2C(=O)COCc1cccnc1 c1(C(N(C2CCN(C(c3c(C)scc3)=O)C2)CCO)=O)ccc2ocnc2n1 C(C(F)(C(=O)N1CC(CC(F)(F)F)C1)C(C)C)NC(C1(C)CC(=C)C1)=O C12(NC(c3c(F)cccc3F)=O)CCCC1CN(C(=O)CCc1cccnc1)C2 Cc1nc(C(N2CC(NC(=O)C(C3(O)CCCC3)F)C2)=O)nn1C c1(C(=O)NC(CCNC(C(C)(C)OC(C)=O)=O)C)c(Cl)nc2ccccn12 C1(S(C)(=O)=O)(C(=O)NCCCN(C(c2cc(O)n(CC)n2)=O)CC)CC1 N1(C(C(COCC)C)=O)CCCCC(CCC(=O)N(C)Cc2cscn2)C1 c1(C(N2CCC(c3ccccc3)C(O)C2)=O)ccc2ncnn2c1 c1(-n2cc(SCC)nn2)cccnc1C(=O)Nc1cccc(C2CC2)n1 N1(C(CCc2ncn(C)c2)=O)CCC2CN(C(=O)C(c3cscn3)=O)CC2C1 C(=O)(C1=NOC2(CCOC2)C1)N(CC(O)CNC(c1cnn(C)n1)=O)C C(C(=O)NCC1CC(C)(O)C1)(C(C)(C)C)NC(C(c1ccccc1)OC)=O C1(CC(=O)NCC=CCC)CN(C(=O)CC2(C#N)CC2)CCO1 C(=O)(CCCS(C)(=O)=O)NC1CC(CNC(CCc2ccn(C)c2)=O)C1(C)C Cc1nc(CO)sc1C(=O)NCCC(C)CCNC(C1(S(N)(=O)=O)CC1)=O N1(C(C=CCC)=O)CC(C(N2CCC3(CC(OC)C3)C2)=O)CC(C)(C)C1 C1(C(=O)NC2CCC(CCNC(C(CC)(CC)CO)=O)C2)CCn2ccnc2C1 C1(C(N(C)CC2OCCN(C(Cc3cnc(C)o3)=O)C2)=O)CCCCNC1=O Cc1ccc(C(C)C)c(CNc2ccc(C)c(-c3nn[nH]n3)c2)c1 C1(NC(CC2CC(OC)C2(C)C)=O)CCC2(CC1)CN(C(c1ccc(Cl)cn1)=O)C2 C(=O)(C(CC(C)CC)NC(=O)CCCC1CC1C)NC1(C(=O)OCC)CC1 C1(CN(CCCC)C(C2CCN(CCc3ccc(C)cc3)CC2)=O)CCCCCC1 CC(C)C(C(=O)N(C1CC1)Cc1nccs1)C(C)NC(=O)CCCC1CCCC1 C1(C(=O)NCCC(C)SC)CC(O)CN1C(C1(c2cc[nH]n2)CC1)=O c1(C(=O)OCC)ncn2c1CN(Cc1cc(OC)cc(OC)c1Cl)CC2 Cn1cnc2cncc(C(=O)NCC(O)CNC(C3(C)C=CCC3)=O)c12 C1(NC(C=CCC)=O)CC(CNC(c2ncc(CCOC)s2)=O)C1(C)C Cc1ccc2scc(C(N3CC=CC(NC(C4CCCC5(CC5)C4)=O)C3)=O)c2c1 c1(C(=O)NCCC(C)N(C)C(C2CCN2C2CCCC2)=O)cc(Cl)c[nH]1 c1(C(=O)NC(C2CCN(C(C(CC)SC)=O)CC2)(C)C)n[nH]c2cccnc12 c1(C(N(CC(C)(C)NC(C2(CO)CC2(F)F)=O)C)=O)cc[nH]c(=N)c1 Cc1cc(C(N2CCN(CCCCCNC(=O)C3=CCC3)CC2)=O)c(C)o1 N1(C(C(C2CN(C(CC3(OC)CCC3)=O)C2)OC)=O)CCCC(C)(F)C1 N1(C(c2c(OC)c(Cl)sc2)=O)CCN(C(=O)C(C)O)CC(O)C1 N1(C(C=Cc2c(C)coc2C)=O)C2CCC1CN(C(C1CCCC(C)(C)O1)=O)C2 c1(C(=O)NCCCCC(C)NC(C=C(C)C)=O)cnc2c(Cl)cccn12 CC1CC(C(N2CC3CC2C3C(=O)NCCC(O)C(F)F)=O)CCO1 C(C(C)(C(=O)NN1CCCC(O)C1)NC(=O)COC(C)(C)C)SC C1(C(=O)NC(CC)CNC(c2cnn(C(C)C)n2)=O)Cc2ccccc2N1C c1(NC(=O)OCCN2CCOCC2)cc(CC2CCCCO2)ccc1F Cc1c[nH]c(C#N)nc1=NC(C)CN(C)C(c1cnc(Cl)[nH]1)=O N1(C(CCSC)=O)CCCC(CCNC(c2ccncn2)=O)CC1 c1(CC)c(C(=O)NCCC(O)CNC(c2csc(C(F)F)c2)=O)cccc1C Cc1ccc(F)cc1NC(c1ccnc(CNC(=O)CC2(C)CCOC2)c1)=O CN1CC(O)CCC1C(=O)NC1(C(=O)NCC(O)C(F)(F)F)CCCCC1 Cc1nc(N2CCCC2CCCNC(=O)C(C)C2CCC2)cc(C#N)n1 CCC(C(=O)NC(C)CN1CCCCC1)N(C(=O)CN(C)C(C)C)C C1(C(N2CCC(N(C)C)C2)=O)(NC(C2CC(SC)C2)=O)CCC(C)(C)C1 c1(OC)cc(C(N2CC(OC)C(NC(C3CC(C#N)(OC)C3)=O)C2)=O)oc(=O)c1 CC(CC(F)F)C(=O)NC1CN(C(c2ccccc2-n2cccn2)=O)CCC1O c1(CC(=O)NC(C2CCOC2)CNC(CC=CC=C)=O)cnn2c1OCCC2 C1(C(N2C(C(=O)NC3CC(CC)C3)CC2C)=O)CC(=O)CCO1 C1(C(=O)OCC2CCCCC2N2CCCC2)OCC2CCOC12 c1(CC)ccc(C(N2CCC(O)(C(C)NC(c3cn(C)cc3C)=O)C2)=O)cc1C c1(C(N2CC3CC(NC(c4c(CC)onc4C)=O)C3C2)=O)cc[nH]c(=NC)c1N C#CCCCCCC(=O)N1CCC2(CC2)CC1C(=O)NCCc1noc(C)n1 C1(C(N2CCC(CN(C(C)=O)C)CC2)=O)CCCC1S(C)(=O)=O c1(C(=O)NC(C2CC(NC(c3cc([N+](=O)[O-])n[nH]3)=O)C2)C)coc2ccccc12 C12(CNC(c3c(C)cncn3)=O)CCC(CNC(C3CC4(C3)CC4F)=O)(CC1)CO2 c1(N(C(C2COCCN2C(=O)CCN2CCOCC2)=O)CCO)ccc(Cl)cn1 c1(C(=O)NC2CN(C(CSCC=C)=O)CC2F)nccc2nn[nH]c12 N1(C(c2cccc(NS(C)(=O)=O)c2)=O)CCC2CN(C(C34CCC3C4)=O)C2C1 CCC(CC1CCCC1)C(=O)N1CCN(C(c2c[nH]c(=N)s2)=O)CC1 c1(C(N2CCC(CNC(COCCCCCC)=O)C2)=O)ccc(F)c(C(F)F)c1 c1(C=O)cc(-c2ccncc2)[nH]n1.N12CCC1C(=O)N(C)CCCCN2C.CCOC c1(C(=O)NC(c2c(C)cccc2)C)ccc2n[nH]c(C)c2c1 c1(C(=O)NCC(CN(C)C(C2CCC2)=O)O)cncc(S(C)(=O)=O)c1 c1(C(N2CCNC(c3cccc(OC(F)F)c3)C2)=O)nc(Br)sc1Cl CC1(C(=O)N2CCCC(NC(=O)CSC(F)(F)F)C2)CCc2ccccc21 C(C1=NOC2CN(C(c3c[nH]c(=N)s3)=O)CC12)NC(Cn1nc(C)n(C)c1=O)=O N1(C(C(C)SC)=O)CCC(C)(NC(=O)CC23CC(C2)C3)C1 N1(C(C#CC(=O)N(C)C)=O)CCN(C(=O)CC2CCCN(C)C2)C(CCN(C)C)C1 c1(C(=O)NCC(C)NC(C2(C)CCSCC2)=O)ccc2c(c1)C=CCC2 N1(C(CCC(C)CN(C)C)=O)CC(NC(=O)CCOCC2CC2)C2CCCCC12 c1(C(=O)NCC(C)NC(=O)Cc2cncc(O)c2)ccnc2[nH]c(O)nc12 CC#CCC(C(=O)NCc1ccc(F)c(O)c1)NC(c1cnsn1)=O C1(NC(=O)CCn2cccc2)CCCC(c2ccccc2)C1 c1(-n2c(CNCC3CCN(C(C(C)CC4CC4)=O)C3)ccc2)cccc(F)c1F Cc1cc(C(N2CCCC(N(CCO)C(C3CCCC(O)C3)=O)C2)=O)nc(C)n1 c1(C(N2CC(C)(NC(c3cn(CCCC)nn3)=O)C2)=O)c(N)cc(Cl)cc1F N1(C(c2nc(NC(C)=O)sc2)=O)CCOC(C(=O)Nc2cnn(C3CC3)c2C)C1 Cc1nc(C(=O)NCC(C)CN(C)C(c2nc(=O)n(C)[nH]2)=O)nn1C C1(C(=O)NC(CCC)(C)CC)CN(C(=O)CC2(COC)CC2)CC(C)(C)C1 N1(CC2CC2C(=O)NC2CC(OC)C2)CCOC2(CC1)CCS(=O)(=O)CC2 c1(C(N2CCC(C(C(N3CC(O)(CC)C3)=O)F)C2)=O)cc(Cl)cc2cccnc12 N1(C(C2CC(CNC(c3c(C)nn(C)c3N)=O)OC2)=O)CCOCC(C)(O)C1 c1(C(=O)NCC(C2CC2)NC(CNC(=O)NC)=O)cc(O)ccc1C c1(OC)ccnc(C(=O)NC(CNC(=O)COC(C)=O)C(C)(C)C)c1 C1(CNC(C23C(C(=O)OC)(CCC2)C3)=O)CC2CCC1N2C(c1ccnnc1)=O C(=O)(C(CC1CCOCC1)NC(C1CCCCS1)=O)N(CC(CN(C)C)O)C C1(NC(CC(=O)NC)=O)C2COCC1CN(C(c1cc(C#N)cc(C)n1)=O)C2 N1(C(C(C)n2cccn2)=O)CCCC(CN(C(=O)CN2CCNC2=O)C)C1 C12(Cn3cc(CCNC(Cc4noc(C)c4Br)=O)nn3)CCCCC1C2(F)F C1(C)(CC)CN(C(C2CCN2C(c2cn[nH]c2)=O)=O)C1 c1(C(=O)NC(C2(O)CN(C(C(C)OCC(C)C)=O)C2)C)cc(=O)cc[nH]1 C1(C(=O)NCCC(C)OC(F)F)CCc2nc(-c3ccccc3)ncc2C1 C1(CC(=O)Nc2c(OCC(C)C)cccc2)CCCCC(C)(C)C1 N1(C(CCCCCC#N)=O)CCC2CCCC(C1)N2C(=O)CN1CC2CC2C1 N1(C(C2CCN(C(CC)=O)C2)=O)CC2C(C(=O)NCC(O)C(F)(F)F)C2C1 C(=O)(C1=CC2(CCN(C(=O)CCOC3COC3)C2)C1)N(C)Cc1cncnc1 c1(C(C)NC(=O)CC2(F)CN(C(C3CNC(=O)C3)=O)C2)ccc(O)cc1 CC1(C)CC(CNC(c2nn(C(C)(C)C)cc2Cl)=O)CN1C(=O)CCF Cc1nn(C(C)(C)C)c(C)c1C(N1CC(N(C)C(C2(F)CC=CC2)=O)C(O)C1)=O c1(C(N2CC3(CCN3Cc3ccc(Br)[nH]3)C2)=O)ccc2c(c1)OCCCO2 C1(CNC(CSCCC(C)C)=O)CC(C(=O)N2CCOC3CC23)=NO1 N1(C(C2COCCN2C(C23COCC2C3)=O)=O)CCC(F)(F)C(O)C1 N1(C(Cn2c(C)c(Cl)cn2)=O)CCC2CCC(C1)N2C(C1CCCC2C1C2(F)F)=O C12(C(C)=O)CCCC1(C(=O)NC(C)(C)CCNC(c1csc(C(=O)N(C)C)n1)=O)C2 c1(OC)nn(C)cc1C(=O)OCCC(O)c1cccs1 N1(C(C(C)=C2CCC2)=O)CCC(CO)CC1C(=O)NCC1([Si](C)(C)C)CC1 N(C1c2ccccc2CC1NC(c1nc(=O)n(C)[nH]1)=O)C(CC=CCC)=O C1(NC(=O)CC2CCCO2)CN(C(C2(C3NC(=O)NC3=O)CC2)=O)CC1F c1(CN2CCC(CN(c3csc(Br)c3)C(=O)O)CC2)cccc2nccnc12 c1(C(=O)NCCN(C(c2nnc(C(C)C)s2)=O)CC)c(C)nn(C)c1OC C1(NC(=O)NC2CCN(c3nc(OC)c(Cl)cn3)CC2C)CCCC(C)(C)CC1 C1(CNC(=O)Nc2ccc(OC)cc2)CC(C)CN(Cc2ccncc2Cl)C1 Nc1ccc(C(N2CCC(NC(C3CCS(=O)(=O)C3)=O)C2)=O)nc1 N1(C(CCN(C)CC)=O)CCC(C2CC(NC(c3cccnn3)=O)C2)CC1 N1(C(C)=O)CCC(C)(C(=O)NC2CN(C(c3ccsc3C#N)=O)CC2C)C1 C(=O)(CCC(=O)C(C)(C)C)N1CC(C(=O)NC2CCc3nnnn3C2)CC(C)C1 NS(=O)(=O)c1cc(C(N2CC3CCN(C(c4cc(Cl)c[nH]4)=O)C3C2)=O)co1 c1(C(=O)NC2CN(C3CN(C(C(=O)NC)=O)C3)C(=O)C2)cc(C)c(C#N)cn1 S(=O)(=O)(c1ccc(NC2CCn3cncc3C2)nc1)NC(CC=O)CN C1(C(=O)NC2C(N3CCN(C(c4cc(C)on4)=O)CC3)CC2)C(F)(F)C12CCC2 Nc1ccc(F)c(C(=O)NCCOC2CCN(C(=O)C3=C(Cl)CCC3)CC2)c1F CCC(CC)(CCN(C)C(C1CC(O)CN1C(=O)C(C)C1CC1)=O)OC C(CCC)(C(=O)NCc1cn(CCNC(=O)Cc2cc(C)nn2C)nn1)=CCC CC(CNC(C1COC(=O)N1)=O)CC(=O)NCC1CC1(F)F C1(OC)CC(C(=O)NC(C)COC2CC2)N(C(c2ncncc2C)=O)C1 C1(NC(c2cnc(CC3CC3)s2)=O)CCCCCC1NC(C1(C2CC2)CCC1)=O C1(NC(C2(C)CC2(F)F)=O)(CO)CCCN(C(c2ccn(C(F)(F)F)n2)=O)C1 c1(C(=O)NCC2CC2NC(c2cnnn2C(F)F)=O)cccnc1OCC(F)F N1(C(CCC2N(C)CCC2)=O)CC(O)CC1C(=O)NCCc1nc(=O)o[nH]1 N1(C(c2c(CC)ocn2)=O)CCC(C)CC1CNC(=O)C(C)(C)C(=O)NC Cc1ccc(F)c(C(N2CC(CCNC(c3scc(C)c3Br)=O)C2)=O)c1 C1(CNC(C(CC)Cc2ccc(N)cc2)=O)N(C(=O)CC2CC2)CCCC1(C)C N1(C(CC=CC)=O)CCN(C(c2ccc(CC3CC3)s2)=O)C(C)CC1C N1(C(=O)NC(c2c(OC)cc(F)cc2)C)CCC2(OC)CCCC12 c1(C(N2CC(NC(c3cncc(C)n3)=O)C(O)C2)=O)c(Br)ccc(N)c1F C1(COC)(NC(=O)Cc2csnn2)CCN(C(c2nccnc2C)=O)C1 c1(C(N2CCC(NC(Cn3c(C)ccn3)=O)CC2)=O)ccnc(Cl)c1F c1(CC)cc(C(=O)OCc2ccc(Br)c(O)c2)cc(N)c1 N1(C(C2CN(C(C)=O)C2)=O)CCOC2(C1)CN(C(=O)CC1COC(=O)C1)C2 C(=O)(NNc1ccc([N+](=O)[O-])c(C)c1)c1nc(C)nn1C1CCOC1 c1(CC)nnc2n1CCCC2C(=O)NC1CC(NC(=O)CC(=O)OC(C)(C)C)C1 C1(NC(C2CCCN(C(c3cc(F)cnc3O)=O)C2)=O)CC2(CCOC2)C1 C1(CNC(CC=C)=O)CN(C(c2cnc(-c3ccccc3)s2)=O)C2CC12 Cc1ccc(N(C)C)cc1NC(=O)Nc1ccc(N(C)C)cc1OC c1(C(N(CC(C)NCCNC(CCC)=O)C)=O)cccc2nc(C(F)F)sc12 C(=O)(C(C(C)C)C(C)C)NC1C(CNC(c2c(C)nc(C3CC3)[nH]2)=O)CC1 C(=O)(C1=NOC2(CCC2)C1)N1CCC(CC)C(NC(=O)OC(C)(C)C)CC1 c1(C(N2C(CN(C(CC=C)=O)C)CCC2)=O)cnn2c1OCC(OCC)C2 C(C(O)C(=O)NCC(C1CCC1)OC)NC(C=C(CC)CC)=O C(=O)(C1=CNC2=NCCCN12)NC1C(C(=O)NCC#C)CCCC1 CN1CCC2(CCN(C(C3CCCCN(C(C4(C)CC5CCC4O5)=O)C3)=O)C2)C1 CC(CC(=O)NCCCN(C(=O)CNC=O)CCO)C(C)(C)C C1(=O)C(C)CCCOC2CN(C2)C(=O)CC2CN1C2.C1(C=C)(CC=C)CCC1 N1(C(C(COC)C)=O)CC2C(CN(C)C(c3sccc3CC#N)=O)C2C1 Nc1cc(Cl)nc(C(=O)NC2CCC2NC(C2CCCC23CC3)=O)c1Cl C1(NC(=O)C=Cc2cccs2)CC2CC1N(C(=O)CC1(O)CCCCC1)C2 C1(C(=O)NCC2CC3(CC(NC(C4(O)CC4)=O)C3)C2)C2CCC3(COC(=O)C13)O2 c1(CC)ncnc(N2CC(C(N3CC4CC3CO4)=O)CC(F)C2)c1F c1(C(C)C)nc(OC)cc(N2CC3C(CNC(=O)CCC4CCCCCC4)C3C2)n1 N1(C(=O)Cc2cncnc2)CC(CO)C2(C1)CN(C(c1cccnc1S)=O)C2 C(=O)(CCC(=O)N1CC(OCCC(N2CC(C#N)C2)=O)C1)NCCC Cc1cc(CCNC(=O)C(C2(O)CN(C(c3cccn3C(C)C)=O)C2)F)no1 CC1(C)CC(O)(C(=O)NCC23CC2CN(C(c2nn[nH]c2Cl)=O)C3)C1 c1(NC=O)nc(O)c2c(-c3ccccc3)csc2n1.C1(O)CCN(CC2CCC(C)N2C)CC1 Cc1ccc([N+](=O)[O-])cc1C(N1CCC2(CCN(c3cnc(C#N)cn3)C2)C1)=O C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCN(C(CNC(CCSCC)=O)C(F)(F)F)CC1 C12(CNC(C3ON=C(C)C3)=O)CCCCC1CN(C(=O)C(C(C)C)C(C)C)C2 Cn1cnc2c(C(N3CC(CNC(C4CC4(C)Br)=O)C3)=O)ccnc12 c1(N2C3CN(C(C(=O)Nc4ncc[nH]4)=O)C(C3)C2)ncnc2occc12 C1(NC(C2C(C)C2(F)F)=O)CC(C)CN(C(=O)C(C2CCC2)C2CCC2)C1 Cc1cc(F)c(CC(=O)NCC(C2CC2)N(C(=O)C(C)C(C)(C)C)C)cc1F CCC(C)(C)CC(=O)NC(C(C(C)C)NC(=O)C1=CCOC1)c1ccccc1 C12CC(=O)N(C1)C1OCCCC(C3CCCOC3)(c3nnnn3C(CC)CC1)NC2=O c1(CC)cccc(CC)c1C(N1CCOCC1CN(C)C(C1(F)CCCC1)=O)=O C1(NC(C=Cc2cn(C)nc2)=O)COCCN(C(=O)CN2CC(C)(C)C2)C1 c1(C(C(=O)NCC2C(C(=O)OCC)CCC2)(F)F)cc(Cl)ccc1Cl CC(C)(CCCO)C(=O)N1CCOC(CNC(C2CCCC23CCC3)=O)C1 CC1(C)CN(C(=O)CC2(O)CCOC2)CC1NC(c1cccn2cnnc12)=O N1(c2cc(CC)nc(C)n2)CC2CC(NC(=O)C(C)SC)CC1C2 c1(NC(C(=O)CCc2ccc(C(=O)OC)nc2)=O)nc2c(s1)C(=O)CCC2 O=C(C1CCc2c[nH]nc21)NCC1(F)CCC(NC(=O)CCc2nccs2)C1 c1(-c2c(F)ncc(SC)c2)c[nH]c2cc(C(=O)N(CCO)CCO)ccc12 C1(C(N2CC(=O)NCC2)=O)C2Cc3cc(Cl)ccc3C12.C12=CC=C(C=C1)C2 c1(CNc2ccc(CC)c(C)c2)cccc2ccccc12 N1(c2c(-c3cc(Cl)c(O)cc3F)cn(C)n2)Cc2[nH][nH]c(=NC(=O)C(C)(C)C)c2C1 Cc1scc(C(N2CC(NC(=O)C3=NOCC3)C3CC23)=O)c1N N1(C(C2C(C)CCC2)=O)CCC(O)C(NC(=O)CCCc2ccccn2)C1 c1(CC(=O)N(CC(C)NC(=O)C=CC2CCCO2)C)cncc(Br)c1 c1(CC(=O)NC(c2cncn2C)C#C)ccc(CCCC)cc1 N1(C(CCCSC)=O)CCN(C(c2coc(Br)c2)=O)CC(C)(C)C1 C1(NC(C2(CC)CC(C)(C)C2)=O)CC12CCN(C(=O)CC1CC3(CC3)C1)CC2 c1(CC(N2CCC(NC(=O)CC3CC=CCC3)C23CC3)=O)cn2cc(F)ccc2n1 C(CCN(C)C(C1C(C)C1C)=O)(C(C)(C)C)NC(c1cc(C)ns1)=O c1(C(=O)NC2(COC)CN(C(c3cscc3F)=O)C2)cccc(C)c1O c1(N2CCC(NC(c3n[nH]c(C)c3C)=O)C(CO)CC2)cc(C)nc2ncnn12 C(CCCC(=O)NCc1ncccc1C(=O)NCC1CCCC1(C)C)NC(C)=O c1(C(C(=O)NC2CCSC2)NC(=O)Cc2cc[nH]n2)cccnc1 CC1(C#CC(=O)N2CCC(O)C(NC(c3ccc(F)o3)=O)C2)CCCO1 c1(-c2c(OC)n[nH]c2)ccccc1CNC(c1noc(C)n1)C Cc1cc(Br)oc1C(N1CC(CNC(=O)Cc2cnc(C3CC3)[nH]2)C(C)C1)=O N1(C(CC2(CNC(C3N(C)CC(O)CC3)=O)CC2)=O)CC2(COC(C)(C)C2)C1 C1(C(=O)OC)CCN(C(=O)C(C(C)C)NC(C2CC(=C3CCC3)C2)=O)O1 CC1(C)CCN(C(=O)CC(Cl)Cl)CC1CNC(C1CCCOC1)=O C1(C(=O)NCC(CCC)NC(C2CC(OC)C2)=O)CC2CCC(C1)C2 c1(CNC2CCC(C(=O)NCC3CCS(=O)(=O)C3)CC2)cnc(Cl)c(F)c1 CCC(C(=O)N(CCC(=O)N(C)Cc1nc(C)no1)C(C)C)NC(N)=O C=CCN=C(NCc1ccc(C)c(F)c1)NC(c1ccccc1)CF C(=O)(C(COC(=O)CSCCc1cccc(C#N)c1)CC(C)(C)C)OC N1(C(CC(CC)C)=O)CC2CCC(C1)N2C(=O)C(O)c1cnc[nH]1 O=S(=O)(c1ccc(C#N)c(NCCCCCCO)c1)N1CCC(C2CC2)C1 C1(NC(CC2CC(C)C2)=O)CN(C(C2CC3CCC2CC3)=O)C(C)(C)C1 Nc1cc(C(=O)NCC2(O)CN(C(c3ccoc3)=O)C2)cnc1Cl C1(C2CC2)(NC(c2ccc(C)c(O)n2)=O)CCN(C(C2CSCCS2)=O)C1 C1(CC(=O)NCCN(C(C(F)=C(C)C)=O)Cc2ccccc2F)CC(=O)NC1=O C1(CNC(C2CCN(C(CC)=O)C2)=O)CCCCCN1C(=O)CC(C)(F)F N1(C(C(=O)NCC)=O)CC2CS(=O)(=O)CC2(NC(c2cc(C(C)C)no2)=O)C1 C(CC(CC)C(=O)N1CCCC1CCNC(=O)CSCCCC)=CC c1(NCC(C)C(F)(F)F)ccc(S(=O)(=O)N2CCOC(c3ccco3)C2)cc1Br CCC(CC(C)C)C(=O)N(CC(C)CNC(c1cc(OC)ccc1N)=O)C N1(C(c2cc(C#N)oc2)=O)CC2(CCC(NC(c3ccc(C4CC4)s3)=O)CC2)C1 N1(C(c2ccc(CC)cc2F)=O)CC2(COC(C(=O)N(C3CCC3)CCO)C2)C1 CC1(C)COC(C)(C(N2CCCC(O)(c3ccccc3)C2)=O)CO1 C(C(=O)NCc1ccc(SC(CO)C(=O)O)cc1)(C(C)C)OCC c1(C(=O)NC2C(NC(Cc3c(COC)cccc3)=O)C2)cc(Cl)c(Cl)n1C C1(CNC(C2(C)CC(=O)C2)=O)C2CN(C(=O)C(C)(C)n3cccn3)CC12 c1(C(=O)NC2CCCC(CNC(COCCOC)=O)C2)c(Cl)ccnc1C c1(N(C(C)C)C(C2CC(NS(=O)(=O)CC#N)C2)=O)ccc(Br)cc1F N1(C(C(c2cccs2)NC(c2cc(COC)on2)=O)=O)CCCCC1CF C12(CNC(C(N3CCOCC3)C)=O)CC(CN1C(C1CC3C=CC1C3)=O)C2 C=CCCCCCCC(=O)NCC1CC1CNC(=O)C(N1CCSCC1)C N#Cc1cc(CN2CCN(C(c3ccncn3)=O)CC2C#N)ccc1Cl C(=O)(C(COC)(CC)CC)N(CCN(C(c1cc(COC)no1)=O)CC)CC C1(CCCNC(CC(C)n2cccn2)=O)CCN(C(=O)CNC=O)CC1 C1(NC(C2CCN(C(C)=O)C2)=O)CCCCC1CNC(c1cc(Cl)ns1)=O N1(C(c2nc(C(C)C)oc2)=O)CCC2CC12C(=O)NC(C(C)(C)O)C1CC1 CC1CCCCC1(CNC(c1ccon1)=O)NC(=O)Cn1nnc(C2CC2)n1 C12(CCCn3cc(CCNC(C(CC=C)(C)O)=O)nn3)CC3CC(CC(C3)C1)C2 c1(OC)ccc(C(F)F)cc1C(N1CCSCC1C1CC1)C(=O)NC1COC1 N1(CCCC(=O)NC2CCN(C(c3cc(C)sn3)=O)CC2C)C(=O)NC(C)(C)C1=O c1(C(=O)NCC2(C)CCN(C(c3c(N(C)C)cccn3)=O)C2)cc(=O)n(C)cn1 c1(N(c2cc(C)no2)C)cc(Br)ccc1S(=O)(=O)N(CCCF)C C(=O)(C(C(C)CC)N(C)C)N1CC(NC(C(C)OCC#C)=O)C(C)C1 C1(C(N(CCC)CCNC(C2(C(N)=O)CCC2)=O)=O)CCCN(C(=O)NC)C1 c1(CNC(C(C(CC)C)C)=O)nc2c(s1)CN(C(c1cc(Br)n[nH]1)=O)CC2 C1(C)(CCCC)NC(=O)N(CC(=O)NC2(C3CN(C(=O)CC4CC4)C3)CC2)C1=O C(=O)(NNc1cc(Cl)ccc1Br)NC(C)Cc1cccc(C#N)c1 N1(C(CCCCNC(=O)C=CC(F)(F)F)=O)CCc2nc(O)[nH]c2C1 CN1CCC(C)(C(=O)NCC2CC(NC(=O)Cc3ccsc3Cl)C23CCC3)CC1 c1(N(C(C)C(N2CCNCC2)=O)C)cccc(CN2CCN(CCCO)CC2)c1 CC1CCN(C(=O)CC(=O)NCC2CC2)C1CNC(=O)Cc1ccco1 c1(C(N(CC(=O)NC(C(=O)NC(C)C)C2CC2)CC)=O)cc([N+](=O)[O-])c[nH]1 N1(C(C(=O)NC2CCN(C(C(CCSC)C)=O)CC2F)C)CCc2ccccc21 C(CNC(=O)C(C)NC(=O)C(C)(C)C)(CCCC)NC(CCC=C)=O N1(C(C2C(CC)C2)=O)CC2(C=C(C(=O)NC3(CO)CC(O)C3)CO2)C1 C(=O)(C1=CCN(C(=O)C(C)=C2CCC2)C1)N1CC(SCCC)C1 CC1CCC(NCC(N2CCC(CF)(NC(=O)C(c3ccc(Cl)s3)C)C2)=O)CC1 c1(C(=O)OC)ccc(C(=O)NCc2c(F)cccc2Br)c(F)c1 N1(C(Cc2c(C)nc(S)s2)=O)CCCCC2C(NC(C3CN(C4CCC4)C3)=O)C12 C1(CN(C(C2(C#C)CC2)=O)C2CC2)CCC(NC(C23CCC(CO2)C3)=O)CC1 C(C(C)(C)CC(=O)NC(C)(C)C(C)NC(=O)Cc1c[nH]nc1C)OC N1(C(C(=O)NCC)=O)CCC2(CC1)CC2NC(c1cnc(C2CC2)[nH]c1=N)=O N1(C(COCC#C)=O)CCCC(C2CC2NC(=O)Cn2nc(C)cc2C)C1 N1(C(c2n(CC)nnc2)=O)CC(C(=O)NC23CC=CC(C2)OC3)CC(C)(C)C1 c1(N2CCOCC(NC(C3CCc4cncn4C3)=O)C2)ccc(Cl)cc1[N+](=O)[O-] C(C(=O)N(CC(N1CC2CC1CS2=O)=O)C1CCC1)(C(C)(C)C)N(C)C C1(C(N2CCCC(n3cc(CC(C)O)nn3)C2)=O)CC(=O)N(c2ccccc2F)C1 C1(CNC(=O)CCc2ccccc2Cl)CCCN(C(C2CC(=O)N(O)C2)=O)CC1 C1(C(N2C(C)C(C(=O)NC3CC(CO)N(C)C3)CC2)=O)CCC(O)CN1C CCCC(CNC(c1ccn(C2CC2)n1)=O)C(=O)N1CC2CC1CO2 c1(C(=O)NCC2N(C(CC(C)(F)F)=O)CC(O)C2)cc2c(Cl)nccc2o1 Cc1ccc(Cl)c(N)c1C(=O)N(C(C)CCNC(=O)CC1CCCC12CC2)C CC1CC(CNC(=O)CCNC(c2ccncc2)=O)CN1C(=O)Cc1cnc[nH]1 c1(OC)ncc(COC2CN(C(=O)C(C)(C(C)C)NC(C)=O)C2)c(C)n1 C1(NC(COCCOC)=O)CCN(C(c2cnc(N(C)C)nc2)=O)CC1O N1(C(c2sccc2F)=O)CC2COCC2(C(=O)NCC23CCC(CC2)CC3)C1 Cc1ccnc(N2CC3C(C(=O)NCCc4cnn(Cc5ccccc5)c4)C3C2)n1 C1(C(N2C(C(C)(C)NC(C3C(C)(C)C3(F)F)=O)CCC2)=O)COC(C)(C)CO1 c1(CC)ncc(C(=O)NCC2COCC2NC(=O)Cc2cccnc2)s1 N(C1c2ccccc2CC1O)c1cc(-c2c(S(=O)(=O)NC)cccc2)c(F)cc1 N1(C(CCNC(=O)OC)=O)CCCC(C2CC2NC(=O)CCS(C)=O)C1 Nc1cc(C(N2CCOCC2CNC(c2cnn3c2CCC3)=O)=O)ccc1Br C#Cc1cccc(C(=O)NCCNC(c2cnn(C3CC3)c2)=O)c1 CC1CN(C(c2cn(C)nc2CC#N)=O)CC1CNC(c1ccn(C(F)F)n1)=O C(=O)(C(O)CC(F)(F)F)NC1CC(CNC(C(c2ccccc2Cl)OC)=O)C1 C1(N(C(C(C(=O)OCC)OC)=O)CC(=O)NCCCN=[N+]=[N-])CCCCC1CO C(=O)(CCCCCC#N)N1CC(CCCC)N(C(c2cc3c(s2)CCC3)=O)CC1 c1(N(C2(CNC(C(CCC)NC(N)=O)=O)CC2)C)nc(Cl)nc(C2CC2)c1F C(=O)(CC1CCc2cc(Br)ccc21)N1CCN(C(CC(=O)OCC)=O)C(C)C1 C(c1ccc(O)cc1)=CC(N1C(C)CC(NC(c2ncoc2C2CC2)=O)C1)=O N1(C(C(C(C)C)C)=O)CCC2(CC1)CCN(C(C1Cc3ccccc3N1C)=O)C2 c1(NC(CNCC2(CS(N)(=O)=O)CC2)=O)cc(F)cc(F)c1 S(=O)(=O)(c1cnn(C)c1)NCC(=O)N(C1CN(C(=O)CNC=O)CC1F)C Cc1cc(C#N)cc(C(=O)NC(C)C(C)NC(=O)CNC(=O)CC(F)(F)F)n1 CC1(CO)CC(F)(F)CN1C(c1ccc(C2CC2)o1)C(=O)Nc1ccccc1Cl N1(C(COC(CC)C)=O)CCN(C(=O)CCC2CCCCCC2)C(CC(F)F)C1 C1(=O)C(CC2CN(C(C3COC(C(=O)NC)C3)=O)C2)N1.CCC(CC)C1CC1 C#CCC(C(=O)NC)NC(=O)CCC1CCN(C(C2CN(C(C)C)C2)=O)C1 c1(C(=O)NC(C2CCN(C(c3c(C)nccn3)=O)C2)C)cc2cnccc2[nH]1 c1(C(C)C)cnc(O)c(C(=O)NC2C=CCN(C(=O)Cc3cccnc3)C2)c1 C1(CNC(c2cc(-c3ccc(F)cc3)[nH]n2)=O)C2CN(C(=O)CCCF)CC12 N1(C(C(COC)N(C)C)=O)CCCC(C2CN(C(=O)Cc3csnc3C)C2)C1 Cc1ncc(F)c(N2CCN(C3CCCC3NC(=O)C(C)CSC(F)(F)F)CC2)n1 Cn1nc(C2CC2)cc1CC(N1CCC(F)(CNC(c2cnn(C(F)F)c2)=O)C1)=O Cc1sccc1CNC(=O)CC(C)N(C)C(c1cocn1)=O C12(CCC(C)(C)C1)C(=O)N2.N1(CCN(CCOC)CC)CCCCCC1 c1(NC(C(C)(C2CCC2)NC(CN(C(C)C)C)=O)=O)cnncc1O C#Cc1ccc(F)cc1C(=O)NC1CCN(C(=O)Cc2ccns2)C(C2CC2)C1 C1(C(N(CCOCCN(C(C=CCC)=O)C)C)=O)CC(C(C)=NO)C1(C)C Cc1n[nH]c(C)c1CCC(=O)NCC1C2CN(C(c3ccoc3C(C)C)=O)CC12 CC(C)CC(O)C(C)C(=O)N1CCC(C)(CC(N2C3C=CCC2CCC3)=O)C1 C1(NC(C2(C(C)N)CCCC2)=O)CC2(CCN(C(c3nccn3C)=O)C2)C1 C1(CNC(C=CC(=O)OCC)=O)CCCN(C(c2nc(C(F)(F)F)sc2C)=O)C1 C(=O)(C(CCC)CC(C)C)NCC1C2CN(C(C(CC#C)C)=O)CC21 c1(NC(CCN(C(CS(=O)(=O)N(OCC)CC)=O)C)C)cc2nnc(C)n2cn1 Cc1c[nH]cc(C(N2CC(CCCCNC(C3CC4CCCC34)=O)C2)=O)c1=O c1(C(=O)NC2CN(C(CCCCOC)=O)CC3(C2)CC3)cnn2c1OCC(O)C2 c1(C(=O)NC2CN(C(C(C)CC(N)=O)=O)CC(F)C2)ccc2cnoc2c1 C=C(C)C1CN(C(=O)C(F)CC2(C3NCC3)CC2)CCO1.C(=O)C(F)OC(F)(F)F n1(CC)ncc2cc(C(N3CC(C)N(C(=O)C(C)=CC(C)(C)C)CC3C)=O)cnc12 Cc1ccn2ncc(C(N3CCN(C(c4c(C5CC5)noc4C)=O)C4CC34)=O)c2c1 N1(C(CCCOC(C)=O)=O)CCC(C2(NC(=O)CN3CCC3C)CCC2)CC1 c12cc(Br)cnc1N2.N12CCC(O)C1C2=O.CCCS(=O)(=O)NCC(F)(F)F c1(CC)ncnc(N(C)CC2CCCCN2C(=O)CC2CCNC(=O)C2)c1F c1(OC(CSCC(N2CCC(NCc3n(C)ncn3)C2)=O)=O)ccc(Cl)cc1 C(=O)(C(Cn1cccn1)N)NC1C(C(=O)OC(C)(C)C)C1.C(C(=O)OCC)=CCC C(c1ccc(C#N)cc1)=CC(=O)NCC1C(NC(c2cnn(C)c2F)=O)C1 C#CC1CN(C(=O)C(CC)OCC)CCN1C(=O)C=Cc1cc[nH]c1 CC(C)(C)CCC(=O)NCC(C1CCCC1)NC(=O)CC1CC2CCC1O2 C1(CNC(C(C2CC2)SC)=O)CCCCCN1C(=O)COCC(F)(F)F Nc1c(O)ccc(Cl)c1C(=O)NCC(O)CNC(=O)CSc1ccsc1[N+](=O)[O-] N1(C(C(CCOC)C)=O)CCC(F)(CNC(C2CN(C)CC2C)=O)CC1 C1(CNC(c2cncc(F)c2)=O)CC2(CCN(C(=O)COCCCF)CC2)CO1 C1(N(C(c2n(CC)ncn2)=O)C)CCN(C(=O)Cn2ccc(C3CC3)n2)CC1C C1(CNC(C(=O)NCCOCCCC)=O)(NC(=O)C(CC)SC)CCC(C)(C)C1 C1(C)(NC(CCC2CC(OC)C2)=O)CCN(C(=O)CC2CC(C)(C)CO2)CC1 C=C=C(C)CC(=O)N1CCOC(CNC(c2cc(C)n(-c3ccccc3)n2)=O)C1 C#Cc1c[nH]nc1C(=O)NC(C)C(=O)OC(C)(C)C.C12(C)CCN(C1)C(=O)OC2 c1(C(C(=O)NC(CC)(C)C)N(C2CCN(C)CC2)C)ccc(C)c(OC(F)F)c1 c12ccc(cc1F)c(=O)[nH]2.c1(SCCN(C(C)=O)C(C)C)cc(C(=O)O)ccc1Br CCC(F)(F)CC(=O)N(C)CC1CCCN(c2nc(CC)ns2)C1 CC1(C)CCN(C(c2ccc([N+](=O)[O-])o2)=O)C1CNC(C1CCCC2(CC2)C1)=O Cc1ocnc1CC(=O)NC1(CF)CN(C(=O)C(C)CC2CCCC2)C1 c12cccc(c1)NC(=O)NCC2.C(C(=O)OC)NC(=O)NC N1(C(Cn2nnc(C)n2)=O)CC2(C1)SCCC2NC(c1ccc2nn[nH]c2c1)=O N1(C(C=CC)=O)CCC(NC(c2csc(C(C)OCC)n2)=O)C(CC)C1 CCCCCCCC1CC(c2nnnn2C2CC2)(NCCCc2cn(C)nn2)C1 C1(CC(=O)NCC(C)(CO)NC(COCc2n(C)ncn2)=O)CCCC1(F)F C1(C(N(CCCNC(CC(C)C)=O)C)=O)C(C)CCN1C(=O)OC(C)(C)C CC(CNC(c1cnc[nH]c1=N)=O)CC(=O)N=c1cc2ccccn2[nH]1 C#CCCCCCCC(=O)NCC1CN(C(c2nnnn2CC)=O)CC12CCC2 N1(C(C2CC(OC)C2)=O)CC2(C1)C(NC(=O)C=CC(C)(C)C)CCS2(=O)=O C1(OC)CCC(C(=O)NCC(C2CCOC2)OC)C1.n12cc(nn1)C2 c1(OC)cc(C(=O)NCC2(C)CN(C(c3coc(Cl)c3)=O)CCO2)cc(F)c1F C1(C(=O)NCC(C2CC2)SC)CCN(C(=O)CC2CCC(C)(C)C2)CC1 C1(CC(=O)NCc2cc(C(N(CC(COC)(F)F)C)=O)no2)CCCN(C)C1=O c1(SCC(=O)OCCCC(C)(C)C)cc(Cl)ccc1Br N1(C(c2c(COC)scc2)=O)CC(NC(=O)CC2CC(SC)C2)CC1C C1(C(N(CCNC(c2nccnc2C)=O)CC)=O)CCCC2(CC2)C1 N1(C(CC(C)(C)OC)=O)CCC2(C=C(C(=O)N3CCC3c3ccccc3)C2)C1 c1(C(N2CC(O)(CCNC(c3cnn(C)c3Cl)=O)C2)=O)c(N)ccc(F)c1F CC(C)CC(C)C(=O)NC1(C(N2CCN(C(C)C)CC2)=O)CC(O)C1 C1(C(N(c2cc(O)nc(C)n2)CCC)=O)Cc2cccc(C)c2O1 C(=O)(CCCCC(C)(C)C)N1CC(C)CC(C(=O)NCc2c(C)c(F)ccc2)C1 C(=O)(CCCCC(=O)NC1CCN(C(c2cnc(S)[nH]2)=O)C(C2CC2)C1)NC C1(NC(c2nccnc2Cl)=O)CCCC12CN(C(C1CCC3C(C1)C3(F)F)=O)C2 c1(OC)ccc(C(=O)NCCC2CCCN2C(=O)CCCC2(C)N=N2)c(Cl)c1 C1(CNC(CCCOC(C)C)=O)CCN(C(=O)C(N2CCCCCC2)C)C12CC2 c1(C(N2C(CN(C)C(c3cn(C)ccc3=O)=O)COCC2)=O)cc2n(n1)CCC2 O=C1CC(C(=O)NCC2CCCC(NC(=O)CN3CCC3)C2)=NN1 Cc1ncc(C(=O)NCC2COCCN2C(C2CC(C)(O)C2)=O)c(C)n1 N1(C(C=C(CC)C)=O)CCC2C(CCN2C(c2ccc(=O)n(CC)n2)=O)C1 C1(C(NOCCOC)=O)CCN(C(=O)CCc2ccco2)C1 CC(C)CC(CC(=O)NCCCn1ccnn1)NC(C1CC=CCC1C)=O C1(C(N(C)CCNC(=O)CCN2CCC(F)C2)=O)CC2CC(O)C(C1)C2 c1(CC(=O)NCC2CCN2C(=O)CSC2CC2)ccco1 S(=O)(=O)(c1cccc2c1NCCC2)NC(c1cccc2cccc(Br)c12)=O N1(C(C2CCC(C)O2)=O)CC2ON=C(CNC(C3CC4CCC3CC4)=O)C2C1 N1(C(c2cc(SC)oc2)=O)CC(C)CN(C(C2CN(C(N)=O)C2)=O)CC1C C(=O)(CCC(C)NC(c1ccc(OC)o1)=O)NCC(C(=O)OCC)C C1(NC(C(C(=O)OC)OC)=O)CC=C(C(=O)NCC(C)(C)OCCO)C1 CC1CN(C(=O)C(C)Cc2cnc[nH]2)CCCN1C(c1ccn2ncccc12)=O C12(NC(C(C)=C3CCC3)=O)CCCC1N(C(c1[nH]c(O)nc1C)=O)CC2 C(C)(C(C(=O)NCC1CCCCN1C)NC(C1CC2(CC2)C1)=O)OC C1(NC(CSCCCC)=O)CCCC(CNC(C2CC(n3cnnc3)C2)=O)C1 N1(C(C(=O)NCCSCC=C)=O)CCN(S(=O)(=O)N(C)C)CC1 C1(NC(C=CC2N(C)CCC2)=O)CN(C(=O)CC2(CO)CCC2)CCC12CCC2 c1(C(=O)NCCC2CN(C(c3onc(C)n3)=O)C2)cn(C(C)(C)C)nc1C CC1=C(C(=O)N2CCC(=CCNC(=O)CCc3cnc[nH]3)CC2)SCCO1 C1(CC)CCCN(c2nnc(C3CNC(=O)C3)n2CCCOC)C1 CC1CC(C(=O)NC(=O)C(C)NCCS(C)(=O)=O)CCN1C(=O)C=CC1CC1 C1(NC(C23OCC(C)(C2)C3)=O)CC2CN(C(c3cnc(Cl)cn3)=O)CC2C1 C1(N(C(=O)CCC2CCCN2C(=O)CCc2ccncc2)C)CC(CO)N(C)C1 N1(C(c2cnn(C)n2)=O)CC(C)(C)OCC1CNC(c1c[nH]nc1Br)=O N1(C(CC(CC)O)=O)CCC2(CCCN2C(c2cc3cccn3cn2)=O)C1 C(N=c1[nH]cnc(Cl)c1C(C)C)C1C2CN(C(c3scc(COC)c3)=O)CC21 c1(-c2ccc(C)cc2F)ccc2c(c1C(=O)NCC(=O)N(C1CC1)CC1CC1)OCO2 Cc1ccc(O)c(N(C2CC(C)(c3nn[nH]n3)C2)C(C(=O)OC(C)C)=O)c1 Cc1cc(CN(C(c2cnccc2C)C(=O)Nc2ccccc2)C)c(F)cc1Br C12(CNC(C(C)CN(C)C)=O)CCC(NC(=O)Cc3ccc(O)nc3)(CO1)C2 c1(C(=O)OC)cc(C(N2CCC(O)C2)C(=O)NC2CCCC2)n(C)n1 C(c1ccc(F)c(F)c1)=C(C(N1CCC(NC(c2cnc(SC)s2)=O)C1C)=O)C C1(C(N(CC(=C)C)C)=O)COCCC1NC(=O)CC12CCC(CC1)C2 N1(C(C(c2cccs2)SC)=O)CC(CNC(=O)C(COC)OC)C2CCCCC12 C1(CCNC(Cc2ccc(C)s2)=O)CN(C(=O)CC(C)C)CCO1 c1(CC)ccncc1NC(=O)CCCNC(=O)C=CC(C)(C)SC N1(C(C(CC)CCOC)=O)CCCC2(CCCCC2NC(C2C=CCC2)=O)C1 c1(C(C)=O)ccc2cc(C(=O)NCc3cnc(C)c(C#N)c3)[nH]c2c1 c1(CC(N2CCC(CCNC(C(C)(C)SC)=O)C2)=O)ccc(C)nc1Cl CC(N=C(NCCOCCS)NC(C)CCC(C)(C)C)c1ccccc1 CCCC(O)(CCC)CC(=O)N(C1CCN(c2nc(Cl)c(C#N)s2)C1)C C1(NC(CC(CN(C)C)O)=O)CN(C(c2c[nH]c(=O)cn2)=O)CC2(CCC2)C1 n1(C(C)C)cnc2c(N3CCOC(C)C3)nc(C(F)(F)F)nc12 C1(NC(C(COC)(C)O)=O)COC2CN(C(C3CC4(CCC4)CO3)=O)CC12 c1(CN(C)CCc2ccon2)cn(CCOCC(=O)NCC2CCC2)nn1 C(=O)(C1CCC(=O)c2ccccc21)N1CCC(C(C)C)CC1.C1(=O)CC(C)N1 C1(NC(C2N(C)C(=O)NC2)=O)COC2(CNC(c3ccc(O)cc3F)=O)CC1C2 C1(C(=O)NC(c2cnn(C)c2)C(=O)NC(C2CSC2)C)CCC2(CC2)C1 C1(C(=O)NC(C(=O)NC(c2ccccc2)C#C)CC2CC2)CC(C(C)C)=NO1 CCC(C)C(O)C(C)C(=O)N1CCC(CC(=O)NCCCC2CC2)C1(C)C c1(C(N(C(C)C(=O)NCCCn2ccnn2)CCC)=O)nccc2[nH]ccc12 c1(CC(=O)NCCCC(C)NC(C(C2CCOC2)OCC)=O)cn2ccsc2n1 C(CC(C)(C)NC(c1csc(C(C)C)n1)=O)NC(C(C1CC1)OCC)=O C=CCCCCCN1CCC(C(C)NC(=O)C(c2ccc(F)cc2)C)C1 N1(C(CSCC)=O)CCCCC(CNC(c2cc(C(F)F)no2)=O)C1 c1(CCC(N2CC(NC(C3(C(F)(F)F)CC3)=O)C(O)C2)=O)csc2ccccc12 C1(CCNC(C2C(C=C)C2)=O)CCCCN1C(=O)C=C1CCOCC1 n1(CCC)cc(C(=O)NCC(C)CNC(c2cc(C)oc2C)=O)c2ccccc12 c1(C(=O)NCCC(C)NC(CSCC(C)C)=O)ccccc1C(N)=O N1(C(OCC(c2cccc(CC(F)(F)F)c2)(C)F)=O)CCCC(C#CC(=O)O)C1 Cc1cc(C(=O)N(CC(C)NC(C2(C3CCC3)CCC2)=O)C)c(O)c(C)c1 Cc1ccc(C(=O)NCC(C)(O)CNC(=O)CC2CCC2C)c(F)c1F C1(CNC(CCC=CC)=O)CN(C(=O)CCc2csc(-c3ccco3)n2)CCO1 C(C(C)(C)CC(=O)N(C)CC1C2CN(C(c3ccc(C(N)=O)o3)=O)CC12)OC CC1CCCN(C(=O)CN(C)C2CC2)C1C(=O)NCC(Cl)C(C)(F)F C1(CNC(C(CC)CC2CCCC2)=O)CC2CCC1N2C(c1ncc(Br)cn1)=O Cc1cc(C(=O)NC(CNC(=O)CSc2nccn2C)C(C)C)ncc1C(F)F N1(CCC(=O)N(C)Cc2cc(CS(C)(=O)=O)on2)CCc2ccccc21 C(=O)(CN=c1ccc(Cl)n[nH]1)NCC1N(C(C(C)C(C)(F)F)=O)CC1 c1(C(=O)NC(CNC(C2(CCOC)CC2)=O)C2CC2)nn(C)nc1C C1(NC(c2n(C)ccc2)=O)CC2CCC1(NC(=O)CN1CCCCCC1)C2 N1(CC=C)CCN(C(C2CCCN(C(C3(CC)CCCC3)=O)C2)=O)CC1 c1(-c2cnc(C(=O)NCC3CCCCC3O)nc2)ccc2occc2c1 c1(C(N2C(CCOC)CCCC2)=O)c[nH]c2nc(F)ccc12 c1(C(=O)NCCCC(C)NC(c2ccoc2Cl)=O)occ2c1CCCC2 c1(C(=O)NCC2(C)OCCN(C(C(C)C#N)=O)C2)cc2cc(F)ccc2cn1 N1(C(C=Cc2ccc(C)o2)=O)CC2CC(NC(C3(C(C)C)CC3)=O)CC1C2 c1(OC)ccc(C(N2CC(NC(c3cccc(C)n3)=O)CC(C)C2)=O)cc1O C(=O)(CC(CC)C(=O)OC(C)(C)C)NC(CCCNC(CN(C(C)=O)C)=O)C N1(C(CCCCC#C)=O)C2CCC1CC(CCNC(=O)C(CC(C)C)N(C)C)C2 Cc1ccccc1SCC(N1CC(CO)(NC(C2CC(=O)N(C)C2)=O)C1)=O N1(C(C(CC)n2cccn2)=O)CCC2(CCCN2C(=O)CCC(F)(F)F)CC1 N1(C(C=CC(=O)NC(c2ccc(F)cn2)(C)C(=O)O)=O)CCc2sccc2C1 N1(C(C2CCN(C(c3ccc(C)cc3Cl)=O)C2(C)C)=O)CCn2nncc2C1 N1(C(C=CC(CC)C)=O)CCSCC1C(=O)NCC(C)(F)F CCCC(CCCNC(=O)C(C)c1ccsn1)NC(=O)CNC=O N1(C(C(CC)C)=O)CCC(C(C)NC(=O)C(c2cnn(C)c2)=O)CC1 C1(N(C(C(C2(O)CN(C(CC)=O)C2)F)=O)C)CC(O)C1(C)C C1(C(=O)NC(Cc2cc(C)[nH]n2)C)CN(C(=O)CC2CC2)C2(CCC2)C1 CC1(C)CCCN(C(C23CC(C2)C3)=O)C1CNC(c1c(F)ccc(Cl)c1O)=O C(=O)(CCC(C)(C)C#N)N(CCCCCC)CCNC(c1cn(CCO)nn1)=O CCC(CC(=O)NCC(C)C(F)C(=O)NC1CCOC(C)(C)C1)C(F)F C(CCCCC(=O)NCC1CC(F)CN1C(=O)C=CCn1cncn1)OC c1(NC2CC(CNC(C(CC)OC)=O)C2)ncnc2scnc12 C1(OC)CC(CNC(=O)C(c2cccs2)NC(=O)CNS(N)(=O)=O)C1 N1(Cc2cccc(C)c2Cl)CCC2CN(c3ncc(C(=O)N(C)C)cn3)CC12 c1(C(=O)Nc2ccc(C(F)F)nc2)ncc(Cl)cc1Br C12(C(=O)NC3CN(C(C(COC)N(C)C)=O)CC3C(F)F)CCN(CC1)CC2 c1(CSC(COC)C)cccc(C=O)c1.c1(SN)nnnn1C C1(C(=O)NC(C#CC)CC(C)C)CN(C(C2CCC2(OC)OC)=O)CCC1(C)C N1(C(CCC2CC(NC(Cc3nc(C)oc3)=O)C2)=O)CCS(=O)C(C)C1 c1(C(=O)NCC(CC(C)C)NC(C2CCC3CC23)=O)ccc(C#N)nc1 C1(C(=O)NC2C(CNC(CN(CC)CC)=O)CCC2)CC2(C1)CC2(F)F Cc1nc(Cl)sc1C(=O)NC1CC(NC(=O)Cc2cc(C)n(C)n2)C1 C(C#CC(=O)NCCCCNC(=O)C(C(C)OC)N(C)C)OCC.CC c1(N2C(C(=O)Nc3c(OC)cccc3Cl)COCC2)nc(C)nc2c1CCC2 c1(Nc2c(OC(C)=O)ccc(CC)c2)c[nH]c2cccc([N+](=O)[O-])c12 Cc1cc2cc(C(N3CCC(CNC(=O)CCc4nccs4)C3)=O)[nH]c2cc1Cl C1(NC(C(CCCC)O)=O)CC(O)(C2CCN(C(=O)CN3CSCCSC3)CC2)C1 C1(C(=O)NCC2CCN(C(C3=NNC(=O)C3)=O)C23CC3)CCC(C2CCCO2)O1 c1(C(=O)NC(CCN(C)C(C2CC2C#N)=O)C(C)(C)C)nc2c(s1)CN(C)CC2 C1(CCSC)COCCN1C(=O)NCc1ccc(OCC(F)(F)F)nc1 c1(C(=O)NC2CC(CCC(=O)N(CCC(C)(C)C)C(C)(C)C)C2)ccncc1Cl C1(c2n(C(C)C)nnn2)(NCc2cccc(N(C)C)c2)CCCN(C)CC1 c1(C(N(CCCNC(CC2(C(=C)F)CCC2)=O)CC)=O)ccc(Cl)cc1C c1(C(=O)NC(C)CCCNC(C2CCCN(C)C2)=O)cnc(Cl)c(N)c1 c1(Cc2nc(C(CC)C)nn2-c2ccnc(Cl)c2)ccc(Br)cc1Br C1(CNC(C(CC#C)C)=O)CCC(C)CN1C(c1cncc(N2CCCC2)n1)=O C(=O)(CCC(=O)c1cc(Br)cs1)NC(C)CNC(C1(NC(N)=O)CC1)=O c1(C(CC(=O)N(C2CN(C(=O)CC3CC4(CC4)CO3)C2)C)C2CC2)ccccc1F C(=O)(CCCCCC#N)NC(CCC(C)C)C(N1CCN(C)CC(C)C1)=O C1(CNC(Cc2cc(C)no2)=O)CN(C(=O)CN(C)C)C2CC12 C1(CNC(c2cc(C)n(C)n2)=O)COCCN(C(=O)Cn2ccnc2C(C)C)C1 c1(CNC(=O)NCC(N2CCN(C)CC2)C(C)C)ccc2ncsc2c1 c1(C(N(CC(C)O)CCNC(C(C=C)(C)O)=O)=O)cnc2sccn2c1=O N1(C(CSCCCC)=O)CCC2CCN(C(c3ccc4ccsc4c3)=O)C2C1 c1(C(=O)NC(CC)CNC(=O)C(C)N(CC(F)(F)F)C)ccc(C(N)=O)cn1 C1(CNC(c2cc(C(=O)C(F)(F)F)c[nH]2)=O)CNCCC12CCOCC2 C=C(CNC(C1CN(C(c2cn(C3CC3)nn2)=O)CC1F)=O)C1CCOCC1 CC12CC(C(=O)NC3CCCC3CNC(=O)Cc3cc(F)cc(F)c3)(CCO1)C2 c1(OC)cccc(S(=O)(=O)NC2CN(Cc3ccnnc3O)CC2F)c1 c1(C(=O)NCC2C3(CN(C(=O)OC(C)(C)C)C3)CC2)cc(Cl)cc2c1CCC2 C#Cc1cncc(C(=O)NCCC2CCC(NC(c3sc(=N)[nH]c3CC)=O)C2)c1 C1(C(N2C(CNC(c3cc(C)n(CCO)n3)=O)C=CC2)=O)CC2(COC(=O)N2)C1 Cc1nc(Cl)ccc1NC(C1CC2CC2N1C(C1CC1(C)C)=O)=O C#CC1(C(=O)NC2CCSC2)CCN(C(=O)C(F)CCCC)CC1 Cc1nc(=N)[nH]cc1C(=O)NCC1CN(C(C23CC(C)C2C3)=O)CC1C(F)(F)F C12(C(N(CCNC(C3(C=C)CC3)=O)C3CC3)=O)CCCCC1CC(F)(F)C2 C1(SC)CCC(C(=O)NCC(O)CNC(=O)CCOC2CCCOC2)CC1 c1(CC(CNC(NNC(=O)C2(N(CC)CC)CCSC2)=O)C)ccc2c(c1)OCO2 c1(OCC(N2CC3(COC)CC2(CNC(C2CC(O)C2)=O)C3)=O)ccc(Cl)cc1F C12(C(=O)NC3CN(C(CCC=CC(C)C)=O)C(C)CC3)C3CCC(CC13)C2(F)F CCCCCCOC(C)C(=O)NC(C)(CNC(C1CCCOS1)=O)CC C(CC(N)=O)(C(=O)NCC1CCC(CCO)CC1)NC(C(=O)N(C)C)=O N1(CC)CCC(NC(c2cccc(F)c2)=O)CC1 C1(C)(CC)CC(NC(c2cscn2)=O)CN1C(=O)CNC(c1ccnn1C)=O Cc1ccc2c(c1)CCN(CC(c1ccc(C)s1)O)C2 C=CCC(C)(C)CC(=O)NCC1CCN1C(C1COCCC1(F)F)=O C1(C(=O)NC(CC(=O)NC)C2CC2)(CC)CCCN(C(c2nc(=N)cc[nH]2)=O)C1 C(C(=O)Nn1nnc(C)c1C)(CC(C)C)C(=O)NC(c1c(C)ncnc1)C C=CC(C)CC(=O)NCC1C=CC(NC(C2(CO)CCCO2)=O)C1 Cc1ccoc1C(=O)NCC(O)C(=O)NCC1CC1c1ccco1 C1(CC(=O)NCCN2CCN(C(=O)CC(F)F)CC2)(OC)CCOCC1 S(=O)(=O)(c1ccc(C)c(Cl)c1)N1CC(N(C(C(=O)NC)COC)C)C1 c1(OC(=O)C(C)(CCC=C)OC)cc(OC)cc(OC)c1 Cc1ccc2sc(C(N3CCN(C(=O)C=Cc4ncco4)CC(O)C3)=O)cc2c1 CCCCC(CNC(c1csc(C)n1)=O)NC(=O)C(C)Cc1cccnc1 N1(C(C(C)S(N)(=O)=O)=O)CC2OCC(NC(=O)C=Cc3cncnc3O)C2C1 c1(OC)cc(C(N2CC=CC2CNC(c2ccc(C)cc2C)=O)=O)cc2ccoc12 CC1(C)Cc2[nH]nc(C(N3CC(CCNC(=O)CCCC4CCCC4)C3)=O)c2C1 CCCCC(O)C(C)C(=O)NCC(O)C(=O)NC1C=CC(C)CC1 N1(C(Cc2ccc(OC)cn2)=O)CC2CC1CC2NC(c1cc(C2CC2)[nH]n1)=O N1(C(C=Cc2c(C)cccn2)=O)CC2(CCN(C(c3cc4n(n3)CC(F)C4)=O)C2)C1 N1(C(CCCOCC)=O)CCC(C)C(NC(=O)CCC2CC2(C)C)C1 C(=O)(CCCc1ncc(C)o1)NCC(C)(C1CC1)NC(CCOCC#C)=O N1(C(C(CC)C(=O)OC)=O)CCC2(CC(NC(=O)Cn3ncnn3)CO2)C1 N1(C(CCOCC#C)=O)CC2CCC(C1)N2C(=O)CCc1csnn1 Cc1oc(C)c(C(=O)NC2(COC)CCN(C(=O)C=CC3CCCN3C)C2)c1C C#Cc1ccc(C(=O)N(C(CC)CC(=O)NC(C2CC2(C)C)CC)C)nc1 c1(OC)cc(I)c(Br)cc1CN(C(Cc1c(C)nn(C)c1Cl)C(=O)O)C=O C1(NC(c2c(OC)nccc2)=O)CN(C(c2nc(C)c(C)s2)=O)CC2(CCC2)C1 n1(CC)cc(Cl)c(C(=O)N(C2CCC(NC(c3cc(OC)cs3)=O)C2)C)n1 C#CC(C(C)C)NC(=O)NCCCN(c1ccccc1)C c1(OC)c(NC(CNC(c2cnc(Cl)c(Cl)c2)=O)C2CC2)ncnc1Cl S(=O)(=O)(c1cccc(Br)n1)N1CCCC(C)(CNC(c2cc(F)cc(Br)c2F)=O)C1 C(=O)(C(C(C)C)C1CCCN(C(C)=O)C1)OC.c12ccc(cc1)C(=O)NNC2=O CCC(COC)C(=O)NCCCCCCNC(c1cnc(C(=O)OC)cn1)=O C12(C(=O)NCC3C(C)CN(C(=O)Cc4cccs4)CC3)C3CCC(CC13)C2(F)F C(C(C)(CO)NC(c1cncn1C)=O)NC(C1CC(C(C)C)C1)=O C1(C(N(C2CCCC2)CC(=O)OC)=O)COCCN1Cc1ncccc1Br C(=O)(C(C)(C)CC(=O)OC)N1CC(CCC)C(C(=O)NCCCSC)C1 c1(-n2ccc(C(=O)NC(C)CN(C)C(C3CC3F)=O)n2)c(Cl)cccc1Cl C(=O)(C(C(C)CC)OCC(C)C)N1CC(N(C(C(C=C)c2ccccc2)=O)CC)C1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)N(c1cc(CC)c2[nH]ccc2c1)C1CC2CC1CN2 CCCCCCCCCCC(=O)NCCOC1CCN(C(=O)C=CS(C)=O)C1 C1(C(=O)NC(C=C)(C)C)CCN(C(=O)C(C2CC2)OC)C12CC2 c1(C(=O)NC(C(=O)NC(c2ccnn2C)C)C2CCC2)cccc(O)c1 c1(CNC(c2cc(Cl)ccc2SCc2ccccc2Br)=O)ccc([N+](=O)[O-])c(O)c1 c1(C(C(=O)NC(C(n2cc(CCSC)nn2)C)=O)O)cccc(Cl)c1 C1(NC(C2(COC)CCC2)=O)CN(C(c2cnn(C)n2)=O)C2(CCOC2)C1 Cc1ccccc1CN(C)C(=O)NCC1CC(CC(F)(F)F)C1 c1(C(=O)NCC2(C)CCN(C(C3N(CC)CC3)=O)CC2)cccn2[nH]c(=N)nc12 O=C1CC(NC(C2(F)CCN(C(C3(c4ncccc4F)CC3)=O)C2)=O)CCN1 CC1CN(C(C2(O)CCC2)=O)CCC1NC(c1cnn(C)c1Cl)=O c1(NC(CCc2ccc(C(N(C)Cc3cnc(CC)s3)=O)[nH]2)=O)ccccc1I C1(CCC(=O)NCC(CNC(=O)C(CSC)OC)OC)CCCCCC1 CC1C(C(=O)N2CC=CC(NC(=O)CCN3CCCC3=O)C2)=Cc2ccccc21 C1(C(=O)NC(C)CC2CCCC2)C=CCN(C(C2CCN2C(C)(C)C)=O)C1 Cn1cc([N+](=O)[O-])cc1C(N1CCC(CNC(C2CC(=C(F)F)C2)=O)C12CC2)=O CS(=O)C=CC(=O)NCC1CCN(C(=O)CCc2cccc(Br)c2)C1 Cc1cc([N+](=O)[O-])ccc1C(=O)NC1(CCCNC(c2ccnnc2C)=O)CC1 c1(C(=O)NC2CC(C)(NC(Cc3cccc(SC)c3)=O)C2)cn(C)c(=O)c(C)n1 C1(C(N(CCCNC(C(CC)=CC)=O)C2CC2)=O)CCc2nc(CC)ncc2C1 c1(OC)ncc(C)cc1C(=O)NC1CC(CNC(=O)CC(C)C)C1(C)C C1(C(=O)NCCC(C)(C)CNC(=O)Cn2cnnc2O)CNC(=O)CC12CCC2 C1(CNC(CCCC)=O)CN(C(c2cnc3n2CCCC3C)=O)CCC12CCC2 CC(C)(CS(=O)(=O)c1cccc(Cl)c1)c1cn(C2CC(NCC3CCCO3)C2)nn1 C#Cc1ccc(F)c(C(=O)NC2CCCC2CNC(C2(C)CCCCC2C)=O)c1 c1(CN(C(c2ccccn2)CC)CC)cc2c(C)cc(Br)cc2[nH]1 c1(CNC(C(=O)NC(C)COc2ccc(F)cc2)=O)cc(Cl)ncc1Cl c1(C(=O)NC2CCN(C(c3nc(C)c(C)s3)=O)C2)cc(=O)c2cc(F)ccc2o1 Cc1ncnc(N2CC3C(NC(=O)Cc4ccc5nn[nH]c5c4)C3C2)c1C#N C#CCC(C)(C)NC(C1C(C)CN1C(=O)C=CC(F)(F)F)=O CC1C(NC(c2ccc(Cl)s2)=O)CC2CCC1N2C(c1sccc1C(F)F)=O C1(C#N)(C(=O)NCc2cc(C(N(C3CC(F)(F)C3)C)=O)n[nH]2)CC=CC1 Cc1nnnn1CC(=O)NCCCC1(NC(c2cnc(C3CC3)o2)=O)CC1 C(=O)(CC(C)(C)CCOC)NCC1CC(F)(CNC(c2cc(CCC)on2)=O)C1 O=C1CCC2(CNC(=O)CC3(C(=O)O)CCCC3)CC3(CC3)CN12 C1(C(=O)NCC2CC(CNC(c3cc(CC)cn3C)=O)C2)CCN(C)C(=O)C1 C(c1ccc(C)cn1)=CC(N1CC(CNC(C=CCOC)=O)C2C1C2)=O c1(C(C)NC(C2C(CN)C2(C)C)=O)cc(OC)ccc1Cl c1(SC)ncc(N)c(C(N2CCC(C)(NC(=O)C=Cc3ccc(SC)o3)C2)=O)n1 C(CN=[N+]=[N-])(C(=O)C(C1C(C)=CCS1)=O)N.C1(C(NC)C)CCC1 C(N=c1nc2sccc2c(N(C)C)[nH]1)C1CC(NC(c2ncco2)C)C1 c1(C(N2C(CN(C)C(C3(C(N)=O)CC3)=O)CCC2)=O)ccnc2c1CC(=O)N2 S(=O)(=O)(c1cnn(-c2c(Cl)ccc(Cl)c2Cl)c1)N1CC(COC)(OC)C1 c1(OCC)nc(NC(=O)NC)co1.C12CCN(C1)C(=O)OC(C)(C)CCC2 C(=O)(CCCCC(C)=O)OC.C1(=O)C(F)C(C)CC(=O)NOCCCN1C C1(C(=O)NCC2(C)CC(NC(=O)C(C3CCCOC3)OC)C2)(OCC)CCCC1 CC(CN(C(=O)CC1(C)CCN(C(c2nccn2C)=O)C1)C)C(F)(F)F N1(C(CCCCN(C)C)=O)CCC(C)(C(N2CCC(CO)C(O)C2)=O)CC1 C1(CNC(Cc2c(C)nccc2)=O)CCN(C(=O)C2=COCCO2)CC1C c1(C(=O)NCCN(C(C(C)C(C)(F)F)=O)CC(C)O)cc2c[nH]cnc-2n1 C(=O)(C1=C(C)OCC1)N1C(C(CC)NC(=O)CSc2cccc(F)c2)CCC1 CC(CS(=O)(=O)c1ccc(F)cc1)C(=O)NC1CC1CNC(C1COC1)=O c1(-c2sc(NC(c3n[nH]cc3[N+](=O)[O-])CC)c(C)n2)ccc([N+](=O)[O-])cc1O c1(N)c(C)cccc1Cl.c1(OC)cc(C(=O)NC2CCCC(NC(=O)CO)C2)n(C)n1 C(C)(CCC(=O)NC(C)(CO)C(=O)N1CCOC(CN=[N+]=[N-])C1)OC N1(C(c2c(C)cc(Br)nc2)=O)Cc2[nH][nH]c(=NC(=O)c3cccc(I)c3F)c2C1 Cc1cc(F)c(C(F)(F)F)cc1CNC(N1CCCC2CC12)=O N1(C(c2n(C)cnc2)=O)CC(NC(=O)CC2CCC2)C(F)C1 C=CCC(CC)C(=O)Nc1cccc(CNC(=O)CC2CCCC3(CC3)C2)c1 N1(C(c2ccc(=N)[nH]c2Cl)=O)CCC2OCCN(C(C3CCCCO3)=O)C2C1 C1(C2CCOCC2)(CNCCCc2c(F)cccc2)CC1 Cc1nnc(C2CCCN2C(=O)NC(c2ccccc2)NC2CCCC2)o1 C1(C(F)(F)F)(OC)CC(C(=O)NC(C2(O)CN(C(=O)C(O)CSC)C2)C)C1 CC(C)(CS(N)(=O)=O)C(=O)N1CC2(C1)CN(C(=O)Cn1nnc3ccccc13)C2 C1(NC(C2(CN(C)C)CCC2)=O)CCCC2CN(C(=O)COc3ccsc3)CC12 C(=O)(C1=CCN(C)C1)NCC(C1CCC1)NC(CC(CC)c1ccccc1)=O C(=O)(C1=CCC(F)(F)CC1)NCCC1(CNC(C(C(COC)C)C)=O)CCC1 Cc1cc(NC(C2NCC(F)C2)=O)cnc1C(F)F CCCCC(C(=O)N(CC)Cc1ccccn1)NC(=O)CC1CCOC1=O Cc1ccc2sc(C(N3CCC(C)(NC(C4CCC4CF)=O)C3)=O)cc2c1 N1(C(c2c(C)ccs2)=O)C2CCC(C2)C1CC(N1CCN(C)CC1CCO)=O C(CCC)(C(O)C(=O)NCC(C1CCCC1)N(C)C)NC(COCCC=C)=O C1(CC)CN(C(=O)Cc2csc3nccn23)CCN1C(=O)Cc1ccc(Cl)s1 N1(C(C(C)(C2CC2)OC)=O)CCC2(CC1)CN(c1ncc(C#N)cc1Br)C2 C1(C(N2C(CC(=O)NCC3C(C)CCC3)CC2)=O)C2CC3C(C2=O)C13 c1(C(N2CC(NC(C(C)NC(CC)=O)=O)C3(C2)CC3)=O)cccc2c(C)[nH]nc12 c1(-c2cc(C(N3C(CCCNC(C=C(C)C)=O)CCC3)=O)sc2)ccc(Cl)cc1 C1(CCC)CCC(C(O)NC(=O)NC(C2CCCC2)C)CC1 C1(C(N(CCOCC#C)C)=O)CCOC1CNC(c1cnn(CC=C)c1)=O c1(C(C)CCc2ccncc2)nc(-c2cnn(C)c2)nn1C1CCCCC1O C1(CNC(C(COCC)C)=O)CN(C(c2nc(O)c(C)s2)=O)CC1C(F)(F)F C=CCC(C)C(=O)NCC1(NC(C2CCC2(C)C)=O)CC(F)(F)C1 CC(C(=O)NC(c1nocc1C(=O)N(C)Cc1cccc(F)c1)C)C(F)F C1(CNCc2c(OCC)cc(Cl)nc2)C2Cc3ccccc3C12 C1(C(=O)NCC(COC(C)=O)O)CCN(C(c2coc(CO)c2)=O)C1 CC(C)CC(C(=O)N1CCC1(C)C(C)C)ONC(c1ccn(C(F)F)n1)=O N1(C(CCNC(C)=O)=O)CC(NCC(N2CCOCC2)C)C2(CCC2)C1 Cc1cc(C2(NC(=O)CCCNC(=O)C=Cc3ccncn3)CC2)cc(C)c1 c1(C(=O)NCC2(CNC(CNC(N)=O)=O)CCC2)cncc(C(F)F)c1 Cc1cc(CN2CCC(F)(C(N3CC4C(C3)C4(F)F)=O)C2)cc2c[nH]nc12 C1(C(N(CC(CN(C)C)O)C)=O)C=CCCN1C(c1cncc(Cl)c1)=O N1(C(C(CC)(CC)OC)=O)CC(Cn2cc(CCN3CCCC3)nn2)OC(C)(C)C1 c1(C(=O)NCCCCN(C(c2cc(C)on2)=O)C)c(C)nn(CCCC#N)c1Cl C1(NC(C(CCC)O)=O)CCC12CN(C(=O)CCCCCc1cccs1)C2 CCS(=O)(=O)CC(=O)N1CC2CC2(C(=O)Nc2ccc(Br)c(Cl)c2)C1 C1(C(N2CC(O)(CCNC(C(C)(C)OC(C)C)=O)C2)=O)CCC12CCC2 Cc1ccc(C(C)(C)C(=O)NCC2CC2CNC(c2cccnc2O)=O)cc1 c1(C(=O)NC2CN(C(c3n[nH]cc3Cl)=O)CC2CC2CC2)cc2ncccc2o1 c1(CC)cc(NC(C2CCCN2C(=O)CC2(OC)CN(C(=O)C3CC3)C2)=O)cnn1 C1(Cn2cc(-c3ccc(C=O)o3)nn2)CCCCC12CCC2 c1(NC(C(N2CC(CNC(C(CC)F)=O)C(O)C2)=O)=O)c(C)cccc1C C1(C)(C(N2CCC(c3n(C)ncc3)CC2)=O)CCN(c2ccccc2)S1(=O)=O c1(CNC(c2nnnn2C2CC2)C2(SCC)CCC2)cnn(C)c1F c1(C(N2CC(CC(C(=O)NCCC)F)C2)=O)cccc(C(=O)O)c1F Cc1ncccc1CC(=O)NCC(C)CN(C(=O)CCCc1nnc(C)n1C)C c1(C(=O)NCC(CCCC)NC(=O)Cc2cc(Cl)cc(Cl)c2)ccc(C)c(C)n1 N1(C(COc2cccc(C)c2)=O)CC2OCC(NC(=O)C(CO)C(C)(C)C)C2C1 N1(C(C(C)C)=O)CC2CCC(C(=O)NC(C)(C)CF)(C2)C1 N1(CC(N)CCC2(O)CCC2)CCOC2(CCSC2)CC1 C1(NC(C(C)SC(C)C)=O)CCC(C)(CNC(=O)Cn2ccccc2=O)CC1 c1(C(N2CC(O)(C(C)NC(C(C3CCOCC3)C)=O)C2)=O)cnn2cnnc2c1 C1(N(C(CCN(CC)CC)=O)CCO)CCN(C(C2(C(C)C)CCCO2)=O)CC1 c1(C(=O)NCCN(C(C2(CC)CC2(F)F)=O)C)cc(C)c2c(c1)CCCN2 N1(C(C#CC2(CC)CC2)=O)C2CCC1CN(C(C1CCC1C(N)=O)=O)C2 C1(CC(=O)NCCC2(C(N3C(C)(CNC(C)=O)CC3)=O)CCC2)CC2(CC2)CO1 C1(CNC(c2nc(C)c(C)s2)=O)CCC2CN(C(=O)C3=CCCC3)CCC2C1 N1(C(c2ccnc(C)n2)=O)CC2CC1CCC2NC(=O)CC1CCC(C)C(C)C1 CCC(C)C(O)C(=O)NC(C)(C)CN(C(=O)Cc1cc(C)cs1)CC C(C(COC)CC(=O)N1CCCCC1CCC(=O)Nc1cc(O)ncc1F)OC c1(C(N(C)CCn2cc(CO)nn2)=O)cccnc1S.C12(CCCO1)C(=O)NC2 CCS(=O)(=O)c1ccc(OC)c(C(N2CCOC(CNC(C3CC3F)=O)C2)=O)c1 CC1(C)CC(CNC(c2ccc(Cl)cc2N)=O)CN(C(=O)CCc2ncc[nH]2)C1 c1(C(=O)NCCOCCN(C(C2CC(C)OC2)=O)C)ccncc1N CCC(F)(F)CCN1CCC(F)(c2cn(C(C(=O)OC)C)nn2)C1 CC(c1cccnc1)=CC(=O)NC1CCCC(CNC(c2[nH]cnc2C)=O)C1 C=C(C)CC(C(=O)N(C)CC)NC(=O)CCC1(C)CC1 C(CN1C(=O)COc2ccccc21)NC(C1CCc2c(ccc(C)c2)O1)=O n1(CC(=O)N(CCCNC(C2CC2CC(C)(C)C)=O)CC)cnnc1 c1(C(N(CC(C)N(C(=O)C(c2cnn(C)c2)O)C)C)=O)cc(O)ncn1 N1(C(c2c(C)csc2)=O)CCN(C(c2cccc(C)c2O)=O)C(C(F)(F)F)C1 C1(C(=O)N(C)Cc2cnn(C)c2)(NC(c2scc(C(C)=O)c2)=O)CCC(C)(C)C1 N1(C(C(NOC)=O)=O)CC2(CCC2)CC1CNC(=O)C(C)(C)CC1CC1 C(c1ccc(F)cc1)=CC(N1C(C(=O)NCCc2n(C)ncc2)C2CCC1C2)=O N1(Cc2c(OCC)cccc2)CC(NC(C2CC=C(C)CC2)=O)C(C#N)C1 N1(C(c2c(OCC(C)C)cccc2)=O)CC(C2CN(C(=O)CC3CC=CC3)C2)C1 c1(C(=O)NC2CC(NC(CC(CC)(F)F)=O)C2)cc2ccc(F)cc2nc1O CC1(C)Oc2cccc(S(=O)(=O)N3CC(CS(C)(=N)=O)C3)c2O1 c1(C(N2CC(NC(=O)CN3CCCC3CO)(CO)C2)=O)ccc(Cl)cn1 C1(NC(=O)CC2CCCS(=O)(=O)C2)CCCCN(C(c2cc(Br)c[nH]2)=O)C1 N1(C(C(C2CCOC2)OCC)=O)CCC(CNC(c2cn(C)nn2)=O)(CC)C1 C1(CC)CCCCCN1CC(=O)NC(C)(C)C.c12ccnn1C2 N1(C(=O)OC(C)(C)C)CCC(C(N2CCCC2C(=O)Nc2cc(C)ns2)=O)C1(C)C C(c1cc2ccccc2o1)=CC(N1CC(C)C(NC(=O)CC2CCOCC2)C1)=O Cc1cccc(CCC(N2CC3C(CN(C(=O)C=Cc4ccco4)C)C3C2)=O)n1 O=C(CCCCCc1ccccc1)NC1CCN(C(C2CC3CCC23)=O)CC1 CC(C)C(C)(F)CNC(=O)C=CCN(C)C(c1cnn[nH]1)=O N1(C(C(c2cnn(C)c2)NC(c2cccc(C)n2)=O)=O)CC2(CNC(=O)N2)C1 c1(C(=O)NCCN(CCCN(C)C)C(c2nc[nH]n2)=O)ccc(CO)o1 CC#CCC(C(=O)NCC1CC(=C2CCC2)C1)NC(=O)CC1CCCO1 N1(C(C(n2c(C)ccn2)C)=O)CC(CNC(c2ccc(C(C)(C)C)[nH]2)=O)C(C)C1 c1(C(=O)NCc2ncc(C)o2)ccc(NC(=O)NC2CCCC2F)cc1 N1(c2nnc(CC)o2)CCC(C)(NC(C2CCC(C)(C)C2)=O)C1 c1(OCC)c(Br)cc(C)cc1S(=O)(=O)NC(=O)NCc1cnc(C(C)C)n1CC C12(CC)CCC(C(=O)N(CCCn3cc(-c4ccsc4)nn3)C3CC3)(CO1)C2 C1(C(N2CCCC(C(C)C)C2)=O)CC2CC1CN(C(c1n[nH]c3c1COC3)=O)C2 c1(CN2CCC(NC(C3CCC(CO)CC3)=O)C2)ccc(N2CCCCC2)cc1 c1(CCC)ccc(C#N)c(NC2CC3CN(C(c4c(OC)cccc4O)=O)CC23)n1 C(=O)(C(C(C)(C)C)Nc1ocnc1C(=O)NOCC=CCl)N(C)C Cc1nn(C)c(C)c1CC(N1CC(CNC(=O)CN2CCCC2C)C(C)C1)=O C=CCC(CNC(=O)C(C1CC1)N(C)C)NC=O.n1(CCC(=O)N)cc(C)cn1 N1(C(c2c(C)cn(C)n2)=O)CC(N(C(=O)C(C)Oc2ccccc2)C)C(C)(C)C1 C12(C(N)=O)CCC(C(=O)NCC3CCCN(C(c4nonc4N)=O)C3)(CC1)CC2 CCCC1C(O)C(=O)NC2CCC3CCN1C23.C(=O)(CCCC(C)CC)N CCC(CC)CCC(=O)NCC1CN(C(C2(N(C)C)CCCC2)=O)CCN1C c1(NC)ccccc1C(N1CCC(O)(CNC(=O)CCc2ccccc2Cl)C1)=O C(=O)(C1=CCN(C(c2cccc(Cl)c2)=O)C1)N1CCC(O)(CC(C)C)C1 C1(C(=O)NC(CNC(=O)CCc2ncc(F)cn2)CC(C)C)(OC)CCCOC1 C1(NC(C(=O)NC2CCN(C)C2)=O)CCC2CC12COC(=O)OC(C)(C)C C1(C(N2CC3CC(NC(C4C(C)CCCC4)=O)C3C2)=O)CC2(C1)CC1(CCC1)C2 c1(C(N(C2CCCC2)CC)=O)c(CNC(C2CC23CCCC3)=O)nnn1C O=C(CCOCCCNC(=O)C=C1CCC1)NOCC=CCl C1(C(N2CC(OC(=O)NCC)C2)=O)C(C2CC2)CCN1C(C12CCC(C1)OC2C)=O N1(C(C(CC)OC)=O)CCOC(C(=O)NC2CCOC2C)C1 N1(C(CSCC=C)=O)CC(C)N(C(=O)CSc2ccccn2)CC1C CC1C(NC(c2cc(Cl)c(Cl)n2C)=O)CC2CCC1N2C(=O)C(F)(F)C1CC1 S(=O)(=O)(c1ccc(Cl)cc1F)NC(C(C(C)C)C)Cc1nc2ccccc2o1 N1(C(c2c(C)ncnc2O)=O)CCCC2(CCCN2C(C2CNC(=O)N2C)=O)C1 c1(CC)cc(NC(C2(C(c3ccccc3)NC(=O)NC)CCOC2)=O)sc1C N1(C(CCCC=C)=O)CCN(Cc2cc(OC)cc(Br)c2)CC1C Cc1ccc(C(=O)NC2CCC2NC(=O)CC(n2nc(C)cc2C)C)nn1 c1(CC(=O)NC2CN(C(c3nc(C)nn3C)=O)CC2C)cnc2c(C)cccn12 C12=NC=CC(=NCC(C)N3CCN1CC3)N2.c1(OC)ccc(SC)c(C)c1OC C1(C)(C(N2CCC(COC)C2(C)C)=O)CN(C(c2ccnc(C)c2)=O)C(C)(C)C1 c1(C(=O)NCCN(C(C2CCCN2C(C)=O)=O)CC)c(C)ccc2nsnc12 C#CC1(CN2CCCC(n3cc(C(C)O)nn3)C2)CCCC1 C1(C(=O)NC(C#CCC)(C)C)CN(C(c2cc(C)sc2N)=O)CC12CCC2 CC(C)C(O)C(C)(C)C(=O)N1CC2(C(=O)N(C)OCc3ccccc3)CC1CO2 Cc1oc(Br)cc1C(N1CCCC1C1(C)CC1)=O N1(C(=O)C=Cc2ccco2)CCN(C(C2CCCS2)=O)CC12CCC2 n1(CC(=O)NC2COCCN(C(C3(n4cncn4)CC3)=O)C2)nnc2c1CCCC2 C#Cc1cncc(C(=O)NC2CC3(C2)CC(CNC(=O)C2=CCSC2)C3)c1 C(c1ccc(O)c(O)c1)=CC(=O)NC1N(C(CC23CC(C)(OC2)C3)=O)CC1 c1(C(=O)NC(CC=C)CNC(=O)CC(=O)NCC(F)(F)F)cccc(N(C)C)c1 CCC(CC(=O)N1CC(NC(=O)CC2(O)CCCOC2)CC2(CC2)C1)C(F)F N1(C(Cn2c(=N)nc[nH]2)=O)CC2(CCC2)CC1C(=O)NC1CCCN(O)C1=O c1(CC)ccc(C(=O)NC2CCCCC2CNC(c2cccc(Cl)c2)=O)c(C)n1 C1(NC(=O)CCNc2ccccc2)CC(O)CN(C(c2cc(Cl)no2)=O)C1 N1(C(Cc2nnc(C)s2)=O)CCCC(CNC(c2cc3ccsc3[nH]2)=O)CC1 c1(NC2C(OC)CN(C(=O)OC(C)(C)C)CC2)cccc2cc(N)ccc12 Cc1ccc(CNCC2(c3ncccn3)CCCC2)c(Br)c1 C12(NC(=O)CCN(C(=O)CC34CCCC3C4)C3CC3)CCCN(CCC1)C2 C1(C(=O)NC2CCC(NC(c3c(C)scn3)=O)CC2)CCC=CCCC1 C(CO)(CC(F)(F)F)NCCCN(C(CC1C=CC(NC(CSC)=O)C1)=O)CCO Cc1nc(Cl)cc(=NCCC2(O)CCN(C(=O)C(C)CC(F)F)CC2)[nH]1 c1(C(N2CC(C3CN(C(C4(C)CCC4)=O)C3)C2)=O)ccc2c(c1)C(=O)CCCC2 O(NC(=O)C(C)N(C(=O)CCCCNC(C1CCC1)=O)C)CCCOC C1(NC(CCCOCC=C)=O)CCCCN(C(=O)CCCC(=O)N(C)C)C1 CC(C)(C#N)CC(=O)N1CCC(CC(N2CCC(C)(CO)C2)=O)C1(C)C C1(NC(C(CC)c2ccccc2)=O)COC2(C1)CN(C(=O)C=Cc1ccco1)C2 c1(CNC(=O)CN2CCC(c3cccs3)C2)ccc(F)cc1Cl.C123CC(C1)(C2)NC3=O Cn1cc(C(N2CC3CC3(NC(=O)CCc3nncs3)C2)=O)ncc1=O c1(NC(C(CC#C)NC(=O)CCC(C)=O)=O)cccc(C#C)c1C CC(C)(CN(C=O)CCC12CCCC1C2)C(N)=O c1(C(=O)NCC(C)(C2CCC2)NC(=O)CCc2cn[nH]c2)ccc(F)c(CO)c1 O=[N+]([O-])c1ccc(CNC(c2nnnn2CCC2CC2)C(C2CC2)C2CC2)cc1 C1(NC(C(C)C#N)=O)CC2CCC1(NC(=O)COc1ccc(F)cn1)C2 C(=O)(C1CCc2ccccc21)NCC(C)(C(C)C)NC(CCC#CC)=O N1(C(C(C)C(F)F)=O)CC2(CCC2)CCC1CNC(C1CC(F)(F)CS1)=O c1(C(N2CCC(CCOC)CC2)C(=O)NCC(F)F)ccc2ncccc2c1 C1(C(=O)NC(C)CC(=O)Nc2ccc(F)cc2)CC2(C1)CC(N)C2 C(C)(C)(C(C)(C)CO)NC(C(C(C)CNC(=O)CN(N(C)C)CC1CC1)F)=O C(=O)(C(F)C(C)(F)F)NC1(CCOC)CCN(C(C2CC2OC)=O)C1 C(C1=NOC2(CCC2)C1)NC(C(N1CCCCC(C)C1)=O)=O n1(C(CC)CC)nc(C(N2CC(N(C)C(C3(C)CCCC3CC)=O)C2)=O)cc1C CC(C)C(C(=O)N1CCC(O)(C(F)(F)C(N)=O)C1)NC(=O)CN(C)C N1(C(C(C(=C)Cl)(C)C)=O)CCCC(C2CCN(C(=O)Cc3cc(C)no3)C2)C1 CC1(C)CC(C(=O)NCCC2COCCN2C(=O)Cc2ccco2)CCO1 C12(C(N3C(CN(C(C(N4CCN(C)CC4)C)=O)C)CCC3)=O)CC(N=[N+]=[N-])C1C2 c1(C(=O)NC(CC(=O)N(C2CCCC2)CC#C)CC=C)cccc2c1CCC2 N1(C(C(CN(C)C)NC(C(C)OC(C)=O)=O)=O)CC(=O)NC(=O)C1C N1(C(c2cnn(C)c2F)=O)CCC2(C1)CN(C(c1cc(CCCO)on1)=O)C2 C1(C(=O)NC2CCCC(NC(C(C)(C)C(F)F)=O)C2)COC2CCCCC12 C=CCC(CC)C(=O)NCC1CCCCN(C(=O)C(C)(C)CCSC)C1 C(C(=O)N1CCCCC1CN(C(=O)Cn1cc[n+](C)c1)C)(C(C)C)NC(=O)NC c1(CC)ccc(NC(=O)CN2CCN(Cc3nc4c(s3)CCC4)CC2)c(C)n1 C(=O)(CN=c1cc[nH]cc1)N(C1CCC(C(N2CC3CC=CC2C3)=O)C1)C C(=O)(C(C)(C)CCNC(=O)Cc1ccnn1C)N(C)Cc1ccncc1 C1(C(=O)NCC(C)N(C(=O)C(C)C2CCOC2)CC)CC2CCC1CC2 C(=O)(C(C)(O)CC)NC(CC)CN(C)C(c1cnc(NC(=O)C2CC2)s1)=O CCC(C)(CNC(=O)CN(C)C(=O)OC)C(=O)NCC(O)C(=O)NC c1(CCC)cc(C(N2CCCC2CCC(=O)NC(C2CCC2)C)=O)ccn1 C(CCCCCC1CC1)NC(C(c1cn(CC)nc1)N1CCCCC1)=O C1(NC(CN(c2ccccc2Br)C(C)=O)=O)CN(C(=O)C(N)=O)CC2(CCC2)C1 N1(C(CCCC#N)=O)CC2(C1)CN(C(c1cc(Cl)ncn1)=O)CC2CO C(=O)(C1CCc2c[nH]nc21)NCCCC(C)(C)NC(=O)Cc1cncnc1 Cc1ccc2c(c1)C(C(=O)NC1(CNC(C3(C4CCC4)CC3)=O)CCOCC1)C2 Cc1cc(CNCC2CC(C(=O)N(C)C3CC3)=NO2)cc(C)c1F c1(C(=O)NCC(C(C)C)NC(c2ccc(C3CC3)o2)=O)nn(C)c2c1CSCC2 N1(C(C=CC(C)NC(C2CCOC2C)=O)=O)CCC(C)C1(C)C c1(C(N2CCC(CNC(C(C3CC3)OCC)=O)C2)=O)cnc(C)c(C)c1 C(=O)(C(C)(C)Cc1ccccc1)NCCCCN(C(C(COC)C)=O)C N1(C(C(C)C2(O)CCC2)=O)CCC(C2(NC(=O)CS(=O)(=O)C3CC3)CC2)CC1 C1(NC(c2cc(C)ncn2)=O)CN(C(=O)CCc2ccncc2)C2(CCC2)C1 c1(CC)ccc(C(N2CCC(O)(CCNC(c3csnc3C3CC3)=O)C2)=O)cn1 Cn1nc(I)c2cc(C(N3CC(NC(c4csc(Cl)n4)=O)CC(F)C3)=O)ccc12 N1(CC(=O)NCC(C)NC(C2C(C(=O)OC)CCC2)=O)C(C)=CC(C)=NS1(=O)=O N1(C(c2c(O)ccc(CC)c2)=O)CCC(NC(=O)CS(=O)(=O)NC)C(F)(F)CC1 c1(NC(C)C)ccccc1C(=O)NCC1(O)CN(C(=O)C(C)(C)C2CCCC2)C1 c1(C(N(C(C)C)CCN(C)C(C2CC(C)(CO)C2)=O)=O)cccc2cnsc12 CC1(CNC(=O)CCC2CCCN(C(c3cn(CCO)nn3)=O)C2)COCCO1 C1(C(=O)NCCC2=CCN(C(C(C(C)(C)C)OC)=O)CC2)Cc2ccccc2S1 Cn1c(Cl)nc2nc(Cl)nc(N3CCCC(C)(NC(C4CC(C)(F)C4)=O)C3)c12 n1(CC)c(C)nn(CC(=O)NCC2CCCN(C(=O)COC(C)=O)C2)c1=O c1(C(N(CCNC(CCCCOCC)=O)C2CC2)=O)cc2c(s1)CCCCC2 CCCC(C)(CCC)C(=O)NCC1CN(C(=O)COCCCOC)CCC1C c1(NCCCSC)cc(NC2COCC2C2CC2)nc(C(C)C)n1 c1(C(=O)OC)ccc(C(N2CCC(N3CCC3CNC(C3COC3)=O)C2)=O)cc1 C1(CNC(C(C)Sc2nncn2C)=O)CN(C(c2nncn2C)=O)CCN1C c1(C(c2n(CCC)nnn2)NC2CC23CCC3)ccc(C(C)C)cc1 C(=O)(C1=CC2(CCOC2)C1)NCC1CC(OC)CN1C(c1cccc(C#N)c1C)=O c1(C(N(C)CCc2cn(-c3cccc(C(=O)O)c3)nn2)=O)n[nH]c2c1COC2 N1(C(c2c(C)cc(F)cn2)=O)CCN(C(=O)C(C)C)C2CSCC12 C(=O)(C(CCC1CC1)ONC(=O)NC(COC(C)C)Cc1ccccc1)OC C(C(=O)N1CC(N(C)C(c2ccc(CC3CC3)s2)=O)C(O)C1)(C(C)(C)C)OC c1(OC)c(F)cc(F)c(C(=O)OC(C)CCc2ccc(O)cc2)c1Br N1(C(C2(SC)CCC2)=O)CCCC(CCNC(C2C(C)(C)C2(C)C)=O)CC1 N1(C(CNC(CC)=O)=O)CCCCC1C(N(C)Cc1csc(C)n1)=O C12(C(N(C3CCC(CO)CC3)C)=O)CCCC1CCN2C(C1C=CC=CC=C1)=O C1(CNC(CC2(OCC)CC2)=O)CC2CCCC2N1C(=O)Cc1cnn(C)c1 c1(C(=O)NCCc2c(CNC(C3C(C)CC3)=O)nco2)cccc2cccnc12 c1(C(N(C(C)CNC(C2(N(C)C)CCCC2)=O)OCC)=O)n[nH]c(C)c1O C1(C(=O)NC(c2ccccc2F)CNC(C=C(C)C(C)C)=O)CC2(CCOC2)C1 C1(NC(CCC(C)N(C(CC2CC(=C)C2)=O)C2CC2)=O)CN2CCC1CC2 c1(N2CCC(C(C)C#N)CC2)ncccc1S(=O)(=O)N1CCCCC1 C1(CCNC(C=C2CCN(C)C2)=O)CN(C(=O)CN2CCC2)CCCO1 c1(C(=O)NCC2(F)CC(NC(c3cc(C(C)=O)on3)=O)C2)onc(C)c1C CC1Cc2ccccc2N1C(=O)CC1CCCCC1NC(c1cnn(C)c1)=O N1(C(c2c(C)cno2)=O)CC2CC2(CNC(=O)C=Cc2cccs2)C1 C(C(C(=O)N(C)CC1(C#N)CCC1)C(C)(C)C)NC(C(C)(C1CC1)OC)=O CN1CCC(=CC(=O)NCC(O)CNC(C2(Cl)CC2(F)F)=O)CC1 c1(OC2(C(=O)NC3C(NC(C(CC=C)(C)CC)=O)CC3)CC2)ccc(Cl)c([N+](=O)[O-])c1 N1(CC(=O)N(C2CCN(C(=O)COc3ccsc3)C2)C)CCCCCCC1=O C(c1cccc(OC)c1)=CC(=O)NC(CCNC(CCC(C)OCC)=O)C C1(C)(CNC(C(COC)(C)C)=O)CN(C(c2ccccc2NC(N)=O)=O)CCO1 C1(NC(C(N2CCC(C)CC2)=O)=O)CCN(C(=O)CC2CC(F)(F)C2)C1(C)C N1(C(Cc2ncc(C)s2)=O)CCCC(F)(CNC(=O)COC2CCCC2O)C1 c1(NC(CCN(C(=O)CC2COCCOC2)CC=C)=O)ccccc1F c1(OC)cc(C)c(C)cc1-n1nc(C(C2CC2)OC)nc1C(C)C(C)O C(c1cc(F)cc(F)c1)=CC(N1CC(CNC(C(CC)C(C)C)=O)CC1(C)C)=O CC(CC(=O)NCCOCCCNC(C1CC12CCCC2)=O)C(F)(F)C(F)(F)F C12(C(=O)NC(C3CC(C)(C)C3)CO)CCC(CC1)N(C(=O)C(C)(C)CC1CC1)C2 N1(C(C(N)CF)=O)Cc2ccccc2C(c2cccs2)C1 N1(C(C2N(C(C3CN(C)C3)=O)CSC2)=O)CCOC2CC12 C(=O)(CCCCC1CC1)N(C(C)CNC(C1CSCCS1)=O)C c1(C(=O)NCCC(C)N(C(=O)Cn2cccc2)C)ccc(-c2ccccc2)[nH]1 CC1CC(CCNC(c2nc(Cl)sc2Cl)=O)CCN1C(=O)CCF CP(C)(=O)C(CC(=O)NC1CCCCC1NC(C1CCNC1=O)=O)P(C)(C)=O c1(C(c2n(C3(C)CC3)nnn2)NC(C2CC(CCCF)C2)=O)ccnc(F)c1 C1(CC(=O)NC(C#C)CCC)CCCC(NC(=O)C#CC2CC2)C1 c1(C(=O)OCC)cnc(NC(C2CCC(C)N2Cc2cc(Br)ccn2)=O)c(Br)c1 c1(C(N2CC3C(Br)C3C2)=O)cc2c(Br)cncc2s1 N1(C(C=CC=CC)=O)CCC2C1CCN2C(c1cc(CC)no1)=O Cc1nn(C)c(N(C)C)c1NC(=O)Cc1ccccc1.C12CCCC1CNC2=O c1(C(=O)NC(c2nccn2C)CC)coc(CNC(c2cc(C)co2)=O)c1 c1(C(=O)NCC(CN(C(C(C)NC(=O)OC)=O)C)C)c(C)cc(F)cc1C C1(C(=O)NCC(C)O)Cc2cc(O)ccc2CN1S(=O)(=O)c1ccc(Cl)cn1 N1(C(c2nc(OCC)oc2)=O)CCCCC1Cn1cc(C)nn1.C(=O)(CC=C(Cl)Cl)N S(=O)(=O)(c1cc(C)cnc1N(C)Cc1cnc(C)cn1)NCC(COC)C C(Cc1cn[nH]c1)(C(=O)NC(c1csc(C)n1)C)NC(C1CN(C(C)=O)C1)=O C(C)(CCCC(=O)NC(CO)C(C)(C)CO)NC(C1(C(=O)OCC)CCC1)=O C1(CNc2cc(C)c(F)nc2)C(C2CC2)CCN1c1nc(OC(C)C)ncc1Cl C1(O)(CCNC(=O)CC2CC2)CN(C(C2CC(O)(C(F)(F)F)C2)=O)C1 Cc1c(C(=O)NC2CCC(CNC(c3cc(Cl)c[nH]3)=O)C2)nnn1C1CCOC1 C(C(=O)NCCCN(C(=O)CC1(C)CC1(F)Cl)C)(C(C)C)OCC(C)C C1(CNC(C(=Cc2ccco2)C)=O)CC(C(=O)NCCCC2CCOC2=O)=NO1 C(CCC(C)(C)C(=O)NCCNC(=O)C(C)C)NC(CCCCC)=O C1(CNC(C(C)=CC)=O)CN(C(=O)CCC2(CC)N=N2)CC1(C)C C(=O)(NNc1cccc(S(=O)(=O)C2CC2)c1)C1CCC(CC)O1 N1(C(C2CC(OC)C2)=O)C(CNC(C2CC(C)C2)=O)CC2CCCC12 CCC(c1ccccc1)=CC(=O)NCC(C)(C)CNC(=O)C(n1nccc1C)C c1(OCC#N)cc(C(=O)Nc2ccc(I)c(C(F)(F)F)c2)cc(Br)c1 CCCC(C(=O)N(CCCNC(=O)C(C)C(F)F)Cc1ccc(C)cc1)N(C)C c1(C(=O)N(CCCC2(NC(C(CO)NC(C(C)C)=O)=O)CC2)C(C)C)ccncc1O c1(OCC)cc(=NC(=O)C(=O)NCC(O)CNC(=O)OC(C)(C)C)[nH]n1C C1(C(N2CC(N(C(=O)C(C)(F)F)C)C2)=O)CCc2ccccc2N1 C(=O)(CCC(C)(C)F)NC1C(C)CN(C(=O)C(C(=O)N(C)C)C2CC2)C1 C1(COC)(C(NC(C2CC2c2nccn2C)=O)C2CC2)CCN(c2nnn(C)n2)CC1 C1(C(=O)NC(CC)CN(C(=O)C(C)SC)C)CC2(C1)CC2(F)F N1(CC)CCN(C(c2cn(C3CCOC3)cn2)=O)C(C)(C)C1=O C12(C(=O)NCC(CNC(c3cccc(C(C)=O)c3)=O)(C)O)CCCC(C)(C1)OC2 CCC(C(=O)N(CCC(=O)NCCn1ccnc1)C)C(F)(F)F CCCCC(O)CC(=O)N(C1CC1)CC1CCCN1C(=O)Cc1nncn1C C1(CC(=O)NC(CCC)CO)C2CCC(C2)N1C(=O)Cc1ccon1 c1(C(=O)OC)cnc(N2CCCC(C)(NC(c3nnc(O)nc3O)=O)C2)cc1C CCCC(CCC)C(=O)N1CC(CC(N2CC(O)CC2COC)=O)(OC)C1 Cc1ccc(-c2nc(C(=O)NC(C3CCCN3C(=O)C(C)C#N)C)cs2)o1 C1(NC(COCCC)=O)CC12CC(NC(=O)C(C)n1cncn1)C2 C(CC(O)CNC(c1ccn(CCC#N)n1)=O)NC(C1(CCC=C)CC1)=O N1(C(C=C(CC)CC)=O)CCC(C)C(CNC(=O)CCN2CCCCC2=O)C1 O=C(C1=C(Cl)CCOC1)NCC1CCN1C(=O)Cn1ncc2cccnc12 C#CCCC(O)CCc1nnc(N2C(C)CN(C3CC3)CC2C)n1CCCOC N1(C(C(C)C2CC2)=O)CCC(NC(=O)Cc2csc(-c3ncccn3)n2)C1(C)C C1(OC)CC(C(=O)N(C)Cc2ocnc2C)N(C(C2CC2(Cl)Cl)=O)C1 Cc1ccc(CNC(CSC2CCN(C(C3COC4CC3C4)=O)C2)=O)cc1.C1(C)CCC1 C(=O)(CCCCN=[N+]=[N-])N1C(C(=O)NCCC2CC(OC)CN2C(N)=O)CCCC1 N1(c2nnc(C(CC)(C)C)o2)C2CCC1C(C)C(NC(c1cc(C)on1)=O)C2 c1(CC)ccc(C(N2CC(CNC(=O)CCF)C(F)(F)C2)=O)cc1C(F)(F)F CC1(C)CCC(N(C)C(=O)Nc2cccc(Cl)n2)CC1 C=C(Br)CCC(=O)NCCC1CC(NC(=O)C#CC(=O)N(C)C)C1 c1(C(N(CC(C)N(C(=O)CCCN(C)N=O)C)C)=O)csc2ncnc(O)c12 c1(N(CCC)C(N2CC(c3cccc(F)c3F)C2)=O)cccc(Br)c1F CC1CC(NC(=O)Cc2cnccn2)CN1C(c1csc(C#N)c1)=O N1(C(C(=C(C)C2CC2)F)=O)CC2CCCC2(NC(=O)Cc2cc(C)ns2)C1 C1(C(C)(C)C)CCOCCN1C(=O)CN1CCNCC1=O C(CC(C(C)(C)C)NC(c1ncc(C)cn1)=O)N(C(Cc1n[nH]c(=NC)s1)=O)C N1(C(C2CC23CCOCC3)=O)CCC2(CC1)CN(C(c1ccsn1)=O)CC2CO Cc1nc(CC(C)C)sc1C(=O)NCC1CC1NC(=O)CC1C=CCCC1 N1(C(Cn2c(C)ncc2)=O)CCC(C=CC(N2CC(=O)NC(C)C2)=O)CC1 C1(C(N2CCN(C(c3c(C)c(Br)cs3)=O)CC2)=O)CCCCC12CCC2 CC(C)(N)CCCNC(=O)NC(Cc1ccc(I)cc1)CO CN1CCC(NC(=O)CCN(C(=O)C(=O)CCc2ccsc2)C2CC2)C1(C)C C1(C(N2CC(NC(CSCC(C)=O)=O)(CO)C2)=O)CCC(O)CC1 C(c1cn(C)c2ccccc12)=CC(N1CC(N(C)C(c2n[nH]c(=N)s2)=O)C1)=O C(=O)(C1(C)CCc2ccccc21)N1CC(C(C)NC(=O)C(C)(C)CC(F)F)C1 N1(C(=O)NC(C)(C)C)CC2CCCCC2(NC(c2c(N(C)C)ccnc2)=O)C1 C1(NC(c2n(CC)ncc2Br)=O)CCCC12CN(C(C1CC13CC3)=O)C2 c1(CC(=O)N(C(CCNC(C=COCC)=O)C)C)ccc([N+](=O)[O-])c(OC)c1 C1(N(C(C(C)N(C(C)=O)C)=O)C)CCCC2CN(C(C3COC(=O)C3)=O)CC12 c1(C(N2C(CNC(C3OCCN(C)C3=O)=O)CC2)=O)cccc2nn(C)cc12 c1(C(N2CC(C)(NC(C3CCCS(=O)(=O)N3)=O)C2)=O)ccnc2ncnn12 c1(OC)ccc(C(=O)NCC(O)CCNC(C2CC(F)(CO)C2)=O)s1 Cn1nc(C(=O)NC(c2ccc(Cl)cc2)C2CCCC2)c2c(Cl)cccc12 Cc1[nH]cc(C(=O)NCC2CCC(C)CN2C(=O)Cc2cn[nH]c2)c(=O)c1Cl N#Cc1cc(C(=O)NC2(c3nc4ccccc4s3)CCC2)ccc1O N1(C(C2CC(=O)NC(=O)N2)=O)CCC2(CC2)CC1C(=O)NCCCN1CCCC1 C1(CC(=O)NC(c2ccccc2)CCC)C2CCCC2N1C(c1ccc(C)[nH]1)=O c1(C(N2C(CNC(=O)CC=C(Cl)Cl)CCCC2)=O)cc(Cl)c(Br)[nH]1 C1(C(N(c2n[nH]c(C)n2)CCOC)=O)CCCN(C(C2CN(C(N)=O)C2)=O)C1 c1(NC(CNC(c2ccccc2F)C(C)C)=O)ccc(F)c(F)c1 c1(-c2c(C)occ2)nc(C2CC23CC3)nn1-c1ccc(Cl)nc1 C1(S(C)(=O)=O)(C(N2CC(C(C)NC(C3C4CC5C(C4)C35)=O)OCC2)=O)CCOCC1 Cn1nc(C(N2CCOCC2c2cn(-c3cncc(Cl)c3)nn2)=O)cc1C(N)=O C1(NC(Cc2nc(C)sc2)=O)(CO)CCN(C(c2cncnc2C2CC2)=O)C1 C1(C(=O)NCC(C)C)COC(CNC(=O)C(c2ccccn2)C)C1 C1(NC(Cc2c(C)cccn2)=O)(CO)CCN(C(c2sncc2C)=O)CC1 C(C)(C)(CC(Br)C(=O)OC)OC.C(=O)(C(F)(F)C(F)F)N1CCC1 N1(C(C=CC(C)C)=O)CCN(C(=O)C=CC2CCOC2)C(CF)C1 CCC(C(=O)NCC(C)NC(c1ccccn1)=O)NC(=O)NC C1(NC(=O)COC2CCOC2)CN(C(c2cnc3n2CCS3)=O)CC1C1CC1 C1(CC)CN(C(c2ccon2)=O)CC1C(N1CC(CO)C1)=O c1(C(N2CCCC(N(C(=O)C(O)CC(N)=O)CC)C2)=O)ccc2nccn2c1 c1(C(N2C(C)CC(OCCN(C)C)C2)=O)ccc(C#N)cc1.C(=O)(COCCF)N C1(CC)C(NC(C2CN(C(=O)OC(C)(C)C)C2)=O)CCN1C(=O)CN1CCCC1=O c1(C(=O)NCC(C)CNC(c2[nH][nH]c(=N)c2Br)=O)cc2n(n1)CC(C)NC2=O N1(C(C(CC=C)(C)N(C)C)=O)C2CCC1CN(C(=O)C1=NN(C)C(=O)CC1)CC2 C(=O)(CC(C)(C)COCC(F)(F)F)N1CC2C(CNC(C(C)NC(C)=O)=O)C2C1 C1(C)(CNC(C(C(C)C)OC)=O)CN(C(c2ccsc2C#N)=O)C(C)(C)C1 C1(C(C)(C)CO)COCCN1CC(=O)N(C1CCC1)Cc1cccc(F)c1 c1(C(N(CCCNC(C2OCCC2C(C)C)=O)CC)=O)cnc(S)n1C C1(CN(C(=O)C(C)(C)C)C)CCCC(NC(c2ccn(C)c2)=O)C1 c1(C(=O)NCC(C(C)C)NC(C2(C=C)CCOCC2)=O)cnc2ncc(Cl)cn12 c1(CNC(c2ccn(C)n2)=O)n[nH]c2c1CN(C(C1CC1(Cl)Cl)=O)CC2 C(=O)(C(CNC(c1cc(O)cc(=O)o1)=O)C(C)(C)C)Nc1c(C)cccc1 N1(C(C#C)C)CCN(C(c2cccc(CNC(=O)C(CCC)OCC)n2)=O)CC1 N1(C(c2c(CC)n(C)nc2)=O)CCC2(CC1)CC(Nc1nc(C#N)c(Cl)s1)CO2 N1(C(c2ccn(C)n2)=O)CCN(C(c2coc(C(N)=O)c2)=O)C(CO)C1 N1(C(c2n(C=C)ncc2)=O)CCCCC(NC(c2ccc(C3CC3)nc2C)=O)C1 C1(C(=O)NC(c2cccs2)C)(NC(c2cnc(CC)s2)=O)CCC(C)(C)C1 C1(NC(C2CC(CCNC(c3ccc(C#N)s3)=O)C2)=O)CC2COCC(C1)C2 C(=O)(CCCC(C)(C)NC(=O)C(C)OCCF)NCCSCC(C)C C(=O)(CCCC(OC)OC)NC1C(C(=O)NCc2cn(CC)nc2)CCC1 C12CC13CC(C3)N2.N1(C2CN(C(CNS(CC)(=O)=O)=O)C2)CCCCC1 c1(CC(=O)NCC2CCN(C(C(C)O)=O)C2)csc2c(Br)cccc12 C1(c2n(C)ncc2)CN(C(C2CC2(C)C(F)F)=O)CCN1C(=O)CSC1CC1 C(=O)(CCCCCC(C)C)NCC1(F)CN(C(C2CC(F)(C(=O)OCC)C2)=O)C1 c1(C(N2C(CC)CN(C(C3(CO)COC3)=O)CC2)=O)ccc2ncnc(O)c2c1 c1(C(=O)NC2CCCC(NC(c3cccs3)=O)C2)cc2nc(Cl)ccc2o1 c1(C(C)(CNC(=O)OC(C)(C)C)NC(C2C=C(C)CS2)=O)ccccc1F c1(-c2cnc(C(=O)OC)nc2)cnc(Cl)c(C(=O)Nc2ccc(Cl)nc2F)c1 c1(CC(=O)NC(C2CCN(C(C=CCN(CC#C)C)=O)C2)C)cccnc1O C1(NC(C(=O)NC2N(C)CC(C)(C)C2)=O)Cc2nc3ccccc3n2C1 c1(NC2(C)CC(NC(CCC(=O)NCCC)=O)C2)nc(C)c(C#N)cc1Cl C1(C(=O)NCc2n[nH]cc2C)(OC)CCN(C(=O)CC(C)C)C1 C1(CNC(CC(C)(C)c2ccc(F)cc2)=O)CS(=O)(=O)CCN1 C1(C(=O)NC(c2nccs2)(C)C)CCC2CCC1N2C(C1CCC1C#N)=O c1(C(=O)OC)cc(NC(c2n(C(COC)C)ccn2)=O)c(C)c([N+](=O)[O-])c1 Cc1cn2[nH]c(=NC(C(C)NC(=O)CNC(=O)CC3CCCC3)C(C)C)sc2n1 C12(CNC(c3c(CC)n(C)nc3)=O)CCCC1N(C(=O)Cn1cnnn1)CCC2 Cc1ccc(NC(c2nnnn2CC2CCOC2)C2(C#N)CC2)cc1F C12(C(=O)NCC3N(C)CCOC3)CCN(C(C3CC(F)C3)=O)CCC1C2 CC(C)(C(=O)NCCC1(NC(=O)CC2CC2(Cl)Cl)CCC1)C(F)(F)F N1(C(c2c(CO)ccc(SC)c2)=O)C(CNC(=O)CN(C)C)CC2CCCC12 N1(C(c2cnn(CC(F)(F)F)n2)C(=O)NCCSC)CCC(C)(C)CC(C)(C)C1 N1(C(c2ncc(OC)nc2)=O)C2CCC(C(N3CC(C)=CC(C)C3)=O)C1CC2 C(=O)(N(OC)C(C)C)C1CC(CCNC(C2C(CC)OCC2)=O)C1.C1(C)CC1 CC1(CNC(c2cc(C3CCC3)on2)=O)CCC(NC(=O)CCn2cccc2)C1 C(=O)(C(COC(C)=O)C(C)C)N1CCN(CC(C)NC(C(C)(C)SC)=O)CC1 N1(Cc2cnc(C)s2)CCN(CC(=O)O)CC1C N1(C(CC2C(=O)CCCC2)=O)CCN(Cc2csc(Br)c2)CC(O)C1 C1(CNC(c2c(CC)ocn2)=O)CN(C(=O)CSc2nncn2C)C(C)(C)C1 N1(C(C2C(C=C)C2)=O)CCN(C(c2ccc(Br)c(C)n2)=O)CC1CC n1(CC(=C)C)nnnc1C(c1cnc(-c2ccccc2)o1)NC1CC1F c1(N(C2CCN(C(C(CC)NC(C)=O)=O)C2)c2ccccc2)ncc(O)cn1 CC1(C)CCC(C(=O)NCCCc2cn[nH]c2)CN1C(c1cnsc1)=O c1(C(=O)NCc2ncc(CO)o2)ncc(-c2ccc(N3CCOCC3)nc2)cn1 c1(C(=O)NC2C(NC(C(C(C)C)NC(N)=O)=O)CCOC2)ccc2c(c1)NC(=O)C2 C1(F)(C(=O)N2c3nccc2n3)CCNCC1.C1(COC)CC1C(=O)OC.C(=O)OC C1(C(C(=O)NCc2snc(COC)n2)C)CCN(C(=O)C=C2CCC2)CC1 c1(C2(NCC(N3CCC(C#CC)CC3)=O)CC2)ccc2oc(S)nc2c1 C(=O)(CC(F)(F)CC)NC1(CC=C)CN(C(=O)C2=CCOCC2)C1 C(C)(C(CC(=O)NCCc1ccsc1)NC(c1cnccc1C)=O)OC c1(C(N2C(C(=O)NCc3ccc(O)cc3)C(O)CC2)=O)cc(F)cc(F)c1Cl C1(CNC(c2occ(C)c2)=O)CCN(C(c2sccc2Br)=O)CC1C c1(N(C)C)nnc(-c2ccccc2-c2ccc(OC3CCC3)cc2)n1C CS(=O)(=O)CCC(=O)N1CCC(Cn2cc(CCSC3CCC4CC4C3)nn2)C1 C12CN(CCO1)C2c1ccc(C)s1.C1(CCN(C(C)=O)CCN(C)C)CCCO1 C(=O)(CCC(C(C)C)NC(c1ccnc(CO)c1)=O)N1CC(C#C)(F)C1 C1(C(=O)NCCC=CC)CSCCN1C(c1ccc(CO)o1)=O O=C(C1=C(Cl)CC1)NCC1C2CC1N(C(c1ncccc1Br)=O)C2 C1(CNC(c2oc(C(C)=O)c(C)c2)=O)(CO)CCN(C(C2CC3CC3C2)=O)CC1 C(=O)(C(F)(F)CC1CCCO1)N(CC(C)CNC(c1n[nH]c(C2CC2)c1Cl)=O)C c1(OC2CN(C(=O)NCc3c(C)cco3)C2)ccccc1O N1(C(CCNC(=O)OC)=O)CC(N(C(=O)Cn2cncn2)C)C(F)C1 C(=O)(C1CCCc2cccnc21)N1CC(=C(CNC(C(C)NS(C)(=O)=O)=O)F)C1 c1(CC(=O)NCC2CCN(C(C3CS(=O)(=O)C3)=O)C2)ccc(C(F)(F)F)nc1 S(=O)(=O)(c1cc(C(=O)NCC2COC(C)(C)CN2C(C)=O)c(C)o1)NC C1(C(=O)NCCC2N(C(CC3(C)OCCO3)=O)CCOC2)CC(C2CC2)=NO1 C1(C(C)C)C(=O)N1.c1(CNC(C)=O)nnn(C)c1C(N1CCOCC1C1CC1)=O N1(C(CCCCC)=O)CC=C(CNC(c2cc(CO)on2)=O)CC1 c1(C(=O)NCC=CC(=O)NCCS(C)(=N)=O)ccc(C#N)n1C c1(C(=O)NC(=O)C(C)C2CCCO2)ncoc1CC.N1(CCC)CCCCC1 CS(=O)c1ccc(C(N2CCC(C)C(NC(c3nc[nH]c3C(C)(C)C)=O)C2)=O)cc1 N1(C(C(=O)NCc2cc(Br)cc(Br)c2)=O)CCC(O)C2(CCC2)C1 c1(C(=O)NC2CCN(C(CNC(C)=O)=O)CC2)cc(Cl)cc(Cl)c1O CC(CC(=O)NC1CN(C(c2ccc(=N)[nH]n2)=O)CC12CC2)C(F)(F)C(F)(F)F c1(N2CC(=C(CNC(C(C3CCCOC3)OCC)=O)F)C2)nnc(O)s1 Cc1ccc(C(=O)NC2CCC2NC(=O)CSCc2csc(C)n2)nc1 C(=O)(C#CC(C)(C)O)NCC(C(N1CC(COC)OCC1)=O)CC1CC1 Cc1cn2c(n1)CC(C(=O)N(CC(C)N(C(=O)C(C)C1CCC1)C)C)C2 C=CCC(CC(C)C)C(=O)NC1CN(C(c2cnn(C)c2)=O)CC1CC(C)(C)C Cc1cccc(C(N2C3CCC2(CNC(=O)C(F)CC2CCC2)CC3)=O)c1C N1(CC(c2nccs2)C)CCOC(C)(CNC(c2cncnc2C2CC2)=O)C1 c1(CNC(C2CC(C#N)C2)=O)ccc2c(c1)CCC2NC(C1(Br)CC1)=O c1(CCNC(CNC(C2C(C)C2)=O)=O)n[nH]cc1C(=O)NCc1cc(O)ns1 C(C(C)(O)CC(=O)NCC(CNC(c1scc(C)c1OC)=O)CO)OC C=CCC(C)C(=O)NC1CCOC(C(=O)Nc2cnccc2C)C1 c1(C(=O)NC(C(=O)OC)Cc2cnoc2)ccc(Cl)cc1F C1(C(=O)NCCN2C(=O)NCC2)CCCN(C(=O)C(C2CCOCC2)=O)C1 C1(C)(CNC(c2c(OC)ccc(C)n2)=O)CN(C(c2oncc2C)=O)C(C)(C)C1 N1(C(CC2CCCN(C)C2)=O)CC(C)(C(=O)Nc2cccc(CO)c2)CC1(C)C C(CCC(=O)N(C)CCNC(=O)CO)N(C(C(COC)C)=O)C c1(CC(=O)NCC2CN(C(C3CC(=O)N(CCOC)C3)=O)C2)c[nH]c2ccccc12 C(=O)(C(C)CC(N)=O)N1CC(N(C(c2csc(C)c2C2CC2)=O)C)C(O)C1 c1(C)ccccc1.C(C(=O)NCCCN(C(=O)CC1(O)CCC1)CCO)(SC)SC C(C)(CCC(=O)N1CC(O)CC1C(=O)NCCc1cnn(C(C)C)c1)OC c12ccc(nc1C)NC(=O)N2.C1(C(=O)NCC)CCCOC1c1cnn(CC)c1 C(C(CC(F)(F)F)NC(=O)C(C1CCCCCC1)O)NC(C(CSC)(C)C)=O c1(N(C(C(=O)NC2C=CCC2)=O)CC(N2CCOCC2)=O)cccc(Cl)c1 Cc1cc(Br)cc(C)c1OCC(N1CC(C)N(C(=O)CC(F)F)CC1C)=O C(CCN=C(NCC1CC2(C1)CC21CCC1)NCC(C)CNC(=O)OC)OCC C1(CNC(CCc2cc(C)no2)=O)CN(C(c2scnc2C(C)C)=O)CC1(F)F C1(NC(C2N(CCC)CCC2)=O)COC2(CCN(C(C3(C4CC4)CC3)=O)CC2)C1 C1(OC)CC(CNC(C2CCC2(C)C)=O)N(C(=O)CCOC2CCOCC2)C1 C(=O)(C1=NNC(=O)CC1)N(C)CCN1CCN(C(c2cnc(Cl)n2C)=O)CC1 CCC(CNC(c1c[nH]nc1C)=O)(CC)NC(c1cccc(CS(C)=O)c1)=O CC(C)C(C)CC(=O)NC1C=CCN(C(=O)C(C)Oc2ccccc2F)C1 c1(C(=O)Nc2cc(C)c(-c3cnc(N(C)C)c(C)c3)cn2)cccc([N+](=O)[O-])c1O n1(CC(C)C)nccc1C(=O)NC(C1CCN(C(=O)Cc2cccn2C)C1)(C)C n1(CCOC)nnnc1C(c1cn(C2CCCC2)nn1)NCCC1(C)CC1 c1(C(=O)NC2(CF)CCN(C(c3c(C)c(Cl)ccc3)=O)C2)ccc(C)c(Cl)c1F C1(NC(C2C(NC(Cc3c(C)nccc3)=O)COC2)=O)CCCCC12CC2 c1(NCc2cc(O)c(C(F)(F)F)cc2)ccc2ncccc2c1 n1(CC(=O)N(CCC)CCNC(c2ncccn2)=O)cc(C(F)(F)F)cn1 c1(OC(C)CNC(=O)CCN2CCCCC2C)ccccc1C#N c1(SCC#C)cccc(C(=O)NC2CCC(C(=O)N(C)Cc3cscn3)C2)c1 c1(OCCCC(=O)NC2(C)CN(C(C3N(C)CC3)=O)C2)cccc(C#N)c1 N1(C(CCN(C(c2n(CC)nnc2)=O)CCO)=O)CCC2C(C(N)=O)C2C1 N1(C(CSCc2nc(C)sc2)=O)CC2CCN(C(=O)C=CS(C)=O)CC2C1 CC1CC2CC2CC1C(=O)NCC1CC2CC2N1C(c1ncc(C(N)=O)cc1Cl)=O Cc1cccnc1CC(=O)NC(C)(C(=O)NCCn1ncccc1=O)C1CCC1 N1(C(C(C)N(C)C(c2cccc3ccnn23)=O)=O)CCOC2(CCC2)CC1 C1(CC)CN(C(c2nc(-c3cccs3)oc2C)=O)CCN1C(=O)C(F)C(C)C C(=O)(CCCCC(N)=O)NC1CCC(CNC(C=C(C)I)=O)C1 N1(C(Cc2c(CC)n[nH]c2CC)=O)C2CC1CN(C(c1snnc1C(C)C)=O)C2 CC(C)CCC(C(=O)N1CCC(C)(F)C1)NC(=O)Cc1cccc(O)c1 Cc1cnc(C(=O)NC2C3CN(C(=O)Cc4n[nH]c(=N)s4)CC23)cc1C c1(C(N2CC(NC(c3cc([N+](=O)[O-])c[nH]3)=O)C(F)CC2)=O)cc2n(n1)CCCC2 c1(C(=O)NC23C(C)OC(CNC(=O)CN(C)C)(C2)C3)ccc2c(c1)COC2(C)C C1(NC(=O)CC2CCCC23CC3)CC2CC(C1)N(C(=O)C=Cc1cc[nH]c1)C2 c1(CC(=O)NCCC(C)NC(CC(CCC)O)=O)c[nH]c2cnccc12 c1(C(=O)NC(CNC(CC2C(C)OCC2)=O)CO)cccc(Br)c1 CCC(C)CCC(O)CC(=O)NCCCN(CCO)C(C1CC(F)C1)=O C1(C(F)(F)C(=O)NC(CNC(=O)CC2CCN(C)C2)C2CC2)(OC)CCCCC1 c1(N2CCC(C)C2CNC(C2(O)CC2)=O)cc(Cl)c(O)nn1 C#CC1(C(=O)NC2CCC(CNC(=O)C=C3CCSCC3)CC2)CCCC1 CN1N=C(CC(=O)NC2COC3CN(C(=O)C=CC(F)(F)F)CC23)CC1=O C1(C(=O)NC2C(NC(CC3(OCC)CCC3)=O)C2)CCCC1F N1(C(=O)OC)CCC(C(=O)NCC(CCOC)NC(=O)C=CCl)CC1.C1(=O)CCN1 CCC(CC(F)(F)F)C(=O)NC1CC1CNC(=O)Cc1cccn(CC)c1=O C1(C)(C(=O)NC(CNC(c2c(C)oc(C3CC3)n2)=O)C2CCC2)CC2(CCC2)C1 N1(C(Cc2cccc(OC)c2)=O)CCC2CCCN(C(c3cnncc3C)=O)C2C1 C(=O)(CCC(C)CC)N1CCN(CC(C)(C)NC(CCSCCC)=O)CC1 N1(C(C(C)N(C)C)=O)CC2CCC(CNC(=O)Cc3cncn3C)C2C1 N1(C(CC2CCC(C)O2)=O)CC(NC(c2ccc(P(C)(C)=O)o2)=O)C2(CCC2)C1 Cc1cnc(C(=O)NC2(C)CCN(Cc3ccc(SC(F)(F)F)cc3)C2)cc1Br n1(CC(=O)N(C2CC(NC(C3CCN(C)C3C)=O)C2)C)nc(Cl)ccc1=O N1(C(C(n2cc(C)nc2)(C)C)=O)CCCC(CNC(c2c(C)ncn2O)=O)C1 C(=O)(C1=COCCC1)Nc1cccc(NC(CC2C(C)(C)C(O)C2)=O)c1 O=C(NNc1nc2cnccc2s1)c1oc2ccccc2c1Cl Cn1c(CCC(=O)NC2CC2C(=O)Nc2ccc(O)cn2)nc2ccccc12 C(=O)(C(C)C(O)C(C)C)NCC(C(=O)NCC(=O)N(C)C1CC1)O N1(C(C(CCC)CCC)=O)CC2CN(C(=O)Cn3nccc3C)CC2(C)C1 CC(C)C(C)C(=O)N(CCC(=O)NCC1CC(O)C(O)C1)C1CC1 Cc1ccc(C(=O)NC2CC(CC(=O)NCC(C)(C)OCC(F)F)C2)cc1O c1(C(=O)NC2(C)CCN(C(C(CO)OC)=O)C2)ccc(O)cc1F C1(CNC(CC2(N(C)C)CCC2)=O)CC2CC1CN(C(=O)C(Cl)Cl)C2 N1(S(CC)(=O)=O)CCc2c(CC)cccc2C1.c12noc(n1)CCS2 C1(CNC(C)=O)Cc2ccccc2CN1C(=O)C(C)C(=O)Cc1ccccc1F C(C)(C(C)C(=O)NCCCCCCF)NC(COC(C)C)=O N1(C(CC2(OC)CC2)=O)CCN(c2ccccc2CNC(=O)CC(C)F)CC1 C1(O)(C(=O)NC2(CNC(Cc3cn(CC)nn3)=O)CC2)CCCCC1 C1(OC)CC2C1CCN2CC(CO)SC c1(CC)ccc(C(=O)NCC2CCCCN(C(=O)CSCCN(C)C)C2)c(Cl)c1 C12(C(=O)NCC(N(C(CC(C=C)C)=O)C)C3CC3)CC3CCC(CC(C3)C1)C2 Cc1ccc(-c2nn(-c3ccccc3)cc2C(N)=O)cc1C C1(C(N2CC3C(CC)(C3)C2)=O)CC2CCC1CN2C(C1OCCC1C(=O)OC)=O Cc1ccc(Cl)c(F)c1CNCC(O)Cc1ccc(F)cc1F Cc1cc(C(=O)NCC(CNC(c2ccn(C3CC3)n2)=O)CO)cs1 N1(CC(=O)NC2CC3CN(c4nc(C#N)c(Cl)s4)CC32)Cc2ccccc2C1=O c1(C(N2CCC(C(C)NC(CCC(CC)C)=O)CC2)=O)cc(F)c(N)c(F)c1 C1(CN(C(C=CC(CC)C)=O)CC)CC(C2CCC2)C1 n12cc(nn1)C(=O)NCC1(CCC1)CC2.C(CC(=O)NCC=C)=CCC N1(C(CCc2cccc(OC)c2)=O)CCN(C(=O)CCC(C)C)CC(C)(F)C1 C(C)(C(C)C(=O)NCCOCC(C)C)NC(c1c(CC)ocn1)=O N1(C(CCN(C(=O)CCS(N)(=O)=O)CC=C)=O)CCC2(CCCO2)C1 c1(SCCCC)cccc(C(=O)NC2CC(C)(CNC(C3CCC(=O)N3)=O)C2)c1 C1(C(=O)NCCc2nn[nH]n2)CC2CCC1(CO)C2 C1(NC(C2OCCN(CC)C2)=O)C(C)CCN(C(c2cc(OC)no2)=O)C1C N1(C(C(N)Cc2ccoc2)=O)CCCCC2(CCC2)C1 c1(CC(=O)NC(C2CCN(C(c3cccc(=O)o3)=O)CC2)C)ccc(Cl)c(Cl)c1 C(=O)(C(C)(C)S(C)(=O)=O)NCCCC(C)NC(CC1(OCC)CC1)=O N1(C(C=C(C)C(C)C)=O)C2CCC1CC(NC(=O)C(F)CC(C)C)C2 C(=O)(CC(F)(F)C(F)F)N1CCC(N(C(=O)CC(F)(F)F)CC)C1 N1(c2n(CCC=C)c(-c3ccc[nH]3)nn2)CC(C(N)=O)C2(CC2)C1 c1(C(N2CC(NC(CSC(C)C)=O)C(CO)CC2)=O)ccc2cc[nH]c2n1 Cc1sc(O)nc1C(=O)N(C)CC=CC(=O)NCC(C)OCCO C1(C(=O)NC2CC(C(C)NC(CNC(=O)OC)=O)C2)CC(C)(C)SC(C)(C)C1 C1(C(=O)NC2(CCCC)CC2)CC2CCC(C1)N2C(=O)CC1CCC1 c1(C(=O)NC2(CNC(C(C3CCCO3)OC)=O)CC2)c[nH]c(Br)c1 C1(C2CCCO2)(C(N2C(CNC(=O)CCCC3OCCO3)CCC2)=O)CCCO1 Cc1nn2c(C(=O)NC3CN(C(c4cccc(F)c4)=O)C(C)(C)C3)c(C)nc2s1 C(c1ccc(C#N)cc1)=CC(N1C(CCNC(C2C(OCC)C2)=O)CSCC1)=O CC1CCC(C(=O)NCCCCCNC(c2cnn3c2CCC3)=O)C(=O)N1 CC(C)(CC(=O)NC1CC2CCC1(CNC(C1CC(OC3CC3)C1)=O)C2)C(F)F c1(C(N(C(CC)C)C)=O)cnn(CCNC(=O)Cc2cnc(C)s2)c1 c1(C(=O)Nc2n(CCN(C)C)ncc2)cccc2[nH]cc(Cl)c12 C1(C(=O)NC(CC)(CC)CO)CC(C)CN(C(C2C3CCC(F)C23)=O)C1 CC1CC=CCC1C(N1CCC(C)(NC(=O)CSCC(N)=O)C1)=O N1(C(C(CCC)C)=O)CCCC12CCN(C(c1ccc(Br)c3cn[nH]c13)=O)C2 c1(C(=O)NCC2N(C(COCC#C)=O)CC(O)C2)ccnc(C)c1C C1(C(N(C2CCN(C(S(C)(=O)=O)=O)C2)CCC)=O)CCc2nn[nH]c2C1 C1(CNC(c2nc(CC)oc2C)=O)CN(C(=O)CCCC2(C)N=N2)CC12CCC2 C1(C(N2CC(C(=O)OC(C)(C)C)C2)=O)CCOCCN1C(C1CC1NC(C)=O)=O Cc1cc(C)c(C(=O)NCC2(F)CN(C(=O)C#CC3CCCO3)C2)cc1N N(C(=NCCCC(F)F)NC(C1CCC1)C)Cc1ccc(OC)cc1OC C1(O)(CC(=O)NC(C)CNC(=O)CSc2ccccc2F)CCCCCC1 C1(C(=O)NCc2ccc(CBr)cc2)Cc2cccc(F)c2O1 N1(C(C(C)(F)F)=O)CCC(C2N(c3ncc(Br)cn3)CC2(C)C)CC1 N1(C(COCCOC)=O)CCC(C)C(CNC(c2c[nH]nc2C)=O)C1 N1(C(c2nc(C)sc2C)=O)CCC(C)N(C(c2cnc3n2CCCC3)=O)CC1 N1(C(c2c(OC)cnc(F)c2)=O)CCC2(CC1)CCN(C(=O)CCS(C)=O)CC2 C12(CCC(=O)NC3(C)CC(NC(c4nc(C(F)(F)F)cs4)=O)C3)CCC(CC1)C2 c1(CCC)cc(C(N2CCC(C(C)NC(=O)C(C)(C)c3cscn3)C2)=O)c(C)o1 C=CC1(CC(N2CCCCC2C2(NC(C3C(C(F)F)C3(C)C)=O)CC2)=O)CCCCC1 C(=O)(C1=CC2(CCOC2)C1)N1C(CCC)CN(C(=O)CN2C(=O)CCC2=O)CC1 c1(CC)ccc(C)c(C(N2CC(CNC(C3(O)CCC3)=O)C(C(F)(F)F)C2)=O)c1 C12CCC3CN(CC3C1)N2.c1(C)cccc(CO)c1.c1(C=O)cnccn1 n1(CC)cnc2nc(N3CCCC(C)(OC)C3)nc(N3CCC(C)(F)CC3)c12 N1(C(CCOC(C)C)=O)CCCCCC(NC(=O)C#CC2(C)COC2)C1 c1(C(=O)NC2C3CCC2N(C(=O)CCc2cnoc2)C3)ccc2cnccc2c1 CC(C)CC(CNC1CCC=CCC1)CC(=O)NC(C1(NC(=O)NC(N)=O)CC1)C N1(CCCNc2ccc(NCc3c(C)n[nH]c3)cn2)CCc2ccccc2C1 Cc1ccc(C(=O)N(CCS(C)(=O)=O)C)c2c1NCCC2 C=CCCN=C(NCC1(C)CC1)N(C)CC1CCC1 C1(C(N2CC(=C(F)CNC(=O)C3=CCSC3)C2)=O)CCC(C(=O)C2CC2)CC1 C1(OCCNC(=O)NCC(CNC(=O)OC(C)(C)C)O)C2CC=CCC12 Nc1ccc(CC(=O)NC2CCCC2C(N2CCC2C(N)=O)=O)nc1 N1(C(c2c(NCCCC)cccc2)=O)CC(C)N(C(c2nocc2C)=O)CC1C CCCCC(O)C(=O)N1CC(=O)CC1C(=O)NCc1nc(C)ccc1C CN=c1ncn(CC(N2CCC(C(F)CNC(=O)C(C)(C)CF)CC2)=O)[nH]1 c1(C(N2CC(C)(C)C(NC(=O)CC3=NNC(=O)C3)C2)=O)cc2c(cc1N)OCO2 c1(N2CCC(C)(CSC)C2)nc(N2CCC3(CNC(=O)C3)C2)nc2ncn(C)c12 CC1(C)CC(NC(=O)C(N2CCOC(c3ccc(Cl)cc3)C2)=O)(CO)CO1 C12CCCN(C1=O)C2=O.c1(OC(=O)Cc2ccsc2)cc(Cl)ccn1 N1(C(C(C)CC2CCCC2)=O)CC(CNC(=O)CN2CCNC(=O)C2)CC1(C)C CCC(CCC(=O)NCC1(C)CCC(C)CC1)NC(=O)C1=CCCC1C n1(CC(=O)NCC(C)NC(=O)CCn2ccnc2)cc(C2CCOC2)cn1 C#CC1(C(=O)NCC(C)C(C)O)CCN(C(C2CC2CC)=O)C1 c1(C(N2CCN(C(C(CCSC)NC(C)=O)=O)CC2)=O)csc2cncn12 N1(C(c2cn(CCC)nn2)=O)CC(NC(=O)CN2C(=O)CNC2=O)CC1(C)C C12(NC(NC(c3ccc(CC(C)C)cc3)C)=S)CCC(CC1)C(C)(C)O2 c1(C(N2CCC(N(C)C(C3C4CCC34)=O)C2)=O)c(F)ccc(Cl)c1F N1(C(CC2CC(SC)C2)=O)CCC(NC(c2ccc([N+](=O)[O-])[nH]2)=O)C(F)C1 C1(NC(CC=C=C)=O)C(C)(C)C(NC(=O)Cc2ccc(F)c(C)c2)C1(C)C Cc1c(C(=O)NC(C)CCNC(=O)Cn2nnnc2C)cnn1CC(F)(F)F CC(C(=O)N(CCCCNC(=O)C(C)C1CCCO1)C)NC(C1CCCC1)=O c1(C(=O)NCC2N(C(c3cn(C)c(Br)c3)=O)CC2)ccccc1S(C)=O N1(C(C(C)Cc2ccccn2)=O)C(C(=O)Nc2cncc(Br)c2)CC2CC12 CC1CCN(C(=O)CCC2NC(=O)NC2=O)CC1NC(C1(C)CNC(=O)C1)=O N1(C(Cc2c(C)scc2)=O)C2CCC1CC(N(C)C(C1(C3CCC3)CC1)=O)C2 c1(C(=O)NCC(CC)C)ccccc1Cn1cc(CCN(C)CCO)nn1 c1(CNC(COCCC=C)=O)nc2c(s1)CN(C(=O)CC1(COC)CC1)CC2 N1(C(c2cc(OC)ns2)=O)CC2C(N(C(=O)CCCN3C(=O)CCC3=O)C)C2C1 Cc1ccc(C(=O)NCC(C)CNC(c2cnc[nH]c2=N)=O)c(F)c1F c1(C(c2nnnn2C)NC(CC)CC2CCCCC2)cc2ccccn2n1 CC(O)C(C)C(=O)N(C)CCOCCNC(c1ccn(C(F)(F)F)n1)=O N1(C(c2ccc(C)n2C2CC2)=O)CC(CNC(c2cnco2)=O)CC(C)C1 N1(CCNC(C(C)Cc2cnc[nH]2)=O)CCN(C(c2cnsc2)=O)CC1 c1(C(C)=O)ccc(S(=O)(=O)NC2CCN(C(C3CC4CCC3O4)=O)C2)cc1 c1(C(=O)NCCC(C)N(C(CCC(=O)NC)=O)C)cnn(C)c(=O)c1 N1(C(C(C)NC(C(C)(C)C)=O)=O)CCC(C2CC2NC(C2CCC3(CC3)C2)=O)CC1 c1(CC)ccc(NCCNC(=O)COCC(C)(C)SCC(=O)NC2CCCO2)cc1 N1(C(c2cccc(OC)n2)=O)CC2(CNC(C3(C)CCNC(=O)C3)=O)CC1CO2 c1(C(=O)NCC2N(C(c3c(SC)ccs3)=O)CCC2)c[nH]c(=N)c2[nH]ccc12 N1(C(CC(C)OC)=O)CCC(C(N2CC(O)(C(C)C)C2)=O)C12CCC2 c1(C(=O)NCCCNC(C=C)=O)ccc(C)c(O)c1Cl N1(C(CC(=O)OC(C)(C)C)=O)CCCN(C(c2ncn3c2CCC3)=O)C(CO)C1 C1(C#N)(CC(=O)N(CCNC(C(C)OCC)=O)CC)CCOCC1 N1(C(Cc2c(C)scc2)=O)CC(CCNC(c2cnsn2)=O)OC(C)C1 c1(C(=O)NC(C(C)C)CCN(C)C(C2CC(O)CN2C)=O)ccc(N)cc1F CCC(CC1CCCCC1)CC(=O)NC1CCC(NC(=O)C=CC(C)(C)SC)CC1 C1(COC)CN(C(=O)C=C(C)C(C)(C)C)CCN1C(c1csc(-c2ncc[nH]2)n1)=O C(C(=O)N1OC2C=CC1CC2)C1CCN(C(CCNC(=O)NC)=O)CC1 C1(N(C(=O)C=CC2(C)COC2)C)C2CN(C(=O)C(F)OC(F)(F)F)CC12 C(=O)(C(C)(C)C(=O)N(C)C)NCCc1cn(C(C2CCCCO2)CC)nn1 C(=O)(C(C)(C)CNC(=O)C(C)(C)C1CCCN1C(=O)CCCOC(C)(C)C)NC C1(CC(=O)NCC(F)CNC(=O)C(c2ccc(Cl)cc2)(F)F)CCCC(=O)N1 C1(C)(C(N2CCC(=C)CC2)=O)CCCN(C(c2ccn(C)c2C)=O)C1 c1(-c2cc(C)[nH]n2)nc2c(s1)CCN(C(=O)CCNC(c1ccncc1)=O)C2 CN1CCCC2CN(C(=O)Nc3cnn(C4CC4(F)F)c3)CCC12 c1(C(=O)NC2C(NC(CC=C=C)=O)CC2)cccc(F)c1C C1(C(N(C2CCC2)CC#C)=O)CCCN(C(=O)C(O)C2CCCC2)C1CC c1(CC(=O)NC(CCNC(c2cc(C)ns2)=O)(C)C)cccc(C(F)(F)F)c1 c1(OC)ccc2c(c1)CCC(NC(c1cccc(C(C)C)c1C)=O)CC2 Cc1cccn2nc(NC(N)=O)cc12.C12(CCCC1)C(=O)N1CCC1CNC2=O c1(OC(C(=O)NC2C(NC(C(CC)(C)C)=O)CC2)C)cc(C)ccc1Cl O=C1CCN(CC2CCC2)C(=O)N1CC1CC(O)C12CCC2 N1(C(c2cc(C(C)C)no2)=O)CCN(C(=O)CSC2SC(=N)NC2=O)CC1 C1(C(C)NC(c2cc(C)on2)=O)CCN(C(c2cn(CC3COC3)nn2)=O)CC1 C1(NCC(=O)NC2CCC2)C(=O)OCC1CO.C1(CN)CC1 c1(C(N2CC(CCNC(C(C)OC3CCCC3)=O)C2)=O)ccncc1C(F)F C(=O)(C1=Cc2ccccc2C1)N1CC2C(CNC(C(F)=CCC)=O)(CCC2)C1 C1(NC(C2CCCOC2)=O)CC2CC1N(C(c1cccc(Br)c1)=O)C2 c1(OC)cc(C(=O)NC2(CNC(=O)COC3CCCCC3C)CCC2)cc(C)n1 CC1C(C(=O)NCC(O)CNC(=O)OC(C)(C)C)C1C CC1(C)Cc2cc(CNC(=O)C(N)CO)ccc2O1 N1(C(c2cccc(C)c2F)=O)CCC2(CC1)CC2CNC(=O)CC1CCCC1O C(C(CC(F)(F)F)NC(C1CN(C)C(=O)N1)=O)NC(CCN(C(C)=O)C)=O c1(N2CC(C)CS(=O)CC2)ccncc1S(=O)(=O)N(CC(O)C1CC1)C C(=O)(C(CN(C)C)C(C)C)NCC1(NC(c2c(C)nccc2)=O)CCC1 Cc1cccn2nc(C(=O)N(C3CCCC3)CCN(C(C3CC3F)=O)C(C)C)cc12 c1(C(N(CC(CC)NC(=O)C(O)Cn2cncn2)CC)=O)ccc(CSC)cn1 C1(C(=O)NCC2C(C)CN(C(c3ccc(F)cc3)=O)C2)CCCC(C#N)C1 C(C)(C)(C#Cc1cn(CCc2cccnc2)nn1)NC(C(CC)OCC)=O C1(C)(CNC(C2N(C(C3N(CC)CC3)=O)CCC2)=O)CC2CC2C1 C(CCC(CCC)NC(=O)C(C(C)C)c1cnn(C)c1)NC(CN(CCC)C)=O C1(C(=O)NC2(CCC)CC2)(CCOC)CCN(C(=O)C(C)O)CC1 N1(C(C(C=C=C)C)=O)CC2CCC(C1)C2NC(=O)C(c1cnn(C)c1)C C1(NC(c2cnc(CC)s2)c2nnnn2C(C)C)CCOCC1(C)C c1(C(C)NC(CCC(CC)OC)(C)c2nnnn2C2CC2)nnc2n1CCOC2 C(=O)(CCC(C)(C)N(C)C)NCc1c(C(=O)NC(CC)C2CCC2)scc1 C=CC(C)(CC)C(=O)NCC1(CNC(c2cc(OC)no2)=O)CCCC1 Cc1nn(CCC(=O)NC(CNC(C2(C)CC(F)C2)=O)CO)c(C)c1C N1(C(C=CC=CCCCCC)=O)CCN(C2CCCN(C(=O)CCSC)C2)CC1 C(=O)(C(F)C(F)(F)F)N1CCN(C2CCN(C(C(C)NC(CC)=O)=O)C2)CC1 C1(C(C)C)C(=O)N1.C1(C(CNC(C)=O)(C)C)CCCN1C(C1CC1C(C)O)=O C1(NC(C(CC)(F)F)=O)CC2CC1CN(C(=O)C(C)Oc1ccccc1F)C2 C1(C(N2C(C(=O)OC)CC2)=O)CN(C(=O)C(C)N2CCCC2)CC1(C)C N1(C(CN(C)CC)=O)CCC(F)(CNC(c2cc(C)ccc2F)=O)CC1 N1(C(c2c(C)nn(C)c2Cl)=O)CCCC2(CC(NC(=O)CSS(C)(=O)=O)CO2)C1 N1(C(c2cc(CC)sn2)=O)CC(CNC(c2cnsc2)=O)C(C)C1 CCCC(O)CC(=O)NC1CCN(C(=O)CCCNc2ccccc2)C1 c1(C(=O)NCCc2ncc(C)nc2)ccc2c(n1)OCC(=O)N2 CCCC(CCCC(=O)NC(CC)CO)NC(=O)CC(CC)C(C)(C)C N1(C(CNC(=O)CCc2nc[nH]n2)=O)CCC(C2CCCC2)C1 C1(C(=O)NCCCOCCN(C(=O)CCCCN2CCCC2)C)C(C)(C)C1(F)F C1(CCCC)CCCN(C(C2CC23CC(NC(C24CCN(CC2)C4)=O)C3)=O)C1 C1(CNC(c2ccn(CCOCC)n2)=O)CC2CN(C(=O)CSC3CCC3)CC12 N1(C(C2(C)CC2)=O)CC(C2CC2)(C(=O)NCCC(O)C2CCCC2)C1 C1(C(=O)NCCC2CN(C(c3c(C)scn3)=O)CC(C)O2)Cc2ccccc2C1 c1(CC)c[nH]c(C(=O)NC2(C3CCCN3C(=O)CCCn3cncn3)CC2)c1 C1(C(=O)NC(=O)C(Cl)(Cl)Cl)CN(C(C2CCC(NC(N(C)C)=O)CC2)=O)CCO1 c1(CC(C(=O)NCCC#C)NC(C2CCN2C(C)(C)C)=O)ccc(Cl)cc1Cl C(=O)(C1=CC2CCCCCC12)NC1CN(C(CC2(C)CCCO2)=O)CC12CCC2 C1(C(=O)NC2(CNC(C3CCCOC3)=O)CCOC2)C2(CCC2)C12CCC2 Cc1[nH]nc2c1CN(C(c1ccc(Cl)nc1NCc1cncc(C#N)c1)=O)CC2 Cc1ccncc1CC(N1CCN(C2CCC(NC(=O)C=CCO)C2)CC1)=O C(C)(C(C(=O)N(C(C)CO)C)NC(=O)C(C)n1cccc1)OC C(C)(C)(CC(=O)NC1(C)CC(NC(C)=O)C1)N(C(=O)CCC(C)C)c1ccccc1 C1(CNC(C2(NC(=O)CN3CCOCC3)CSC2)=O)CCCC2(CC2)C1 C1(C(N2CC(n3cc(CNS(N)(=O)=O)nn3)(C(=O)OC)C2)=O)CC2CC1CC2O Cc1ccc2c(c1)C(C(=O)NCCC1CCCN(C(c3ccoc3)=O)C1)C2 c1(N)cc2ccccc2nc1N1CCCC1.O=C(CO)NCC1CC1.C1CN1 c1(C(=O)NCC2(C(F)F)CCN(C(C(C)C(F)F)=O)C2)cc2n(n1)C(C)CCC2 N1(C(CC2CN(C(C)=O)C2)=O)CC=CC1(C)C(=O)NC(C)CN1CCOC1=O C1(CC(N2CCCC(C(C)NC(COCCC#C)=O)C2)=O)CC2CCC1CC2 c1(CC)nn(C)c(C(=O)NCC(O)CCNC(=O)C=CCn2cncn2)c1Cl C1(C(C)NC(C2(C)CC2(F)F)=O)CCCN(C(C2CCC(F)C2)=O)C1 Cc1nccnc1C(=O)NCC1CC(F)(CNC(=O)CC2CC2C2CC2)C1 CCCCC(C(=O)NCC(C1CCCC1)NC(=O)CCc1cccs1)N(C)C C(=O)(CCC(=O)CC)N1CC(C=C)(CC(=O)NOCCn2ccnc2)C1 c1(SC)cc[nH]c(=NCCC23CCC2CN(C(c2c[nH]nc2C)=O)C3)n1 C1(C(C)C)CN(C(=O)C=CSCc2ccco2)CCC1NC(C1(C#N)CC1)=O C1(NC(c2cnoc2C2CC2)=O)CCSC12CN(C(c1c(F)ccnc1Cl)=O)C2 C1(SCCNC(=O)NCCC(COC)OC)CC1C1CCCCC1 c1(C(=O)NC2CCC(NC(C3CC=CCO3)=O)C2)nc[nH]c2nccc1-2 c1(CCNC(C2CC(c3ccccc3)NC2=O)=O)c[nH]c2ccccc12 N1(C(CCC(CC)C)=O)Cc2[nH]nc(C(N3CC(OC(F)F)C3)=O)c2C1 C(N=c1[nH]cnc(Cl)c1CO)C1(F)CCN(C(CN(C2CCOC2)C)=O)CC1 C1(CNC(CCCN(C)C)=O)C2CCC(C2)N1C(=O)CC1OCCCC1(C)C CC(C)CC(O)CC(=O)NC1C(C(=O)NC2CCNC(=O)CC2)C1(C)C c1(OC)ccc(Cl)c(NC(C2CCCN(C(c3cc(Cl)ncc3Br)=O)C2)=O)c1 c1(C(CNC(C2CC2(F)F)=O)NC(c2ccncn2)=O)cccc(Cl)c1 C(=O)(CCCCCC(C)O)N1C(CNC(c2c(C)n(CCO)nc2)=O)CC(O)C1 C=CC(F)(F)C(=O)NCc1ocnc1C(N1CC(c2cnn(C)c2)C1)=O C1(C(N2CC(=C(CNC(CNC(c3cn(CC)nc3)=O)=O)F)C2)=O)C2CCC1CC2 c1(C2(C(N3CC(C(c4ccccc4)=O)C3)=O)CC2)ccc(Cl)c(Cl)c1 C1(COC)(CNC(=O)C=CCO)CCN(C(c2cc(C)ccc2Cl)=O)CC1 C1(NC(c2ccc(CC)[nH]2)=O)CCC2(CC1)CN(C(=O)C(C)(C)O)C2 Cc1c(NC2CN(C(=O)CN3CCCCC3C)C2)cccc1N1CCCC1=O c1(C(N2CCCC(C(C)NC(c3cccnc3F)=O)C2)=O)cccc(O)c1Cl C(C(CC)(CC)CO)NC(CCC1(C)N(C(C(CC)SC)=O)CCC1)=O Cc1nc2nc[nH]n2c(=O)c1CCC(N1CC(NC(=O)C(C)O)CC1(C)C)=O C1(C(N2CCC(C)(NC(=O)CC3CC4CCC3O4)CC2)=O)CCc2nncn2C1 N1(C(CC)=O)CCC2(CC2C(=O)Nc2ccc(Oc3ccccc3)nc2)C1 N1(C(c2cc(C)nnc2)=O)CCCCC(NC(C2CCCN(C)C2)=O)C1 c1(OC)cc(C(N2CC3C(N(C(=O)C(CSC)OC)C)C3C2)=O)ccc1[N+](=O)[O-] N1(CCOC)CCN(C(C2CC3CCC2C3)C(=O)NC2(C)CC2)C(C)C1=O c1(C(N2C(C)CN(C(C3CCCN3C)=O)CC2)=O)noc2c1CCCCC2 c1(C(=O)NCC2CCN(C(=O)Cc3ccccn3)C2)nc(C(F)(F)F)ccc1F N1(C(CCC=CC)=O)CCC(N(C(=O)C(C=C)CC)C)CC1 C1(C(=O)NCC2N(C(c3nc(C)c(C)s3)=O)CCC2C)CCC2(CC1)CC2 C1(NC(c2nc(CCOCC)oc2)=O)CC(C)N(C(c2cccc(=S)[nH]2)=O)C1 CC1CC(C)N(C(c2conc2C2CCC2)=O)CCN1C(c1nn[nH]c1Cl)=O N1(C(C(CCC)C)=O)CCC(C#N)(NC(=O)Cn2ccccc2=O)C1 c1(C(N2C(C(C)C)CN(C(=O)C(F)C3CCCC3)CC2)=O)cc(O)cc(C#N)c1 C1(CNC(=O)C(=Cc2c[nH]cn2)F)CCCN1C(=O)CN1CC2CC2C1 C1(C)(OC)CC(NC(=O)CN(C(c2ccoc2C)=O)C(C)C)C1(C)C C=CCC(CC(F)F)C(=O)NCC(C)CN(C(=O)C(C)C1CCCC1)C C12(CNC(=O)Cc3cncs3)CC1CN(C(C1COCCO1)=O)C2 N1(C(C)=O)CCC(CC(=O)N(C2CC(CNC(=O)CN3CCOCC3)C2)C)C1 n1(CC(C)C)ncc2cc(C(=O)NC(C)CCNC(=O)Cc3cccs3)cnc12 C1(NC(c2c(C)noc2)=O)CC(NCC(N2CC=CC2)=O)C12CCC2 N1(C(C(CCN(C)C)O)=O)CCC(NC(c2csc(CO)n2)=O)C(F)C1 Nc1cc(F)cc(Cl)c1C(=O)NCCCNC(c1ccc2c(c1)CC2)=O c1(NC(=O)NC(CN(CC)CC)C)cccc(CC(F)(F)F)c1 C12(CC)CC(C(=O)N(C)CC3CCCN(C(c4ccnnc4C)=O)C3)(CO1)C2 C(CCNC(C)(C)C)(C(=O)N=c1cc[nH][nH]1)c1c(OCC)cccc1[N+](=O)[O-] C1(C(N(CCC=C)CC)=O)CCC2(CC2)N1C(C1CCC2(CCC2)O1)=O C12(C(=O)NC(CCC)CCC)CCCC1CN(C(C1CC3(CC3)CO1)=O)C2 Cn1cnc2ncnc(N3CCCC34CN(C(c3cc(CO)cc(Br)c3)=O)C4)c12 N1(C(C(C)OCC=C)=O)CCC(N2CCN(C(=O)C(C)=C(C)CC)CC2)CC1 N1(CC)CCCC1C(=O)NC(C)(C)C(C)NC(=O)CCc1cc(OC)no1 c1(OC)ccc(OC)c(C2(NC(=O)NC(C)C3CC3)CCC2)c1.c1(N)cc(C)cc(C)n1 c1(C(=O)NC2(CN(C(C3CCCC4CC34)=O)C3CC3)CC2)ccc2cccnc2c1 C(c1ccc2c(c1)CCO2)=CC(=O)NC(CCCCNC(c1c(CC)ncs1)=O)C c1(CNC(=O)COc2ccc(-c3ccccc3)cc2)cc(Cl)cnc1F N1(C(C2(CC)CCCC2)=O)CC2(CNC(=O)Cc3nnc(O)s3)CC1CO2 C1(NC(CC(CC)(C)C)=O)CCC12CCCN(C(=O)C=CCOCCOC)C2 CC(C)(C)C(=O)CCc1cn(C2CCC(NC(c3nc(O)[nH]c(=O)n3)=O)C2)nn1 C1(NC(c2ccsc2)=O)CC(F)CN(C(c2cccnc2S)=O)C1 n1(CCC#C)c(N2CCC(C(C)(C)C)C2)nnc1-c1ccc(CCO)cc1 C1(CN(C)C)CCCN(C(C2CCC=CC2NC(=O)CNC(=O)CN(C)C)=O)C1 c1(C(=O)NCC(CO)NC(CSCCOC)=O)ccc(CC(C)C)nc1 C1(CC(=O)OC)COC(CN(S(=O)(=O)CC2CCNCC2)CCC(=O)O)C1 c1(C(=O)NCC23C(CN(C(c4cc(COC)sc4)=O)C2)C3)ccc(O)c(N)n1 c1(C(N2C(CC)C(NC(=O)C=Cc3ccco3)CC2)=O)cc(Cl)ccc1N c1(C(N2CCCC(CNC(=O)Cn3cncn3)C2)=O)n[nH]c2c1CCCCC2 CCCCCC(C)(CC)C(=O)NC1CC2(CCN(c3ccncc3C#N)CC2)C1 CC1CCc2sc(C(=O)NCCNC(c3cc(C(F)(F)F)no3)=O)cc2C1 Cn1cc(C(=O)NCC2CCN2C(C2CC2c2ccccc2)=O)c(Br)n1 C1(C(C)NC(COCC#C)=O)CCN(C(=O)COC(C)C)C1 C1(CC(=O)NC2(CNC(CCOCCCOC)=O)CCC2)CNC(=O)C1 C1(c2n(CC)nnn2)(Nc2ccc(NC(=O)CCCSC)cc2)CCN2CCCC12 c1(C(c2n(C(CC)C)nnn2)N(CCn2cccn2)C2CC2)cncc(Cl)c1 C1(CCNC(c2cnc(C)o2)=O)COCCN1C(=O)C(c1nc(C)cs1)C Cc1cc(C(=O)NC2CC(O)CN(C(C3(F)C(C)(C)C3(C)C)=O)C2)c(F)cc1F C(=O)(CC(O)CC(C)(C)C)NCCOC(CNC(c1cccc(C)n1)=O)(C)C N1(C(c2c(C(C)C)ccs2)=O)CC2CCC(NC(c3cc(O)nc(Cl)c3)=O)(C2)C1 c1(CN2CCN(CC(N3CC(C)(C)NCC3)=O)CC2)cc(I)cc(I)c1O C1(C(=O)Nc2c(C)ccnc2)CC2CN(C(C3(C)C=CCC3)=O)CC2C1 C1(CC(=O)N(C2CCN(C(c3n(C)ccn3)=O)C2)CCO)Cc2ccc(Cl)cc2C1=O C1(CNC(c2cnc(C)o2)=O)CCC(C)(C)CN1C(c1cnn(C)c1N)=O c1(C(N2CCC(n3nc(C)c(C(=O)OCC)c3C)C2)=O)cccc2c1CCN2Br c1(C(N2C(C(C)NC(c3occc3F)=O)CCCC2)=O)ccc(N)c(Cl)c1 C(=O)(C1CCCn2cnnc21)NC(CC1CN(C(C=C(C)C(C)C)=O)C1)C N1(C(COCCOCC)=O)CCC(C)C1C(=O)NC1CCNC1=O C(C)(C)(C(=O)NC(C1(O)CN(C(=O)C(C)Sc2ccccc2)C1)C)OC(C)=O N1(C(c2c(C)nn(C)n2)=O)CC2CCCC2(NC(C2CC(=O)NC(=O)N2)=O)C1 c1(N(CCN(C(C2C(CC)OCC2)=O)C(C)C)C)cccc(I)c1 Cc1sc(Br)nc1S(=O)(=O)NC1CCNC12CCC2 c1(C(N(C)CC2CCN(C(=O)CC3(C#N)CCC3)C2)=O)ccc(F)c(C(F)F)c1 C1(C(N(CCNC(=O)Cc2cncnc2)CC)=O)(C(F)F)CCCCC1 c1(C(C(=O)NCC2CC(NC(C(C)CO)=O)C2)(F)F)ccc(Br)cc1 CS(C)(=O)=NCC(=O)NC1CC1CNC(c1conc1C1CCCC1)=O c1(CSC)ccccc1-n1ccnn1.C12(F)CN(C1)C(=O)N(C)C2=O c1(C(C(=O)N(CCNC(c2c(C)oc(C(F)(F)F)n2)=O)C)C)cc(F)cc(F)c1 c1(OCc2cn(CC(=O)NC3CCNC3)nn2)ccc(Cl)c(O)c1 C1(C(N(CC)Cc2cccs2)=O)C2CC1N(C(=O)CCC1CC1(C)C)C2 C=CCC(CNC(C1(C#N)CC1)=O)NC(=O)C(C)c1cccs1 Cc1nnc(C(=O)NCC2COC(CNC(=O)C(c3cccn3C)=O)C2)s1 Cc1c(Cl)ccnc1C(=O)NCC(C1CCCC1)NC(c1cccn1C(C)C)=O CC1c2ccccc2CC1NCC(=O)Nc1c(F)cc(Cl)cc1F c1(C(N2C(CN(C(C(CCCC)O)=O)C3CC3)CCC2)=O)nc(C)c(C)nc1C c1(C(=O)NC(CNC(CC(C=C)C)=O)CC)cc(C#N)c2n1CCCC2 N1(C(CC(C)C2CC2)=O)CCCCC(C(N2CC3(C2)CN(C2CC2)C3)=O)C1 Cn1nc(C(=O)NCC2(C)CCC(NC(=O)C(C)(C)N3CCCC3)C2)cc1C#N c1(OC)ccc(C(N2CC(CCNC(C3CC4CCC3C4)=O)=N2)=O)cc1Cl C(C)(C)(CCC(=O)N1CCCC1CF)NC(C1CN(CC)C(=O)C1)=O N1(C(c2cc(C(C)C)no2)=O)CC(NC(c2ccn(CCF)n2)=O)CC1(C)C C(=O)(CCS(N)(=O)=O)NC(CC(C)C)CNC(=O)CC(O)Cc1ccccc1 C1(OC)CC(CNC(=O)CSc2cscn2)N(C(C2CC3CC3C2)=O)C1 C(CCCC(=O)N1CCCC1CN(C(=O)C(C)O)C)n1c(C)ncc1 Cc1ncccc1CC(=O)NC1(CN(C(=O)C=CC(=O)N(C)C)C)CC1 N1(C(c2c(C)nn(CCO)c2)=O)CCCC(C)(NC(c2ccc[nH]2)=O)C1 c1(NC(C2CCN2C(=O)Cc2c(F)cccc2F)=O)ccc(F)c(F)c1O Nc1ccc(C(O)C(=O)OCC(=O)NCCNC2CC2)cc1 N1(C(CC(C)C)=O)CC(CC(=O)NC2(C)CCSCC2)CC1C C1(NC(C2CC(CCF)C2)=O)CC2CC(C1)N(C(=O)COC1CCCCCC1)C2 C(CCC(N)=O)(C(=O)NC1CCCN(C)C1)n1cc(-c2ccc(C)cc2)nn1 n1(CCOC)ccc(C(=O)NC2CC(CCNC(c3cc(C)cs3)=O)C2)n1 C1(NC(C=CC)=O)CN(C(=O)CCc2cc(Cl)cc(Cl)c2)C(C)(COC)C1 c1(C(=O)NCc2nnn(C)c2C(=O)NCCCN(C)C)nnc(O)nc1O c1(CN(C(CC=C=C)=O)C)cccc([N+](=O)[O-])c1.C12(O)CCN(C1)C2=O c1(C(=O)NCC2(CNC(c3c(C)[nH]nc3Cl)=O)CC2)cc(O)nc2ccccc12 C1(CCC)CC(C(=O)NC2(C)CN(C(=O)Cc3cnccn3)C2)CCO1 N1(C(CC=C)=O)CCC(CCCCNC(=O)C(c2ccc(Cl)cc2)CC)CC1 C1(CNC(CNC(CNC(c2n(CC#C)ccc2)=O)=O)=O)CN2CCC1CC2 CN=c1[nH]cc(C(N2CC=CC2(C)OCC(N2CCC(c3ncc[nH]3)C2)=O)=O)o1 c1(N2CC(NC(C=C(C)C(F)F)=O)CC3(C2)CCC3)c(Br)cncc1[N+](=O)[O-] CCCN=c1[nH]c(N2CC(CC)C(CO)C2)nc2c1CCCCC2 Cc1cc(CC(=O)NC2CCN(C(=O)C(C)Oc3ccc(CO)cc3)C2)c(C)s1 c1(OCC(=O)OCC)cccc(NC(C23CCC(CO2)C3)C)c1 CC1C(NC(=O)C(=O)N(C)C)CCN1C(=O)Cn1cc(C2CC2)cn1 N1(CCCC)CCOCC1C(=O)NCC(CNC(c1nccn1CC)=O)CO c1(C(=O)NC2CC3CN(C(C4CC(=C)C4)=O)C(C2)C3)ccc2c(c1)CC(=O)N2 N1(C(c2c(C)cc(O)nc2C)=O)CCC2(CC1)CCN(C(c1cnns1)=O)CC2 c1(CNC(C(C=C)O)=O)cccc(C2CC2)c1C c1(C(=O)NCCC(=O)N2CC(C(C)N)C2)cccc2cncn12.CC(=O)OC Cc1ccc(C)c(C(N2CC(C)N(C(c3nn[nH]c3Cl)=O)CC2C)=O)c1N C(N=c1[nH]c(C)ncc1C)C1C(C(F)(F)F)CCN(C(c2cccc(C)n2)=O)C1 C1(C)(CNC(C2CC(C)OC2)=O)CCCN(C(c2cnoc2C(C)C)=O)C1 CCCCCCCCC(=O)N1CC(CNC(=O)C(CC)C2CCOC2)(COC)C1 CCC(C)(F)C(=O)NCC1CC1CNC(=O)CCc1nc(C(F)(F)F)n[nH]1 C1(N(C(c2ccnc(CC(C)C)n2)=O)C)CN(C(=O)CC2CCCO2)CC12CC2 C(=O)(C(C#N)C(C)C)NC1C(OC)CN(C(c2cn(CCCF)nn2)=O)C1 N1(C(C(C)C#N)=O)CCCC(O)(CN(C)C(c2cccc(F)c2)=O)C1 c1(C(=O)NCC(C)(C2CCC2)NC(c2cnc[nH]2)=O)ccc2n[nH]cc2n1 C(=O)(CCC(C)(C)C(=O)N1CCCC1CNC(c1cnn(CC(C)C)c1)=O)OC c1(C(N2CC3(C(NC(=O)C(F)F)CCC3)C2)=O)cnc2n1CCCCC2 c1(C(=O)NCCC2CCN(C(C(C)=C3CCCC3)=O)C2)ccc(F)cc1Cl N1(C(CCCC)=O)CC2CCN(c3c(OC)ccc(CC=O)c3)C(C2)C1.O(C)CC N1(C(CN(CCC)C)=O)CCC(NC(=O)CC2(C)CC2(Cl)Cl)CC1C C(c1ccc(F)c(F)c1)=C(C)C(=O)N(C(C1CCCCC1)Cc1ncccn1)C C1(OC)CN(C(C)=O)CCC1CO.C1(=O)C(C)(C)COC(=O)C2CCC2N1 C1(C(=O)NCC2C(NC(=O)C3=CCCC3)CCCC2)CCC2(CC1)CC2 CC1(C)CC(C(=O)NC2(CCC(=O)Nc3ccc(F)cc3)CCC2)=NO1 CCC1=NOC(C(=O)NC(C)CCNC(=O)CCc2ccccc2C(N)=O)C1 c1(C(COC)NC(CCN(C2CC2)CC)=O)ccc(NC(=O)CC)cc1 CC1CN(C(=O)C(O)Cc2ccccc2)CCN1C(C1CC2(C1)CC21CC1)=O c1(CNC(C2CCC(C)O2)=O)nnn(C)c1C(=O)NC(C)C(=O)N(C)C C=CC(C)CC(=O)NCCCOCCNC(c1ccc(C(C)(C)C)cc1)=O C1(C(C)C)CN(C(c2cc(C3(C)CC3)on2)=O)CCN1C(=O)C=C1CC1 Cc1ccc(Cl)c(F)c1C(=O)NCC1CC2COCC2N1C(C12CC(F)(C1)C2)=O C(=O)(C(C#N)(CC)CC)NC1(CNC(C(CCCC)N(C)C)=O)CCC1 c1(C(=O)NCc2cccnc2-c2cnc(N3CCC3)nc2)ccc(O)cc1Br c1(N2CCC(NC(C3CCCN(C)C3)=O)C(O)C2)ncnc2c1cnn2CCO C(C(C(=O)NCC(=C1CN(C(C2(CC(F)F)CCC2)=O)C1)F)OC)OC C(C(CC)(CC)CO)NC(C(C1CN(C(c2cccc(CC)c2)=O)C1)O)=O O=S(=O)(c1ccc(NC(CO)C2CC2)nc1)Nc1nc(C2OCCO2)cs1 CC(C)C(C)(CN=c1ccc(-c2ccncc2)n[nH]1)NC(c1csc(Cl)c1)=O CC1CCCN(C(=O)C(N2CCC(C(=O)NC(=O)CSc3cnn(C)c3)C2)=O)C1 C1(CC)(NC(=O)NC2CC(C(N3CCC(c4ccon4)C3)=O)C2)CCCC1 C(=O)(C(C)(C)C(=O)N1CC(NC(c2coc(C(C)(C)C)n2)=O)C(F)C1)OC N1(C(c2cn(CC)nc2C2CC2)=O)CCCC(NC(C2CCCOC2)=O)C1C Cc1nc(C)c(C(=O)NC2CCCC2NC(c2nn[nH]c2Cl)=O)[nH]1 Cn1cnn(CCNC2CC(CO)N(C(=O)Cc3cccnc3)C2)c1=O c1(CC)ccc(C(N2CC(CNC(=O)C(C)C3CCCC3)C(C)(C)C2)=O)c(C)n1 c1(N(CCN)C(c2ccncc2Cl)=O)cnc2c(c1)CNCC2 Cc1cc(Br)ccc1-n1nc2nc1C1CC(=O)N2C1.c1cnn(C)c1 C(=O)(CC(CC)CC(C)C)N1C2(CNC(C(CCC)C)=O)CC(C1)C2 C(=O)(C(CO)c1ccccc1)NC(CC)CNC(=O)CCC1OCCO1 C(CC(=O)N1CCCCC1CC(C)C)(C(F)(F)F)NC(CCCC#CC)=O N1(C(C(C=CC)O)=O)CC2(CCC2)CC1CNC(c1c(NC)cccc1Cl)=O c1(CC)nc(C)c(C(=O)NC(C)(C)C(C)NC(=O)Cc2ccc(Br)nc2)s1 N1(C(CCc2c(C)noc2)=O)CCCC1(C)C(C)(C)CNC(=O)CCNC(N)=O c1(COC)ccnc(C(N2CCC2C(=O)NCCC2CC2C2CC2)=O)c1 c1(C(C)(C)C)nc(N2CC3CC2CN3C(c2cc(C(F)F)[nH]n2)=O)[nH]c(=N)n1 C#CCCCCC(=O)N1CCC(C)C(CNC(c2cnn(C3CC3)c2)=O)C1 C1(CCNC(Cn2c(C)ncc2)=O)CN(C(=O)C(=O)Nc2ncc[nH]2)CC1C CC1CN(C(C2CC=CC2)=O)CCC1CNC(=O)Cc1c(F)cccc1F CC1CC(CCNC(C2CN3CCN2CC3)=O)CCN1C(=O)Cc1cn[nH]c1 c1(CC(=O)N(CCCC(=O)N2CCC(CO)C2)C)cccc2c1OC(C)(C)C2 n1(CC)nc(C(N2CCCC(N(C)C(c3c(C)ncnc3O)=O)C2)=O)ccc1=O N1(C(c2cnc(C)nc2)=O)C2CCC1CC(O)(CNC(=O)CC(C)F)C2 CC1OC(C)C(C(N2CCC(CNC(=O)CSC(F)(F)F)C2)=O)C1C c1(C(=O)NCC(C)N(C(C(CSC)C)=O)C)cc(Cl)c(F)cc1Br c1(CNC(C2(CNC(C(C)OC)=O)CC2)=O)ccc(C2CCC(=O)N2)cc1 C(C)(C)(C(=O)N1CC(C(=O)NCC(C(=O)NCCNC(C)=O)O)C1)NC(C)=O C1(NC(c2n(C=C)ncc2)=O)CN(C(=O)CC(O)C2CCCC2)CCC12CCC2 C1(C(=O)NC(CNC(C2C(=C)CC2)=O)(C)C)CCc2ccc(F)cc2C1 Cc1cccc(C(=O)NCC(F)CNC(c2cccnc2-n2ccnc2)=O)n1 c1(C(N2CC3C(NC(c4cn(CCC)nc4)=O)(CC3)C2)=O)c(C)cc(C)nc1O C1(C(N(C2CN(C(C=CC)=O)C2)C)=O)CCC(OC)CC1 C=Cc1ccc(C(=O)NC(CNC(C2CC(COC)C2)=O)C2CC2)cc1 CC1CCCCN1CCC(=O)N1CC(CN(C(=O)CC2CCCN2C)C)C1 C(CCNC(=O)O)(C(C)C)NC(CN(C1CC1)CC)=O.C1CC(F)(F)CS1 Cc1c(C(=O)NCCCN(C(=O)C(C)C2CC2)C2CC2)sc2ccsc12 c1(C(CO)NC(C2CN(C(CNC(=O)NC)=O)C2)=O)csc(=N)[nH]1 C1(C(=O)NC(CC=C)C(=O)OC)CCN(C(=O)C(C)CC2CC2)C12CC2 c1(OCC)ccc2nc(C3CCCC3)nc(N3CCC(N4CC(C)(C)C4)C3)c2c1 n1(CCC)ccc(C(=O)NC2(C(=O)NCc3cnn(CCF)c3)CCSC2)n1 Cc1cc(Cl)ncc1CC(=O)NCC1CN(C(=O)C=Cc2cscn2)CC12CC2 N1(C(C=C(CCC)C)=O)CC(C)N(C(=O)CC2(NC(C)=O)CCCCC2)CC1C N1(C(c2nc(C#C)sc2)=O)CCC2CCC(C1)N2C(=O)C1=CC1.C(C)(=O)OC N1(C(C(C)=CC2CC2)=O)CCC(n2cc(CNC(c3csc(Cl)c3)=O)nn2)C1 C(=O)(C1CCCc2ccnn21)NC1CN(C(CN(C(C)=O)C)=O)C2C1CCCC2 C12CCCC(C1)NC2=O.C1(OCC(=O)OC)CCCCC1.c1(C(=O)N)ncsc1CC c1(C(=O)NC2CCC(C(=O)NCC(CO)SCC)CC2)c(F)ccc2n[nH]cc12 C(=O)(C(CC(=O)N1CCCN(C(c2csnn2)=O)CC1)C(C)=O)OCC N1(Cc2cn(C)nc2-c2nn(C)nc2Br)CCC2(CC1)COC(=O)N2 n1(CC(=O)NCC2N(C(C(F)=CC)=O)CCOC2)cc(P(C)(C)=O)cn1 C1(CNC(COCCCC)=O)CN(C(c2cc(C)c(O)nn2)=O)CCN1C C(=O)(CC(CC)C(C)(C)C)N1CCC(N(C(COCCCC#C)=O)CCO)C1 C1(OCC(N2CCCC2c2ncccn2)=O)CNCC12CC2 C1(C(C)C)N(C(=O)C(C)OCC2CC2)CC12CCN(C(=O)C(C)(O)C1CC1)CC2 N1(C(CC=CC=C)=O)CCN(C(=O)CC2(CC)CC2)C(c2cccc(OC)c2)C1 C1(NC(Cc2onc(C)n2)=O)C2CCC1CN(C(c1cccn3cncc13)=O)C2 c1(CCNC(C2(CNC(CC3CC(=O)C3)=O)CC2)=O)ccncc1F C1(N(CCC(=O)OCCCC(=O)OC(C)(C)C)CCCCCO)CCN(C)C(C)C1 c1(C(C)N(CCCCN(C(=O)CNC(=O)Cc2cccs2)C)C)nnnn1C C(C(=O)N1CCCCC1CNC(c1coc(Cn2cccn2)c1)=O)(C(C)C)OC c1(NC(C2(C)CCN2C(c2ccc(=O)n(O)c2)=O)=O)cnc(C#N)cn1 C1(C(=O)NC2(COC)CCOCC2)CCc2cc(F)ccc2O1 N1(C(C2CC3(CC(=C)C3)C2)=O)CCC(C2CC2)C1CNC(c1cc(OC)ns1)=O Cn1cnnc1CCCC(=O)NC1(C)CC(NC(C2(C)C=CCC2)=O)C1 n1(CCOC2CCC(C)(C)C2)cc(P(C)(C)=O)cn1 C(=O)(CC(O)CC(C)(C)C)N1CCCC(NC(CC(=O)OCCC(C)C)=O)C1 C12CC3(C1)CC(C3)N2.C1(C(=O)NCCNC(N)=O)CCCN1C(N)=O C1(CC)CN(C(C2CC(F)CN2C(C2CCOC2)=O)=O)CC(=O)N1 N1(C(C(=O)NCCOC)=O)CC(NC(C2CCC(=O)N2C)=O)CC2(CC2)C1 CCCCC(O)C(=O)NC1(C2CCCN2c2nnc(C(N)=O)s2)CC1 Nc1nccn2ncc(C(N3CCCC(NC(C4C(F)(F)C45CCC5)=O)C3)=O)c12 C1(NC(C2(CC#C)CCN(C(C3CCSC3)=O)C2)=O)CCCN2CCCC12 C1(C(N(C(CC)C)CC)=O)CCCN(C(C2(F)CCCCC2)=O)CC1 C1(N(C)C(=O)OC(C)(C)C)CN(C(c2coc(C3CNC3)n2)=O)CC1F C1(NC(c2cc(C)ncc2)=O)CN(Cc2cc(O)cc(Cl)c2)CC(F)(F)C1 C1(CNC(c2ccc(CC#N)cc2)=O)CCN(C(c2cnco2)=O)CC1O N1(C(c2c(N)cncc2)=O)CC2CC1CCC2NC(=O)C(O)C1CCCC1 C1(c2nnnn2CCCOCC)(NCc2ccc(C)cn2)CCN(C)C1C C1(CC)(NC(c2cc(C(F)F)no2)=O)CCCOC1 c1(C(N2CC(C3(NC(c4cc(OC)n[nH]4)=O)CC3)C2)=O)cc(F)c(Cl)cc1F CC(CC(C)(C)C)C(F)C(=O)NC1CCN(C(=O)C2=NOCC2)C12CCC2 C(CCCC(=O)N1CC(NC(c2nc(Cl)oc2C)=O)C(C)C1)OCCC=C O=C(C1=CC2CCCC12)N1CCC(CCNC(C23CC=CCN2CCC3)=O)C1 N1(CC(=O)NCC(CCNC(=O)C(C)=C2CC2)OC)CCc2ccccc21 c1(C(=O)NCC2OCCN(C(CC(C=C)C)=O)C2)nn(CC)c2c1COCC2 Cc1cc(C(=O)N(C)CC2COCCN2C(=O)C(C)CCO)c(C)n1NC(N)=O CN=C(NCc1cnc(-n2cccn2)s1)NCC(C)(F)F N1(C(c2c(CC)[nH]cc2)=O)CCC2C1CCCN2C(=O)Cn1cnnc1O N1(C(C(C)NC(CC)=O)=O)CCCC(n2cc(CNC(=O)C(C)(C)O)nn2)CC1 c1(C(N(C)CC2N(C(C=NOC)=O)CCCC2)=O)cccc(C(F)(F)F)c1Cl N(C(=NCCNc1ccc(Cl)cc1Cl)NC1CC(=O)NC1C)CCC(=O)OC CC1(C)CC(NC(C2CCCC(F)C2)=O)CN(C(C2(C(=O)NC3CC3)CC2)=O)C1 N1(C(CCCCCOC)=O)CCCCC(NC(c2cn(CCN(C)C)nn2)=O)CC1 C12(CNC(C3CCC34CCC4)=O)CC(CO1)N(C(=O)CSc1ccccc1)C2 CCCCCC(O)C(C)C(=O)NC1CCC(CNC(C2CC(N=[N+]=[N-])C2)=O)C1 Cc1cc(C(=O)NC(C)(C)C(C)NC(C2CC3(CCC3)CO2)=O)cc(C)c1C#N c1(C2(CNC(C3C(OC)(OC)CC3)=O)CC2=S)cccc(F)c1 c1(CN2CC3(CC(CC(=O)Nc4cccnc4O)C3)C2)cc2c(Br)cccc2s1 N1(C(c2c(C)nn[nH]2)=O)CCC(NC(c2cnc(C3CC3)nc2)=O)C(CO)CC1 CC(Cc1ccc(Cl)s1)N=c1[nH]c(N2CC(C)OCC(C)(C)C2)nc2c1SCC2 N1(C(C2(NC(C)=O)CCC2)=O)CC(C(=O)NC(C)C(=O)NC(C)C)C(F)(F)C1 Cc1cc2cc(C(=O)NC(CCN(C(=O)C(C)SC(C)C)C)C(C)C)ccc2[nH]1 C(C(CC)(CC)C(F)(F)F)NCC1(C)N=C(C)SC1 CC(c1ccccc1C)=CC(N1CC(NC(=O)C(C)CC(C)C)CC2(CC2)C1)=O C1(NC(CC=C=C)=O)CN(C(=O)Cn2cc(-c3cnccc3C)nn2)CC1CC c1(C(=O)NC(C)CN(C(=O)Cc2ncn(-c3ccccc3)n2)C)cncc(F)c1 C(=O)(CC(O)CC(C)C)N(CC(=O)NC(c1ccc(C)cn1)C)C C(C(C)CC(=O)NC1(CC2CCC2)CC1)NC(C1(COC)CC=CC1)=O c1(CCn2c(C(C3CCCCC3)NC3(CC=C)CC3)nnn2)cccc(Br)c1 CC(C)(C)C(=O)C(=O)N1CC(CNC(C2(C)CC3CC3C2)=O)C(F)(F)C1 C(=O)(C1=NOC2(CCN(C(c3cc4c(C)cccc4o3)=O)C2)C1)N(CCO)CC CC1CN(C(=O)CCC2CC2C)CCCN1C(c1cccc(OCC(F)F)n1)=O C1(C(=O)NCC23CCC(NC(CCC=C)=O)(C2)CO3)CCC([N+](=O)[O-])CC1 c1(C(=O)OC)cc(NC2C(CCNc3cccc(F)c3)C2)cc(Cl)c1 c12ccc(c(C(C)C)c1)C(c1nnnn1CC1CCCO1)N2.C1(CC)(CC)CC1 N1(C(c2cc(C(C)C)n(C)n2)=O)CCC(NC(C2OCC2(C)C)=O)C(O)C1 C1(CC(=O)NC2(C3N(C(CCCC=C)=O)CCC3)CC2)OCCCC1(C)C c1(C(C(=O)NCC(F)F)N(CC(=O)NC)CC(=O)NC)cscc1Br N1(C(c2c(C)nncc2)=O)CC2CC(C(=O)N(CC(C)(C)O)C)CC2C1 C1(C(c2n(CC)nnn2)NC2(C)CN(Cc3ccccc3)C2)CCCCC1OC c1(C(N2CC(NC(C=CS(C)=O)=O)C(CO)CC2)=O)ccc(O)c(F)c1F c1(C(N(CC(C)O)CCNC(C23CC(OC)C2C3)=O)=O)cccnc1O C12(C(N(CCN(C(c3cc(SCC)ncc3)=O)C)C(C)C)=O)CC(N=[N+]=[N-])C1C2 C1(NC(CC=O)=O)CCN(C(=O)C=CC(F)(F)F)CC1F.c1(C)cccc(F)c1 CC1C(NC(=O)C(C)(C)CN2CCOCC2)CCCN1C(c1nncn1C)=O c1(OC)ccc(F)c(C(=O)NCC2CCCN2C(C2OCCC2C(C)C)=O)c1F c1(C(=O)NCC(CC)NC(=O)C(CC)NS(C)(=O)=O)c(F)ccc2c1OCC2 c1(-n2cc(CN(C(C3CCCC3(F)F)=O)CC)nn2)ccc(C(=O)O)nc1 C1(NC(C2(CC)CCC2)=O)CC(CO)N(C(=O)COCC2CCCCO2)C1 CC(C)(C)CCCNC1(c2nnnn2CC2CC2)CC1(C)C.c1ccco1 c1(C(=O)NCCCOCCN(C(CC2(OC)CC2)=O)C)ccc(O)c(F)c1F N1(C(CCCC#C)=O)CCN(C(c2nnsc2-c2ccccc2)=O)CC1C(F)F c1(C(c2n(C3(C)CC3)nnn2)NC2(C)CCCCC2)cc2c(nc1Cl)CCCC2 OCC1=CC2CCC(C1)N2Cc1cc(Cl)ccc1-c1ccc(F)cc1[N+](=O)[O-] CC1(C)CCC(C(N2CCC(CN=[N+]=[N-])C2)=O)CN1C(=O)CCC1CCOC1 c1(C(N2C(CNC(C3CC=CCO3)=O)CCCC2)=O)onc2c1CCCC2 CC1ON=C(C(=O)NCc2cccc(NC(=O)C(C)(C)CN(C)C)c2)C1C CC(C)CC(C)(C)CNC(C1CCCC(NC(C2CCCC(C#N)C2)=O)C1)=O Cn1cc(C(N2CCC(c3cn(-c4ccc(F)c(N)c4)nn3)C2)=O)c2ccccc12 N1(C(CSSC)=O)CCC2(CC1)OCCC2NC(C1CCNC(=O)C1)=O c1(SC)cc(C(=O)NCCC2CN(C(=O)C(F)CC3CCOC3)C2)ccn1 C1(=O)C(CC)CCO1.c1(COCC(=O)Oc2ccsc2)scnc1C c1(OC)cc(C)c(C(=O)NC2CN(C(=O)CSC(C)(C)C)C(C)(C)C2)c(C)c1 CCCCCCCCCCCCS(=O)(=O)N1CC2C(C1)N2Cc1cccc(Cl)n1 C1(CNC(C(C=C)CC)=O)N(C(=O)COc2ccsn2)CCCC1(C)C c1(C(N(C)NC)=O)ccc(CNC(c2ccc(SC(C)C)cc2)=O)cc1 C(=O)(C#CC1CCCCO1)NCC1(F)CC(CNC(C(c2cccnc2)C)=O)C1 C#CCC(C)(C(=O)NCCC1CCSC1)NC(=O)C=CCO C1(O)(CN(C)C(C2CCC(C)O2)=O)CCN(C(C2CC23CCCC3)=O)CC1 C1(CC(=O)NCC2(CCNC(C(C)C3CCC3)=O)CC2)CCCC1(F)F N1(CC(C)(C)NC(C2CCSCC2)=O)CCN(C(C2CC3C=CC2C3)=O)CC1 CC1=C(C(=O)NCCC2COCCN2C(C2CC(F)(F)CS2)=O)CCC(C)(C)C1 c1(CCC(N2CC(C(F)(F)F)C3(CC3)C2)=O)cc(O)cc(Br)c1 C1(C)(CNC(CCC=C(C)C)=O)CCN(C(c2cc(CO)c(C)o2)=O)C1 C=CCC(C)(C)CN.C(CC)(CC)OC(=N)O c1(C(N2CCC(CC=C)(NC(=O)CCC(C)C)C2)=O)c[nH]c2cc(Cl)ccc12 C(=O)(C(C)CC(C)(C)C)NC(c1c(C(=O)NCc2ccc(C)cn2)con1)C C1(c2cn(CC(CSC)O)nn2)CCN(C(C2(CN(C)C)CC2)=O)CC1 C1(NC(CSCCC)=O)C2CC1CN(C(C1C=CCCC1)=O)C2 CCCS(=O)(=O)CC(=O)N1CCCC(F)(CNC(C2(N(C)C)CC2)=O)CC1 N1(C(CC2(C=C)CCC2)=O)CCCCC1C1CCCN1Cc1cc(Cl)ncc1Cl N1(C(=O)CCCCn2cc(CCCCO)nn2)CCC2CCCC(C2)C1 c1(CC(N2CC3CC(C2)C3NC(C2CC(F)C2)=O)=O)ccc2ccccc2c1 C1(CNC(CCCOCC=C)=O)CN(C(=O)COCC(=O)NC)CCC1(C)C C1(C(=O)NCCN(C(=O)CCc2ccc(Cl)nc2)C2CCCC2)(SC)CCOCC1 N1(C(c2ccc(F)c(OC)c2)C(=O)N(C)C2CC2)CCc2ccccc2C1C(C)C c1(OCC)ccc2nc(Cc3noc(C(C)OCC)n3)[nH]c2c1 c1(N2CC3C(CN)(C3)C2)ccnc2cc(Br)nn12.C(=O)OCC N=c1ccc(C(N2CCC(F)(CNC(c3nn[nH]c3Cl)=O)C2)=O)c(Cl)[nH]1 C1(OC)CCC2(C(N3CC(O)(CCNC(C4CCCN4S(C)(=O)=O)=O)C3)=O)CC12 C1(NC(C2CC3CCC2O3)=O)COCCN(Cc2cnc(Br)s2)C1 N1(CC(=O)N(C)CC2(CNC(c3c(C)snc3)=O)CC2)CC2CCC1C2 C#CCC(C)(CC)C(=O)N1CCC2(C1)CN(C(c1cc3scnc3[nH]1)=O)C2 C1(CNC(CN(C(C)C)C)=O)CCCC2CN(C(=O)CC(C)C(C)C)CC12 c1(C(=O)NC2(CNC(c3ccc(C#C)cc3)=O)CCOC2)ccc2nn[nH]c2n1 N1(C(C(C)C)=O)CC=CC(NC(c2ccn(Cc3ccc(Cl)cc3)n2)=O)C1 C1(C(=O)NCc2cc(C(N(C)CC3CC4(CC4)C3)=O)sc2)CCCCC1(C)C C1(CNC(C=CCOC)=O)CN(C(=O)CC(F)F)CCN1C c1(CC)occ(C(F)(F)F)c1C(=O)NCC1CC(O)(CNC(C2CC(C#N)C2)=O)C1 CCCCS(=O)(=O)CC(=O)NCCC(C)N(C(=O)CCCOC(=O)CC)CC Cc1nc(C2CCCO2)sc1C(=O)NCC[Si](C)(C)C C(CC(=O)N1CCN(C(CNC(=O)CNC(N)=O)C(F)F)CC1)(C(C)C)OCC C1(NC(C(C)OC)=O)CCC(C)(CNC(c2ccncc2)=O)CC1 C1(F)(C(N2C(C(=O)OC)C=CC2)=O)CCN(C(c2n[nH]c(C)c2O)=O)CC1 N1(C(C2CCC(Cn3cc(CCCCC)nn3)C2)=O)CCC(O)C(O)C1 C1(NC(CCC=CC)=O)CCN(C(=O)CCCn2cccn2)C(C)C1 c1(CC)nc2ccccn2c1C(N1CC2CC(NC(C3CCOC3)=O)C1C2)=O c1(C(=O)NC(CCNC(C(CC)NC(N)=O)=O)C)cnc(N)c(CO)c1 c1(Cn2cc(C3(C)N(C(C(C)OC)=O)CCC3)nn2)ccc(Cl)cc1Cl C1(C(N2C(CC)COCC2)=O)CC(O)CCN1C(=O)Cc1cccc(O)c1 C(=O)(C1Cc2ccc(F)cc21)NCC1(F)CC(NC(C(CC)(F)F)=O)C1 C1(N(C(C=C(C)C(F)F)=O)CC2CC2)CCN(C(C23CC(CF)(CO2)C3)=O)CC1 C=CCC(C)(CNC(C1CCC(O)CN1C(=O)CCC(C)N(C)C)=O)CO C(C)(C)(CCC(=O)N1C2CCC1CC2)NC(C1C(C)CC1)=O C(=O)(C#CC(C)(C)CNC(=O)CC(O)CN(C)C)NC1CCC(CC(C)C)C1 N1(C(C2(C#N)C(C)(C)C2)=O)CCC(NC(=O)CCNC(=O)C=CCl)C2(CCC2)C1 Cc1c(NC(C2CN(Cc3ccccc3Br)C2)=O)ccc(Br)c1F N1(C(C(C=C)(C)O)=O)CC(NC(=O)C(CC)NC(c2ccco2)=O)C(C=C)C1 C1(C(N(CC(C)O)CCNC(=O)C(Cl)=CCl)=O)CCCC2(CCC2)O1 c1(OC)ccc(SCC(=O)NC2CN(C(=O)Cc3cc(Cl)n(C)n3)CC2O)cc1 C1(C(C)C)CN(C(=O)C(=CC2CCCCC2)F)CCN1C(=O)C(F)=C1CCC1 C1(C(=O)NCCCCC=C)CN(C(=O)C(C(C)O)N(C)C)CCC1(C)C N1(C(C)CO)CCP(C)(=O)CC1.c12cccnc1CNn1cc(nn1)CN2 C1(CNC(=O)CCOCC(F)F)CCC2CN(C(c3ccnnc3)=O)CC12 Cc1ccnc(C(=O)NOCC23CNC(C)(C2)C3)c1C C1(C(N(C)CC2(C)CC2)=O)CCCCC1(C)NC(c1n[nH]c(O)n1)=O C1(NC(C2(NC(c3c(C)snn3)=O)CCSC2)=O)CCCC1(F)F N1(C(CC(C(=O)OC)C)=O)CCN(C(=O)C=Cc2cn(C)cn2)CC(C)(F)C1 N1(C(Cn2nnc(C)n2)=O)CC2(C1)CN(C(c1cc(Cl)n(C)n1)=O)C2 c1(OC)cc(C(N2CCC(O)(C(C)NC(C3(C)CC=CC3)=O)CC2)=O)cnc1C C1(C(N2CCC(F)(C(N3CCC(CO)C(O)C3)=O)C2)=O)OCC2CCCC12 N1(CC2CCC(C)(C)C2)CCN2C(=O)CCC2C1 CC1(C)CC(C(=O)NCC2(CNC(=O)COC3CCOCC3)CC2)CNC1=O C#CC(C)(C)C(=O)NC1CN(C(=O)Cc2cnc(C)s2)CC1C c1(C(C)C(=O)N2CCCC2)ccc(S(C)(=O)=O)cc1.c12cn(cn1)CC(=O)N2 C(CNC(=O)Nc1ccc(CC(C)C)cc1)(C(C)C(C)C)OC c1(CC(=O)NC(CNC(C(CC=CC)C)=O)C(C)C)ccc2cnccc2c1 C(CCC(=O)NC(CNC(C1CCCC1C(F)(F)F)=O)CO)N(C)C c1(C(C(=O)NCCN(C(C2CC3(CC3)C2)=O)CC)(C)C)ccc(Cl)nc1 c1(C(N2C(C)CC(NC(=O)CC(F)(F)F)CC2)=O)cccc2c1nnn2C c1(NC(C(CNC(c2ccc(OC)nc2)=O)N(C)C)=O)c(C)nn(CCO)c1C C(=O)(C1CCc2snnc21)NC1C(C)(CN(C(c2n(CC)ccn2)=O)C)CCC1 N#CC1CCC(C(=O)NC2CC(NC(c3cccc(OC(F)F)c3)=O)C2)C1 Cc1coc(C)c1C=CC(=O)NCC1CC(NC(c2ccc(C(F)(F)F)o2)=O)C1 Cc1sc(C(=O)NC2CN(C(C3CC3CC(C)C)=O)C2)c(Br)c1C C=CC(C)(O)CC(=O)NCC1CCC1NC(=O)Cc1ccc(C(F)(F)F)c(F)c1 C1(CNC(C=C2CCN(C)C2)=O)CN(C(C23CC(C2)C(C(F)(F)F)O3)=O)CCO1 C(=O)(C1CCc2cccc(F)c21)NC(CCCC)CNC(=O)C1=CC(C)(C)C1 c1(C(N2CCC(CCC(=O)OC)CC2)=O)ccc2[nH]cc(Br)c2c1 CC(C)CCC(O)C(=O)N1C2CCCC1CC(N(C(=O)C(O)CC(N)=O)CCO)C2 Cc1cc(C(=O)N(C)CCNC(C2OCCCO2)=O)nn1C1CC1 N1(C(C2CC3(CC(=C)C3)C2)=O)CC(NC(C2(C)CCCCO2)=O)CC2(CCC2)C1 C=CC(F)(F)C(=O)NCCCC(=O)NC1CC(C)(C(N)=O)C1 C1(N2CC3(CN(c4c(C#N)cncn4)C3)C2)CCOC2(CCCOC2)C1 c1(C(=O)NCC23CC2CN(C(c2ccsc2Cl)=O)C3)cn2ccccc2n1 CCC(C)(C)CNC(=O)C=CCC1(NC(c2ccon2)=O)CCC1 N(C(=NCCNS(=O)(=O)NCC(F)(F)F)NCCNCC)C(c1c(Cl)cn(C)n1)Cl C(=O)(C(F)C(C)CNC(=O)CCSCCOC)NCc1cn(CC)nc1 c1(C2CCN(C(CCCC#C)C(=O)NC)C2)ccc2c(c1)OCCO2 CCC1=NOC(CC(N2CC=CC2C(N2CCC2(C)C(=O)NC)=O)=O)C1 C1(NC(C(CC)C2CCOCC2)=O)CCN(C(C2(CF)CC2)=O)CC1F c1(C(=O)NC2CC(N(C)C(C3CC4C=CC3C4)=O)C2)ncnc2c1ccn2C c1(C(=O)NCC2N(C(c3occ(C)c3C)=O)CC2)ccc2c(c1)C(C)CO2 Cc1nn(C)c(Cl)c1CC1CCN(C(=O)CCN2CCOCC2)CC1 CC1(C#CC(=O)NC2CCCN(C(C3CC4CCC(C3)O4)=O)C2)CC1 c1(C(=O)NCC(CNC(CN(CCCCCC)C)=O)F)cc(C)ccn1 c1(-n2cc(C(N(C(c3ccoc3I)=O)CC)C)nn2)cnn(C)c1C(C)C c1(C(=O)Nc2cccc(NC(C3CC3F)=O)c2)ccc2c(c1)CCCO2 N1(C(C)=O)CSCC1C(=O)N(C1CC1)CC1C=CCN1C(=O)C=Cc1cnc[nH]1 CC(C(C)C(=O)NCC(O)COC(C)C)NC(C1CC1(F)Cl)=O c1(C(=O)NC(C)CCN(C(=O)Cc2cc(Cl)cc(Cl)c2)C)ccn2nccc2c1 c1(CC)ccc2c(c1)CCN2C(CCCF)=O.N12CCC(C1)C2C(=O)NC c1(C(=O)OC)cc(C(=O)NCC(O)CNC(c2nocc2C)=O)cc(Br)c1 c1(-c2cn(NC(=O)NC(CCSC)C)nn2)cc(F)cnc1Cl C(=O)(C1=CCCCCC1)NC1N(C)CCN(C(C(C)C(F)F)=O)C1 Cc1nc(C(=O)Nc2cccc(C(C)O)c2)ccc1-c1cccs1 Cc1ccc(C(N2CCC(O)(CNC(C34CCC3C4)=O)CC2)=O)c(=O)n1C c1(CC)ccc(C)c(C(N2CCC(CC)C2CNC(C2CC2C(N)=O)=O)=O)c1 Cc1cc(C)c(CC(N2CCCCC2CNC(c2ncn(C(C)(C)C)n2)=O)=O)s1 c1(C2(C(=O)NCCC3CCC(NC(c4cnc(C)o4)=O)C3)CC2)cccc(F)c1 Nc1cc(C(N2CCC3CCC23)=O)ccc1F.C12CCC1C(=O)N2 c1(CN2C(C(=O)NC3(CC)CC3)CC2)cncc(Br)c1 C1(OC)CC2CC(C(=O)NCCC(C)(C)NC(c3ccc(N)c(N)n3)=O)CC12 N1(C(CC2OCCN(C(C3CC4(CCC4O)C3)=O)C2)=O)CC(F)(F)C(F)(F)C1 c1(C(=O)NCC2(O)CCN(C(C(CC)F)=O)CC2)ccc2c(c1)CCC2(C)C C1(C(=O)NC2(CC=C)CN(C(=O)C(C)(C)n3cccn3)C2)C2CCCCC12 Cc1ncc(C(C)NC(c2cn(CCNC(=O)CCc3cccnc3)cn2)=O)s1 N1(C(=O)NCCC(=O)OCC)CCN(C(=O)C(CC2CC2)CC2CC2)C(CO)C1 CC(CC(=O)NC(C)(C)C(C)NC(c1ccc(N(C)C)nc1)=O)C(F)(F)F N1(C(C(=O)NCCOC)=O)CCOCC1CN(C)C(c1cscc1C)=O Cc1ncc(F)c(N2CCC(C)(C(=O)Nc3cnn(CCO)c3)C2)n1 C(=O)(CCCCCCc1ccccc1)N1CCC(NC(C=C(C)C)=O)CC1C1CC1 c1(CN(C(=O)Nc2cnc3n2CCC(C)C3)CC)cn2cc(Cl)cc(C)c2n1 C(=O)(C#CC1CCC1)N(C)CC1(O)CCN(C(=O)C=CCCc2ccccc2)C1 N1(C(CSCC=C)=O)CCC2(CC1)COC(C)C2CNC(C)=O CCCN(Cc1ccc(F)cc1Br)N1CCCC(OC(F)F)C1 C1(CCNC(C2CC2c2ccco2)=O)(NC(CCC(=O)NO)=O)CCCC1 c1(C(=O)OC)scnc1NC(=O)C(C)COc1ccccc1 C(=O)(C1CCCn2cnnc21)NCC1C(NC(=O)CNC(=O)Nc2ccsc2)C1 c1(C(=O)NCC2N(C(C3(C)C=CCC3)=O)CCN(C)C2)cc2nc(=O)ccn2[nH]1 C(CNC(=O)C(C)=CCNC(=O)C(C)N1CC(C)C1)(C(F)(F)F)OC c1(C(C2CCCN(C(c3ccc(Br)s3)=O)C2)O)cc(F)c(F)c(F)c1 N1(C(C2(CC#C)CCC2)=O)CCC2CN(C(=O)Cc3cnccn3)CC2CC1 C(=O)(C(F)C(=O)OC)N1CC(CNC(C2C(OCC)COC2)=O)(OC)C1 N1(C(c2c(CC)scn2)=O)C(C)C2CC1C2NC(c1ccc(F)cc1)=O C1(NC(C2(C(C)NC(c3c(C)n(C)cn3)=O)CC2)=O)CCN2CCC1C2 N1(C(C(CC)N(C)C)=O)CCN(C(=O)Cc2cc(C)ns2)CC1C1CC1 Cc1noc(C)c1CC(N1CCC(N(C)C(C2CC(C)(C(C)(C)C)C2)=O)C1)=O N1(C(=O)OCC)CCCC(CC(N2CC(C(=O)Nc3cnns3)C2)=O)C1 C1(C(N2CCCC(C(C)C(=O)NCCc3cc[nH]n3)C2)=O)NC(=O)OC1(C)C c1(C(=O)NC2C(C(N(C)CC3(O)CCC3)=O)CCCC2)sccc1S(=O)(=O)N(C)C C1(NC(=O)C#CC2CC2)CCN(C(c2ccc(C(F)(F)F)nc2)=O)C12CC2 C1(C(c2n(CCOCCOC)nnn2)NC2CC2)OCCOC1(C)C Cc1cc(C(=O)Nc2c(C)cc(Cl)cc2C)cc(C)c1C#N CCC(CC)CCCC(=O)N(C)CC1(CNC(=O)CC2CCCCC2O)CC1 c1(NC(N2CCCC(CC3CCCCC3)C2)=O)cccc(C2CC2)c1 c1(C(=O)NC(C(C)NC(CCC=C)=O)(C)C)cn2c(n1)SCC2 C1(CNC(COCCC(C)C)=O)CN(C(=O)CC23COC(C)(C2)C3)CC1C C1(C(=O)NCCCN(C(=O)CN(C)C)CCC)CCCCO1 C1(C(=O)NC2C3CN(C(c4c(CC)c[nH]c4)=O)C2C3)CCc2nc[nH]c2C1 CC(CS(C)(=O)=O)C(=O)NC(C)(C)CNC(=O)CNC(c1cccs1)=O C12(C(=O)NCCOCCCN(C(C(C)C3CCOC3)=O)C)CCC(CC1)C2(C)C C(=O)(CC(C)C1CC1)NCC1CN(C(C(N2CC(C)C2)C)=O)C1.C(=O)(C(C)(C)C)N CCCCC(C(=O)NC1(c2nc(C)no2)CC1)NC(C1(CC)CC1)=O Cc1ncc(C(N2CCSC(C(=O)Nc3cnc(I)cn3)C2)=O)cn1 C1(c2ccccc2)(CNC(CSCCCC)=O)CCN(C(C2CCCC2C)=O)CC1 C=CC1(C(=O)NCCCC(C)NC(=O)C(c2cscc2Br)=O)CCC1 c1(C(=O)NCC(CN(C)C(c2ccc(=N)[nH]c2Cl)=O)(C)C)cn(C)c(=O)cn1 N1(C(CSCC#C)=O)CCC2(CCC(N(C(=O)CC3(O)CCC3)C)CC2)C1 C1(C)(C(=O)NC(C23CC(CO2)C3)C)CN(C(c2cnsc2)=O)C(C)(C)C1 N1(C(COCCOCC)=O)CCCCC2(C1)CN(C(=O)C(S(C)(=O)=O)C1CC1)C2 C1(C(=O)NC(CC#C)CC)CCCCCN1C(C1CN(CC)CCO1)=O S(=O)(=O)(c1cccc(-c2cnnc(O)c2)c1)NCc1ccc(C)c(Cl)c1Cl C(C#Cc1cccnc1)NC(C1(C)N(C(CC2CC(=C)C2)=O)CC=C1)=O C(=O)(C(C)CCCOC)N(c1cc(CC)ncc1)C.C1(O)CC=CC1.C1(=O)CO1 C1(C(=O)NCCCOCCN(C(C(C)n2cccn2)=O)C)CCn2ncnc2C1 c1(C2C(C(=O)NC(C(C)NC(c3cc(C)sc3C)=O)CO)C2)c(F)cccc1F N1(C(c2c(F)cc(C(F)F)cc2F)=O)CCCC2(CCC(NC(=O)CCF)C2)C1 c1(C(N2CCC(NC(c3cnc(OC)s3)=O)C2)=O)ccnc(SC2CC2)c1 N1(C(C2CCCC2C(=O)OC)=O)CC2OCCN(C(=O)C(F)=CC3CC3)C2C1 C1(NC(C(C)(C)NC(=O)NCC)=O)CN(C(=O)C(F)=CCCF)C2(CCCC2)C1 C(=O)(C(C)(F)C(C)(C)F)N1CCN(C(c2cc(OCC)no2)=O)CC1 c1(C(N2CC(NC(C3(C(F)(F)F)CC3)=O)C(CC3CC3)C2)=O)ncc(F)cc1F c1cc2nc(N3CCC4(CC3)CSC4)[nH]c(=NCC34CCC(C3)C(=O)N4)c2[nH]1 CC1CC(NC(c2c[nH]nc2Br)=O)CN1C(=O)C(=O)NC1CC1 c1(COC(C(C)SCc2ccc(OC)cc2)=O)ccc(Br)c2cccnc12 C1(NC(c2ccc(OC)nn2)=O)CN(C(C2CN3CCC2CC3)=O)CCC1CO c1(C(=O)NC2(CCC)CCCN(C(CCCC#C)=O)C2)cc(C)c2[nH]cnc2c1 c1(C(=O)NC2CC(N(C(c3cc(C)cc(C)c3)=O)C)C2)ccc2cc[nH]c2c1F Cc1nc(C)c(-c2cn(Cc3ncoc3CNC(C3COC(=O)N3)=O)nn2)s1 Cn1ccc2cccc(C(=O)NCC34CC3CN(C(=O)CC(C)(C)O)C4)c12 C1(N(C(C(C2CCOCC2)OC)=O)C)CCCCN(C(C2(O)CCCC2)=O)C1 C(=O)(CCCCC(F)(F)F)N1CCN(C(C(COC(C)C)(C)C)=O)C(C)C1 CC12CN(C(C3C4CCC3(c3cccnc3)C4)=O)CC1C1C=CC2CC1 N1(C(c2c(C)oc(CNC(=O)CN3CCC(C)C3)n2)=O)CC2CCC(C1)N2C c1(NC(C23CC2CN(C(c2n(C)ccc2)=O)C3)=O)cc(Br)ccc1OC(F)(F)F C1(CC(N2C(CC)CN(C(c3nnc(C)s3)=O)CC2)=O)CC2(CCOCC2)CO1 C(C)(C)(CC(F)C(=O)NCC(c1ccncc1)C)NC(CC1CCCC(C)O1)=O C1(NC(C(=O)NCCC(C)Nc2cc(N(C)C)ccc2F)=O)CCCCC(=O)C1 c1(C(=O)Nc2ccc(N(C)SC)cc2)cc(CCOC(C)C)n(C)n1 Cc1c(C(=O)Nc2cccc3c(C)cccc23)[nH]c2c(Cl)cccc12 C(=O)(CCCCCOC)N(C1(O)CCN(C(c2cccc(F)c2F)=O)CC1)CC Cn1cncc1C(=O)NC1CCC(NC(c2cnn(Cc3ccccc3)c2)=O)C1 c1(-c2cc(OC(C)C)cc(F)c2)cc(C(=O)Nc2cccs2)cc2[nH]ncc12 N#Cc1ccc(C(N2CCC(O)(CNC(C34CCCC3OCC4)=O)C2)=O)c(O)c1 C1(C(=O)NCC(C(C)C)CO)C2CC3C(C2NC(=O)CCc2cnn[nH]2)C13 c1(CNC(c2nc(C(C)(C)C)[nH]n2)=O)ccc2cccc(F)c2n1 C1(=O)C2=NOC(C2)CN1.c1(C(N(c2ccc(CC)cc2)C)=O)cn2c(n1)CCC2 C1(CC)CCCN1C(c1sccc1CNC(c1ccn(C)n1)=O)=O c1(C(=O)NC2CCCC2n2cc(C(=O)O)nn2)cc(I)sn1 c1(CC)c(C(=O)NC(C)CCCNC(C2CN(C(N)=O)C2)=O)ccn1C CC(C)(CO)C(C)(C)NC(C12CC(CN1C(=O)Cc1cc[nH]c1)C2)=O C1(C(C)C)N(C(=O)C(F)(F)C(F)(F)F)CC12CCN(C(=O)CCc1cnco1)CC2 C1(C(=O)OC2CN(C(=O)NC(C3CCC3)C)C2)CCCCCC1 CC(CC=O)C(F)F.C1N(CC(C2CCCC2)O)CCOC(c2ccccc2)C1 N1(C(c2cn(CCC)nc2)=O)C2COCC1CC(NC(=O)Cc1csc(C)c1)C2 C1(CCNC(C=C(CC)CC)=O)CN(C(c2cnc(C(C)C)[nH]2)=O)CC1C c1(C(N2CC(C(C)NC(C=Cc3cnc(C)s3)=O)C2)=O)ccc(N)c(F)c1 Cc1cccc(COC(C)C(=O)NCC2CC(F)CN2C(=O)Cc2cnns2)c1 C1(C(N2CCC(NC(=O)C=Cc3ncco3)(CF)C2)=O)CCc2nccn2C1 c1(CNC(C)=O)ccc(C(=O)NC(C2CCOCC2)CC2CCOC2)cc1F N1(C(N2CCCCCC(CCn3ccnn3)C2)=O)CC2CCCC(O)C2C1 CCC(CNC(=O)NCCCOCCN(C)C)(CC)C(=O)Nc1ncc[nH]1 c1(C(=O)NC(C)CN(C)C(C2CCNC(=O)C2)=O)cc2ccccc2cc1Cl CC1(C)CCN(C(c2cccc(N)n2)=O)C1CNC(=O)C(F)(F)C1CCCC1 N1(C(c2cccc(N)c2O)=O)CCN(C(C2(C(N)=O)CC2)=O)C2(CCC2)C1 N1(C(Cn2ccc(C)n2)=O)CC(NC(c2cc(O)ncc2Br)=O)CC(C)C1 c1(OCC)ncc(NC(C2CC(OC(C)(C)C)C2)=O)cn1 c1(C(N2CCC(n3cc(CN4CCCC4)nn3)C2)=O)cccc2[nH]ncc12 C1(CCC=C)CCCC1N=c1[nH]c(=NCc2nc(C)c(C)[nH]2)[nH]c2c1CSC2 Cc1csc(=NCC(=O)NCC(CNC(=O)C(c2ccc(F)c(Cl)c2)O)CO)[nH]1 C1(CNC(c2cc(C(N)=O)[nH]n2)=O)C2CCCC1N(C(C1(C(=O)NC)CC1)=O)C2 c1(CC(N2C(C(C)NC(CC=CC=C)=O)CCC2)=O)csc2nccn12 C1(C(=O)NCC(C)NC(C2(C)CCC(F)(F)CC2)=O)CN2CCN1CC2C c1(C(=O)NCCOCCCN(C(c2c(C)nn[nH]2)=O)C)cc(C)n(C)c(=O)c1 c1(OC)cccc2sc(C(N3CCC(C)(NC(=O)C(C(=O)OC)OC)C3)=O)cc12 N1(C(c2cccc(C(=O)NC)c2)C(=O)NC(CC)C)CC(C)c2ncccc21 C(=O)(C(C(C)(C)C)n1cc(CC2CCOC2)nn1)NC1(CCOC)CCNC1=O C#CCC(CC(=O)N1CC(O)(C(C)C)C1)NC(c1cc(O)ccc1F)=O C12(C(N3C(CC#C)(C(=O)NCCCCC#CC)CCC3)=O)CC(C)(CCO1)C2 N1(C(c2c(C)csc2)=O)CC(C(=O)NCC23CCCN2CCC3)C(F)(F)C1 C12(NC(CCCC)=O)CCCCC1N(C(=O)CCc1ccc(OCC)cc1)CC2 c1(C(=O)NCC2C(NC(Cc3c(C)occ3)=O)C2)ncnc2cc[nH]c12 Cc1ccsc1C(N1CCC(OCC2CCOCC2)C1)C(=O)NC1CCC1 c1(COC2CC3CC(CNC(c4nnnn4C)COC)CC32)cc(F)cc(F)c1F C1(CNC(CC2CCC(C)CC2)=O)CC2(CO1)CN(c1ncc(O)cn1)C2 c1(NC(C(=O)NCC=CCSC)=O)ccc(NCC#N)cc1 C1(OC)CN(C(c2cscn2)=O)C(C)(CNC(c2cnccn2)=O)C1 c1(OCC)cc(Cl)ccc1C(=O)NCC1COCC1NC(=O)C(C)OC(C)C C1(NC(c2c(C)ccs2)=O)CC1C1CCCN(C(=O)Cc2cnsc2)C1 C1(C(=O)NCC(CC=C)NC(c2nccc(CO)n2)=O)CCC(=O)N(C(C)C)C1 CCCCCC(O)CNC(C1(C(C)C)CCN(C(c2nnsc2N)=O)C1)=O C1(Cc2c(C)nc(C)o2)CN(C(c2nn[nH]n2)C)CC1(C)C C(=O)(C1=C(Cl)CCCC1)N1CCC(NC(C2C(C#C)C2(C)C)=O)C1 C1(CC(=O)NC2(CCCNC(c3cc[n+]([O-])cc3)=O)CC2)CCCS1(=O)=O N1(C(CC2N(C(C)C3CC3)CCC2)=O)CC2CCC(C1)N2C(=O)CCC1CCCOC1 N1(C(CCC(C)NC(N)=O)=O)CCN(C(C2(N(C)C)CC2)=O)CC1CCOC C1(C(=O)NCCOC2CC(C(CCNC(C)(C)C)=O)C2)CC1(F)F.C(=O)OC C1(C(=O)OC)OC(C(=O)NC2(CNC(=O)CC3CC4CC4C3)CCOCC2)CC1C CCC(CCC(=O)NCc1cc(C(C)C)no1)NC(c1nc[nH]n1)=O C(=O)(C(C(C)OC)N(C)C)NC(C(C)C)CNC(C1SCCCS1)=O C1(CNC(C2C=C(C)CS2)=O)C(C)CCCN1C(=O)Cc1c[nH]nc1C C1(C(=O)NCCOC)CC2C=CC1N(C(C1CCC(C)O1)=O)C2 N1(C(C(C)OCC)=O)CCC2(CCC2)C(NC(c2cc([N+](=O)[O-])cc(C)n2)=O)C1 CC1(C)CCCC(NCC2N(c3ccnc(N4CCSCC4)n3)CCOC2)C1 CC(F)(F)C(F)C(=O)N1CCCCC1C(=O)NCCC12CCC(CC1)C2 CCCC(C(=O)NCC1CC(NC(C23CCC(C2)OC3)=O)C1)NC(N)=O N1(C(Cc2n(C)ccn2)=O)Cc2n[nH]cc2C1C(=O)N(C)C(C1CC1)CC1CC1 C(CCCC(=O)N1CCC(n2cccc2)C1)N(C)C(c1cccs1)=O S(=O)(=O)(c1csc(C(N2CC(CCO)(NC(c3cc[nH]c3)=O)C2)=O)c1)N(C)C N1(C(CCC(=O)c2ccc(C)s2)=O)CCCN(C(C2(CC3CC3)CC2)=O)C(C)C1 C(=O)(C(C)C(C)NC(c1snc(C)c1N)=O)NCC1N(CCC)CCC1 c1(CCC(=O)NC2CCCN(Cc3cc(C)on3)C2C)nc2ccccc2[nH]1 C12(CNC(c3c(C)nn(C(C)C)c3)=O)CCC1CN(C(c1[nH]ncc1C#N)=O)C2 C1(C(=O)NCCCNC(CCC2CCC(C)O2)=O)CC(F)C(=O)N1C CC1(C(F)F)CC1C(=O)N(CCC(=O)NCCN1CCCC1)C1CC1 C1(CC(=O)NCC(C)CNC(=O)Cn2cc(C3CC3)cn2)CCCC1(F)F O=C1CCC(N2CC(C(=O)NCCOc3ccc(Br)cc3)CC(F)C2)C(=O)N1 c1(COC(C(c2c(OC)cccc2Br)(F)F)=O)cc(C)c(OC(F)F)c(C)c1 Cc1oc(C#N)cc1C(=O)NC1CCN(C(=O)Cc2ccc(F)cc2Cl)C(C)C1 C#CC(C)(C)C(=O)NCC1CCCCN1C(=O)C(C)NC(c1cnoc1C)=O N1(C(C(C)C(C)O)=O)CC2CCCC(C1)N2C(=O)CCOc1ccccc1C#N Cn1cc(C(=O)NC2CCCC2NC(=O)COC(C)(C)C)c(O)nc1=O c1(CN(CCC(N2CCC(CC(=O)O)C2)=O)C2CC2)cncnc1C.C(=O)OC C12(CC(=O)NC3(CO)CN(C(C(C(C)(C)C)OC)=O)C3)CC3CC(CC(C3)C1)C2 c1(CC)ccc(C(=O)NCCc2nc(-c3ccccc3)cs2)cc1F C(C)(CCC(=O)NCC(C)NC(C1(c2ccccc2)CC1)=O)OC N1(C(C(CCCC)O)=O)CCC2CCN(C(=O)CCc3cncs3)CC2C1 c1(C(c2n(CCOC)nnn2)NCC(c2ccncc2)C)sc(C)cc1Cl C12(NC(C(CC)(C)F)=O)CCCC1CN(C(=O)CCOc1ccccc1Cl)C2 C(CC(C)CCNC(=O)C(O)CN1CCOCC1)NC(CC(=O)OC)=O C(=O)(C(C)C(C)(C)C)N1CC(CC(C(=O)N(CC(=C)C)CC(=C)C)F)C1 c1(C(N2CC3(C(NC(CC4ON=C(CC)C4)=O)CC3)C2)=O)ccc2c(n1)CCO2 C12(CNC(C3CC(N(C)C)C3)=O)CC(C1)C(C)(C)O2.C1(C2CC2)(NC=O)CC1 CC1CCN(C(=O)CCc2ccncn2)CC1CC(N1CCc2n[nH]cc21)=O CCCCC(O)C(C)C(=O)N1C(C(=O)NOCC2(F)CCC2)CC2CC12 C1(OC)CC12CCN(C(C1CC3CCC(C1)N3C)=O)CC2 c1(C(=O)NCC2CCCC(NC(COCC(C)(C)C)=O)C2)ccc2cncn2c1 C1(NS(CC)(=O)=O)CCOCC1NCCN1CCCC1 C(=O)(C1CCCc2nnn(C)c21)N(CCNC(C(CC(C)(C)C)OC)=O)C c1(C(=O)NC(CC)CNC(=O)C(C)(C)CC2CC2)ccc(OC)c(N)n1 c1(OC)ccc2cc(C(N3CC(CCNC(=O)C4=CCCOC4)C3)=O)[nH]c2c1 C1(C(=O)Nc2ccccc2O)CC1C1CCCN(C(=O)CSc2nncn2C)C1 c1(C(N=c2nc(C(=O)OC)[nH]s2)=O)cc2c([nH]1)CCN(Cc1ccccc1)C2 C1(C(N(CC(=O)N(CC)CC)C)=O)CCC2(CC2)N1C(=O)Cn1nccn1 C(=O)(CC(C)NC(=O)C(C)(C)N(C)C)N(CCN(CCC)C)CC C1(C2CN(C(COC(C)(C)C)=O)C2)CN(C(c2cccnc2F)=O)CCO1 C1(NC(CCCn2ncc(C)c2)=O)CCOC(CNC(=O)Cc2c(C)cnn2C)C1 c1(C(N(c2cc(F)cc(C)c2I)c2ccccc2)=O)cc([N+](=O)[O-])ncc1Br N1(Cc2nccc(C(N(CCCOC)C)=O)c2)CCCC(C)(NC(=O)CCCF)C1 O=C(N=c1c(Cl)c[nH]cc1Cl)C(=O)Nc1nnc(C2C3CC4C(C3)C24)o1 c1(C(NOCCCCC)=O)cc(C(C)C)on1.C12(CCC1)C(=O)NC2 c1(C(N2CCCC(N(C)C(C3CCCC3CF)=O)C2)=O)c(N)cccc1Cl C(=O)(C(c1ccco1)N(CCOC)Cc1cccs1)NCCCOC=C C(CS(=O)(=O)CC(=O)NC12CC1CN(C(c1nc(C3CC3)cs1)=O)C2)OC C(C)(CCC(=O)NCCn1cc(C(N2CCCCC2C2(O)CC2)=O)nn1)SC N1(C(CC2(C=C)CCC2)=O)CC(NC(c2cc(Br)no2)=O)C(C)C1 C(CC(C(=O)N1CCC(C(F)(F)F)C1)NC(=O)COCC1CCCC1)N(C)C N1(C(CC2(COC)CC2)=O)C2CCC1CC(NC(C1CCC(C3CC3)C1)=O)C2 c1(C(N2CCN(C(c3cc(C)sc3)=O)CC(O)C2)=O)ncn2c1CCCCC2 C1(C)(C(N(C(C)CNC(=O)CCN(c2ccncc2)C)C)=O)CC(C2CC2)=NO1 O=C1C2CSCCCN2C(=O)N1c1ccc(F)cc1F c1(C(N2CC(C)C(CNC(=O)CN3CCCS3(=O)=O)C2)=O)ccc(O)c(O)c1 c1(C(=O)OCC)cnc2sncc2c1NC1CC(NC(c2cnsn2)=O)C1 N1(CC(N2CC(CC(=O)Nc3ccn(CCO)n3)C2)=O)CCC(F)CC1 c1(C(N(C2CCS(=O)(=O)C2)CC(N)=O)=O)cc2c[nH]cnc-2n1 N1(C(CCC#C)=O)CC2C(NC(C3C(C)(C)C3(F)F)=O)C2C1 c1(C(=O)NC(CN(C(=O)C(O)CF)CC)C)cnn(C)c1-c1ccc(C)cc1 c1(CN2CCC(NC(C3(CC#C)CCOC3)=O)C2)ccc(S(=O)(=O)N)cc1.C1CC1 C1(CCNC(c2n(C(C)C)nnc2)=O)CN(C(=O)CC2(C)CCCCC2)CCO1 CC(F)(F)C(C)(C)CC(=O)NCC1CCN(C(C2COCC2(C)C)=O)C1 N1(C(C2(COC)CC2(F)F)=O)CCN(C(c2ccc(C(F)F)cc2Cl)=O)C(C)C1 C(N=c1[nH]c(=NCc2ccc(N)cn2)[nH]c2c1CCC2)C1CCN(C(C)C)C1 c1(C(N2CCCC(N(C)C(c3ccc(CO)o3)=O)C2)=O)cc(O)c(F)cc1N c1(C(=O)NCCC2CC(C(=O)NC(CC(=O)NC)C3CC3)C2)nccc(C)c1F c1(C(=O)NC(C)CCCNC(=O)Cc2nc[nH]n2)coc(C#N)c1 C1(C(=O)NC2CN(C(=O)NC)C2)CCC(F)(F)CN1 CCC(F)(F)CC(=O)NC(c1ccccc1)C(C)NC(c1cc(C)c(C)o1)=O Cc1cccc(OCCCN(CC(N(C(C(=O)NCC(C)C)=O)C)C2CC2)C)c1 c1(CC(=O)NC2(CC=C)CN(C(=O)C(C#N)C(C)C)C2)ccc2n[nH]cc2c1 C1(C(=O)NCCNC(C(CC)C)=O)Cc2cc(Br)ccc2O1 c1(N2Cc3n(cc(C(F)(F)F)n3)CC2)nccc(=NC2CC3(C2)CC3(F)F)[nH]1 C#Cc1cncc(C(N2CCCC(CNC(=O)CCCNC(N)=O)CC2)=O)c1 N1(C(c2n(CCC(=O)OCC)nnn2)CC)CCSC(C)(C)C1.c12csc(n1)CC2 C(C(CC)(CC)C(=O)OCCCO)NC(CCCCCNCC)=O N1(C(C2=CC(C)(CC)C2)=O)CCC2(CC1)CCN(C(c1coc(C(F)F)c1)=O)C2 C1(CC)CCN(C(c2c[nH][nH]c2=N)=O)C1C(=O)NC1CN(C(C)=O)C1 Cc1ccc2c(c1)C(C(=O)N1CC(NC(=O)CSCc3ccccn3)C1)C2 c1(-c2ccccc2)cncc(C(=O)NCC2(CNC(C3CCC(=O)N3)=O)CC2)c1 Cc1cccc(C2CC2C(=O)NCC(C)NC(c2ocnc2C2CC2)=O)c1Cl CC(C)(C(=O)NCCn1cc(CC(CO)C2CCC2)nn1)c1ccccc1 CCC(CCC(=O)N1CC(N(C)C)C(C)(C)C1)NC(c1c[nH]c(=NC)o1)=O CC1(C)CCC(=CC(N2CCN(C(c3n[nH]cc3Cl)=O)C(CC3CC3)C2)=O)CC1 CC(C)(C)C(CO)C(=O)NCCC1(C)CCN(C(c2cnc(Br)s2)=O)C1 N1(CCc2cn(CC(=O)NC3(C)CC(C)=C(C)CC3)nn2)CC2CC3CC2C1C3O C12(C(N(C)NCC34CC(NC(COCCC#C)=O)(C3)C4)=O)C3CC(CC13)C2(F)F C(=O)(CCCCC(C)(C)C)NCC(C1CCC1)NC(C1(CC)CCCCO1)=O C(CCC(=O)NC1(NCC(C(C)C)OC)CSC1)NC(=O)OC c1(C(=O)NCCCN(C(c2ccc(OCC(=C)C)cc2)=O)C)ncc(F)cc1C Cc1cnncc1C(=O)NCCN(C(=O)C(C)NC(C1CCOCC1)=O)C(C)C CC(C)(C)S(=O)(=O)CC(=O)NCC=CCN=c1[nH]nc(COC(F)F)s1 C1(C(C)NC(=O)CC2COCCO2)CN(C(=O)CC2SC(=N)NC2=O)CCO1 N1(C(c2cc(CC)sn2)=O)CC2(CC(C(=O)Nc3cccc4c3CCC4)CO2)C1 C=CC(C)(C)CCCNC(=O)NCCc1cccc(OC(F)(F)F)c1 C12(NC(CC3CN(C)CC3O)=O)CCC(CC1NC(=O)CN1CC3CC3C1)C2 N1(C(C2CC(OC)C2)=O)CC(N(C(=O)C(n2ccc(C3CC3)n2)C)C)C(O)C1.C1(C)CC1 O=C(O)C1c2ccsc2CN1C(=O)NCCC1CCC(c2ccccc2)CC1 CCCC(C)CN=c1[nH]c(N(CCC#N)C)nc2cc(C(F)(F)F)ccc12 c1(C(N2CCC(CC=C)(NC(=O)Cn3ncnn3)C2)=O)cccc2nc(C)[nH]c12 c1(C(C)NC(=O)NCC(O)CO)ccc(Cl)cc1C(F)(F)F.c12sc(nc1C)[nH]2 C1(C(=O)OC)(CNC(=O)NCCc2nccc(C#N)n2)CCCNS1(=O)=O S(=O)(=O)(c1ccc(F)c(F)c1F)NC1CCCC(SCC)C1 c1(C(=O)NCCC(CNC(C2(C)CC(F)C2)=O)OC)ccn2ccnc2c1 N1(C(=O)C=CC(F)(F)F)CCC2(CCCN2C(C2CCC([N+](=O)[O-])CC2)=O)C1 N1(C(COC(C)C)=O)CCCCCCC1C(=O)NCC1CCOC(C)(C)C1 S(=O)(=O)(c1ccc(NCc2ccc(F)cc2)nc1)NC(c1ccncc1F)C c1(C(=O)NCCC(CCNC(C2C(OC)C2)=O)C)c[nH]c(=N)nc1C C1(CC)CN(C(c2[nH]cnc2C)=O)CCC1NC(C1(NC(C)=O)CCC1)=O C(=O)(CCCC(F)(F)F)N1C2C(NC(C(N3CCN(C)CC3)C)=O)CC(C2)C1 c1c[nH]c2cc(F)ccc12.C1(c2n(C(CC)(C)C)nnn2)(N)CCC1C1CC1 Cn1ncc(C(N2CCC(CC(=O)NCC3(CF)CCC3)C2)=O)c1Cl C=C1CC2(C1)CC(C(N1CCN(C(c3c[nH]c(=NC)s3)=O)CC1C1CC1)=O)C2 c1(CNC(CCn2c(=O)cc(C)nc2)=O)nc2c(s1)CN(C(=O)CC1CC1)CC2 C(=O)(C(O)CC(F)(F)F)NC(C(N1CC(N(C)C)C1)=O)C1CCC1 CC1SCCCC1C(=O)NC(c1ccccc1)C(=O)NC1CON(CC)C1=O.CC=O c1(CN(C(CCC)=O)CCNC(=O)CCc2cnco2)cccc(OC)c1 c1(NC(=O)NNCC2CC=CCC2)ncc(Br)cc1CO c1(CC(N2C(CNC(CC3C(C)(C)C3)=O)CC3CC32)=O)cn2ccsc2n1 N1(C(C(c2cccc(Cl)c2)CC)=O)CCN(C(C2(c3ccno3)CC2)=O)CC(O)C1 c1(C(C2(c3ccccc3F)CC2)=O)ccc(-c2ccccn2)nc1O N1(C(c2ccc(SC)o2)=O)CC(NC(=O)C(c2cncn2C)=O)C2(CC2)C1 N1(C(C(C)(C)SC)=O)CCC2CCN(C(C3CCN(C(C)C)C(=O)C3)=O)CC2C1 N1(N2CC(c3c(C)con3)C2)CCCC(n2cc(SC(=N)O)nn2)CC1 C12(NC(c3occc3F)=O)CCOCC1CN(C(c1scnc1Cl)=O)C2 N1(C(COCC=C)=O)CCC2CC2(C(=O)NC2CN(C3COC3)C2)CC1 c1(C(=O)NCC2C(NC(C(C3CCC3)OC)=O)C2)ccc(OCCF)cc1F c1(C(N(CCN(C(CSCCCC)=O)C)C)=O)cc(C2CC2)ccn1 C1(CCCNCCCCCN)(CO)CCOCC1 n1(CC(=O)NC(CNC(C2(OC)CCCC2)=O)C)nc(O)ccc1=O CC(C)C(CC(=O)N1OC2C=CC1CC2)NC(=O)CC(C)C(C)(C)C C1(C(=O)NCC2(NC(c3ccc(OC)c(C)c3)=O)CC2)Cc2nn[nH]c2C(C)C1 C(CCCCCCCO)=CC=O.CC(C)C(O)CN(C(=O)C(=O)N(C)C)CCN(C)C C(CCc1ccccc1)(C(C)NC(c1cnc(=N)[nH]c1)=O)NC(C(C)SC)=O c1(CNC(CCc2cnc(C)s2)=O)nc(C(=O)N(C)CC2CC2)c(C)o1 C(=O)(C(C)(C)N=[N+]=[N-])NC(CCC)C(=O)NC1C(C)CCC1C c1(OC)cccc(S(=O)CC(=O)NCCN(C)C(c2cc(C)ccc2F)=O)c1 c1(C(=O)NC2C(CNC(c3cc(C)n(C(C)C)c3)=O)COC2)ccn(C)c(=O)c1 c1(CC(=O)N(C)CC2(O)CCN(C(=O)Cc3cnn(C)c3)C2)cccc(F)c1F C(=O)(CC(C)C(=O)N(CCC(C(C)C)NC(=O)CC(O)C1CCCC1)C)OC c1(C(=O)OC)cc(CC(=O)NCC(C)NC(C2COCCO2)=O)cs1 C1(N2CCOCC2)(CC(=O)NCC(C2CCOC2)OCC)CCOCC1 c1(C(=O)NC(C)CCNC(=O)CC2(CO)CC2)nccnc1N N1(C(CNC(C(CC)CC)=O)=O)CCC(NC(=O)CC2CCCOC2)C(O)C1 C12(C(N(C(CCO)C(F)F)C)=O)CC1CCN2C(=O)CN1CCC(F)CC1 C12(NC(c3cnn(CC(C)C)c3Cl)=O)CCCCC1CN(C(=O)CC1CCC1)C2 C1(C(=O)NCc2cn[nH]c2)CN(C(=O)C=CC2CCCCC2)CCO1 N1(C(c2c(C)occ2)=O)CCC(C)(NC(c2cc[nH]n2)=O)C1 C1(CNC(CNC(=O)OCC)=O)CN(C(c2c[nH]nc2Br)=O)CCO1 C12(CN(CC(C)(C)C)C(Cc3cc(C)nn3C)=O)CC(C1)C(NC(=O)C)CO2 c1(C(=O)N(CCCCCO)CC2N(S(C)(=O)=O)C3C(C2)C3)cc(I)cnc1Cl C(C1=COc2ccccc2O1)(c1nnnn1-c1cccc(Cl)c1)CC(F)(F)Cl Cc1ccc(C(N2CC3CC3(CNC(=O)CC3CCC(=O)NC3)C2)=O)c(N)n1 c1(N2CC3CN(C(c4c(OC)ccc(Br)c4)=O)CC32)ncnc2[nH]c(C)nc12 c1(C(=O)NC2CCN(C(c3c(OC)n(C)nn3)=O)CC2O)cc2sc(Cl)cc2s1 C(=O)(CS(=O)(=O)C1CCCC1)N1C2CCN(C(C=C(COC)C)=O)CC2C1 CCCCC(F)C(=O)N1CCOC(Cc2cn(C3CCCC3O)nn2)C1 C(C(O)CN=c1cc(C)[nH]cc1C(=O)N1CC(O)CO1)OCC C(C(N=[N+]=[N-])C(=O)NC(C(=O)N(CC(O)CO)C)C1CC1)OCC C1(NC(C(CCSC)NC(=O)CC2CSC2)=O)CCCCCC1(C)C C=CCN=C(NCc1cccc(CN2CCCCCC2)c1)N1CCC(C)C1C C1(N(C(C(C)SC)=O)CC2CC2)CCN(C(=O)CNC(=O)CC)C1 c1(CC(=O)NC(c2ccccc2)CNC(CC2(C=C)CC2)=O)ccc(F)c(F)c1 c1(CC)c(C(N2CCC2CNC(=O)C2=NOC(CN)C2)=O)[nH]c(C)c1C(=O)OC c1(C(=O)NCC2(CNC(C3C(C)(C)CC3)=O)CCCC2)c(Cl)ccc(F)c1F CC1CC2(C(N3CCCC3CN(C(=O)Cn3cccn3)C)=O)CC12 C1(CCn2cc(CCCSC)nn2)CCCN(C(C(C)C2CC2)=O)CC1 CC(C)C(F)(F)CCNC(=O)CCc1cn(C2CCOC2C(C)C)nn1 C1(C(=O)Nc2nc3ccccc3[nH]2)CC12CCN(C(=O)Cc1nc[nH]n1)CC2 CC(C)C(C)(CN=c1nc[nH]s1)NC(=O)CCOC1CC1 C1(C)(C(N(CCN(C(C2CCC(OCCC)CC2)=O)C)C)=O)CCCCCCC1 c1(C(=O)NC2C3CCN(C(CC(=C=C)C)=O)C32)ccc(S(C)(=O)=O)cc1 C1(C(=O)NC2(CC#C)CCCC2)CCC(C)N1C(C1CC2(CC2)C1)=O C1(CC(=O)NCCOCC#C)C2CCC(C2)N1C(=O)C(C)(C)n1cccn1 N1(C(c2c(CC)[nH]nc2Cl)=O)CC2(CCCC2Nc2nc(Cl)nc(C)c2Cl)C1 n1(CCCC)cc(C(=O)NCC2CC(NC(C3(N(C)C)CC3)=O)C2)nn1 c1(C(=O)NCC2C(C)CN(C(=O)C(F)=CC3CC3)C2)ccc(N)c(Cl)n1 C12(C(=O)NCc3cccc(C)n3)CC(C)(CN1C(=O)C(C)SC(C)C)C2 N1(C(C2N(C(C3(C)CC3(F)F)=O)C3(CC2)CC3)=O)CCn2ncc(O)c2C1 C(=O)(C1=CCC(F)(F)CC1)N(CCCNC(c1cc(C)c(Br)o1)=O)C c1(NC2C(NC(C(CC=C)C)=O)CCCC2)c(C#N)cnc2c(F)cc(F)cc12 C1(C(=O)NCC2(CCC)CC2)CC=CCC1NC(c1cc(C)c(C)[nH]1)=O N1(C(c2c(C)nc[nH]2)=O)CC2CCN(C(=O)C(C)(O)C3CC3)CC2C1 Cc1cc(C)c(NC(N2CC(NC(C3(O)CC3)=O)C(C)C2)=O)c(C)c1 c1(CNC(C2C(C)(C(C)C)C2)=O)cc(C(=O)NCC2(C)CCOCC2)n(C)n1 Cc1cc(N2CCCN(Cc3cccs3)CC2)nc(=NCCC(=O)N(C)C)[nH]1 c1(C(=O)NCC2N(C(CN(C(C)C)C)=O)CCCCC2)n[nH]c2ccc(O)cc12 c1(NCCC(C(=O)OC)(C)C)cccc2c1CNC2=O C1(NC(c2cnc(Br)s2)=O)CCCN(C(C2CCCC23CC3)=O)C1 C=C=CC(C)C(=O)NC1C=CCC(C(N2CCOCC2C2(C)CC2)=O)C1 c1(C(=O)NC(C(=O)NCCCNC(C)=O)C2CCCO2)cncc(O)c1 c1(OC(C)C(=O)NCC2(CNC(=O)CC3CCC(=O)N3)CC2)ccccn1 C1(CNC(C2(OC)CC2)=O)CCCCC1NC(=O)C(C)(C)CN(C)C n1(CC(=O)N(CC(C)CNC(=O)CSc2cn[nH]c2)C)cc(S(C)(=O)=O)cn1 C1(CNC(=O)CC2CSCCS2)CCN(C(C2CC=CCO2)=O)C12CC2 N1(C(c2cc(CC)on2)=O)CC(CNC(c2nc(C)sc2C)=O)CC12CCC2 C1(C(=O)NC2CC(F)(CNC(c3ncncc3Cl)=O)C2)CCc2nc[nH]c2C1 c1(C(=O)NCC(CO)NC(c2cn(C(C)(C)C)nc2)=O)cnc2ccsc2c1 Cc1cc(C(=O)NCCC2CCCCN2C(c2cc(CO)c(C)o2)=O)cc(F)c1 C#CC(C(C)OC)NC(c1coc(CNC(C2CCC(C(N)=O)O2)=O)n1)=O C(=O)(C(CC(F)F)N(C)C(c1cncc(C#N)c1)=O)N(CCCCCC=C)C C1(OC)CN(C(c2ccc(SC)cc2)=O)CC1NC(c1csc(=N)[nH]1)=O C#Cc1cnc(C(=O)NCC(C2CCC2)NC(=O)C(C2(O)CCCC2)F)c(C)c1 C(=O)(CCS(N)(=O)=O)N1CCCC(CNC(CCC2OCC(C)(C)C2)=O)C1 n1(CC(=O)NCCC(C)NC(c2c(NC)nccc2)=O)nc(Cl)ccc1=O c1(C(N(c2cccc(C(=O)Nc3ncc(Br)cc3Cl)c2)C)=O)ccc(F)c(Cl)n1 c1(CN)cccc2sc(=O)n(C)c12.c1(OCOC(C)C)cccc(C)n1 Cc1ccc(CC(=O)NCC2(C(C)NC(c3cc(C)c(C)o3)=O)CC2)cc1F C=CCC(C)(CC)C(=O)NCC(C)(O)CNC(=O)CC1(OCC)CCC1 C(CN=c1nc2scnc2c(N2CCC3(CCC3)C2)[nH]1)(C1CCCO1)OC c1(C(N2CCCC(NC(CC3(C#N)CC3)=O)CC2)=O)[nH]c2ccccc2c1C1CC1 Cc1cccc(C(N2CCC(CCCNC(=O)C=Cc3cncs3)CC2)=O)n1 n1(CC(=O)NCCC(C)NC(C(C2CC2)SC)=O)cc(C)c2ccccc12 c1(C(N(CCN(C(C(CC)CC)=O)C)C)=O)ccc(C(C)C)nc1C c1(-c2c(C)csc2)cncc2sc(C(=O)Nc3nccc(C)c3F)cc12 C1(NC(CSCCOC)=O)C2CCN(C(C3(C#N)CCCOC3)=O)CC12 N1(C(CC(C)c2ccncc2)=O)CCN(C(c2cnn(C(F)F)c2)=O)CC(O)C1 N1(C(CCCC(=C)C)=O)CCC2CCN(C(c3cnc(C)nc3C)=O)CC2C1 N1(C(c2c(CC)n(C)nc2)=O)CCN(C(c2coc(C(F)F)n2)=O)CC1C(C)C N1(C(C=CC(C)C)=O)CC(C(=O)Nc2ccc(C3CCN(C)CC3)cc2)C(O)C1 C1(C(=O)NC(C#C)C)CC=CCN1C(c1ccc(F)s1)=O N1(C(C(COC)(F)F)=O)CCCCC(C(N2CCC(c3cc[nH]n3)C2)=O)C1 c1(CC(=O)N(CCNC(c2c(OCC)scc2)=O)C)cn2c(C)csc2n1 CCCC(C(O)C(=O)N1CCCC(F)(CO)C1)NC(c1ccc(CO)nc1)=O CCC(C(=O)N1CCC(N(C(=O)CC(=O)OC(C)C)CCC)C1)c1ccccc1 C1(NC(=O)Nc2cnn(C)c2CO)CCS(=O)(=O)CC1 CC1CCCCCCN1C(=O)CC1CC(C)N(C(c2cc(Cl)cs2)=O)C1 N1(C(C(C(C)C)n2cnnc2)=O)CCCC(NC(C2(C)CC2)=O)CC1 c1(C(N(CC(N2CC(O)(CC(C)C)C2)=O)CC(N)=O)=O)cccn2nccc12 C1(C(=O)NC2(COC)CCN(C(=O)Cc3nc(C)c(C)s3)C2)CCC(C)(C)OC1 c1(C(N2C(CNC(C3CN(C4COC4)C3)=O)CC(OC)C2)=O)nnc(O)cc1O Nc1snnc1C(=O)NCc1cn(CC(N2CCCC2C(=O)O)=O)nn1 C1(c2nc(C)nn2-c2ccc(C3CC3)cc2)Cc2cccc(C)c2O1 C1(NC(=O)C(O)C(F)F)CN(C(=O)CCc2cc(Cl)ccc2Cl)C2(CCC2)C1 c1(C(=O)OC)ccc(C(=O)NC2CCN(C(=O)CCN3CCCCC3)C2)s1 C1(NC(c2c(OC)ncc(C(N)=O)c2)=O)CCCC2(C1)CC2(F)F C(=O)(C1CCc2scnc21)NC1CC(NC(C(C(C)C)C(C)C)=O)C(O)C1 CC(C)CC(C(=O)N(C1CCCN(C(C2CCCOC2)=O)C1)C)N(C)C c1(CNC(C2C(C)(COC)C2)=O)cnn(C)c1C(N1CC(O)(C(C)(C)C#N)C1)=O N1(C(C(C)OCCC=C)=O)CCC(CNC(C2CCC(C(N)=O)CC2)=O)C(C)C1 C1(C(N(C(c2ccccc2)CNC(CC=CCC)=O)C)=O)CCCCNC1=O C1(CNC(C2CCN(C(C(CCC)NC(C)=O)=O)C2C)=O)CC(=O)NC(C)C1 N1(C(CCCCC#C)=O)CCC(NC(c2nccc(N)c2Cl)=O)C(C)(C)C1 CC1CN(C(=O)C=CCF)CC2(CCN(C(C3CCCC(=O)N3C)=O)C2)O1 CCC(COC)C(=O)NC(CCN(C)C(c1ccccc1SC(F)F)=O)C(C)C c1(N(CC(=O)NCCCC(C)NC(CCCN(C(C)=O)C)=O)C)ccc(Cl)nn1 c1(OC)nn(C)cc1C(=O)NC12CC1CN(C(=O)CC1CCC(=O)N1C)C2 C1(CC=CC)CCCN(C(=O)C(C)(C)CNC(=O)COC2CCOC2)C1 CC1CN(Cc2ncn(C)n2)CCC1NC(C1CN2CCC1CC2)=O C(=O)(CC1=CCCCC1)N1CCC(O)(CCNC(C(C)N2CCC2)=O)C1 Cc1cc(C(=O)NC2CC2CNC(c2cnn(C)c2CC(C)C)=O)c(C)n1C C(C(CC(=O)N1CCC2(CC1)CC2NC(C12CCN(CC1)CC2)=O)C(F)F)OC C(=O)(C1=CCOC1)NCCN(CCCN(C)C)C(=O)CNc1ncccn1 c1(NC(=O)NC(c2nc(CC(F)(F)F)cs2)C)csc(Cl)c1 C1(S(C)(=O)=O)(C(=O)NCCC2(O)CN(C(C=C(C)CN3CCCC3)=O)C2)CCC1 CCCCCCN(C)C(C1CN(C(=O)COC(C2CC(C)=NO2)=O)C1)C1CCCO1 N1(C(C(CCCCC)C)=O)CC2CC(NC(=O)C(C)C)CC(C2)C1 N1(C(C2CCC(CC)O2)=O)CCCC12CCN(C(C1CC3(C1)CC(O)C3)=O)C2 N1(C(C2C(C)CCS2)=O)CCC2(C1)CN(C(=O)CNC)C2.c1(O)cc(F)cc(Cl)c1 CC(C)(CN1CCOCC1)C(=O)NCCCC(CO)CNC(=O)CCC1CCC1 c1(C(N2C(C(CNC(C3(CC)CCCC3)=O)(C)C)CCC2)=O)csc2nccn12 CCC(CC(=O)NCC1(C(=O)N(CCCN(C)C)CC)CC12CCC2)C(C)C C1(C(=O)NCC(=O)NC(c2cn(Cc3onc(CC)n3)nn2)C)CN(C)CCO1 N1(C(CC(COC)C)=O)CCCC(F)(CNC(c2csnn2)=O)C1 c1(CC(=O)NCC2C(NC(CNC(C(CC)CC)=O)=O)C2)cc2ccccc2s1 CC1CN(C(C23CC(F)(C2)C3)=O)CCC1NC(=O)Cc1ccc(F)cn1 C1(NC(COCCCCCC)=O)CCN(C(=O)Cc2cnn(C)c2)C12CCC2 c1(CCC)ccc(CC(N2CC(N(C)C(c3onc(C)c3C)=O)C(F)C2)=O)cc1 N1(CCOC)CC(NC(N2CCOC(CC(=O)OC(C)(C)C)C2)=O)CC1=O C1(OC)CN(C(C2CN(C)C(=O)N2)=O)CC1NC(=O)CCc1cnc(O)[nH]1 CC1CN(C(=O)C(C)C2CCCC2)CCCN1C(c1cccc(C(F)(F)F)c1)=O C12(NC(C(CC)N(CC)CC)=O)CCC(CN(C(c3n[nH]c(C)c3C)=O)C1)C2 C1(=O)C(C(C)C)CN1.c1(C(N(CC(COC)(F)F)C)=O)cccnc1OC C12(C(=O)NC3COCCN(C(CNC(CC(C)C)=O)=O)C3)CC1COC21CCC1 c1(C(N(CC(=O)Nc2csnn2)CC)=O)csc(CC(C)C)n1 N1(C(C2=CC(C)(CC)C2)=O)CC(NC(=O)CCOC2CCCC2)C2CCCC12 c1(CN2CC(C)N(C(c3ccc(Cl)cc3)=O)CC2)ccc2cncn2c1 N1(C(CC(C)CNC(C2(COC)CC2)=O)=O)CC(O)C2(CCCC2)C1 C1(CC=C)(NC(=O)C(c2cccc(Br)n2)C)CCN(C(=O)C(C)(C)C#N)C1 N1(C(c2nc(CC)oc2C)=O)C2CCC1C(NC(=O)CN1CC(C)(C)C1)C2 Fc1ccc(F)c(C(N2CCCC2)CNC(=O)NCCc2csnn2)c1Br C#CC1CCCC(NC(C2(NC(=O)C(C)CC3CC3)CC2)=O)C1 c1(NC(=O)CC2CN(Cc3nccc(O)n3)CCO2)cnc2c(Br)cc(Cl)cn12 c1(C(=O)NC2CC(C(C(=O)N(CCCCCCC)C)F)C2)cc(F)cnc1O c1(SCC(=O)NCCN(CCOC)C(c2nnc(S)n2C)=O)ccc(Cl)cc1 C1(CC)CN(C(C2(SC)CCC2)=O)CCN1C(=O)C(CC1CCC1)OC C1(CC(=O)NCC2CN(C(=O)Cc3ccc(F)cc3F)C2)COCC2(CCC2)O1 CCCC(C)(CC)C(=O)Nc1cccc(NC(=O)C(F)CC)c1 C(C(C)(F)C(C)C)NC(C1(C(=O)O)CCC1)C.c12cn(nn1)CCNC2=O C(C)(C)(CC(=O)NC1CCCCN1C(=O)COCCOCCO)SC N1(C(C(n2cc(CCC3CCC3)nn2)C)=O)CCC(C2CCNCC2)C1 CC(C)(C)CCCC(=O)N1CC2(CC2)CC1CNC(c1ccc(F)c(C(F)F)c1)=O C1(CC#C)(C(=O)NCCC2(CNC(=O)CCCc3nccs3)CC2)CCCCO1 c1(C(N2CC(N(C(C=CC(=O)OCC)=O)C)C(F)C2)=O)cc(Cl)c(F)cc1F C1(C2CCCN(c3ncnc(Cl)c3Br)C2)(NC(C2CC3CCC(C2)C3)=O)CC1 N1(C(C=C(C)CNC(=O)CN2CCCNC2=O)=O)CCOCC(O)C1 N1(C(C2CC(=C)C2)=O)CCN(C)CC1CNC(=O)Cc1ccc(Cl)c(Br)c1 N1(C(Cn2nc(C)c(Cl)c2)=O)CCC(NC(c2ncc(F)cc2F)=O)C(O)C1 C1(NC(c2c(OC)cccc2)=O)CN(C(=O)C=Cc2cncn2C)CC12CCC2 C1(C(=O)NC2CC3C(NC(C4(CC=C)CC=CC4)=O)C3C2)CCC(F)(F)CC1 C(=O)(C(C)(CC(=O)NNC(=O)NCC)CC)OC1C(c2cn(CC)nc2)OCC1 C1(O)(C(=O)O)CCN(c2cncc(C(=O)NCCS(=O)(=O)CC3CC3)n2)CC1 CC1(C)CC(NC(C2(F)CC=CCC2)=O)CN1C(=O)Cc1cc(C2CC2)no1 n1(CC(N2CC(OCC)(CNC(=O)CCCN3CCOC3=O)C2)=O)cccnc1=O CCCC1C(O)C(=O)N1.C(C)(C(C)SC)NC(C1CC1C(C)(F)F)=O Cc1cc(C(=O)NCC2CC(C)(C)CN2C(=O)CNc2cccnc2)cc(C)n1 c1(NC(=O)NC(C)CCCc2ccccc2)cc(O)nn1C C1(SC)CN(C(=O)CC2(C)CCCCC2)CC1NC(=O)C(=C1CCCCC1)F C1(NC(C2CCN(C(C)C)CC2)=O)CCCN(C(=O)CC2(C)CC2(F)Cl)C1C c1(C(=O)NCC(CNC(C(CC)SC)=O)F)cccc2c1OCCN2C C1(C(=O)NCc2cn(CCC)nn2)CC(C)CN(C(C2CCC(C)(C)CC2)=O)C1 CC(CC(=O)N(CCCNC(C1CC(=C2CCC2)C1)=O)C1CC1)C1CCCCC1 C1(NC(=O)Cc2cc[nH]c2)CCC(NC(c2cnc(C(F)(F)F)s2)=O)CC1 N1(C(CC)C)CC(C(=O)NCC2CCC(NC(C3CC3C3CC3)=O)CC2)CC1=O N1(C(CN(CC)CC)=O)CC2CCCC1(CNC(c1cnc(Cl)[nH]1)=O)C2 C1(C)(CNC(CCC(=O)NCCC)=O)CC(F)(F)CN1C(=O)CCCCC1CC1 C1(NC(C=C(C)C(C)C)=O)CCN(C(c2ccccc2-n2cccc2)=O)CC1F C1(O)(C(N(CC)Cc2nc[nH]n2)=O)CN(C(=O)COCCOC)C1 N1(C(C2(C)C=CCN2C(=O)CN2CC3CC3C2)=O)CCC2CCC(C1)S2 C(=O)(CCC(C)NC(=O)Cn1cc(C#N)cn1)N(C(CSC)C)C C1(CO)CN(N(C)C(C2(C(=O)NC(C)(C)C)CC2)=O)CCO1 N1(c2snc(C(C)C)n2)CCC(NC(=O)CCCNC(N)=O)C(C)C1 N1(C(c2n(C)nc(C3CC3)c2)=O)CCC2CCNCC2C1 C1(CC)(CO)CCCN1C(=O)C(CN(C)C)NC(=O)CCCn1cncn1 c1(OC)c(C)cc(C(N2CCN(C(C3(NC(C)=O)CCCC3)=O)C(C)C2)=O)cc1Cl CC(C)(C#CC(=O)N1CCC1CC1CCCC1)CNC(=O)C(C)(C)C1CCOC1 CC(C(=O)NC(CNC(c1ccn(C2CCCCC2)n1)=O)C(C)(C)C)C(C)(C)O c1(C(=O)NC(C)CC2CN(C(=O)Cn3cnnc3)C2)cc2n(c1)CCSC2 C1(NC(CN2CC(C)(C)C2)=O)CC12CCN(C(c1ccoc1C(F)(F)F)=O)CC2 c1(C(C)C)ncc(C(N2CCC(CCNC(=O)C(C)N3CCC3)C2)=O)n1C O=C(CS(=O)(=O)C12CC(C1)C2)NC1CN(C(=O)CO)CC1O C1(O)(CNC(c2ccc(-n3cccn3)nc2)=O)CCN(Cc2c[nH]ccc2=N)C1 CC(C)(C)CCCCCC(=O)N1CCC(NC(c2cc3sccc3[nH]2)=O)C1 CC(C)(C)C(C(=O)N1CC(F)(CF)C1)NC(c1sccc1Cl)=O c1(C(N2C(CN(C)C(C3(CO)CC3(F)F)=O)CCC2)=O)cccc(F)c1N C(=O)(C(CC1CCCO1)C(F)(F)F)N(CCCNC(C1(C)CC1)=O)C1CC1 Cc1cc(F)ccc1C(CNC(=O)CC1CC1)NC(=O)CC1C=CS(=O)(=O)C1 N1(C(c2cnc(S)n2C2CC2)=O)CC2CC(Nc3cc(C(F)F)ncn3)C2C1 N1(C(c2c(CC)cnn2C)=O)CCC(NC(=O)C(CC)(CC)CO)C(C)(C)C1 c1(N2CCC(CNC(C(CC)N(C)C)=O)C2)nc(C)ncc1C(C)=O C(=O)(CC(CC)C(F)F)N1C(C(N(CCCC=C)CC)=O)CCC1C1CC1 c1(N(C(C)C)C(C2CC3(C2)CC3(F)F)=O)cc(F)cc([N+](=O)[O-])c1 C1(C(=O)NCc2nc[nH]n2)(OC)CCN(C(=O)CC2CCCC(C)C2)C1 c1(C(=O)NC2C(C)(C)N(C(=O)C3=CCCOC3)CC2)cc(F)cc([N+](=O)[O-])c1 c1(NCc2ccc(C(N(c3cc(COC)ccn3)CC)=O)[nH]2)ncc(F)cc1Br C=C(C)CC(C(=O)NCc1ccc(C#N)cn1)NC(c1cc(Cl)cn1C)=O c1(CC)[nH]c(=N)sc1C(N1CCC(OCC(=O)Nc2cc(C)cnn2)C1)=O c1(C(=O)OC)c(NC(=O)COc2ccc(NCCO)cc2)sc2c1CCCC2 N(C(=S)NNC(=O)c1cccc2c1CN2)C(C=C)C.c1(O)ccccc1.OCC N1(C(C2(O)CCSC2)=O)CC2(CO)CC2(CNc2nccc(CO)n2)C1 c1(C(N2C(CO)CC(NC(C(CC)COC)=O)C2)=O)snc2ccccc12 CC#CCC(C)N=c1[nH]c(=NCc2cccc(F)c2)c2cccc(F)c2[nH]1 c1(C(N2CCN(C(CC(C)SC)=O)CC(C)(F)C2)=O)ccc2c(c1)CCNC2=O c1(NC(C2(C(N)=O)CCC2)=O)cccc(NC(=O)C(CC2CC2)N2CCCCC2)c1 Cc1cc(N2CC(C)OCC(C)(C)C2)ncc1S(=O)(=O)NC1CCC([N+](=O)[O-])CC1 C12(C(=O)NCC(C)C(C)(F)F)CCC(NC(C3CCCN3C3CC3)=O)(CC1)C2 N1(C(C(C)C)=O)CCCC(C(C)C(N2CCN(C(=O)C=CC(C)(C)C)CC2)=O)C1 c1(C(=O)NC2CCCC(N(C(C3=C(C)CCC3)=O)C)C2)ccnc2ccccc12 N(C(=NCC1CCC1)NC(C)CCc1ccc(F)cc1)C(COCC)C1CCC1 C1(CCN(C(C2(C(C)NC(c3c(CC)c[nH]n3)=O)CC2)=O)COC)CCC(C)(C)O1 CC(C)CC(C)(C)C(=O)NC1CCCC1CNC(c1snnc1C1CC1)=O c1(C(=O)NC(CC)CN(C(=O)Cc2cnnn2C)C)ccc([N+](=O)[O-])cc1Cl C=CC(C)(C)CC(=O)N1CCC(C(=O)NCCc2cnn(C)c2)C1C(C)C CC(CC(=O)NC(CCOCCO)C(=O)NCC1=CCCCC1)C(F)F c1(C(=O)NCC(C)NC(=O)Cc2ccn(CC(=O)O)n2)cn2cccnc2n1 C(C(C(C)(C)C)NC(C)=O)NC(COCCC=C)=O C(CC1CC1)(CC(=O)NCC1CC=CCC1)NC(C(C)O)=O C1(N(C(C2C(C)OCC2)=O)C)CN(C(C2(c3ccsc3)CC2)=O)CC1O c1(COC)cc(=NCC2CN(C(c3cc4c([nH]3)CCC4)=O)CCC2C)[nH]cn1 c1(CNC(c2n(CC)ccn2)=O)ccccc1CNC(=O)C(C)(C1(C)CC1)OC N1(C(Cn2ncc(CC)c2)=O)CCC(NC(c2cccc(OC)c2C)=O)C(C)C1 C1(NC(c2c(C)n(C3CCC3)nc2)=O)C2CCN(C(=O)C(F)(F)C3CC3)CCC12 CC1CCN(C(=O)Cn2nccn2)CCN1C(c1ccc(C#N)cc1)=O c1(CC)cc(C)c(OCc2nnc(N3C(CO)CCC3)n2CC2OCC2(C)C)[nH]1 C(N=c1[nH]nc(C2CC2)s1)C1CN(C(C(C)c2ccco2)=O)C1 Cn1cnnc1C(=O)NCC1CC1CNC(c1cc(-c2cccnc2)no1)=O C1(NC(c2cncc(Cl)c2Cl)=O)CC2CC(C1)N(C(c1ccc(Cl)cc1F)=O)C2 CC1=C(C(=O)N2CC(C)N(C(=O)C(c3cncnc3)C)CC2C)C(C)(C)CCC1 CCC(CO)(C(=O)N(CC(C)C)C1CC1)OCC(=O)Nc1ccc(OC)c(O)c1 CN1CC2CN(C(=O)CC(C(F)(F)F)NC(=O)C(Cl)Cl)CC2(C)C1 N1(C(CCc2n(C)ncc2)=O)C2CCC(C2)C1C(N1CCC(C(C)(C)O)C1)=O c1(C(N(CC(C)NC(=O)CCCNC(N)=O)C)=O)csc(-c2ccccn2)n1 N1(C(C)=O)CCCCC1C(=O)N(C)CC1COCCN1C(=O)CC1(C#N)CCC1 C12(C(=O)NC3(N(C)Cc4c(C)noc4Cl)CCCC3)CCCCC(=O)N1CCC2.CN n1(C(CC)CC)ccc(C(=O)NC2CC(NC=O)C2)n1.C1(CC(=O)N)OCCO1 N1(C(c2cc(C)sn2)=O)CC2CCCC1C2CNC(=O)CN1CCC(=O)NC1=O c1(NC2C3N(C(C4CCC(N=[N+]=[N-])C4)=O)CC(CC3)C2)ncc2c(n1)CCOC2 C1(CC=C)(NC(C2CC2(C(=O)OC)C(C)C)=O)CN(C(c2nn[nH]c2Cl)=O)C1 C=CCCC(C(=O)N1CCOCC1C(C)O)NC(c1cc(NC)no1)=O N1(C(C(CC)CC)=O)CCN(C(C2CC(C)(O)C2)=O)CC1c1ccc(F)cc1 C1(NC(C2(OC)CC2)=O)CN(C(c2cnc3cc(C)[nH]c3c2)=O)C2(CCOCC2)C1 C1(C2C(NC(C(C)C#N)=O)CCO2)CCN(C(=O)CCCc2ccsc2)CC1 C1(NC(C(C=C)O)=O)Cc2ccccc2C1NC(c1cnn(C(C)(C)C)c1N)=O N1(C(c2n(CC#C)ccc2)=O)CC2CC1(CNC(c1cc(SC)c(C)o1)=O)C2 Cc1nc(-c2ccccc2)oc1C(=O)NC(C)CNC(=O)C(C(C)O)NC(N)=O c1(N2CC(CC(C)NC(C3(C(F)(F)F)CC3)=O)C2)ncnc2c1nnn2C(C)C N1(c2nc(OC)nc(C)c2)CC(CNC(=O)C(C)C2CCOC2)OC(C)(C)C1 N1(C(CCCNC(=O)OC)=O)C2CCC(C(=O)N(CC(C)O)CCO)C1CC2 CN(C[Si](C)(C)C)C(=O)C(=O)NC1CC(C(=O)NCC(F)F)C1(C)C Cc1cc(C(=O)NCC2CN(C(=O)C(C)(C)CF)C2)oc1C C(=O)(C#CC1(C)CCCO1)N.C(CCCC(=O)C(CC1CCCC(N)C1)=O)OCC CC1(C)CN(C(=O)Cc2cnccn2)CC1NC(C1CC(=C2CC2)C1)=O C(=O)(C(F)CC(C)(C)NC(=O)CC1CCCC(=O)N1)NC(CC)C(N)=O CS(=O)(=O)CCCC(=O)N1CCC2CN(C(C3CCCC34OCCO4)=O)C2C1 c1(C(N2CCC(O)(CCNC(c3cnc(OCC)s3)=O)C2)=O)ccc(Cl)c(F)c1 C(C1CCN(C(=O)C2=CCSC2)CC1)=CC(N1CC=CC(O)C1)=O n1(CC(=O)NCC(C)(C2CCC2)NC(C(C)NC(C)=O)=O)cc(CN(C)C)nn1 C1(CC=C)(C(N2CCC(CN(C)C)C2)=O)CCCN1C(c1ncn(C)c1C)=O C12(C(N3CC(C)(NC(c4cc(C)sn4)=O)C3)=O)CCCC1C2(F)F N1(C(CCN(C(=O)C2=CCCC2)C2CC2)=O)Cc2cncnc2C1 c1(N(C(c2c(OC)nccc2)=O)CC2CCNC2)ncc2c(Br)cccc2n1 C(=O)(NNc1ccccn1)NC1(NCc2nc(C)sc2)CCC(C)(C)CC1 C1(=O)C(C(=O)OC(C)(C)C)NC(=O)C2CC2CN1.n1(C(CC)CC)ccnc1CC C(CN=c1[nH]cnc2cccc([N+](=O)[O-])c12)(C(C)(C)C)NC(c1c(C)ocn1)=O C(=O)(C(C(C)(C)O)NC(C1C2C3CCC(C3)C12)=O)NC(CC#C)C(N)=O C1(C(N)=O)CN(C(c2sccc2Cl)=O)CCC1NC(=O)C1=CCOCC1 CC1CC(C(=O)NC2CC(N(C)C(c3cc(O)n(C)n3)=O)C2)CCS1 C1(C(=O)NC2(C)CN(C(c3coc(CS(C)(=O)=O)n3)=O)C2)CC2CCCCC2O1 c1(OC)cccc(F)c1C(=O)NCC12CCC(CN1C(=O)C1=CCCSC1)C2 C=CCC(CNC(=O)CC1CC2(C1)CN(C(c1conc1C)=O)C2)CC(C)C c1(C(N(CCC(=O)NCc2ccc(OCC)cn2)C2CC2)=O)ccc(F)c(O)c1 Cn1cc(-n2cc(C3(C)CNC(=O)C3)nn2)c(C(F)F)n1 c1(CC(=O)N(CC(C)OC(C)(C)C)C)ccc(N2CCOCC2)cc1 C(=O)(C1=CC(C)C1)N1CC(OC)(CNC(C2CC(=C3CC3)C2)=O)C1 C(=O)(C1=NOC2(CCOC2)C1)N1C(C(C)(C)OC)CN(C(=O)C2=CCCSC2)CC1 CC(C)CCCC(=O)NCCOCCN(C(=O)C(C)NC(C)(C)C)C C1(NC(=O)CCOCC2CC2)CN(C(C2(c3ccno3)CCC2)=O)CC1C1CC1 c1(C(N2CCC(C(=O)NCCC(=O)Nc3cccs3)C2)=O)cnc2n1CCOC2 C=CC1CN(C(=O)Cc2cnnn2C)CC1NC(=O)COC(c1nccn1C)C c1(C(c2n(C(CC)C)nnn2)NCc2conc2C(C)C)ncc(F)cc1C Cc1cc2sc(C(=O)NCCOCCNC(=O)CC3(C)OCCO3)cc2s1 N1(Cc2nn(CC)nc2C)CCOC(C)(CNC(=O)CCc2cnn(C)c2)C1 Cc1ccc(F)cc1C(N1CCCC(C(C)C(=O)N(CCO)CCO)C1)=O N1(C(C23CC(CN(C(C(C)SC(C)C)=O)C2)C3)=O)CCC2(CCOC2)C1 C1(C(N(C(CC)CC(=O)N2CC=CC2CF)C)=O)C2CCC(C2)C1C CC1OCCN(C(C23COC(C2)C(NC(c2cnn(C(F)F)c2)=O)C3)=O)C1CO c1(C(N(C2CCN(C(=O)C(F)(F)CC)C2)CCC)=O)c[nH]c2cccnc12 N#Cc1nc[nH]c1C(=O)NC1C=CCN(C(c2ncsc2-c2ccccn2)=O)C1 Cc1ncc(Cl)cc1C(=O)NCC1CN(CCN2CCNC2=O)CCCO1 c1(C(=O)NC2CN(C(c3c(C)nn[nH]3)=O)C3(C2)CCC3)cc2nc(F)ccc2o1 C1(C2CCN(C(=O)CC(CC)c3ccc(C)cc3)C2)(NC(C(C)=CC)=O)CC1 CC(O)C(F)(F)C(=O)N1CCC(CC(N)=O)(NC(=O)C=Cc2cccnc2)CC1 C1(NC(c2cc(OC)no2)=O)CC(F)CN(C(C2Cc3nccn3C2)=O)C1C C1(OCC)CN(C(=O)NCCC(C)(C)CN(C)C)CC12CC2 C(=O)(C1=CCCN(C(c2ccn(C(C)C)n2)=O)C1)N(C)CC1N(CC)CCC1 CC(CC1CC1)C(C(=O)NC(C)(C)C)N1CCC(N(CCO)CC2CC2)C1 C1(CNC(C2C(CC)OCC2)=O)(NC(=O)COC2CCC2)CCCCC1C c1(C(CNC(=O)CC2CSC2)CNC(=O)CCC2CC2(F)F)ccccc1 c1(C(=O)NC(CN(C(=O)CCC2CCCCC2)CC)C)n[nH]c2c1C(=O)CCC2 Cn1cc(C(=O)NC(C)(C)CCNC(c2ccnc(C(N)=O)c2)=O)nc1C(F)F C1(C(N(C2CCN(C(=O)COCCO)C2)CCC)=O)CNC(=O)CC1(C)C CC1C=C(C(=O)N2CCC(CCNC(=O)CCn3cc(Cl)cn3)CC2)CC1 N1(CC=C)CCC(N2CCNCC2)CC1.C12C3CN(CC13)CCNC2=O C=CCC(CC)C(=O)NC1(CCC(=O)NC2CCCC2CN(C)C)CCCC1 N1(C(CCC#C)=O)CC(CNC(c2cnn(C3CC3)c2)=O)CC1(C)C C1(C(N2CC(CCC)C(NC(c3ccc(OC)s3)=O)C2)=O)CCC(F)(F)CC1 c1(C(=O)NC2CCN(C(COCC)=O)C2)cccc(-c2nc(=O)o[nH]2)c1 C(C)(C)(CC(=O)NCCC1CCC2CC12)NC(c1ccc(C(C)C)o1)=O Cc1ccc(C(C2CC2)NC(C2CCC(NC(=O)C(O)C(C)C)CC2)=O)cc1 C1(CC(=O)NCC2CC2(F)F)CN(C(C2CCC(=O)O2)=O)CCO1 c1(OC)c(Cl)cccc1S(=O)(=O)Nc1ccc(C)c(NCC)c1.C12(CC1)C(C1CC1)N2 CCC(CC)(C(=O)NC1CC(NC(=O)CCc2cscn2)C1)OC N1(C(C2OCCN(C(c3c(CC)ccs3)=O)C2)=O)CC2CCCC2C1 C(=O)(CCCCCCCC(=O)O)N1CCN(C(C)Cc2cc(Cl)ccc2Cl)CC1 c1(NC(c2ccc(-c3c(OC)ncc(C)c3)cn2)=O)nc(O)ccc1[N+](=O)[O-] C#CCC(O)C(=O)NCC1CCN(C(c2csc(COC)n2)=O)C1 N1(CC)CCOC(C(N2CCC(C)C2CNC(=O)C(C)(C)n2cccn2)=O)C1 CC(C)CC(C)(CNC(=O)CC1CCC(=O)N1C)NC(=O)CN1CCOCC1=O N1(C(C=C(CC)C)=O)CCC(C2CCCN2C(c2cocn2)=O)C1 N1(CC(=O)NCCc2nnc(NCC3CCOCC3)s2)CCS(=O)(=O)CC1 c1(C(=O)NCC2(C(=O)Nc3cncc(Br)c3Cl)CC2)ccc(Br)c([N+](=O)[O-])c1 Cc1ccc(-c2cc(SCCCN3CCC(OC(F)F)C3)on2)cn1 c1(NC(C(C2CCCO2)NC(c2cc(C)[nH]n2)=O)=O)c[nH]ccc1=O c1(C(N(CC(CN(C)C(c2ncccc2Cl)=O)O)C)=O)snc2ccccc12 Cc1ccc2c(c1C(N1C3CCC1CC(CNC(C1CC1F)=O)C3)=O)CCCN2 c1(C(N(C2CCCC2)CCNC(c2ncn(CC)n2)=O)=O)nnn(C2CC2)c1C C1(C(=O)NC2CN(C3CCCCC3)C2)CCC(O)CN1C(c1ccc[n+]([O-])c1)=O C12(C(=O)NCC(c3cn(CC)nc3)=O)COCC1CN(S(C)(=O)=O)C2 c1(C(N2CCC(C)(NC(=O)CC3CC4CCC3C4)C2)=O)ccc2c(c1)COC2 CC1(C)CC(NC(=O)CC2CCC2)CN(C(=O)C#CC2CCCC2)C1 C=CC(C)(CCOC)C(=O)NCC(C)NC(C1OCCOC1C(=O)OC)=O C1(C(=O)NCCCOCCCC)C(O)CCN1C(=O)C(COC)OC CC(C)(C)CCCCC(=O)N1CC2C(NC(C3(F)CC3c3ccccc3)=O)C2C1 C(=O)(CCS(N)(=O)=O)NC(C(=O)NCCC(C)C)CCOCCO c1(C(C(=O)NCC)N(CC(C)C)CC)cnn(CC)c1C CCCCS(=O)(=O)N1CCCCC1C(=O)NC(CCN(C(=O)C(F)F)C)C(C)C Cc1cc(=NCC(C)NC(=O)CN(C)C(=O)C2CC2)[nH]cc1C#N c1(C(=O)NC(CNC(COC(C)(C)C)=O)C2CC2)nccnc1Cl C(c1cccc2cccnc12)=CC(=O)NCC1C2CN(C(CCC=CC)=O)CC21 C1(NC(CCCS(C)(=O)=O)=O)CN(C(=O)CN2CCSCC2)CCC12CCC2 c1(CNC(c2ccc(-c3cc(C(F)F)ccn3)cc2)=O)nc(Cl)ccc1F c1(CNC2(CO)CC(F)(F)C2)ccc2ccc(Br)cc2c1 C(C)(C)(CCCCC(=O)NC1CC(Nc2ccc([N+](=O)[O-])c(C)n2)C1)OC.C(C)=O N1(C(C(C)NC(N)=O)=O)CC2COCC(C1)N2C(C1CCN(C)C1)=O c1(CC)cncc(C(=O)NCC2CCC(NC(c3cc(C)n(CC4CC4)n3)=O)C2)c1 c1(C(=O)NCC(C)N(C(=O)C(C(=O)C2CC2)SC)OCC)cc(C2CC2)ncn1 N1(C(CSCOC(C)=O)=O)CCC(NC(=O)C=CCn2cncn2)C(F)C1 C(C1=NOC2COCC12)C(C(c1c(F)ccc(C)c1)(F)F)=O C(=O)(C(C)CC(F)(F)F)NC(C1CCN(C(C2(COC)CCC2)=O)C1)C C(C(F)(F)C(C)(C)O)NC(C(CCC)NC(c1ccnn1CCF)=O)=O c1(C(N(CCN(C)CC)CC)=O)cc(Cl)ccc1Sc1cccnc1 N1(CC)CCCC(ONC(=O)CCN(C)C(c2snnc2C(C)C)=O)C1 c1(C(N2CCOC(c3cccc(Br)c3)C2)C(=O)NC)cc(F)c(F)cc1F c1(-c2cc(=N)[nH]cc2)ccc2nc(Nc3nccc(N4CCOCC4)n3)[nH]c2c1 CC1CC(NC(c2ncn3c2CCC3)=O)CN(C(=O)Cn2cc(Cl)cn2)C1 N1(C(C(C)CC2CCCCC2)=O)CCC(CO)(CNC(C2(C(N)=O)CCC2)=O)C1 C12(COC)CCC(C(=O)Nc3ccc(N)cc3Br)(CC1)CO2 C(=O)(CC1CN(C)c2ccccc21)N1CCCN(C(CC(C)SC)=O)CCC1 C1(CNC(CP(C)(C)=O)=O)CC2(CO1)CN(C(c1ccccc1Br)=O)C2 c1(C(c2n(CC=C)nnn2)NCc2nc(CC3CC3)cs2)ccc(Br)nc1 N1(C(c2ncn(C)n2)=O)CCCC(C2CCCCN2C(C2CCNC2=O)=O)C1 CCC(CC(=O)N1CC(O)CC1CNC(C1(CN(C)C)CCCCC1)=O)C(C)C C(CN=C(NCc1ccc(Cl)o1)NC1CCCC1)CNC(N(C)CC1CCCO1)=O N1(C(c2ccc(C(C)C)nc2O)=O)CC2CCC(C1)C(NC(C1(C)CC1F)=O)C2 C(=O)(CS(=O)(=O)CCO)N(CCN(C(=O)C(F)(Cl)c1ccccc1)CC)CC CS(=O)(=O)c1cnc(N2CCCC3(NC(=O)CS(N)(=O)=O)CC3C2)c(Cl)c1 C1(C(=O)NCC2(CC)CCC2)CC2CCC1N2C(c1cccc(OC)c1O)=O Cn1cnc2cc(C(=O)NCC3CC(NC(=O)CCC4CC4(F)F)C3)cnc12 c1(CCCCC(=O)OC)ccc([N+](=O)[O-])cc1 c1(C(=O)NCC2CN(C(COCc3occ(C)c3)=O)CC2C)ccc(O)c(Cl)n1 CCCC(C(=O)NCCCCCC=O)C(=O)N1CCN(C2CC2)C(C)C1 S(=O)(=O)(c1ccc(NCC(C)(C)C#N)cc1Br)NC1CC(C)(C)OC1 C1(C(=O)NC2CCN(C(C(n3cc(Cl)cn3)C)=O)CC2)CCC2(CCCCC2)C1 C12(CNC(CSS(C)(=O)=O)=O)CCC1CN(C(c1cccc(Cl)n1)=O)C2 C12(NC(C(C)(C)OC(C)=O)=O)COC(NC(=O)CC3CSCCS3)(C1)C2 c1(C(=O)NCC(CN(C)C(C2CC(F)C2)=O)O)cc(Cl)ccc1O N=c1nc(C2CC2)nc(N2CC3C(CNC(c4cc(C5CC5)no4)=O)C3C2)[nH]1 CCCC(C(=O)OC)C(=O)NC1CC(NC(=O)CC2CC2)C1.c12cccc(c1)S2 C=CC1(CC(=O)N(CC(CC)NC(=O)CCC2(N(C)C)CCCC2)C)CCC1 N1(C(C2(C=C)CCC2)=O)CCCN(C(=O)C=CC(c2ccccc2)=O)C(C)C1 N1(C(CCCC(=C)C)=O)C2CCC1C(C)C(NC(C1CCCN1S(C)(=O)=O)=O)C2 N1(C(CCc2ncn(C)c2)=O)CCCCC1C(=O)NCC1CCN1C(C)(C)C N(C(=NCC1CC1)NCC(c1ccc(F)cc1)(F)F)CCCOOC c1(OC)ncc(Cl)cc1C(N1CCC(N(C(=O)CCc2ccccc2)C)C1)=O N1(C(C2CC=C(C)CC2)=O)CCC2(CC1)CC(Nc1ncnc(O)c1Br)CCO2 c1(C(=O)OCC2CCc3ccc(Br)cc3O2)cc2ccccc2oc1=O c1(CCC(=O)NC2(C)CCN(C(C3(C)COC(=O)C3)=O)C2)cc(Cl)cc(Cl)c1 N1(C(CCNC(CC(C)C)=O)=O)CC(N(C(=O)CC2OCCC2C)C)C2(CC2)C1 c1(CC)conc1CC(N1CCC(N(C(=O)CC2CCNC2=O)CCO)C1)=O C12(CNC(CCC3CC(C)C3)=O)CCCCC1N(C(=O)CC(F)F)CCC2 N1(C(C(C)(C)C2CC2)=O)CCOC(CCNC(c2nocc2C(C)(C)C)=O)C1 c1(C(N2C(C)CCC(NC(c3occc3C3CC3)=O)C2)=O)ccn2nccc2n1 c1(CC)[nH]nc(C(N2CCC(NC(C34CCC(C3)C4)=O)C2C2CC2)=O)c1Cl C1(NC(C(CC)CO)=O)CCCN(C(=O)C=Cc2cccn2C)C1C C(=O)(CCCC(F)(F)F)N1C(CC(=O)NC(=O)CSc2ccncc2)CC(O)C1 c1(CCNC(c2n(CC=C)nnn2)c2nnc(C(F)F)s2)ccc(Cl)c(C)c1 c1(OC)c(F)ccc(C(=O)NCCC2(CNC(=O)CCS(N)(=O)=O)CC2)c1F CC#CCCCC(=O)NCC(C1CCCCN1C(=O)C(C)N1CCCC1)(C)C C1(C(C(CNCC(C)C)OC)=O)CC2(CC(NC(=O)COC3CCCC3)C2)C1 C(=O)(C(C)(O)CCC)NC(CCNC(CN(CCCCCC)C)=O)C c1(C(N2CC3CN(C(c4scc(CC)n4)=O)C3C2)=O)cc(F)cc(Br)c1C c1(OC)ncc(C(=O)NCCCCNC(c2ccccc2Br)=O)c(C)n1 c1(C(=O)NCC(CO)NC(c2c(OCC#C)nccc2)=O)ccc(C)c(Cl)c1Cl Nc1cc(F)cnc1C(N1CC(NC(c2csc(Cl)n2)=O)C2CC12)=O c1(C(=O)OC)cc(C)c(C(=O)NC2CC=CCC2)o1 C1(C(N2C(CNC(c3ccc4c(n3)CCC4)=O)CC2)=O)CC2CC1CC2(F)F C(C(C(C)(C)C)NC(=O)C(O)Cc1ccccc1)NC(Cn1c(C)cnc1)=O Cc1cccc(C(N2CC3(CC3C(=O)Nc3ncn(C)n3)C2)=O)c1F C1(C(=O)NCC(CNC(C(CC)OC)=O)OC)(OC)CCC(C)CC1 c1(CNC(C(C(=C)C)(C)O)=O)nc2ccccn2c1C c1(C(N2CCC(CCNC(C(C(C)C)SC)=O)CC2)=O)cccc2c1CCCN2 C1(N(C(=O)CCc2ccc(F)nc2)C)CN(C(c2cc(N)ccn2)=O)CC1(C)C S(=O)(=O)(CCC(=O)N1CCSCC1C1CCN(C(=O)CCCN=[N+]=[N-])C1)NC N1(C(c2n(C)nc(C)c2Cl)=O)CCC2(CCCN2C(=O)C#CC(=O)N(C)C)C1 N1(C(C=Cc2cccc(C)c2)=O)CCC2(C=C(C(=O)NCCC3(C)N=N3)C2)C1 Cc1cn2c(n1)CCC(C(=O)NCC1(NC(c3cnoc3)=O)CCCC1)C2 c1(CN(C(C)(C)CCc2cccn2C2CCCNC2)CCN)ccc(Cl)c(Cl)c1 C1(NC(Cc2c(C)nc(S)s2)=O)CC2CN(C(=O)CCC3CCCO3)CC2C1 Cc1cccc(F)c1CNC(=O)NC12COC(C1)C(NC(=O)OC(C)(C)C)C2 C12(C(=O)OC)C(N3CCCCC3)C1CN(C(c1n[nH]c(C)c1Cl)=O)C2 c1(OCC)nc(C(=O)NCCCCCN(C)C(c2conc2C)=O)co1 N1(C(c2cn(C)nc2I)C(=O)NC(C(=O)OC)C)CCS(=O)(=O)C(C)(C)C1 c1(C(N2CC(CC(=O)NCc3csc(O)n3)C2)=O)ccc(Cl)cc1[N+](=O)[O-] N1(C(CCCSC)=O)CC(F)CC1CNC(=O)CN1CC(=O)NC1=O C1(CC)C(NC(=O)CCN(CCC(C)(C)C)C)CCCN1C(=O)C(=O)N(C)C C1(c2cccc(-n3c(C)c(N4CCC(C#N)CC4)nn3)c2)CC(C)CC(C)(C)C1 c1(CN2CC3CC(NC(C4C(C)(C)C4)=O)CC3C2)cccc(S(C)(=O)=O)c1 Cc1ncc(C(=O)NCCCCC(=O)NCC2CC[Si](C)(C)C2)n1C C(=O)(C(C)(C)CCC#N)N1CC(C(C(=O)NCc2cn(CC)nc2)OC)C1 c1(C(=O)NCCCC(C)NC(=O)CCSCC(N)=O)nnc2n1CCCC2 C1(C(=O)NCCCCCNC(C2Cc3nncn3C2)=O)Cc2ccncc2N1 C#Cc1ccc(C(=O)N(CC(C)NC(c2cncn2C)=O)C)c(C)c1 c1(C(=O)NC(CC)CN(C)C(C2C3CC4C(C3=O)C24)=O)cccc2cnsc12 C1(CC)CN(C(c2cn(CC3CCOC3)nn2)=O)CCN1C(=O)CCn1cnnn1 C1(C(=O)NCCC=C=C)CNC(=O)CN1C(=O)CC1CC(CC)C1 C1(N(C(c2c(C)c(-c3ccccc3)[nH]n2)=O)C)CCCCN(C(=O)CC(C)F)C1 CC(C)(C)C#CC(=O)NC(Cn1cccn1)C(=O)NCCn1cnnc1 CC1(C)C2CCC(C(N3CCC4CCC(NC(C5CCCN5N=O)=O)C34)=O)C1C2 c1(C(=O)NCC2C(CNC(=O)Cc3ccno3)C2)nc2cccnc2s1 Cc1nocc1CC(C1CCN1CCc1ccccc1)NC(C1CNC1)=O c1(C(N(CC(C)C(=O)N(CC(C)(C)C#N)C)C)=O)c[nH]nc1[N+](=O)[O-] c1(OC)c(F)ccc(F)c1C(=O)NC1CC2CN(C(=O)Cc3cnns3)CC2C1 C1(C(N(C2CCN(C(=O)CN3CCOC3=O)CC2)CC)=O)CC(=O)N(C2CC2)C1 N(C(=NCC1CC1)NCC(CC)CC)CC(C1CC(F)(F)C1)OC c1(C(=O)NCC(CN(C(C(COC)(C)C)=O)C)(C)C)ccc(C)c(C2CC2)c1 C1(NC(C(CC#C)NC(=O)CCC2CCC2)=O)CCn2nccc2C1 c1(SC)cc(F)ccc1C(N1CC2CCCC12)=O C1(C(=O)NCCN(CCOC)C)CCC(C)CN1C(c1cc(Cl)c[nH]1)=O C(=O)(CC1NC(=O)c2ccccc21)C(C)=O.c1(OCCO)c[nH]c(N)cc1=O CC(Cc1ccco1)C(=O)NC(CC1CCOCC1)C(=O)NCC1(C(N)=O)CC1 c1(CC)cc(C(=O)NC(C)CN(C)C(c2cccc(CC)n2)=O)ccn1 N1(C(CC2(OC)CC2)=O)CC2CCC(CNC(C3CC34CC(C)(C)C4)=O)(C2)C1 c1(OC)c(Sc2ncc(Cl)cn2)cc(F)cc1F N1(C(CCSC)=O)CCCC(O)(NC(=O)C(C2CCCCCC2)C)C1 C(=O)(C1=CCCC1)NC1CCC(CC(N2CC(CCO)(CC)C2)=O)C1 C1(C(=O)OCC)(CC)CN(CCN(C(C)C(=O)N(C)CCO)CCOC)C1 c1(CC(=O)NC(C2CN(C(C3(n4ccnn4)CC3)=O)CCO2)C)ccc(C#N)cc1 c1(C(N2CC(NC(C(C)=C(CC)C)=O)C(SC)C2)=O)cc(C)c(=O)n(C)c1 c1(C(=O)NCC2C(CNC(c3c(C)cc(Br)o3)=O)C2)cc2c(F)cccc2[nH]1 Cc1nc(Cl)c(NC(c2nc(NCc3cc(Br)c(C)cn3)cn2C)=O)cc1Br c1(C(N(CCN(C2CCCC2)CC)C(C)C)=O)cccc2sccc12 CN1CCCC(Cn2c(N3CCC(CC(=O)OC(C)(C)C)C3)nnc2CO)C1 CC1CSCCCN1C(C1(C)CCCN(C(c2cnns2)=O)C1)=O N1(C(c2cnc(CC)s2)=O)C2CCC1C(CNC(=O)CC1OCCO1)C2 CCCCCC(C)CC(=O)N(C)CC=CC(N1CCC(c2nc[nH]n2)C1)=O N1(C(C(CCCC)O)=O)CCC(C)N(C(=O)CC2CCC3CC23)CC1 N1(C(c2noc(CC)c2C)=O)CCC(NC(=O)C(C)SC)C(CO)C1 C=CCC(CC(F)F)C(=O)N1CCOCC1CNC(c1cc(F)c[nH]1)=O c1(C(N2CCOC(C(C)(C)O)C2)C(=O)NC2(C)CC2)nccc(Cl)c1Cl CC1CC2CN(C(c3cnnn3C3CC3)=O)CC2N1C(C1CCCC1(C)C)=O c1(C(=O)NCCCN(C(C2C(CC)CCC2)=O)C(C)C)cnc2ncccn12 c1(C(C(=O)NCc2ccccc2)N(CCC(=O)NC)C)ccc(OC(F)F)cc1 CN1CCC(NC(=O)COC(C)(C)CNC(C2(C3(O)CCC3)CC2)=O)C(C)(C)C1 Cc1ccn2cnc(C(=O)NCC3(C)CCN(C(C4(C5CC5)CCC4)=O)C3)c2c1 Cc1onc(Br)c1C(=O)NC1COCC1NC(C1(O)CCOCC1)=O Cc1cc(C(=O)NC(C)CN(C(=O)Cc2ccn(C)n2)C)cc2ccsc12 C1(C)(C(=O)NC(CC)(C)C)CCCN(Cc2occc2C(=O)NC)C1 Cc1ccc(N2CCCC(C(=O)NCC3CCCN3C(C3CC(F)C3)=O)C2)nc1 C1(NC(c2csc(-c3cnc[nH]3)n2)=O)CN(C(c2cc[nH]n2)=O)C2(CCC2)C1 N1(C(C(F)=CCC)=O)CCC(NC(=O)CCCc2cc(F)ccc2F)C(C)C1 CC1CN(C(=O)C=Cc2nccs2)CCC1NC(c1cncn1C)=O c1(NC(C2CCN(C(=O)Cc3cscn3)CC2)=O)cc2ccc(Br)cc2s1 N1(C(C(C)C)=O)CCN(C(C2CCC2c2cncn2C)=O)CC1 c1(C(N(C2CCN(Cc3c(Br)cc(Br)cc3Br)C2)C)=O)ccc(O)c([N+](=O)[O-])c1 S1(=O)(=O)c2cccc(c2)C(=O)N2CC(C2)N1C.C(CSC)(OC)N.C1(CC2CC2)CC1 C(c1cccc(F)c1)=CCC(N1C(CNC(C(CC)C)=O)C=CC1)=O CC1=CCN(C(C23CC2CCN3C(=O)CN2CC(=O)NC2=O)=O)CC1 c1(CCC(=O)N(CC(CC)NC(=O)C(CC2CCC2)OC)CC)cnn(C)c1 CC1(C)COCCC1C(=O)NC1CCCC1CC(N1CCCC1)=O N1(C(c2ccc(C)nc2)=O)CCN(C(=O)CCOCC(F)F)CC1C1CC1 N1(C(c2cnc(C)o2)=O)CC(C(=O)NCC(c2cccnc2)O)C(C)C1 C1(C(C)C)CN(Cc2cccc(F)c2Cl)CCN1Cc1ccc(I)o1 C1(OC(C)C(=O)N(CCNC(c2ccc(CN(C)C)cc2)=O)C2CC2)CCCCC1C C1(OC)CC(NC(=O)CSc2nncn2C)CN(C(c2cc[nH]c(=N)c2)=O)C1 N1(C(C(C)N(C(C)=O)C)=O)CCC(N(C(=O)Cc2cccnc2C)CCO)CC1 C(=O)(C1=NOC(C)C1)NC(C1CCCN1C(c1cc(Cl)n(C)n1)=O)C C(=O)(CCC(=O)NCC1CC(O)CN1C(c1cc(OC)n[nH]1)=O)OCCC c1(C(N2CCN(C(CCC#C)=O)C(CC)C2)=O)ccc2oc(S)nc2c1 CC1=CCC(C(=O)NC2CN(C(c3cccn3C(C)C)=O)CC2C(F)(F)F)CC1 C(=O)(C(C(C)C)n1cc(Br)cn1)NCCC(C)NC(c1c(CC)nc[nH]1)=O C1(NC(=O)CNC(c2ccccc2O)=O)CCCCN(C(c2cc(F)c[nH]2)=O)C1 c1(C(=O)NC2CC(NC(=O)CCc3nc[nH]n3)C2)cn2ncccc2n1 C1(C(N2C(CNC(C(CC)(O)c3cccc(Cl)c3)=O)CC2)=O)OC2CCC1CC2 c1(C(N2CC(C(C)NC(c3c(C)nccn3)=O)C2)=O)ccc(Br)cc1C#N CC1(C)CCOC1CNC(C1CC(CNC(=O)Cc2ccc(O)nc2)C1)=O C1(C(=O)NC2(C(=O)NCC3CC(CSC)C3)CCC2)CCN(C)C1C C12(C(N3CCC(CC)(CC)CC3)=O)C(N)C3CCC1C2C3 N1(C(c2n(C=C)ncc2)=O)CCCC(F)(CNC(=O)Cn2cc(C(F)F)cn2)C1 n1(CC(=O)NC(CNC(COCC(=C)C)=O)(C)C)cc(-c2cccs2)cn1 N1(C(C(c2c(C)nn(C)c2C)=O)=O)CCN(C(C2CCS2(=O)=O)=O)CC2(CC2)C1 c1(CC(=O)NCCCOCCCNC(=O)CCC2CCCCO2)nc([N+](=O)[O-])n[nH]1 c1(C(=O)NC2CCC(CCNC(c3c(C)oc(Cl)n3)=O)C2)cc(S(C)(=O)=O)cs1 c1(C(N2CCC(O)(C(C)C)C2)=O)ccc2c(c1)[nH]c(=N)n2C CC1OC2(CNC(=O)CN(C)C(=O)C3CC3)CC1(NC(C1CCNC1=O)=O)C2 C1(CC(=O)NCCNS(NC)(=O)=O)CN(C(=O)C2=NOCC2)CCO1 CCC(C#N)C(=O)NC(C(=O)NCc1ncn(C(C)C)n1)c1ccco1 C(CC(=O)NCC1C=CCN1C(c1ocnc1C(F)(F)F)=O)(C(F)(F)F)OC N1(C(c2cncc(NC)n2)=O)CC2CC1CC2NC(c1coc(C(N)=O)c1)=O N1(C(C2(CC)COC2)=O)CCC2CN(C(=O)C(C)(O)CC(C)C)CC2CC1 C1(C(N2C(COC)CCCC2)=O)CN(C(c2ccc(C)nn2)=O)CC1(C)C c1(C(=O)NCC(F)CNC(=O)CC2CCCC2)ccccc1C1CC1CC Cc1csc(CCC(=O)NCCC2CN(C(c3csnc3Cl)=O)C2)n1 CCC(C)C(C)C(=O)N1CCOCC(CNC(c2cncc(F)c2Cl)=O)C1 Cc1cc(C(N2CC(C(=O)NCCSC(C)C)CC(F)C2)=O)ccc1C(C)C C1(NC(C=C(C)C(C)C)=O)COC2(CNC(C3COC4(CCC4)C3)=O)CC1C2 N1(C(C(C(C)C)O)=O)CCC(CNC(=O)C(N2CCN(C)CC2)C)C(F)(F)C1 C1(C2CCN(C(=O)Cn3ccnn3)CC2)(NC(c2cccc(C#C)c2)=O)CC1 C#CCCCC(C)C(=O)N1CC(O)(CNC(=O)C(O)CC)C1 Cn1ccc2cnc(N3CC(C(=O)NCc4ccc(O)cc4Cl)C3)nc12 c1(NCC2(NC(C3CCCCC3)=O)CC2)ncnc2sc(C(C)C)cc12 CCCC(CC)CCC(=O)N(C)CCOCCN(C(=O)C(C)(C)c1cc[nH]n1)C Cc1cc(C(=O)NC2COCC2CNC(=O)CCCn2ccnc2C)c(O)nn1 N1(C(c2c(C#C)c[nH]n2)=O)CCC2CCCC12CNC(c1cc(C)c(C)[nH]1)=O c1(C(N(C)CC2(O)CN(C(c3[nH]cc(C)c3)=O)C2)=O)cccc(C(F)(F)F)c1C CCC(CC)(CCNC(C1CSCCS1)=O)NC(c1ccc(C(C)(C)C)cn1)=O C1(NC(C(C)OCC#C)=O)CN(C(c2ccc(S(C)(=O)=O)[nH]2)=O)CCC12CCC2 C1(CNC(c2cc(C)oc2)=O)CCCCC1NC(=O)CCC1CC1 C=CC(C)CC(=O)N1CCCC1(C)C(=O)NCC(n1ccnc1)C c1(OC)cc(-c2ncsc2C(=O)Nc2cc(-c3ccccc3C)cs2)c(OC)cn1 C1(CNC(c2cc(C)[nH]n2)=O)CC2(CCC2)CN1C(c1cc(N)c(C)cc1C)=O c1(C(N2C(CC(N3CC(C(=O)OCC)C3)=O)CCC2)=O)cc(Cl)cc(C(F)F)n1.SCC c1(OC)ccc(OCC(=O)NCC2CN(C(=O)CN(C)CCO)C2)c(Br)c1 c1(C(=O)NCCC2CCCN(C(C(C)O)=O)C2)ccc(Br)c(Br)c1 c1(CN2CCC(Cc3ccc(OC)cc3F)CC2)cc(OC)cc2cccnc12 C1(CN(CC(=O)NCCC)C)CCCN(C(c2ccc(-c3nc[nH]n3)cc2)=O)C1 C1(c2c(C(=O)OC)n[nH]c2)CCN(C(=O)CNC(=O)Cc2ccccc2Cl)CC1 Cc1cnc2cc(C(N3CC(CNC(=O)C(C)C4CCC4)C4(CC4)C3)=O)nn2c1 N1(C(=O)C2CC2)CC(F)(F)CC1C(=O)N(c1nccs1)CCCn1ccnn1 N1(C(CN(C(C(C(C)C)O)=O)C)=O)CCCC(C)C1CO N1(C(C(COC)(C)C)=O)CCC(NC(C2C=CCOC2)=O)C(O)C1 C1(C(=O)NC(CNC(c2cc(C)ncc2)=O)C2CC2)CCc2ncc(C)n2C1 CCC(CC(F)(F)F)C(=O)NCC12CC(NC(=O)C=Cc3ccsc3)(CCO1)C2 c1(C(N2CC(CCOC)N(C(=O)CC3(C#N)CC3)CC2)=O)ccc(Cl)c(C#N)n1 CC1OC(=O)NC1C(N1CC(CF)(NC(C2CCCS2(=O)=O)=O)C1)=O Cc1ccc(N)c(C)c1C(N1CCC(C)(NC(=O)CC(C)C(C)(C)C)C1)=O c1(CC(=O)NCC(C)N(C)C(C2CCCCS2(=O)=O)=O)ccc2c(c1)CCN2C c1(NC(CCCN(C(CN(CCC)C)=O)C)=O)ncn2c1CCC2 C(=O)(C(F)(CNC(c1cnccn1)=O)C(C)C)NC(CC)(C)CCO Cc1c(C(=O)NC2CC(C)N(C(c3ccsc3C#N)=O)C2)sc2cncn12 c1(C(N2CC(NC(c3c(C)nc(O)[nH]3)=O)CC2(C)C)=O)ccn2nnnc2c1 c1(C(=O)NCC(C)NC(c2coc(C(F)F)c2)=O)csc(C(F)(F)F)n1 CCCCCCC(C)C(=O)NC1CC2CC(NC(=O)CCCn3cncn3)CC12 N1(C(c2ccc(SC)cc2)=O)CCN(N2CCC(N3CC(O)C3)CC2)CC1 C(=O)(C(F)(F)c1ccccn1)NCC(C1CC1)NC(C(C)N(CC(F)(F)F)C)=O CC(C)CCCC(=O)N1CC(CNC(=O)C(C(C)(C)C)NC=O)CCC1C c1(CCC)noc(CN(CC(=O)NCC2CC2C(F)(F)F)CC)n1 C(CO)(CCCCNC(C1CCN(C)C1)=O)NC(c1c(C)[nH]nc1Br)=O CCC(C)(CO)C(=O)NC1CCN(C(=O)CC(=O)NCCCCOCC2CC2)C1C C=Cn1nccc1C(N1CCC(CNC(=O)CCOCCC)(OC)C1)=O c1(C(=O)NCC2(F)CN(C(C3(C(=O)NC)CCC3)=O)C2)cnn(C(C)(C)C)c1C N1(C(C(C)NC(C2CCCC2)=O)=O)CCC2(CCCN2C(=O)CO)CC1 N1(CC(=O)NC2CN(C(c3cc(F)c[nH]3)=O)C3CC23)CCCCS1(=O)=O C(=O)(C1=C(C)CCC1)NCc1cn(C2CN(C(C3(OC)CCCCC3)=O)C2)nn1 CCCC(C)C(=O)NCC1(C(=O)NCC2CCSC2)CC1 C1(=CC(=O)N(CCCN(C)C(C2CCCCC2F)=O)C)CN2CCC1CC2 N1(C(C2CN(CC)C(=O)N2)=O)CC(NC(C2CCN2C(C)(C)C)=O)CCC1C N(C1c2ccccc2CC1C(=O)NCCN(C)C)C(CCCCN(C(C)C)C)=O C(=O)(C(F)CCC(C)C)NCCNC(CNC(C1=C(C)CCC1)=O)=O C1(NC(C2CCS(=O)CC2)=O)CC2CCC1(C(=O)NCC(O)C1(Cl)CC1)C2 c1(OCC(=O)NCC2(C(N)=O)CN(C(C3CC3Cl)=O)C2)ccc(F)cc1Cl c1(S)ccc(C(=O)Nc2ccccc2)cc1F.C(=O)(CNC(C1(CO)CC1)=O)OC CC1(NC(c2cc(CF)on2)=O)CCCN(C(C2CC(F)C2)=O)C1 C=CCC(CC=C)C(=O)N1CC=C(C(=O)NC(CC=C)CCOC)CC1 N1(C(C(Cc2ccco2)N(C)C)=O)CC2CC1(c1cn(C(C)(C)CO)nn1)CO2 c1(C(C(=O)OC)N(CC(CCC)C)C)cncc(F)c1 c1(C(N2CCN(C(C(C)(C)O)=O)C(C)C2)=O)c(F)cc(Br)cc1Br C1(C(=O)NCc2cc(C)ns2)CC2CCCC2N1C(=O)C(C)(C)C C1(CN(OC)C)CCCC(CN=C(NCC(F)(F)Cl)NC2CCC2)C1 N1(C(c2c(C)ccnc2)=O)CCC2C(C(=O)NCC(F)(F)C(F)F)C2C1 C(=O)(CCC(=O)N1CCN(C(=O)CC(C)Nc2c(C)noc2C)CC1)OCC Cc1nnccc1C(=O)NCC1CC1CNC(C1CCNC1C(C)(C)C)=O c1(C(N2CCN(CCNC(C=C(C)C)=O)CC2)=O)cc(C)c2ncccc2c1C c1(OC)ccc2c(c1)N(C(c1cnn3ccccc13)=O)CC2C Cc1cncc(CCC(=O)N(C)CCNC(C2CC(C)(C)C2)C2CC2)c1 Cn1cnc(C(=O)NC2CC(C)(C(=O)NC3CC4CCC3O4)C2)cc1=O C1(NC(Cc2cn(CC)nc2)=O)CCCN(C(C2(CC3CC3)CC2)=O)CC1 C(=O)(CCCCC1CC1)N1CC(C(C(=O)N)O)C1.C#CC(C)(C1CC1)CC c1(-n2c(CONC(COC)=O)ncc2)ccc(OC)cc1C N1(C(c2c(C)nsc2)=O)C2CCC1C(C)C(NC(=O)CSCC1CCCCO1)C2 Cc1noc(CNC(=O)CC2CCCC2C)n1.C12(CCC1)CC(=O)N2C N=c1cc(C(=O)NCC2CN(C(C3CCSC3)=O)CC2C(F)(F)F)nc(Cl)[nH]1 N1(C(CC(C)C)=O)C2CCC1C(NC(=O)C=Cc1ccoc1)C2 c1(OC)cccnc1C(N1CC(C)(C(=O)Nc2ccc(C(F)F)nc2)C1)=O C1(NC(C2C=CC(NC(Cc3cccc(C#N)c3)=O)C2)=O)CC2(COCCO2)C1 C12(NC(CN(C)CC3CC3)=O)CC(C1)N(C(C1(Cc3cccs3)CC1)=O)C2 C(C(C)(C)C(=O)NC(C)C(c1ccccc1)NC(c1cnc[nH]1)=O)NC(C)=O c1(CC(N2CC(N(C(=O)CC3CC3C)CC)C2)=O)csc(C)c1 c1(C(N2CC3CCN(C(=O)CC4CCC4)CC3C2)=O)cc2c(Br)cncc2s1 Cc1cc(C(=O)NCC2(C)CCCN(C(=O)C(C)CN3CCC3)C2)cc(O)n1 C(C)(C)(CC(F)C(=O)N1CCC1(C)CC)NC(C=CC(=O)OCC)=O CNS(=O)(=O)N1CCC(C(=O)NCCN(C)C(C2CC3(C2)CC3F)=O)CC1 C1(CCOC)CN(C(C2CC(C#N)C2)=O)CCN1C(=O)CCn1cc(C)cn1 N1(CC(c2nnnn2C2COC(C(F)(F)F)C2)(C)NCC(CO)F)CCCCC1 Cc1cnc(Cl)c(C(=O)NCC(F)(F)Cn2cc(CC3CCCCNC3=O)nn2)c1 C1(NC(C(C)C(=O)OC(C)(C)C)=O)CC2CCC(C1)N2C(c1cc(F)n(C)n1)=O C1(NC(C(C=C)OC)=O)CN(C(C2CCOCC2(C)C)=O)CC1C=C c1(C(=O)NC2(CN(C)C(c3coc(C(F)F)n3)=O)CC2)ccc2ccnc(Cl)c2n1 c1(C(=O)NCCCCCCN(C(=O)C(F)CC2CCCC2)C)cnc(O)c(F)c1 Cc1c(C(=O)NCC(C)C(F)C(=O)NCCc2ccncn2)cncc1F N1(C(c2n(CCC)ccc2)=O)CCN(C(C2C(C)(C)C2(C)C)=O)CC1CC1CC1 c1(C(N2CC(C)(CNC(c3ccccc3-c3ncc[nH]3)=O)C2)=O)cc2scnc2[nH]1 C1(CC#C)(C(=O)Nc2ccccc2CC)CCN(C(C2CSCCO2)=O)C1 N12CCc3nc(sc3C1)C(=O)NCC2=O.CCC(O)C(=O)OCC(C)(C)C N1(C(=O)COCC(C)C)CC(NC(COc2cccc(C)c2)=O)CC(O)C1 c1(CNCCN2CCN(C(Cc3cccc(CC)c3)=O)CC2)cccc(F)c1Cl Cc1noc(C)c1C=CC(N1CC(C)(C)CC1CNC(C1CC(=O)N(C)C1)=O)=O C1(=O)C2=NOC(C2)C(C)N1.C(CCCCCO)NC(C1CN(CC(F)F)C1)=O C(=O)(C1=CCC(C)CC1)NC(CNC(c1c(C)occ1-c1ccccc1)=O)C [N-]=[N+]=Nc1cncc(C(N2CCC3(CNC(=O)CSC(F)(F)F)CCCC23)=O)c1 CC1CC(CNC(c2coc(Cl)c2)=O)CCN1C(=O)CC1COCC(C)(C)O1 C1(C(N2CC3C(NC(=O)CSCC4CCCCO4)(C3)C2)=O)CC12CCSCC2 CC1(C)C(O)CC12C(=O)N2.C(CCCN1CCC1)NCCCO Cc1cccc(-c2nc(C)c(C(N3CCC(NC(C4C=CCC4)=O)C3)=O)[nH]2)c1 Cn1cc(C2=CCS(=O)(=NC(=O)C3CCCC(C(=O)O)CC3)CC2)cn1 C1(NC(CCCNC(C2(OC)CC2)=O)=O)CN(C(c2ccccc2)=O)CC1OC C(=O)(CC1=NN(C)C(=O)C1)N1C(C)(C(NOCCCC=C)=O)C=CC1 C1(NC(Cc2c(C)nc(C)s2)=O)CCCCN(C(c2cc(N)c(Cl)cn2)=O)CC1 C1(CNC(C(CC)OC)=O)CN(C(=O)C(C)(C)NC(=O)C(F)(F)F)CC12CCC2 Cc1nn2cc(C(=O)NC3CCC4CN(C(C5CC=CCC5)=O)CC4C3)nc2s1 C=CC1(C(=O)NCc2cnsc2)CCN(C(c2cc(C)cc(C)n2)=O)CC1 C1(NC(CCSC)=O)CCN(C(=O)COC2(C)CCC2)C(c2ccccc2)C1 c1(CC(=O)NCC(CC)NC(=O)C(C)(C(C)C)N(C)C)ccc([N+](=O)[O-])cc1 C1(NC(c2ccc(OC3CCOC3)cc2)=O)CC12CCC(NC(=O)C1CC1)CC2 c1(CCC(=O)NCC(=O)NCCCF)nc2onc(-c3ccccc3)c2c(=O)[nH]1 c1(C(=O)NCC2(C(C)NC(c3cc(C#N)no3)=O)CC2)cc(Cl)ccc1Cl c1(OC)ccc(C(=O)NC2(C)CCN(C(C3CCCN3CC(C)C)=O)C2)c(C)n1 C1(NC(CC(COC)COC)=O)CN(C(=O)CN2CCC(C)CC2)CC2(CC2)C1 C(=O)(CCCCCCCCN)N1CCC(CCNC(C)=O)C1 c1(C(=O)NC2COCCN(c3ncnn4cccc34)C2)cc2cccnc2s1 CCCCC(O)C(C)C(=O)NC1CCC(CNC(c2c(CC)cccc2F)=O)C1 N1(CC)CC2(CN(C(=O)C3=CCN(C(C4(C)CCCN(C)C4)=O)C3)C2)C1 N1(C(C(CC)C)=O)CCC(C)C(CNC(C2CN(C)CCO2)=O)C1 N1(C(c2ncn(C)c2)=O)CC2CCC(C1)C2NC(c1c[nH]c(C#N)c1)=O C(=O)(C(F)CC(C)(C)C)N1C(C(C)NC(c2nn(C)cc2Cl)=O)CCC1 CCCCC(C(=O)N(C1CCCC1)C)NC(=O)CN(C)C(=O)CC C(C)(C)(C(C)CC(=O)NCC(C)(C)F)NC(C(c1cnn(C)c1)C)=O CCCC(CNC(=O)C(C)(O)C1CCC1)C(=O)Nc1c[nH]ccc1=O N1(C(CC=CC)=O)CCC2(C1)CN(C(=O)CC1(C)CCC1)C2 c1(C(N)=O)c[nH]c(C(=O)NCC(O)CNC(C2(Cl)CC2)=O)c1 Cc1ncc(Cl)c(C(=O)NC2(CCCNC(C3CCCN3N=O)=O)CC2)n1 N1(C(C(CCC)=CCC)=O)C2CCC1CC(NC(=O)C(C)Cc1ccccn1)C2 N1(C(C(c2ccccc2)OC)=O)CC2CCCC2(NC(=O)CCOC2COC2)C1 c1(CC(=O)NC2C(CNC(c3cnn(CCO)c3)=O)CC2)cccc(F)c1Cl Cc1csc(C)c1C(N1CCOC(C(=O)NC(C)CS(C)(=O)=O)C1)=O Cc1nc2c(C)cc(C(=O)NC3(C)CCN(C(=O)Cc4ccccn4)C3)cn2n1 C1(=O)C(F)(F)CN1.C(C)(C)(CN(C(=O)C=CC1CC1)C)OC(C)C C(C)(CCC(=O)NCC1CC1c1ccoc1)NC(CCc1c(C)noc1)=O N1(C(C2(CC)CCC2)=O)CC(C)OC2(CCN(C(c3ccc(C)cc3)=O)CC2)C1 C1(CCN(CC(=O)Nc2ccccc2)CCC)CCCN(CCCCCF)C1 C(CC(C)C)(C(=O)N1CCC1C(=O)N(C(C)(C)CO)C1CC1)NC(C)=O N1(C(c2cccc(CC)n2)=O)CCC(C(=O)NC(CCO)C2CC2)=C(F)C1 c1(C(=O)NC(CNC(C(N)=O)=O)Cc2ccccc2)cccc2c[nH]nc12 Cc1ccc(Cl)cc1-n1cc(CC(C)NC(C2CCC2C(=O)O)=O)nn1 C1(CNC(=O)NC2(C)CCOC3CC23)CC2(CC(OC(C)(C)C)C2)C1 C1(CNC(C=CC)=O)(CO)CCN(C(C23CC(c4ccccc4)C2C3)=O)CC1 c1(C(=O)NCC(CNC(c2csc(C(N)=O)n2)=O)OC)ccn(C)c(=O)c1 c1(-c2ccc(SC(=O)NCC(C)(C)N(C)C)cc2)ccn2ncnc2c1 C=C(Cl)CCC(=O)N1CC(C2CCN(C(=O)C(C(C)C)OCC(C)C)CC2)C1 c1(C(=O)NC2CC(NC(C=CC(CC)C)=O)CC2O)cc(C)ccc1O c1(C(=O)ON(CCOCCC2CCC23CCC3)CC)sc(-c2ccccc2)cc1N C1(C(=O)NC2C=CCN(C(c3cc(C(C)C)sn3)=O)C2)Cc2cccnc2C1 c1(C(N2CCCCC(NC(C(C)=C(C)C)=O)C2)=O)nccc2c1NCCC2 C(=O)(CCCS(N)(=O)=O)N1CCN(C(C(COC(C)C)(C)C)=O)CC1C N1(C(Cc2c(OC)cccc2Cl)=O)CCCC12CCN(C(C1(C)CC1(C)C)=O)CC2 c1(C(N(C)CC2CCCN2C(C2CCCN2C)=O)=O)nc(Cl)ccc1N C(=O)(C1=NOC2(CCC2)C1)N1CCCC(NC(C(CCCC)CC)=O)C1C C(=O)(C1CCCn2cnnc21)NC1CC(C)CN(C(C2CC(O)C2)=O)C1 N1(C(=O)Nc2c3n(nc2)CC(C)CO3)CCCCCC(S(C)(=O)=O)C1 N1(C(c2nn(C(CC)CC)c(C)c2)=O)CC(C)N(C(c2n[nH]cc2C)=O)CC1C c1(CC(=O)NC(c2ccccc2)C2CCCCC2)ccnnc1O C1(CC)CN(C(=NCCN(C)C)N(C)Cc2ccc(Cl)c(F)c2)CCO1 c1(NC(C(=O)NCC(C(=O)NC2CCC(C)CC2)(C)O)=O)cccc2ccoc12 N1(C(C(CC(N)=O)O)=O)C2CCC1CN(C(c1cc(C3CC3)ns1)=O)CC2 C1(COC)CN(C(=O)C(c2ccccc2F)C)CCN1C(c1ccc(O)nc1)=O O=S(=O)(c1cnc(NCc2ccc(C(F)(F)F)s2)c(Cl)c1)NCCc1cnoc1 N1(CC(=O)NC(CNC(CCCN(C)C)=O)(C)CO)CCCNS1(=O)=O Cn1nccc1C(=O)NCC1COC(CNC(=O)CCc2ccccc2)C1 N1(CCNC(c2ccn(CC#N)n2)=O)CCN(C(c2cnc(Cl)s2)=O)CC1 N1(C(C(CC)C(=O)OC)=O)CCC(C2CN(C(c3nocc3C)=O)C2)CC1 C(C)(CCC(=O)NC(C(=O)NC(CO)C(C)NC(=O)OC(C)(C)C)C(C)C)SC C(=O)(C(=O)N(CC#C)CCOC)NCCCNC(=O)CNC(C)=O.C(C)=O C1(NC(c2c(C)cc(CC)o2)=O)CCN(C(c2ccc(N)c(Cl)n2)=O)CC1O Cc1ccc(-c2nc(C(=O)NC3CCNCC3O)cs2)cc1 C1(OC)CCC(N=c2[nH]c(=NCCn3cc[nH]c3=O)nc(-c3ccsc3)[nH]2)CC1 c1(C(C)=O)cc(C(=O)NC2CN(C(C3(C)C=CCC3)=O)CC2C(F)(F)F)c(C)o1 C(=O)(C(C(C)(C)C)N1CCCCC1=O)NC1N(C)CCCC1.N12CCC(C1)C2 C1(NC(c2c(SC)cnn2C)=O)CN(C(=O)C(C)Oc2ccccn2)CC1(C)C C(=O)(C1=NOC(CNC(=O)C(C)C2CCOC2)C1)NC(CCC(=O)OCC)C N#Cc1cccc2[nH]cc(C(N3C4CCC3C(CNC(c3ccsn3)=O)C4)=O)c12 c1(C(C(=O)N(C2CCN(C(c3c(C)csc3)=O)C2)CCO)O)ccc(Cl)cc1F C(C1CCOCC1)=CC(N1CC(C(C(=O)NCCCc2cnc[nH]2)OC)C1)=O C1(NC(c2cc(COC)on2)=O)CCCC(NC(C2CC(C#N)C2)=O)C1 Cc1nc2[nH]c(C(=O)N(CC(C)NC(c3cc(Cl)c(F)cc3F)=O)C)cc2s1 N1(C(CCN(C(=O)Cc2cc[nH]n2)CC#C)=O)CCC2(CNC(=O)C2)C1 C1(C(=O)NCCSCC=C)CN(C(C2CCC=CCCC2)=O)CC12CCC2 C(=O)(C(C)(CC)C(F)F)N1CCC(CCNC(C=CCC)=O)C1 C1(C(N(CC(C)NC(c2ccc3n[nH]cc3c2)=O)C)=O)CN2CCCCC2CO1 c1(CC)nocc1C(N1CC(C(=O)NC(C2(C(C)(F)F)CC2)=O)C1)=O C(=O)(C1=CCC(C)(C)CC1)N1CCN(C(c2c(C)oc(Cl)n2)=O)CC1C(C)C N1(C(c2cc(C)n(C)c2C)=O)CC2CN(C(=O)C(C)OCCC(C)C)CC2(C)C1 N1(C(c2c(OC)c(=O)cco2)=O)CC=C(CCNC(=O)CCC(C)SC)CC1 C1(C(=O)NCCN(C(=O)C(C)(C)F)C)OCC2CCCC1C2 C1(C(=O)NC(COC(C)(C)C)C(=O)OCC)(C(N(C(CC)C)CC)=O)CCOCC1 c1(C(=O)NC2C(OC)CN(C(c3c(C)nn(C)c3F)=O)C2)cccn2ccnc12 Cn1c(Cl)cnc1C(=O)NC1CCC(NC(=O)CCC2CC2(F)F)CC1 C(=O)(C(CC)C(C)C)N(CCOC)CCN(C(=O)CCC=CC(C)C)C(C)C C12(C(=O)NCCSCC(=O)NCC3CCCCCC3)CCCC(CO1)C2 c1(C(N2CCC(NC(CCCCC#C)=O)C(C(C)C)C2)=O)onc2c1CCCC2 c1(C(=O)NC2C(NC(C3OCC(C)(C)C3)=O)CCC2)c(Cl)cccc1[N+](=O)[O-] c1(C(=O)OCC)cc(NC(C2C3CC2N(Cc2ccc(C)o2)C3)=O)c(O)c(F)c1 N1(C(CCC=CCC=C)=O)CCC=CC1C(=O)NCCC(=C)C c1(CC)cc(NC(C2CCCCC2n2cc(CSCC)nn2)=O)c(C)nn1.C(C)(C)S C1(NC(Cc2[nH]c(=NCc3c(OC)cc(Cl)cc3)sc2)=O)C2CCC1CN(CC)C2 N1(C(C(CCN(C)C)NC(=O)Cc2cccn2C)=O)CCC2(CCCN2C)C1 C12(C(=O)NC3CC(CCNC(c4ccn(CCC)n4)=O)C3)CCC(CC1)C2(C)C CC(C)C(C(C)NC(=O)CN1C(=O)CNC1=O)NC(=O)Cc1cnns1 CCC(C)C(C(=O)N1CC=CCC1C(=O)NC)N(C)C(C1C=CCCC1CO)=O C1(C(=O)OCC)(C(=O)NCCCNC(=O)CC2CCCC2C)CCCC1 c1(CC(=O)NCC(CCC)NC(C2CC(CF)C2)=O)noc2ccccc12 N1(C(C2(C)CCC(C)CC2)=O)CCC(NC(=O)CC2CC2C)C(CO)CC1 C1(CCOC)(NC(C=COCC)=O)CCN(C(c2ccc(Cl)cn2)=O)C1 Cc1cncc(C=CC(N2CCN(C(C3COC3)=O)C(CC(C)(C)C)C2)=O)c1 CCCCC(CNC(=O)C(C)Sc1cccc(Cl)c1)NC(=O)C(C)(C)CN(C)C c1(NC(C2N(c3nc(SC)c(Br)cn3)CCC(O)C2)=O)cc(C#N)ccc1Br C1(C(=O)NCCCC(C)O)CCCC(NC(c2cccn2C)=O)CC1 N(C1CCc2c(F)cccc21)C(N1CC(C)C(c2ccc(Br)cc2)C1)=O Cn1cnnc1CC(=O)N(C1CC(NC(=O)COCC2CCOCC2)C1)C NS(=O)(=O)c1cc(C(N2CC3C(C2)N3C(=O)CC2CCCCC2)=O)c(O)cc1Cl c1(N(C(C2CCCC2NC(=O)CNC(=O)C(F)(F)F)=O)CC)ccc(Cl)cc1 C1(NC(=O)CCCNC(C2CCCO2)=O)CC2CC1N(C(c1ccc(Cl)[nH]1)=O)C2 C(=O)(C(CO)NC(=O)CC1CCCN1C(=O)CCNC(N)=O)N(C)C c1(CN(CC)CC)cc2cccnn2c1.C(=O)CC(N)C(C)C N1(C(C(COC)C)=O)CCC(CNC(c2ccc(C(C)=O)[nH]2)=O)(COC)CC1 C1(CNC(c2cccnc2O)=O)CCCN(C(=O)C(C2CCCCC2)O)CC1 N1(C2(Cc3cn(CCC=C)nn3)CC2)CCN(C(=O)CSCC(C)C)CC1 C1(N(C(Cc2scc(C)c2)=O)C)CN(C(=O)Cc2ccsc2C)CCC1C c1(NC(C2CC3CC3N2Cc2cc(O)c(O)c(Cl)c2)=O)nc2ccc(Br)cc2s1 CC(C)C(C(=O)NCC1CC1NC(C1(SCc2ccccc2)CC1)=O)N(C)C c1(C(=O)NC2CC(C(C)NC(CCc3onc(CC)n3)=O)C2)cnc(C)cn1 CC(C)C(F)C(=O)N1CCCCC1CCCNC(c1cnn(CC(F)F)c1)=O Cc1oc(S(C)(=O)=O)cc1C(=O)NC1COCCN(C(=O)C(F)(F)C(F)F)C1 c1(CCCNC(C2C(NC(=O)CNC(C3CCC3)=O)CC2)=O)ccccc1 Cc1cccc(C(N2CC3C(C(N4CCSC(C)CC4)=O)C3C2)=O)c1N N1(C(CCNC(C2(COC)CC2C)=O)=O)CCC(C)(O)C(O)C1 CC1CN2CCN1C(C(=O)NCC1(Nc3ncccn3)COC1)C2 C(=O)(C1CCCc2scnc21)N1C(C)C(NC(=O)CCc2ccc(F)cc2)CC1 N1(c2ccnc(C)n2)CCCCC(CNC(=O)CC(C)C)C1 C=CC1(C(N2CCC3(CC2)CC3)=O)CCN(C(=O)CNC(=O)C(C)(C)C)C1 C(C(C(=O)NCc1ccnc(Cl)c1)C(C)C)NC(c1c(CC)nccn1)=O C1(CC=C)(C(=O)NCC(F)CNC(c2ccoc2C2CC2)=O)CCCCC1 N1(C(C2C(CC)OCC2)=O)CC2CCCC(NC(c3cncnc3)=O)C2C1 CC1(CNC(=O)CCOCC(F)F)CC(F)(F)CN1C(c1cnc2[nH]ncc2c1)=O CC(C)(C)CCC(F)C(=O)N1CC2(CCC2NC(C2CCC3(CCC3)O2)=O)C1 S(=O)(=O)(c1c[nH]c(C(N2CCCC(CNC(=O)CNC(N)=O)CC2)=O)c1)NCC CCC(C)C(C)(c1nnnn1CCCF)NCCC1CCCC1(C)C Cc1n[nH]c(=NC2CC(F)(CNC(c3cc(C(F)(F)F)ncc3)=O)C2)s1 C1(CC)(CO)CCN(C(=O)C(C)(CNC(=O)CC2(C#N)CC2)CC)CC1 c1(C(=O)NCC2C(C)(C)N(C(C3CC(F)(F)CS3)=O)CC2)n[nH]c2c1COCC2 C1(C(=O)NC2CCC(NC(c3c(OCC)scc3)=O)C2)C2CCC1(C)C2(C)C C1(C(N2CCCC(CCO)C2)=O)CC2(CCC2)CN1C(C1CCCCC1)=O C(C)(C)(CCC(=O)NC1(CNC(C2CCCC(CC(=O)O)C2)=O)CCOC1)OC CP(C)(=O)C1CCCCC1C(=O)NCCCNC(=O)CCc1ccsc1 Cc1nc(Cl)ccc1CC(N1CC(N(C)C(C2CCCO2)=O)C2(CC2)C1)=O C1C(OC)CC(=O)N1.C1C(C)CN1CCCC.CCCCOC(C)=O Cc1ccc2c(c1)CC(C(=O)NCC(C)(CO)NC(=O)Cc1cc[nH]n1)O2 C(=O)(C(C)(C)CC(=O)N1CCCC1C(C)NC(=O)CNC(=O)C(C)CC)OC C1(CNC(C(C)C(F)F)=O)CC2CCC(C1)N2C(c1sc(N2CCCC2)nc1Cl)=O c1(C(N2CC(F)CC(NC(C3(CC#C)CCCO3)=O)C2)=O)cccc2sccc12 C(CO)(C(F)(F)F)N1C(=O)c2c[nH]nc2C1.C1(C(=O)NC2CC2)CCCCC1F c1(C(=O)NC(C(C)C)CCN(C)C(c2cn(C)cn2)=O)cn2cc[nH]c(=O)c2n1 C1(CC=C)(C(=O)NCc2cncc(C)c2)CCN(C(=O)CCC2CCCCO2)C1 c1(C(N(C(CC(=O)NC(C#C)C(C)OC)C)C)=O)nccc(C)c1N N1(C(c2c(CC)non2)=O)CC2CCC(C1)N(C(=O)CCCOC)C2 C1(C2(O)CCOC2)(C(=O)N(C2(CNC(CS(=O)(=O)NC(C)(C)C)=O)CC2)CC)CC1 CCCCCCCCC(=O)N1CC2(CCC2)CC1CNC(C1(COC)C=CCC1)=O C1(c2n(CC)ncc2)NC(=S)N(c2ccc([N+](=O)[O-])cn2)C2=C1C(=O)NC(CC)C2 C1(C(=O)NC(C2(CNC(=O)Cc3ccco3)CC2)C)(OC)CCCC(C)(C)C1 C1(NC(CCCOC)=O)CC(NC(=O)Cc2ccno2)CC1O S(=O)(=O)(c1ccc(N2CCCCC(O)C2)c(Br)c1)NCCC(=O)NCC c1(C(=O)OCCCS(=O)(=O)NC2CCCCC2)cc(Cl)ccc1C(F)(F)F C1(C(N2C(CN(C)C(C3(C)CSC3)=O)CC(F)C2)=O)CCn2nnnc2C1 C#CCC(CC(F)F)C(=O)N1CCCC(C(N2CCCC(CC)C2)=O)(CO)C1 N1(C(COCC)=O)CCOCC1CN(C)C(c1c[nH]nc1C1CCC1)=O N1(C(=O)CC2CCCOC2)CCC(C(N2CC=CC2CF)=O)C(O)C1 c1(C(N2CCCC(CCNC(c3nc(C)oc3)=O)C2)=O)cc(C(C)C)cnc1O C1(NC(C(C)(C)F)=O)CN(C(=O)CNC(c2ccccn2)=O)CC1C1CC1 C1(C(=O)NCC(CCCC)NC(C2(CC)COC2)=O)CC2(CC(C)=NO2)C1 C(=O)(C(C)C(O)C(C)C)N(C1CCN(C(=O)Cc2ccc(Cl)nc2)C1)CCC C1(C2CC2)(C(N2C(CC)CC2)=O)CN(C(c2cc[nH]c2C)=O)C1 c1(C(N2CCCN(C(CNS(C)(=O)=O)=O)CCC2)=O)cc2cc(Cl)cnc2[nH]1 N1(C(C#CC2(CC)CC2)=O)CCC2CCCC(C1)N2C(c1cncc2sccc12)=O N1(C(CC(C=C)O)=O)CCCC2(CCN(C(c3c[nH]nc3C)=O)C2)C1 N1(C(CN(c2ccccc2)C)=O)CCC2C(CCN2C(C2CCCS2(=O)=O)=O)C1 C1(CNC(c2c(C(C)C)occ2)=O)C(C)CCN1C(=O)C1=CCCC1 CCCC(C(=O)N(CCNC(C1CCC(=O)N(CC(F)(F)F)C1)=O)CC)C(C)C C(CC(C(=O)NC1CC2C=CC1C2)NC(=O)C=CC1CCCN1C)OC c1(CNC(c2c(OC)nc(C)cc2)=O)cc2nccnc2[nH]1 C1(NC(=O)Cc2ccnc(F)c2)CN(Cc2ccc(C(F)(F)F)nc2)CCC1(F)F N1(C(CC=C)=O)CC2C(C(=O)NCCCCC(N)=O)C2C1 C(=O)(CCCS(N)(=O)=O)N1C(SCC(=O)NC(c2n(C)ccn2)C2CC2)CCC1 CCC(C)CC(=O)C(=O)NCC(C)(C)C#CC(=O)NCc1cc(C)ccn1 c1(C(=O)NC(CNC(c2c(CC)ncnc2)=O)C2CC2)cc2ccc(C)cn2n1 N1(C(c2cc(OC)nc(C)c2)=O)CC2CCCN(C(c3coc(C4CC4)n3)=O)C2C1 N1(C(c2c(Cl)cn(C(C)(C)C)n2)=O)CCC2(CCCN(C(=O)C3=CCCC3)C2)C1 c1(OC)ccc2c(=NCC=C(C)C)[nH]c(N3CCCS(=O)(=O)CC3)nc2c1 N1(C(c2cc(C(C)C)no2)=O)CCN(C(C#N)C(C)C)CC1 c1(OC)ccc(C(=O)NC2CC2C(=O)NC(c2ccc(Cl)cc2)CO)cc1O c1(C(=O)NC(C2CCCN(C(c3[nH]cc(C)c3)=O)C2)C)cc2nc[nH]c2cc1N C1(CNC(c2n(CC)c(O)nc2)=O)CC(F)(F)CN1C(=O)CCc1cnn[nH]1 c1(OC)cccc(C(=O)NC2CCC(CC3CC4CC3CN4)CC2)n1 C(=O)(C1=NOC2(CCC2)C1)NC1CC2C(NC(C3(CC#C)CCCCO3)=O)C2C1 C1(CC(=O)NC(C2CCOC2)C)CCCN(C(=O)CCc2nccn2C)C1 C12(CNC(CC(CCC)C)=O)CN(C(c3cc(CF)on3)=O)CC1CS(=O)(=O)C2 c1(-c2cn(C(C)=O)nn2)ocnc1C(=O)N(CC(O)CN(c1sccc1C)C)C c1(C(=O)NC2C(N(C(CCOCCCOC)=O)C)CCC2)ccc(OC)cc1C N1(C(C(=O)OCC=C)C(C)C)CC(C(=O)Nc2ccsc2)OC(C)C1 C12(NC(CCc3ncc(C)[nH]3)=O)CCC(C1)N(C(C1C3COCC13)=O)C2 C1(C(=O)NCC(C)NC(=O)C(=O)NCCC(N)=O)CC(C)(C)C(C)(C)C1 Cc1ccc(C(=O)NC(CNC(C2(C(C)(F)F)CCC2)=O)C2CCC2)cc1C C(CCC(C)(c1nnnn1-c1ccccc1OC)NCC1CC1(C)C)OCC c1(C(=O)NCC(CC)NC(C2C(COC)C2(C)C)=O)cccc(OC)c1[N+](=O)[O-] C1(C(=O)NC(C(C)NC(Cc2c(C)nc[nH]2)=O)CO)CCN(C2CC2)CC1 CCC(C)C(CC(=O)N(C(C)CO)C)NC(=O)CN(c1ncccn1)C C1(NC(C(C)OCCOC)=O)CCCN(C(c2cc(C#N)on2)=O)C1C N1(C(c2nc(CC)sc2)=O)CC(NC(=O)CSCc2cccc(C)c2)CC(F)C1 C12(C(=O)NCCS(CC)=O)CC1CN(C(=O)CCN(CCO)CCO)C2 Cc1noc(C2CC2)c1C(=O)NC(C)CCCNC(=O)C(C)n1cncn1 N1(C(C(F)=CC)=O)CCC2(CCC(NC(c3sccc3SC)=O)C2)C1 Cc1ccc(O)c(CC(=O)NCC2CN(C(C3CC(O)(CO)C3)=O)CC2(C)C)c1 c1(C(=O)NC(C)CNC(c2c(C(F)(F)F)ncn2O)=O)ccc2nn[nH]c2c1 C=C(C)CC(C(=O)NCC1(CO)CCC1)NC(=O)CSC(F)(F)F c1(C(=O)NCC(C)NC(C2(CO)CCCO2)=O)cccc2ccnn12 C(=O)(C(CCC1CCCOC1)N(C1CCOCC1)CCOC)NCC=C N1(C(C(COC)OC)=O)CCN(C(=O)CCc2nc(O)n[nH]2)CC1CO c1(C(=O)NCC(CCCC)NC(C2(Cl)CC23CCC3)=O)ncc2[nH]ncc2n1 CC(C)S(=O)(=O)CCN=c1[nH]c(=NCCc2csc(=N)[nH]2)[nH]c2ccccc12 N1(C(C2CCCN(CC)C2)=O)CCC12CN(C(=O)C(C)(C)Oc1ccccc1)C2 C(=O)(C1=CS(=O)CCC1)NCC1(NC(CNC(c2ccc(C)cc2C)=O)=O)CCC1 CC1(C2CCN(C(C3CC4CC3CN(C(C3CCNC3=O)=O)C4)=O)CC2)CC1 c1(-c2c(OCC)cccc2F)cnc2[nH]cc(C(=O)Nc3nc(=O)o[nH]3)c2c1 CC1(C)CC(CNC(=O)Cc2cc(F)cc(F)c2)N(C(C2(CO)CCCO2)=O)C1 CP(C)(=O)c1ccc(C(N2CC3C(NC(=O)C(c4ccc(F)cc4)F)C3C2)=O)o1 Cc1cc(Br)cc(C)c1CC(=O)NC1CCCCN(Cc2ncccn2)C1 c1(C(N(C(C(=O)NC(C(=O)OC)C2(O)CCC2)C)C2CC2)=O)conc1C c1(C(=O)NCC(CC=C)NC(c2cnc3[nH]ncc3c2)=O)ccc2nonc2c1 Cc1nc(Cl)cc(=NCC(C)(CC(C)C)NC(=O)CN(c2ncccn2)C)[nH]1 c1(C(N2CCC(O)(C(C)NC(CS(CC)=O)=O)CC2)=O)cc(C)c(C)nc1O CCCC(C)(O)CC(=O)NCc1cn(CC(=O)NCCCCCCCO)nn1 c1(C(C)NC(C2(CNC(C3CC3Cl)=O)CC(=C)C2)=O)ccc(F)cc1 C1(C(N2CCCC(N(C(c3c(C)occ3)=O)C)CC2)=O)CCOC2(CCCC2)C1 C1(NC(=O)C=Cc2cscn2)CCCC(NC(C2(CF)CCC2)=O)C1 N1(c2nnccc2)CC(N=c2nc(N3CCC4(CCC4)CC3)c3c([nH]2)CSC3)C1 N1(C(CCOC)=O)CCC(C(=O)NCC(C)(F)C(C)C)C12CC2 C(=O)(CCN=c1ccc(C)c[nH]1)NC1CN(C(c2ccc(OC)nc2)=O)C(C)C1 c1(-n2cc(CNC(C3CCCS3(=O)=O)=O)nn2)cncc(C(=O)NCC2CC2)c1 c1(OC)ccc2c(C(=O)NCC3CCC3NC(C3CN(C(C)=O)C3)=O)cnn2c1 Cn1cc(CC(c2ccccc2)NC(c2cc(-c3cccnc3)n[nH]2)=O)cn1 c1(C(=O)NC(C=CC(=O)N(CCCOC)CCO)(C)C)cc(C)n(C)c1C Cc1ccccc1COC(C)C(=O)NC(C1CN(C(=O)CCc2cncs2)C1)C C1(CCNC(c2c(C)nc(C)o2)=O)CCCN(C(c2ccc(C(N)=O)[nH]2)=O)CC1 C(=O)(CCS(=O)(=O)Cc1ccccn1)NCC1(NC(c2cc(C)sn2)=O)CC1 CCCCC(C(=O)NCc1ccc(Cl)s1)N(C)Cc1cccs1 c1(C(N2CCC(NC(CCC=C)=O)C(C(C)C)C2)=O)nc2cnccc2s1 Cc1[nH][nH]c(=N)c1C(=O)NCc1cccc(NC(C2CC23CCC3)=O)c1 c1(C(N2C(CN(C)C(C3CCC(C)O3)=O)CC(F)C2)=O)cc(N)ccc1Cl C(=O)(C1SCCc2ccccc21)NCC(CNC(=O)CC(=O)Nc1nccs1)O Cc1ccc2c(N3CCN(CCO)CC3)nc(N(C)Cc3ccn(C)n3)nc2c1 c1(C(N2CCC(CNC(C3CC4CC4C3)=O)C23CC3)=O)ccc2ncccc2n1 N1(C(c2cc(C)c(O)cc2)=O)CC2CCC(C1)C2N=c1ccnc(Br)[nH]1 N1(C(CNC(C(CC)C)=O)=O)CCN(C(c2nccc3c[nH]nc23)=O)CCC1C C1(C(N2CC(CC=C)(NC(=O)C=CC3CCC3)C2)=O)CCC(=O)C(C)C1 C1(NC(c2cn(CC=C)nc2)=O)CN(C(c2occc2Cl)=O)CCC1CO N1(C(c2c(C)ccc(OC)n2)=O)CCCC12CCN(C(C1(C)CCNC1=O)=O)C2 C12(CNC(=O)CCC3CCCCO3)CC1CN(C(=O)Cc1cncnc1)C2 C1(CC)CC(C)CN(C(c2ccc(-n3cc(C(C)(C)C(N)=O)nn3)cc2F)=O)C1 C1(C(N2CCS(=O)(=O)CC2)=O)CCN(C(=O)C(c2ccc(F)cc2)F)C12CC2 Cn1c(O)ncc(C(=O)NC2CC3CN(C(=O)C#CC(=O)N(C)C)CC3C2)c1=O c1(CC)ccncc1C(N1CC(F)CC1CNC(=O)CN1CCCCC1)=O C1(NC(C2(O)CC(CF)C2)=O)CC(CNC(C2(CCO)CC2)=O)CC1O c1(C(=O)NC2CN(C(CCSC)=O)C(C)C2)nccc2[nH]nc(C(C)C)c12 C1(NC(COC2CC(C)(C)C2)=O)CCN(C(c2cn(C)c(=O)cn2)=O)C12CC2 c1(N(C)CCC2CC2)ccc(S(=O)(=O)NCC2CCCC(O)C2)c(Cl)c1 C=C(C)CCC(=O)NC1CCC1C(N1CCC(C(=O)Nc2ccccc2)CC1)=O C=CC1COCCN1C(=O)C(C(C)OC)NC(C1CN2CCC1C2)=O c1(CNC(C2(C)CCN(C(c3cncc(C)c3)=O)C2)=O)cnc(O)c(C)c1 C1(C(N(CC(C)N(C(c2cn(CCC)nn2)=O)C)C)=O)CC(OC)C(OC)C1 CC(C)CCC(C(=O)NC1CCC1)NC(c1cncc(Cl)c1)=O c1(C(=O)OC)c(N(C(C)=O)CC2CCCOC2)ncn1C.n12cc(nn1)[nH]c2=O C1(NC(CN(C(C(C)C)=O)C)=O)CC2(C1)CC(NC(=O)COCP(C)(C)=O)C2 C1(C(N(c2ccsc2)C)=O)CC1C1CN(C(C2CCCCS2)=O)C1 c1(C(=O)OC)c[nH]nc1S(=O)(=O)N1CCC(c2cccc(NC(C)=O)c2)CC1 N1(C(C(C2CCOCC2)C)=O)CC2(C(N3CC(CO)C(O)C3)=O)CC1CCO2 N1(C(C(C)c2cccs2)=O)CCOC2(CCN(C(C34CC(CO3)C4)=O)CC2)C1 C(=O)(CCCCCCN=[N+]=[N-])N1CCCC(N(C(c2ccnc(C)c2C)=O)C)C1 C1(C(C)NC(Cc2cc(C)[nH]n2)=O)CCCN(C(=O)Cc2ccsc2)C1 CCS(=O)(=O)CC(=O)N1CCN(C(=O)CC2(C#N)CCC2)C(C2CC2)C1 c1(COC)ccc(C(=O)N(C)CC2CN(C(=O)CC3CCCOC3)C2)cc1 N1(C(C(CC)n2cncn2)=O)CCC(F)(C(=O)NCCC(C)OC)CC1 C(=O)(C(Cc1cccs1)NC(C)=O)NCCC1(NC(C(C)OC)=O)CCC1 C1(N2CCC(NC(C(=O)NCCC(C)N3CCC3)=O)C2)CCN(C)CC1 N1(C(CN(C(c2cnn(C)c2N)=O)C2CC2)=O)CC2CCCC1C2CO N1(C(CC(C(C)OC)NC(C2CCCN2C)=O)=O)CC2(CCC(=O)NC2)C1 Cc1cc(C(N2CCC2CNC(=O)COc2c(C)nn(C)c2C)=O)nc(O)c1 C(=O)(CC(C)(C1CCC1)NC(c1cn(CC2CCCCC2)nn1)=O)OC N1(C(=O)CC2(O)CCOC2)CC2CN(C(C34CC=CCN3CCC4)=O)CC2C1 CC1(C)CC(NC(c2c[nH]c3cnccc23)=O)CCN(C(=O)C(O)CF)C1 C12(C(C=C(C)C(F)F)=O)CCCCC1N(C(C1(c3ccn(C)n3)CC1)=O)CC2 C(=O)(C1CCCc2sc(C)nc21)N1C(CNC(COCC)=O)C(C)(C)CCC1 C1(=O)C(C2CC2)NC(=O)N(NCCSC)CC(=O)N1.c1(C)cccs1 c1(C(N2CC3CCC(CNC(COC(C)=O)=O)(C2)C3)=O)cc2c(C)cccc2[nH]1 C(c1cccc(F)c1)=CC(=O)NC(C1CCOC1)CNC(c1nc(C(C)=O)sc1)=O C1(NC(CCSCC(C)C)=O)CCC(C)N(C(c2cccc(F)c2C(F)F)=O)C1 c1(CNC(C)=O)ccc(C(N2CCC(CNC(=O)CC3CC34CC4)C2)=O)c(F)c1 N1(C(C23CCC(CC2)CC3)=O)CCC(c2ccccc2)C(CO)C1 Cc1cccnc1C=CC(N1CC(N(C(=O)COCCN(C)C)C)C(F)C1)=O C1(C(=O)NCCc2ncon2)CC2CCC1N(C(=O)C(O)CC(=O)O)C2 n1(CCC(N2CC3(CN(C(C4C(=C)C4)=O)C3)C2)=O)c(C2CC2)nc2ccccc12 C12(NC(c3cccc(Cl)c3Cl)=O)CN(C(=O)CCCCNCC)CC1CS(=O)(=O)C2 C1(CC)CN(C(c2ccn(C(C)C)n2)=O)CCC1NC(c1ncncc1F)=O N1(C(C2N(CCC)C(=O)CC2)=O)CC2(CCN(C(c3ccc(F)n3C)=O)CC2)C1 c1(C(=O)NC2CC(NC(C3CCN(C)C3)=O)C2)ccnc2ncccc12 c1(OC)cc([N+](=O)[O-])cc(Br)c1CNC(c1cc(OC)c(O)c(I)c1)=O C1(N(C(C2CCN(C(C)=O)CC2)=O)CC)CC(NC(=O)C(F)(F)CO)C12CCC2 c12cnn(C)c1C(=O)NC2.C1(C)(C(=O)OC)CC(NC(=O)CC2(C)CC2(F)Cl)C1 N1(C(C2CCCS2(=O)=O)=O)CCCN(C(C23CC(C(F)(F)F)(C2)C3)=O)CC1 N1(C(CCC=C=C)=O)CCC(F)(CNC(=O)C(c2ccc(OCCC)cc2)=O)CC1 N1(CCC(=O)NCC2CC(CNC(c3csc(CO)n3)=O)CO2)CCCS1(=O)=O c1(NC)cnc(C(=O)NC(Cc2cn[nH]c2)C(=O)N(C2CCC(F)(F)C2)C)cn1 C1(NC(CCN(C(C)=O)C)=O)CN(C(=O)CNC(=O)CC2CCCCC2)CC1O c1(C(=O)NC2CCN(C(C(CCC(C)C)=O)=O)C2)cnn2c1S(=O)(=O)NCC2 S(=O)(=O)(c1ccccc1Cl)N1C(C)(C)CC(O)C1 Cc1ccc(CC(N2CC(CN(C(=O)C(C)N3CCC3)C)C3(CC3)C2)=O)cc1C C1(C(=O)NC2C(NC(c3c(C)nsc3)=O)C2)Cc2cccc(F)c2O1 CC1=C(C(=O)NC(CCC2CC2)C(=O)NCC(C)(O)C2CCC2)CCCO1 N1(C(c2nc(C(=O)OC)oc2)=O)CCC(C)(C(=O)NC2C=CCCCC2)C1 C(c1cccc(F)c1F)=CC(=O)NC(CC)CNC(c1cc(Cl)cnc1O)=O C(C(=O)N(CCC(=O)NCC1OC2CCC1C2)OC)OCC C1(NC(c2ccc(C)s2)=O)CC2(C(=O)NC(c3n[nH]c(C)n3)C)COC1C2 C#Cc1cnn(CC(N2CC(C(=O)N(C)Cc3cn(C)cn3)(CC)C2)=O)c1 c1(C(=O)NCCCC(C)NC(C2CCN(C)C2=O)=O)ccnc(C(C)(F)F)c1 c1(C(C(=O)NC2CCOC2)N(C(c2ccccc2)C)C)cc2n(n1)CCCC2 N1(C(C(C)CO)=O)CC2CCN(C(=O)CC(C)(O)C(F)(F)F)C2C1C Cc1c(C(N2CC3CC2C3C(=O)Nc2ccc(Cl)cc2)=O)cccc1O N1(C(C(CC#C)O)=O)CC2CCN(C(=O)CCN3CCN(C)CC3)CC12 c1(C(N2CCCC(CN(C(c3c(C)nc(C)o3)=O)C)C2)=O)ccc2occc2n1 C=CC1(C(=O)NCC(CC)N(C(=O)CCc2nnc(C3CC3)o2)C)CCCCC1 C12(C(N3CCCC(NC(=O)CC4CCSC4)C3)=O)CCCC1C2(F)F C1(NC(CC2(CC=C)CCCC2)=O)CC(F)CN(C(=O)C(C)(C)NS(C)(=O)=O)C1 C1(C(N2CCCC(CNC(c3ccc(F)cc3F)=O)C2)=O)CC12CCCCCC2 C1(CC)CN(C(=O)CC2CC(C)(C)CO2)CCN1C(C1CCC(=C2CCC2)CC1)=O c1(C(N(C(CC)CNC(=O)CC(C)(C)C2CC2)C)=O)ccc(C)cc1C CC1CN(C(=O)CCC2CCN(C)CC2)C(C)CCO1 c1(C(=O)NC(CNC(C(F)=C(C)C)=O)CO)oc(-c2ccccc2)nc1C C1(CNC(C(C(C)C)F)=O)CCN(C(c2ccc(C3CCCO3)[nH]2)=O)C1(C)C C1(CC=C)(NC(=O)CC(C)(C)OC)CCCN(C(=O)C(C)OC)C1 c1(C(N2CCC(C(=O)NCC(C)C3CC3)C2(C)C)=O)cccc2[nH]ncc12 N1(CC)CC(C(=O)N(C2CCN(C(=O)CC3CNC(=O)C3)CC2)CCO)CC1=O C(N=c1nc(C2CC2)[nH]s1)C1(F)CC(NC(CCOCC)=O)C1 C1(C(=O)NCC2C(C)(C)CN(C(c3ccncc3Br)=O)C2)CCOC2(CCC2)C1 CC12CC(C(=O)NOCC(=O)NCc3cccc(CO)c3)(CCO1)C2 C(=O)(C(C(C)(F)F)c1ccccc1)N(CCNC(C1CC(CCC)C1)=O)CCC Cc1cc(C(=O)NC(C(=O)NCC2COC(=O)N2)C2(C)CC2)c(C)s1 c1(CC(=O)NC2C(NC(CN3C(C)CCC3)=O)CCC2)cc(Cl)ccc1[N+](=O)[O-] c1(C(=O)NC(C2CCN(C(C3CNC(=O)N3)=O)C2)C)nnc2ccccc2n1 Cc1ccc(N2CCCC2C(=O)NCC(C)CF)cc1 N1(C(C2C3CN(C(c4ccnc(O)c4)=O)C2C3)=O)CCC2(CC1)COC2 N1(C(C2CCN(C)CC2)=O)CC2CC(NCCNC(c3ccc(CO)s3)=O)C1C2 c1(CC(=O)NCC2C(NC(c3c(SC)cn(C)n3)=O)C2)oc2ccccc2c1C c1(NC(CCC#C)=O)ncnc(N(C)C)c1[N+](=O)[O-].C123CC1CN(C2)C3 CC1C(C)N(C(=O)Cc2c[nH]ccc2=O)CCN1C(=O)CCc1cn[nH]c1 c1(C(=O)NCC(C)N(C(CC2(NC(C)=O)CCCCC2)=O)C)c(C)cccc1N n1(CC)ncn(NC(=O)C23CC2CCN3C(=O)OC(C)(C)C)c1=O C1(N(CC(C)C)CCC)CCC(C)N(C(=O)Nc2nc[nH]n2)C1 c1(OC)ncncc1NC(C1CCN(C(c2n[nH]c(C)c2C)=O)CC1)=O N1(C(c2cnc(OCC)s2)=O)CCOCC1CNC(C1(C(F)(F)F)CC1)=O C1(C(=O)NCCN(C(C(CC)n2nccc2C)=O)C)CC(C)(C)SC(C)(C)C1 C1(NC(COC(CC)C)=O)C2CCC1N(C(c1cc(C(F)F)cs1)=O)C2 Cc1nc2cnn(C)c2cc1C(=O)NCC1CCCN1C(=O)C(CO)N(C)C c1(CC(=O)NCC2COCCN2C)ccc(C)c(O)c1.C12(COC)CN(C1)C2=O c1(C(N2CCC(N(CCC)C(C3CC(F)(F)C3)=O)C2)=O)c[nH]c2ncccc12 c1(C(N(C(c2ccc(Cl)cc2)CNC2CC2)C)=O)cc(Cl)ccc1OCC(F)F c1(C(N2CCOCC2c2nc[nH]n2)C(=O)NCCCC)n[nH]c(C)c1C CC(O)CCCCCC(=O)N(C1CCN(C(C2CC2C)=O)CC1)CCO O=C(CCCCN1CCCC1)NCC1CN(C(c2cccc(CCO)c2)=O)C1 C1(C)(C(N2C(CC#C)CCCC2)=O)CC(O)CN1C(=O)CC1(OC)CCCCC1 C(=O)(CC(C)C(F)(F)F)N(CCCCC(=O)NC1CC(C)(CC)OCC1)C N1(C(CCC=CC)=O)CC(NC(c2cncc(C(C)C)c2)=O)C(CC(C)(C)C)C1 c1(OC)ccc2cc(C(N3CC(NC(=O)C=CCO)CC(F)C3)=O)cnc2c1 C12(C(=O)NCCC3N(C(C(C)SC)=O)CCCC3C)CCC(N(C)C)(CC1)CC2 N1(C(=O)OC)CCCC(C(=O)NC2COCC2NC(c2cc(CO)n(C)n2)=O)C1 Cc1ccc(S(N)(=O)=O)c(C(=O)NCCC(C)NC(=O)C(O)C(C)C)c1 C1(CNC(C2CC2(F)F)=O)CCCCN1C(=O)C(c1cccc(F)c1)=O c1(C(N2CC(NC(C3CC(CF)C3)=O)CC(O)C2)=O)onc2ccccc12 C1(c2cn(CCOC)nn2)CN(C(c2cc(C)c[nH]2)=O)CCO1.C(C)(=O)O CC(CC(F)F)C(=O)NCC1CC1NC(c1cnc(-c2ccccc2)nc1)=O CCC(CC(=O)N1CCC(C)N(C(c2ccc(OC)nn2)=O)CC1)C(C)C Cc1ccnc(C(=O)Nc2c[nH]nc2C2CCN(C(=O)CCN3CCC3)CC2)n1 c1(C(=O)NCC(CN(C)C(C2CC3(CCC3)C2)=O)O)nc(=O)n(C)[nH]1 N1(C(CSCCCC)=O)CC2CN(C(=O)C=Cc3cccc(CO)c3)CC2(C)C1 c1(CC)ccc(C(c2nnnn2-c2ccc(F)cc2)NC2CC23CCC3)nc1 Cc1c(Cl)ccc2c1CN(C(c1nnn3c1CSCC3)=O)CC2 C1(C(=O)Nc2cnccc2C)(CC)CCN(C(=O)Cc2cc[nH]n2)CC1 Cc1cc(C)c([N+](=O)[O-])cc1C(=O)NC(CNC(c1cc[nH]n1)=O)C(C)(C)C c1(C(C)C)cccc(C(N2CCCC(CNC(=O)CNS(=O)(=O)C3CC3)C2)=O)n1 CC1COCCC1N(C)C(C1CC(F)CN1C(=O)CC1CC2C=CC1C2)=O c1(C(=O)NC(CCNC(CCC=CC(C)C)=O)C)cc(F)c(F)c(F)c1 CCCC(CC1CCCCC1)C(=O)NC1C2CC1CN(C(C1CCSCC1)=O)C2 N1(C(c2ncc(OC)cn2)=O)CC2CCC1CC2NC(c1c[nH]nc1C(C)C)=O CC1(C)CCc2c1n[nH]c2C(=O)NCCC1(O)CCN(C(C2C=CCCC2)=O)C1 N1(C(C(c2ccc(Cl)cc2)CC)=O)CCCN(C(C2CCC3(CCC3)O2)=O)CC1 C1(CN(C)C(C2CCN(C(N)=O)C2)=O)CCN(c2nnc(C(C)(C)C)o2)CC1 c1(C(=O)NCC(C)NC(C2CCN(CC(C)C)C2)=O)cncc(Cl)c1 CCC(CC)(CO)C(=O)NCCC1(O)CCN(C(c2sc(=N)[nH]c2C)=O)C1 N1(C(c2cc(C#N)c(Cl)cc2)=O)CC(NC(=O)CCC2CC2)C2(CCCC2)C1 C(=O)(C1=NOC2(CCC2)C1)NCCCOCCC(N1CCCC(C)(O)C1)=O Cc1ccc(C)c(S(=O)(=O)N2CC(NCc3cc(F)c(Br)cc3C)C(C(=O)O)C2)c1 Cc1cccc(-c2cn(C3CCCN(C(=O)C(C)CC(N)=O)C3)nn2)c1F c1(CN(C)C(c2ncc[nH]2)=O)cc([N+](=O)[O-])ccc1Cl N1(C(C(C)CCC(C)(C)C)=O)CCCc2cc(Cl)cnc21 N1(C(Cc2ccn(C)n2)=O)CC2(CC(CNC(=O)CC3CC(C4CC4)C3)C2)C1 C1(CNC(CC=CCC)=O)CCCC1NC(c1ccnn1Cc1ccccc1)=O CC1CCC(C)(NC(C2CC(O)CN2C(=O)C(F)F)=O)C1 N1(C(c2cc(CO)ccn2)=O)CCC2CCN(C(C3(C(F)(F)F)CC3)=O)CC2C1 C(CCCC(=O)NCC(C)(O)CNC(c1cccc(N(C)C)c1)=O)N(C(C)=O)C C1(NC(C2CC(CF)C2)=O)CC2CCC1C2.CC1(C)C(=O)N2C1CCC2 N1(C(CC2CC(=O)C2)=O)CC(NC(=O)CC2CC=CCC2)Cc2ccccc21 C1(CNC(=O)C(N2CCCC2CC(F)(F)F)C2CCSC2)CCC(F)(F)CC1 N1(C(=O)COCCF)CCC(CC2COCCN2C(=O)Cc2ccco2)CC1 C(C(C(=O)NCC(O)C1(C)CC1)NC(N)=O)OC(C)(C)C C12(C(N3CCC(N(C(=O)CCOc4ccccc4)C)C3)=O)CCC(C)(C1)OC2 N1(C(C2CCCN2Cc2cnc(-c3cccnc3)s2)=O)CCS(=O)(=O)CC1 O=C(CCCCN(C)C)NCc1cc(C(=O)NCC2CC2[N+](=O)[O-])co1 C1(O)(CN(C(c2c(C)cns2)=O)C)CCCN(C(c2nnc(C(F)(F)F)s2)=O)C1 C12(C(N(C)CCO)=O)C3CC1C1C(C(=O)Nc4ccc(C(=O)O)cc4)C3C21 N1(CNC(C(C2CC(CC)C2)N(C)C(C2CC2)C)=O)CCOCC1.CCO N1(C(CCCC=C)=O)CCN(C(=O)C(c2ccc(F)cc2)C)CCC1C C1(COC)(NC(=O)Cc2ccccc2Br)CCCN(C(=O)CCP(C)(C)=O)C1 c1(CN(C(=O)NCc2c(C)ncnc2)C)cccc2ncccc12 C(=O)(C(O)C1=CCCCC1)N1CC(CC(=O)N(CC(F)F)CCF)(OC)C1 N1(C(CCC(=C)C)=O)CCC(C)N(C(=O)Cc2ccc(C)cc2)CC1 c1(OC)cc(C)ccc1OCC(=O)NC1CC1NC(=O)C1=CSCS1 C1(=O)CC(CC2CC2)N1.C(=O)(C(C)CC1CC1)NCC(=O)OCC=C CCC(CC)C(C(=O)NC(C)CNC(=O)Cn1nccc1C(F)(F)F)OC C1(CC(=O)NC(C2(O)CN(C(c3cnn(CC(F)F)n3)=O)C2)C)CCC(C2CC2)O1 C=CC(CCC)CC(=O)NCCCCC(C)(C)NC(C1CCCN1S(C)(=O)=O)=O C(=O)(C(CC(C)(C)C)NC(=O)C(=O)NOC)NC1CCN(CC)CC1 N(C(=NCc1ccco1)N1CCC(OCC)C1)Cc1cccc(CC)c1 c1(C(C(=O)Nc2c(C)cccc2)N(C)Cc2ccon2)cccc2c1CCC2 C(=O)(C(CC(C)C)NC(=O)C(F)C1CC(NC(C2CC(C)CCO2)=O)C1)NC CCCC(C(=O)N(C(C)CCNC(c1sccc1S(N)(=O)=O)=O)C)C(C)C CC1CCn2cc(C(N3CCC(CF)(NC(C4CC(Cl)(Cl)C4)=O)C3)=O)nc2C1 C1(C(N2CCC(OCC#C)C2)=O)CCN(C(=O)Cn2cccn2)O1 Cc1cc(C(N2CCOCC2CC(=O)NC(CN(C)C)C(C)C)=O)nnc1C c1(C(=O)NCC2N(C(CCCCC=C)=O)CCOC2)cccc2nn(C)cc12 N1(C(C=CCOC)=O)CCC(CNC(C2CC(=O)NC(=O)C2)=O)C1(C)C C=C1Cn2c(C(N3CCN(C(c4ccoc4Cl)=O)CC3C)=O)nnc2S1 S(=O)(=O)(c1c[nH]ccc1=NCCCCCF)N(CCC(C)(C)C)C CC1CCN(C(=O)CC(C)(F)F)CC1NC(c1ccc(OC(F)F)c(Cl)c1)=O c1(CC)ccc(C(=O)NC2CC(C)(NC(c3ccn(CCF)n3)=O)C2)cc1Br N1(C(c2ccc(C)c(O)n2)=O)CCCN(C(=O)Cn2ncccc2=O)C(C)C1 C1(C(C)NC(c2cc(OC)n[nH]2)=O)CN(C(c2cc(CO)c(C)o2)=O)CCO1 CCC(C)(C(=O)NC(C(=O)NC)C1CC1)OC.c12ccc(o1)c(=O)[nH]2 N1(C(C2C(C)CCC2)=O)CC2(CCCN(C(C3(C(F)(F)F)CC3)=O)C2)C1 C1(C)(C(N(CCNC(C2(CCOCC)CCC2)=O)C)=O)COC(C)(C)CO1 Cc1c(O)c(=O)ccn1C(c1ccc(I)cc1Cl)=O C1(C(=O)NC2CC(C)N(C(c3ccccc3O)=O)C2)CC2CCC1CC2 C12(C(=O)NC3(C)CC(NC(=O)C(F)(F)c4cccnc4)C3)CCCC1CC2 C(=O)(C(O)CCn1cncn1)N1CC(O)(C(C)NC(=O)COCC2CCC2)C1 C1(CC=C)(NC(C2(C3CCCO3)CC2)=O)CCN(C(c2cnccc2C)=O)C1 c1(COC)ccsc1C(N1CCC(C(C)NC(c2ccnn2CCOC)=O)C1)=O c1(SCCC(=O)NC2C(NC(c3c(C)nsc3)=O)CCC2)ccc(F)cc1 n1(CC)cc(CCC)nn1.C(C(=O)NCCOCC)(C1CC1)NC(N)=O.COC C(CCCCCCS(C)(=O)=O)NC(=O)NC1CN(c2cn(C)nc2)C(=O)CC1 C1(CC)(NC(=O)CC2(CC(=O)OC)CC2)CCN(C(=O)C=Cc2sccc2C)CC1 c1(C(N2CC=CC(NC(C=CCCC)=O)C2)=O)nc2nc(C)cc(C)n2n1 c1(C(N2CCC(N(C(=O)CSC3CC3)CC)C2)=O)cc2c(nc1N)CCCC2 c1(C(=O)NC(CC(C)NC(C(C)=C(CC)C)=O)C)cccc(Br)c1OC c1(CC(=O)OCC)cccc(CC)c1.c12cnn(c1CC)C13CC(C1)(C3)NC2=O CC(C)C(O)Cc1cn(C2CN(C(=O)C(C)C)C2)nn1 CCC(C)C(C(=O)OC)NC(C)=O.n12cc(nn1)C(C)(C)NC1CC(C1)C2 C12(C(=O)NCCCc3cc(C)no3)COC(C1)C(NC(c1ccn(C)c1C)=O)C2 c1(OC)c(C(=O)NC2CCN(C(c3[nH]cnc3C)=O)C2(C)C)cccc1C(F)F c1(C(=O)NC(c2oc(C(=O)OCC)c(C)n2)C)cc(C)c(Cl)cc1Cl c1(CN(C(C2(F)CCN(Cc3c[nH]ccc3=N)CC2)=O)CC)ccc(O)cc1O c1(NCCNC(CCSCC)=O)ccc(NC(=O)CC(C)F)nc1 c1(C(N2CCC(CC(N3CC(CO)C(F)C3)=O)C2)=O)ccc(Cl)cn1 Cc1nc(CC(=O)NCC(C)CNC(C2CC(=C(F)F)C2)=O)[nH]c1C C(c1ccc2c(c1)CCO2)=CC(=O)NCC1CCN1C(c1coc(Br)n1)=O C(=O)(C(F)(CNC(=O)Cn1[nH]cnc1=N)C(C)C)Nc1ccc(OC)c(F)c1 N1(C(C=C(COC)C)=O)CC(C(F)(F)F)OC(CNC(c2cncc(Cl)c2)=O)C1 N1(C(=O)OC(C)(C)C)CC2(C)CN(C(C3(C)CCC3)=O)CC2(C)C1.C12=CC(C1)C2 c1(CCC)cccc(C(=O)NC2CCC(C(=O)N(CC(F)F)C)C2)c1 C1(CNC(C2(C)CCSCC2)=O)C2CCCC1N(C(c1ccc(N)c(N)c1)=O)C2 N1(c2nc(CC)cc(CC)n2)CCC2C(CCCN2C(C2CCCN2C=O)=O)C1 N1(C(C(C)(C)OC)=O)CC2CCC1CN2C(c1sccc1CCOC)=O CCCN=C(NCCC1CCCOC1)NC(c1ccc(OCC2CC2)cc1)C N(C1CN(C(=O)CC2CCC(O)C2)CCc2ccccc21)C(C1CCCCO1)=O N1(C(c2c(C)coc2C(C)(C)C)=O)CC(CNC(=O)C(C)(O)C(C)C)CC1(C)C c1(C(C(=O)OCC(CC(=O)OC)C)(F)F)nc2ccccc2s1 C1(N(C(=O)C=CCF)C)CCC(NC(C2CC(C)(O)C2)=O)C1 N1(C(C2CCCN(C(C)C)C2)=O)CCC(C)C(NC(=O)C2=CCCCO2)C1C c1(CC(N2CCC(CNC(CC=CC)=O)C23CC3)=O)ccc2c(c1)CC(C)O2 c1(NC(C2(C)N(C(C(C)=O)=O)CCC2)=O)ccc2c(C)n(C)nc2c1 C(CCCCC(=O)NCCC1CN(C(=O)CSCC(C)C)CC1C)OC c1(C(=O)NC(CNC(C(C)OCC)=O)C(C)(C)C)cc(C)ccc1F c1(C(=O)NC(CC)CNC(c2cncn(C)c2=O)=O)noc2c1CC(C)(C)CC2 C1(O)(CNC(=O)Cc2cnccn2)CCCN(C(c2cc3[nH]ccc3s2)=O)C1 c1(OC)cc(Cl)c(C(N2CCN(C(C3CC(O)C3)=O)CC2CF)=O)cc1Cl C(=O)(CCC(=O)N1CCC(F)(CNC(c2cc(OC)ccn2)=O)C1)NC CC1=C(C(=O)N2CCCC(CO)(NC(c3cc(Cl)cc(F)c3F)=O)C2)CCCC1 N1(C(C2CCC(=O)O2)=O)CCOCC1CCNC(C1(CO)CCOCC1)=O c1(OC)cc([N+](=O)[O-])c(OC)cc1C(=O)NCC1(O)CN(C(C2COC2)=O)C1 C1(CCC)CN(C(C2CC2CC)=O)CCN1C(=O)CC(O)C1CCC1 C1(NC(C(C)OCCOC)=O)CC2CC(NC(=O)Cc3cc(F)ccc3Cl)C2C1 O=C1CCC(C(=O)N2CC3C(CCNC(CC(N4CCOCC4)=O)=O)C3C2)=NN1 C1(NC(c2c(C(C)C)n[nH]c2)=O)CN(C(=O)Cc2ccc(O)c(O)c2)CC1(C)C N1(C(=O)OC(C)(C)C)CCCC(O)(CNC(C2(C(=O)O)CC3CC3C2)=O)C1 Cc1nc2nc(=S)[nH]n2c(C)c1CCC(=O)NCCC(C)NC(C1CC1CF)=O N1(C(COCCCC)=O)CCC2CC12C(N1CCN(C2CC2)CC1)=O c1(OC)ccccc1C(C(=O)NCC(C1CCC1)NC(c1cc(Cl)no1)=O)OC N1(C(c2c(N)nccn2)=O)CC(NC(c2cccc(OC(F)F)c2)=O)CC(O)C1 c1(CN2CCC(NS(CC(=O)OC)(=O)=O)C(C)(C)C2)ccc2ccncc2c1 c1(CC)ccoc1C(=O)NC1COCC1NC(c1coc(SC)c1)=O N1(C(C2(C)CC(F)(F)C2)=O)CC(NC(c2ccc(N3CCC3)cc2)=O)C2(CC2)C1 Cc1[nH]nc(C(=O)NC2CN(C(=O)C=Cc3cnccn3)C3CC23)c1C N1(C(C(CC)(C)COC)=O)CCC(C)(C)C(C(N2CCCCCCCC2)=O)C1 C(=O)(CCCC(=O)NC1CCN(C(c2cc(C(F)(F)F)cn2C)=O)C1)NCCC C(C(=O)N1CC(F)(F)CC1)(C(C)CC)NC(CC(C=C)C)=O N1(C(CCc2cc(C)nn2C)=O)CCCC(F)(CNC(=O)C2=C(Cl)CC2)C1 C1CCN2CCC1NC(=O)CCC2=O.C1(CCN(C)C)(COC)CC1 C1(C(N(CCOCC)CCOC)=O)CCC2CCC1N2C(=O)CC1CCC(=O)N1C CCC(N=c1[nH]c(N2CCc3ccccc3CC2)nc(=N)[nH]1)c1cccnc1 c1(C(C(N2CCC(F)(Cn3cc(C4CC4)nn3)C2)=O)O)ccc(F)c([N+](=O)[O-])c1 c1(C(N2CC(N(C(c3ccc(C)s3)=O)C)C(F)C2)=O)cc2cc(Cl)ccc2n1C c1(C(=O)NCCN(C(C)C)C(c2cc(CC3CCC3)c[nH]2)=O)ccnc(F)c1N c1(OC)cnc(C(=O)NC(C2(O)CN(C(C3(CF)CCNC3=O)=O)C2)C)c(F)c1 C1(NC(c2c(C)onc2C(F)(F)F)=O)CCN(C(c2cnoc2C)=O)C(C)C1 C1(C(=O)NCC2CCCN(CC)C2)CC(F)(F)CN1C(=O)C(CC)OC N1(C(=O)CSn2cc([N+](=O)[O-])cn2)CC2CCC1C1CNCC21 N1(CCCCC)CC(F)(F)CC1C(=O)NCc1cnc(C(=O)OCC)cn1 C1(C(N2C(C)C(NC(c3cn[nH]c3)=O)CCC2)=O)CC2C=CCC(C1)C2 c1(CC)cccc(NC(C2CC2CNC(c2cncc(F)c2)=O)=O)c1 c1(C(=O)NC2C3CN(C(Cn4ccc(=N)[nH]4)=O)CC32)cnc2[nH]nnc2c1 N1(C(CNS(N)(=O)=O)=O)CCC(C2CCCN(C(c3cccc(F)c3F)=O)C2)C1 c1(OC)ccc(CC(N2CCC(NC(=O)CCC3CC(F)(F)C3)CC2)=O)cc1 c1(OC)ccn2c(C(=O)NCCC(C)(C)NC(=O)CCNC(N)=O)cnc2c1 c1(SCC(=O)N(CC(C)NC(c2nc(C(C)(C)C)no2)=O)C)cnn(C)c1 C1(C(C)C)CC(C(=O)NCC2(NC(c3cnc(C(C)C)[nH]3)=O)CCC2)CCO1 CCCC(C)C(=O)N1CCC(OCCN)CC1.C(=O)(C(=O)NC)C(=O)Cc1cnco1 N1(C(c2cc(CCC)ncc2)=O)CCC(NC(C2CCC2C(F)(F)F)=O)C(F)C1 c1(CC(=O)NCC=CCNC(=O)CCn2cncn2)ccccc1Cl C(=O)(C1=CC2C=CC(C1)C2)NC(C(=O)Nc1ccc(OC)c(C)c1)C(C)(C)C C(=O)(C(C)(C)CC(=O)OC)NCC1C(NC(CNS(CCCC)(=O)=O)=O)CC1 C(=O)(CC(CNC(=O)Cc1nocc1C)C1CCC1)N1C(C(=O)OC)CCC1 Cc1c(Br)sc(NC(=O)C(N2CCCC2C(c2ccccc2)O)=O)c1C Cc1ncc(C(N2CCC(C(=O)NC3(CO)CC3(C)C)CC2(C)C)=O)cc1C#N C12(C(N3C(COC)C(C)(C)C3)=O)CCC(CC1)N(C(c1cnoc1)=O)C2 C1(N(C(=O)C(C)C2CCC2)CC#C)CCN(C(C2CCS(=O)(=O)N2)=O)CC1 C(=O)(C1=C(c2ccccc2)CCC1)N1C2CC(NC(=O)CC3CC3)C(C)C1CC2 c1(C(N2CCC(C(=O)NCc3n(CCC)ncn3)C2)=O)cc(C)ccc1F O=C1CC(C(=O)NCc2ccc(C(=O)NC(CO)CCCF)nc2)CCN1 O=C1CN(CC(=O)NCC(O)C(=O)NC2CNC(=O)OC2)CCN1 C#CCCN=C(NCc1ccccc1SC)NCC1OCCC1(C)C C(CCCCCN=c1cc(NCc2ccc(-n3ccnc3)cn2)nc[nH]1)N(C)C n1(CC)ncc(C(N2CCC(c3n[nH]cc3CNC(=O)CC(CC)OC)C2)=O)c1C C=C=CC(C)C(=O)N1CCN(CC(C)(C)NC(=O)C(C)C(C)C)CC1 C=C1CC(C(N2CCC(c3ccc(Br)cc3)C2)=O)N(CC2(N(C)C)CCC2)C1 C1(CNC(C2(C3(C)CC3)CC2)=O)C2CC1N(C(=O)CN1CCOCC1=O)C2 c1(COCCNC(N2CCCC(OC(C)=O)C2)=O)cc(C)ccc1F c1(C(N2C(C(N(CCN3CCCC3)CC)=O)C(C)(C)CC2)=O)ccc(C)nc1C c1(-c2c(C(=O)Nc3ccc(F)cc3C(F)(F)F)ccnc2)ccc([N+](=O)[O-])cc1 CS(C)(=O)=NC(=O)C(=O)NCC1CC(F)CN1C(c1nc(Cl)sc1Cl)=O C=CCC(CC(C)C)C(=O)NC(c1nocc1C(N1CCOC(C2CC2)C1)=O)CC C1(C2CN(C(c3csc4nccn34)=O)C2)(NC(C(C)c2ccsc2)=O)CC1 C1(SC)CN(C(C2ON=C(C)C2C)=O)CC1NC(C1CC(=O)N(CCC(C)C)C1)=O c1(CNC(N2CCC(COC)CC2)=O)csc2nccn12 c1(C(=O)NCC(=O)NC2C(CNC(CC3(CC)CCCC3)=O)C2)cc(C)nn1C N1(C(CCN(C(C2N(CC)CCOC2)=O)C)=O)CCCC(C)(C)CC1 C(CC(C(C)(C)C)NC(=O)CCCCCSC)N(C(C1(CC)CCCC1O)=O)C CCCC(C)CC(=O)N1CCC(CNC(=O)CN2CCCCC2=O)(OC)C1 C1(C(=O)NC2CCC(NC(C3C(C=C(C)C)C3(C)C)=O)CC2)CCCS(=O)(=O)C1 N1(C(CC2CCC(C)(C)O2)=O)CC(C(N2CCC(C)(C)C2)=O)C2(CC2)C1 c1(C(=O)NC(C(C)NC(C2(CC)CCCC2)=O)C)ccc2occc2c1 C1(NC(CC2CN(C(C)=O)C2)=O)CCC(CCN(C(=O)C(C)n2cncn2)C2CC2)C1 C12(NC(c3ccc(NC4CCC4)nc3)=O)CCCC1N(C(=O)COC(F)F)CC2 CC1=NOC(=O)C1CC(=O)NC1C=CC(CNC(=O)C(C)(C)c2cccnc2)C1 C1(C)(C(c2n(CCOCC)nnn2)NCC(C)(C)COC)CC=CCC1 C1(CNC(C2CCCC23CC3)=O)CCCCN1C(c1cnc(CC2CC2)s1)=O C(=O)(C#CC1(C)COC1)NC(CC)C(=O)NCC1(C(C)(F)F)CC1 n1(CCNC(C(C)n2ccnc2)=O)ccc(C(=O)NCCC2COC(C)(C)C2)c1 N1(c2cc(NC(C)(C)CNS(C)(=O)=O)ncn2)CC(=O)Nc2ccccc21 N1(C(c2ccc(C=C)cc2)=O)CCC2(C)CN(C(=O)C(c3ccnn3C)C)CC12 Cc1cccc(C(=O)N(CC(=O)NC2CC(CC(=O)OC(C)(C)C)C2)CCO)c1F n1(CC(=O)NC2CCC(F)(CNC(=O)CCC3CC3)C2)cccc([N+](=O)[O-])c1=O C(c1ccc(=N)[nH]c1C)=CC(N1CCN(C(C2CC(C#N)(OC)C2)=O)CC1)=O c1(C(=O)NCC(C)NC(=O)Cc2cc(Cl)ccc2Cl)c(Cl)c([N+](=O)[O-])nn1C C1(C(N(C(C)(C)C)CC#C)=O)CC2CC1CC2NC(=O)CC1CSC1 C1(NC(c2cc(CSCC)on2)=O)C2CCC1N(C(=O)C=Cc1nccs1)C2 c1(C(=O)NC2CCC(C)N(C(c3cc(C#N)ccc3F)=O)C2)cc(S(C)(=O)=O)co1 C1(C(=O)NCC2CC(NC(c3ccncc3Br)=O)C2)CCOC2(CCC2)C1 C1(C)(C(c2nnnn2CCCSC)NC(C(=O)OCC)COC)CCOCC1 CCC(CC)CC(F)C(=O)NCc1ocnc1C(=O)N(C)C(c1nccs1)C CCCCC(C)(F)C(=O)N(C)CC1CCCN(C(=O)Cc2cnn(CC)c2)C1 C(=O)(C(CO)NC(C1COCOC1)=O)N(CC(CC)O)C c1(C(C)C)nccc(N2CC(C)(C(N3CCC(N(C)C)C3)=O)C2)n1 N1(C(C(C)CC2CCC2)=O)CC(C(N2CC3(C2)CN(C)C3)=O)C2(CCC2)C1 Cc1c(CC(=O)NCCCN(C)C(C2CCC(=O)N(C)C2)=O)cccc1[N+](=O)[O-] N1C(NCc2ncc[nH]2)=NCCCCCCC1C1CC1.FC(F)CNC1CC1 CCC(C(=O)N(C1CN(C(c2cnsc2)=O)C1)C)Oc1ccccc1 c1(C(=O)Nc2c(C)cn(C(F)F)n2)cc(S2(=O)=NCCC2)ccc1F C=C(C)CCC(=O)NC(C1CN(C(C2(N3CCOCC3=O)CC2)=O)CCO1)C c1(NCC(c2ccccc2)NC(c2ccc(CC)o2)=O)nn(CC)cc1[N+](=O)[O-] n1(C2(CC(=O)N(CCCN(C(COCC(C)C)=O)C)C)CC2)cncn1 c1(C(=O)NCC2N(C(C(CC)OCC)=O)CC2)cc(Cl)cc(Cl)c1 C1(CC(=O)NNC(=O)C2CC3(C2)OCCO3)(C(=O)OC(C)(C)C)CCCS(=O)(=O)C1 c1(C(N2C3CN(C(c4c(C)ccnc4C)=O)CC2C3)=O)nc2ccccc2[nH]1 c1(C(N2CC(O)(C(C)NC(C3CCC(C)O3)=O)C2)=O)ccc(-c2cccs2)cn1 CCC(C)(C(=O)N1CCN(c2ccccc2NC(C2C3CCC23)=O)CC1)OC C(=O)(C1=NN(C)C(=O)CC1)NCC(N(C(=O)C(O)C1CCC1)C)C1CC1 c1(C(C(=O)NCC(CC)NC(=O)C(C)NC(N)=O)=O)ccc(C)cc1 c1(C(N2CCN(C(CNC(=O)OC)=O)C(C)C2)=O)cn2nc(C)cc2[nH]c1=O CC1(C)CCCN(C(c2nnn3c2COCC3)=O)C1CNC(c1cncs1)=O Cn1ncc2cccc(C(=O)NCCC3CCN(C(=O)CCC(F)(F)F)C3)c12 c1(C(N2CC(NC(CC3CCCC(C)C3)=O)C(C)CC2)=O)cn2c(n1)CCCC2 C1(C)(CNC(C2(NC(C)=O)CC2)=O)CCN(C(=O)C(C)Cc2ccccc2F)C1 c1(N2CC(C)CS(=O)CC2)nc2ccccc2nc1N1CCC(F)CC1 C1(C(=O)NCCCC)CN(C(=O)C=C(C)C2CC2)CC1(F)F Cc1cc(Br)ccc1C(=O)NC1CCCC1NC(=O)CC1CCCC(=O)N1 C#CC1CC2CCC1N(C(=O)CC1COCCN1C(=O)CSCCOC)C2 C#Cc1ccccc1CC(=O)N(C1CCN(C(=O)C(CC)CC=C)CC1)CC#C N1(C(C(C=C)O)=O)CCCN(C(c2ccc(F)c(F)c2Br)=O)CCC1 C1(C(=O)NCC2C(C)CCN(C(=O)COC3CCOC3)C2)CC2CCCCN2C1 N1(C(C(C)OCC#C)=O)CC(O)(CCNC(=O)C(C)OCC(C)C)C1 C12(C(=O)NCc3c(C4CN(C(CCS(N)(=O)=O)=O)C4)ocn3)CCC(=O)N1CCS2 C1(C(N2CC(CC=C)(NC(c3ccccc3OC)=O)C2)=O)CC2(CC2)CN1C C(=O)(C(C)(O)CC(C)C)N1CC(O)(CCNC(C(CC)C)=O)C1 CC1CCCN(C(c2cc(CN3CCCC(O)C3)nn2C)=O)C1 C=C1CC2(C1)CC(C(N1CCC(CCNC(C3(O)CCCCC3)=O)C1)=O)C2 Cn1cc2c(C(N3CCC(CF)(NC(=O)CC4CNC(=O)C4)C3)=O)cccc2n1 Cc1cc(C(=O)NCC2(O)CCCCC2)c2c(c1)CCCN2 n1(CC(=O)N(CCn2cc(-n3c(C)cc(C)n3)nn2)C)cc(Cl)c(O)nc1=O CC1CC(N(C(=O)C=CC2CCN(C(=O)CCc3ccoc3)CC2)C)CC(C)O1 c1(CN2CCC(NC(C3N(C(=O)NC)CCC3)=O)CC2C)cc2ccncc2[nH]1 c1(OC)nccc(C(N2CCC(c3n[nH]c(C)n3)CC2)=O)c1Br C1(c2ccc(C)cc2)CC(F)(F)CN1C(=O)NC1CC1c1ccccc1Cl c1(OC)cc(C=CCNCC(c2ccccn2)C)ccc1F c1(C(N(CC(N2CC(SC3CCCC3)C2)=O)C)=O)ccc2c(c1)NC(=O)CCN2 N1(C(c2c(C(C)NC(=O)Cc3ccc(F)nc3)noc2)=O)CCCC(F)CC1 c1(C(C)NC(C2CCN(C(=O)Cc3cccc(F)c3)C2)=O)ccnc(F)c1 CCCC(C)(O)CC(=O)N1CCC(NC(C2CCC=CO2)=O)C(CO)CC1 C12(C(N(C3CCC(NC(C4(F)CC=CCC4)=O)C3)C)=O)CC3CC1(CO)CC3C2 Cc1cc(C(=O)NCC(C)(C)OCCNC(C2CCCN2C)=O)ccc1[N+](=O)[O-] Cc1c(C(=O)N(C2CN(C(C3(C)CC4CCC(C3)S4)=O)C2)C)nn2ccccc12 c1(C(C)OC)nc(N2CCOCC(NC(=O)Cc3cc(C)nn3C)C2)cc(Cl)n1 CC1CC(NC(=O)CCN2CCCC2)CCN1C(=O)C(C(C)(C)C)n1ccnn1 CC1(C)C2CCC1(CCOC(=O)CCCc1cnn[nH]1)CC2 CC(=O)CCCC(=O)N1CC=CC(NC(=O)C(F)(F)C2CCOCC2)C1 C1(CCNC(C(C)(C)OCCC)=O)CCCN(C(=O)Cn2nccc2C)C1 C1(n2cc(-c3cnc(C)o3)nn2)CCCN(C(=O)Cc2csc(Br)n2)C1 Cc1coc(C=CC(=O)N(CCCNC(=O)Cc2ccnn2C)C(C)C)n1 Cc1c(C(=O)N(c2ccccn2)C(C2CCC2)=O)cnn1CC(F)F c1(C(N2CC(CCNC(CC3(OC)CCC3)=O)C2)=O)cccnc1CC(C)C N1(C(C(CC(C)C)C)=O)CCCCC2(CCN(C(c3nccn3C)=O)C2)C1 CC(CO)(CO)C(=O)NC1COCCN(C(c2c(O)cccc2Cl)=O)C1 c1(-n2c(C(=O)OC)c(F)cn2)cccc(S(=O)(=O)OC)c1 N1(C(c2cc(C)ncn2)=O)CC=C(CNC(c2ccc(N(C)C)cc2)=O)CC1 C1(NC(=O)CC2CC23CC3)C2CC1CN(C(c1ncccc1F)=O)C2 c1(CC)cc(C)c(C(=O)NCC2C3CN(C(C4CCSC4)=O)CC23)o1 CN1CCC(C(=O)NC2(C)CN(C(c3n[nH]cc3Br)=O)C2)CC1=O c1(NC(=O)OC(C)(C)C)c[nH]ccc1=NC(=O)CCc1cccc(F)c1 CCCC(C(=O)OC)C(=O)NCC(O)C(=O)NCC1(c2ccon2)CC1 c1(SC)cc(C(=O)NCC(CO)NC(c2cccc(Cl)c2)=O)c(C)o1 C1(C(=O)NCC2(CNC(c3cn(C4CCOC4)cn3)=O)CC2)(COC)CCOC1 CC(=O)CCN=C(NCc1nnc(CO)s1)N1CCC(c2nncs2)C1 N1(C(C2N(C(C(C(=O)OCC)OC)=O)CCC2O)=O)CCN2CCOCC2C1 C1(C(C(=O)N(C(C)CSC)CC)O)CCN(C(c2cccnc2)=O)CC1 c1(C(=O)NC(C)CCCNC(C2(O)CC2)=O)cc[nH]c(=N)c1[N+](=O)[O-] N1(C(C2C3CC(=O)CC32)=O)CC(C2CC2)(C(=O)NC2CCC(c3ncc[nH]3)CC2)C1 N1(C(C2CCC(=C)CC2)=O)CC2(C1)C(NC(=O)COC1CCCCC1)CCS2(=O)=O N1(C(COCc2cc(C)on2)=O)CCN(C(c2cc(C(F)F)n(C)n2)=O)C(C)C1 n1(C(COC)C)nc(-c2cc(C(F)(F)F)ccn2)nc1-c1sc(COC)nc1C C1(C(N2C(C)CCC(NC(c3cccnc3N)=O)C2)=O)CCc2nnnn2C1 C1(C(N2C(C(=O)NC3CCC(O)C3)CC(F)CC2)=O)CC2CCCCCC12 c1(C(N2CC(NC(CC(c3cccnc3)N(C)C)=O)C2)=O)cc2sccc2s1 CCC(CC(=O)NC1CN(C(c2cc3oc(C)cc3[nH]2)=O)CC12CC2)C(F)F N1(C(CCc2c(OCC)nccc2)=O)CCC(CNC(=O)COC2CC2)C(O)C1 C(=O)(C(=O)N=c1cc(C)o[nH]1)N1CC2(CN(C(C3C(c4c(C)ccs4)C3)=O)C2)C1 CC(C)CC(C(=O)NC(C(=O)NCC(F)CC)C(C)O)C(C)C N1(C(C(C2CCCCC2)C)=O)CCN(C(CCS(N)(=O)=O)=O)C2CCC12 N1(C(c2cc(CC)sc2)=O)CCN(C)CC1C(=O)NCC1CSC1 CC1CN(Cc2cccc(NC(=O)C(N3CCC(C)(CN)C3)=O)c2)CC(C)O1 c1(C(=O)NC2CC(CNC(c3cc(F)c[nH]3)=O)C(O)C2)c[nH]c2cc(F)ccc12 C(=O)(C(O)CC(F)(F)F)NC(C)CCNC(c1ccccc1-c1cncnc1)=O C1(NC(c2c(OC)cc(Cl)cc2)=O)CC2(CCN(C(C3(C)CCN(C)C3)=O)C2)C1 CC(C(=O)NC1CC=CCC1C(N1CC(CC23CC(C2)C3)C1)=O)C(C)(C)C Cc1cc(C(N2C(C)(CCC(=O)Nc3ccc(C)nn3)CCC2)=O)cc(O)c1 C1(NC(c2ncn(CCNC(CSCC)=O)c2)=O)CC(C)(OC)C1(C)C CC(C)C(F)C(=O)N(CCCOCCNC(C1C2CCC1(c1cnco1)C2)=O)C Cc1ccn2ncc(C(=O)NC3CC(NC(=O)Cc4nn(C)cc4Cl)C3)c2c1 CC1(C(=O)NC2CCCCC2NC(c2ccc(NCCO)nc2)=O)CCCS1(=O)=O c1(C(=O)NCCN(CCC)C(c2cccs2)=O)ccccc1S(=O)CC C1(NC(C2C(OC)(OC)CC2)=O)CCN(C(=O)CCN(CC(C)C(C)C)C)CC1 C1(NC(COCCOCC#C)=O)COCCC1NC(=O)CN.C(=O)C(CC)CC C1(C(=O)NCc2c(C)noc2)CCCCC1(C)NC(=O)C(c1ccn(C)n1)C c1(C(N2CCC(CNC(c3cc[nH]n3)=O)C2)=O)cnc2c(c1)CNC2=O c1(C(=O)NCC2(O)CCN(C(C3CC(CC)C3)=O)C2)cc2ccccc2cc1F N1(C(c2nc(OCC)oc2)=O)CC(C)CN(C(c2cc(CC)oc2C)=O)CC1C Cc1cc(Cl)c(CNC2CCNCC2)cc1C C1(O)(C(=O)NCC(CC)(C)NC(c2cc(C)sc2C)=O)CN2CCC1CC2 C=CCC(C)(C(=O)NCC1(C)CCCN1C(=O)Cc1ccc(C=C)cc1)N(C)C C1(c2ccccc2)(NC(C(C2CCOCC2)C)=O)CCN(C(c2ccco2)=O)C1 c1(CC(N2CCC(N(C(COCCOCC)=O)C)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 N1(C(CC=CC(C)(C)C)=O)CCC(C)(CC(=O)NC2CCCC2O)C1 C=CCCCCC(=O)NC1CCN(C(=O)CCC(C)OC)CC1O C=CCCCC(C(=O)N1CCC(CC)C1)NC(C1CCCN(C)C1)C N1(C(c2cncc(C(C)C)c2)=O)C2CCC1CN(C(c1cc(Cl)cnc1O)=O)C2 c1(C(N2CC(CC)C(NC(C3CC(=O)NC(C)C3)=O)C2)=O)cc(C)c(F)c(C)c1 c1(C(N2CCC(C)(C(=O)NCCC(CC)(F)F)C2)=O)ncn2ccccc12 S(=O)(=O)(c1cc(C=CC#N)ccc1OC)NCC.C(C)(CSC)NC(C1(C(N)=O)CC1)=O C(=O)(C1CCCc2nc[nH]c21)N1CC(O)(CNC(=O)C#CC2(CC)COC2)C1 c1(CC(C(=O)OC)NCc2cc(C(C)=O)c[nH]2)ccc(SC)cc1Cl c1(CN(C(=O)Cn2cc(CN3CCC3c3ncon3)nn2)CC)ccc(C)cc1 C1(CC(=O)NC(C)(C)C=CC(=O)NCCCC2(O)CCC2)(OCCOC)CCC1 CC1OC(C)C(C(=O)NC(C)(C)CNC(c2cnc(Cl)c(N)c2)=O)C1C C1(C(N(C)CCC2CCN(C(=O)COC(F)F)CC2)=O)Cc2cncn2C(=O)N1 C(=O)(C#CC1(C)CCCO1)NCC(C(N1CCCC1(C)CCCO)=O)N(C)C C1(NC(=O)C(c2ccccc2)F)CC2C1CCN2C(=O)CCc1cccc(Cl)c1 C(N=c1[nH]c(C)cc(=NCCN2CCP(C)(=O)CC2)[nH]1)C1CCC(CCC)CC1 C1(C(=O)NC(C)(C)CC)CC(NC(CCCCOCC)=O)C12CCC2 N1(C(C2N(C(C3CCN(C)C3)=O)CC2)=O)CC(CC2CCC2)C1(C)C C1(NC(C(COC)N(C)C)=O)CCSC12CN(C(c1cc3sccc3[nH]1)=O)C2 C(CCCC(=O)NC(C1(O)CCN(C(C2SCC=C2C)=O)C1)C)SC c1(C(=O)NC(CNC(c2c(C)coc2)=O)C(C)C)cccc(CC(C)C)c1 c1(CN(C(C(CC)O)=O)C2CCCC2)ccc(C)n1-c1cccc(C(F)(F)F)c1 Clc1nsc(CC2CCN(c3nccc(Oc4ccccc4)n3)C2)c1Cl N1(C(C2CN(C(C3N(C)CC3)=O)CC2F)=O)CC(C)(C)C2CCCC12 N1(c2c(C)c(NN3CCC(C(=O)N(C)C)C3)ncn2)CCOc2cc(F)ccc2C1 c1(OC)c(C)cc(C(=O)N(C2CCCCC2)Cc2cccnc2)cc1Cl c1(C(N2CCC(NC(CCC=CC)=O)C2)=O)ccc2cc(Cl)ccc2n1 CC(C(=O)NC1(CF)CCN(C(c2cc(Cl)cs2)=O)C1)C(F)F c1(C(N2CCCCC2C(F)(F)C(F)(F)F)=O)ccc(I)c2c1OCCO2 C1(NC(c2c(C(=O)OC)nco2)=O)CCCC2CN(C(C3CC4(CC4)C3)=O)CC12 c1(CC)ccc(C(N2CCCC2C2(O)CN(C(C3CC3C3CCCO3)=O)C2)=O)s1 C1(C(N(C)CC2(NC(=O)COc3ccc(Cl)cc3)CC2)=O)CNC(=O)C(C)(C)C1 C1(O)(C(=O)NC(CNC(c2nc(OCC)oc2)=O)C)CCC(C)CC1 CC(C(=O)Nc1cc(C(=O)NOCC(F)F)on1)C(F)(F)F.c12cn(nn1)C2 C1(NC(c2c(CC)onc2C)=O)COC2(CCN(C(c3cocn3)=O)C2)C1 c1(C(=O)OC(CNC(C(C(CC)C)=O)=O)=O)ccc2c(c1)OCCO2 N1C2CCCC1CC(n1cc(CN(C)C)nn1)C2.Cc1nc(O)c(F)c(Cl)n1 c1(OC)cc(F)ccc1C(N1CC2CC1C2C(=O)Nc1cccc(C#N)c1)=O N1(C(C(C(C)(F)F)(C)C)=O)CCC(C2(NC(C3CCCC4CC34)=O)CC2)CC1 N1(C(C2CC2F)=O)CCN(C(=O)CCCF)CC1c1cccc(F)c1 N1(C(CN(C)C(N)=O)=O)CCC2(CCCC2NC(c2ccn(CC(F)F)n2)=O)C1 N1(C(c2c(COC)scc2)=O)CC2CC1CC2CNC(c1ccccc1)=O c1(C(C)(C)C#N)cc(NC(=O)NC2CCC(C(N)=O)C2)cc(C(F)(F)F)c1 c12cccc(c1)NC(C)CC(C)NS(=O)(=O)C2.c1(C(=O)CC)nn[nH]c1Cl.C(=O)N Cc1cc(C)c2[nH]c(C(c3nnnn3C3CC3)NCc3ccc(I)cc3)cc2c1 c1(N(C)C(C2CC(O)CN2C(=O)C(O)CC(N)=O)=O)cc(O)cc(F)c1 c1(C(=O)NC2CC(C(N3CC(COC)C3(C)C)=O)C2(C)C)ncc(F)cc1C N1(C(=O)CCF)CCC(CCC2CCCCN2C(=O)CCn2ccnn2)CC1 C(=O)(C(F)(F)C(F)(F)C(F)F)N1CC(CNC(c2c(COC)cco2)=O)C(O)C1 C1(NC(C(=O)OC)=O)CCN(C(=O)CCCOc2ccc(F)cc2Cl)C(C)C1 N1(C(c2ccc(OC)s2)=O)CCC(O)C(NC(c2cc(Cl)ccc2OC)=O)C1 C1(CC)CCCC1C(=O)NC(C1CN(C(c2ccnn2C(CC)CC)=O)C1)C N1(C(C(C)OCC)=O)CCN(C(c2nc(C(C)C)ncc2Br)=O)CC1CO C(=O)(C1=C(C#N)CCC1)NC1CC(C)(C)N(C(c2cccc(OCCF)c2)=O)C1 c1(CC)sc(C(=O)NC(C)CC(C)NC(=O)C(C)(C)C)cc1C C1(C(=O)NCCOCCN(C(CN(CCC#C)C)=O)C)CC(C(C)C)C1 c1(C(N(C(CN(C(c2c(COCC)cc[nH]2)=O)C)C)C)=O)sc(C)c(C)c1C c1(OCC)ncc(Cl)cc1C(N1CC(NC(=O)Cn2cc(C#N)cn2)C1)=O C(=O)(C1=CCCN(C(C2CN(C)C2)=O)C1)Nc1ccc(C)nc1 Cc1nc(C)c(CNC(C2(CNC(=O)CC(C)F)CC=CC2)=O)o1 C1(NC(C(F)OC)=O)CCOC2(CCN(C(c3coc(Cl)c3)=O)CC2)C1 O=C(C(O)CC1CCOCC1)N1CC(c2ccccc2)(C(F)(F)F)C1 c1(C(N(C2CN(C(C3(C)CCCC3O)=O)C2)C)=O)ccc(F)c(CO)c1 S(=O)(=O)(c1cnc(Nc2ccc(F)cc2)c(Cl)c1)NC(CN(C)C)CO.CC1CO1 CC1(CNC(C2(C)CC(NC(=O)Cc3cncnc3)C2)=O)CC2CC2C1 C1(NC(C2OCC(=C)C2)=O)CCCCC1c1nc[nH]n1 OCCCCC(Cc1ccccc1)Nc1nsc(CSc2ccccc2)n1 C(C(C)(C)C#CC(=O)N(CC(O)COCC)C)NC(CC(=C=C)C)=O c1(SCC)cccc(CC(N2CC(CNC(=O)CN(C)C(C)=O)CC2C)=O)c1 Cc1cc(C(N2CCCC2CN(C)CCNS(C)(=O)=O)=O)ccc1Cl C1(C(=O)NC(CC(C)C)CNC(=O)C2=NOCC2)CCN(C2CC2)S1(=O)=O C(CC(F)F)(C(=O)N(C1CCOCC1C)CC)N(C(C1N(CCC)CCC1)=O)C c1(NC(C2C3CCC(C3)N2C(c2cccc(I)c2Cl)=O)=O)c(F)cc(I)cc1F N1(C(C(C(C)C)(C)O)=O)CCC2C(CCCN2C(c2ccsc2C#N)=O)C1 N1(C(c2cc(C)ncc2)=O)CC2(CCCN(C(c3oc(C)cc3C)=O)C2)C1 C(=O)(C(CCC=C)NC(=O)CC1C(=O)NN=C1C)N1C(C#C)CCC1 C1(C2(C(=O)NC(C)C(N)=O)CC2)CCCN1C(=O)CCc1ccoc1 c1(C(N2C(C)C(NC(=O)COc3ccon3)CC2)=O)n[nH]c2ccc(Cl)cc12 C(=O)(CCCCCC#N)N1C(C(=O)NCC2CCC(C)(CC)O2)(C(C)C)CCC1 Cc1sc(C(=O)NCC2C3CN(c4nnc(C#N)s4)CC23)nc1O c1(CC(=O)NC2CC(NC(c3csnn3)=O)C(O)C2)nsc2ccccc12 c1(C(=O)NCC2(F)CCC(NC(c3scc(CC)c3)=O)C2)cc(Cl)cc(F)c1F c1(C(C)C)ccc(C(N2CCOC(CNC(c3cn(C4CC4)nn3)=O)C2)=O)cn1 C1(CC)CN(C(=O)CN2CCCCC2)CC1C(=O)NOCC1(C)CC1 c1(C(=O)NC2C(NC(CC(C)SC)=O)C2)cc(C(F)(F)F)n(C)n1 c1(CN2C(CC(N3CCCC(F)C3)=O)COCC2)cnc2ncccn12 c1(C(=O)NCCCC(C)NC(C(C)NC(N)=O)=O)c[nH]c(=O)c2ccncc12 c1(OC)nccc(I)c1C(c1nnnn1C(C)C)CN1CC(OCCO)C(O)C1 N1(C(c2cc(C)cc(O)n2)=O)CCCN(C(=O)C(c2ccc(Cl)s2)C)C(CO)C1 c1(CCC)cccc(NC(=O)CCN(C(=O)CC2CCCN(C)C2)CCO)c1 n1(CCNC(C(=O)NC(C2CC23CCC3)CC)=O)nc(C)ccc1=O C(=O)(CCCCC(=O)N1CC2CC(NC(c3ccnc(C(F)F)c3)=O)C2C1)NC C1(NC(Cc2c(C)ncs2)=O)CCN(C(c2c(Br)noc2C)=O)CC1 N1(C(c2nc(COC)oc2)=O)CCC(C)(CC(=O)NCCCCCO)C1 O=C1NCc2cc(N(C(=O)C(=O)C=Cc3ccccc3)Cc3cn[nH]c3)ccc21 c1(OC)ccc2[nH]c(C(=O)N(C)CCN(C(=O)C(F)C(C)C)C)cc(=O)c2c1 CC(C1=CCN(C)CC1)NC(=O)CC(CNC(C1CC2CC2C1)=O)C1CCC1 CCC(C)C(O)C(=O)N(C1CCC(CNC(=O)COC2CCCOC2)CC1)C CCCCC(C(=O)Nc1ccc(O)cc1Cl)NC(=O)CNc1ccccn1 Cc1cc(C(=O)NCC2CCC(NC(c3csc(C(F)(F)F)n3)=O)C2)nnc1O C1(NC(C=CSC)=O)CC2(CCC(NC(C3Cc4ccccc4O3)=O)CC2)C1 C(=O)(NNC(=O)C1CCOCC1)NC1(CC=C)CC1 C(C)(CCC(F)(F)F)NC(c1cc(C)nn1-c1ccccc1Br)=O C1(CCC)CN(C(c2cc(O)nn2C)=O)CCN1C(=O)C(O)Cn1cncn1 c1(C(N2C(CN(C(COCC(C)C)=O)C3CC3)COCC2)=O)cc(Cl)ncc1O CCC1=C(C(=O)N2CC(C(N3C4CCC3CC(C)C4)=O)(CC)C2)CCCO1 C1(C(N(C(C2CCC2)C)CC)=O)CN(C(=O)C(C)(C(C)C)OC)CCC12CCC2 C=CC(C)(O)CC(=O)NCC1CC(COC)CN1C(=O)CCc1cnn(C)c1C N1(CC(=O)NCc2cnc(N3CCOCC3)s2)CCCOCC1 N1(C(C=C(CC)C)=O)CC(N(C)C(c2ccc(C(=O)OC(C)(C)C)cc2)=O)C(O)C1 C(C(C)(C)C(=O)NC1CN(C(=O)CCCOc2ccccc2)CC1O)OCC c1(SC)ccnc(-c2nc(CCCF)n(C(c3ccc(C)s3)C)n2)c1 C1(CC2CCC(NC(C3CCC(C(=O)OC)CC3)=O)C2)CNc2ccccc2C1 C=CCCC(C)(C)NC(=O)NCCn1ccnc1-c1ccc(F)cc1 Cc1cccc(C(C)(CO)NC(=O)NCCc2c(C)cccc2Br)c1C N1(C(C(CC=C)c2ccccc2)=O)CCOC(C)(CNC(=O)CC2(OC)CCC2)C1 c1(CC(N2CC(N(C(CCC(CC)C)=O)C)C2)=O)ccc2ccncc2c1 c1(C(=O)NC2C(NC(c3c(C)cccc3F)=O)C2)cn(C)c2ccccc12 CC1CN(C(=O)CC2CCN(C(c3ccnn3CCF)=O)CC2)CC(C2CC2)O1 C(=O)(C1=CC(O)C(NC(c2nnc(S)n2C)=O)C1)N(C)Cc1cnn(C)c1 N1(C(CSc2n(CC)cnn2)=O)CCC2(CC1)CCN(C(=O)COCC(C)C)C2 N1(C(C(c2ccn(C)n2)C)=O)CCCC(NC(=O)CCc2cnccn2)CC1 CC(C)C(CNC1CC1)C(=O)NCC1(CNC(c2ccc(CO)cn2)=O)CC1 C12(CNC(C(n3c(C)cc(C)n3)C)=O)CCC1CN(C(=O)CN1CC(C)C1)C2 N1(C(C(=O)N2CC(c3cc(Br)cs3)C2)=O)Cc2ccncc2C1 C1(CNC(CCSc2nc(C)[nH]n2)=O)(CO)CCN(C(=O)C(C)NC(N)=O)CC1 C1(C(=O)NCC=C2CCN(C(C3(C)N(C)CC(O)C3)=O)CC2)CC2(C1)CC1(CC1)C2 N1(C(C(COCC)C)=O)CC2CCC(C1)C(NC(c1sc([N+](=O)[O-])cc1Cl)=O)C2 CCCC(C)(O)C(=O)N1CC(CO)(NC(=O)Cc2cc(F)ccc2F)C1 CN1C2CCCC1CC2.C(CCNCC)C(C)(F)F c1(CC(=O)N(CCOC)CCNC(c2cccs2)=O)cnc(C(F)(F)F)s1 c1(C(C)NC(=O)NC23CC(C(=O)NC(C)(C)C)(C2)C3)ccc(Cl)cc1F c12nnnn1C2.C(C(C)NC(=O)C1CC1)NC(=O)OC c1(C2C(=O)NCCN2CC)cc(OC)ccc1SC1CC1.C1(CN(C)C)CCC1 C#CCC(C)(C)C(=O)NCCC1C(C)CCCN1C(=O)CC1CCC(C)CC1 N=c1ccc(C(=O)NC2(CF)CCN(C(c3cnn(CC4CC4)c3)=O)C2)c[nH]1 c1(CC)ccc(C(=O)NCC=CCNC(c2c(C(N)=O)cccc2C)=O)c(Cl)c1 N1(C(=O)Cc2cccnc2O)CC=C(c2ccc(Cl)cc2)CC1 CC1C(NC(=O)CC(C)NC(N)=O)CC2CCC1N2C(=O)CC(=O)N(C)C c1(C(=O)NCC2N(C(C3C(OC)CCC3)=O)CCC2)c[nH]c2cccc(C#N)c12 Cc1cc(Cl)c(C(N2CCC(NC(=O)CCC3CCOC3)C23CC3)=O)cc1C C(CN=c1[nH]c2ccccc2o1)C1CCN(C(C(c2ccccc2)C)=O)CC1 N1(C(CSCC(=O)OC(C)C)=O)CCCC(NC(C23CCCC2CCC3)=O)CC1 Cc1cc(N(C(C2CCN(C(C3CCC(CO)CC3)=O)CC2)=O)C)n(C2CC2)n1 C12(CC)CCC(C(N3CCC(CNC(=O)C=CBr)(OC(C)=O)C3)=O)(CC1)CO2 N1(C(C(CC)NC(N2CCC(O)C(O)C2)=O)=O)CCn2cc(C(F)(F)F)nc2C1 C1(NC(C(C)SC)=O)CCCC1(C)CN(C(=O)CCCc1cccs1)C N1(C(Cc2nc(C)[nH]n2)=O)CCCC1C1CCCCN1C(C1CS(=O)(=O)C1)=O c1(CN2CC3N(C(=O)Cn4cc(Br)cn4)C(C3)C2)n[nH]c2ccc(Br)cc12 c1(C(N2C3(CN(C(C(n4cc(Cl)cn4)C)=O)C3)CC2)=O)cc2cccnn2c1 c1(C(N2CCC(NC(c3cc(C)c(C)s3)=O)CC2C)=O)ccccc1N=[N+]=[N-] c1(C(=O)NC(C)CNC(C23CCCC2CC3)=O)ccccc1SCc1ccccn1 C(c1ccc(Cl)cc1F)=NCC1(N(C(C(CC(C)C)C)=O)C2CC3(CCC3)C2)CC1 N1(C(C(C)SCC)=O)CCN(C(c2occc2CC)=O)CC1C(C)C C#CC1CC1C(=O)N(CCCN(C(=O)CCNC(=O)CO)C)C c1(CC(=O)NC2C(CNC(CSCCCCC)=O)CC2)cnc(C)nc1O c1(C(N2C(CN(C)C(C3OCC3(C)C)=O)CCCC2)=O)cc(O)cc(O)n1 c1(C(CC(=O)NCC2(O)COC2)NCCSc2cccnc2)ccc(F)cc1 C1(C(=O)NCc2cc(Cl)cs2)CCC2(CC2)N1C(=O)CCCN1CCCC1 Cc1noc(C)c1C(c1nnnn1C1(C)CC1)NCC1CCC(F)(F)C1 C(C(O)C(=O)NCCCN(C(c1ccn(C)n1)=O)CC1CCCC1)SC CC1CC=C(C(=O)NCCC2(O)CN(C(c3cc(C4CC4)nnc3O)=O)C2)CC1 CCC(C)CCC(=O)N1CCCC(NC(c2cc(C(C)(C)C)c[nH]2)=O)CC1 N1(C(C2N(CC)CCC2)=O)CC2CC(NC(C3(CCOC)CCCC3)=O)C(C2)C1 c1(C(F)(F)Br)csc(-c2ccsc2)n1.C1(C(C2CC2)N)CCCC1.CCC CN1CC2(C)CN(C(c3cc(-c4cccc(F)c4)c4cn[nH]c4c3)=O)CC2(C)C1 N1(c2nc(Cl)nc(C)c2F)CCOC2(CCS(=O)(=NC(=O)C(F)CC)C(C)C2)C1 C(=O)(CCCC1CCCCC1)NCCC(C)N(C(=O)C(O)C1CCC1)C C1(C(=O)NCCN(C(c2ncc(C)nc2)=O)CC2CC2)CC(C)CC(C)C1 CCS(=O)(=O)CC(=O)N1CC(NC(C2C=CC(C)(C)CC2)=O)C(SC)C1 c1(C(N(C(=O)NC(C=COC)=O)C)=O)cc(Br)ccc1N.C1(C)(C)C=CCN1 n1(CC)ncn(NC(=O)C2(C)CN(C(C3CCC(=O)CC3)=O)C(C)(C)C2)c1=O c1(C(N2C(C(=O)NCc3nc(C)on3)CC(O)C2)=O)ccc([N+](=O)[O-])o1 S(=O)(=O)(c1ccc(NC2C3Cc4ccc(Cl)cc4C23)c(Br)c1)NCCN(C)CC CC(C)N=c1nc(N2CCOCC(C3CC3)C2)[nH]c(=NCCC2=CCOCC2)[nH]1 C1(c2ccccc2Cl)(CNC(C2CCC(NC(C)=O)C2)=O)CCOCC1 c1(N(C)C)ncc(C(C(=O)NC(C)(C)C)N(C2CCCC2)CC2CC2)o1 N1(C(CCOCCN(C(c2c(C)snc2)=O)C)=O)CCSCCC1C CON(CCC(=O)NCCC1NC(=O)NC1=O)C(=O)c1cnc(C)o1 N1(C(c2nc(C)on2)C)CCC2(CC1)CC(C)N(C(=O)C(C)OCC1CC1)C2 C1(NC(CN(C)CCO)=O)CCN(C(c2ncccc2CO)=O)C12CC2 CC(=Cn1ccnn1)C(=O)N1CC(N(C(=O)C=Cc2ccc[nH]2)C)C2(CC2)C1 N1(C(C(C)OCC#C)=O)CCCCC1CN(C)C(c1sccc1-n1cnnn1)=O C(CC(O)CC(=O)NC1CC(C)N(C(=O)C(O)Cc2cnc[nH]2)C1)SC C(CCCCC(=O)NC1(C)CCN(C(=O)CCCN2C(=O)CCC2=O)C1)N(C)C N1(C(CC2CC(=C)C2)=O)CCCC(C(=O)NC2CC2C2CC2C)C1C N1(C(C2CC(CC)C2)=O)CC2CC2C1C(=O)NCc1noc(C(C)C)n1 c1(C(=O)NCC2CCN(C(c3cc(C)[nH]n3)=O)C2)ccnc2c(Br)cccc12 C1(CNC(c2sc(C)c(Br)n2)=O)CN(C(C2CCCS2)=O)CC12CC2 N1(C(c2c(CC)csc2)=O)CCN(C(=O)Cn2cc(CC3CC3)nn2)CC1CO N1(C(C(C2CCOCC2)OCC)=O)C2CCC1CN(C(c1ccc(C#N)n1C)=O)C2 CC1=CCSC1C(=O)NCC(C1CCC1)NC(c1nnn(C(C)(C)C)n1)=O c1(NC(C2COCCO2)C)cc(=NCc2ccnc(O)c2)[nH]c(C(C)C)n1 C1(C(N(CC(O)CN2CCC(CC3CC3)CC2)C(C)C)=O)CCCC(=O)C1 c1(OC(C(=O)NC(CC)(C)CNC(C)=O)COC)ccccc1CCC(F)(F)F c1(-c2ccc(C(N(CCCCNC(c3cnc(C)s3)=O)C)=O)o2)cccc(O)c1 CC(C)(C)CCC(F)C(=O)N1CCC(C(F)CNC(=O)CN2CC(C)(C)C2)CC1 C(=O)(C(O)CCC(C)C)N(CC(CNC(c1cnn(CCCC)c1C)=O)O)C C(CC(=O)N(CCCC(C)(F)F)C)(C(F)(F)F)NC(C1(OCC)CCOC1)=O C(=O)(C(CC(C)C)NC(=O)NC1CC2(CC2)CCC1)NCC1CC(OCC)C1 c1(OC)cccc2c(C(=O)N(C)CCNC(c3cn(C)c(C)cc3=O)=O)n[nH]c12 N1(Cc2ccc(OC)c(Br)c2F)CCC2(CC1)CCN2C(=O)C(C)(F)F C(CC(C)(C)C(=O)NCc1cncnc1)NC(c1c(C)cc[nH]1)=O N1(C(Cc2n[nH]c(=N)s2)=O)CC2CCC(C1)C(NC(=O)CCn1cccn1)C2 N1(C(CN2C(=O)CCCC2)=O)CCC12CN(C(=O)Cc1cnc[nH]1)C2 C1(CCC)CN(C(c2ncncc2Cl)=O)CCN1C(=O)CCC1CCCO1 CCCCCCCCC(=O)NCCC(O)CNC(c1ncc(Br)cn1)=O c1(C(N(CC(C)NC(c2cc(C)[nH]n2)=O)CC)=O)cn2cc(Cl)cnc2n1 C(CCCCCNC(=O)COCCN(C)C)NC(C(C)SC(C)C)=O C1(CCOC)(NC(=O)CCc2ccsc2)CN(C(=O)NCCOC)C1 C(=O)(CC(C(C)OC)NC(=O)CSc1ncc[nH]1)N(C)CC N1(C(C)=O)CCC2CCCN(C(c3csc(S)n3)=O)C2C1.c1ccc2ocnc2c1 C1(C(=O)NC(C(C)(C)NC(CSCC=C)=O)C)CCCCN(C)C1=O Cc1cccc(C(N2CCCC2C2(O)CN(C(c3ccn(C)n3)=O)C2)=O)c1Cl c1(OC)c(NC(C2C(O)CCN2Cc2csc(C)n2)=O)ccc(F)c1F C1(C(N2CCN(C3CCC(NC(=O)C=CSC)CC3)CC2)=O)(OC)CS(=O)(=O)C1 c1(C(=O)NCC23C(CN(C(CSCCN(C)C)=O)C2)C3)ccc2cnn(C)c2c1 c1(C(=O)Nc2ccc(C)cc2)c(C)ccc2c1NC(=O)C2=O C1(NC(c2cn(CCO)c(=O)nc2O)=O)CCc2cnccc2C1 c1(NCC=CC)ccc(S(=O)(=O)NC2(CSC)CCOC(C)(C)C2)cc1Cl C=CC1(C(=O)NC2CCCOC2)CCN(C(c2ncc(F)cc2F)=O)C1 c1(Cn2cc(C(C)NC(=O)Cc3cocc3Br)nn2)c(Cl)cccc1Cl c1(C(C)(C)C)cc(C(N2CC(CO)(NC(=O)CC3CC(F)(F)C3)C2)=O)no1 C12(CNC(C3CC(CC(C)(C)C)C3)=O)CC(CO1)N(C(=O)C#CC1CC1)C2 c1(C(=O)NC2CC3CC2CC3(F)F)cn2cccc(Br)c2n1 c1(C(=O)NC(CNC(C(CC=C)C)=O)(C)CO)ccc([N+](=O)[O-])c(C)n1 CC1=CCC(NC(=O)C(c2cnn(C)c2)NC(=O)CCC2CC2(F)F)CC1 C1(C(=O)NCC2CC(OC)CN2C(C2CC(=O)N2)=O)CCCCCCC1 CC1(C)C2CCC1(CC(=O)NCCCCNC(C1C(Cl)(Cl)C13CC3)=O)CC2 C1(C(N(C)CC2CCN(C(C)(C)C)C2)=O)C=CC(N=c2cncc[nH]2)C(=O)N1 c1(C(=O)NCC2(OC)CN(C(C(CC(=O)OC)C)=O)C2)cc2nc(Cl)ccc2s1 N1(C(CCOC)=O)C2CCC1CN(C(C1CC3C=CC1C3)=O)C2 C=C(C)c1cccc(NC(=O)CC2CCCN2C(C2CC23CCC3)=O)c1 C1(NC(C=C(C)Cl)=O)CCC2(CC1)CC(NC(c1cc(C)c(C)c(C)c1)=O)C2 Cc1nnc(=NCCCCC(C)N(C(=O)C(C)OCCN(C)C)CC)[nH]c1C N1(C(Cc2c(SC)cccc2)=O)CCC12CCN(C(C1CCCC(C)C1)=O)CC2 C1(COC)CCCN(c2nnc(C3CC3Cc3ccsc3)n2CC)C1 C(CC(C)C(=O)N1CCC(NC(C2(N)CC2)=O)C1)=CC Cc1nc(CCC(=O)N(C(C)CNC(c2occc2-c2cccs2)=O)C)oc1C CCCC(C(=O)NCc1nc(C(=O)NC2C=CCC2)c(C)o1)OCC C1(C(=O)NCC(C(C)C)NC(c2cn(C)nc2C2CC2)=O)CCCC(C#N)C1 N1(C(C2OCCC(C)(C)C2)=O)CCC2C(C1)CN2C(c1cccc(CCO)c1)=O C1(CC)CC(=O)OC1(C)C.C12C(C(=O)NC3(C(=O)OC)CC3)CCN1C2=O N1(C(CCCC(C)C)=O)CCCN(C(c2ccn(C)c(=O)c2)=O)CC1C(C)C C(=O)(CCC(CF)CF)N1CCN(C(=O)COC2CCCOC2)CC1 C1(OC)CN(C(=O)CC2CC2)C(C)(CNC(=O)CC(C)(C)c2cccs2)C1 N1(C(C(c2cccc(C)c2)O)=O)CC(N(C(=O)CC2(C(F)F)CC2)C)C2(CC2)C1 N1(C(C(C)O)=O)CCOC2(CCN(C(c3ccc(S(N)(=O)=O)cc3F)=O)C2)C1 c1(C(N2CCC3(CCCOC3)C2)=O)ccc(Br)c(S(=O)(=O)N2CCCC2)c1 C1(CNC(C(C(C)C)OCC)=O)CC(C)CN(C(c2sc(F)cc2Cl)=O)C1 c1(NC)scnc1C(=O)NC(CC(=O)NC(C1CCOCC1)C)C1CC1 C12COCCC13CN(C3)C2=O.CC1(CC(=O)Nc2ccc(C(F)F)s2)OCCO1 Cc1ccc2c(CNC(=O)CC3(C)CN(C(=O)OC(C)(C)C)CC3C)coc2c1 c1(OC(C(=O)NCC(CC)NC(c2cnc(O)s2)=O)C)ccc(C)cc1 c1(C(=O)NCC2CN(C(c3cc([N+](=O)[O-])n[nH]3)=O)CC2O)c[nH]c2ncccc12 N1(C(C(C)=O)=O)CCn2ncc(CNC(=O)CCC(C)(C)O)c2C1 c1(NC(C)=O)cnn2ccccc12.C12C3CCCC3CN1c1cc(C)nc(n1)SC2 C1(C(=O)NC2C(CNC(C(=Cc3ccncc3)C)=O)C2)CC2(CCCCC2)CO1 c1(C(=O)NCC2CC2N)c[nH]cc(Cl)c1=O.C12(OC)CC(C1)C(=O)N2.OC C(=O)(C=C1SCC(=O)N1C)NC(C1CC1NC(=O)CSc1ccccc1Cl)C C(CC1CCC1)(C(=O)NC1(C(N(C)CC2CCOC2C)=O)CSC1)OC C(=O)(C1=CCOCC1)N1CC(C(C)NC(=O)CC=CC(C)(C)C)OCC1 C1(NC(C(=O)NCC)=O)CC2CCC1(NC(C1CC1CC)=O)C2 C1(NC(c2c(C)nc(C(C)(C)C)s2)=O)CC2CC(NC(=O)CC(C)N(C)C)CC12 CN=c1[nH]cc(C(N2CC(=O)CC2C(=O)NCc2conc2C2CC2)=O)s1 CC1CN(C(=O)CSc2ccccc2)CCC1NC(=O)CN(C)CCO CCC(C)(C(c1nnnn1CCCC1CC1)NCCNC(C)=O)N1CCCC1 O=C(CS(=O)(=O)CCO)NCCC1CCN(C(C2CCCCC2O)=O)C1 C(=O)(C=C1SCC(=O)N1C)NC1CN(C(Cn2c(C)ccn2)=O)C(C)(C)C1 C1(C(=O)NCCOCCN(C)C(c2cccc(=O)n2C)=O)CCCCC(F)(F)C1 c1(CC)ccccc1OCCC(N1CCC(N(C(=O)Cc2ncoc2C)C)C1)=O C1(C(C)Cn2cc(-c3cccnc3NC(=S)NC3CCCC3)nn2)COCCN1C(C)C C12(C(=O)NC(C3N(C(c4nc(C(C)C)sc4)=O)CCC3)C)CC3CC(CC1C3)C2 N1(C(CC2CCC(=O)NC2)=O)CC(NC(=O)Cc2csnn2)C2(CCOCC2)C1 c1(C(C)NC(C(C)C2CC2c2ccc(F)cc2Cl)=O)ccc2c(c1)OCCO2 C(=O)(C1=C(C#N)CCC1)N(C(C)C(=O)NCC1CC1(C)C)CC c1(C(N2CCN(C(=O)Nc3cc(Cl)c(F)c(Br)c3)CC2)=O)ccc2c(c1)OCO2 N1(CCC)CCN(C(c2ccc(CNC(=O)NC(C)C)cn2)=O)CC1 C1(NC(C(CCNC(c2cncc(C)n2)=O)OC)=O)CCC(C)(C)CC1C c1(N2CC3CCS(=O)CC3C2)nc(=NC2CCSC2)[nH]c2cc[nH]c12 C1(CNC(C2C(C(C)NC(Cc3c(C)nn(C)c3)=O)C2)=O)OC(=O)CC1(C)C N1(C(c2c(C)nn(C)c2)=O)CC(CC(=O)NC(c2ccsc2)C)CC1(C)C S(=O)(=O)(CC(=O)N(CCCN(C(=O)C(C1CC1)N(C)C)CC)C)NCC c1(Nc2nc(Cl)ccc2[N+](=O)[O-])ncc([N+](=O)[O-])cc1O.CC12CCN1C2=O N1(C(CC=C(C)C)=O)CC2CCC2(CC(=O)N(CCCN(C)C)C)C1 Cc1ccncc1C1CC1C1N(C(N2CCNCC2c2ccccc2)=O)CC(O)C1 CCC(C)C(CO)NC(C1(C)CCN(C(=O)C(O)CSC)C1)=O C(=O)(C1=CC(O)C(NC(c2cccc(F)c2N)=O)C1)NC(CC)C(C)(C)C CC1(C)CN(C(=O)Cc2ccn(C(F)F)n2)CC1CNC(C1CCCC12CC2)=O C1(C(=O)NC(C(=O)N(C)C)Cc2ccccc2Br)CC2COCC(C1)C2 N1(C(C=CS(C)=O)=O)CCN(C(=O)COC2CC=CC2)CC1CC(F)F N1(C(c2cc(C3CC3)cs2)=O)CCC(OC(F)F)(CNC(C2(F)CC2)=O)C1 c1(CNC(C2(CC)CC3CCC2CC3)=O)ccc2c(c1)NC(=O)C(C)O2 c1(NC(C(C(C)NC(c2n[nH]c(CC)c2Cl)=O)C)=O)cccc2c1OCO2 c1(OC)cc(C(=O)NCC2(CS(N)(=O)=O)COC2)cc(CNCC(C)=O)c1O C1(CN(C(c2n[nH]c(C)c2C(F)(F)F)=O)CC)CCCCN1C(=O)C(C)SC N1(C(C(CCC)N(C)C)=O)CCC2CN(C(c3sc(CC)nc3C)=O)C2C1 Cc1nc2ccc(C(=O)NCC(C)(O)CNC(C3CCC(=O)C3)=O)cc2n1C N1(C(COC2(C)CCC2)=O)CCCC(NC(c2cc(Cl)c[nH]2)=O)CC1 N1(CCNC(C(=O)N(CC(C(C)C)OC)C)=O)C(=O)CN(C)C1=O c1(C(C)C(=O)NCC2CCCC2NC(=O)Cn2nccn2)ccc(Br)cc1 c1(C(=O)NCC(C)CC(N2CCN(C)C(=O)C2C)=O)ccc2c(c1)OCO2 c1(CC)n[nH]c(=NCC2CC(CNC(c3scnc3C(F)(F)F)=O)CO2)s1 c1(C(=O)NCC(C2CCCN2c2ncc(F)cn2)(C)C)cnc2n1CCOC2 c1(C(=O)NC2C(C(=O)NC3CCN(C(=O)NC)C3)CCC2)cnc2n1CCOC2 Cc1sc(NC(=O)COC2CCCCC2C(C)(C)C)c(C#N)c1C N1(C(c2n[nH]c(C)c2C)=O)CCC(C2(O)CN(C(=O)Cc3cccs3)C2)CC1 C(=O)(C(CC)N(C)C)NNC(=O)C=CCCC1(CCOCC)CCC1.C.N c1(OC)cc(F)ccc1CC(N1CCC(N(C)C(c2c[nH]nc2F)=O)C1)=O C(=O)(C1CCCc2sccc21)NCC1(NC(CC(=O)NCC)=O)CCOC1 N#Cc1cc(Br)ccc1CN1CCN(c2nccc(Br)n2)C2CC12 C1(CC(=O)NC2CC(CNC(c3nc(OCC)oc3)=O)C2)CCC2(CCC2)O1 CC1=NOC(=O)C1CC(=O)NCC1CN(C(=O)CCc2ccnc(Cl)c2)CC1O C1(C(=O)NC2C(C)CN(C(=O)CNC(N3CCCC3)=O)C2)C2CCC1(C)C2(C)C CCC(C(=O)OCOC)C(=O)N1CC(F)CC1CNC(c1cc(C)ns1)=O C(c1cccc(C)c1)=CC(=O)NC1(C(=O)NCC2(CCC=C)CC2)CCCC1 c1(C(=O)NCCC2(NC(=O)C(C3(O)CCCC3)F)CCC2)c[nH]c2cccnc12 CC1=NS(=O)(=O)N(C)C=C1C(=O)NC1(C)CCCN(C(c2ccc(F)o2)=O)C1 c1(C(=O)NC2C(C)CN(C(=O)C(C)(C)C#N)CC2)cnn2cc(C(N)=O)cnc12 C(=O)(C(C)(O)CNC(=O)CC1(C)CCN1C(=O)C(C1CCOCC1)C)OC C=CCN=c1[nH]cc(C(N2CCC(C(C)NC(C3(COC)CC=CC3)=O)C2)=O)s1 c1(CC(=O)NCCC)cc(F)ccc1C.C1(C)(C(N(CC)CC)=O)CCOC(C)C1 N1(C(CSCCNC(=O)C(F)C2CCOC2)=O)CCc2n[nH]cc2C1 c1(SC)ncc(C)c(=NCCC2(NC(C3CC3(F)Br)=O)CCOCC2)[nH]1 C1(C2CCN(C(=O)CN3CCOCC3)CC2)(NC(C2NC(=O)C(F)C2)=O)CC1 c1(CC)ncc(Br)cc1C(=O)NCC#CCNC(=O)C(F)C1CCOC1 c1(CN2CCC(NC(C(CC)(C)C)=O)CC2)cn(CC(C)C)c2ccccc12 C12(NC(CC(CC)(F)F)=O)CCCC1CN(C(=O)C(n1nc(C)cc1C)C)C2 c1(C(=O)NCC(C)CN(C)C(c2n[nH]cc2Cl)=O)cn(C)c2c(Cl)cccc12 C(CCCCCN=c1cc(Cl)nc(O)[nH]1)NC(c1cnc(OC)nc1)=O C=CC(C)(C)CC(=O)NC1(CN2CCN(C(c3cc(C#N)on3)=O)CC2)CC1 C(=O)(CCCCC(N)=O)NC1CN(C(C2(C(C)C)C(C(=O)OC)C2)=O)CCC1F C12(CC)CN(S(=O)(=O)CC(C(F)F)N3CCOCC3)CC(Cc3ccccc3)(C1)C2 c1(CC(=O)NC(CN(C(CCN(C(CCC)C)C)=O)C)C)cc(Cl)cs1 C1(C(N(C(c2ccccc2)CNC(c2cscc2Br)=O)C)=O)CN2CCN1CC2 C1(C(N2C(CNC(c3ccnn3CC(F)F)=O)CCC2)=O)CCS(=O)(=O)C1 N1(C(c2c(C)nn[nH]2)=O)CC2CCCN(C(=O)CCC3CCCO3)C2C1 n1(CC)nc(C(=O)N(C)CC2(CNC(=O)C(c3cnn(C)c3)O)CC2)ccc1=O NC(=O)CC(O)C(=O)N1CC(CCCCNC(=O)CCOC2CCCOC2)C1 N1CC2c3ccoc3CN2C1.Brc1ncsc1-c1nnc(Cc2ccccc2)o1 N1(C(c2nnn(CC)c2C)=O)CCCCC12CN(C(=O)C(C)C(F)F)C2 C1(C)(C(=O)NCCCC(C)NC(c2cc(C)n(C(C)C)n2)=O)CCCCNC1=O Cc1cn2[nH]c(=NC(=O)c3ccc(-c4ccncc4)nc3)cc(C)c2n1 N1(C(C2C(OCC)C2C)=O)CC2(C1)SCCC2NC(=O)Cc1cc(C)sc1C N1(C(C2CCCCC2O)=O)CCC2CCCC12C(N1CC2CC=CCC2C1)=O C1(NC(c2c(CC)cns2)=O)C=CCN(C(=O)C=CC2CCOC2)C1 C1(c2c(C(=O)OC)cccc2)CC(N=c2[nH]c3cccnc3s2)CCO1 C1(CNC(=O)CSC(F)F)CC2(CCC2)CN1C(=O)CN1CCCCCC1 C1(NC(c2ncc(C)nc2)=O)CCN(C(c2cc(C3(C)CC3)n[nH]2)=O)C1(C)C C1(NC(c2cnc(C(C)=O)s2)=O)CN(C(C2CCC(O)C2)=O)C2(CCCOC2)C1 C(CC(C)C(=O)N1CCCC1CN(C(=O)CC12COCC(C1)C2)C1CC1)=CC C1(CN(C(C(C)C2CC2)=O)C)CCN(C(=O)CC(F)(F)Cl)CC1 C1(COC)(NC(=O)Cc2c[nH]ccc2=O)CCCN(C(C2(c3cccs3)CC2)=O)C1 N1(C(C(C)OCCOC)=O)CCN(C(=O)C=CC2CCC2)C(C2CCCC2)C1 CC(C)(C)CC(O)C(=O)NCC1(F)CN(C(c2ccn(C3CCCC3)n2)=O)C1 c1(NC(=O)Nc2ccc(C)c(CO)c2)ccc2c(c1)C(=O)N(C(C)C(C)C)C2=O C(=O)(C(C1=CCC(C(C)(C)C)CC1)N1CCC(C(=O)NC2CCCC2)C(F)C1)NC c1(OC(C(=O)NCCC(C)N(C(CC(=C=C)C)=O)C)C)ccc2ccccc2c1 c1(CC(=O)N(C2CN(C(c3n[nH]c4c3CCCC4)=O)C2)C)n[nH]c2c1CCCC2 N1(C(C2C(C)C2)=O)CC(CC(=O)NCc2ncc(F)cc2F)C2(CC2)C1 CCCCCC(O)C(=O)NCC12CC1CN(C(=O)Cc1ccc(C)c(OC)c1)C2 N1(C(c2cc(C(=O)Nc3cc(Cl)c(Br)c(Cl)c3)[nH]n2)=O)CCC2(CC1)OCCO2 C1(COC(C)(C)C)CN(C(N2CC(F)(CC)C2)=O)CC(C)(C)O1 N1(C(CCCCN(C)C)=O)CCCC(O)(CCNC(c2ccnc(Cl)n2)=O)C1 N1(C(COc2cncc(C)n2)=O)CCN(C(=O)CCc2ccccc2)C(C#N)C1 C1(CNC(CSCC(N)=O)=O)CC(CNC(=O)C(O)C2CCCC2)C1 C(=O)(CC1C(=O)Nc2cc(OC)ccc21)NC(CNC(C(C#C)(C)C)=O)CC=C N1(C(CC2CC(OC)C2)=O)CCOCC(NC(C2(n3nccn3)CC2)=O)C1 C1(C)(CNC(COCCCC)=O)CC(CC)CN1C(c1cn(CC(F)F)cn1)=O c1(C(N2CC(NC(CN(CCOC)C)=O)C(F)C2)=O)ccnc2nc(C)nn12 c1(C(N(C(CNC(CCCOC)=O)C)C)=O)cnc2nccn2c1 CC(C)C(CCN(C(=O)C(C)(C)C1CC1)C)NC(C1(C)CC(=O)C1)=O Cc1noc(C)c1CC(=O)NCC12CC(NC(c3cnc(C4CC4)[nH]3)=O)(CO1)C2 C(=O)(C(C)(C)CF)NC(CC)CN(C(C1CN(CC(F)(F)F)C1)=O)CC C1(C)(C(=O)NCC(CC)NC(c2cc(CC3CCC3)c[nH]2)=O)CCSCC1 C1(NC(C(COC)O)=O)CN(C(c2cc(Br)n3cc[nH]c23)=O)CC12CCC2 N1(C(C(COC)C)=O)CCCC(CO)(NC(c2cc(C)nc(O)n2)=O)C1 CC(CC(=O)ONC(c1ccc(P(C)(C)=O)s1)=O)C(C)(C)C.N1CCOCC1 C(c1ccc(Cl)cc1)=CC(=O)Nc1scc(C(=O)NC2CCC(OC)CC2)n1 c1(C(=O)NC(C2CCCCN2C(=O)CCc2cncn2C)C)cc(O)cc(F)c1 C1(C(=O)NC(C)CNC(C2CCC(C)(C)OC2)=O)CCc2nccn2C1 C=CC1(C(=O)NCC(CCOC)NC(N2CCC(SC)C2=O)=O)CCOCC1 N1(CCCNC(c2c(C)coc2)=O)CCN(C(=O)CCc2cncs2)CC1 C1(CC(=O)NC(C(C)C)c2ncc[nH]2)CN(C(=O)C=CC(F)F)C(C)(C)C1 CC1CCCC=C1C(=O)N(C)CC1(O)CN(C(=O)CCC2CCCC(=O)N2)C1 CC1CCCN(C(=O)CCc2ncc(F)cn2)C1CNC(=O)Cc1csc(S)n1 C1(O)(C(C)(C)NC(C=C(C)C(F)F)=O)CN(C(=O)COCc2ccncc2)C1 CCC(C)C(=O)C(=O)N1CC2C(C(=O)Nc3cnccc3OC)C2C1 C1(C(=O)NC(C2(O)CN(C(c3ccsc3Cl)=O)C2)C)Cc2nccn2C1 Cc1nncc(CNC(C2CCCN(C(c3c(F)cccc3F)=O)CC2)=O)c1C C(=O)(NNc1ccc(S(C)(=O)=O)cc1)NCCc1c(OC)ccc(O)c1 C1(O)(CNC(CCNC(=O)C=CCl)=O)CCCN(C(c2ccc(CO)s2)=O)C1 c1(C(=O)NCC(C)(C2CC2)NC(C2N(CC)CC2)=O)ccc(C2CC2)nc1O c1(CC(C(=O)NC(c2noc(CCc3ccccc3)n2)C)=O)ccc(Cl)cc1 C(=O)(CC1CCOc2ccccc21)NCCn1nc(C)n(CC)c1=O c1(C(=O)NCCCN(C(C)C)C(C2C(F)(F)C23CC3)=O)cnoc1-c1cccs1 C#CCCCCCCC(=O)NC(C)(C)C(C)CC(=O)NCCc1c(C)noc1C N1(C(C(CC2CC2)OC)=O)CCN(C(=O)C(=O)Nc2ccccc2)CC1C c1(N(C)C(=O)NCCNC2CCCN(c3cccc(F)c3)C2)cc(Br)ccc1Cl C1(CC)CN(CS(=O)(=O)CF)CCN1C Cc1ccncc1C=CC(=O)NCC1CN(C(=O)CCOCC2CC2)CCN1C C(=O)(C1=NOC(C)(C)C1)NC1CCC(C)(NC(C2(C)CC3CCC2O3)=O)CC1 CC1C=C(C(=O)N2CCN(CCCNC(c3coc(C4CCC4)n3)=O)CC2)CC1 S(=O)(=O)(c1c(C)noc1C)c1nnc(-c2c(C#C)nc(Cl)cc2)o1 N1(C(C(C)NC(C2CCCCS2)=O)=O)CC2CCC2(C)C1 C(=O)(C1=CC2CCCCCCC12)NC1(CCNC(c2c(C)csc2)=O)CC1 Oc1cccc(CNCC2CC23CCOC3)c1 C(=O)(C1CCCc2nn[nH]c21)NCCC(C)N(c1cc(=O)n(C)c(=O)n1C)C c1(CNC(C2CCCCC2(F)F)=O)cccc(Cl)c1O.C12CCC1C(=O)N2 c1(C(=O)NC(C(C)NC(C(C(=C)C)(C)C)=O)C)cc2c(Br)cccc2cn1 c1(C(=O)NC2(CO)CCCN(c3nnc(C(N)=O)s3)C2)ccnc2[nH]cnc12 Cc1nc(C(C)(C)C)ncc1C(=O)NCC(C)N(C)C(C1CCCCC(=O)C1)=O c1(OCC(=O)NCCN(C(Cc2c(C)cc(F)cc2)=O)C)c(C)cc(Cl)cc1C C=Cc1cncc(C(N2CC(CCO)(C(N3CCC(COC)CC3)=O)C2)=O)c1 c1(C(N2CC(C(C)NC(c3c(OC)cc(O)nc3)=O)C2)=O)cc2cc(Cl)sc2[nH]1 C(C(C)(C)C(=O)OCC)(c1nnnn1CCCOC)NC1C(CC=C)CCC1 N1(C(C(CCC)C)=O)CCc2sc(-c3cccc(NC(C)=O)c3)nc2C1 c1(C(=O)NCC2CN(C(C3CC(OC)(OC)C3)=O)CC2C)ccn2cccc2c1 Cc1ccc(C(F)(F)F)cc1NC(=O)NCC(N1CCOCC1)C N1(C(c2nc(C)sc2)=O)CCOCC1CNC(C1CCCN1C(=O)C(C)C)=O C1(OC)CN(C(C2(C#N)CC2)=O)CC1NC(c1cc(CC(C)C)c[nH]1)=O c1(C(=O)OC)cc(=NC2CCn3c(O)nnc3C2)nc2[nH][nH]cc1-2 N1(C(Cn2c(CCC)ncc2)=O)CCN(C(C2(F)CCOCC2)=O)CC(C)C1 c1(N2CC(C(=O)OCC)C3C(C2)CCCC3)nc(O)n(C)c(=O)c1[N+](=O)[O-] c1(OCCOC)ccc(CC(=O)NC2CC2NC(C2CC23CC(O)C3)=O)cc1 Cc1cccc2[nH]c(C(=O)NC3CC(CO)N(C(c4ccon4)=O)C3)cc12 n1(CCC)cc(Cl)c(C(=O)NCC2CC2NC(=O)C2=NOCC2)n1 CCCCC(C)(F)C(=O)N1CC(C(=O)NCCC(C)N2CCC2)C2(CC2)C1 C1(C)(CC(=O)NC(CN(C(=O)CCOc2cccnc2)CC)C)CCC(=O)N1C C1(NC(C2(CC=C)CN(C(c3cc(Cl)ns3)=O)C2)=O)CC(C)(C)C12CCC2 N1(C(C2C(C)(C(C)C)C2)=O)CCC(CN(C)C(C2CCCCN2C)=O)CC1 c1(C(C(=O)NCC(C(C)C)NC(c2ccoc2)=O)OC)c(F)cccc1F C1(F)(CNC(c2cnc(C)s2)=O)CCC(CNC(C2(Br)CC2)=O)C1 N1(C(C2CCN(C(C(CCC)NC(N)=O)=O)C2C)=O)CCOCC(C)(C)C1 Nc1cc(Cl)ncc1C(N1CCN(C(c2cnnc(O)c2)=O)C2CC12)=O c1(C(=O)NC(C)C(CO)NC(=O)C(=O)NCC(F)F)ccc(C2CC2(F)F)cc1 c1(OC)cccc(N2CCN(C(=O)CSc3occc3Br)CC2)n1 c1(C(=O)NCC23CCC2CN(C(=O)CC(F)(F)F)C3)ccc2nccn2n1 Cc1ccccc1OCCCN(C)CC1CCCN(C(C2CC=CCC2)=O)C1 Cc1ccc(C)c(C(C2CC2)NS(=O)(=O)CC2CCCCO2)c1 CC1(C)CC2(CC(NC(C3CCN(C(=O)CN4C(=O)CCC4=O)C3)=O)C2)C1 c1(C(=O)NCC(C2CCC2)NC(CCC(CC)OC)=O)n[nH]c2c(C)cccc12 N1(c2nccc(C)n2)CC2(COC(CNC(C3NC(=O)CC3C)=O)C2)C1 c1(C(N)=O)cccc(C(=O)NCCC2CCC(NC(c3nsnc3O)=O)C2)n1 c1(C(=O)NCC2(c3cncs3)CC2)c[nH]c2cc(F)ccc12.C12CC(C1)C(=O)NC2 c1(C2CCN(c3nnc(C(C=CCC)O)n3CC)CC2)cccc(F)c1F Cc1[nH]nc(C(N2CC3C(NCc4cccc(C(F)(F)F)c4)C3C2)=O)c1C c1(C(C)(C)C)cc(CNC2CCCNC2)on1 C1(CNC(C=C(C)C)=O)CCCC1NC(c1cn(C(C)C)nn1)=O c1(C(=O)NC2C(C)CCN(C(=O)CC3CCC4CC34)C2C)ccc2ccccc2n1 C1(CNC(CC(C)(C)SC)=O)CC2(CCC2)CN1C(c1ccc(C(F)F)cc1)=O C=C(F)C1(CC(N2CCC=CC2C(=O)NCC2(C)COCCO2)=O)CCC1 c1(CC(C(=O)O)NC(=O)C=Cc2ccsc2)ccc2[nH]ccc2c1 c1(C(=O)NC(CCNC(C#CC(C)C)=O)C)ccc2c(n1)NCC(=O)N2 N1(C(C2N(CC#C)CCC2)=O)CCN(CCCCCNC(=O)C=CC=CC)CC1 C1(C(=O)NC(C2CCCN2C(C2CCC(C)(C)CC2)=O)C)Cc2ccncc2N1 CC1=C(C(=O)N2CCC(CNC(C3(CC(C)C)CCCC3)=O)C2(C)C)CCCO1 N1(C(C2CC(CC)OCC2)=O)CCC(C2(NC(C3(F)CCOC3)=O)CC2)CC1 C1(NC(Cc2c(C)noc2)=O)CC(NC(=O)C(C)OCCC(C)C)CC1O c1(C(=O)NCC2(C(N)=O)CN(C(c3ccc(SC)o3)=O)C2)c(C)ccc(C)c1O c1(C(=O)OC)cnc(N(CC(C)CNC(=O)Cc2ccc(F)cn2)C)cn1 c1(C(=O)OC)cc(F)c(NC(=O)C(=O)NCC2(CC(F)F)CC2)c(Br)c1 C1(C(CNC(C(C)NC(CC)=O)=O)C)CCN(C(c2nc(Cl)sc2C)=O)CC1 C1(NC(C2ON=C(C(C)C)C2)=O)(CNC(c2cncs2)=O)Cc2ccccc2C1 c1(NC(c2c(C)ocn2)=O)nc(Cl)ccc1C(=O)NC(CO)C1CC1 C(=O)(C1=CC2(CCOC2)C1)N1CCC(N(CC#C)C(c2ncc(F)cc2C)=O)C1 Cn1cnc(Cl)c1C(N1CCC(C(N)=O)C1)C(=O)NCC1CCCO1 c1(C(=O)NCC2(O)CCN(C(C(C(C)C)n3cnnc3)=O)C2)cccc(N)c1F C1(C(C)(C)C)COCCN1C(C(=O)NC1CC1)C1CCCC1 C1(NC(Cc2c(C)nc[nH]2)=O)CCN(c2nc(C(C)C)ns2)C1(C)C c1(C2C(NC(C(C)NC(CC)=O)=O)CCC2)cccc(C(=O)OC)c1F O=C1CCC(NC(=O)Cc2csc(-c3ccccn3)n2)C(=O)N1 C1(NC(C(c2cccc(OC)c2)N(CCCCC)CCC)=O)CC2CCC(C1)C2 C1(NC(c2c(CC)onc2)=O)CCN(Cc2cn(-c3cc[nH]c(=N)c3)nn2)CC1 N1(C(Cc2cc(CC(C)C)on2)=O)CCCN(C(=O)CC2CCCCN2C)CC1 C#CC1(F)CN(C(C2CCOC2CNC(=O)CC2CCSC2)=O)C1 c1(OC)ccc(NC(N2CCCCC2CC2CCCN2C)=O)c(Br)n1 C(=O)(C(CC1CCCC(OC(F)(F)F)C1)CC(C)C)NCCC(CCC)C1CC1 CC(CC(=O)NC1CN(C(c2ccnc(OC(C)C)c2F)=O)CC1C)C(F)(F)F N1(C(C2C=CCC2)C)CCC2(CC1)CN(C(=O)C(F)(F)C(F)(F)F)CCO2 c1(OC)cccc(C(C)C(N2CCCC(NC(C3CC(=C4CC4)C3)=O)C2)=O)c1 S(=O)(=O)(c1cc(Br)c(Br)s1)N1CC2N(C(c3ccc(F)cc3Br)=O)C2C1 N1(C(c2cc(CC)n(C)n2)=O)CCCC(CC)(NC(=O)C=Cc2ccccc2)C1 CC1(CNS(=O)(=O)CC2(C)CCCN2)Cc2ccccc2C1 Cc1cc(C(=O)NC2CC(NC(C3CCCC(C)(C)O3)=O)C2)cc(C)n1 Cc1nnnn1CC(=O)NCCC(C)N(C(=O)C(C)N1CCC1)C c1(CC)cc(C(=O)NC2C3CC2N(C(c2cnccc2C)=O)C3)cc(F)c1 CCC(Cc1ccccc1)C(=O)N1CCC(CNC(=O)CSCc2ncc[nH]2)C1 c1(C(N2C(CCNC(C(C)NC(=O)OC)=O)CCCC2)=O)ccc2c(c1)CCC2 CC1CN(C(=O)CCCN(C)C(N)=O)CCN1C(C1CNC(=O)O1)=O C1(CNC(C(CC)SC)=O)(NC(=O)CC(=O)N(C)C)CC2CCC1C2 c1(OC)ccc(CC(N)C(=O)N2CCC2(C)CCO)c(OC)c1OC c1(C(=O)NC(C2N(C(C(C)c3ccsn3)=O)CCC2)(C)C)ccnc2[nH]ncc12 N1(c2nnc(C(C)(C)C)o2)CC(C)(C)CCC1CNC(=O)C(C1(O)CCCC1)F C(CC(F)F)(C(=O)N1CCN(CC)C(C)C1)NC(C(CCC)N(C)C)=O N1(C(c2scc(COC)c2)=O)CCOCC(NC(C2CCCCN2C)=O)C1 Cn1nc(C(=O)NCCNC(c2ccnc(-c3ccco3)c2)=O)cc1C(F)(F)F C(C)(C)(C=CC(N1CC(c2cc[nH]n2)C1)=O)N(C(C1C(=C)C1)=O)CC CC1CCN(C(c2ccc(Cl)c(F)c2N)=O)C(C)C1NC(c1ccccc1O)=O Cc1cnc(C(=O)NCC2(C)CCN(C(=O)C(C)(C)c3ccsc3)C2)nc1 N1(C(CCC2(C#N)CCC2)=O)CC2(CCN(C(c3cnc4n3CCCC4)=O)C2)C1 C1(CC)CC(C(N2CCC(F)(C(N3CCN(C(=O)CO)CC3)=O)C2)=O)CCO1 C=C(CNC(=O)CCC1CCN(C(=O)CC2CC2C2CC2)C1)c1ccccc1 C(=O)(CC(C(C)(C)C)NC(c1n[nH]cc1C)=O)N1CCC(CCCC)C1 Cc1cc(C(N2CC(F)(F)CC2C(N2CC(C)C2)=O)=O)c(Br)cc1F C12(CNC(C=CC=CCC)=O)CN(C(c3n[nH]cc3Cl)=O)CC1(C(F)(F)F)C2 C1(CNC(c2cnc(C)s2)=O)CC2(CC2)CN1C(c1cncc(C(F)(F)F)c1)=O c1(C(N2CC3C(NC(=O)CCc4cncnc4)(C3)C2)=O)c(F)cc(Cl)cc1F c1(COC)cc(C)nc(N2CCC(C(C)(C)C)(C(=O)OC)C2)n1 n1(CC)cnnc1C1CCN(C(c2csc(C)n2)C(=O)NCCCSC)C1 N1(C(C2(C=C)CCN(C(=O)C(C)OC(C)=O)C2)=O)CC2CC(C1)C2(C)C c1(C(N2CC(C3(NC(c4c(C)cns4)=O)CC3)C2)=O)cccc2ncc(C)n12 C1(CC(=O)NC2CCCN(C(c3ccc(C(F)(F)F)s3)=O)C2)CCCC(F)(F)C1 C(=O)(C=C1SCC(=O)N1C)N1CC(NC(C(C)P(C)(C)=O)=O)C(F)C1 N1(C(COCC=C)=O)CCOCC1CCNC(=O)C=CCC(C)(C)OC n1(CCC)c(CNC(c2c(I)cnn2C)=O)nc2ccccc12 C(=O)(C1=C(C)CCC1)N1C(C)(CC(N2C(C(CC)O)CCC2)=O)CC1 Cc1[nH]c(C(N2CCC(O)(CN=c3[nH]nc(O)s3)CC2)=O)c(C)c1[N+](=O)[O-] CC1CC(NC(=O)COCC2CC2)CCN1C(C1CC1c1cnccn1)=O CCCCCC(CC)C(=O)NOCCN(C(=O)Cc1csc(COC)n1)CC.O CCCCCC(C)(CC)C(=O)NC(C)C(C)NC(=O)CCCNC(N)=O C1(C)(CNC(c2c(CC)ncs2)=O)CN(C(=O)CC(=O)Nc2nccs2)CCO1 C(=O)(N1CCCO1)NC(C1CC(OC)(OC)C1)=O.c1csc(C(C)=O)c1 c1(COC)nc(-c2ccnc(Sc3ccncc3)c2)n(C(C)COC(C)(C)C)n1 CC(C)(C)C#CC(=O)NC12CCC(C1)N(C(=O)CC1(N(C)C)CCCC1)C2 N1(C(c2c(OC)cccc2)=O)CC(C)(C)CC1CNC(=O)C(C)CC(C)C CC(C)(CC(=O)N1CC(NC(=O)CC2CCCCCO2)CC(F)C1)C(F)(F)F N1(C(CC(C)(F)F)=O)CCCN(C(C2CCC=CO2)=O)CC1 C1(C(N2C(CNC(C3(C(=O)NC)CCC3)=O)CCC2)=O)CC(=O)N(C(C)(C)C)C1 c1(C(N2CCN(C(C=CSC)=O)C(C3CCC3)C2)=O)cc(N)cc2ccccc12 C1(C(=O)NC(CN(C(C2CCC(=O)N2C)=O)CC)C)CCC(=O)N(CCOC)C1 CCC(CCCC(=O)N(C)Cc1ccn(C)c1)NC(c1oc(C)cc1C)=O N1(S(=O)(=O)C2CC(Cc3ccccc3)C2)CCOc2cc(F)ccc2C1 n1(CCC)ccc(C(=O)N(C2CCC(NC(c3nc(Cl)cs3)=O)C2)C)n1 C1(CC)CC(C)CN(C(C2CC(CNC(=O)C(O)CCSC)C2)=O)C1 C(=O)(C1=CCCCC1C)N1CC(CNC(c2c(C)noc2)=O)OCCC1 Cc1cc2cc(C(=O)N=c3cc(-c4ccccc4NCC4CC4)o[nH]3)ccc2[nH]1 C(=O)(C(F)(CNC(c1cnnn1CC)=O)C(C)C)N1CCC(=C)C1 C1(N(C(=O)CC2CSCCO2)C)CCCC(NC(=O)CC(C)(C)C2CC2)C1 C1(C(C)NC(=O)CCC2CC2)CC(C(C)(C)C)CN(C(c2cncn(C)c2=O)=O)C1 C1(C(=O)NC2CC(c3ccccc3)(NC(C(C)OCC)=O)C2)CCC(C#N)CC1 c1(CCC(=O)N(C2CCN(C(C3CCC(CC)C3)=O)CC2)C)ccc(N)c(F)c1 C1(C(=O)NCCN(C(CC2C(C)CCO2)=O)C2CC2)CC2C=CC1C21CC1 c1(CNC(=O)Cc2ccnc(Br)c2)cc(F)c(N2CCOCC2)c(F)c1 C(CCNC(C1CCC2(CC2)C1)=O)(C(=O)N1CC(OC(C)C)C1)OC C(C(O)C(C)(C)C)NC(C(CNC(c1c(CC)occ1)=O)N(C)C)=O Cc1ccsc1C=CC(=O)N(C(C)CNC(C1(NCCO)CC1)=O)C C1(NC(CC2C(C)(C)CCO2)=O)CC2CCC1N2C(c1ccnc(CO)c1)=O c1(C(=O)NCC(C)(CO)NC(C(COC)N(C)C)=O)cncn(C)c1=O c1(C(N(CCCN(C)C(C2(c3ccn(C)n3)CC2)=O)C)=O)ccc(F)nc1 C(C)(N=c1[nH]c(Cl)nc(CC)c1Cl)C1CN(C(C(CC)OC2CCCC2)=O)C1 C1(NC(=O)Cn2cnc(Br)c2Br)CC(C(=O)OC(C)(C)C)(C(=O)O)C1(C)C C(=O)(CC(O)CNC(=O)Cn1nc(C)cc1C)NC(CCCC)C C1(C)(C(=O)NC(CCCC)CC)CN(C(c2ncn(C(C)C)n2)=O)C(C)(C)C1 Cc1ccc2c(C(N3CCCC(CNC(=O)C(F)=C4CCC4)C3)=O)cnn2c1C c1(NC(C2CCCC(NC(C(CC)C)=O)C2)=O)cc(Cl)ccc1I c1(OCC(=O)NCC2(F)CC(CNC(=O)C3=CCC3)C2)ccccc1Cl CC1CN(C)CC(C(N2CCN(CCN(C)C(c3cn[nH]c3)=O)CC2)=O)O1 C12(CCNC3CCN(C(C)CC4CCCC4)CC3)CCC(CC1)C2(C)C c1(SC)nc2nc(C)c(CC(=O)NC3CCC3CNC(=O)C(C)C)c(C)n2n1 C12(C(=O)NCc3ccc(-c4ccccc4F)s3)C3C4C1C1C2C3C41 C1(CNC(Cn2cc(C(C)=O)nc2)=O)CN(C(C2CC3CCC2C3)=O)CC1C C1(C(C)C)C(=O)C2CCCCCC(CC)C(C)(C(=O)N2CC)N1 c1(C(=O)NC2C(NC(C3(CCCC)CC3)=O)CCC2)cc(CC)c(C)s1.C(=O)(C1CC1)N O=C(C1=CCN(C(c2sccc2CO)=O)C1)N1CC2CC1CN2C CS(=O)(=O)c1cccc(O)c1C(N1CCCC2(C1)CN(C(c1cnc[nH]1)=O)C2)=O CN1C(=O)NCC1C(=O)NC(CNC(c1cnc(CC2CC2)s1)=O)C1CCC1 C1(C(N(CCNC(=O)C=CC(F)(F)F)Cc2ccccc2)=O)CC=CCC1 C(=O)(CC(C)(O)c1ccccc1)NCCC(=C)CNC(=O)CCC(=O)NCC CCCC(C)(O)C(=O)N1CCC(NC(=O)CCCn2nc(C)nc2C)C(C)C1 c1(-c2scc(C(=O)OC)c2)ccc2oc(CC(C)C)cc(=O)c2c1 c1(C(=O)NCCCc2ccc(C#N)cc2)ccc2nc(C3CC3)[nH]c2c1 c1(C(N(C2CCN(C(CCC=C)=O)C2)C)=O)sc(N(C)C)nc1Br C1(CN(C(C2(CC#C)CCCC2)=O)C)COCCN1C(c1cc(Cl)n[nH]1)=O Cc1nc(C(F)(F)F)oc1C(=O)NCC(C)(CO)NC(C1CCC(C)O1)=O C(=O)(CCCC(F)(F)F)NC(C(C)NC(c1cc(CO)[nH]n1)=O)(C)C Cc1cc(C(=O)N(CCC(C)NC(c2nc(C(C)(F)F)cs2)=O)C)co1 N1(C(CN(CCC)C)=O)CC(NC(c2ccn(CC(F)F)n2)=O)C2CCCCC12 CCCCCCCC(=O)NCCC1C(C)CCCN1C(c1cc(OC)ncn1)=O C1(NC(C(C)C)=O)CCC(N2CCN(C(C3CC4(CC4)CO3)=O)CC2)CC1 c1(C(N2CC(NC(c3cc(CC)n(C)n3)=O)C2)=O)ccc2cc(O)ccc2n1 N1(C(C2(CC)COC2)=O)CCC(C2CN(C(C3(C)CCCOC3)=O)C2)CC1 N1(C(C2CCC(=O)O2)=O)CCN(CC(N2CCCC(Cn3cncn3)C2)=O)CC1 c1(C(=O)NCC2(C)N(C(CCC(=O)OCC)=O)CCC2)cn2c(n1)COCC2 Cc1noc(CCCC(=O)NC2CC(NC(=O)C(C)NC(=O)C(C)(C)C)C2)n1 c1(NC)ncccc1CNC(=O)COCc1cccc(OCC2CCOCC2)c1 Cc1nc(NCC(C2CCCC2)C)cc(N2CCOC(c3ccc(F)cc3)C2)n1 c1(C(=O)NC(CC)CN(C)C(C2(C)C=CCC2)=O)ccc([N+](=O)[O-])cc1C C1(C)(CNC(C(c2ccc(Cl)cc2)C)=O)CCCN1C(=O)CNc1nccs1 C1(NC(C(C(C)(F)F)F)=O)CC2CC(NC(=O)C=Cc3ccoc3)CC2C1 C1(NC(c2nc(C(C)C)oc2)=O)CS(=O)(=O)CC1NC(c1cc(C(N)=O)c[nH]1)=O C(=O)(C1CCCc2n[nH]cc21)N(CC(C)(C)NC(C(CCCC)NC(N)=O)=O)C c1(C(=O)OCC)cc(Br)c(-c2nn[nH]n2)cc1F.c12nnn(CC)c1NC2=O C1(C(C)(C)C)CC(CNC(=O)Cc2cccc(F)c2)CN(C(c2occc2Br)=O)C1 c1(CNC(N2CCC(N(CC)CC)C2=O)=O)c(F)c(F)c(F)c(F)c1F c1(CC)cnccc1C(=O)N(C)CCN(C(C1SCCC1C)=O)C(C)C C1(NC(COCCC)=O)CN(C(c2cc(S(C)(=O)=O)oc2C)=O)CC2(CCC2)C1 C(=O)(C1=C(Cl)CC1)NC(C1N(C(C(c2cnccn2)C)=O)CCC1)C N(C1CCCc2ncccc21)C(=O)NCC1CCC(SCCC(=O)OC)CC1 C(c1ccccn1)=C(C(=O)NCC12CC(NC(Cc3snc(C)n3)=O)(C1)C2)F N1(C(C2N(C(C)=O)CCC2)=O)CCN(C(C2COC(C)(C)C2)=O)CC(O)C1 C1(OC)CCN(C(=O)COCCO)CC1.C1(=O)CC(C2CCCCC2)N1.C1(S)CC1 CCCCC(CC)C(=O)N(CCCNC(C1COCCN1C)=O)CCO c1(C(=O)NC(C2CCCN2C(c2ccncc2F)=O)(C)C)cc2n(c1)CCSC2 C(=O)(C(C)(C)CCCF)NC1CC(CC(=O)NCc2cnc(OCC)nc2)C1 c1(C(=O)NC2(CF)CCN(C(c3nc(OC)oc3)=O)C2)cc2n(n1)CCO2 CCCCC(O)CC(=O)NCC(C(=O)NC(C)C(=O)OC(C)C)N(C)C C1(C(=O)NC2CCC(CCC(=O)N(CC(C)O)C)C2)CC2(CCC2=O)C1 c1(OC2(C(=O)NC(C)C(C)NC(=O)CCn3cccc3)CC2)ccccc1 c1(CC)cc(C(=O)N(CC(C)C#N)CC(C)C)c(C)o1 C1(NC(c2cncc(OC)c2)=O)CCCC2CN(C(=O)CCC(CF)CF)CC12 N1(C(C=CC)=O)CCC2(CCC2)C(CNC(=O)Cc2cnc(Cl)cc2C)C1 C(=O)(C(C(C)C)N(C)C)NCC=CCOC.C12CCCC1CNC(=O)C2 CC1(C)CC(O)C(O)CN1C(N1CC2(CCC2)C1(C)C)=O C12(NC(C(CCSC)NC=O)=O)CCCC1N(C(=O)CCCn1cncn1)CC2 CCC(CC(=O)N(CCCC(=O)N1C(C(=O)OC)CC1C)C)C(F)F c1(C(=O)NCC(CN(C)C(c2nn(C)cc2Cl)=O)(C)C)ncccc1O CC1(C)CCCC1(c1nnnn1-c1ccc(Cl)cc1)NCCCF c1(N(CC(F)Cl)C)nc2ccc(S(=O)(=O)NCC3CC(O)CCO3)cc2s1 c1(OC)cc(CC(N2CCC3(NC(=O)C(C4CCC4)OC)CC23)=O)c(F)cc1O c1(C(=O)NC(C2(O)CN(C(=O)CC3CC(O)C3(C)C)C2)C)cccc2c1nnn2C N1(C(=O)CCOC2CCCC2NC(C2CCCC2)=O)CCOC(CF)C1 C(C(C)C(C)C(=O)NC1CC(CC(N)=O)C1)OC.C12CCCCC1CCC(=O)N2 C(C(=O)NC(c1cc(C)on1)C)(C(C)CC)N(C(c1c(NC)scn1)=O)C C1(NC(Cc2c(C)cnn2C)=O)CCCCC12CCN(C(c1cccnc1)=O)C2 C(=O)(CC(CC(C)C)NC(C1CCC(=O)NC1)=O)NCC(=O)OCC#C C1(NC(c2c(CNC(c3cc(C)nnc3)=O)n[nH]c2)=O)CCCC1N=[N+]=[N-] c1(OC)ccc(Cl)c(C(=O)NC2CN(C(c3cc(C4CC4)nn3C)=O)CC2(C)C)n1 C1(NC(C2C(C)C2)=O)CCN(C(=O)C=C2CCC(C(C)(C)C)CC2)C(C)C1 Cc1ncncc1C(N1CCOC(Cn2cc(CNC3CCC3)nn2)C1)=O N1(C(C2(COC)COC2)=O)CCC2CN(C(=O)Cc3cc[nH]c3)CCC2C1 C(=O)(CCC(F)(F)C(F)(F)F)N1CC(CNC(C2N(C)CCC2)=O)OC(C)(C)C1 Cc1ccc(C(=O)NCCOCCNC(=O)C(N2CCC(C)C2)=O)nn1 Cc1cc(C(=O)N(C)CC2CCCN2C(c2nocc2C)=O)cnc1OC(F)F CCC(F)(C(=O)OC)C(=O)N1CCN(C(=O)C#CC(C)(C)O)C(CCO)C1 N1(C(Cc2c(C)nc(C)s2)=O)CCC(NC(=O)CSCCN(C)C)CC(O)C1 CC(C)C(C(=O)NCC1(F)CN(C(=O)CC2CCC(C)(C)O2)C1)c1ccccc1 c1(C(=O)NC(CC(C)NC(C(CCC)N(C)C)=O)C)ccc2oc(O)nc2c1 C#CC1(CNC(C2C(CC)CCN2C(=O)C(C)S(N)(=O)=O)=O)CCOCC1 CC1(C(=O)NCC(C)(C)CNC(=O)CC2(N(C)C)COC2)CCC2(CC1)CC2 c1(C(=O)NCC(=O)N(O)Cc2cn(CC(F)(F)CO)nn2)ccc(Br)c(Br)c1 CC1CCN(C(=O)CCc2ccoc2)C1C(=O)NCCc1cccc(F)c1 C12(NC(COC(C)C)=O)CCCC1N(C(=O)C(F)(F)c1cscn1)CC2 c1(C(N2CCN(C(C(CC)OCC)=O)C(C)C2)=O)cccc2[nH]c(=N)oc12 N1(C(C(CONC(=O)OC(C)(C)C)F)=O)CCN(OC(C)(C)C)CC1CC(F)F C(C)(CCC(=O)NCC(C)(C)CN(C)C(c1cccc(F)c1)=O)OC N1(C(C23CC(NC(=O)CC4(O)CCC4)(C2)C3)=O)CCN2C(=O)OCC2C1 N1(C(C(c2n(C)cnc2)O)=O)CC2OCC(NC(=O)C=CC3CCC3)C2C1 O=C(C#CC1CCOC1)N1CCN(C(=O)Cc2cc[nH]n2)C(c2cn[nH]c2)C1 CC1CC(CNC(=O)CN(C)C(c2ccoc2)=O)CN1C(c1cc[nH]c(=N)c1)=O CC(CN(C)C)CCC(=O)N1CCOC(C(=O)NCC2OC(=O)CC2(C)C)C1 c1(C(=O)OCC)cccnc1N1CCC(CN(C)C(C2CCOC2)=O)C1 C(C)(CCC(=O)NC1(C(=O)NCCCCSC)CC(O)C1)OC C(=O)(CC(C)(C)C)N1C(CCc2cn(C(CC)CC)nn2)CCC1 C=C(C)CC(=O)NC1CCCC1NC(c1ccn(C)c1)=O C#CC1N(C(C2(C3CN(C(=O)COC)CCO3)CC2)=O)CC1(C)C N1(C(c2cncc(OC)n2)=O)CC2OCC(NC(=O)C(C)c3ccco3)C2C1 C=CC(CC)CC(=O)NC(C)(C)CCCNC(=O)C(c1cccc(Cl)c1)O C1(C(=O)Nc2c(O)ccc(C)c2)CCN(C(=O)Cn2nccc2C)O1 C=CC(C)CC(=O)NCC1(O)CCN(C(c2cc(Cl)c(Cl)[nH]2)=O)C1 C(C(C(C)(C)C)NC(C1CCN(C(C)C)CC1)=O)NC(C(C)OCCC(C)C)=O c1(C(=O)NCC#CCNC(C2(C)CC2)=O)ccc(-n2cc(Br)cn2)nn1 N1(C(C(CC)CC(F)(F)F)=O)CCCC2(CCN(C(C3(O)CCOC3)=O)CC2)C1 C(=O)(C(O)C(F)F)NCC(COC)NC(c1ccc(-n2ccnn2)cc1)=O C1(C(N2C(Cn3cc(-c4cn(C)nc4)nn3)C=CC2)=O)CC12CCOC2 c1(OC)ccnc(-c2n[nH]cc2CN2CCCC2C(=O)NC(CO)C(=O)OC)c1 c1(C(C(=O)NC2C(CNC(C(C3CCN(C)C3)C)=O)CC2)(F)F)ccc(F)c(F)c1 N1(C(=O)CC2CC2c2ccccc2)CC2CCN(C(C34CC(F)C3C4)=O)CC12 C(=O)(C(F)(F)c1ccccc1)NCC(CN(C)C(C12CC(F)C1C2)=O)O CC1(C(=O)N(CCCNC(c2ccc(C#N)o2)=O)CCO)CC=CCC1 C1(NC(c2ccnc(Cl)n2)=O)CC2CCC(C1)N2C(=O)Cc1ccccc1F c1(CC2CCN2N(C)Cc2c(OC)ccc(C(=O)OC)c2)ccc(C#N)cc1Br C1(C(=O)NCC(N2CCCC2)C)CC(=O)CN1C(=O)C=Cc1cnccn1 Cc1cc(C(N2CC(C)C2C(N2CCC(F)(F)C2)=O)=O)c(C)o1 C12(C(N(CC(CNC(Cc3nc(CC)sc3)=O)O)C)=O)COCC1C2(F)F C1(C(=O)NC(C)CC2CN(C(C34CCC(CC3)O4)=O)C2)CC2(CCCC2)CO1 CC1CCC(C(=O)N(CCN(C(=O)CCCc2nc(C(C)C)no2)C)C(C)C)S1 N1(C(c2c(C)nc(SC)o2)=O)CC2CC(N3CCOC(C(=O)OC)C3)C1C2 N1(C(Cc2c(C)nn(C)c2)=O)CCOCC(C(N2CC3(CC3)CC2C)=O)C1 c1(C(=O)NC2CC3CC(NC(C4C(C)(C)OCC4)=O)C3C2)cc2ccncc2o1 C1(NC(c2c(CC)[nH]cc2)=O)CN(C(c2cc(Cl)cnc2O)=O)C2CCCC12 N1(C(C(CC)F)=O)CCC(NC(C2CCCCN2C(C2CCCC2)=O)=O)C(F)C1 c1(CC(=O)N(CC(CN(C(C2C(OCC)C2)=O)C)O)C)cc(C)cc(F)c1 N1(C(CCC(COC)C)=O)CC2CCC(C1)N2C(=O)C(O)C(F)(F)F C(=O)(C(C)C(C)(F)F)NCC(C)N(C(c1ccc(C(=O)OC)cn1)=O)C N1(C(C(NOC)=O)=O)CCC(C)(C)C1CC(=O)NC1CCSC1 Cn1cnc(S(N)(=O)=O)c1C(=O)NC12CCC(CC1n1cc(CC3CC3)nn1)C2 C(=O)(C(CC(C)C)ONC(C1C2CCC(F)C12)=O)NCC=CCOC c1(CC)ccc(OCC(F)F)c(N2C3N(C4C(C3)C4)C2=O)c1.C(C(F)(F)F)OC N1(C(CCOC)=O)CCCC(N2CCN(C(c3cscn3)=O)CC2)C1 Cc1ccnc2c(NC(=O)Nc3ccc(CN4CCOCC4)cc3)cnn12 N1(C(C(C)C(C)(C)C)=O)CCCC2(CNC(c3cc(F)n[nH]3)=O)CCCC12 c1(CC(=O)OC(c2cc(Br)sn2)C)ccc(F)c(F)c1F c1(C(N(C(=O)C(C)(C)C2CC2)CCF)=O)nn(CC)cc1Cl C1(C(N2C(CC(=O)NC)CC2)=O)C2CC2CN1C(C1CC(=O)N1)=O c1(CC(N2CCC(C)(NC(=O)Cn3cnc(=N)[nH]3)C2)=O)ccc(S(N)(=O)=O)s1 N1(C(c2c(OC)nsc2)=O)CCC2(COC(CNC(=O)CC3(C)CC3(F)Cl)C2)C1 c1(OC)cc(C(F)(F)F)nn1CC(=O)OCC(c1ccc(I)cc1)(C)C C(=O)(C(F)(F)C(F)(F)F)N(C1CN(C(CCn2c(C)csc2=O)=O)CC12CC2)C N12CC(C(C)C1)N(C)CCC2=O.C1(C(C)=O)CCC1 c1(C(N2CCCCC(NC(CC(CC)OC)=O)C2)=O)c(O)cc(F)cc1F c1(CC(N2CC(CNC(C(C)=O)=O)OCC2)=O)cccc2cnccc12 c1(C(=O)NC(C2CCCN(C(CS(=O)(=O)NC)=O)C2)(C)C)cccc2nn[nH]c12 CCS(=O)CC(=O)N1CC(N(C)C(C2(c3ncco3)CCC2)=O)C(O)C1 CCC(C)(CNC(C1(C2CCCO2)CCCC1)=O)NC(=O)C(=O)NC1CC1 Cc1cccc(OCCSCc2cc(C(C)C)on2)c1 N1(C(C(CC(=C)Cl)NC(=O)Cc2cnns2)=O)CCC2(CCCC2)CC1 N1(C(C2(N(C)C)CCCC2)=O)CC2CC1CCC2NC(C1CSCC(=O)N1)=O c1(C(=O)NC2CC(C)(NC(c3cccc(CO)c3)=O)C2)cccc(Cl)c1Br c1(CN(C(=O)Cn2cc(CNC(C3CC3C(C)(F)F)=O)nn2)C)ccncn1 C1(CNC(C(C)OCC(F)(F)F)=O)(NC(=O)CCC2CCC2)CCC(C)(C)CC1 C1(NC(C2C(C(C)(F)F)C2)=O)CCCC(CC(=O)NCC(O)CCC2CC2)C1 N1(C(C2N(C)S(=O)(=O)CC2)=O)CC2=C(C1)CN(C(=O)C(Cl)=CCl)C2 C(=O)(C1=CC2(CCOC2)C1)NCC1N(C(C2(CCF)CC2)=O)CCN(C)C1 C(CC(C)(C)C(=O)N1CCC(CNC(=O)C(C)n2cnnn2)C(C)C1)OC C1(NC(C(CC)CC)=O)CC2CN(C(C3(OC)CCSC3)=O)CC12 N1(C(CCC=C)=O)CC2CCC1C(NC(c1ccc(S(N)(=O)=O)s1)=O)C2 C1(NC(C(C)OCC2CC2)=O)CN(C(=O)CCC=CBr)CC12CCCC2 c1(OC)ccc([N+](=O)[O-])cc1-c1nc(Cn2cncn2)nn1C(C)C(C)C Cc1nnn(CC(=O)NCC2CCCN2C(=O)CC2CC2)c(=O)c1CCN(C)C Cc1nc(C(=O)NC2CCN(C(=O)CCCN3CCCC3)C2)c(=O)[nH]c1C c1(C(=O)N)ccc(Cl)cc1.C(CC(=O)NCC1(N(C(=O)CCc2ccsc2)C)CC1)OC C(CCC(C)C(=O)NC1COCCC1C(=O)N(C)CC1CCN(C)CC1)OC N1(C(c2cc(CNC(C(C)OCC)=O)on2)=O)CCOCC(F)C1 C#Cc1ccc(C(=O)NC2CCN(C(c3cccc(F)c3Cl)=O)C2C)nc1 Cn1cc(C(=O)NC2CNCC2(C)C)c(-c2cnn(C)c2)n1 C1(c2ncc(C(=O)OC)s2)CCN(C(C)C(=O)NCCOCCO)CC1 C1(CNC(C2C=CCC2)=O)CC12CCN(C(C1CC1c1ccccc1)=O)CC2 CCCCS(=O)(=O)CC(=O)NC1CCCC1CNC(c1cnc(C)s1)=O C1(CC)CN(C(=O)CCc2nc(O)n[nH]2)CCN1C(=O)C(C(C)C)n1cnnn1 C12(CNC(Cc3cnc(C)[nH]3)=O)CCC1CN(C(c1cc(C(C)C)n(C)n1)=O)C2 c1(C(=O)NCCCCN(C)C(C2CC(F)CN2C)=O)cccc2ccsc12 N(C(=NCCCNc1cnnn1C)NNC1CC1C(C)(F)F)C(C)C N1(C(C2CC(=O)NC2)=O)CC2(CCOCC2C(N2CCC3COCC3C2)=O)C1 CN1C2CCCC1CC(CNC(=O)CCCOc1cccc(F)c1)C2 c1(C(N2CCC3(CC2)CC(O)C3)=O)cc(Br)cc2[nH]ncc12 N1(C(C(CCC)N(C)C)=O)CC(O)(C2(CNC(c3cc(C)n(CC)n3)=O)CC2)C1 N1(C(C(CC(C)=O)(C)C)=O)CC2(CCC2)CC1CNC(c1ccn(C(C)C)n1)=O C1(C(=O)NCC(c2cccc(F)c2)OCC)CCc2nnc(C)n2C1 C1(CNC(C=CC(CC)C)=O)CC(F)CN1C(c1cc(CN(C)C)c[nH]1)=O c1(C(=O)NC)cccc(NC(COCC#C)=O)c1.C12CCCN1C(=O)C21CC1 c1(C(=O)NC(C2CCN(C(C(CC)(C)F)=O)CC2)C)cc(NC(C)=O)cnc1O C1(NC(CSc2cn(C)nc2)=O)CC2CC(NC(C3CCCCO3)=O)CC12 C1(=CC(=O)NC(CC=C)CNC(C2(C)CCOC2)=O)CCN(C)CC1 N#Cc1ccc(-c2cn(CC3CC34CCSCC4)nn2)nc1 CCCC(C(=O)NCC1CCC(NC(c2sc(CC(F)(F)F)nc2C)=O)C1)OC C(=O)(C1OCCc2cc(C)ccc21)Nc1c(OCCC)ccc(F)c1 c1(C(N2CCC(C=C)(O)C2)C(=O)NC2CCC2)cc2ccccc2cn1 C1(C(CC)(C)C)CCC(C(N2CCC(O)(CNC(C3(C)CC=CC3)=O)C2)=O)CC1 C(C(C)CC(=O)NC1CN(C(c2cc(-c3cccn3C)[nH]n2)=O)CC1C)OC c1(C(N(C(C(=O)N(CCC(=O)NC)C)C)C)=O)ccc(CO)cn1 C1(NC(=O)NCCCC#C)CN(C(=O)C(C)Sc2ccccc2)CCC1(F)F N1(CC(C2CCC2)OC)CCC2(NC(C3CN4CCC3CC4)=O)CCCC12 C(CC(C)(C)C(=O)N1CC2CC(NC(c3ccc(F)cc3Cl)=O)C1C2)OC N1(C(C(F)OC)=O)CCOC2(CCC(NC(C3C=CCCC3)=O)CC2)C1 c1(C(N2CCCCC(NC(c3n(CC)ccc3)=O)C2)=O)cc(Cl)c(Br)cc1N Cc1ccc(F)cc1C(=O)OC1CC=CC1.C12CC(C1)CNC2=O C1(COC)CN(C(C23CCCC(C2)OC3)=O)CCN1C(=O)Cc1cnccc1C c1(N2C(CCNC(C3C(OC)C3)=O)CCCC2)cc(Cl)nc(-c2nccs2)n1 O=C(C1CCCc2ncccc21)NCCc1cc(Cl)c2c(c1)OCO2 Cc1c(C(N2CCC(NC(c3csnc3Cl)=O)C(CO)C2)=O)sc2ccccc12 C#CC1(C)CCN(C(C23CCCC2CCN3C(=O)COc2ccsc2)=O)CC1 c1(C(C)(O)C(=O)NCCC2CCN(C(=O)CCC3CC3)C2)ccc(Cl)cc1 C1(CNC(c2n(CC)cc(Cl)c2)=O)CCN(C(=O)Cn2nccn2)C(C)C1 c1(CN(C(=O)C=CCO)C)cnn2c1CN(C(C1CC(OC(F)(F)F)C1)=O)CC2 C(=O)(C1=NNC(=O)C1)NC1C(CC(=O)N(C(C(=O)OC)C)C2CC2)CCC1 c1(C(N2CC3N(C(c4c(C)nn(CC)c4C)=O)C3C2)=O)cccc2cnccc12 Cc1noc(Cl)c1CCC(=O)NCC(CO)NC(c1ccc(C2CC2)cn1)=O C(=O)(CC(O)CNC(c1ccc(Cl)cn1)=O)NCCN(C1CC1)CC C1(C(=O)NC2CCN(C(=O)C3CC4CC4C3)O2)OCC2CCC1C2 C1(NC(COC(CC)C)=O)CCC2CN(C(=O)C(C)SC(C)(C)C)CC2C1 CCC(CCC(=O)NC(COC)C(C)(C)C)NC(c1ccsn1)=O C1(NC(C(C=C)(F)F)=O)CC2(C(=O)N(CCC3CC3)CC)COC1C2 c1(OCC(=O)NCC2CCC(c3ccccc3)C2)ccc(Cl)cc1F c1(C(=O)NC(CCC)C(=O)NCC(N2CCOCC2)C)cnn(C)c(=O)c1 c1(OC)ccc(Cl)c(Cl)c1CC(=O)NC1CC2CC(C1)N(C(=O)C(C)O)C2 c1(NC(C2CCCN(C(=O)OC(C)(C)C)C2)=O)ccc(NC(=O)CC2CC2)cc1 CC(CC(=O)NC12CC(CNC(C3CCCS3)=O)(C1)OC2(C)C)C(C)(C)C C1(OC)CC(CCNC(c2ccnn2C)=O)N(C(C2CCC(C(N)=O)O2)=O)C1 N1(C(c2cc(C)[nH]n2)=O)CCCC12CCCN(C(c1cccc3nc[nH]c13)=O)C2 C12(NC(C(C)OC)=O)CCCC1CN(C(C13CCCC1CCC3)=O)C2 C1(CC(=O)NCC2(C(=O)NC3(CO)CC(C)C3)CCCO2)CCOC1(C)C c1(N2CCOCC(CNC(C(COC)(C)C)=O)C2)ccnc2ncnn12 c1(OC)ccc(CC(C)C(=O)N2CC(CN(C(=O)CC(C)C)C)C2)cc1 c1(CN(C(c2cc(F)ccc2OC)CC)C)ccc(C)cc1Br.OC C1(C(N2C(NC(c3c(C)con3)=O)CC2)=O)CCCCN1C(N1CSCC1=O)=O C(COC(C)C)(C(=O)N1CCCC1C(C)NC(=O)C(C)(C)N(C)C)NC(C)=O Cc1c(C(=O)N(C)CC2CCN(C(C3(C)CC(C)C3)=O)CC2)c(Cl)nn1C C1(CCNC(C2(C(=O)OC)CC2)=O)CCN(C(c2[nH]cnc2C2CC2)=O)C1 C(=O)(C(O)CCC(F)(F)F)NCC1CCCN(C(COCc2cc(C)on2)=O)C1 c1(C(=O)NCCCN(C(C(Br)=C(C)C)=O)C(C)C)cc(N)ccc1F C(c1c(C)cc(C)cc1C)=CC(=O)N(CCNC(c1cccc(CO)c1)=O)CC CC1N(C(C23CCN(C(=O)Cc4ccn(C)c4)CCC2C3)=O)CCCC1(C)C N1(C(CCC#C)=O)CC2ON=C(CNC(c3cn(C(C)C)nc3C(F)F)=O)C2C1 C#Cc1ccc(C(N2CCN(C(c3ocnc3C)=O)CC2CC)=O)cc1C c1(OCC(=C)C)ccccc1C(=O)NC(C)(CNC(=O)CCCF)Cn1cccn1 Cn1cc(C(=O)NC2(C(=O)NC3(c4cc[nH]n4)CC3)CC2)c(C2CC2)n1 C1(CC=C)(NC(c2ccns2)=O)CCN(C(C2(c3cc[nH]n3)CC2)=O)C1 N1(C(C(C=C=C)C)=O)Cc2ccccc2C(CNC(C2(C(C)(C)C)CCC2)=O)C1 C1(CNC(c2cc(C)n(C)n2)=O)CCN(C(c2ccc(F)c(F)c2)=O)C12CCC2 C1(NC(CC(C)(C)CNC(C2CN3CCN2CC3)=O)=O)CC2CC1C(O)C2O c1(C(N2CC=CC(NC(C(C)OCCN(C)C)=O)C2)=O)ccnc2c1OCC2 CC(C)(C#CC(=O)N1CCCC(C)(C#N)C1)CNC(C1CC2(CCO1)CC2)=O C1(C(C)(C)CNC(C2CCCCO2)=O)CCN(C(=O)CNc2nccs2)CC1 C(=O)(C1=CCCC1)Nc1scc(CNC(=O)C=CC2CCCC2)n1 c1(OC)cc(C)c(C(=O)N(C(C)CCNC(C2(C(F)F)CCCC2)=O)C)c(C)c1 N1(C(C=CCNC(C2CC(C)OC2)=O)=O)CCCC2(CCC2)C1 Cc1cccc(C(C)NC(c2cn(C)nc2C2CCCNC2)=O)n1 N1(C(c2cc(CC)cc(Cl)c2)=O)CCC2CCN(C(=O)CCCCOC)C2C1 C#CCCCCC(=O)NCC12CC(CO1)N(C(=O)CC1(O)CCOCC1)C2 N1(C(C(c2ccccc2C)OCCC)=O)CCOC2(CCC(=O)NC2)C1 c1(C(=O)NCCN(C(C(C)SCCCC)=O)CCOC)cc(CC)no1 CCC(CC)C(C)C(=O)NC(CO)CCCNC(C1CN(C)C(=O)N1)=O c1(C(N2CCCC(N3CCOCC3)C2)C(=O)NCCSC)nn(C)c(Cl)c1Br C(=O)(C(O)C(C)C(CC)CC)NCC(=O)NCC(=O)NC(C#C)C N1(C(CC2(OCC)CC2)=O)CC(NC(c2nn[nH]c2C(F)(F)F)=O)CC(O)C1 C1(C(=O)NCc2c(C(N3CCCC4CC34)=O)scc2)CC(=O)C12CCC2 C(CN=C(NCc1occc1C)NCC1CCCC(C)(C)O1)OCC C1(NC(c2noc3c2COCC3)=O)CN(C(C2CCCC2)=O)C2(CCCOC2)C1 c1(CC(=O)NC(C(C(C)C)OC(C)(C)C)C)nc2c([nH]1)CCCC2 Cc1nc2ccc(C(=O)NCC3(C)CC(NC(C4(CO)CCCC4)=O)C3)cc2[nH]1 N1(C(C23CN(C(c4ccnc(C)c4O)=O)C(C2)CO3)=O)CC2CCC(CC2)C1 CC(C)C(CNC(c1cc(CCCO)on1)=O)NC(=O)C(O)C1CC1 CCCC(O)CC(=O)NC1CC(CNC(C2CCN(CC)C2)=O)C1 Cc1c(C(N2CC3(CCN3C(=O)CCc3ccoc3)C2)=O)ccc(Br)c1F c1(C(=O)NCC2CCN(C(C(CC)(C)F)=O)C2)cc(-n2cccc2)ccc1Cl N1(C(CCc2cnc(C)s2)=O)CCC2C1CCCN2C(=O)C(C)OCCN(C)C C1(SCC)CN(C(C2CCNC2=O)=O)CC1NC(C1(C(=O)OC)CCC1)=O c1(C(=O)NCC2CN(C(c3cnn(CC(F)F)c3)=O)C2)ccn2c1CCCC2 C1(C(=O)NCC2(C(N)=O)CN(C(c3ccncc3F)=O)C2)CCCC2CCCN12 c1(CCC(=O)N(CCOC)CCNC(=O)C(C)n2ccnn2)cnn(C)c1 c1(CNC(C2(OC)CCC2)=O)cccc(CN(C(=O)C(C2CCC(=O)N2)F)C)c1 C1(CC=C)(NC(=O)Cc2n[nH]c(C)n2)CCCN(C(c2[nH]c(C)nc2C)=O)C1 c1(OCOC)ccc(-c2ccc(COC(c3ccc(OC)cn3)=O)s2)cc1 C1(C2(NC(c3nsnc3O)=O)CC2)CCCCN1C(=O)Cc1ccnc(Cl)c1 Cc1ncncc1C(N1CCCC1C(C)C(N1CCC(C(=O)N(C)C)C1)=O)=O c1(C(N2CC(CNC(c3ccc(C(C)(C)C)[nH]3)=O)C2)=O)c(N)cccc1[N+](=O)[O-] N1(C(CCCN=CC)=O)CCCC2(CCCN2C(C2CCC(CCC)CC2)=O)C1 N1(C(CC(CC)SC)=O)CC(C(=O)N(C(C(N)=O)C2CC2)C)C2(CCC2)C1 C1(CNC(C=CCN(C)C)=O)CC2CCC(C1)N2C(c1ncnc2sccc12)=O C1(CC=C)(NC(c2cnc(CC)s2)=O)CCN(C(c2cc(CC3CC3)[nH]n2)=O)C1 c1(C(N2CC(OCCNC(C3CC3c3occc3Br)=O)C2)=O)cccc(F)c1 n1(CC(=O)N(CC)CCS)cc(C2CC2)nn1.C1(C(=O)CCC2CCC2)CCC1N c1(C(N2C(C)CC(CNC(=O)Cc3ccno3)C2)=O)cc(F)cc(N)c1N CC(CCCNC(C1C2COCC12)=O)NC(=O)CCOC1CCC1 c1(NC(C(c2ccccc2)OC)=O)c(F)cc(C(F)(F)F)cc1F c1(C(=O)NCC2CCC(C(=O)NC3(C)CCCOC3)O2)cccc2cncn12 N1(C(C(N(C(Cc2nc(C)sc2)=O)C)C2CC2)=O)CC2C(C(N)=O)C2C1 n1(CCCCC)nc(-c2ccc(F)cc2)nc1-c1cn(C2CC2)nc1C C12(C(N(C3CCCCC3)CCNC(c3cncc(OC)c3)=O)=O)COCC(C1)OC2 c1(C(=O)NC(CNC(CC)=O)(C)Cn2cccn2)nc(C)sc1C(F)(F)F Cc1cc(C(N2CC(C)(C)CC2CNC(c2[nH]cnc2C)=O)=O)c2occc2c1 c1(C(=O)NC(CC)CN(C(=O)Cc2cc[nH]n2)C)ccnn1C(C)C c1(C(N2C(CN(C)C(c3cnns3)=O)CCC2)=O)ccccc1C(F)(F)F c1(C(N2C(C3(C)COC(=O)N3)CCCC2)=O)cc(Br)cc2[nH]ncc12 N1(C(CN2CCC(C)CC2)=O)CCC2(NC(=O)CN3CCS(=O)(=O)CC3)CC2C1 CCC(CCCC(=O)NC1CCN(C)C(=O)C1)NC(C1C2CC(=O)CC12)=O Cn1cnc(C=CC(=O)NC(C(=O)NCCCC2(C)CC2)C2(C)CC2)c1 N1(C(CC(C)=C2CC(=C)C2)=O)CCCC(C)(CNC(=O)CCCOC)C1 C12(CNC(Cc3cnc(C)[nH]3)=O)CCCC1CN(C(c1c(C)cncc1C)=O)C2 c1(N(C(C2CC3CC2CN3)=O)CC2CC2(F)Cl)cncc(C(F)(F)F)n1 Oc1c(C)cc(F)cc1Cl.c1(C[SH](=O)=O)ccc(C(F)(F)F)cc1 N1(C(CCCN(C(C)=O)CC2CC2)=O)C2CCC1CC(O)(c1cnnn1C)C2 Cc1ccc(CNC2N(C(C3(N4CCCC4)CCC3)=O)CC(C)(C)C2)cc1F c1(CC(N2CCC(N(C(=O)C(C)NS(C)(=O)=O)CC)C2)=O)ccc(F)c(Cl)c1F N1(C(c2c(CC)nc(C)[nH]2)=O)CCN(C(C2CC2COC)=O)CC1CC(C)(C)C C1(=O)CCC(=O)NC(C)CN1.c1(C(=O)OC)nnc(C)s1.C1CN(C(C)C)C1=O c1(CCC)cc(C(=O)N(CC(=O)NCc2n[nH]cc2C2CC2)C(C)C)no1 Cn1ccnc1CNC(c1occc1CNC(C1CCC(F)C1)=O)=O c1(C(=O)NCC(C2CCN(C(=O)C=C3CC3)CC2)(C)C)ccn2ncccc12 c1(C(C(=O)NC(CC)(C)CNC(c2ccnn2C(C)C)=O)C)ccc(OC)cc1 Cn1ccc(C(F)=CC(=O)NC2CCCCC2NC(c2cc3c(s2)CCC3)=O)n1 c1(OC)cc(C(N2CCCC2CNC(c2cncn2C)=O)=O)nc2ccccc12 N1(CC(=O)NCC2CC(NC(C(C)OCCOC)=O)C2)CCOCC1=O C1(C(=O)NCCNC(C2CN(C(c3c(C)cns3)=O)C2)=O)CC=CCC1C c1(OCC)cc(Br)ccc1C(=O)NCC1(NC(=O)Cc2ccnc(Cl)c2F)CC1 C1(C#N)(C(=O)NCCOC2CCN(C(c3cc(OC)no3)=O)C2)CCCO1 C=C(C)CC(C(=O)N1CCCC(O)(C(C)C)C1)NC(c1cncc(O)c1)=O C1(C(CNC(C2C(C=C)C2)=O)NC(=O)Cn2ncnn2)CCCCC1 c1(CC(=O)NC2C=CCN(C(c3cnc(C)[nH]3)=O)C2)cccc(S(C)(=O)=O)c1 c1(C(=O)NCC2C(NC(C(C)CC3CC3)=O)C2)c(F)cc(Br)c(F)c1F N1(C(c2c(CC)occ2C)=O)CCC(CNC(C2(C(F)(F)F)CCC2)=O)C(C)C1 c1(CN2CC(F)CC(C(=O)NC3CC(C)C3)C2)cc2ccc(C#N)cc2[nH]1 C1(NC(C2C(C(=O)OC)C2)=O)CC2CCC(C1)N2C(c1cc(CC(C)C)[nH]n1)=O C=C(C)CC(C(=O)N1CC(NC(=O)CC2(C)CCC2)C(C)(C)C1)NC(C)=O N1(C(C(C)N=[N+]=[N-])=O)CC2CCCC2(C(N2CCCC(C(C)(C)O)C2)=O)C1 C1(NC(C2C(CC)CCO2)=O)CN(C(c2ncn(C)c2C)=O)CC1F C1(C2CCN(C(=O)CCC3CCCO3)CC2)(NC(C2(S(C)(=O)=O)CC2)=O)CCC1 c1(OC)cc(Cl)ccc1C(N1C(C(=O)Nc2cc(Cl)ccn2)CC2CC12)=O c1(C(=O)NC(CC)CNC(=O)CC2OCCCO2)ccc2nc(C)cn2c1 c1(C(=O)NCCOCc2ccoc2)ccc(B(O)O)cc1.CC1C(=O)N1 C1(CNC(C(C)C2CC2)=O)CCC2(CCC2)CN1C(c1cc(F)cnc1O)=O C1(C(=O)OC)CN(C(=O)C(O)CCNCc2c(C)cn(C)n2)CCN1C N1(C(C(Br)=C(C)C)=O)CC(N(C(=O)C(C(C)C)c2ccncc2)C)C(O)C1 c1(C(=O)NC2CCCCC2NC(=O)C(O)C(F)(F)F)cc(C(F)F)ccc1F N1(C(c2c(C)nc(CC)s2)=O)CCN(C(=O)C=CC(F)(F)F)C2CC12 CC(C(=O)NC1CCC(NC(=O)CCCc2ccc(F)cc2)C1)C(C)(F)F N1(C(c2c(N)nccc2)=O)CCCC2(CC(NC(=O)C3Cc4ccccc43)C2)C1 CC1(CNC(=O)Cc2cccs2)CCCN1C(=O)COCC1CCCOC1 CC(CC(C(F)F)c1ccccc1)NC(c1cncc(C)c1)=O c1(OC)c(N)ccc(C(=O)NC23CCCC2CN(C(=O)C(C)(CO)OC)C3)c1F n1(CC)cc(C(=O)NCCC2(O)CN(C(C3CCC(=O)C3)=O)C2)c(C(C)C)n1 C(CNC(=O)CN(C)CCO)(CCNC(=O)C(F)C1CCOC1)OC Cc1cc2[nH]c(C(=O)OCCCCC(=O)O)cc2o1 CCCCCCCCCC(O)C(=O)N1CCSCC1CCNC(=O)Cc1ccoc1 Cc1sc(S(N)(=O)=O)cc1C(=O)NC(CNC(=O)Cn1cnc(=N)[nH]1)C(C)(C)C C=Cc1ccc(C(=O)NCC(C)CC(=O)NC2CCCN(O)C2=O)cc1 c1(CN2C(C(=O)Nc3cn(COC)nc3)C=CC2)cnc2ccccc2c1 C1(CCNC(CCSCC)=O)C(C)CCCN1C(=O)CNS(=O)(=O)CC C(CC(C)(C)C)(C(=O)NCC(C1CC1)NC(c1ncoc1-c1ccco1)=O)OC C1(C(=O)NC2C(CNC(c3cc(CC)cc(F)c3)=O)C2)CCCC(C)(C)CC1 c1(C(=O)NCC2CCC(NC(c3ccc(F)cc3)=O)C2)cccc2c1CCN2 C(=O)(C1CCCc2ccnn21)NCC1N(C(Cc2cc(C)c(Cl)cc2)=O)CC1 C1(C)(C(=O)NC(c2ccccc2)C(C)NC(c2cccs2)=O)COCCO1 C1(CNC(C2CN3CCC2CC3)=O)CC(C(=O)NCC2CC3(C2)CC(O)C3)=NO1 N1(C(C=C(C)C(C)(C)C)=O)CCC(O)(CN(C(=O)CC2COCC(C)O2)C)CC1 CC12CCC(C(N3CCC(NC(C4CCCS4(=O)=O)=O)C3)=O)(CC1)C(C)(C)O2 Cc1cc(C(=O)NCC2CCCCN2CC(c2ccco2)O)cc(I)c1 CCC(CC(=O)NCC(C)CC(=O)N1CC(c2cc[nH]n2)C1)C(C)(C)C c1(CCC)nnc(S)n1CC(=O)NC1CCCC1CNC(C1CC1CSC)=O c1(-n2cc(CC(Cc3ccco3)NC(C3CN(C)C3)=O)nn2)ccccc1N C1(C(N2CCC(C)C2)=O)CC2CCC1N2C(c1cccc(C2CCC2)c1)=O c1(NC(N2CC3C(CNC(=O)Cc4nc[nH]n4)(C3)C2)=O)ccc2[nH]ccc2c1 c1(C(N2CC(C(C)(C)O)(CNC(=O)CC3CCC(O)C3)C2)=O)ccc(F)nc1 c1(CNC(=O)CC2CC3CN(C(c4ccncn4)=O)CC23)cc(Cl)ccc1[N+](=O)[O-] Cn1c(C(=O)NC2COC3(C2)CN(C(=O)Cc2ccco2)C3)cc2sccc12 C(C)(C(=O)NCC(C)(C1CCC1)NC(c1cn(CC(F)(F)F)nn1)=O)(C1CC1)OC N1(C(c2c(OC)csc2)=O)CC(OC)CC(NC(C2NC(=O)OC2C)=O)C1 N1(C(CCCC(C)=O)=O)CCC2CCCN(C(c3c[nH]cc(Cl)c3=O)=O)C2C1 N(C(=NCCC(C)C)N(C)CCOC)c1c(CC)cc(F)cc1OC c1(C(c2ccncc2)NC(N(C(CC)C2CC2)C)=O)ccc(Br)cc1 n1(CCCn2c(C(C3CCCCC3)CCC#C)nnn2)ncc(Cl)c(Cl)c1=O C(=O)(C(C(C)(C)C)NC(C1CCCCN1C)=O)N1CCCC(COC)C1 Cc1ccc(C=CC(=O)N(CCCNC(=O)C(C)Oc2ccc(OC)cc2)C)o1 n1(C(C)C)cc(C(=O)NCC#CCNC(c2c[nH]nc2-c2ccoc2)=O)cn1 N1(C(C(CCC)C#N)=O)CC2CCC1C1CN(C(c3nc(Cl)sc3C)=O)CC21 CC1CCC(CC(=O)NC(c2nocc2C(=O)N(C)Cc2ccns2)C)OC1 C1(CC)CN(C(C2CC(F)(CF)C2)=O)CCC1NC(=O)C=C(C)C(F)F N1(C(c2cccc(C(=O)NC)n2)=O)CCCC(NC(=O)C=CC(F)(F)F)C(F)C1 N1(C(C(=O)NCC)=O)CC(NC(c2nn(C)cc2N)=O)C(C)C1 c1(OCCC)ccc(OC(c2ccco2)=O)cc1.c1(N)cc(C(N)=O)ccc1C N1(CC)CCN(CC(=O)NCCCC(CO)NC(C2CCC(C)C2)=O)CC1 c1(CC(=O)NCCN(C=O)CC)cccc2nsnc12.C1(=O)C(C)O1.C(C)(C)(C)O N1(C(CSCCCC)=O)CCCC(CN(C(=O)C(CC)n2cncn2)C)C1 C1(C(=O)NC(CCNC(C2(OC)CCCC2)=O)C)CC(F)(F)C1(F)F c1(C(N2C3(CN(C(c4n(C)cc(Cl)c4Cl)=O)C3)CC2)=O)ccc2cnoc2c1 C1(C)(C(=O)NC(COC)CNC(c2cc(CO)[nH]n2)=O)CC(C)(C)C1 CC1CN(C(=O)CC(C)(C)c2cn(-c3cccc(F)n3)nn2)C(C)CO1 C1(CNC(C(C=C)O)=O)CCCN(C(c2cc(I)c[nH]2)=O)CC1 C1(C)(C(N(C)Cc2nnc(C)s2)=O)CN(C(c2ccc(O)nc2)=O)C(C)(C)C1 CC1CC(NC(c2scnc2C(F)(F)F)=O)CN1C(=O)CSc1nncs1 C1(C(N2CCC(C=C)(O)C2)=O)CC2(CCN1C(c1ccc(C)c(C)c1)=O)CC2 C1(NC(CC=C)=O)CCCC12CCN(C(=O)CCCc1ccc3ocnc3c1)C2 C1(C(C(=O)OC)(C)C)CCCCN1C(=O)C(C)OC1COC1 C1(CC=C)(NC(C2CC(F)C(=O)N2)=O)CCN(C(C2(n3cc(Br)cn3)CC2)=O)C1 C=CC(C)(CC)C(=O)NC1(CO)CN(C(c2ccc(-c3ccco3)o2)=O)C1 N1(C(CCC(=O)NC)=O)CC(CN(C)C(C2CCCCN2C)=O)C2(CC2)C1 N(C(=NCCCC(C)(C)C)NC1CC1CF)C(c1ccc(OC)c(Cl)c1)C NC(=O)CCCCC(=O)NC1CN(C(c2sc(C(=O)O)cc2Br)=O)CC1O C1(CC(=O)NCCCC(C)NC(=O)Cn2nccn2)CCn2cncc2C1 C=CCCCCCC(=O)NCC1(NC(=O)CCCC(C)(F)F)CCOC1 C1(NC(=O)CCCC2CC2)CS(=O)(=O)CC1N=c1nc(-c2ccccc2)[nH]s1 C1(CN(C(c2cnc(C)cn2)=O)CC)CCCCN1C(=O)C=CSC C1(C)(CC)C=C(C(=O)N2CCCC(F)(CNC(c3cc4sccc4s3)=O)C2)C1 c1(OC)ccc(CC(=O)NC2C3CC(O)C2N(C(=O)C=CBr)C3)c(Cl)c1OC c1(C(=O)NC2CCCCC2n2cc(C(=O)O)nn2)cc2cc(Cl)cnn2n1 C1(CC(=O)NC2CC(C(C)C)C2)CN(C(=O)CCC2CCCN2C)CCO1 c1(CN)nn2c(c1C(N1CCN(c3ccccc3F)CC1)=O)CCC2 N1(C(C(C=C)(C)O)=O)CCN(C(=O)CCc2ccc(OC)cc2)C(CO)C1 C=CCC(CC(=O)NC1COCC1CC)NC(C1CC(=O)N(OC)C1)=O C(=O)(CC(C)C(F)(F)F)NCC1(C)N(C(CCn2ncc(C)c2)=O)CCC1 C(=O)(CCC(CF)CF)NCC1CC(CNC(c2c(NC)scn2)=O)C1 C(C)(C(=O)NCCCN(C(c1cccc(O)c1F)=O)C1CC1)(C(C)C)OC N1(C(C2(N(C)C)CC2)=O)CCC2(CC1)CC2NC(=O)C(F)CC1CCCC1 C(c1ccc(=N)[nH]c1)=CC(N1CCC(O)(C(C)NC(c2cnn(C)n2)=O)C1)=O c1(NC(N2CCN(C(C(=O)NC(CC)C)=O)CC2)=O)ccc(S(C)(=O)=O)o1 c1(OC)noc(C(N2CC(C)(NC(c3cnc[nH]3)=O)C2)=O)c1Br CC(O)C(F)(F)C(=O)NC1CC(NC(=O)C(CC(F)F)c2ccccc2)C1 c1(C(=O)NC2CCC(C(N=c3cc(C)o[nH]3)=O)OC2)ccc2c(Cl)ccnc2c1 c1(CC)c(C)nc2ncnn2c1N(C)CC1CCCCN1C(=O)CC(C)COC C1(C(N(CC(=O)NCC2CN3CCC2C3)CCC)=O)CCCCN1C C12(CNC(C(C(C=C)C)C)=O)CCC(CNC(c3scnc3CC)=O)(CC1)CO2 C1(C(=O)NCC2C(CNC(c3c(C(C)C)n(CCO)nc3)=O)C2)CN2CCC1CC2 C1(C(N2C(C(N(CCC(=O)OC)CC#C)=O)CSC2)=O)CC=CC(O)C1 C(c1ccc(F)cc1)=CCC(=O)N(C(CNC(c1c(CC)nn[nH]1)=O)C)C c1(OCC)ccc(CCC(=O)NCCNC(C2CC(SCC(F)(F)F)C2)=O)cc1 C(=O)(CS(=O)(=O)NC)N(CC(CO)NC(COCCCCC)=O)C C(=O)(CCCCCC#N)N(CC(CO)(CO)NC(CC1N(C(C)C)CCC1)=O)C C#CCC(CC(=O)N(CCCN(C(=O)CNC(N)=O)CCO)C)c1ccccc1 N1(CC(=O)NC2C(NC(C(=O)NC(C)C)=O)COCC2)CCCCC(O)C1=O Cn1c(I)cc2c(N3CCCC(NC(c4c(Cl)ccc(Cl)c4F)=O)C3)ncnc12 C1(C(c2c(OC)cncn2)c2nnnn2C2CCCOC2)(OC)CCOC1(C)C N1(C(C2CCCN(C(N)=O)C2)=O)CC2CCC1C1CN(Cc3ccsc3)CC21 c1(C(=O)NC2CCN(C(CC(CC)C3CCC3)=O)C2C)cc2n(n1)CCCC2 CC(C)(C(=O)N1CC2CC(C1)C2NC(=O)C=CC(F)(F)F)C(N)=O Cc1cccc(C(C)N(C)C(=O)NCC2(c3ccc(F)cn3)CC2)c1 C1(NC(c2cn(CCCC)nc2C)=O)CN(C(c2cnn(C)c2)=O)C(C)(C)C1 C1(CC)CN(C(C2CCCC(CF)C2)=O)CC1C(=O)NCC=C(Cl)Cl C(=O)(C(C)(C)C(=O)NC(c1nccn1C)CC1CCC(F)(F)CC1)NC C1(C(=O)NC2C(NC(c3[nH]cc(CC)c3)=O)CS(=O)(=O)C2)CCC2CC1C2(C)C C1(CN(C)C(C2CC(CF)C2)=O)CCCC1C(=O)NCC1(F)CCCC1 C1(NC(C(C)OCCC=C)=O)CCCN(C(c2ccnc(C(C)(C)O)c2)=O)C1 c1(N2CCCC(CCNC(C=CCCC)=O)CC2)ncnc2c1cnn2C c1(CN(CCCC(O)CO)C)ccc(Br)c(C#N)c1 C1(CNC(C(CCC)NC(C2CCCO2)=O)=O)OC(=O)NC1(C)C CC(=O)CCCC(C)C(=O)NC(C)CC(=O)Nc1cn(C)nc1C1CC1 C(c1c(Cl)cccc1Cl)=CC(=O)NCCN(CCC)C(c1cc2sccc2[nH]1)=O CCC(C)C(=O)C(=O)NCc1cccc(C(=O)NC(C)(CC)CCC)n1 CC1Cn2nccc2CN1C(c1c(Br)ncn1C)C(=O)NCC1CCOC1 c1(CN(CC(=O)OCC)C(=O)CC2CCCCO2)ccc([N+](=O)[O-])cc1Br c1(C(=O)NCCCCN(CCOC)CCO)c2c(nn1C(C)(C)C)CCCC2 c1(-c2c(C)nc(C)s2)ccc(S(=O)(=O)Nc2cnccc2C#N)s1 n1(CC=C)c(N(C)CC2COC(=O)O2)nnc1-c1cncc(OC)n1 N1(C(C=C2CCC(C)C2)=O)CCCCC(NC(=O)CN2C(=O)CCC2=O)C1 C1(C(=O)NCC(CC)NC(c2cc3c(s2)CCSC3)=O)Cc2cccnc2C1 c1(NC)cncc(C(=O)N(C)CC2CN(C(c3ccc(F)s3)=O)CCO2)c1 N1(C(c2scc(CNC(c3cc(SC)oc3)=O)c2)=O)CCOC(C#N)C1 C1(C(C)C)CN(C(c2nccc(Cl)c2F)=O)CCCN1C(=O)CC(C)(F)F CC1(C)CC=C(C(=O)N2CC3CC(NC(c4cn(C5CC5)nn4)=O)C2C3)CC1 C1(CNC(c2c(C)noc2C2CC2)=O)CC(F)(F)CN1C(=O)C(CO)N(C)C c1(C(=O)NC2C(CNC(c3c(C)cco3)=O)C2)cnc2c(Cl)c(Cl)ccc2c1 c1(C(c2n(CCC)nnn2)NCCOCC2CC2)cccc(F)c1I CC(F)(F)CCCC(=O)N1CC(F)(CNC(=O)C=Cc2cccnc2)C1 c1(OC)ccc(S(=O)(=O)CCC(=O)NCC(O)CNC(C2OCCC2C)=O)cc1 Cc1ncc(CC(=O)NC(C2CN(C(C3(C)CC=CC3)=O)C2)C)s1 c1(N2CCC(C(C)NC(=O)CCc3cccnc3F)C2)nc2cc(F)cc(F)c2o1 CC1(CNC(=O)C2=C(Cl)CCC2)CCC(NC(C2CCOCC2)=O)CC1 CCC(CS(C)(=O)=O)NCC(c1ccc(C#N)nc1)=O C1(CCOC)(NC(c2cnn(C)c2Cl)=O)CCN(C(C2CCCC(F)C2)=O)CC1 C(CNC(c1ccc(C#N)s1)=O)(CC(=O)N1CC(CCN(C)C)C1)OC C1(CCNC(=O)NCC(=O)NC2CN(C(=O)C=Cc3cccs3)C2)CCCCC1 CC(C)C(CC(=O)N1CCC(O)C(O)C1)NC(C1CCC(=O)N(C)C1)=O N1(C(C2CCCN(C(Cc3scc(C)c3)=O)C2)=O)CCCC12CCNC2=O C=C(CNC(=O)CO)CCNC(=O)CCNC(=O)C(CC)N(C)C(C)=O c1(C(N(CC(CNC(C(C)O)=O)(C)C)C)=O)ccn(C)c1C1CCC1 c1(C(=O)NC2CCC(NC(C3CCC4(CC3)CC4)=O)C2)c(F)cncc1F C1(SCCNC(C2(C)CC(=C)C2)=O)CN(C(=O)C(C(C)(C)C)C2CC2)CC1c1cn[nH]c1.O N1(C(C(C)=O)=O)CC(NC(c2cccc(C3CCOC3)c2)=O)C(C)C1 C1(C(N2CCOC(C3CCC3)C2)=O)(CNC(C(C)=C2CC2)=O)CCCCC1 c1(C(=O)NCCCC2CN(C(C3CC4CC4C3)=O)CCO2)cncc2c1CCC2 Cc1cnc(NC(C)CCC2CC2)c(S(=O)(=O)NC2(C)CC(C)(C)C2)c1 N1(C(C(CC)C)=O)CCC2(CC1)CC(NC(=O)Cc1nc(C)cs1)C2 c1(-c2cn(CC3N(C(C=CC(C)C)=O)CCOC3)nn2)cc(OCCO)ccn1 c1(OCC(=O)Nc2c(CNC(CCC(C)OC)=O)cccn2)ccc(C)cc1Cl c1(C(=O)NC(C2CN(C(c3cccc(OC)c3N)=O)C2)C)nn(C)cc1[N+](=O)[O-] c1(C(=O)NC2(C)CCN(C(c3c(COC)scc3)=O)C2)cccc2oc(O)nc12 C1(NC(CNC(CN(C)C)=O)=O)CCCN(C(=O)CCN2CCCC2)CC1F c1(C(c2n(CC)nnn2)NCc2cscc2C(F)(F)F)cccc([N+](=O)[O-])c1C Cc1ccncc1C(N1CCC(C(C)(C)NC(=O)CC2CCCCO2)C1)=O N1(C(c2cc3nc(C)sc3[nH]2)=O)CCC2(CCN(C(=O)Cc3n[nH]c(=N)s3)C2)C1 c1(SC)ccc(C(=O)NC2CN(Cc3ccc(N(C)C)cn3)CC2O)cc1 C(CCCCCNC(C1CCCN1S(C)(=O)=O)=O)NC(C(C)(C)N(C)C)=O CC1=C(C(=O)NCC2CCCCN(C(=O)C(c3c(C)n[nH]c3C)C)C2)COCC1 C(CCSC)(C(=O)N(CC(C)O)CC(C)O)NC(C(CC)NC(C)=O)=O N1(C(C2NC(=O)OC2)=O)CCC2(CC1)CC(NC(c1cc3sccc3s1)=O)C2 C1(C)(CNC(C(c2scc(C)n2)C)=O)CCCN1C(=O)Cc1csc(Cl)c1 N1(C(C2CC(CC)C(=O)CC2)=O)CCC2(CC1)CN(C(=O)Cn1nnnc1C)C2 C1(CNC(C(C2CCCOC2)OC)=O)C(C)CCN1C(c1ccncn1)=O c1(C(=O)NCCCc2onc(-c3cccc(C)c3)n2)nc2ccccc2cc1F C(=O)(C1=NOC2(CCN(C(c3ncccn3)=O)C2)C1)NC(C1CCCO1)C C1(NC(C(CC)NC(C)=O)=O)CCCC(N(C(=O)CCCc2csc(=N)[nH]2)C)C1 c1(C(C)NC(CC)CN(S(C)(=O)=O)CC)ccccc1OC C(C)(C)(C(C)CC(=O)NCCCSCC)NC(CCC(CC)C)=O c1(OC)ccc(C(=O)NC23CCC2CN(C(c2cscn2)=O)C3)cc1Cl C1(C)(CC(=O)NC(C2CCN(C(C3CCC(=O)N3C3CC3)=O)C2)C)CCOCC1 c1(OC)cc(C(=O)NC(Cn2cccn2)C(=O)NCCC2CCOC2)n(C)n1 n1(CC(=O)NC23CCCC(NC(CCCCC)=O)(C2)C3)nc2c(n1)CCCC2 C1(C(=O)NC(C(C)NC(=O)Cc2ccc(C#N)cc2)CO)CC2(CCOCC2)C1 CC1(C)CC=C(C(=O)NC2(CCCNC(c3ccccc3F)=O)CC2)CC1 c1(CC(=O)NCC2C(NC(C(CC)Oc3ccccc3)=O)C2)cccc(F)c1 C1(CC(=O)NC2(CC(=O)O)CN(C(Cc3nc(C)sc3)=O)C2)CC2CCCC2C1 c1(C(N2CC(F)(CNC(C34CC(c5ccccc5)C3C4)=O)C2)=O)nnc(O)nc1O c1(C(=O)NCCC2CN(C(C3C4CC4C4CC34)=O)C2)ccc2nnnn2c1 N1(C(C(C2CN(C(C3CCC(=O)O3)=O)C2)OC)=O)CCC(C2CC2)C1 C(CC(C(C)(C)C)NC(=O)Cc1cnnn1C)N(C)C(c1cccc(O)c1)=O C1(F)(CNC(C2(SC)CCC2)=O)CCN(C(c2coc(C3CCC3)n2)=O)CC1 N1(C(CC2CC(=O)C2)=O)CCN2CCC1CC2 N1(C(C=CC(c2ccccc2)=O)=O)CC2CCC2(C(N2CCC(O)C(O)C2)=O)C1 c1(CNC(C2CC3CC3N2Cc2c(OC)cco2)=O)cc(Cl)nc(Cl)c1 N1(CC(=O)NCCC2CCCN(C(C(C3CCC3)OC)=O)C2)CCCCCC1=O N1(C(c2ncccc2O)=O)CC2CC(C1)CN(Cc1cc(O)ccc1F)C2 C1(NC(CC(C=C)C)=O)C2CC1CN(C(c1n[nH]cc1C(F)(F)F)=O)C2 Cc1nnc2c(C(N3CCN(C(=O)Cc4c[nH]ccc4=O)C4CC34)=O)cccn12 N1(C(CC(C)c2cccnc2)=O)CCCC(C)(NC(=O)C=Cc2nccs2)C1 C1(C(=O)NC2CCC2c2ccc(Cl)cc2)CCCCC(F)(F)C1 C(N=c1ccc(C2(C)CC2)n[nH]1)=C1CCN(C(c2ccn(C)n2)=O)CC1 N1(C(C(C)(C)CCCO)=O)CCOC2(CCCN(C(=O)C3=CCCS3)C2)C1 C1(CCNC(=O)COC(F)(F)C(F)(F)F)CC(F)(F)CN1C(=O)CC1CC1 CCC(CC(=O)N1CCC(C(C)C(=O)NC2CCCC2N=[N+]=[N-])CC1)CC(C)C CCCC(C(=O)OC)C(=O)NCC1CCN(C(C2CCCC(O)C2)=O)CC1C C1(NC(CSc2cn(C)nc2)=O)CCCC2(C1)CC2(F)F c1(OCC(=O)NC2CCOCC2NC(C23CCCC2CC3)=O)ccc(Cl)cc1 c1(C(CC)C)ccc(C#N)c(NC2CN(C(=O)Cc3ccc(C)cc3Cl)CC2C)n1 C(C1CCCN1C(=O)C(C)=C1CC1)=CC(=O)NCC(=C)C N(C(=NCCCF)NC1CC1(c1ccc(Br)c(OC)c1)C)CCOC N1(C(C2CN(C)C(=O)N2)=O)CC2CN(C(=O)COC3CCCCC3)CC(C1)O2 c1(C(=O)NC(C(C)C)CNC(C23CC(F)C2C3)=O)cccc2c1NC(=O)CO2 C1(C(N(CCCN(C)C(C2CNC(=O)N2C)=O)C)=O)Cc2ccncc2C1 c1(Cn2cc(C3N(C(CNC(N)=O)=O)CC3)nn2)c(F)cccc1F c1(NS(c2cccc(C)c2)(=O)=O)n[nH]c(=NC2CC3CCCCC23)s1 N1(c2ncnc(C)c2Br)CCC2(CC1)CC(NC(C1COCCO1)=O)C2 CC1CCC(NC(N(C)CCC2CC(C(F)F)C2)=O)C1 N1(C(CCC(C)=O)=O)CCC2(CC1)CC(C(=O)NCc1cccc3c1CCC3)CO2 C1(C(N(C)Cc2ncc(C)o2)=O)CCC(C)(C)N(C(C2CC(C)CC(C)C2)=O)C1 N1(C(c2c(N)ccc(C#N)c2)=O)C2CCC1CN(C(c1coc(Br)c1)=O)CC2 C12(NC(CSCC=C)=O)CCC(C1)N(C(C1(c3cc(C)ccc3C)CCC1)=O)C2 n1(CC(N2C(CNC(c3cc(-c4ccns4)on3)=O)CC2)=O)cnnc1O N1(CC(N2CCC(N(C(C(CC=CC)C)=O)CCO)C2)=O)C(=O)CC(C)(C)C1=O C1(NC(C2CCC(C)O2)=O)CN(C(C2C(C)(C)C2(C)C)=O)CCC1O CCCC(C(=O)N(C)Cc1ccccc1)NC(=O)CC(C)=C(C)C c1(C(=O)NC2C(CO)CCN(C(CNC(CC)=O)=O)C2)cncc2nc[nH]c12 O=C1CC2(CC(=O)N2C(c2ccccc2)C(N2C3CCC2CC(O)C3)=O)N1 CCC(C(=O)OC)C(=O)NCC(C)(O)CNC(c1ccc(Cl)c(C)c1)=O c1(C(N2CC(CO)(Cc3nc(C(C)(C)C)sc3)C2)=O)cccc(Cl)c1Cl Cc1ccc(C)c(C(=O)NCc2cccc(NC(C3CCC(=O)NC3)=O)c2)n1 N1(CC(=O)NCC2CC3CCC2N3C(C2CC=CCC2)=O)CCCCCC1=O C1(C(N2C(CNC(COCC(=C)C)=O)CC3CC32)=O)COC2(CCC2)CO1 N1(C(Cc2c(C)n(C)nc2)=O)CCCC(F)(C(=O)NC2CCC3(CC3)C2)C1 c1(CCN(C(CCC2CC=CCC2)C(=O)NCC2CCCO2)C)ccc(F)nc1 C(=O)(C1=CC2C=CC(C1)C2)N(C(CC(C)C)C(=O)NCC1COCCO1)C N1(C(CC=CC)=O)CC2(NC(=O)C(O)CCSC)CCC1C2 c1(CN=C(NC(COC)C2CC2)N(C)CC(F)F)cc(F)c(F)c(F)c1F c1(C(=O)NCCN(CCOC)C(C2CC23CC3)=O)cncn1-c1ccccc1 c1(C(=O)N(C2CCN(C(=O)Cc3nc[nH]n3)C2)CCO)cccn2cncc12 C=CC1(C2(C(=O)NC3CCC4(CC3)CN(C(=O)C(C)(C)F)C4)CCC2)CCC1 C1(NC(C2C(CC(C)(C)C)C2)=O)CC2CC1CN(C(=O)CN1OC(C)(C)CC1=O)C2 C1(CN(C)CC2(C(N3CCCC(COC)C3)=O)CCCC2)CCS(=O)(=O)CC1 N1(C(c2csc(C)c2C)=O)CCCC(O)(CNC(C2(C#N)CCCOC2)=O)C1 C1(C(=O)NC(C2N(C(c3c(C)ccs3)=O)CCC2)(C)C)CC12CCOC2 C(=O)(CC(O)CN(C)C)NCC1(C)CCN1C(=O)CC1(C(=O)OC)CC1 C(=O)(CC1=Cc2ccccc2C1)NCC1(C)N(C(CC(COC)(C)C)=O)CCC1 C1(C)(CNC(C2(C)CC(=C)C2)=O)COCCN(C(c2cccc(NCC)c2)=O)C1 C1(C)(C(=O)NC2(C(N3CCC(C)(CCC)C3)=O)CC(O)C2)CC2C=CC1C2 N1(C(CS(CC)=O)=O)CC2CCCCC2(CN=c2[nH]c(C3CC(OC)C3)nc(=N)[nH]2)C1 c1(CC)ccc(C(=O)NCC=CCC(=O)NC2(CO)CCC(C)(C)C2)cc1 Cc1cc(C(=O)NC(C)CNC(=O)CCc2nc(-c3ccoc3)no2)ccc1F N1(C(C2CC(O)(CNC(CCCOCC=C)=O)C2)=O)CCOCC1CO c1(C(N2CCC(NC(CCCC)=O)C(O)C2)=O)ccc2nc(O)[nH]c2c1F c1(OC(C)C)cnccc1CN1CC2C(C(N3CCC(C(=O)O)C3)=O)C2C1 c1(C(=O)NC2CCN(C(CC(CC)C3CCC3)=O)CC2)ccc(F)c(CO)c1 C(=O)(C(O)C1=CCCCC1)N1C(C)CC(CNC(c2ccc(C)c(C)c2N)=O)C1 N1(C(C(=O)N(C(Cc2ccccc2)CC(F)(F)F)C)=O)CC(N)C2(CC2)C1 CCC(CCC(=O)N1CCCc2nccn21)NC(=O)CC(C)(C)COC Cc1ccc(SCC(=O)NCCC2CN(C(=O)CC34CCCC3C4)C2)c(C)c1 C1(NC(c2cc(C)sn2)=O)CC2CN(C(c3cc(F)n(C)n3)=O)CC2C1 C1(N=c2cc(C)c(C#N)c[nH]2)(C(=O)NC2CC(C)=C(C)CC2)CCCCC1 C1(F)(CNC(COc2c(C)cccc2)=O)CCN(C(=O)CCC(N)=O)CC1 N1(C(CC2C(C)(C)N(C(C3CC3C(F)(F)F)=O)CC2)=O)CC2CCC(CC2)C1 Cc1oc(CNC(C2CCC2(F)F)=O)nc1C(=O)NC1CC(=O)N(O)C1 S(=O)(=O)(c1ccc(NC2CC=CCC2SC2CC2)c(Br)c1)N1C(SC)CCCC1 c1(C(N(CC(C)NC(c2nc(O)[nH]c(=O)n2)=O)C)=O)ccc(F)c2ccccc12 C1(CNC(=O)CCN2CCCC2)CC(F)(CNC(=O)CNS(N)(=O)=O)C1 c1(C(N2CC(N(C(CC(n3ccc(C)n3)C)=O)C)C2)=O)n[nH]c2c1CCOC2 c1(C(=O)NC)cc(Cl)ccc1N.N1(C(CCN(CCC)C)=O)CCCC(C)C1 c1(C(=O)NC2CCN(C(COCC(C)C)=O)CC2)nn(C)c2c1CSCC2 C1(C(=O)NCC2C(C=C)CC2)CC2(C1)CN(C(=O)CCCCOCCO)C2 N1(C(Cc2ccc(CC)cn2)=O)CCc2sc(CO)cc2C1 C=Cn1nccc1C(=O)NC1CCN(C(=O)C(N2CCOCC2C)C)C1 c1(CC(=O)NC(CCNC(c2c(COC)nn[nH]2)=O)C)cccc(F)c1Cl CC(C)C(C)(CNC(c1cnc(O)s1)=O)NC(=O)CC1(C)CCC1 C1(NC(c2cc(C)no2)=O)CCN(C(c2cc(C(F)F)on2)=O)C(C2CC2)C1 c1(CC)cc(C(N2CCCC2C(C)NC(C2C3CC(=O)CC23)=O)=O)n(C)n1 c1(-c2nc(CNC(=O)NCC(C)OCC=C)sc2)c[nH]c(=N)nc1C(C)C C1(NC(c2c(C)noc2C(F)F)=O)CCN(C(=O)Cc2ccc(Cl)s2)CC1C N1(C(C2(C)CCSCC2)=O)CC2(CCCC2NC(=O)C(=O)C2CC2)C1 c1(NCC2C(C(C)(C)C)NCC2)ccnc(OC(F)F)c1 CCC1=C(C(=O)N2CCN(C(C3OCCO3)=O)C3CC23)CCCO1 C(C1CN(C(C2(SC)CC(=O)C2)=O)Cc2ccccc21)NC(C=CC=CC)=O c1(OC(C)C)ccccc1C(C(C)N)NC(C1CC1Br)=O c1(NC(C2CN(C(c3cnc(Br)o3)=O)CCC2O)=O)cn2c(Br)cccc2n1 C12(NCc3cccc(C(C)C)c3)CCCCCC1N(C(=O)OC(C)(C)C)CC2 CCCC(C(=O)NC1CCCC12CN(C(=O)Cn1nccc1C)C2)C(C)C C(c1ccccc1C)=CC(=O)NCC(C1N(C(CCNC(C)=O)=O)CCC1)(C)C C1(C)(NC(C23CC(OC(C)=O)C2C3)=O)CCCC1NC(=O)CCCC1CCC1 c1(C2(C(C(=O)N3CCC3CC(n3ccnn3)=O)(F)F)CC2)cccc(Cl)c1 c1(C(=O)NC(C(C)NC(=O)CN2CCS(=O)(=O)CC2)C)ccn2ncnc2c1 C1(NC(c2ccco2)=O)CN(C(c2cc3ccccc3o2)=O)CC12CCCC2 Cc1c([N+](=O)[O-])c(C(=O)NC(C)CN(C)C(C2CC3CCC3C2)=O)nn1C c1(C(=O)NCC2CCCCN(C(C3CC(CC)C3)=O)C2)ccc(OC)c(F)c1O CC1(C)CC(=O)NCC1C(N1CC(NC(c2ocnc2C(F)(F)F)=O)C(F)C1)=O C1(C(=O)Nc2ccc(-c3ccc(C)cc3)cc2)CCC(=O)N(C)C1 N1(C(C(C)=CC)=O)CC(C2CCN(C(C3CCC3n3cccn3)=O)CC2)C1 O=C1CC2CCCC2(C(N2CC3CC2(CNC(C2CCC4(CCC4)O2)=O)C3)=O)C1 C1(CNC(CSCC=C)=O)(OC)CCN(C(c2cc(CC)nn2C)=O)C1 c1(C(=O)OC)cccc2nc(CNC(C3CC(C)(C)CCO3)=O)cn12 N1(C(c2c(Br)ccc(C(C)=O)c2)=O)CCC2(CC(C(=O)NC3(C)CC3)=NO2)C1 c1(COC)nc(NCC(CC2CC2)CO)cc(N2CCCC(OCC3CC3)C2)n1 C1(NC(C2(C=C)CCC2)=O)CC1C1CCCN(C(c2oncc2CC)=O)C1 C=CC1(CC(=O)NC(c2nc(C)no2)CO)CN(C(C2CC3CC3C2)=O)C1 S(=O)(=O)(c1c[nH]c(=NCc2cc(C)ccc2OC)cc1C)NC(COC)C(C)C C1(C(=O)NC(CC2CN(C(C(C)OCC(C)C)=O)C2)C)CC(=O)NC(=O)C1 CCC(C)(CO)C(=O)NC(C)C(CO)NC(c1cccc(C(F)(F)F)c1O)=O c1(C(c2n(CC3(CC)CC3)nnn2)NCC(C)C)nc(F)ccc1Br C(CNC(=O)CCCN(C)CCSC)(C(C)C)NC(C(C)OCCC#C)=O C(=O)(CS(=O)(=O)CCC(F)(F)F)NCC(=C)CCNC(=O)C1=NN(C)C(=O)CC1 N1(C(c2c(N)n(C)nc2)=O)CCc2ccccc2C(NC(=O)CC23CC(C2)C3)C1 c12cccc(c1)C(=O)O2.C1(NC(CC)=O)C2CC(NC(C(=O)NCC)=O)CC12 N1(C(CCCN(C)C)=O)CC2(CCN(C(=O)C(C)(F)c3ccccc3)CC2)C1 N1(C(C2N(C(CCC=C)=O)CC(=O)C2)=O)CC2(CCN(C)CC2)C1 N1(C(C2CCC(=C)CC2)=O)CCC(NC(=O)CNC(=O)C(F)(F)F)CC1C C(=O)(C(F)C(C)(C)O)N1CC(OCCNC(C=C2CCN(C)C2)=O)C1 N1(C(c2sc(CC)c(C)c2)=O)CC2CCCN(C(=O)CC(C)C(C)C)C2C1 Cc1ccc(COCC(=O)NCCN(C2CCCC2)C(=O)CC2OCCO2)cc1 Cc1ccc2nc(C(N3C(Cn4cc(C(C)OC)nn4)C4CCCC34)=O)cn2c1 c1(C(=O)NC2CN(C(c3cc(OC)no3)=O)CC2(C)C)coc2c(F)cccc12 C1(CN(C(=O)CCC2CC2(Cl)Cl)C)CCN(C(c2cc(C#N)on2)=O)CC1 C(=O)(CCC(O)C(C)(C)C)NC(C1CN(C(=O)COc2cn[nH]c2)CCO1)C N1(C(c2c(C)nns2)=O)CC2CN(C(C3C(C)(C)C3(C)C)=O)CCC2(CO)C1 CC1(C)CC(CO)CN(C(=O)C(Cc2ccoc2)NC(C2CCCC2O)=O)C1 CC(C)C(O)C(F)(F)C(=O)NC1CN(C(=O)CC#N)CC1(C)C N1(CCNC(CSCC#C)=O)CCN(C(=O)CCc2nc[nH]n2)CC1 C(=O)(NNC(=O)C1CCN1C(C)(C)C)c1ccc(C)s1 c1(C(=O)NCc2cn(C3CN(C(C4C(C(C)C)C4)=O)C3)nn2)cnc2n1CCS2 c1(NCCc2cc(C)on2)nccc(CN2CCCO2)n1 CC1(C)CCC(C)(C(=O)NC2CC3CCC2C(NC(C2CCOC2)=O)C3)CC1 N1(C(=O)OC(C)(C)C)CCCC(O)(NC(=O)NC23COC(C2)C(O)C3)C1 c1(NC(CNC(=O)NCC(c2ccccc2)CC)(C)C)cccnc1 C1(C)(NC(CCSc2n(C)ccn2)=O)CCN(C(=O)Cc2cnns2)CC1 N1(C(C(CSC)OC)=O)CCC(=CCNC(C2CCCN(C)C2)=O)CC1 C1(OC)CC(CNC(c2nnn(C)c2C(F)F)=O)N(C(C2CCN(C)CC2)=O)C1 N1(C(CN(C)C(N)=O)=O)CCN(C(c2cccc(-c3cc[nH]n3)c2)=O)C2CCC12 C12(NC(Cc3nc(C(C)C)sc3)=O)CCC(C1)N(C(c1ccnnc1)=O)C2 N1(C(C23CC(c4ccccc4)C2C3)=O)CCN(C(c2ccnn2CCCO)=O)CC1 N1(C(c2cc(C)sc2)=O)CCOC(C(=O)N(C(C)C(N)=O)C)CC1 CCCC(C(=O)NC1CN(C(c2cnccc2Cl)=O)CC1n1ccnn1)C(C)C C1(CNC(CCN2CCN(CC)CC2)=O)CC(C)(C)CN1C(=O)C(O)CCSC C1(NC(C2C(C(=O)OC)CC2)=O)CN(C(c2nccnc2N)=O)CC2(CCC2)C1 CS(=O)(=O)c1cccc(-c2ccc(CCn3ccnc3)cc2F)c1 N1(C(COc2cccc(C)c2)=O)CCCCC(NC(=O)CSCCN(C)C)CC1 c1(C(=O)OCCC)ccc(OCCNC(=O)CCNC(N)=O)c(OC)c1 Cc1cc(NC(C)C(=O)N(CCC#N)Cc2ccccc2)nn1-c1ccccn1 c1(C(=O)NCC2(F)CN(C(=O)C(c3ccccc3F)F)C2)ccc(F)c(CO)c1 C(Cc1ccoc1)(C(=O)SCC=C)N(CC(=O)NCc1cnsc1)CC N1(C(CC)=O)CC2CN(C(=O)C(n3cc4ccccc4n3)C)CC2C1 C(=O)(C#CC(C)(C)O)NCC(C)(C)C(=O)N1CC2(C1)CNC2.CC(=O)OC CN1CCN(C(C2(CO)CC(C)(C)C2)=O)CC1C(=O)N(C1CSC1)C c1(C(N2CC(NC(C3C4CCC3CC4)=O)C(F)CC2)=O)nccc2ncccc12 c1(CNC(C2N(C(C=CC(C)(C)C)=O)CCC2)=O)cncc(F)c1 Cc1nc(C(=O)N(C2CC(C#N)C2)CC(=O)NC2CC(O)C2O)sc1C C#CC1(C(c2nnnn2CCC2(C)CC2)NCC2(CCO)CC2)CCCC1 C1(c2cccc(C(=O)O)c2)C2CCCCCC12.c12ccc(c(F)c1)-n1nc-2nn1 Cn1ncc2c1CC(C(N1CC3CCC(C1)N3C(c1n[nH]c(=N)s1)=O)=O)CC2 CCCCC(O)CC(=O)NCC1CN(C(=O)C(c2ccc(F)cc2)(F)F)CC1O C=CC(CC)C(=O)N1CC(F)(C(N2CCC(CN=[N+]=[N-])C2)=O)C1 C(CC(CC)C(=O)NC(CNC(=O)Cc1cncc(F)c1)CC(C)C)=CC c1(C2N(C(c3ccsc3C)C(=O)NC)CC2)nc(C)ccc1C(=O)O CC(C(=O)NC(=O)CSc1nnc(S)s1)S(=O)(=O)c1ccc(F)cc1 C(=O)(C(CC)CC)NCC1C(NC(C(C)OCCC=C)=O)C1 N1(C(c2cc(N)cc(C)c2F)=O)CCCC2(CCN(C(=O)CC(C)C)CC2)C1 C1(C(=O)NC2C=CCN(C(C(Cc3ccc(C)cc3)C)=O)C2)CCCC(C)CC1 c1(C(C)NC(c2cccnc2)C(C)OC(C)(C)C)ccc(CCO)cc1 CCC(C)C(O)C(C)C(=O)N1CC=C(C(=O)N(CCC(=O)N(C)C)C(C)C)C1 c1(C(C)C)ccc(C(N2CCC(C(C)NC(c3nsnc3O)=O)C2)=O)s1 C(=O)(C#CC1CCOCC1)N1C(C)CC(NC(=O)COc2cccc(Cl)c2Cl)C1 C1(CN(C(C(CC)n2cncn2)=O)C)CN(C(=O)C2CC2)CC12CC2 c1(C(N2CC(CCNC(COCC#C)=O)OCC2)=O)ccc(C2CC2)nc1C CC(C)C(O)C(C)NC(=O)N(C)C(c1ccc(-n2cccn2)cc1)C C(=O)(CCC(=O)N1CCC(NC(c2ccc(CC(C)C)s2)=O)C1)NCC C1(CNC(COCCCC)=O)CC(C)N(C(c2cnccn2)=O)C1 N1(C(C=CCCC(C)C)=O)CCC(C)C1C(=O)N(CCCO)C C1(C(N2CCC(CC#C)C2)=O)CC=CCN1C(C1CN(C)C1)=O c1(C(N(CC(C)(C)CNC(C2(S(N)(=O)=O)CC2)=O)C)=O)ccc2ncsc2c1 c1(NC(C2(N)CCC(C)C2)=O)ccc2ncn(C)c(=O)c2c1 N1(Cc2cc(OC(C)C)cc(C)c2)CCCCc2ccccc2C1 c1(N(C(CC2N(C(COC(C)=O)=O)CCC2(C)C)=O)C2CC2)c(C)cc(C)cc1C S(=O)(=O)(CCN=c1[nH]c(=NCC2CC2c2cccc(Cl)c2)[nH]c2c1SCC2)NCC CC1CN(C(=O)C#CC2CC2)CC1CC(=O)NCCCc1cnccn1 C1(NC(c2cc(C)[nH]n2)=O)CCC12CN(C(=O)C(N1CCSCC1)C)C2 C1(CNC(C(C)=C2CCC2)=O)(CNC(CCC(C)C)=O)CC12CCC2 N1(C(=O)CC2CCCCO2)CCC2(C(=O)NCCCCC3CC3)CCCC12 C(=O)(C1CCc2nccn21)N1C(CC(N2C3CC(OC)CC2CC3)=O)CC(O)C1 C1(CC)CC(C(=O)NCC2CC(C)N(C(C3CCC(=O)CC3)=O)C2)CC(=O)N1 C(=O)(C(C)(CC)C(=O)NCC1COCCN1C(c1ccc2nn[nH]c2c1)=O)OC N1(C(C=CC=CC)=O)CCC2CC(C1)CN(C(c1cncc(C#N)c1)=O)C2 CCC(CC)C(C(=O)NCC(CC(=O)NCC12CC(CO)(CO1)C2)C1CC1)OC C(C1OCCc2sccc21)NC(c1cc(CC)c(F)cc1)=O c1(NCC(C)OC(C(c2nnnn2CC2CC2)N(C)C)SC)cccc(C2CC2)c1 c1(CNC(C=CCN(C(=O)CC2CCN(C)C2=O)C)=O)ncc(F)cc1F C=C(C)C(C)(C)C(=O)N1CCC1C(=O)NCC1(O)CCN(C)C1 c1(-c2n(C(n3cncn3)C)nc(Cn3nc(Cl)ccc3=O)n2)cc(C(F)F)ccc1F Cc1cc(C)c(C(N2CCCC(CO)(NC(=O)C(C)S(N)(=O)=O)C2)=O)c(S)n1 C(=O)(C(F)CC1CCC1)N(CC(=O)O)NC(=O)CCc1nncs1.C1(N)CCCC1 C(C)(C)(CC=CC(=O)N(C)CCn1cncn1)NC(C(C)OCC#C)=O c1(CCC(=O)NCC2C3CC2N(C(c2conc2C2CC2)=O)C3)cccc(Cl)c1 CCC(CNC(=O)COCCN(C)C)(CC)C(=O)NCc1ccc(O)c(C)c1 N1(C(C2(NC(C)=O)CCC2)=O)CCC(NC(c2c(N)cccc2F)=O)C(CO)C1 c1(COC(c2c(CC)cc[nH]2)=O)c(I)ccnc1O C12(NC(Cc3nc(=N)[nH][nH]3)=O)CCCC1CN(C(c1cocn1)=O)C2 Cc1ccccc1OC(C)(C(=O)Nn1cc(C2CCCNC2=O)nn1)C1CC1 N1(C(C(C(=O)OCC)F)=O)CC2CC(CNC(=O)C(C)(C)CCCO)CC1C2 C1(NCCNOC)CN(C(=O)OC(C)(C)C)CC12CC2 CCCCC(O)C(=O)N1CCC(F)(C(=O)NCC(C)(O)C2CCC2)CC1 c1(OCC)ccccc1NC(C1(NC(=O)CC(C)(C)OC)CC1)=O N1(C(c2cc(CCC)on2)=O)CC2CCC(CNC(=O)CC3CCC(=O)N3)C2C1 c1(C(=O)NCC(CCCC)NC(C2CCCN2C)=O)cc(Cl)cc(Cl)c1[N+](=O)[O-] Cc1ccc(-n2cc(C(=O)NCCCCC3CCOC3=O)nn2)cc1C c1(CC(=O)NCC(C)(C)NC(=O)CNC(=O)C2CC2)coc2cc(Cl)ccc12 N1(C(c2ncn(CC)n2)=O)CCOC2(CCN(c3ncccc3C(=O)OC)C2)C1 CC(C)C(CNC(=O)CC(C)(C)C)C(=O)NCC1CC(C(C)(C)C)C1 c1(CN(C)C(c2cnc(CNC(c3ccccc3Cl)=O)nc2)=O)cccc(O)c1 CC1C(CNC(C)(C)C)CCN1C(C12CC(Cc3ccccc3)(C1)C2)=O Cc1ccc(C(N2CC(CC(N3CCC3C(=O)N(C)C)=O)C3(CC3)C2)=O)cc1O N1(C2CCN(C(C3C(=C)CC3)=O)C2)CCN(C(c2ncccc2N(C)C)=O)CC1 C=CCCCC(C(=O)N1CCOC(C2(C)CC2)C1)NC(c1cnc(C)c(C)c1)=O CCC(C)(CO)C(=O)N1CCOC(CNC(c2ncc(OC(C)C)cc2F)=O)C1 c1(C(=O)NC2CC(CNC(C(CCC)C)=O)OCC2)cccc2c1OCCO2 N1(C(C2C(CC)CCO2)=O)CCN(C)CC1CNC(=O)CCN1CCCCC1 c1(NCC(C)N(C(c2ccc(OC)c(F)c2)=O)C)ncc(C#N)cc1F n1(CC(N2CC3(N(C(CCC#N)=O)CC3)C2)=O)ccc2ccccc12 c1(C(=O)NCC(CNC(C2N=C(C)SC2)=O)O)cc(C)cnc1Cl N1(C(CCOC)=O)CC(CNC(=O)CCCNC2CCCCC2)CC12CCC2 C(=O)(C(C)(C)CCC(=O)NC(C1CCOC1)CNC(c1sc(F)cc1C)=O)OC N1(C(c2cncc(C)n2)=O)CC2CCC2(CNC(c2cc(Cl)c(C)cn2)=O)C1 c1(NC(C2(O)CCN(Cc3c(C)nc(C)[nH]3)CC2)=O)cc2c(cc1C)OCO2 C1(NC(=O)NCc2ccn(CC(C)C)n2)CCCCC1c1nc[nH]n1 CCC(C)C(C(=O)NCC1(F)CN(C(=O)COCCN(C)C)C1)NC(C)=O N1(C(C(C)SCC)=O)CCN(C(c2cc([N+](=O)[O-])n[nH]2)=O)CC12CC2 C=C(C)CC(C(=O)NCC(C)(Cl)CC)NC(=O)Cc1ccsc1C C(=O)(C(C)(C)C(=O)N(C)CC1(CNC(=O)CCCSc2cccs2)CC1)OC Cc1c(C)n(C)c2ccc(NC(=O)CNC(C)Cc3ccc(Br)s3)cc12 c1(CC)cc(C(=O)NCC2CC(NC(C3C4CCC3CC4)=O)C2)ncn1 c1(C(N2C(CNC(C3(C#C)CCC3)=O)CCC2)=O)sc2ccc(F)cc2c1C CC1(CC(=O)NCCC(O)CNC(c2ccnc(C(N)=O)c2)=O)CC(F)(F)C1 C=CCCC(C)(c1nnnn1-c1ccccc1OC)NCC1C(C)(C)C1(C)C N1(C(C(C2CCOCC2)OCC)=O)CCOCC(F)(CNC(=O)CC(F)F)C1 n1(CCC(=O)NCC(C2CC2)NC(c2cnc(S)[nH]2)=O)ccc2cc(Cl)ccc12 C1(CNC(c2c[nH]nc2Cl)=O)CCCCN(C(=O)CCc2ccoc2)C1 c1(CC)cncc(C(=O)NC2CC(C)N(C(=O)Cc3cn(CC)nn3)C2)c1 C(=O)(C(CC1CC1(F)F)N(C1CC1)CC1CC1c1ccco1)NC CC1CCC=C1C(=O)NC1CCCCC1CC(N1CCCC1C1CC1)=O S(=O)(=O)(c1c(Cl)cc(Br)cc1Cl)NCCC(=O)Nc1ccc2c(c1)OCCO2 N1(C(c2cnc(SC)s2)=O)CC(C)N(C(=O)CCc2cc[nH]n2)CC1C CC(C)CC(C(=O)NC1CC1NC(=O)C1=CCOC1)NC(=O)OC(C)(C)C C(=O)(C1=CCCOC1)NC(C)CCN(C)C(C1(C)CCN(C)C1)=O CN=C(NCC(C)C(F)F)NCC1CCC(C(F)(F)F)O1 C1(NC(CC=CC)=O)CCCCC12CCCN(C(=O)Cn1nccc1C)C2 C1(C(=O)NC2CC(C(=O)NCCc3cncs3)OCC2)CC(C2CC2)=NO1 CN1C(=O)CCCC1C(=O)NCCOC(C)(C)CNC(C1CCCN1C=O)=O c1(OCCOC)ccc(CC(=O)NCCN(C)C(c2ccc(C(N)=O)o2)=O)nc1 C1(N(C)CCn2cc(C3CCOC3)nn2)CCN(S(C)(=O)=O)CC1 N1(C(c2cc(C(C)(C)C)oc2)=O)CCC(Cc2cn(C3CCCCC3)nn2)CC1 CCCCC(F)C(=O)NC1CC(C(C)NC(c2[nH]nnc2CC)=O)C1 N1(C(c2cc(C)ncn2)=O)CCC(C)C(NC(=O)CCC2CCCO2)C1C CN1CC=C(CC(=O)N(C)CC2CCCN(C(C3(C)CCCS3(=O)=O)=O)C2)CC1 c1(N(CC(C)(C)C2CC2)C(=O)CCC2CCCC2)cccc2ccccc12 c1(NC(=O)C(N2CCC(c3nccs3)CC2)=O)ccc(F)c(Br)c1 CC1(C)COCC1CC(=O)NC1COCC1CNC(c1cnc(=N)[nH]c1)=O C(c1ccoc1)=CC(=O)NC(C1CCCC1)CNC(C(C1CCC1)OC)=O Cn1c(NC(c2ccc(S(N)(=O)=O)s2)=O)nc2ccc(Cl)cc12 C1(C(=O)NC23CC(CNC(c4c(C)ncs4)=O)(C2)C3)CCCN(c2nccs2)C1 c1(CNC(=O)NC(C)(C)COC(C)(C)C)ccc(CNC(C)=O)o1 c1(OC)ccc(CCN(C)C(=O)NCCc2cccc(OCC#N)c2)cn1 c1(C(N(CC(CC)NC(=O)CC(F)(F)Cl)CC)=O)cnc2[nH]nnc2c1 C1(CC)CC2CCC(C1)N2C(c1cccc(CO)n1)C(=O)NCCCSCC1CC1 C(=O)(C(C)(C)CC1CCOC1)N(CCCCNC(c1cn(C(F)(F)CO)nn1)=O)C c1(C(N2CC(NC(c3c[nH]c(=O)cn3)=O)CC(C)C2)=O)cc([N+](=O)[O-])ccc1Cl CC1(C)CC1(C#N)C(N1CCC(C)(CC(=O)NCCN2CC(CF)C2)C1)=O C1(CC)CCC(=O)N1.C(C(=O)NC(C)COC(C)=O)SCC c1(COC(c2cc(F)ccc2C2CC2)=O)ccc2c(n1)COCC2 C1(CC#C)(C(=O)NC2COCC2NC(=O)Cn2ccnn2)CCCC1 CC1CN(C(=O)CC(C)(F)F)CCCN1C(c1cccc(C(F)(F)F)c1)=O N1(C(c2cncc(C)c2)=O)CCCC2CN(C(=O)CC3CCC3)CCCC12 CC(C)C(C(=O)NCc1ccc(Br)s1)N(C)C(=O)OC(C)(C)C.C1C(=O)N1CCO C=C1CCC(C(=O)NCC=CCNC(C2CCCN2C(=O)C(C)C)=O)CC1 N1(C(C(=O)NC(c2ccc(SC)c(Br)c2)C)=O)CC(F)(F)CC2(CCC2)C1 CCCCC(C)(F)C(=O)N1CC(CNC(C2CCCS2)=O)(COC)C1 N1(CCCCOC)CCCN(C(=O)C(N)C(C)C2CC2)CC1 N1(C(C(C2CC2)OCC)=O)CC2CCN(C(=O)C=Cc3csc(C)n3)C2C1 c1(-c2c(COC(C)C)cccc2)cc(=O)n(C)c2ccc(Br)cc12 CC1CN(C(C2CCC(=O)C2)=O)CC1NC(c1cc(CF)on1)=O C(=O)(C(C)CCCc1ccccc1)N(CC(C)CNC(C1(P(C)(C)=O)CC1)=O)C C1(CNC(=O)C#CC2CCOC2)CCC2(CO1)CC(O)C2 C1(C(=O)NC2(COC)CN(C(=O)C=CC(C)(C)C)C2)CC(C)CC(=O)N1 N1(C(CSCCCC)=O)CC(O)(C(C)(C)CNC(=O)C=CC2CCCO2)C1 N1(C(c2ccc(OC)[nH]2)=O)CCC(C2CCN(CCn3cc[nH]c(=O)c3=O)C2)CC1 n1(CCCC)nnnc1C(c1cnsc1)NC(c1ccn(-c2ccccc2)n1)C CCC(CCC(=O)NCc1ccnc(C)n1)NC(=O)CCCCSC C1(OC)CN(C(c2scc(C)c2Cl)=O)CC1NC(=O)C(F)(F)C12CC(C1)C2 c1(CC)oc(C)cc1C(=O)NCCC1CCCN(C(=O)C(n2ccc(C)n2)C)C1 C1(C(C)C)CN(C(c2cnn(CCF)c2)=O)CCCN1C(C1CC=CCO1)=O N1(C(CCCOCC=C)=O)CC2(C(=O)NCc3nn(C)cc3CO)CC1CO2 c1(C(=O)NC2C(CNC(CC3CN(C(C)=O)C3)=O)CCC2)oc(Br)nc1C C(=O)(CC(C)(C)CNC(=O)C(c1ccccc1)F)N1CC(C)(C(=O)OC)C1 c1(CC)ncncc1C(N1CCC(N(C(=O)C(O)CCc2ccccc2)C)C1)=O N12CCSC(C1)OCCNC2=O.C1(OCCO)CN(CC(F)(F)F)C1.C1CO1.C1CO1 C1(CC(=O)NC2CCC(CO)C2)C2CCC(C2)N1C(=O)C=Cc1cc[nH]n1 CC(CS(C)(=O)=O)C(=O)NC(C)C(C)NC=O.c1(N)csc(=NC)[nH]1 c1(C(O)CNC(=S)NCC2CC2(Cl)Cl)ccccc1Br C1(CC(=O)NCC(N2CCCC2CO)=O)C(SCC2CC2)C1(F)F.C1C(=O)N1 N#Cc1ccc(C(N2CCC(CC(N3CC(N(C)C)C4(CC4)C3)=O)C2)=O)cc1 C1(NC(c2n[nH]c(C)c2Cl)=O)C2CCC1CN(C(=O)C#CC1CCOC1)C2 C1(NC(CCCCOC)=O)CN(C(C2CC23CC(C)(C)C3)=O)CC(C)(C)C1 c1(OC)cc(C)c(C)cc1C(N1CC(N(C)C(C2(F)CCOC2C)=O)C1)=O N1(C(CCCNC(=O)OCC)=O)CCC(NC(=O)C2=CSCS2)C12CCC2 c1(C(C)(C)C)nccc(C(=O)OCc2csc(I)n2)n1 C1(N(C(C2N(C(c3ccc(OC)s3)=O)CC(F)C2)=O)C)CCCC(C)C1C c1(COC(C2CC3CC3N2)=O)cccc(Oc2ccccc2)c1 Cc1c(CC(N2CCN(Cc3nn[nH]n3)CC2)=O)nc(Br)n1C c1(C(=O)NC2(CC=C)CCS(=O)(=O)CC2)cnc2c(c1)NC(=O)CS2 N1(C(CC(=O)OCC)=O)CCC(NC(=O)CC2OCCCC2(C)C)C(C)(C)C1 C1(N(CC(CNC(CNS(CC)(=O)=O)=O)C)C)CCN(CC(F)(F)F)C(=O)C1 Cc1cc(C(=O)NC(C2CCCC2)CNC(C2CCCCN2C)=O)c(F)cc1N c1(CCC=C=C)nc2nn1c1ccccc21.C(CCC)S N1(C(c2c(CC(=O)OCC)cccc2)=O)CCCCCCC1CC c1(C(=O)NC(C)CN(C)C(c2cnn(C3CC3)c2)=O)cc2ccsc2n1C c1(C(=O)NC2CC(CNC(c3ccc(C#C)cc3)=O)C2)onc2ccccc12 c1(C(N(CCCNC(C2(OC)CCC2)=O)C2CC2)=O)nc(O)[nH]c1 c1(N2CC3C(C(N4CCCC(CO)C4)=O)(C3)C2)ncnc2c1CCC2 C=C(C)CCCC(=O)NC1CCN(C(C2CN3CCC2CC3)=O)CC1F C1(N(C(COCc2cc(C)no2)=O)C)CCCC(NC(=O)CCC2CCCC2)C1 N1(C(=O)Nc2ccnn2C(F)(F)F)CCOc2cc([N+](=O)[O-])ccc2C1 c1(C(N(C)CC2CCOCC2)=O)cc(CCNC(=O)C(O)C2CC2)on1 c1(CC)onc(C(N2CCC2CC2CCCN(CCn3cc(C)cn3)C2)=O)c1C c1(CCC)cn2ccccc2n1.c1(OCC)nnc(CN(C)CCOCCO)s1 C1(C(=O)Nc2c(C)cccc2C)Cc2nccnc2CN1Cc1ccc(F)cc1 C(c1cnc(C)s1)=CC(=O)N(CCN(C(=O)CCN1CCCCC1=O)CC)CC C1(CCC)CC(C(=O)NC2CCC(C(=O)Nc3nnc(C)n3CC)CC2)CCO1 N1(CC)CC(C(=O)NCC(C)NC(=O)C(F)C2CCCC2)CCC1=O C1(NC(C2(SC)CC2)=O)CCN(C(=O)C(=C2CCCCC2)F)C1 c1(C(N(C2C3CN(C(C(C)(C)SC)=O)CC32)C)=O)ccnc2nc(C)nn12 C1(C(=O)NC2CN(C(c3c[nH]cc(F)c3=O)=O)CC2O)CC1C1CCOCC1 CC(CC(=O)N1CCCC1C(C)C)NC(=O)C=CC(C)(C)C.C(N)=O C1(COC(=O)Cc2ccc(N3CCCCCC3)cc2)CCCC(F)(F)C(=O)N1 CN1CCCC1(C)C(=O)NC1CC(CC(=O)N(C2CC2C2CC2)C)C1 C1(C(=O)NC2C(C)(C)CN(C(=O)OC(C)(C)C)C2)(CO)CCS(=O)(=O)CC1 N(C1CN(C(C2(CF)CC2)=O)Cc2ccccc21)C(C1CC(C(=O)OC)C1)=O C12(CNC(c3ncc(CC)cn3)=O)CCC(CC1)N2C(=O)C(C)c1cccs1 Cc1[nH][nH]c(=NC(=O)c2ccc(CNC(=O)CC(O)c3ccccc3)cn2)c1C c1(C(N2CC(C(C(=O)NCC3CC(F)(F)C3)O)C2)=O)coc(C2CC2)n1 c1(C(N(C(C)CNC(=O)C=CC(=O)NC)CC)=O)ccc2c(c1)CCCC(=O)N2 c1(N(C)CCc2nccs2)nc(=NCC2CCCO2)[nH]c2c1CCCCCC2 c1(CC)cccc(C(N2CC(F)(F)CC2CCO)C(=O)NCCCF)c1F C(=O)(C#CC1(C)CCCO1)NC1CC(NC(C2C(C)(C)NC(=O)C2)=O)C1 C1(C(=O)NCC2CCN(CC)C2)CN(C(C2CN3CCN2CC3)=O)CCN1C N1(C(c2scc(C)n2)C(=O)NCC2CCCO2)CCCC12CCOCC2 N1(C(CC(OCC)OCC)=O)CCCC(C)(C)C1CNC(c1nc(C)ccc1O)=O Cc1ccc(C)c(CCN2CCOC(C)C2)c1.N12CCCC(C1)C(=O)NC(=O)C2 C1(C(=O)NCC(CC(C)C)NC(C(CC)F)=O)CC2CC(O)CC(C1)C2 CC1CCCC1(C(=O)NCC1(F)CCOC1)NC(=O)C=Cc1ccncn1 C#CCC(C)C(=O)NCC1CN(C(=O)C(C)Cc2ccccc2)CC1C N1(C(C(C(C)C)OC)C(=O)NCCSC)CCOC2COCC12 N1(C(CC2C(NC(CCCOC)=O)CC2O)=O)C2CCCC1CC(O)C2 c1(C(=O)NC(CCN(C(CCSCC)=O)C)C)cc2cc(F)c(F)cc2[nH]1 N1(C(COCCC#C)=O)CCN(C(c2cc(Cl)ccc2Cl)=O)C2(CC2)C1 C(C(=O)N=c1ccn(C(F)F)[nH]1)C1(NC(C2CC23CCCCC3)=O)CCC1 Cc1c(C(=O)NC2(C(=O)NC3CC(=O)N(C)C3)CCN(C)C2)cccc1F C1(NC(CC=C)=O)Cc2ccccc2C1NC(C1CCCCC1n1cccn1)=O c1(C(C(C)(C)C)NC(=O)NCC(C)OCCC)cccc(Br)c1 C1(NC(=O)NCC(CNC(COCCOCC)=O)CO)CCC2(CC1)CC2(F)F C12(C(=O)NCC3(c4ccc(OC)cc4)CCOCC3)CCCC(CO1)C2 C1(C2CCN(C(c3ccnn3CCC)=O)C2)(NC(C(CCC#C)O)=O)CC1 C1(C(=O)NC(C(C)NC(C2(C(N(C(C)C)C)=O)CC2)=O)C)CCS(=O)(=O)C1 n1(C(C)C)ccc(C(N2CC(NC(=O)CC3CSC3)CC(F)C2)=O)cc1=O N1(C(C(CCC)O)=O)CC2CC(NC(c3ccc(CC(F)(F)F)cc3)=O)C(C2)C1 C(CO)(CN=C(NCC1(F)CC1)NC1CCCC1)c1ccc(C)o1 C1(CNC(C(C)(C)OCCC)=O)CCC2(CCC2)C1O c1(CCNC(=O)NCc2nc(-c3cccc(I)c3)n[nH]2)cnn2c1C(=O)NCC2 C(=O)(C(CO)C(F)(F)F)NC(C(N1CC(C#C)C1)=O)CO C1(CC)CN(C(C2CCCN(C(=O)C=CC(=O)N(C)C)CC2)=O)CC(=O)N1 C(=O)(C(C)(C)C(=O)NCCCNCCCC(C(=O)NCCOC)C)NC N1(C(C2CC(C)N2C(C2CCC(C3CC3)C2)=O)=O)CCN2CCC1CC2 c1(C(=O)NC(C(C)C)OC(=O)NCCNC(=O)OC(C)(C)C)sccc1Br C=CCC(CC(=O)NC1CCCN(C)C1=O)NC(=O)Cc1cccc(F)c1 C1(CNC(CC(CC)OC)=O)CCCCCN1C(=O)Cc1cc(C(F)(F)F)ccn1 CC1CCC(OCC(=O)N(C(C)CCNC(C2(C)CCC2)=O)C)CC1 c1(CNC(CC)(CC2CC2)c2nnnn2-c2ccc(Br)cc2)c(C)cc(O)cc1C C=CC(CC)C(=O)NCc1cc(C(=O)NC2CC=C(C)CC2)on1 CC1CN(C(c2cn(CC3CNC(=O)O3)nn2)=O)CCN1C(c1ccoc1Cl)=O N1(C(C2(CCC)CC2)=O)CC2(C)CC1(C(=O)NCCC1(C)N=N1)C2 c1(C(N2CC(=C(CNC(C(C)N3CCCC3)=O)F)C2)=O)ccc(=O)n(C)n1 N1(C(=O)C=Cc2cnccn2)CC2CCCC2(N=c2[nH]ncs2)C1 CC(C)CC(C)(CO)NC(C1CCCN(C(=O)C(O)C(C)C)C1)=O N1(C(CC(C)C2CCCCC2)=O)CCCC(N(C(C2CC(O)C2)=O)CC2CC2)C1 C1(NC(c2c(OC)c[nH]n2)=O)CCCN(C(C2CC(c3ccccc3)CO2)=O)C1 C1(NC(C2C(C)(C)CCCO2)=O)CC12CCC(NC(=O)CSCC(F)F)CC2 c1(CC)cccc(C)c1C(N1CC2CC2(NC(=O)CC2(C)CC2(F)F)C1)=O N1(C(c2cncnc2)=O)CC(C2CC2C(N2CC(O)(C(F)(F)F)C2)=O)C1 c1(NC(C2CCCN2Cc2cccc(Cl)c2F)=O)cccc(F)c1CO C1(O)(CNC(C2CCOC2)=O)CN(C(c2ccoc2Br)=O)C1 c1(C(N)CO)cccc(C(=O)Nc2cscc2Br)c1 N1(C(c2c(C(C)C)noc2)=O)CCOCC(F)(CNC(c2ccnnc2)=O)C1 C1(COC)(NC(c2cn(C)c(C)n2)=O)CCN(C(c2ccc(C)nc2C)=O)CC1 C1(NC(C(C)N(C)C(C2CC3(CCC3)C2)=O)=O)COC2(CCCC2)C1 Cc1nc(C)c(C(N2CCC2c2cn(C(C3CCOCC3)C3CCCC3)nn2)=O)o1 N1(C(CCC(CC)C)=O)CCC2(CCCC(CNC(c3csc(Cl)n3)=O)O2)CC1 C1(C(=O)NC)CCC(CNC(N2CCC(c3nccc(C)n3)CC2)=O)CC1 c1(SCCc2ccc(C(=O)NC(c3ccc(C)s3)C)cc2)ccc(F)c(F)c1 N1(C(COC(C)=O)=O)CCC2(NC(=O)CCOc3cccnc3)CCCCCC12 C(=O)(C#CC(C)(C)O)N1CC(CCCNC(C(C)(C)C2CCCCO2)=O)OCC1 CC(C)CC(C(=O)N1CCCC1CCNC(=O)CC1CCCC(C)(C)C1)N(C)C Cc1ccc(C(=O)NCC2CCN(C(c3oc(Br)nc3C)=O)CC2C)cc1O C1(NC(CSCCC)=O)CN(C(c2ccc(N)c(Cl)c2)=O)CCC1CO N1(C(C=CCNC(c2ncc(NC)nc2)=O)=O)CCCCC(CO)C1 N1(C(CC2N(C(C3CC(C(C)C)C3)=O)CC2)=O)CCC2(CC=CCO2)C1 C(C(C)(CC(C)C)NC(=O)Cc1nncn1C)NC(c1nc(C)oc1C)=O c1(C(=O)NC(CCC)CNC(=O)CCC2CCCOC2)ncccc1N C(N=c1[nH]cncc1F)C1(C(F)(F)F)CN(OC(C2(NC(C)(C)C)COC2)=O)C1 N1(C(C2OCCN(CC)C2)=O)CC2CCC(C1)N2C(c1ccc(F)cc1O)=O N1(c2ccnc(C(C)(C)C)n2)CC(NC(=O)Nc2ccc(Br)nc2)CC(C)C1 c1(OCC(=O)NC(C2CCN(C(C3(F)CCCOC3)=O)C2)C)ccc(Cl)c(F)c1 c1(SC)cccc(F)c1C(=O)NC1CC(NC(=O)C(C)(C2CCOC2)NC(C)=O)C1 C12(NC(C(CCC)C#N)=O)CCCC1CN(C(c1[nH]nc(C(F)(F)F)c1C)=O)C2 C(N=c1cc(NC(C)CN2CCCCC2)nc[nH]1)c1cc(C)cc(C)c1 N1(C(c2ccc(C(C)C)o2)=O)CCCN(C(c2scc(Cl)c2Cl)=O)CCC1 CCCC(C)CC(=O)NC1C2CC3C(C2)C13C(N1CC2(CC2)CC1CO)=O c1(C(=O)NC2(CNC(C3(C(C)C)CCC3)=O)CC2)cccc2oc(N(C)C)nc12 c1(C(=O)NC2CC(NC(CCCOC)=O)CC2O)cc2sc(C(=O)OC)cc2[nH]1 C1(CNC(C(C)(C)NC(=O)OC)=O)CC2(CCN(C(c3nnc(C)s3)=O)C2)CO1 C1(C(=O)NC(C)CCCNC(=O)CSc2nncs2)CC2(C1)CC(F)(F)C2 c1(C(=O)NCC2C(C)CCN(C(C3CC(OC)C3)=O)C2)cc(C#N)c(N)cc1O CN1C2CCCC1CN(C(CCC1CCCCC1)C(=O)NCC1CCOC1)C2 CC(C)(CNC(=O)CN1CC2CC2C1)CCNC(=O)Cc1n[nH]cc1Br C1(C(=O)NCC(CC(=O)N(CCC(=O)NC)CC)C)CC(=O)NC(=O)C1 c1(OC)ccc(CNCC(c2cccc(C)c2)F)cc1 C(C(CC(C)C)C(=O)N(C)CCOCCN(C(=O)C(C)(CO)N(C)C)C)OC c1(C(=O)NCCC(=O)NC2C(CN(C)C)C2)cc(F)cc(F)c1 C(=O)(C(C)(C)COC)NC.C1(OCC(N2CC=CC2)=O)CN(C(N)=O)C1 C12(n3cc(CCCC(=O)OC)nn3)CN(C(=O)C(C(C)O)OC)CC1(N(C)C)C2 N1(C(c2c(CC)onc2C)=O)CCC(C)C(NC(=O)CSCc2cccnc2)C1 N1(C(C23CC(NC(c4c(C(=O)OC)cnn4C)=O)(C2)C3)=O)CC2(C1)CN(C)C2 N1(C(C=CCOC)=O)CCC(C(=O)N(C)Cc2ccc(F)cn2)C(C)C1 S(=O)(=O)(c1ccccc1)NC(C(=O)NC1CC(CNC(C2(CC=C)CC2)=O)C1)C CCCCCC(=O)NC1CN(C(=O)C(c2cccc(OC)c2)(F)F)CC1C C1(C(N(C)CC2CN(C(C3CC(n4ccnc4)C3)=O)C2)=O)CCCN1S(C)(=O)=O CC(F)(F)C(F)(F)CC(=O)NCc1ccc(F)cc1CO C1(CC(=O)N(CCCNC(c2c(C)nsc2C)=O)CCC)CC2(CCO1)CC2 c1(C(=O)NC(CN(C)CC)C)ccc(OC(F)(F)F)cc1C C1(N(C(C2CCN(CC)C2)=O)C)CCN(C(=O)CCn2cccc2)CC1 N1(C(C2CCSC2)=O)CCCC1C1CCCCN1C(C12CC3CC1C2C3)=O C1(C(N2CCN(CCN(C(=O)C(F)OC(F)(F)F)C)CC2)=O)CCC2(CCC2)OC1 c1(OC)cccc(C(CF)NC(=O)NCC2CCN(CC(C)O)CC2)c1 N1(C(CC(C)(C)OC)=O)CCC2CN(C(=O)Cc3c(C)cccc3C)CCC2C1 c1(C(N2C(CNC(C(C)NC(C)=O)=O)CCCC2)=O)c(C)nn(CC(F)(F)F)c1Cl C1(CC(=O)N(c2ccsn2)CC)CCCN(C(=O)CCCC2CCCC2)C1 C1(C(Cn2cc(CN(C)CC)nn2)C)CCN(C(=O)Cn2c(C)csc2=O)CC1 C(C(C(=O)N1CC2COCC(C2)C1)C(C)(C)C)NC(CCCC=C)=O C1(C(N2CC(NC(c3nc[nH]c3C(F)(F)F)=O)C(O)C2)=O)CC2(CCOC2)C1 C=CCCCC(C(=O)N(C)Cc1csnn1)NC(c1ccoc1)=O C1(C(=O)NCCC2(O)CN(C(C=CC(CC)C)=O)C2)CCn2c(C)nnc2C1 c1(C(=O)NC(CC)CNC(c2ccnn2C(C)C)=O)ccc(CC(F)(F)F)cc1 C1(NC(CCN(C(=O)CS(=O)(=O)CCOC)CC)=O)CCn2cnnc2C1 C1(NCCN(C)C(C)C)=NC2=CC(=NCC(C)(C)N2)N1.C(C)(C)(C)OC c1(OC)c(C)csc1C(=O)NCC1CC(NC(c2cc(-c3csc(C)n3)c[nH]2)=O)C1 C1(C(=O)NC(CN(C(C(c2ccc(OC)cc2)=O)=O)C)C)CCC2CC1CO2 C1(NC(C(C)(C)NC(C)=O)=O)CCCC(C(N2CCCC2(C)C(C)(C)C)=O)CC1 CP(C)(=O)c1cc(Br)ccc1CNC1CCOC(C2CC2)C1 N1(C(c2c(CC)cc[nH]2)=O)CCC12CC(C(=O)NOCC(C)(C)O)C2 C1(C(=O)NC(c2cccc(OCC(=O)O)c2)CC)CCC(S(C)(=O)=O)C1 N(C1CC(C)Oc2cc(F)ccc21)CCn1cc(-c2c3ccc(C)cc3sc2)nn1 C(C(C)(C(C)C)NC(=O)Cc1ccccc1Cl)NC(C12CC(C(=O)OC)(C1)C2)=O C1(CNC(C2CCC(C)O2)=O)CCC(CNC(c2cnn[nH]2)=O)CC1 N1(C(CCC)C(=O)NCc2nnn(C)n2)CCC2CC1(C(=O)OCC)C2 Cc1cc(C)cc(S(=O)(=O)N2CC(N(C)C(c3cc(Cl)c(O)cc3O)=O)C2)c1 c1(C(N(C)CC2CCCN(C(C(C(C)O)N(C)C)=O)C2)=O)cnn2ncccc12 CCCCC(C)(F)C(=O)N(C)CCN1CCN(C(C2C3CCC2CC3)=O)CC1 c1(C2(C(N3C(C)C(NC(C4CCC4(F)F)=O)CC3)=O)CCC2)ccc(F)c(F)c1 C1(CNC(CCOC)=O)CC(C)(C)CN1C(=O)CCCNC(C1CCCCO1)=O C1(NC(C2N(CC)CCOC2)=O)CN(C(=O)C(c2ccccc2)F)CCC1CO CCC(C)CC(C(=O)NCC)NC(=O)C(C)(Cl)Cl.c12ccc(cc1)CN(CC)C2 C1(C(N(CCCO)CC#C)=O)CCOCCN1C(=O)CCCF C1(C(=O)NC(C)CNC(c2nc(C(C)(F)F)cs2)=O)CNC(=O)C(C)(C)C1 N1(CCC(=O)NC(CC(C)C)C)CCC(O)C(NC(=O)CNC(=O)C(C)(C)C)C1 C1(C(C)C)CN(C(=O)C(O)Cc2cnc[nH]2)CCN1C(=O)C=Cc1ncc[nH]1 Nc1ccc(C(N2CCCC2CCC(=O)NCCCc2cccs2)=O)nc1 CCS(=O)(=O)CC(=O)NC1CCC(CCNC(c2csnc2C)=O)C1 N1(C(C(CC2CC2)NC(CNC(CN(C)C)=O)=O)=O)CCNC(=O)C1C C(=O)(C1=CCN(C)C1)NC(C(=O)N(CC)Cc1cccnc1)COC CCCC(O)CC(=O)N1CCCC(C)(CNC(C2(c3ncco3)CC2)=O)C1 C1(C(N2CC(CC=C)(NC(C(C=C=C)C)=O)C2)=O)CCC(C#N)CC1 N1(C(c2c(C)noc2)=O)CC(CC(=O)N(C2CN(C)CC2O)C)CC1C CCC(C(=O)N1CC(NC(=O)CCc2cccc(OC)n2)CCC1C)C(C)O c1(CNCCc2nnc(C)s2)cc2scnc2[nH]1 C(=O)(C(CO)C(C)(C)C)NCCCC1N(C(c2ccc(OC)cc2N)=O)CCC1 c1(C(N2CCC(N(C(=O)OC)C)CC2)C)ccc(OCc2ccc(Br)cc2)cc1 N1(S(c2scc(C)c2)(=O)=O)CC2CN(C)CCC2(c2ccc(CNC3CC3)cc2)C1 Cc1cc2[nH]c(C(=O)NC(CNC(=O)CC3NC(=O)NC3=O)C3CCC3)cc2o1 C=CCC(CC(=O)NC(C)(C)CF)NC(=O)CCc1cncs1 O=C(C1=COCCO1)NCCC1(NC(C2CC2c2cccc(Br)c2)=O)CC1 C1(CC=C)(NC(=O)CNC2CCOC2)CCCN(C(C)=O)C1 c1(NC(C(CCC)C)C)cc(C(=O)N(C)Cc2ccccc2)ccc1Cl c1(C2C(C(=O)NCC(C)(C3CC3)N(C(c3csc(Cl)n3)=O)CC)C2)cccc(Cl)c1 n1(CC)nc(C(N2CCC2C(=O)NCc2cscn2)=O)cc1C C1(C)(C(N(C)Cc2ncc(C)o2)=O)CCCN(C(c2nccnc2N)=O)C1 CC#CCCCC(=O)NC1CCN(C(C2(F)CC3(CCC3)C2)=O)CC1CO C(=O)(CCCCC(C)(C)C)N1CC(NC(C(CC(C)C)N(C)C)=O)N(C)CC1 c1(C(=O)NCC2CCCN2Cc2ccccc2Cl)ccc2nc(O)[nH]c2c1 c1(S)ccccc1.C(F)(C(=O)N(CC(C)N(C(=O)C(O)C1CCC1)C)C)=C(C)C c1(C(=O)NC2C(C)CCN(C(c3csnc3Cl)=O)C2)ccc2ncnn2c1 C1C(C)(C)C(=O)N1.Cc1ccoc1C(=O)NCCC(C)N(C)C(C)C c1(N(C(c2oc(C)c(S(N)(=O)=O)c2)=O)CC2CC2)ccc(Br)c2cccnc12 c1(NC(C2C3CN(Cc4cnc(CCC)s4)C2C3)=O)cc(F)c(F)c(F)c1Br C1(NC(c2n(CC)cc(Cl)c2)=O)CCN(C(c2csc3ccsc23)=O)C1C C1(CS(=O)(=O)N(c2ccc(C#N)cc2)CC(C)C)Cc2ccccc2C1 c1(CCC(=O)NC(c2ccccc2Cl)(C)C)ccc2ccccc2c1 c1(C(=O)NCC2N(C(CN3CCC(C)C3)=O)CC(C)(C)C2)ncnc2ccsc12 Cn1cc(C(=O)NC2CC2CNC(=O)CC2CC(F)C2)c(=O)n(C)c1=O N1(C(C2(SC)CC2)=O)CCC2(CCCC2CNC(c2cc(C)ccn2)=O)CC1 Cc1nccc(C(=O)NC(C2CCCC2)CNC(c2nc(Cl)cs2)=O)c1C c1(C(=O)NCC(CC)(C)NC(C2CCCCNC2=O)=O)cccc2nn[nH]c12 C1(CC)CCC(C(=O)NCC2COCCN2C(c2cn(C)cn2)=O)CC1 c1(OC)ccc2[nH]cc(C(=O)NC(CCN(C(=O)C=C3CCC3)C)C(C)C)c2c1 c1(C(N2C(CN(C(C3C(C=C)C3)=O)C)CCCC2)=O)cccc2c1OCC2 c1(C(N2CC(CCNC(CC(C=C)(C)C)=O)C(C)C2)=O)c[nH]c2nc(F)ccc12 C(=O)(C(CN(C)C)C(C)C)NC(CC=CC)C(=O)NC1CCC(C(=O)OC)C1 N1(CCOC)CC(C(=O)NC2CCCC2NC(=O)C(F)(F)C2(OC)CCC2)CC1=O CC1CCC(NC(c2nc(Br)cnc2N)=O)CN1C(C1(C2CC2)CCC1)=O C1(NC(c2c(C)snc2)=O)CC2CN(C(c3cnc(N)c(CO)c3)=O)CC12 CC(C)C(C(=O)N1CC(C(=O)NCc2ccnn2C)C(F)C1)n1ccnc1 C12(C(N3CC(CCC)C(NC(C4CC(C(C)C)=NO4)=O)C3)=O)CCCC1C2(F)F C1(c2c(C(=O)OC(C)(C)C)c[nH]n2)CCN(N2CC3(CCN3C3CC3)C2)CC1 n1(CCCC)nnnc1C(c1ccoc1)NCC(c1ccc(Cl)s1)C C1(CC(=O)NC)CCCCC1N=c1[nH]c(=NC2CN(C)C2)[nH]c2cc(C)ccc12 N1(C(C2(SC)CC2)=O)CCN(C(=O)C(S(C)(=O)=O)C2CC2)C(CCO)C1 CCC(C)(C)C(C)CC(=O)N1CCC(CNC(c2cc(C)n(C)c2)=O)(OC)C1 Cc1cc(C)c(C#N)c(N2CC3(CCCC(CNC(C4(O)CCC4)=O)O3)C2)n1 N1(C(C(CSC)C)=O)CC2(CCC(NC(C3(C)CCC(C)C3)=O)CC2)C1 c1(C(=O)NC(CC)CNC(=O)C2=C(C)OCCS2)nn2ccccc2c1Br C1(CNC(COC(CC)CC)=O)N(C(=O)C(C)C#N)CCC1(C)C CC1CC(C(N2CC(O)(CO)C2)=O)N(C(=O)CC(O)C2CCCC2)C1 C1(C)(C(N(CCOC)CCNC(=O)COc2cccnc2)=O)CS(=O)(=O)C1 c1(OC)ccc(C2(C(N3CCCC(CN4CCC(C)C4)C3)=O)CCC2)c(F)c1 Nc1cnn2ccc(CC(N3CCC(c4nn[nH]n4)(C(=O)O)CC3)=O)cc12 Cc1cccc(C(CO)NC2(CC(=O)NC(c3ccc(S)cc3)=O)CCC2)c1 c1(C(=O)NC(COCCCNC(C(CC)F)=O)(C)C)cnc(C(C)(C)C)nc1 c1(OC)cc(OC)cc(C(O)CNCc2cc(C3CCCO3)n(C)n2)c1 CC1(C(=O)NC2CCC(CC(=O)NOCCCF)C2)CCCCC1 CCC(O)(C(=O)N1CCC(NC(c2cncc(F)c2)=O)C1)c1ccccc1 C12(C(N3C(CCC)CCC3)=O)CCCC1CCN2C(=O)CC(C)(C)C N1(C(c2c(C(C)(C)O)cncn2)=O)CCC(c2ccccc2)C(c2ccccc2)C1 CC#CC1CCN(C(C2CC23CCN(C(=O)C(n2ccnc2C)C)C3)=O)C1 CC1(C)CN(C(C2CCCN2C2CC2)=O)CC1NC(C1CC2C=CC1O2)=O C1(COCC)CN(C(=O)CCCN(C)C)CC1CC1CC1 c1(NC(C=CCNC(CCC#C)=O)=O)cccc2occc12 C1(O)(CC(=O)NC2CC(CNC(CC3CC(CC)C3)=O)C2)CCCOC1 c1(CNC(C2CCCN(c3ccc(Br)cc3)C2=O)=O)cccc(F)c1Cl Cc1nc2c(s1)CCCC2C(=O)NCC1CN(C(=O)C(C)O)CCC12CCC2 C(C(C(C)C(C)C)NC(=O)CC1CSC1)NC(C(=Cc1ccncc1)C)=O C1(NC(CC=C)=O)CCOCC1NC(C1CC(CC2CC2)C1)=O c1(SC(C2CCCC2CN(c2nnc(CCCC)s2)CCC#N)=O)ccccc1Cl N1(C(C(C#C)(C)C)=O)CC(CN(C(C2(C)CCNC(=O)C2)=O)C2CC2)CC(C)C1 Cc1ccc2c(c1)C(C(=O)NCCCNC(c1ncn3c1COCC3)=O)OCC2 c1(CC(=O)NCC2(OC)CCN(C(c3c(C)nc(C)o3)=O)C2)cnc(Cl)cc1C c1(CC(N2CC(O)(CNC(C(CC(N)=O)O)=O)C2)=O)cc2ccccc2nc1O C1(C(=O)NCCN(C(C(C=C)(F)F)=O)C)(COC)CCC(F)(F)CC1 C1(NC(C23C(CN(C(CCNC(C)=O)=O)C2)CC3)=O)CC2(CNC(=O)O2)C1 CC(C)CCCCCC(=O)N1C(C(=O)N(C)Cc2cn(C)nn2)CCC12CC2 Cc1cnccc1C(C)C(=O)NC(C)CC1CN(C(=O)C=Cc2cncs2)C1 c1(C(N2CC(C(C)NC(C3C(CC)C3)=O)C2)=O)ccc(C2CC2)nn1 C12(CNC(c3c(C)nn[nH]3)=O)CC1CN(C(C1CCC(=C3CCC3)CC1)=O)C2 CC1CCN(C(C2CC(C)(C)CO2)=O)CCN1C(C12CCCN(CC1)C2)=O N1(C(C(C)(F)F)=O)C2CCC1CN(C(=O)Cc1cc(Br)ccc1O)CC2 c1(C(N2CC3CCN(C(C4CCCCS4)=O)CC3C2)=O)ccccc1C#CC1CC1 N1(C(C=CCCC=C(C)C)=O)CC2CCC2(CCNC(=O)C#CC(C)(C)O)C1 C(C(O)CNC(C1(F)CCC1)=O)NC(CN(C)C(c1ccoc1)=O)=O C1(CNC(C(C)n2cnnn2)=O)CN(C(C2OCCC2C(F)(F)F)=O)CCCO1 C(=O)(C1=NNC(=O)CC1)NCC1CC(NC(c2ccc(C)[nH]2)=O)C1 c1(C(=O)NC(C)CCNC(c2nnc(S)n2C)=O)cnn2cc[nH]c(=O)c12 C1(NC(C(CCOC)C)=O)CN(C(=O)CC2CC(C)(C)C2)CC12CC2 C1(NC(C2CC(OC3CC3)C2)=O)COC2CN(C(c3cc(F)cs3)=O)CC12 c1(OCC)cc(C(=O)N(CC(O)CN(C(=O)Cc2ccoc2C)C)C)ccn1 c1(C(=O)NC2C3CCN(C(C=C(C)Cl)=O)C32)cc2cc(F)cc(F)c2[nH]1 c1(C(=O)NCCC(C)NC(=O)CCc2ncccn2)cnnn1C1CC1 C1(NC(C(CC)COC)=O)CCC2CCN(C(=O)CC(Cl)Cl)C1C2 c1(C(c2ccccc2)N(C)C(=O)NCc2ccc(Cl)cc2)ccc(I)cc1 N1(C(C=CC(CC)C)=O)CCC(CCOC)(C(=O)NC2CCOC(=O)N2)CC1 C1(NC(c2nc(C)nc(O)c2)=O)CN(C(=O)CN2CSCC2=O)C2CCCC12 C1(O)(CNC(C(Cc2cnc[nH]2)NC(Cc2c(C)ocn2)=O)=O)CCN(C)C1 C1(C(N(C2CCN(C(c3c(C)nc(C)o3)=O)C2)C)=O)CS(=O)(=O)CC12CC2 N1(C(C(C)Sc2ccccn2)=O)CCC2CN(C(C3CCC3(F)F)=O)CC2C1 c1(C(N(C(c2cscn2)=O)CCF)=O)cccc(NC(C2CCC3CC23)=O)c1 c1(CCC)ccccc1NC(C1CCN(C(=O)C(c2cccn2C)=O)C1)=O c1(C(N2CC(NC(C(C)CN(C)C)=O)C(C)(C)C2)=O)ccc2c(c1)COCCN2 C1(C(=O)NCCCCn2cc(-c3cccc(C(=O)OC)n3)nn2)CC1C1CCCC1 c1(C(N(CC(CNC(c2cc(CCC)n(C)n2)=O)O)C)=O)cc(C)cc(C)n1 c1(C(C)(C)C)cc(N)ccc1C(=O)NC1CCCCC1NC(c1ccc(Cl)o1)=O c1(C(N(C(C)CNC(=O)C=Cc2ccccn2)C)=O)cc2cc(F)ccc2s1 C12(C(N3CCN(C(c4cocn4)=O)CC3)=O)CCCCC1CS(=O)(=O)C2 N1(C(C2(OCC)CC(F)(F)C2)=O)CCC(C(=O)NC2CC2C2CCC2)CC1 C1(N(C(=O)CCc2cncnc2)C)CCCCC1N(C(=O)CC1CCCO1)CCCO N1(C(CCSC)=O)CCCC(C)C1CNC(=O)C(C)NC(c1ccccn1)=O C=C(C)C1CN(C(=O)CC(CNC(=O)C(CCC)C(C)C)OC)CCO1 N1(C(CCN(CCC)C)=O)CCOC(C(C)NC(=O)CCc2cnn(C)n2)C1 c1(COc2ccc(C(C(=O)OCCC(c3cccs3)OC)C)cc2)ccccc1F CC(CCCCNC(C1(C)CC(F)C1)=O)NC(c1ccc(CC2CCC2)cc1)=O C1(NC(CCSCCC)=O)CCCN(C(=O)Cn2cc(C)cn2)CC1 CC1=CCC(C)(C(N2CC(O)(CNC(c3ccnc(C(=O)OC)c3)=O)C2)=O)CC1 c1cc([N+](=O)[O-])cc2c1OC(F)(F)O2.c1(C(N)=O)n[nH]cc1S(=O)(=O)N N1(C(C(CCC)OC)=O)CCC2(CC1)CCN(CCOc1cccc(C)c1)CC2 N1(C(C2(C)CCCO2)=O)CCOCC(C(=O)NC2CCCC2CF)C1 C1(C2CCCOC2)(NC(C2C3(CC(NC(C4CN(CC(F)F)C4)=O)C3)C2)=O)CC1 Cc1nc(C2CCCC2)sc1C(=O)NCC(C)N(C(=O)C(C)OCCC(C)C)C N1(C(C2N(C(Cc3c(C)con3)=O)CC=CC2)=O)CC2C(=O)NC(=O)C2C1 c1(C(=O)NCCCCC(C)NC(=O)C(F)=C2CCCC2)cc(Cl)c(F)cc1N C(=O)(C1c2c[nH]nc2CN1C(=O)CC1CCC(=O)C1)NC1CN(C)CC1(C)C N1(C(C2CCC(C)CC2)=O)CC2CCC1C(C(=O)Nc1csc(=N)[nH]1)C2 Cn1nc2c(c1C(=O)NC1CN(C(C3CCS3(=O)=O)=O)C1)CSCC2 N1(CC(=O)NC(C(C)C)CNC(=O)CCc2ccon2)C(C)CCCC1C Cc1nn(C)cc1C(=O)NCC1(C(=O)NCCN2CC(OC)CC2)CC12CCC2 c1(NCCNC(CN(C(=O)C(n2nccc2C)C)CC)=O)cc(OC)cc(Br)c1 C(C(=O)NCC1CC(CNC(c2cnsn2)=O)C1)(C(C)C)SC N1(C(COC)=O)CCC(C(N2CCOCC2c2cn(CC3CCCO3)nn2)=O)CC1 c1(Nc2cc(CS)ncn2)ccc2cnnn2c1.C(CC(C)C(C)C)NC(C)=O c1(OC(C2CCCC2)CC)csc(C(=O)NCC2CC(C(=O)NC)C2)c1 CCCC(CCCNC(=O)C=CC1CCOC1)NC(c1cc2sccc2[nH]1)=O C1(F)(C(=O)NCCCC2(C)CN(C(c3cccc(C(F)F)c3)=O)C2)CCOCC1 c1(C(N(CCNC(C(C)=CC)=O)CCOC)=O)ccccc1OCC(N)=O c12cccc(c1)NC(=O)CCN(C)Cc1cn-2nn1.C1(CCO)(CO)COC1 Cc1cc(C(N2CCC(CC(C)NC(c3ccoc3)=O)CC2)=O)c[nH]c1=N N1(C(c2c(C)cc(O)cc2)=O)CCC2(CC1)CN(C(c1c(Br)cncc1Br)=O)C2 N1(C(c2nc(Br)cs2)C(=O)Nc2c(OC)cccc2)CCCC(C2CNC(=O)C2)C1 N12CCN(CC1)C2.N1(C(COCCCOC)=O)CC(CC=O)C1.C1(CO)CC1 C1(C)(NC(c2c(C)noc2CO)=O)CCCN(C(c2cnc(C3CC3)nc2)=O)C1 N1(C(C2CCC(CC)O2)=O)C(C)CC2CN(C(c3cncc(NC)c3)=O)CC12 c1(NC(C(n2ncc(C)c2)C)=O)cccc(NC(=O)NC2CCC=CCC2)c1 C1(C(=O)NCc2c(CC)cccc2)CCN(C)C12CCCN(C(C1(C)CC1)=O)C2 C1(CNC(C(C)SCC)=O)CCC2(CCN(C(c3cn(C)nc3O)=O)CC2)CO1 C1(C(=O)O)CC(C(N2CCC(n3cccn3)C2)=O)CC(C(F)(F)F)C1 c1(CCC(=O)NCC(C(C)C)NC(c2nnc(C)s2)=O)n[nH]c2ccccc12 CCC(C)(C(=O)OCc1conc1C)NC(=O)NCc1ccc(F)cc1 C1(CNC(COCCC(C)C)=O)CCC12CN(C(=O)C#CC(C)C)C2 N1(C(CN(C(C2CCCN2CC)=O)CC)=O)CCC(O)C(C)C1 C12(C(=O)NC(CC3CN(C(C4C(C)CCC4)=O)C3)C)CC3CC1C2C3O c1(OC)cc(N)c(Cl)cc1C(N1CCC(COCCC(=O)NC2CCOC2)C1)=O Cc1ccsc1-c1cn(C(C)C(=O)NCC(Cc2ccoc2)CO)nn1 CC1CCN(C(C2CC(=O)N(C)C2)=O)C(C(=O)NCCC2CC(C)(C)C2)C1 c1(CCNC(C2C(C(N(CC(F)(F)F)CC)=O)C2)=O)cc(F)c(Cl)cc1Cl CC1C(F)(F)CCN1C(=O)NC1CCC1C(F)(F)F N1(C(C2C(COC)C2)=O)CC(NC(c2nc3cnccc3s2)=O)CC12CCCC2 c1(C(N2CC(C)C(NC(=O)CC3C=CCCC3)C2)=O)cc(N)cc([N+](=O)[O-])c1 C(=O)(C(C(C)C)N1CCN(c2sc(=O)n(C)c2Cl)CC1)NCC=C C1(C(N2C(CN(C(CCCNC(C)=O)=O)C)CCC2)=O)CCN(C2CC2)C1=O c1(C(N2CCC(N(C(C3C(CCC)C3)=O)CC)C2)=O)ncncc1Cl N1(C(COC(C)C)=O)Cc2ccc(NC(c3cccc(Br)c3[N+](=O)[O-])=O)cc2C1 N1(C(C2CC(SC)C2)=O)CC2CC(NC(=O)CCCCN3CCOCC3)CC2C1 CCC(F)(F)C(C)(C)NC(C1COC(CNC(C2CC(C)C2)=O)C1)=O c1(OC)cc(C(=O)NCc2ncoc2CCNC(=O)Cc2n[nH]c(=N)s2)ccn1 c1(C(N(C(C)CNC(=O)Cc2csc(S)n2)C)=O)ccc(F)c(CO)c1 C(CCCOC)(C(=O)NCC(O)CNC(N)=O)NC(C(CC)COC)=O c1(C(=O)NCC(CN(C(Cc2c(C)nc(C)s2)=O)C)O)noc2ccc(Cl)cc12 C1(C(=O)NCc2c(C(N3C(C(C)C)CCCC3)=O)con2)CC(C)(C)CN1C C1(CCC)CN(C(C23CSCC2C3)=O)CC1C(=O)NC(C)COCC C1(C(=O)NCCNC(C(C)(C)C2CC2C(F)(F)F)=O)CCS(=O)(=O)C12CCC2 c1(C(=O)NC2(CNC(CCc3c(C)ncs3)=O)CCCC2)cc(F)ccc1C#N n1(CC(N2CCCC(CNC(CS(CC)(=O)=O)=O)CC2)=O)ccc2ccccc12 N1(C(CCCC#CC)=O)CCCC2(NC(c3cnn(CC4CC4)c3)=O)CC2C1 C1(C(=O)NC(CCCC)C)CN(C(=O)CC(O)C(C)C)CCC1(C)C c1(SC(C)C(=O)N(C2CCNCC2)C)ccc(Cl)cc1 C(=O)(C(CO)C(F)(F)F)NC(CN(C(Cc1cncc(C)c1)=O)C)C c1(C(=O)NC2C(CNC(c3cn(CCOC)nc3)=O)CCC2)cccc(O)n1 c1(C(N)=O)cc(C(N2CCC(OCC(=O)NC3CC=CC3)C2)=O)n[nH]1 C1(NC(C2(CC)CCC2)=O)CC(C(N2CC(CCO)C2)=O)C12CCC2 Cc1cc(NC(c2n[nH]c3c2CN(C(=O)CNC(C)C)C3)=O)cn2c(C)nnc12 C1(C)(C(N(CCCNC(C(C2CCN(C)C2)(C)C)=O)C)=O)CCC2CC2C1 C1(C(=O)N(c2ccc(F)c(Cl)c2)CC(F)(F)F)CC2(CCCCO2)C1 C1(N(C)C)CC2CC1N(C(=O)Nc1c(C)n(-c3ccc(C(F)(F)F)cc3)nc1)C2 CCC(CCOC)C(=O)NCC(F)(F)Cn1cc(C(n2cncn2)C2CC2)nn1 c1(C(N2C(C3(NC(C=C(COC)C)=O)CC3)CCC2)=O)cccnc1C(N)=O N1(C(c2[nH]c(=N)sc2)=O)CC2CC(NC(=O)C3=CS(=O)(=O)CCC3)CC(C2)C1 N1(C(C2CCN(C(=O)OCC)CC2)=O)CCC12CCN(C(c1ccoc1)=O)CC2 C(=O)(CCCC(=O)n1sccc1=O)N1CC2(N(C(CNC(CC)=O)=O)CC2)C1 Cc1ccc(C(=O)NC(C2CCCN2C(c2nc(Cl)oc2C)=O)(C)C)nc1C CCCCC(CC(=O)NC1CCC(=O)N(C)C1)NC(C1(CC(=O)OC)CC1)=O N1(C(C(COCC)C)=O)CCCC(O)(CNC(=O)C(C)(C)CC2CC2)CC1 N1(C(C(CC)(O)c2ccccc2)=O)CC2CC(NC(=O)C(C)C3CCC3)CC2C1 C(C1(CO)CCc2ccccc21)Nc1nc(CCC)sn1 c1(OC)ccc(C(=O)NCC2CC2NC(=O)C(=Cc2c[nH]cn2)F)cc1Cl c1(C(=O)NC2CC(OCC(N3CCCC3)=O)C2)ccc(CO)c(F)c1 N1(C(CC(C)CC2CC2)=O)CC(NC(c2ccc(N(C)C)nc2)=O)C(C)(C)C1 c1(C(=O)NC(CC)C(F)(F)F)ccc(NC(c2occc2C)=O)c(C)c1 N1(C(c2ccc(COC)cc2)=O)CCC(CO)(CN(C)C)CC1.c1cccnc1 CCCCCCCCCCC(=O)NC1CCCC(N(C(=O)COC)C)C1 Cc1cc(Cl)cc(C(=O)NC(CO)C(C)NC(=O)C=Cc2cccnn2)c1O c1(C(N2CC3C(CNC(C4C(C)(C)NC(=O)C4)=O)(C3)C2)=O)cnc2cccnn12 N1(C(c2ccc(CC)c(C)c2)C(=O)NCCCF)CC(C(N)=O)CC(O)(CC)C1 N1(C(C(C2CCN(C(C34CC(F)(C3)C4)=O)CC2)C)=O)CCCN2CCCC2C1 N1(C(C=C(C)C)=O)CCC(NC(=O)C=Cc2cnccc2C)C(CO)CC1 N1(C(c2ccc(CC)cc2)=O)CCC2(CC1)CC2(C)C(=O)N(C)CCOC(F)F C1(NC(C(CCOC)C)=O)CCCCN(C(=O)CC(c2ccc(F)cc2F)C)C1 C1(C(=O)NCCC(C)NC(c2cn(C)nc2Br)=O)CCCC2CCCCC12 c1(C(=O)NC(C)C(C)NC(=O)COC2(C)CCC2)cn(CC(F)(F)F)nn1 N1(C(CC2(C=C)CN(C(=O)CCCCOC)C2)=O)CCC(O)CC1CC CC(C)(C)CC(C)(C)C(=O)NC1CCCC(NC(C23CCC(CC2)OC3)=O)CC1 Cc1nnc(CN(CC(=O)NC2CCC3CC23)C)n1C.C12CCCN1C2=O c1(Cn2cc(-c3occ(F)c3)nn2)noc2c1COCC2 c1(OCCNC(C(c2cccs2)NC(c2cnc(CC)s2)=O)=O)cccc(F)c1 c1(NC(C(C)(C)NC(=O)NC)=O)cncc(CNC(=O)CCN2CCCC2)n1 CCC(C)CC(C(=O)NCc1nc[nH]n1)NC(=O)C(O)CC(C)(C)C c1(C(C)=O)ccc(S(=O)(=O)N(CCC(c2ccccc2C)C)C(C)C)cc1 N1(C(C(N2CCCC(C(F)F)CC2)=O)=O)CCOc2cc(Cl)ncc2C1 C1(S(N)(=O)=O)(C(=O)NCC(CNC(c2c(SC)scc2)=O)F)CC1 Cc1ccc(F)c(C(=O)NC2CCCC2CNC(c2nc(C)c(C)[nH]2)=O)c1 CCC(C)C(C(=O)NC1(C(=O)NC(C)C(C)(C)C#N)CCOCC1)OC N1(C(CCCn2cc(C(C)O)nn2)=O)CCCC2(C1)C(O)CC2O N(C1CN(C(=O)CC(C)CF)CCc2ccccc21)C(C1N(C(C)=O)CCC1)=O C#CCCCCCC(=O)NC1CCN(C(c2cn(C)nc2C)=O)C(C2CC2)C1 c1(C(=O)OC)cccc(C(=O)NC2CCCC2NC(=O)CSc2ccccn2)n1 CC1CCN(C(C2(CO)CC(F)(F)C2)=O)CC1NC(=O)COCc1nccs1 C1(C(=O)NCc2c(C(=O)NCCC(CC)CC)nco2)CCC2CC1CO2 c1(N(C(=O)COCCOC2CC(NC(C3CCCOC3)=O)C2)CC)ccccc1C c1(C(=O)NC2CCN(C(C3(CC4CC4)COC3)=O)C2)ncccc1Cl C(=O)(CCC1CCc2ccccc21)NC(C)CCNC(C1CCC(=O)N(C)C1)=O C(=O)(CC(C)(C)C(C)=O)N1CCC(=CCNC(c2c(CC)[nH]cc2)=O)CC1 Cc1nn(CCCl)c(Cl)c1C(c1nnnn1CC1CC1)NC(C1CCOCC1)C C(=O)(C(CO)C(F)(F)F)NC1CC(OC(CC)(C)COc2ccccc2)CCO1 C(=O)(C(CCOCCO)NC(c1nccnc1N)=O)NC(C(=O)OCC)C C=CC(F)(F)C(=O)N(CCCCN(C(=O)C(C)(C)OCCN(C)C)C)C C1(CNC(c2n(CC)nnc2)=O)CCCCN(C(=O)CN2CSCC2=O)C1 CC(C)CC(C(=O)N(CCCS(C)=O)CC(C)(C)C)ONC(=O)C1CCCC1 c1(CC)nccnc1C(=O)NCC(C)(C)CC1CN(C(C2CCCC2O)=O)C1 N1(C(C(C2CC2)OC)=O)CCCC12CCN(C(C1(C)CS(=O)(=O)C1)=O)C2 c1(COC)ccc(-c2cn(C3CCC(C(=O)NC4CC(C)(O)C4)CC3)nn2)cc1 C(=O)(C(C(=O)NOC(CC(C)C)C(=O)NC1CCC1)OC)OC Cc1nc2c([nH]1)CC(C(N1CCC3(CCC3NC(=O)CC(C)(C)O)CC1)=O)CC2 Cc1cc(-n2cc(CCNC(=O)Nc3cccc(OC(F)F)c3)nn2)ccc1F C(=O)(C1=COCCC1)NC(C(CO)NC(c1ccc(-n2ccc(C)n2)cc1)=O)C C1(CNC(C(COC)OC)=O)CN(C(c2ccc3c(c2)CC3)=O)CC12CC2 c1(NC(N2C(c3cccc(OC)c3)C(C)(C)C2)=O)ccc(F)c2[nH]ncc12 C1(NC(CC)=O)CCC(N(C(=O)C=Cc2cccs2)C)CC1 CN1CCCC(CC(C(=O)O)NC(=O)C(O)CC2CCOCC2)C1.C12CN(C1)C2 N1(C(=O)CC2CCCO2)CCc2sc(-c3cnn(C4CCOC4)c3)nc2C1 N1(C(C=C(C)Cl)=O)CC(CNc2nccc(N3CCCC3)n2)CC1(C)C c1(OC)ccc(CC(=O)NC(C)C(C(C)C)NC(=O)Cn2cnc(=N)[nH]2)nc1 C(=O)(CCP(C)(C)=O)N1CCC(C(C)C)(C(=O)N(C)CCC2CCOCC2)C1 C1(NC2CCCCC2)CCCN(C(C2(NC(C(C)(C)C3CCCO3)=O)CC2)=O)C1 c1(NS(c2occ(C(=O)O)c2)(=O)=O)ncc2c(n1)CCCCC2 c1(C(C(=O)NC(CNC(=O)C=CC=C(Cl)Cl)CO)=O)ccc(F)c(F)c1 C(N=c1[nH]c(N2C3CCC2CC(=O)NC3)nc2c1SCC2)c1c(C)cncc1 CC(C)C(O)CCN=c1cc[nH]cc1S(=O)(=O)N(C1CCC(C)(C)C1)C CC1(C)CCN(C(=O)C(O)Cn2cncn2)C(C(=O)NC(C(O)CO)C2CC2)C1 C1(C(=O)NCCN(C(C)C)C(c2ccc(OC3CC3)s2)=O)CCCC(F)C1 C(C)(CCCCNC(c1cnn(CCOC)c1)=O)NC(c1c(OC)scc1)=O C12(NC(c3ccc(OC)s3)=O)CC(C1)N(C(c1cc(C3CC3)no1)=O)C2 C1(COC)(NC(c2nsnc2O)=O)CCN(C(c2c[nH]c(=N)cc2C)=O)CC1 c1(N2CC(n3c(=O)ccnc3)C2)nc(=NCCCCc2ncc[nH]2)[nH]c2c1CCC2 Cc1cccc(CCC(=O)NC2CCC2NC(c2cccc(N(C)C)n2)=O)c1 O=[N+]([O-])c1ccc(Br)cc1CNC(C1(CNC)CC1)=O.C12CC(F)CN1C(=O)OC2 c1(C(=O)NCC2N(C(C(C)O)=O)CC2)cc(S(C)(=O)=O)cnc1O C=CCCCCCC(=O)NCCC1CCN(C(c2cnoc2CC)=O)C1 C(=O)(CCCC(C)(C)NC(c1cscc1Cl)=O)NC(CCC)C C1(C(=O)NC2CN(C(C34OCC(C)(C3)C4)=O)C2)CC(c2cccc(Cl)c2F)=NO1 N1(C(c2c(C)cc(C)o2)=O)CCN(C(=O)C(O)C2CC2)CC1c1cccc(F)c1 Cc1cc(Cl)c(C(N2CC(CNC(=O)C=C3CCC3)C2)=O)cc1[N+](=O)[O-] N1(C(=O)OC(C)(C)C)CC(C(=O)Oc2cccc(Cl)c2I)CCCC1C CCCC(C)(C)C(=O)NCC1CCCN1C(=O)CCC1CC(F)(F)C1 CC(C)(C#CC(=O)NCC1CC(O)C(O)C1)CNC(c1ccc(Cl)s1)=O C1(C(=O)NCCCOC)CN(C(c2ccn(C)c2)=O)C2(CCC2)C1 C=CCC(CC=C)C(=O)N1CC(O)(CNC(c2c[nH]cc2-c2cnn(C)c2)=O)C1 c1(C(=O)NCCCN(C(C(CC)C)=O)CCO)cc(C)n(C(C)(C)C)n1 N1(C(CSc2ccc(C)cc2)=O)CCOCC(CNC(c2cn[nH]c2)=O)C1 c1(OC)cc(Br)c(Cl)cc1NC(=O)N(Cc1ccc(F)cc1)Cc1ccccc1 c1(OC)cccc(O)c1C(N1CCC(CNC(C2CCC(=O)N2C)=O)C1)=O C=C=CC(C)C(=O)NCCCCC1CCN(C(=O)C=CC)CC1 C=CCC(CC(=O)NC(C)CC(N)=O)NC(c1cccc(F)c1F)=O C(=O)(C(CO)NC(N)=O)NC(C(=O)NCCC(=O)NCCOC)C1(C)CC1 c1(C(N2C3(CNC(C(C)OCC)=O)CC(C2)C3)=O)cccc(C)c1C(F)(F)F C1(C(=O)OCCOCC(=O)OCC)(COC)CCCCC1 C=CC(CCC)CC(=O)NC(C)(CNC(C1(Cl)CC1(F)F)=O)CO C1(C(=O)NC2C(NC(c3n[nH]c(CC)c3Cl)=O)CCCC2)CCc2ccccc2N1 C(=O)(CC(O)CNC(c1n[nH]cc1C1CC1)=O)NC1C(OC)C(O)C1 C1(C)(NC)CC(OC)CN1C.CCCCCN1C(=O)NCC1 N1(C(c2scc(OC)c2)=O)C(C)CN(C(c2nn(C)c3c2CCC3)=O)CC1C C1(CC(=O)NCC(CC)NC(c2cnc(C)s2)=O)Cc2cc(F)ccc2O1 CCC(CC)CC(=O)NCC1CC(NC(c2cnn(CCO)c2N)=O)C1 C(=O)(CCCC(=O)N(C)C)NCC(Cn1nccc1C)OC C1(CC(=O)NC(CC(C)NC(c2cnc(C(C)C)[nH]2)=O)C)CCN(C)CC1 CCCCCCC(C)C(=O)N1CC2CC2(NC(c2cc(C)cnc2C(F)F)=O)C1 c1(C(=O)NC2CC(NC(C(CCC)CC(C)C)=O)C2)cccc2cccc(OC)c12 c1(CC)cc(C(=O)N(C)CCN(C(=O)C(CO)N(C)C)C(C)C)cc(Cl)c1 c1(OC)cc(C(=O)N(C)CC2CCCN2C(=O)C(F)=CC2CC2)c(Cl)nc1Cl C1(NC(C(F)OC)=O)CN(C(C2CCCN(C(=O)C3CC3)C2)=O)CCC1C c1(C(N(CCNC(C2CNC(=O)N2CC)=O)CC)=O)cccc2cnsc12 N1(C(C2(C=C)CCC2)=O)CC(C2CN(C(=O)Cc3c[nH]nc3O)C2)C1 CC(CCCCN(C)C)OC.C(=O)(CCCc1ccccn1)NCC=O CCCCCS(=O)(=O)CC(=O)NCCC(CNC(c1c[nH]c(=NC)s1)=O)OC c1(C(=O)NCC(CC)NC(=O)C(CC)CCOC)cc2c(cc1N)CCC2 C=CCCCCC(=O)NC12CCN(C(c3cc(Cl)ccc3Br)=O)CC1C2 N1(C(c2c(CC)cno2)=O)CCN(C2CCC(NC(=O)CC3CC=CC3)C2)CC1 C(=O)(C#CC1CCCCO1)NCCN(C)C(C1(C)C(C)(C)C1(C)C)=O C1(CCNC(=O)NCC(COC)OC)CCCC1C Cc1ccnnc1C(=O)NCC1COC(CNC(=O)CC2CC3(CC3)C2)C1 CC(C)(O)C(F)CNC(C1C=CCN(C(C2CN(C(C)C)C2)=O)C1)=O C1(N(C(C(F)OC)=O)CC2CC2)CCN(C(c2scnc2C)=O)CC1 C1(C(=O)NC(CC)CO)CCN(C(=O)Cc2ccc(CO)cc2)O1 c1(CNC(=O)NC2CCN(C3CC3)C2=O)cccc(N2CCOCC2)c1 c1(C(=O)NC2CN(C(C3(CCC)CC3)=O)CC23CCC3)cc([N+](=O)[O-])ccc1N c1(C(=O)NC2CC3CN(C(COCC(=O)N(C)C)=O)CC32)cccc2[nH]ccc12 Cc1ccc2cc(C(=O)NC3CC(C)CN(C(C45CC4C5)=O)C3)ccc2c1 N1(C(C2(CC)COC2)=O)CCC(C)(CNC(=O)C(C)Oc2ccc(Cl)cc2)C1 c1(CC)nc(C)c(C(=O)NCC(C)C(C)(C)C)o1.C12(O)CC(C1)C(=O)NC2 c1(C(N(C(C)CNC(=O)CCCCC#N)CC)=O)cnc2[nH]nnc2c1 C1CCCCCNC(=O)C(C)O1.C1(NC(=O)CNS(C)(=O)=O)CCOCC1 C1(NC(CN(C)CCO)=O)CN(C(C2CCCN2C2COC2)=O)C(C)(C)C1 C1(C(N(CC(=O)NC2(CCC)CCNC2=O)CC)=O)CC2CCCC2C1 CC(CCCCNC(=O)C(C1(C)CC1(Cl)Cl)C)NC(=O)Cc1cnoc1 CCC(C(F)F)NC(=O)C(c1cccs1)NC(=O)OC(C)(C)C c1(NC(C2C=CC(NCc3ncn(C)n3)C2)=O)cc(Cl)cc(Br)c1 c1(NC(c2ccc(F)cc2F)C)nc2ccccc2nc1NC1CC=CC1 C1(CNC(c2cc(CC)on2)=O)CCN(C(c2ncc(Cl)cc2O)=O)CC1(F)F c1(OCC)c(C=CC(=O)N(C2CN(C(=O)CN(C)C3CC3)CC2F)C)ccnc1O N1(C(C2(O)CCN(Cc3c[nH]nc3Cl)CC2)=O)CCN2C(=O)OCC2C1 c1(CNC(C(C(COC)C)C)=O)cnn2c1CN(C(c1ocnc1C(F)F)=O)CC2 C(=O)(C#CC1CCC(=O)CC1)N1CCC(OC2CCCN(C(=O)COCCF)C2)C1 n1(COC)ncc(C(=O)NCC(CO)NC(=O)COCCCF)c1C C1(NC(C2(C)CCCN2C(=O)CC2(O)CCOCC2)=O)CCCCC1(F)F Cc1nccc(C(=O)NCCCCCCN(C(=O)C(F)=C2CCC2)C)c1C c1(NC(C)(C)C)ccc(CCNC(CO)C(O)c2cccs2)cc1 C1(NC(C2C(C(C)(C)C)C2)=O)CC2CCC1CN2C(C1CC2C=CC1CCC2)=O N1(C(C(CC=C)NC(C)=O)=O)CC2CN(C(c3cc(Cl)cs3)=O)CCC12 CC1(C)CN(C(=O)CCN(C(=O)CCC2CCCC2)CCCO)C12CCC2 C1(CN(C)C(C2CC2c2ccsc2)=O)CCCCN1C(=O)CCCOC(C)(C)C CC(C)C(C(=O)NCCCC1CC1C)NC(C1CCN(C)C1=O)=O c1(C(=O)NCC2(CCC)CN(C(C3CC3OCC)=O)C2)cccc(C(N)=O)n1 c1(C(C)(C)OCC)cccnc1C(=O)N(C)CCc1ccncc1 C1(NC(CC(C)C2CC2)=O)CN(C(C2CCN2C(C)(C)C)=O)CC12CCOCC2 Cn1c(O)nc2c(C(=O)NCCCNC(=O)Cc3cncn3C3CC3)cccc12 Cc1ccccc1C#CCOC(C12CCC(CF)(C1)OC2)=O N1(C(c2ccc(Cl)c(Cl)c2)C(=O)NC2CCCC2)CCN2CCOCC2C1 c1(OC)cc(CNC(=O)NCCNc2snnc2C)cc(F)c1 C1(NC(c2c(SC)csc2)=O)CCCN(C(=O)CN2CCC(NC(C)=O)CC2)C1 c1(C(=O)OCC)c[nH]ccc1=NCC1CCN(C(=O)C(c2cnn(C)c2)O)CC1 C12(C(N3CC(OC)(CNC(c4cncc(N)n4)=O)C3)=O)CCOC1CC(=O)NC2 CCC(CC)(C(=O)N1CCC(C(C)NC(c2cc(C3CC3)ncn2)=O)C1)OC C(=O)(C(O)CC(C)C)NCCC(=C)CNC(c1cccn(C)c1=O)=O C=C(C)CC1C(=O)N1.C1(=O)C(C(C)O)NCC(C)C(=O)N1.C(C)(=O)OC C1(C(N2CC(F)(CNC(c3cc4cccnc4s3)=O)C2)=O)Cc2ccccc2S1 N1(CC(=O)N(CC(C)NC(c2nccc(C(F)(F)F)n2)=O)C)CCCCCC1 C(CC(C)(C)C(=O)NC1CC(F)(F)C1(C)C)NC(C=CC=CCC)=O O=C1NC(C(=O)NC2CCC2CNC(c2ocnc2C2CC2)=O)CO1 C1(CNC(C(C)(C)NC(=O)C2CC2)=O)CC2COCC2N1C(C1CCOCC1)=O N1(C(CCC(=O)OC)=O)CCC(CNC(=O)CN2CCCC2CO)C(F)(F)C1 CCCC(C)CC(=O)NCC1C=CC(NC(=O)CC=CC(C)(C)C)C1 N1(C(C(CCC)OCC)=O)CCC(C)(C)C(NC(=O)CC(C)(C)O)C1 c1(C(N2C(C)(C(=O)Nc3ncc(Cl)cc3Br)CC2)=O)cc2ccccn2n1 c1(CC)[nH]nc(C(N2CCN(C3CN(C(C4CC4C(F)(F)F)=O)C3)CC2)=O)c1C c1(N(CC(F)F)C)nc(N2CCC3(C)C(C2)C3(Cl)Cl)nc2c1CCC2 CCC(CCCCC(=O)NCCC)N=c1cc[nH]c(=NCCCCOC)[nH]1 c1(OC)cc(C(=O)NC2CCN(C(=O)CN3C(=O)CCC3=O)C2)ccc1Br c1(C(N(C(C)CCNC(=O)CN(C)C2CC2)C)=O)ccc(O)c(Br)c1 C1(CNC(C2C(C)=C2)=O)COCCN(C(=O)COc2cc(C(C)C)on2)C1 N1(C(COC)OC)CCN(C(=O)CCCCc2cc(OC)cc(OC)c2)C(C)C1 CC1CN2CCC1NC2=O.C1(C)(C(=O)Oc2ccc(C#N)s2)CC2CCC1C2 CCC(O)C(F)(F)C(=O)N1CCOC(CNC(=O)CCCc2cnn[nH]2)C1 CC1OC2(CNC(=O)C(C)(C)C(N)=O)CC1(NC(C1CCCCS1)=O)C2 C1(C(N(C)C)=O)CCCCN1C(=O)N(C)CCN(C)C.C12(CC1)C(=O)O2 C1(O)(CC=C)CCN(C(C2CSCCN2C(=O)C(C)O)=O)CC1 C1(CC(N2CC(CN(C(CCOCCC)=O)C)C2)=O)CCC(=O)NC1=O C1(C(N(CCNC(CC(C)SC)=O)C)=O)CCS(=O)(=O)C1(C)C O=C(C1=CCc2ccccc21)NC1CCCC1NC(c1ccc(C(F)F)s1)=O c1(N(CCCNCC2CCCN(C3CC3)C2)C)nc2ccccn2n1 C1(NC(c2csc3cncn23)=O)CCCC(N=c2[nH]nc(C(F)(F)F)o2)C1 C1(C(=O)NCCC(C)F)CC12CC(NC(C1(C)CCC1)=O)C2 c1(C(=O)NCC2OCCN(C(CC(=O)NCC#C)=O)C2)cn2cc(C)nc2s1 C1(NC(CN2CC(=O)NCC2)=O)CN(C(c2ccc(Cl)s2)=O)C2CCCCC12 C1(NC(c2cc(F)ccc2Br)=O)CC2CCC1N(c1ncc(O)cn1)C2 C=C1CC2(C1)CC(C(=O)NC13CCN(C(c4cc(CC)on4)=O)CC1C3)C2 CC(CC(=O)NC1(CNC(c2cc(C(F)(F)F)c[nH]2)=O)CC1)N(C)C C1(C#N)(C(=O)NCC(C)(C)NC(c2csc(-c3ncccn3)n2)=O)CC2(CCC2)C1 C(=O)(C(C)S(=O)(=O)C(C)C)N1CCC(C)(CNC(c2c(C)onc2Br)=O)CC1 C(=O)(C(C)(C)C1=CCN(C(=O)C(C2CCOCC2)C)C1)NCc1nc(C)c(C)o1 N1(C(c2n(CC)nc(C(C)C)c2)=O)CCCC1C1CCCN1C(=O)CCC(N)=O c1(C(=O)NCC(CO)NC(C2CC(F)C(=O)N2)=O)cc(Cl)c(F)c(Cl)c1 C=C(Cl)CCC(=O)N1CC=CC(NC(c2ccc(CC(N)=O)cc2)=O)C1 c1(C(=O)NCC2CC(C)N(C(c3ccns3)=O)C2)coc2c1CSC2 N1(C(C)C)CC(NC(=O)C(C2CCOC2)NC(=O)COCC2CCC2)C(C)C1 c1(CSCCNC(C(N)CC2CC2)=O)cc(Br)cc(C(F)(F)F)c1F C(=O)(CC(C)CC(=O)NCCn1cc(NC(C23CCCN(CC2)C3)=O)cn1)OC C1(CC(=O)NCC(C)(C(C)C)OCC)CCC2(CC1)COC2 C(=O)(C1=CCCC1C)NCC(CN(C(CCCC=C)=O)CC)(C)C C1(NC(c2ccc(C)c(Cl)c2)=O)CC2(C1)CC2N=c1[nH]ccnc1F c1(SCC(=O)NCC(CN(C(=O)CN2CCCC2=O)C)(C)C)cc(Cl)ccc1Cl c1(CC(N2CC(C(C)NC(=O)C(C)(C)CF)OCC2)=O)c[nH]c2ccccc12 CCC(CC1CCC1)CC(=O)N1CC(C2CN(C(=O)CCC(F)F)CCO2)C1 c1(CC(C)C)cc(N2CCC(CCNC(=O)C(C)(C)C3CCCCC3)C2)ncn1 n1(Cc2ccc(C(=O)NCCSCc3ccccc3)o2)cc(C(C)(C)C#N)nn1 c1(C(N(CCCO)C)=O)c(C)noc1C(F)F.C(CC)(C(=O)NCCOCC)CC C=CCCC(C)(C)C(=O)N(C1CCCN(C(C2(O)COC2)=O)C1)CC1CCCO1 C1(NC(c2ccn3cnnc3c2)=O)COC2(CCN(C(=O)C3=C(Cl)CC3)CC2)C1 C1(C(N2CCN(C)CC2CNC(=O)C(C)(C)NS(C)(=O)=O)=O)CCCC1S(C)(=O)=O c1(CC(C)C)n[nH]c(=NCC2CC(CNC(=O)CC3CCCCCC3)CO2)s1 N1(C(C2(Cl)C(C)(C)C2)=O)CCC(C(F)(F)F)C(NC(c2cccs2)=O)C1 C(=O)(C(F)CC1CCCC1)N(CC(CC)NC(=O)C(C)(C)c1cncnc1)C CC1CCN(C(C2CC(C)(F)C2)=O)CC1NC(C1CCC2(CCC2)C1)=O c1(C(C)C(=O)NC(CNC(c2cnc(Br)s2)=O)CO)cccc(C#N)c1 CCC(C)(C)CCNC(=O)C(c1ccco1)NC(=O)C(CC)NC(C)=O N1(C(C(C)=CC)=O)CCC2CN(C(c3cc(OC)c(C)cc3N)=O)CC2C1 c1(N(CCCC)C(C2CCN(c3cccc(Br)c3)C2=O)=O)ccccc1CCC C(CN=c1[nH]c(=NCc2nccc3ccsc23)[nH]c2ccsc12)=CCCC C1(C(=O)NCCCCCn2cc(CN3CCCC3=O)nn2)CCC(F)(F)C1 c1(C(=O)NC(CNC(CC2(C)CCCO2)=O)CO)cccc2nonc12 c1(NC(C(=O)N(C2CN(C(C3C(CCC)C3)=O)C2)C)C(C)C)ccc(Cl)cc1 N1(C(c2c(CC)cccc2)=O)CCCC(CC(=O)N(CC)Cc2ccccc2)CC1 N1(C(c2cccc(C)c2)=O)CCC(NC(=O)Cc2cc(C(C)C)no2)C12CC2 C1(N(C(C(=Cc2ccco2)C)=O)C)CN(C(=O)CCCc2csc(=N)[nH]2)CC1F N1(CCC(=O)NC(CNC(CCCOC(C)=O)=O)C2CC2)CCC(O)CC1 C1(CC#C)(OC(C)C)CCN(C(=O)C(c2cccc(NC(=O)C=CC)c2)(F)F)C1 c1(C(N2C(CN(C(=O)CCc3ccc(OCF)cc3)C)CCC2)=O)cc(Br)n(C)c1 CC(Cc1cnn(C)c1)C(=O)NCC(F)CNC(=O)C=Cc1cnc[nH]1 C(Cc1ccco1)(C(=O)N1CCC1C1(O)CCCC1)NC(C(C1CC1)SC)=O C(C(=O)N1CCC(C(=O)NOCC2(C#N)CC2)O1)(OC)OC N1(C(c2c(C#C)c[nH]n2)=O)CC2CC1CC2NC(c1ccc(=O)n(C)c1)=O c1(C(N(CC(C)NC(c2c(F)cccc2F)=O)C)=O)ccnc2ncccc12 CC(C)(C)C(O)C(=O)N1CC(C)(C(=O)NCC=Cc2cccc(CO)c2)C1 N1(C(c2c(C)[nH]cc2)=O)CC2CCCC(C1)N2C(=O)C(c1ccn(C)n1)C C1(N(C(C(COC(C)=O)C)=O)C)CC(=O)N(CCn2cccnc2=O)C1 C12(C(N(C3CCN(C(=O)CN(c4nc(C)cs4)CC)C3)CC)=O)CCN(CC1)C2 C(=O)(C1=CS(=O)(=O)c2ccccc21)N1CCN(C(C(C)C)=O)C2C1CCC2 c1(OC)cnccc1C(=O)NCC(c1ccc(F)cc1)NC(=O)C(C)C(C)C N1(C(C=C(C)c2ccccc2)=O)CC2CCC1CC2NC(c1nscc1C)=O Cc1cnc(C(=O)NC2CCC(CCNC(c3cscc3C(F)(F)F)=O)C2)nc1 C(=O)(C=CS(C)=O)NC(C)C(CO)NC(c1cn(C)cn1)=O CC(C)CC(CNC(c1ccc(F)cn1)=O)C(=O)NC1CCOC12CCCC2 C(=O)(C#CC(C)(C)C)N1CCC(C(=O)NC(C2CCCCC2)C)(CC)C1 N1(C(c2cccc(C(=O)OC)c2)=O)CCC2C(CCN2C(c2cnc(C)[nH]2)=O)C1 C(C(C(=O)NCCC12CCCC1C2)C(C)C)NC(c1cn(CC=C)nn1)=O c1(C)csc([N+](=O)[O-])c1.N1(CCN2C(CC(=O)OCC)COCC2)CCC(C)(C)CC1 N1(C(CCC(C)SC)=O)CCCC(NC(c2cnccc2C)=O)C1C n1(CC)nc(C(N2CCC(CNC(=O)Cc3ccoc3C)CC2C)=O)ccc1=O N1(C(c2c(OC)c[nH]n2)=O)CC2(CCC2NC(=O)CC2CCCOC2)C1 C1(NC(c2ccc(C)c(CO)c2)=O)C(C)CN(C(=O)CC2(O)CCC2)CC1C C1(C(=O)NC2CC(NC(c3c(C#N)ccs3)=O)C2)CCC(=O)N2CCCC12 Cc1c[nH]c(C(N2CC(O)(C3CCN3C(C3CCSC3)=O)C2)=O)c1 C(=O)(C1c2ccccc2C2CC1C2)N1CCC(OCCNC(COCC(C)C)=O)C1 c1(C(=O)NCC2N(C(C(CC(C)C)OC)=O)CCC2)cc(F)cc(C)c1N C(=O)(C(C)C(O)C(C)C)N1CCC(N(C(=O)C(C)SCC)CCC)CC1 n1(CCOC)cc(C(=O)NC2CC(O)CN(C(c3cnsc3)=O)C2)c(=O)cc1C Cc1[nH]nc2c1CCC(C(=O)NC1CCCC1NC(=O)CSCCC#N)C2 c1(C(=O)NC2CC(NC(=O)CCc3nc[nH]n3)C2)cc(=O)c2ccc(Cl)cc2o1 N1(C(C2(CC)CC2)=O)CCC(F)C(NC(=O)CCc2sccc2C)C1 C(CNCC1CCNCC1C)(CC(=O)Nc1cc(OC2CCOCC2)ncn1)OC CC1CN(C(C2CC3OC2C2CC32)=O)CCC1NC(c1ccc(C(F)F)cc1)=O CCCCC(C)C(=O)NCC(C)(C)C(N1CCC2(CC1)N=N2)=O C1(C(=O)NC2C(C(=O)OC)CC2)CC(O)CN1C(=O)CC1CC2CCC1O2 C(=O)(C#CC1(C)CCCO1)NCC(CNC(c1cn(C)c(=O)cn1)=O)O Cc1cc(Cl)c(C(=O)NC2C=CCN(c3ncnc(Cl)c3C#N)C2)cc1C Cc1cc(C(=O)NC2C3CCN(C(=O)CCc4cn[nH]c4)C23)c(F)c(Br)c1 CCCCS(=O)(=O)CC(=O)NCC1CCCN1C(c1ccc(C#N)cc1OC)=O N1(C(c2cn(CCCC)nn2)=O)CC(CNC(C2CC2CF)=O)C(O)C1.C(=O)OC c1(CN(C(=O)CC2(NC(C3CC(CC)(CC)C3)=O)CCC2)CCC)ccccn1 N1(CC(N2CC(C)(NCc3cnc(C)s3)C2)=O)CCCC(O)C1 CC1(c2cn(-c3ccccc3)nn2)COCCN1C(c1csc(C#N)c1)=O N1(C(C(C)CN(C(=O)CC(C)N(C)C)C)=O)CCC2CCC(C1)N2C c1(OC)cnc(OC)c(C(N2CCC(NC(c3cnn(C(C)C)c3F)=O)C2)=O)c1 c1(C(N2C(CCNC(C(CC)N(C)C)=O)CC(OC)C2)=O)cnc(O)cc1C c1(C(N2CCC3(CC3)C2)=O)ccc(S(=O)(=O)NCc2ccccc2Cl)cc1 C(CCCC(=O)NCCC(C)N(C)C(C1(C#N)CC1(C)C)=O)OC c1(C(C)N(CCO)C(C2(C#N)CCCCC2)=O)ccc2ccccc2c1 c1(C(C(=O)OC)C)ccc(C)cc1.C12CN(C1)C(=O)N2CCC c1(CC)nc(N2CC(NC(=O)CCNS(C)(=O)=O)CC2C)cc(C)n1 N1(C(C2(OC)CCC2CO)=O)CC2CC1CN2C(c1ocnc1C(F)F)=O C1(C(=O)Nc2c(CC)cccc2)COC2(C1)CN(C(c1noc(C)n1)=O)C2 CCC(CC)C(C(=O)NC(CNC(c1ccc(C(C)C)cc1)=O)C1CC1)OC C1(NC(C(CC(C)C)C)=O)CCOC2(CCN(C(=O)COC(F)(F)F)CC2)C1 c1(NC(CCN(c2ccc(Cl)cc2Cl)C(C)C)=O)c(Br)ccc(Cl)c1F N1(C(CS(N)(=O)=O)=O)CC(C2CN(C(c3c(F)ccc(O)c3O)=O)C2)C1 CCC(CNC(c1cn(CC2CCCO2)nn1)=O)(CC)NC(C1CCNC1=O)=O Cc1cccc(Cl)c1OCC(N1CC2(CCC2CNC(=O)CCN2CCC2)C1)=O C(=O)(CC(CC)CC)N1CC(NC(C2(CCOCC)CCCC2)=O)C(F)C1 N1(C(c2n(C)c(O)nc2)=O)CCCC2(NC(=O)CC(O)C3CCCC3)CC2C1 N1(C(C(C=C)OC)=O)CC(NC(c2ccc(F)c(F)c2)=O)C(C)(C)C1 Cc1c(C(N2CCC(NC(=O)CC(=O)N(C)C)C(C)C2)=O)c(C)n2ccncc12 N1(C(C2(C)C=CCC2)=O)CC(NC(=O)C(c2ncccc2Br)(F)F)C(O)C1 c1(C(=O)NCC2N(C)CCN(C(C(CC#C)(C)C)=O)C2)cnnc2ccccc12 c1(C(=O)NCC(CC)NC(=O)CC2NC(=O)NC2=O)ccccc1NC(N)=O C1(NC(=O)CC2CC3(CC3)C2)CC1C1CCCN(C(=O)CCC2CCOC2)C1 C1(C(=O)NC(CNC(=O)NC)=O)CCCC(N=c2[nH]c3c(F)cc(Cl)cc3s2)C1 C(CCC(C)CC(=O)N1CC2CC2(NC(=O)C(CN(C)C)C(C)C)C1)=C(C)C c1(C(=O)NCC(=O)N(CCC)C)ccc2c(c1)COB2O.CC1CC1C(=O)NC N1(C(C(COC)C)=O)CCC2(CCN(C(c3ccc(CNC(C)=O)s3)=O)C2)C1 N#Cc1ccc(C(N2CCCCC2CCNC(C23CCCC2C3)=O)=O)c(O)c1 N1(C(C(n2cnc(C#N)n2)C)=O)CC2CC1CN(C(C1CCCC(CF)C1)=O)C2 N1(C(C(CCC)O)=O)CCC2C(CCN2C(c2coc(CO)c2)=O)C1 C(C(C)C(C)(C)C)NC(CC1(NC(c2nc(C)oc2)=O)CCC1)=O N1(NC(=O)CC)CC(OC)C2(CC2)C1.C=C1CC2(C1)C(=O)NCC(=O)NC2 C(C(=O)N1CC(CNC(=O)C(CC)CC)C(C)C1)(C(C)C)OCCOCC C1(NC(c2cccc(CCCCO)c2)=O)CCCN(C(=O)C(F)(F)C2CC2)C1 C1(C)(CCC(=O)NCCCN(C(=O)C(Cl)=CCl)CCOC)CCC(=O)N1.CC N1(CC=C)CCCC(C(=O)N(CCC(C(C)C)Nc2ccnc(Cl)n2)C)C1 N1(C(C(n2ncc(C)c2)C)=O)CCCCC(C(C)C(=O)NOC2CCC(O)C2O)C1 CCC(C)(C(=O)NCCNC(=O)CC1CC(C)(C)C1)OC c1(C(N(CCCCNC(=O)CC(C)(C)C)C)=O)cc(S(N)(=O)=O)c[nH]1 C12CCC(CC1)COC1CN(C1)C2=O.C1(O)(C(CCCCC)=O)CC1(C)C Cc1nnc2n1CCCC2NS(=O)(=O)c1cccnc1NC1C2CCCCC1CC2 C=C1CCN(C(C2CCOC2(C)C)=O)C(C(=O)NCC(C)C(C)(C)C)C1 C1(CNC(C(CC)O)=O)CC2CCC(C1)N2C(=O)C(c1cccc(F)c1)(C)C C1(C(N)=O)(C(=O)O)CCN(C(=O)Nc2ccc(OCO)nc2)CC1.n12cc(nn1)C2 N1(C(Cc2c(C)nn(C)c2)=O)CC(C)OC2(CCN(C(c3ccns3)=O)C2)C1 C1(C(C)C)CN(C(C2CCNC(=O)C2)=O)CC1C(=O)NCCC(O)C(F)F c1(N(CC(CC(=O)NC)C)C)nc(N2CCC(F)CC2)c2c(n1)CCC2 c1(CC)ccc(C(N2CCOC(CNC(=O)CC3SC(=N)NC3=O)C2)=O)c(F)c1 C12CCCN(C1)C(=O)c1ccc(o1)C(=O)N2CC.C1(CNC)CCC(O)CC1 c1(CN2CC(F)(C(N3CC(O)C3)=O)C2)ccc(Br)c(Cl)c1Cl C(=O)(C1=CCCOCC1)N(C)CC1(O)CCN(C(C2CCCC2)=O)C1.C1(=O)CN1 c1(C(N2CCC(NC(c3cccc(Cl)c3)=O)C2)=O)cc(Br)c2ccccc2n1 N1(C(C(CC)OC)=O)CCC(CCNC(=O)C=CCF)CC1.C1C(=O)N1 C12C=CCN(C1)C2=O.C(CO)(C(=O)NCC1CCCN1C1CC1)N(C)C c1(C(N2CCCC(N(C(c3cnn(CC)c3Cl)=O)C)C2)=O)cc(OC)ccc1F C1(CC)CC(CC(N2C(C(N3CCCC(CN(C)C)C3)=O)CCC2C)=O)CCO1 c1(C(=O)NC2CCCN(c3n(C)ccn3)C2)cc2cc(Br)cn2cn1 Cc1c[nH]cc(C(N2CCN(C(=O)CCC=CC(C)C)C3CC23)=O)c1=O N1(C(CC=CCC)=O)CC(=O)CC1C(=O)NC(C)Cn1ccnc1 CCC(C(=O)NC1CC(CC(=O)NCC(O)CF)C1)n1cncn1 C1(NC(c2ncc(NC)nc2)=O)CCCCCC1NC(=O)C(C)OCCC(C)C N1(C(C(C=C=C)C)=O)CCCN(C(=O)Cc2cc(C(C)C)no2)CC1CO N1(C(CCCSC)=O)CCCC(C)C1CNC(=O)CCc1cccc(O)n1 C(C(C)C)(C(O)C(=O)NCC(C)(C)Cn1cc(C2CCC2)nn1)OC N1(C(CC(C)(C)F)=O)CCOC2(CCN(C(=O)C3CCCn4nccc43)C2)C1 N1(C(CCc2n(C)cnc2)=O)CCC(F)(CNC(C2CCCN2N=O)=O)C1 N1(C(CCCSc2cc(C(F)(F)F)nn2C)=O)CCCCC1C1CCCN1CC c1(C(N(CC(CNC(c2nc(C)oc2C)=O)O)C)=O)c(C)sc2ccc(Cl)cc12 CCS(=O)(=O)CC(=O)NCC1CCN1C(c1cccnn1)=O Cc1nc(CNC(=O)CONC(c2cc(Cl)ns2)=O)c(C)s1 C1(CCC)(NC(=O)CCS(C)(=O)=O)CCN(C(C2CCC2C(=O)OC)=O)CC1 c1(CCC(=O)N2CC(=C3CCOCC3)C2)ccc(O)nn1.C1CCSC1 N1(C(C(C)OC2CCCC2)=O)CC(NC(c2cnsc2)=O)C2CCCCC12 N1(C(c2c[nH]ccc2=O)=O)CCN(C(c2cc3n(n2)CCO3)=O)C(CF)C1 N1(C(c2c(C)c[nH]c2)=O)CCCC(NC(c2csnn2)=O)C(F)C1 N1(C(CCSCCCC)=O)CCC2CCC12CNC(c1cc(O)cc(=O)o1)=O C12(CNC(CC(C)n3cccn3)=O)CCCCC1N(C(=O)C1=CCCCC1)CC2 c1(C(=O)NC2CN(C(c3n(CC)nc(C)c3)=O)CC2C)cccc(O)c1C C1(CNC(C2C(C)C2C)=O)CCCCN(C(c2ccccc2O)=O)C1 C1(CNC(CNC(=O)CO)=O)CC12CCN(C(=O)CCCN1C(=O)CNC1=O)CC2 C1(C)(NC(CN(C(=O)OC)C)=O)CCN(C(=O)CCN2CCC2)C1 c1(C(N(C(C)CCNC(C23CCC2CC3)=O)C)=O)cccc(N)c1O N1(C(c2c(Br)cnc(C)c2F)=O)CCC(C)N(C(c2cnn3c2CCC3)=O)CC1 N1(C(CC(C(C)C)O)=O)CCCC2(C1)CN(C(c1cc3ncccn3n1)=O)C2 C1(NC(C)=O)CCCC(CNC(=O)C(=O)NC2CCCCC2CN)C1 c1(OCC)ccc(Cl)nc1C(=O)NC(C)CC1CN(C(=O)C(C)c2cc[nH]n2)C1 C1(CCC)CC(C(=O)NCC(C)(C)CN(C(=O)CN(C)C2CC2)C)CCO1 C1(NC(CSCC#C)=O)CCN(C(=O)C(C)(CO)NC(=O)COCC2CC2)CC1 C1(C(=O)NCCCC2(NC(=O)CSc3cc[nH]n3)CC2)CC2(CCOC2)C1 c1(C(N2CCC3C(NC(c4c(C)cn(C)c4)=O)C32)=O)ccc(F)c(F)c1 N1(C(c2ccc(CNC(C3CCC(C)C3)=O)o2)=O)CCC(CN=[N+]=[N-])CC1 C1(NC(Cc2c(CC)noc2CC)=O)CN(C(C23CC(F)(C2)C3)=O)CCC1(C)C n1(C(C)C)cc(C(=O)NC2(CCCNC(C3(C)CC3(F)Cl)=O)CC2)cn1 CON(C(=O)C1CC12CCN(C(c1ccn(CCF)n1)=O)C2)C1CCCC1 CC1CC(=O)NCC1C(c1ccc(C(=O)NCN=c2nc(C3CC3)[nH]s2)cc1)=O C12(NC(C3CC34CCOCC4)=O)CCCC1N(C(=O)C=Cc1ccoc1)CCC2 N1(C(C(CCC)C(C)C)=O)CC(CO)C2(C1)CN(C(c1occ(C)c1C)=O)C2 C1(COC)(NC(=O)COCCCN(C)C)CCN(C(c2sc(C)cc2C)=O)C1 c1(C(C(=O)NC2CCCC2)N(CCCC)Cc2ccoc2)nccnc1C N1(C(C=CC(C)C)=O)C2CCCC1CN(C(c1cc(S(N)(=O)=O)cs1)=O)CC2 C(C)(C(=O)NCCN(C(=O)CCSC)CC1CCCC1)(C1CCOCC1)OC C1(NC(=O)C(O)C2CN(C(C3CC(=C4CCC4)C3)=O)C2)CCC2CCC12 C1(C(N(C(C(C)C)C)C)=O)COCCN(C(c2ncc(F)cn2)=O)C1 N1(C(C(C#C)(C)C)=O)CC(N(C)C(C2CC3CCC3C2)=O)C2(CC2)C1 C1(C(N(CCCNC(CCN(CCCCC)C)=O)CC)=O)OCCC1C(F)(F)F C1(C#N)(CSC(C)(C)C)CCOCC1.C1(=O)CS(=O)(=O)C(=O)NC(C)(C)CN1C C(C(C(=O)N1CCCC(C(C)NC(C2CCCC(C)CC2)=O)C1)C(F)(F)F)OC C1(=O)C(CCC(N)=O)N(C)C2CN1C2.CCS(=O)(=O)CC(=O)NC1CC12CC(O)C2 c1(CC)cnc(C(=O)N(C2CCC(NC(C3(C(F)(F)F)CCCC3)=O)C2)C)s1 C12(C(=O)NC(C3CCN(C(C4(COC)CC=CC4)=O)CC3)C)CC(C)(C1)OC2C C(=O)(C1CCc2cccnc21)NC1CC(NC(C(c2ccc(C)cc2)C)=O)C1 c1(C(=O)NC2C(NC(CC(C(N)=O)NC(C)=O)=O)CCCC2)ccc([N+](=O)[O-])n1C C1(C(NOC(C)(C)C)=O)CCCC(NC(c2ccn(C)c2)=O)C1 N1(C(CNC(C2=C(C)OCCC2)=O)=O)CCN2CCCCC2C1 C1(NC(c2sc(C)c(O)n2)=O)CCN(C(c2nn(C)cc2N)=O)C12CC2 c1(C(N2CC(O)(CNC(C(CCC)C)=O)C2)=O)c(C)nc(C)n1O C1(CNC(C(CC)SC)=O)CN(C(c2ccc(CSC)o2)=O)CC2(CCC2)O1 C(=O)(C(F)C(C)(F)F)NCCC(=C)CNC(c1nccn1CC)=O C12(C(=O)NCC3(CCOC)CCC3)CCCC1CCN2C(=O)C1=CCN(C)C1 C1(NC(c2ncccc2F)=O)(CO)CCN(C(=O)CCOCC2CCC2)C1 N(C(=NCC(=O)N(C)OCC)N1CCN(c2cccc(C)c2)CC1)C(C=C)C c1(C(=O)NCC(C2CCCCC2)NC(CCC(C)OC)=O)ccc(C#N)n1C C1(C)(CNC(c2n(CCCOC)nnn2)c2cocn2)C2CCC1CC2 C1(C(=O)NC(C2CN(C(C(C)N3CCC3)=O)C2)C)CCC(C(N)=O)CC1 N1(C(C(COC)O)=O)CCC(C2(NC(C3CCC(C(F)(F)F)CC3)=O)CC2)CC1 C1(CNC(C(C)SC)=O)CN(C(=O)COC(F)F)CCO1 C1(OC)CCC(C(=O)NCc2nc(CCC(c3nncn3C3CC3)=O)cs2)CC1 N1(C(C(C)OCCOC)=O)CCN(C(=O)CCc2ccoc2)C(c2cn[nH]c2)C1 C1(C(N(CCN(C(=O)CC2CCCCC(=O)N2)C(C)C)C)=O)CC(=O)NC(=O)C1 CCC(C)(C)CC(=O)NCC1CC1CNC(C1(c2c(F)cccc2F)CC1)=O c1(C(=O)NCCN(C(=O)CCc2ccc(C)s2)CCC)cc(Cl)nnc1O C1(OCCCC(=O)Nc2cccc(OCCC(=O)OCC)c2)CCC2(CCC2)C1 n1(CC)cc(CC(N2CCOC(CCNC(c3csc(SC)n3)=O)C2)=O)c(C)n1 C(=O)(CCC(C)(C)C)NC(=O)C=O.CC(C)CCC(C)C1CCCN1N1CCC(SCC)C1 c1(C(C2CC2)NC(C(=O)NC(C)C(C)n2cncn2)=O)ccccn1 C1(C(=O)NC(CCC)C2CCC2)CCCCC1NC(C1CC=CC(O)C1)=O N1(C(Cc2cn(CC)nc2)=O)CC(C)(C)CC1CC(=O)NCC(C(C)C)OC C1(C)(C(=O)NCC2C(CCC)C2)CC(O)CN1C(c1cnc(S)nc1)=O C#CCCC(O)C(=O)N1CCCC(N(CCO)C(c2cc(Cl)c(Cl)s2)=O)C1 N1(C(C(C)OCC)=O)CCN2CCOCC2(CNC(=O)CSC(F)F)C1 C(=O)(C(F)C(C)C)N(C(CNC(c1nc(CC(C)C)sc1)=O)C)C(C)C C1(CC)C(C(=O)NCCN(C(=O)CC2(C)CCC2)C)CCN1C N1(C(C23N(C(c4c(C)coc4)=O)CCC2CCC3)=O)CCC2(COC(C)C2)C1 C1(NC(CC=CC=C)=O)CC(C)(NC(=O)CCCOC)C1 C1(NC(C(CC)=CC)=O)CCS(=O)(=O)C12CN(C(=O)CSCC(N)=O)C2 C1(C(=O)NCC(C)(C)C(C)C)(CC)CCN(C(C2CCS(=O)(=O)C2)=O)C1 S(=O)(=O)(c1cccc(F)c1C)N1CCCC(C(=O)NC(C(CC)C)CO)CC1 Cc1nccc(Cl)c1C(=O)NCC1(C(C)(C)C)CCN(C(C2C=CCS2)=O)C1 C1(CNC(C2CCCN(C(CC)=O)C2)=O)CCN(C(c2ccc(F)o2)=O)C12CC2 CC1(CCNC(=O)COCC(F)F)CCN1C(=O)CN1CSCC1=O C=CCCCC(=O)N1CC(NC(C23CC(OC)(CO2)C3)=O)C(C(=O)OC)C1 c1(C(N(CCNC(C2CCC(CSC)C2)=O)CC2CC2)=O)cccc(F)c1 CCCCC(C)CCC(C)NC(=O)CCC(C)c1nn[nH]n1 C1(C(F)(F)F)(C(=O)NC2C(NC(c3c(C)cno3)=O)CC2)CC2C=CC1CC2 C1(C(=O)NCC23CCCC(C2)C3)(CC)CCCN1C(=O)CC1(C#N)CC1 Cc1nnc2n1CCN(C(=O)CC13CCC1CN(C(=O)C=CC1CCCC1)C3)C2 CCC(CCCC(=O)NC1COCCC1(F)F)NC(=O)C(=O)C(C)C CC1CC(NC(=O)Cc2c(Br)cnn2C)CN1C(=O)Cc1c(Cl)cnn1C C1(CC#C)(NC(C2(CF)CCN(C(C3C4CCCC34)=O)C2)=O)CCOCC1 N1(C(C2N(C)C(=O)NC2)=O)CCC(C)N(C(C2CC(N(C)C)C2)=O)CC1 C1(NC(Cc2c(C)cco2)=O)CCC(C)N(C(c2ccc(CCN(C)C)cc2)=O)C1 O=C(C1=Cc2ccccc2C1)NC1CN(C(=O)C(F)(F)C(O)C2CC2)C1 CCCC(C)(CC)C(=O)NCC1(C)CC(F)(F)CN1C(c1cc2ccsc2s1)=O C1(CCOC)(NC(=O)CCCC#N)CCN(C(=O)Cc2ccc(F)cc2Cl)CC1 CC1CN(C(c2ccc(C#N)n2C)=O)CCCN1C(=O)CN1C(=O)CN(C)C1=O C1(NC(C2C(CC)C2)=O)CN(C(=O)C(C)(O)Cc2ccccc2)CCC1O Cc1ncc(C(=O)NC2CCC2NC(c2cc(C(N)=O)cs2)=O)s1 CCC(C)(C)CCCC(=O)NC(C)C=CC(=O)NCC1CC(F)(F)CO1 N1(CC(=O)NC2(N(C(CCCN(C(C)C)C)=O)C)CC2)CCC(C)(O)C1 C(CCO)(C(F)(F)F)NC(C1N(C(C(C)OCC=C)=O)CC(F)C1)=O c1(CC)onc(C)c1C(N1CC(OCCC(=O)NCC2COC(C)(C)C2)C1)=O N1(C(CC=C)=O)CC2CCC2(CC(=O)NCC2(C(=O)N(C)C)CC2)C1 C1(NC(=O)CC2CC3CCC2O3)C=CCN(C(c2ccsc2Cl)=O)C1 N1(C(CCc2c(C)ccs2)=O)CCN(C(C2CCCCC2(C)C)=O)C(C(C)C)C1 C1(C(=O)NCC2C(CNC(CCC)=O)C2)CCc2nnnn2C1 N1(C(=O)Cn2cnnc2)CCCC2(C1)CN(CC(O)CC(F)(F)F)CCO2 c1(CC(C(=O)NC(C2CCN(C(=O)C=Cc3ncc[nH]3)C2)C)C)ccc(Cl)nc1 N1(C(c2ccc(COC)nc2)=O)CCCOC(C)C1.c1(OC)ccccc1 C(c1cccc(C)c1)=CC(=O)NCCC1CCCN(C(Cc2nnc(C)o2)=O)C1 C1(NC(COc2c(C)cccc2)=O)CCN(c2ccc(C#N)nc2)C(C)C1 C1(C(=O)OC)(NC(CC=C)CNC(=O)CN(C)CC)CCCOC1 N1(C(=O)C2=C(Cl)CCOC2)CCCC(C2CCN(C(=O)C3CC3)C2)C1 c1(C(N2CC(CC=C)(NC(c3cc(Br)no3)=O)C2)=O)c(C)ncn1O c1(NC(C)=O)cc(F)ccc1C(=O)NCC1(F)CN(C(=O)C(C)S(N)(=O)=O)C1 C(=O)(C(C)(C)SC1CCCO1)N(CCCOCCNC(=O)C=CBr)C C12(C(=O)NC(CN(C)C(=O)NC(C)(C)C)C3CC3)COCC(C1)C2 C1(O)(C(CNC(C2(CSC)CC2)=O)C)CCN(C(=O)CCCC2CCC2)C1 C1(NCc2n[nH]c(=N)s2)CC(NC(C23CCC(CC2)CC3)=O)C12CCOCC2 C(CC(=O)NCC1Cc2nccn2C1)(C(C)(C)C)NC(CS(CC)=O)=O CC1CN(C)CC(C(N2CCC(CC(=O)NC34CC(C)(C3)C4)C2(C)C)=O)O1 N1(C(C(CC#C)NC(=O)CC2(C)OCCO2)=O)CCCCC(C)(F)C1 c1(C(=O)NCC(=O)Nc2cccc(SC(F)F)c2)cc(F)ccc1O N1(C(C(CCC)NC(N)=O)=O)CC2CCCC2(NC(=O)C(C2CCOCC2)O)C1 C(=O)(CC1=CCN(C(c2ccnn2C(C)C)=O)CC1)NCc1onc(C)n1 Cn1cnc2ncnc(N3CC4(CN(Cc5cc(F)ccc5Br)CCO4)C3)c12 c1(C(=O)NC2(C)CN(C(C3(C#N)CC4(CC4)C3)=O)C2)cccc2c1CCC(=O)N2 C1(C(=O)Nc2cn(CC(C)C)nc2)CCC(C2CC2)N1C(C1CC12CC2)=O C(=O)(CCCCCF)NC1CC(CCC(=O)NCCS(=O)(=O)NC)C1 c1(C(N(CCCNC(=O)CCOCC(F)F)C)=O)cn(CC2CCCO2)nn1 C1(F)(CNC(=O)CCOCC2CC2)CCN(C(c2ccc(C(F)F)nc2)=O)C1 C(=O)(CC(C)(C)CNC(=O)CC(C)(C)COC)N1CC(N(C)CC)C1 C1(CNC(c2ccc(CSCC)cc2)=O)CN(C(C2CCOC2)=O)CC12CC2 N1(C(C2(CC)COC2)=O)CC2CC(NC(c3ncoc3C3CCC3)=O)C1C2 C12(C(N(c3ccc4occc4c3)CCOC)=O)CCC(CC(=O)C1)S2(=O)=O C(=O)(CC(C)(C)COC)NC1(CNC(Cc2cc(CC)no2)=O)CC1 C(=O)(C(CO)OCC=C)NC(=O)CC1(C)OCCO1 CCCC(C)(C)C(=O)NC(C1CCOC1)CNC(c1cncc(C(F)F)c1)=O C(CCN=C(NCC1CCC1)NCn1cnnc1C)SC N1(C(CCCC)=O)CCC2(CC1)CCN(C(=O)CCOc1cc(F)ccc1F)C2 C1(COC)(NC(=O)C(F)C(C)C)CCN(C(C2CC(C)N(C)C2)=O)CC1 n1(CC)ccc2cc(SCC(N3CC(c4ccsc4)OCC3C)=O)ccc12 C1(C2(NC(C(C=C)O)=O)CC2)CCCCN1C(=O)CCc1ccncc1 C(=O)(CS(=O)CCC(F)(F)F)N1CCC(c2nc(C3CCCC(N)CC3)on2)C1 C1(NC(C(C=C)(F)F)=O)CC12CCN(C(=O)COc1c(Cl)cccc1Cl)CC2 c1(OC)cc(C(=O)NC2CC(CNC(=O)CCC(N)=O)C2(C)C)ccc1Cl N1(C(COCC)=O)CCN(C(=O)CC2(C)OCCO2)CC1OC(c1ccccc1)C Cc1cccc(OCC(N2CCCC2C2CCN(C(=O)CC3CC3)CC2)=O)c1 c1(C(=O)NCC2(C)N(C(c3cn(CCC)nc3)=O)CCC2)ccc2nc[nH]c2c1 c1(C(=O)NCCC(C)N(C(C(C=CCCC)O)=O)C)cc2c(F)c(Cl)ccc2[nH]1 Cc1noc(C)c1C(=O)NCCOC1CCN(C(=O)CC2CCC(=O)O2)C1 N1(C(c2ncc(C)nc2)=O)CC2(C1)CN(C(c1nn(C)nc1C)=O)CCO2 c1(NC(=O)NC2CCC(CC)CC2)nc2ccc(F)cc2s1 c1(C(=O)NC2CCCCN(C(C3(C)CCCCO3)=O)C2)cnc(S(C)(=O)=O)s1 c1(C(N2CC3C(NC(CCc4n(C)ncc4)=O)(C3)C2)=O)c[nH]ccc1=O c1(C(=O)NCCNC(C(C)Cn2ccnc2)=O)ccc(C(F)C(F)(F)F)cc1 C1(C(=O)NCCCOCCN(C(Cc2c(C)ocn2)=O)C)CC1C1CCCC1 C1(C(=O)NCCn2cc(C(=O)NC(CSC)(C)CO)nn2)CCCC(C)(C)C1 Cc1ncc(Br)c(C(=O)NC2CC3CCC2N3C(=O)Cc2cccc(C#N)c2)n1 N1(CC(=O)N(CCCCC)CCN=[N+]=[N-])CCCC(C)(OC)C1 N1(C(=O)Cn2cc(-c3ccccc3)cn2)CCOCC(C(F)(F)F)C1 c1(-c2onc(CC(=O)OCc3ccc(C)cc3F)n2)cc2cnccc2n1C c1(C(=O)NCCOC2CCN(C(C3(F)CCC3)=O)C2)nc2cc(O)ccc2[nH]1 C=CCC(C)(C)C(=O)NC1CNC(Cn2cnnc2)C1 N1(CC(C(=O)NCC(=C)C)NCC(C)C)CCCC(C(=O)OC)C1 c1(NC(N(c2nc(C(=O)OC)sc2)CC)=O)cccc(Br)c1[N+](=O)[O-] N1(CC)C(=O)CCC1CC(N1CC(NC(=O)CCC(=O)OC)C(C(F)(F)F)C1)=O c1(C(=O)NCC2C3CN(C(C4CCC(C)(CC)O4)=O)CC32)cc2ncccc2o1 CC1CC(NC(c2coc(CO)c2)=O)CN1C(c1cc(C2CC2)nn1C)=O c1(CNC(=O)N(c2c(O)cccc2O)Cc2cccnc2)ccc(O)c(CO)c1 C1(C(=O)NCC(CNC(Cc2cccc(C(N)=O)c2)=O)O)CC12CCSCC2 N1(C(C(C)OCC#C)=O)CCC(C(CO)NC(=O)C(C(C)C)n2cnnc2)CC1 c1(CNC2(CC(=O)NN3CCNC3=O)CCC2)c(F)cccc1Cl c1(C(=O)NC(=O)CC2CCCN2)c[nH]nc1C1CCCNC1 c1(CC)ccc(CC(C)(O)C(=O)NC)cc1.n12nnnc1N1CCC(C1)C2 c1(C(=O)NCCCNC(=O)CC2CCS(=O)(=O)C2)c[nH]c2c(F)cccc2c1=O Cc1ccc(C(C)NC(=O)CC2CC(NC(=O)CC3CSC3)C2)s1 CC1CC(CC(=O)N2CCC2)CN1C(c1c[nH]nc1Cl)=O N1(C(c2n(CC)ncc2Cl)=O)CCC(NC(=O)COC)C(O)C1 N1(C(C(C)Oc2ccc(F)cc2)=O)CCC(NC(=O)CCP(C)(C)=O)C(O)C1 C1(C(=O)NCCCC(=O)NO)(CC)CCCN1C(=O)CN1CCCC1 N1(C(C(N2CCC(C)CC2)=O)=O)C2CCC1(CNC(=O)CCCCC1CC1)CC2 c1(CCC)c(C(=O)NCC(C)(CC)NC(=O)CO)cnn1C N1(C(C(C2CCCCC2)OC)=O)CCC2CCN(C(C3CCC=CCC3)=O)CC12 C(C)(C(C(C)C)NC(=O)CC1CCN(CC(F)F)CC1)NC(c1c(C)ccs1)=O N1(C(C(CCCC)CC)=O)CCCC2(CCC2NC(c2coc(CO)c2)=O)C1 C1(N(C2(C(F)(F)C(F)(F)F)CC2)C(C)=O)CC(C)CN(C(c2c[nH]cc(C)c2=O)=O)C1 C1(CC)C2CCC(C2)C1NC(=O)N(c1c(SCC)cccc1)Cc1cc(C)ccn1 c1(OC)ccc(C(=O)NCC(F)CNC(=O)C(C)CSC)c(OC2CC2)c1 c1(OC)cc(C(=O)NCCC2(NC3CC3C(F)(F)F)CCCC2)cc(OC)c1C C1(C2CC2)(C(N2CCC(OCCN(C(CCCNC(C)C)=O)C)C2)=O)CC=CC1 CC1(C)CC(C(N2C3CCC2CC(NC(=O)CC2OCCO2)C3)=O)CNC1=O c1(OC)c(NC(=O)NC2CC3(CCC(C(N)=O)CC3)C2)ccc(F)c1F CCC(CC)(CCNC(c1ccc(Cl)cc1C)=O)NC(c1ccn(C)c1C)=O Cc1cc(C(N2CCC(C3OCCC3NC(=O)CCC3CCC3)CC2)=O)ccn1 c1(C(=O)NCC2CN(C(C)=O)C(C)CC2)cc2ncccc2o1 c1(OC)cc(C)cc(C(=O)NC2CN(C(C3OCCO3)=O)CC2(C)C)c1C c1(N2CCC(NC(C3COCC4(CCC4)O3)=O)C2)ncc2scc(Br)c2n1 C1(C(=O)NC2CCCCC2O)CCCC12CCN(C(C1CC3CCC1O3)=O)C2 CN1CCN(C(=O)C(=O)NC2CCC3CCCC23)CC12CCC2 N1(C(C(C)OC2CCOC2)=O)CCN(C(C2(C#N)CCC2)=O)CC1COC CC1CCC(C)(C(N2CCC2CC(=O)NCC2C=CCCC2)=O)CC1 C1(NC(C(C)OCC2CCCO2)=O)CN(C(=O)COCC2CCCC2)C2CC12 c1(OC)cncc(C(N2CC3CC3C2)C(=O)NCc2ccncc2F)n1 N1(C(C(CCC)CCC)=O)CC(NC(=O)C=Cc2ccccn2)CC2(CCC2)C1 N1(C(c2conc2OC(F)F)C(=O)NCC(C)C)CCCC(CO)C1 c1(CS(C)=O)ccc(S(=O)(=O)NCCc2ccccc2N2CCCCC2)cc1 Cc1cc(Cl)cc(Cl)c1-n1cc(CC(C(=O)O)NC(=O)CCOCC(F)F)nn1 N1(C(CC=CCC)=O)CCC2(CC1)OCCC2NC(=O)C=Cc1cncs1 C1(CNC(C=CC(C)C)=O)CC2CN(C(=O)CNC(=O)CN(C)C)CC12 C12(C(=O)NCc3c(C(=O)NC(c4onc(C)n4)(C)C)c[nH]n3)CCCCC1C2 C1(C(=O)NC(c2ccc(F)cc2)CNC(=O)CCC2CC2)CC2C=CCC(C1)C2 N1(C2(C)C(C)(CC)NC(COC)C2)Cc2ncccc2NC(=O)C1C c1(OC)cc(C)cnc1C(=O)NCC1(O)CCN(C(c2nc(C)[nH]c2C)=O)C1 C#CCCCCC(=O)N(CC(C)N(C)C(C1CC(N(C)C)CCO1)=O)C C1(C(=O)NC2CCCC(CNC(c3cnc[nH]3)=O)C2)CCc2ccccc2O1 c1(C(N2CC(C)(NC(CCC3CCC(C)O3)=O)C2)=O)ccc(F)cc1Cl N1(C(CCc2cnc(C)s2)=O)CCC(NC(=O)CC2CC=CC2)CC(O)C1 C(=O)(C(C)(O)C(C)c1ccccc1)N1CC(O)(C(C)NC(=O)CC(C)(C)C)C1 C1(OC)CC(CNC(=O)CCC2NC(=O)NC2=O)N(C(c2nc(C)sc2C)=O)C1 c1(NC(c2cc(F)ccc2OC(F)F)c2n(C)nnn2)cc(Br)cc(O)c1 C1(NC(C2C(C)OC(=O)N2)=O)CC2CCC(C1)N2C(C1CC(C)(C)C1)=O [N-]=[N+]=NCCCCC(=O)N1CCC(CCNC(C2CC3CCCC3C2)=O)C1 n1(CC(=O)NCC2CC2NC(c2ocnc2C(F)(F)F)=O)ncccc1=O CN1CC(N=c2[nH]c(N3CCC(C)(C)C3)nc3ccc(OC(F)F)cc23)CCC1=O C(=O)(CCC(C(C)C)NC(=O)CC1CCCC1O)N1CCCC(CC=CC)C1 C=CCC(C(=O)N1CCC(CNC(=O)CCn2c(C)csc2=O)CC1)OC C(=O)(C1CSc2ccccc21)N1CC(SC)C(NC(=O)Cc2ccns2)C1 c1(OCC)ccc(CNC(=O)C(=O)NCC(c2ccc(F)cc2F)F)cc1OC Cc1noc(CC(=O)NCc2cnn(C3CN(C(C4(C)CC4(F)F)=O)C3)c2)n1 N1(C(CNS(CC)(=O)=O)=O)CC(CNC(=O)Cn2cnc(=N)[nH]2)C2(CC2)C1 C1(CNC(CC=C)=O)CCCCCN1C(=O)C=Cc1ccc(C(N)=O)o1 N1(C(CNC(=O)OCC=C)=O)CCCC(NC(=O)Cc2ccc(C)nc2Cl)CC1 N1(C(CN(C(C(C)C)=O)C)=O)CC(O)C(O)C1NC(C(C(C)N)CC1CC1)=O CON(CC1CC1)C(=O)C(CC(F)F)N(C(=O)CC1CC1C)C C(CCCCCC(=O)N1CCC(O)C(C)C1)NC(c1c(C)nc(C)o1)=O Cc1cccc(OCC(=O)NC2C3CC2N(C(=O)CC(C)c2ccncc2)C3)c1 C1(C)(C(N(C(C(=O)NCC(C)Cn2cccn2)C)C2CC2)=O)COCCO1 C12(CNC(CC=C=C)=O)CCCC1N(C(c1ccc3nc(C)cn3c1)=O)CCC2 N1(C(C2C(NC(C(CC=C)OC)=O)CCO2)=O)CCC(F)(F)C(F)C1 c1(C(=O)NC(CN(C(C2(C=C)CCC2)=O)C)C)c(NC(C)=O)cccc1F c1(C(=O)NCC(C)N(C(C(C)NC(=O)NC)=O)C)c[nH]c(=O)cn1 C1(C)C(=O)NNC(=O)C2C(=O)NCCN12.CCCCSC(C)=O C(=O)(C(CC)C(=O)NC1(C(=O)NC2CC(=C3CCC3)C2)CC1)OCC c1(CC(=O)NC(CCNC(c2c(C)scc2)=O)C)cc(F)cc2ccccc12 c1(N(C(c2ccccc2)CNC(CCC)=O)C)ncc([N+](=O)[O-])cn1 CC(C)CC(C)(C)CNC(c1ccnc(CNC(C2CCN2C)=O)c1)=O c1ccnc2ccccc12.c1(C(C)CNC(=O)NCC=CCN)ccc(F)c(Br)c1 c1(CNC(CCCOCC=C)=O)cccc(CNC(C2(S(N)(=O)=O)CC2)=O)c1 Cc1cccc(C)c1-c1cn(C2CCN(C(=O)CC3(C)NC(=O)NC3=O)CC2)nn1 C1(C(N2CC(CO)(NC(C3CCOCC3)=O)C2)=O)(COC)CC(F)(F)C1 C1(NC(CN(CCCCCC)C)=O)(CF)CCN(C(C2CCCCCC2)=O)C1 C1(F)(CNC(c2c(C)onc2)=O)COCCN(C(C2(S(N)(=O)=O)CCCC2)=O)C1 C1(C(=O)NCCC2(NC(CCOCC(C)C)=O)CC2)CC2(CCC2O)C1 c1(N2CC(CN(C)C)OCC2)nc(=NCC2OC(=O)NC2(C)C)[nH]c2c1COC2 c1(C(=O)NCC2C(NC(C(F)=CCC)=O)CCC2)nn(C)cc1C c1(C(=O)NC2CCN(C(C3N(C)CCC3)=O)C2)c(Br)ccc2ccncc12 c1(CC=C)cccc(C(=O)NCCC2(O)CN(C(=O)CCOC3CCOC3)C2)c1 C1(NC(CC2(C)CC2(F)Cl)=O)CCN(C(=O)CCn2ccnc2)CC1F Cc1ccc(N)c(C(N2CCC3(NC(c4[nH]ncc4C#N)=O)CC3C2)=O)c1 CN1CCC(NC(=O)C2CC2)C12CCCNC2.C12(COC1)CN2 C1(n2cnnn2)(C(N2C(CNC(c3c(C(C)C)con3)=O)CCC2)=O)CCOCC1 C1(CN(C)C(C2CNC(=O)N2)=O)CC2CCC(C1)N2C(=O)Cn1ccsc1=N C(C1CN(C(C2CC=CC2)=O)Cc2ccccc21)NC(c1cc(Cl)ncc1Cl)=O n1(CCC(=O)NC(C(C)NC(C2(CC#C)CCCO2)=O)C)ncn(C)c1=O c1(C(=O)NCCN(C)C(C2Cc3nccn3C2)=O)c(N)ccc(Br)c1F CCC(C(=O)N1CCC1CNC(C1(OC(C)=O)CCCO1)=O)N1CCCC1=O C(=O)(CP(C)(C)=O)N1CCC(CCCCNC(Cc2nc(C(C)C)sc2)=O)C1 C1(CNC(CC=C(C)C)=O)CC2(CCN(C(C3CC(n4ccnc4)C3)=O)C2)CO1 C(N=C(NC(c1ccccc1)C)N1CCN(C(C)C)C(=O)C1)C1CC(OC)(OC)C1 CC(C)CC(C)(CNC(=O)CNC(=O)C1CC1)NC(=O)N(C)C CCC1=C(C(=O)NCCC2CCCN(C(=O)Cc3cc(C)on3)CC2)SCCO1 Cc1cc(Cl)ccc1CC(=O)NCCOCCCN(C(=O)CCCC(C)C)C c1(CC(CSC)N(CC(O)C(F)F)CC(=O)OCCC(=O)O)ccccc1 c1(C(N2CCC(COC)(NC(c3cc(Br)c[nH]3)=O)C2)=O)cccc2nsnc12 c1(C(=O)N(C2CC(CCNC(C)=O)C2)C2CC2)cnc(-c2ccsc2)s1 C1(NC(CNC(CC)=O)=O)CC(CNC(=O)CCC(C)C)C(O)C1 c1(CC)[nH]ccc1C(=O)NCC1CCC(NC(=O)C(CC)n2cncn2)C1 N1(C(C=Cc2ncn(C)c2)=O)CCN(C(c2nc3ncccn3n2)=O)CC(O)C1 C(=O)(C(CO)C(C)(C)C)NC12CCC(CNC(CCCCCC)=O)(OC1)C2 Nc1cc(N2CCNCC2)ccc1N1CCNC1=O.C1(C(=O)O)CCN1 c1(C(=O)NC(CNC(C2C(C=C)OCCC2)=O)C)coc2c1N(C)C(=O)CCC2 S1(=O)(=O)c2ccc(cc2Br)C(=O)N1.C1(N(C)C)(CO)CC2CCC1CC2 N1(C(Cc2nc(=N)[nH][nH]2)=O)CCN(C(C2CCCO2)=O)CC1C(F)F c1(N2CCC(O)(CN3CCC(C=C)CC3)C2)cc(SC)nc(S(C)(=O)=O)n1 C#CCC(C)(C(=O)NC1CNC(=O)C12CC2)NC(=O)CCSC c1(C(=O)NCC(CC)NC(=O)CCn2ccnn2)ccc(CN2CCCC2)o1 C(=O)(C(C)CC(F)(F)F)OCC.S(=O)(=O)(CC(=O)NCC1CCN2C1C2)NCC c1(C(=O)NCCC2(C(=O)NC(CO)C3CCC3)CC2)cccnc1O N1(C(c2ccc(NC)cc2)=O)CCOCC(F)(CNC(=O)CCC(C)(F)F)C1 Cc1c(C(N2CC(NC(c3c[nH]c(C(N)=O)c3)=O)C(O)C2)=O)noc1C1CC1 CC(C(F)C(=O)N(CCCCCCNC(C12CCCN1CCC2)=O)C)C(F)(F)F C1(N2CCN(c3n(CC)c(C4CCOCC4)nn3)CC2)C(C)CCCC1(C)C N1(C(Cc2cc(OC)c(F)cc2)=O)CC2CC(NC(=O)C=C3CCSCC3)C(C2)C1 C1(F)(C(=O)NCC(C)(C)OCC(=O)NCC2CCC(C#N)C2)CCCCC1 C=CC(C)(O)CC(=O)NC(C)(CNC(=O)C=Cc1ccccc1Cl)CC c1(C(N2CCCC(NC(CNC(C)=O)=O)C2)=O)ccc(Cl)c(F)c1 N1(C(c2cc(C)nnc2)=O)CCN2C(=O)C(NC(c3cccnc3)=O)CC2C1 c1(C(C)C)ccc(C(N2CCC(C(C)NC(c3c[nH]c(C#N)c3)=O)C2)=O)nc1 C(=O)(C(C)(C)C(=O)NCC1CCCCN1C(=O)CC(F)F)OC(C)(C)C n1(CC(=O)NC2(C)CN(C(=O)CN3CCCCC3)C2)cnc2ccc(F)cc2c1=O C12(C(=O)NCCCN(C(c3ccc(CC)cn3)=O)CC)CSCC1C2(F)F CC1CCC(C)N1C(C)C(=O)NC(C1CCN(C(c2cnoc2)=O)CC1)C C1(C(=O)NCC(CC)NC(c2cccn2CC)=O)CCCCC1C(=O)OC C(=O)(CCCCC(N)=O)NC(C(C)C)(C)CNC(=O)Cc1cnccc1Cl c1(CC)cc(C)c(C(=O)NCC#CC(=O)NCC=CCO)o1 c1(C(=O)NC(CN(C(=O)Cc2cnoc2)CC)C)cn(C)c(=O)cn1 C(=O)(CCCC(=O)N1CCCC(CN(C)C(C2CC(C)(C)C2)=O)C1)OCC c1(C(C(N2C(CNC(c3cnc(C)s3)=O)CC2)=O)O)ccc(CC(C)C)cc1 N1(C(=O)CSn2nnc(C3CC3)n2)CCCN(C(c2ccccc2F)=O)CCC1 c1(NC(=O)NCC2C(Nc3ncc(C#N)cc3Cl)C2)ccc(C#CCCO)cc1 C(C1CN(C(=O)CNC(C)=O)CC1C(=O)NCC(C)N)=CC C#CC1(O)CC(C(N2CCC(C(C)(C)NC(c3scnc3C(F)(F)F)=O)C2)=O)C1 N1(C(CCCC(=O)OC)=O)CCCCC(N(C)C(C2CC(C3CC3)C2)=O)C1 N#Cc1ccc(NC(c2ccn(CCNC(=O)CSC3CC3)c2)=O)c(O)c1 C#CC1(C(=O)NC(C)(C)C)CCN(CCOCCN2CCCS2(=O)=O)CC1 n1(COCC)nnc(C(=O)NCC2CN(C(=O)C(C)NS(C)(=O)=O)C2)c1N CC(CNC(=O)C(F)=CCCF)(CO)NC(=O)CC1CCC(=O)N1 c1(OC)ccc(CNC(c2coc(C)n2)c2nnnn2CC2CCCO2)cc1Br Cc1nn(C)cc1C(O)C(=O)NC(C)CNC(c1csc(N2CCCCC2)n1)=O C#CCC(C(=O)NCC(C1CC1)SC)NC(C1CC12CCCC2)=O c1(C(=O)NCC(C)NC(=O)CC(C)CC(C)(C)C)cncc(P(C)(C)=O)c1 C(=O)(C(C)(C)C(C)O)NC(CNC(Cn1c(C)c(Br)cn1)=O)CO N1(c2n(C)c(CCn3cnc4ccccc34)nn2)CC2CC(O)CC2C1 N1(C(CN(C(=O)OC)C)=O)CC(NC(c2[nH]cc(C)c2C)=O)CC1C C(=O)(CC(C)(C)C#N)NCC1(COC)CCN(C(=O)CCOC2CC2)C1 CCCCC(CNC(c1cnn(C)c1F)=O)NC(=O)COC N1(C(CCC#N)=O)CCC2(CCC2)C(CNC(=O)CCC2CCCOC2)C1 C(=O)(CCCCCCS(N)(=O)=O)NC12CC(CNC(C(C)(C)C)=O)(C1)C2 C1(C(N2CCC(NC(c3ccc(C4CC4)cc3F)=O)C2)=O)CCCC1C1CC1 Cc1cc(C(N2CCC(NC(=O)Cc3ccc(C#N)cc3)C2)=O)c(C)cn1 N1(C(CNC=O)=O)CCCCC1C1(O)CN(C(=O)CCc2cccc(Br)c2)C1 N1(C(C(COC)OC)=O)CC(NC(c2ncccc2O)=O)CC(C)C1 C(=O)(CC(C)CC(C)C)N1CC(NC(C2(C#C)CCOCC2)=O)CC1(C)C C1(CNC(C(C)CCO)=O)CC2(CCN(C(c3cnc(C(C)O)s3)=O)CC2)CO1 c1(C(=O)NC(CNC(CSCC(N)=O)=O)CO)cccnc1S(=O)(=O)C(F)(F)F c1(C(N2CC(C)(NC(=O)Cc3cccnc3)C2)=O)csc(=NC2CCOCC2)[nH]1 N1(C(C2C(CC)C2)=O)CC(C2CN(C(=O)CCc3cc(Br)ccc3C)C2)C1 C=CCC(C(=O)OCC)NC(C1(O)CCN(C(c2ccncc2C)=O)C1)=O N1(C(Cc2c(C)noc2)=O)CC(CNC(c2cnco2)=O)C(F)(F)C1 C1(N(C(C2(NC(Cc3c(C)occ3)=O)CC2(C)C)=O)C2CC2)CCN(C)CC1C C1(C#N)(NC(c2c(C)nsc2)=O)CCN(C(C2(C)CCC2)=O)C1 C(=O)(C(CO)C(C)(C)C)N.C1(OCC)CCCC(NC(C2(CO)C(C=C)C2)=O)C1 C12(NC(CNC=O)=O)CCOC(CO)(C1)C2.c1(C(=O)N)ccnc(N2CCCC2)n1 CCC(CC)CC(=O)N1CCC(C2CCCN2C(=O)COC2CCOCC2)CC1 N1(C(=O)C=C(Cl)Cl)CCCCC1NC(=O)CCNS(=O)(=O)C(F)(F)F CC1(C)CC(C(=O)NC(CO)C2CC2)CCN1C(C1CCC=CCC1)=O c1(C(N2CCC(NC(c3cc(O)cc(F)c3)=O)CC2)=O)cnc2ccccc2c1 c1(OC)c(C(=O)NC(C2COCCN2C(C2COC(=O)O2)=O)C)nc(O)nc1O N1(C(Cn2ncc(CC)c2)=O)CCN(C(c2cnn(CC3CC3)c2)=O)CC1CC CC1Cn2nc(C(=O)NCCC(C)NC(C3CC=CCC3)=O)cc2C(=O)N1 n1(CC(=O)NCC(CNC(C(C)SCCCC)=O)O)cc(CO)nn1 C1(CNC(C(C)(C)COCC(F)F)=O)CC(F)(F)CN1C(=O)CCc1ccc[nH]1 CC(CN=c1nc2c(ncn2C)c(NCc2ccc(C#N)cc2Br)[nH]1)C(C)(C)C Cc1c(C(=O)N(C2CCCOC2)C2CC2)cnn1CC(C)(C)O C1(NC(c2ccsc2)=O)CC2CCC(C1)N2C(C1CCc2n[nH]cc2C1)=O N1(C(C2C(OC)CCC2)=O)CCCCCC1CNC(=O)C(c1cccnc1)O CCCC(CC)CCC(=O)NC(C1CCCC1)CNC(c1cc(C)co1)=O C(=O)(C1CCCc2c(O)cccc21)NCC1N(C(c2c(C)oc(C#N)c2)=O)CC1 C(CC)(CCCO)N(C(C(C)N(CC(=O)NCCCO)CC)=O)C1CC1 c1(OC(C)C(N2CCC(CCNC(C34CCCC3C4)=O)C2)=O)ccccc1Cl CC(CC(F)(F)F)C(=O)NC1CC2CC1N(C(c1csc(Br)c1)=O)C2 C(C(=O)NCC1(C(F)F)CCN(C(=O)CCCc2cnccn2)C1)(C(C)C)OC c1(C(C(=O)NCCC)N(C(C)(C)C)CCC2CC2)ccc(C2CC2)s1 N(C1CCc2cccnc21)CC(c1cc(Cl)ccc1Cl)O CC1CCN(C(C2CN(C(C3CC4C=CC3C4)=O)CCO2)=O)CCC1O N1(C(C(CC)CC2CCCC2)=O)CC2(CNC(=O)CCC3CC3(Cl)Cl)CC1CCO2 N1(CCCCOC(C)=O)C2CCCC1CC(N=c1nc[nH]cc1C#N)CCC2 c1(C(N2CCN(C(C(C)O)=O)CC2c2cn[nH]c2)=O)cnc2c(n1)CCCC2 C12(C(N3CCC(O)(CCNC(c4ncccn4)=O)CC3)=O)CCCC1C2(F)F C(=O)(C1=NOC(CNC(c2cncc(O)c2)=O)C1)N(CC(C(C)C)C)C C1(CSC2CC2)CCN(C(=O)Cc2cn(NC(CC(C)OCCO)=O)nn2)C12CC2 c1(C(=O)NCC2CC(NC(Cc3cc(CC)no3)=O)C2)ccc(O)c([N+](=O)[O-])c1 Fc1cc(Br)c(CSCc2ccc(I)cc2)cc1F C(=O)(C1=CCCCCC1)NC1(CO)CCN(C(C2C(C)(C(F)F)C2)=O)CC1 c1(C(N2C(CNC(CC3CC(C(=O)OC)C3)=O)CC2)=O)cc(C)c(N)cc1Cl c1(C(=O)NCC(C(C)C)NC(c2cccc(SCC#C)c2)=O)cc2sccc2[nH]1 C1(C(=O)NCC2CCC(NC(CCNC(=O)C=CCl)=O)CC2)CCN2CCOCC12 C1(NC(C2(CC)CCOC2)=O)CCCCC1NC(C1C=CCS1)=O c1(C(=O)NC2CCN(C(CCCCC=CC)=O)C2)ccc(Cl)c2ncccc12 C1(N(C(C2CCC(C)C2)=O)C)CCN(CCNC(=O)C(C#N)=CC(C)(C)C)CC1 Cc1cc(F)c(C(=O)NC2CCN(C(c3ccc(C#N)o3)=O)C(C)C2)cc1F c1(C(C)C(N2CC(C)CC2C(N2CC3CCC2CC3)=O)=O)ccc2c(c1)COC2 c1(SC)ncc(C#N)c(N2CC3CCC(C(=O)NOCc4ccc(C)cc4)C3C2)n1 O=C(CCC1CCOC1)NCC1CC(NC(=O)CCc2cccs2)C1 c1(N2C(CNC(C3CCCC(C)C3)=O)CCC2)ccc([N+](=O)[O-])c2cccnc12 C(=O)(C1CCCc2ccnn21)N1C(C2CCN(C(C(C)O)=O)CC2)C(C)(C)C1 N1(C(CC(C)(F)F)=O)CCCCC(CNC(=O)CCOC2CCOCC2)C1 N(C1CCc2c(Cl)cc(F)cc21)C(c1cc(-c2ccc(F)cc2)nn1C)C C(=O)(CCCCCC(C)C)NCC1CCC(CN(C(C2C(COC)C2)=O)C)CC1 C1(CNC(C(C)(C)CO)=O)CC2(CCOCC2)CN1C(=O)C1=CCCOC1 C(CCN(C(=O)CSc1ccccc1C)C)(C(C)C)NC(c1ncn(CC)n1)=O N1(C(C(CC=C)(C)O)=O)CC2CN(C(c3ccn(C4CC4)n3)=O)CCC12 c1(COC)nc(C(=O)NCCN(C(c2c[nH]nc2C2CCC2)=O)C2CC2)co1 n1(CC(=O)NC2(CNC(C3CCC(C)C3)=O)CCC2)ccc2ccccc2c1=O C(=O)(C1CCCc2nnn(C)c21)N1CC2CN(C(C3CC(C)SCC3)=O)CC2C1 C1(SCCOC2(C(=O)O)CCN(C(C(CC(C)C)O)=O)C2)CCc2ncnn2C1 N1(C(CCCNC(=O)OC)=O)CCC(C)(C)C1C(=O)NCCN1CC2CC2C1 c1(SC)cn(C)nc1C(=O)NCC1(CCNC(=O)C=C(C)C(C)(C)C)CC1 C1(CC(=O)NCC(N(C(C(CN(CC)CC)F)=O)C)C2CC2)OC(C)(C)OC1=O N1(C(N(c2nc(C)sc2)C(C)C)=O)CC(F)C(F)C1 c1(C(=O)NC(C)CN(C(=O)CNc2nccs2)C)cccc(CC#N)c1 CCCCC(O)C(=O)N(C1CCN(C(C2CCCN2C(=O)OCC)=O)CC1)CC c1(OC)cc(C(N2CC3CC2(CNC(C2CCCC(C)CC2)=O)C3)=O)ccc1Cl c1(C(C)NC(c2cccc(NC(CCc3ccsc3)=O)c2)=O)ccc(Cl)cc1F N1(C(C(C)NC(C)(C)C)=O)CCN(C(=O)Cc2cc(F)cc(Cl)c2)CCC1C Cc1cnc2n1CCC(C(N1CC3CC1CN3C(c1n[nH]c3ccccc13)=O)=O)C2 c1(OC)cccc(Cl)c1C1CC1NC(=O)CNC1CCOCC1 C1(N2C(CNCc3ccccn3)CCC2)CCC2(CCCC2)C1.n12cc(nn1)C2C1CC1 c1(OC)cc(C2CC(=O)N2)ccc1C.S(=O)(=O)(C(C)C)NC C(=O)(CCCCCN1CCCC1)NCCCOCC(C)C C1(CN(C(=O)Cn2cncn2)C)CN(C(c2ccsn2)=O)CCC12CCC2 N1(C(CC(C)(C)N(C(c2ccc(OC)nc2)=O)C)=O)CCCC(C2CC2)CC1 c1(C(=O)NC2(C)CN(C(c3ccc(F)cc3)=O)C2)ccc(-n2cnnn2)c(Cl)c1 N1(CC(=O)NC2CCC(C)N(C(c3nc(Br)c[nH]3)=O)C2)CCc2ccccc21 C=CCC(C)(C)CC(=O)N(C(C)(C(=O)NCCOCCF)C1CC1)C c1(OC)cncc(C(N2CCCCC2CN(C)C(C2OC(C)CC2C)=O)=O)c1 c1(C(N2CC(C(=O)NC3CCOC(C)C3)(COC)C2)=O)cc2ccccn2c1 C1(CNC(CC2CN(C)C2)=O)CC(NC(=O)COCc2ccncc2)C12CCC2 C12(NC(CCSc3n(C)ncn3)=O)CCC1CN(C(C1CC3CC3C1)=O)C2 c1(C(N2CC(CCOC)C2)=O)cc2cccnc2cn1.C12(CCC1)C(=O)N2 CN1N=C(CC(=O)NCC2CC3(C2)CN(C(c2ccc(F)cc2F)=O)C3)CC1=O N1(C(CNC(CC)=O)=O)CCC2CCN(C(=O)C#CC3(O)CC(CC)C3)C2C1 C(C(C)C(C)C(=O)NCCC(C)(C)NC(=O)C(C)Cc1cnn(C)c1)OC c1(C(=O)NC23CC(NC(C(c4cncnc4)C)=O)(C2)C3)nn(C)c2ccccc12 C(=O)(C(CC(C)C)C(C)C)N1C(CC)(CC)CC(NC(c2cc(N)ccn2)=O)C1 c1(C(=O)NCC2CCN(C(CC(C)O)=O)C23CC3)cnc2c(F)ccc(F)c2c1 O=C(Cn1ccnc1S(=O)(=O)N1CCOC1=O)NNC(=O)N1CCCC1 Cc1cnc(C(=O)NCC2CN(C(=O)C(c3ccnn3C)C)CC2C)cc1C c1(CNC(c2cc(C(=O)NCC3(C)OCCO3)ccn2)=O)nc2ccccc2o1 c1(CN(C(CN(C(COC)=O)C)=O)C)cccc(CNC(C2CC2(C)C)=O)c1 C(=O)(C1=CC2(CCOC2)C1)N1CC(OCCNC(CCc2n(C)ccc2)=O)C1 Cc1cc([N+](=O)[O-])ccc1NC(=O)CCOC(=O)CC1CC(O)C1(C)C c1(CC)ncoc1C(=O)NCCCOCCCNC(C1CNC(=O)N1)=O Cc1cnc(C(=O)NCCC2COCCN2C(=O)CCCCCF)c(C)c1 C1(CNC(C(CCOC)C)=O)CCCCN(C(=O)C(C)Cc2cccc(F)c2)C1 C1(NCCO)CN(C(=O)NCCNc2cccc(F)c2)CCC2(CCCC2)CO1 N1(C(c2c(C)nc(O)cc2)=O)C(C(=O)NCCn2cnnn2)C2CC(O)C1C2 c1(C(=O)NCC(CNC(c2cc(CCOC)on2)=O)C)cccc(C(F)(F)F)n1 C1(C(=O)NC(CCCCC)C2CC2)CN(C(c2ccnc(C)n2)=O)CC(F)(F)C1 C(CN=c1cc(NCCCc2csc(C)n2)nc[nH]1)n1c(C)nc(C)n1 CCC(F)C(=O)NCCC1(NC(=O)COCC2CC2)CCC1 C(C1=CCN(C(c2sc(Cl)nc2Cl)C(=O)NC(C)CC)CC1)OCC CC(C)C(C(=O)N1CCC(CN(C)C(C23CC(CF)(C2)C3)=O)C1)N1CCCC1=O C(=O)(CC1=CCCC1)NC1(CC=C)CCN(C(C2(C#N)CC(C)C2)=O)C1 C1(C(N2CC(=C(CNC(C(CC)N(C)CC)=O)F)C2)=O)CN2CCN1C(C)C2 C(=O)(C1=CCCN(C(=O)C(CC)(CO)OCC)C1)N1C(CCCC)CCC1 C(CC(CNC(=O)CSc1ccncc1)NC(=O)C(C)C1CCCC1)OC C1(C(=O)NC(C(=O)NCC(C2CC2)SC)(C)C)CCc2c[nH]nc2C1 C(CNC(c1sccc1Br)c1nnnn1CSc1ccccc1)(C(C)C)OC C=CCCCCCCCC(=O)N1CC(NC(c2cccc(CO)n2)=O)C1 CC1(C)CCC(C(=O)NCCN(CCOCCO)C(c2ncn3c2CCC3)=O)CC1 C(C(=O)N=c1cco[nH]1)N1CCC(NC(c2cccc(Br)c2O)=O)C1 C1(C(=O)NC2CC=C(C)CC2)CC(C)(C)CCN1C(=O)CCCC(=O)N(C)C c1(C(=O)NCC2(CN(C(C3(C#C)CCCC3)=O)C)CC2)ccc2ccccc2c1F N1(C(C2(OCC)CCOC2)=O)CC2CC1(C(=O)NCC=Cc1ccco1)C2 Cc1ccc2c(=O)c(C(N3CCC(NC(=O)CCS(C)=O)C3C)=O)c[nH]c2c1 C(=O)(C(CC1CC1)NC(C1CCCS1)=O)N(C1CCOC1=O)C C1(C(N(C)Cc2nc(C)sc2)=O)CCC2(CC2)N1C(c1sccc1C#N)=O C1(NC(c2n(C)nnn2)c2cn(C3CCCC=C3Br)nn2)CC2CC1C1CCCC21 N1(C(CC(C=C)CCC)=O)CCC2CCN(C(C3CCCN3C=O)=O)CC12 C1(C(=O)NCCN(CCO)CC)CC(C)N1C(=O)C(C1CCCCC1)O C1(CNC(c2c(SC)snn2)=O)CN(C(c2cc(C)c(N)cn2)=O)CCCO1 C12(NC(=O)NCC3C(C)CCC3)CCC(CN(C(=O)OC(C)(C)C)C1)C2 C12(C(=O)NCCC(C)(C)NC(c3cocn3)=O)CC(CO)(C1)OC21CCC1 C(=O)(CC(O)C(C)C)N1C(CCNC(Cc2c(C)nc(C)s2)=O)CCC1 CC#CCC(C(=O)N(CC)OCC)NC(=O)C=Cc1cncn1C CC(N=c1[nH]c(=NCc2ccncc2Br)[nH]c2c1CSC2)c1cc[nH]n1 n1(CCCOC)nnnc1C(C1CCCO1)NCc1cnc(-c2cccnc2)s1 c1(CC(=O)N(C(C(F)(F)F)C2CC2)C2C(C(=O)OCC)COC2)ccc(C#N)cc1 C1(C(=O)NCCC(C)NC(=O)CC2CCOC2(C)C)(OC)CCCCCCC1 c1occc1Br.c1(C(=O)NC(CNC(C2(C)CC2)=O)C2CC2)csc(CC(F)(F)F)n1 C1(C(=O)NCC2C(NC(C(CNC(=O)OC)(C)C)=O)C2)CN2CCCN1CC2 c1(OC)cnc(C(F)(F)F)c(NS(=O)(=O)CC(C)C2CCCC2)c1 C1(NC(C2OCCN(CC)C2)=O)C2CC1CN(C(C1(OC)CCC1)=O)C2 C=CCC(CC)C(=O)N1CCC(N(C(=O)Cc2csc(CC)n2)CC)C1.C(C(C)(C)C)=C Cc1ccc(C(=O)N(C2CCN(C(=O)C(O)Cc3cnc[nH]3)C2)C)cc1 N1(C(c2c(OC)c(C)sc2)=O)C2CCCC1CN(C(C1CCN(C)C1=O)=O)CC2 C1(CNC(c2c(CC)scn2)=O)CCN(C(=O)COc2cncc(Cl)n2)CC1C C(C(=O)NCC1CCN(C(c2cnn(C)c2C2CC2)=O)C1)(C(C)(C)C)OC C1(C(=O)NCC(N2CCOCC2)=O)CSC2(c3ccccc3)CCC(=O)N12 c1(CNC(NCC(C)(C)C)=NCCN2CCCOCC2)cccc2c1CCCC2 N1(C(C2(C)C=CCC2)=O)CC(C2CN(C(c3nocc3Br)=O)C2)C1 c1(C(N(CCCNC(=O)C(F)OC(F)(F)F)C(C)C)=O)cc2cccn2cn1 Cc1sc(N)c(C(N2CCCCC(NC(=O)C(O)C(F)F)C2)=O)c1C c1(CN2CC(NC(c3cnc(C)nc3)=O)C(F)C2)ccc2c(c1)OCCO2 c1(CC(N2CCC(NC(CC)=O)C(C(C)C)C2)=O)nc2ccccc2s1 C(=O)(C1=CCCCCC1)N1CC(NC(C(C)Sc2c(OC)cccc2)=O)(CO)C1 N1(C(C2N(C(c3cc(F)cc(F)c3)=O)CCC2)=O)CC2CCN(CC34CC(C3)C4)C2C1 C1(C(=O)NCC2CCCN(C(c3n(C(C)C)nnc3)=O)C2)COC2(CCC2)C1 N1(C(CC#C)=O)CC2CN(C(=O)C(c3ccccc3)I)CC2C1 C1(C)(NC(c2cnc(CC)[nH]2)=O)CCN(C(=O)Cc2cccc(O)c2)C1 C12(CC(O)C1)C(=O)N2.C(=O)(CCC=CC(C)C)N(C)CC1CC(OC)C1 C1(N(C(CCSC)=O)C)CCN(C(c2cc(C#N)cs2)=O)CC12CC2 C(=O)(C1=NNC(=O)CC1)NCC(CNC(C1C(C)N(C)CC1)=O)C(F)(F)F C12(CCNC(C3CCC(NC(=O)CC(F)(F)F)CO3)=O)CC3CC(CC(C3)C1)C2 [N-]=[N+]=NC1CCCN(C(C(=O)NCCCc2cn[nH]c2)C2CCOC2)C1 c1(OC(C(=O)NC(C(=O)OCC)Cn2cc(C)cn2)C)ccc(NC)c(C)c1 C(CCC)(C(=O)N(CC(C)NC(=O)C(C(C)C)Sc1ccccc1)C)=CCC CC1CN(C(C2CC(=O)C23CCC3)=O)CC(C)CN1C(C1CCC(C)C(C)C1)=O C(=O)(CCCC(C)(C)CC)N1CC(NC(c2ccc(CC)[nH]2)=O)C(CC2CC2)C1 c1(C(CN(C)C(=O)NC2(O)COC2)O)cc(Cl)cc(Cl)c1 c1(C(=O)NC2(CCCNC(c3ccc(C(C)=O)[nH]3)=O)CC2)ccc(Cl)cc1C C1(NC(CC(C)c2nn[nH]n2)=O)C(C)(C)C1(C)C CC1OC2CCC1(C(N1CC(O)(CN(C)C(C3(C)CC4CC4C3)=O)C1)=O)C2 c1(C(C)C)cc(C(=O)NC2CCC2NC(C2(C#N)CC23CCC3)=O)ccc1F C1(NC(C2C(=O)NCC2)=O)C=CCN(C(C2CCCN(CC(F)(F)F)C2)=O)C1 C1(N(C(c2occ(C)c2)=O)C(c2ccno2)C)C2CCC1CNC2 Cn1ccc(C(=O)NCC(C)(C)CNC(C2(C)CC2Br)=O)c1 c1(C(CC)C)ccc(NC(N2CCN(c3cccc(O)c3)CC2)=O)cc1 Cc1cc(Cl)ccc1C(N1CC(N2CCCC2C2CCC(=O)CC2)C1)=O N(C1CCc2cccc3cccc1c23)CC1CCCCC(N)C1 N1(C(CC(=C)Br)=O)CC(CNC(=O)COc2cccc(C#N)c2)C2(CCC2)C1 C12(CNC(C(CC#C)C)=O)CCC(CNC(C3CC3c3cccs3)=O)(CC1)CO2 CC1(NC(c2cc(C(N)=O)c[nH]2)=O)CC(NC(=O)CCc2ccoc2)C1 c1(C(=O)NC2C(CNC(C(CC)N(C)C)=O)COC2)ccc(OC)c(Cl)c1 C1(CC(=O)N(C2CCC(CNC(c3c(C)c[nH]c3)=O)CC2)C)CC2(CCC2)CO1 c1(C(C)NC(=O)C(C)(C)n2cnnn2)ccc2c(c1)OC(C)(C)C2 C1(COC)(NC(=O)CCc2cccs2)CCN(C(c2ncccc2F)=O)C1 C(=O)(CCC(=O)N1CCOC(C2CCOCC2)C1)OCC C1(C(N(C)CC2CCCN2C)=O)CCCN(C(C2CNCC(F)C2)=O)CC1 c1(C(=O)NCCOCCN(C(=O)CC2(O)CCC2)C)onc2ccccc12 c1(COC)c(C(N2CC(CC(COC)NC(=O)C3=CCOC3)C2)=O)cnn1C c1(C(C(=O)NC(COC)CO)C)cn(C)nc1C CC(C(CO)NC(=O)CCn1ccnn1)NC(c1csc(CC(F)F)n1)=O C1(C)(C(N(CC=C)CCC)=O)CCCN(C(=O)C(C2CCOCC2)O)C1 c1(CC)ccccc1OCC(N1CC2CC2(CNC(C2(F)CCC2)=O)C1)=O Cc1c(C(N2CCC(CO)(NC(=O)CC(C)N3CCCC3=O)C2)=O)ccn1C CC1CC=CCC1C(=O)NCC(C)(C)CN(C)C(C1(O)CCC1)=O CCC(C)N=c1nc2c(ncn2C)c(NC(c2cn[nH]c2)C)[nH]1 C1(NC(CCOC(C)=O)=O)CCC(C)N(C(c2cc(C)c(C)[nH]2)=O)C1 CC(CN(C)C)N=c1[nH]c(=NCC2(C)CCCCC23CCC3)[nH]c2ccsc12 Cc1cc(F)sc1C(=O)NC1CC(C)(C(N2CCC(C#N)C2)=O)C1 c1(CC)nc(C(C)NC(C2(CNC(=O)Cn3cc(CCO)nn3)COC2)=O)n[nH]1 c1(C(N2CCC(N(C(=O)CCCCCF)CC#C)C2)=O)cc(C(C)C)ccc1F N1(C(c2cnc(CC)[nH]2)=O)CC2COCC2(C(=O)NC(CC)C(C)O)C1 Cc1sc(C(=O)NC(C2CCN(C(=O)Cn3ccnn3)CC2)C)nc1O C1(NC(C2CC(=C)C2)=O)CC(C(=O)NCC(c2ccccc2F)O)CC1O CC(C)C(C)(O)C(=O)N(C)CC1CN(C(C2CC(C3CC3)=NO2)=O)CCO1 C1(C(=O)NCCOCCNC(c2cc(C3CC3)on2)=O)CCCCC1O Cc1nn(CC(F)F)cc1C(=O)Nc1cn(C)c(C(=O)Nc2ccc(Br)nc2)n1 CC(C)C(C(=O)NCCN1CCC(F)CC1)N(C1CCCC1)C1CCC1 c1(C(=O)NC2C(CNC(c3cc(CC)c(C)s3)=O)C2)cc(Cl)c(OC)c(Cl)n1 N1(C(c2c(SC)cnn2C)=O)CCCN(C(c2ncnc3c2CCC3)=O)C(C)C1 Cn1c(O)nc(NCC2CCCCN(C(=O)C=Cc3cccc(Cl)c3)C2)cc1=O Cc1ncc(F)c(=NCC(C)(C)CNC(c2occc2C2CC2)=O)[nH]1 N1(C(C=CC(CC)=CC)=O)CCN(C2CCCN(C(C3CC3C3CCC3)=O)C2)CC1 Cc1ccc(CC(=O)NCC2CC(F)CN2C(=O)CC2CCC(F)(F)C2)c(C)c1 C1(NC(c2ccn(CC)c2C)=O)(CC)CCN(C(=O)COC2CCOCC2)CC1 N1(C(c2nccc(C)c2)=O)CC(O)(C2(CNC(c3c[nH]c(C#N)c3C)=O)CC2)C1 C1(OCCNC(c2c(N)non2)=O)CCN(C(=O)CCn2cnnn2)CC1 Cc1cc(C)c(C(=O)NCC2CCC(NC(C3(C)CCNC3=O)=O)CC2)[nH]1 N1(C(=O)CCc2nncs2)CC2(CCC2)CC1C(=O)NC1CN(CC2CC2)C1 c1(NC(C2CCC(NC(c3ccc(CCC)cc3)=O)CC2)=O)cc(Br)ccc1Cl CC1CCN(C(C2CCC(C)C2)=O)C1C(=O)N(C)CCc1ccccc1 C1(C(=O)NCC(N(C)C(c2ccccn2)=O)C2CC2)CCc2nncn2C1 N1(c2ccnc(COC)n2)CC2CCC1C(NC(=O)CCc1ccc(F)cc1)C2 CCC(C)CC(C(=O)NCC(=O)OCCOC)NC(C1OCCC1C)=O N1(Cc2ccc(NC(C)=O)cc2)CCN(S(=O)(=O)CC#N)C(C#N)C1 c1(OC)ncc(C(N2CCCC2(C)C(=O)NCCC2CCCN2C)=O)cc1F c1(C(=O)NC(CN(C(=O)CC2CCCOCC2)CC)C)ccc2ccsc2c1 CC(=O)C(C)CC(C)C(=O)NCC(O)CC(=O)Nc1cnccc1CO CC1CN(C(C2CC2c2ccco2)=O)CCC1NC(=O)CC(O)n1cccn1 C#CCC(C(=O)NCC(C)(COC)CO)NC(C=CC(=O)OCC)=O C1(C(CC)NC(=O)Cc2cc(-c3cccc(OC)c3)n[nH]2)(OC)CCOC(C)(C)C1 CC1CN(C(=O)C(=O)Nc2ncc(Cl)cc2Cl)CC1(F)F C12(C(=O)NC(c3nn[nH]n3)CC)CC(CN(C(=O)COC3(C)CCCC3)C1)C2 c1(NC(C(c2ccoc2)NC(C(CC)O)=O)=O)cn(C)nc1C#N CC(O)(CNC(=O)NC(c1ccc(C#N)cc1)CF)C(F)(F)F C1(C)(C(N(CCCCN(C(=O)COc2ccccc2Cl)C)C)=O)CCCS1(=O)=O N1(c2nnc(CC(C)C)s2)CCC(NC(C2CC(O)C2)=O)C(F)C1 CC1CC(C)N(C(C2CC(C)(F)C2)=O)CCN1C(c1ccc2scnc2c1)=O C(=O)(CCCC(=O)OC)N1CCC(N(CC=CC(=O)NC)CC)(CF)C1 N1(C(CCN(C)CC)=O)CC(NC(C2CN(C(=O)OC(C)(C)C)C2)=O)CC1(C)C C1(SCC)CN(C(=O)C(OC)OC)CCC1NC(=O)CCC1CCOCC1 c1(CC(=O)NC2(COC)CN(C(=O)CC3CCOC3)C2)ccc2c(cnn2C)c1 C12(CNC(c3cccc(C)n3)=O)CCCCC1N(C(c1csc(C)c1)=O)CC2 c1(OC)cc(CC(=O)NC2CN(C(=O)CC3CSC3)CC23CC3)ccc1O C(CCC(C)C(=O)N1CC2CC(C(N3CC(CSC)C3)=O)(C2)C1)OC c1(C(=O)NCCC(C)NC(=O)CC23COCC(C2)C3)ccnc(F)c1N C(=O)(C(C)(C)C(N)=O)NCCCCC1CN(C(CCC(=O)NCCC)=O)C1 C(=O)(C(O)C(C)C)NC1CC(OC)C1.C(C(CNC(C)=O)N(C)C)OC(C)C CCCCN(CC(=O)NCC)C.C(=O)(COCCOCC1CC1)OCC C1(NC(c2ccc(F)cc2C2CC2)=O)CCOC2(CCN(c3nnnn3C)CC2)C1 c1(CC(C(=O)NCC2(NC(c3cc(C)on3)=O)CCOC2)O)cccc(Cl)c1 N1(C(C(CC)C#N)=O)CC2CCCC(CNC(=O)CC3CC(O)C3(C)C)C2C1 N1(C(CN(C)C(N)=O)=O)CC2CCC(N(C)C(C3CCCN3N=O)=O)C2C1 CC1(C)CCCOC1CNC(=O)C(c1ccoc1)NC(C1(O)CCCCC1)=O c1(C(C)C(=O)NC2CC(O)(CNC(=O)CCS(C)=O)C2)ccc(F)cc1Br CCCC(C(=O)NCCC1(CNC(C2(c3cc[nH]n3)CCC2)=O)CCCC1)N(C)C c1(NC(N(C)CC2CC(OC)C23CCC3)=O)ccc2c(O)nnc(O)c2c1 C1(C(=O)NCC(CC=C)NC(=O)CCc2ccoc2)CCn2ccnc2C1 C(=O)(C1=NOC2(CCC2)C1)N(CCCCCNC(C1CCOC1C(F)(F)F)=O)C C=CC1(NC(C2CC(C)(C)CN2C(C2CCC=CCCC2)=O)=O)CCCCC1 c1(CCC(=O)NCCOCCC2CC2)ccc([N+](=O)[O-])cc1.C(=O)C(F)(F)C(F)F N1(C(c2ccc(CC)o2)=O)CCC(C)(CCNC(=O)C(c2cnn(C)c2)C)CC1 C1(CC(N2CCC(=CCC)C2)=O)CC(NC(=O)CC(C)n2cccn2)C1(C)C C(=O)(CCS(C)(=O)=O)N1CCCC(CN(C(C(c2cccc(Cl)c2)CC)=O)CC)C1 N1(C(C(n2cc(C(N3CC(SCC4CC4)C3)C)nn2)C)=O)CCC=CC1C(F)(F)F.CCO N1(C(C=CC)=O)CCCC(N(C(=O)Cc2nonc2C)C)CC1 c1(CN2CCC(=O)N(Cc3ccc(C)cc3C)C2)ccc(S(C)(=O)=O)o1 C1(NC(COCc2cc(C)on2)=O)C2CC1N(C(c1cn(C)nc1C(C)C)=O)C2 C(CCC(=O)N1CCCC1CN(C(c1cnnn1CC)=O)C1CC1)OCCC c1(C(=O)NC(c2cccnc2)C(=O)NCCC2C(C)C2)c(C#N)cnn1C N1(CC2CCC3(CC3)C2)CCN(C(=O)Nc2cccc(OC)c2)C(C)(C)C1 C1(C(=O)NCCCN(C(C2COCC2C)=O)CC)OCC2CCCC12 c1(C(CN)C)ccc(F)cc1.c1(N2C(=O)CNCCC2)ccc(F)cc1.CCO c1(CC(C)C)ccc(C(=O)NC2CC(CNC(=O)C(c3cncn3C)O)C2)cc1 C(=O)(CC1=NNC(=O)C1)NC1CCCN(C(C(C(C)C)c2cc(O)no2)=O)C1 C1(NC(c2c(C)ocn2)=O)CC2CCC1N(C(c1cc3c(s1)CCC3)=O)C2 C(=O)(CCCCN(C)C(C1CCN(C(c2cncnc2C)=O)C1)=O)OC C(=O)(N=c1cc(C(N)=O)n(C)[nH]1)C1C(CCC)CN(C(c2nn[nH]c2CC)=O)C1 Cc1oc(C(C)(C)C)cc1C(=O)NC(C)C(CO)NC(C1CC2C=CC1O2)=O C1(CC=C)CCCCC1(c1nnnn1CCSC)NCCNS(C)(=O)=O c1(C(N2CCN(C3CN(C(CC4C(C)(C)C4)=O)C3)CC2)=O)ccnc2[nH]nnc12 CCCCCC(O)C(=O)N(C(C)CCNC(c1cccc(CC)c1C)=O)C c1(CC(=O)NCC(C)NC(=O)CCn2ncn(C)c2=O)ccccc1C(F)(F)F c1(C(C)C(=O)Nc2ncc(I)s2)ccc(S(N)(=O)=O)cc1 c1(NC(=O)Nc2cccn2Cc2cccs2)ccc(F)nc1Br S(=O)(=O)(c1ccc(NCC2(CO)CC23CCC3)cc1Cl)NC1C(C)(C)C(F)(F)C1 c1(C(=O)NC(c2cn(Cc3c(OC)ccs3)nn2)C(C)C)cccc(C(C)=O)c1 C1(NC(CCc2ccn(C)n2)=O)CC2CC1CN2C(c1cc(C(F)(F)F)cs1)=O c1(C2CCN(C(CCNC(C(=O)OC)=O)Cc3ccccc3)C2)ccc(Br)cn1 C1(NC(c2n(CC)ncc2)=O)CCC2(CC1)CN(C(C1CC1C)=O)C2 c1(N2C3CC(CC)CC2CCC3)nc2ccccc2c(=NCc2cccs2)[nH]1 c1(N(C)C(=O)OC)ccc2c(c1)CN(CC(C1CCOC1)N(C)C)C2.C(C)(C)(C)O C(CC(C)(C)C#N)(c1n(CCCC)nnn1)NC1CC1Cc1ccccc1OC n1(CC)cnc2nc(=NCC3(C(C)C)CC3)[nH]c(NCCCS(N)(=O)=O)c12 c1(CC)cc(C(=O)NC(CO)C(=O)NC2CCCN(C3CC3)C2)n(C)n1 C1(NC(C2(C(F)F)CC(=C)C2)=O)CCCC(C(=O)NCCN(CC2CC2)CC)C1 c1(C(=O)NCC(=O)NCC(=O)NCC(CC)n2cccn2)ccc(Cl)o1 c1(CCC=C)ccc(C(=O)NCC2(C)CC(NC(=O)CCOC3CC3)C2)cc1 N1(C(=O)NCCC2CCCCO2)CCCC(N2CCC(O)CC2)CC1 CC(C)(CCC(=O)N1CC(CO)(NC(C2CCCC3CCCN23)=O)C1)[N+](=O)[O-] c1(C(N(C2CCCN(C(C3CCCCO3)=O)C2)C)=O)cnn2ccncc12 c1(C(N2C(CN(C(C(C)=C3CCC3)=O)C)CC(F)C2)=O)c[nH]cc(F)c1=O C1(C)(CC(=O)NCCC2(CC)CCC2)CCN(C(=O)CC2CC=CCC2)C1 c1(C(=O)NCC2(C(C)NC(=O)CCc3cnn[nH]3)CC2)cc(S(N)(=O)=O)c[nH]1 C#CC1(C(=O)NC2(CCOC)CC2)CCN(C(c2cnnc(C)c2)=O)CC1 C(CCCCNC(c1cnn(C(F)F)c1)=O)N(C)CC.C1(=O)C(C2CC2)N1 N1(C(C2N(CC)CCOC2)=O)CC(NC(c2cccc(CCO)c2)=O)C2(CC2)C1 C1(C(N(CC(CN(C(C=CCC)=O)C)O)C)=O)CCOC1C c1(C(CN(C(=O)NC(c2n(CC)ncc2)C)CC)C)ccc(NC)cc1 c1(OC)ccc(OCC(N2CC(NC(=O)C(C)(F)F)C(C(F)(F)F)C2)=O)cc1 C1(SC)CN(C(=O)CC2C(C)C2(F)F)CC1NC(c1cc(C(F)F)[nH]n1)=O Nc1c(F)cc(OCC(=O)NC2CC3CCC(C2)N3)cc1Br c12ccc([N+](=O)[O-])c(c1)C(=O)NCCCN(C(C1CC1F)=O)C2.CC(C)(C)C c1(CC(=O)NCCCN(CCCCNC(=O)C(F)C2CCOC2)C)ccnnc1 Cc1coc2c(NC(=O)C(=O)NCC3CCC4CC34)cccc12 Cc1cc([N+](=O)[O-])ccc1C(=O)NCCC1CCN(C(c2cnn(C)c2F)=O)C1 Cc1ccc2c(c1)CCC2NC(=O)CCC1(C)CCN(C(=O)OC(C)(C)C)C1 c1(-c2cccc(OC)c2F)cccc2[nH]cc(C(=O)NC(C3CCCCC3)C)c12 Cc1ccc(CCC(=O)NC2CCN(C(=O)CCc3ccon3)CC2C)c(C)c1 C(=O)(C(O)C1=CCCCC1)N1CCC(NC(c2ccc(C(F)F)s2)=O)C(F)C1 N1(C(CC(C)O)=O)CC2(C=C(C(=O)N(CCN=[N+]=[N-])C)CO2)C1 C(CCCCC(=O)NC1CCCC1NC(C1(NC2CCC2)CC1)=O)OC C(C(COC)CC(=O)NCC1CCN1C(c1scnc1C(F)(F)F)=O)OC CCCCC(=O)C(=O)NCCOCCN(C(=O)C(C(C)C)n1cnnn1)C N(C(=NCCCF)NC1COCC1F)CC(CCN(C)C)OCC c1(C(C)C(=O)NCC(CC(=O)O)C2CCCC2)ccc(F)cc1Br N1(C(CC2(C(=O)OC)CC2NC(=O)CN2CCCC2C)=O)CCCC2OCCC2C1 c1(CNC(=O)NCC(C2CCCCCC2)C)cnn2c1NCC2 c1(SC)ncc(N)c(C(N2C3CCC2C(NC(=O)C=Cc2ccco2)C3)=O)n1 C(=O)(C1=CCCS1)NC(c1ccccc1)CNC(C1(OCC)CCC1)=O CC1=C(C)CN(C(=O)CC2CCN2C(C2CC(N3CCCCC3)C2)=O)C1 c1(C(N2C(C)CC(NC(=O)CCC3(C)CC3(F)F)CC2)=O)ccc(F)c(F)c1F C(=O)(C(CC(F)F)N(C)C(C1CCC(C2CC2)C1)=O)N(C1CCCCC1)CC#C C1(C)(C)C(C)CC(=O)N1.CCCC(CNC(=O)CSCC)CCO N1(C(C(C)S)=O)CCC2(CC1)CC(C(=O)NC(C)C#N)=NO2 CC(C)CC(CNC(C1CCC1C)=O)C(=O)N(C)CC1CC1(F)F n1(CC)cnnc1CNC(c1sccc1CNC(C12CSCC1C2)=O)=O C1(C(N(C)Cc2cc(C)no2)=O)CN(C(=O)CC2CCC(C)(C)C2)C(C)(C)C1 C1(C(N(CCNC(c2cnc(C)nc2)=O)C2CC2)=O)CC2COCC(C1)C2 CON(C)C1CCN(C(=O)CC2CCCN(C(=O)CN3C(C)CCC3C)C2)CC1 C1(C(N2CCC2CNC(C23CCCCC2OCC3)=O)=O)CCn2nccc2C1 C#Cc1ccc(CC(N2CC(CCNC(=O)Cn3cnc(=N)[nH]3)(OC)C2)=O)cc1 Cc1cc(C(=O)NC2CC(CCNC(=O)C(C)(C)CC(C)C)C2)c2n[nH]cc2c1 c1(C(N2CCCC3(CC(O)C3)C2)C(=O)NC(CC)(C)C)cc(Cl)c2c(c1)OCO2 N1(C(c2c(C)nns2)=O)CC2CC1CN2c1ncns1 c1(NC(N2CCC(c3snc(N(C)C)n3)CC2)=O)cc(Br)c(F)cc1C C1(C(=O)Nc2c(-c3cn(CCF)nc3)nccc2)CCc2cc(F)ccc2O1 C1(C(=O)NC(CN(C(CSCC(=O)OC)=O)C)C)SCC=C1C C12CCCCN1C(=O)c1c[nH]c(c1)C(=O)N2.N1(C(C)(C)C)CCC(C(C)(C)C)C1 CCC(C(=O)NCC1COCCN1C(c1cc(C(F)(F)F)nc(Cl)c1)=O)C(C)C C1(C(=O)NC2CCN(N3CCC3)C2)CCN(C(C2(Cl)CC2(F)F)=O)CC1 Cc1c(Br)cc(C(=O)NC2CC(C)N(C(c3ccccc3Cl)=O)C2)cc1Br Cc1ccc2c(c1)CC(C(N1CCC(CNC(c3cncc(O)c3Cl)=O)C1)=O)S2 N1(C(CC)=O)CC2CC(NC(=O)C(C(C)(C)C)c3ccc(C)c(C)c3)C(C2)C1 N1(C(C(CC)NC(C)=O)=O)CCC(C(=O)N(CCCCCO)C)(CC)C1 CN1CCN(C(=O)C(C(C)(C)C)CNC(=O)CCC2OCCO2)C(C(C)(C)C)C1 C(C1=NOC2CN(C(c3c(C)noc3C)=O)CC12)NC(c1cc(C)nc(Cl)c1)=O CCCC(O)CC(=O)NCCC1(NC(C2CC=CCO2)=O)CC1 n1(C(C(=O)NCC2CN(C(C(CCC)C#N)=O)C2)C)nc(C)c([N+](=O)[O-])c1C Cc1ccc(CN2CCC(NC(c3ccc(C(C)(C)C)cc3O)=O)C2)c(O)c1 c1(C(N2CCCC(C(=O)NC)C2)=O)ccc2c(c1)C(CC=O)C(=O)N2 c1(-c2c(C)csc2)cc2c(C(=O)N(C)CCO)nccn2c1 CC(CCCCNC(=O)COC1CCCC1)NC(=O)C(C)OCOC C1(C)(C(=O)NCC23CC(NC(C(C)(Cl)Cl)=O)(C2)C3)CCC(=O)N1 N1(C(c2cn(C)nc2Cl)=O)CCN(CCNC(C23CC(F)(C2)C3)=O)C2(CCC2)C1 C1(OC)CC(CNC(=O)Cc2ncccc2C)N(C(C2CNC(=O)N2C)=O)C1 N1(C(c2c(C(=O)OC3C(OC(C)=O)C3)c[nH]n2)=O)CCC2C(NC(C)(C)C)CC12 c1(C(N2C(CNC(c3cn4ccnc4s3)=O)CCCC2)=O)cc([N+](=O)[O-])sn1 C(=O)(C#CC(C)(C)C)NC1(CC=C)CCN(C(=O)CN2CCC(OCC)C2)C1 c1(NC)ccc(C(N2CCC(F)(CNC(=O)CCc3ccnc(C)n3)C2)=O)cc1 c1(C(C(N2CCC(CC(=O)NC3CC4CCC3C4)C2)=O)O)ccc(F)cc1 c1(CC(=O)N(CCCCN(C(=O)CCn2cncn2)C)C)ccc(F)cc1 C1(F)(CNC(C2(CC=C)CC2)=O)CCCN(C(c2ccc(F)cc2O)=O)CC1 Cc1cnc(NCCSCc2ccc(F)cc2)c(S(=O)(=O)NC2(C)CCCC2)c1 Cc1cc(COC)oc1C(=O)NC1CCCC1NC(=O)CC1CCN(C)C1=O c1(C(N2C(CNC(C(C(C)C)C(C)C)=O)CCC2)=O)cnc2c(c1)NC(=O)CS2 Cc1cc(CCNC(c2nnnn2CC(F)F)CCC2CCCCCC2)ccc1F c1(OC)cc(NC(=O)C(N2CC=CC(C(=O)OC(C)(C)C)C2)=O)nc(Cl)c1 C(=O)(C(CO)C(F)(F)F)N(C(C)C)CCN(C)C(C1CCCC(=O)CC1)=O C12(C(=O)NC3C(C)CN(C(C4(C)COC4)=O)C3)CCC(C#N)(CC1)CC2 C1(C)(C2(CNC3(c4nnnn4C)CN(C(=O)OC(C)(C)C)C3)CC2)COCCO1 C1(C2CCCO2)(C(N(CCC(C)NC(c2ccc(C#N)s2)=O)C)=O)CCCCC1 C1(CCNC(=O)C(=O)NCC(C2CCCCC2)NC(N)=O)CC1C1CC1 c1(C(=O)NC2CC(N(C(c3c(C)nc(C(C)OC)s3)=O)C)C2)cc(C)nc(O)c1 N1(C(c2cncc(C#C)c2)C(=O)Nc2ccccc2C)CCCC2CC(O)CCC12 S(=O)(=O)(c1ccccc1C(N1CCN(C(=O)NC2CCCCC2)CC1C)=O)NCC N1(C(c2cn(CCNc3ccc(C(=O)OC)s3)nc2)=O)CCC(C)(C)C1C C(CNC(C1CC(C(C)C)C1)=O)(CC(F)(F)F)NC(c1ccc(OCC)nc1)=O c1(CC=CCNC(C(=O)NC(c2cccc(C)c2)CC)=O)ccccc1Cl C(=O)(C(C)CC(C)CC)N1CCC(CC=C)(NC(C2CCCC(O)C2)=O)CC1 C1(C(=O)Nc2c[nH]nc2Cl)COCCC12CN(Cc1ccnc(Cl)c1Br)C2 N1(CC)N=C(C(=O)N2CCc3nn(C)c(=O)cc3C2)Cc2ccccc21 CCCC(CNC(c1ccncc1NC)=O)C(=O)NCC(O)CC(C)(C)C c1([SH](CC(=O)NCCC(O)CNC(c2ccncc2)=O)C)ccc(OCCF)cc1 C=C(C)c1ccccc1N(C(=O)C(C)(O)C(F)(F)F)C(=O)CCCN1CCCC1 C1(OC)CC(CNC(c2ccc(CC(N)=O)cc2)=O)N(C(c2cnc(C)s2)=O)C1 O=C(C1=CCOC1)NCC(c1ccccc1)CNC(c1cscc1Cl)=O c1(NC(C2CC3CC3N2Cc2ccnc(O)c2)=O)cccc(CC(F)(F)F)c1 C1(C(=O)NC(C)CC(O)NC(C2CC3(C2)CC32CCC2)=O)CCc2nncn2C1 C(CS(=O)(=O)CCN=c1ccc(Br)c(S(=O)(=O)N2CCCS(=O)(=O)CC2)[nH]1)OC c1(C(N(CC(CNC(CCCOCCC)=O)O)C)=O)cncc(C(C)(F)F)c1 C12(NC(c3c(COC)cccc3)=O)CCC(CN(C(c3ncc[nH]c3=O)=O)C1)C2 C(=O)(C1=CNS(=O)(=O)N=C1C)NC1CC(NC(C(C)N(CCC)C(C)=O)=O)C1 c1(C(N2CCC(CO)(NC(=O)COC3CCCOC3)C2)=O)cncc(C(F)F)c1 C1(O)(C(C(=O)NCC2(C(N(C(C)C(=O)OC)CC)=O)CCC2)F)CCCC1 Cc1cnc(CCNC2CCOC2C)c(C)c1 C1(C(=O)NC(=O)CCC2CCCC2)CCC(C)CO1.C1CC(CCCOC(C)=O)N1 CC(C)(C)C(C(=O)Nc1cnn(C2CCCCCC2)c1)Sc1cc(Cl)ccc1F C1(NC(C(C)N(C)C)=O)CN(C(c2nnn3c2COCC3)=O)Cc2nccn2C1 c1(C(N(CC(C)N(C(=O)COCc2ccc(Cl)cc2)C)C)=O)cc(O)ncc1F CC(CC(C)(C)C)C(=O)NC1CC2CC(NC(C3(CF)CC4(CCC4)C3)=O)C2C1 c1(C(C)=O)cc(NC(=O)C(=O)NC(C2CCCO2)C)ccc1C C1(SC)CN(C(c2ncnn2C)=O)CC1NC(=O)C(C)(C)Cc1cnn[nH]1 c1(SCC(=O)NC(CCCCNC(C2(C#C)CCC2)=O)C)ccc(F)cc1F C1(F)(C(=O)NCC(C)CC2CCCC2)CCCN(C(c2ccccc2CO)=O)C1 c1(NC(N2CCCC(CN(CC)CC)CC2)=O)ccc2nc(Cl)nn2c1 C1(CC)CN(C(=O)C(F)(F)c2csc(=N)[nH]2)CCC1NC(=O)C(C)C1CCC1 C1(CNC(C(CCCCC)O)=O)CCCC12CCN(C(c1ncoc1C)=O)CC2 C1(CC(=O)NCC2(NC(C(CC=C)(C)C)=O)CCOC2)CSc2ccccc2O1 Cc1nc(CC(C)C)sc1C(N1CC(C(C)NC(=O)C(O)c2ccco2)C1)=O c1(NC(c2n(CC=C)nnn2)(C)CC2CCCO2)ccc(CC)c(Cl)c1 c1(C(N2CC=CC(NC(CSCC(N)=O)=O)C2)=O)nnn2c1CCCC2 C1(C(N2CC(CNC(C3C4CC5C(C4)C35)=O)OCC2)=O)CC2(C1)CC1(CCC1)C2 C1(C(C)C)N(CC(c2ccccc2)O)CC12CCOCC2 c1(C(N(C2CCCN(C(C3(C=C)CCC3)=O)C2)CC)=O)ccc(C)nc1OC c1(C(N(C)CC2CCCN(C(CCCOCC=C)=O)C2)=O)cnc(OC)c(F)c1 C(=O)(C(O)CCC(C)C)N1C(CC)CN(C(c2ccnc(S)c2)=O)CC1 N1(C(c2c(C)nncc2)=O)CC(NC(c2csnc2C)=O)CC(C)C1 c1(CCN=C(NC(C=C)C)NCC(C2CC2)OC)ccc2c(c1)CCN2C CC1CCNC(=O)C1CNC(=O)CN(C)C(C12CC(F)(C1)C2)=O C=CCCC(C)C(C(=O)Nc1nnn(C)n1)N1CCN(CC(F)(F)F)C(C)C1.OCC CC1(C)C(NC(c2nc(F)ccc2Cl)=O)CCN1C(=O)CC1OCCO1 CC(=O)CCC(=O)N1CC2CC1(C(N1CC(OC(=N)O)C1)=O)C2 N1(C(C2CC(F)(F)C2)=O)CCN(C(=O)C=Cc2cnc[nH]2)C(c2cccnc2)C1 C(C(C)(C)CC(=O)NCC(C1CCCN1C(C1CCCCCCC1)=O)(C)C)OC c1(OCC)cc(Br)cc(C(N2CC3CC2CN3Cc2ccccn2)=O)c1N C1(C(F)(F)F)(C(=O)NCCN(CC(C)O)C(C2CC2[N+](=O)[O-])=O)CC(C)(C)C1 c1(C(N2C(CNC(C(c3c(C)noc3C)C)=O)CC2)=O)cc(N)nc(Cl)c1 Cc1ncc(Br)c(C(N2CC(CC(=O)Nc3cccc(C#N)n3)C2)=O)n1 N1(CC2CCCC(C)C2)CCC(C(=O)Nc2nccc(Cl)c2I)C(O)C1 c1(NC(C(c2cccs2)N(CCOC)C)=O)cncnc1.C1CC(=O)NC12CC2 CC(F)(F)C(C)(C)CNC(=O)C(O)CCNC(c1nnc(O)nc1O)=O N1(C(c2c(F)ccc(C)c2Cl)=O)CCC2(CCCC2C(=O)Nc2ccns2)C1 c1(C(=O)NC2C(NC(C=Cc3cn(C)nc3)=O)CCC2)ccc(=O)n(C)c1 C1(NC(C(CC)OC)=O)(CNC(=O)CC2(OC)CC2)CCCC1C Cc1nc(N2CCC(C(C)(C)C)(CNC(C3CC3F)=O)C2)c2scc(C)c2n1 C=CC1CN(C(C2(C)CC2)=O)CC1NC(C1CC(n2cnnc2)C1)=O c1(CC(=O)OCC)cccc(C(=O)Nc2cn(-c3cccc(C(N)=O)c3)nn2)c1 C1(NC(CCCC=C)=O)CC(C)CN(C(=O)Cc2ccc(F)cc2C)C1 CC1CN(C(=O)COCCF)CCC1N(C(=O)C(=O)Nc1ncccn1)C Cc1sc(C)c2sc(C(=O)NC3CC3NC(=O)Cc3cncn3C)cc12 c1(C(=O)NCC2OCCC(NC(C=C(C)Cl)=O)C2)oc2ccc(F)cc2c1C C(=O)(C(CC1CC1)OC)NC(C)C(C1CC1)NC(C=CC(=O)NCCCC)=O C1(COC)CN(C(=O)CCOCc2cccnc2)CCN1C(=O)C(F)OC C1(NC(C2CC(=O)NC2)=O)CCN(C(c2csc(C3CC3)n2)=O)C12CCCC2 n1(CC(=O)NC(C2(O)CCN(C(C3CC3F)=O)C2)C)ccccc1=O N1(C(C(COC)O)=O)CCN2CCOCC2(CNC(c2cccc(F)c2F)=O)C1 C1(C(C)C)CCCCC1N=c1nc(N(CCO)Cc2cnc[nH]2)c2[nH]ccc2[nH]1 O(C1CCCc2cccnc21)Cc1c(C)n(Cc2ccc(F)cc2)nn1 N1(C(C2C(NC(CNC(=O)OCC)=O)COC2)=O)CC2CCCC12 CC1(C)CCC(CN(c2nnc(-c3ccccn3)n2Cc2ccccc2)C)CC1 c1(C(N2CCC(C(=O)NCc3c(C)noc3)C2)=O)ccc(SC(F)(F)F)nc1 C1(NC(=O)C(O)Cc2ccccc2)CC(CO)N(C(C2CC(Cl)(Cl)C2)=O)C1 c1(NC(C2C(C(=O)NC(c3cccc(Cl)c3)COC)C2)=O)cc2cn[nH]c2cn1 Cc1ccc(C)c(NC(=O)NC2(C)CCN(C(=O)C(C)(F)F)CC2)c1 c1(C(N(CC(CN(C(c2c(C)c[nH]c2)=O)C)O)C)=O)ccc(F)c2occc12 CC1(F)CCCN(C(C2CC23CC(NC(=O)CC2C=CCC2)C3)=O)C1 C(=O)(C(C)(C)C(C)O)NC1CCC(CNC(c2cc(C(=O)OC)no2)=O)CC1 C12(C(N3CC(C)(CNC(CCSCCC)=O)C(C)C3)=O)CC3CC(CC(C3)C1)C2 C#Cc1cncc(C(N2CCC(CO)C(NC(c3ccnc(CC)c3)=O)C2)=O)c1 c1(C(CC)N(C(=O)CCCC2CCCO2)CC)ncc(C)[nH]1.C12CC(C1)NC(=O)C2 Cc1nc(C(N2CCOC(CN(C)C(c3ncccn3)=O)C2)=O)c2ccnc-2[nH]1 c1(-c2ccccc2)nocc1.CC(C(=O)NC1(CCNC=O)CC1)OCC1CC1 C1(C(=O)NC(CCC)C(N)=O)N(C(=O)C=CC(C)(C)C)CCC1(C)C C1(NC(=O)CCC2CCCCCC2)CC2CN(C(=O)Cn3ncnn3)CC2C1 C(C(F)(F)C(F)F)CCC(N1C(CNC(C(N2CCN(C)CC2)C)=O)CC1)=O C1(CC(=O)N(C)CCN(C(=O)Cn2cnc(C#N)n2)C)CCCCC1(C)C C1(N(S(=O)(=O)c2cn[nH]c2)c2ncc(CC)s2)CC2CCCC(C1)N2 CCCCC(=O)C(=O)NOC(=O)C(C)N1CCOC(C(C)(C)O)C1 N1(C(CNC(CC(C)C)=O)=O)CCC(CNC(=O)C(C2CCOCC2)C)C1C Cc1ccc(C2C(C(N3CC(F)CC3NC(CNS(C)(=O)=O)=O)=O)C2)cc1 CC1CC(NC(=O)C(F)C(C)(F)F)CCN1C(C1CC2(CSC2)C1)=O C(=O)(C1=CCCC(C)(C)C1)N1C(C)CCC(C(N2CCOC(CCF)C2)=O)C1 c1(C(=O)NC2(CNC(CCC=C)=O)CCOCC2)n[nH]c2c1CC1CC21 N1(C(Cc2cc(OC)c(F)cc2)=O)CC(C2CN(C(C3(CF)CC3(F)F)=O)C2)C1 C(C)(C)(CCC(=O)NC(C(C)NC(=O)Cc1cc(F)cc(Cl)c1)C(C)C)OC C1(O)(C(=O)NCCCN(C)C)CCN(Cc2ccc(Cl)o2)CC1 C(N=c1[nH]c(NC2CC2C2CC2)nc2ccsc12)C1CC(C)(C)OC1(C)C C=C(C)CC(C(=O)OC)NC(=O)C(C1CCN(C(c2csnc2C)=O)CC1)C Cc1ncc(Cl)c(C(N2CCC(C(C)(C)NC(=O)C=Cc3nccs3)C2)=O)n1 c1(C(=O)NCCCC(C)NC(C(=C(C)C2CC2)F)=O)cnc2sccn12 C1(CC(=O)N(C2CCN(C(=O)CC3(C)CC3)C2)CC#C)CC2CCC1C2 O=S(=O)(c1cccnc1NCc1ccc(F)cc1)NCc1cn2ccccc2n1 N1(C(=O)N(C2CCNCC2)C2CC2)CCCCC12CCC(F)(F)CC2 CCC(C(C)CN(C)C1CC1)NC(=O)CCN(CCCO)C(C1CCCC1)=O c1(C(N2C(CNC(CC(C)SC)=O)CC2)=O)ccc(-n2ccnc2)c(F)c1 C1(c2cccc(OC)c2)CN(C(=O)C(O)C(F)(F)F)CCC1O Cc1ccc(C#N)cc1NC(C1(F)CCN(C(=O)CCc2ccc(F)cc2)C1)=O C1(C(=O)NCC2CC[Si](C)(C)C2)N(C(=O)CCc2cscn2)CC12CCCC2 c1(NC(CC)=O)cccc(C(N2CCC(Cn3cc(CCO)nn3)C2)=O)c1 CC(=O)CC(C)(C)CC(=O)NC1CCCC(CNC(C2CCCC2(C)C)=O)C1 c1(C(=O)NC(c2nocc2C(=O)NCC2CC3CCC3C2)C)c[nH]nc1[N+](=O)[O-] C1(F)(C(=O)NCC(F)(F)F)CCCN(C(=O)C(=O)NCC2CC2)C1 N1(C(C(C)C2CC2)=O)CCN(C(=O)C(N)=O)C(OC(=O)OC(C)(C)C)C1 c12nc(n(-c3ccc(Sc4ncc(F)cn4)cc3)n1)C2.C1(C)(C(C)OCC)CC1 C1(NC(C(C(C)NC(=O)C2=CCCSC2)C)=O)CCn2cnnc2C1 c1(CCC)cc(C(=O)NC2(C)CC(NC(c3c[nH]c(Br)c3)=O)C2)ccn1 C1(C(N2CC(CC(=O)OC)C2)=O)CC(O)CN1C(c1csc(O)n1)=O N(C(=NCCC(C)(O)C(F)(F)F)NCc1nc[nH]n1)C(COCC)C(=O)OCC Cc1cc(COCC(N2CCN(C(=O)Cc3cc(C)ns3)CC2)=O)n(C)n1 CC(C)(C)C(O)CC(=O)N1CC(CCc2cn(C3CCCNC3=O)nn2)C1 CC(CC(N)=O)C(=O)N1CCC(NC(=O)CC2(N3CCCC3)CC2)C(F)C1 C1(NC(c2ccc[n+]([O-])c2)=O)CCCC(C(=O)Nc2cnns2)CC1 c1(C(N(CC(CC)NC(C2CC=CCC2)=O)C)=O)cc(Br)c2c(c1)CCO2 C12(NC(=O)CSCC(F)F)CCCC1N(C(=O)C(c1ccccc1)C1CC1)CC2 C1(CNC(C(C(CC)C)OC)=O)CC2CCC1N(C(C1(C#N)CC1(C)C)=O)C2 C12(CNC(CC(COC)C)=O)CN(C(=O)CCCSC)CC1CCO2 C12CCN(C1)C(=O)C1CC(C)(C1)C(=O)C(=O)C1(CC1)NC2=O.CCN.OCC C1(C(N2CCCCC2)=O)(NC(C2CC(Cl)(Cl)C2)=O)CCCCC1 C(=O)(CC(C)(C)CC(=O)N1CCC(Oc2cccc(OCC)c2)C1)C(=O)C=CS(C)=O Cn1ncc2c1CCC(C(=O)NCC1CC(NC(c3nn[nH]c3Cl)=O)C1)C2 C1(CNC(C2CCN(C)C2=O)=O)CN(C(=O)CCn2cccnc2=O)CCCO1 CN1CCN(C)C(CNC(=O)CC(C(F)F)NC(c2cnn(C(F)F)c2)=O)C1 c1(C(N2CC3C(NC(CC(C)(C)CC(F)F)=O)(C3)C2)=O)ccc2cccnc2n1 N(C1CSc2ccc(Br)cc21)C(N(CC=C)Cc1ccccc1Br)=O c1(C(=O)NC(CNC(CCCC(C)=O)=O)C(C)(C)C)cc2c(nc1O)CCC2 c1(C(=O)NC2C(CC)CN(C(=O)C=CC(=O)N(C)C)CC2)c(C)nc(C)nc1C C(=O)(C(F)(F)C(F)(F)F)N(CCC(C(C)C)NC(C1CC(C)(C)OC1(C)C)=O)C N1(C(C=CCC)=O)CCC(C)N(C(=O)C(c2ncc(Cl)n2C)(F)F)CC1 c1(C(=O)NCC2CC(O)(CNC(=O)C(c3ccccc3)F)C2)cccc[n+]1[O-] N1(C(CC(C)CC(F)(F)F)=O)CC2(C1)CN(C(=O)C(F)(F)C(C)(C)O)CCO2 C(=O)(CS(=O)(=O)CCO)N1C(CNC(=O)C=Cc2cncc(O)c2)CCC1 c1(OCC)ccc(C(=O)NC(C)CC(C)NC(c2cnc(Cl)[nH]2)=O)cc1C c1(C(=O)NC(CCC)CNC(=O)CC2CSCCO2)cc(N)ccc1O C1(OC)CC(CNC(C2CC3(CSC3)C2)=O)N(C(=O)CCc2cnn(C)n2)C1 C1(C)(CC)CCCN(C(c2sccc2CNC(c2cccn2C)=O)=O)C1 C1(NC(c2cc(C)ns2)=O)CN(C(=O)C(C(C)O)N(C)C)CC1C(F)F C(=O)(C1=Cc2ccccc2OC1C(F)(F)F)N1CCC(Oc2ccc(C)cn2)C1 N1(C(c2c(C)oc(C3CC3)n2)=O)CC(C)(C)OC2(C1)CN(C(=O)CC(C)C)C2 N1(C(C=CC(C)(C)C)=O)CC2CCC1CN2C(=O)C#CC1CCC1 c12cc(OC)ccc1OC1CC1CNC2C.c1(CCC(=O)OC)nnc(C)o1 c1(SC)cc(C)c(C(=O)N(C2C3CN(C(c4coc(C#N)c4)=O)CC23)C)o1 c1(OCC(=O)NC(CC=C)CNC(=O)CN(C2CCC2)C)ccccc1[N+](=O)[O-] N1(C(C(c2cn(C)nc2)O)=O)CC2CC(NC(c3cccs3)=O)CC2C1 C1(C)(C(N2CC(CNC(c3c(C)nc[nH]3)=O)C(O)C2)=O)Cc2ccccc2C1 C(=O)(CCCCCCNC(=O)CCS(N)(=O)=O)N(C1CS(=O)(=O)C1(C)C)C C12CC(C13CCC3)C(=O)NC1(CCC1)CC(=O)N2.c1(COC)cnn(CCF)c1 C1(CCN(C(CSCCN(C)C)=O)C2CC2)CCN(C(C2CC2[N+](=O)[O-])=O)CC1 c1(N(C)CC2CCCN(C(c3ccc(OC)nc3)=O)C2)nc2ccc(N)cc2s1 c1(CC(=O)NC2C(NC(CC(C)SC)=O)C2)cc(Cl)ccc1Br c1(C2(CSC)CC2)ccc(N(C2CCN(C(CN(C(CC)C)C)=O)C2)C)c(F)c1 C1(C(=O)NC(C)CC2CCN(C(=O)OCC(C)(C)CO)CC2)CCC2(CC1)CC2 C#Cc1ccccc1CC(=O)NCC(CO)NC(=O)CC1CCCCC(=O)N1 C1(NC(c2cc(Cl)cs2)=O)CC2CC(NC(c3cc(=O)cc[nH]3)=O)C2C1 C1(N(C(C(CC)OC)=O)C)CCCCC1NC(c1csc(-c2cnn(C)c2)n1)=O C1(NC(c2ccn(CCCC)n2)=O)CCC12CN(C(C13C=CC(CC1)C3)=O)C2 C(CCN=C(NCC1(C)CCC(=O)NC1)NCC(c1cccc(C)c1)(F)F)SC CC(CCCCNC(=O)CCC(F)F)NC(c1coc(C2CCCCC2)n1)=O C1(NC(C2CCCOC2)=O)CN(C(=O)CC2CCCCC2O)C2CCCCC12 CC1C2CC(C2NC(=O)CCC2NC(=O)NC2=O)N1C(=O)CC=C(Cl)Cl Cc1cc(C(N)=O)c(NC(C2CCN(C(c3oncc3C)=O)CC2)=O)s1 CCC(CC(C)CO)Nc1cc(-n2nc(C)nn2)ccc1OCCN1CCCS1(=O)=O N1(C(C2CC(C)C2)=O)C2CCC1CC(CNC(C1CCc3ccnn3C1)=O)C2 N1(C(c2csc(O)n2)=O)CC(F)(F)CC1CCNC(C1(n2cnnn2)CC1)=O c1(C(N2CC3C(CNC(c4c(C)nc(C)o4)=O)(C3)C2)=O)cccn2c(O)nnc12 c1(OCCN(CCCNC(COC)=O)C(C2CC2(C)CCOC)=O)ccccc1 N1(C(C(COC)(C)C)=O)CCC(O)C(C(=O)NCC(O)CCl)C1 CCCCCC(CC)C(=O)NC1CC(CNC(c2ccc(C3COC3)cc2)=O)C1 C=C1CCC(CNC(=O)Nc2ccc(-c3cccc(Cl)n3)cc2)CC1 C1(C(=O)NCC(C)CNC(c2cccc(CC3CCC3)c2)=O)CCCCC(=O)N1 c1(N2C(C)CCC(NC(C3(C(F)F)CCCCC3)=O)C2)ncnc2c1nnn2C C(C(CC(C)C)C(=O)NC(c1csc(C)n1)C)NC(C1(CCC=C)CC1)=O c1(C(CNC(C2N(CC)CC2)=O)NC(=O)CS(N)(=O)=O)cc(F)cc(Cl)c1 C=CCC(CC)C(=O)NCC1CCN(C(=O)CCc2nc(=N)[nH][nH]2)C1(C)C CC1CCC(C)(CNC(C2CCCN2C=O)=O)C1.C1C=CCN(C(N)=O)C1 Cc1cncn1CC(=O)NCC1(NC(=O)CC2CCCO2)CCCC1 C1(NCC(=O)Oc2cnccn2)CS(=O)(=O)CC12CC2 c1(C(=O)NC2C(C)CN(Cc3cccc(C(F)(F)F)c3)C2)ccc(I)c(F)c1F CCCCC(CC(=O)NCc1cn(C2CC2)cn1)NC(=O)C(C)(C)CCC CC1CC(CC(=O)NC2CC(CNC(=O)C(F)=CC3CC3)C2)C(C)O1 N1(C(N(S(CC)(=O)=O)C)=O)CCC(c2nnnn2Cc2cccs2)(NC)CC1 N1(C(C2CCC(=O)N2C2CC2)=O)CC2CC(Nc3ccn4nccc4n3)CC1C2 C=C(C)CC(C)C(=O)N(C1CCCCN(C(c2nccn2CC)=O)C1)C C=C(Cl)CC(C(=O)N1CC(CCCC)C1)NC(C1CCC1N(C)C)=O N1(C(CNC(CC)=O)=O)CCC(O)(CCNC(c2conc2C)=O)C1 c1(C(=O)NC2CC2NC(C2CC(F)(F)C2)=O)ccn2ccccc12 c1(OC)cccc(C(=O)NCCCN(C(=O)CC(C)C2CC2)C)c1OC C1(NC(CC2(N(S(C)(=O)=O)C)CC2)=O)CC(O)C1CC(=O)NC1CC(C#N)C1 C1(CC)CCC(C(=O)N(C(C)C(=O)NCCOC2CC2)C)CC1 C1(C(N(CC(CNC(Cc2c(C)nsc2)=O)(C)C)C)=O)CCC2CCC1O2 CC(CCCCNC(=O)C(C)N(C)C)NC(=O)C(C)CNS(C)(=O)=O CC1(C)CC(=O)OC1CNC(=O)NCc1cccc(C[Si](C)(C)C)c1 N1(C(CCCC#CC)=O)CCC2CCCC12C(=O)NCCC(=O)N(CC)CC Cc1cncc(C)c1C(N1CC(F)(F)CC1C(=O)Nn1ccnn1)=O C(=O)(C1=NNC(=O)C1)NC1CCN(C(c2c(C)cn(-c3ccc(F)cc3)n2)=O)C1 n1(CCNC(=O)CCc2nncs2)cnc(C(=O)NC2(c3ccsc3)CC2)c1 N1(C(C(F)=CC)=O)CC2(CCC(CNC(=O)CSc3cccc(C)c3)O2)C1 C(=O)(C(CNC(=O)CNc1cccnc1)N(C)C)NCC(C)Cn1cccn1 C1(C)(OCC)CCN(C(=O)C(C2CC=CCC2)NC(=O)C2=C(C)CC2)CC1 Cc1nc(C(=O)NC(C)C(=O)NCCCOCCN(C(=O)CCF)C)n[nH]1 C(=O)(CC(C(F)F)C(C)(C)C)NC12CC(NC(C(C)OCCC(C)C)=O)(C1)C2 c1(C(N(CCCCNC(=O)COC2CCOCC2)C)=O)ccc2ccnn2c1 C1(NC(C)C(=O)N(C)Cc2cc(-c3ccccn3)nn2C)CCS(=O)(=O)CC1 N1(C(c2ccc(C(N)=O)s2)=O)CCC2(CC1)CN(C(C1CC1F)=O)C2 C1(C(=O)NCCCNC(c2coc(Br)n2)=O)CCC2(CCC2)OC1 N1(Cc2cc(OC)ns2)CCCC(NC(c2ccc(Cl)cc2)c2ccccc2)C1 C(=O)(CCCC(=O)N(C)C)N1CCCC(N(C(C(C=C)C)=O)CC)C1 C(C)(C)(CC(=O)NCc1cn(CC2CCCN2C(=O)CC2(C)CC2)nn1)OC n1(CC(=O)NC(CC=C)CNC(=O)CC(C)C2CCC2)nc(C(C)C)cc1C N1(C(C(C)c2ccsc2)=O)CCN(C(c2ccccc2CN(C)C)=O)C(C)C1 N1(C(C2(CCCC)CCCC2)=O)CC2(CC(NC(=O)CN3CCS(=O)CC3)C2)C1 Cc1cncc(C=CC(=O)N(C2CN(C(=O)CNC(=O)N(C)C)C2)C)c1 Cc1cc(Cl)c(C(=O)NCC2CN(C(=O)C=Cc3cncs3)CC2C)s1 n1(CCC)nccc1C(N1CC(C)(CCC(=O)NC(C)CCCO)C1)=O C1(CNC(C2(CC)CCC2)=O)(N)CCCC1.n1(C(C(=O)C=O)C)cc(C)cn1 O=C(CC(O)C1CCCC1)NCC1(NC(c2cnn(CC3CCC3)c2)=O)CCOC1 C1(C(=O)NCC(C)N(C(=O)Cc2nnn(C(C)(C)C)n2)C)CCCC2(CCC2)C1 c1(C(C)C)cc(C(N2CCC(NC(=O)Cc3ccccc3)C2)=O)on1 c1(CCC(=O)NCC(C)(C)CNC(=O)CC(C)(C)C)ccc(Cl)c(Cl)c1 CCCCC(CNC(=O)C(c1cnn(C)c1)O)NC(=O)COC1CCC(C)CC1 c1(CN2CCOCC(NC(c3c(C)cc(F)nc3)=O)C2)c[nH]c2ccc(O)cc12 N1(C(C2CC(OC)C2)=O)CCOCC1CCNC(c1ccc(C(F)F)cc1)=O C(=O)(CCCCCCCBr)N1CCC(C#N)(NC(c2cc(C)c(Br)cc2C)=O)C1 N1(c2nccc(C)n2)CC(C(=O)NC(=O)CCCC(N)=O)CC2(CC2)C1 c1(C(N2CC(C)N(C(c3cc([N+](=O)[O-])ccn3)=O)CC2)=O)nccc2cccnc12 c1(OC)cc(Br)c(C(N2CCCC2CNC(c2n[nH]c3ccccc23)=O)=O)cc1O C(C(F)(F)C(=O)N1CCC(N(C(c2c[nH]c(C(F)(F)F)c2)=O)C2CC2)C1)N(C)C N1(C(c2c(CC)non2)=O)CCC(C(=O)NC2CCCC(C)(C)C2)C1(C)C N1(C(=O)NCCc2c(CC)con2)CCn2c(cc3ccccc23)C1 C(=O)(C1=COCCO1)N1CCC(C(C)(C)C)(CNC(=O)Cc2c[nH]nc2O)C1 c1(N(CC(C)C(C)(C)C)C)nc(NCC2Cc3ccccc32)nc2c1cnn2C C1(NC(c2c(C)occ2)=O)CN(C(=O)COc2cc(F)cc(F)c2)CC2(CC2)C1 CN(C(=NCc1ccc(Cl)c(Cl)c1)NC1CCCC1)Cc1ncc(Cl)n1C CCC(CC)C(C(=O)N1CC(C)(NC(=O)CC(C)SC)C1)OC CCC(CCCC(=O)Nc1cccc(F)c1C)NC(c1sccc1Cl)=O C1(C(=O)NCCN(C(C2CN(C(=O)NC)C2)=O)C2CC2)NC(=O)CC1C c1(C(=O)NCCNC(c2c(C)ncc(C)c2)=O)cccc2[nH]ncc12 C(CCC(=O)NC1CNC(=O)C1(C)C)(C(C)C)NC(C(CCCC)O)=O CNS(=O)(=O)N1CCC(C(=O)NCCOCCN(c2cnn(C)c2Br)C)CC1 N1(C(C2CC(C)(O)C2)=O)CCCCC2(C1)CN(C(c1ccc(Br)c(O)c1)=O)C2 S(=O)(=O)(c1ccc(Br)cc1NCC=Cc1cccnc1)NC1C(C)C2CCC1C2 c1ccc2c(NCC(c3ccc(Br)cc3)N)cccc2c1 N1(C(CS(CC)=O)=O)CCC(C2(O)CN(C(=O)CCC3CC(OC)C3)C2)CC1 C1(C(=O)NCCC(C)N(C(c2ccc(COC)s2)=O)C)CC2CCCCCCC12 Cc1nn(C(C)C)cc1C(=O)NCC1(CNC(C2(O)CCCC2)=O)CC1 C(=O)(C1=C(Cl)CC1)NCCN(C(C1CN(C(C)C)C1)=O)C(C)C c1(NC(CCC)C)cc(N(C)Cc2cc(C)n(C)n2)nc(C(C)C)n1 C1(NC(c2cn(C(C)C)nn2)=O)CCC2(CC1)CC(NC(c1c[nH]c(=N)o1)=O)C2 N1(C(CC(CC)CC)=O)CC2COCCC2(NC(=O)C=CC(F)(F)F)C1 c1(CNCN(C2C(C)C2)C)ccc(SC(C)(C)CO)cc1 c1(CN(C(=O)CC(N)Cc2ccc(C(C)C)cc2)CC)cc(C)c(Br)c(C)c1 CC(C)(O)C(F)(F)C(=O)NC1CCCC(Sc2ccccc2C(N)=O)C1 C(=O)(C1CCc2cccc(F)c21)N(CCCCN(C(=O)CC1CCC(=O)N1)C)C N1(C(c2c(C)nc(-c3ccc(C)cc3F)s2)=O)CCC(CN)c2ccccc21 c1(C(C(=O)NC(C)C(=O)NCC=CCOCCOC)(C)C)scnc1C(=O)OC CC1C(NC(c2cc3ccccc3s2)=O)C(C)CCN1C(=O)CCCCO C1(C(=O)NCCCC2(C)CCCC2)CC(O)CN1C(c1ccon1)=O c1(C(=O)NC2CCN(C(C3CCC(C)NC3=O)=O)CC2)nc2cnccc2s1 CC(C)(C)C(O)C(=O)N1CCCC1CC(=O)Nc1cncnc1O N1(C(CC(C)(C)OC)=O)CCCC2CN(C(C3(C(F)(F)F)CC(O)C3)=O)CCC12 CC1CN=C2NNC(C(=O)Nc3ccc4[nH]ccc4c3)=NC12.c12cccc(c1)CO2 c1(C(=O)NCC23C(CN(C(C4(CC)CCC4)=O)C2)C3)csc2ncnc(O)c12 C1(NC(c2cncc(F)n2)=O)(CO)CCCN(C(=O)Cn2ccnn2)C1 C(=O)(CC(=O)NCC1C(C(=O)NC2CC(O)C2O)C1(C)C)OC(C)(C)C c1(C(=O)OC)cc(C(=O)NC2CCC(NC(c3ccc(F)cc3)=O)C2)cc(F)c1 C=CCC(CC=C)C(=O)N(C1CCN(C(C2CCCC2C(F)F)=O)C1)CCC C1(C(=O)NCCOCC(N)=O)COCCC1NC(c1ncccc1Cl)=O CC1=C(C)CC(C)(NC(C2CCN(C(c3ncccc3C)=O)CCO2)=O)CC1 c1(C(=O)NC(C)(C)C)nnc2n1CCN(S(C)(=O)=O)C2 C=C1C(C(=O)OC)CC1C(=O)N(CC(C)(C)CNC(=O)C(F)CC)C N1(C(c2ccnc(OCCO)c2)=O)CC2CCC(C1)N2C(C1C=CCC1)=O N1(C(COCCOC)=O)CC2(CCN(C(=O)Cc3c[nH]ccc3=O)CC2)CC1C n1(CC(=O)NC(C(C)C)CNC(C2CCCN2C)=O)ccc([N+](=O)[O-])n1 c1(C(=O)NCC(C)CN(C(=O)CC2CCN(C)C2=O)C)cccc2c1NCCC2 C1(C(=O)NC2CN(C(C)C)C2)CC12CCN(C(=O)C(N)=O)CC2 C(Cc1ccccc1)(C(=O)NC1CCC(CNC(=O)C=C2CCCCC2)C1)OC c1(C(C)C(=O)NCCC2CCC2)cc(Cl)ccc1Nc1ccccc1 C1(NC(C=CC)=O)CCC2(CC1)CC(NC(=O)C1=NOC(CC3(O)COC3)C1)C2 N1(C(c2occ(C)c2)=O)CCC2CN(C(C3CC3c3cccc(F)c3)=O)CC2C1 C(=O)(C(F)CC(C)(C)NC(=O)Cc1ccc(F)cc1)NCC(C(C)C)C(C)C CCC(COC)C(=O)NCC=CCCC(=O)NCCCC(O)C(C)C C1(C(=O)NC(C)Cc2cccc(F)c2)CC(F)CN(C(c2ccc(=N)[nH]n2)=O)C1 Cc1c(NC2CCCC(CN)C2)ccc2ccccc12 C(=O)(C(C)CN(C)C)NCC1N(CC(=O)NCC(=O)NC)CC1 c1(C(=O)NCC(CC=C)NC(=O)COc2ccsc2Cl)cnc2nccn2c1 C1(CC)C(CC(=O)NC2(CNC(c3ccn(C(C)(C)C)c3)=O)CCC2)C1(F)F N1(C(C(CC)O)=O)CC(CNC(=O)CC2OCCO2)C2(CC2)C1 C1(NC(C(CC)O)=O)CCC2(CC1)CN(C(c1cncc(C)c1Cl)=O)C2 N1(C(c2ncc(OC)nc2)=O)CCCC(C)(CNC(c2ccno2)=O)C1 C1(C(C)NC(c2cc(O)ccc2O)=O)OCC2CCN(C(C3CC3(F)F)=O)CC12 c1(CNC(C(C(C)C2CC2)NC(C)CCCCO)=O)cn2cccnc2n1 c1(CC)conc1CC(=O)N(C1CC(NC(c2c[nH]nc2C2CC2)=O)C1)C c1(C(c2ncc(C(=O)NCCNC(C3(C)C=CCC3)=O)s2)=O)cnn(CC)c1.CC C12(CNC(C3(C)CCC3)=O)CN(C(C3CC4CCC3C4)=O)CC1CCO2 N#Cc1cccc(OCC(N2CC3C(C2)N3C(c2cc(F)cc(Cl)c2)=O)=O)c1 N1(C(COC(C)C)=O)CC2(CCN(C(=O)CC(C)(C)C3CC3)CC2)CC1C N1(C(=O)CSC)CCCC(n2cc(C3(c4ccc(Br)cc4)CC3)nn2)CC1.C1CCC1 N1(C(CCOCC#C)=O)CC(CNC(=O)Cc2ccccc2Cl)CC12CCOC2 c1(C(N2CCC3(C(NC(CC4CCC(C)CO4)=O)C3)C2)=O)nc[nH]c2ncnc1-2 C(C)(C1OCCc2ccccc21)NC(c1c(NC(=O)OC)cccc1)=O C1(CN(C(C23CC(C)C2C3)=O)C)CN(C(c2cc(C(F)F)[nH]n2)=O)CCO1 c1(C(C)C)cnc(Cl)nc1N1CCC(CN(C(=O)CSS(C)(=O)=O)C)CC1 Cn1cc(NC(=O)NNC(=O)C2CC(c3ccccc3)C2)c(=O)c2sccc12 c1(C(=O)NCC2(NC(Cc3cc(C)sc3)=O)CCC2)cnc(O)c2c1NCCC2 Cc1sc(C)c2sc(C(=O)NC3CC4CCC3C(NC(c3ccccn3)=O)C4)cc12 C1(CCOC)(C(N2CC(CS(C)=O)C2)=O)CC(C)(C)C1.C12CC(C1)CC(=O)N2 N1(C(C(=O)NCCC)COc2ccccc2)CCOC(c2n[nH]c(C(C)C)n2)C1 c1(C(N2CCC(OC(C)CN(C)C)CC2)=O)ccc2c(Br)cccc2c1 CS(=O)(=O)c1ncccc1NC(=O)NCCNc1nc(O)sc1C#N c1(CC)c(C(=O)N(CCCCCCNC(=O)CC2CCCC(O)C2)C)nnn1C c1(C(C(C2CC2)N)C2CC2)ccc(F)cc1C(c1nnnn1C1(C)CC1)OC.C1CC1 c1(C(N(C2CCN(C(c3cc(CCC)on3)=O)C2)C)=O)c(OC)ccnc1F c1(NC(C2C(C)C2)=O)cc(NC(c2ccco2)=O)no1.C123CC(C1)(C2)NC3=O C1(CC(N2CCOC(C3CC(F)(F)C3)C2)=O)CCCOCC1 C(=O)(C(CN=[N+]=[N-])NC(C1CCC=CCCC1)=O)NC1CCN(CC)C1 N1(C(CC(=O)NCC(C)N(C(c2c(C)ncs2)=O)C)C)CCCCC1=O c1(C(=O)NCC2C(NC(c3cc[nH]c3)=O)CC2)nc(C2CC2)ncc1Br C1(CNC(C2N(C(C3C(CC(C)C)C3)=O)CCCC2)=O)CC2CCC1CC2 c1(C(=O)NCC2CC(n3cc(-c4c(SC)cccc4)nn3)C2)cncc(C)c1Cl C(CC1=CCN(C(c2cncs2)=O)CC1)NC(C(C)C(C)c1ccccc1Cl)=O C1(NC(CCC=C(C)C)=O)CC(C)CN(C(C2(c3cccs3)CC2)=O)C1 N1(C(C(C(C)O)NC(C(CC)=CCCC)=O)=O)CCCC2(CCC2)C1C CCC(CCCC(=O)NC1CNC(=O)C12CC2)NC(=O)C(C1CCCCC1)F C1(CNC(C2CN(C(C)=O)C2)=O)CCC(C)(C)CN1C(=O)C=CC(F)(F)F C1(NC(C2C(CC)C2)=O)CN(C(C2CCn3cc(C)nc3C2)=O)CC2(CCC2)C1 C#CC(CC(C)(C)C)OC(=O)Cc1ccc(Oc2ccc(C(=O)O)cc2)cc1 Cc1ccc(CNC(=O)C(c2ccccc2OCc2ccccc2F)O)n1C N1(C(C(C)Cc2ccccn2)=O)CC(C2CC2)(C(=O)N(C)Cc2ccon2)C1 C(=O)(C(C)S(C)(=O)=O)NC1(CN(C(c2c(C)n(C(C)C)nc2)=O)C)CC1 C(CC(C(=O)NOC1CCC1)NC(C1CCN(C)C1=O)=O)OCC N1(C(c2nccc(OC)n2)=O)CC(C)CCC1CNC(C12CC(CC(C)C)(C1)C2)=O c1(C(=O)NC2C(OC)CN(C(C3(C)CC(C)=NO3)=O)C2)cccc2nc[nH]c12 Cc1nc(C(=O)NCCC2CCN(C(=O)C(=O)N=S(C)(C)=O)C2)ccc1[N+](=O)[O-] c1(CN(CC(=O)NCC(C2CCCN2C)C)C(C)=O)ccc(C)cc1 c1(C(N2CC(CCC)C(NC(=O)CC3=CCOCC3)C2)=O)ccc(N)c(F)c1F N1(C(c2ccc(=NC)[nH]c2)=O)CCC2(C=C(C(=O)NC3(COC)CCCC3)C2)C1 CC(C)C(C)C(=O)N1CCOC(CC(=O)NC(C)(C)C(C)(C)O)C1 C1(N(C)C(c2ccnc(C(F)(F)F)c2)=O)CCC(=O)NC1=O CC(C)C(C)C(=O)NC1CC12CC(NC(=O)C(=O)NCCSCCO)C2 Cc1cncc(C(=O)NCCC(C)(C)CNC(=O)CC2COC(=O)C2)c1C C1(CN(C(=O)Cc2n[nH]c(C)n2)CC)CCCN(C(C2CC(C)(C)CO2)=O)C1 C(C)(C(C(C)C)NC(c1cnoc1C1CCC1)=O)NC(C=C(C)Cl)=O C1(C(N(C(CNC(CCCOC)=O)C)C)=O)CC(O)CN1C(C)=O CCCC(C)C(=O)NCCC(Cc1ccccc1)NC(C1CCC(OC)CC1)=O Cc1cccc(C(=O)NCC2CCN2C(c2cccn2Cc2ccccn2)=O)c1C N1(c2n(CCC=C)c(-c3[nH]nc(Br)c3C)nn2)C2CCCC(O)C1CC2 c1(C(N(CCN(C(C2CC(C(F)(F)F)CO2)=O)CC)CC)=O)cc(F)ccc1C Cc1cn(C)nc1C(=O)N(CCNC(=O)C=Cc1ccco1)CC1CC1 c1(C(=O)NCC2N(C(CCCCSC)=O)CCCC2C)c(C)[nH]c2ccccc12 C1(C=O)CCC2CC1CO2.C1(C(=O)NCC2(OCC(N)=O)CC2)CCC(CO)CC1 N1(C(CN(C)CCO)=O)CCCC1C(C)(C)CNC(c1ncc(C(F)(F)F)s1)=O C(=O)(C1=CCCC1(C)C)NC(C1CCCC1)CNC(CC1CCCC(C)O1)=O N1(C(C(C)NC(=O)OC)=O)CCC(F)(CNC(c2ncccc2SC)=O)C1 C1(C(=O)NC(C2CCCC2)C#C)CCCCN(C(C2CCC(N(C)C)C2)=O)C1 C(=O)(CCCC(=O)NCC1(C)CCCN(c2ccnc(C)n2)C1)NCCC N1(C(c2n(C)c(Cl)nc2)=O)CC2CC(C1)CN(C(c1ccc3c(c1)NCC3)=O)C2 Cc1ccn(C)c1C(=O)NCC1(C)CC(NC(=O)CCC2CCCCC2)C1 Cc1c(C(=O)NCCC(C)NC(c2cc([N+](=O)[O-])n[nH]2)=O)oc2ccccc12 C1(NC(C2(CNC(C3N(C)CCOC3)=O)CCCC2)=O)CCn2nccc2C1 N1(C(CC(CN(C)C)O)=O)CC=C(CNC(c2cnn3c2CCC3)=O)CC1 C(=O)(C(C)C(C)CC)NCc1ccc(C(C)NC(C2(COC)CC2)=O)cc1 C1(CNC(C(C(C)C)F)=O)CCN(C(=O)C(c2cccc(C#N)c2)C)C(C)C1 c1(NC(=O)NCc2c(C)cccn2)ncnc2sc(I)cc12 C1(NC(CC2CN(C)CC2O)=O)CN(C(c2cnco2)=O)C(C)(C)C1 C(=O)(CCCC(=O)NC1CC2(C1)CC2OC(C)C)NC(CC)C(C)O O=C(N1OC2CCC1CC2)C1CCC(C2CC2)N1C(=O)CSC1CC1 C#CC(C)(C)C(=O)NC1CC(C(F)C(=O)N2CC(C(C)CC)C2)C1 C1(CS(C)(=O)=O)CN(Cc2coc(C3CCCC3)n2)CCO1 N1(C(c2c(C)cc(C)s2)=O)C(C)CN(C(c2cc3scnc3[nH]2)=O)CC1C C1(C)(CC)C(C(N2CC(F)C2)=O)CC1N N1(C(C(C(C)(F)F)F)=O)CCC(C2CC2)C1CNC(c1n[nH]c2c1COCC2)=O c1(C(N2CCCC(N(C(C3N(C)C(C(N)=O)CC3)=O)C)C2)=O)ccc(F)c(F)c1 CCC(C)C(O)C(C)C(=O)N1CCC(C(=O)NCC2CN(C3CC3)C2)C1 C1(NC(C(CC(C)C)O)=O)CCN(C(c2cc(-c3ccns3)on2)=O)CC1(C)C c1(NC)cncc(C(=O)NCC(C)(C)OCCC2C(C(=O)NC)C2)n1.C(CO)O S(=O)(=O)(c1cc(C)cc(Br)c1)NC1C(C(=O)Nc2c(OC)ccc(C)n2)C1 C1(C(N(CCNC(=O)C(C)n2cncn2)CC)=O)CCCCC1(F)F N1(C(C(C)Sc2ccccn2)=O)CCN(C(c2cc(F)cnc2Cl)=O)CCC1C C1(CC(=O)N(CC#C)CCF)CC(O)CN1C(=O)CC1CCOCC1 N1(C(CNC(CC)=O)=O)CC2CC(NC(C3COC4COCC34)=O)CC2C1 O=C(CCS(=O)(=O)C(F)(F)F)N1CC2CC(O)CC1C2 c1(C(=O)OC)cccc(NC(c2ccc(OC(C)=O)cc2)c2ccccc2)c1 C1(C(=O)NC(C)CCN(C)C(c2ocnc2C(F)F)=O)CC(C)(C)CCO1 c1(NC(C(CC2CN(C(C=C(CCC)C)=O)C2)F)=O)cnn(C)c1C1CC1 c1(C(N2CC(CNC(C3CN(C(C)=O)C3)=O)CCC2C)=O)ccc(F)c(N)c1F N1(C(c2ccc(C)cc2)=O)CCC(C2CCCN(c3ccnc(C)n3)C2)C1 c1(C(=O)NC(CNC(c2cnc(OC)nc2)=O)C)cc(Cl)c(OC)c(Cl)c1 C1(C(=O)OC(C2CCCCO2)C)CCCN1Cc1ccsc1 c1(NCC(C)S(C)=O)cc(Br)ccc1S(=O)(=O)N1CCC(=O)N(C)CC1 N1(C(C(C)OC2CCC2)=O)CC2(CCN(C(=O)Cc3cnc[nH]3)C2)C1 C12CCC(CC1)OC1CC(NC(=O)C3CC3)(C1)C2.C(C)(C)(C)OC(=O)OC c1(C(N(CCC(C)NC(=O)Cc2ccsc2Cl)C)=O)cccc(N(C)C)c1 c1(C(N(CCCCN(C(C2CC(OC)C2)=O)C)C)=O)c[nH]nc1-c1ccnn1C C1(C(=O)NCC(=O)NC)CC12CCN(CC1OCCC1(C)C)CC2 C1(CCC)CN(C(=O)COC2CCC2)CCN1C(=O)C(C)Cc1ccncc1 C(=O)(CC(c1ccccc1)N(C)C)NC1C(NC(C2(OC)CC2)=O)CC1 c1(C(N2C(Cn3cc(CSC)nn3)CCCC2)=O)cc2oc(C)c(C)c2[nH]1 Nc1c(F)ccc(Cl)c1NC(C1CCCN(C(=O)C(=O)NC2CCOCC2)C1)=O C(=O)(C(C)S(N)(=O)=O)NCC1CCC(C(=O)NCCc2nc(C)[nH]n2)C1 C1(NC(c2ccc(SCC)cc2)=O)CCCCN(C(c2csc3cncn23)=O)C1 CC(C)CC(C)C(=O)N(C(C(N1CCC(C#N)CC1)=O)C1CC1)C Cc1cc(F)c(C(N2CC(C(=O)NCCCO)CC(F)C2)=O)cc1F c1(C(N2CCC(CC=C)(NC(=O)C=C(C)C)C2)=O)cccc2oc(C)nc12 c1(C(=O)NC2(CC)CN(C(C(CC)C#N)=O)C2)ccn2c1CCCC2 C(=O)(CC(C)(C)O)N(C1CCCN(C(c2ncc(C(F)(F)F)s2)=O)C1)CC Cc1oc(Br)cc1NC1(c2nnnn2C2CCCC2)CCCCC1 N=c1[nH]c(CC(=O)NC2CC2NC(c2ccc(-c3ccccn3)o2)=O)cs1 c1(C(N2CC3CN(S(=O)(=O)CCCl)CC3C2)=O)nc2ccccc2[nH]1 c1(CC)cccc(C(=O)NC(C)C(=O)N(C)Cc2ncnn2C)n1 CCCC(C)CC(C)NC(=O)NCC(O)CCOC c1(CC)nc(C)c(C(=O)NCC(O)CNC(=O)CCOC2CCCOC2)s1 c1(OC)c(C(=O)NCC2CN(C(=O)Cc3ccccc3O)CCO2)csc1Cl N1(C(c2nnc(C)s2)=O)CCC2CCN(C(=O)C(N(C)C)N(C)C)CC2C1 n1(CC=C)nnnc1C(C)(CN(CCCC1CC1)CC)N(C)C.C1(CO)(C)CCCC1 c1(NCCN(C(=O)CC2(C(F)(F)F)CC2)C)ncnc2sc3c(c12)CCC3 Cc1cc(O)cc(C)c1CN(C1CCN(c2nccnc2Cl)CC1)CC1CC1 c1(C(=O)NCCC2(NC(c3cc(C)c(Cl)cc3)=O)CCC2)cccn2nnnc12 C(=O)(CCCCCNC(=O)C(c1cccc(I)c1)O)OCC c1(OC)ccc(CC(N2CCN(CCN3CCOC3=O)C(=O)C2)=O)c(Cl)c1OC c1(C(=O)NCC(C)(CC)NC(COCCC#C)=O)cc2ccc(Cl)cc2[nH]1 C(CC(C(C)C)NCC=O)(N(CC(F)(F)F)C(C)(C)C)OC.CO C(CN=c1[nH]c(C2CCCC2)nc2c1CCC2)NC(N(C(CC)(C)C)C)=O CC1CCSC1C(=O)NC1(C)CC(NC(=O)CC(Cl)Cl)C1 n1(CC(=C)C)nnnc1C(c1ccnn1CCC)NCC1CCCO1 c1(C(C)NC(C(N2CC(CC=C)OCC2)=O)=O)ccc2c(c1)OCCO2 Cc1cc(F)c(C(N2CC(CCNC(c3cccc(=O)n3C)=O)C2)=O)c(F)c1 c1(C(N2CCCC(N(C)C(C3CC(n4cnnc4)C3)=O)C2)=O)cncc(Cl)c1Cl CCCC(C)CC(=O)N1CC(F)CC1CNC(c1cc2scnc2[nH]1)=O Cc1ccc(N)c(C(N2CC(C(N)=O)(CNC(=O)CCC3CCC3)C2)=O)c1 C(CCCCNC(=O)C(C)C1CCOC1)C(C)C(=O)Nc1nsnc1O c1(N(C(CCc2cc(C)on2)=O)C2CC(NCCCCCl)C2)ccnc(S(C)(=O)=O)n1 C(CC(C(=O)NC1CC(F)(CNC(C2(CO)CC2)=O)C1)N(C)C)SC C12CCCC3(C1)CC3CC(C)=NC=CC1=NC(CCOCC)(C(=O)N1)N2 c1(C(=O)NC(CC)CNC(c2cc(C3CCCCC3)[nH]n2)=O)ccc(C)c(O)n1 C1(COC)CN(C(=O)C(c2ccccc2)=O)CCN1C(C1C=CCCC1)=O c1(C(=O)NCCN(C(C23CC(C(C)C)(C2)C3)=O)C2CC2)n[nH]c2ccccc12 CC1CCc2n[nH]cc2C1C(=O)NCC1COC(C)(C)OC1 c1(CC)nn(C)cc1C(=O)NC(C)C(C)C(=O)NCC1CC1Cl CC(CC(=O)N1CCC(N(C(=O)C(F)C(C)(C)O)C)CC1)CC(C)(C)C N1(C(C)C)CCC2(CC1)CN(C(=O)Nc1ccc(Br)o1)C1COCC21 Cc1nccn1C(C)C(=O)NCc1ccoc1C(=O)NC1CC(F)(F)C1 c1(C(C)C)ccc(C(=O)NCCC2CCN(C(c3cnc(O)o3)=O)C2)s1 c1(CC(=O)NCC2(O)CC(CNC(CC(C(C)C)C)=O)C2)ccc2n[nH]cc2c1 c1(OCC)ccc2[nH]c(CN3CCC4OCCN(CC(=O)OC)C4C3)c(C)c2c1 C1(C(=O)NC2C(NC(C(CCOC)C)=O)CCCC2)(C(=O)OC)CC2(CCC2)C1 Cc1coc(C)c1C(=O)N(C)CC1C2CN(C(c3ccccc3Br)=O)CC12 Cc1c(C(N2CCCC(CC(=O)NCc3ccccc3)C2)=O)cccc1[N+](=O)[O-] c1(C(=O)NC2CCC(C)(OC)CC2)cnc2n1CCC(C)C2 CC(C(CCc1ccccc1)NC(c1cccc(Cl)c1)=O)NC(=O)C=CC(F)(F)F C1(CNC(CCSC)=O)C(C)CCCN1C(C1CCN(CC(C)C)CC1)=O C(CN=c1[nH]c(=NC)[nH]c(=NCC(C)(C)SC)[nH]1)c1cc(OC)cc(C)c1 CCC(C(=O)NCC(C)NC(=O)C=Cc1cn(C)nn1)C(C)(F)F c1(C(=O)NC(C(=O)NC(C=C)C(F)(F)F)COC(C)C)ccc(C)c(O)n1 CC1CCN(C(c2ccc(CSC)cc2)=O)C1CNC(=O)CN(C)C c1(C(N(C(CCNC(CCOCCC)=O)C)C)=O)cccc(NCCNC(C)=O)c1 C(=O)(C(C)CC(C)(F)F)NC(C1CN(C(=O)CCc2cc(F)cc(F)c2)C1)C c1(C(=O)NCC(C)CNC(=O)C#CC2(C)CC2)c(C(C)(C)C)nc2ccccn12 N1(C(C2C(C)CC2)=O)CCC(C)(CNC(c2cc(Br)no2)=O)C1 C1(NC(CC=CCCCCC)=O)CN(C(=O)C(C)NC(=O)NC)C(C)(C)C1 c1(C(=O)NCC(C)NC(CC2(C=C)CCOCC2)=O)cc(Cl)c(Cl)cc1O c1(CC)nn(C)cc1C(=O)NC1CC(NC(C2CC(O)CN2C(C)=O)=O)C1 C1(NC(CCSC)=O)COC2(CNC(=O)Cc3ccc(Cl)cc3C)CC1C2 C1(CC)C(NC(c2cc(C(C)(F)F)on2)=O)CCN1C(=O)C(C)COCC C(CCC(CO)NC(C1CN(C2COC2)C1)=O)OC N1(C(C(C(C=C)O)(C)C)=O)CCC2(CCC(NC(=O)CC(=O)NC)C2)CC1 C1(NC(c2cc(C)n(C)c2)=O)CC2(C(=O)NCCC(N)=O)COC1C2 C1(NC(c2ccnc(N(C)C)n2)=O)CCCN(C(=O)CCC(=O)C2CC2)CC1 COC=CC(=O)NCCC(C)N(C(=O)CSCC(=O)OC(C)(C)C)C CC1=C(Br)CCN(C(=NCc2nc(C)cs2)NC(C2CCCCC2)C)C1 C1(NC(c2cc(N)c(-c3cccnc3)cc2)=O)Cc2ccccc2C1 C1(NC(c2n(C(C)C)cc(Br)c2)=O)CC(O)CN(C(=O)Cc2cnoc2)C1 C(=O)(C(C(C)(C)C)c1ccccc1)N(C)CCNC(C1CC2CC2C1)=O C(=O)(C1Cc2ccccc21)N1C2C(CNC(=O)CC3CC3(Cl)Cl)C(CCC2)C1 N1(C(CC=C)=O)CC2CCCC2(NC(c2cccc3c2OCC3)=O)C1 C(=O)(CCC(C)(C)NC(C1CCCCS1)=O)N1CC(CC)C(F)C1 N1(C(C)=O)CC(C(F)(F)F)OCC1C(=O)Nc1ccc(N2CCCC2)nc1 C1(C(=O)NCC(CNC(C(COC(C)=O)C)=O)(C)F)CC1C1CCC1 C=C1CC2(C1)CC(C(=O)N(C)CC1(O)CCCN(C(c3c(C)ccn3C)=O)C1)C2 N1(C(Cc2c(C)ccnc2)=O)CC2CCN(C(c3cc(C#N)c[nH]3)=O)CC2C1 C1(P(C)(C)=O)(C(=O)NCCCNC(C2C(C)(COC)C2)=O)CC1 S(=O)(=O)(c1cccc(-c2cscc2C(=O)NOC2CC2)c1)CCC(C)C C1(C(=O)NCCc2c(CNC(CS(C)(=O)=O)=O)nco2)CCCC2(CCOC2)O1 c1(NCC(c2ccc(Cl)cc2)(C)NC(C(C=C)O)=O)nccc(SC)n1 c1(C(N2CC3C(CNC(CC(C)OC)=O)(C3)C2)=O)ccc2c(C)n(C)nc2c1 c1(C(=O)NC(C2CN(C(C3CCN(CC#C)CC3)=O)C2)C)cc(Cl)cc(Cl)c1 C(=O)(CC(C)(C)C(=O)NC(CO)CCCCNC(=O)CCc1ncccn1)OC c1(C(=O)NC(CC=CC)C(=O)NCCC#CCC)cc(C)c(C)cn1 C1(NC(C2C(C(=O)OC)C2)=O)CC=C(C(=O)NCC(=O)NCCF)C1 C1(C)(C(=O)NCCCC(C)NC(c2ccnn2C)=O)CC(C)(C)C1 CC1=C(C(=O)NC2CCC(NC(c3coc(O)n3)=O)C2)CCO1 c1(OC)ncc(Cl)c(C)c1C(N1CCCC(N(C)C(c2cc(C)c[nH]2)=O)C1)=O C1(NC(CCOCCOC)=O)CN(C(=O)CSCC2CCCO2)CC2(CC2)C1 N1(C(CN(C(C)=O)C)=O)CCCC1CC(=O)NCCc1[nH]cnc1C CSC=CC(=O)NC(C)CC1CN(C(=O)COCC(C)C)C1 c1(OCCOC)cc(OC)ccc1C(N1CCC(CCNC(=O)C(C)O)C1)=O C(=O)(C(C)(C)CF)NC(c1cnn(C)c1)C(=O)NCCC(C)N(C)C C1(NC(CSCCOC)=O)CC(C2CCN(C(C3Cc4nnsc4S3)=O)CC2)C1 C1(CC#C)(C(=O)NCC2(C)CC(C)(C)C2)CCN(C(=O)C(C2CCC2)OC)C1 N(C1c2ccccc2CC1NC(=O)CC1CCC1)C(CC1(C=C)CCCCC1)=O N1(C(CCCC#C)=O)CCCC(C2CN(Cc3ccc(-c4cc(C#N)cs4)s3)C2)C1 N1(CC(=O)NCC2CN(C(C(C)OC)=O)CC2O)CCc2ccccc21 c1(CC)c(C(N2CC(N(C(=O)CC3C=CCCC3)C)C2)=O)cnn1C(CC)CC C(=O)(CC(C)C(F)F)NCC1N(C(C(=O)NCCOC)C)CCC1 C1(CNC(CCOCCOC)=O)CCN(C(c2csc(C)n2)=O)C12CCC2 N1(C(CC2(C=C)CN(C(c3ccn(C)c3)=O)C2)=O)CCC(C)C(C)(C)C1 c1(C(N)=O)ccc(NC(=O)CC2CCN(C(N)=O)C2)c(CCO)c1.n12cc(nn1)C2 C1(NC(=O)C=CC2CC2)CCC12CN(C(c1cc(O)nc(Cl)c1)=O)C2 Cc1nc(C(=O)NCCNC(=O)C(C)(C)O)sc1-c1ccc(OCC(F)F)cc1 N1(C(c2cnn(C)n2)=O)C(C(=O)NC(C(F)F)C(C)(C)C)C2CC(O)C1C2 C12(CNC(c3ccncc3F)=O)CC1CN(C(C13CCCC1C3)=O)C2 C(C(Cc1ccccn1)C(F)(F)F)n1cc(-c2c(C)ccs2)nn1 CN1CCCC(CCC(=O)NCCC2CCCCN2C(=O)CCc2nncs2)C1 N1(C(c2ccc(OC)nn2)=O)CC(NC(C2CCC2)=O)CC(C)(C)C1 C=CC(O)C(=O)N1CCCC1C(N1CC2CC2C1)=O CCC(C#N)(CC)C(=O)NC1CC12CCC(O)CC2 c1(C(=O)NC2CCN(c3nnc(Cl)s3)CC2O)ccc2nncn2c1 c1(C(=O)NCC(C)(C2CC2)NC(=O)CCc2ccoc2)cc2c(F)cccc2[nH]1 Cc1ccnc(O)c1C(N1CCN(C(=O)CNC(C2CC3(CC3)CO2)=O)CC1)=O N1(C(CC2(OC)CCCC2)=O)CCN(C(=O)C=C2CCN(C)CC2)C(COC)C1 N1(C(C(CCC)OC)=O)CCCC2(C(N3CCN(C(=O)CO)CC3)=O)CC2C1 N1(C(C(COC)C)=O)CCC(NC(=O)CN2CC(=O)N(C)C2=O)C12CC2 CC(C)CC(C)CC(=O)NC1CN(C(C2CC(=O)N(C3CC3)C2)=O)C1 N#Cc1ccc(C(N2CCCCC2CCNC(=O)CC2CCOCC2)=O)[nH]1 N1(C(C2C(C)(C)CCCC2)=O)CCC2C(C1)CN2C(=O)CCCc1nccs1 C1(C(NOCCCCC=C)=O)CCN(C(=O)CC(COC)C2CCC2)O1 c1(C(N(CCC)CCNC(c2cc(OC)ccn2)=O)=O)ccc2c(c1)C(C)CO2 Cc1nn(CC(N2CC=CC(NC(c3cnc(C4CCC4)s3)=O)C2)=O)c(=O)n1C c1(CNCC2(OCC)CCC2)nc(NC(C2CCCCC2)=O)cc(C)n1 C1(C(=O)NC(C#C)C(C)(C)C)CC(C)CN(C(c2cncn2C2CC2)=O)C1 CN(O)C(=O)CNC(=O)C(CC1CCCC1)NC(C1CCCN1C1CC1)=O CC1(C#CC(=O)NCC2(F)CN(C(C3CN(CC(F)(F)F)C3)=O)C2)CCCO1 Cc1nccc(=NC(C)C2CN(C(=O)C(c3cccc(F)c3)C)CCO2)[nH]1 Cc1ccc(SCCC(N2CCC(NC(=O)CC34COCC(C3)C4)CC2)=O)cc1 c1(OC)cc(C)sc1C(=O)N(C1CCCC1)CCNC(C1CC(C)CCO1)=O c1(N(C)Cc2noc(-c3cccnc3)n2)ccccc1C(=O)NC(C)C c1(CCC(=O)N(C)CC2N(C(C(C)=CC)=O)CCC2)cc(C)sc1C C1(NC(=O)CC2CC2)CC2(C(=O)N(CCC(O)CO)CCO)COC1C2 N1(C(c2cnc(C)[nH]2)=O)CCN(C(=O)CC(C)(C)CN(C)C)CC1C CC1OC(C)CC1C(=O)NCCNC(c1cccc(N2C(=O)CCC2=O)c1)=O c1(C(N(C2CCN(C(=O)CN3CCCCCC3=O)C2)C)=O)csc([N+](=O)[O-])c1 C1(NC(COCCCC)=O)CCS(=O)(=O)C12CN(C(c1nccc(Cl)c1C)=O)C2 n1(C(C)C)ncc(C(=O)NCC2CC(NC(C3(C)CCC3)=O)C2)c1N N1(C(CN2C(C)CCC2)=O)CCCC(C(N2CC(CCCCCCN(C)C)C2)=O)C1 C(C(C)(C)C#CC(=O)N1CC2C(CC(=O)OC)C2C1)CC.N12CCOCC1C2=O c1(C(=O)NCCCCCNC(C2CCC(CC)O2)=O)cc(F)ccc1C1CC1 C(=O)(CCCCC(=O)NCC(CO)NC(=O)C(C(C)C)c1ccn(C)n1)NC c1(OC)ccc(Cl)c(C(=O)NC2CC(NC(c3c[nH]cc3C(F)(F)F)=O)C2)c1F N1(C(Cc2cnc(C)s2)=O)CCN(C)CC1CNC(c1c[nH]nc1Cl)=O CC(C)(C#N)CC(=O)NCC(C)(C)CNC(C1CC(CCF)C1)=O c1(OC)cncc(C(=O)NC(CCOC)C(=O)N2CC(F)(CO)C2)n1 CCCC(C)(O)C(=O)N1CCC(CC(=O)NCCN2CCC3CC23)C1 CCCCCC(O)CC(=O)NCCNC(=O)CCc1ccc(C#N)cc1 c1(OCCC(N2CCC(CCN(C(=O)COC)CC)CC2)=O)ccccc1C#N N1(C(C2CCN2C2CCCC2)=O)CCC(NC(C2CC(N3CCCC3)C2)=O)C12CC2 c1(CC(=O)NCC(CC=C)NC(=O)CN2CC=CC2)cccc(C(C)C)c1 c1(C2(C)CC2C(N2CCC(NC(=O)Cn3nnc(=O)[nH]3)C2)=O)ccc(Cl)cc1 C(=O)(CCCCCC(C)C)NC(CCCCNC(C(CC)n1ccnc1)=O)CO C1(NC(c2cc(CC)c(C)s2)=O)CCCCCN(C(c2nocc2C)=O)C1 N1(C(=O)NC(c2ccc(Cl)c(Cl)c2)C)CCC2(CC1)C(O)CC2O c1(C(=O)NC(CCNC(C(C(=O)OCC)F)=O)C)sc2cc(C)ccc2c1Cl c1(C(N2C(C(=O)Nc3cnc(Cl)cn3)CSCC2)=O)c(F)ccc(I)c1F C(C)(C(CO)NC(C1(C)CC1C)=O)NC(C1CN(S(CC)(=O)=O)C1)=O c1(OC)nccc(C(=O)NCC2(F)CC(NC(=O)C(C)n3cnnn3)C2)n1 c1(N(C)C)ccc(NCCNC(=O)CCC2(C)N=N2)nn1 c1(C(=O)NCC(C(C)C)NC(C2CCc3nnnn3C2)=O)ncnc2ccsc12 C12(C(=O)NC(c3ccccc3)C#C)CC(CN1C(=O)CC1CC(=O)NC1=O)C2 Cc1cc(=NC2CCCC3CN(C(C4CC(F)(CO)C4)=O)CC23)[nH]c(Cl)n1 CC1(C)C(C)(C)C1(F)C(N1CCC2(NC(=O)CCc3ccc(Cl)cc3)CC2C1)=O C1(C(=O)Nc2c(CC)csc2)CN(C(=O)CCCC(=O)N(C)C)CCN1C C1(C(=O)NCCC(C=C)C)CCN(C(=O)CCCC2CCCC2)C(C)C1 c1(C(N)=O)cc(F)ccc1C(=O)NC1CCCN(C(=O)CCc2cccs2)C1 C(CC(=O)NCC1(C)C=CCCC1)(C(F)F)NC(CCCC)=O CC(CC(=O)NCCCCNC(=O)CCc1nnc(C2CC2)o1)C1CC1 c1(C(=O)NC2CN(C(Cc3nnc(C)o3)=O)C(C)C2)cc2c(=O)[nH]ccn2n1 C(CO)(CO)(CO)NC(C1CC(C)N1C(=O)CC1(N(C)C)CCC1)=O N1(C(C(C)C)=O)CCC(C(=O)OC(C)(C)C)CC1C.C12(CCCC1)CCC(=O)N2 N1(C(C2N(C(=O)CC3CCOC3)CCCCC2)=O)CCN2C(=O)OCC2C1 c1(C(=O)OC)nc(N2CCCC2CNC(=O)Cc2cccnc2)[nH]c2ncnc1-2 CCCCC(F)C(=O)NC(C)(C(=O)NC1(CO)CC(F)C1)C1CCC1 N1(C(C2CCC(C)C2)=O)CC2(CCC2)CC1CNC(=O)C=C1CN2CCC1CC2 c1(CNC(C2C=C(C)CS2)=O)ccc(C(=O)NCC2C(C)C2C)nc1 C=CCC(CC)C(=O)N1CC2CC(C(=O)N(C3CCOC3)CCO)(C2)C1 N1(CC)CCOC(C(=O)NCCOC2CN(C(c3ccccn3)=O)C2)C1 c1(C(CC(=O)OCCOC(C)(C)C)Nc2cnsn2)ccccc1Cl c1(N2CC=C(C)CC2)cc(N2CCC(OCC3CCCC3)C2)nc(C(F)(F)F)n1 C1(CNC(C2C(C(C)C)C2)=O)CCN(C(=O)CC23COC(CF)(C2)C3)CC1C C1(OC)CCN(C(c2cnc(O)cc2C)=O)C(C)C1.c12ncc(s1)C=CCO2 C1(C(N2CC(C)(NC(CCN(C(CC)CC)C)=O)C2)=O)CCCC(OC)C1 CC(C)(C)CC(=O)NCC1(O)CN(C(c2cccc(-c3cccs3)n2)=O)C1 C(C(C)C)(C(O)C(=O)NC1CC(N(C(=O)Cc2cnn(CC3CC3)c2)C)C1)OC Cc1cc(C(F)F)n(CC(=O)OCC2CC23CCC3)n1 N1(C(c2nc(CC)oc2)=O)CCCC12CCN(C(c1cc(C(C)=O)on1)=O)CC2 C1(C(N(CCCC)CC(N)=O)=O)CCC2(CC2)N1C(C1CCCCS1)=O CCC(C)CCCC(=O)N1CC(C(N2CCC(n3ccnn3)C2)=O)CCC1C CC(C#N)CN=c1[nH]c(=NC2CCC(N3CCCCC3)C2)[nH]c2c1CCCCC2 N1(C(C(c2ccc(C)o2)C)=O)CCC2CCN(C(=O)C(O)CC3CC3)C2C1 CCC(CC(C)C)C(=O)NCC(CC(C)C)NC(c1ncc(F)cc1C)=O Cc1ncc(C(=O)NC2C=CCN(C(=O)Cc3csc(Cl)c3)C2)cc1N C1(OC)(CNC(=O)CCC#N)CN(C(C2CN(C(N)=O)C2)=O)C1 C(CC(CNC(=O)C(=Cc1cn[nH]c1)C)NC(=O)C(c1ccn(C)c1)C)OC CN(C(=NCCNS(C)(=O)=O)NCc1ncc(Br)s1)Cc1ccsc1 C1(NC(c2c(Cl)nc(OC)s2)=O)CCN(C(=O)CC23CCCN2CCC3)C12CC2 C12(CNS(=O)(=O)C1)CC(=O)N2.C(C(=O)OCC)(OC(F)(F)F)OC C(CO)(C(=O)NC1CCCC1CC(=O)NCc1ccnnc1)NC(N)=O C1(C)(CNC(C(C=C)C)=O)CN(C(C2CC3(CCCO3)C2)=O)CC1C O=C(CS(=O)c1ccc([N+](=O)[O-])cc1)NC1COCCN1C(=O)CO C1(C)(C(=O)Nc2c(CC)cccc2)CCCN(C(c2ncccn2)=O)C1 C12(C(=O)NC3CCN(C(c4nc(CC)oc4C)=O)C3C(C)C)COCC1C2(F)F c1(CNC(C2CCC(O)(C(F)(F)F)C2)=O)cccnc1N1CCCCC1 Cc1nsc(N)c1C(=O)NCC#CCNC(=O)C(C(C)C)c1ccc(F)cc1 N1(C(C(C2CCN(C(C=CCN(C)CC)=O)C2)(C)C)=O)CC(CO)C(C)(C)C1 N1(C(CCCC)=O)CCC2CCCN(C(c3csc(C4CCC4)n3)=O)C2C1 C=C=CC(C)C(=O)N1CC(O)CC1C(=O)NC(C)C(=O)NCCF C1(C(N(C(=O)Cc2cc(C)[nH]n2)CC)=O)CCCN(C(=O)CN(C)C(C)C)C1 C(=O)(CC(O)CNC(c1cnc(OC)s1)=O)NC(c1nc(=O)o[nH]1)C c1(C(=O)NCCCc2nccc(C)n2)snc2ccc(Br)cc12 N1(C(COC(C(c2ccc(C(F)(F)F)cn2)(C)C)=O)=O)Cc2ccccc2C1 c1(C(=O)NC2C(OC)CN(C(c3cnc(SC)s3)=O)C2)cccc(SC)c1Cl Cc1cc(C(C(=O)NCSc2cc(F)cc(F)c2)Nc2ccc(F)cc2)cc(F)c1 c1(OC)cc(NC(=O)CC2CCCN(Cc3cccn3C)C2)cc(OC)c1C N1(C(Cc2c(C)con2)=O)CCSCC1CCNC(C1(CC2CC2)CC1)=O c1(NCC2C(NC(c3nc(OC)oc3)=O)CCCC2)ncc2scc(Br)c2n1 C1(NC(c2nc(C)[nH]c2C(F)(F)F)=O)CCN(C(=O)CCc2ccc[nH]2)CC1C n1(CC#C)cnnc1C(N1CC(C)(CCC(N2CCC(CO)C2)=O)C1)=O Nc1nn2ccccc2c1NC(=O)NC1CCC2SCCSC12 c1(CC(=O)NCCNC(c2ccn(C3CC3(F)F)n2)=O)cc(C2CC2)ccc1F c1(C(=O)NC2COCC2NC(C2CC2(F)F)=O)snc2ccccc12 C(=O)(C(C)(C)CCNC(c1cnn(CCO)c1)=O)NC(CC)CN(C)C c1(CN(C(c2cc(C(=O)NCCC)ccn2)=O)CC)ccncc1Cl.C(=O)OC C1(C(=O)NCCCCN(CC)CC)OC(=O)NC1(C)C.N12CC(C(F)C1)C2=O N1(C(Cc2c(Br)cn(CC)n2)=O)CCN(C(C2CC2F)=O)C(CF)C1 C=CCC(C(=O)N(CC1(C(=O)OC)CC1)Cc1cccc(C)c1)NCC(N)=O c1(CCC)cnnc(C(=O)NCC(CC)NC(=O)CCOc2ccccc2CC)c1 C1(OC(C)C(=O)N(C)CC2CCCN2C(=O)CCc2cc(O)no2)CCCCC1 c1(C(=O)Nc2ccccc2O)ccc(CN(C)CCO)cn1.c1(S)ccccc1 O=P1(c2ccc(NC(=O)CCc3nnc(C(F)F)o3)cc2)CCCCC1 N1(C(c2nn(C)c3c2CCCC3)=O)CC2CCN(C(C3CC(=O)N3)=O)CCC2C1 C1(C(=O)NC2C(NC(Cc3ccc(OC)cc3)=O)CCC2)CC(C2CCC2)C1 c1(C(N2CCCC(N(C(CCC)=O)C)C2)=O)nn2c(c1Br)CCC(C)C2 C1(CCC)CN(C(=O)Cc2csc(Cl)c2)CCN1C(=O)Cn1cnnn1 C(CC(C)C(=O)N(CCCCC(=O)NC1CCC(OC)C1)C)OC Cc1ccn2cc(C(=O)N(C)CCNC(c3sncc3C)=O)nc2c1 Cc1c(NC(CF)CF)ncnc1NCCCc1ncc[nH]1 N1(C(C2C3(CCC3)C23CCC3)=O)CC2CC(C1)CN(C(c1csc(Cl)n1)=O)C2 c1(NC)ccc(F)cc1C(N1CCC(O)C(NC(c2cc(C)c(C)cn2)=O)C1)=O C(=O)(CC(O)Cc1ccccc1Cn1cc(-c2c(C)ccs2)nn1)NCC1CC1 N1(C(C(C)N(C(C)=O)C)=O)CCC2C1CCN2C(c1cc(I)cnc1Cl)=O c1(CC)cc(OC(=O)Nc2ccccc2C#N)cc(C)c1 N1(C(C2(C(C)C)CCN(C(c3ccc(=N)[nH]c3)=O)C2)=O)CC2CCCC2C1 c1(C(=O)NCC2(F)CN(C(C3CC(OC)C(OC)C3)=O)C2)ccc2c(c1)CC2 C1(NC(C2C(NC(c3c(C(C)C)occ3)=O)CCC2)=O)CC1C1CCCC1 Cc1nc(C(C)(C)C)[nH]c(=NCC2C3CN(C(C4CN(C(N)=O)C4)=O)CC23)c1C Cc1nocc1CNC(c1occc1CNC(=O)CNc1ncccn1)=O C=C(C)C(C)(O)C(=O)NC(CNC(=O)CC1(COC)CCCC1)C(C)(C)C C1(COC(c2c(C#N)cc(F)cc2)=O)CC2(CCOCC2)C(=O)O1 N1(C(=O)NC(C2CCCCO2)C)C2CCC1c1ncccc12 Cc1cncc(CN2CC(NCCCc3nnnn3C)C(C)C2)c1 Cc1c(C(=O)O)cnn1-c1ccc(NC(C)C(CO)NC(=O)OC(C)(C)C)cc1 N1(C(C(N2CC(c3cncc(Br)c3)(F)C2)=O)=O)CCOC(CC2CCC2)C1 C12(CNC(CCCCC#C)=O)CN(C(C3CCCOC3)=O)CC1CS(=O)(=O)C2 C(=O)(C(C)C(=O)OC)NC.C1(CC(=O)N(CCC)C2CC2)CCC(O)C1 c1(NC(C(CCC=C)NC(=O)C=C(C)c2ccco2)=O)cc(C)c(O)cc1C c1(C(=O)NCC=CCCC)c(C2CC2)nsc1N N1(C(C)=O)CCC(C)(C(=O)NCCC(C)NC(C2CCOC2C(F)(F)F)=O)C1 c1(C(=O)NCCCN(C(C2C(C)(COC)C2)=O)CCO)cc2n(c1)CCC2 CC(C(=O)N1CCCC(O)(CN(C(=O)COCC(F)F)C)C1)C(F)(F)C(F)F Cn1ncc(Cl)c1C(=O)NCCCN(c1nccc(C(=O)OC)n1)C1CC1 C1(OC)CC(C(=O)NC2C3CC(NC(C4CCCN4C(C)C)=O)CC23)C12CCC2 C1(CC)CCN(C(=O)CN2CCC(=O)CC2)C1C(=O)NCCCCc1cnc[nH]1 C1(C(N(CCCCN(C)C(C2(O)CCC2)=O)C)=O)CCCC(C)(C)CC1 C1(C)(C(=O)NCc2cc(C)on2)CN(C(C23CCC(CC2)CO3)=O)C(C)(C)C1 C1(C(=O)NCC(CC)CCO)CN(C(C2CC2Cl)=O)CC12CC2 S(=O)(=O)(c1ccc(NCCCS(N)(=O)=O)c(Br)c1)NC(CC)CO c1(OC)ccc(F)c(C(N2CCC(C(C)(C)NC(=O)CS(N)(=O)=O)C2)=O)n1 Cc1ccc(COCC(=O)NCC2COCCN2C(=O)C(F)C(C)C)cc1 c1(C(N2CC(CC(N3CCC(=C)CC3)=O)OCC2)=O)cc(I)ccc1F c1(C(N2C(CNC(COCCC#C)=O)C=CC2)=O)ccc(F)c(Cl)c1N c1(CC(=O)N(CC(C)N(C(CC(CC)OC)=O)C)C)nc([N+](=O)[O-])n[nH]1 CN1CC2(CCN(c3ncnc4ccc(F)cc34)C2)CC1=O C1(NC(=O)Cc2nnc(O)s2)CC1C1CCCN(C(c2cn(C(F)F)cn2)=O)C1 n1(CCC(=O)NCCC2CCC(NC(c3c(OC)csc3)=O)C2)c(C)ccc1C c1(C(=O)NC(C2CCN(C(C(CC#C)(C)C)=O)C2)(C)C)ccc2c(c1)COB2O C1(C(=O)OC)CC2CC(NC(C3(Cc4cncnc4)CCCC3)=O)C2C1 c1(C(=O)NCC(CC)NC(=O)C(O)CC[S+](C)C)c(N)cc(F)cc1F Cc1cccc(CN2CC(N(C)C(c3ccccc3O)=O)C2)c1Cl N1(C(COCCC(C)C)=O)CCN(C(=O)Cc2ccnn2C)CC(CO)C1 c1(C(N2CC3C(CNC(C(CC)COC)=O)C3C2)=O)ccn2c(C)cnc2c1 C1(N2CCCN(C(C(=O)NCC=C)c3ccns3)CC2)CC2CC3CC(C2)CC1C3 C(C1=CCCCC1)NC(C(C1CCCO1)NC(c1cc(C)[nH]n1)=O)=O N1(C(Cc2c(C)ccc(C)c2)=O)CCC2CN(C(C3CC(=O)NC(=O)N3)=O)CC12 N1(c2nnc(C(=O)NCC3CCC(C(C)(C)C)O3)s2)CC(C(F)(F)F)CC1C C(=O)(C1=NOC2(CCC2)C1)N1CCN(C(CCCc2cc(C)sc2C)=O)C2C1C2 C(CC(C(C)(C)C)NC(=O)CCC1CCCC1)N(C(=O)CC1(O)CCOC1)C c1(C(=O)NCC(CN(C(C(C)OCC)=O)C)(C)C)cc(C)nn1CC(F)(F)F c1(CNC(C(C(C)C)NC=O)=O)coc2ccccc12.c12cccc(c1)NC2=O Cc1ccc(C(=O)NCc2ccsc2C(=O)NC2CC(=O)NC2=O)n1C Cc1csc(C(=O)NCC(C)(O)CNC(c2ccc(C(C)=O)nn2)=O)c1C N1(C(Cc2cn(CC)nc2)=O)CCC(CC(CO)NC(C2CCCCN2C)=O)CC1 N1(C(C)C(N)=O)CCC(CN(C(=O)CCc2ccc(Cl)cc2)C2CC2)CC1 C=CCCC(C)(C)C(=O)NCC1(F)CN(C(C2OC3CCC2C3)=O)C1 CN1CCC2CCN(C(C3CCN(C(=O)C4=CCCCC4)C3(C)C)=O)C2C1 C(CC)(CCC(=O)N(CCOC)CCOC)NC(c1n(CC)ccn1)=O c1(CNC(C2(NC(C(CC)SC)=O)CCSC2)=O)ccc(Cl)cc1 c1(OC(C)C)ccc(N(c2ccccc2)C(=O)NCCC(C)(O)CN)cc1 Cc1cc(C)c(OCCC(=O)NCC(c2c(C)cccc2F)(C)O)c(Br)c1 c1(N2CC(C(C)NC(CCS(=O)(=O)NC)=O)OCC2)ccc2c(n1)CCC2=O CCCC(C)(CC)C(=O)NCC1(C(N)=O)CN(C(C2CCCSC2)=O)C1 C1(NC(C2CCNC2=O)=O)CC2CN(C(=O)CCCCCc3cccs3)CC2C1 c1(NCC(C(CC2CCN(C(CC(C)(C)O)=O)C2)=O)C2CC2)cccc(Cl)c1Cl CC(C)CC(C(=O)N1CC(C#N)(CCF)C1)N(C1CC2CC(=O)C1C2)C C1(NC(c2nc(C)oc2)=O)CCC(N(C(=O)CC2CCC(=O)O2)C)CC1 C(CN=C(NC(C1CC1[N+](=O)[O-])C)N1CCC(CSc2ccccc2)C1)SC c1(C(=O)NC2CC(C(N3CCN(CCC)CC3)=O)C2)c(C)cc(Br)cc1C N1(C(=O)CCc2cnn[nH]2)CC2(C1)CN(C(C1CC3CCC1O3)=O)C2 Cc1nc(NC(=O)CCCN(C)C)cc(SC(C)C)n1.C12CCN(C1)C2=O C(=O)(CC1=CCCCC1)N1CCCC(C)(CNC(C2(C)CCCC2(F)F)=O)C1 C1(NC(C(CCCC)O)=O)CC2COCC(C1)C2NC(c1[nH]c(O)nc1C)=O CCCC(C)(CC)C(=O)NCCC(CNC(c1cc(C)cc(C)c1O)=O)OC Cc1cc(CCC(=O)NCCCC(C)NC(c2ncc(C(F)(F)F)s2)=O)c(C)s1 CCC(CCOC)C(=O)NC1CC=C(C(=O)NCCCCc2cnc[nH]2)C1 c1(C(=O)NCCCC(C)NC(C2C(=C)C2)=O)c(C)oc(C)c1Br C1(C(=O)OC)C(O)CCN1C(c1conc1C(C)NC(c1ccc(OC)o1)=O)=O C(N=c1[nH]c(=NCc2cccnc2)[nH]c2c1CCCC2)C1(OC)CCCC1(C)C CC1(C)CN(C(C2(CNC(=O)C#CC(=O)O)CC2)=O)CC(C)(C)O1 N(C(=NCc1cnn(CC2CC2)c1)NC1CC1C1CC1)Cc1ccccc1 Cc1cccc(-c2cn(C3CC(CN(C(=O)CN4CCCC4C)C4CC4)C3)nn2)c1F C1(OC)(CNC(=O)Cc2conc2C)CCN(C(=O)CCCCc2cnc[nH]2)C1 O(NC(=O)CN(C(=O)C(C1CCOC1)S)CC1CC1)CCCC#C.OCC c1(C(N2CC(CN)CC(C(=O)OC)C2)C(=O)OC)cc(Cl)cc(Cl)c1Cl c1(C(=O)N(C(=O)C(F)OC(F)(F)F)C(C2CCOC2)CO)ccn2nccc2c1 C1(F)(CNC(C2CC(C#N)(OC)C2)=O)CCN(C(=O)Cc2cc(C)[nH]n2)CC1 C1(NC(c2ccc(C)c(CO)c2)=O)CC2CCC1N(c1cc(O)nc(C)n1)C2 N1(C(C(C)NS(CC)(=O)=O)=O)CCCC(CC)(NC(c2csc(C3CC3)n2)=O)C1 c1(C(=O)NCC(C)(O)CNC(=O)C(O)Cn2cncn2)ncc(Br)cn1 CC1C2CCCCC2CN1C(=O)C(C)(C)NC(C1C2CC(=O)CC12)=O c1(OC)ccc2c(c1)nc(CNC(=O)CN(C)CP(C)(C)=O)n2C N12CCOCC13CCN(C3)CCNC2=O.C1(O)CCC(C)CC1.Cc1ccc(C)s1 N1(C(C2CCN(C)CC2)=O)CCOC2CCN(C(=O)CC3CCOC3=O)CC12 Cc1ccc(=O)n(CC(=O)NCC=CCNC(c2cc(C(C)(C)C)c[nH]2)=O)n1 C1(C(=O)NCC2CCC3CC23)(CNC(C2CC(OC)C2)=O)CCCCC1 c1(CN2C(C)(C(=O)Nc3cc(OC)c(O)cc3)CC2)ccc(O)c(C)c1O C1(C(=O)NC2C(CC(=O)NC(c3nc(C)sc3)C)COC2)CC2(CCC2O)C1 c1(C(=O)NC(CNC(C2(C(F)F)CCCC2)=O)C2CCC2)c(Cl)csc1Cl N1(C(CC(CC)O)=O)CCC2(CC1)CCN(C(C1CCC1CN(C)C)=O)CC2C C1(NC(COC(CC)CC)=O)CC12CCC(NC(c1ccoc1Br)=O)CC2 CCCC(C#N)C(=O)N1CC(C(=O)NCCCOC(F)(F)F)C(C)(C)C1 c1(CN2CC(CNC(CCN(C(=O)OC(C)(C)C)CC)=O)C2)c(C)cc(C)nc1S C1(C(N(CCCN(C)C)CCN(C(C=CC(CC)C)=O)CC(O)=O)=O)CCCOCC1 C12(C(N(CC(=O)OC(C)(C)C)C)=O)CCCC1CN(C(=O)OC1(C)CCC(C)C1)C2 C=C(C)CCCC(=O)N1CC2CC2(NC(=O)CCCC(=O)NCCC)C1.C(=O)(C1CC1)NCC CN1N=C(CC(=O)N(C)CC2(O)CN(C(C3CS(=O)(=O)C3)=O)C2)CC1=O C1(CNC(C2N(CC)CC2)=O)CCCN1C(c1ccc(CN(C)C)s1)=O C1(C(=O)NCC23CN(C(c4c(NC)scn4)=O)C(CC2)C3)OC(C)(C)OC1(C)C C1(CC)CCN(C(c2cccnc2NC)=O)C(C(=O)NCC(C)C2CCC2)C1 C1(NC(c2n(C=C)ncc2)=O)CC2CC1N(C(c1c(C(F)(F)F)noc1C)=O)C2 c12nc(no1)CCCNC(=O)CC2.O=C(CCOCC1CCCO1)NC1CC1 C1(CNC(CCC(=O)NC23C(CN(C(C)=O)C2)C3)=O)C2C3CCC(C3)C12 C(=O)(C(C)C(F)(F)F)NCC(C(C)C)NC(=O)CCc1cncn1C S(=O)(=O)(c1ccc(Br)cc1N1CCCCCCCC1)N(C1CCC(C)CC1)C1CCC1 Nc1c(F)c(F)cc(CN2CCC(C(N3CCCC3)=O)CC2)c1Cl Cc1nn(C)c(C(=O)NC2CCC2CNC(C2CCCOCC2)=O)c1Br C1(C(=O)OCC(C)CC2CCC2)CCCC(C(F)(F)F)C1 C12(CC(=O)NCC3C(NC(CCc4c(OC)cccc4)=O)C3)CCC(CC1)OC2 C1(CNC(C2CCN(C(=O)CSC3CC3)C2)=O)CCC2(CC1)CC2 C1(CC=C)(NC(c2cn(-c3ccccc3)nc2C)=O)CCN(C(c2cnns2)=O)C1 Cc1nc2ccccc2nc1C(N1CC(O)(C(C)NC(=O)Cc2cnoc2)C1)=O N1(C(c2cc(OC)c(F)cc2)=O)Cc2ccc(C(N3CCC(C)C3C)=O)cc2C1 N1(C(C2C(=C)C2C(=O)NCC)=O)CCOCCC1C(=O)N(CC)CC CC(CSC1CCC1)N=c1[nH]c(N2CCC3(CCCN(C)C3)C2)nc2c1SCC2 N1(C(CNC(C2C(C)C2)=O)=O)CCCC(C(=O)NCC2CC23CCC3)CC1 CCCCCCNC(c1cc(-c2ccccc2)co1)=O.C1(C(=O)NCC)CC1 CCC1CC(=O)C(=O)N1C.C1(Cl)(C(C2CC2)N)CC1(F)F.c1(S)ccon1 N1(C(CCc2onc(C)n2)=O)CC(F)(F)CC1C(=O)NCCCNC(=O)C(C)C c1(NCCOCCOCC)nc(N2CCOC(C)(COC)C2)c2sccc2n1 C(=O)(CCCCc1cnn[nH]1)N(C1CN(C(c2csc(C3CCCO3)n2)=O)C1)C CC(C)C(F)(F)CC(=O)N(C(C)CN(C(=O)COC1(C)CCCC1)C)C N1(C(=O)OC(C)(C)C)CCOCC(C(N2CCCC2(C)Oc2ccc(Cl)cn2)=O)C1 Cc1ccc(Cl)c(C(N2CCOCC2c2cn(CCc3ccccn3)nn2)=O)c1 C1(C(C(=O)NCC(C)NC(=O)CN(C)C2CC2)C)CCOCC1 c1(NC(=O)Nc2cccc(-c3ccc4c(c3)NCC4)n2)cccc2ccccc12 C(=O)(CCCCC(C)(C)OC)N1C(CNC(CCCCCC)=O)CC2CC21 CC(C)(C)C(CO)C(=O)NCC(CNC(c1cnc2n1CCS2)=O)C(F)(F)F c1(OC)ccccc1C(C(=O)NC1CC1NC(C1CC2C=CC1C2)=O)OC C(CC(C)CCNC(C1(N(C)C)CCCC1)=O)NC(C(C)Cc1ccccc1)=O c1(CNC(C(CCC)C)=O)ccc(OC)c(OC)c1.C12CCN(CC1)NC2=O.C1CC1 c1(C(N2C(CCNC(COCC=C)=O)COCC2)=O)cncc2cc(Cl)ccc12 C1(OC)CC(NC(c2cc3n(n2)CCO3)=O)CN(C(C2CCCCC2)=O)C1 Cc1ccc(C(=O)NC(C)Cn2cc(CCS(C)(=N)=O)nn2)c(C)c1 CC(C)CCC(F)C(=O)N1CC2CCCC2(NC(c2ccccn2)=O)C1 c1(CNC(C(C)SC)=O)ccc(CC(C)NC(c2cc(C3CCC3)[nH]n2)=O)cc1 C1(C(=O)NC2CC(NC(=O)CCOC3CC3)C2)(NC2C(C)C2)CC12CC2 N1(C(CCCC(=O)OCC)=O)CCCC2(CNC(c3ccc(Cl)s3)=O)CCCC12 Cc1ccc(C(=O)NC(CCC2CC2)C(=O)NC(C(O)CO)C2CC2)cc1 c1(CNc2c(C(=O)Nc3ccc(Br)nc3I)cc(Cl)nc2)ccc2c(c1)CCO2 c1(C(=O)NCC(C)CN(C(=O)CC(C)(C)C2CC2)C)nccc2cccnc12 CCC(C)(C)CC(=O)N1CCC(CCNC(c2cc(C3CC3)on2)=O)C1 Cn1ccnc1S(=O)(=O)C(=O)NC1(CO)CCCCCC1 O=C(CC(Cc1cccc2c1OCO2)NC(C1CC1F)=O)N=c1cc[nH]cc1F CN1CC(N(C(=O)CCN(C(C2CCN(C)C2=O)=O)C2CC2)C)CCC1=O c1(C(=O)NCC=CCNC(C2N(C(C)=O)CCCC2)=O)ccc2n[nH]cc2c1 c1(CC2CCN(CC)CC2)cc(Cl)ncc1C(=O)N(C)Cc1ccnc(C#N)c1 c1(C(N(C)CCNC(=O)COC2CCCC2)=O)cnn(C2COC2)c1 N1(C(C(C2(O)CN(C(CCOCC)=O)C2)F)=O)CCN(C)C2(CCC2)C1 c1(NC(CC2N(C(c3c(CC)ccs3)=O)CCC2)=O)cc(O)ccc1OC C(=O)(CN1C(=O)Cc2ccccc21)NC(C(C)NC(=O)Cc1csc(Cl)n1)C C12CCC3CN(CCC3C1)C2=O.c1(OC)ccc(C(C)OC)cc1F c1(NCc2cnc(NC(c3cccc(N4CCCC4=O)c3)=O)s2)ccc(Cl)cc1 N1(C(c2nnn(CC)c2C)=O)CC2CC(NC(c3ccncc3F)=O)C(C2)C1 c1(C(=O)NC2(CC)CCCN(C(c3ccncc3Cl)=O)C2)cc2ccncc2[nH]1 Cc1nscc1C(N1CCC(CN(C)Cc2ccc(-c3ccncc3)s2)C1)=O Cc1nn2cc(C(=O)N(C)CCNC(C3C4CCC3(c3ccco3)C4)=O)nc2s1 Cn1cc(C(N2CCC(CCNC(C3(CCF)CC3)=O)C2)=O)cc1S(N)(=O)=O N1(CCC(=O)NC(c2ccccc2)C#N)CCN(Cc2sccc2Cl)CC1=O c1(OC)cc(C(=O)NC2CCN(C(=O)C=Cc3cccnc3)CC2)cc(C)n1 CCC(C(=O)NC(C(=O)NC1CCCC1SC)C(C)C)C(C)C c1(C(N2CC3OCCN(C(=O)C=CCO)C3C2)=O)cc2cncn2c(O)n1 CCCCCCOCC(=O)N(CCCOCCNC(=O)C(C)(C)C1CCCO1)C Cc1ccc2n[nH]cc2c1C(N1CCCN(C(c2cccc(F)c2)=O)C(C)C1)=O C1(=O)CCCC(C)N1.C1(OCCOC)CCN(C(=O)C(F)F)C1 CC1(C)CC(C(=O)NCCC2(CNC(c3coc(-c4ccccn4)n3)=O)CC2)O1 c12ccc(cc1OC(C)=O)C(=O)NCCCN(C)C2=O.c1(OC)cccc(CO)c1 Cc1c(C(=O)NCCNC(C2CC(=O)N(CSc3ccccc3)C2)=O)cnn1C C1(NC(C2CC(O)CN2C(=O)Cc2ccc(F)cc2)=O)C2CCCC1CC2 c1(CNC(N(C2CCC(O)C2)C)=O)ccc(N2CCOCC2)c(C#N)c1 C(C)(C(C(=O)N(C)CC1COCCO1)C(C)C)NC(C1C(C(C)C)CCO1)=O Cc1cc(C(N2CCCC2CN(C(C2CN(C)CCO2)=O)C2CC2)=O)nc(O)c1 c1(C(=O)OC)cc2n(n1)CCCC2NC(=O)Cc1cnc(C)o1 CON1CCC(C(=O)NC2(COC)CN(C(c3cn(CCO)nc3C)=O)C2)CC1 C1(C(=O)NC(CC(C)C)CCO)CC2CCC1N(C(=O)CNc1ccccc1)C2 CC1(NC(=O)CC2(C#N)CCC2)CCN(C(c2cnc(-c3cccs3)o2)=O)CC1 C(=O)(C1=C2CCCN=C2NN1)NC(C(C(C)C)C)CNC(=O)CCS(N)(=O)=O CC1CCN(C(=O)CCCC2CC2)CC1NC(=O)CCOc1ccc(F)c(Cl)c1 N1(C(CN(CCOC)C)=O)CC2CC(N(C(=O)C(n3nc(C)cc3C)C)C)C1C2 c1(NCC2N(C(C(C3CCCC3)OC)=O)CCCC2)cc(C)nc2c(C)cnn12 c1(C(=O)NCCCC(C)NC(c2c(CC)con2)=O)ccc(=O)n(CCO)c1 c1(C(N2CCC(CNC(c3cc(=NC)[nH]cc3)=O)CC2)=O)cccc2c1CCO2 N1(C(CC(=O)NCC#C)=O)CCN(C)CC1C(=O)NC(CC)C#C C1(NC(c2sccc2-n2cnnn2)=O)CCCN(C(c2cc(Cl)no2)=O)C1 CC(=O)CCCC(C)C(=O)NCc1cc(C(=O)NCc2ccc(C)nn2)on1 N1(S(=O)(=O)CC2CCCO2)CCCC1c1ccccc1 CCCCC(O)CC(=O)N1CCN(C(c2sccc2SC)=O)C(CC(C)(C)C)C1 N1(C(c2ccc(CNC(COC(CC)CC)=O)o2)=O)CC(C)C(C)C1C CC(C)CCCOCC(=O)NC(CCCNC(=O)C(C)Cc1ccco1)C1CC1 N1(C(C(C2CCC2)OCC)=O)CC(CN(C(=O)CCS(C)(=O)=O)C)C2(CC2)C1 C1(NC(C(C=C)c2ccccc2)=O)CN(C(c2cc(Cl)cs2)=O)C2(CCOCC2)C1 CC(C(=O)N1CC(N2CCN(C(C34CCCN3CCC4)=O)CC2)C1)S(N)(=O)=O CC1(C)COCC1C(=O)NC(C(=O)NCC12CCN(CC1)C2)C1(O)CCC1 C(CCC(C)(C)C(=O)NCc1ccc(C)o1)NC(C(C=C)O)=O C#CC1CN(C(C2CC2[N+](=O)[O-])=O)CCN1C(c1cc(O)cc(=O)o1)=O O=C(COC(c1ccc([N+](=O)[O-])cc1)=O)N=c1c2ccccc2[nH]n1CCO CC1CN(C(c2cnnn2C)=O)CC1(C)C(=O)N(C)CC1(CO)CCC1 c1(C(=O)NC(C2OCCN(C(c3ccn(CC)n3)=O)C2)C)ccc(O)cc1Cl CC(C)C(O)C(F)(F)C(=O)NCC12CC(CO1)N(C(c1cnsn1)=O)C2 c1(C(N(C2CCCC2)CCCNC(CCC=C=C)=O)=O)ccc(=O)n(CCF)n1 N1(C(c2cc3nc(C)sc3[nH]2)=O)CC2(C1)CN(C(=O)C(C)C(C)(C)C)CC2CO C12(CNC(C(C3(C)CC3)NC(C3CCCCO3)=O)=O)CC=CC(C1)OC2 CC(CC(=O)NC1C2CC1N(C(c1c(N)ccnc1F)=O)C2)CC(C)(C)C C1(CC)CCC(C(=O)NCC=CCNC(=O)C(C)(O)C2CCOCC2)O1 C1(CNC(c2cc(C(C)(C)C)no2)=O)CC2CC2N1Cc1ccnc(Br)c1 C1(NC(C=C2CCC(C)CC2)=O)CC2(C1)CC(C(N1CCCC(C)(F)C1)=O)C2 C1(NC(c2ccc(CC)[nH]2)=O)CN(C(c2cncc3ccsc23)=O)CC2(CC2)C1 C1(NC(C2(CCCC)CC2)=O)C2CCCN(c3noc(SC)n3)C2C1(C)C N1(C(c2c(C(C)C)scn2)=O)CC(NC(=O)C2=COCCO2)C(C)(C)C1 C1(CNC(Cc2c(C)nccc2)=O)CCC(C)N(C(=O)CN2CC3CC3C2)C1 C(=O)(C(C)CCCC(C)=O)N1CC(CNC(c2cncc(NCC)c2)=O)C1 C12(NC(C3CN(C(C)=O)C3)=O)CCC(CN(C(C3CCCN3C=O)=O)C1)C2 C(=O)(C1=CS(=O)(=O)c2ccccc21)N1CC(CNC(=O)C(F)Cc2ccccc2)C1 C1(C)(N(C2CC(OCC)C2)C(=O)C(N2CCn3ccnc3C2)=O)CCC(C)C1(C)C CCCC(C(O)C(=O)NCC1C2CCCCCC12)NC(=O)C(C)(C)C(N)=O CCC(CC(=O)NC1CCC(NC(=O)Cc2cccc(OC)c2)C1)C(C)C c1(C(=O)NC(C)C(CO)NC(c2csc(CO)n2)=O)c(Cl)ccc2c1OCO2 C=CCCC(F)(F)C(=O)N1CC(CCCCNC(c2nc(C)sc2C)=O)C1 c1(CNC(c2cnn(C)c2)C(C)C)csc2ccccc2c1=O Nc1cc(C(=O)NCC(CNC(=O)C(F)CC2CCOC2)S(C)(=O)=O)ncc1F c1(CC)cccc(C)c1C(=O)NCC1COC(CNC(C2OCCO2)=O)C1 CC(C)C(C)C(CNC(=O)CC(=O)N(C)C)NC(C1CCC=CCC1)=O C1(CNC(Cc2n(C)c(S)nn2)=O)CN(C(=O)C(C)(F)F)CCC12CCOCC2 C(=O)(CC(C(C)OC)NC(C1C2CCC(F)C12)=O)N(CCCC)CCCC CC1CCC=C1C(=O)N1CCN(C(c2ccn3ccsc23)=O)C(C2CCC2)C1 C1(C(=O)OC)CCN(C(=O)NCc2ccn(C(F)F)n2)C12CCC2 c1(OCC(=O)NCCCN2CCCCC2)cccc(F)c1F c1(C(=O)NCC(CN(C(C(C)OCCOCC)=O)C)C)cccc2c(C)[nH]nc12 N1(C(C2(c3cccnc3)CC2)=O)CCN(CCCNC(C23CCCC2C3)=O)CC1 c1(NC(c2nnnn2C2CC2)CCOC)ncnc2c(F)c(Br)ccc12 n1(CCC(=O)NCCOC(CNC(CC(C)(F)F)=O)(C)C)cc[nH]c(=O)c1=O C1(NC(c2ccnn(C)c2=O)=O)CC2CN(C(=O)CN3CCC(C)(C)C3)CC2C1 c1(C(=O)NC2(C3N(C(C(C)CO)=O)CCCC3)CC2)csc2ncnc(O)c12 CCC(CCCC(=O)NC1CC1(C)N(C)C)NC(C1CCOC1C(C)C)=O N1(C(CSCC)=O)CCC(NC(c2ccc(-n3cncn3)cc2)=O)C(O)C1 C(=O)(C(CC1CCCC1)NC(C1(SC)CC1)=O)NC(CC)CN1CCCC1 N1(C(C=CSC)=O)CCC(NC(c2cc(C(C)(C)C)oc2C)=O)C2(CCC2)C1 O=C(N=c1ncc(F)c[nH]1)NC1CCC(c2nc3ccccc3[nH]2)CC1 C(c1ccc(F)cc1)=C(C)C(=O)NCC(C(C)C(C)C)NC(=O)CCCC(C)=O c1(OC)cc(C(N2CCN(C(=O)C3=CCSC3)C(C)C2)=O)ccc1C C1(COC)(CN(C)C)CCCN1C(=O)CC1(C(=O)NC2CCCC2CF)CCC1 C1(CNC(COCC(C)C)=O)CC(F)(CNC(=O)CNC(=O)CSC(F)F)C1.C1CC1 c1(C2C(C(=O)NCC3CCCCO3)C2)nc(-c2cccs2)nn1CCC(F)(F)F N1(C(C23CCC(CC)(OC2)C3)=O)CC2(CCN(C(C3C=CCC3)=O)C2)C1 c1(C(=O)NCC(CN(C(CSC)=O)C)O)ccc(OCC(F)(F)F)cn1 N1(C(c2ccc(C(C)C)o2)=O)CC(NC(=O)CS(=O)(=O)CCO)CC(C)(C)C1 N1(CC(C)C)CCC(C(=O)NCC2(O)CN(C(c3nc[nH]c3C(F)(F)F)=O)C2)C1 N1(C(CCN(CC)CC)=O)CC(NC(c2cc(C)c(C)[nH]2)=O)CCC1C c1(CN2C(C)CCC2C(=O)O)cc(Cl)cc([N+](=O)[O-])c1 c1(OC)ccc(CC(=O)NC2CCCC(CCNC(=O)C=C(C)C)C2)cc1O c1(C(=O)NC(CNC(C(CCOC)C)=O)(C)C2CC2)cn2ccsc2n1 Cc1nc(C(C)C)sc1C(=O)N(CC(CO)(CO)NC(=O)C(C)CF)C CCCC(C(=O)OC)C(=O)NC(C(=O)NC1CN(C)C(C)(C)C1)C(C)C n1(CC(N2C(CNC(C3CCC(C(F)(F)F)CC3)=O)CCC2)=O)ncccc1=O c1(C(N(CC(C)NC(C=NOC)=O)C)=O)nn(-c2ccc(F)cc2)cc1C c1(C(=O)NC(CC(=O)NCC(COCC)C)C2CC2)ncccc1N N1(C(C(CO)OC)=O)CC(C)N(C(c2ccc(F)s2)=O)CC1C N1(C(Cc2c(C(C)C)con2)=O)CC2CC1CN2C(C12CCC(CO)(CC1)C2)=O c1(OC(C(=O)NCC2(NC(C(CC)C)=O)CCCC2)(C)C)c(F)cccc1F Cc1nc(CSCCC(=O)NCC2=CC2)cs1.c1(C(=O)N)cc(C(F)(F)F)cs1 C12(C(N3CCN4CCC3CC4)=O)CCOC1CS(=O)(=O)C2 n1(CC)nnnc1C(c1nnc(CNCc2cn(CCSC)nn2)s1)NC(N)=O C(=O)(C(CC(F)F)NC(=O)CC1CCC(=O)N1)NCC(C)(C)F c1(C(N2CCOCC(CNC(=O)Cc3cnns3)C2)=O)coc2c(F)cccc12 Cc1cccc(C(C)NC(=O)C(CCF)NC(=O)C#CC2CC2)n1 CP(C)(=O)c1cncc(C(=O)NC2CC2CNC(c2ccoc2)=O)c1 c1(C(=O)NCCN(CCOC)C(C2CC(F)(F)C2)=O)ccc(C(C)(F)F)nc1 N1(C(C(C=CC)O)=O)CC(CNC(=O)CC(=O)Nc2ccc(Cl)cc2)OC(C)(C)C1 C12(NC(COC(CC)C)=O)CC(C)(C1)OC21CN(C(=O)CC2C=CS(=O)(=O)C2)C1 N1(C(c2cc(OC)ns2)=O)CCC2CN(C(=O)C(C)=C(C)C)CCC2C1 C12(CC)CCC(C(=O)NC3CC(NC(=O)CC4(C)CC4)C34CCC4)(CC1)CO2 N1(C(Cn2ncc(C)c2)=O)CCC(O)(Cc2cn(C3CCCC3O)nn2)C1 C1(C)(CNC(CC2N(C(CC)=O)CCOC2)=O)CCCC(=O)N1 C1(NC(Cc2ccc(C#N)cc2)=O)C2CC3C1C3(NC(=O)COC1CCOC1)C2 C=CCC(C)(C)CN=c1[nH]c(=NCc2cnnn2C)[nH]c2ccsc12 C1(CNC(C(C#C)(C)C)=O)N(C(c2ccnc(OCC)c2)=O)CCC1(C)C c1(OC)ccc(CC(=O)NCC2(O)CN(C(c3c(Cl)c(C)nn3C)=O)C2)c(F)c1 N12CCC(=O)N(C1=O)Cc1ccc(c(F)c1)-c1ccc(cc1)C2.C=CCOC(=O)C N1(C(C(C2CC2)OC)=O)CCC2(CCCN(C(=O)C=Cc3cncs3)C2)C1 c1(C2C(=O)N2)c(C)cccc1Br.c1(C(N2CCC(COCC)C2)=O)[nH]cc(C)c1C C(c1ccccc1)=CCCC(=O)NCC1(C(C)NC(C(C)OCCCC)=O)CC1 c1(OC(c2[nH]nc(C(=O)OCC)c2[N+](=O)[O-])=O)cc2c(=O)[nH]ccn2n1 N1(C(Cc2c(C)nc(S)s2)=O)CC(NC(=O)CC2CCCO2)CC2(CC2)C1 c1(OC(C)C(=O)NC(C)CNC(c2cc(C3CCCC3)[nH]n2)=O)ccc(Cl)cc1 c1(C(C)C)oncc1C(=O)NCCC1CN(C(c2cc(Cl)no2)=O)C1 c1(C(=O)NC2CCC(CNC(c3c(C)nncc3)=O)C2)cc2cc(F)ccc2s1 c1(C(N(C2CCN(C(C3CC3C#N)=O)C2)CCC)=O)cn(CC)cn1 C(C(C)C(=O)N1CCCC1C(C)NC(c1ocnc1C1CCC1)=O)OC c1(NC(=O)Nc2ccc(C(=O)OCC)nc2)cccc(C#N)c1O Cc1ccc(C(=O)Nc2ncnc(C3CC3)n2)c(F)c1Br C(=O)(CC(C)(O)C1CC1)N1C(C(C)NC(C(C)(C)OC(C)=O)=O)CCC1 CC(C)C(C)CN(CCC(=O)N(C)CCN(C(=O)C(C)Cc1cnn(C)c1)C)C Nc1ccc([N+](=O)[O-])cc1C(=O)NC(C1CCOC1)CNC(C1CCCC1)=O Cc1cnc(C(N2CCC(C(N3CCC(CN(C)C)CC3)=O)C(O)C2)=O)c(F)c1 N1(c2nc(-c3cc(N(C)C)nc(C)n3)on2)CC(C)C(CN)C(C)C1 c1(N2CC(C(C)NC(c3cc(C)n(C)n3)=O)OCC2)ncc(S(C)(=O)=O)cc1Cl c1(C(C)C)cc(C(N2CCC(O)(CN(C)C(c3ccsc3)=O)C2)=O)ccc1F c1(C(=O)NCC(CNC(CCc2ccn(C)c2)=O)(C)C)cc2c(cn1)CCCC2 CCCC(C)(C)CC(=O)NC1C2CN(C(=O)COc3cc(F)cc(F)c3)CC12 c1(NC(C2C3CCN(C(C4CCC=CCCC4)=O)CC23)=O)ccn2nccc2c1 C=C(C)CC(C)C(=O)N(C1CCN(C(C23CC4CC2C3C4O)=O)CC1C)C c1(-n2cc(C(C)N(C)C(c3cc(Br)cn3C)=O)nn2)cccc(Cl)c1F C=C(C)C(CC(=O)NCCC1(C(=O)NC(CC)C(C)(C)O)CCC1)OCC C(C1=CCN(CC(=O)Nc2cc(C)on2)CC1)NC(C(C(C)C)OCC)=O C1(C=O)CCN(N2CCC(N(C(=O)C(C)CC3CCCC3)CC#C)C2)CC1.CC c1(C(=O)NC(C2CCN(C(c3ccc(F)s3)=O)C2)C)cccc2oc(O)nc12 C1(C(=O)NCC(C=C)O)CCN(C(C2CCCC(CF)C2)=O)C12CCC2 C1(NC(CCc2c(C)noc2)=O)(CNC(c2ccsn2)=O)CCC(F)(F)CC1 c1(C(N2CCC(CC(C)NC(C(C)OC)=O)CC2)=O)cnc2cc(Br)ccn12 CCCCC(O)CC(=O)NCC(=O)NCC(=O)NCC1CCCCN1C C1(COC)(NC(c2ccn(C(C)C)n2)=O)CCN(C(c2cn(C)c(=O)[nH]2)=O)C1 CC1Cc2cccc(C(=O)NC3CN(C(c4sccc4-n4ccnn4)=O)C3)c2O1 c1(C(N2C(C)CC(NC(C3CCCCC3)=O)CC2)=O)onc2c1CCCC2 C1(O)(COC)CCN(C(c2cc(CNC(=O)CC(C)(C)C)[nH]n2)=O)C1 C12(CNC(C3(C)C(C(C)C)C3)=O)CC(NC(=O)CSN3CCCCCC3)(CO1)C2 CC(C)CC(C(=O)N(C)C)C(=O)Cn1cc(C2(C)CCOC2)nn1 c1(CC)nc(C)c(C(=O)NCC2CC(O)CN2C(=O)CCC2CCCOC2)s1 c1(C(=O)NCc2c(C(=O)O)csc2)ccc(COc2ccccc2)cc1 C1(NC(C(COCC)C)=O)CC(F)CN(C(c2cnc(C)nc2)=O)C1 CC1=C(C(=O)NCC23CC(CN2C(C2CCC(=O)C(C)C2)=O)C3)CCC1 CCCC(C)C(CO)NC(=O)C(O)CCNC(c1ccc(Cl)s1)=O N1(C(C=C(C)C)=O)CCC2CCN(C(=O)Cn3cc(-c4ccccc4)cn3)C2C1 c1(-c2nc(C3N(C(C4(C(F)F)C(C(=O)O)C4)=O)CCC3)on2)cccc(F)c1Br C1(C(N(CCCNC(=O)C(C)(C)CCF)C(C)C)=O)CCn2nnnc2C1 C(=O)(CS(=O)(=O)C1CCCC1)NCCCCC1CN(C(C(COC)(C)O)=O)C1 c1(Cn2cc(CC(C)O)nn2)ccc(C(N2CCCC2C)=O)c(Cl)c1 C1(CN2CC(n3cc(CNC(C4C(OCC)C4C)=O)nn3)C2)CCCCC1O C#Cc1ccc(C(=O)NC2(CF)CCN(C(=O)CCSCC(N)=O)C2)cc1F C=CC1(C(=O)NCC2CCN(C(c3cc(Cl)ns3)=O)C(C)C2)CCOCC1 Cc1cc(=NC2CC=C(c3ccccc3)CC2)[nH]c(NC2CCCCCC2F)n1 C(C)(C(=O)N1CCCC(CNC(c2ccc(F)cc2Cl)=O)C1)(C(C)C)NC(C)=O O=C(N=c1cnc2ccccc2[nH]1)C1(F)CCN(Cc2ccc(Br)cc2O)CC1 C1(NC(C(F)OC)=O)CCC2(CC1)CN(C(C1CCSC(C)C1)=O)CCO2 Cn1c(C(N2CCC(C3CC3)(NC(=O)CC3COCC3O)C2)=O)cc2ccsc12 C1(NC(c2cc(OC)no2)=O)CN(C(c2oc(C)nc2C)=O)C2(CCCCC2)C1 N1(C(CSCC=C)=O)CCC(NC(c2c(C(F)(F)F)noc2C)=O)C(OC)C1 c1(COC2(Cc3c(Cn4cc(Cl)cn4)cccc3)C(OC)C2)cc(Cl)c([N+](=O)[O-])[nH]1 C(=O)(CS(=O)(=O)C(C)(C)C)NC1(CCOC)CCN(c2nnc(SC)s2)C1 Cc1c(C(=O)NC(C2(O)CN(C(=O)C(F)C(C)(F)F)C2)C)cc(C2CCC2)n1C Cc1cc(C(=O)N(C)CCN(C(=O)CS(=O)(=O)NC(C)C)C)c2cnccc2c1 C1(NC(CNC(CC)=O)=O)C2CN(C(C3(C(F)(F)F)CCC3)=O)CC12 CCC(C)C(CNC(=O)CC1(C)CCN(C(c2cc(C)n(C)c2)=O)C1)CO C1(C(=O)NC(C)Cc2nc[nH]n2)CC(F)CN(C(=O)CC(C)c2ccco2)C1 C1(CNC(C=NOC)=O)CN(C(c2nccnc2C(=O)OC(C)(C)C)=O)CCC1C C(=O)(CCCCCC(C)O)NCC(C)(C(C)C)NC(CC(C=C)(C)C)=O N1(C(C2(CCOC)CC2)=O)CCCC2(CCN(C(=O)C3=CS(=O)CCC3)CC2)C1 C1(C=O)COCCC1=O.c1(C(=O)NOCCO)cc(C(F)F)cs1 Cc1c(C(=O)NC2(CNC(=O)C(C3CCCCC3)=O)CCOC2)cnn1CCO c1(CC(=O)NCC2CCCC2C(F)(F)F)ccc([N+](=O)[O-])c(OC(F)F)c1 C(=O)(C1=CCCC1(C)C)N(CC)CC1CCCN1C(=O)COc1ccc(Cl)cc1 N12CCC(C1)NC(=O)C2C.c1(C(=O)NNC(C2CCCC2)=O)n[nH]c(=N)[nH]1 c1(OC)cc(F)ccc1C(=O)O.C1CCC(=O)N1.C1CC(F)Cn2cc(nn2)CO1 c1(C(C2CCCO2)NC(=O)NCC(Cc2ccc(F)cc2)N(C)C)cc(Br)n(C)n1 N1(C(c2ccc(CC)c(C)c2)=O)CC2CCC1CN(C(c1cc(F)n(C)n1)=O)C2 CC1N(C(=O)Nc2c(OC(F)F)cccc2F)CCC12CCOCC2 C(=O)(CCN=C(NCCC=Cc1ccccc1)NC1CN(C2CC2)CCC1C)NC CCOCCNC(=O)C(=O)N(C1(N)CCOC1)C1CC1.C1CN1 C#CCCCC(=O)NC1CCCC1CC(=O)NC1CC(=C)C1 c1(C(N2CCOC(CC)C2)C(=O)NC(CC)C2CC2)cc(OC)ccc1OC c1(C(=O)NCC2(C(C)(C)O)CN(C(=O)C3=CCCCO3)C2)cc(N(C)C)ccc1Cl N1(C(c2ccc(OC)cc2)=O)CC2(C1)CN(CC1(c3ncccc3F)CC1)C2 C1(NC(c2ccc3c(c2)CC3)=O)CN(C(=O)Cc2cnc[nH]2)C2(CCCCC2)C1 N1(C(C2OCCN(C(C3(F)C(C)(C)C3(C)C)=O)CC2)=O)CC2(COC(=O)C2)C1 c1(N(CC(=O)NCC(c2nn[nH]n2)(F)F)Cc2ccccc2)ccc(Cl)cc1 CC(C)CCCC(=O)N1CCN(C(=O)CCC(C)(C)c2ccccc2)C(C)C1 C1(C(=O)NC2CC(NC(Cc3c(OC)nccc3)=O)C2)Cc2nccn2C1 C1(C(=O)OC)(OC(=O)CCc2ccc(OC)cc2)COCC12CCC2 C1(NCc2c(C)nn(-c3ccccc3)c2Cl)COc2ccccc2C1O c1(C(=O)NCC2N(C(C3(CC)CCCC3)=O)CC2)c(C)[nH]c2ccccc12 C1(OCC)CN(C(=O)C(=Cc2ccccc2)C)CC1CNC(c1cccn1C)=O c1(C(N2CC(CCOC)N(C(c3ncoc3C)=O)CC2)=O)ccsc1S(N)(=O)=O c1(NC(=O)CSc2cncc(-c3cccc(CO)c3)c2)ccc([N+](=O)[O-])cc1 CC1CC(NC(=O)CCn2cnnn2)CN(C(c2c(Cl)cncc2Cl)=O)C1 c1(OCC(N2CCC(N(C(c3c(CC)cc[nH]3)=O)CC)C2)=O)ccc(C)cc1F C1(CN(C2CCCC2n2ccnn2)C)CCCN1C(=O)C(=O)N1CCCC1 c1(C(N2CC(CN(C)C(C3(C)CCC(=O)C3)=O)C2)=O)nc2cnccc2s1 c1(OC)ccc(C(C)C(N2CC3CC2CN3C(=O)CCCC2CCC2)=O)cc1F C(CCC(C(=O)N(CCC(O)CO)C)NC(c1ccc(O)nc1)=O)OC c1(C(=O)NCC2C(CNc3nc(SC)c(C)cn3)C2)c(C)nc2cccnn12 C1(C(C)NC(CCNC(COC)=O)=O)CCN(C(C2CCNC2=O)=O)CC1 CCCC(C(=O)NC1CC(CCC(=O)NC(C)C(C)(C)C2CC2)C1)OCC Cc1ccc2c(c1)SC(C(=O)NCC=CCNC(C1CCn3nncc3C1)=O)C2 O=C(C1CCCc2nc[nH]c21)NC1CCN(C(c2cnsn2)=O)CC1F c1(C(CCC(=O)NC2CC2CNC(=O)C2CC2)=O)ccc(F)c(F)c1 c1(C(=O)NC2CCCC(NC(CN(C(C)C)C)=O)C2)ccc(Cl)c(O)c1N c1(CC(=O)N(CCCN(C(CC(CC)(C)C)=O)C)C)c(C)nc2ncnn2c1C c1(C(=O)NCCCC(C)NC(CCCC=C)=O)cn(CCO)c(=O)nc1O C(=O)(N=S(=O)(c1cccc(Br)c1)C1CC1)C1CCC(OC(CC)C)CC1 N1(C(C(C2CC(F)(F)C2)OCC)=O)CCN(C(c2csc(=N)[nH]2)=O)CC(C)(C)C1 CC1(C(=O)NCC(C2CCOC2)NC(=O)Cc2cccc(F)c2)CCNC1=O N1(N2C(CC=C)C(C)CCC2)CCC2(CCOC2)C(CO)C1.C(=O)NCC c1(OCCC(=O)NCC(CCOC)NC(c2cc(Cl)ns2)=O)ccc(C)c(C)c1 CCCCC(O)C(=O)N1CC(F)CC1C(=O)NCC12CCCN1CCC2 C1(CC)CC(C(N2CC(CNC(=O)CCNC(=O)C(C)(C)C)CC2C)=O)CCC1=O c1(C(=O)NCCn2cc(-c3cccc(F)n3)nn2)cccc(N2CCOCC2)c1 C(=O)(C1=CC2(CCOCC2)C1)NCC12CCN(C(C3(C(N)=O)CCC3)=O)C1CCC2 C(=O)(C1=CCCN(C(C2CC2F)=O)C1)N(C)CC1(N(C)C)CCCC1 C(CCC(C)(C)C(=O)N1CCC(F)(CF)C1)NC(C(C(C)C)F)=O c1(C(=O)Nc2cc(O)ncn2)ccc2ccccn12 n1(CC(N2CC(NC(CCC#C)=O)C(C(F)F)C2)=O)nc(C2CC2)n(C)c1=O c1(C(=O)NCC2(C(C)(C)O)CN(C(C3(CC)CCOC3)=O)C2)cnc(SC)n1C c1(C(=O)NC2CN(C(C(C)NC(COC)=O)=O)C2)ccc(S(C)(=O)=O)cc1 C1(C(N(C)CC2CCCN2C(=O)CCc2ccncn2)=O)CN2CCN1C(C)C2 c1(OC)c(C(C)NC(c2nc(O)n[nH]2)C)cccc1F c1(C(N(CC(C)NC(c2nn(C)cc2C(F)F)=O)C)=O)cc([N+](=O)[O-])cn1C c1(C(c2nnnn2-c2ccccc2)NCc2cccnn2)cnc(COC)s1 c1(-n2c(C(C)NC(C(C)(C3CC3)OC)C)nnn2)ccc(C)cc1 CC1CN(C(c2ncncc2Cl)=O)CCCN1C(=O)Cc1ccc(Cl)cc1Cl C1(C(=O)NCc2onc(COC)n2)CN(C(c2ccnc(O)c2)=O)CC1(F)F c1(COC)ccnc(C(=O)NC(CNC(=O)C(c2cnn(C)c2)C)C(C)C)c1 CC(C(C)C(=O)NC1CC(n2ccccc2=O)C1)NC(=O)CCn1ccnn1 C1(c2nnnn2CCNC(=O)NC(C)(C)C)(NCC=C)CCOC(C)C1 N1(C(CC(CCC)(C)O)=O)CCN(C(c2cn(C(C)(C)C)nn2)=O)C2(CCC2)C1 c1(CC(=O)NC2C(CNC(C3(c4cc(C)no4)CCC3)=O)CC2)cc(Cl)n(C)n1 N1(C(Cc2nc(C)oc2)=O)CCOC(C)(CNC(c2cc(C(N)=O)co2)=O)C1 C1(C(N(C2CCN(C(C3CCCCNC3)=O)CC2)CC#C)=O)CC(CC)=NO1 C(C)(C(=O)N1CCOC(CCNC(=O)CC2CC(=O)NC(=O)C2)C1)(C(C)C)OC N1(C(c2nn(CC)c(=O)cc2)=O)CCC2CN(C(C3CNC(=O)N3C)=O)CC12 N1(C(CN(CC)CC)=O)C(C(=O)NCCCCCN=[N+]=[N-])C2CC(O)C1C2 O=C(NN1CCCC1C(=O)NCC1CC2(CC2)CO1)C1C2CCC(F)C12 C(=O)(C1CNC(=O)c2ccnn21)NCC(C1CCCN1C(=O)Cc1nncs1)(C)C C12(C(=O)NCC3(NC(COCCCC)=O)CCOC3)CCC(N=[N+]=[N-])C1C2 c1(CC)[nH]c(C(=O)NCC(C(C)C)NC(=O)CCC(C)C#N)c(C)c1C(=O)OC c1(C(=O)NCC(C)NC(c2ncoc2C2CCCO2)=O)cn2cccc(Cl)c2n1 N1(C(=O)C=CC(F)(F)F)CCCC2(CCN(C(=O)C(N3CCSCC3)c3cccnc3)CC2)C1 N1(C(CC(C)(C)O)=O)C2CCC1CC(NC(c1cc3ncccc3[nH]1)=O)C2 N1(C(CC2C(=O)NCC2)=O)CC2CC1CN2C(c1cc(C2CC2)[nH]n1)=O C1(CNC(COCCC#C)=O)OCCC1C(=O)NCCCN1CCC1 Cc1ncc2n1CCC(C(N1CCC1CNC(c1ccc(C(C)C)cc1)=O)=O)C2 c1(OC)c(C(=O)NCC2CCN2C(C2CCC(n3ccnn3)C2)=O)cccc1F C1(O)(CN(C(c2ccc(COC)o2)=O)C)CCCN(C(C2CCCC(CF)C2)=O)C1 C1(N(C(=O)CC2(NC(C)=O)CC2)CCC)CCN(C(C2CC3(C2)CC3F)=O)CC1 CCCCCC(C)(C)C(=O)NC1CN(C(c2cc(OC)no2)=O)C2(CCOC2)C1 C1(NC(C(CC=C)OC)=O)CC=C(C(=O)N2CC(O)CC2(C)C)C1 C1(NC(C2(C(N(C)C)=O)CC2)=O)C2CC1CN(C(c1cnc(C3CC3)s1)=O)C2 CC1(C)OC(=O)CC1C(=O)NC1C2CCC(C2)C1C(=O)NCC1CCC(=O)N1 C(=O)(C(CCC(C)(C)C)N1CC(COC(C)(C)C)C2(COC2)C1)NC1(C)CC1 c1(C(=O)NCCC2CN(C(c3c(C)ncn3O)=O)C2)nc(O)nc(O)c1N CC(C(=O)NCC1CCCN1C(C1(C)CCC(O)CC1)=O)P(C)(C)=O c1(CNC2(NC(Cc3ncn(C)c3)=O)CC2)ccc(CO)cc1 c1(OCC)cc(C(=O)NC2CC2CNC(c2cncc(C)c2)=O)ccn1 N1(C(C2N(C(C(CCC)C)=O)C3C(C2)C3)=O)CCC(C)(O)CC1C c1(OC)cc(CC2CC2C(N2CC(F)(C(=O)N(C)C(C)C)C2)=O)ccc1I C1(F)(CNC(CC=CCC)=O)CCN(C(=O)C(CCC)NC(C)=O)C1 c1(CNC(C=CC)=O)ccc(NC(=O)C(O)C2CC2)o1.C1C(C)(SC)CCCO1 N(C(=NCCN1CCCC1)NC1CC(=O)N(C2CC2)C1)CCSCC C12(NC(Cc3nnc(C)o3)=O)CC1CN(C(=O)CC1CCC(C)CC1)C2 c1(CC)ccc2cc(NC(=O)OC(C)(C)C)[nH]c2c1.C1(=O)C(CC(F)(F)F)N1C C=C(C)C1CCC(C)C(c2nnnn2CCSCC(C)(C)C)(NC(C)(C)CC)C1 C(=O)(C(C)(C)C#N)N(CCOCCN(C(C1(CC#C)CC1)=O)C)Cc1ccccc1 C(C(=O)N1C2CCC(C2)C1CC(=O)N(C)Cc1ccoc1)(C(C)(C)C)OC c1(C(N2C(CNC(Cc3ccn(CC)n3)=O)CC2)=O)cnc(F)cc1C C(C)(CC(=O)NC1(CCNC(=O)CSC(F)(F)F)CCC1)NC(=O)OC(C)(C)C C1(C(=O)NCC(F)C2CCC2)CCCCN1C(c1ncc[nH]1)=O N1(C(C(C(C)C)O)=O)CC2(C1)SCCC2NC(c1cnc(CC(C)(C)C)s1)=O Cc1nc2nccc(C(N3CC(N(C(=O)C(O)CC4CC4)C)C4(CC4)C3)=O)n2n1 c1(SC)n[nH]c2c1CN(C(C1COCC1N1CCN(C(=O)OC(C)(C)C)CC1)=O)C2 C1(NC(C(C(C)C)n2cnnc2)=O)CCCCN(c2nc(C3CCOCC3)ns2)C1 c1(C(=O)NC(CCCC)CNC(=O)Cc2ccc(F)nc2)c(F)cc(F)cc1F c12noc(c1C(C)C)NC2=O.c1(CC(C2CCCC2)OC(COCC)=O)nc[nH]n1 C(CN=c1[nH]c(Cl)ncc1[N+](=O)[O-])c1ccc(CNC(C2CCCSC2)=O)cc1 N#Cc1ccc(OCC(=O)NC2CC2NC(c2ccc(Br)c(Cl)c2Cl)=O)c(Cl)c1 C1(OC)CN(C(=O)CNC(c2cnoc2C)=O)CC1NC(=O)C=C(C)C(C)(C)C N1(C(C(CC)F)=O)CC(CNC(c2ncoc2-c2ccccc2)=O)CC1C Cc1nn(CC(F)F)c(C)c1C(=O)NCC1CC(NC(C2CCC(=O)N2)=O)C1 C1CCC2(CCCN(CC3CCCN(c4cccnn4)C3)C2)OC1 CC1N(C(C23CC(NC(C4CCCC(F)C4)=O)(C2)C3)=O)CCCC1(C)C c1(C(=O)NCC2(CCNC(c3c(CC)nns3)=O)CC2)cc(C)c(C#N)[nH]1 N1(C(C(C(C)C)NC(C)=O)=O)CC(N(C)C(C2CN(CC(C)C)C2)=O)C2(CC2)C1 c1(CN2CC(CC(=O)Nc3cc(Cl)nnc3Cl)C2)cccc2c1OCCO2 c1(C(=O)NC2CC(CO)N(C(=O)C(O)CN3CCOC3=O)C2)cc2cccn2cn1 Cc1nn(C)c(C)c1CC(N1CC2CC2(CNC(=O)Cn2nnc(=N)[nH]2)C1)=O N1(C(CCOC)=O)CCCC2C1CCN2C(C1(OC2CCCOC2)CC1)=O c1(CC(=O)NC(CNC(CCC(C)SC)=O)C2CCC2)cccc(Cl)c1F Cc1nc(C)c(C(=O)NC2(CO)CN(C(c3c[nH]cc3-c3cnn(C)c3)=O)C2)o1 c1(NC(CC)CN(C)C)ncnc(NCCOC(C)C)c1C CC1COC2(CCC2)CN1C(=O)C#CC(C)(C)CNC(=O)C#CC(C)(C)O Cc1cc(CN(CCC(=O)Nc2cc(C)nn2C)CC2CC2)cc(Br)c1 c1(C(=O)NC23CCCN(C(C(C(C)C)(C)O)=O)CC2C3)c(Cl)ccc2c[nH]nc12 Cc1c(C(=O)NC2CCC3(CCOCC3)CC2)sc2ccc(C#N)cc12 C1(C(=O)NCC2(C(N)=O)CN(C(c3c(CC)nc[nH]3)=O)C2)CC2C=CCC(C1)C2 C1(C(=O)NCCCOCCNC(CC(C)(C)C2CC2)=O)CC2(CCC2)CO1 C1(C)(NC(Cc2cn(C)nn2)=O)CCN(Cc2cc(F)ccc2F)CC1 C(=O)(C1=C(Cl)CCCC1)NCC(C(C)C)C(=O)NC(CC1CC1)C1CC1 c1(N2CC3CC(NC(C=CCC)=O)C3C2)nn(C)c(C(F)(F)F)c1[N+](=O)[O-] CCCC(CNC(C1CCN(Cc2nc(C#N)cs2)C1)=O)C(=O)OCC C1(CNC(CCOCC)=O)CCC(CO)CC1.C12CCC(C1)CC(=O)N2 c1(C(=O)NCCCN(C(c2cnc[nH]2)=O)CC)cc2nccc(Cl)c2s1 N1(C(CC(=O)NCC#C)=O)CC2CC2(NC(=O)CC(CC)c2ccc(Cl)cc2)C1 CC(C)C(O)C(=O)NC(C1CCN(C(c2cc(C3(C)CC3)on2)=O)CC1)(C)C c1(C(=O)OC)ccc(C(N2CCOC(C3CC3)C2)C(=O)NC2CCCOC2)c(F)c1 C1(CC(=O)NC2(C(=O)OC(C)(C)C)CCC2)CCCN1C(=O)Cn1cc(Cl)cn1 C1(C(=O)NCC2C3CN(C(C4(CC=C)CC=CC4)=O)CC32)CCc2c[nH]nc2C1 c1(OC)cc(CO)ccc1C(=O)NCCCCCNC(c1ccc(Cl)c(C)c1)=O C1(C)(C(=O)NCC=CCNC(C2C(C(=O)OCC)C=C2)=O)CCCN1C N1(C(=O)C#CC2CC2)CCc2c(-c3cn(CCCO)nn3)noc2C1 c1(C(N2C(C(N3C(C)CC(O)C3)=O)CC2)=O)ccc2ocnc2c1 N1(C(C(CC=C)OC)=O)CC2CC1CC2NC(c1ccc(OC)s1)=O C(=O)(CCCCC(C)C)N1CC2C(NC(C3(C(F)F)CC(=C)C3)=O)(C2)C1 Cc1nc2n(n1)CC(NCC1CC(F)(F)C1)CC2 C(=O)(C(CC(C)C)NC(=O)C(N1CC(O)C(C)(C)C1)c1cccnc1)OC C1(NC(C2(C)CCN2C(=O)COC2CCCOC2)=O)CCCC12CC2 N1(C(CCCN=[N+]=[N-])=O)CC2CC(NC(C3CCCC(CF)C3)=O)C(C2)C1 C1(NC(c2cc[nH]c3nccc2-3)=O)CC2CCC(C1)N2C(C1(CF)COC1)=O C=CCN=C(NCc1cc(Br)cs1)NC(C)(C)CCC CC(N=c1nc(N2CCCOC(C)C2)c2cnn(C)c2[nH]1)c1ncc(F)cc1F C=Cc1cccc(C(C)NCc2ccc(C(C)C(F)(F)F)cc2)n1 c1(C(N(C(CCNC(C(F)=CC)=O)C)C)=O)cnc2cccnc2c1 CC(CF)CC(=O)NCC1(F)CN(C(C2(CCO)CC2)=O)C1 c1(C(=O)NC2CC(NC(c3n(CCCC)ncc3)=O)C2)cc2c(C)nn(C)c2s1 CON1CC(C(N2C(CC(N3CC(OCC(C)(C)C)C3)=O)C3CCCC23)=O)CC1=O CC1(C)C=CC(NC(=O)C(C2CCCO2)NC(C2CCC3(CCC3)C2)=O)CC1 Cc1cc(NC(=O)CC23CCC2CN(C(C2(CO)CC2)=O)C3)cc(C)c1F N1(C(C2(C(=O)OCC)CC2)=O)CC2CCN(C(c3ccoc3Br)=O)CC2C1 c1(CC)ccc(O)cc1CCNCCC(C(CS)=O)OC(=O)OC(C)(C)C C12(C(N3CC(O)(C(=O)OC)C3)=O)CC1CCN2C(=O)CCc1ccsc1 c1(COC)cc(NC(c2cnn(C(C)C)c2-c2ccccc2)=O)ccc1Cl c1(C(=O)NCC(C)N(C)C(c2cnc(Cl)c(N)c2)=O)cc2ccncc2c(O)n1 c1(N2C(CSC)CCC2)ccc(S(=O)(=O)NC2CCC3(CCCC3)C2)c(Cl)c1 N1(C(=O)NCCCC(C)c2ccccc2)CC(C)(C)CCC1CO CC(N=c1ccnc(NC2CCN(C3CCOC3)CC2)[nH]1)c1ccsc1 C(=O)(C(C)C(=O)NCC1CN(C(C2(CCO)CC2)=O)CC1C)OC C1(NC(C(C)(C)C)=O)CCN(C(c2ncnc3cc[nH]c23)=O)CCC1CO CC12CC1CCCN2C(c1ccc(-c2ncccn2)cc1)=O.N12CCC(C1)C2=O C(=O)(C1=C2CCN=C2NC=C1)NC1CC(CNC(c2cccc(C)c2Br)=O)C1 C1(C(=O)NCC#CC(N2CC(F)(C(=O)OC)C2)=O)CC(O)C(F)C1 C=CCC(F)(F)C(=O)N1CCC(C(F)(F)F)C(NC(=O)CC=CCC)C1 C=CC1CN(C(C2CCCC2(F)F)=O)CC1NC(C1CC(O)C1)=O CC(C)(C)CCCCC(=O)N1CC(NC(=O)C(C)(C)C2CC2)C2(CCCC2)C1 N1(C(C2CCCC2C(c2cccc(Br)c2)=O)=O)CCC(c2ccc(O)cc2)CC1 c1(COC)cccc(OC2CCCC2SC)c1.c12ccc([nH]1)C(=O)NOCC(=O)N2 c1(C(=O)NCC2CN(C(Cc3cc(OC)ncc3)=O)CC2F)cc2sccc2[nH]1 C1(C(N2CCC2CNC(C2(Br)CC2)=O)=O)CC(O)(c2cccnc2)C1 N1(C(C2C(C(=O)OC)C2)=O)CCC=C(C(=O)N2CC3=C(C2)CN(C(C)=O)C3)C1 CC(C(=O)NC1(CNC(=O)CCN2CCCCCC2)CCC1)C(F)(F)C(F)F N1(C(=O)OC(C)(C)C)CC2CC(C1)C(F)(C(=O)NCCCc1cn[nH]c1)C2 c1(C(N2C(CS(C)(=O)=O)CC2)=O)c(F)cc(C(F)F)cc1F N1(Cc2nc(NC(=O)Nc3coc(Cl)n3)sc2)CCC(F)(F)CC1 C1(NC(c2c(N)cccn2)=O)CC2CCC(C1)N2C(c1cocn1)=O c1(C(=O)NC2CCC2NC(=O)C(O)C(F)(F)F)cncc2ccccc12 C=Cc1ccc(C(=O)NOCC(=O)NCCCc2cnoc2)cc1 c1(C(N2CCCC(NC(C34CC(F)(C3)C4)=O)CC2)=O)cccc2cc(O)ncc12 C1(CNC(c2ncc(F)cc2F)=O)CC(C(=O)NCC2CC23CCCCC3)=NO1 C1(NC(C2C(C)CCC2)=O)CC2(C1)CN(C(c1ccc(=O)oc1)=O)C2 C1(NC(C2CCC(SC)C2)=O)CC2CC(C1)N(C(=O)CCc1c(C)noc1Cl)C2 N1(C(CCN(C(c2cc(CC)ncc2)=O)C(C)C)=O)Cc2ccc(C)nc2C1 CC1(C)CCC(C(N2CC(C)(CCC(=O)NC3CCCC3(F)F)C2)=O)CC1 C1(C(N(C(c2ccccc2)CNC(c2cc(O)n(C)n2)=O)C)=O)CCC2(C1)N=N2 O=S(=O)(Oc1cccc2ncccc12)c1ccc(-c2ccc(F)s2)cn1 C1(C(=O)NC(C(=O)NCC(C#C)(C)C)CC2CCCC2)CCCN1C=O N1(C(CN(C(C2C(OC)(OC)CC2)=O)C2CC2)=O)CCCC(C)(N(C)C(C)=O)C1 CCC(CCOC)C(=O)NCC1CCCCN1C(c1nn(CC)cc1Cl)=O c1(CC(=O)NC2CCCC2C(N2CCC(O)(CO)CC2)=O)ccc([N+](=O)[O-])cc1 C1(NC(c2cccc(F)c2F)=O)COCCN(C(c2ccccn2)=O)C1 CC1c2ncc(C(=O)CCC3CCCC4(C3)N=N4)n2CCN1c1cc(N)ncn1 N1(C(c2nc(C)sc2)=O)CCN(C(=O)CCc2cccn2C)CC(CO)C1 C(=O)(CCCCCC(C)(C)C)N1CC(CNC(C(C)c2ncco2)=O)C(C(F)(F)F)C1 c1(C(N2CCC(NC(C(CCCCC)O)=O)C(C)C2)=O)cc(C)cn2ccnc12 N1(C(=O)Nc2nc(-c3cccc(C)c3)sc2)CC(CC(=O)O)OCC12CCC2 C1(CCC)COCCN1C(c1sccc1C)C(=O)NC1CCCCCC1 CC(C)(CCNC(C1(C)CC1(F)Cl)=O)NC(=O)C(c1cccnc1)O C(=O)(NNc1ccc(Cl)cc1Cl)C1CC(n2cc(-c3ccc(C#N)s3)nn2)OC1 N1(C(c2c(C)occ2)=O)CC2CC(NC(=O)C(C)OCCN(C)C)C1(C)C2 C1(CNC(Cc2ccn(C)n2)=O)CC2(CO1)CN(C(C1CCS(=O)(=O)CC1)=O)C2 CC(C)CC(CNC(C1CC(C)CCO1)=O)C(=O)N(C1CCC(CO)CC1)C C1(OCC)CC2(C1)CC2C(=O)Nc1cccc(C(=O)N(C)Cc2ccon2)c1 C1(C(N2CC(C)(NC(=O)CC3CC3(C)C)C2)=O)Cc2ccccc2S1 Cc1cc(F)c(F)cc1NC(=O)CC1CCN(C(c2cccc(Br)c2N)=O)CC1 C1(C(=O)NC2CCC2C(=O)NC(C2CCN(C)C2)C)(COC)CC=CC1 C(C1(C)CCOCC1)=CC(N1CCC(COC)(NC(C2CC(F)(F)CS2)=O)C1)=O N1(C(C2C3(CN(C(C(C)=CC)=O)C3)C2)=O)CC(F)CC(F)C1 CC1=CC(NC(=O)C(CNC(c2cncc(C)c2)=O)N(C)C)CCC1 C(C)(c1cccnc1)=CC(=O)NCC(CC=C)NC(=O)Cc1ccoc1 C1(C)(NC(C=C(COC)C)=O)CCN(C(=O)CCc2c(C)n[nH]c2C)CC1 C1(NC(c2c(Cl)cn(CCC)n2)=O)CC2CC(NC(c3cnsc3)=O)C2C1 Cc1ccc(C=CC(=O)NC2CCC(CCNC(=O)Cn3cnnc3)C2)cc1Cl c1(-c2cc(C)cc(F)c2)ccc2[nH]c(NC(=O)CSc3ncccn3)nc2c1 N1(CCC(CCC=C)=O)CCC2(CC1)C1CC3CC(C1)CC2C3 C1(CC(=O)NC(C2CN(C(Cn3ccc(C)n3)=O)C2)C)CCS(=O)(=O)C1 C1(C(N2CC(C(=O)NC)C2)=O)CN(C(=O)CN(c2ccc(F)cn2)C)CC12CC2 C1(CCC(N2CC(N(C)C(c3nc(C(N)=O)co3)=O)C2)=O)CC2CCC1C2 C1(NC(CCCN(C)C(C2CC3(CCC3O)C2)=O)=O)CCC2(CC1)N=N2 Cc1ccc2c(c1)C(=O)OC(C)(C(=O)N(CC(C)NC(=O)C(C)(Cl)Cl)C)C2 C1(NC(C2(CC#N)COC2)=O)CC(NC(c2cncc(Cl)c2Cl)=O)C12CCC2 N1(c2nc(C#N)cc(C)n2)CCCC2CCCC(O)C12.c12ccc(cc1)c(=O)[nH]2 c1(C(N2CCC(COC)(NC(C3CC(n4ccnn4)C3)=O)C2)=O)ccc(F)cc1O c1(C(=O)NC2C(NC(CC(C)C3CCCC3)=O)CC2)cnn2ccccc12 Cc1cccc(OCC(=O)NCC2(CNC(=O)CCOC(=O)CO)CCOC2)c1 c1(C(=O)NCC(CNC(=O)C=Cc2cnc[nH]2)F)cccn2cncc12 c1(C(=O)NCC(CC=C)NC(c2c[nH]nc2CCC)=O)cc(Br)n(C)c1 C(C(C)N=c1[nH]c(=NCC2(CF)CCC2)c2ncccc2[nH]1)OC C1(C(N2CC(N(C)CC)C2)=O)N(C(c2snc(C)c2N)=O)CCCC1(C)C c1(Cc2cncc(C)n2)ccc(F)cc1Cl.c12ccoc1CNCCCOC2=O c1(N(CC(F)(F)F)C)ccncc1S(=O)(=O)NCC1(CN(CCC#N)C)CC1 C1(NC(CCN(C)CCO)=O)CCC12CN(C(=O)CN1CCCCS1(=O)=O)C2 c1(C(=O)NC2CCCN(C(Cc3c(SC)cccc3)=O)C2)c(C)cc(C#N)cc1C c1(CC(=O)NCC(C)(C2CCC2)NC(c2[nH]cc(C(C)=O)c2)=O)cnccc1Cl c1(CC(=O)NCC2CCN(C(CC=C)=O)C2)ccc(Nc2ccccc2)cc1 C1(NC(c2ccc(C)c(O)n2)=O)CCCC12CN(C(c1n[nH]c(C(C)C)n1)=O)C2 C=CC1(C(=O)NC2CC2C(=O)NCc2cccc(OC)n2)CCOCC1 c1(CCCOC)cc(Cl)c(C(=O)NC2(CC(C(=O)CSC)C3CC3)CC2)cc1Cl CC(C)CC(F)C(=O)Nc1cnn(C2CCN(Cc3cc(Cl)ccc3O)CC2)c1 C1(CNC(c2c(C)ncnc2C)=O)CN(C(C2CC3CC3C2)=O)C2(CCC2)C1 C1(C(N2CC(n3nccc3C(F)(F)F)C2)=O)CCC(C(=O)NCCC)CC1 N1(C(CCSCCC)=O)CCCC(C(=O)Nc2cc(O)ccc2F)C1CC CCC(CNC(c1cc(C)ns1)=O)(CC)C(=O)N1CCCC1C(=O)OC C12(C(=O)NCCCc3cn(CC(F)(F)F)nn3)CCCN1S(=O)(=O)CC2 C12(CNC(C=C(C)C(C)(C)C)=O)CC(CO1)N(C(c1cnn(C(F)F)c1)=O)C2 N#CC1CCC(CC(=O)NC2CN(C(=O)NCc3conc3C3CCCC3)C2)C1 Cc1nn(C)c(C)c1SCC(N1CC(CNC(=O)CCc2cnoc2)C1)=O N1(C(c2cn(C)nc2)=O)CCNC(=O)CC1.N12CCC(C1)OCC2=O C1(C(N2CC(O)CC2CNC(=O)CCC2CC(C)C2)=O)(OCC)CCOCC1 N1(C(c2c(C)snn2)=O)CC(NC(=O)C(F)C2CCC2)C(C(F)F)C1 C1(CNC(CCSCC)=O)CC2CCC1N(C(=O)C(C)Oc1ccc(N)cc1)C2 CCC(CC(=O)NC1CC1NC(=O)CC1CCN(C)CC1)OCCOCCOC c1(CCC(=O)NC2(CNC(c3cnc[nH]3)=O)CCC2)c(F)cccc1F C1(C2CC2)(CNC(C(C)OC)=O)CCN(C(C2(OC)CCS(=O)(=O)C2)=O)C1 N1(C(COCC#C)=O)CCN(C(c2cccc(Cn3cncn3)c2)=O)C(CC)C1 C1(C)(COC(C2C(OCC)C2)=O)CCCN(C(c2nn(C)cc2Br)=O)C1 c1(C(=O)NC2CCN(C(CC3(C#N)CCC3)=O)C2)csc2nnsc12 CCCCS(=O)(=O)NCC(=O)N(C1CCN(C(=O)CS)CC1)C.C1(CS)CCCO1 C1(C(N2C(CNC(C3(O)CCOC3)=O)CC(C)(C)C2)=O)CCc2cncn2C1 c1(C(C)O)ccc2c(c1)OCCO2.c1(C=O)nnc(C(F)F)o1 c1(CC)cccc(C(N2CCC(O)(CCNC(=O)C3=CCCC3C)C2)=O)c1O c1(CN(c2cc(NC(C)CN3CCN(C)CC3)ncn2)C)nnc2n1CCOC2 C12(CNC(=O)Cc3ccon3)CCC(NC(C3CCCSC3)=O)(CO1)C2 N1(C(CC(C(F)F)NC(C(CCC)OC)=O)=O)CC2(COCC(=O)N2)C1 c1(NC(C2N(C(c3cccc(C)c3Cl)=O)C(C)CC2)=O)cc(Br)c(F)cc1I C1(C(N(CCOC)CCNC(C2CCCOC2)=O)=O)CCC(CC(C)C)C1 C(=O)(C1=CCCCCC1)N1CCCC(C(N(C)Cc2snc(C)n2)=O)C1C C#CC1CN(C(c2ncn(C)n2)=O)CCN1C(=O)CCc1nncn1C c1(OCC)cc(C(=O)NCC2CCC(NC(C3CCCC3(F)F)=O)C2)cc(F)c1 N1(C(C(C2CCCC2)OC)=O)CCC(O)(Cn2cc(C3CCN(C)CC3)nn2)C1 Cc1ccc2c(c1)C=C(C(=O)N1CCC(NC(=O)Cn3nc(C)cc3C)C1)CO2 N1(C(c2ccc(COC)[nH]2)=O)CC(NC(=O)CC2C=CCC2)CC(C)C1 c1(C(N(C2CN(C(C3CC3c3cccc(F)c3)=O)C2)C)=O)cc2n(n1)CCCC2 Cc1cc(C(N2CCC2CNC(c2c[nH]nc2C)=O)=O)c(N)c(Cl)c1 N1(C(C2(OC)CC2)=O)CCN(C(=O)CCC2CCCCO2)C(C2CCC2)C1 C1(NC(c2c(CC)ncs2)=O)CCN(C(c2cc(S(N)(=O)=O)cs2)=O)CC(O)C1 c1(NC(=O)Nc2c(C(N(OC)C)=O)cc(C)cn2)nccc2ccccc12 C1(NC(c2cocn2)=O)CC2CC(C1)CN(C(C1CC(O)C(F)C1)=O)C2 Cc1cc(C(C)(C)NC(N2CCCC(n3nccn3)C2)=O)ccc1Br c1(N(c2sccc2Cl)C(C(N2CCCC(N(C)C)C2)C)=O)ccc2c(c1)OCCO2 C12(CNC(C3CCCCCC3)=O)CC1CN(C(N1CC3C=CC1C3)=O)C2 N1(C(CCc2nc(C)sc2)=O)CCC(C)(C)C(CNC(c2ncc(Cl)n2C)=O)C1 C1(CNC(=O)C(Cl)=CCl)CN(C(C2CNc3ccccc3O2)=O)C2COCC2O1 C1(NC(C2C(OCC)CC2)=O)CCCC(NC(c2nnn(C)c2CC)=O)C1 Cn1ccc2nc(Cl)[nH]c(=NC=O)c12.COCC(=O)NC12CCCC1CCC2 c1(C(C)=O)ccc(C(N2CCCC2CCNC(=O)CCc2cnco2)=O)c(Cl)c1 c1(C(=O)NCCC(CNC(C2CCN(OC)CC2)=O)O)cccc2sncc12 C1(C(=O)NC(C2CCCCC2)C(=O)N2CC(OC(F)F)C2)C2CCCCC12 N1(C(COCCC)=O)CCCC2CN(C(c3cnc(N)cc3C)=O)CC12 c1(NC(CCCCC)=O)cc(OC)ccc1NC(n1ccnc1)C1CC1 c1(C(=O)NC(C)CNC(C2C(C)CC2C)=O)ccc2c(n1)NC(=O)CO2 C(N=c1ccnc(N(CCC(C)(C)C)C)[nH]1)c1c(OC)nn(C)c1 n1(CCC)nc(C)c(C(c2nnnn2C(C)(C)C)NC(C)C(C)S(C)(=O)=O)c1C C1(C)(CNC(C2C(=C)CC2)=O)CC(NC(=O)CC2CC(C)=NO2)C1 C1(OC=O)COc2ccccc2O1.N1(N(C)C)CC2CC(C=O)C(C2)C1 C12(NC(CCOCC#C)=O)CCC(CNC(=O)C(C)n3ccnc3)(C1)OC2 N1(C(CCC)=O)CC(O)CC1(C)C(N1CC(CC(F)F)C1)=O n1(CC)cc(NC(=O)C(C)CN(C)C(=O)Nc2ccccn2)c(C)n1 N1(C(CC2CCC(C)(C)C2)=O)CC2CC1CCC2NC(=O)Cc1cnns1 c1(C(N2CC(O)(CNC(C(C)(C)F)=O)C2)=O)nccc2c(Cl)cccc12 C1(C(N2CC(=O)NCC2C)=O)(OC)CCN(c2nnnn2C)CC1 C1(CNC(CC(C)C)=O)CN2CCN2C1.C1(C#N)(C=O)CC=CC1 C1(NC(C2CCC(=C)CC2)=O)COC2CN(C(C3(CF)CC3(F)F)=O)CC12 n1(C(C)C)cnc(C(=O)NCC(C2CCCC2)CNC(=O)C2CC2)c1 C1(F)(CNC(CN(CC(C)C)C(C2CCOCC2C)=O)=O)CCCCC1 CCS(=O)c1ccc(-c2ccc(NC3CCN(CC)C3=O)o2)cc1 c1(C(N2CCC(CNC(=O)C(O)Cn3cncn3)C2)=O)csc2nccn12 CC1(C(F)(F)F)CCC(C(=O)NC2C3CN(C(=O)C(F)(F)c4ccccn4)CC23)O1 N1(C(COC(CC)C)=O)C2CCC1C1CC1(NC(C1OCCC1(C)C)=O)C2 C1(O)(CCNC(C2C(C)OCCO2)=O)CCCN(C(c2ncccc2F)=O)C1 C(=O)(CC(F)(F)CS(C)(=O)=O)NCC(N(C(=O)CCn1ccnn1)C)C1CC1 N1(C(CN(OC)Cc2cccc(-c3sccc3C#N)c2)=O)CCC(O)(CO)C1 CCC(C)(CNC(=O)C(C)C1CCCC1)C(=O)N1CCN(CCF)CC1 c1(C(=O)NCC2(C)C(C)CN(C(COCCC=C)=O)C2)c[nH]c2cc(Cl)ccc12 c1(OC)ccc2c(c1)nc(NC(=O)Cn1ncc(Br)n1)n2C C1(NC(C(N2CCOCC2)C)=O)C2CC(O)C1N(C(=O)CCP(C)(C)=O)C2 C1(CNC(C2C(C)=C2)=O)CC2CCC(C1)N2C(c1sc(OC(=O)N(C)C)nc1C)=O C1(C(=O)NC2CCC(CNC(=O)CCCC3CCCC3)C2)CCC2C1C2(F)F C1(NC(C2C(C)C2C)=O)CN(C(c2cccc3[nH]ncc23)=O)CC2(CC2)C1 Cn1cc(NC(=O)NCC23CC=CCN2CCC3)cc(Br)c1=O C12(C(CO)NC(c3n[nH]cc3CNC(C3OC4CCC3C4)=O)=O)CCC(CC1)C2 c1(C(=O)NCCN(CCOC)C(c2cnc(Cl)cn2)=O)cnc2c(c1)CCOC2 C=Cc1cncc(C(N2CC(C(F)(F)F)C(CNC(=O)CC(=O)N(C)C)C2)=O)c1 N1(C(CSCCCC)=O)CCC2CN(C(=O)C(C(C)C)OC)CC12 C1(N(C(C=CC(CC)C)=O)C)CCCN(C(=O)CN2CCC(C)(C)C2)CC1 c1(CNC(COC2CCN(C(CCCSC)=O)C2)=O)cc(O)cc(F)c1 N1(CC(=O)NCC(CO)NC(C(COC)OC)=O)CCC(NC(=O)OC)CC1 c1(C(N2CC(C(C)NC(C(CC)C#N)=O)OCC2)=O)cnc2sccn2c1=O N1(C(C(F)=CCC)=O)CCC(N(C)C(c2cc(C(F)(F)F)cc(Cl)c2)=O)C(C)C1 C12(C(=O)NCCCC#C)CCC(CC1)N(C(C1OCCCC1(C)C)=O)C2 N1(C(COCCCC(C)C)=O)CC(NC(C2CC2C2CCCO2)=O)CC1(C)C C1(C(C)C(=O)NCC2CCCC2C#N)CCN(C(=O)CC#N)CC1 C(=O)(CC(C)C(F)(F)F)N1CC2C(C(=O)Nc3c(C)nsc3)(CC2)C1 N1(C(c2ncc(C)c(C)c2)=O)CCC(NC(c2cc(C)c(C)o2)=O)C(CO)CC1 Fc1cc(NCc2cc(Cl)sc2Cl)ccc1NCC(F)(F)F O=S(=O)(c1ccc(NCCCCF)cc1Cl)NC(c1cnccn1)c1ccccc1 C1(N)CC2CC(NC)CC12.C1(C(C(=O)C(c2cnc(C3CC3)o2)=O)O)CCOCC1 C(=O)(CC(C)(O)COC)N(C(C)CNC(c1csc(-c2cn[nH]c2)n1)=O)CC CCC(COC)C(=O)NC(CNC(c1ccc(OC)s1)=O)CCOC C(C(C)(O)C(C)(C)C)NC(C(C)OC)=O.C(=O)CC=C(Cl)Cl N1(C(c2c(C)nn(C)c2)=O)CC2(CCC(NC(C3OCC4CCCC34)=O)CC2)C1 CC1=C(C(=O)N2CCC(O)CC2)CCO1.C1(N)CCC(c2cn(C(C)C)nn2)CC1 c1(CC)c(C(=O)NCCOCCCNC(=O)C(C)CN2CCCCC2)nnn1C C1(O)(COC)CCSC1C(=O)NCc1cc(C)oc1C c1(OC)cc(F)c(CC(=O)N(C(C)CNC(=O)CC(C)n2cccn2)C)c(F)c1 c1(C(C)(C)C)cn(O)nn1.C1(CC2CNC2)CCCN1C c1(C(=O)NCC(C)N(C(C2(N3CCCC3)CC2)=O)C2CC2)ccnn1CC(F)F C1(CNC(C2N(S(C)(=O)=O)CCC2)=O)CC(F)(F)CN1C(=O)CC1(C)CCOC1 C#CC1CC2CCC1N(C(C1CCN(C(=O)CC(C=C)CCC)CC1)=O)C2 C1(CNC(C2CCC(=C)CC2)=O)CC2(CCN(c3nc(OC)ncc3Cl)C2)CO1 C1(N(C(CN(C(C(C)C)=O)C)=O)C)C2CN(C(=O)CC(C)(C)C)CC12 C=CC(C)CC(=O)NCCC1CC(NC(c2c(C)noc2C(F)(F)F)=O)C1 N1(C(c2c(OCC)scc2)=O)CCC2(NC(=O)CCSc3ccc(C)cc3)CC2C1 N1(C(CCOCCCNC(Cc2nc(C)oc2)=O)=O)CC(CO)C(C2CC2)C1 c1(C(N(C)C)=O)cc(C(=O)NC2(CNC(=O)CCCSC3CC3)CCOC2)ccn1 c1(C(N2CC(C)(NC(C(C)Cc3ccccc3)=O)C2)=O)n[nH]c2c1NCCC2 C1(C(=O)NCC(C)(O)CNC(C2(C3CC3)CC2)=O)CCC(=O)N(C2CC2)C1 C1(C(N(CCC)CCNC(C2CCCN2S(=O)(=O)CC)=O)=O)CCS(=O)(=O)N1 CC(C)(CO)C(=O)N1CC(C)(NC(=O)CSCc2ccccn2)C1 c1(C2N(C(C(C)NC(C=C(COC)C)=O)=O)CC2)ccccc1 N1(C(c2nn(C)c(F)c2)=O)CCN(C(=O)C(C)(C)C2CC2)CC2CCCCC12 C(c1ccc2cc(F)ccc2n1)=CC(=O)NC1C(CNC(c2c(C)onc2)=O)C1 C1(C(N(CC(C)CNC(c2cnn[nH]2)=O)C)=O)CC2(CCOC2)C1 C(=O)(CCCCC(C)(C)OC)N1CC(CCC)N(C(c2ccncc2C)=O)CC1 C1(C(N2CC(CNC(CN3CCC(OC)C3)=O)C(C)C2)=O)CCCC(=O)N1C c1(C(C(=O)OC(C(CN(C)C)c2ccccc2)=O)(F)F)cccc(F)c1F Cc1cc(C(N2CC3C(CNC(=O)C=CC4CCCC4)C3C2)=O)c(C)nc1C c1(CCC(N2C(C)(NC(=N)NCC(F)F)CC2)=O)ccc(Br)cc1.CO c1(C(N(C(C)CNC(c2cc(N)ccc2F)=O)C)=O)coc2c(Cl)cc(F)cc12 c1(C(=O)NCC(CNC(=O)C=CCF)OC)c(Cl)ccc2c1OCO2 N1(C(CSCC#C)=O)CC(C(=O)NC2(C(=O)OC)CCC2)CC2COCCC12 Cc1nn(C2CC2)cc1C(=O)NCCNC(c1cnc(S)o1)=O.C1(CN)CCSC1 CC1CN(C(=O)CCn2cnnn2)CC1NC(=O)CCn1cnc(=N)[nH]1 CC(c1ccsc1)=CC(=O)NCC1N(C(=O)OC(C)(C)C)CC1(C)C C(=O)(CS(=O)(=O)C1CCCC1)N1CC2(CC)CC1(CNC(=O)C=CC(C)(C)C)C2 C1(C2N(C(Cc3n(CC)cnn3)=O)CC2)CCN(CCCC(N)=O)CC1 C1(OC)CN(C(=O)C(C)(C)c2cccs2)CC1NC(C1CCC1)=O c1(C(=O)NC2CCC(C)N(C(=O)CN3CCCCCC3)C2)cnc2sccc2c1 C=C(C)CCC(=O)NC(CNC(=O)C(c1cnccn1)C)CCCC N(C1COc2ccc(O)cc21)Cc1cc(C)nnc1C Cc1cc2nccnc2cc1C(=O)NCCC(C)(C)NC(c1ccccc1O)=O CCC(C(=O)N(C1CCCCC1)CCNC(C1COC(=O)O1)=O)C(C)(C)CC c1(CC(=O)NCC(C)NC(CC(=O)NCC)=O)cc[nH]c(=N)c1 c1(C2(C(=O)NC3CCC(N(C)C(C4SCCCS4)=O)C3)CC2)ccc(F)cn1 c1(C(=O)NCCCNC(c2c(C)nc(=N)[nH]c2)=O)nc(Br)c2n1CCCC2 C(C(=O)NCC(C1CCCC1)NC(=O)CC1NC(=O)NC1=O)(C(C)(C)C)OC C1(C(=O)NCCOC(C)C)CCCC1CNC(c1cc(Cl)c[nH]1)=O N1(C(CCOCC#C)=O)CC(C(=O)NC2CN3CCC2C3)C(F)C1 Cc1cnc2nc(C(=O)NCC3C=CCN3C(C3CCN(C)C(=O)C3)=O)nn2c1 c1(NC(CC2CCN(Cc3nc(CC)sc3)C2)=O)ncc(F)c(N(C)C)n1 C1(CNC(c2cn(C)nc2Cl)=O)(NC(c2ccncn2)=O)CC2CCC1CC2 C12(C(=O)NCC3CC(C)N(C(=O)C4=CCC4)C3)CCC(N(C)C)(CC1)CC2 CC(C)(CO)C(=O)NCCCNC(=O)Cc1ccnn1C1CCOCC1 C1(C(N2C(CNC(CS(N)(=O)=O)=O)CCCC2)=O)CCCC2CCCCC12 C(=O)(CCCCC(F)(F)F)NCC1(C)CC(NC(=O)Cc2cncs2)C1 c1(C(=O)NC2CC(NC(CCC#CC)=O)CC2O)ccc2c(c1)CC(=O)NC2 c1(C(=O)NCC(CC)NC(c2cnc(O)c(C)c2)=O)ccc(O)nc1Cl c1(C(C)=O)cc(C(=O)NCC2CCCCC2NC(c2ccc(F)s2)=O)ccc1O CC1(C)CC(=O)N(CC(=O)NCCNC(=O)C(O)CCCc2ccccc2)C1=O c1(NC(C2(c3ccccc3)CCO2)=O)ccc(-n2ncc(O)c2)cc1 S(=O)(=O)(c1cccnc1N1CCN(C2CC2)C(C)C1)N1CCCC(CC=C)C1 CCCCC(C(=O)NC(C(N1CC(F)(C#N)C1)=O)c1ccoc1)C(C)C C1(CCC=C)CCCN(C(c2cc(-c3cccnc3)nn2CC)=O)C1 CCCCC(C(=O)NCCc1cnco1)NC(c1cnnc(C)c1C)=O C1(NC(C=NOC)=O)CCCC(NC(=O)C(c2cscc2Br)=O)C1 C=CCC(C)(C)CNC(C1CCC1CNC(c1ccnc(CO)c1)=O)=O CC(C(CO)NC(C1CCCN1C)=O)NC(=O)COCCN(C)C S(=O)(=O)(c1cc(Cl)cc(Cl)c1)N1CC2(CN(C(CCC(=O)NC)=O)C2)C1 C1(C(N(CC(F)(F)F)CC)=O)CCN(Cc2n(CC=C)nnn2)c2ccccc2C1 c1(C(C(=O)NC(CC)C)N(C)CC2CCN(CCO)CC2)cnc(C)n1C(F)F C(=O)(C1=CCC(C)(C)CC1)NCC1C(NC(c2c(C)nn(C)c2N)=O)C1 CC(C)(O)CC(=O)N1CCC(CC(=O)NC2COC(C(F)F)C2)CC1 C(=O)(CC1=NN(C)C(=O)C1)N1CCC(=C)CC1C(N1CCCCC1COCC)=O C1(NC(c2ccc(C(F)(F)F)o2)=O)CCCCC1NC(C1CC12CCC2)=O c1(C(F)(F)F)ccc(N2CC(c3ccc(F)nc3)C2)nc1 N(C1CCC(NC(c2cc(C)nnc2O)=O)c2ccccc21)C(CC(=O)OC)=O CC12CC(C(N3CCC(NC(=O)C4=COCCO4)C(C)(C)C3)=O)(C1)C1(CCC1)O2 c1(CC(=O)NCC=CCNC(C(c2n(C)ncc2)(C)C)=O)ccccc1S(C)=O C1(Cn2cc(C(CC)(C)O)nn2)CN(C(=O)Cc2ccnc(C(F)(F)F)c2)CCO1 Cc1nc(-c2cc(Cl)sc2Cl)sc1NS(=O)(=O)CCBr N1(C(CC(C)F)=O)CC2C(c3cn(CC4CCCCCC4)nn3)C2C1 N1(C(c2c(OCC)cc(Cl)cc2)=O)CCC2C1CCCN2C(=O)C1=CCCSC1 C1(CC)CN(CC(=O)Nc2cccc(OCC(Cl)(Cl)Cl)c2)CCO1 c1(C(=O)NCCCN(C(=O)CC2CCCC(F)(F)C2)CC)cncc2sccc12 N1(C(CCCN(C)C)=O)CCn2ncc(S(C)(=O)=NC(=O)C(O)CN(C)C)c2C1 C1(NC(c2cnc(CCC)s2)=O)CCCC(NC(=O)Cn2cc(C3CC3)cn2)C1 N1(C(C2COCC(C)O2)=O)CCC(C(=O)NCC(C)OC(F)F)C(O)C1 N1(C(CNC(=O)OCC)=O)CCC(n2cc(-c3cnn(C(C)(C)C)c3)nn2)CC1 C1(NC(CC(C)CF)=O)CC2CCC(C1)N2C(C1CC(C(F)(F)F)C1)=O C=CCC(CNC(C1(CSC)CC1)=O)NC(=O)C(C)CC1CC1 C1(NC(C2CCOCC2)C#C)CCN(C(=O)CCS(N)(=O)=O)CC1(C)C N1(C(COCC#C)=O)CC2CC(NC(=O)C(c3ccc(F)cc3F)(C)C)CC2C1 c1(CC(N2CCCC(OCCC=C)C2)=O)cc(F)ccc1Br C#CCCC(C(=O)Nn1cc(C2CC2)nn1)NC(c1cccc(CSC)c1)=O c1(C(N2C(COC)(CNC(=O)CC3CC3(Cl)Cl)CCC2)=O)cccc2scnc12 N1(C(C(CC)=CC)=O)CCCC(NC(C2CCCN2C2CCCCC2)=O)CC1 C1(CNC(c2cc(C)c(Cl)s2)=O)CC2(CCN(CCc3ccoc3C)CC2)CO1 C1(C(=O)NCC2(OC)CN(C)C2)N(C(=O)C(O)CC(N)=O)CC12CCCC2 c1(N2CCCC(CN(C)C(c3ccc(C(N)=O)nc3)=O)C2)ncnc2c1CCC2 CC(C)(CC(F)C(=O)NC1COCC1O)NC(=O)C(O)CC(F)(F)F C=CC1(CC(=O)NCc2nc(C3CC3)no2)CN(C(=O)CC(C)F)C1 C(CC)(CC(F)(F)F)NC(COCC(N1CCC(CCC(=O)CCC)C1)=O)=O CC1(CCCC(=O)NCCC2(CNC(=O)CNc3nccs3)CC2)NC(=O)NC1=O N1(C(C(CC)CCN(C)C)=O)CC(C2CN(C(C3(C(=O)NC4CC4)CC3)=O)C2)C1 N1(C(c2c(C)scn2)=O)CCC2(CC1)CC(NC(C1(F)CCCOC1)=O)CO2 C12(NC(C(C)NC(N)=O)=O)CCCC(NC(C3C(C)C3C)=O)(C1)C2 c1(CC(=O)OC)ccc2c(c1)CCOC2C(=O)N1CCC(C)c2ccccc21 C(=O)(C(F)(F)C(C)(C)O)NCC1(C)CCCN(C(c2nccc(CC)c2)=O)C1 c1(CC)nnc(C)cc1C(=O)OC1CC(F)CN1CC C1(C(=O)NC2CCN(C(C3C(C)CC3)=O)C(C)C2)COC2(CCC2)CO1 c1(CCC(=O)NC2CCN(C(C(C(C)C)NC(COC)=O)=O)C2)nnc(O)nc1O c1(CC)ccc(C(=O)NC2CC(NC(c3cc(C4CCOC4)[nH]n3)=O)C2)c(O)c1 Cc1ccc(C(=O)NC(C2(O)CCN(C(=O)C(C3CC3)C3CC3)C2)C)nc1C Cc1cccc2oc(N3CC4(C3)SCCC4NC(=O)CC3CC4(CCC4)CO3)nc12 CCCC(C(=O)NC1(CNC(=O)C(c2cnn(C)c2)C)CCCC1)C(C)C C(=O)(C1=CCC2(COC2)OC1)NC1C(NC(C(C)(C)C2CCC2)=O)CCC1 C(=O)(CS(=O)(=O)C1CC1)NCC1(CC=C)CN(C(=O)C=C(C)c2cccnc2)C1 N1(C(C(C(C)C)NC(C)=O)=O)CC2CCN(C(C3(NC(C)C)CC3)=O)CC2C1 C=Cc1cncc(C(N2CCCC(CC(=O)NCC=CC(C)(C)C)CC2)=O)c1 Cc1nn(C)c(C)c1CC(=O)N(C1CC2CC1N(C(c1ccncc1)=O)C2)C c1(C(=O)NCc2cccc(OC(F)F)c2)cc(Cl)c([N+](=O)[O-])cc1F C(=O)(C(O)CCC(C)C)NC(CCC)CNC(C1CCC(=O)N(C)C1)=O N1(C(c2c(SC)nn(C)c2)=O)CCCC12CCN(C(=O)C1=CC3CC=CCC13)C2 C1(C(N(CC(=O)Nc2scc(C)c2OC)CCOC)=O)CCCC(OC)C1 S(=O)(=O)(CCC(=O)NCCCCNC(=O)CN1CCCNS1(=O)=O)N(C)C C(=O)(C1=CC2(CCOC2)C1)NC(C1(O)CN(C(C2C(C(=O)OC)C2)=O)C1)C c1(COCCNC(C(n2cc(Cn3ccnn3)nn2)C)=O)ccc(C#N)s1 c1(OC)ccc(C(=O)NCc2c(C)nsc2Br)c2c(C)[nH]nc12 c1(C(N2CCCC(CN(C)C(c3c[nH]c(C#N)c3)=O)C2)=O)cc2scnc2[nH]1 CC1(C)C(NC(C)CCCc2ccccc2)CC1(F)F N1(C(C2(NC(C(C(CC)CC)C)=O)CCSC2)=O)CCCC(C2CCC2)C1 C1(C(N2C(C)CN(C(c3ccc(O)cc3Cl)=O)CC2)=O)CCCN(S(N)(=O)=O)C1 C=CCC(CC(F)F)NC(=O)CN(C(=O)C(C)C(F)F)C CCC(C)(C#N)C(=O)N1CCOC(C(=O)NOCC2CCOCC2)CC1 c1(C(N(C)CC2(O)CN(C(CCCC(=O)N(C)C)=O)C2)=O)ccc2snnc2c1 C1(=O)C(CC(C)C)ONC(=O)C2CCC2N1.N1(CCC)CCC(COCC)C1 C(=O)(C1c2ccccc2C2CC1C2)N1CC(CN(C(CSC)=O)C)OCC1 C1(C(=O)N)C2CCC(C2)N1C(c1ccnn1CC(C)C)=O.c1(OC)ccccc1CO CN1CC(C(N2CCC(n3cc(CC(C)(C)C4CCC4)nn3)C2)=O)CCC1CO N1(C(CC(=O)NCC#C)=O)CCCN(C(c2nc(C(F)(F)F)ccc2F)=O)CC1 c1(C(=O)NCCCCC(C)NC(C=C(C)C)=O)cc2n(c1)CCOC2 C1(F)(CNC(c2c(OC)cncn2)=O)CCCN(C(c2nccnc2C)=O)C1 CC1OCCN(C(=O)CCCn2cccc2)C1C(=O)NCCC(C)(O)C1CC1 N1(C(c2sc(C)c(Br)c2)=O)CCN(C(=O)C=CC2CC2)C(CC(C)(C)C)C1 [N-]=[N+]=NC1CCN(C(=O)CC2C3CCCC3N2C(=O)CCc2cncs2)CC1 c1(CN2CC(CNC(C3CC4COCC4C3)=O)C3(C2)CC3)cnc2ccccn12 CC1=C(C(=O)NCC2CCCCN(C(C3CCCC3O)=O)C2)CCC1 c1(C(N(C(CNC(C(CC)F)=O)C)C)=O)cccc(CC)c1N N1(C2CCCN(C(C(C)N(C)C)=O)C2)CCN(C(C2(C)COC2)=O)CC1=O CCC(N=c1[nH]c(=NCCc2nccnc2C)c2sccc2[nH]1)C1CCC1 c1(C(=O)NCC2CCCC(NC(C3CC(N(C)C)C3)=O)C2)nc2cc(F)ccc2s1 C1(NC(CC)=O)CCCC12CCN(C(c1cc(Cl)c(Cl)c([N+](=O)[O-])c1)=O)CC2 c1(CC(=O)N(CC(C)NC(=O)C(F)(F)c2cnnn2C)CC)cccnc1C c1(C(=O)NCCCN(C(C(CCC)CC)=O)C2CC2)ccc2nnc(O)n2c1 c1(-c2ccc(C)cc2)ccc(F)c(OC)c1.C1(C)(C(=O)NCCOC)CCN1CO CC(C)(CC(=O)N1CC=CC(NC(C2CC2CF)=O)C1)CC(=O)c1ccccc1 C1(CNC(C(CC#C)C)=O)(CO)CCN(C(c2cc(C(N)=O)co2)=O)CC1 C1(C)(C(N2CCC(N(C(c3c(CC)nccc3)=O)CC)CC2)=O)CCCC(F)(F)C1 c1(C(=O)NC2CC(CNC(C(C)N(C)C)=O)C2)ccnc2c1CCO2 C(CC(C)C(=O)NCC(C)(C)NC(=O)CC1COCCN1C)=CC C1(C(=O)NC2(CNC(c3cc(O)cs3)=O)CCC2)COc2ccc(Cl)cc2O1 S(=O)(=O)(c1ccc(N2Cc3cccc(F)c3C2)c(Cl)c1)NC1(C)CCOC1 C1(NC(N2CC(CC(N)=O)C2)=O)CCCC(CC2CC2)C1 C(c1cccs1)=C(C)C(=O)NC1CCC(CNC(C2CC(=C3CC3)C2)=O)C1 N1(C(c2cc(C)nn2C)=O)CCC2(CC1)CC(C)N(C(=O)CSc1nc[nH]n1)C2 c1(C(=O)NC2CCC(NC(c3n[nH]cc3Cl)=O)CC2)cc(C(F)(F)F)ccc1O c1(C(N2CCCC(COC)(NC(=O)CS(N)(=O)=O)C2)=O)csc2ncnc(O)c12 N1(C(C=Cc2ccc(C)cc2Cl)=O)CCCC2C1CCN2C(=O)CS(C)(=O)=O CCCCCCCCCC(=O)NC(CNC(c1scc2c1OCCO2)=O)CC C#Cc1ccc(C(=O)NC2(C)CCN(C(C3CCC(C)(C)OC3)=O)CC2)cc1F C(CCCC(=O)N1CCC1CCC(=O)N(C)Cc1ccc(F)cc1)NC(C)=O N1(C(C=CC)=O)CCC(NC(C2CC(CC3CC3)C2)=O)CC(O)C1 C1(C(=O)NCC(C)C)CC12CCN(C(=O)C(C)CC1CCC1)C2 CC1(C)COC(CC(=O)NCC(O)CNC(c2cnn(-c3nccs3)c2)=O)CO1 CC1=C(C(=O)NC(C(=O)NC(CC2CCCC2)CO)C2CCC2)CCCO1 Cc1nn(C)c(Cl)c1CC(=O)NC(CNC(C1(CO)CCC1)=O)C1CCC1 c1(CCC)ncoc1C(=O)NC1CCCC1NC(c1conc1CC)=O C(CC(C(=O)NC1(CC(=O)NC(CO)C2(C)CC2)CCCCC1)OC)OC c1(CNC(CN(C)C(N)=O)=O)cc(C(=O)NC2(CC3CC3)CCC2)n(C)n1 C1(NC(C2CC(F)(CO)C2)=O)CC(F)CN(C(c2ccccc2)=O)C1 c1(OC)cc(Cl)c(Br)cc1C(N1CCC(C)(CCO)C1)C(=O)NC1COC1 C1(NC(c2n(C)nnc2)=O)CN(C(=O)CCc2cc[nH]n2)CCC1(C)C c1(OC)cc(OC)c(N)c(C(=O)NC(C)CN(C)C(C2(F)CCOC2)=O)c1 c1(C(=O)NCC(C)NC(c2cc(C)nn2C)=O)ccc2[nH]c(=N)oc2c1 N1(C(CC2(C)CCOCC2)=O)CC2CCCCC2(NC(=O)CCCCC2CC2)C1 N1(C(CC2ON=C(CC)C2)=O)CCCC(N(C)C(c2cc(C)c(C)o2)=O)CC1 N1(C(C=CCCC(C)C)=O)CCN(C)CC1C(=O)NCC1CNC(=O)CO1 CCCCC(O)CNC(=O)CC(C)NC(c1c(C)noc1N)=O C1(C(N2C(COC)CCCC2)=O)CCCN(C(c2ccc(I)c(F)c2)=O)CC1 C(=O)(C(F)CC(C)C)N1CC(NC(CC(CC)C2CCC2)=O)(CNC(C)=O)C1 CCC(F)(F)C(=O)N(C)CCN1CCN(C(C2CCC(F)(F)C2)=O)CC1 c1(OC)cccc(C(=O)NC2COCCN(C(c3nccc(Cl)c3O)=O)C2)c1C C12(C(=O)NCC3(C)CCC(C)CC3)CCCCCC1OCC2 c1(C(N2CCCN(CCOC)CC2)C(=O)NCCCF)sc(=O)n(C)c1Cl N1(C(c2nc(COC)sc2)=O)CC(C)(C)CCC1CNC(=O)CSc1cn[nH]c1 C1(C(=O)NCCCCCNC(Cc2cn(CC)nc2)=O)CCCC(O)C1 N1(C(c2c(C)nns2)=O)C(C)CC2CN(C(C3CCCN3C3CCCC3)=O)CC12 c1(C(Cc2nc(CCCC)sc2)=O)nc2cc3c(cc2[nH]1)OCO3 c1(C(N2CC(CCC)N(C(=O)CC3CCCCO3)CC2)=O)c(N)cc(Cl)cc1Cl Cc1nc(C)n(O)c1C(N1CCCC(F)(CNC(=O)C2=CCCOC2)C1)=O C#Cc1ccc(C(=O)NCC(CCNC(=O)C(C)N(CC(F)(F)F)C)OC)cc1C N1(C(c2cc(COC)nn2C)=O)CCN(C(=O)CSCc2cscn2)C2CC12 C(C(C(=O)NCC(C)CN(C)C(C1CC(C)(CC)C1)=O)OC)OC c1(C(N2C(C(C)NC(c3ccc(CC)cc3)=O)CCC2)=O)cnc2nccn2c1 N1(Cc2c(C)ccc(Br)c2)CC2CCN(C(c3c(C)ccc(I)c3C)=O)CC2C1 C1(C(=O)NC(Cc2ccccc2)CO)CCCCN1C(C1CC2CCC1O2)=O N1(C(C2CCCC(C)C2)=O)CCN(C(C2CCCO2)=O)C(C(C)C)C1 C1(F)(C(=O)NC(C)CCNC(C2CC(C(C)(C)C)C2(C)C)=O)CCC(F)(F)CC1 c1(C(N(C2CN(C(C(C(C)C)N3CCCCC3)=O)C2)C)=O)ccc(I)c(F)c1F CC1CCN(C(c2cncc3c2CCC(C(=O)O)C3)=O)CCc2ccccc21 c1(NCCc2ccc(C)cc2F)nccc(=NC2CCc3nn[nH]c3C2)[nH]1 c1(OC)cccc2[nH]c(C(=O)NCCCN(C)C(C3(C)CC3F)=O)cc12 c1(NC(C(N2CC(C)SCC2)=O)=O)ccc(Oc2ccc(F)cc2)cc1F c1(C(=O)NC2(CO)CCN(C(c3cc(C)nnc3)=O)C2)cc2c(nn1)OCCS2 C(CCC(C)NC(c1cnc(C(C)(C)C)s1)=O)NC(C1C(=C)C1)=O.c12ocnc1C2 N1(C(C(C(C)C)N=[N+]=[N-])=O)Cc2n[nH]cc2C1C(=O)NCC1C(CO)C1(C)C c1(C(N2C(C(N3CC(C#N)(F)C3)=O)CCC2)=O)ccc2cc[nH]c2c1 C#CC1(CNC(=O)C2=NNC(C(F)(F)F)C2)CCOCC1 N1(C(C2CC3(CC(NC(CCNC(C)=O)=O)C3)C2)=O)CCC2(CC1)COC(=O)N2 c1(NC(=O)NC(C(=O)OC)C)ccnc(NC(C2C(O)CCOC2)=O)c1.C(C)C c1(C(N(CCCCCNC(C2CC2(C)C)=O)C(C)C)=O)ccn2cncc2c1 CC1(C(N2CC(CC(C)NC(=O)C3=CCCSC3)C2)=O)CCC(O)CC1 c1(CC(N2CCC(NC(C(CCC)(C)C)=O)C(C)C2)=O)cn2c(n1)CCCC2 C1(CC)C(C(=O)NCC(C)(C)C2CCC2)CCN1C(=O)CCN(C1CCCC1)C N1(c2nc(=NC)[nH]c(=NCC3CC4(CCC4)C3)[nH]2)CCS(=O)(=O)N2CCCCC12 CCC(CC)CC(C(=O)NCCCF)N(C)Cc1cnc(OC)cn1 CC(=NO)c1cc(C(N2CCC(C)C(NC(c3nccn3C)=O)C2)=O)cnc1O N1(C(C2N(CCC)CCOC2)=O)CCC(C)N(C(=O)CC(F)(F)CC)CC1 Cc1cccc2c1OC(C(=O)NCC1CCN(C(c3c(CO)cnn3C)=O)C1)C2 C(=O)(C(C#N)C(C)(C)C)NCc1nnc(-c2nc(C)oc2C)n1-c1ccc(Br)cc1 CC1CCN(C(=O)CSc2cccc(F)c2)CCN1C(C1C=CCS1)=O C(N=c1cc(C(F)(F)F)nc(C)[nH]1)C1CN(C(c2c(CC)nns2)=O)C1 CC1CCc2nc(N3CCCC(CO)C3)[nH]c(=NCC3SCCS3)c2C1 c1(CN2CCC(n3cc(-c4c(C)cc(F)cc4)nn3)CC2)[nH]cc2c1CCCC2 CCS(=O)(=O)c1cccnc1C(N1CCC1CNC(=O)C=Cc1cccs1)=O C12(CNC(c3c(CC)noc3C)=O)CN(C(C3(O)CCC3)=O)CC1(C(F)(F)F)C2 C(=O)(CC(C)(C)NC(=O)CCc1nc(=N)[nH][nH]1)NC1CCN(C(CC)=O)C1 c1(SCC(=O)NC(CC)CNC(=O)CN2CC=CC2)cccc(C#N)c1 c1(COC(=O)Cn2cnnc2O)cc2c(cc1Cl)OCCO2 c1(C(=O)NCC2CC(CNC(c3c(C)nc(C)s3)=O)OC2)ccn2nnnc2c1 C1(F)(CNC(C2CC(F)(F)CS2)=O)CC2CCC(C1)N2C(c1ccccn1)=O c1(OC)cc2c(cc1OC)NC(C(=O)NCc1cc(C)cc(OC)c1Br)C2 C(=O)(CC(C)P(C)(C)=O)N(CCCCN(C(C=CC(CC)C)=O)C)C C1(O)(CN(C(C(F)=CCC)=O)C)CCN(C(c2cnoc2C(C)(C)C)=O)C1 C(=O)(CC(C)C(C)(C)NC(=O)CC1OCCO1)NCCC(C(C)C)N(C)C N1(C(Cc2nc(CC)sc2)=O)CCC2CCN(C(c3cnc(Cl)s3)=O)CC12 C1(C(=O)NCCNC(c2ccsn2)=O)CC2CC12 C(=O)(C1=NOC2(CCC2)C1)NCC1C(C(=O)NCC=C=C)CCO1 CCC(C)(CO)C(=O)N1CCC1C(=O)NC(c1ncc[nH]1)CO C(c1c(F)ccc(Cl)c1F)=CC(=O)N(C1COC2(C1)CN(c1ncccn1)C2)C c1(C(N2CCC(C)(CNC(=O)CC3CC3)CC2)=O)cccc2c1C1CCC2CC1 C1(OC)CN(C(=O)C(C)CSC)CC1C(=O)NC(C1CCCCO1)(C)C CCC(F)(F)CC(=O)NCC1CCN(C(c2nc(C)ncc2Cl)=O)C1(C)C C1(C(N2CC(CCCCNC(CCCC=C)=O)C2)=O)CNC(=O)CC12CCOC2 N1(C(C(F)OC)=O)CCC(O)(CCNC(=O)C(C(C)O)Nc2ccccc2)CC1 c1(C(C(=O)NCC2CC(NC(c3n(CC)ncn3)=O)C2)=O)c(C)nn(C)c1C C(=O)(C1CCc2ccccc21)NC(C1(O)CCN(C(=O)C(C)S(N)(=O)=O)CC1)C c1(C(=O)NCCNCCn2cc(C3CC3)nn2)cnn(Cc2ccccc2)c1I c1(CC(=O)Nc2cscc2C(=O)O)ccc(F)cc1F c1(C(C(=O)NCCC)N(C)Cc2cnco2)cc(I)ccc1F N1(C(C(CC)(C)C)=O)CC(C(=O)NCc2cccc(F)c2F)C2(CC2)C1 c1(CC)cc(C(=O)NC2CCCCC2NC(c2cc(NC)ccn2)=O)ccc1F CCCC(CNC(C1CCCC(=O)N1)=O)C(=O)NC1(C)CCCCCC1 CCN=C(NCCC(C)c1cn[nH]c1)N1CC(O)C(C)(C)C1 S(=O)(=O)(c1ccc(Cl)cc1)NC(C)C(N1C(C(=O)O)CSC1C1CC1)=O c1(CC(N2CC(C(C)NC(C3CC4C=CC3C4)=O)C2)=O)nc(F)c(F)cc1F C(c1ccccc1)=CCC(C)(C)NC(C1CN(C(=O)Nc2ccccc2)CCO1)C C1(n2cc(C(CC(C)O)(C)C)nn2)CC2CCC1(N(C(C1CCCCC1)=O)CC)C2 CCN=C(NCc1ccc(NC)cn1)N1Cc2ccc(F)cc2C(C)(C)C1 Cc1ccc(O)c(C(=O)N(C(CC(F)F)C(=O)NC(CO)C(=O)N(C)C)C)c1 C1(NC(CCCCOCCN(C(=O)C=CC2CCCCC2)C)=O)CC(C)(C)CCO1 C1(NC(C2N(C(C)C)CCC2)=O)(CNC(C2(C)CC2(F)F)=O)CCCCC1 c1(C(=O)OCC)cnc(=NCc2cccnc2N(C(C2CC2F)=O)CC)[nH]c1 c1(C(=O)NC(CNC(c2ccc(C)cc2)=O)C2CC2)c(Cl)ccc2c1OCO2 N1(C(CC(C=C)(C)C)=O)CCN(C(c2cn(C)nc2C(C)C)=O)CC(CO)C1 c1(C(=O)OCC)nc(=NC2CCCN(C(=O)C(O)C3CCC3)CC2)cc[nH]1 N1(C(c2ccc(NC(=O)CCCCF)s2)=O)CCCC(NC(C)=O)C1C c1(C(N(C2CCN(C(C34CC(O)C3C4)=O)C2)C)=O)cc(CCCO)on1 C1(NC(C2C=C(C)CS2)=O)C(C)CN(C(=O)CNC(c2ccccc2)=O)CC1C N1(CC=C)CCC(C(=O)NCC#CC(=O)O)CC1 CCCCC(CNC(c1cnc(C2CCOC2)s1)=O)NC(C1(C)CCC(C)C1)=O N1(C(CNC(=O)OC)=O)CCN(C)CC1CNC(c1csc(C)c1OC)=O CS(C)(=O)=NC(=O)C(=O)NCC1CN(C(c2cncs2)=O)CC12CCC2 N1(C(CCCC#C)=O)CCC2(CC(NC(c3sccc3CC#N)=O)CO2)C1 C1(NC(C(c2cnn(C)c2)OC)=O)CCN(CC(C)(C)NC(=O)C(C)C)CC1 C(c1ccc2[nH]ccc2c1)=CC(=O)OCc1sccc1Cl C1(C(=O)NC(c2nc(O)n[nH]2)CC)(CO)CCN(C(=O)CC2CC(C)(C)CO2)C1 C1(NC(C(C(C)(C)C)O)=O)CC1C1CCCN(C(c2cc3ncccc3s2)=O)C1 C1(C(=O)NCC2(OC)CCCC2)CC2CC1CN(C(C13CCC(CC1O)C3)=O)C2 Cc1cc(F)c(N)cc1C(=O)NCC(O)CNC(c1cnc(C2CCCO2)s1)=O C1(C(=O)NCC)CN(S(=O)(=O)CC(C)(C)OC)CC1C1CC1 Cc1ccc(F)c(C(=O)NCC(C)CN(C(=O)CCc2ccccc2Br)C)n1 C1(C(C)NC(C(C)NC(C)=O)=O)CCCN(C(=O)C(O)CCN(C)C)C1 C(=O)(C(F)CC(C)(C)C)N1C(CCNC(c2n[nH]c(C)c2C)=O)CSCC1 CN1CCC(NC(N2CCC2C2CCC2)=O)C(C#N)C1 N1(CC(=O)N(C2CCN(C(c3c(C)onc3)=O)CC2)CCO)CC(=O)N(C)C1=O CC1CCN(C(=O)CC2CCNC23CCC3)CC1(F)F N1(C(C2C(C=C)C2)=O)CCCN(C(=O)CS(C)(=O)=O)CC1C c1(C(=O)NC2C(NC(c3[nH]cc(CC)c3)=O)CCC2)ccc2ccc(O)nc2n1 CCCCC(C)C(=O)NC1NCCC(CN2CCCCC2)C1 C(=O)(C(C(C)C)NC(=O)C(=O)Nc1ccc(Cl)n1C)NCC#C c1(CCC(=O)NC(C2CN(C(c3csnc3C3CC3)=O)C2)C)nc(C2CC2)no1 c1(C(=O)NC(CNC(c2c(CC)c[nH]n2)=O)C)c[nH]c2ccc([N+](=O)[O-])cc12 Cc1cn2c(n1)CC(C(N1CCCC(CO)(NC(=O)C3=C(Cl)CCCC3)C1)=O)C2 C1(NC(C2(CC(C)C)CC2)=O)CCCC1NC(=O)CN1CCCC1CN(C)C N1(C(C(C2(O)CN(C(C3CC(SC)C3)=O)C2)F)=O)CC2CCCC2C1 c1(C(=O)NC2CN(c3nc(C4CCCC4)nc(=N)[nH]3)C2)nccc2cc[nH]c12 C12(NC(CCCCCOC)=O)CCCC1N(C(C1CCOC(C)C1)=O)CC2 C1(NC(c2c(C)coc2)=O)CCCCCN(C(c2[nH]c(O)nc2C)=O)C1 c1(N)ncccc1S(=O)(=O)N.c1(C(CC(CO)N2CCCC2)C)ccccc1[N+](=O)[O-] C1(OC)(CNC(=NCCCCl)NC2CCOC(C)(C)C2)CCC(C)(C)CC1 C1(C(N2C(C)(COC)CC2)=O)CC(F)(F)CN1C(C1CCSC1)=O c1(NC(C(=O)NCC2CCCC2c2ccccc2)=O)cccc(SC)c1.c1nc[nH]n1 c1(C(=O)NC2CC(NC(C3(C)CCCCCC3)=O)C2)ccc2ncncc2c1 Cc1sc(C)c(C(N2CCC23CCC3)=O)c1C#N C1(C#N)(C(=O)NC2CCC(N(C(Cn3ncc(CC)c3)=O)C)C2)CCN(C)CC1 c1(C(=O)NCc2ccc(C(N(C)CC3COCCO3)=O)s2)cnc2ccccn12 C1(=O)C(C(C)C)C(=O)OCCCN1.CCCCCCN(CCCOC(COC)=O)C C(C1=NOC2CN(C(=O)Cc3ccc(CC)cc3)CC12)NC(CCC=CC)=O C1(OC)CC2CC(C1)N(C(=O)CCCN(C)C(C1CC(C(C)C)C1)=O)C2 C=CCCC(C)(C)C(=O)NCCSCC(=O)NCC(=O)NCCOC C1(C(N(C)CC)=O)CCCCN1C(C1CC(O)CN1C(C1CC(=O)N(C)C1)=O)=O CC1(CNC(c2sccc2Cl)=O)CC(NC(C2CC2CF)=O)C1 CC1CC(CC(=O)NCC=Cc2cccnc2)CN1C(=O)Cc1nc[nH]n1 c1(C(N(CCN(C(=O)C(C)SC(C)C)CC)CC)=O)nc(F)c(F)cc1F.CC N1(CC(=O)NC(CC)=O)CCN(C)C(=O)C1C.N12CCN(C)C(C1)CNC(=O)C2=O N1(C(C2C=CC(NC(c3cc(Cl)ncc3Br)=O)C2)=O)CCc2c(O)noc2C1 C1(CNC(c2c(CC)oc(C)c2)=O)CC2CCC(C1)N2C(=O)Cn1nccc1N c1(C(=O)OC(=O)C(CC2CCOCC2)SC(F)(F)F)ccnc(C(F)(F)F)c1 C1(OC)(OC)CC(C(=O)NCC(N2CCCC2CCO)=O)C1 CC1(C)CC(NC(c2ccc(C(C)(C)C)nc2)=O)CCN(C(C23CCC2C3)=O)C1 c1(C(=O)NC(C2(O)CN(C(C3CCC(C)(CC)O3)=O)C2)C)ccc(Cl)nc1O CC1CCCC(C)N1CCC(N1CCCC1(C)CNC(c1cccnc1O)=O)=O N1(C(c2cc(COC)on2)=O)CCN(C(c2cccc(C(N)=O)c2N)=O)C(C)C1 N1(CC(=O)NC(CN(C(C2C(C(=O)OC)CCCC2)=O)C)C)CCCCCC1=O N1(C(c2cn(C)nn2)=O)CCCC12CCN(C(=O)CCc1ccc(=N)[nH]c1)CC2 N(C)(C1CCc2ccc(Br)cc21)CC(=O)OCCC C(=O)(C=NOC)N(CC(=O)NCC1CCNC1)CC#C CC1CN(C(=O)C(F)=CCCF)CC1CNC(C1(C2CCCO2)CCOCC1)=O C=CC1(C2(C(N3CC4CCN(C(CNC(=O)OC)=O)CC43)=O)CCC2)CCC1 c1(C(CC(C)C)NC(=O)NCC(CSC)OC)ccc(C(C)C)c(Br)c1 C(CC(=C)C)(C(=O)N(C)CC1CCC1C)NC(C(C)OCCC=C)=O n1(CC(=O)NC2(C)CCN(C(c3ccsn3)=O)C2)ccc(O)nc1=O CC1CN(C(=O)CN(S(C)(=O)=O)C)CC1NC(=O)CCCCC1CCCCC1 C1(N(C)C(C2CCCCC2)=O)CN(C(C2CC2C2CC2)=O)CC12CC2 C(=O)(C1=C(C)OCCS1(=O)=O)NCCN(C(C1C(=C)CC1)=O)C(C)C N1(C(CCSC(=N)N)=O)CCC(Cc2cn(C3CCOC3)nn2)C1 N1(C(CNC=O)=O)CC2CC1C2NC(=O)COc1ccc(C(C)(C)C)cc1 C1(C(=O)NC2(CNC(C(C3CCC3)OC)=O)CCC2)CCN(c2ccccc2)C1 c1(C(NOCc2[nH]nc(CC)n2)=O)cccc(-n2cc(C(C)OC)nn2)c1 c1(OC)ccnc(N(C)CCN(C(=O)CC(C)N(C)C)CC2CC2)n1 c1(C(=O)NCCC2(OC)CN(C(C3CCC(C)O3)=O)C2)ccc2nc(C)[nH]c2c1 c1(C(N2CCCC(N(C(=O)CC(C)OC)CCC)C2)=O)ccc(OC)c(OC)c1 C1(C(=O)NCC(CC(F)(F)F)NC(Cc2cnc(C)[nH]2)=O)CCC(=C(F)F)CC1 C1(NC(c2cc(C(=O)OC)no2)=O)CC(NC(C2CCC(O)C2)=O)C12CCC2 N#Cc1ccc(C(N2CCCC(CNC(C3CCCC3O)=O)CC2)=O)cc1O C(C1=NOC2CCCC12)NC(C1(C2N(C(CN=[N+]=[N-])=O)CCC2)CC1)=O c1(SC)cccc(CN2CC(O)CC2c2cn(CC(=O)OC)nn2)c1 c1(C(=O)NCC(CCCC)NC(C(CC(=C)C)C)=O)cn2c(n1)CC(OC)CC2 C1(N(C(C(C(C)O)C)=O)C)CC2CCC(C1)N2C(=O)CC#N N1(C(C(CCOC)NC(C(C)OCCCC)=O)=O)CCCNC(=O)C1C CCCC(CC)C(=O)N1CCC(CC(=O)NCC(C)(C)SC)C1 c1(NC(CC2(NC(C(CN(C)C)O)=O)CCC2)=O)cccn2nccc12 c1(C(=O)NCC(CCC)(C)O)ccc2c(n1)CN(C(=O)CN1CCC(F)C1)CC2 N1(C(C(c2ccc(Cl)cc2)C)=O)CCC(F)C(NC(c2cc(C(N)=O)c[nH]2)=O)C1 O=C(CCCN=c1ncc(I)c[nH]1)N1CCN(CC2CCOC2)CC1 C(CCC1CCC1)(C(=O)N1CC(c2cscn2)C1)NC(C(C)SC(C)C)=O c12cc(c(Cl)cc1Cl)NC2=O.c1(SC)cc(C2CC2)ccc1F.C12CC1C(=O)N2 C1(N(C(C(C)NC(COC)=O)=O)C)CCC(NC(=O)C=CC2CC2)CC1 C1(NC(C2C(=C)C2)=O)CCN(C(c2c[nH]nc2-c2cnn(C)c2)=O)CC1C c1(C(=O)NC2CN(C(c3c(CC)[nH]c(=N)s3)=O)CC2C)cnc2ccnn2c1C CC1(C)COC(CCC(=O)NCC2(F)CC(NC(=O)CC(F)F)C2)C1 O=C(CCCCc1cnc[nH]1)N(C1CCN(C(=O)CC2CNC(=O)C2)CC1)CCO CCCN=C(NCC(C)(C)O)N1CCC(NC(N)=O)C1 c1(CC)ncc2n1CCC(C(=O)NC1CCC1NC(c1n[nH]c(C)n1)=O)C2 N1(C(C#CC(C)(C)C)=O)CCC(CNC(c2ccc(Cl)s2)=O)C(F)(F)C1 C1(NC(=O)NCCC2N(C)CCOC2)CC2CCC1(c1ccncc1)C2 CN1CCC(=CC(=O)NCCN(C2CC2CC(=O)O)Cc2ccccc2)C1 C(=O)(C(F)(CNC(=O)CC1CC=CC1)C(C)C)NCCn1c(C)ncc1 N1(C(c2c(C)sc(Cl)n2)=O)CCC(C2CC2)(CNC(C2CCCC2C)=O)C1 c1(C(N(CC(C)NC(C2CC(=O)NC2(C)C)=O)CC)=O)cc(F)c2cn[nH]c2c1 CCCCC(F)(F)C(=O)NC(CNC(c1[nH]c(C2CC2)nc1C)=O)CC(C)C c1(CCNC(C2CCNC2c2ccc(F)cc2)=O)cc(F)ccc1Cl C(=O)(C1=NOC2(CCC2)C1)NCC(C)NC(CNC(=O)NC)=O c1(-c2scc(CC)n2)cccc(NC(=O)C(CC2CCCCC2)OC)c1 Cn1[nH]c(=N)cc1C(=O)Nc1cccc(C(=O)OC(C)(C)C)c1.C12CN(C1)C2 N1(C(C2C(CNC(C(C(CC)C)N(C)C)=O)CCC2)=O)CCCC2(C=CCO2)C1 N1(C(C(c2nc[nH]n2)CO)=O)CCCC(O)(CNC(CC(CC)C2CC2)=O)C1 N1(C(CC)=O)CCC(NC(=O)C(c2cn(C)nn2)NC(=O)CC2CCCN2C)C1 c1(OC)cc(OC)cc(N2CCC(C)C2)c1.C(=O)(C=CC(C)C)NCCC1CC1 C1(NC(c2ccccc2C)=O)CCOC(CNC(C(C)N(CC)CC)=O)C1 C(=O)(C(F)C(C)CNC(=O)Cn1cccnc1=O)NCC1(SC)CCC1 NS(=O)(=O)c1ccc(C=Cc2ccc(OCC(F)(F)F)cc2)cc1 N1(C(c2c(CCC)n[nH]c2)=O)CC(NC(C2CNC(=O)C2)=O)C(C2CC2)C1 C1(NC(CSCC)=O)CCCC(C(=O)NC(C)CC2CC(C)=NO2)C1 N1(C(c2cc(CC)on2)=O)CC2CN(C(C3CC(CF)C3)=O)CCC12 c1(OC)ccc(N2CCC(NC(c3cncc(C)n3)=O)C2)cc1 CC1CN(C(c2ccc(N)c(Cl)n2)=O)CCN1C(=O)CCc1cncnc1 C1(C(=O)NC(C)CN(C)C(C2SCCCS2)=O)COC2(CCC2)CO1 CCCC(CCC)C(=O)N1CCCC(NC(c2cc(CCOCC)on2)=O)C1 C1(C(N2CC(C)(NC(=O)C(F)C3CCC3)C2)=O)CCc2nnc(O)cc2C1 c1(C(N(C(C)CNC(=O)Cc2cc(C(F)F)on2)C)=O)cc2ccoc2cc1F N1(Cc2c(C)nn(CC(=O)OCC)c2C)CCC2(CCC2)C1.CC c1(C(=O)NC(C2CCOC2)CNC(c2nnc(C)s2)=O)ccc(C(C)C)cn1 N1(C(c2n(C)c(S)nc2)=O)CC2CCC1CN2C(C1CC=CCO1)=O c1(C2C(C(N3CCOCC3)C(=O)NCC3CCOC3)C2)cccc(O)c1 C1(CC)C(C(=O)N(c2cccc(C)c2)CC)CCN1C(c1cnsn1)=O C(C)(CNC(=O)CCc1ccc(OC)cc1)(C(C)C)NC(C1C(C#C)C1)=O C1(C(N2C(C(N(C(CO)C3CC3)C)=O)C=CC2)=O)CC2C=CC1CC2 N1(C(CC)=O)CCCCC1CCC(=O)N(C1CC(C(=O)OC(C)(C)C)C1)C C1(C(=O)NC2CC(F)(CNC(CCC)=O)C2)CC2CCC1CC21OCCO1 C(=O)(CCCCC#N)N1CCC(NC(C(Cc2ccc(C)cc2)C)=O)C1C1CC1 C1(CCNC(C2(OC)CCCC2)=O)CN(C(C2(C(C)C)COC2)=O)CCS1(=O)=O c1(CCC(=O)NC(CC)CN(C(=O)C(c2ccccc2)O)CC)ccccc1C Cc1ccc2cc(C(N3CCC(O)(C(C)NC(=O)C#CC4CCC4)C3)=O)[nH]c2c1 CCCCCCC(C)C(=O)NCC1CCC(F)(F)CN1C(c1cocn1)=O c1(C(N(CC(C)N(C(=O)C=C(F)c2ccccc2)C)C)=O)ccn(C)c(=O)c1 c1(Cn2c(NCc3cc(OC)cc(OC)c3)nnn2)cccc2c(C#N)c[nH]c12 Cc1ccc(C(N2CC(NC(=O)CCc3ccc(C)nc3)CCC2C)=O)c(O)n1 N1(C(c2nc(C)oc2)=O)CCN(C(=O)CNC(=O)NC(c2ccco2)C)C2CC12 C1(C(N2CCC(NC(C)=O)C2)=O)CC12CC(NC(=O)OC(C)(C)C)C2 C1(C)(C(=O)NC2(CCCN(C)C(c3coc(C(F)F)n3)=O)CC2)C=CCCC1 CC(C)C(N)CCNC(=O)NCC(c1ccsc1)O c1(C(C)(C)NC(C(C)N(C(=O)O)CC)=O)ccccc1F.N1(CC(C)N)CCC1C C#CCC(CC(=O)N(CCN(C)C)CC)OC1CCC(C(=O)NCC=C)C1 C1(CC)CCCC1(C)C(=O)Nc1ccc(CN(C)C(=O)OC(C)(C)C)cc1 CC(C)C(CNC(=O)C(C)n1cccn1)NC(c1cnc(C(C)(C)C)s1)=O c1(N2C(C(=O)NCCC)CCC2)nc(Cl)c2c(ccn2C)n1 c1(C(C)NC(C2CCC(O)C2)=O)ccc(C(=O)O)cc1F c1(CNC(C2(S(N)(=O)=O)CC2)=O)cc2n(n1)CCN(C(=O)C1=NOCC1)C2 N1(C(CCSCCC)=O)CCC2CCN(C(=O)CCc3cnn(C)c3C)C2C1 N1(C(C(CC)C)=O)CCC2(CC1)CN(C(=O)C(C)n1cccn1)C2 c1(C(N2CCCCC2c2cncnc2)C(=O)NCCOC)cc(SC)ccc1Br N1(C(C2(CNC(c3noc(CC)c3C)=O)CCC2)=O)CCn2ncnc2C1 N12CCC(F)(C1)C2C(=O)NCCC.c1(CCCNC(=O)OC(C)(C)C)ccccc1 C(=O)(CCC(=O)NN(C)C)NC1CN(C(C(C)(C)OCC)=O)CC1n1ccnn1 c1(C(=O)NC(C2(CNC(C3(C)CC3Br)=O)CC2)C)cccc([N+](=O)[O-])c1O N1(C(CSC(C)C)=O)CC(N(C(=O)CCc2cn(C)nn2)C)C(O)C1 C1(C(=O)NC(C2(O)CN(C(c3ccc(C)nc3O)=O)C2)C)CCn2nnnc2C1 c1(N(CCCN(C)C)C)nc2c(F)cccc2c(=NC=C2CCN(C)C2)[nH]1 N1(Cc2c(C)ccs2)CCC(CNC(=O)COC(F)(F)F)C(C)C1 c1(OC)cnnc(C(N2CCC(=CNC(C3CCC(C)CC3)=O)CC2)=O)c1 N1(C(C(CC)Br)=O)C2CCC1CN(C(c1cc(C)[nH]n1)=O)CC2 CC1(C#N)CCN(C(C2(NC(=O)CCOCCN3CCC3)CC2)=O)CC1 N1(C(CCCC#C)=O)CCN(C(c2ccc(F)c(OC)c2)=O)CC1C1CCC1 N1(C(c2cc(CC)oc2C)=O)CCCC(C)(C(=O)NC(C2CC3(CCC3)C2)C)C1 c1(CCC(=O)NCCCN(C(=O)CC2(O)CCOC2)C2CC2)cccc(F)c1Cl Cc1nn(C)c(=O)c(C(N2CCC(C(C)NC(=O)C(C)C3CCC3)CC2)=O)c1C CC(=O)C(C)CC(C)C(=O)NC1CC=C(C(=O)N2CCS(=O)(=O)CC2)C1 c1(CCC)ccc(C(=O)NC(C)(C)C(=O)OC(CC2CC2)C(=O)OC)cc1 CCCC(C)(CC)C(=O)N1CC(NC(C23CC(C2)N(C(C)=O)C3)=O)C(SC)C1 C1(C(=O)NCC(C)NC(c2c(F)ccnc2Cl)=O)CC2CCCCN2C1 N1(C(CC(C)C2CC2)=O)CCOC2(CCC(Nc3cnc(O)o3)CC2)C1.S(C)(=O)(=O)N C=CC1(CC(N2CC3C(C(=O)OC)C3C2)=O)CN(C(C23CC(CO)(C2)C3)=O)C1 Cn1cc(S(N)(=O)=O)cc1C(=O)NC1CCSC12CN(C(=O)C(F)CC1CC1)C2 CC1CN(C(=O)C(=O)NC2CC2)CC1CNC(c1cnc(C2CC2)nc1)=O O=C(CCc1cccc(C2CC2(F)F)c1)N=c1ccn(C2CC2(F)F)[nH]1 C(=O)(CC1=NN(C)C(=O)C1)NC1CCC(CC(N2CC(C)N(C)CC2C)=O)C1 C1(CC)CCN(C(=O)CCCC2CCC2)C1C(=O)N(C1CCC(C)(C)C1)C c1(C(N2CC(NC(C3(C)CSC3)=O)CC23CCC3)=O)cccc2[nH]nc(O)c12 C12(NC(C(=O)NCCOC3CC3)=O)CCCCC1N(CCC1(OC)CCC1)CC2 c1(CC(N2C(C(=O)NCc3ccon3)C=CC2)=O)ncccc1F c1(C(N(CCCCNC(C2(F)C(C)OCC2)=O)C)=O)c(Cl)ccc(F)c1F C12(CNC(=O)Cc3csc(Cl)c3)CCC(CN(C(C3CC4(C3)CC4(F)F)=O)C1)C2 N1(C(C2C(C=C)CC2)=O)CCC(C)N(C(c2ccsn2)=O)CC1 N1(CC)N=C(C(=O)N2CCC(NC(c3cnn(C)c3Br)=O)C2C)CCC1=O c1(N(C(CC)C(=O)N2CCC2(CO)CO)C)ccc(C(=O)NCC(N)=O)cc1 c1(OC)cc(O)ncc1C(=O)NCC1(CO)CN(C(C2CCC(=O)C(C)C2)=O)C1 Cc1ccc(C(=O)NCCN(C(=O)CCn2cc(Cl)cn2)CC(C)O)s1 C1(CC(=O)N(C)Cc2cncn2C)COCCN1C(C1CC1C(C)(F)F)=O C1(CNC(C)C(C)(C)CO)C2CC(F)C1N(C(=O)OC(C)(C)C)C2 C#CCC(CC#C)C(=O)N1CCN(CCNC(C2(C3CCCO3)CCC2)=O)CC1 CC1=NS(=O)(=O)N(C)C=C1C(=O)NC1CN(C(=O)C(F)=C2CCCC2)C2CC12 C1(C(N2CCCC(NC(C34C(C(N)=O)(CCC3)C4)=O)C2)=O)C2CC3C(C2=O)C13 Cc1cccc([N+](=O)[O-])c1C(N1CCC(C2CCCN2C(=O)C(=O)C2CC2)C1)=O c1(C(N2CC(C(N(CC#C)C(C)C)=O)C(O)CC2)=O)ccc2sccc2c1 Cc1[nH]c2ccccc2c1C(CC(C)C)S(=O)(=O)CC1CS(=O)(=O)C1 c1(CC)nn(C)cc1C(N1CC(OC)C(NC(c2ccccc2NC)=O)C1)=O c1(CCNC(c2c(CNC(C(COC)N(C)C)=O)cco2)=O)cnccc1C C1(C(=O)NCC(C(C)C)NC(C2(C(=O)N(C)C)CC2)=O)CCC(C)(F)CC1 Cc1cc2c(Br)ccc(C(=O)N(CCCNC(=O)CC(C)(C)C)C)c2o1 CC1CCC(C)(C(=O)NCCN(C(=O)C(C)(C)c2cc[nH]n2)C)C1 C1(NC(C2C(NC(=O)C(F)CC3CC3)CC2)=O)CC2CCCCCC12 C12(CNC(=O)C3=CCCSC3)CCC(CN(C(c3ccc(Cl)s3)=O)C1)C2 N1(C(c2cc(OC)c(C)nc2)=O)CC2CC(C)N(C(=O)CC3CCCCO3)C2C1 N1(C(C2C(C)C2)=O)CCC2(CC1)CC(C)N(C(c1cc3ccnc(Cl)c3[nH]1)=O)C2 c1(C(=O)NC2CCCN(C(C3NC(=O)OCC3)=O)CC2)cc2cc(Cl)ccn2n1 N1(C(c2cc(C)[nH]n2)=O)CCOCC(C(=O)N2CC=CCO2)C1 c1(CNC(c2ccc(CNC(CC3N(C)CCC3)=O)o2)=O)[nH]ccc(=O)c1O c1(C(=O)NCCC2CCN(C(c3c(OC)scc3)=O)CC2)c(C)cc(=O)oc1C C(C(COC)CC(=O)NCC(C)(O)CNC(=O)C(c1cc(C)cc(C)c1)C)OC C1(NC(=O)CCc2cn(Cc3ccccc3)nn2)CCn2c(O)nnc2C1 c1(C(=O)NCCN(C(=O)CCC2CCC2)CC)ccc(C(N)=O)nc1 C1(C(=O)NCC(C)(CO)NC(c2cc(Cl)ccc2F)=O)CCCCC12CCC2 N1(C(c2n(C)nc(CNC(C3CC=CCC3)=O)c2)=O)CC(C2CCCCC2)C1 CON=CC(=O)NC1CC1CNC(=O)C=Cc1cocn1 c1(CNC(C(C)C2CCCO2)=O)c[nH]nc1C(=O)N(C)Cc1nncn1C C1(NC(CCCC#C)=O)CN(C(c2ccc(C(=O)CC)cc2)=O)CCC12CCC2 C1(O)(CN(C(=O)CCC2CCC2)C)CCCN(C(C2CC2(Cl)Cl)=O)C1 C12(CNC(C(CCC)O)=O)CN(C(C3(CO)CCCO3)=O)CC(F)(C1)C2 C1(C)(NC(CCC2(C)CC2)=O)CCCN(C(c2cccc(-n3cccc3)c2)=O)C1 c1(CC(N2CCCC(N(C(=O)C3=CSCS3)CCF)C2)=O)ccnc(O)c1 N1(C(C2(c3ccc(Cl)cc3)CC2)=O)CC2CN(Cc3ncc(Cl)cc3F)C2C1 c1(CC)cc(NC(C2CCCCN2C(=O)C(C2CC2)SC)=O)cc(O)c1 CC1CCCC(C(N)CN2CCN(C3CCN(c4ccc(CO)cn4)C3)CC2)C1 C(=O)(CCC(=O)N(C)C(c1n[nH]cc1Cl)=O)NC.C1C(C)(C)CN1C N1(C(CCCC#C)=O)CCCOC(CCNC(c2cn(C(C)C)cn2)=O)C1 C(=O)(C(C)(C)CCSC)N(C)CC1CCCN(C(C2(C(F)F)CC(=C)C2)=O)C1 Cc1nc(CC(N2CC3C(NC(=O)Cc4cc[nH]n4)C3C2)=O)c(Cl)s1 C1(NC(CCCCCCC)=O)CCC12CCN(C(C1(C)CC(=O)N(C)C1)=O)CC2 C(=O)(CCC[N+](=O)[O-])N1CC(O)(C(C)NC(CCC=CC(C)C)=O)C1 N1(C(CC(C)(C)SC)=O)CCc2ccccc2C1CNC(c1cncc(F)n1)=O C1(CNC(=O)CSc2cn(-c3ccccc3O)nn2)CC2OCCCC12 CC1(C)CCC=C1C(=O)NC12CC1CN(C(C1(C3CC3)CC1)=O)C2 c1(CCC(N2CC=CC(NC(C3CC(N(C)C)C3)=O)C2)=O)ccc([N+](=O)[O-])cc1 Cc1ncsc1CC(=O)NC(C)(C)CCNC(c1nc(C(F)(F)F)cs1)=O c1(C(=O)NCC2N(C(CCCCC=C)=O)CC=C2)ccc2nc(N(C)C)sc2c1 C1(OC)CN(C(C2(F)CN(C(=O)CCc3cncnc3)C2)=O)C2(CCC2)C1 C1(CC(=O)NCC2N(C)CCC2)CN(C(=O)CCc2cccnc2)CCO1 N1(C(CN2CC(C)(OC)C2)=O)CCOCC(C(=O)NCC23CC(CCO2)C3)C1 N1(C(CCn2c(C)cc(=N)[nH]2)=O)CCC2CN(C(c3ccc(Cl)cc3)=O)CC2C1 C(=O)(C1CCC(=O)c2ccccc21)NC(C)CCNC(c1cc(C(N)=O)no1)=O c1(C2(C)CCO2)cccc(NC(=O)NC2(c3cccs3)CCOCC2)c1 N1(C(C(CCC)OC)=O)CC2CCN(C(=O)C(C)(C)CC(C)C)CC2C1 N1(C(C(CC)C2CCCCC2)=O)CC2CC(O)C1C2COC CC1COCCCN1C(C1(NC(C2CCCCC2O)=O)CCN(C)C1)=O N1(C(C2CC(SC)C2)=O)CC2(CCC(CNC(C3CC3C3CC3C)=O)O2)C1 c1(C(C)C)cncc(C(=O)NCCC2(CNC(c3cncc(N)n3)=O)CC2)c1 c1(C(=O)NC(CNC(=O)C=C2CCCC2)CO)c(Cl)oc2ccccc12 CC(C)(C(=O)N1CC(CCNC(c2ccc(-n3cnnn3)cn2)=O)C1)C(N)=O c1(NC(C2CC2C(F)F)=O)cccc(CN(C)C(C2CCC(C(N)=O)C2)=O)c1 N1(C(CNC(=O)NC)=O)CCC(C(=O)OC)CC1.c1(C(=O)N)cc(C)ns1 C1(C(N2C(CNC(CCCc3n(C)ncn3)=O)CC2)=O)C2CCC(=O)C12 C12(C(N(C)CC3CCCC(C)C3)=O)CC(CO)(CN1C(=O)Cc1cnsc1)C2 Cc1c(C(N2CC(CCCCNC(=O)C(C)S(C)(=O)=O)C2)=O)nn2ccccc12 c1(C(=O)NC2CC3(C(NC(C(C)SCCCC)=O)C3)C2)cc2c(s1)CCOC2 c1(C(=O)NCCN(C(C)C)C(c2cncn2-c2ccccc2)=O)cc(Cl)c[nH]1 C(C(C)C(C)C(=O)NCC1CN(C(=O)C(C)(C)C(C)C)C1)OC Cc1ccc(-c2ccc(-c3nccn3C(C)C(=O)Nc3cn(C)cn3)nn2)cc1 C=CCC(F)(F)C(=O)N1CCN(C(C2(c3ccncc3)CC2)=O)C(COC)C1 Cc1ccc(CCNC(=O)C(N2CCCC2C(C)(C)C(=O)OC(C)(C)C)=O)s1 C1(NC(N(C)Cc2cc3cnccc3[nH]2)=O)CCCCC12OCCO2 N1(C(C)C)N=C(C(=O)N2CC(NC(=O)Cc3ccco3)CCC(O)C2)CCC1=O C(C(=O)N1CC=CC(NC(c2scc(C)c2Cl)=O)C1)(C(C)O)NC(=O)OC c1(C(=O)OC)ccc2sc(=NC3CCN(c4cc(C)ncn4)CC3)[nH]c2c1 c1(C(N(CCCCNC(=O)Cn2nccn2)C)=O)cn(CC2CC=CCC2)nn1 C(=O)(C(C)(O)CC(C)C)NCC1CC(NC(COc2cc(C)c(F)cc2)=O)C12CCC2 C#Cc1c[nH]nc1C(=O)NCC(C1CC1)NC(=O)COc1cccnc1C(Cl)(Cl)Cl C1(F)(C(N(C)CC2CCN(C(c3cn(CC)nn3)=O)CC2)=O)C2CCCCC12 C1(NC(c2c(C)ccs2)=O)CCCN(C(=O)C(C)c2ccco2)CC1 CCC(C)(CNC(c1cc(C)nn1C)=O)C(=O)N(C1CCOC(C)(C)C1)C N1(C(CC(C)NC(N)=O)=O)CCC(C)(CCNC(=O)CC2(CO)CC2)C1 c1(CCC(N2C(CNC(=O)CCOC3COC3)CC(F)C2)=O)cc(F)cc(F)c1 Cc1cc(C)c([N+](=O)[O-])c(C)c1C(N1CCCC(CNC(=O)C2CC2)C1)=O Cc1cccn2cc(CC(=O)NCCN(C(=O)C(F)C3CCOC3)C(C)C)nc12 c1(C(=O)NC2CCN(C(C(C)c3cc[nH]n3)=O)C2C)ccc2occc2n1 c1(CNC(c2nc(CNC(c3cc(CCC)[nH]n3)=O)oc2)=O)ccc(C)c(F)c1 C1(NC(=O)CC2CSCCS2)CCS(=O)(=O)C12CN(C(c1c[nH]nc1C(F)F)=O)C2 N1(C(c2cn(CCOC)nc2)=O)CCC2(CC1)OCC(C)(C)CO2 CC(N=c1nc2scnc2c(C(F)F)[nH]1)c1ccc(S(C)(=O)=O)cc1.C12(CC1)NC2 c1(OCCC(=O)NCCC(C(C)C)NC(C(C)SCC)=O)cccc(CC)c1 c1(C(=O)NC(C)CN(C)C(C2(C)CC2(Cl)Cl)=O)ccc(-c2cccc(C)c2)n1C C12(NC(c3c(C)c(Cl)ccc3)=O)CCCC1CN(C(=O)C=Cc1ccncn1)C2 Cc1cc(CNC(=O)CC2CN(C(c3cc(C#N)c[nH]3)=O)CCO2)c(C)s1 CC(=O)C(C)(C)CC(=O)NC1C(C(=O)NCC2CCCC2)C1(C)C c1(C(=O)NC(CC)CNC(=O)CCc2ncco2)ccc(Br)c(Cl)c1F C1(NCC(=O)NCC(Cn2cc(CCOC)nn2)(F)F)CC(C(=O)O)C12CCC2 C(=O)(CCN(C(=O)CN(CC)CC)C)NCCOCCC#C CC1(C)CN(C(=O)C(O)NC(=O)Cc2cc(-c3ccco3)[nH]n2)CCC1C1CC1 CC1CN(C(=O)CCCOCC(C)(C)C)CC1(C)CNC(C1CC1F)=O C=C(C)CCCC(=O)N1CC(CCNC(=O)C=CC2CCOC2)(OC)C1 C1(C(N(CCCC)Cc2cccc(F)c2)=O)CC2(CCC(F)(F)CC2)C1 N1(C(c2nc(C(C)OC)oc2)=O)CC2COCC(C1)C2NC(=O)C=CCl C=CCC(CC(C)C)C(=O)N1CCN(C(c2ccn(CC)c2C)=O)C(CO)C1 C1(NC(C(C)c2ccco2)=O)CN(C(C2CC3(CSC3)C2)=O)CCC1(C)C c1(C(=O)NCc2coc3c(Cl)cccc23)ccc2c(c1)CCCO2 N1(C(C2CCC(SCC)CC2)=O)CC(C(N2CC(=O)NCC2C)=O)CC(F)(F)C1 N1(C(C(CCCC)O)=O)CCC2(CC1)CC2C(=O)NC(C)(C)C(C)(C)O C(=O)(C#CC1CCC1)N(CCC(=O)N(C)CCn1cncn1)C.C12CC(C1)N2 c1(C(=O)Nc2c(C(N3CC(F)CC(C(=O)OC)C3)=O)scc2)cc(Br)c(C)c(Br)c1 c1(CC)ccc(C(=O)NC(CNC(=O)Cn2nc(C)oc2=O)CCOC)nc1 C1(=CC(N2CC(C(C)NC(=O)C3=NNC(=O)C3)OCC2)=O)CCCCC1(C)C C1(C)(CNC(c2c(C)onc2CO)=O)CN(C(=O)C(C)(C)n2ccnn2)CC1C Cn1c(I)cc2c(N3CCCC(C4CCCC4)C3)ncnc12 C1(C2CCN(C(=O)C(C)CCO)C2)(NC(C2CCN(C(C)C)CC2)=O)CC1 CC1CN(C(C2(Cl)CC2)=O)CCC1CNC(=O)COc1ccc(F)cc1O c1(C2C(C(c3cccc(-n4cnnc4CO)c3)=O)C2)ccc(F)cc1Cl C1(NC(C2CC(O)(CC#C)C2)=O)CC=C(C(=O)N(C)Cc2cccc(C)n2)C1 N1(Cc2c(N(C)C)cccc2)CC2(CCN2C(c2cc(C(F)(F)F)cc(Cl)c2)=O)C1 C(=O)(C1CCCc2oc(C)nc21)N(CCC(C)NC(c1cc(SC)c(C)o1)=O)C CCCC(C(O)C(=O)NC(C)C(N)=O)NC(=O)CCC(C)N(C)C c1(C(N2CC(C(C)NC(C(C)(C)OC)=O)OCC2)=O)cnc2c(C)cccc2c1 c1(OC)ccc(C(=O)NC(CNC(=O)C(=O)N(C)C)CO)cc1OC(F)F CC#CCCCC(C(=O)NCC(C)C)N1C(C)COCC1C C=CCC(C(=O)N(C)CC1(O)CCN(C(=O)Cn2c(C)csc2=O)C1)C(C)C C1(NC(COCc2onc(CC)n2)=O)CCN(C(C2CCC3CC3C2)=O)C(C)C1 c1(C(N2CC(F)CC(NC(CCCCC)=O)C2)=O)cc2sccc2n1C CCC1=C(C(=O)N2CCCC2(C)CNC(C2CCC([N+](=O)[O-])CC2)=O)CCCO1 c1(C(=O)NC(CNC(CCCOCC)=O)C2CC2)cc2n(n1)CCN(C)C2 c1(C(N2CC3C(CNC(=O)Cc4cncc(F)c4)C3C2)=O)cc(Cl)cc(Cl)c1O C(N=c1[nH]c(N2CCN(C)C(=O)C2)nc(=N)[nH]1)c1n(CC)nnn1 C(=O)(Nn1nnc(C)c1C)c1c(CNC(c2cnc(CC)s2)=O)n[nH]c1 C1(NC(=O)C=CC2CC2)CCC2(CC1)CC2NC(=O)Cn1ncc(O)nc1=O c1(OC)ccc(N2CCN(C(C3COC(C)C3)C(=O)N(C)C)CC2)cc1F Cc1c(C(=O)N(C2CCC2O)C)nnn1-c1ccc(N(C)C)cc1 N1(C(c2ccc(CO)s2)=O)CCCC2(C1)CN(c1nnco1)CCO2 c1(C(=O)N(C2CCCC2)Cc2ccc(F)cc2Br)ccc2c(n1)CCO2 c1(C(=O)NCC2CCN(CC(=O)N(C)C)CC2)ccc2c(n1)C(O)CC2 c1(OC)cnc(C(N2CC3(CNC(=O)CC(C)C4CCCO4)CC2CO3)=O)c(F)c1 C(C(=O)N1CCCC(N(C)C)CC1)(C(C)(C)C)NC(C(CC)NC(C)=O)=O N1(C(C=C(C)C)=O)CC2(C1)C(NC(=O)C(C1CCCCCC1)O)CCS2(=O)=O c1(CC)cccc(C(=O)N(CC(C)CNC(=O)CCF)C)c1O C1(C(N2CCOCC(NC(C3OCC(=O)C3)=O)C2)=O)CNc2ccnn2C1 CC(C)(C)C(C)(C)C(=O)NCCC1CN(C(=O)C#CC2CCCO2)CCCO1 c1(C(=O)NCC(CCCC)NC(c2cc3ccsc3s2)=O)cc(C)c(N)cn1 O=C1CC(CC(=O)NCC2CCN(C3CCCCC3)C2)CCCN1 Cc1cc[nH]c(=N)c1C(=O)NCC1CC2CCC1N2C(C1CC2(CC(=O)C2)C1)=O Cc1cc(CNC(=O)CCC(C)CNC(C2CC(O)C(F)C2)=O)nc(C)c1 C(=O)(CC(CC#N)c1ccccc1)NCCCNC(C(COC)C)=O N1(Cc2c(C#N)cccc2)CC2NC(NC(=O)C3=NNC(=O)CC3)=NC2C1 C1(C(=O)NCCC2CN(C(=O)COC(C)C)C2)(CC)CCC1 c1(C(N2CC(CCNC(=O)CN3CCNC3=O)(OC)C2)=O)cccc2c1COC2 C1(C(N2CCC(OCCNC(C3=CCCC3C)=O)C2)=O)COC2(CCC2)CO1 C1(C(N2CCOC(C3CC3)C2)=O)(CC)CCCN1C(C12CCC(C1)C2)=O N1(C(c2cc(C)c(Br)cc2)=O)CCC2CCN(C(c3nc[nH]n3)=O)C2C1 C1(NC(C=C(C)Cl)=O)CC2CC(NC(=O)Cc3cccnc3Br)CC2C1 C(=O)(C(CC)C(F)(F)F)NC(CC=C)CC(=O)NC(CCO)C(C)(C)O CC#CCCCC(=O)OCc1ccc(-n2cncn2)cc1 N1(C(C(C)OC)=O)CCCC(N(C)C(c2csc(Cl)c2)=O)CC1 N1(C(C(C)(C)C2CCOC2)=O)CCC(N=[N+]=[N-])(C(=O)NCc2cncc(F)c2)C1 c1(C(N(CCOC)CCNC(=O)CC2(C(F)(F)F)CC2)=O)ccc2n[nH]cc2c1C C1(C(=O)NC(C(C)C)C(C)NC(=O)C(C)(C)C(=O)N(C)C)CC2(C1)CC(O)C2 C(c1cc(Cl)c2c(c1)OCO2)=CC(=O)CSC(F)(F)F.c1nccc2occc12 c1(CNC(C(C)C)C(F)F)cc(Br)ccc1Cl c1(C(N(c2cccc(C#N)n2)C2CCC(N)C2)=O)ccc2c(c1)OCO2 c1(CN2CCN(c3ncc(CCC)cn3)CC23CC3)ccc2ccn(C)c2c1 N1(C(c2c(C)snc2)=O)CC(NC(=O)C2=CCCOC2)CC(C)C1 c1(C(=O)NC(c2ccccn2)C)nc2ccc(-c3ccc(F)c(F)c3)cc2o1 C1(n2cccn2)(C(=O)NCC(CC)(CC)OC)CCN(C(c2occc2C)=O)CC1 C1(CNC(C(CCSC)O)=O)CCCCCN1C(=O)Cn1ncn(C)c1=O C(C)(C)(CCC(=O)NCCC(O)CNC(=O)CSc1ccccc1Cl)N(C)C C1(C(=O)NCCCCCO)CC12CN(C(c1cccc(-n3cncn3)c1)=O)C2 Cc1ccc(F)c(C(N2CCC(CCNC(=O)Cc3csc(C)n3)(N(C)C)C2)=O)n1 c1(C(N2C(c3cn(CC(=O)N(CC)CC)nn3)CCC2)=O)ccsc1OC c1(C(=O)NCC(CC(C)C)NC(C=C(C)C(C)(C)C)=O)cc(N)ccc1F C1(CNC(CCC2CN(C)C(=O)C2)=O)Cc2cc(O)ccc2CN1C(=O)CC#N c1(C(N(C(C(=O)N2CC(c3ccccc3O)C2)C2CC2)C)=O)ccc(O)nc1 CC(CNC(c1cc(=O)cc[nH]1)=O)C(F)C(=O)NCCOc1cccnc1 c1(C(=O)NCC2(F)CC(CNC(C3C(C(C)C)C3)=O)C2)ccc(F)c(O)c1 c1(C(=O)NCC2(C)C(C)CN(C(CSCC=C)=O)C2)cc2cccn2cn1 C1(C)(CNC(c2c(NC)scn2)=O)CC2CC2C1.C12(OC)CC(C1)C(=O)N2 CC1(NC(=O)COC2(C)CCOCC2)CCC(NC(C2CC3CCC2C3)=O)CC1 c1(OC)ccc(C(C)C)c(C(N2CCC(NC(=O)CCc3cccs3)C2)=O)c1 CCC(CC)C(C)C(=O)Nc1cccc(Nc2ncccn2)c1 C12(C(N)=O)CCC(NCc3ccc(I)o3)(CC1)CC2.c12cncc(c1)NC2=O C(=O)(CC(O)CC(C)C)NC(C(=O)NC(CCCCC)C)C(C)(C)C C1(CC)(CC)CC(NC(C2CCCC(=O)N2)=O)CN1C(=O)C(=O)NC1CC1 c1(N(C(C2CCCC2)CNC(CNC(CN(CCC)C)=O)=O)C)cc(C)n(C)c1 c1(NC(C2(O)CCN(Cc3n(C)ccn3)CC2)=O)cccc(Cl)c1C#N C1(CCC)CCCCN1C(C1CNCC(C(=O)O)O1)=O c1(C(C(=O)NCC=C)N(C)CC2CCCN2C)cc(Cl)cc(Br)c1OC c1(N2CCCC(C)(C(=O)NC(C(=O)OCC)C(C)O)C2)ccc(C#N)nc1O c1(COC)cc(N2CC(O)(C(C)NC(C3(c4ccccc4)CC3)=O)C2)ncn1 c1(C(c2nnc(N(CCOC)C)n2CCC#N)O)cccc2[nH]ncc12 N1(C(c2cncc(CC)c2)=O)CC(CNC(c2ccc(F)cc2)=O)N2CCC1C2 c1(C(=O)NC(C2N(C(c3c(C)c[nH]c3)=O)CCCC2)C)nnc2ccccn12 C1(NC(CCCOC)=O)C2CN(C(c3ccc(CF)cc3)=O)CC12 CCCS(=O)(=O)CC(=O)NC1CCN(C(C2CC2Cl)=O)CC1 CCCC(CCc1ccc(Cl)cc1)n1nnc(-c2cccc(OC(F)F)n2)n1 CC1CN(C)CC(C(N2CC(O)(C(C)NC(c3nccs3)=O)C2)=O)O1 C1(OC)CC(N(C(c2ccc(CF)cc2)C(=O)NCC2CCCO2)C)C1(C)C N1(C(C(C(=C)C)(C)C)=O)CC(C)C(N=c2[nH]c3ccc(OC)cc3s2)C1 c1(CC(=O)NC2(CNC(CC3ON=C(CC)C3)=O)CC2)cc(C)ccc1Br C(=O)(CCCCCN(C)C)NCC1N(C(C2(C)CCC(C)C2)=O)CCC1 C(=O)(C1=C(C)Oc2ccccc2C1)N1C2C(NC(C(C=C=C)C)=O)CC(C2)C1 c1(C(=O)NCC2CCN(C(c3n(C)ccc3)=O)C2)cc(C(F)(F)F)ccc1F C=CCC(C)(CC=C)NC(=O)C(C)N(C(C1CC(O)C(F)C1)=O)CC c1(CC)cc(CC(N2CCC(O)(CNC(c3cccc(Cl)c3)=O)C2)=O)n(C)n1 C(=O)(C(=O)CCC(C)(C)C)NC(C(C(C)C)C)CNC(=O)CN1CCCNC1=O c1(C(N2CC(N(C(C3N(S(C)(=O)=O)CCC3)=O)CCO)C2)=O)cccc2ccnn12 C(C(C)(C)C(=O)NCCC1CCN(C(=O)Cc2nc(C)sc2Cl)C1)OCC c1(C(=O)NCCC2N(C(c3nc(C)oc3)=O)CCSC2)n[nH]c2c1COCC2 CC1c2c[nH]nc2CCC1C(N1CCCC(CNC(=O)C(C)n2ccnc2)C1)=O O(N1CCC(NC(C23CCC(CC2NC(c2ccnnc2)=O)C3)=O)CC1)CC C1(NC(Cc2nc(C)[nH]n2)=O)CCC2(CC1)CN(C(c1ccc(C)c(O)n1)=O)C2 C(CN=c1cc(C(C2CC2)C2CC2)nc[nH]1)N(C(c1cc(OC)n[nH]1)=O)C N1(C(CC(=C=C)C)=O)CCCCCC(NC(=O)CC2SC3=NCCN3C2=O)C1 CCCCCOCC(=O)NC1CCC1NC(=O)CSCCC c1(NC(C2(C)N(C(C(C(C)C)SCC)=O)CCC2)=O)cnc2ccnn2c1 C=CC(C)CC(=O)N1CCCC1C(=O)N(CC)Cc1nnc(O)n1CC C1(C(N(C)CC2CCCN2C(=O)Cc2nnc(O)s2)=O)CCC2(CC1)CC2(F)F c1(OC)ccc(C(=O)N(C(CNC(=O)Cc2cc(C(N)=O)no2)C2CC2)C)c(C)n1 C(CC(C)CCNC(c1ccc(-c2ccco2)[nH]1)=O)NC(C(C)N1CCC1)=O N#Cc1cnn(CC(=O)NC2CCCCC2NC(c2ccn(C3CC3)n2)=O)c1N c1(N2CC3CC(NC(c4ncc(OC)cn4)=O)C3C2)c(Cl)cccc1[N+](=O)[O-] N1(C(CC2CC(OCCOC)C2)=O)CCC(C)C(NC(=O)CC(O)CN(C)C)C1C Cn1cc(C(O)C(=O)NCC2CC2CNC(c2cc(C(N)=O)c[nH]2)=O)cn1 N1(C(c2nccc(N)c2)=O)CC2CC1CCN2C(C1C2CCCCCC12)=O CC(CCC(C)(C)C)C(=O)NC(C1CCCCC1)CNC(=O)C(O)C1CCC1 N1(C(c2cnn(C)c2N)=O)CCCC2(C1)CN(C(C1CC(O)C(F)C1)=O)C2 c1(C(N(CCC(=O)NCC(CCC)(C)C)C2CC2)=O)c(C#N)cnn1C c1(C(N2CC(CCNC(C(C)OCOC)=O)C(C)C2)=O)cnc2scnc2c1 N1(CCC)CCCC(C(=O)NCCC2(NC(=O)CC3CC3C)CC2)C1 N1(c2nnc(CC)c(CC)n2)CCC(NC(=O)Cc2cccc(C)c2)C(C)(C)C1 CCC(C)(C)CC(=O)NC(CC(C)C)C(=O)N(C12CC(C1)C2)CC c1(C(=O)NCC2(CN(C)C(C3CC3(C(C)C)CF)=O)CC2)noc2ccccc12 C(CC(=O)NCC1CCCOC1)(C(C)OC)NC(c1c(OC)n(C)nc1)=O N1(C(=O)CC2CCCCC(=O)N2)CC2(CCN(C(C3N(CC)CC3)=O)C2)C1 CCC(CC)C(F)C(=O)NC(C1CCN(C(C2CC3(CCC3)C2)=O)C1)(C)C C(=O)(CC(O)CNC(=O)CC1CCC(=O)N1)NC1CCN(CCOC)C1 C1(C(=O)NC2CCS(=O)(=O)C2)CC12CCN(C(C1CC3CC1CC3=O)=O)C2 c1(-c2cc(C)cc(OC)c2F)ccc2[nH]c(C(=O)Nc3ccno3)nc2c1 c1(CC)cc(N)ccc1C(N1CC(O)(C(C)NC(=O)CC(C)(C)O)C1)=O C1(C(=O)NC(COCC)C(=O)NCc2cnn(C)c2O)CCCC12CCC2 Cn1cc(N(C(C2(C)CC(=O)C2)=O)C(c2cccc(F)c2)=O)c(OCC(F)F)n1 CN1CCC(NC(c2sccc2CNC(C2(C)CCC2)=O)=O)C(C#N)C1 N1(C(CNC(=O)NC2CC2)=O)CCN(C(c2ccoc2)=O)C(CC(F)F)C1 c1(CC(=O)NC2CC3(CCN(C(CCSC)=O)C3)C2)ccc(S(C)=O)cc1 C1(C(N2C3CC(NC(CSCC(N)=O)=O)C(C3)C2)=O)CC2COCC(C1)C2=O C1(NC(=O)CC2(C(=O)N)CC2)CC2(CCN(C(=O)COc3cccs3)C2)C1.CCO CC1(C)CCN(C(C2C3CCC(F)(F)C23)=O)C(C(N2CCC(O)(C(N)=O)C2)=O)C1 c1(OC)ccc(C(N2CCCC(NC(C3(N(C)C)CCCC3)=O)C2)=O)c(I)c1 C1(C#N)(CC(=O)NCC(CC(C)C)NC(C2(F)CCCN(C)C2)=O)CCCCC1 c1(C(=O)NC(CC)CC(=O)NCCC2CCSC2)cc(C)nnc1C C(=O)(CCCC(F)(F)Br)N.N1(C(c2c(C)coc2)=O)CCCCCC1C N1(C(C(CO)NC(C)=O)=O)CCC(CCN(C(C2(Cl)CC2(C)C)=O)C(C)C)CC1 N1(C(c2cc(C(N)=O)[nH]c2)=O)CC(NC(=O)CC2CNC(=O)C2)CCC(O)C1 Cc1cc(CN2CCOCC2C(=O)Nc2cccc(C#N)c2)cc(O)c1 n1(CC(N2C(CNC(CN3CC=C(C)C3)=O)CC(O)C2)=O)cnc([N+](=O)[O-])c1 c1(CC)cc(F)ccc1C(=O)NC1CCCC1NC(C1CCCCC1C(=O)OC)=O C(CCC(=O)N(C)C(C)C1CC1)NC(C=C(C)C(C)C)=O C1(C(=O)NC(c2c(C(=O)NCc3onc(CC)n3)con2)C)COCCC1C C1(N(C(c2ccc(C(=O)NC)nc2)=O)C)CN(C(=O)CC(C)(C)OC)CCC1C c12nnc(N3CCCC3c3cn(-c4ccc(Cl)cc4)nn3)n1C2.CC(C)(C)C1CC1 N1(C(C(c2c(C)cccc2Br)NC(c2nc(C)sc2C)=O)=O)CCS(=O)C(C)C1 C1(CNC(C2C(C)C2C)=O)CC2CCC(C1)N2C(=O)CCc1nc(=N)[nH][nH]1 c1(C(=O)NCC2(NC(=O)CCC(=O)c3cccs3)CC2)ccc(OC)c(F)c1F N1(C(CSC)=O)CC(N(C)C(c2c[nH]c(C(N)=O)c2)=O)C(C)(C)C1 c1(C(=O)NC(CNC(C2(CCC=C)CC2)=O)CC(C)C)cccn2nccc12 CN1C(=O)C(=O)N(CC(=O)NCCOCCNC(C2COC3(CCC3)C2)=O)C1=O Fc1cc(-c2nn[nH]n2)ccc1CN1CCC(C2CCCCO2)CC1 C12CCCCN1C2=O.c1(C(=O)NC)nnn(C2CN(C(C3(F)CCC3)=O)C2)n1 c1(CCC(=O)NC2(CCNC(CN3C(C)CCC3)=O)CCC2)ccc(C(F)F)cc1 c1(CC)cccc(OCC(C)NC(=O)Nc2ccnn2C)c1.C(CN(C)C)O C(=O)(C1=C(Cl)CCCC1)N1C(COC)CN(C(c2cc(=O)n(C)cn2)=O)CC1 Cc1noc(C(F)F)c1C(=O)NC1COCCC1NC(=O)C(C1CCOCC1)C Cc1ccc(SCC(=O)NCC2CCC2NC(=O)CCC(C)C)cc1C C1(N(C)C(C2CC3CCC2O3)=O)CCCN(Cc2ncc(C(C)(C)C)o2)CC1 c1(CC(=O)NCCC(C)(C)NC(C(n2cc(Cl)cn2)C)=O)ccccc1OC(F)F CC(CC(=O)NCC(O)CN(C)C(C1CCN1C)=O)C1CC1 C1(CC(N2CCCC2CCO)=O)CCCCN1C(C1C2COCC12)=O C1(CNC(C(CCC)C)=O)CCC2CN(C(c3cscc3C(N)=O)=O)CC12 N1(C(CCSCC)=O)CCC(C(=O)NCCC(C)(C)C)C(C)(C)C1 C1(CCC(=O)OC)(CNC(C2CCC(C)(C)C2)c2nnnn2C(C)C)CCOCC1 c1(CC(=O)N(C2CCCN(C(=O)CC3CCC3)C2)CC)ccc(F)c(Cl)c1 C1(C(N2CCC(CNC(c3cncc(CO)c3)=O)C2)=O)Cc2ccc(F)cc2C1 N1(CC(=O)NCCCCCCNC(C2(C)CC3CC3C2)=O)CCn2ccnc2C1 c1(C(N(CCNC(C(CC)C(C)C)=O)CC)=O)coc2c1C(=O)NCC2 c1(CC(=O)OC)cc(SC2CCN(C)C2=O)c2c(c1)CCO2 c1(C(=O)NCC(CNC(c2cc(=O)cc[nH]2)=O)F)cncc2nc(O)[nH]c12 CS(=O)(=O)c1coc(C(N2CCC(O)(CNC(=O)C(O)CF)CC2)=O)c1 N1(C(C2ON=C(C)C2)=O)CCCC(N(C(=O)CN2CCCNC2=O)C)CC1 N1(C(c2c(CCC)nsc2N)=O)CCCC2C1CCCN2C(c1ns[nH]c1=O)=O C1(C(=O)NCC2CC(C)N(C(=O)CC3(CO)CCC3)C2)COc2ccccc2O1 N1(C(c2ccc(OC)cn2)=O)CCC(C2(NC(C3CC34CCOC4)=O)CC2)C1 C1(C(=O)NCC2=CCN(C(C(C)O)=O)CC2)CC(C)(C)OC1(C)C C1(C(N2CC(CCNC(=O)C(O)CC3CCOCC3)C2)=O)CC2CC1CC2O Cc1ccc(CNC(C2CCCC(NCC3(C#N)CC3)C2)=O)cc1Cl c1(C(N2CC(CCC)C(NC(=O)CN3CCC(C)(C)C3)C2)=O)csc2nccn12 N1(C(C(C)=CC)=O)CCN(C(=O)C(c2cccs2)SC)CC(C)(F)C1 C(=O)(C(F)C(C)CNC(C1(CCOC)CCC1)=O)N(c1ccccc1)CC#C N1(C(CCC2CCN(C(Cc3c(C)nsc3)=O)C2)=O)CCCC12CCN(C)C2 O=C(C#CC1CCCOC1)NCC1C=CCN1C(c1ccc(N2CCC2)nc1)=O C(c1cc2ccccc2n1C)=CC(=O)NC1(CNC(C2C(C)C2C)=O)CCCC1 c1(NC)nc(C)ccc1C(=O)NCCC1(C)CCN(C(c2cc(CO)[nH]n2)=O)C1 C1(CCC)(C(=O)NC(C)C(CO)NC(=O)Cc2cc(C3CC3)no2)CCNC1=O C(=O)(C1CCCc2nncn21)N1CC2N(C(C#CC(C)(C)C)=O)CC(CC2)C1 c1(C(N2CCC(N(C(=O)CP(C)(C)=O)CC#C)CC2)=O)ccc(F)cc1C#N c1(C(N2CCC(O)(CN(C(=O)CCC(=O)NC3CC3)CC)C2)=O)cc(C#N)[nH]c1C C(CCO)(C(C)(C)O)NC(CCN(CC=C)C(C1CCCN1C=O)=O)=O CN1N=C(C(=O)NCC2CCN2C(C2CC3(C2)NC(=O)NC3=O)=O)CCC1=O C(C(CC(F)(F)F)NC(c1cccnc1N)=O)NC(C(C=CC)O)=O c1(NC(N2C3CN(S(CCOC)(=O)=O)CC32)=O)ccc(F)c(F)c1[N+](=O)[O-] c1(Cc2n(CC)c(N3CC4(OC)CC3C4)nn2)cc(C(F)(F)F)cc(Cl)c1.C(=O)OC N1(C(CCN(C)C(c2cc[nH]n2)=O)=O)CCCC2(C=CCO2)C1 N1(C(CC=C=C)=O)CC(CNC(c2cc(C)nn2-c2ccccn2)=O)C2(CC2)C1 C1(NC(c2cc(C)cc(C)c2)=O)CCN(C(=O)C2=CC(O)CCC2)CCC1(F)F C1(NC(c2n(CC)ccc2)=O)CCN(C(c2cccc(=S)n2O)=O)C(C)C1 C1(C(N(C(C=C)C)C)=O)CC2CC1CC2NC(=O)C(COC)COC c1(C(N2CCOCC(NC(c3ccc(Cl)cc3)=O)C2)=O)cccc2c1OCO2 CC1C(C)N(C(c2cn(C)cn2)=O)CCN1C(=O)CCNc1ccc(F)cc1 C12(CC(=O)NCC3C(NC(C(C)NC(C)(C)C)=O)C3)CCCN1CCC2 C(=O)(C(C)(F)C(F)(F)F)N1CCC(OCCNC(C2(CCCC)CC2)=O)C1 Cc1nn(CC(N2CC=CC2CNC(c2csc(C(N)=O)n2)=O)=O)c(C)c1C c1(N2CCC(CC#C)C2)ccc(CN=C(NC(C)C)NC2CC3(CCC3)C2)cc1 C(CC(C)(C)C(=O)N1CCC1CNC(=O)Cn1ccc(=O)cc1C)OC c1(C(=O)NCCC2(O)CN(C(C(C)OCCOC)=O)C2)cc(C2CC2)cc(Cl)c1 c12cccc(c1)O2.C1(NC(C2(OC)CCOC2)=O)CNCCOC1 Cc1ccc(CN2CCC(=CC(=O)NC3CONC3=O)CC2)c(O)c1 CC1(C)CCC(CNC(=O)CCc2ccco2)N(C(=O)C(C)(C)F)C1 N#Cc1ccc(=NCC2CN(C(C3CC3C(N)=O)=O)C2)[nH]c1 C1(CCC)(NC(=O)CCCOC)CCCN(C(c2cnn(C(C)(C)C)c2)=O)C1 C1(C(N2CCCC2Cn2cc(COC3CC3)nn2)=O)CCc2ncncc2C1 c1(C(=O)NC(CCNC(C2(C=C)CC2)=O)C)ccc(S(=O)(=O)N2CCCCC2)o1 c1(CC(N2CC(N(C)C(C3CCCC3)=O)C2)=O)cccc([N+](=O)[O-])c1 CC(F)(F)C(C)(C)C(=O)NCC1CN(C(c2csc(CO)n2)=O)CC1O C1(NC(C2C(C)(C)CC2)=O)C2CCC1CN(C(C1CC1C(F)(F)F)=O)C2 c1(OC)cccc(C2CC(C)CN2C(c2cncn2C)=O)c1 Cc1ccn(CC(N2CCN(C(=O)CCCC3CCCC3)C(C)C2)=O)c(=O)c1 N1(C(CCCCCCCSC)=O)CC2C(CO)C2C1.C12(CC1)CC(=O)NC2 C1(NC(Cn2ccc(C)n2)=O)CC(C)CN(C(=O)NC2CC2c2ccno2)C1 c1(C(=O)NCC(CNC(c2cncc(C)n2)=O)CO)c(C(F)F)cccc1N c1(C(=O)NC(CCNC(c2ccn(CC(C)C)n2)=O)C(C)C)cc(O)ncc1F CC1(C)CC(NC(=O)C(O)CCCc2ccccc2)CN(C(c2cncs2)=O)C1 N1(C(c2c(CC)con2)=O)CCC(NC(c2cc(-c3ccco3)c[nH]2)=O)C(O)C1 C1(C(N2C(C3(NC(C(F)OC)=O)CC3)CCC2)=O)CC12CCOC2 CC(CCCCNC(=O)C1=C(Cl)CC1)NC(C12CC(CO)(C1)C2)=O CC1(C)CC(NC(=O)C(=O)NC2CC3CC2CC3(F)F)CCS1(=O)=O C(C(=O)N1CCC(CCCO)C1)(C(C)O)NC(C1CC(C(C)C)C1)=O N1(C(=O)Nc2c(CC(C)C)nc(C)s2)CCC(C(=O)OC(C)(C)C)C1(C)C C(=O)(C1=NN(c2ccccc2)C(=O)C1)NCC(c1scc(C)n1)C c1(C(=O)NCC2CC(NC(C(c3ccc(C)cn3)(F)F)=O)C2)cccc(C)c1F C(c1cccc(F)c1F)=CC(=O)NC1C=CCN(C(C2(Cl)CC2(F)F)=O)C1 CC(C)(CC(=O)NCC1CCC(F)C1)n1cc(CC2CCSCC2)nn1 C1(CC)CN(C(=O)CCC(C)OC(C)(C)C)CCC1NC(C1CCCOC1)=O c1(C(=O)NCCC(C(C)C)NC(CSCCCC)=O)ccc(C(F)(F)F)c(C)c1 C(=O)(C(O)CC(N)=O)N(c1nnc(NC(=O)C(F)CC2CCCC2)s1)C Cc1nsc(CN(C)C(C2(CNC(=O)CC3CCSC3)CCC2)=O)n1 C1(OC)(CNC(=O)CCCN(C)C)CN(C(C2OCCC2C)=O)C1 CC(C)CC(=O)N1CCCC1C(N1CCC(CN=[N+]=[N-])C1)=O Cn1nc(C2CCC2)cc1C(=O)NCC1(O)CC(NC(=O)CC#N)C1 N1(C(C2CC(C#N)C2)=O)CCN(C(=O)CC2CCCOC2)CC1CC(F)(F)F c1(NC(C2(C)N(C(C(C3CCC3)OC)=O)CCC2)=O)cnc(F)cc1C Nc1ccnc2c1CN(N1CCC(Cc3c[nH]c4ccc(F)cc34)CC1)CC2 C1(NC(c2cc3sccc3s2)=O)CN(C(c2ccc(F)cc2Br)=O)CCC1O CC(CC(C)(C)C)C(=O)OCc1ccc(Cl)cc1 CC(C)CCC(=O)N(C1C=CC(C(=O)NC2CCN(CC(C)C)C2)C1)C(C)C C(=O)(CCC(C)(F)F)NCC1N(C(CCNC(=O)OC)=O)CCCC1 n1(CC(=O)N(C2CCN(C(=O)CC(=O)NC3CC3)C2)CC)cccc(N)c1=O C1(C(=O)Nc2ccccc2-c2nn[nH]n2)CN(CC2CC3CCC2O3)CC1(F)F c1(C(=O)NC(C)CNC(c2csc3nnsc23)=O)cc2cn[nH]c2cn1 c1(CC)ncnc(CC)c1C(=O)N(CC(O)CNC(C1(C)COC1)=O)C C12(C(=O)NCCC(C)NC(c3c(C)n(C(C)(C)C)nc3)=O)CCN(C1)S(=O)(=O)C2 c1(C(=O)NCCC2CCCN(Cc3ncc(OC)cn3)C2)nc(C)c(C)nc1C C12(CC)CN(CCO1)C(=O)N2.c1(COC)nnc(C(F)F)s1 Cn1nc(C(N2CCOCC2C(C)(C)C)=O)c2c1CCC(F)(F)C2 C1(NC)CCC(C(=O)OC)CC1.c12ccc(cc1)CCNC(=O)CC2C Cc1ccc(C2(C(=O)N)CC2C(=O)NC2C=CCN(Cc3ccccc3)C2)cc1 N1(C(CC=C=C)=O)CCC2CCN(C(=O)C(C)(C)CCOC)CC2C1 N1(C(C2C(C)C2)=O)CCC2CN(C(c3ccc(CC4CC4)s3)=O)CC12 C(=O)(CCCN(C)N=O)N1CCC(N(C(CC2CN(C)C2)=O)C)C1 c1(C(N2CCC(NC(C(N3CCOCC3)C)=O)C2C)=O)cccc(Cl)c1F c1(C(N(CC(CC)CC)CC)=O)n[nH]c2c1CCCCC2 Cc1cccc(O)c1C(=O)N(C)CC1CN(c2ncc3c(n2)CCC3)C1 c1(C(=O)NCC(C2CCCN(C(C=NOC)=O)C2)(C)O)cnc(O)n(C)c1=O N1(C(c2c(OC)csc2)=O)CC(NC(=O)Cn2cnnc2)CC(O)C1 Cc1cnc2c(C(=O)NC3CC(N(C)C(C4CC(C5CC5)C4)=O)C3)cccc2n1 c1(C(=O)NCC(C)(C2CC2)NC(=O)Cn2cnnn2)cnn(CC2CC2)c1 N1C(C)CCC12CCC2.C(c1ccncn1)=CC(=O)NC=O Cn1ccc(C(=O)NCCCC(=O)Nc2ccc(Cl)cc2)c1CC(=O)O N1(C(CNC(CCC2C(C)C2)=O)=O)CCN(C(C2CC2CC(C)(C)C)=O)CC1 c1(CC)cnn(CC(=O)NC2(CCNC(=O)CC3(O)CCC3)CCC2)c1 CC1(C)CCCC1(C)NC(=O)CC12CCC1CN(C(C1CCCN1C1CC1)=O)C2 N1(C(c2cncc(OC(C)C)c2)=O)CCC2(CCC2)C(NC(=O)C(F)C(C)C)C1 Cc1cccc(CC(N2CCN(C(=O)CNC(C3SCCC3C)=O)CC2)=O)c1F C1(CC(N2CC(N(C)C(C3NC(=O)C4CC34)=O)C2)=O)Oc2ccccc2NC1=O CCCC(C)(C)C(=O)NCC1CC(NC(c2cc(=N)[nH]n2C)=O)C1 c1(C2(C(N(CC(C)(C)NC(C=C(C)C)=O)C)=O)CC2)ccc(C)c(C)c1 N1(C(C(COC)OC)=O)CCC(C(C)(C)NC(c2csc(C)c2)=O)CC1 c1(CCC(=O)NCC(C)N(C)Cc2cc(C)n(C)n2)nnc(O)nc1O CC1(CN2CC(c3cn(CC(=O)NC4CC(N)CCO4)nn3)(O)C2)CCCOC1 C1(OC)CC(CNC(=O)CCC(F)F)N(C(=O)CCC2(C)CC2(F)F)C1 Cc1nn(C)c2c(NCC(F)(F)Br)nc(N3CC4CCC4(C)C3)nc12 C(=O)(C(C(C)C)OCC)N1C(N(C(CC=CCC)=O)CCO)CCC1 c1(C(=O)N(C(c2c(CC)cccc2)CNC(=O)C=CSC)CC)cc(C)ccc1Cl C1(NC(C(CC=C)(C)C)=O)CC1C1CCN(C(c2cc(C#N)cn2C)=O)CC1 C1(CC(C)C)(C(=O)NCCOC2CN(C(=O)CC3CC3(Cl)Cl)C2)CCCCC1 C1(C(=O)OCC(O)C(F)(F)F)CCC2C1C2(F)F C1(OC)CC(C(=O)NCc2ccc(CO)o2)N(C(c2coc(C)n2)=O)C1 C1(CCC)(NC(C2CSC2)=O)CCCN(C(=O)CCc2cnoc2)C1 CC1CC(NC(C2CCCC2(C)C)=O)CN1C(c1cc(-c2cnn(C)c2)on1)=O c1(OCC)ccc(NC(=O)C(=O)NC2CCC(C(C)(C)C)C2)cc1.C1CC(=O)N1 C=CCC(C(=O)NCC(C1CC1)N(C(=O)C=CCN1CCOCC1)C)C(C)C c1(CN(C(=O)C(=O)N(C)C(c2ccccn2)C)C(C)C)cccc(F)c1I N1(C(CN(CCOC)C)=O)CCC2CCC(NC(C3(c4cc[nH]n4)CC3)=O)C1C2 C1(CC(=O)N(CCOCCNC(c2c(CC)non2)=O)C)COCC1(C)C Cc1sc(C)c(S(=O)(=O)NCCNOCc2cc(F)cc(F)c2)c1C(F)(F)F N1(Cc2nc(C(C)C)on2)CCCC(C(C)NC(c2cc(F)n(C)n2)=O)C1 C12(CN(C=O)Cc3c(CC)noc3)CC(CCO1)C2 c1(C(N2CC(CC)N(C(C3C4CCCCCC34)=O)CC2)=O)cc(C)nc(C)c1O N1(C(c2c(C)[nH]cc2)=O)CC2(CCC2)CC1C(N1CCC(CCF)CC1)=O N1(C(C(C)SC(C)C)=O)CCCCCC(NC(c2cc(CC3CC3)on2)=O)C1 c1(C(=O)NC2CN(C(c3n(CC(=O)OC)nc(C)c3)=O)C2)cc(C)cc(C)c1 C1(C)(COC)CCCN1C(=O)CCC1CN(C(=O)CCCOC(C)=O)C1 c1(C(N(CC(C)NC(c2ccc(COC)o2)=O)C)=O)c(F)cc(F)cc1F c1(NC(=O)NC2CCCC(F)(F)CC2)cc(Cl)c(OC(F)F)c(Cl)c1 C1(C(=O)NCCC(CNC(c2csc3nnsc23)=O)O)Cc2cccc(F)c2O1 CC1CN(C(=O)C(c2ccc(O)cc2)=O)CC(C)N(C(=O)CN(S(C)(=O)=O)C)C1 N1(C(c2n(C)ccc2)=O)CCC(C2CC(NC(c3ncccc3Br)=O)C2)C1 N1(C(C(C2CCCOC2)OC)=O)CCC(CNC(=O)CC(F)(F)F)C(F)(F)C1 N1(C(CC(CC)SC)=O)CC(OC)C(C(=O)NC2(N3CCCCC3=O)CC2)C1 c1(C(=O)NC(c2ccccc2)C(=O)NCC(C)N=[N+]=[N-])cn2c(n1)CCC2 N1(CC(=O)N(CC(CN(C(c2c(CC)csc2)=O)C)O)C)CCCNS1(=O)=O Cc1cn2c(n1)CCC(C(N1CCC(C)C(NC(=O)CCC3(C)CC3)C1C)=O)C2 C(=O)(CC(C)C(C)C(C)C)N1CCN(C(Cn2ccc(C)n2)=O)C(C(C)C)C1 c1(C(=O)NC(C(C)NC(C2CC(=C)C2)=O)C2CC2)ccc(CCC)cc1 CC(CCCNC(c1cc(Cl)ns1)=O)NC(C1(Br)CC1)=O C#CC(C)(C)C(=O)NC1C=CC(C(N2C(C)CC2(C)C)=O)C1 CN1CCCC(F)(C(=O)NCCCC2CCCCN2C(C2(F)CCC2)=O)C1 CCC(COC)C(=O)N1CC(CCNC(=O)CC(C)(C)O)(OC)C1 c1(C(=O)NCCCCc2ccccc2Br)cc([N+](=O)[O-])ccn1 c1(CC)cccc(CC)c1CC(N1C2CN(C(=O)OC(C)(C)C)CC12)=O.C(C)(=O)O Cc1oc(C(C)(C)C)cc1C(=O)NC(C1(O)CCN(C(c2ncn(C)n2)=O)C1)C N1(C(C2CCC(=O)NC2)=O)CC(NC(c2csc(C(F)(F)F)n2)=O)C2CC2C1 C1(C(=O)NCC(=Cc2cn(C)nn2)F)CC(NC(c2cncnc2)=O)C12CCC2 C(=O)(CCC(C)S(C)(=O)=O)NCC1CN(C(C(CCC)C#N)=O)C1 N1(C(C2(c3ccccc3)CC(F)(F)C2)=O)CC2(CCN2C(C2COC(=O)C2)=O)C1 c1(N2CCC(C)C2CNC(=O)CC2=CCN(C)CC2)nc2cccc(F)c2o1 C1(NC(N2CC(N(C(CC3(OC)CCC3)=O)C)C2)=O)CCCC12CCC2 C1(C(=O)NC2(C3N(C(C4CC(=O)NC4)=O)CCC3)CC2)CN(S(N)(=O)=O)C1 C(=O)(C1=CN=C2N=CNN2C1)NC1C(C)CN(C(C2CC(N(C)C)C2)=O)CC1 C(CC(O)C(=O)Nc1ccnc(OC)c1)NC(CCN(CCC)C)=O C(CNC(=O)C(=C1CCCCC1)F)(C(=O)NC(C(N)=O)C1CCCC1)N(C)C O=C(CC(F)(F)C(F)F)NCCC1(O)CCCN(C(C2CC2(F)Cl)=O)C1 c1(C(=O)NC2C(NC(CCOC(C)C)=O)CCC2)noc2c1COCC2 C1(CN(C(CCOC(C)=O)=O)C)CCCCN1C(C1CCC1(C)C)=O C1(CC(=O)NC2C(O)CCN(C(c3c(CC)c[nH]n3)=O)C2)CC(C)CC(C)(C)C1 c1(CC(=O)NC(CC)CNC(c2nn(C)cc2C)=O)cccc2c(C)csc12 c1(C(=O)NCC(CNC(CC(C)F)=O)F)ccc(-c2ccncc2)cc1 c1(COCC(=O)NC2C(NC(COC(CC)C)=O)CC2)nc(C)no1 C1(OCC)CCN(C(C2CC2C(c2c[nH]c(C(F)(F)F)c2)N(C)C)=O)CC1 CCC(C#N)(CC)C(=O)N1CC2CN(C(=O)Cc3ccc(SC)cc3)CCC12 c1(C(N2CCC(CC(C)NC(C3CCCCO3)=O)CC2)=O)cc(N)cc(F)c1 C1(N(C(CCCSC)=O)CC2CC2)CCN(C(C23CCC2C3)=O)CC1 C1(CNC(c2ccc(OC)cc2F)=O)CN(C(=O)C2=CCC2)C2(CCOCC2)C1 c1(C(N2CCC(C(N(CC)CC)=O)C2)=O)cc(C)sc1C c1(NC(CC(N2CC=C(CNC(COC)=O)CC2)=O)=O)ccc(Cl)cc1C c1(CNC(c2nnnn2C)C2C(C)(C)C2)cnn(CC(F)(F)F)n1.CC(F)(F)F N(C(=NCCOC)N1CCCC(CC=C)(NC)C1)C1CC(C(=O)OCC)C1 C(=O)(CC(C(C)(C)C)NC(c1ccnnc1)=O)NCCC(C)CCO C(C)(C)NCC=CCOC(C)=O.C(C)=O N1(C(C2CCCOC2)C(=O)OC)CCC(NC(=O)COCCO)CC1 CCC(C)(C)C(O)C(=O)N(C(C)(C(=O)N(CC(C(C)C)OC)C)C1CC1)C c1(CNC(=O)C=Cc2ncc[nH]2)cccc2c1CCN(C(C13CC(O)C1C3)=O)C2 C1(Cn2cc(-c3cccc(Br)c3)nn2)C2(CCC2)C12CCC2 C1(C(NOC(C=C)C)=O)CCC(C)(C)N(C(c2nnc(O)nc2O)=O)C1 C(=O)(C(C)(C)C(=O)N1CC(CC(N2CC3(CCN3C)C2)=O)C2(CC2)C1)NC c1(C(N(CCCN(C(C2(OCC)CCC2)=O)C)C)=O)ccc(N)c([N+](=O)[O-])c1 C1(C(=O)Nc2cncs2)CC(O)CCN1Cc1cccc(Br)c1Cl c1(C(N2CCC(N(C(=O)CCC3CC3(Cl)Cl)CCO)C2)=O)ccc2c(c1)OCC2 Cc1n[nH]c(Cl)c1CC(=O)NC1CCCC(NC(=O)C=CCN2CCCCC2)C1 C(=O)(C(CC(C)C)NC(c1cc(CNC(C2CC2Cl)=O)on1)=O)NC c1(C(=O)NCC2(F)CCN(C(Cc3cc(OC)no3)=O)C2)cnc(C)nc1C N(C(=NCc1noc(C(C)(C)C)n1)NC1CCC1)C(C)CF CC1=C(C(=O)NCCC2CSCCN2C(c2cnc(N)c(N)c2)=O)CCCC1 C1(=O)C(CC2(C#N)CC2)N(C)CC(C2CCCO2)N1.N1(CC)CC(C)(C)C1 c1(C(C)C)nocc1CNC(C1(CNC(=O)C(N2CCOCC2)C)CCCO1)=O C1(C)(C(=O)NCCOCCCNC(c2c(C)cco2)=O)CCN(C(=O)N(C)C)C1 c1(C(=O)NCC2(O)CC(CNC(COCCCC(C)C)=O)C2)cn(C)nc1O CCC1(C)CNC(=O)C(C2CCCC2)N1.c1ccccn1.C(=O)(CSC(C)C)N C(C(O)(CNC(C1(CNC(=O)C(C2CCC2)OC)CC12CCC2)=O)CO)OC CCCCC(C(=O)N1CC(CC(F)C(=O)NOCCOCCO)C1)OCCO c1(CC)ncncc1C(=O)NCCN(C(c1cc(C)ns1)=O)CC N1(C(=O)NCCc2ccco2)C2CCC1CC(OCF)C2 C(=O)(C#CC1(C)CCCO1)NCC1C(CNC(c2c(C)noc2C2CC2)=O)C1 Cc1cccc(C2CC2C(=O)NCCCC2CCCN2C(c2cnc[nH]2)=O)c1 C=CCC(C(=O)N1CCCC1c1cn(C(c2cccnc2F)C)nn1)C(C)C N#Cc1ccsc1C(=O)NCC1CCC1NC(c1ccnc(-n2cccn2)c1)=O CCCCC(CCC)(c1nnnn1C1CCOCC1)NC(COC)C1CC1 C(=O)(C(Cc1cc[nH]n1)NC(C1CCCN1C)=O)N1C(C(N(C)C)=O)CC1 C1(C(=O)NCC2C(NC(Cc3cn(C)nc3)=O)COC2)COC(C)(C)C1 C1(NC(=O)Cc2cc(C3CC3)on2)CC2CC1N(C(=O)C(O)C1CCCC1)C2 C=C=CC(C)C(=O)NC1CCCCC1NC(C1(CS(N)(=O)=O)COC1)=O c1(N2CC(C(C)NC(C=C(C)C(C)C)=O)OCC2)cncc(C#N)n1 C(CCCCC(=O)NC1(CC2CC2)CCC1)NC(C=CC(C)C)=O C(=O)(CCCC(=O)NC)NC1CC(CNC(C2C(C(=O)NCC#C)C2)=O)C(O)C1 C(c1ccccc1)=CC(=O)N(CC(C)NC(=O)C(C)Cc1ccnn1C)C c1(OCC(=O)N(C(CN(C(CSS(CC)(=O)=O)=O)C)C)C)ccccc1Cl N1(C(c2ccc(CC)o2)=O)CCC(CO)C(NC(=O)C(C(C)C)NS(C)(=O)=O)C1 CC1CC(C)CC(c2nnnn2CCCOC)(Nc2cnsc2)C1.C1(C)CC1 C1(CNC(C2(CC#C)CCCC2)=O)CC(F)(F)CN1C(c1ccncc1Br)=O C(=O)(CCC(F)(F)C(F)F)NCCC(C)N(C(C(CC(C)C)NC(=O)OC)=O)C C(c1ccc(C)cc1)=CCC(=O)NCC1(C)N(C(CC)=O)CCC1 C(=O)(C1=CCCCO1)NC(COC)CNC(=O)Cc1cccn1C O=C(C1CCc2c(Cl)cccc21)Nc1cnn(-c2ccncc2)c1 CCCC(C)(C(=O)OC)NC(c1occ2c1CCC2)=O c1(-c2ccc(CCC)s2)cc(C(=O)NCCNC(=O)N(C)C)c(F)cc1C C(N=c1[nH]c(Cl)ncc1C(C)=O)C1C(NC(c2cc(SC)oc2)=O)CCCC1 c1(C(=O)NCCN(C(=O)C(C)=C2CCCC2)CCOC)ccnc2cc[nH]c12 CC1CCN(C(=O)C(C)(F)F)CCN1C(=O)CNCc1cccc(C(C)(C)C)c1 N1(C(c2c(C)ncn2C)=O)CC2(CC2)CC1CNC(=O)C=CC(C)C c1(C(N2CCC(CO)C2)C(=O)NCCC)cc2ccnc(Cl)c2s1 C1(CNC(C2C(CCC)C2)=O)CCCN(C(c2csc(Br)c2)=O)CC1 c1(C(=O)NC(C)CC(C)NC(=O)COC2CCC2)cc(O)cc(=O)o1 C1(C(=O)NC(c2ccncc2)C)C2CCN(C(C3COCCC3C)=O)CC12 N1(C(C(C)=CC2CC2)=O)CC(C2CC2C(N2CC(C(C)C)C2)=O)C1 Cc1c(C(N2CC(CO)(NC(C3C(C)(C)C3(C)C)=O)C2)=O)ccc2ccccc12 N1(C(C2C(=O)OCC2)=O)CC2CC1CN(C(c1cc(Br)co1)=O)C2 Cc1sc(O)nc1C(=O)NC1CCC(CNC(c2cn(CC(N)=O)nn2)=O)CC1 C1(NC(C(C)NC(N)=O)=O)CCCN1C(C1(NC(=O)OC)CCCC1)=O CCC(C)C(O)C(C)C(=O)N(C1CCN(C(=O)CNC(=O)C(C)CC)CC1)C C1(CC(=O)NC2(CCCCNC(C(C)c3cccs3)=O)CC2)CCCNC1=O c1(C(N(CC(C)(C)CNC(=O)Cc2csnn2)CC)=O)cc2n(n1)CCCC2=O c1(C(N2C(C(=O)NCCOc3cn[nH]c3)CCC2)=O)ccc(N2CCC2)nc1 N1(C(c2c(CC)sc(=N)[nH]2)=O)CCC2CCCN(C(=O)C=C3CCCC3)C2C1 C1(C)(CC)CCCN(C(=O)C(F)C(C)CNC(=O)CSC2CC2)CC1 CC(C(=O)N(CC(C)Nc1ncnc2c1ncn2C)C)C(C)S(C)(=O)=O c1(N2C(=O)NCC3(C4CC4)CC(C3)C2)cccc(C(CCCC)=O)c1.C(=O)N.OCC Cc1c(C(N2CCCC(CNC(c3ncc(Cl)n3C)=O)C2)=O)cccc1Cl C=CCC(CC)N=c1[nH]c(N2CCOC(C(=O)NC)C2)nc2cc([N+](=O)[O-])ccc12 c1(OC)c(C(=O)N(CCCCCNC(=O)C2=CCOC2)C)cccc1Br N1(C(c2ccc(COC)o2)=O)CCSCC1C(=O)NC(c1ccc(C)s1)C C1(O)(CN(C(=O)C2=CCCCO2)C)CCCN(C(C23CC(C(F)F)(CO2)C3)=O)C1 c1(-c2nnc(C(=O)N(CC)CC)n2-c2ccccc2)csc2cccc(OC)c12 C=CC1CN(C(C2CC2C(=O)NCc2ccccc2)=O)CC1NC(=O)CSC1CC1 C1(C)(C(=O)NC(COC)CCO)CCCN(C(=O)CN=[N+]=[N-])C1 CN1CCC(CO)(CNC(C2CCC(NC(=O)Cc3cn(C)cn3)CC2)=O)CC1 c1(NC(CCN(C)C(C2(O)COC2)=O)C)ncnc2[nH]c3ccccc3c12 C(=O)(CCC(N)=O)N(C(CN(C(C(C)n1ccnc1)=O)C)C)C c1(C(=O)NCC2N(C(C3(C)CCCC3O)=O)CC2)cc(C2CC2)cc(F)c1 C1(C(N(CC(CNC(c2cc(SC)oc2)=O)O)C)=O)CC(=O)N(C)C1 CCC(F)(F)C(C)(C)C(=O)N1CC(CCNC(c2ncoc2C(C)C)=O)OC(C)C1 CCCCC(CCCC)C(=O)NCCC(C)NC(=O)CC1CSC1 C1(SC)CCN(C(C2CCC(Cn3cc(C(C)(C)NC(C)C)nn3)C2)=O)C1 C1(C(N(CCCNC(c2cnco2)=O)C2CC2)=O)CCOCC12CCC2 Cc1cc(C)c(C(N2C(C(=O)NCc3cnc(Cl)s3)CC3CC23)=O)cn1 CCC(CC)C(C)C(=O)NC1CN(C(C2CCN(C(=O)OC)CC2)=O)CCC1F Cc1nnc(NC2CC(NC(C3(CCF)CC3)=O)C23CCC3)nc1C c1(NC(C(C)C)=O)ccc(Cl)c(C(=O)N(C)CCN(C(=O)C(C)CF)C)c1 C1(NC(=O)Nc2c(C)coc2)C2C=CC(c3ccc(C(F)(F)F)cc3)C12 c1(SCC2CN(C(=O)CCc3ncco3)C2)cccc(Br)c1 CC(C)CCC(C)N(C)C(C1C(C)CCN1C(c1cncn1C)=O)=O C1(NC(C(c2ccc(Cl)cc2)CC)=O)CCCCC1NC(=O)CC(C)(C)C1CC1 c1(SC)nn(C)cc1C(=O)NCC(C)N(C)C(C1CCN(C)C1C)=O N1(C(CCN(C(=O)CCC2CCCOC2)C2CC2)=O)CC2(CCC1CO)CC2 c1(C(N2C(CN(C(COC)=O)C)CCC2)=O)cccc(-n2c(C)nnc2O)c1 C(=O)(CCC(=O)NCC1C(C)CCN1C(c1cnc(C(C)C)nc1C)=O)OCC C12(C(N3CCCC(CO)(NC(C4CCCOC4)=O)C3)=O)C3C4C1C1C2C3C41CO c1(OC)cc(C(=O)NC(C2C(NC(c3scc(CO)n3)=O)C2)=O)cc(C)c1 Cc1cc(F)c(CC(=O)N(CCC(C)NC(C2CCC23CCC3)=O)C)cc1F C(=O)(C(C)(CNC(=O)CCC1CCCCO1)CC)NC(CC=C)C C(=O)(CCC(C)(C)C)N1CC(C(=O)NC(c2cc(C)on2)C)(SC)C1 C#Cc1ccccc1CC(N1CCOC(CNC(=O)Cc2ccsc2C)CC1)=O Cc1cc(C(N2CCCC(CNC(=O)C(C)SC(C)C)C2)=O)ncc1C#N C1(NC(C2(Cl)CC2)=O)CCCCC12CCN(C(C1CC1(F)F)=O)C2 C(C(C(=O)NCCC1CC1)N(C)Cc1ccc(OCCO)cc1)(C1CC1)OC C1(CNC(=O)C=C2CCC2)C2CN(C(c3ccccc3)=O)CC12 C1(NC(c2cc(CC)on2)=O)CCN(C(C2COC2)=O)CCC1c1ccccc1 C=C(C)CC(C)C(=O)N1CC(CC)(NC(=O)CCN2C(=O)CCC2=O)C1 N1(C(c2cc([N+](=O)[O-])sn2)C(=O)NCCOCC)CCOC2(CCCC2)C1 C1(C(N2CC(C)(CC)C2)=O)(CNC(C2SCC=C2C)=O)CCCCC1 N1(C(CC(C=C)CC)=O)CCC2(C=C(C(=O)Nn3cncn3)C2)C1 N1(C(CCc2cnn(C)n2)=O)CC2CC(C1)N(C(c1cc(Cl)nnc1O)=O)C2 c1(C(=O)NC(CCCC)CNC(C23CC(CN2C2CC2)C3)=O)cc(Cl)ccc1O C1(C)(NC(C(C)Oc2ccc(OC)cc2)=O)CCCN(C(=O)CCCC2CC2)C1 C1(C(=O)NCC2C3CN(C(c4c(C)cc(C)nc4)=O)CC32)CC2(CCC2)CCO1 Cn1ncc(Br)c1S(=O)(=O)NC1(C(=O)Nc2cccc(Br)c2)CC1 c1(OC)ccccc1C(N1CCC(C(=O)N(C)CCF)(CO)C1)=O Cc1nccc(Cl)c1C(=O)NC(CO)CCCNC(c1ccc(Cl)c(N)c1)=O c1(CC)ccc(Cl)c(C(=O)NCCCCNC(c2ccc(C(F)F)c(F)c2)=O)c1 c1(CNC(C2CC(C)CN(C(=O)CC#N)C2)=O)cc(Br)cc(C#N)c1 C1(NC(=O)Cc2ccsc2)CCN(S(=O)(=O)Cc2ccccn2)C1 c1(C(N2CC(COC)N(C(c3cnns3)=O)CC2)=O)c[nH]c2ccc(O)cc12 N1(C(CN(C(=O)C(C)CF)CC)=O)CCC(C(C)(C)CNC(C(C)=CC)=O)CC1 C(=O)(CCCC(=O)NCC1CCC(NC(=O)COC2CCCOC2)C1)OC c1(CNC(=O)NCCc2n(C)nnn2)cccc2cn(C(C)(C)C)nc12 Cc1ccc(C(N2CC(C(=O)NCCOc3ccon3)CC(F)C2)=O)c(F)c1 Cn1cc(Br)c2c(NCC(c3ccccc3)NC(c3c[nH]c(=N)s3)=O)ncnc12 N1(C(C(CCC)OC)=O)CCC2C(C1)NC(=O)CN2C(c1cn(C(C)C)cn1)=O C=CCN=c1[nH]c(C(=O)N(CC(O)CN(C)C(C2COC(C)(C)C2)=O)C)cs1 N1(C(C(C)(F)F)=O)CC(NC(C2(Cc3ccc(F)cc3)CC2)=O)C2CC2C1 C1(NC(C2CCC(C)(C)C2)=O)CN(C(c2cnccn2)=O)CCC1F C1(NC(CC2CCN(C(C(C)OCCC=C)=O)CC2)=O)CCCCC12CC2 C=CCCCCCC(=O)N1CCC(NC(=O)COC(F)(F)F)C(CO)CC1 C1(NC(c2c(CC)ocn2)=O)CN(C(c2cc(Cl)cn2CC)=O)CC2CCCC12 C1(OCC(=O)NC(C(=O)N(CC(=O)N(C(C)C)C)C)C)CCCCC1 c1(C(C(C(C)C)NCC(O)Cc2cccnc2)c2ccco2)ccc(C#N)cc1 N1(C(CC=C)=O)CCCC(CCC2CCCN2C(c2cnn(CCCC)c2C)=O)C1 N1(C(c2cn(C(CC)C)nc2)C(=O)NCc2ccco2)CCC(C)C(F)(F)C1 C1(CC(=O)NCCNC(COCCC=C)=O)COCCO1 N1(C(CCC2CC(NC(CC(CN(C)C)O)=O)C2)=O)CCn2c(O)nnc2C1 C(=O)(C1=NOC(CNC(C23CCCC2CCC3)=O)C1)C1CC(CC)(COC)C1 c1(C(=O)NCC2(NC(c3cc[nH]c3)=O)CC2)cc(Cl)n(-c2ccccc2)n1 c1(CNC(C(C)C2CCC2)=O)nc(CNC(c2ccc([N+](=O)[O-])o2)=O)cc(O)n1 Cc1cocc1C(=O)NCC1CC(NC(C2CC2(C)C(F)(F)F)=O)C1 c1(NCC(C(C)(C)O)(C)C)nccc(=NCCCC2CC2)[nH]1 N1(C(C(CC)SC)=O)CCC(C(=O)NC2CC(CC(=O)O)C2)(CO)C1 c1(CC)ccc(C(=O)N(CCNC(C2CSCCS2)=O)C(C)C)c(C(F)(F)F)c1 C=C1CC2CC1CN2C(=O)C1=NOC(CNC(c2c(CC)cccc2F)=O)C1 c1(C(N2CC(N(C(C(c3ccc(F)cc3)CC)=O)C)C2)=O)[nH]cc(C)c1C C(=O)(C(F)(F)C(C)O)NC1CC(NC(C=CC=CC)=O)C1 C(=O)(CC(C)(O)C(F)(F)F)NCCCCNC(C(CC)n1cncn1)=O N1(C(CNC(CC)=O)=O)CCC(O)C(NC(c2ccnn2C)=O)C1 C1(C(N(C2CCCN(C(C3N(CC)CCOC3)=O)C2)CC)=O)CCC2(CCC2)O1 N1(C(C(c2ccccc2)C)=O)CCC2(Nc3nccc(OC(F)F)n3)CCCC12 c1(C(N2CC(C)(C)C(CNC(=O)COC3CCOC3)C2)=O)ccc2[nH]ccc2n1 N1(C(CCN(CC)CC)=O)CCN(C(=O)C(O)C(C)c2cccs2)C(C)C1 C(C)(CNC(=O)CC1(N(C)C)CCCC1)(C(C)C)NC(c1ncc(C)[nH]1)=O N(C1COc2ccccc21)C(NNC(=O)C1CCN(c2ncccc2F)CC1)=O Cc1cc(C(=O)NNC(=O)OC(F)(F)F)sc1C Cc1c(C(N2CCC(O)C(NC(=O)CNc3ccc(O)cc3)C2)=O)cccc1F CC1(C(=O)Nc2ccc(SC(F)(F)F)cc2)CCCN(C(C2CCCCO2)=O)C1 Cc1cnc(S(C)(=O)=O)[nH]c1=NC1COC2(CCN(Cc3ncc[nH]3)CC2)C1 CC1CCCC=C1C(=O)NCC1(C)CCCN1C(c1cc(Br)co1)=O c1(OC(C23CCCCC2CCC3)=O)ccc2nc(Cl)cnc2c1 CC(CC(C)(F)F)C(=O)N1CC(C(C)NC(c2csc(C(F)(F)F)n2)=O)C1 O=C1CC(NC2(CO)CCOCC2)CC(=O)N1 c1(C(N2C(CNC(c3cc(C)sc3)=O)CCC(C)C2)=O)cccc2oc(C)cc12 N1(C(C(CC)OC2CCCC2)=O)CC2CC2(NC(c2cnc(C)nc2)=O)C1 C(=O)(C(F)(F)C(C)O)N1CC(O)(C(C)(C)NC(c2scc(C)n2)=O)C1 C1(CCNC(c2c(C)cc[nH]2)=O)CCN(C(c2cc(Br)co2)=O)C(C)C1 CC(C)(C(=O)NC1CC(OCC(=O)NCCCCCCF)C1)C(F)(F)F N1(C(CCCCC)=O)CCC2C(CCN2C(=O)CCc2c(C)nn(C)c2C)C1 C1(C(=O)NCCN(CC(C)O)C(=O)Cn2nc(C)oc2=O)(CC)CNC(=O)C1 C1(NC(c2scnc2C(F)F)=O)CCC(CC(=O)NCCC2CC(C(=O)OC)C2)O1 C(=O)(CCCCC(=O)N1CC(NC(C2(C)CC2C(F)(F)F)=O)C(O)C1)NC c1(OCC)ccc(CC)cc1.C1(C(=O)N)(O)CCC1.C12(CC1)C(=O)N(C)C2 c1ccc(SC(F)F)cc1.C(CC(CNC(=O)CC)NC(=O)CN1CC=CC1)OC C1(N(C(C(CC)C)=O)C)CCN(Cc2cccc(F)c2)CC1 N1(CC)CCCCC1CNC(=O)CC1CCCN(C(c2cncc(Cl)c2)=O)C1 N1(C(CC2CCC(NC(C(N3CCCCCC3)C)=O)C2)=O)CC2CCC(O)C2C1 c1(C(=O)NCC(CC)(CC)NC(c2cncc(OC)n2)=O)scc2c1CCCC2 C1(NC(C2CSC2)=O)CC(F)(F)CC1NC(=O)C=Cc1ccccn1 C1(O)(C(=O)NC2CN(C(c3cc(CC)sn3)=O)C(C)C2)CCC(C)(C)CC1 CCC(CCC(=O)N(C)OCC(O)CO)NC(C1(C(=O)OC)CC1C)=O CN1C(=O)OCC1CNC(=O)C=CCNC(=O)CC1CC(O)C1(C)C C1(C(=O)OC)C2CC1N(N(CC1CC1)CCc1cccc(C(N)=O)c1)C2 N1(C(CN2CC(C)C2)=O)C2CCC1C(NC(=O)CCF)C2 c1(NC(=O)Nc2c(C)ncs2)ccc2cc(CN3CCCCCC3=O)ccc2c1 C(c1cc(C)no1)=CC(=O)N(C1CCN(C(C2CN(S(C)(=O)=O)C2)=O)C1)C C1(C(=O)NC(Cc2cccc(C)c2)C)C2CCC(C2)N1C(=O)C=CC(F)(F)F C1(OC)CCC(c2cn(CC(c3ncoc3C(C3CC3)C3CC3)=O)nn2)CC1.CC(=O)O c1(C(=O)NCCCNC(CC2C(=O)NC(=N)S2)=O)cc(C2CC2)ccc1F N1(C(c2nccc(N(C)C)c2)=O)CC2CCC2(CNC(c2ccccc2Cl)=O)C1 N1(C(c2cn(CC)nc2)=O)CC2CN(C(c3n[nH]cc3Br)=O)CC(F)(F)C2C1 C1(CC=C)(NC(=O)CSc2cn[nH]c2)CCN(C(c2ocnc2C2CC2)=O)C1 C#Cc1ccc(C(=O)N(CC(C)CNC(c2cnn(C)c2)=O)C)nc1 N1(C(=O)NCc2n[nH]c3c2COC3)CCc2nnnn2CC1 C1(CNC(c2cn(CC=C)nc2)=O)CC(OC)CN1C(c1csc(C)c1)=O CC1C2CC(C2NC(C2(F)C(C)(C)C2(C)C)=O)N1C(=O)C=CC(F)(F)F C(CCCCC(=O)N1CC(O)(CCNC(=O)CCN(S(C)(=O)=O)C)C1)SC CP1(=O)CCN(CC(N2CCC(CCNC(c3cccc(F)c3)=O)CC2)=O)CC1 Cc1c(C(=O)NC(C)CC2CN(C(C3(C#N)CC(C)C3)=O)C2)sc2cncn12 c1(C(N(C)CC2(CNC(C3CCC(C(F)(F)F)O3)=O)CC2)=O)cscc1C#N c1(C(N2CC(O)(C(C)NC(=O)Cn3cccc3)C2)=O)cc2ccccc2o1 C(=O)(C(O)CC(F)(F)F)NCCN(C(c1cnc(NC2CC2)s1)=O)CC C(=O)(C1=NOC2(CCC2)C1)NCC1CCCN(C(CCN2C(C)CCCC2)=O)C1 c1(C(=O)NCC=CCNC(=O)CCc2nc[nH]n2)c[nH]nc1-c1ccoc1 c1(C(=O)NCC(C)NC(Cc2ccc(C(C(=O)OC)(C)C)s2)=O)cc(=O)n(C)cn1 N1(C(c2c(C)nns2)=O)CCCCC(CCC(=O)NC(C(F)(F)F)C2CC2)C1 C1(CC(=O)NCC(CN(C(C(F)OC)=O)C)C)Oc2ccccc2NC1=O CC1CCC(SC(C)C(=O)OC(C2CC(=C(C)C)C2)=O)CC1 CC1NC(=O)C2=C1N(CC1CCCO1)C(=S)NC2c1cnn2c1CCCC2 N1(C(CC(CNC(c2cc(C)oc2C)=O)C)=O)C2CCCC1CC2 C1(CNC(C2C(C)=CCS2)=O)CC(C(F)(F)F)CN1C(C1CC1F)=O C1(CNC(CC=CC)=O)CCCC12CCN(C(=O)Cn1ncccc1=O)CC2 CCCCC(=O)C(=O)NCCC(C)NC(c1cccc(C(F)F)c1F)=O c1(OC)ccc(CN2CC3C(C(=O)Nc4ccc(Cl)nc4OC)C3C2)c(C)c1 c1(C(=O)NC2CC(NC(CCN(CC)CC)=O)C2)cn(C2CC2)nc1C c1(C(N(CC(C)(C)C)CC)=O)cc(CNC(=O)C(O)C2CCCC2)nn1C c1(CC(=O)NCC2CCCCCN2C(c2cncc(Cl)c2)=O)cccc(F)c1F c1(C(N2CC(C)C(NC(c3cc(O)cc(O)n3)=O)C2)=O)cccc(Cl)c1Cl c1(OC)cccc(C(N2CC=CC2(C)CNC(c2c(C)coc2C)=O)=O)n1 N1(C(CC2N(C(c3c(N)cncn3)=O)CC(F)C2)=O)CCCC2OCCC2C1 c1(C(=O)NC(C(C)C)CO)ccc(OCCN(C)C)cc1 CC1(C)C(NC(=O)CCc2cccs2)CCN1C(=O)CCc1ccc(F)cc1 CCCC(CNC(=O)C(C1(O)CCCCC1)NC(=O)C(F)C(C)(F)F)CCC C1(C(=O)NOCCO)CC(O)CN1C(=O)CCn1cncn1 C1(C)(C(=O)OC)CCCN1C.c12ccc(o1)[nH]c2=O.n12cc(nn1)CNC1(CC1)C2 C1(NC(C(CC2CC2)OC)=O)CCOCC1C(=O)NCC(F)(F)C(C)C N1(C(C2CC(SC)C2)=O)CC(C)CN(C(c2nc(CC(C)C)sc2C)=O)CC1C c1(C(=O)NC2C=CCN(C(C=C(C)C(C)C)=O)C2)cc(C)c(C)nc1C c1(C(=O)Oc2c(CCC)nnn2-c2ccccc2)ccc2c(c1)CCNC2=O N1(C(C2CCCN(CC)C2)=O)CC(C(=O)NCC2(C)CC3CC3C2)C(C2CC2)C1 N1(C(C=Cc2cn(C)nc2)=O)CCCC2CN(C(c3nocc3Cl)=O)CCC12 C(=O)(C1CCOc2ccccc21)N1C(C(C)NC(CCSCC(C)C)=O)CCC1 CN1CCC(C(=O)NC(CNC(c2ccc([N+](=O)[O-])s2)=O)C2CCC2)CC1=O C(C)(C)(CCC(=O)NCC(CO)NC(C1C2CCC1CC2)=O)N(C)C Cc1nc(O)nc(O)c1CC(=O)NCCOCCN(c1ccco1)C C=CC(C)(CC)C(=O)N1CC(CCNC(=O)CCCOC)C2(CC2)C1 CCCN=C(NCCc1nc2c(s1)COCC2)N1CCC(C(F)F)CC1 C1(NC(C2CCC(C)CC2)=O)C2CC1N(C(=O)CN1CCC(CO)CC1)C2C c1(C(C)C(N2CCC(C)(CNC(=O)COCC3CC3)C2)=O)ccc(Cl)c(Cl)c1 C(=O)(C(C)(CO)NC(c1ccc(O)nc1)=O)NC(c1c(C)ncs1)C c1(C(=O)NC(C(=O)NCc2c(C)cn(C)n2)CO)cc(C)ncc1C C1(S(C)(=O)=O)(C(=O)NCC2CCN(C(CCCOCC=C)=O)CC2C)CCCC1 C1(N)COCCN(C=O)C1.C1(C(=O)NC(C2CCCC2)=O)(CC)CC1(F)F C1(CC(=O)NC2(CCNC(CCC=CCC=C)=O)CCC2)CCCC(F)(F)C1 C(=O)(C1=CCC(C)(C)CC1)NC1C2CN(C(c3ccc(C)cc3C(=O)NC)=O)C1C2 N1(c2nnc(C)o2)CCC(C2(NC(C3CCC3(C)C)=O)CC2)C1 Cc1cn2c(n1)CC(C(N1CC3CC3(CNC(=O)CCCC(F)F)C1)=O)CC2 C=Cn1nncc1C(=O)NC(CO)C(C)NC(c1ncc(OC)cn1)=O C#CCC(CC(F)F)C(=O)N1CC2(CCC(CNC(C3CC34CCC4)=O)O2)C1 N1(C(CC)=O)CC2OCCN(C(c3ccc(C4CC4)cc3)=O)C2C1 CC(C1CC1)=CC(=O)NC1(CNC(=O)CNC=O)CC1 c1(OCC)nc(N2CCC(CNC(c3cc(Cl)n(C)n3)=O)C(C)C2)ncc1Cl c1(N2C(CNC(C=C(C)C)=O)CC3(CCC3)C2)ncc2scc(Br)c2n1 C1(O)(CC(=O)N(C(C)CNC(=O)CN(C2CC2)CC)CCC)CCC1 Cc1[nH]c(NC(C2CSCCN2Cc2ccc(C(C)(C)C)cc2)=O)c(C#N)c1C N1(C(c2sc3cc(C)sc3c2)=O)CCCC2(CC(NC(=O)C(=O)NC3CC3)CO2)C1 N1(C(C)C)CCN(C(C2CC=CCN2C(C2CCN2C(C)(C)C)=O)=O)CC1 c1(C(=O)NCC2C3CN(C(c4coc(C(F)F)c4)=O)CC23)c(O)ccc(Cl)c1F CCC(O)C(C)(C)C(=O)N1CCC(CO)C(NC(=O)Cc2c(F)cccc2F)C1 N1(C(c2cnc(CC)s2)=O)CC2COCC2(C(=O)NCCc2ccccc2)C1 C1(F)(C(=O)NCCCC(CCC)NC(CCCC=C)=O)CCC(F)(F)CC1 C1(CC(=O)NC(Cn2cc(CNC(C(CCC)O)=O)nn2)C)CC2(CCO1)CC2 n1(CC)nc(C(N2CC(CC(C)NC(=O)Cn3nnc(=N)[nH]3)C2)=O)cc1O N1(C(=O)CSC(F)F)CCC2(CC1)CN(C(C1(Cc3cccc(F)c3)COC1)=O)C2 c1(OCC)cc(C(F)(F)F)ccc1-c1nc(Nc2ccc(Cl)cc2OC)cs1 c1(NC(=O)OC(c2ccc(C)cc2)CN(C)C)ccc(F)cc1F CCCC(CNC(=O)C(C)(O)CC)C(=O)NCC1(C)CC2(CC2)C1 c1(C(=O)NC2C(NC(C(C3CC3)OC)=O)CCCC2)ccc(N)cc1Cl c1(OC)c(F)ccc2[nH]c(C(=O)N(CCCNC(C3(C)CCCC3C)=O)C)cc12 C1(NC(=O)Nc2ccc(CN3CCOCC3)s2)CCN(C2CC2)CC1 CC1=CCC(C)(C(=O)NCCC2CCN(C(c3cn4ccnc4s3)=O)C2)CC1 C1(N(C(CCC)=O)C)CCCCN(C(c2ccc(C(F)(F)F)cc2)=O)C1 C#Cc1cc(NC(C2CCCCCCN2C(=O)C(O)CN(C)C)=O)ccc1C c1(NC(C(C)NC(c2ccc(C)o2)=O)=O)ccc(O)c(Cl)c1 C1(CNC(Cc2n(C)ncc2)=O)CCC2(CN(C(c3cc4sccc4[nH]3)=O)C2)O1 N1(C(C(C(CC)O)C)=O)CCC2CN(C(c3ccc(C(C)C)s3)=O)CC2CC1 c1(C(N(C(C)C)CCN(C(=O)Cc2ccc(Cl)cn2)C)=O)cc(Br)cnc1N c1(C(N(C)CCN(C)C(c2ccncn2)=O)=O)cc2ccnc(Cl)c2s1 C(N=c1[nH]c2ncc(Cl)cc2o1)C1C(C)CN(c2ccc([N+](=O)[O-])cc2F)C1 N1(C(c2cncc(OC)c2)=O)C2CCC(C2)C1CC(=O)NCC1C=CCC1 C(=O)(CCC(=O)N1CCC(OC2CCC(NC(c3ccns3)=O)CC2)C1)NCC C(CCCCCC(=O)NCC1C=CCN1C(=O)CC12COC(C)(C1)C2)SC C1(C(N2CCC(OCCNC(C3CC(O)C3)=O)C2)=O)CCc2ccc(F)cc2O1 Cc1nn(CCCl)c(Cl)c1CNc1nc(-c2ccc(Cl)cc2Cl)cs1 c1(C(N2CCC(C)(CNC(=O)Cn3cccc3)C2)=O)ccc2c(=O)ccoc2c1 C1(C(=O)NCC2CC(=C)C2)CCN(C(=O)c2cnncc2O)O1 c1(C(=O)NCC(C)(C)NC(Cc2c(C)nc(Cl)cc2)=O)cc2cccnn2c1 N1(C(C(CC)C(C)O)=O)CC2CCC1C(Nc1cc(C)ncn1)C2 C1(COC)(CNC(=O)C(F)OC(F)(F)F)CCN(C(=O)C(CC)SC)CC1 C1(NC(c2noc(CC)c2C)=O)(CNC(=O)CC(C)(C)C)CCCCC1C c1(C(=O)NC(C)CC(=O)NCCC2CCOC2)nccnc1N c1(C(N2CCC(NC(c3cc(SC)c(C)o3)=O)CC2)=O)cnc2ccccn12 C1(n2ccnn2)C(=O)N1.C1(OCCN(C(C2(C(=O)NC)CC2)=O)C)CC1(F)F C1(C(=O)NCCC(C)(C)N(C)C)CN(C(=O)C(C)(C)n2cncn2)CCO1 C(CCCN=c1ccn2ncc(S(=O)(=O)NCCCCOC(F)(F)F)c2[nH]1)SC N1(Cc2ccccc2)CCNCC12CCOCC2.C(c1ccccc1)=CCCC(=O)N c1(C(N(CC(CC)NC(CC=C=C)=O)C)=O)ccc(-c2nnc(S)o2)cc1 N1(C(c2c(C)ccn2C)=O)CC2CC(C1)CN(C(=O)CCCCCCN=[N+]=[N-])C2 C1(C)(C(=O)NCCn2ncc(CC)c2)CCCN(C(=O)C(C)NC=O)C1 C1(CCC(N2C(COC)CC2)=O)CCC(NC(c2scnc2C)=O)C1 N1(CC)CCOCC1C(=O)NCC(C)=CC(=O)NC1CCC(CCO)CC1 N1(C(C)C)CC(C(=O)NC2CCC2NC(=O)C=Cc2ccc[nH]2)CCC1=O c1(C(=O)NC2CCCC(NC(C(C)OCCOC)=O)C2)c(F)cncc1Br CCCCCC(O)C(=O)N1CCCC1(C)C(=O)NCc1ccc(CO)o1 c1(C(N(C2CCCN(C(C3ON=C(C)C3)=O)C2)CC)=O)cccc2nc(O)oc12 N1(C(C(=O)NC(C)C)=O)CC2CC2(C(=O)NCC(C)(C)C2CCOC2)C1 C(CC(=O)NCCN(C(c1sccc1C(C)=O)=O)C(C)C)(C1=CCCC1)OCC c1(C(=O)NCCC(C)N(C(C(C)NC(C)=O)=O)C)cc2cnccc2o1 N1(C(C(c2cncnc2)C)=O)CC(C)(CNC(c2ccns2)=O)C1 C(=O)(C(O)C(C)(C)C)NCC1N(C(c2cnc(C(C)(C)C)[nH]2)=O)CC1 Cc1ccc(F)c(C(=O)NCC(=C2CN(C(=O)CC3CCCC(F)(F)C3)C2)F)c1 C(=O)(C#CC1(C)COC1)NCC(C(C)C)NC(C1CCC(=O)N(C(C)C)C1)=O C1(CC(C)NC(C2CCCC(=O)N2)=O)CC2CCC(C1)N2C=O.C1CC1C1CC1 c1(C(C)C)c[nH]nc1C(=O)NCC1CCCC1NC(=O)CNC(c1cscn1)=O c1(C(=O)NCC2(NC(C(C=C)OC)=O)CCOC2)ccc(-c2nccs2)cc1 CC(C(CCc1ccccc1)NC(=O)C(F)F)NC(=O)CS(N)(=O)=O N1(C(CNC(C)=O)=O)CCC(F)(C(=O)NCCn2cnnc2C(C)C)CC1 C(=O)(C1=CCN(C(C23CC(F)(C2)C3)=O)C1)NC(C)C(F)F C#Cc1cnc(C(N2CCSCC2C(=O)NC(CO)C2CC2)=O)c(C)c1 C#Cc1ccc(C(=O)NCC2(OCC)CN(C(c3ccc(COC)cc3)=O)C2)o1 c1(C(=O)NC(CC)CNC(=O)C(C(=O)OC)OC)cccc(C#N)n1 C(=O)(CC(Cc1cccs1)NC(c1cc[nH]c1)=O)NC(C(=O)OCCC)C C=CCC(CC(=O)NCCC1CCN(C)C1C)NC(=O)COC C(=O)(C1CCCc2ccnn21)NCC1=CCN(C(C(CSC)C)=O)CC1 CCCC(C(O)C(=O)NCC(F)(F)CC1CC1)NC(=O)C(C)OCC(C)C C(C(C(=O)Nc1ccc(O)c(CO)c1)C(C)(C)C)NC(CCNC(COC)=O)=O C1(C#N)(C(N2CCC(C(C)NC(C(CC)CC)=O)CC2)=O)CC2C=CC1C2 C(=O)(CCC(C)(C)C#N)N1CCN(C(C)CNC2CC3(CCC3)C2)CC1 c1(C(N2CC(CC(C)NC(c3nnc(C)s3)=O)C2)=O)cnc2ccnn2c1 CCC(CC(=O)N1CCC(C)C(NC(=O)Cc2ccnnc2O)C1)CC(F)(F)F C1(C(N(CCN(C(Cn2c(C)ccn2)=O)C)C(C)C)=O)CCCCN1C c1(C(=O)NCC(C)CNC(C2CCN(CC(F)F)CC2)=O)cc2c(s1)CCCC2 C1(C(=O)NCC23CC(CNC(C4CC5CCC4O5)=O)(OC2)C3)CCC2(CCC2)C1 CC1(C(=O)NC(C(=O)NCCc2ncccc2F)C2CC2)CC(F)(F)C1 c1(CCC)nsc(N(C)CCOC2CN(C(c3cnc(C)[nH]3)=O)C2)n1 N1(C(c2cccc(C#C)c2F)C(=O)NCCC)CCc2ccc(C#N)cc21 c1(C(=O)NCCCCCN(C(=O)COCCF)C)cccc(C=C(F)F)c1 N1(C(C2C(C=C)C2)=O)CCC(C2CC2)(CNC(c2cc(Br)nn2C)=O)C1 c1(CCC)n[nH]cc1C(=O)N(C(C)CN(C(=O)C(C)SCC)C)C Cc1ccc(OCC(=O)NCCOCCN(C)C(C2CC(C)C2(C)C)=O)c(F)c1 C=C1CC(C(=O)NCC(c2ccsc2)C)(CNC(c2cc[nH]n2)=O)C1 Brc1cccc(CCn2cc(C3CCOCC3)nn2)c1.N12CCCC(C1)OCC2 C1(NC(c2nc(OCC)oc2)=O)CCCN(C(c2conc2C(C)(C)C)=O)C1C c1(OC(C(=O)NCCCCn2cc(SCC(=O)OC)nn2)C)ccc(F)cc1 C1(C(=O)NCC#C)CCN(C(=O)Cc2cnsc2)CCO1 C(=O)(C(COCC1CC1)N(c1ccccc1)C)N(C1CCCN1C)C C1(NC(C(CO)N(C)C)=O)CN(C(c2nncs2)=O)CC1O N1(C(CC(C(C)C)(F)F)=O)CCCC(C2CCN(C(=O)CC3CCC(=O)C3)C2)C1 c1(C(=O)OC)oc(C(=O)Nc2cn(C)c(C(=O)NC3(CC4CC4)CCC3)n2)cc1C C(=O)(C(CCC=CC(=O)O)N1CCOCC1C)NC(C)(C)C.c1(C(=O)N)ccco1 c1(-c2c(C(=O)NCCC(C)N(C(C=CC)=O)C)c[nH]n2)ccc(F)cc1F C(=O)(N=c1[nH][nH]c2ccccc12)C1(F)CC(N(C)Cc2ccc(C)c(Cl)c2)C1 CC(C)(CCCO)C(=O)NC1CCCC1NC(c1cc2n(n1)CCC2)=O c1(NCC(=O)NCCC(C)NC(=O)CCN(C)C2CC2)ccc([N+](=O)[O-])cc1 N1(C(CSCC#C)=O)CCC2(CCOC2)C(CNC(c2scc(OC)c2C)=O)C1 c1(C(N2C(CNC(C(C)Oc3c(C)cccc3)=O)CCC2)=O)cnc(Cl)cc1Cl c1(N2CCC(N(C(c3ccc(CC)cn3)=O)CC)C2)nc(C#N)c(Cl)s1 c1(CC(=O)NCC(C)NC(=O)CC2CCCC(=O)N2)cc(C2CC2)nn1C C=C(C)CC(C(=O)N1CCCC1CCC)NC(=O)C#CC1CCC1 Cc1nccc(CNC(C2(NC(=O)NC(C)(C)C)CCN(C)C2)=O)n1 CCCC(C)(O)CC(=O)NC(CNC(c1cnc(O)cc1C)=O)CC(C)C C12(CNC(C(CC)COC)=O)CN(C(=O)CC3(NC(C)=O)CC3)C(CO)(C1)C2 C1(CC(c2cn[nH]c2)(C)O)CCCN(C(c2cnc(N3CCCC3)cn2)=O)CC1 c1(C(N(CCN(C(=O)CC2(O)CCCOC2)CC)CC)=O)cc([N+](=O)[O-])c[nH]1 CC1CCCC1(C(=O)NC1(c2ncc[nH]2)CC1)NC(=O)C=Cc1cncs1 C(C(C)(C)CC(=O)N1CCC(C)C(NC(=O)C(C(C)C)c2ccccc2)C1)OC c1(CC)nc(C)c(C(=O)NCCCN(C(c2cncn2C)=O)CC)s1 C1(C(N2CCC(OCCF)C2)=O)(CC)CCN(C(c2[nH]nnc2CC)=O)C1 N1(C(C(N2C(CN(C(c3n[nH]c(C)c3Cl)=O)CC)CCC2)=O)=O)CCCC(C)C1 C(CCCCC(=O)NCC(O)CO)N(C(C(C)c1cncs1)=O)C1CC1 c1(N(CC(C)C)C(=O)NC2C(CC)C2)cc(-n2cccc2)ccc1C C1(C(=O)NCC2C(C)CN(C(C3CCCSC3)=O)CC2)CCC2CCCCN12 C1(NC(C2CC(N(C)CC)C2)=O)CCCCCN(C(=O)CC2CC3C=CC2C3)C1 C1(C(N2CC(N(C(C=Cc3c(C)ccnc3)=O)C)C2)=O)CCC2C(CC1)C2(F)F c1(C(N2CC(CNC(C3CC4CC4C3)=O)OCCC2)=O)cccc2c1CCO2 C1(O)(CNC(=O)CSc2cccc(Cl)c2)CCN(C(=O)CCc2ccc[nH]2)CC1 c1(C(=O)NCC(C2CC2)NC(C2CC3CC3C2)=O)ccc2cccnc2n1 Cc1ccc(-n2cc(C3CCC(NC(=O)CC4COC(=O)N4C)CC3)nn2)cc1 c1(C(=O)NC2C(NC(=O)Cc3ccc(Cl)s3)CC2)ccc(F)c(Cl)c1F C(=O)(C1=CCCC1C)NCC1(COC)CN(C(c2c(C)[nH]nc2C(F)F)=O)C1 C1(NC(C(CC)(C)OC)=O)CCC2(CC1)CN(C(=O)Cc1cnns1)C2 C1(C)(CNC(c2c(OC)nn(C)c2)=O)CCCN(C(c2cc(C(=O)OC)cs2)=O)C1 c1(C(=O)NCC2CC(CN(c3nnc(C)s3)C)C2)nc2ccccc2o1.C(C=O)N c1(CC(N2CCC(O)(CNC(CC3(C=C)CC3)=O)C2)=O)cc(C)ccc1F c1(OC)ccc(C(C)C)cc1CCSCC1(Br)CCC1 C(=O)(C1CCCc2scnc21)N1CCC(C)(NC(C23CC(CC(C)O2)C3)=O)CC1 c1(NC(C2(C(=O)OCC)CC2)=O)cc(C(=O)Nc2cc(Br)cnc2Cl)ccc1Br Cc1c(C(N2CC(NC(c3nn(C)cc3N)=O)C2)=O)nnn1-c1cccc(Br)c1 C=CCC(CC(C)C)C(=O)N1CCC2(CC1)CC2C(N1CC(O)(CN(C)C)C1)=O C12(NC(Cn3c(C)ncc3)=O)CCC(NC(=O)Cc3cn(C)nn3)(CC1)C2 C1(O)(CNC(C(C)N(C(C)=O)C)=O)CCN(C(c2cc(C#N)cs2)=O)C1 C(=O)(C(C)CC(=O)NCCC(C)(C)C(=O)N1CCC(N(C)C)CC1)OC CCCCC(O)C(C)C(=O)NCCC1(O)CCCN(C(c2cncc(C)c2)=O)C1 C(c1cnc(O)nc1O)=CN1CCN(C(CC2CCCN(C(C)=O)C2)=O)C(C)C1 C12(NC(CC(=O)N(CC)CC)=O)CN(C(=O)C(Cl)=CCl)CC1CS(=O)(=O)C2 N1(C(CC2C(C(=O)OC)C2)=O)CC2CCC(C1)N2C(C1CN(C(=O)N(C)C)C1)=O c1(SC2CCN(C(c3ccc(CC)s3)C(=O)NC)C2)ccccc1C C1(C(=O)NC(C2(O)CCN(C(=O)CC3CCOCC3)CC2)C)CC2CCCCC12 C1(F)(CNC(C2C(=C)C2)=O)CCN(C(=O)CCc2ccccc2C)CC1 CN1CCN(C(c2ccc(Cl)c(Cl)c2)=O)C(CNC(c2cc[nH]n2)=O)C1 O=C1CC(C(=O)NCC2CCCN(C(=O)CCCn3ccnn3)C2)NC1=O N1(C(C(C)OCC=C)=O)CCN(C(=O)Cc2cccnc2)CC1CCC C1(O)(C(=O)NC2CC(C)(CNC(C3CC3F)=O)C2)CCCCCC1 c1(C(=O)NC(CNC(C2ON=C(C)C2)=O)C(C)C)cccc2[nH]nc(O)c12 CC1CN(CCN2CCCCC2C2CC2)CCC1CC(=O)O C1(C(N2CC3N(C(C(CC(=O)OC)C)=O)C(CC3)C2)=O)CCc2ccccc2O1 c1(COC)ccccc1CC(=O)NC1CC1NC(=O)C(c1ccc(F)cc1)C c1(C(=O)NC(CNC(CC=CC=C)=O)CCOC)ncccc1C(C)=O C12(C(=O)NCC3CN(C(c4cc(C)ns4)=O)C(C)C3)CC(C)(CCO1)C2 c1(C(N(CCCNC(Cn2c(C)ccn2)=O)CCO)=O)cc(N(C)C)ccn1 C(=O)(C(C(=O)N(C1CCCC1)C1(CNC(=O)CCC(N)=O)CC1)C1CC1)OCC c1(CC)cc(C(N2CC3CCC2CN3C(=O)C=CC2CCOC2)=O)cn(C)c1=O Cc1cc(C(N2CCC(NC(c3c(C)cncc3C)=O)C2)=O)cc(C)n1 c1(CNC(C(C)C2CCC2)=O)ccccc1CNC(c1ccn(C2CCC2)n1)=O C(=O)(C1=CCN(C(C2CC3(CC3)C(=O)N2)=O)C1)NCc1ccn(CC)n1 C12(CNC(C(COC)C)=O)CC(NC(c3ccc(OC)cn3)=O)(C1)C1(CCC1)O2 N1(C(=O)Cc2c[nH]nc2O)CCCC(N(CCF)C(C2COCC2C(F)F)=O)C1 c1(C(=O)NCCCCC(C)NC(C(COC)C)=O)ccc2c(c1)COCCN2 N1(C(C23CC(C)(C2)C3)=O)CCCC(CCNC(c2ccncc2F)=O)C1 c1(CC)cc(C(N2CCOC(CCNC(=O)C=C(C)Cl)C2)=O)ccc1Cl C(=O)(CCCNC(=O)CC1CCSC1)N(C)CC1(O)CCC1 N1(C(COCC(=C)C)=O)CC2CC(N(C)C(c3cnccc3C(C)(C)C)=O)C1C2 N1(C(c2cccc(C(C)C)c2)=O)CCN(C(C2CCC2(C)C)=O)CC1CCO Cc1ccnc(O)c1C(=O)NCC1(O)CCN(C(=O)C(C)Sc2ccccc2)C1 CCCCCC(C(=O)N1CCN(C(C2CCC(=O)O2)=O)C(COC)C1)C(C)C c1(C(=O)NC2CN(C(C34C(=O)CCC3C4)=O)C2)cc(F)c(O)cc1Br Cn1cc(C(N2CCC2CNC(=O)CC(F)F)=O)c(-c2ccnn2C)n1 CCCCCCCC(=O)N1CCCC(CNC(=O)COc2ccsc2)C1 C#CC1CN(C(=O)C(F)C(C)(F)F)CCN1C(c1nonc1N)=O N1(C(C(c2cn(C)nc2)=O)=O)CC(CNC(C2CCC23CCC3)=O)CC1(C)C c1(C(=O)NC2CN(C(C3N(C(C)=O)CCCCC3)=O)C2)cc2n(n1)CC1(CC1)C2 CCCC1CO1.c1(NC(=O)COCCF)nc(=N)[nH][nH]1 C1(CC=C)(NC(c2sc(C)cc2Cl)=O)CCN(C(C2(CC(C)C)CCCC2)=O)C1 N#CC1(CC(N2CC(O)(C(C)Cn3cc(CCN4CCCC4)nn3)C2)=O)CCC1 C1(NC(C(CC)C)=O)CCN(C(c2csnc2C2CC2)=O)CC1CC CC1(C)CN(C(c2csc(-c3ccsc3)n2)=O)CC1NC(C1CCCOC1)=O C(CCCCC(=O)NCC(C)(Cl)CC)NC(C(CSCC)C)=O c1(C(=O)NCC2CC(NC(C3CCC(=O)N3)=O)C2)cccc2sncc12 C1(C(=O)NCC(CC)NC(=O)C(C)OCC2CC2)CCCCC1C(N)=O C(=O)(C(CNC(=O)CC1C=CCCC1)C(C)C)NCCc1cnc(C)s1 N1(C(C(CCC)CCC)=O)CCC2CCCC(C1)N2C(=O)Cc1cc(C)oc1C c1(N(C)Cc2cn(COC)nc2C(F)(F)F)ccc(Cl)c(F)c1.c12cnn(c1)C2 CCC(CC(=O)NC1COCC1NC(c1coc(C(=O)OCC)n1)=O)C(C)C Cc1nn(C2CC2)cc1C(=O)N(C)Cc1cccc(NC(C2CCO2)=O)c1 c1(SC2(CC(=O)N(C)CCn3cc(C4CCN4C)nn3)CC2)cccc(Br)c1 C(=O)(CCCCCC(C)O)NCC1N(C(Cc2c(CC)cccc2)=O)CC1 C(C)(CN=[N+]=[N-])NC(=O)NC(c1coc(Cc2ccccc2)n1)C c1(C(N(CC(CN(C(C2N(C(CCC)=O)CCC2)=O)C)O)C)=O)c[nH]c(=O)cn1 N1(C(CC2CCC(NC(C(CC)SC3CCCCC3)=O)C2)=O)CCC(C(N)=O)CC1 c1(N2CC(CC(C)NC(c3c(C)ccnn3)=O)C2)nc2ccc(Cl)cc2s1 CC1(CNC(c2ncc(Br)cn2)=O)CCN(C(c2cnn[nH]2)=O)C1 C1(NC(C2CN(C(C)C)C(=O)C2)=O)CCC(C)N(C(=O)C(F)=CCCF)C1 N1(C(C(C2CCCC2)NC(c2ccc(C)s2)=O)=O)CC=C(CO)CC1 C(N=c1[nH]c(=NCCCSC(F)(F)F)c2cccc(F)c2[nH]1)C1C(O)COC1 c1(C(CC)OC)ccc(OC(=O)C(C)N(C2CCC2)C)cc1 C#CCCCCCC(=O)N1CCC2CC2(C(=O)Nc2ccc(Cl)cc2NC)CC1 C1(C)(CN(CCN(C)C)Cc2ccccc2)CC2(CCC2)C1 C(C(COC)CC(=O)N1CCCCC(NC(=O)COC2CCC(C)CC2)C1)OC C1(C(=O)NC(C2CCCN2C(=O)CCCc2ccncc2)C)(CC)CCCC1 c1(C(C(=O)NCCCC)N(CCC)Cc2cccc(Cl)c2)ccccc1C(=O)OC N(C(=S)N1CCCC1)c1n(C)c(C2CN(S(=O)(=O)c3cccs3)C2)nn1 CC1(C)CC=C(C(=O)NCCCN(C(c2cnn[nH]2)=O)C2CC2)CC1 c1(CC(=O)NC(C(C)NC(c2cncc(C)c2)=O)C)cccc(C)c1F CC1CCN(C(c2ccncc2N=[N+]=[N-])=O)CCN1C(c1coc(CO)c1)=O C1(NC(CCCC#N)=O)CN(C(c2cnccc2-n2cccn2)=O)CCC1CO C1(NC(C(C(=O)N(C)C)(C)C)=O)CN(C(=O)CCC(N)=O)C2CCCC12 c1(C(=O)NC(C(C)C)CNC(C2CC23CCOCC3)=O)cnc2ccoc2c1 c1(C(N2CC(C)C(NC(=O)CN3CCCC3=O)CC2)=O)cc(F)c(Br)cc1F C1(OC)(CNC(c2sccc2CN(C)C)=O)CCN(C(=O)CC2COC(=O)C2)C1 c1(OC)n[nH]cc1C(=O)NC1CC(NC(C2(F)CCC2)=O)C1 Cc1nc2sc1c(=O)[nH]2.C1(C)(CC(=O)NCCn2cnnn2)CCCO1 CN1N=CC(CC(=O)NCCCC2CCCCN2C(c2ccsc2C#N)=O)C1=O Cc1noc(Cl)c1CCC(=O)NC(CNC(C1COCCO1)=O)C1CC1 C(=O)(CCCCOC)NC1C(NC(CC)=O)COC1 Cc1cc2c(ccc3ccccc23)cc1NC(c1cn2ccc(C)cc2n1)=O N1(C(C(C)Cc2ccncc2)=O)CCCC(CN(S(C)(=O)=O)C)C1 C1(CN(C(c2c(CCC)n[nH]c2)=O)C)C2CN(C(c3noc(CC)c3C)=O)CC12 c1(N(C(=O)NCCN(CCC)CCC)C(C)C)cc(-c2cnn(C)c2)no1 C1(CC)CN(C(c2cc(Cl)n(C)n2)C(=O)NCC(C)C)CC(C)O1 C12(C(N(CCC(C)NC(C(C(=C)Cl)(C)C)=O)C)=O)CCCN1CC(OC)C2 C1(NC(c2c(CCC)nns2)=O)C2CCC1CN(C(C1CC=CCO1)=O)C2 Cc1oc(CNCCN(C)C)cc1C(=O)NC(C)Cc1csnn1 N1(C(CC)CNC(=O)NCc2csc(CNS(C)(=O)=O)n2)CCOCC1 C(=O)(C(C)C(O)C(C)CC)NC1C2CCN(C(Cc3ccc(C#C)cc3)=O)C21 C(=O)(C(C)CC(N)=O)NC1C(C(=O)Nc2cccc(C(C)=O)c2)CC1 Cn1nc(C2CCC2)c(C(F)(F)F)c1C(=O)NCC#CCNC(=O)C1=CCCCO1 C(CCCN=c1[nH]c(Cl)c(C#N)s1)NC(C(C)C1CCOC1)=O O=C(C1Cc2ccccc21)NCC1CC2CC2N1C(=O)CNS(=O)(=O)C1CC1 C1(NC(c2ccc(C)o2)=O)CC(O)CN(C(=O)C=C2CCC(C)(C)CC2)C1 CCC(C(=O)N1CC2CC1C2NC(=O)Cc1cnccc1Cl)C(C)C c1(CN(CC)CC2CCCC2N(C)C)ccc(F)cc1 c1(-c2nc(-c3ccc(C)o3)nn2CCC(C)(C)C)nc2c(Br)cccn2n1 CCCC(C)(O)CC(=O)C(C)=O.N12CCCOC(C1)C2=O.C1CCOCCNN1 N1(C(c2c(C)cnn2C)=O)CCC2(CCCN(C(=O)C(=O)CCCl)C2)C1 N1(C(c2cccc(C(C)=O)c2)=O)CCCC(NC(=O)C2=C(C)CCC2)C1C C1(CC=C)(C(=O)OC)CN(C(C2C(CNC(C3CC(=O)CS3)=O)C2CC)=O)C1 C1(C(N2C(CNC(CN(CC)CC)=O)CC2)=O)CCc2c[nH]nc2C1 C1(CCCC)CN(C(c2n[nH]cc2C)=O)CCN1C(=O)COCC1CCCC1 Cc1c(C(=O)NCC(C)CN(C)C(c2cccc3c2CCC3)=O)ccc(Cl)c1Cl Cc1cc2c(N3CCCC3)ncnc2[nH]1.c1ccccn1 c1(CC)ccc(CN2CCC(O)C2C(=O)Nc2cc(C)c(Cl)cn2)c(F)c1 N1(C(C(=O)NCC2CC2)=O)CC(C(=O)NC2CCn3cnnc3C2)C(C2CC2)C1 c1(OCC)cc(Cl)ccc1NC(=O)NC1CCN(C(=O)C(CC(C)C)N(C)C)CC1 N1(C(C2(CNC(c3ccccn3)=O)CC3(CC3)C2)=O)CCN(CCO)C(=O)C1 C1(C)(OC)CC(NC(c2cc(CNC(=O)CCC3(C)N=N3)cs2)=O)C1(C)C N1(c2nnc(NC(=O)Nc3cncc(OC)c3)s2)CCC2(CCCCC2)C1 c1(C(C)(C)C)ccc(Br)c(OC(C2CC3CCC3C2)=O)c1 c1(CC)oc(C(=O)NCCOCCCNC(C2CCCC2SC)=O)cc1C C1(C(=O)NC(C2CN(C(c3nc(CC)sc3)=O)C2)C)(COC)CCCCC1 C1(C(N(CC(CN(C(C(CC)CN(C)C)=O)C)O)C)=O)CC2(C1)CC(O)C2 n1(CC#C)ccc2cc(NCCCC)ccc12.c12ccc(cc1)[nH]c2=O c1(-c2n(CCC)ncc2)nc2c(s1)CCN(C(c1cc(O)ccc1C)=O)C2 c1(C(=O)NC2CC(NC(C(CC)F)=O)C2)ccc2oc(CC(F)(F)F)nc2c1 C(=O)(C#CC(C)(C)CNC(=O)C(O)C(F)(F)F)N(CC(O)CF)CC Cc1[nH]nc(Br)c1C(c1nnnn1C1(C)CC1)NCc1c(C)coc1C C1(CNC(CCCCOC)=O)CN(C(=O)C(O)CCCc2ccccc2)CCN1C c1(NC(C2N(Cc3ccc(C(=O)O)cn3)C3C(C2)C3)=O)nc(O)c2nc[nH]c2n1 C(=O)(C#CC1(CC)COC1)OCC=C.C12(C)CC(C(=O)N1)c1ccc(cc1)CN2 c1(C(=O)NCC(n2cccn2)C)ccoc1CNC(c1cnn(C2CC2)c1)=O Nc1ccc2c(c1)CCC(n1cc(-c3cc(C(F)(F)F)cnc3F)nn1)C2 CC1(C)CCCC(O)(C(=O)NCC2CN(C(c3ccc[nH]3)=O)CCCO2)C1 N1(C(c2ccn(CC(F)F)n2)C(=O)NCCCSC)CCC(SC(F)(F)F)CC1 N1(C(C(CC)C)=O)CCC2CN(C(c3c(C)ccnc3O)=O)CC2C1 C1(NC(=O)CS)COCC1NC(C12CC(F)(C1)C2)=O.C1(C2(N)CC2)CCCCO1 c1(-n2cc(CCNC(=O)C3=COCC3)nn2)c(F)c(F)c(Br)c(F)c1F N1(C(C2CS(=O)(=O)C2)=O)CCC2CC2(C(=O)NCCC#CCO)CC1 Cc1cc(F)c(CNC(Cc2ccoc2)C(=O)O)c(Br)c1 c1(C(=O)NC(CCOCC)C(=O)NC(C)CS(C)(=O)=O)cc(O)ccc1OC C(=O)(C(F)C(=O)NC(C1CC(NC(=O)C=C(C)C(C)(C)C)C1)C)OCC C1(NC(CC(CC)(F)F)=O)CCCC12CN(C(C1COCCN1C(C)=O)=O)C2 C1(C(N(C2(C(=O)NCCCO)CCC2)CCCN(C)C)=O)CC(O)(SCCO)C1 CCCC(O)C(=O)N1CCC(C2CCCN2C(c2ocnc2CC)=O)C1 N1(C(CN)=O)CC2(CC(N)CO2)C1.O=C(CCCCO)C(c1cc(Cl)c(Cl)s1)=O N1(C(=O)C=Cc2cc[nH]c2)CC(COC)C2(C1)CN(C(C1CCC1)=O)C2 C1(N(C(C)CCO)C(=O)CCc2cccs2)CCC2(CCNCC2)CC1 C1(CC)(CC)CC(C(=O)NC2(CCNC(=O)C(C)n3cccn3)CC2)C1.C(C)(=O)N C(CCC(N)=O)(C(=O)NCCC1CC(C(=O)NCC2CCC(=O)NC2C)C1)SC Cc1cc(=NC(=O)C(Cn2cccn2)NC(c2cscn2)=O)[nH]n1C1CC1 c1(C(N2CC3C(N(C)C(C4CCCCC(=O)N4)=O)C3C2)=O)nc2ncccn2n1 c1(CC)nc(C)cc(=NC2CC(F)(CNC(=O)Cc3[nH]cnc3C)C2)[nH]1 N1(C(c2n[nH]c(CC)c2Cl)=O)CC2(C1)CN(C(c1ccc(CC)c(C)c1)=O)C2 C1(F)(C(=O)NCC2COCC(C)O2)CCN(C(=O)Cc2cncnc2)CC1 C1(CNC(C(CC=C)C)=O)CCN(C(=O)Cn2cnnc2)CC1(F)F C1(NC(C(C)=C2CC2)=O)CC2(C(N3CC(CO)C(CO)C3)=O)COC1C2 C1(CC)CN(C(=O)C(C)(C)CCSC)CCC1NC(=O)CCC1(C)N=N1 N1(C(CN(C(=O)OC)C)=O)CC(CO)CC1C.c12c[nH]cc1C(=O)NC2 N1(C(CC(CC)C)=O)CCCC2(CC(NC(=O)CCc3ccccc3F)C2)C1 C12(NC(CCC)=O)CCOCC1CN(C(=O)Cc1scnc1C)C2 C(c1ccc(F)nc1)=CC(=O)N(C)CC1CCCN(C(c2cc(C)oc2)=O)C1 C(=O)(C#CC1CCCO1)N1CCC(CN(C(=O)CN2CCCSC2)C)C1 N1(C(C2C(OC)C2)=O)CCOCC1CNC(C1(CO)CCOCC1)=O CCCC(C)(O)CC(=O)NCC1CC(NC(C2(P(C)(C)=O)CC2)=O)CCO1 c1(C(=O)NC2(C3N(C(C(C=CC)O)=O)CCCC3)CC2)ncn2c1CCC2 c1(C(=O)NC(C)C(C)(C)NC(C2CC2C(F)(F)F)=O)ccc2c(c1)[nH]c(=N)n2C Cc1cc2c(cc1C)C(C(=O)OCCOc1cccc(Cl)c1)CO2 C(=O)(C(C(CC)=Cc1ccsc1)N1CCCC1CC(C)C)NCCCCCC c1(C(N2CCCC(O)(CNC(c3n(C)ccn3)=O)C2)=O)cccn2cnnc12 C1(CNC(COCC(C)C)=O)CN(C)CCN1C(=O)CN1CCCNS1(=O)=O C(=O)(CC(C(F)F)c1ccccc1)NCC1N(C(CC(=O)OC)=O)CC=C1 C(c1ccc2c(c1)CCO2)=CC(N1CCC(C)C(CNC(=O)CCC#N)C1)=O c1(CC)c(C(N2CCCC(C(C)NC(c3cc(Br)n[nH]3)=O)C2)=O)cnn1CC c1(C(=O)NCCCCNC(C2(c3ccno3)CCC2)=O)ccn(C2CC2)n1 C1(F)(CNC(C2CCC(C)(C)O2)=O)CCCN(C(C2CCCC2)=O)C1 C1(NC(CC2CC(OCC)C2)=O)CCN(C(=O)C(c2ccc(Cl)cc2)C)C12CC2 c1(C(N2CCN(C(C=CCC)=O)CC2CCCC)=O)cc(OCC)c(F)c(F)c1 N1(C(C23CCN(C)C2CCC3)=O)CCN(C(=O)CCc2cccs2)CC12CCC2 C1(CC)CN(C(C2CC(=O)CN2C(C2CC(=O)N(C)C2)=O)=O)CCS1 C12(C(=O)NCC3N(C(CC(COC)COC)=O)CC3)C3C4C1C1C2C3C41C(N)=O N1(C(C2C(CC)N(C(C3C4CCC(F)C34)=O)CC2)=O)CCc2ncn(C)c2C1 N1(C(c2ccc(N)c(F)n2)=O)CCC2CCN(C(=O)CS(=O)(=O)C3CC3)CC2C1 C1(C(N2CCC(C)CC2CNC(=O)CC#N)=O)COc2ccc(Cl)cc2C1 c1(N2CC3N(C)C(CC3)C2)nc(=NCc2cc(Cl)n(C)n2)[nH]c2c1CSC2 CC(CC(=O)NCC(=O)NCCN(C(C)C)C(C)CN(C)C)c1ccccc1 CC1CN(Cc2ccc(-c3ccccn3)nc2)CC1NC(=O)C(C)C1CCC1 Cc1cccc(CNC2CCN(C(C3CN(S(=O)(=O)C(F)F)C3)=O)C2)c1N C1(OC)CCCCC1C(=O)N(C)CC1(NC(c2ccnc(OC)c2)=O)CC1 c1(C(=O)NC2CCCC(N(C(=O)C=Cc3cn[nH]c3)C)C2)cc(P(C)(C)=O)cs1 C(C)(C)(CCC(=O)NC1CC2CC1CC2C(N1CC2CC=CCC2C1)=O)OC C(c1csc2ccccc12)=CC(=O)NCCCCNC(c1nnc(C)s1)=O N1(C(C=CCN(C)C)=O)CC(CCN2CCC=CC(O)C2)CC1(C)C C12(C(=O)NC3CC(C)(NC(c4c(COC)nc(C)nc4)=O)C3)CCCC1CCC2 C1(CC(=O)NC(C=C)COC)CN(C(C2(CO)CCOC2)=O)CC12CC2.C(C)(=O)O c1(C(=O)NC(CNC(C(C)SCCCC)=O)CC(F)(F)F)coc(S(C)(=O)=O)c1 C(=O)(C#CC1CCCOC1)NCC1CCN(C(C(CN(CC)CC)F)=O)C12CC2 C(CNC(c1occc1Cl)=O)(CC(F)(F)F)NC(CCn1c(C)ncc1)=O c1(OC)cc(O)ncc1C(=O)NCC(C(C)C)NC(c1cnn(C)c1)=O C1(C(C)C)CC(C)(NCC(N2CC(C)(NC(=O)C(C)Oc3ccccc3)C2)=O)C1 Cc1nc(Cl)ccc1CC1CN(C(=O)C(C)C)CC12CC2 N1(C(COCCOC)=O)CCC(C)(NC(=O)C(C(C)C)NC(=O)CC(F)(F)F)C1 n1(CC)nc(C)cc1NC(C1C=CC(CC(=O)NC)C1)=O.N12CCOCC1C2 C=CCC(CC)C(=O)NC1CCCCC1NC(C1(F)CCCC1)=O CCC(C)CC(c1nnnn1-c1ccccc1)NCC1CCCCS1 Cc1csc(C(C)N(CCC2CC2)C2CC2)n1.C(C)(C)(C)OC(=O)NCC Cc1cc2ccc(C(N3CCN(C(=O)CC4CCOC4)CC3C)=O)cc2[nH]1 CC1CCc2[nH]c(=NCC3(C)CCCO3)[nH]c(=NCc3cc4c(s3)CCC4)c2C1 C1(=O)C(C)(CC)CN1.c1(C(N(CCC)CCN(C)C)=O)ccc(C)n1C C(CC1=CCOCC1)NC(c1ccn(CCNC(C2CCC(O)C2)=O)c1)=O C1(NC(C(C)N(C(c2ccnn2C)=O)CC)=O)CC(O)C(F)C1 Cc1[nH]nc2c1CC(C(N1CC(CCCCNC(C3CCC3(C)C)=O)C1)=O)CC2 CC(C)(C)CCCCC(=O)NCC1C2CCN(CC(C)(C)C)CC12 C(=O)(C(C#N)C(C)(C)C)N(CC(C)O)CCNC(c1ccc(C(F)(F)F)cn1)=O c1(C(N2CCCC2CNC(=O)C(C)(C)OC)=O)cncc(C(=O)OC)c1 CCCCC(O)C(C)C(=O)NC1CCC(CC(N2CCC(F)(C#N)C2)=O)CC1 C12(CC(N3C(c4cn(CCOCC)nn4)CCC3)=O)CCC(C1)C2(C)C C1CCS(=O)(=O)CC1.C1(C#N)(COC)CCCO1 N1(C(C(C(C)C)c2ccc(F)cc2)=O)CC2(CCN(C(=O)CCCF)C2)C1 C(C(CC(=O)NC12CC(NC(=O)CC3CCCN3C)(C1)C2)C(F)F)N(C)C CC(C)(C)CCC(=O)NC1(C)CCCN(C(=O)C(c2ccc(C#N)cc2)O)C1 C1(C(=O)NCCC(C)N(C)C(c2cccc(F)c2F)=O)CCC(=O)N(C)C1 CC1CCCC=C1C(=O)NCCn1cnc(C(=O)NCC2(C)NC(=O)NC2=O)c1 C1(CCCCCC)CCCN(C(c2cn(C)nn2)C(=O)Nc2ccc(F)cc2)C1 C1(C(=O)NCCOCC(=O)NCC2CCC=CO2)CCCN1C=O Cn1ncc2c(=O)n(CC(=O)NC3CCC3NC(=O)CCC(N)=O)cnc12 Cc1cnc2c(C(=O)NC3CC3CNC(=O)C=Cc3cccn3C)cnn2c1 c1(C(=O)NCC2(F)CC(NC(CC)=O)C2)nccc(C)c1O C1(NC(c2c(C)cc(CC)o2)=O)C2CC3CN(C(=O)Cc4cc[nH]c4)C1C3C2 N1(C(Cc2cc(C(=O)OC)cc(OC)c2)=O)CCC(P(C)(C)=O)C1 C1(F)(C(=O)NC2C(NC(CCCCC#N)=O)CCC2)CCS(=O)(=O)C1 C1(NC(C(C(=O)OC)C)=O)CC=C(C(=O)NCCC2CCN(C)CC2)C1 c1(CNc2cn(C)nc2)cc(S(=O)(=O)N(c2ccccc2)CCN(C)C)c[nH]1 O=C1CCCC2CN(C(=O)C(NC3CCc4ccc(F)cc43)=O)CC2N1 C1(OC)CN(C(=O)CC2(OC(C)C)CCC2)C(C)(CNC(=O)C(F)(F)CO)C1 C1(CC(N)=O)(NC(c2cc(C3CC3)on2)=O)CCN(C(C2CCOCC2)=O)CC1 CCC(C#N)(CC)C(=O)N(C)CCNC(=O)CC1CCCC1(F)F O=C(C(O)CC(F)(F)F)N1CCCCC1C1CCN(C(C2CC(Cl)(Cl)C2)=O)C1 N1(C(C(c2cnccn2)C)=O)CCN(C(C2CC(F)(CO)C2)=O)CC1CO c1(C2(C)C(CNC(=O)NCC3(C)CC(C)C3)C2)cccc(F)c1 C1(C(C)C)(C(N2CC(C)(c3cn(CCCO)nn3)C2)=O)CNC(=O)C1 C(=O)(CC(O)CC(C)C)NCC1(CNC(C=CSC)=O)CC1(F)F c1(C(N(CCCNC(C2(C(=O)OCC)CC2C)=O)C)=O)cc(N(C)C)n(C)n1 Cc1ccc(C(N2CC3CC3(CNC(c3cccnc3Cl)=O)C2)=O)cc1I N1(C(c2c(C)noc2C)=O)CC(C(N2CCOC(C)CC2)=O)CC1(C)C CC1CCN(C(=O)C(C)NC(N)=O)C1C(=O)N(C1(C)CCCC1)C C1(C(=O)NCCC2CCN(C(C(c3cnn(C)c3)C)=O)C2)CC2C(C1)C2(F)F C(C)(C)(CCC(=O)N1CCC(NC(c2ccccc2SCCO)=O)CC1)OC CCC(CC(=O)N1CCCC(N(C(=O)C(C)C(C)C)CC)C1)OC N1(C(C(C)=CCC)=O)CCC(C(=O)NC2CSC2)(C(C)C)C1 c1(C(N2CCC(N(CCC)C(C3C(C)C3C)=O)C2)=O)cccnc1OCC CCCC(C(=O)OC)C(=O)N(C1CN(C(=O)C=Cc2ccc(SC)cc2)C1)C C1(CNC(C2CC2C#N)=O)CC2(CC2)CN1C(C1C(C=C(C)C)C1(C)C)=O c1(C(N2CC(CN(C(c3c(C)nsc3C)=O)C)OCC2)=O)nn(C)c2c1CCC2 C1(C)(CC)C=C(C(=O)N(C2CCCCC2NC(c2cc(C#N)cn2C)=O)C)C1 c1(C(=O)NC2C=CC(C(=O)NCC(C)(C)C#N)C2)ccc(Cl)cc1 C(C)(C(=O)N=c1[nH]nc(Cl)c2ccccc12)SCC1(C(=O)NCC)CCC1 c1(CC(=O)NCC(CC)N(C)C(C23CCC(C2)C3)=O)cccc(F)c1F c1(C(=O)NCC(C)(C)NC(C2CCC2C(N)=O)=O)csc(C(F)(F)F)c1 CC1CC(C)N(C(=O)C=C2CC2)CCN1C(N1CCP(C)(=O)CC1)=O c1(C(=O)NC(CC(=O)OC)(C)c2cccc(OC)c2)ccc2ccccc2c1C N1(CC(=O)OCC)CCN(CC2CCN(C=Cc3ccc(F)cn3)CC2)CC1=O N1(C(CCCC(C)C)=O)CC(CNC(=O)CSC2CCOC2=O)C2(CCC2)C1 C1(C(=O)NCCN(C(C2N(C)CCC2)=O)CC2CC2)CC2CCC(C1)C2O S(=O)(=O)(c1ccc(NC(c2cc(C)no2)(C)C)c(F)c1)N1CCC(OC)C(C)C1 Cn1cc2cc(NC(c3n[nH]cc3-c3ccncc3)=O)ccc2n1 C(=O)(C1=CCC(C)CC1)N1CCC(CC=C)(NC(=O)CC2CCC=CCC2)C1 C1(CNC(C(C(C)C)F)=O)(NC(=O)C(O)CCN2CCOCC2)CCCCC1C c1(C(=O)Nc2ccc(NC(CC(=O)OC)=O)cc2C)csc2c1CCCC2 C12(C(=O)NCCCCC#C)CCC(CC1)N(C(=O)CC1(C)CCOCC1)C2 C1(C)(CC)CC(NC(=O)CCN2CCCCC2)CN1C(c1nnc(O)cc1O)=O C1(CCC)(CNC(=O)NC2CC(CO)C2)CCC1 CN=c1[nH]cc(C(=O)Nc2cc(OCC(N3CC(OC)C3)=O)co2)s1 C1(CNC(CCOC)=O)CN(C(c2ccccc2SC(C)C)=O)CCC1(C)C N1(C(c2c(O)cc(C)nn2)=O)CC2CCN(C(c3cc(O)nc(Cl)c3)=O)C2C1 Cc1cc(Br)c(C(=O)NC(CO)C(C)NC(=O)CC(F)(F)F)s1 CC1(C)CC2(CC2C(=O)NCC2(C)CCN(C(=O)COc3ccc(F)nc3)C2)C1 c1(CC(N2CCC(C)C2CNC(=O)CP(C)(C)=O)=O)c(Cl)cccc1Cl c1(C(N2C(C(N(CC)CC3CCC3)=O)CCC(O)C2)=O)ccnc2cc[nH]c12 N#Cc1ccc(O)c(C(N2CC(F)(CNC(c3cnc4cccnn34)=O)C2)=O)c1 C(=O)(C1Cc2ccc(F)cc21)N1CC(C)C(NC(c2c(O)cc(O)cc2O)=O)C1 c1(C(N(CC(CN(C(=O)C=Cc2nccs2)C)O)C)=O)occc1Br CP(C)(=O)C1COCCN1C(c1nnc2n1CCC2)C(=O)NCCOCC1CC1 C(CCC(=O)NCCC1CCCN1C(=O)CNC(C1CCCO1)=O)=C(C)C C1(OC)CC(C)CN(c2ncnc(NCCN(C)CCF)c2C)C1 C1(C(=O)NCC(C)(C)CNC(C2CCC(C)(C)OC2)=O)OCCOC12CCC2 c1(C(C(=O)N(CC(C)NC(C2CC2)=O)CC)C)c(C)n[nH]c1C.c1(C)cc(Cl)no1 C1(CC(=O)N(CCOCCN(C(C2C(C)C2C)=O)C)C)NC(=O)CNC1=O CCC(CCC(=O)N1CC=CC1(C)C(N1CCC1C(=O)CC)=O)OC C1(C(N(CC(=O)OC)C)=O)CCN(C(=O)CC2CCC(C)(C)C2)C12CC2 Cc1c(C(=O)NC2CCC(CNC(c3coc(O)n3)=O)C2)ccn1C1CC1 CCCC(F)(F)C(=O)NCC1OCCC1C(=O)N(c1ccccc1)C1CC1 C1(CC(=O)NC2CCC(O)C2)CCCCN1C(=O)Cc1ccc(F)cn1 CC(C(C)(C)C(=O)NCCOc1ccsc1)NC(=O)Cc1ccon1 CCC(C(C)CN(C)C)NC(C1C=CCN(C(=O)CC2CC2)C1)=O c1(C(=O)NCC2CC(NC(Cn3c(C)c(Br)nn3)=O)C2)cc(N)ccc1Br C1(C(=O)NC(C)CNC(c2cn[nH]c2)=O)(OC)CCSC1 C1(C(N(c2cccc(C)c2)C)=O)CCN(C(=O)C(n2ccnc2C)C)C(C)C1 N1(C(c2cc(F)c(F)c(F)c2)C(=O)OC)CCOc2cc(Cl)ncc2C1 C1(COC)(CNC(=O)C(C2CCOCC2)C)CCN(c2nnc(C(F)F)s2)CC1 N1(C(C(CN(C(C2(CCC)CC2)=O)C)C)=O)CCN(C(C2C(C)CC2C)=O)CC1 CC(O)(CNC(C1(C)CCN(C(c2ccsc2)=O)C1)=O)CCO Cc1nnsc1C(=O)NC1CC(NC(=O)C(c2ccccc2)n2cccc2)C1 CC(C)(C)CCCC(=O)NCC1CCN(C(c2cncc(Cl)c2)=O)C1 c1(CN(C(=O)CC2CCN2C(=O)CCN2CCOCC2)CC)cc(F)ccc1F C1(CNC(=O)Cc2cnn(C(F)F)c2)CC2(CCC2)CN1C(C1SCCCS1)=O CCCCC(O)CC(=O)NC(CC)CCC(=O)N1CCC(C)(C)CC1 C(C)(C)(CC(=O)N(CC(C)(C)CNC(C1CCCC1(C)N(C)C)=O)C)OC CCCC(CCC)CC(=O)NCC1=CCN(C(C2CCCC23CC3)=O)CC1 C1(NC(C2(NC(CC(CN(C)C)O)=O)CC(F)C2)=O)CCCC1C1CC1 c1(SC)ncc(NC(=O)CC2(C)CCN2C(=O)C(=O)N(C)C)cn1 C#CCC(C)C(=O)N=S1(=O)CCC2(CC1)NC(=O)N(CCOCC)C2=O C=C=C(C)CC(=O)NCC1(C(C)(C)C)CCN(C(=O)CN2CCOCC2)C1 c1(OC)ccc(NC(COC(C)(C)C)C(=O)OC(C)(C)C)cc1Br n1(CC)nc(C)c(C(=O)NC(C)CC2CN(C(c3[nH]c(O)nc3C)=O)C2)c1C C(=O)(C(=O)N=c1cc(C)o[nH]1)NC1CC(CNC(C2(C)CC(=C)C2)=O)C(O)C1 Cc1c(C(=O)NC2CCN(c3nnc(C(F)(F)F)s3)CC2F)cnc2ncnn12 N(S(=O)(=O)N1CCOC(C)(C)C1)OC.C123CC(CO1)(C2)C(=O)N3 C(C1OCCc2ccccc21)NCc1ccc(Cl)c(C)c1Cl Cc1ccc(N(CCC(N2CC(NC(CS(C)(=O)=O)=O)C3C2C3)=O)S(C)(=O)=O)cc1 N1(C(c2cc(C)oc2)=O)CCC2CCCC12C(=O)Nc1ccccc1 c1(C(=O)NC2C(C)N(C(=O)CCc3cccnc3F)CC2)cc(Cl)ccc1F N1(C(C=CC)=O)CCC2(CCCN(C(=O)C=Cc3cccc(Cl)c3)C2)CC1 C12(C(C)C)CCCN1C(=O)COC1CN(C1)C2=O.C1(O)CCCC1.c1(CC)ccoc1 c1(C(N2CC3CC2(c2cccnc2)C3)=O)ccc2sncc2c1 C1(NC(COCCC)=O)CCN(C(=O)CCSc2cccnc2)CCC1CO c1(C(=O)NC(C)(CNC(=O)CCc2cncs2)C2CCC2)ccc(O)c(Cl)n1 Cc1nsc2ncc(C(=O)NCC3CN(C(=O)COCCC(C)C)C3)cc12 c1(C(=O)NCC(C)CNC(C2CCCC(C(F)(F)F)C2)=O)c(F)cc(Cl)cc1F c1(CC)cc(C(=O)NCC(CC)NC(=O)CC2COCCO2)cn(C)c1=O C1(NC(C2(CC#C)CCCO2)=O)CN(C(=O)CCOC(C)=O)CC1CCC C(C)(C(C(=O)NC1CCCOCC1)Nc1ccccc1)NC(=O)OC(C)(C)C N1(C(CN2CCC(n3c(C)cnn3)CC2)=O)C2CCC1(CO)CC2 C1(CNC(CS(C(C)(C)C)(=O)=O)=O)CC2(CCOCC2)CN1C(=O)CC1CC1 C1(CNC(CC(CC)OC)=O)CN(C(=O)C(C)(C)N2CCCCC2)CC12CC2 c1(OCC(N2C(CN(C(CC(=C=C)C)=O)CC)CCCC2)=O)c(C)cccc1C C=CC1(CC(=O)NCC(C)(CO)NC(c2ccc(C(C)C)nc2)=O)CCCCC1 CC1CCCC(C(=O)NC(C(=O)NC(C)Cn2ccnn2)C2CCCC2)C1 C1(C(=O)NC2(C#C)CC2)CCCN1C(=O)C(C)N1CC(C)C1 C(=O)(C(O)(C(C)C)C(F)(F)F)N1CCC(CNC(c2cc(CC)ncc2)=O)CC1 N1(C(C(CC)F)=O)CC(C)OC2(CCN(Cc3c(C)cccc3C)C2)C1 Cn1c(C(=O)NCC2(F)CCN(C(=O)Cc3n[nH]c(=N)s3)C2)cc2sccc12 Cc1cc(Cl)ccc1CNCC1COCCN1C(=O)Cc1c(F)cccc1F Nc1cncc(-c2noc(C3CC3(c3ccc(Br)cc3)F)n2)n1 N1(CCCNC(c2ncn(C(C)C)c2)=O)CCN(C(=O)C(CN(C)C)N(C)C)CC1 O=C(C(CCc1ccc(F)cc1)N1CCC(O)(CC(=O)OC)C1)NCc1cccs1 C1(CNC(c2cc(C)oc2C)=O)CC(C)CCN1C(c1[nH]nnc1C)=O N1(C(C23CC(Nc4ccc(CC)cn4)C2C3)C(=O)NC)CC2CSCC(C2)C1 S(=O)(=O)(C(F)(F)F)NCCC(=O)NCCOC1CN(C(Cc2cn(C)nc2)=O)C1 C(=O)(C(CC(F)F)N(C)C(c1ccc(SC)o1)=O)N(CCO)CC C1(c2nc(-c3cc4c([nH]3)CCCC4)no2)CCNC12CCC2.FC(F)F c1(OC)ccc(C(C)C(=O)NC2(C)CCN(C(c3ccnnc3S)=O)C2)cc1 Cc1nc2c(s1)CCCC2C(=O)NC1C(N(C(=O)CNC=O)C2CCC2)CC1 c1(-n2ccc(CNC(=O)NCC=C(C(=O)OC)C)n2)ccccc1Cl c1(C2CCN(C(c3c(NC)ncnc3)=O)C2)ccc(Cl)cc1Cl CC1=NOC(C)(CNC(=O)CC2CCCC2NC(=O)C(C)(C)CF)C1 N1(C(C=C(C)c2cnn(C)c2)=O)CC(NC(=O)C(O)C(C)C)C(N=[N+]=[N-])C1 N1(C(C2(c3cn(CCCCCO)nn3)CC3(CC3)C2)=O)CCC(O)(CF)CC1 Cc1cccn2cc(C(=O)NCC3(F)CCC(CNC(=O)C(CCO)SC)C3)nc12 C(=O)(C(C(=O)OC(C)(C)C)C(C)C)NC1(CCO)CN(C(C=C(C)C)=O)C1 c1(C(C)C)cc(C(=O)N(C2CCCC3(CC3)C2)C)nn1-c1ccc(F)cc1 N1(C(C(c2cnn(C)c2)C)=O)CCCC(NC(=O)CCC2CCCO2)C1C c1(CCSC)nc(-c2ccn(C(C3CCCO3)C)n2)n(C2CCC2)n1 CCCC(C)CCCC(=O)N1CCC2(CC2NC(=O)CCOCCOC)C1 C1(O)(C2CN(C(CC(OCC)OCC)=O)C2)CCN(C(=O)C=C(Cl)Cl)CC1 N1(C(C(CCCC)C)=O)CCC2CN(C(c3cncc(OC)c3C)=O)CC2C1 C(=O)(CC(CCC)NC(=O)C(C)(C)CCOC)NCC1CCN(C(CCC)=O)C1 C[Si]1(C)CCN(C(C2CC3CC(N)C3C2)=O)CC1 CCCCCCCCCCCCNC(N1CCC(c2nccn2C)C1)=O C1(C(N2CC3(OCC(NC(CCC#CC)=O)C3)C2)=O)Cc2cc(F)ccc2O1 c1(C(=O)NC2C(CNC(c3c(C(=O)OC)con3)=O)C2)ccc2c(c1)nnn2C C(=O)(C(O)C(F)(F)F)N1CCC(OCC(=O)NC(c2cnccn2)(C)C)C1 C(=O)(CC(C)C(F)F)NC(Cn1cc(-c2n(C=C)ncc2)nn1)C C1(c2nc(CC3(CCOC)CC3)nn2C2CCCCCC2)CC2CC1CC2(F)F C(=O)(C1CCCc2scnc21)NCC1(OC)CN(C(C2(Cl)CC2(C)C)=O)C1 Cc1cn2c(n1)C(C)CC(C(=O)NCC(C1CCC1)NC(=O)C=C1CCC1)C2 C(CNC(=O)Cc1sccc1C)(CC(=O)Nc1cc(C)sc1C)OC C(C(C)CN(C(=O)CC1CC12CC2)C)NC(C1(CC(=O)OC)CC1)=O c1(C(=O)NC(CC)CNC(=O)CSc2nnc(S)s2)cc(OC)ccc1Cl N1(C(C2(CC)CCCN2C(=O)COC(F)(F)F)=O)CCC2(CCN(C)C2)C1 N1(C(c2ncc(CC)nc2)=O)CC(NC(c2csc(CC)n2)=O)CCC1C c1(C(=O)NC(CN(C(=O)COC(F)F)CC)C)ccc2c(n1)CCC(C)C2 c1(C(=O)NCC2(C)CCN(C(c3c(C#C)c[nH]n3)=O)CC2)cc2n[nH]cc2cc1C C1(NC(CN(C(=O)CCn2cncn2)CC#C)=O)CCCC1C(C1CC1)OC c1(C(=O)OC)cc(-c2cn(CC(=O)NCCCc3nc(C(C)C)no3)nn2)c[nH]1 N1(C(C(C)C)=O)CCN(C(=O)CC(C)(C)CNC(=O)CC2(C)CC2)C2CC12 CC1CCC(C(C)NCCC2C=NN(C)C2=O)CC1 Cc1nc2ccc(C(=O)NC3CCN(C(=O)CCC#N)CC3C)cc2o1 C(CCCCCNC(c1cc(C(F)(F)F)nn1C)=O)NC(CC1CN(C)C1)=O N1(C(c2ccccc2)=O)CC2(CC3(C(=O)O)C(C)(C)CCC3)CCC1CC2 C1(CNC(C(C)NC(N)=O)=O)CC(C)N(C(=O)CCN2CCCCCC2)C1 Cc1cc(CC(N2CC3(C2)CN(C(c2cnc(C4CC4)nc2C)=O)C3)=O)cc(F)c1 N1(CC#C)CCC(n2cc(CC3C(NC(=O)CC(=O)NC)CCC3)nn2)CC1 CCC(C)C(C)OC.C12(CC1(C)C)C(=O)N2.c12cn(nn1)CCNC2=O C(=O)(CCC(CC)OC)NCCC(=C)CNC(c1cncn1CCC(F)(F)F)=O c1(CC(=O)NCC#CCNC(C(C(C)C)NC(N)=O)=O)ccc2ncsc2c1 Cn1nccc1Cn1cc(C2CCCN2C(c2cn(C(F)F)cn2)=O)nn1 N1(C(c2c(C)cc(O)nc2)=O)CCC(N=c2[nH]nc(C3CC3)s2)C1 N1(C(C(C)(C)C)=O)CCC(NNC(=O)NCc2c(C(C)C)occ2)CC1 C(=O)(C(O)C(O)C(F)(F)F)N(C12CCC(C#N)C1CC2)Cc1ccccc1 N1(C(c2c(NCC=C)cccn2)=O)CCCC(C)(CNC(c2coc(Cl)n2)=O)C1 C(=O)(CC(CC)C(=O)OCC(N1CCN(C(C)C)CC1)=O)NC1(C=C)CCCC1 C(CC(C(=O)NCC(=C)CC)NC(c1ccc(C)s1)=O)=CC C1(CN(C(N2CCC(C(=O)NCCC(OC)OC)C2)=O)C)CC2(CCC2)C1 C(=O)(C(O)C(N)CC1CCCC1)Nc1cnc(C(=O)NC)nc1 c1(C(N(CC=CC(=O)N(CCCC)C)C)=O)nonc1N C1(NC(CC2(CC(=O)OC)CC2)=O)CN(C(c2ccn(CC(F)F)n2)=O)CC1C S(=O)(=O)(c1ccc(C#N)c(NC)c1)N(C(N(C(CCC)=O)C)C)CCOC(F)F C1(CNC(c2ccc(C)cc2)=O)CC(F)(F)CN1C(c1cc(O)cnc1N)=O N1(C(C2CC2[N+](=O)[O-])=O)CC2OCCN(C(c3cc(-c4ccoc4)[nH]n3)=O)C2C1 C1(C)(CC(=O)NCC(COC)OC)CCN(C(C2OCCC2C)=O)C1 C1(NC(C(CC)CC)=O)CCN(C(c2cc(C(F)(F)F)n(C)n2)=O)C12CCC2 c1(C(N2C(CNC(=O)CC(F)(F)F)CCC(C)C2)=O)cc2c(o1)CCCC2 CN1CCN(C(C2OCCC2C(F)(F)F)=O)C(CNC(=O)C(C)(C)C(N)=O)C1 N1(C(C2CCCC(C(F)(F)F)C2)C(=O)NC(C(=O)OC)C)CCC(P(C)(C)=O)C1 C(CN=C(NCC(C)(CO)OC)N1CCC2(CCCN(C)C2)C1)OC c1c(F)cc(F)c(OC)c1[N+](=O)[O-].N12CCC3CN(CC13)CC=CC2=O.CO CCCC(C)N(C(=O)CNC1CC1(F)F)C c1(C(C)N(C2CCS(=O)(=O)C2)C)nnc(Cc2cnn[nH]2)n1C C=CCCC(C)(C)C(=O)N1CCN(C(=O)CN(C)C(C2CCCC2CCC)=O)CC1 C1(N(C)C(c2csc(F)c2)=O)CCCN(C(c2cnc(Br)s2)=O)CC1 C1(C(N2CCC(NC(c3c[nH]c(Br)c3)=O)C2)=O)Cc2ccccc2N1 c1(C(N(C(=O)C=Cc2ncc[nH]2)Cc2n(CC)cnc2)=O)ncncc1C c1(C(N2CCC(NC(C=C(COC)C)=O)C(O)C2)=O)cnc2ncccc2c1 N1(C(C23N(C(CN(C(C)C)C)=O)CC(C2)C3)=O)CCC12CCCOCC2 N1(Cc2snc(C(C)C)n2)CCCC(NC(C2CCCCO2)=O)C1C C12(CNC(c3ccncc3O)=O)CCC1CN(C(c1cccc(Br)c1F)=O)C2 C1(CNC(=O)Cc2cncnc2)CC2(CO1)CN(C(c1cc(F)ccc1Cl)=O)C2 Cc1ccccc1OCC(=O)NC1CCOC1NC(c1ccc(C(C)C)s1)=O N1(C(=O)C(O)Cc2cnc[nH]2)CCCC(C2CCN(C(C3(Cl)CC3(F)F)=O)C2)C1 C1(O)(C(=O)NCC2C(NC(c3c(N(C)C)cccn3)=O)CC2)CCC(C)(C)CC1 C1(C)CN=C(N(C)CC2CNC(=O)O2)NCCO1.c1(NC(C(C)C)=O)ccccc1 c1(C(N2CCC(NC(C3(C)COC3)=O)C(O)C2)=O)ccc2ncc(Br)cc2c1 C(=O)(C(CN=[N+]=[N-])NC(=O)CCc1ncnn1C)Nc1c(C)nn(C)c1 CN1C(=O)C(=O)N(CC(N2CCC(CO)(NC(=O)C=CC3CCCO3)C2)=O)C1=O c1(C(N(C(CCNC(c2c(C)ncn2C)=O)C)C)=O)ccc(C#N)cc1F Cc1cnc(C)c(C(N2CC(NC(=O)C3=CC(C)(C)C3)CCC2C)=O)c1 C1(C(N2CC(CNC(C(C(C)C)n3cncn3)=O)C2)=O)CCc2[nH]nc(O)c2C1 C1(CNC(C2(SC)CC2)=O)CCCN(C(c2c(Cl)c(C)nn2C)=O)CC1 n1(CCC)nc(C(C)COC)nc1-c1ncn(C)c1C C(=O)(C1CCCc2scnc21)NC1C(NC(C(C)Sc2ccccn2)=O)CCC1 C12(CNC(C)=O)CN(C(=O)CC3(CO)CCOCC3)CC1CCO2 N1(C(C(C)CO)=O)CCC(CCCN(C)C(c2cn(C3CC3)cn2)=O)CC1 c1(C(=O)NC23CC(C(N(C)CC4CCOC4)=O)(C2)C3)cc2ccccc2n1C N1(C(CC(CCC)CC)=O)CCC2CCN(C(=O)CN(C)CCO)C2C1 CC(C)C(F)(CNC(=O)CCC1CCC(=O)C1)C(=O)NC1CCN(CCO)CC1 S(=O)(=O)(c1cncc(Br)c1)N1CCC(CNC(C(C)C)=O)C(F)(F)C1 c1(C(=O)NC2C(CO)CCN(C(C3CC(C)C3)=O)C2)cc2c(cn1)NC(=O)CS2 c1(C(N2CCNC(c3cccc(F)c3)C2)=O)cc2cc(I)ccc2s1 c1(CNS(N)(=O)=O)ccc2c(O)nccc2n1.CC1(C)CC2N(C1)C(=O)NC2 n1(CC)ccnc1C(=O)NC(CC1CCC1)C(=O)NC1CCCC1F C(=O)(C1Cc2ccc(Cl)cc21)NCC(C)NC(=O)CCSc1ccccn1 c1(C(C)C)cncc(C(=O)NCC2CC(CNC(C3(N=[N+]=[N-])CC3)=O)CO2)c1 c1(NC(=O)CCc2ccccc2Cl)c[nH]c2cc(-c3ccc(C(=O)O)cc3)cnc12 C(CCCCC(=O)NC1CCN(C(=O)NCC=C(C)C)C1)OCC c1(NC(C#C)=O)cccc(C(=O)NCCCCNC(=O)CCOCC(F)(F)F)c1 N1(C(c2ccc(C)s2)=O)CCC(C)(NC(=O)C(C)Cn2ccnc2)C1 N1(C(CCCC(CC)NC(C2CCCC23CCC3)=O)=O)CCC2(COC(=O)N2)C1 CC(C)CC(C(=O)NCc1ccoc1C(=O)N(C)C(CC(C)C)C)C(C)C C(=O)(CS(=O)(=O)C(C)C)N(C(C)C)CCNC(=O)CS(=O)(=O)NCC1CCCO1 CC1ON=C(C(=O)NC2CCC(NC(c3nc(C(C)(F)F)cs3)=O)CC2)C1C N1(C(c2ncc(C)s2)C(=O)NC2CCCC2)CCOCC(CO)C1 S(=O)(=O)(c1cccnc1NC(c1c(C)cccc1C)C)NCc1c(C)nc(C)s1 C=CCC(CNC(=O)C(F)(F)CO)C(=O)N1CCCC(O)CC1 CCCCC(O)CC(=O)N1CC(CC(=O)NCc2cnc3n2CCC3)CC1(C)C C(=O)(C1=NOC2(CCC2)C1)N1CCCC(C(C)NC(c2nccnc2N)=O)C1 C1(C(C(=O)NCCNC(c2nc(COC)oc2)=O)F)CCC(=O)CC1 N1(C(C(CCCC)O)=O)CCC2(CC1)CN(C(c1snnc1C1CCC1)=O)C2 Cc1cc(C(=O)NCC2CN(C(=O)C(F)=CC3CC3)CC(C)(C)O2)cc(C)c1F C(=O)(C(C#N)C(C)(C)C)N1C2(CN(C(C=C(C)C3CC3)=O)C2)CC1 c1(C(N(CCCNC(C(C(C)C)N(C)C)=O)C(C)C)=O)cc(C(C)C)cc(F)c1 Cc1cccc2sc(NC(N3CC(c4ccccc4C#N)C3)=O)nc12 C12(C=O)C3C4C5C3C1C5C24.N1(C2(C(N3CC(O)C3)=O)CC2)C(=O)CCC1=O c1(C(=O)NC(CC2OCCN(C(c3ccc(C)nn3)=O)C2)=O)cc(Cl)ccc1Cl N1(C(C=CSC)=O)CCCC(C)(NC(C2CCN(c3ccc(Cl)cc3)C2=O)=O)C1 C1(O)(C(C)CN(C)C)CCN(C(=O)C(C(C)O)NC(=O)Cc2ccnn2C)C1 c1(CC)ccnc(CNC(=O)CN(C(=O)Cc2cnns2)CCOC)c1 c1(CCNC(c2cnn(C(C)C(C)C)c2C)=O)cccc(NC(C(C)OC)=O)c1 C1(CC(=O)NC2CC2c2cccc(Br)c2)Cc2ccc(Cl)cc2C1 N1(C(CC(=C)C)=O)CCN(C2CCCC2NC(=O)CC(CC)SC)CC1 N1(C(C2C(C)C2)=O)CCC(C2CCCN2C(C2CCN(C)C2)=O)CC1 Cc1cc(CC(N2CC3C(CNC(=O)CCc4cnc(C)s4)C3C2)=O)cc(C)c1 C1(=O)CC(C)N1.C1(C(=O)OC)CCN1C(=O)COCc1nc[nH]n1 C1(N(C(C2(C(C)C)COC2)=O)CC)CCCN(C(=O)C=CC2CCC2)C1 N1(CC(=O)N(C)CC2CCN(C(C3(CN(C)C)CCC3)=O)C2)C(=O)CNC1=O C(CCC=CC(=O)OCC=CCC)=CCOC(C)(C)C.C1C(C)=CC1 c1(C(=O)NCCCNC(C2CC(=O)N(CC3CC3)C2)=O)cc2ccnc(Cl)c2s1 C12(NC(CC3ON=C(CC)C3)=O)CCC(C(C)NC3CC3CC(C)(C)C)(C1)OC2 N1(C(=O)Cc2ccsc2)CCN(C(C2COCCC2(F)F)=O)CC(O)C1 C1(CNC(C2C(C(=O)OC)C2)=O)CCC2CN(C(c3nccc(Cl)c3F)=O)CC12 Cc1cc(COC(c2c[nH]nc2-c2ccoc2)=O)nn1C N1(C(c2c(CCC)[nH]cc2)=O)CCOCC(CNC(=O)Cn2cc(Cl)cn2)C1 Cc1nc(Cl)ccc1C(N1CCC(Cc2cn(CC3CC3)nn2)C1)=O Cc1[nH]nc2c(C(=O)NCC3(F)CC(NC(c4csc(=N)[nH]4)=O)C3)cccc12 c1(C(=O)NCC2CCCN(C(COC3(C#C)COC3)=O)C2)csc2nnsc12 c1(C(=O)NC(CNC(C=C(CC)C)=O)(C)Cn2cccn2)cc(C)ccc1Cl C1(NC(c2nc(C)nc(O)c2)=O)CCSC12CN(C(=O)CC1CC=CC1)C2 C12(CNC(C3C(CNC(=O)CCOC4CCC4)C3)=O)CCC(CC1O)C2 N1(Cc2cncc(OC)c2)Cc2ccccc2C1C(=O)N1CCCCC1C N1(C(CC=C=C)=O)CC2(CO)CC1(C(=O)Nc1cncc(C3CC3)c1)C2 N1(C(C(c2c(OC)cccc2)=O)=O)CCC2CN(C(c3ccc[n+]([O-])c3)=O)C2C1 Cc1cncc(C)c1C(=O)NCC1CCC1NC(c1c(C)nn(C)c1Br)=O c1(C(=O)NC(COC)C(=O)NC(c2noc(C)n2)C)ncc(C)cc1F C1(CNC(c2c(CC)nco2)=O)CCCN(C(c2c(C)noc2C)=O)CC1 N1(C(C2CC(CCCC)C2)=O)CC(N(C(=O)C(C)SC)C)C(F)C1 N1(C(CCCOCC=C)=O)CC(C)(C)CC1C(=O)N(C1CCC(F)(F)C1)C C1(C(N2CCC(C(C)(C)NC(CC3N(C)CCC3)=O)CC2)=O)CC(=O)NC(=O)N1 C1(C2CCC2)(CNC(=O)Nc2ccc(-c3onc(C)n3)cn2)CCC1 C1(C(=O)NCCc2c(C)ccnc2)CN(C(C2SCCS2)=O)C2(CCC2)C1 Cc1ccccc1CSCC(N1CCC(C)C1CNC(=O)CCC1CC1)=O Cc1cc(C)nc(SCC(=O)NCC2(C)CCN(C(C3CC34CCCC4)=O)C2)n1 c1(C(=O)NC2C(NC(C=C(C)C(C)(C)C)=O)CCC2)cccc(Br)c1 N1(C(CN2CCN(C)CC2)=O)CCCC(CC(=O)N(C2CCCC2(C)O)C)CC1 CC1(C)CC(CCO)CN1C(c1ccnc(CNC(c2cc(Cl)no2)=O)c1)=O C#CCCCCCCC(=O)NC1CC(C(F)C(=O)Nc2cn(COC)nc2C#N)C1 N1(C(CCc2c(C)nccc2)=O)CCC(C(=O)O)c2ccccc21 N1(C(CCOCC#C)=O)CCCC1C(=O)N(C)C(C1CCCCC1)C N1(C(=O)CCSC(F)(F)F)CCOC2(CCN(C(C3CC3C(F)F)=O)CC2)C1 c1(C(N(C(C)C)CCNC(=O)C=CBr)=O)cccc2nsnc12 N1(C(c2c(C)nc(CC)s2)=O)CCCC2(C1)CN(C(c1ccnc(OC)c1)=O)C2 c1(N2CCC(C(=O)NC3C(CCC)C3)(CF)C2)nc(OCC)c(F)c(C)n1 N1(C(c2c(Cl)ccc(C#C)c2)=O)CCC2(CC1)CCN(C(=O)C(C#N)CCC)CC2 O=C(C#CC1CCCC1)NC1CCCN(C(C23CCCC(CO2)C3)=O)CC1 c1(C(=O)NCC(CC)N(C)C(c2cncnc2)=O)ccc2oc(O)nc2n1 CCCC(C)(C)C(=O)NC1CN(C(c2cccc(CS(C)(=O)=O)c2)=O)CC1C Cc1oc(C(=O)NC2C3CC2N(C(=O)CC2OCCCO2)C3)cc1CO C1(NC(c2cncc(C(F)(F)F)c2)=O)CN(C(=O)CC2CC=CCC2)CCC1O c1(CNC(=NCCn2nccn2)NC2CC3CCC2O3)nc(O)c2ccccc2n1 N1(C(c2c(CC)nc[nH]2)=O)CCC(NC(=O)CCc2ccsc2)C(F)(F)CC1 c1(C(N2CC3C(CNC(CC(CC)C4CC4)=O)C3C2)=O)cc(N)cc(N)c1 N1(C(C2(C#N)CC2)=O)CC2CC(NC(c3csc(C4CC4)n3)=O)CC(C2)C1 C(=O)(C(CCCC)NC(C1CSC(=O)N1)=O)NC(C=C)C c1(OC)cc(CN2CCC(O)(C(=O)NCc3cccc(CO)c3)CC2)ccc1C#N C1(CCC(=O)NC2CCN(C(c3cnc(CC(C)C)s3)=O)C2)NC(=O)NC1=O C(=O)(CC(C1CC1)C1CC1)NC1CC(NCC2(C)C(C(=O)OC)C2)C1 C1(CNC(c2nc(C)oc2)=O)CN(C)CCN1C(=O)C(F)Cc1ccccc1 C#Cc1ccc(F)c(C(=O)NC(C2(CNC(=O)C=CCCC)CC2)C)c1 N1(C(C2(CNC(=O)C(CC)C3CCC3)CC(=C)C2)=O)CC2CCCC1C2CO C1(CC(=O)N(CC(CNC(C2CCC(C)(CC)O2)=O)(C)C)C)CN2CCC1CC2 N1(C(C2NC(=O)OC2)=O)CC=C(CNC(C2CC3(CCCO3)C2)=O)CC1 c1(N2C(C(=O)OC)(CNC(C(C=C)(C)O)=O)COC2)nn2cc(C)nc2s1 c1(C(=O)NCC2C(NC(C(C=C=C)C)=O)CCCCC2)cccc2c1NCC2 N(C1CCCc2n[nH]cc21)C(CN(C)C(c1cc(Cl)cn1C)=O)=O c1(C(=O)NCC=CCC(N2CCC(C(C)C)C2)=O)cnc2n1CCC2 C1(CC)CN(C(c2cncc(I)c2)=O)CCC1NC(=O)C1CC1 c1(C(N(CC(O)CNC(c2ccoc2Cl)=O)C)=O)ccc(OCC2CCCO2)cc1 c1(OCC)ncc(C(N2CC3CC3(CNC(=O)C(C)c3cc[nH]n3)C2)=O)cc1Cl c1(CC(=O)NC(c2ccccc2)C2N(C(C3C(C=C)C3)=O)CC2)c(C)cnn1C N1(C(C23N(C(C(CC)n4ccnc4)=O)CC(CO)(C2)C3)=O)C2CCC1CN(C)CC2 CN1CCC=C(CNC(=O)CCC2CCCN(C(C3(C)CCCC3O)=O)C2)C1 n1(CCC)nnnc1CNC(C1CC(C)C1)C1(C)CC1.c1(C2(SC)CC2)ccccc1 c1(OC)ccc2occ(C(N3CCCC3CNC(=O)Cn3cnnc3)=O)c2c1 C(C(=O)NOC1CCOCC1)(C(C)(C)C)NC(c1c(C)non1)=O c1(C(N2C(CN3CCCCC3)CC2)=O)cccc(C=C(F)F)c1.O=C1CC2(CC2)N1 NC1CCCc2[nH]c(C(=O)Nn3ccnc3C(F)(F)F)cc21 c1(C(N2C(CNC(CCSC)=O)C(C)(C)CCC2)=O)c(C)c(C)nn(C)c1=O C12(C(=O)O)CCC(CN3CC(O)C(O)C3CF)(CC1)CC2 C1(NC(C2C(CCC)CCC2)=O)CCCC12CN(C(=O)C(C)CF)C2 C1(NC(C2CCC(C(C)C)CC2)=O)CCCC12CN(C(c1cc(C#N)cs1)=O)C2 n1(C(C(=O)Nc2c(OCC)nccc2)C)cnc2ccccc12 c1(C(N2C(CNC(Cc3scc(C)c3)=O)CC(O)C2)=O)cc2ccccn2c1 C(=O)(C(C)CS(C)(=O)=O)NC1CC2CN(C(C(C)C)=O)C1C2 C1(Cc2ccc(OC)cc2)NC(=O)N(CC2OCCOC2(C)C)C1=O N1(C(c2cccc(OCC)c2)=O)CCC12CN(C(=O)CC1CCC(C)CO1)C2 CCC(C)CCCC(=O)NCC(C)(C1CCC1)NC(=O)Cc1n[nH]c(C)n1 N1(C(C2CN(c3c(OC)c(Cl)ccc3)C(=O)C2)=O)CCC2(CC1)COC2 c1(C(N(C)Cc2ccc(Oc3ccccc3)cc2)=O)c(O)ccc(Cl)c1Cl C1(C(NOCC(N2CC(C)(OCC)C2)=O)=O)C2CC(=O)CC12 N1(c2nnn(C)n2)CCCC(S(=O)(=O)CNC(c2cc(Cl)cnc2O)C2CC2)C1 N1(C(CCN2C(=O)CCC2)=O)CC2(C1)CN(C(C1CC13CC3)=O)CC2CO CC1(CNC(C2CN3CCN2CC3)=O)CN(C(C2OCCO2)=O)CCO1 S(=O)(=O)(c1cccnc1Nc1nccs1)N(C(COC)C)C(C)CC1CCCCC1 C1(CNC(CCCCOC)=O)CN(C(c2cc(C(N)=O)[nH]n2)=O)CCC12CCC2 N1(CC(C)(C)NC(C=NOC)=O)CCN(C(=O)CCc2ccsc2)CC1 C(C1CN(C(=O)CCC(C)(C)OC)CC1C(=O)NCC(C)C(F)(F)F)=CC c1(C(N2CCC(C)(CC(=O)NCc3scc(C)n3)C2)=O)ncc(N)cc1C C1(NC(C2(C)CC3CCC2C3)=O)COC2(C1)CN(C(=O)CCC(N)=O)C2 C1(=O)CCCCCCCCN1.CC(CCCNC(c1ncoc1C1CC1)=O)N(C)C CCC(CCCC(=O)NCc1c[nH]ccc1=O)NC(c1cc(OC)cnn1)=O N1(C(C(COCC)C)=O)CC(C2CC2)(C(N2CCCOCC2C)=O)C1 Cc1nc2cc(CNC(N3CCCC(C)(C#N)C3)=O)cnc2[nH]1 Cc1cccc(CCNC(C2CCN(CCC(=O)OC(C)(C)C)CC2)=O)c1I c1(CCC(=O)N(C2CCN(C(=O)CC3CCCSC3)C2)CC)cc(Cl)cc(Cl)c1 c1(C(=O)NC(COC)CNC(c2cnc(=N)[nH]c2)=O)cc(C)nnc1C c1(C(=O)NC2C(NC(c3cnc(O)o3)=O)CCC2)cccc2ccoc12 c1(-c2ccc(C(C)(C)O)cc2)cc(F)c(NC(c2cc(O)ccc2F)=O)c(F)c1 O=C1CC2(CCC2)C(C(N2CCCC(NC(C3CC4C=CC3CC4)=O)C2)=O)CN1 C1(CCOCC)(NCCCCC(c2cn[nH]c2)C)CCO1 Cc1c(C(N2CC(NC(C3COC(=O)N3)=O)CC(C)C2)=O)[nH]c2ccccc12 c1(OCC)ccc(CC(c2nnc(N(C3CCCO3)CC3CC3)n2C)(C)C)cc1 CN1CCOC(C(=O)NC2(C)CCN(C(=O)C(O)CN3CCCC3)C2)C1=O C1(CCNC(C2C(NC(c3n(CC)ccc3)=O)CCO2)=O)CCOC1(C)C CCC(F)(F)CC(=O)N1CC(C2CN(C(c3coc(C4CCC4)n3)=O)CCO2)C1 C(=O)(C1CCc2nccn21)NCC1N(C(C(C)CSC(F)(F)F)=O)C2C(C1)C2 C1(CNC(C(CC2CC2)NC(C)=O)=O)CCCCCN1C(=O)Cc1cnns1 CCC(CC(=O)NCCC1CCN(C(=O)CSc2n[nH]c(C)n2)C1)C(C)(C)C c1(C(=O)NCC2C(NC(c3cnc(CC)nc3)=O)CCC2)cccc(Cl)c1C CON(CCC(=O)NCC(Cl)C(C)(F)F)C(=O)c1ncn2c1CCC2 C(=O)(C1=NOC(C(C)(C)C)C1)NCC1CC(NC(C(C)CF)=O)C1 C1(CN(CCOCCOCC)CCc2ccc(Br)cc2)CN(CC)CCO1 C12(C(N(CCNC(CCCC#C)=O)CCOCCO)=O)CC3CC1C2C3O c1(-c2n(C(C=C)C)nc(Cn3nccn3)n2)ccc(C)c(CO)c1 N1(C(CC(C)N(C)C)=O)CCCN(C2CC2)CC1.C(CCC=O)NC C12(CNC(CNC(=O)NC)=O)CCCC1N(C(c1ccc(N)cc1Cl)=O)CCC2 CC1OC2CCC1(NC(=O)C1=NOC(CN(C(=O)CCCC3CCCC3)CC)C1)C2 C#CCC(O)C(=O)NC1CCN(C(c2cn(C(C)C)nc2C(C)(C)C)=O)CC1 C(=O)(C(O)CC(F)(F)F)N(C1CCCN(C(C2CC3(CC3)CO2)=O)C1)CC1CC1 C(=O)(CCC(=O)NCCCC1CCCN1C(=O)CCn1c(C)ccc1C)OCC c1(CC(N2C(CNC(C(C(C)C)SC)=O)CC2)=O)cc(C(F)(F)F)ccc1C C1(C(=O)NC(c2ccoc2)COC(C)=O)CN(C(C2CCCN2C)=O)CC1(C)C Cc1nc(F)ccc1CNC1CN(C(c2ccc(F)cc2OC(F)F)=O)CCC1F C(=O)(C1CCc2cccc(O)c21)NC(c1cc[n+]([O-])cc1)C.c12cccc(c1)CO2 C1(C2CN(C(C(=O)OCC=C)C)C2)C(C)(N)C(=O)N1.C1(C#N)(SC)CC1 c1(C(=O)NCCC2CN(C(=O)OCC)C2)csnc1C1CC1 c1(CC(=O)N(CCC)CCNC(=O)CC2(O)CCCC2)coc2cc(Cl)ccc12 N1(C(Cc2n(C)ncc2)=O)CC(NC(c2ncccc2Cl)=O)C2(CCOCC2)C1 C12(NC(C3(F)CCCN(C(C4CC(C#N)C4)=O)C3)=O)CCC(C1)C(O)C2O C(C(CNC(c1cc[nH]c1C1CC1)=O)S(C)(=O)=O)NC(C1N(C(N)=O)CC(O)C1)=O C1(C(=O)NCC2(CC(=O)OC)CC2)CN(C(=O)CC2CSC2)CC1CO C#CCCCCCCC(=O)NC1CCN(C(=O)Cc2ccc(OC)cn2)CC1C N1(C(C=CC)=O)CCCC(N(C(c2ccc(C3CCCOC3)cc2)=O)CC)C1 C#CC(C)(C)C(=O)N1CC(O)(C2CCCN2C(=O)C(C)C2CC2CC)C1 N#CC1(C(=O)NC2CCC(NC(c3ccc(F)s3)=O)CC2)CCSCC1 CCCCC(O)C(=O)NCC1CCCN1C(C1CN(C)CC(C)O1)=O c1(CC(=O)NC2CCCN(C(C(CC)C(C)C)=O)CC2)nn(C)cc1[N+](=O)[O-] c1(C(=O)OC)cnc(NNC(=O)C2CCC23CCOCC3)nc1C CC1CN(C(=O)CC2(OCC(=O)Nc3cnc(S)nc3)CC2)CCS1=O Cc1cc(C(N2C3CCC2CN(C(c2nccs2)=O)C3)=O)c2nccn2c1 C(=O)(C(C)(C)CC(F)(F)F)N(C)CC1N(C(CCC(=C)C)=O)CCOC1 CC1CC(C(=O)OC(C)C(=O)Nc2cc(Cl)cc(Cl)c2)CC(C)C1 C(c1ccccc1C#N)=CC(=O)NC(C(C)C)(C)CNC(=O)Cc1cccnc1 C1(C(N2CCN(Cc3cncc(Cl)c3)CC2)=O)C2CCC(C2)C1N c1(NC(c2ccnn2CCCO)=O)ccc2c(c1)CCC(c1ccc(Br)cc1)O2 Cc1ccc(C(=O)NCC(C)N(C)C(C2CC3CC3C2)=O)c(Br)c1 C(=O)(C(C)(C)CC(=O)N1CCC(CF)(NC(c2ccnc(F)c2F)=O)C1)OC c1(C(N=c2cc(C)n(C)[nH]2)=O)n[nH]c2c1CCN(Cc1cnc(N(C)C)nc1)C2 C1(NC(C(C(=O)OCC)F)=O)CC=C(C(=O)NC2C=C(C)CCC2)C1 C(N=c1[nH]c2cc(F)ccc2o1)C1(CNC(=O)C=CCN2CCC2)CCCC1 N1(C(c2c(CC)cno2)=O)CC(C(=O)NCC(c2ccncc2)C)C(C)(C)C1 N1(CC)CC(NC(=O)CC2CN(C(C3C=CC3C(=O)OC)=O)CC2C)CC1=O C(N=c1cc(C)[nH]c(=NCCc2cc(Cl)cc(Cl)c2N)[nH]1)c1ccc(C)cc1Cl C1(C(=O)NCC(O)CC(=O)N(C(COC)CC)C)(CC)CCCCC1 Cc1ccc(C(N2CCC(CNC(=O)CC3CCC34CCC4)CC2)=O)c(C)n1 N1(C(COCCOCC#C)=O)CCCC1CCCNC(=O)C(C)SC(F)(F)F C1(CNC(C(C)(C)F)=O)CCN(C(c2csc([N+](=O)[O-])c2)=O)CC1C(=O)O C1(C(N(CCCF)CC)=O)CC12CC(NC(=O)CCCn1ccnn1)C2 c1(C(N2CCC(NC(CCc3ccc(C#C)cc3)=O)C2)=O)cc(O)c(F)cc1N C12C=CC(C1)C(=O)N2.C1(C(=O)N(C2(C(N)=O)CC2)C2CC2)CCCC1O c1(CCC(N2CCC(NC(C3CC4CCC3O4)=O)C2)=O)ccnc2ccccc12 CN1CCN(C(C2(C)CCCN(CCCC3CC3)C2)=O)CC1=O c1(CC)ccc(NC(=O)C(C(C)C)NC(c2nccn2C(F)F)=O)cc1 C#Cc1ccc(F)cc1C(N1CCCC(C)(NC(=O)C(C)OCCOCC)C1)=O c1(C(N2CCCN(CCNC(CC3C(CC)C3)=O)CC2)=O)ccc2nnc(S)n2c1 c1(C(=O)NC2CCN(C(C3(C)CCCNC3=O)=O)C2)cc(S(N)(=O)=O)c(Cl)o1 c1(C(=O)NC2(CC=C)CCN(C(=O)CC(C)(C)CC)CC2)nccc2ccsc12 c1(NC(C23C(CN(C(C(CC)(C)O)=O)C2)C3)=O)cc(Br)cc(C#N)c1 C1(C(=O)NC(C(C)O)CO)COCCN(C(c2cc(Br)ncc2Br)=O)C1 c1(OCC(=O)NCCC(C)OCCCF)ccccc1C(=O)N(C)C Cc1csc2c(NC3CN(C(=O)Cn4cc(CO)nn4)CC3C)ncnc12 C12(CC(=O)N(C)CC3(C)C(C)(C)C3(C)C)CCC1CN(C(=O)C=CC(F)(F)F)C2 CCCCCCCC(F)C(=O)N1CCCC1c1ccncc1.C1C(=O)N1 Cc1cnc(C(=O)NCCCN2N(C)CC(C)C2=O)cc1C C1(Nc2c(C(C)C)scc2)CCC2(CC1)CCN2C(=O)OC(C)(C)C C(=O)(C1CCc2c(Cl)cccc21)NCC(CC)NC(=O)C(N)=O Cc1ccnc(C)c1CNC(=O)CC(C)CNC(=O)C(C)O C1(CCc2cn(C(C(=O)OCC)C)nn2)CCN(C(=O)Cc2cn[nH]c2)C(C)C1 C1(C(c2nnnn2C2(C)CC2)NC(c2cncs2)C)CCCSC1 N1(C(c2cc(OC)ncc2)=O)CC2CCN(C(=O)CCOCCN(C)C)CC2C1 C(=O)(C1=CCCCO1)NC1CCC(CCNC(c2c(CC)ocn2)=O)C1 N1(C(C2CCN(C(c3c(C)cccn3)=O)C2C(C)C)=O)CC(C#N)C2(CCC2)C1 C=Cc1cc(C(N2CC3CC2(CNC(=O)CCc2cn[nH]c2)C3)=O)cc(F)c1 C1(NC(=O)C=Cc2ccoc2)CN(C(=O)CCc2cnc[nH]2)CC12COC2 c1(SCCN2CCC(C(C)NC(=O)Cc3ccoc3)C2)ccc(Cl)cc1 c1(NC(C2C(OCC)C2)=O)cc(NCC2CC(c3ccon3)C2)nc(C)n1 N1(C(C(C)OCc2ccccc2)=O)C2CC1CN(C(C1CCCC(C#N)C1)=O)C2 N1(C(C)=O)CC(C2CCCN(CCC3CC3)C2)C1 c1(C(=O)NC2(C(=O)NC(COC)C)CC2)ccc(C)c(C)c1O CC1CCCN(C(c2ccccn2)=O)C1CNC(c1csc(C2CCCO2)n1)=O C(C)(C)(C(F)(F)F)N(CC(CC)(C)Cl)C.C(=O)OCCO Cc1cnccc1C=CC(=O)NC1CC(F)(F)CC1NC(c1cnnc(O)c1)=O N1(C(Cc2c(C)n(C)nc2)=O)CCC2CC(C(=O)NCC(C)(C)CN(C)C)C2C1 CCC(Cc1ccccc1C)C(=O)NC1CC(O)(CNC(C2(CCO)CC2)=O)C1 Cc1nc2cc(C(N3CCC(NC(=O)Cc4nccn4C)C(C)C3)=O)cnc2s1 N1(C(C2C(C)=CCS2)=O)CC(C(F)(F)F)OC(CNC(C2CC(=O)N2)=O)C1 N1(C(c2nc(C)nc(O)c2)=O)CC2CCC1CN2C(c1cc(C2(C)CC2)on1)=O c1(C(=O)NCC#CCNC(C2C(C(=O)OC)CC2)=O)cc2c(s1)CCSC2 C(CNC(C1(CSC)CCCO1)=O)(C(C)(C)C)NC(C(C)OCCC#C)=O C1(c2n(CC=C)nnn2)(Nc2ccc(CC3CCCO3)cc2)CCC(CCC)C1 C1(N(C(=O)C(CC2CCCC2)NC(c2sccc2F)=O)C)CCCC(O)C1 CC1CCCC(N=c2[nH]c(=NCc3cocn3)[nH]c3ccsc23)C1 C(=O)(C(=O)CCC(C)C)NCC(CC(C)C)NC(c1c(Cl)cc(C)s1)=O CC1C2CCC(C2)C1C(N1CC(C)C(C)(C(=O)NC(c2cccnc2O)C)C1)=O c1(N(CC(=O)NCc2cnn(C)c2)C)ccnc(C(C)C)n1 N1(C(CN(CCOC)C)=O)CC(NC(c2cnc(CC(C)C)s2)=O)CC(O)C1 N1(C(CN(C)C)=O)CCC2(CCC(CC(=O)Nc3cc(F)ccc3O)CC2)CC1 C(CCC(CCC)NC(c1nnccc1C)=O)NC(CC(C=C)C)=O c1(C(N2CC(C(=O)Nc3cccc(C#C)c3)C2)=O)ccc2c(n1)OCCO2 N1(C(C(Cn2cncn2)NC(=O)C=CC2CCCCC2)=O)CCC2CCCC2CC1 C1(CNC(c2cc(OC)n[nH]2)=O)CC(C)(C)CN1C(=O)CC1CCN(C)CC1 C1(NC(C2(C3CC3)CC2)=O)(CF)CCN(C(C2(n3cnnn3)CC2)=O)C1 C(=O)(C1=COCC1)NC(CC(C)NC(=O)C(C1CCCCC1)C)C N1(C(c2scc(Cl)c2Cl)C(=O)NC(C)C)CCC2(CC1)OCC(C)(C)CO2 C(CC(C)C(=O)NCC(C)(C)OCCNC(=O)C(C(C)C)n1cnc(C)c1)=CC C(=O)(CCCC(=O)NC)NC1(C(=O)Nc2cn(CC=C)nc2)CCCC1 C1(NC(C(CCC=C)(F)F)=O)CCC2(CCCN(C(C3(CN(C)C)CC3)=O)C2)C1 c1(CNC(c2cnc(C)[nH]2)=O)cccnc1CNC(C1NC(=O)CC1C)=O C1(C(=O)NC(C)CN(C)C(c2ccccc2N(C)C)=O)CCC2CC2CC1 c1(C(=O)OC)nsc(N2CCC(CCNC3CCN(CS(C)(=O)=O)C3)C2)n1 Cc1c(C2CC2C(=O)NC2CCC(CNC(c3cc(Cl)no3)=O)C2)cnn1C C(=O)(C(C(C)C)n1cnnn1)N(CCC)CCNC(=O)C=CCCC=C(C)C C1(N(C(c2ccc(C#C)o2)=O)C)CN(C(c2cc(Cl)nnc2O)=O)CC12CC2 C1(C)(CNC(C2N(CC)CCC2)=O)CCN(C(c2cc[nH]c2CC)=O)CC1 CC1CN(C(=O)COCC(F)F)CCC1NC(=O)CC1(N2CCCC2)COC1 C1(CC(=O)N(C(C)CNC(C2(Cc3ccccc3)CC2)=O)C)NC(=O)NC1=O Cc1cc(F)c(C(N2CCC(CC(C)NC(=O)CN(C)C)CC2)=O)c(Cl)c1 N1(C(CC2(C=C)CC2)=O)CCN(C(c2cocn2)=O)CC(CO)C1 Cc1cc(Cl)ccc1CC(N1CC(NC(=O)COCc2ccnn2C)C(C)C1)=O Cc1cccc(CC2C(=O)NCC(C)N(C)N2C2CCCC2)c1.n1(C)cncn1 N1(c2n(CC=C)c(COC(C)C)nn2)CCC2NC(=O)CCC2C1 C12CCN(CC1)C(=O)C=CCN2.C1(Cl)(C(N(C)CC)=O)CC1(F)F.C(C(F)(F)F)N N1(C(c2c(COC)cccn2)=O)CCCC12CN(C(=O)CCc1cccnc1)C2 N1(C(Cc2cn(C(C)C)nc2)=O)CCC2CN(C(C3CCN(C)C3=O)=O)CC2C1 c1(NC(=O)NCC(F)(F)Br)cc([N+](=O)[O-])cc2c1OCOC2 c1(CNC(CC(C)C(C)(C)C)=O)nn(C)c2c1CN(C(=O)C1=CCOC1)CC2 N1(C(=O)Nc2n(C(C)(C)C)nc(C3CC3)c2)CCC2C(F)(F)C2(F)C1 C1(C(=O)NC(C)C(C)NC(c2cc[nH]n2)=O)CN(S(=O)(=O)N(C)C)C1 C1(CC(=O)NC2C(NC(C3(N(C)C)CCCCC3)=O)CC2)OC(C)(C)OC1=O C(=O)(C(F)C(C)(C)O)NCCN(C(C1CCCSC1)=O)CC N1(C(C(C(=O)OC)C)=O)CC2CCN(C(c3ccc(N(C)C)cn3)=O)CCC2C1 C(C(C)(C)CC(=O)NCC1COC(CNC(=O)CNC(=O)C2CC2)C1)OC c1(C(N2CCCC(CNC(C3C(C#N)C3)=O)C2)=O)csc([N+](=O)[O-])c1 c1(N(CC)CC)ccc(C(=O)NC(CNC(=O)C(O)C2CC2)C(C)(C)C)cn1 c1(C(=O)NCC2OCCN(C(C(Cn3ccc(C)n3)C)=O)C2)c[nH]cc(C)c1=O N1(C(c2ccc3c(c2)CC(C(=O)O)C3)=O)CCOc2ccc(Cl)cc21 N1(C(c2ccc(SC3CC3)cc2C(F)(F)F)=O)CC2(CF)CCC2(CO)C1 CC1(C)CN(C(c2ccc(O)c(CO)c2)=O)CC1NC(C1CC2CCC12)=O Cc1cc(C)c(C(=O)NC(c2ccccc2)CNC(C2CCCO2)=O)[nH]1 Cc1ccc(C(N2CCC2(C)CC(=O)NOCC2CC3CCC3C2)=O)nc1C C1(NC(CCCNS(CCC)(=O)=O)=O)COCCN(C(=O)C(C)(C)SC)C1 N1(C(C(C)OC(C)(C)C)=O)CCC(CO)(NC(C2CCCCC2)=O)CC1 C1(CNC(C(CC=C)(C)N(C)C)=O)CC2COCC2N1C(C12CCCC1C2)=O Cn1cnnc1CCC(=O)NCC(C1(NC)CCCC1)(C)NC(=O)CCCC(F)F C1(NC(C(C2CCCC2)NC(=O)CCCC2CCC2)=O)CC2(C1)CC21CCC1 c1(C(N(CC)CC)C)cccc2cnccc12.C12CCCN(C1)C(=O)C(=O)N2 c1(C(=O)NC2C(CNC(c3cc(C(=O)OC)no3)=O)CCC2)cc2c(s1)CCC2 N1(C(C2(C(=O)OCC)CC2)=O)CC(NC(c2ccn(C)c2)=O)CC2(CCC2)C1 C=CCCCC(=O)NC(CCSC)C(=O)NCC(c1ccc(OC)cc1)O Cn1nc(C(=O)NCCc2ccc(C(=O)NCCCN(C)C)cc2)cc1O c1(OCC(N2CC(SC)C(NC(c3nccn3C)=O)C2)=O)ccc(C#N)cc1 c1(-c2nc(-c3c(OC(C)=O)ccc(OC)c3)on2)cc(C)cc2c(=O)c(C)c[nH]c12 c1(NC(Cc2cccc(C)n2)C)ccc(S(=O)(=O)NC(c2ccoc2)C)cc1F Cc1cc(C(=O)NCC2CCN(C(=O)C(F)C3CCOC3)CC2)cnc1C(F)F C1(S(C)(=O)=O)(C(=O)NC(CN(C(c2n(C(CC)CC)nc(C)c2)=O)C)C)CCC1 Cc1oc(CO)cc1C(=O)N(C(C)CNC(=O)Cc1ccnn1C)C C(C(C)(C)C(=O)N(C1CCCCCC1)C1CC2CC2C1)N(C)C(C1CCCC1)=O c1(OC)cc(C2CCN(CCc3cnn(C)c3C)C2)cnc1F c1(C(=O)NC2CN(C(c3c(C)nc(C)s3)=O)C(C)C2)cc(N)cc(O)c1C Nc1c(C(N2CCCC(O)(CNC(=O)C(F)(F)CO)C2)=O)cccc1[N+](=O)[O-] C(=O)(C(C)(C)S(C)(=O)=O)NC1C(O)CCN(C(c2cccc(CCC)c2)=O)C1 C12(CC13CCC3)CNC(=O)c1ccc(s1)C2.C1(CCCC)(CNC=O)CCC1 c1(C(N2CC3CCN(C(C=C(CCC)C)=O)CC3C2)=O)ccc([N+](=O)[O-])c(C#N)c1 Cc1cc(C(=O)NC2CCCC2CNC(=O)CCc2ccco2)c(C)n1C c1(C(=O)NCCN(C)C(C2CCCS2)=O)cc(Cl)c2ccccc2n1 C(=O)(C#CC1CCCOC1)N1CCCN(C(C(C=C)(C)C)=O)CC1C Cc1cncc(CC(N2CCC(C)(NC(=O)COCc3ccccc3C)C2)=O)c1 C1(C(=O)NC(C)(C)CCNC(=O)CC2CC3CC3C2)CCC(F)(F)C1 C(c1cccc(CO)c1)=CC(=O)N(C1C2CN(C(C=C(C)C(C)(C)C)=O)CC21)C C(=O)(CC(O)CCC(C)CC)NCCCCCN1CCN(C(CCOC)=O)CC1 Cc1nn2cc(C(N3Cc4cnc(C(C)(C)C)nc4C3)C(=O)N)nc2s1.N(C)C CC(CC(=O)N1CC(CC(C)NC(=O)C(C)CN(C)C)C1)CC(C)(C)C c1(C(N2CC(NC(=O)CSCC(F)(F)F)C(F)C2)=O)ccc2cccnc2c1 CC(C)C(O)CC(=O)NCc1cn(-c2ccc(Oc3ccccc3)cc2)nn1 c1(C(CC)C(=O)N(CCOC)CC2(F)CN(S(=O)(=O)CC)C2)ccc(OC)cc1 C1(NC(C2CS(=O)(=O)C2)=O)C2CCN(C(c3ccnnc3)=O)CC12 CC1COC2(C1)CN(C(N1CC3(F)C(OC(C)(C)C)(CCC3)C1)=O)C2 n1(CC)cc(C(N2CC(O)(CN(C)C(C3(C(F)(F)F)CCC3)=O)C2)=O)cn1 C12(C(N(CCNC(C(C)C3CCCO3)=O)CC3CC3)=O)C3C4C1C1C2C3C41C C(C)(C)(CC(=O)NC1C=CCCCC1)N(C(C1(CC#C)CCCO1)=O)C C1(OC)CC(C(=O)NC(c2nnc(C(C)(F)F)s2)C)N(CN)C1 N1(C(c2c(SC(C)(C)C)nco2)=O)CC(c2ccccc2)C(N)C1 c1(C(=O)NCCOC2CCN(C(C3CCOC3)=O)C2)cc(C(F)(F)F)ccc1O C1(N(C(C=CC(C)C)=O)CCO)CCCN(C(=O)Cn2cncn2)C1 c1(C(=O)NCC2=CCN(C(C(C)C(C)(F)F)=O)CC2)cc(Cl)c2n[nH]cc2c1 C(C1CCCCC1)=CC(N1C(CN(C(CC2C(C)CCC2)=O)C2CC2)CCC1)=O C1(CC(N)=O)(NC(c2scnc2Cl)=O)CCN(C(C2CC2[N+](=O)[O-])=O)CC1 C(=O)(CCCC(=O)N)NCC1CCCC(NC(COCC)=O)C1.C1(=O)CN1.C(C)(=O)NC C(c1ccccc1)=C(C(=O)NCC(CCOC)NC(C1C(COC)C1)=O)C N1(C(C2CC3C=CC2O3)=O)CCC2CCN(C(c3cc4n(n3)CCCN4)=O)C2C1 c1(CN(C(=O)CC2CN(C(c3ccc(C(C)(C)C)[nH]3)=O)C2)CC)cc(C)[nH]n1 N1(C(C=CCC)=O)CCN(C(=O)CCC[N+](=O)[O-])C(CCO)C1 C(C(COC)CC(=O)NC(C1CCCCN1C(c1cscc1F)=O)C)OC CCC(C)C(C(=O)N1CC(NC(c2cnccc2C)=O)C1)OC.C(C)(=O)O C1(CN(C(C(C)NC(CC)=O)=O)C)CCCCN1C(=O)CC(C)(C)O Cn1nc(CCC(=O)NS(=O)(=O)CCC2CC3CCC2C3)c2ccccc12 N1(C(c2c(COC)ncs2)=O)CC(CNC(=O)CCC2CC2(F)F)CC1(C)C CC1(C)OCCOC1CC(=O)NC1(CF)CN(C(c2ccon2)=O)C1 Cc1nc(N2CCC(CC(C)(C)C)CC2)nc(N(C)C)c1Br C1(CNC(C=CCOC)=O)CC2CCC1N2C(C1CN(CC(C)C)C1)=O C1(NC(c2cc(C(F)(F)F)n[nH]2)=O)CCCN(C(c2ccc(F)o2)=O)C1 c1(C(=O)NC2CN(C(=O)NCCOc3ccon3)C2)ccc(OCC(F)F)nc1 c1(CS(=O)(=O)NCC2CCC(NC(CCOC)=O)CC2)ccc2ccsc2c1 Cc1ccc2c(CC(N3CCC(N(C(=O)CC4(F)CC4)C)C3)=O)coc2c1 C(=O)(C(O)CC(C)(C)C)NCCC(C)NC(c1cc(N)cc(O)c1)=O c1(C(N2CCCC(NC(=O)Cn3ncccc3=O)C2)=O)ccnc(Cl)c1O C1(CNC(c2cc(OC)ns2)=O)CCCCCN1C(=O)CC1(C)CC1 Cc1nc2ccccc2c(C)c1C(=O)N(CC(O)CN(C(=O)C(C)(C)N(C)C)C)C N1(C(COc2cccc(C)c2F)=O)C(C)CN(C(=O)CC(C)N(C)C)CC1C c1(CC)cccc(Br)c1C(=O)OC(C)(C)C.C12(CC1)CNC(=O)N2 C1(NC(C2C3CN(Cc4ccc(OCC)nc4)C2C3)=O)COc2ccccc2O1 C1(C(=O)NCCCC2(NC(CCCCOCC)=O)CC2)CCC2(CCC2)O1 n1(C(CC)C)ncc(NC(=O)NC(C(=O)O)c2nccs2)c1C c1(C(N2C3C(NC(C4=CCCC4C)=O)C(C3)C2)=O)cncc2c1CCCC2 C1(N(C(c2cn(CCCC)nn2)=O)C)CN(C(C2(C(N)=O)CCC2)=O)CC1O c1(C(=O)NC2C(CC(=O)NC3CCC(COC)CC3)CC2)cc(F)ccc1F c1(C(N(CCN(C(=O)COc2ccc(F)c(F)c2)C)C)=O)ccc2ccoc2c1 N1(C(C(N(C)C)C2CC2)=O)CC(CNC(c2cc(CO)on2)=O)C2(CC2)C1 C(=O)(C1=C(C)OCC1)NC(C(=O)N(C1CCOCC1)CC#C)CC1CC1 N1(S(c2ncc(C)o2)(=O)=O)CC2(CCC2)c2ccccc21.C12CCC(CC1)CC2=O C12(NC(C=C(C)C(C)C)=O)CCCCCC1N(C(=O)CN1CCOCC1)CC2 C1(CCNC(C(C)NC(N)=O)=O)CN(C(c2csc(C#N)c2)=O)CCO1 C(CCC(=O)NC(C)CNC(c1ccn(C(F)F)n1)=O)=CCC=C C(CC(=O)N1CCCC(N(C)C)C1)(C(C)(C)C)NC(C(COC)OC)=O c1(C(=O)NCC2N(C(COC)=O)CC2)ccc(CNc2cnc(Cl)cn2)nc1 C(=O)(C1=CCOCC1)NCc1nccc(C(=O)NCC2C(C)CCC2)c1 c1(C(=O)NC(C(C)C)C(=O)NC(C(N)=O)C2CC2)ncn2c1CCC2 N1(C(c2c(C)nsc2)=O)CCC(NC(=O)CCSCC(C)C)C(CO)C1 C=CC1CCN(C(=O)CC(Cc2cccs2)NC(C2CCCCCC2)=O)C1 N1(C(CCN(c2ccccc2)C)=O)CC2CC1C2C(=O)NCc1ccnnc1S Cc1cc(C)[nH]c(=NCC2CCN(C(c3c[nH]nc3C(C)C)=O)CC2C)n1 c1(CC(N2C(CC=C)CC(F)C2)=O)cc(CO)c([N+](=O)[O-])c(F)c1 c1(NC(C2(NC(C(CC)C#N)=O)CCN(C)C2)=O)ccc2ncccc2c1 N1(C(c2ccc(CC)o2)=O)CC2CN(C(=O)CCc3ncc[nH]3)CC2(C)C1 N1(C(CCCCN(C(C2(C)C(C)OCC2)=O)C)=O)CCC(C)(CO)CC1 C(=O)(C#CC(C)(C)CNC(c1csc(O)n1)=O)NCc1c(C)cccc1C c1(C(=O)OC)cc(Cl)c(Cl)[nH]c1=NC1CS(=O)(=O)CC1NC(=O)CSC1CC1 N1(C(c2cc(C)ncc2)=O)CCCCC(NC(=O)C(C(C)(C)C)N2CCCC2)C1 c1(C(N2CCC(NC(c3cccc(Cl)n3)=O)C2)C)cnc2[nH]ccc2c1 C1(NC(C(c2ccn(C)n2)(C)C)=O)CC(NC(c2cc(C(F)F)cs2)=O)C(O)C1 Cc1ccncc1C=CC(N1CC(C(F)(F)F)C1)=O.C1(=O)C(F)=CCN1 C1(N(CCC)C(c2cc(Cl)ns2)=O)CCN(C(=O)C(c2cnn(C)c2)OC)CC1 c1(C(=O)N)ccc(CCC2(C(=O)OC(C)(C)C)CC2)cc1.C=CC(O)C(=O)N(C)C N1(CC)CCOCC1C(=O)N(C)CC1(NC(=O)Cn2ccnn2)CC1 C1(C(N2CCN(C(COCC(=O)OC)=O)C(C)CC2)=O)Cc2cc(Cl)ccc2O1 N1(Cc2ccc(OC(C)C)nc2)CCC(NC(c2ocnc2C(F)F)=O)C(C)C1 C1(NC(CC(CN(C)C)C(F)F)=O)CC1C1CCN(C(C2(F)CCC2)=O)CC1 C12(NC(c3cc(N(C)C)ncc3)=O)CN(C(C3(O)CCC3)=O)CC1CS(=O)(=O)C2 CC1=NOC2(C1)CC(C(=O)NC1CCOCC1NC(C1(c3cccs3)CC1)=O)C2 C#CCCC(O)C(=O)NCC.C1CCOCCO1.C(=O)CSC(C)(C)C C(=O)(C1=NN(C)C(=O)CC1)N1CC(NC(c2cc(C)sc2C)=O)C2(C1)CC2 C1(C(=O)NCCC2C(C)CN(C(C3(C#N)CC4CC4C3)=O)C2)CC2(CCO1)CC2 c1(C(=O)NC(CNC(C(C(C)O)N(C)C)=O)C(C)(C)C)cccc2c1ccn2C C1(CC)CC(CNC(C2CCCN2C)=O)N(C(=O)CN(C)S(N)(=O)=O)C1 c1(C(=O)NCC(C)N(C)C(c2ccc(C(F)(F)F)o2)=O)cnc(C(F)(F)F)c(F)c1 CC(C)(C)C(C#N)C(=O)N1CC(c2ocnc2CNC(C2(C)CCCCO2)=O)C1 CC1OCCCC1C(=O)N(CC(O)CN(C)C(c1ccnc(F)c1)=O)C C1(CNC(CN(C(C)C)C)=O)CC2CCC(C1)N2C(C1CC2(C1)CC21CC1)=O c1(C(=O)NCC2CC(O)(CNC(C(CC)(C)O)=O)C2)cc(OC)c(O)c(Cl)c1 c1(OC)cccc2c(=O)c(C)c(NCC(=O)Nc3ccsc3Cl)[nH]c12 C(=O)(C1=C(Cl)CCC1)N1CC(CCCNC(C(C)OC2CCCC2)=O)OCC1 CC1CN(C(=O)C(CC(F)F)NC(C2CCSCC2)=O)CC(=O)N1 N1(C(C(C)(C)n2cccn2)=O)CCC(c2nc[nH]n2)CC1.C1(=O)C=CS1 C1(C(=O)NCC(CCOC)NC(=O)Cc2cc[nH]n2)CCCC(=O)N1 C(=O)(CCCS(N)(=O)=O)NCCCCNC(CC1CN(C(C)=O)C1)=O C(=O)(CCCC(C)(C)CC)N(C)CC1N(c2nnc(C)s2)CC(F)C1 c1(CC)cnc(O)c(C(N2CC(N(C(=O)CC3CCCC3O)C)C(O)C2)=O)c1 C1(C(=O)NCn2ccc(C3CC3)n2)(NC(C2CCN(CC)C2)=O)CCC(C)(C)C1 N(C)(C(=NCCSc1ccccc1)NCC1CCCS1)C(n1cc(CCC)cn1)C.C C(=O)(C(CN(C(=O)C(C)SC)C1CC1)C(C)C)N1CCC(OC)CC1 C(C(O)(C(F)(F)F)c1ccccc1)NC(Cc1nc(C)c(-c2ccc(Cl)cc2)o1)=O N1(C(C2CSCN2C(=O)CCCF)=O)CCn2ccnc2C1 C#CCC(CN=c1[nH]c(=NCC2CCOCC2(C)C)[nH]c2cccc(F)c12)OC C1(CNC(=O)COC2CCCOC2)(NC(C(=O)NCCOC)=O)CC1(F)F N1(C(CC(CC)C)=O)CCC(NC(=O)CCCNC(N)=O)C1(C)C C(=O)(C(O)CC[S+](C)C)NCC1(C(C)NC(C2(OCC)CCC2)=O)CCCC1 CC1(CNC(c2cc(F)cs2)=O)CCN(C(c2sccc2C(F)F)=O)CC1 CC1CCCc2cc(C(=O)N(CCCCNC(C3CCCCCCC3)=O)C)nn21 C(=O)(C1CCc2nccn21)N1CCC(C(N(C(C)C2CC2)C)=O)CC1 c1(OCCC)ccc(C(=O)NCc2n[nH]cc2COC(=O)C(C)C(C)O)cc1 CC1CCC(C(N2CC(O)(CN(C(=O)Cc3nncn3C)C)C2)=O)O1 CN1CCC(NC(=O)CN2CCC(=O)CC2)C12CCCN(C(C1CSC1)=O)C2 CN1CC(CNC(c2ccc(CNC(=O)CNC=O)nc2)=O)CC1=O C(C)(CCC(=O)NCCN1CCC(NC(=O)CC2COC3CC2C3)CC1)SC C1(C)(CNC(CC(COC)C)=O)CC(F)(F)CN1C(c1cc(C)c(O)c(N)c1)=O N#CC1(c2ccccn2)CC(C(=O)NC2(CNC3CCCO3)CC2)C1 C1(C(=O)NC23CCC(CC2n2cc(C4CC4)nn2)C3)CCc2nc[nH]c2C1 CC1CCN(C(=O)Cc2cn[nH]c2)CC1CNC(C1C2CCC1CC2)=O N1(CC(=O)Nc2ccoc2)Cc2ccnn2CC(C(N2CCC(O)CC2)=O)C1 c1(OC)cc(Cl)ccc1C(=O)N(C)CC1(CNC(=O)CCN2CCC(F)C2)CC1 Cc1ccc(C)c(C(C2(SC)CCCC2)NC(=O)NC2CCCC(C(N)=O)CC2)c1 c1(OCCCCC)cc(C(N2CC3C(N(C)C(c4cocn4)=O)C3C2)=O)ccn1 C1(C(=O)NCC(=O)N(C)C)(CNC(c2c(C)cc[nH]2)=O)CC(C)(C)C1 Cc1ccc(F)cc1C(=O)NCC1CCCN(C(=O)CC2(C#N)CCCCC2)C1 C=CCC(CNC(=O)C=CC1(C)COC1)C(=O)NCc1ncn(C2CC2)n1 C12(NC(C(C(C)C)C)=O)CCC(CC1)N(C(=O)CCCC1CCC1)C2 n1(CC)ncc2c1CC(C(=O)NCC#CCNC(c1ccn(CC)c1C)=O)CC2 c1(C(N2CCC(NC(=O)Cc3cnco3)C(F)C2)=O)cnc2scnc2c1 CC1CCNC(=O)C1NC(c1ccc(CNC(=O)Cc2c(F)cccc2F)o1)=O N1(C(c2cnc(C)[nH]2)=O)CC2CN(C(C3(C4CCCO4)CC3)=O)CCC12 N1(C(C(C=C)(C)CC)=O)C2CCCC1CN(C(C1CC(C)CO1)=O)CC2 C1(O)(C(CNC(c2ccc(C)o2)=O)C)CCN(C(=O)C=Cc2scnc2C)C1 c1(C(=O)NC(C2CCN2Cc2noc(C3CC3)n2)C)cc(C2CCCC2)no1 C1(C(=O)NCC2(F)CC(NC(c3c(CC)occ3C)=O)C2)CCC2C1C2(F)F C(=O)(CCCC(F)F)N(CCCCN(C)C(c1cnc(CN)[nH]1)=O)C c1(CCC)cc(C(N2CC(O)CC2CNC(=O)C(C)(C)n2cccn2)=O)ccn1 C=CC(CC)C(=O)NC1C=CC(CNC(c2cn(C(C)C)cn2)=O)C1 C1(NC(c2c(C)[nH]cc2)=O)COCCC1NC(=O)CCC1CCC(C(N)=O)O1 c1(NC(c2ncc(Br)nc2I)=O)nccc2[nH]ccc12 CN1CC2CC2(CNC(C2(C3CCCN3C(=O)C3=CCCC3)CC2)=O)C1 C(C)(C)(CCC(=O)N1CCCC(O)(CNC(=O)C=Cc2ccncn2)C1)OC CCC(CCc1ccccc1)C(=O)NCCN(c1cc(O)nc(C)n1)C1CC1 N1(C(c2ccc(C)cc2)=O)CC2CN(C(c3occc3Br)=O)C2C1 N1(CC(=O)NC2CCC(NC(=O)Cc3ccoc3)C2)Cc2ccccc2C1=O c1(C(N2CC(COC)(CNC(=O)C(C)N(C)C)C2)=O)cc(C(C)C)n(C)n1 c1(OC(C(=O)OCC)=NOCc2noc(C3(F)CCC(CN)C3)n2)c(C)occc1=O C(C(C(=O)N1CCC1CC(=O)NCCCc1nncs1)N(C)C)OC CCCC(C(=O)OC)C(=O)N1CCCOC(CNC(=O)CCc2ccncn2)C1 N1(C(c2ccc(CF)cc2)C(=O)NCCCSCC)CCN2CCCC2C1 N#Cc1cncc(C(N2CCOCCC2C(N2CCC(CC3CC3)C2)=O)=O)c1 c1(OC)cc(C)ccc1NCC(N1CCCC(C)(C(=O)NC2CCCCC2)C1)=O Cc1cc(C(=O)NCC(C)CN(C(=O)C(CC(F)F)C2CCC2)C)ncc1N c1(C(N(C)CC2CCCCN2C(C2C3COCC23)=O)=O)c(Cl)ccc(O)c1N C(CC)(C(=O)N1CC(C(C)CC2CCC2)C1)N(C(C=CCC)=O)C c1(CC)cnc(C(=O)NC(C2CCCN(C(=O)Cc3cc(C)ccn3)C2)C)nc1 C1(CCN(CC(=O)NCC=C)C)CCN(C(C2(CC)CC=CCC2)=O)CC1 C(C1c2ccsc2CCN1C(C1CC1C1CCC1)=O)NC(c1ccc(CO)s1)=O CCCC(C)(C)C(=O)NC1CCOCC1NC(c1csnc1Br)=O CN1CC(NC(C2C=CCN(C(C3SCCS3)=O)C2)=O)CCC1=O c1(-n2cc(C(=O)OC)nn2)cccc(S(=O)(=O)N(C)CCc2cccc(Br)c2)c1 c1(N2CCCC3(C(=O)Nc4snc(SC)n4)C(C2)C3)[nH]cnc2nc(Cl)cc1-2 n1(CCC)ccnc1C(F)(F)C(=O)N(C)CCN(C)C(C1(F)CCCC1)=O c1(CNC(C(=O)NCCOC)Cc2ccccc2)ccc([N+](=O)[O-])cc1 C12(C(N(CC(=O)NCC(C)(CC)CO)CC#C)=O)CCCC1C2(F)F c1(CCC)occc1C(=O)N(C)CC1(NC(C23CCC(C2)C3)=O)CC1 c1(CN2C(CCC(N3C4CCC3COC4)=O)CCC2)ccc(I)c(F)c1F C1(C(=O)NC2(C)CCN2C(c2ccc(N=[N+]=[N-])cc2)=O)CC2(COCCO2)C1 CC1CC(C)N(C(=O)Cn2cc3ccccc3n2)CCN1C(c1ccon1)=O c12cc(OC)cc(c1)C(C1CCOC1)NC2.c1(OCC)nn(C)cc1OC C1(NC(c2cc(C)cc(C)n2)=O)CCCC12CN(C(=O)CN1CCCC1CO)C2 C1(NC(COCC)=O)(COC)CCN(C(c2ccnc(C(C)(C)C)n2)=O)C1 N12CCOC(C1)C(=O)N1CCC(CC1)C2.S(=O)(=O)(Cc1ccon1)CN(C)CC FC(F)(F)C(F)(F)CCCCNCc1c(Br)nsc1Br C1(C(F)(F)F)(COC)CN(C(c2nc(-c3cccc(F)c3)sc2C)=O)CCO1 c1(C(=O)NCC2(OC)CN(C(C(CCOC)C)=O)C2)cc(S(N)(=O)=O)ccc1F C1(OC)CC(C(=O)N(CCCO)CCO)N(C(=O)Cn2ccnc2C)C1 C1(O)(CNC(CC(=C)C)=O)CCCN(C(C2CCN(C(=O)C(C)CC)CC2)=O)C1 Cc1cc(C)c(C(N2CC(CNC(=O)C(O)C(F)(F)F)C3(CC3)C2)=O)c(O)c1 c1(C(N2CCN(CCC)CC2)c2ccccc2)ccc(Cl)cc1C(F)(F)F n1(CC#C)cc(NC(=O)CC(c2cccs2)c2nccs2)cn1.c12nnnn1C2 C(CN=c1nc2scnc2c(NCc2cnn(CC(F)F)c2)[nH]1)c1nnn(C)n1 O=C(C1=CCCCC1)N1CCCCC1C1CCN(C(c2ncncc2Cl)=O)C1 C1(O)(CN(C(c2ccc[n+]([O-])c2)=O)CC)CCCN(C(=O)CCCCN2CCC2)C1 c1(C(=O)NC(CNC(C(CSC)O)=O)(C)C)ccnc(C(F)(F)F)n1 C1(CCCNC(CCSCCCC)=O)CCCN1C(=O)CCCc1csc(C)n1 C(=O)(C1OCCc2c(O)cccc21)N1C(CC)CN(C(=O)C=CC(C)C)CC1 c1(C(N2C(C)CCN(C(=O)Cc3ccsn3)CC2)=O)ccc2c(c1)B(O)OC2 c1(C(N(C)Cc2cccc(CNC(C(C=C)(C)C)=O)c2)=O)cc2n(n1)CCO2 c1(C(=O)NC2(C)CCCN(C(C=C(C)C3CC3)=O)C2)nc2nc(C)cc(C)n2n1 CC(CNC(c1cscn1)=O)(Cn1cccn1)NC(C1CC(C(F)F)C1)=O Cc1nnc2c(NCc3ccncc3-c3cccc4nccnc34)cc(Cl)nn12 C(=O)(C(F)(F)C(F)F)NCC(CC(C)C)NC(=O)CC1OCCC1C C(=O)(CC=CCNC(=O)CCN(C)CCC)N(CC#C)CC1CC1 N1(C(c2ccc(C)cc2F)=O)C2CCC1C(F)C(NC(C1CC(CCO)C1)=O)C2 Cc1oc(C(F)(F)F)nc1C(=O)NC(C1CN(C(=O)C(C)C2CC2)CCO1)C C1(NC(C(N2CCOC2=O)C)=O)CCCCC1NC(c1ccncc1)=O c1(C(N2CCC(F)(CNC(c3cn[nH]c3)=O)C2)=O)c[nH]c(=O)c2ccncc12 C1(NC(C2(CF)CCN(C(C3N(C)CCC3)=O)C2)=O)CC2CCCC2C1 c1(C(=O)NCCN(CCOC)CC)nc(C)n(C)n1.c1(C)ccc(C(C)CC)cc1 Cc1c(C)c(CNC(=O)Cn2cc(CC3CCCC(F)(F)C3)nn2)c(C)c(C)c1Br C1(CC(=O)NCCSC(F)(F)F)CC(CO)N(C(=O)CCn2cc(Cl)cn2)C1 Cn1ccc2cc(C(=O)NC3CC3CNC(C34CC3CCC4(F)F)=O)cnc12 C1(C=C)(C(=O)NCC(CC=C)NC(=O)CCCCN2CCOCC2)CCCCC1 c1(C(=O)NCC2(O)CCCN(C(C(C)CC(F)F)=O)C2)cc2cnc(Cl)cc2s1 n1(CC(C)C)cc(C(=O)NCCC2(CNC(=O)CC3OCCC3C)CCC2)cn1 C1(C(C)C(=O)N2CC(C3CCOCC3)C2)CCN(C(C2CCS(=O)CC2)=O)CC1 N1(C(CCCC#C)=O)CC2ON=C(CNC(=O)C=Cc3cocn3)C2C1 Cc1cccnc1C(C)NC(C1(NC(C2CN(C)CCO2)=O)CCCC1)=O c1(CC(=O)NC2CCCC(NC(C(CC)(C)F)=O)C2)cccc(Br)c1Cl c1(C(=O)NCC2N(C(CCN(C(CCC)C)C)=O)CC2)ccc(S(=O)(=O)NC)s1 O=C(CC1=CCCC1)NCC1OCCC1C(=O)NCC(O)C1CC1 c1(CCN2CC(NC(C(C3CC=CCC3)NC(C)=O)=O)C2)ccccc1 c1(C(=O)NCC(F)(F)F)cccc(Cl)c1N.C1C(C)(C)CNC(=O)C(C)N1C C1(C(=O)NCC2CC(NC(=O)CCc3nccs3)C2)CCCS1(=O)=O N1(CC(C2CCC(C(=O)OC)C2)=O)CC=CC1(C)C c1(C(NNC(c2n(C)cc(Br)c2)=O)=O)c[nH]c2ncc(F)cc12 CC(C)(C)CCCC(=O)NC1CCC(F)(CNC(=O)Cc2cc(Br)ccc2F)C1 c1(C(N2C(C3CCN(C(CCC=C)=O)CC3)CCC2)=O)c[nH]nc1[N+](=O)[O-] C1(NC(CN(C)S(N)(=O)=O)=O)CCC(NC(=O)CC2(C(F)(F)F)CC2)CC1 Cn1ccc(C(=O)NCC2C(O)C(O)CN2C(c2ccnn2CCF)=O)cc1=O C(=O)(C(C)(O)CCc1ccccc1)NCC(CNC(C1OCCN(C)C1)=O)(C)C Cc1cc(C(=O)NCC(O)CNC(=O)C(C)c2ccsc2)c(C)n1C(C)C N1(C(C2CC(SC)C2)=O)CC(NC(=O)COc2cc(Cl)ccc2Cl)CC1(C)C C(=O)(CCNCCN(CC)CC)NC(C)C(=O)NC c1(C(=O)NCC(CN(C(c2c(C)nc(C)[nH]2)=O)C)O)cc2c(C)ccc(F)c2o1 CC(C)CC(C(=O)N1CCOCC1CN(C)C(c1ccn(CCN(C)C)n1)=O)N(C)C C1(N(C(=O)CN2CCCC2CSC)CCC)CCN(C(C)=O)CC1.C1(C)C(=O)N1 Cc1cc(NC(c2cccc(C#N)c2)=O)ccc1NC(c1ccoc1C1CC1)=O c1(NCCCN(C(c2nccc(C)c2)=O)C)ncnc2c1nnn2CC1CC1 S(=O)(=O)(c1cnc(NC23CCCC2C3(F)F)c(Cl)c1)NCC1CCCN(CC)C1 C1(CNC(C=C(CCC)CCC)=O)CCCCCN1C(=O)CC1CC(C)(C)C1 C1(NC(c2cnc3c(n2)CCCC3)=O)CCC2CN(C(C3CC(F)C3)=O)CCC2C1 N1(CC)CCC(C(=O)Nc2cc(N3CC(C(=O)OC)C3)ccn2)C1=O C(c1ccc(OC(C)C)c(C)c1)=CC(=O)NC(CCNC(C(C(C)C)SC)=O)C C(C(O)CN=c1[nH]c2cccc(F)c2o1)NC(C1(O)CCOC1)=O N1(C(=O)Cc2cnoc2)CCN(C(=O)CN2CCOCC2=O)C2CCCCC2C1 C1(CC(=O)N(CC(CNC(C(C)CCN(C)C)=O)C)C)CCC2(CC2)CO1 C1(CC)CN(C(=O)CN(C)C(C)C)CCC1NC(c1ccc(OC)nc1)=O Cc1cccnc1C=CC(=O)NC1CC(CNC(C2(S(N)(=O)=O)CC2)=O)C1(C)C c1(CNC(=O)NCc2ccc(Cn3cnnc3)cc2)cnc(Cl)c(Cl)c1 C12(C(=O)NCCCOCCCNC(c3cc(OC)no3)=O)CC1COC2C C1(N(C(=O)CC2OCCCO2)CC#C)CCN(C(c2cccnc2)=O)CC1 c1(C(=O)NC2CCCN(C(CC3CC(SC)C3)=O)C2C)sc([N+](=O)[O-])cc1Cl CCS(=O)CC(=O)NCc1cc(C(=O)NCc2ncc[nH]c2=O)ccn1 CCC(CC(C)C)C(=O)NCC(C)CNC(=O)Cc1cccc(OC(C)C)c1 CC1CC2(CC(CNC(=O)C(CCF)NC(=O)C3=CCCOC3)C2)C1 Cn1ncc2cc(C(=O)NCC3CC4CCC(C3)N4c3ncc(F)cn3)sc12 N1(C(C2CN(C)C2)=O)CC2CC2(NC(=O)CNc2ncccn2)C1 N1(c2snc(C(C)(C)C)n2)CCC2(CCCN(C(=O)CC3CCCCO3)C2)C1 C(c1ccc(F)cc1)=C(C)C(=O)NC1CN(C(c2c(C(F)(F)F)ncn2O)=O)C1 O(C1CCCc2ccccc21)CC(=O)N(C1CCN(C(C)=O)C1)C c1(C(=O)NC)cc(F)ccc1NC(=O)CCc1ccc(C(N2CCCC2)=O)[nH]1 N#Cc1ccccc1CC(N1CCCC(NC(=O)C(C2CCCCCC2)O)C1)=O c1(C(=O)OC)cc(C(N2CCCCC2CNC(c2ccc(C)cn2)=O)=O)c(C)o1 N1(CC(=O)N(C2C(NC(CCCCOCC)=O)CCCC2)C)CCCCCC1=O C1(C(=O)NCC2CCN(Cc3c[nH]c(Br)c3)C2)CC2CCNCC2C1 c1(N2CC(CNCCOC(=O)CNC(C)=O)OCC2)cnc(O)c2ncccc12 c1(OC)ccc(-n2nnnc2C(c2cc(C)nn2C)NCCCC2CCC2)cc1 c1(C(=O)NCC(CCC)NC(CN(CCC#C)C)=O)nccnc1C c1(OC(CC)C(=O)NC(C)(C)CN(C(=O)CN(C)CC)C)ccccc1F Cc1nn(C)c(Br)c1C(=O)NCCn1cc(CNC(C2CCCS2)=O)nn1 c1(C(=O)NCCCOCCNC(CS(N)(=O)=O)=O)cc2cc(Cl)ccc2[nH]1 c1(COC)noc(COC(=O)CONC(=O)Cc2nc(CO)no2)n1 C(C(=O)NCC1CCCC1NC(C1CCN(CC(F)F)CC1)=O)(C(C)(C)C)OC c1(C(N2CCC(OC)(CNC(=O)C(F)C3CCC3)C2)=O)cc2ccccc2[nH]1 C(=O)(NNC1CCCC1)NC1CCN(C(C)=O)CC1 C#Cc1cncc(C(=O)N(C2CC(NC(C3CC3(c3ccccc3)C)=O)C2)C)c1 C12(NC(C3C(CCC)C3)=O)CCCCC1CN(C(c1ccc(S(N)(=O)=O)o1)=O)C2 C1(C(=O)NCC2N(C)CCN(C(Cc3ccc(C)s3)=O)C2)C2CCCCCCC12 c1(CNCCCC(C2CCCC(C(=O)NCc3occ(C)c3)C2)C)cnn2c1CCC2 C(=O)(N=c1cc(C2(C)CC2)[nH][nH]1)NCc1cc(C(C)C)cc(C(C)C)c1 N1(C(C2(CC=C)CCCC2)=O)CC=C(C(=O)N2CCC(O)(C(N)=O)C2)CC1 CCC(CC)C(C(=O)NC1CCCN(C(c2cnc3n2CCC3)=O)C1)OC C1(C(=O)NC2CCN(C(C3N(CC)CCOC3)=O)C(C)C2)CN2CCN1C(C)C2 N1(C(C(CC)NC(N)=O)=O)CCC(NC(=O)Cc2ccc(F)cn2)C12CC2 C1(C(=O)NCc2n(CC)ncc2)CC12CCN(C(=O)C(F)CC)CC2 c1(OCC)cccc(C2CC2C(=O)N(C)CCNC(C2CSC2)=O)c1 CC(C)C(CO)C(=O)N1CCC(C(C)NC(=O)CC2C=NN(C)C2=O)C1 C1(NCc2cn(CC(C)NC(C(C)NS(C)(=O)=O)=O)nn2)CCS(=O)(=O)N1 C1(C(=O)NC2CC(F)C2)CC(F)CN1Cc1cnc(Cl)s1 CC1CC(CNC(=O)CC23CC4CC2C3C4)CN1c1ncc(I)cn1 C1(OC)CN(C(c2ccc(O)nc2)=O)CC1NC(=O)CCCNC(=O)C(C)(C)C C(=O)(C#CC1(C)CC1)NCC1CC(OC)CN1C(C1CC(OC(F)F)C1)=O c1(C2C(C(=O)NCC34CC(CNC(C(C)SC)=O)(OC3)C4)C2)cccc(F)c1F N1(c2c(OC)cc(OC)c(N)c2)Cc2nn(C)c(CO)c2C1.C(=O)O c1(C(=O)OC)ccnc(C(=O)NCC2CCC(NC(C3CCSCC3)=O)C2)c1 Cn1cc(CCn2cc(C3(O)CN(C(=O)CC4OCCO4)C3)nn2)cn1 C1(C(N2CCN(C(CC)=O)C(CC3CC3)C2)=O)Cc2ccccc2CO1 CC(C)C(CNC(C1CC2(CCC2)C1)=O)C(=O)NCC1C(C)(C)C1(F)F c1(NC(c2cccc(-c3cn[nH]c3)c2)=O)[nH]nc2c(Br)cnc(F)c12 CCCC(C)(O)CN(C(=O)CCC1CCN(C(=O)COCCC(C)C)C1)CCOC C1(CNC(c2snnc2C2CC2)=O)CN(C(c2cc[n+]([O-])cc2)=O)CCC1(F)F c1(C(C)C(=O)N(CC(C)(C)NC(C2CCCO2)=O)C)cccnc1 C(CC(=O)NCc1cc(C)ccc1F)(C(F)(F)F)NC(C(C)=C1CCCC1)=O c1(C(=O)NCc2scc(C(N3C(C(C)C)CCCC3)=O)c2)ccc(F)c(O)c1 N1(C(C=CSC)=O)CCC2CCN(c3nc(Cl)ncc3C(C)C)CC2C1 c1(C2(C(=O)NC3C(OC)CN(C(=O)C(C)C(C)C)C3)CC2)cc(F)cc(C#N)c1 N1(C(C)=O)CC(NC(c2cc(-n3ccnc3)ccn2)=O)C2(CC2)C1 c1(OC)ccc2c(C(N3CCOC(CNC(=O)C(O)C(F)(F)F)C3)=O)cnn2c1 N1(C(C2(CC=C)CCCN2C(C2C(C)C2C)=O)=O)CCc2cccnc2C1 CC(C)C(CC(=O)NC1CC(NC(C2CC23CCCCC3)=O)C1)c1ccccc1 c1(C(N2CCC(C(C)(C)C)(CNC(C(C)CO)=O)C2)=O)coc2ccc(F)cc12 c1(C(=O)NC2(C)CN(C(C3CC=CCC3)=O)C2)cc(C#N)ccc1O N1(C(c2c(C)nccc2Br)=O)CCOC2(CCN(C(=O)C=CC(C)C)CC2)C1 c1(C(=O)NCC2C(NC(c3ccnc(OC)n3)=O)CC2)ccnc2cc[nH]c12 C(C1=NOC2CN(C(C3CC4CCC(C3)C4)=O)CC12)NC(c1nc(C)sc1C)=O C1(NC(CCc2c(C)noc2Cl)=O)CCN(C(c2nocc2C2CC2)=O)CC1F n1(C(C)C)ccc(C(=O)NC2CCC(CC(=O)NC(c3nc(CO)n[nH]3)C)C2)c1 CCC(C(=O)N1CC=CC1CNC(c1sccc1CN(C)C)=O)C(C)(F)F C1(C(C)NC(=O)CCn2cccn2)CCN(C2CCCC2)C1 N1(C(c2c(C)cncc2)=O)CC2(CC2)CC1CNC(=O)CC(=O)NC1CCCC1 C(=O)(CCCC(=O)N(CCNC(C1CCCNC1=O)=O)CCOC)NCC C1(C(=O)OC)CC12CCCN(C(=O)NCc1csc(Br)c1)C2 N1(C(Cn2c(C)csc2=O)=O)CCCOC(CNC(c2cnc(Cl)cn2)=O)C1 Cc1cc(C(N2CCCC2C2(O)CN(C(C3CCC3C)=O)C2)=O)ncn1 C(=O)(CCC(C(C)C)NC(C1CC(O)C1)=O)NC(COC)C(=O)OC C(C(F)(F)C(=O)NC(C)CC1CN(C(=O)C(c2cncn2C)OC(C)=O)C1)OC c1(CC)cc(C(=O)NCC2CCN(C(=O)Cc3ccoc3C)CC2C)c(C)nn1 c1(CNC(C23CC(NCc4ccc[nH]4)(C2)C3)=O)ccc(Cl)cc1 C1(NC(C(N2CC(C)C2)C)=O)(CNC(=O)CNC(c2cccs2)=O)CCCCCC1 C1(NC(c2c(C#C)cn(C)n2)=O)CC1C1CCN(C(=O)C(C)(C#N)CC)CC1 N1(C(C(C(=O)OCC)(C)C)=O)CCC(C)N(C(=O)Cc2cc(C)on2)CC1 n1(CC)ncc(Cl)c1C(=O)N(C1CCCN(C(c2cc(C(N)=O)co2)=O)C1)C(C)C N1(C(C(C(C)C)OC)=O)Cc2cc(Br)cnc2C1 c1(C(N2CC3C(C(=O)Nc4c(OCC)nccc4C)C3C2)=O)cccn2ccnc12 C1(CNS(C)(=O)=O)CCC(CNC(=O)COCCC(=O)NC2CCC2)CC1 C1(CNC(C(C(C)C)F)=O)CCC(C)(C)CN1C(c1ccc(Cl)cc1)=O c1(C(=O)OC)c(C(=O)N(C)CC2CCCCN2C(c2nocc2C)=O)n[nH]c1C C12(CNC(C3CN(CCC)C(=O)C3)=O)CCC(CC1)N2C(C1SCCS1)=O c1(C(CC)C)ccc(C(=O)NC2CC23CC(NC(=O)C(F)(F)CSC)C3)cc1 C(=O)(C1Cc2ccccc21)NCC1CCCN(C(c2c(OC)cccn2)=O)C1 Cn1cc(S(=O)(=O)N2CCOCC2C(=O)Nc2cc(Br)ccc2I)cn1 N1(C(C(C=C)OC)=O)CC(N(C)C(c2cc(C)nn2C)=O)C(F)C1 C1(C(=O)NCC2C(NC(c3ccc(C)o3)=O)COC2)CCCN1N=O C(=O)(C1CCC(=O)c2cccn21)NC1(CC)CCN(C(CC(C=C)CC)=O)CC1 C(=O)(C(CCC)N(C)C)NCCn1ccc(C(N(CCCC)C(C)CC)=O)c1 C1(C(=O)NC2(C(=O)OC)CCC2)COC2CN(C(c3coc(C)n3)=O)CC12 c1(CNC(C(=O)NCCC(N2CCCC2)C)=O)cc(S(C)(=O)=O)ccc1F N1(C(c2c(Cn3cc(CC(=O)OC)nn3)cccc2)=O)CCC(C2CC2(F)F)C1 Cc1c(NCCCC2CCNC2=O)c(C(N)=O)c(C)n1C Cc1cc(C(=O)NCc2cccc(NC(=O)CC3CCC4CC34)c2)n(C)n1 CCC(F)(F)CC(=O)NC1CN(C(c2c(Br)ncn2C)=O)CCC1O c1(C(=O)NC(CNC(C(C)OCC(C)C)=O)CO)cc(S(=O)(=O)N(C)C)c[nH]1 C1(C(C)CNC(=O)CC2(C)CC2)CCN(C(=O)Cc2ccsc2)C1 n1(CC)ccc(O)nc1=O.C(C(C)c1ccccc1)(C(=O)OC(C)(C)C)N(C)CCBr C12(C(=O)OCC)CCCC1CCN2C(C12COCC1C2(F)F)=O C1(NC(C(CC)C)=O)CN(C(=O)Cc2ccc(C(C)(C)C)cc2)CCC1F c1(-n2ccc(C(N3CCC(C(C)(C)NC(C(F)=CC)=O)C3)=O)n2)ccc(F)cc1 N1(C(c2[nH]cc(CC)c2)=O)CCC(NC(C2(F)CCCC2)=O)C1C C1(NC(C2CC(OC)C2)=O)(CNC(c2cnccn2)=O)CC2CCC1CC2 c1(N2CCN(C(Cc3ccc(C#N)cc3)=O)C3C2C3)ncnc2occc12 C(=O)CC1CCc2ccccc21.C=CC(C1CCC1)NC(=O)OC.OC N1(C(=O)NCc2cc(S(N)(=O)=O)oc2)CCOc2cccc(Br)c2C1 N1(C(c2[nH]cc(C)c2)=O)C2CCC1CC(NC(c1c[nH]nc1C(F)F)=O)C2 CC1=NS(=O)(=O)NC=C1C(=O)NCC(C1CCC1)NC(C1(C)COC(=O)C1)=O N1(C(C=C(CC)CC)=O)CCC(NC(=O)Cc2ccc(F)cn2)C(C)(C)C1 N1(C(CC(C)N2CCCC2=O)=O)CCN(C(c2ccc(N)cn2)=O)CC1CCO C(CCC(C)CC(=O)N1CCN(C)C(CNC(c2ccccc2CO)=O)C1)=C(C)C O=S(=O)(c1ccc(Br)c(Cl)c1)NC1CCN(Cc2ncccc2F)CC1 C1(CCNC(CC2ON=C(C)C2)=O)CCCN(C(c2cn(C3CC3)cn2)=O)C1 C(C(=O)NCCOCCNC(c1cn(CCO)nc1C)=O)(C(C)C)SC C1(C(=O)NCC(CCOC)NC(c2ccccc2N(C)C)=O)CCC(F)(F)CC1 c1(OC)nccc(Cl)c1CN1CC2C(C1)N2C(c1ccc(C)cc1)=O Cc1c(Br)c(C(=O)NC2C3CCC2N(C(C2(O)CCCC2)=O)C3)nn1C N1(C(C(C)C#N)=O)CCOC2(CCCN(C(=O)Cc3cc4ccccc4o3)C2)C1 c1(C(=O)OC)ccc(S(=O)(=O)NCC(C)(CN)OCC2CC2)cc1 N1(C(CN2CC(CC)C2)=O)C2CCC1C(CNC(C13CCC(OC)C1C3)=O)C2 c1(C(N2CCCN(C(c3n4c(nn3)SC(=C)C4)=O)CC2)=O)cn2c(n1)CCCC2 c1(C(N2CCCC(NC(=O)Cc3ccoc3)C(F)C2)=O)cc2c(F)cccc2s1 N1(C(=O)NCc2ccc(C)cc2)CCCN(C(C)C)CC1C.C123CC(C1)(C2)N3 C(C)(C1CCCCC1)=CC(=O)NCCN(C(C1(C)CC=CCC1)=O)CC C=CCC(C)(C)CC(=O)NC(Cc1cn[nH]c1)C(=O)NC(C)CCN1CCCC1 C1(N)(CC(N2CCC(N(C(=O)CO)C)CC2)=O)CCS(=O)(=O)C1 CN1CCN(CC(N2CCCC(C)(CNC(C3(CC(F)F)CC3)=O)C2)=O)CC1=O C1(CCC)CN(C(=O)Cc2c(Cl)cnn2C)CCN1C(=O)C1=CSCS1 N1(C(CCC(=O)OC)=O)CC(NC(C2COCCC2(F)F)=O)C2(CC2)C1 c1(C(=O)NC2(C)CC(NC(C3C(C=C)CC3)=O)C2)ccc(-c2ccco2)nc1 CC(C)(CC(=O)NCC1CCN1C(c1ccc(C(F)F)nc1)=O)c1ccccc1 C1(N(C(CCN(C(C(C)OCCCC)=O)CC)=O)C)CCN(C)CC1.C(CO)O CN1CC(C(=O)NC2(CNC(C3(C(C)C)CNC(=O)C3)=O)CCCC2)CC1=O c1(C(N2C(C(N(CC(C)C)CCOC)=O)CC2C)=O)ccnc2cc[nH]c12 c1(C(=O)NCC(CO)NC(c2cc3ccccn3n2)=O)n[nH]c2ccccc12 c1(C(=O)NC2(COC)CCN(C(=O)C(C)=C3CC3)C2)cnc2ccccc2c1C N1(C(C2(F)CCN(C(CC#C)=O)CC2)=O)CCC2(CC1)CC2(F)F c1(C(N2CCN(C(CC(C)c3ccccc3)=O)CC2C)=O)ncccc1[N+](=O)[O-] C1(C(=O)NCc2occ(C(N3CC(CC(C)(C)C)C3)=O)n2)CC2CCCCC12 c1(C(=O)NC(C2CN(C(C3CC=CC3)=O)C2)C)cnc2c(cnn2C)c1N C(=O)(C1=CC2CCCC12)NCC1CN(C(CCn2ncc(C)c2)=O)C(C)C1 c1(CC(=O)NC(CN(C(C2CC(F)C2)=O)CC)C)occc1C(=O)NC c1(CC)nc2sc(C)cn2c1C(=O)NC1COCCN(C(=O)C(C)COC)C1 C1(NC(C2C(NC(C3C(C)C3)=O)CCOC2)=O)C2C3CC4C1C1C2CC3C41 C1(CNC(C2CC(CCO)C2)=O)CCN(C(=O)C(F)(F)CO)CC1C1CC1 C(=O)(C1=CNC2=NCCC2=C1)N1C(C)CCC(CNC(Cc2c(C)nc[nH]2)=O)C1 N1(C(c2c(C)noc2)=O)CCC(C)(CNC(=O)C(N2CCOCC2)C)C1 c1(OCC#C)cc(CN)ccc1O.N1(C(C)CN(C)C)CCCC(CCSC)C1 CN1CC(C(=O)NCCN(C(c2occc2C2CC2)=O)CC2CC2)NC1=O CCC(C(=O)N1CCC(NC(c2ccccc2CN(C)C)=O)C1C)NC(N)=O C(=O)(C(CC(F)F)NC(C1COC(=O)N1)=O)NCC(C(C)(C)C)O CCC(O)C(C)(C)C(=O)N1CCN(C(=O)CC2CC(F)C2)CC(C)C1 C1(OC)(OC)CCCCC1NC(=O)CC1CCC2CNCC12 CS(=O)(=O)CCC(=O)NCCC1CN(C(=O)CCOCCN(C)C)CCO1 c1(C(c2nnnn2C)NCc2nc(CC)on2)cc(C)c(=O)n(C)c1 C1(C(=O)NC(CC(C)NC(c2n(C(C)C)ncc2Br)=O)C)CCC(=O)CC1C c1(C(=O)NC(CC)CNC(C2CC=C(C(C)C)CC2)=O)cc(F)c(C)c(N)c1F CCC(C)C(C(=O)N(C(C)CNC(N)=O)C)NC(=O)Cc1ncc(Cl)s1 C1(C(N2CC(N(C(CCc3c(C)n[nH]c3C)=O)C)C2)=O)Cc2ccccc2C1 c1(C(=O)NC(CNC(C(C2CCC2)OC)=O)C)cccc(C(C)=O)c1 c1(N(CC(C)NC(=O)CCc2ccccc2F)C)nc2cc(Cl)ccc2s1 C1(NC(C(C)C(C)O)=O)CCCN(C(c2ccc(C3(O)COC3)cc2)=O)CC1 c1(C2(NC(c3ccc(C4CCC4)nc3)c3n(CC)nnn3)CCC2)ccc(Cl)cc1 c1(OC(C)C)cccnc1C(=O)OCc1csc(CC(F)(F)F)n1 n1(CCC(=O)NC(C2CCN(C(C3CC(CC)(CC)C3)=O)C2)C)cnccc1=O CC1CCC(CO)N(C(C2CCN(C(c3nccn3C(C)C)=O)CC2O)=O)C1 c1(C(=O)NCCN(C(c2c(C)nns2)=O)C2CC2)cc2n(n1)CCNS2(=O)=O CC1CN(C)CC(C(N2CCC(NC(C3(C(=O)NCC4CC4)CC3)=O)CC2)=O)O1 c1(C(=O)NC(CC(C)NC(c2ocnc2C2CC2)=O)C)ccc2c(c1)CCC2=O Cc1cc(CC(=O)NC(C)(C)CCCNC(=O)C(C)C2CCCO2)ccc1Cl N#CCS(=O)c1ccc(C(N2C3CCC2C3CO)=O)cc1 N1(C(CC=CCNC(C2(CC)CCCC2O)=O)=O)CC2CC(C1)N(C)C2 C1(C(=O)NCC2CCCN(c3nc(OCC)cc(C)n3)C2)CN(CC)CCN1C N1(CC2(NC(CCOCCC)=O)CC2)CCN(C(=O)C(C)(Cl)Cl)CC1 c1(NC(CC2(C=C)CN(C(=O)Cc3cncnc3)C2)=O)cnc2ncnn2c1 c1(C(=O)NC(CN(C(c2cc(OC)no2)=O)C)(C)C)ncc(F)c2ccccc12 c1(C(=O)NC2CN(S(C(C)C)(=O)=O)CC2F)cc2sccn2c1 N1(C(C(CSCC)N(CCN(C)C)CC)=O)CCC2(CC1)CC2CO N(C(=NCc1cc(C(F)(F)F)sn1)NCC1(SC)CC1)C(COC)C CCC(CC)(CC(=O)OC)C(=O)N1CC2(CC(NC(c3coc(Cl)n3)=O)CO2)C1 N1(C(c2c(C)nc(CO)nc2)=O)CC(NC(=O)CC2CSCCS2)CC12CCC2 CC1CN(C(c2cnco2)=O)CC(C)N(C(=O)C2=CCCC2)C1 N1(C(C2(C(C)(C)C)CCCC2)=O)CC2CC(NC(=O)C=CC3CCOC3)C1C2 [N-]=[N+]=NCCCCC(=O)N1CC(CC(=O)NCC2(O)CC=CC2)C2(CC2)C1 c1(C(=O)NC2C(NC(C3CCC(OC)C3)=O)CCC2)ccc(CCC(N)=O)cc1 CC1(NC(c2coc(CNC(C3CC3C3CC3)=O)c2)=O)CCC(O)CC1 N1(C(c2c(C)cn(C)c2)=O)C2CCCC1CN(C(=O)Cc1sccc1C)CC2 CC(CC1CC(F)(F)C1)C(C(=O)NCC1CCCO1)N1CCC(O)(C(N)=O)CC1 C1(C2CCN(C(C3CC4CC(C3)N(C3CCC(=O)NC3=O)C4)=O)CC2)(OC)CC1 C12(CC(=O)NC(CC(=O)NC)(C)C)CC3CC(C1)CC(O)(C3)C2 C(=O)(CCC(F)F)NC(C1CCCC1)CNC(CCCN(C(=O)OC)C)=O c1(CCC)ncc(C(N2CC(F)(CNC(=O)CCNC(N)=O)C2)=O)s1 C(=O)(C1=CS(=O)CCC1)N1CCN(C(=O)CCCCc2ccccc2)CC1CO N1(C(C(C)=CC)=O)CCC(CCNC(c2cc(C)sn2)=O)CC1 N1(C(C#C)=O)CCC2(CC1)CC(C(N1CC3(C1)OC(=O)NC3C)=O)CO2 c1(OC)ccc2nc(C)[nH]c(=NCCc3ccnc(C)n3)c2c1 N1(C(C(CC)CC)=O)CCN(C(c2cc(Cl)ccc2F)=O)C2CCCCC2C1 c1(C(N(CCNC(CN2CCC(C)CC2)=O)C2CC2)=O)cnn2c1OCC2 C1(CNC(c2cc3ccsc3s2)=O)CC2COCC2N1C(=O)CCC[N+](=O)[O-] Cc1cc(=NCCOCc2ccccc2)[nH]c(=NCCCn2cccn2)[nH]1 c1(CNC(C2C3CC3C3CC23)=O)cc(Br)cc2c1CCCC2 C1(CNC(c2nc(C)oc2)=O)CC(O)CN1C(c1cc(C)c(C)o1)=O C1(C(=O)NC(CC#C)CC=C)CC(F)(F)CN1C(c1sc(C)nc1C)=O C1(C(N2CC3CC(NC(=O)CCCCCF)C3C2)=O)(OCC)CCCCCC1 Cc1cnn(C)c1C(=O)NCCC1CN(C(C2(O)CCCCC2)=O)CC1C C1(N2C(=O)NC(C3(c4ccccc4)CCC3)C2=O)COC2(CCOCC2)C1 c1(C(C(=O)NCC(CNC(CSc2cc(C)on2)=O)F)=O)ccc(F)cc1 S(=O)(=O)(c1ccc(NCC2CCC=CCCC2)c(Br)c1)N1C(COC)C=CCC1 c1(OC)ccccc1C(O)C(=O)N(CCCN1CCCOCC1)C=C(C)C N1(CC(N2CCC(C)(CCNC(=O)Cc3cn[nH]c3)C2)=O)C(=O)CCCC1=O c1(C(=O)NCC2N(C(C(CCC)=CCC)=O)CC(OC)C2)cc(C)cnc1OC N1(C(c2n[nH]c(C)c2O)=O)CC(C(N2CC(F)C(F)C2)=O)OC(C)C1 c1(C(=O)NCC2OCCN(C(C=C(CC)C)=O)C2)c(S(C)(=O)=O)cnn1C N1(C(C2C(C#C)C2)=O)CCC(CNC(c2ccc(Cl)nc2OC)=O)C1(C)C N1(C(c2c(C)ncs2)=O)CCCC(C)(C(N2CCC(c3ccccc3)C2)=O)C1 C1(CNC(C(C)OCC=C)=O)CCC2CN(C(=O)COCc3ccncc3)CC12 CCC(C(=O)OC)C(=O)Nc1cccc(NC(=O)C=CC(C)(C)SC)c1 C1(C(N2CC(C(N)=O)C2)=O)CC(NC(=O)CSCC2CCCO2)C(O)C1 N1(C(c2n(CC#C)ccc2)=O)CC(O)CCC1C(=O)NCCCC1CCC1 C1(NC(c2n(C)nnc2)=O)CCC2CN(C(=O)CCC3CCCO3)CC12 C1(C(N2CC3CCC2C3)=O)CC(O)CN1C(c1cncc(CO)c1)=O CCC(C)C(CN(C)C)NC(=O)C=C(C)CNC(C1(C)COC(=O)N1)=O c1(CC)cccc(C(=O)NC(C)(C(=O)NC2CCC(O)C2)C2CCC2)n1 O=C(CCCN1CCCCC1)NCC1CCC(NC(=O)C(F)CC2CC2)C1 CC(C)(CC(=O)N1CCC(C)(C)C1CNC(c1coc(Cl)n1)=O)C(F)F N1(C(C(C)=C2CCC2)=O)CC2CCCC2(CNC(=O)CN2CCC(C)CC2)C1 C#Cc1cccc(C(=O)NC2C=CCN(C(C3(C)CC4CC4C3)=O)C2)c1C C=CC1(C(=O)NCC(CNC(=O)C(c2cncc(F)c2)(C)C)CO)CCOCC1 c1(C(N2CC(N(C(Cc3cc(C)[nH]n3)=O)C)C(C)CC2)=O)cnc2ncccn12 N1(C(CSC)=O)CC2CN(C(=O)CC(C(F)(F)F)NC(c3ccco3)=O)CC2C1 c1(C(N2CCOCC2C(F)(F)F)=O)cccc2[nH]cc(Cl)c12 c1(C(N2C(CNC(CN3C(=O)CN(C)C3=O)=O)C=CC2)=O)cc2cc(Cl)sc2[nH]1 Cc1ccc(Br)c(F)c1C(=O)NCC(CO)NC(c1ncsc1C(C)C)=O C1(CNC(CCC)=O)CN(C(C2CCOCC2(C)C)=O)C2(CCC2)C1 C=C(C)CC(C(=O)NCCCc1c(C)noc1C)NC(C1CC1(C)C(F)F)=O c1(C(=O)NC2C(NC(c3ccncc3Cl)=O)C2)ccc2snnc2c1 C(=O)(C(F)(F)C(O)C(C)C)NC1CCN(C(c2ccc(CCC)[nH]2)=O)CC1 CC1CCN(C(c2cc(O)cs2)=O)C(C(N2CCC(O)(C(F)F)C2)=O)C1 c1(Sc2ccc(-c3n(C)c(C(F)(F)F)nn3)c(Cl)c2)c(Cl)cccc1I c1(C(N2CCC(NC(C(C)OCCOC)=O)C(O)C2)=O)noc2c1COCC2 C(=O)(C(CCS(C)=O)N(C)C)N(CC(CN(C(=O)CCCNC(C1CC1)=O)C)O)C C(CC(C(C)C)NC(=O)CC12COCC(C1)C2)NC(C1C(CCC)C1)=O Cc1cccc(C(N2CCC(C(F)F)(CNC(C3CCC(C)CC3)=O)C2)=O)n1 c1(C(=O)NC2CC(C(=O)NC(c3ccsc3)C)C2)cccnc1O c1(C(=O)NCC2(O)CCN(C(=O)Cc3ccoc3)C2)cc2c(s1)CCCCCC2 C1(C(=O)NCCC(C)(C)NC(c2cnc(C(C)O)s2)=O)CCS(=O)(=O)N1 CCC(CC(=O)N(C)Cc1cn[nH]c1)N(C)C(c1coc(C(N)=O)c1)=O CCCCC(CNC(=O)CCc1ccc(CO)cc1)NC(=O)C(C(C)O)N(C)C C1(NC(c2scnc2C2CC2)=O)CC2CC(C1)N(C(c1cnc(C3CC3)s1)=O)C2 C1(CNC(CN(CCC)C)=O)CC2CCC(C1)N2C(C1CC1c1ccsc1)=O N1(C(C(c2cccc(O)c2)C)=O)CC(NC(c2nnn(C)c2N)=O)C(C)(C)C1 N1(C(c2cncc(N(C)C)c2)=O)CCC2CC2(NC(=O)CC2CCC3CC23)CC1 c1(CNC(C(=O)NC(C)CC2CCNC2)=O)ccccc1OCCO Cc1nc(NCCCCC(=O)NC2(CNCN)CC2)nc2ccccc12 c1(C(=O)NCC(c2ccccc2)NC(CCC#N)=O)cc(Cl)c(O)c(Cl)c1 C12CC3(C1)C(C1CCC3C1)NC(=O)N2.C(C(C(F)F)N1CCOCC1)OC c1(C(=O)NC23C(n4cc(CC(C)O)nn4)CC(CC2)C3)ccc2c(n1)OCO2 C1(C(N(CCC(C(C)C)NC(C2CCCOCC2)=O)C)=O)CCC2(CCC2)O1 n1(CC)cc(NC(=O)CCC2CCN(C(C3CCOC(C)C3)=O)CC2)c(C)n1 C1(CCC(=O)N(CC(CC)OC)C)CCCN1C(c1coc(C2CC2)n1)=O C1(CNC(C2CCC(C)O2)=O)C(C)CCCN1C(=O)CN1CC(=O)NC1=O C1(NC(=O)C(O)C2CC2)(COc2ccccc2)CN(C(C2CCC2)=O)C1 Cc1ccc(-c2nccc(C(C)NC(C3CN(S(C)(=O)=O)C3)=O)n2)cc1 N1(C(CN(CC(C)(C)C)C)=O)CCC2(CCCN2C(=O)CCCNC(N)=O)CC1 C#CCCCCC(=O)N1CC2CC2(NC(C2CC(=O)N(c3ccccc3)C2)=O)C1 Cc1cccc(CCOC(C2C=CC(CO)C2)=O)n1 C(C)(CO)(C1CCC1)NC(CN(C(=O)CC1CCC1)CC#C)=O c1(C(=O)NCC2CC(C)N(C(C3CC(F)(F)CS3)=O)CC2)n[nH]c2c1CC1CC21 c1(CNC(C2CCN(C(C(C)CC3CCC3)=O)C2)=O)ccnc(F)c1 N1(C(C(CC)C)C(=O)NCC(=O)OCC2CC2)CC(C)(C)OCC1CC C1(=CCNC(C2CC(SC)C2)=O)CCN(C(c2cc(C(N)=O)co2)=O)CC1 N1(C(C(C)OC(C)(C)C)=O)CCC(C(=O)N(C(C)CO)C)C(C)C1 c1(CNC(C(F)=CC)=O)cccc(CNC(c2cccc(CC#N)c2)=O)c1 Cc1ccc(OCCCC(=O)NC2CCCN(C(c3cc[nH]c3C)=O)C2)c(Cl)c1 CCCCC(CC(=O)NC1CC2(CCOC2)C1)NC(=O)C(CN(C)C)N(C)C c1(OC)cccc(F)c1CNc1cccc(C(=O)NS(C)(=O)=O)c1 C1(NC(C(C(C)C)N(C)C)=O)C2CC1CN(C(C1(F)C3CCCC13)=O)C2 CC(C)C(O)CC(=O)NCC(O)CC(=O)N(C1CCCCC1)C C=CCC(CC(=O)NC1(CO)CC(C)C1)NC(c1cn(CC)cn1)=O C1(CNC(c2c(CC)[nH]nn2)=O)CN(C(=O)C(O)C2CC2)CC1(F)F.C(C)(C)(C)O c1(C(=O)NC(C(=O)N2C(CN=[N+]=[N-])CC2)C2CCCC2)cncc(CO)c1 c1(C(CNC(C(C)N(C(=O)OC(C)(C)C)CC)=O)(C)C)ccccc1 S(=O)(=O)(c1ccc(NCC2COCCO2)c(Br)c1)N(C)Cc1cnsc1 CC(C)C(C)(F)CNC(=O)C(CNC(=O)C=CC1CCOC1)CC1CC1 c1(C(=O)NC2C(C)CN(C(=O)C(C)(C)C)C2)cnc2c(c1)c(=O)n(C)c(=O)n2C CC(=O)CCCC(=O)NC1CCN(C(=O)C(c2ccc(Cl)cc2)CO)C1(C)C Cn1ncc2[nH]c(C(N3CCC(C)(C)C(CNC(C4CC(C)(O)C4)=O)C3)=O)cc12 CCCC(C(O)C(=O)NCC(F)CO)NC(c1scc(C)c1C)=O CC1OC2(C(=O)NC(C3CN(C)CCO3)C)CC1(NC(=O)OC(C)(C)C)C2 c1(OC)nc(C(=O)NC2CCC(CNC(c3ncc(Cl)s3)=O)C2)cc(O)n1 N1(C(=O)NC)CCN(C(=O)N(C2CCOCC2)CCCNC(C)=O)CC1 C1(C)(C(N(CCNC(=O)Cn2cc(C#N)cn2)CC)=O)CCC(C)(C)CC1 CC1CN(C(c2csc(F)c2)=O)CCN(C(c2nn(C)cc2Cl)=O)C1 N#CC1(CNC(C2CC(F)CCN2C(C2CN3CCC2C3)=O)=O)CCOCC1 c1(NC2(CNC(C(C3CCC3)OC)=O)CC2)ncc([N+](=O)[O-])cc1F N12CC=C(CC1=O)CC2.C(=O)(C(C)(O)CC)NC1C(c2cn(CC)nc2)OCC1 C(=O)(C1=C(F)CN(C(=O)CC2(C)CCC2)CC1)N1C(C)CN(C)CC1 N#Cc1cncc(C(=O)NC(CNC(=O)CCCc2cccs2)C2CCC2)c1 c1(CC(N2C3CCC2C(NC(=O)C2=C(Cl)CCC2)C3)=O)ccc([N+](=O)[O-])cc1F CCC(C)C(C(=O)N1CC(C)=CC(C)C1)N(C)C(c1c[nH]cc1C)=O C1(NC(CN(C2CCC2)C)=O)CCC2CCN(C(=O)CC3CCCC3)C1C2 CCCCC(C(=O)N1CC(CO)(CF)C1)NC(=O)CC1C=CCCC1 c1(CC(=O)NCCCN(C(c2nccn2C)=O)CC)n[nH]c2ccccc12 FC1(F)CCCCCCC1NCCOc1ccc(-c2cccc(Cl)c2)nc1 CCCCC(O)C(=O)NCC(CC)NC(c1ccccc1CN1CC2CC2C1)=O CC(=O)CCC(F)(F)C(=O)NCCn1cc(CNC(=O)Cc2nncs2)nn1 C(CCO)(C(F)F)NC(C(CC1CN(C(CNC(N)=O)=O)C1)F)=O O=C1CCN(CC(=O)NC2CC3CN(C(C45CCCC(C4)OC5)=O)CC23)C(=O)N1 C1(C(=O)NC(C)(C)CNC(C23CCC(CO2)C3)=O)COc2cc(F)ccc2C1 c1(OC)ccc(Cl)c(C(N2CC(OC)C(NC(=O)CC(C)(C)C)C2)=O)n1 Cc1ccc(CNC(=NCCCC(C)O)NCCSC2CCCO2)c([N+](=O)[O-])c1 N1(C(c2n(CC)ncc2)=O)CCC2CCCC12C(N1CCC2CCC(C1)S2)=O C(=O)(CCS(C)(=O)=O)NC(CC)CNC(c1n[nH]c(CC)c1Cl)=O C1(CCC=C)(C(=O)NCC2CCCC2)CN(C(c2cn[nH]c2)=O)C1 C(C(=O)NC(CCNC(=O)CC=C(C)C)C(C)C)(C(C)(C)C)OC CC1C(NC(c2cnn3cc[nH]c23)=O)CCCN1Cc1cc(C2CC2)no1 c1(CC(=O)NCC#CCNC(C23CCC(OC)C2C3)=O)cn2c(C)csc2n1 c1(C(=O)N(c2nc(Br)cnc2Br)C2CNCCC2(F)F)sc(C=O)c(Br)c1Br c1(C(=O)NC2CCCN(C(C=C(C)C(F)F)=O)CC2)c(C)nn2cc[nH]c(=O)c12 C(=O)(CC(C)(C)C(=O)OC)N1CC(NC(C2C(CC)C2)=O)C2(C1)CC2 S(=O)(=O)(c1ccc(C#N)c(N2CCC3(CCCCO3)C2)c1)N(CCC=C)CC O(NC(=O)C#CC1CC1)CC(=O)OC.CCCCC1COC1 C1(C(=O)NC2(CN(C)C(c3cccc(F)c3F)=O)CC2)CCC2(CCCCC2)C1 C#CCCCC(C)C(=O)NCC1CN(C(=O)C=CSC)CCN1C Cc1ccc(-n2cc(C(C3CCN(C(=O)C4=CCCC4C)C3)C3CC3)nn2)c(C)c1 c1(CC)ncccc1C(=O)NC1CCN(C(c2nscc2Br)=O)C1 C(C(C(=O)NOC)NC(=O)C(C1(O)CCCCC1)NC)OCC CCC(C)C(C)C(=O)NC(CCOC)C(N1CC2(CSC2)C1)=O c1(C(N(CCCOCCNC(C(C(C)C)C)=O)C)=O)ccc2c(c1)NC(=O)CS2 Cc1ccncc1C(=O)NCC(C)(CO)NC(=O)C(C)SC(F)(F)F Cc1ccc(C)c(C(=O)N(CCCNC(=O)C(C)(C)n2cnc(C)c2)C2CC2)c1 N1(C(c2ccc(CC)nc2C)=O)CCN(C(=O)Cn2ccsc2=N)CC(C)(F)C1 c1(N(C)C)ccc(C(N2CCN(CCNC(=O)CCCC3CCC3)CC2)=O)cn1 C1(NC(CCc2cc(C)[nH]n2)=O)CN(C(C2CCC2(F)F)=O)C2(CCCC2)C1 CCCC(CC)C(=O)N1CCC(COC)C(O)C1 CC1(C)CN(C(C2(O)CC3CCC2C3)=O)CC1C(=O)NCC1CSCCO1 Cc1nc(N2CC(C)(NC(c3conc3C)=O)C2)c2ccsc2n1 C1(=CC(=O)NCC(CC)(CC)NC(=O)CC2(OC)CC2)CN2CCC1CC2 c1(C(N2CCC(N(C)C(c3ccc(C(C)(C)C)[nH]3)=O)C2)=O)cc2c(ccn2C)s1 C#Cc1cccc(C(=O)N(CCNC(=O)C(C)(O)C2CCCCC2)C(C)C)c1F c1(CC=C)cccc(C(N2CCC(C(=O)NCC(F)CC)C2)=O)c1 c1(OCCC)ccc(CNC2CC3(CCCCN3)C2)c(OC(F)F)c1 C1(CC(=O)NC2CCC(NC(C3(CC)CCCC3)=O)CC2)COC2(CCC2)CO1 c1(CC(=O)NC(C)C(C)NC(C2CC3CCC3C2)=O)n[nH]c2ccccc12 c1(OC)cc(CNC23CC2CN(C(c2c(Cl)cnn2C)=O)C3)ccc1Cl S(=O)(=O)(c1ccc(NCCOC(C)C)c(C#N)c1)N(CCCCF)C.C(C)(C)(C)O C(=O)(CS(C)(=O)=O)N(C)CC1(NC(c2cnc(C(N)=O)cn2)=O)CC1 c1(C(=O)NCCN(C)C(c2ncn3c2CCC3)=O)ccc(C2CC2)cc1Cl O=C1NCc2ccc(C(=O)NC3CCCCC3NC(=O)C(F)C3CC3)cc2N1 C(=O)(CCS(=O)(=O)Nc1ccnn1C)NCC(=O)NC(C)CCCCO C1(NC(C(CC)OCC)=O)CCN(c2cc(C3CCCCC3)ncn2)CC12CC2 C1(C2CCN(C(=O)CCCCO)CC2)(NC(=O)CCC(F)(F)F)CC1 O=S(=O)(c1ccc(NCC2COCCO2)c(F)c1)N1C2CCCC1COC2 c1(NC(CC2CN(C(c3c(OC)ccc(Cl)c3)=O)C2)=O)cc(F)c(Cl)c(Br)c1 C(=O)(C(CC)C(=O)N(CC(C)NC(=O)CC1CC2CC1C1CC21)CC)OCC N1(C(CC2ON=C(C)C2)=O)CC(NC(=O)Cc2csnn2)C(CC(C)(C)C)C1 C(C(C)(O)CC(=O)N(CCC(N1CC(O)CC1CO)=O)CCCO)OC N1(C(C2C(OC)C2)=O)CCC2OCCN(C(=O)CC3(C)OCCO3)C2C1 C(=O)(C1=CCS(=O)(=O)C1)NC1C(NC(c2oc(CC)c(C)c2)=O)CC1 CCCC(C)(O)CC(=O)NCC1CCC1C(=O)Nc1cccc(C)c1CO C(=O)(C(CCC1CC1)NC(=O)C=Cc1ccc[nH]1)NC(C)C(F)F C(=O)(C(CC)C(=O)OCC)OCCC(Cc1cn(C)cn1)NC(=O)CC C(=O)(CC(C)CN(C)C)NC(C(=O)NC(C(=O)NC)CC1CCC1)(C)C c1(C(=O)NCC23CC(CN2C(=O)CC2CCCCCC2)C3)cccc2sncc12 Cc1ccc(C(CNC(C2CC2(C)C)=O)NC(c2n[nH]c(C)c2C)=O)cc1 N1(C(c2cc(CC)no2)=O)CC(NC(c2cccc(OC)n2)=O)C(N=[N+]=[N-])C1 c1(C(=O)NC2CC(C)N(C(=O)C=CCN3CCCC3)C2)cc(Cl)cnc1O c1(NCC2(CNC(C3CCCN3C(CC(=C=C)C)=O)=O)CC2)cccc2c1ncn2C c1(C(N(CCN(C(CNC(=O)OCC=C)=O)C)C)=O)cccc2c1C(C#N)C2 CC1(C)CN(C(C2CCc3nn[nH]c3C2)=O)CC1C(=O)NC1CC2CC2C1 Cc1cnc(C(=O)N(C2CN(C(c3nnn(C)c3N)=O)CCC2C)C)cc1Cl C1(O)(CNC(c2cn(CCF)nn2)=O)CCN(C(C2(CC(F)(F)F)COC2)=O)C1 c1(C(CC)(F)F)ccccc1NC(=O)C(=O)NC(CNC(=O)C(F)OC)CO C1(NC(CCCOC(C)C)=O)CN(C(c2ccc(Cl)nn2)=O)CC12CCOCC2 C(=O)(C(O)C(C)CC)NCc1ccc(-c2cccc(NC(CCC)=O)c2)cn1 CN1C(C(=O)NC2CN(C(c3c(C(F)F)nn(C)c3Cl)=O)C2)CCS1(=O)=O C1(C(=O)NCCNC(c2c(CC)csc2)=O)Cc2ccc(F)cc2O1 C1(S(N)(=O)=O)(C(=O)NCC2N(C(CCCOCCC)=O)CCC2C)CCC1 c1(C(=O)NCC2CCCN2C(=O)CSc2ccccc2)ncc2c(F)cccn12 Cc1cc(NC2CCn3ncnc3C2)ncc1S(=O)(=O)N1CCC=C(Cl)C1 C1(CC(C)NC(=O)COc2cn[nH]c2)CCCN(C(=O)C(O)Cn2cncn2)C1 CCC(CC(=O)N1CC(C(=O)NC2(C)CS(=O)(=O)C2)(COC)C1)OC N1(C(c2n(C(C)C)ccn2)=O)CC(C)C(NC(c2c[nH]c(=N)s2)=O)C(C)C1 C(=O)(C1=CNS(=O)(=O)N=C1C)N1CC2CC(NC(c3n(CC=C)ccc3)=O)C2C1 Cc1ccccc1C1(C(N2CCC(C(C)(C)NC(=O)CC3CCOC3)C2)=O)CC1 c1(NC(=O)NCc2ccc(CCOC)cc2)cccc2ccc(Cl)nc12 N1(C(C(N2C(C)C(C(F)(F)F)CC2)=O)=O)CCc2cc(C(C)(C)C)ccc2C1 C1(CC(=O)N(CC(C)(C)NC(C(C)=CCC)=O)C)CCC1(C)C C1(C)(C(=O)NCCN(CC(C)O)C(c2ncccc2F)=O)CCC(C)(C#N)CC1 C1(NC(C2C(OCC)C2)=O)CC(C)CN(C(=O)C=Cc2cncs2)C1.c1ccccc1 C1(CCC(=O)NCc2cn(CC#C)nn2)CCCCN1C(=O)C(O)COC c1(C(N2CCC(NC(C(C)(CO)OC)=O)C2)=O)c(F)ccc(C)c1Br N1(C(C(=O)NCCCCCC)CCCOCC)CCN(S(N)(=O)=O)CC1 C(=O)(C(CCC(C)C)NC(=O)C=Cc1ccsc1)NC(c1nc(C)oc1C)C CC(C)CCC(=O)C(=O)NCC(O)C(=O)NCC(N1CCCCC1)C C(=O)(C1=CCN(C(C2CCCC(=O)N2)=O)C1)NC(CCN(C)C)(C)C Cc1ccc(S(=O)(=O)N2CCC(CC(N3CCC4(C3)CC4(F)F)=O)C2)cn1 c1(Nc2ncnc(C)c2Br)ccc2c(c1)nc(O)n2C#N C1(CNC(CCC(C)OC)=O)CN(C(c2cnc(CC(C)C)s2)=O)CCC1(F)F N1(C(Cc2cn(CC)nc2)=O)C(CC(=O)NC2CCN(C)C2)C2CCCC12 C1(NCc2c(OC)cc(C)s2)CN(c2cc(C)nc(C3CCC3)n2)CC(C)(C)C1 CC1(C)CCOC(CC(=O)NC2CC3C2CCN3C(=O)CCc2nncs2)C1 C(CC(C)(C)C)(C(=O)NCCC1CC(C(=O)Nc2nc(N(C)C)n[nH]2)C1)OC N1(C(CC2C(C)(C)C2)=O)CCN(C(c2cccc(C(F)F)n2)=O)CC1 N1(C(C2C(CCOC)C2)=O)CCC(C)(C)C(CNC(C2CC(=C3CCC3)C2)=O)C1 C1(C(=O)NC(c2cnc[nH]2)C)CCCCN1C(=O)C=Cc1ccncn1 C(CCF)(C(=O)N(C1CCSC1)C)NC(C(C)OCC=C)=O N1(C(CC)=O)CCC(C(=O)NC2CCN(C(C3CCCOCC3)=O)C2)CC1 C1(NC(C2C(C)(C)CC2)=O)CC2(CCN(C(=O)C3=CCCS3)CC2)C1 N1(C(=O)Nc2nc(C)c(C)s2)CCOC2(CCSC2)C1 c1(C(=O)NC(C(C)C)CNC(C2CN(C(N)=O)C2)=O)ccnc2ncnn12 c1(C(=O)NC(CC(=O)NC(CC#C)CO)C2CC2)cccc2ccoc12 c1(C(=O)NCC(CC)(C)NC(=O)COc2ccc(F)cn2)cn(C)nc1C(F)F C=CCC(CC=C)C(=O)NCC1CCC(C)CN1C(c1coc(C2CC2)n1)=O N1(C(C)C)CCC(CC(N2CCC2CNC(C2(F)CCOC2)=O)=O)C1 N1(C(c2c(CC)c[nH]n2)=O)CCC2(CCCC2NC(C2(C)CC2)=O)C1 c1(-c2cn(-c3cc(C)cc(C)c3)nc2)n[nH]c(=NC2CCC(C)C2)o1 c1(C(=O)NCC2N(C(c3c(C)ncn3O)=O)CCC2)cc2c(nn1)CCCC2 CCC(C)CCCCC(=O)NC(C)CC1CN(c2nnc(C#N)s2)C1 c1(C(=O)NC2C(C)N(c3ncc(Cl)cn3)CCC2)ccc(S(C)(=O)=O)o1 CC(C)C(C)(O)C(=O)NCC1CN(C(C2CC(F)(CO)C2)=O)CCO1 c1(CN2CCN(c3c(OC)cnc(SC)n3)CC2)cccc2c1sc1ccccc21 C(=O)(C1CCSc2ccccc21)NCCN(C(=O)C(C(C)C)NC(N)=O)CC CC(CN=c1[nH]c2ccc(S(=O)(=O)NCCCn3cncn3)cc2s1)N(C)C CC(F)(C(=O)NCC1CC1CNC(=O)CCc1cccc(F)c1)C(F)(F)F c1(C(C)=O)ccc(C(=O)NCc2ncc(C(N3CC(O)(c4cc[nH]n4)C3)=O)o2)o1 C(=O)(CCC(=O)N1CC(N(C(=O)CC2CC2C(F)(F)F)C)C1)NC C12(NC(C(c3c(C)n(C)nc3)N)=O)CCCC1CCC2 N1(C(C(C)O)=O)CCCC(C2CCN(C(c3c[nH]c(=N)nc3O)=O)C2)C1 CC(CN(C)C)CC(=O)NCC1(NC(=O)CP(C)(C)=O)CC(OC)C1 c1(C(=O)NCCC2CCN(C(C(CC#C)O)=O)CC2)c(F)ccc(OC)c1Cl Cc1ncc(C(=O)NCC(CC2CC2)C(=O)NC[Si](C)(C)C)c(C)n1 N1(C(C(CCC)OCC)=O)C2CCC1C(CNC(c1ccnc(C3CC3)n1)=O)C2 C1(NC(c2c(C)nncc2)=O)CC2CCC(C1)N2C(=O)CC1CCC(C)(O)CC1 N1(C(C(=O)N(CCc2nccn2C)CC)=O)CCCC(C2CC2)CC1 C(CC(CC)C(=O)NCC(C(=O)N1CC2(C1)CN(C)C2)C(C)C)=CC N1(C(C2CCN(CC)C2)=O)CCC2(C1)CN(C(C1CC(F)(CO)C1)=O)C2 c1(C(=O)NCC(CNC(CNC(=O)OC)=O)(C)O)ccc(OC)c(C(F)F)n1 CC(C)CC(C)(C)CNC(C1CCC(C)CN1C(=O)CNc1ccccn1)=O C1(NC(C2(OC(C)=O)CC2)=O)CCCCN(C(=O)C(C)C(=O)c2cccnc2)C1 N1(C(C=C(C)C(C)C)=O)CC(NC(=O)CCCc2nncn2C)CC(C)C1 CC(C(=O)NC1(CNC(c2cc(-c3ccc(Cl)s3)on2)=O)CC1)C(C)(F)F C=C(C)CC(C(=O)N(C)CC1CCN(C(=O)CN2CCOCC2)C1)NC(C)=O Cc1nnc2n1CC(C(N1CCCCCC1CNC(=O)CC(C)(C)F)=O)CC2 CC1OCCC1CC(N1CC(CCCCNC(C2(n3cc(Cl)cn3)CC2)=O)C1)=O Cn1c(C(=O)NC2CCCCC2NC(c2cc(=N)[nH]c(Cl)n2)=O)cc2occc12 c1(CC(=O)NC2CCCN(C(=O)CNC(c3ccncc3)=O)C2)ccc(Cl)cc1 N1(CC(=O)NCC(C(C)C)NC(C2(n3cnnn3)CC2)=O)CCC(C)(C)C1 c1(C(=O)NCCN(C2CC2)CC)coc(C2CC2)n1.C1(C=O)CCC(F)C1 N1(C(C(C)CC2CC2)=O)CCN(C(c2ccn3c2CCCC3)=O)CC(C)(C)C1 CC1CC(C(=O)NCc2ncco2)CN(C(=O)C(O)Cn2cncn2)C1 C1(C(N2CCCC2CCCNC(c2cocn2)=O)=O)(COC)CC=CCC1 N1(Cc2c(C)nn(C)c2)CC2CC(C1)N2C(=O)Cc1ccccc1F c1(OC)cc(NC(=O)CNC2CC(C(F)F)C2)ccc1C(F)(F)F Cn1cc(CC(N2CC(C)(C(=O)NC3CC(=C4CCC4)C3)C2)=O)cn1 c1(C(=O)NC2CN(C(C(N)=O)=O)CC(O)C2)cccc2ccc(Br)nc12 O=C1CN(CC(N2CCC3(CC2)CN(CC(F)(F)F)C3)=O)C2CNCC2N1 CC1(C)CN(C(=O)CCOC(=O)NC2CC2)CC(CC(N)=O)O1 c1(C(=O)NC(CC=C)CNC(=O)CC(C)(C)CN(C)C)cnn2c1CC(F)(F)C2 c1(NC(CC2(NC(C3C(C)=C3)=O)CCC2)=O)cnc(C)c(C)n1 C1(C)(C(N(CCCCC)CCO)=O)CCN(C(=O)CNc2ncccn2)C1 N1(C(C2(C)CC=CC2)=O)CCCC2C(NC(C3CC(F)(CO)C3)=O)C(C)(C)C12 N1(C(C2(C=C)CCC2)=O)CCCCC1CN1CCN(C(=O)Cc2cc[nH]n2)CC1 C(=O)(N=S1(=O)CCC2(C1)NC(=O)NC2=O)c1cc(OC)c(F)cc1F N1(CCNC(c2c(C)coc2)=O)CCCN(C(c2onc(C)c2C)=O)CC1 c1(C(=O)NC2CC(NC(=O)CCc3ccsc3)C2)ccc2nc[nH]c2c1F C1(NC(C=CCN(CC)CC)=O)CCCN(C(=O)Cc2csc(C(C)C)n2)CC1 C1(CC(=O)NCC2CCN(CCC)C2)CCCCN1C(c1ccn(C2CC2)n1)=O C(=O)(CC(C)CC(C)(C)C)NCCCOCCC(=O)N(C)CC1C(C)C1 c1(C(=O)NC(C)(CNC(=O)C(F)C2CC2)CO)cc(Cl)cc(Cl)c1O C(Cn1cccn1)(C(=O)NCCCCN1CCCC1)NC(=O)CCC1OCCO1 n1(CC(N2C(C)CC(NC(c3ccccn3)=O)CC2)=O)c(=O)oc2ccccc12 CCCCC(C(=O)N1CC(F)(C(N)=O)C1)NC(C1CCN1C)=O N1(C(C2C(C(C)(F)F)C2)=O)CCCC1(C)CNC(C1CCC(C(F)(F)F)O1)=O N(C(=NCCCCC(F)(F)F)NC(C)COC)Cc1c(CC)onc1C N1(C(C(C(CC)(C)CC)F)=O)CCC2C(CCCN2C(=O)C=C2CCC2)C1 c1(C(=O)NC2(CNC(CC(C=C)C)=O)CCOCC2)cc(NC)ccc1Cl CCC(CC(=O)N1C(C(=O)NC2C(=O)OCC2CO)CC2CCCC12)CC(C)C C=CCC(CC=C)C(=O)NC(CNC(c1cc(OCCOC)n[nH]1)=O)C(C)C(C)C C1(C)(CNC(c2c(C)onc2C(F)(F)F)=O)CCN(C(C2CNC(=O)C2)=O)CC1 N1(C(C2C(=C)C2)=O)CC2CCC(CNC(c3c(C)nsc3N)=O)C2C1 CC1C(NC(=O)C=CC2CCCCC2)CCCN1C(C1CCC(O)C1)=O N1(C(c2ccn(CC)n2)=O)CCOC(CN(C)C(C2CCC(=O)NC2)=O)C1 c1(C(N2CCC(NC(C34CCOC(CF)(C3)C4)=O)C2)=O)c(F)ccc2[nH]ccc12 N1(C(=O)OC(C)(C)C)CCN(C(N(N2CCOCC2)C(C)C)=O)CC1CO Cn1cnc2c1CCC(NC(C1CN(C(=O)CSC(C)(C)C)CC1C1CC1)=O)C2 N1(Cc2c(C)ccc(F)c2)CC2CC(NC(C3CCCOC3)=O)CC2C1 c1(C(N2CCC(N(C(=O)CC3CCOC3)CCC)C2)=O)sc(C(C)OC)nc1C CCCC(C)(C)C(=O)N1CC(CCCCNC(c2cc(Cl)ncc2F)=O)C1 C(C)(C(C(=O)N1CCOC2CCCC12)C(C)C)NC(CCC=CCC=C)=O C1(C(=O)NC2CN(C(C)C)C(=O)C2)(CO)CCc2ccccc2O1 Cc1ccc(C(=O)NCC2CCCN(C(c3snc(O)c3Cl)=O)C2)cc1C CCC(CC)(CO)C(=O)N1CC(NC(c2ccn(CC(F)F)n2)=O)CC2(CC2)C1 n1(CCC)nccc1C(=O)NC(c1ccccc1)C(=O)N(C)CCc1cnc[nH]1 N1(C(c2cc([N+](=O)[O-])cnc2O)=O)CCC(c2nn[nH]n2)C(F)(F)CC1 Cc1ncnc2c1CC(C(N1CC3CC1CN3C(c1cc(O)n(C)n1)=O)=O)CC2 c1(C(=O)Nc2cc(N3CCOC(CNCC)C3)nc(C)n2)cnc2ncccn12 C1(C(=O)NC2CC3CN(C(C=C(C)C(C)C)=O)CC2C3)CCc2nnc(C)n2C1 N1(C(c2ccn(CC)n2)=O)CC(NC(C2CCCCN2C)=O)C2CCCC2C1 C(CCN=C(NCC(N1CCOCC1)C)NC1CCCC(F)(F)C1)OC c1(C(=O)NCC(CC)NC(c2cnc(C(C)(C)C)nc2)=O)c(O)ccc(Cl)c1O c1(C(N(CCC(C)NC(c2c(CC)nccc2)=O)C)=O)ncc2ccccn12 Cc1cc(C(N2CC(NC(=O)CCCNC(N)=O)C(O)C2)=O)nnc1O CCCC(C)(O)C(=O)N1CCN(Cc2cn(CC3CC(F)(F)C3)nn2)CC1 CC1CN(C(C2COCCN2C=O)=O)CCN1C(C1CCCO1)=O c1(CC(=O)N(CC(C)O)CCNC(=O)CC2CN(C)C2)ccc(Cl)cc1Cl C1(OC)CC(NC(=O)CN2C(=O)CCC2=O)CN(C(C2CN(C)C(=O)N2)=O)C1 C1(C)(C(N(C(C2CCCC2)CNC(c2ccnn2CC2CC2)=O)C)=O)CC1(F)F CC(C)CCCC(C)C(=O)N1CCCC1CNC(c1cccnc1OC(C)C)=O n1(CCCC(=O)N(C)CC2(O)CN(C(C3(C(C)C)CC3)=O)C2)ccccc1=O c1(C(=O)NCCOC2CN(C(c3c(C)cnn3C)=O)C2)ccn(C(C)C)c(=O)c1 C(CC(C)C)(C(=O)Nc1nnc(C#N)s1)NC(CCNC)=O c1(CNC(c2n(CC(=C)C)nnn2)c2nocc2Br)ccc(C)nc1Cl c1(SCCNC(=O)C(N2CCCC2C2CC2)=O)noc2cc(F)ccc12 C1(C(C)NC(c2nc(-c3ccco3)oc2C)=O)CCCN(Cc2cccs2)C1 c1(C(N(CCNC(c2cncc(NC)c2)=O)C2CC2)=O)cc([N+](=O)[O-])ccc1Cl C1(C#N)(COC)CN(C(c2cc(CCNC(=O)C=CC(C)C)on2)=O)C1 C=CCCN=C(NCc1nn(-c2ccccc2)c2c1COCC2)NC(C)C c1(CNC(C2CCCCO2)CC)cscc1C(=O)O N1(C(c2cc(C)c(Br)o2)=O)CC(NC(=O)CC2(O)CC2)CC12CCC2 C12(NC(C3CCC(c4cn(CCCCCC)nn4)C3)=O)CCCCC1OCC2 N1(C(CC)=O)CC(NC(=O)C(C)(C)C2CCOCC2)C(CC)C1 CCC(C)(C)C(=O)N1CCOCC1C(=O)N(C)CC1CCOC1 CC1CC(C(=O)N2CCN(C(c3c[nH]cc3Br)=O)CC2c2cn[nH]c2)=NO1 C(C1C(C(N2CC(c3nccs3)C2)=O)C1(C)C)=C(C)C c1(SC)ccc(C(=O)NCC(c2ccc(CCN3CCC(CC)C3)o2)=O)cc1.N(C)C.N C(CC(C)(C)C(=O)N1CCCC1)N1CC(c2onc(C)n2)C1 c1(OC)cccnc1-c1noc(C(C)(CCc2nc[nH]n2)n2nnc(C3CC3)n2)n1 N(C(=NCCCF)NC1CCC1n1ccnc1CN1CCc2ccccc21)CC N1(C(CCC(C)=O)=O)CC=C(C(C)(C)C(=O)N2CCCC2C(C)(C)C)C1 N1(C(C2CC(CCC)C2)=O)CCCCC12CN(C(c1n[nH]c3c1CSCC3)=O)C2 CC1C(NC(c2cc(Br)c[nH]2)=O)CCCN1C(c1cc2n(c1)CCC2)=O CC1CCC(CNC(=O)CN2CCCCC2)CN1C(c1cnn(C2CCC2)n1)=O c1(OC)c(C(N2CCC(=CCNC(=O)CC3COC(=O)C3)CC2)=O)ccnc1Cl c1(C(C)C)cc(C(=O)NC2CCC2CNC(=O)CCCC2CCCCC2)no1 C1(NC(CC(C)NC(c2n[nH]c3c2COC3)=O)=O)CCc2c[nH]nc2C1 c1(C2CCN(C)C2)cc(C(N2CCC3CC23C)=O)cnn1 c1(CC(=O)N(CC(C)NC(C2(CCC)CC2)=O)C)cc2ccccc2cc1O S(=O)(=O)(c1ccc(NCC2CCC(F)C2)c(Br)c1)NC1CC2(C)OCC1C2 c1(C(N(C2CCN(C(=O)C(C)N3CCC3)C2)CC#C)=O)sccc1F CC(C)C(CNC(c1ccc(C#N)[nH]1)=O)C(=O)N(C)CC1CCSC1 N1(c2cc(C#N)ncn2)C(CNC(c2csc3nnsc23)=O)CC2COCC12 C(=O)(CCS(C)(=O)=O)N1CC=CC(SC(C)(C)C(=O)NCc2ccccc2)C1 N1(C(C(C)C2CCC2)=O)CC2CCN(C(C3COC4COCC34)=O)CCC2C1 c1(C(N2C(CNC(C(F)OC)=O)CCC2)=O)cc(C(C)(C)C)ccc1O C1(CNC(CCCCC=C)=O)CN(C(=O)CCCNC(=O)C2CC2)C2CCN1C2 C1(C(=O)NCC(CC)C)CCN(C(=O)c2ccc(CO)cn2)O1 CC(CC1CCC1)C(C(=O)NCC1CCCO1)N1CCC(C2CC2)OC1 Brc1ccc(C2(CNc3nccc(I)n3)CC2)nc1 c1(C(N2CC(NC(C34CC(F)C3C4)=O)CC(C)C2)=O)cccn2cncc12 c1(C(=O)OCC)c(C)sc(N(NC(=O)NC2CN(C3CC3)C2)CC)c1C c1(C(=O)NCC(CC=C)NC(=O)CCOCC)cnc2n1CCC(C)C2 C(=O)(C1=C(Cl)CCOC1)N1C(C(N2CCC(C)(C(=O)NC)C2)=O)C=CC1 O=CS(=O)CCc1cn(NC(C2(CC3C(Cc4ccccc4)C3)CC2)C2CC2)nn1 C(=O)(C(C)(C)C(N)=O)NC(CC1CN(c2snc(SC)n2)C1)C N1(C(=O)OC(C)(C)C)CC(C(F)(F)F)OCC1CNC(C1(C)CCCC1)=O c1(C(N2CC(CNC(C(C(=O)OC)C)=O)C2)=O)cc(N(C)C)ccc1Br C(CNC(c1cccnc1OCCO)=O)(C(C)(C)C)NC(Cn1nnc(C)n1)=O c1(C(=O)NCCSC)c(F)cc(F)c(F)c1N C1(NC(CC2N(C(CCc3cnc(C)o3)=O)CC2)=O)CCCN(C)C1C C1(C(C(=O)NCC(C2CCCC2)NC(C2(OC)CCC2)=O)OC)CC(F)(F)C1 C1(NC(CCc2cc(C)[nH]n2)=O)CN(C(=O)Cc2cscn2)CC1C C=CCC(CC(C)C)C(=O)NCCN(CCOCC)C(c1ccc(OC)nn1)=O O=C(C1=COCCO1)NCC1CCCCN1C(=O)Cn1cnc(C(F)(F)F)c1 c1(CC)ccc(C(=O)NC(C(=O)N(CC(C)O)C)C2CCCC2)nc1 C1(C(C)NC(COC(C)C)=O)CCCCN1C(=O)Cc1cnn(C)c1 Cc1ccc(C)c(C(N2CCC(NC(c3sccc3CN(C)C)=O)C(C)C2)=O)c1N C(=O)(CCCCCc1cccs1)NCC1(N(C)C(C2CCC3CC3C2)=O)CC1 N1(C(C=C(CC)CC)=O)CC(NC(=O)CCCCNC(N)=O)C2(CC2)C1 CCC(C)(C)C(C(=O)N1CCCC1CN(C)C(c1cnc(O)c(F)c1)=O)OC N1(C(c2c(C)sc(Cl)n2)=O)CCCCC(NC(C2(C)CCCOC2)=O)C1 C1(C(=O)NC(c2ccc(F)cc2)C2CCC2)CC2(CC(NC(C3CC3)=O)C2)C1 CC(C)(O)C(F)C(=O)N1CCCCC1CNC(c1ccc(Cl)nc1N)=O N1(C(Cc2cc(OC)no2)=O)CCC(NC(=O)CCc2cn(C)nn2)C1(C)C C1(NC(C=CC(C)(C)NC(=O)CCc2cscn2)=O)CCn2cnnc2C1 C1(C2CC2)(CNC(C(CC)N(C)C)=O)CCN(C(=O)CCOCC(F)F)C1 Cc1cc(F)ccc1C(F)(F)C(N1CCC(F)C(NC(C2CC(C#N)C2)=O)C1)=O C=C1CCC(C(=O)NCCN(C(=O)CNC(c2ccc(OC)cn2)=O)C)CC1 c1(C(N2CC(F)CC(NC(C3CC(C#N)(OC)C3)=O)C2)=O)c(C)cc(Cl)cc1C C(=O)(C(F)C(F)(F)C(F)(F)F)N1C(CNC(c2onc(C)c2C)=O)C=CC1 C1(F)(C(N(CCCO)CC#C)=O)CN(C(c2cc(F)c[nH]2)=O)C1 C(C)(C(C(=O)NCCC1CCSC1)NC(=O)C(F)C(C)C)OC C(=O)(C1OC(=O)c2ccccc21)N1C2CC(CC(NC(C(C)NC=O)=O)C2)C1 c1(N2C(C)(C(N3CCCC(C)CC3)=O)CC2)cc2ncnn2cn1 C1(CCCCNC(C=C(C)C(C)C)=O)CCN(C(=O)Cn2cc[n+](C)c2)CC1 c1(N2CC(OC)(CNC(C3CC3(C)C(F)F)=O)C2)cc(C(C)C)nc(C(C)C)n1 C=C=CCCC(=O)NC(c1ccnn1C)C(=O)NC12CC(C1)C2 C1(CC(CNC2CC(N)C2)O)CCCCC1 C(C(C)C)(CC(C)C)C(N(CC(C1(O)CCCOC1)(C)C)C(C)=O)=O CCC(C)(CO)C(=O)NC(C)(C)C.C123CN(C(C(=O)OC)(C1)C2)C(=O)OC3 c1(C(=O)NC(CN(C)C)(C)C2CC2)ccc(NC(=O)C(O)C(F)F)c(F)c1 C1(C(=O)NCC(CC(=O)NC(CCOCC)C)OC)CC(=O)N(OC)C1 CC1=C(C(=O)N2CCC(C3CCN(C(=O)CC#N)CC3)C2)C(C)n2ncnc2N1C c1(C(=O)NCC2(O)CC(CNC(c3nc(C)sc3)=O)C2)nnc(O)nc1O CC(C)C(F)(CNC(=O)CCNC(=O)CO)C(=O)NCC(C)(O)C(C)(C)C Cc1nc2c(s1)CCCC2C(=O)OC(C)(C)C.C12CCN(C1C(=O)O)C2=O C(=O)(CS(=O)(=O)CCO)N1C(C)CN(C(=O)C=CC2CCCO2)CC1 C1(C(=O)N(C2(CNC(=O)CN3CCOCC3)CC2)C)(OC)CC(C)CC(C)C1 C12(CNC(=O)Cn3cnnc3O)CCCN(C(c3ccoc3Cl)=O)C1C2 CC1CN(C(=O)C(=O)NCc2nnc(C(C)(C)C)s2)CCC1(F)F C1(NC(C(N2C(COC)CCC2)=O)=O)CC2CN(c3nc(C(F)(F)F)ns3)CC12 C1(C(=O)NCC2(CCC)CC2)(CNC(=O)C=C(C)C(C)C)CC(C)(C)C1 c1(CC(=O)NC(C2CCN(C(=O)C(c3ccccc3)C)C2)C#C)ccc(Cl)cc1 C(CCN=C(NN1CCOCC1)N1CCC(C)(CN(C)C)C1)OCCOCC C(=O)(CC(C)(C)CC(=O)NC1CC1CNC(c1cc(Br)c[nH]1)=O)OC CCC(C)(CC)C(=O)NCC1CCC(C)N(C(c2cc(-c3ccco3)on2)=O)C1 C1(NC(C(CSC)(C)C)=O)CN(C(C2(OC)CCCOC2)=O)CC(C)(C)C1 N1(C(c2scc(OC)c2)=O)C2CCC1CN(C(C1CC3OC1C1CC31)=O)C2 C1(NC(CS(CC)(=O)=O)=O)CCN(C)C12CCCN(C(C1(O)CCOCC1)=O)C2 C1(F)(C(=O)NC(CNC(c2nc(C)[nH]n2)=O)C2CCC2)CCCN(C)C1 N1(C(CSc2ccc(OC)cc2)=O)CC2CC1CN2Cc1ccn(CCF)n1.C1(CN)CC1 C1(CC)CNC(=O)C(C)(C)C1.C(=O)(C(C)(C)C(=O)NCCNC(=O)OC)NC(C)(C)C N1(C(C)C)CCC(CNC(=S)Nc2ccc(-c3cn(CCC(F)(F)F)nn3)o2)C1 c1(C(=O)NC2C3C(C)N(C(=O)CCC4CC(F)(F)C4)C2C3)ccc2nccn2n1 Cc1cc(CNC(=O)C(CC2CCOCC2)NC(=O)CCC2CCOC2)c(C)s1 N1(C(C2(COC)CCCO2)=O)CC=C(CNC(C2CCCC(OC)C2)=O)CC1 C1(N(C(C(C)N(C(C)=O)C)=O)C)CCCCC1N(C(=O)CCN1CCOCC1)C c1(C(=O)NCC(CO)NC(c2scc(C)c2)=O)cccc(Cc2nnc(C)s2)c1 N1(C(C=CCC)=O)CC(O)(C(C)(C)CNC(c2c[nH]c(=N)s2)=O)C1 C1(C)(C(=O)NCC(C(=O)NC)O)CC(NC(=O)C=C(C)C)CCO1 c1(C(=O)OC)cc(NCCC2CCCC3CC23)c(F)cc1Br N1(c2cccc(C(=O)OC)c2)C(=O)NC(C(c2ccccc2)C)C1=O N1(C(CC(CC)C2CC2)=O)CCC(NC(c2ccc(C)cc2C)=O)C1(C)C c1(C2(NC(=O)NC(CC(=O)OCC)c3ccccn3)CCC2)ccc(Cl)cc1 Cc1nn2c(C(F)(F)F)c(NC(=O)CCC3CCNC(C)(C)C3)nc2s1 c12nc(OC)cc(n1)N1CCCN(CC1)CCN2.C1(C(=O)OC)CCOC(C)C1 C1(C(=O)OCC)CCOC2(CCN(C(c3c(C)nn(C4CC4)c3C)C)CC2)C1 C=Cc1cnn(C)c1C(N1CCN(C(=O)C(C)OCC)C(CC2CC2)C1)=O c1(C(=O)NC2CCN(C(C(CC(=C)C)OC)=O)C2C)cc(C#N)ccc1C C1(C(ONC(c2cn(CCOc3ccc(O)cc3)nn2)=O)=O)C2C3CCC(C3)C12 CC1CCCCC1(CO)NC(c1ccc(NC(=O)C(C)(C)c2cscn2)nc1)=O N1(C(C(N2CCC(C)C2)=O)=O)CC=C(CCNC(C2(C)COCCO2)=O)CC1 Cc1nn(C)c(=O)c(C(=O)NC2CCC(CNC(=O)CCCCC(F)F)C2)c1C c1(C(N2CC(NC(C3CN(C)C3)=O)C3(C2)CC3)=O)ccc2nc(O)nc(S)c2c1 C(CNC(=O)CC(c1ccc(C)nc1)N)(CC(C)(C)C)OC c1(C(C2CCCC2)=O)cccc2c1ccn2-c1ncccn1 CC1CC(CC(=O)NCc2ncccc2Cl)CN1C(=O)CCc1cnn(C)c1 c1(N)ncccc1OCC(F)(F)F.c1(C2(C(N(CC)CC)=O)CCC2)ccn(C)n1 C1(F)(C(=O)NCC2C3CN(c4cc(CC)ncn4)CC32)CCC(C)CC1 c1(C2(C(=O)NC3(CO)CN(C(CCC=CCC=C)=O)C3)CC2)cc(F)ccc1C Cc1cccc(O)c1C(N1CCCC(CN(C)C(c2cc(O)ccc2I)=O)C1)=O C(=O)(CCCC(C)O)N1CC=CC(NC(c2cn(CCC)nc2)=O)C1 C12(NC(C3C(N)C=CCC3)=O)CCOCC1CNC2 C1(NC(c2n[nH]cc2Cl)=O)CN(C(c2n[nH]cc2-c2ccccc2)=O)CCC1O N1(C(C2(C(=O)OC)CC2)=O)CC2(C1)CN(C(=O)C(C)CC(F)F)C2 c1(C(N2CC(NC(C3(C(F)F)CCCO3)=O)C(O)C2)=O)ncn2c1COCC2 c1(NC(C)C)ccccc1S(C)(=O)=O.C12CN1CC2c1ccccc1 c1(CC(=O)NCCCCCNC(c2nc(COC)oc2)=O)ccc2c(c1)CCC2 C1(C(C)C)CCCC2(CN(NC(C(CCOCC)C)=O)C2)O1.C12CC1C2 C(=O)(C(C)(O)CC(C)C)N1CC2CN(OC(C34CC(CC)(C3)C4)=O)CC21 c1(-c2cc(C(=O)Nc3cc(OC)c(OC)cc3)ncc2)cnc2[nH]cnc2c1 N1(C(CCCCCSC)=O)CCC2CN(C(=O)C(c3cncn3C)O)CCC12 C(=O)(C1=CSCCO1)N1C(C(C)(C)NC(C=CCN(C)CC)=O)CCC1 CCCCC(CCCC)C(=O)NCCOCCCNC(=O)CCP(C)(C)=O c1(CC)ccc(C)c(C(=O)NC(C)CC(C)CC)c1 c1(C(=O)NC(CCCCNC(c2c(C)csn2)=O)C)scc2c1CCCC2 c1(NC(=O)CC2CC2CNC(C=C(C)C2CC2)=O)ccc(Oc2ccsc2)cc1 Cc1cccc2c1C(NC(=O)C(C)OCC(C)C)CCC2 C#Cc1ccc(F)cc1C(=O)NCCN(C(=O)C(C)CC(N)=O)CC1CC1 C1(CNC(C(COC)O)=O)CC2CC1CN2C(c1cn(C(C)C)cc1C)=O c1(CN(CC(C)C)C(=O)NCC2CCC(F)C2)nc(O)nc(O)c1F C12(N)COC(CN)(C1)C2.C1(N(CC(=O)OC)C(C)=O)CCN(C=O)C1 N#Cc1cccc(C2CCCN(C(c3ccccc3)C(N)=O)C2)c1 CC1C=C(C(=O)N(C)CC2CCCN2C(=O)CCCSC(C)(C)C)CC1 N1(C(CC)CC)CC(C(N2CCCC2CNC(C2(SC)CC2)=O)=O)CC1=O c1(C(=O)OC)c[nH]c(C)cc1=NC1CCCCN(C(=O)C2=CCCC2)C1 C12(CNC(c3c(C)c(CO)ccc3)=O)CN(C(c3ccncc3)=O)CC(F)(C1)C2 C(=O)(CCCCCCSC)N1CC(c2nnnn2CCCF)(C(=O)NC)C1 C(=O)(C(C)CS(C)(=O)=O)Nc1c(CC=C)nco1.N12CCC(C=C)(C1)C2=O C(=O)(C(CNC(=O)CCC(C)CC)CC(C)C)N(CCOCC)CC Cc1cccc(C(N2CCOC(C(C)NC(=O)C(CO)NC(N)=O)C2)=O)c1C C=C=CC(C)C(=O)N1CCCC1CN(C(c1cc(C)c[nH]1)=O)CC c1(C(=O)NC(CNC(C2(C)ON=C(C)C2)=O)(C)C(C)C)ccn2c(C)cnc2c1 c1(C(=O)NCC(C2CCC2)NC(c2cc(COC)sc2)=O)ccncc1O N1(C(c2ccc(CC)s2)=O)CCCCC(NC(=O)CCCC(C)C)C1 c1(C(N2CC3(C(C(=O)Nc4c(C)noc4)C3)C2)=O)cnn2cccc(F)c12 c1(C(=O)NC2CC3(C(NC(CCC(C)SC)=O)C3)C2)ccc2cncn2c1C CC(C)C(COCc1ccccc1)NC(C1(CC(=O)NCCCN(C)C)CC1)=O [N-]=[N+]=NCC(C(=O)NCc1c[nH]nc1C(=O)O)NC(=O)CC12CCC(CC1)C2 C1(NC(c2ccc(CC)[nH]2)=O)CC(CC(=O)NCC(C)(F)F)C1(C)C n1(C(N2CCN(CC(c3ccccc3)O)CC2)C)cnc2cccnc12 C(=O)(C(C)CCC(C)(C)C)NC1(C)CN(C(c2ccc(C(=O)OCC)cc2)=O)C1 C1(NC(c2cn(CCC)nn2)=O)CC1C1CCCN(C(c2oncc2CC)=O)C1 C(=O)(CC=C(Cl)Cl)N1C(C(=O)NC(c2cccnc2)CC)CC1C c1(CSCC(=O)NCCC(=C)CNC(c2csc(=N)[nH]2)=O)cc(C)n(C)n1 c1(CNC(c2cccc(CSCC(=O)OC(C)(C)C)n2)=O)c(F)cc(Br)cc1F C#Cc1cc(C(=O)NCC2CN(C(c3ccc(C)cc3SC)=O)C2)ccc1C CC(C)(C)C(O)C(=O)N1CC(NC(=O)C(O)c2ccco2)CC(F)C1 CCC(C)(C(=O)NCC1CC(O)CN1C(c1sc(C2CC2)nc1C)=O)C(N)=O c1(NC(C2CN(C(=O)C(F)OC(F)(F)F)CC2F)=O)ccc(Br)cc1F c1(CC(=O)NCC(CN(CCOCC)C)(C)C)ccccc1NC(C(C)OC)=O C1(NC(=O)C(O)Cc2cnc[nH]2)CC2C1CCN2C(c1cnns1)=O C1(NC(C2(C)CCC2)=O)CCCC(NC(=O)CN2CCOCC2=O)CC1 C1(NC(C2CC3CC3N2Cc2ccnn2-c2ccccc2)=O)CCS(=O)(=O)CC1 C(C(=O)C(C)(C)NC(C)(C)C)NC(=O)OCC(CC)c1cnsc1 Cc1cc2nc(C(N3CC=CC3CNC(=O)C(Cl)=CCl)=O)ccc2c(=O)n1C C1(c2n(C)ncc2)CN(C(=O)Cn2ccnn2)CCN1C(C1CCCCC1(C)C)=O C(=O)(C(CC(F)F)OC)N(CCCO)CC.C1(=O)CC(=O)SCCN1 C12(NC(c3c(C)sc(O)n3)=O)CCCC1(F)CN(C(=O)CCc1ccc[nH]1)C2 C1(OC)CC(CNC(=O)C(C)(C)C#N)N(C(=O)COc2cccc(Cl)c2)C1 c1(C(C)CNCc2cccc(NC(C3CC4C=CC3C4)=O)c2)cc(Cl)cc(Cl)c1 c1(C(=O)NCCC(C)NC(=O)CC2CC=CCN2C)cnc2cc[nH]c2c1 C1(CC(N2CC(NC(c3ccc(C(N(C)C)=O)cc3)=O)C2)=O)COCC(C)(C)O1 c1(C(=O)NCC2C(NC(C(C3CC3)OCC)=O)CCC2)ccc2oc(S)nc2c1 N1(C(C(CC(C)=O)(C)C)=O)CCC2(CCN(C(=O)Cn3cncn3)CC2)C(C)C1 C1CC(=O)N(OC)C1.C(=O)(CCOC)N1CCC1.C(C(F)(F)F)OCCC c1(N(c2nc(OC)c(C)cn2)Cc2c[nH]c(=NC)s2)cc(Cl)c(O)cc1Cl N1(C(Cc2nccc(OCC)n2)=O)CCCN(C(C2(OC)CC2)=O)CC1C c1(CCC(N2CC(CNC(c3c(CC)cco3)=O)C(O)C2)=O)ccc(F)cc1Cl C(C)(C)(C(C)CC(=O)NCC1CCN(CCF)C1)NC(CCC(C)OCC)=O C#Cc1ccc(C(=O)NC(C2CN(C(=O)C(O)C=C)CCO2)C)o1 C1(N(C(C2C(C(=O)NCc3n(CC)ncc3)C2)=O)C)CCC(OC)CC1 c1(OC)c(C(N2CC3CC2CN3Cc2cc(F)nc(F)c2)=O)cc(Cl)cc1Cl N1(C(CC2CCN(C(C=CC(CC)C)=O)C2(C)C)=O)CC2(CC(C(=O)NC)CO2)C1 c1(C(=O)NCC2(c3cc(F)cc(Br)c3)CCC2)ccc(Cl)c(N2CCCC2)n1 N1(C(CCC2N(C)CCC2)=O)CC2CC2(NC(=O)CNC(C2CCCC2)=O)C1 C1(CNC(=O)CC2CCCC2)CN(C(c2csc(-c3cnccn3)n2)=O)C2CC12 C1(CC(C(=O)NCC(C#C)CC)C)CCN(C(=O)CCC(C)OCC)CC1 c1(OC)ccccc1.C1(C2CCOC2)C(=O)N1.C12(CC1)C(=O)N2.C1(CO)CC1.C1CN1 C(=O)(C1=C(Cl)CCOC1)NC1CCN(C(C2(CC=C)CCCCC2)=O)CC1CC Cc1cc(N2CCC(C(c3ccon3)N(C)C)CC2)nc(Cl)c1C(F)(F)F CCC(CC)(CCNC(=O)CSC(F)(F)F)NC(c1cc(C(F)F)on1)=O c1(C2C(C(=O)Nc3cc4ccn(C)c4cc3)C2)cccc(C2=COCC2)c1 c1(C(=O)NC(C)C#N)cc2nc(-c3cccc4ncn(C)c34)ccc2[nH]1 N1(C(C(CC=C)OC)=O)CC2(CNC(c3oc(C(C)C)nc3C)=O)CC1CCO2 C(c1ccc(CN2C(NC(c3cccc(I)n3)=O)CC3CC23)cc1)=CC(=O)O N1(CC(=O)NCC2CC(F)(CNC(C3CC3(Cl)Cl)=O)C2)CCCCCC1 c1(C(=O)NC2(C(=O)NC(C(CC)O)c3ccco3)CC2)ccccc1OC1CC1 N1(C(c2ccn(C)n2)=O)CCC(C)(C)C1CC(=O)NCc1nccs1 c1(C(=O)NCCOC2CCN(C(C(CC=C)C)=O)CC2)ccc2c(n1)NCC2 CC(C)(C)C(CN=c1[nH]cnc(Cl)c1[N+](=O)[O-])NC(=O)COC(F)(F)F C1(C(N2CC(C3CC3)(OC)C2)=O)CC2C=CC1N(C(=O)CCCC1CC1C)C2 C=C(C)CCCC(=O)N1CCC(CF)(NC(c2cc(C)cc(F)c2)=O)C1 CCC(F)(F)CCNC(C1(F)CCN(C(C2CC(C)(C)C2)=O)C1)=O CC(C)C(O)C(F)(F)C(=O)N(CC(C)CNC(c1coc(-c2cccs2)n1)=O)C N1(C(C=CC(C)(C)SCC)=O)CCCC(NC(=O)Cc2csc(C(C)OC)n2)C1 c1(NC(C2CN(C(C3CCC(NC(CC)=O)C3)=O)C2)=O)ccc(C#N)cc1C N1(C(C(C=C=C)C)=O)CC(C(=O)NCC2CCCC(C)(C)O2)C2(CC2)C1 C(=O)(CC(C)F)NCCN(C(=O)CCNC(=O)OC(C)(C)C)CC(C)O c1(C(N2CC(C)N(C(c3ccccc3)=O)CC2)=O)c(OC(F)(F)F)cc(Cl)cc1Br C1(OCC)CN(C(=O)C(C(C)C)OC)CC1CNC(=O)CCc1csnn1 c1(C(=O)NCC2C(NC(CC(COC)(C)O)=O)CCC2)csc2c1CCCC2 C1(OC)CCC(N(C2CCCCC2)C)CC1.C12CC(C1)NC2=O CCC(C(=O)NCC1(F)CCCN(C(c2coc(C)n2)=O)C1)C(C)C C1(C(C)NC(CNS(CC2(OC)CCC2)(=O)=O)=O)Cc2ccccc2C1 c1(C(=O)NCC2CC(CNC(c3cc(C)oc3C)=O)OC2)ccn2cncc2c1 N1(C(c2c(C)ncnc2C)=O)CCC(NC(C2(C)CCOC2)=O)C(CO)CC1 c1(CC)ccc(C(C(=O)OC(C)(C)C)NC(=O)NCc2nonc2N)o1 C=CCC(C)(C(=O)NC(C)CCNC(=O)CC1CCC(=O)C1C)N(C)C N(C)(S(=O)(=O)N(C)C)CC(=O)NC1CCC(CNC(C=CSC)=O)C1 C1(CC)CN(C(C2CC(NC(=O)C(C)CC#N)C2)=O)CCCO1 C(=O)(C(C)C(C)C)NCCC1CC(NC(CSCCN(CC)CC)=O)C1 c1(OCOCC(F)(F)F)ccccc1CCOc1nn[nH]n1 C1(NC(C(C)OC)=O)CN(C(c2cc(Cl)c(F)cc2Cl)=O)CCC1(C)C N1(C(c2c(C(C)C)ocn2)=O)CC2CN(C(C3CC(O)C3)=O)CCC2(CO)C1 C(CCCCC(=O)N1CC(C)(C(=O)N(C2CCCC2C)C)C1)OC c1(CC(=O)NC2CC2CNC(=O)CSc2ncccn2)cccc(O)c1F N1(C(CSC)=O)CCC(C)C(CNC(=O)C(C)(C)c2nccs2)C1 N1(C(c2c(C)nc(Cl)s2)C(=O)NC2COC2)CCC2CCC2C1 N1(C(CC)=O)CCCCC1C(N1CCC(CNC(c2cc(C)c(C)o2)=O)CC1)=O C(=O)(CC(CC1CC1)OC)NC(COCC)C(=O)Nc1ccc(C)cc1 c1(C(=O)NCCCC(C)(C)NC(C(CC)(C)OC)=O)cccc(F)c1OC N1(C(C(C(C)C)OC)=O)Cc2cccn2CC(C(=O)NCCCCC(C)CO)C1 N1(C(c2cc(C)nc(C)n2)=O)CC(NC(=O)CCC2CCC(=O)N2)C(C2CC2)C1 C1(NC(c2c(N)cncc2)=O)C2CC3C1C3C2C(=O)NC(c1nc[nH]n1)CO C(=O)(CCC1CC1)N(C)CCOCCNC(N)=O.C(=O)(CCC1CCCO1)N C1(NC(c2cnn(C(C)C)c2Cl)=O)CC2(CCCCN2C(=O)C(F)(F)CO)C1 c1(C(C(=O)NC(C(F)(F)F)c2ccccc2)NC(=O)OCCC)ccc(F)c(F)c1 c1(C(C)(C)C)n[nH]c(=NCCCCC(C)NC(=O)C=Cc2ccsc2)s1 N1(C(COCCCC(C)C)=O)CC2CC1C2NC(C1CCC1)=O N#CC1CCCCC1N1CC2CC2C=NC(c2ccccc2)=N1 n1(CCC)ncc(C(=O)NC2CC3(C2)CC3NC(c2ccc(CC)[nH]2)=O)c1C N1(C(=O)CC2(O)CCCC2)CCCC(CCC(N2CCCC2CCCO)=O)C1 C1(CC=C)CCC2(CCCC2)C1.C1(=CC)CCCN(CCC)C1 C1(C(=O)OCC)CCN(Cc2cc(N)ccc2Br)CC1Cc1ccccc1 c1(C(CC)N(C(c2sccc2OC)C(=O)NC2(C)CC2)C)ccc(F)cc1 c1(CNC(=O)NC2(c3ccc(C)cc3)CCC2)cnn2c1OCCCC2 C1(CN(C(=O)COc2cccc(F)n2)CC)CCCCN1C(=O)C=CCF C1(C)(NC(C(c2ccccc2)OC)=O)CCN(C(c2sc(Cl)nc2C)=O)CC1 Cc1cc(CO)ncc1C(=O)NCCC(C)CCNC(=O)C(F)F.C1(C=O)CCCO1 N1(C(C=C(CC)C)=O)CCC(CC2CCOC2)CC1.C12(CC1)C(=O)N2 Cn1cnc2c1CCCC2C(=O)N1CCN(C(c2cnc(Cl)[nH]2)=O)C2COCC12 N1(C(C(N)=O)=O)CC2(NC(=O)Cn3cnc(Br)n3)CCC1C2 CCCCC(F)C(=O)N1CC(CNC(c2cc(C)c[nH]2)=O)CC1(C)C C1(C(=O)Nc2cccc(CC)c2)CC(C)(C)CCN1C(C1CC1CCOC)=O N1(C(Cc2ccc(C(=O)OC)s2)=O)CCCC(n2cc(CNC3CCCC3)nn2)C1 c12ccc(cn1)CNC2=O.CC(CC1CC1)C(=O)NC1CCOC1 c1(N2C(CNC(Cc3cc(OC)ncn3)=O)COCC2)ccc(Cl)c(Cl)c1 C(=O)(C(C)(C)C(=O)OC)NC(C)CC1CN(C(=O)CC2(O)CCCC2)C1 O=C(Cc1cccs1)NNC(=O)C1(F)CCNC1 N(C(=NCCCCl)NCC(N1CCOCC1)C)C(C)CC1CNC(=O)O1 c1(C(=O)NC(C)CCN(C)C(C2CCC2)=O)ccc(Br)c2c1OCCC2 c1(C(=O)NCCN(C(C2CCCCC2C)=O)CC)cc(Cl)c([N+](=O)[O-])[nH]1 C(=O)(CS(=O)(=O)CC1CCCC1)N(C(C)CNC(=O)CCOCCN(C)C)C C1(CNC(CCOC(CC(C)C)C)=O)CCN(C(c2ccc(F)cn2)=O)C12CC2 N1(C(=O)NCC)CCC(C(=O)NCC2CCCN2C(=O)C(C)(C)OC(C)C)CC1 c1(CNC(C2(NC(=O)CCN3CCCCC3)CCC2)=O)cccc(O)n1 c1(NC(C2CCC(NC(CC(C)(C)C)=O)CO2)=O)ccn2nccc2c1 N1(C(C2=C(C)OCCC2)=O)CCCC2(CCCCC2NC(=O)C2=CCOCC2)C1 c1(C(=O)NCCC(=C)CNC(c2ccnn2C=C)=O)ncc(F)c(OC)n1 N1(C(CC2(OCC)CCC2)=O)CCC(C(=O)NCC(O)C(C)O)C1 c1(CC)csc(CNC(=O)C(=O)NC(c2ccnn2C)C)n1 n1(CCC=C)cc(C(=O)NC(C2(O)CN(C(=O)C(F)(F)c3ncccn3)C2)C)nn1 N1(C(C(c2cccnc2)OC)=O)CCC(C)(NC(C)=O)C1 C=CCCCC(C(=O)N(C)CC1CCC(CC)CC1)NC(=O)C=NOC C1(C)(C(=O)NCCC2CCN(C(c3c(CC)nn[nH]3)=O)C2)CCC(=O)N(C)C1 C(=O)(C(C)C(=O)NCCN1CCN(C(C2(F)CCCC2)=O)CC1)OC Cc1ccc2ncc(C(=O)NC3(CNC(=O)CCC4CC4(F)F)CC3)c(=O)n2c1 Cn1nnc2cc(C(N3CC4CC3CN4C(c3cccc(C(F)F)c3F)=O)=O)sc12 C1(NC(c2cc(C)ns2)=O)CC12CCN(C(=O)CC1COCC1O)C2 C=C1Cn2c(C(N3CC(C(N)=O)(CNC(C4CC5(CC5)C4)=O)C3)=O)nnc2S1 C(=O)(CCCCC(=O)N(C)C)NCC(CC)NC(=O)CC(C)(C)C1CCCC1 C1(N(C(CCOC(C)=O)=O)CCO)CCN(C(C2(C)CC2(F)F)=O)C1 n1(C2CCN(C3CC(C)CC(O)C3)CC2)nnc2c1CCCC2 C1(NC(C2(CCC=C)CC2)=O)CCN(C(=O)C=Cc2scnc2C)CC1C C12(C(=O)NCC3(NC(CC(CC)C4CCC4)=O)CCCCC3)CCC(F)(CC1)C2 c1(C(=O)NC(C(C)NC(c2ccc(=N)[nH]c2)=O)C)csc2cccnc12 N1(C(C2CC(=O)C2)=O)CCn2c(Cc3cn(CCC4CC4(Cl)Cl)nn3)nnc2C1 c1(OC)ncc(F)cc1-c1cn(CCC(=O)NC2CCCN(C)C2)nn1 C1(NC(C2(C)CCCCO2)=O)CC2COCC(C1)N2C(=O)CC1CCC(=O)NC1 c1(NC2C(F)(F)COCC2)nccc2c1OCC2 C12(CNC(CCN(C)CC)=O)CCCC1N(C(C1CCC1(C)C)=O)CCC2 c1(C(=O)NCC2COCCN(C(CCCCC#N)=O)C2)cccc2nc(Cl)cn12 N1(C(=O)NCCN2CCOCC2C2CCCC2)CCC(CC(F)(F)F)CC1 C1(C(=O)NC2CC(CCC(=O)NCC(F)(F)CO)C2)CC(C2CC2)=NO1 C1(NC(C=C(C)c2cccs2)=O)CN(c2nccc(C#N)n2)CCC12CCC2 Cc1cccc(C(C(=O)NCC2CC2)N(C2CC23CCC3)C)c1F N1(C(c2nc(CNC(c3cc(C)c(C)s3)=O)oc2C)=O)CC(C)C(F)(F)C1 C(C)(CNC(=O)C(O)C(C)C)(CC(C)C)NC(C(CC)=CC)=O C(C1=CCN(C(C2CCC3(CCC3)C2)=O)CC1)NC(c1c(C)onc1C1CC1)=O c1(CC)cnc(CC(=O)NCC2C=CCN2C(C23CC(C(C)=O)(C2)C3)=O)[nH]1 C1(C(=O)NC(C)CCCO)CCC2(CC2)N1C(c1cc[nH]n1)=O C1(C)(NC(CC(=C)C)=O)CCCN(C(=O)C(C)N(CC)CC)C1 c1(C(=O)NCC2(C)CC2(F)Cl)ccnc(N2CCN(CCCNC(=O)C3CC3)CC2)n1 C#CCCCCC(=O)NCc1cn(Cc2ccc(C)cc2Br)nn1 Cc1cc(C(N2CC(O)CC2(C)C(N2CC(F)(C3CC3)C2)=O)=O)cc(C)c1 c1(SCC(=O)NC2C(NC(C(C=C)(C)O)=O)CC2)ccc(C#N)cc1 C1(NC(C2CC3(C2)CC(O)C3)=O)CN(C(=O)CS(=O)(=O)CC2CCCO2)CC12CC2 C(N=c1cccc(S(=O)(=O)NCC(C)(C)C#N)[nH]1)c1cccc(SC)c1 C(=O)(CC1COCc2ccccc21)NC(CN(C(COCC=C)=O)C)C c1(CCC)cc(C(N2CCC(N(CCC)C(c3ocnc3C)=O)CC2)=O)nn1C Cc1nc(CC(N2CCC2CNC(c2ccc(CO)s2)=O)=O)c2ccccn12 c1(C(=O)NCC(C)N(C(=O)Cc2nonc2C)CC)ccccc1Br c1(C(=O)NC2C(NC(C(=Cc3cccs3)C)=O)CC2)cnn(C(C)C)c1F c1(C(N2C(CNC(=O)CC3CC4(CC4)CO3)CC2)=O)nc2cccnc2s1 S(=O)(=O)(c1cccc(Cl)c1)NC(C(=O)N(CC(C)NC(=O)COC)CC)C Cc1cccc(F)c1CNC(=O)CCN(C(C1OCCOC1C)=O)CC1CC1 Cc1ccc(CC(C(=O)NC2CN(CCO)C2)O)cc1.c1(OCC)ccccc1 c1(CC(=O)NC2CC(F)(CNC(CC3(C)CC3)=O)C2)nc(-c2ccco2)oc1C CC1=C(C(=O)NC2(CNC(c3nc(C)n(C)n3)=O)CC2)Cn2nnnc2N1C C1(CC(=O)N(C)CCNC(=O)CC(=O)NCC2CC2)CCCC(=O)N1 c1(OCC(n2cc(CNC(C(c3ccccn3)C)=O)nn2)C)ccc(F)cc1Br C(CC(N)=O)(C(=O)NCCC1CCCCC1O)NC(c1cc(CCC)[nH]n1)=O N1(C(C(C2CCCC2)OC)=O)CCOC(CNC(=O)CN2CCCC2)C1 N1(CC(=O)NC(C)C(=O)NC2CSC2)CCCCCC1 c1(SCC(=O)NC2CN(C(=O)C(CO)c3ccccc3)C2)cccc[n+]1[O-] c1(C(=O)NCCCC(C)NC(c2sc(F)cc2Br)=O)cc2ccncc2[nH]1 N1(C(c2cn(C)nn2)(C)C)CCC(=CCNC(=O)C(C)(C)C)CC1 c1(NC(C2CN(C(=O)CN3CCC(n4cccn4)C3)C2)=O)ccc(C(F)F)cn1 N1(C(CC2ON=C(C)C2)=O)CC2COCC(C1)C2NC(=O)CCc1cc[nH]n1 CC1(C)C(NC(C2CC3CC3C2)=O)C2CCCN(c3ncnc4[nH]ccc34)C12 C12(NC(c3c(C(N)=O)c[nH]n3)=O)CN(C3CC3)CC1COC2 c1(N(C)C(c2nnnn2C)=O)ccc(C(F)(F)F)cc1-n1cccc1 C(=O)(CC(C)(C)C(F)F)N(CC(CO)NC(CCC(C)CN(C)C)=O)C1CC1 C12(NC(C(c3cc(F)cc(F)c3)C)=O)CCC(C1)N(C(C1(CF)CC1)=O)C2 C1(C(=O)NCCCOCC=C)CCC(C(C)C)N1C(=O)C(O)CCSC Cc1ccc(C)c(-n2nc(-c3ccccc3)nc2C2CCC(C)O2)c1 c1(C(=O)N)c[nH]c(C#N)c1.C1(C(=O)NC(CC)CN2CCCC2)(C)CCCCC1 C1(F)(CNC(Cc2n(C)ncc2Cl)=O)CCCN(C(C2CC(=O)NC(=O)N2)=O)C1 N1(C(C(C)(C)O)=O)C2CCC1(Cn1cc(CC3CCCCO3)nn1)CC2 C(C)(C(C(C)C)NC(C(C)=CC1CC1)=O)NC(c1ccc(Cn2ccnn2)o1)=O C(=O)(C(C)(C)C(C)(F)F)NCC(C(=O)NC(c1cnc[nH]1)C)O C1(C)(COC)CC(NC(=O)CC(C)(F)F)CN1C=O.c1(C(=O)OC(C)(C)C)nncs1 N1(C(C(COCC)C)=O)CCC2(CC1)CN(C(=O)C(=O)C(C)(C)C)CCO2 CC1CC(=O)NCC1C(=O)NCC1CC2(CC(NC(=O)CSC(F)F)C2)C1 N12CC3CCC1C(C3)N(CCC=C)C2=O.c1(SC)cc(Cl)c(OC)cc1F C1(C(=O)NC2CCNC2=O)(OC)CCN(CC(=O)N2CCC2)CC1 c1(C(N2C(CNC(C(CCC)OCC)=O)CCC2)=O)cc(OC)cc2c1CCCC2 c1(C(=O)NC(CNC(C(CCC)C)=O)CC)ccc2c(c1)C(=O)CCN2 CC(C(=O)NC(C)CC(=O)N(C1CC1)CC1CC=CCC1)C(F)(F)F c1(OC)ncc(C(C)(C)NC(c2cc(Cl)ccc2Cl)=O)cc1-c1cccc(CO)c1 C1(C)(CCN)CCOC1=O.C(C(C)C(=O)NCc1cn(CC(=O)CC)nn1)OC C(CS(=O)(=O)CC(=O)N1CCCCC1C(=O)NC1CC(C)(C)C12CC2)OC C1(NC(CN2CC(C)C2)=O)CC12CC(NC(=O)CC1CC3CC3C1)C2 c1(C(=O)NCCC2N(C(c3c(C)c(N)ccc3)=O)CCC2)c(Cl)ccc(F)c1C c1(C(N(CCN(C(C(CC)C)=O)C)C(C)C)=O)nnc(O)c(Br)c1O CN(C)NC(=O)CCC(=O)NCC1CC1C(=O)NCC1CC=CC1 N1(C(C(=O)N(C(C)C(C)C)CCCC)=O)CCC(OCCC)C(C)(C)C1.C1CN1 c1(C(C(=O)NC)N(C)C(C)C)cc2c(Br)ccc(OC)c2o1.CCCCCOC c1(NC(CC2(C)CCN(C(C(CC)CC)=O)C2)=O)cnc(C)c(C)c1 CCCC(C(=O)NC(C)Cn1cc(CS(=O)(=O)CCOC(C)=O)nn1)C(=O)O N1(C(Cc2nc(C)sc2Cl)=O)CCC(C)CC1CNC(c1cc(F)c[nH]1)=O C(C)(CCCCNC(c1nonc1N)=O)NC(CN(C(C(C)C)=O)C)=O c1(C(N2CCC(C(=O)OCC3CC(OC)(OC)C3)C2)=O)[nH]c2ccc(F)cc2c1Cl N=c1nc(N2CCC(CN3CCOCC3)C2)[nH]c(N2CCCC(CC(N)=O)C2)n1 CC(CNC(=O)CN1CCOC1=O)(CO)NC(=O)C(O)CN1CCCC1 CC(C)(C)C(=O)NCC1CCN1C(C1CC1C(C)(C)C)=O C=C1CC2CCC(C1)N2C(=O)CC(C)C(C)(C)NC(=O)Cc1ccc(F)cc1 C1(C(=O)NCC2CC(F)(CNC(CCCOCCC)=O)C2)CCCC(O)C1 CC1(C)CCCCC1NC(C1CC1C1CN(C(=O)CC2CCCC2)C1)=O c1(CS(N2CCCCC2C2CCC2)(=O)=O)ccc2ccccc2c1 c1(C=O)cc2n(n1)CCCC2.C1CCCN(N(C(C(C)C2CC2)=O)C2CC2)C1 C12(COC)CC(NC(=O)CCP(C)(C)=O)(CN1C(=O)CSC(F)(F)F)C2 c1(CNC(=O)NCC(CC)NC2CCN(C3CC3)C2=O)ccccc1F c1(C(=O)NC2C(NC(c3cncc(OC)c3)=O)CC2)ccc(Cl)c(F)c1O c1(CC)cc(C(=O)NC2CCCC2NC(=O)CCC(N)=O)c2c(c1)CCO2 CC1=NN(C)C(=O)C1CC(N1CC(CNC(C2(O)CC2)=O)CC1(C)C)=O C1(C(=O)NCCN(CCO)CC)CCC(C)N(C(=O)CC2CCCC2)C1 N1(C(C)=O)CCC(C)C1CNC(c1cc(-c2ccccc2)ns1)=O C1(CNC(C(=Cc2cccs2)C)=O)C2CCC1CN(C(c1ncoc1C)=O)C2 CC(CC(C)NC(=O)CC1(N2CCOCC2)CC1)CCNC(=O)Cc1ccns1 c1(CSCCC(=O)NC(C)CO[Si](C)(C)C(C)(C)C)csc2ccccc12 N1(C(C2(C)CCCN(C)C2)=O)CC2=C(C1)CN(C(c1ccc(Cl)s1)=O)C2 S(=O)(=O)(c1cccnc1N1CCOC(CC)CC1)NCC1(COC)CCC1 Cc1coc2ccc(C(N3CCC(NC(=O)CN4CC(C)(C)C4)C(O)C3)=O)cc12 CC1CCCC(O)(C(=O)NC2CCCCC2CNC(c2cc(F)ccc2F)=O)CC1 C1(C(=O)NCCCCC2CN(C(C3(SC)CC3)=O)C2)C2CCC1C2 C1(NC(Cn2ccc(C(=O)OC)n2)=O)CCCN(C(=O)Cc2csc(C)n2)C1 c1(CCNC(CC2N(C(CCCOC)=O)CC2)=O)ncccc1C n1(CC(=O)NCC2OCCC(NC(CCC=CC)=O)C2)cccc(C)c1=O N1(C(c2ccc(C)n(C)c2=O)=O)CCCC2(C1)OC(=O)NC2=O N1(C(c2cncc(C(C)C)c2)=O)C2CCCC1CN(C(=O)CC(C)(C)O)CC2 CC1CN(C(C2COC(=O)N2C)=O)CC(C(=O)NCC2C3CC4C(C3)C24)O1 Cc1c(CC(N2CC(CC(=O)NC3CCC(O)CC3)CC2C)=O)cnn1C C1(NC(CC(CC)O)=O)CC1C1CCCN(c2nc(Cl)nc3c2SCC3)C1 C1(CNC(C(N2CCCCC2)C)=O)CCN(c2cccc(F)c2C#N)C12CC2 CN1CCC(C(=O)NC23CCC(CC2)C3)(NC(c2cnn(C)c2N)=O)C1 O=C1OCc2cc(C(N3CCCCC(NC(C4CC(O)C4)=O)C3)=O)ccc21 N1(C(C#CC2(C)CC2)=O)CC(CNC(c2cc3c[nH]cnc-3n2)=O)N2CCC1C2 C1(NC(C2C(N=[N+]=[N-])COC2)=O)CCN(C(C2CC3CCC3C2)=O)C12CCC2 C1(C(N2CCC(O)(C(C)NC(C3(CC(F)F)CC3)=O)C2)=O)CCN(C)C(=O)C1 c1(C(N(CC(CNC(Cn2ncc(C#C)c2)=O)O)C)=O)cc2cc(C)ccc2[nH]1 c1(N(C(CCSCCC)=O)CC2CC2)c(C)ccnc1O.C12C=CC(C1)C(=O)N2 C1(NC(c2c(C)nc(O)[nH]2)=O)CN(C(c2cncc(Cl)c2)=O)C(C)(C)C1 C(C)(C(=O)N1CC(N(C(=O)CS)C)C1)(C1CC1)OC.c1(C2CCOC2)ccccc1 c1(CC(=O)NC2(CO)CCN(C(C(N)=O)=O)C2)nc2ncccn2n1 N1(C(C2CN(C(C)=O)C2)=O)C2CCCC1CC(NC(C1CCCC3CC13)=O)C2 c1(CC(=O)NCC2(CCNC(c3ccn(C)n3)=O)CC2)ccc2nc(O)[nH]c2c1 Cc1cc(CN2CC(NC(C3CC4C=CC3C4)=O)C3(CC3)C2)ccc1Br N12CC(=O)NCC1C2=O.C=CCC(C)C(=O)OCc1nc(N2CCOCC2)n[nH]1 Cn1ncc(CNC(=O)CC2CCOC2(C)C)c1C(=O)NCCC1(C)CCC1 c1(C(=O)NC2CN(C(c3[nH]cc(C)c3)=O)C(C)C2)cc(Cl)cc2ccncc12 CN1CC=C(CCNC(C2CC3C=CC2N(C(=O)C=CCN2CCC2)C3)=O)CC1 N1(C(CCc2cc(C)on2)=O)CC(C(=O)NCCCSC(F)F)C2(CCC2)C1 c1(C(N2C(C)CCC(NC(c3ccc([N+](=O)[O-])[nH]3)=O)C2)=O)ccnc2[nH]nnc12 C1(NC(CCCC(C)OC)=O)CC2CCC1CN(C(=O)CCc1n[nH]c(=N)s1)C2 c1(C(=O)NCC2CC2NC(=O)C(C2(O)CCCC2)F)nccc2[nH]ccc12 N1(C(c2c(N)c(Cl)ccc2)=O)CC=C(CCNC(C2CC(O)C(F)C2)=O)CC1 C1(C(N2C(c3ccc(OC)cc3)CCC(C)C2)=O)CN(C)C(=O)CN1C c1(C(N2CCCC(CCNC(C(C=C=C)C)=O)C2)=O)ncc(F)c2ccccc12 CN=c1[nH]cc(C(N2CC(NC(c3cnn(C)c3C)=O)C(c3ccnn3C)C2)=O)o1 CC(C)(C(=O)NCC1C=CCN1C(=O)C(O)Cc1ccccc1)c1cscc1Cl CCC(C)CCC(=O)N1CC2(C1)CN(C(c1ccc(COC(C)C)cc1)=O)C2 c1(C(=O)NCCC(C)NC(C2CCCCC2C)=O)cc(Cl)c(F)cc1O CC(C(C)C(=O)N1C(C(=O)OC)CC1C)NC(=O)CC1CCOC1=O c1(CC)nocc1C(=O)NCC(C(C)C)NC(C1CCCC1SC)=O C1(N(C(C(C)OC)=O)C)CCC(NC(C2CC23CCCO3)=O)CC1 c1(C(=O)NCCCCN(C(C2C(F)(C(=O)OCC)C2)=O)C)ccc(OC)cc1Cl N1(C(CCCSCC=C)=O)CC2ON=C(CNC(c3cccc(F)c3C)=O)C2C1 c1(OC)cc(C(N2CCC(N(CCO)C(C3CC(C#N)C3)=O)CC2)=O)ccc1C C1(N(C(C(C)=CC)=O)C)CCCC2CN(C(C3CCC(=C(F)F)CC3)=O)CC12 C1(NC(c2cn(CC)nn2)=O)CC(NC(c2ccccc2C)=O)C1(C)C c1(OC)ccnc(C(=O)N(C2CCCCC2)CCNC(=O)C(C)(C2CC2)OC)c1F c1(C(=O)NCCC(C)NC(C(CCOC)C)=O)cn2ccc(C)cc2n1 C(=O)(C1CCc2ccc(Cl)nc21)N1CCC(N(C(CC2CC(OC)C2)=O)C)CC1 C1(NC(C(CC)NC(C)=O)=O)CN(C(=O)C=Cc2scnc2C)C2(CCC2)C1 Cc1[nH]nc2c(C(=O)NC3CCC(N(C)C(c4cn[nH]c4)=O)C3)cccc12 C(=O)(CCS(=O)(=O)N(C)C)N(C1CCCN(C(C=C(C)C)=O)C1)C c1(NC(=O)NCCC(C(C)C)OC)ccc(N)cc1OCCCC#N c1(C(=O)NCCCC(C)(C)NC(c2c(OCC)nccc2)=O)[nH]nc2c1COC2 Cc1cn2nc(C(N3CC(C4CN(C(c5c[nH]c(=N)o5)=O)C4)C3)=O)cc(C)c2n1 c1(C(N2C(CN(C(C(=CC3CCCC3)C)=O)C)CCC2)=O)cn2cc(C)sc2n1 C1(C(=O)NCC(C(=O)OC)O)CCCN(C(=O)Cc2csnn2)C1 Cc1ccc2nc(C)c(N3CCC(C(=O)NCCC4CCCCC4)CC3)nc2c1 C1(C(=O)NCC2(OC)CCN(C(=O)C(C)(C)Br)C2)CC2CCC(C1)O2 C(=O)(CC(C(=O)NC1C=CCN(C(C2(CO)CCOCC2)=O)C1)N(C)C)OC C(C(C(=O)NC1CCC1NC(=O)Cc1cncnc1)N(C)C)OC C1(C(N(CC(C)C(F)(F)F)C)=O)CC2CCC(C1)N2C(=O)C=Cc1cscn1 Cc1[nH]c2ccccc2c1CC(N1CC(NC(=O)CC2CCCCC2C)C1)=O Cn1nc(C(=O)NC2CCCN(c3cncc(Cl)n3)CC2)c2c1CCOC2 c1(OC)cccc([N+](=O)[O-])c1C(N1CCC(O)C(C(=O)NCC(C)(F)F)C1)=O N1(C(c2ccc(SC)cc2)=O)CC2CC1CN2C(C12CCC(C1)C2)=O N1(C(C2CCCN(C(C)=O)C2)=O)CC2(CCCCN2C(=O)OC(C)(C)C)C1.OC C1(NC(C(C)=CC=C)=O)CCCCCC1C(=O)NC1(CC2CC2)CC1 Cc1[nH]cc(C(=O)NCC(C)(O)CNC(=O)CC2(C)CCCC2)c(=O)c1Cl c1(SC(c2ccc(F)cc2)C(=O)N(C(C)C)C)ccc2ccccc2c1 CCC(C)(C)CC(=O)N1CCCCC1CN(C(c1cc(C(C)(F)F)n[nH]1)=O)CC Cc1ccc(COCC(=O)N(CCCCCNC(c2ccnn2C)=O)C)cc1 C1(NC(COC)=O)CCN(C(=O)C(C)Oc2cccc(C#N)c2)CCC1CO c1(C(=O)NCC2(F)CC(CNC(C(C(C)O)C)=O)C2)cccc2c[nH]nc12 C1(NC(=O)Cn2cc(C3CCNCC3)nn2)CC12CCN(C1CC3C=CCC13)CC2 Cc1ncc(F)c(NC(CCN(C(=O)Cn2cnnc2)C)C(C)C)n1 C1(CNC(CC2(C=C)CCC2)=O)CC(F)CN1C(C1CN(S(=O)(=O)C(F)F)C1)=O Cc1ccc(F)c(OCC(=O)N(CCCCCCNC(C2(F)CC=CC2)=O)C)c1 C1(NC(CCOCCOCC)=O)CCCC1NC(c1cc(C(N)=O)cs1)=O c1(C(N2C(CC(=O)NC3C(OC)CCC3)CCC2)=O)cc(F)cc([N+](=O)[O-])c1 c1(CNC(N2CC(NC(CNC(CNC(C)=O)=O)=O)C2)=O)ccc(O)cc1F C=CC(CC)CC(=O)N1CC(NC(c2sc(Br)cc2C)=O)C(F)C1 N1(C(Cc2scc(C)c2)=O)CC2CCCC(N(C(=O)CC3(C)CCC3)C)C2C1 C(=O)(C1=CC2(CCOC2)C1)N1CCC(COC)(NC(c2ccncc2F)=O)CC1 C1(C(=O)NC2(C)CN(C(c3c(OCC)nccc3)=O)C2)CCCC2(C1)CC2(F)F C(=O)(C1=C(C#N)CCC1)NC(C1CCCCC1)C(N1CC=C(COC)CC1)=O CC(CN(C)C)CC(=O)NC1CCC(NC(c2c[nH]c(=N)o2)=O)CC1 C1(C(N(C)CCn2cc(C3CCCC3)nn2)=O)C2Cc3cc(Cl)ccc3C12 N1(C(C(N2CC(NC(c3ccn(CC)n3)=O)C(C)C2)=O)(C)C)CCS(=O)(=O)CC1 CCC(CC(=O)N1CCC(N(C)C(c2cc(Cl)ns2)=O)C1C(C)C)SC N1(C(CNC(C(N2CCN(C(C=CS(C)=O)=O)CC2)=O)=O)=O)CCSC(C)(C)C1 C(=O)(CC(C)CC(C)(C)C)N1CC2OCC(NC(C=CCN(C)CC)=O)C2C1 Cc1c(NC(=O)N(C)Cc2cn[nH]c2)cccc1Br CN=c1[nH]nc(CC(N2CC(NC(=O)C=CC=CC=C(C)C)CC2C)=O)s1 c1(C(=O)NCCN(C(C)=O)C)ccc(F)cc1.N12CCCC1C2=O C(=O)(C1=CC(C)(c2ccccc2)C1)NCCCCN(C(C1C(C#C)C1(C)C)=O)C CCC(CC)(CO)C(=O)N(C)CCOCCN(C(=O)Cc1ccc(C)c(C)c1)C CCCCN=C(NCCN1CCCCC1)NCC(C)Nc1ccccc1.S(C)(=O)(=O)N Cc1cc(N(C2CNCC2C#N)C(c2cc(Cl)ccc2F)=O)n2nc(C)cc2n1 N1(C(C=CCOCC=CCCCCC)=O)CC2(CC(NC(=O)C3=CC(C)(C)C3)C2)C1 C(=O)(CCC[N+](=O)[O-])N(C1CCN(C(=O)NC2CCC(C)C2)CC1)CC C1(NC(COCCCC)=O)CC2CC(NC(c3nocc3C)=O)CC2C1 C12CCN(C1)C2=O.C1(F)(CN(C(CNC(=O)NC)=O)C)CCOC1 C(=O)(C(C)(F)C(F)(F)F)NC(C(C)NC(C1CCC(CO)CC1)=O)CO c1(C(=O)NCC(C)(C)NC(C(CCSC)NC(N)=O)=O)ccc(S(C)(=O)=O)o1 C(=O)(CC(N)c1nccn1C)N(C1CCCC1Cn1cccn1)C c1(C(=O)NCC(CC)(C)NC(C2(COC)CC2)=O)ccc2c(c1)C(=O)OCC2 c1(C(c2nnnn2C)NCc2scc(CC)n2)cccc(S(F)(F)(F)(F)F)c1 c1(OC)cc(C#N)ccc1C(C(=O)NC1COC1)N(C)Cc1ccccc1SC Cc1cc(CCCC(=O)N(C(CNC(=O)CC2CCCOC2)C2CC2)C)on1 C#Cc1ccc(C(=O)NC(C2CN(C(=O)C(F)CC3CC3)C2)C(C)C)cc1C c1(C(=O)NC(C2CCCC2)CN(C(=O)C(F)C2CCCC2)C)cc(C2CC2)no1 N1(C(=O)OC(C)(C)CO)CCCCC1.C12CC1C(=O)O2 C1(C(N2CC3C(CNC(C(c4ccc(C)o4)C)=O)(C3)C2)=O)CC(=O)NC(=O)C1 Cc1ccc2c(N3CCCN(C)CCC3)nc(=NCc3csc(C)c3C)[nH]c2c1 C1(C(N2C(C)(CCC(=O)NCC(=C)Cl)CCC2)=O)CCN(C)C(=O)C1 N1(CC)CCC(NC(=O)CNC(=NC)NC2CC2)C(C)C1 c1(C(=O)OC)cc(OC)cc(CC)c1.N12CC(CC1=O)N(C)C(=O)C2.CCO c1(C(=O)NCC(CCCC)NC(=O)CC2CC2)c[nH]c2ccc(OC)cc2c1=O CC12CN(C(c3cnc(S)n3C3CC3)=O)CC1(C)CN(c1cc(C(F)F)ncn1)C2 CC1CCOC1CC(=O)NC1CC(CCNC(c2ccnn2C(F)F)=O)C1 C1(C(CC(=O)OCC)NCCc2ccc(Br)s2)CCOC(C)C1 N1(C(c2cc(OC)c(O)c(Cl)c2)C(=O)NC)CCCCC1C1(C)CCCO1 CCCC(C)(O)C(=O)NC(CNC(C1CCN1C(=O)OC(C)(C)C)=O)CC(C)C C1(NC(=O)C=C2CCC2)(CNC(c2cnc(C3CCCO3)s2)=O)CCOC1 N1(C(C(C=C)c2ccccc2)=O)CCN(C(=O)C=CC(=O)NC2CC2)C(CO)C1 C(=O)(C(C)(C)CS(N)(=O)=O)N1CC(C)N(C(c2coc(CO)c2)=O)CC1C N1(C(C(CC)C(C)C)=O)CCC2CCCC12C(=O)N(CC(C)C#N)CC c1(N2CCN(C(CNC)=O)CC2)cc(-c2ccc3nncn3c2)cc2cc[nH]c12 C(CCC)(C(=O)NCCCCNC(=O)CC1CCOC(C(C)C)C1)=CCC N1(C(CCC#C)=O)CC2CC(C1)C2NC(C1(C)C=CCCC1)=O CC1CCN(C(c2cn(C)c(=O)n2C)=O)CC1NC(=O)C(=O)C(C)(C)C C=CCC(C(=O)N(C)C)NC(=O)CN(C(=O)COCC1CCCO1)C c1(C(N2CCC(C(CNC(C(CC)OCC)=O)F)CC2)=O)ccnc2[nH]cnc12 C(=O)(C(O)CCNC(c1cccc(O)n1)=O)NCCNS(C)(=O)=O CC1(C)COCCN(C(=O)C(Cc2ccoc2)NC(=O)Cc2cncnc2)C1 C1(C(=O)NC2(CO)CN(C(c3c(N)nccn3)=O)C2)CCC2(CCCC2)CC1 C=CCC(CNC(C1CCCC1CC1CC1)=O)C(=O)N1CC2CCCC2C1 c1(CC(C)C)onc(C)c1C(N1CC(NC(=O)CSCc2ncc[nH]2)C(O)C1)=O C1(C(=O)NCC2(CO)CCCN2C(c2cc(C(N)=O)[nH]n2)=O)CN(OC)CC1O c1(C(N2C3CC(CNC(=O)CC4CCC4)C2CC3)=O)cc2ccccc2o1 C12(CC)CCC(C(=O)NCC(C(C)C)NC(=O)C=Cc3cc[nH]n3)(CO1)C2 N1(C(c2c(CC)csc2)=O)CC2CCN(C(=O)C#CC3(CC)COC3)CCC2C1 c1(C(N2CCC(CN(C)C(=O)OC(C)(C)C)C2)=O)cc(F)c(F)c(Cl)c1 N1(C(C(C=C)OC)=O)CCCC(N(C(=O)C(C)SCC(C)C)C)CC1 c1(CC(=O)N(C(C)CNC(C2CC2COC)=O)C)ccnc(O)c1 Cn1ncc(C(c2nnnn2C2CC2)NC2CC(c3cccc(F)c3)C2)c1Br N1(C(=O)OCC)CCC(c2nnnn2C(C)C)(NC(CCO)C(C)(C)C)CC1 CC(C)(C)C(CNC(c1cc(C#N)on1)=O)NC(=O)C=CC1CCCCC1 C1(NC(C(C)SCC)=O)CCC(O)CN(C(C2CCCN2CC(C)C)=O)C1 C1(COC(C)(C)C)CCN(N2CC(Cc3ccccc3)C2)CC1 C1(NC(C=C(COC)C)=O)COC2(CCN(C(c3[nH]cnc3C#N)=O)C2)C1 C(=O)(CCCCC(=O)N1CCC(NC(=O)Cn2nc(C)c(Cl)c2C)CC1)NC Cc1nc(O)ccc1C(N1CC=CC1CNC(c1cc(C(C)(F)F)n[nH]1)=O)=O C1(NC(C(COC)(C)C)=O)CN(C(c2ccc(=O)n(C)n2)=O)CC2(CC2)C1 Cn1cccc1C(=O)C(=O)NCC1N(C(c2ocnc2-c2ccccc2)=O)CCC1 C1(NC(c2c(C)cco2)=O)CC2(CCCN(C(c3cc(C)c(C)nc3O)=O)C2)C1 C1(CNC(C=CC=CC)=O)CC2(CCN(C(=O)Cc3cnccc3C)CC2)CO1 c1(NCCC2CCC(NC(c3c(Cl)ccc(C)c3)=O)C2)ncnc2c1SCCC2 C(c1cc(Cl)c2c(c1)OCO2)=CC(=O)N(CC(C)N(C(C=C(C)C(F)F)=O)C)C C12C3CC4C(C3NC1=O)C24.c1(C(C)CNC(C2(CCN(C)C)CC2)=O)cn[nH]c1 n1(COC)c(C2C3CCOC(C3)CN2)nc(Br)c1Br.c1(CC2CC2)ccccc1 c1(CC(=O)N(c2c(C)noc2C)CC)ccc(N2CCNC(=O)C2)cc1 S(=O)(=O)(N=c1cc(Br)[nH][nH]1)CC1(C)CN(C(c2cc(C(C)C)nn2C)=O)C1 C(=O)(C1CCc2scnc21)NC1CC(NC(c2ccn(CC#N)n2)=O)C1 CCC(N=c1nc2scnc2c(NCc2ccc(C3CC3)cc2)[nH]1)C1CCOC1 N1(S(=O)(=O)CCOc2ccccc2I)CC2CC(C1)C2O C1(C(NOCCC#C)=O)(CNC(C2CCC(=O)C2)=O)CC(C)(C)C1 C1(CC(=O)NCCCCNC(c2cncc(C(F)(F)F)n2)=O)CCC(F)(F)CC1 c1(-c2nc(CC)[nH]n2)cccc(C(=O)N(C)CCNC(C2CCO2)=O)c1 N1(C(CC(C)CF)=O)CC(O)(C2(CNC(=O)CCc3cnco3)CC2)C1 CS(=O)(=O)C1CC(C(N2CCC(CCCCNC(=O)C3=CCC3)CC2)=O)C1 C=CCC(C)(C)CC(=O)N1CCC(F)(F)C(CNC(=O)C2=CC(C)CC2)C1 N1(C(C(CC2CC2)OC)=O)CC(C(F)(F)F)CC1CNC(C1(C)CCC(=O)C1)=O C1(N(C)C(c2cn[nH]c2)=O)CCCN(C(c2cnc(N(C)C)s2)=O)CC1 c1(OC)ccc(C(=O)NCCC(O)CNC(=O)CCc2cccc(C)c2)nn1 Cc1cc(C)c(C(=O)NC2C3CN(C(C4CC5C(C4)C5(F)F)=O)CC23)c(S)n1 C1(C(=O)NC2CCC(NC(c3ccc(C#N)[nH]3)=O)CC2)CCn2c(O)nnc2C1 C(C(=O)NC1CN(C(=O)Cc2cncc(C)c2)CC1OC)(C(C)C)OC Cc1cc(CC(=O)NCC2C3CC2N(C(=O)Cc2cnns2)C3)c(C)s1 CS(=O)(=O)C1CCCN(C(=O)CC2CCN2C(c2cc(C#N)c[nH]2)=O)C1 C1(C(N2CC(C(=O)OC)C2)=O)CCCCCCN1C(=O)CC1C=CCCC1 C#CC1(NC(=O)C(CC(=C)Cl)NC(=O)C(N2CCNC2=O)C)CC2CCCC12 c1(C(=O)NC2CN(C(CCC#CC)=O)CC2CC(C)(C)C)cc(F)cc(Cl)c1O N1(C(C2CCC=CO2)=O)CC2CCN(C(C3CC4C=CC3C4)=O)CCC2C1 c1(C(N2CC(CNC(CCSCCCC)=O)(OC)C2)=O)cc2n(n1)CCCO2 C1(NC(C(C)SCCCC)=O)CCN(c2nccc(CC(=O)OC)n2)CC1F C1(NC(C(C)NC(CC)=O)=O)CCCCCCC1C(=O)NC1(CC2CCC2)CC1 N1(C(C2N(C(C)=O)CCC2)=O)CCC(CF)(NC(=O)Cn2nnc(O)n2)C1 C1(NC(=O)Cc2cnoc2)CN(C(c2ccc3nsnc3c2)=O)C2(CCOC2)C1 c1(C(=O)O)ccc(Cl)c(CNC2CC2NC(c2cccc(-c3cccs3)n2)=O)c1 N1(C(C(C)(C)n2cnnn2)=O)CCC2C(C(=O)NCCC3CCC4CC34)C2C1 c1(CC(N2CCOCC(NC(c3nc(C)nn3C)=O)C2)=O)c[nH]c2ncccc12 Cc1nc2c(C(=O)NCC(C)(C)NC(C3CCCNC3=O)=O)ccnc2[nH]1 N1CC(NC(C2(CN(CC)CC)CC2)=O)CC(O)C1.c1cccc(-c2cccs2)n1 CC(=O)CCCC(=O)NC(C1CC=CCC1)C(=O)NCCCCN(C)C(C)C C(=O)(C1c2ccccc2C2CC1C2)N1CCC(C)(CNC(=O)C=CCF)C1 c1(C(C)NC(c2ccc(N(C)C)c(F)c2Br)=O)ccc2c(n1)NCCC2 c1(CC)cc(NC(C2(CNC(c3ncccn3)=O)CCCO2)=O)cc(O)c1 N1(C(c2n(COC)ncc2)=O)CCOC2CCN(C(c3ncsc3C(C)C)=O)CC12 Cc1nc(C(=O)NCCC2CN(C(c3cc(F)cnc3O)=O)C2)c(C)n1C C(=O)(C1=CC2CCC(C1)C2)N(CC(C)(C)CNC(C1(C)CCCS1)=O)CC c1(C(=O)NCCOC2CN(C(CC(=O)OC)=O)C2)sc(CC(F)(F)F)nc1C N1(C(C(CC)N(C)C)=O)CCOC(CN(C(=O)CCCOCCOC)C)C1 C#CC1(CNC(=O)C(C2CCCN(C(=O)CC3(O)CCCC3)C2)F)CCCC1 C(=O)(C1=CCCCC1)NCC(CNC(c1ccc(C(CC)=O)cc1)=O)F C1(CC(=O)NC(CNC(C(C2CCCCC2)OC)=O)C)CCCOCC1 N1(C(CCC)=O)CC(NC(=O)C(n2cc(-c3ccccc3)cn2)C)C(C)C1 C1(C(N(C)CC2CCN(C(c3ccoc3C(F)(F)F)=O)C2)=O)COCCN1C=O C=CCCCCN=C(NCCc1ccc(C)c(F)c1)NCCF N1(C(C2(OC)CCC2)=O)CCCN(CCNC(=O)C(CC)(CC)NC(C)=O)CC1 CCC(C)C(=O)C(=O)NC(C)CNC(c1cn(C)nc1O)=O S(=O)(=O)(c1cccc(-c2ccccn2)c1)NCCC1CC(CC)C1 C1(C(N2C(CN(C)C(c3cccn3C3CC3)=O)CCCC2)=O)CC2COCC2C1 C1(CC)(CNC(=O)C(c2ccoc2)NC(=O)COc2cccs2)CCCC1 C1(=CC(=O)NC(CC)C)CCN(C(=O)Nc2cccc(SC)c2)CC1 C=CCCCC(C(=O)NC(CCC)C(C)(C)C)NC(=O)C(C)CC1CCC1 C=C(C)c1cncc(C(C(=O)NCCN(CCC)CC)NC2CCC(F)(F)C2)c1 N1(C(c2c(OC)scc2)=O)CCOCC1CNC(c1ccc(CS(C)(=O)=O)o1)=O C1(NCc2onc(C)n2)CCCN(C(=O)C(N2CCC(C(F)(F)F)CC2)=O)C1 c1(NCC(CCC=C)(C)C)nccc(=NCc2ccc3c(c2)OCO3)[nH]1 C(=O)(C(C)C(C)(C)C)N(C(C)CCNC(c1cc(C(C)(C)C)c[nH]1)=O)C N1(C(COCCCC#C)=O)CCN(C(c2ccc(F)s2)=O)C(CO)C1 N1(C(c2c(NC)c(F)ccc2)=O)CCC2(CCCCN(C(=O)CC3CCC3)C2)C1 C1(CC(=O)NC(C#C)(C)C2CCOC2)CN(C(c2c(C)cncc2C)=O)CC12CC2 c1(C(N(CC(CC)NC(c2c[nH]ccc2=O)=O)C)=O)c[nH]cc(C)c1=O Cc1cc(C(=O)N(C)CC2CCCN(C(=O)C(C)Cn3ccc(C)n3)C2)ccn1 c1(C(N(C2CCCN(C(C3(OC)CC3)=O)C2)CCF)=O)ccc2c(c1)OCCC2 N1(C(C2(C(=O)OC)CC2)=O)CCc2ccccc2C(NC(=O)C(F)=C2CCC2)C1 N1(CNCc2c(C)nn(Cc3ccccc3)c2C)CCn2c(CC(N)=O)cnc2C1 N1(C(CCc2c(C)ncs2)=O)CCC2C(CCN2C(c2ccc(O)nn2)=O)C1 Cc1c(C(=O)NC(C)C(=O)O)oc2c1C(=O)CC(C)(C)C2 C1(C(=O)NCC(CCNC(C(C)(Cl)Cl)=O)O)CC2(C1)CC1(CC1)C2 c1(C(=O)NC2C(CNC(c3cscn3)=O)CCCC2)cccc2c1CCCC2 Cn1ncc(S(=O)(=O)NCC)c1C(F)(F)F.C(C(C)(CO)N)NC(=O)OC(C)(C)C c1(CC)cc(C)ccc1NC(=O)C(C(C)O)NC(C1CCC(F)(F)C1)=O C#CC12CCC(C(C3CN(C(=O)CN4C(=O)Cc5ccccc54)C3)=O)(CC1)CC2.NNCC C(=O)(CCC(C)CC(=O)OC)N(CCN(C(CCN(CC)CC)=O)C)C C1(n2c(=O)c2=O)CCc2ccccc2C1.c1(CC#C)cc(C)nn1C1CCC1 c1(C(N2C(C)CCC2)=O)cnn(C)c1F.CC1C(=O)OCCOCCO1 N1(C(CC(C)c2ccco2)=O)CCCC(NC(=O)COc2ccc(Cl)cc2)CC1 N1(C(c2ccc(C#N)cc2)C)CC2CC(C1)CN(C(=O)CNC(c1nccs1)=O)C2 C(CC(C)C)(C(=O)NOC)N(C(CSCCC)=O)C.C12(CCOC1)CO2.O c1(NC(CCN(c2cc(C#N)ncn2)CC)=O)ccc(C(C)O)c(F)c1 n1(CC)nc(C)c(CC(=O)NC2CC(C)N(C(c3ccc(C(=O)OC)[nH]3)=O)C2)c1C C1(C(=O)NCC(c2ccccc2F)(C)C)CC2CCC1N(C(=O)Cn1cnnc1)C2 c1(NCCN(OC)C)nc(N2CCCC(C(C)(C)C)C2)nc2c1ncn2C c1(-c2n(CC=C)nc(-c3cccc(OC)n3)n2)ccc2c(OC)nccn12 N1(C(C=CSC)=O)CCC2CCN(C(=O)COCc3cccnc3)C2C1 Cn1cc(C(=O)NCC2(CNC(=O)CCC3(C#N)CCC3)CC2)n(C)c1=O c1(CC(N2C(CCNC(CCC=C=C)=O)COCC2)=O)ccc2nc(O)[nH]c2c1 C1(OC(C2CCC2c2nc[nH]n2)=O)CCCCC1c1ccccc1 C1(C(C(=O)N(CC(=O)OC)C)C)CCN(C(c2csnn2)=O)C1 c1(C(=O)NCC(C)NC(=O)CC2CCOC2)cscc1F c1(C(N(CC)CC2CCN(C(c3cc(Cl)c[nH]3)=O)CC2)=O)cnn2ccncc12 c1(C(=O)NC2CN(C(CS(CC)(=O)=O)=O)C(C)CC2)cc(O)c2[nH]c(C)nc2c1 n1(CC)cc(C(=O)NCC2CCC(NC(=O)CC(C)(F)F)C2)c(C)n1 c1(CN(C(=O)CC(N2CCCC(CO)C2)=O)C(C)(C)C)cc2ccoc2cn1 C1(C(=O)NC(CN(C(C(C=C)(C)C)=O)C)C)CCN(C2CC2)S1(=O)=O c1(C(CC(=O)NC(CN(C(=O)C=Cc2nccs2)CC)C)O)cccc(F)c1 C1(C2C(=O)N2C2CC2)CCSCC1.c1(C)nc(Br)cs1.C1(N)CC1 C1(NC(c2nn(CC)c(C3CC3)c2)=O)CC2(C1)CC(NC(=O)CC1CC1)C2 C(C(C)(O)C(=O)N(CCCN(C)C)CCNC(C1CC1c1cccc(Cl)c1)=O)OC CCC(C)C(C(=O)N1CCC(O)(CCNC(c2cc(C#N)cs2)=O)C1)NC(N)=O C(c1cccc(Cl)c1)=C(C)C(N1CCC(NCc2ncccc2C)C(F)C1)=O c1(C(C)NC2C3CN(C(C(C)n4cncn4)=O)CC32)cccc2ccccc12 n1(CC(=O)NC(C2(O)CCN(C(C3C(C)=C3)=O)C2)C)nc2ccccn2c1=O CCCC(O)CC(=O)N1CCN(C(C2CN(C(=O)C(CN(C)C)CC)C2)=O)CC1 C=CCC(CC)N=c1[nH]c2c(c(=NCC3(CC(C)C)CCC3)[nH]1)CCCCCC2 C12CC3(CO1)CN(C3)CC2.N1(C(=O)OCC(=O)NC2CC=CCC2)CCCCC1 C1(CC=C)(NC(=O)C=CI)CC2CCC(C1)N2c1cncc(Cl)n1 C1(F)(CNC(CC2(OC)CCCC2)=O)COCCN(C(=O)Cn2nnc(=O)[nH]2)C1 C1(C(N2CCC3CCCCC3C2)=O)CCC(F)(F)c2ccccc2N1 CCC(CC(=O)NCC(C(C)(C)C)NC(c1cccn(C)c1=O)=O)CC(F)(F)F C1(C(N2CC3CC3(NC(C3CC(F)C3)=O)C2)=O)CCN(C(N2CCCC2)=O)CC1 c1(C(=O)NC(C)CCN(C)C(c2coc(Cl)n2)=O)ccc(F)c(Cl)c1 C1(CNC(c2n[nH]cc2Cl)=O)CC2(CO1)CN(C(c1cc(CF)on1)=O)C2 N1(C(c2ccn(C)c(=O)c2)=O)CC2(C1)CN(C(c1ncoc1C1CC1)=O)CCO2 c1(NC(=O)NC(c2ccc(NS(C)(=O)=O)cc2)C)ccc(S(=O)(=O)F)s1 c1(CC)ccc(C(=O)NC2CCCC2CNC(=O)CCCNS(C)(=O)=O)[nH]1 N1(C(C(C=C)O)=O)CCN(C(=O)C(n2cnc(C#N)n2)C)CC1 C(=O)(C1=NNC(=O)CC1)N1CC(C)C(CNC(=O)CC2CC2)CC1 C1(C(N(C)CC2(NC(=O)Cn3cnnc3O)CC2)=O)OCC2CCCC12 CC(C)(C)C(O)C(=O)N1CCCC(C(=O)NC2(CNS(=O)(=O)C(F)(F)F)COC2)C1 C1(C(CNC(=O)Cc2ccoc2)NC(COCCOCC#C)=O)CCCCC1 N1(C(CC(C=C)CCC)=O)CCN(C(=O)C(C)C2(O)CCC2)CC(C)(C)C1 N1(C(C(C)Cc2cnc[nH]2)=O)CCCCC1CNC(=O)C=CC=C(Cl)Cl C(CNC(C1CCCC1C)=O)(CC(=O)NCC)OC.C1(C)(C(=O)O)N=N1 c1(C(N(C)Cc2cccc(CNC(C3(C4CC4)CC3)=O)c2)=O)cc(O)ccc1F N1(C(C2(C(C)C)CCC2)=O)CC(O)(C(=O)NCCS(C)(=O)=O)C1 c1(CC(=O)NC2C(NC(c3c(=N)cc[nH]c3)=O)CCC2)cc(O)ccc1Br C1(C)(CNC(C(C)N2CCC2)=O)CCN(C(c2cncc(N)c2)=O)C1 C1(C(=O)NCCC2C(C)(C)CCO2)CCC(C)(C)N(C(C2(CO)CCC2)=O)C1 C12(n3cc(I)cn3)CN(C1)C2=O.C1(c2ccccc2)(C(=O)OC)CC1(Cl)Cl N1(C(CC2(OC)CC2)=O)C(C(=O)N(C2CC2(F)F)C2CC2)CC1C C1(O)(CNC(Cc2scc(C)n2)=O)CC2CCC(C1)N2C(=O)CC1(C)CC1(Cl)Cl c1(C(C(=O)N(CCC)CCNC(C2CN(C)CC2C)=O)(C)C)ccc(F)c(F)c1 n1(CC(=O)NC(CC)CC2CCN(c3ccnc(Cl)n3)CC2)nc(C)c(Cl)c1C C1(NC(C(C2CCC2)OC)=O)CCC(CNC(=O)CCc2ccccn2)C1 CC1(C=CC(N2CCCOC(CNC(C3CC(F)C3)=O)C2)=O)CCOCC1 N1(C(c2ccccc2)=O)CCN(C(C2CC3(C2)CC3(F)F)=O)C(CCO)C1 c1(C(=O)NC2CC(C)(CNC(c3c(C)cc(N)cc3)=O)C2)cnn2c1OCCC2 CC(C)C(CC(=O)N1CC(NC(c2cc(Br)cc([N+](=O)[O-])c2)=O)C1)C(C)C O=C1OCc2ccc(-c3cn(CC4CC5CC4CC5O)nn3)cc21 c1(OC)c(C(=O)NCCNC(c2ccc(C(C)=O)o2)=O)nc(O)nc1O N1(C(CN(S(C)(=O)=O)C)=O)CCC(O)(C(C)CNC(=O)Cc2ncc(Cl)s2)C1 C1(CC#C)(C(=O)NC2CCN(C(c3cnccn3)=O)C2C2CC2)CCOCC1 CC(C)C1=NOC(C(=O)NC(C)C(CO)NC(c2cc3n(n2)CCO3)=O)C1 N1(C(CNC(CCCCC)=O)=O)CC(C(=O)N(C(C)CC)CC)CCC1C N1(C(=O)CC2CCCOCC2)CC2CCC(C1)N2C(c1csc(Cl)c1)=O c1(CC)cc(C(=O)NCCCCC2CN(C(=O)CCOCCOC)C2)ncn1 C12(C(=O)NCC(CC)NC(=O)C(CC(C)C)n3ccnc3)CCC(C1)C2(C)C C1(N(C(CNC(C(C)OCC)=O)=O)C)CCN(C(c2ccccc2)=O)CC1 CC1CCN(C(=O)CC2C=CS(=O)(=O)C2)CC1CNC(=O)CC1CCNC1=O C(=O)(C(F)CC(C)(C)C)NCC1CN(C(C(C)(C2CC2)OC)=O)C1 CC1(C)CN(C(=O)Cc2csc(Cl)c2)CC1NC(c1nccnc1N)=O N1(C(=O)C=C(C)C(C)(C)C)CCC(C(C)C(=O)Nc2n(CC)ncc2)CC1 c1(OC)cc(C(N2CCN(C(C3(F)CC3)=O)C(C(C)C)C2)=O)ccc1Br C1(CC(=O)NC(C2CC3(CCC3)C2)COC)Oc2ccccc2C1C N1(C(C(CCC)C)=O)CCC(O)(CNC(=O)C=Cc2ccc(Br)cc2)CC1 N1(C(CCCCOC)=O)CCC(C2CC2C(=O)Nc2ccc3c(c2)COC3)CC1 C(=O)(CS(=O)(=O)C(C)(C)C)NC1CC2(CN(C(c3ccnc(C)c3C)=O)C2)OC1 C#CC1(C=C)COCCN1C(C(=O)NCc1ccnn1C)C1CCCO1 c1(C(N2CC(NC(c3c(CC)nc(C)[nH]3)=O)C3(C2)CC3)=O)cc2n(n1)CCCN2 C(CS(=O)(=O)CC(=O)NCC1(F)CCCN(C(=O)C(F)(F)C(O)C2CC2)C1)OC C#CC1CN(C(=O)Cc2csc(CC)n2)CCN1C(C1CC=C(C)CC1)=O C=C(N)CN=C(NCC1(OCC)CCC(C)CC1)NC1CCC1 n1(CC)nccc1C(=O)NC(Cc1cn[nH]c1)C(=O)NCC1CC1c1ccoc1 N1(C(C(=O)NCC(C)C)C2COC2)CCC(OC(C2CCCO2)C2CCOC2)CC1 c1(OC)n[nH]c(C(N2CCCC2CN(C(=O)CC2CC(C)(C)C2)C)=O)c1Cl C12(CNC(c3c(C)cno3)=O)CCC(CN(C(C3CC(=O)OC3(C)C)=O)C1)C2 N1(C(CC=CCC)=O)CC2CCN(C(=O)Cc3ccc(Cl)c(OC)c3)CC2C1 C12(C(=O)NCC3N(C(C4CCSC4)=O)CCCC3)CCCN1S(=O)(=O)CC2 CC1CCC(C)(C)CN1C(C1CC2C=CC1N(C(=O)C1=CCCCC1)C2)=O N1(C(C2CCC(=O)NC2)=O)CCC2CN(C(c3cc(-c4ccccn4)ns3)=O)CC12 N1(C(Cc2c(C)cccc2C)=O)CCCC2(C1)CN(C(c1ccns1)=O)CCO2 O=C1COC2(CN1)CN(C(=O)CC1(NC(C3C4CC5C(C4)C35)=O)CC1)C2 C1(OC)CN(C(c2ccc(=N)[nH]c2)=O)C(C)(CNC(=O)C=Cc2sccc2C)C1 c1(CC(=O)N(C2CCC(NC(=O)Cc3ccc(C)s3)C2)CC)cncc(Br)c1 c1(-c2nc(NC(=O)NC(C=C)C(F)(F)F)sc2)ccc(F)cc1C(F)(F)F N1(C(CCCOC(C)C)=O)CCC(O)(CNC(=O)CCOCC2CC2)C1 c1(C(N2CC3(C)CCC3(C)C2)C(=O)NCCCSCC)cc2c(s1)CCCCCC2 N1(C(c2c(C)nco2)=O)CCCC2CN(C(=O)CS(=O)(=O)NC(C)(C)C)CCC12 N1(C(Cc2ccc(C#N)cc2)=O)CC2(C1)SCCC2NC(=O)Cc1cnns1 c1(C(C(=O)NCCCNC(=O)CC2CC2C2CC2)=O)cc(Cl)c(F)c(Cl)c1 N1(C(c2cc(CC)sn2)=O)CCCCC1C(C)(C)NC(c1ccc(COC)o1)=O C1(CCNCCCNC(C(C)SCC)=O)CCN(C(=O)C(C)(C)C2CC2)CC1 N1(C(=O)OC(C)(C)C)CCOC(C2CCCC2)(CO)C1.C12(C=CCC1)C(=O)N2 C1(NC(=O)COC2CC2)CC2CC1N(C(C1(c3ccc(Cl)s3)CC1)=O)C2 N1(CC)CC(C(=O)NC2CCCCC2NC(c2ccc(O)cc2Cl)=O)CCC1=O N1(C(C2C(=C)CC2)=O)CC2CCC(C1)N2C(c1ccncc1Cn1cccn1)=O Cc1nnccc1C(=O)NCCCOCCC(=O)NCc1cnnn1C c1(N(C(=O)CN(CC)CC2CCCN2C(C)=O)CC)cncc(CC2CC2)c1 c1(C(=O)NC2CN(C(C3(CF)CC(F)(F)C3)=O)C2)occ2c1CCC2 Cc1c(Cl)cnn1CC(=O)NC1CCC(n2cc(CNC3CCOC3)nn2)C1 c1(C(=O)NCCC2OCCCN(C(C(C)O)=O)C2)cccc2c1OCCO2 C1(C(=O)Nc2cc(OC)c(C)cc2)CCC2CCC1N2C(C1CC(=O)N(C)C1)=O N1(CC)C(=O)CCC1C(=O)NCCOCCNC(=O)CC(c1c(C)n[nH]c1C)C c1(NC(=O)OC)ccnc(-n2cc(CNC(=O)C(C3CCCCC3)F)nn2)c1 C1(NC(c2ccc(COC)[nH]2)=O)CC2(CCN(C(c3coc(C(F)F)n3)=O)C2)C1 Cc1ccc(=O)n(CC(=O)NC2CC(CNC(c3ccoc3Br)=O)C2)n1 C1(n2cc(CNC(C3CCCC3)=O)nn2)CCN(C(C2CCC3CC23)=O)CC1 C1(NC(c2cccs2)=O)CC12CC(NC(C1CN(c3nncs3)C1)=O)C2 CC(C)CCC=CC(N1CC(O)(C(C)CNC(=O)Cc2nocc2C(C)C)C1)=O C1(NC(c2ccn(COC)n2)=O)CCCC(NC(=O)Cc2cncc(Cl)c2)CC1 c1(CCCC)cn(CC2CC(NC(=O)CCc3nc(C(F)(F)F)n[nH]3)C2)nn1 C12(NC(CC)=O)CCC(C(N3CCN(C4CCOC4)CC3)=O)(CC1)CC2 C1(CC)CCOCCN1C(C1CCN(C(c2cccc(F)c2O)=O)C1)=O N1(C(C(C#N)=CC2CCC2)=O)CC2C(CNC(=O)C(c3cccc(Cl)c3)O)C2C1 Cc1cccc(COC(C)C(N2CCC(N(C(=O)CSC3CC3)C)CC2)=O)c1 C1(C(N(CC(C)NC(c2cc(C(C)=O)c(C)o2)=O)C)=O)CCc2nc(O)[nH]c2C1 c1(C(=O)NC2C(C(N(C3CCC(F)(F)C3)C)=O)OCC2)cc(C#N)ccc1N c1(NCCNC(C2(C)CCC(F)(F)C2)=O)ncnn2cccc12.N1CC(=O)NC1=O C(C(=O)NCc1ccc(C)c(F)c1)(C(C)CC)N(C(C(CCC)F)=O)C C(=O)(C1CCNc2c(C)cccc21)NCC1C=CCN(c2cc(C)nc(Cl)n2)C1 N1(C(c2cnn(CC)c2C)=O)CCC2CCN(C(C3(F)CCS(=O)(=O)C3)=O)CC12 C12(NC(C3CC(=C)C3)=O)COCCC1CN(C(c1csc3ccccc13)=O)C2 c1(OC(C)C)ccc(C(=O)NCC(O)CNC(c2cocn2)=O)cc1 N12CCC(CC1)C2=O.c1(C(=O)O)cc(CCNC2CCCN2CC(C)(C)O)on1 c1(C(N2CC(C)(NC(COCCC#C)=O)C2)=O)cn2cccc(Cl)c2n1 C1(CC(N2CC(CC)(NC(=O)C(C3CCCCC3)O)C2)=O)CCCCC1O C1(NC(=O)CC2CCCOC2)CC1C1CCCN(C(=O)COc2ccsn2)C1 C1(C(=O)NC(c2c(C)noc2C)C)CCN(C(=O)C(C2CCOCC2)=O)C12CC2 N1(C(C2(CC(N)=O)CCN(C(CC(CC)O)=O)CC2)=O)CCC12CCN(C)C2 CCCC(CCC)C(=O)N1CCCC(C(C)C(=O)N(C2CCC(OC)CC2)C)C1 n1(CC(N2CC(CC(C)NC(C(CC)SC)=O)C2)=O)cnc2sccc2c1=O C(=O)(C(C)(C)C#N)NC1CCC(N(C(CCc2cc(OC)no2)=O)C)C1 Cc1nc(C(N2CCCC2Cc2ccco2)C(=O)NCc2cccs2)nn1C c1(CCCCCC)c(-c2cccc(N3CCNC(=O)C3)c2F)ccnc1O C1(C(=O)NCc2n(C)nnn2)CC2(CCN(C(C3(C#N)CC34CCC4)=O)CC2)C1 CCC(C)(C)C(O)C(=O)NC1CCN(C(=O)C(c2cccc(F)c2)(C)C)CC1F C1(C(=O)NC2CC(NC(C3N(C(C)=O)CC(O)C3)=O)CC2O)Cc2nccn2C1 CC(C)CC(C(=O)N1CCCC1CC1CC1)NC(=O)C=Cc1cocn1 c1(CC(=O)NC2CCN(C(c3cc(CCC)n(C)n3)=O)C2C)cc(C)ccc1C C(=O)(CC(C(F)(F)F)c1c(Cl)cccc1Cl)NCCCCNC(C(CC)O)=O Cc1ccc(CC(=O)NCCNC(=O)CC(C)C)c(F)c1F.c12ccccc1N2 N1(C(c2c(C)ncnc2O)=O)CCC2(C1)CN(C(=O)CC1(O)CCCCC1)C2 C1(CN(C(CC(=O)NCC)=O)C)CCCCN1C(C1OC(C)CC1C)=O c1(C(=O)NC(C2CCN(C(C(CC)COC)=O)CC2)(C)C)ccccc1S(C)=O N1(C(C(COC)C)=O)CC2CCC1C(CNC(=O)CCCCC1CCCCC1)C2 C(CCCCCNC(c1cc[n+]([O-])cc1)=O)N(C(=O)CCCCNC(N)=O)C C12(C(=O)NC(C)CCNC(C3(C)CCCOC3)=O)C3C4C1C1C2C3C41C(N)=O c1(C(C)=O)ccc2nc(NC(=O)NCC3CC3c3ccc(F)c(F)c3)sc2c1 Cc1cc(C(=O)NC2C3CCC2N(C(c2c(C)ncnc2C)=O)C3)ncc1CO C1(C)(CCC(F)(F)F)c2nnnn2C2CC(C2)O1.c1(C(=O)OC)cncn1C(C)C C(=O)(C(C)CCC(C)(C)C)NC(CC=C)CNC(=O)CSCCC(C)C C12(CCNC(c3cn4ccnc4s3)=O)CCC(C1)N(C(=O)C1=COCCC1)C2 C(=O)(C(C)(C)C(=O)N1CCC2(CC2C(=O)NCc2csc(C)c2)C1)NC N1(C(C(C)N(C(C(CC)C(=O)OC)=O)CC)=O)CCC2(CCSC2)C1 C(=O)(CCC(C)(C)C)NC1CC(C(=O)NC(CCSC)CO)C1 C(C)(C)(CCCC(=O)NC1CCC(O)C(O)C1)NC(c1ccc(C#C)o1)=O C(=O)(CC(C)C(C)C(C)C)N1CC(C)N(C(c2cnn[nH]2)=O)CCC1 C1(n2cccn2)(C(=O)NC(CNC(CC(C)c2ccco2)=O)C)CCOCC1 CC1CN(C(=O)NCC2CCOC2)Cc2ccccc2O1 C12(C(N(OC)CCO)=O)CCC(CC1)N(C(c1c(C)cccc1C)=O)C2 c1(NNC(=O)NCC(C)(C)C2C(CC)C2)ccc(N(C)C)nc1.c1(S)ccccc1.SS C1(C(=O)NC2COCC2O)C2CCC(CC2(F)F)N1C(=O)Cn1nccn1 Cc1c(C(=O)NCCN(C)C(C2CCCC23CCC3)=O)sc2ccc(F)cc12 C1(C)(NC(C(COC)OC)=O)CCCN(C(c2ccc(C(C)(C)C)o2)=O)C1 N1(C(c2cn(CC=C)nn2)=O)CCCC(F)(CNC(=O)CC2CCCC23CC3)C1 CCCC(C(O)C(=O)N1CCOCC1CC1CCC1)NC(C1CCC(C)CC1)=O N1(C(c2ccc(COC)[nH]2)=O)CCC(CCNC(=O)CN2CCSCC2)CC1 C1(CNC(C2CN(C(=O)Cn3cc(C(F)(F)F)nn3)C2)=O)CCCCS1 CCC(C)(C)C(=O)N1CC(N2CC(NC(=O)CSCC3CCCO3)CC2=O)C1 C1(CN=[N+]=[N-])CCN(C(=O)Nc2ccsc2CNC2CCC2)CC1 C1(C(=O)NC2CC(F)CN(C(=O)CCn3cc(Cl)cn3)C2)CC2CC(O)C(C1)C2 CC(C)(C)CC(=O)NC(C(=O)NC1CCCCC1CO)c1cccs1 c1(C(=O)NCCCCC(C)NC(c2cn3ccnc3s2)=O)nc2ncccn2n1 C1(NC(CN(CC(C)OC)C)=O)CC2CC1CC2NC(c1ncoc1C)=O Cc1c(CCC(=O)NC(CNC(=O)Cc2ccccc2Br)CO)cnn1C N1(C(C(CC2CCCC2)NC(COC(C)=O)=O)=O)CC2CCCCCC2C1 C12(NC(CC=CC=C)=O)CCCC1N(C(c1sc(Br)nc1C)=O)CC2 C1(NC(c2c(CC)nco2)=O)CCC2(CCCN(C(=O)C(F)(F)C(C)(C)O)C2)C1 N#Cc1c2c([nH]c(=NC(=O)NOCC(O)C(F)(F)F)c1)CCCC2 C(=O)(C(C)(C)C(C)(F)F)NCC1CN(C(c2cc(C)ncc2)=O)C(C)C1 c1(CNC(C(C)C2CC2)=O)ccc(CNC(C2CC2C)=O)c(F)c1 c1(CC(=O)NCCOCCN(C)C(C23CCCC2CC3)=O)nc2ncccn2n1 N1(C(C(CCCC)NC(N)=O)=O)CCCN(C(=O)Cn2nnnc2C)CCC1 N1(C(C2N(C)CC2)=O)CC(O)(C2(CNC(C34CC(C3)C4)=O)CC2)C1 N1(C(CC2C(c3n(C)ncc3)OCC2)=O)CC(CO)c2ccccc21.[nH]1ccnn1 Cc1ccc(CNC(=O)C(C)CNC(=O)COCc2nc[nH]n2)nn1 c1(C(=O)OCC(=O)NCCc2ccc(F)c(F)c2)cc(Cl)cc(Cl)c1 N1(C(C2C(CCC)CCC2)=O)CCN(C(=O)CCC2CCC2)C2(CC2)C1 Cc1ccc(C(N2CC(C)(OC(C)C(=O)NC3(C(=O)O)CC3(F)F)C2)=O)s1 c1(C(N2CCC(N(C(=O)C(C)SC)CCC)C2)=O)ccc(SC)cc1OC C12(CNC(CC(C)c3ccco3)=O)CCCCC1N(C(c1cc(O)no1)=O)CC2 c1(C(=O)NC2CN(C(c3ccc(CC)cn3)=O)CC23CC3)cccc2nccn12 N1(C(C(CCC)CNC(c2ccns2)=O)=O)CC(C)OC(C)(C)C1 c1(NC(C)=O)cccc(C(=O)NCCCNC(=O)C=NOC)c1 c1(C(C)C)ccc(NC(=O)CN2CCN(C(=O)C(C)CN(C)C3CC3)CC2)cc1O C(C(C(C)(C)C)NC(=O)CCc1cc(C)n(C)n1)NC(C1C(CC)OCC1)=O c1(OC)c[nH]c(C(N2CCC(NC(=O)COc3cn[nH]c3)C(F)C2)=O)cc1=O CC1CC(C)CCN(C(c2coc(CNC(C34CCC(CC3)CC4)=O)n2)=O)C1 C1(OC)C=CCN(C(CCC2(C)CC2)C(=O)NCC2CCOC2)C1 n1(CC)ccnc1C(=O)NCC1CCC1NC(=O)C(C)COC c1(C(c2n(C(CC)C)nnn2)NCCc2ccc(F)cc2Cl)cc(Cl)ccc1Br N1(C(C(F)=CCC)=O)CCCC12CCN(C(=O)Cc1cccc(C(F)(F)F)c1)C2 Cc1ccc2[nH]c3c(c2c1)C(Nc1cc(N(CC(C)C#N)C)ncn1)CCCC3 CCS(=O)CC(=O)NCC1CC(F)(CNC(C2(n3ccnn3)CC2)=O)C1 Cc1c(C(N2CCc3ccccc3C2)=O)[nH]c2c1CCCC2 c1(OC)nc(Cl)ccc1C(N1CC(NC(=O)CNC(=O)C2CC2)CC(C)C1)=O N1(CC(=O)NC(C(C(C)C)NC(=O)CCC(C)(C)F)C)C(=O)CC(C)(C)C1=O c1(C(N2CCCC(C(N3Cc4ncsc4C3)=O)C2C)C)ccc(F)cc1F c1(C(=O)NCC2OCCN(C(C3CC4(CC(=O)C4)C3)=O)C2)cccc2cc[nH]c12 C1(CNC(c2c(C)con2)=O)CCC2(CN(C(C3CCCC3C(=O)OC)=O)C2)O1 c1(C(=O)NC(C2CCCN(C(=O)CCc3ccccc3O)C2)C)cccc(CF)c1 c1(C(c2n(C3(C)CC3)nnn2)Nc2ccnc3ncnn23)ccc2ccnn2c1 N1(C(C(CC)SC)=O)CC23CCCC2(C1)CN(C(=O)CC1CC=CC1)C3 C1(NC(c2cc(-c3ccco3)no2)=O)C2CCN(C(c3ccsn3)=O)CCC12 c1(N2CCN(C(C(COC)C)=O)CC23CC3)ncc2ccc(Br)cc2n1 N1(C(C(C)C2CCCC2)=O)CC2CC2(CNC(c2ccnc(OC(F)F)c2)=O)C1 C1(CC)(CNC(=O)CCCN(C(=O)C(CCC)OC)C)CCC(=O)N1 CC1CCN(C(c2cc(CCNC(=O)CC3C=CCC3)on2)=O)CC1O N1(C(=O)CC2CN(C(c3ccc[n+]([O-])c3)=O)CCO2)CCCC12CCOCC2 OC1CCc2sc(CN=c3[nH]c(-c4ccc(F)cc4)cs3)cc21 N1(C(c2cccc(C#C)c2)=O)CCC2(CC1)CC(C)N(C(=O)CNC(N)=O)C2 C1(NC(C#CC(C)(C)C)=O)CCN(C(=O)C(F)CC2CCCCC2)CC(O)C1 c1(OC)cc2c(C(=O)NC(CNC(c3cscn3)=O)CSC)cc1[nH]2.C(F)F CC1(C)CN(C(=O)Cc2ccc[nH]2)CC1C(N1CC2C=CC2C1)=O N1(C(C=CCCC)=O)CCC1C(=O)NCC(F)F Cc1ccc(F)cc1CN1C(=O)NCc2n[nH]c(n2)C1.C(C)(C)(C)OC(=O)N C1(C(=O)NC2CN(C(C3(C(=O)OCC)CC3)=O)C3CC23)CCC(C(N)=O)CC1 N1(C(C(C(C)C)OC)=O)CCC2(CC1)CC2C(=O)NCc1cnn(C)c1 N1(C(C2(c3cccs3)CC2)=O)CCCN(NC(C2CSC2)=O)CC1.C12CCCC1C2 CC1(C)C2CC1CC(=O)N2.C1(C(=O)NC2(CC3CCC3)CC2)CCCC1O Cc1cc(C)c(C(N2CCC2CNC(c2nc(C3CC3)cs2)=O)=O)c(=O)o1 C1(C2CC2)(CC(=O)NCC(CNC(=O)C(F)n2ccnc2)OC)CC1 N1(C(c2cccc(C)c2)=O)CC2CN(C(c3cc(C4CC4)ncn3)=O)CC2C1 C=CCC(CNC(=O)CC1CC1(C)C)C(=O)NCC1CN(C(C)C)C1 c1(C(=O)NC2C(NC(C3CCC(=C)CC3)=O)CCCC2)cc(CCO)ccc1O C12(CNC(CCCC#CC)=O)CN(C(C34CC(C)C3C4)=O)CC1CCO2 C12(C(=O)NC(CSCC)C)CC(CCO1)N(C(=O)CC1(SC)CCC1)C2 N#CCCCCCC(=O)NCC1CC(F)(CNC(=O)CSC(F)(F)F)C1 C12(C(=O)OCC)CNCCC1CN(Cc1cc(F)ccc1I)C2 c1(OC(c2ccccc2)C)c(C(F)(F)F)cccc1Cl.C1C(O)CC(=O)OC1=O CC(C1CC1)=CC(=O)NC(C(=O)N(CC(C)O)CCN(C)C)c1ccco1 c1(N2CC(C(=O)OC(C)(C)C)OCC2)nccc(=NCc2cc(Cl)cc(Cl)c2)[nH]1 N1(C(C(CC)NC(C)=O)=O)CC2CC1CC2NC(=O)Cn1cncc1.C(C)(=O)OC C1(NCc2c(C(=O)OC)scn2)CCCN1NC(=O)CN1CCCCC1 C=CCCCC(=O)NC1CCCC(c2cn(CC3CCCO3)nn2)C1 c1(C(C)(C)C)ccncc1C(=O)NCCNC(C1CCCC(O)C1)=O C1(NC(c2nc(C(=O)OC)sc2)=O)CC2(CNC(C3CCS(=O)CC3)=O)CC1C2 CC(C)(C#CC(=O)N1CC(C#N)(C(N)=O)C1)CNC(=O)CCc1nccs1 N1(C(CCCC=C)=O)CCC(CNC(=O)CN(C2CCCC2)C)CC1C1CC1 N1(C(COCC)=O)CCC(CNC(C2(C3CCCO3)CCC2)=O)(COC)CC1.C(F)(F)F c1(C2CCC(C(=O)NC3CN(C(Cc4c(C)scc4)=O)C3)C2)ccc(F)cc1 Cn1c(C(=O)NC23CC(C2)N(C(C2CCCC(=O)O2)=O)C3)c2n(c1=O)CCCC2 C1(NC(C(C)OC2CCCC2)=O)CN(C(=O)C(C)(C)c2ccccn2)CC1F N1(C(CCSCC)=O)CCCC2(CCCN2C(C2CCC(C)CC2)=O)C1 Cc1c(Br)ccc(NC(C2CCC3(CN(c4ccncn4)C3)O2)=O)c1C c1(C(N2C(CNC(C(C)Cn3cccn3)=O)C=CC2)=O)ccc(C2CC2)cc1 c1(C(N2CCC(N(C(C(C)C)=O)CCO)C2)=O)ccc2c(c1)CCC(O)C2 C1(NC(c2cc3c[nH]nc3s2)=O)CCN(C(=O)CCF)C(c2ccccc2)C1 C1(C(=O)NC)CCC(C2CCCC2)CC1.C1(C(=O)NCC2(OCC)CC2)CCC1 C(=O)(C(F)(F)C1=CCOCC1)N(CCCCC)C(c1ccc(C)nc1C(=O)OC)=O C(CCCCn1cc(CCO)nn1)NC(CCOCC(C)C)=O Cc1c(Cl)ccc(C(NCC(C2(C)CC2)N(C(=O)CCNC(=O)CO)C)=O)c1N C1(CNC(Cc2cnc(C)o2)=O)C2CCCC1N(C(C1(C)CCN(C)C1=O)=O)C2 n1(CCCC(=O)NC(CNC(C(C=C)(C)CC)=O)C)c(=O)n(C)c2ccccc12 C(=O)(CCCCC(C)(C)C)N(CCN(C1(CC)CC1)CC)NC(C(CC)CC)=O Nc1cc(F)cc(C(=O)NC2CC(NC(C3CCCC(C(F)(F)F)C3)=O)C2)c1F N1(C(c2nncc(CCC)c2)=O)CC(N(C)C(c2c(C)coc2C)=O)C(C)(C)C1 CC1CCC=C1C(=O)NCC1C2CN(C(c3ccc(C(F)F)o3)=O)CC12 C(=O)(CC1OCc2ncccc21)OCC(C)C(C)(C)C Cc1nn(C)c(Cl)c1CC(=O)NCCC1CCN(C(C2(C)CS(=O)(=O)C2)=O)C1 c1(C(N2C(C(=O)NCc3cc(C)on3)CC(O)C2)=O)cc(O)ccc1I C(=O)(C(N)C1CCc2ccccc21)NCCc1cc(OC)nc(OC(C)=O)c1 c12cc(F)ccc1C2.C=CC1(CS(=O)(=O)OCO)CCC1 Cc1ccc2c(C(N3CC4CC3(CNC(C3(C)CNC(=O)C3)=O)C4)=O)c[nH]c2c1 N#CC1CN(C(=O)Cc2c(Br)cccc2Br)CCN1c1ccncn1 C(CCCC(=O)NC(CC1CC1)CO)N(C)C(C1(C#N)CC(C)C1)=O C1(C(N2CC(CNC(CCCC(C)C)=O)OCCC2)=O)CC2CCCCCC12 C(C(=O)NCCC1(NC(=O)C(C)C2CCC2)CCC1)(C1CC1)OC c1(C(=O)NCCC2N(C(C3(F)C(C)OCC3)=O)CCC2)cc(O)ncc1Br c1(C(N2CCCC(OCc3cn(CCN(C)C)nn3)C2)=O)cccc(F)c1Cl c1(CC(C(N2CCC(N(C(=O)CCNC(N)=O)CCC)C2)=O)O)cccc(Cl)c1 c1(C(=O)NC(C)(CNC(c2cc3scnc3[nH]2)=O)CO)nc(O)nc(O)c1F CC(C)CCCCC(=O)N1CCOC(CNC(C2(C#N)CC3(CCC3)C2)=O)C1 N1(C(CNC(C)=O)=O)CCCC(C)(N(c2ccco2)C(C2(C3CCC3)CC2)=O)C1 Cc1ccc(C#N)cc1C(N1CC(C)(C)C1C1CCN(C(=O)C=CI)CC1)=O CCC(CO)C(=O)NC(C1CN(Cc2nncs2)C1)C.c12csc(n1)C(=O)N2 C#Cc1ccc(CNC(=O)C(C2(O)CCC2)NC(c2ccc(C(N)=O)[nH]2)=O)cc1 C(=O)(C1=NN2CCCN=C2N1)NCCC(C)NC(Cc1cc(CC)nn1C)=O c1(OC)ncc(C(N2CC(NC(C3(CF)CC3)=O)C(SC)C2)=O)cc1Br N1(Cc2c(-c3cccc(C#N)c3)n[nH]c2)CCCC2(CC(NC(=O)CCBr)CO2)C1 C1(NC(c2cccc(O)n2)=O)C2CC3CN(C(=O)CCc4cncs4)C1C3C2 C(=O)(C(C)CC#N)NC(C(CO)NC(CC=C)=O)C CC(C)CCCCCC(=O)N1CC2(CCCC2)C1C(N1CCCC(CCO)C1)=O C1(CN(C)C)CN(C(=O)OC(C)(C)C)CC(C)(C)C1.C12(CCCC1)C(=O)NC2 c1(C(N2C(C)C3CC2C3NC(c2ccsn2)=O)=O)cc(F)c(F)c(F)c1N N1(CC(=O)NC(CCCCC)C)CCC(NC(c2nccnc2C)=O)C(C)(C)C1 c1(C(C(=O)NCCCC)N(C2CCC2)C2CC2)oc(C(=O)O)cc1Br C=C(C)CCC(C)N=c1nc(N2CCOCC(C)C2)c2c([nH]1)CSC2 CC(C)(O)C(=O)N1CCCC1C(O)C(=O)NCCCc1ccccc1 C(C(CCNC(=O)CCC1OCCO1)OC)NC(C1CN(S(CC)(=O)=O)C1)=O N1(C(C2C(=C)CC2)=O)CCC(CCNC(C2C3COCC23)=O)C(F)(F)C1 c1(C(=O)NCCC)cn2ccc(F)cc2n1.C12CN(C(=NC)NC1)C2 C#Cc1nc(C(=O)NC2CC2CNC(=O)C(C)C2CCCC2)cs1 C1(C(NNC(C2Oc3c(C(=O)OC)cccc3C2)=O)=O)COc2ccccc2O1 N1(CC)CCOC(C(N2CC(O)(CN(C(=O)C(=O)NCC3CC3)C)C2)=O)C1 c1(OC)c(F)ccc(CN(C)C(=O)NC(c2cccc(Cl)c2)CF)c1F c1(NC(c2ccc(CCC(=O)Nc3cncs3)[nH]2)=O)cnc(I)cn1 C1(NC(c2cnc(S)nc2)=O)CC2CC(NC(=O)C(F)CC3CC3)C1C2 C#Cc1cc(C(=O)NCCOCCCNC(=O)C(COCC2CC2)CC)cc(F)c1 C1(C)(C(=O)NCCC2(CNC(C(COC)NC(C)=O)=O)CC2)C(C)(C)C1(C)C CCC(C(=O)NC(C1CCCN1C(c1ccoc1Cl)=O)C)Oc1ccccc1 Cc1nn(C)c(C)c1C(C)C(=O)NC1(CNC(=O)CCC(C)CN(C)C)CC1 c1(SC(C)COC)nc(-c2cccc(Cl)n2)nn1CCC1CCCCC1 N1(C(CSc2n(C)ccn2)=O)CCC2CCN(C(=O)CCc3ccncn3)C2C1 c1(NC(=O)CC2CN(Cc3ccccc3C(=O)O)CCO2)cc(F)c(F)cc1F C#CC1CCC(C(=O)N(CC(C)O)CCNC(=O)CCC=C(C)C)CC1 N1(C(CCSC)=O)C(C(=O)NC(C)CC2CCC2)C2CC(O)C1C2 c1(C(N2CC(NC(CC(C)(C)C3CC3)=O)C(F)C2)=O)cc2n(n1)CCCCO2 Cc1csc2cc(C(N3CCCC(CN(C(=O)CCS(C)=O)C)C3)=O)[nH]c12 C1(NC(CCCN(C(C)=O)C)=O)CCN(C(=O)C2=CCCCO2)CC1O CC(O)(CC(=O)NCCCCNC(C12CCCCC1CCC2)=O)C(F)(F)F CC1CN(C(c2ccc(Cl)cc2N)=O)CCC1C(=O)NCC1(C(N)=O)CC1 N1(C(c2nc(COc3ccccc3)oc2C)=O)CCN(C(C2(OC)CC2)=O)C2CC12 C1(O)(CCNC(C(C)NS(CCC)(=O)=O)=O)CCCN(C(C2(C#N)CC2)=O)C1 C#Cc1ccc(C(=O)NC(C(=O)N(C2CCCC2)CCOC)C2CCC2)o1 C1(C(N2CC(CC)C(C(N3CC4C(N(C)C)C4C3)=O)C2)=O)CN2CCC1CC2 Cc1c(C(N2CC=CC2C(=O)NCCCC2C=NNC2=O)=O)[nH]ccc1=O c1(N2CC(CN(C(CC(CCC)O)=O)C)OCC2)ncnc2c1CCO2 c1(C(=O)N)ccc2occc2c1.c1(C(=O)N(CC2(C)CC2)C)n[nH]cc1C1CCCC1 C1(NC2C(c3c(C)cccc3)CCNC2)CC2(CCCCC2)C1 N1(C(CC2C(C(=O)OCC)C2)=O)C2CC1CN(C(C1CCC(C)=C(C)C1)=O)C2 C(C)(CC(=O)NC1(C)CCN(C(=O)Cn2cnc(C(N)=O)n2)C1)(C(F)F)N(C)C c1(OC)c(Br)ccc(NS(=O)(=O)Cc2c(F)cccc2Cl)c1C c1(N2CC(C)(CC(=O)NCC(C)CO)C2)ccc([N+](=O)[O-])cc1 c1(C(=O)NCC2OCCN(C(CC(C)c3ccco3)=O)C2)cc2c(ncn2C)[nH]1 C1(C(=O)NCCOCCN=[N+]=[N-])(CNC(CC2CC(C)C2)=O)CC12CCC2 C1(C(=O)NC(C(N2CC(C)(OC)C2)=O)COC(C)C)CSCC(=O)N1 CC1(C)CC(NC(c2cc(C#N)cs2)=O)CN(C(=O)CCc2ccc[nH]2)C1 C1(N(C(=O)CC(C)C)CC)CCCN(C(c2cnn(C3CCOCC3)c2)=O)C1 N1(C(CCOCCNC(CN(CCC#C)C)=O)=O)CC(OC)CCC1C c1(NCC2(CNC(C3C(CC)OCCC3)=O)CC2)c(Br)cccc1[N+](=O)[O-] C1(NC(CSC(C)(C)C(F)(F)F)=O)CCCCN(C(=O)CC(=O)OC(C)(C)C)C1 c1(CNCC2N(C(c3n(C)ncc3)=O)CC=C2)cccc(F)c1C(F)(F)F c1(CC)c(NC(=O)CCN(CCO)C(c2snnc2CC)=O)cnn1CC CN1C(=O)C(CC(=O)N(O)Cc2cn(-c3ccccc3)nn2)c2ccccc21 N#Cc1cc(CN2CCCC2c2nc3ccccc3[nH]2)ccc1Br Cc1cnc2n1CCN(C(C1CCCCC1CNC(=O)Cn1cnnn1)=O)C2 CCC(C)(CO)C(=O)N(CC(C)(C)CC1CN(C(c2cccc(=O)n2C)=O)C1)CC N1(C(CSCCC)=O)CCCC(NC(C2CC(C)(C)C2)=O)CCC1 C(Cc1ccccc1)(CCNC(=O)Cc1cnccn1)NC(C1(N(C)C)CC1)=O c1(CCC(=O)NC2(CNC(C3(C=C)CCC3)=O)CCC2)cccc(F)c1 c1(C(=O)NCCNC(=O)C2CCOc3ccccc32)ccc2c(c1O)CCCC2 CC(C)(CC(=O)N1CC2CC2(NC(c2cnn3c2CC(F)(F)C3)=O)C1)C(F)(F)F C#Cc1cccc(CN2CCCC(n3cc(CNc4ccccn4)nn3)C2)c1 N1(C(c2scc(C)c2C)=O)CCC(NC(=O)CSC(F)(F)F)C(F)(F)CC1 C=CCCN=C(NCCc1c(C)n[nH]c1C)NCc1ncccc1OC C(=O)(C(C)(C)CC(F)F)NCC(C1CCC1)NC(C(CC)(C)CC)=O C1(CCNC(c2cn(CC)nc2)=O)CN(C(C2CNC(=O)CC2C)=O)CCCO1 C1(S(=O)(=O)N2CCCC2C(C)(C)C(=O)O)(COC)CCC1 C(=O)(C(C(C)NC(=O)CSC(C)(C)C)C(C)C)N1CC(F)(CC)C1 c1(C(N(C2CCN(C(C3(CF)CC(F)(F)C3)=O)CC2)CC)=O)nc(O)sc1C C=CCCN=C(NCc1cccc(C#N)n1)NCC1(c2ccccn2)CCCC1 C(CN=c1[nH]c(=NCc2cc(=O)cc[nH]2)c2ccccc2[nH]1)N(S(C)(=O)=O)CC C1(NC(C=CCN(C(C2C(C)SCCC2)=O)C)=O)CCC(N=[N+]=[N-])CC1 C1(NC(c2ccno2)=O)CCN(C(C2CC2c2cccc(F)c2)=O)CC(O)C1 c1(C(=O)NC(C)CCCCNC(=O)C=CC2CCOCC2)ccc2nsnc2c1 Cc1n[nH]c2cnc(C(N3CCC(NC(c4cc(C(N)=O)cs4)=O)C3)=O)cc12 c1(OC)cc(C(=O)NCCCCCNC(C2CC2(F)F)=O)cc2c1OC(C)C2 C12(C(=O)NC3CCN(C(=O)COCC(F)F)CC3F)CCC(CO)(CC1)CC2 CCCC(C)(CC)NC(=O)C(=O)NCc1nccc(C(=O)OC)n1 C12(NC(C3C(=C)C3)=O)CCCCCC1N(C(c1coc(-c3ccsc3)c1)=O)CC2 CN=c1[nH]c(=NCC(C(C)(C)C)c2ccccc2)[nH]c(=NCC)[nH]1 c1(-n2cc(CN(CCC(=O)OC)Cc3cc(I)c[nH]3)nn2)cc(NC)ccc1F CC(F)(CC1CCCC1)C(=O)OCC1CCCCCC1.N12CC(C1)C2=O N1(C(Cc2[nH]c(=N)sc2)=O)C2CCC1CN(C(c1cc(F)oc1C1CC1)=O)CC2 N1(C(C2CCC(=C)CC2)=O)CC(C(=O)NCC2CC2(F)F)C2(CC2)C1 N1(C(C(COC)(F)F)=O)CCCC2(CCN(C(c3cnc(S)nc3)=O)CC2)C1 c1(C(N(CC(CC)NC(c2scc(C)c2Br)=O)CC)=O)cnccc1C C(N=c1cc(Cl)nc(C)[nH]1)C1C(NC(CN(CC)CC)=O)C2(CC1)CCC2 N1(C(C)=O)CCCc2cc(C(=O)N(CCCNC(=O)CCN3CCC3)C)ccc21 c1(C(N2CC(CC)N(C(=O)C3=C(C)CCC3)CC2)=O)cc2nc(=O)ccn2[nH]1 CN1CC2OCCN(C(=O)C(CO)NC(c3ccco3)=O)C2C1 CC1CNC(=O)CN1C(=O)NCCNC(=O)C(c1cncnc1)N CCC(O)(CC)CCNC(=O)NCC(c1nccn1C)(C)C N1(C(=O)OCCNC(C(COC)OC2CCC2n2ccnc2)=O)CCC(C)CC1 c1(NC(=O)CC(F)F)ccc(CCCNC2(CO)CCCC2)cc1 C(=O)(C(C)CCO)N1CCC(CCNC(c2c(-c3cn(CC)nc3)n[nH]c2)=O)C1 N1(C(C(C)(C)N(C)C)=O)CC23CCCCC2(C1)CN(C(c1cccnc1O)=O)C3 c1(OC)ccc(C(F)(F)F)cc1C(N1CCCC1)=O.C1(C(=O)N)(CN)CC1(F)F CCC(C)CC(N)C(=O)NC(Cc1cccc(OC(F)(F)F)c1)CO C1(C(=O)NCCCC2(NC(c3c(C)coc3)=O)CC2)Cc2ccccc2S1 c1(C(N2CC(CCNC(=O)CC3CC3(C)C)(OC)C2)=O)ccnc2c1ncn2C N1(C(C=CCOCCOCCOC)=O)CCC(C#N)(CC(C)C)CC1 C1(CC(C)NC(c2cc(Cl)c(Cl)s2)=O)CC2CCC(C1)N2C(C1CCN(C)C1)=O Cc1ccc(OC(C)C(=O)NCC2(O)CN(C(C3(C)CC4CC4C3)=O)C2)cc1 C(CCCN)(C(=O)O)NC(c1cnn(CC)c1C(F)(F)F)=O N1(C(C(CC)(C)F)=O)CC2(C1)CN(C(c1cc(C)ns1)=O)CCO2 C1(CCC)CN(C(=O)C(F)CC)CC1NC(C1CN(C)C(=O)N1)=O O=C(C1CCCc2ncnn21)N1CCC1c1cn(C2CCOC2)nn1 N1(C(c2ccc(C(C)=O)nc2)=O)CC2(CCCN(C(=O)C=C(C)C(C)(C)C)C2)C1 C1(NC(c2c(COC)cccc2)=O)CCN(Cc2cccc(C#N)n2)CC1O c1(C(N(CCNC(C2C(C)SCCC2)=O)C)=O)cccc(C(C)(C)C)c1O c1(C(=O)NCCNC(c2c(CC)ocn2)=O)sc(C)c(Br)c1C.C1C(=O)N1 c1(NC(C2N(C(c3nccc(OC)c3)=O)CC(C)C2)=O)ccc2[nH]nc(I)c2c1 C1(N(C(CCc2cc(C)[nH]n2)=O)C)C2CN(C(C3CC=CCC3)=O)CC12 N1(Cc2c(OC)cc(C)cc2)CCC(C(=O)Nc2ccc(OC)nc2)C(C)(C)C1 C1(NC(C(COC)(F)F)=O)CCC(C)N(C(=O)C(C)CSC)C1 C(=O)(CC(C(C)C)c1ccc(F)c(F)c1)NCCCN(C(c1cnc(C)s1)=O)CC c1(C(N2CCCN(C(=O)CC3CC4CC4C3)CC2)=O)cc2cccnc2o1 C1(CNC(c2cccc(C3CCCC3)c2)=O)CN(C(=O)COC(F)(F)F)CC1(F)F Cc1ccc(C(=O)NCC2COC(CNC(c3ccncc3Br)=O)C2)nc1 N1(C(c2n(CC=C)ccn2)=O)CCC(C)C1CNC(c1ccoc1Cl)=O c1(C(C(=O)NCCN(C(COC)C)C)C)ccc(I)cc1 c1(N(C(=O)NC2CCCCN(C)C2)CC)ccc2c(c1)CCC2 c1(C(=O)NCC2CC(NC(CCCOCC)=O)C2)cnn2c1C(C)CCC2 N1(C(=O)CC2CCCCC2O)CC2CCCN(C(C3CSCCS3)=O)C2C1 CCCC(CCC)CC(=O)N1CCC2CCN(C(=O)C3=NOC(C)C3)C2C1 C1(CNC(=NC)NCCc2cccnc2)CCOC(CC)C1 C1(C(N(CCNC(c2snnc2C2CC2)=O)CC2CC2)=O)CC2(CO1)CC(F)(F)C2 c1(C(C)(C)C2CC2)nc(C2CCCO2)n(CCN2CCOCC2)n1 c1(C(N2CC(O)C(F)C2)=O)cnc2c(C3=CCC(O)CC3)cnn2c1 CC1CN2CCN1C(C(=O)NCC(C)(C)NC(C1C(C3CC3)C1(F)F)=O)C2 C1(CNC(C(COCC)n2cc(CO)nn2)=O)CCC2(CO1)CC(O)C2 Cc1cnc(C(C)NC(=O)CCN(CCO)C(c2ccnn2C(F)F)=O)o1 N(C(=NCC(C)N1CCCCC1C)NCc1ccc2ncsc2c1)C(C)C Cn1c(=O)c(C(N2CCN(C(C3(CO)COC3)=O)CC2)=O)c(O)c2ccccc12 CC1(C)CC(CNC(c2nc(-c3cnn[nH]3)no2)=O)N(C(=O)CCS(N)(=O)=O)C1 c1(SC(=O)CN2CC(C3CCCO3)C2)ccc2c(c1)CCCC2 c1(OC)ccc(C(C)C(=O)N(CCCCN(C)C(C2CN(C)C2)=O)C)cc1F N1(C(COCC=C)=O)CCN(C(=O)C(C)(C)C)CC1CS(C)(=O)=O C1(C(NNC(C2N(CC)CC23CCCC3)=O)=O)CC1C1CC(N=[N+]=[N-])C1 C1(Nc2ncc(C(=O)OC)s2)CCCC(N2CCOCC2)C1 Cc1nc(Br)sc1C(=O)NCc1cn(C2CCN(C(=O)C(C)C)C2)nn1 N1(C(C(=O)NC2N(CC3(C=C)CCC3)CC2)=O)CCC2(CCOCC2)C1 C1(CCC2N(C(C(COC)O)=O)CCC2)CCN(C(C2(N(C)C)CC2)=O)CC1 CC1NC(=O)CCC1NC(=O)CC=CCNC(=O)CCCC1CCCC1 C=CCC(CC=C)C(=O)N(C1CCC2CN(C(C3CCCOCC3)=O)CC12)C C1(NC(C(C(=O)OCC)F)=O)CC2(C(=O)NCCC(C)C(C)C)COC1C2 C1(NC(c2scc(C)c2Cl)=O)CN(C(c2ccnc(C)c2N)=O)CCC1C C(=O)(CC(O)C(C)C)N1C(COC)(CNC(c2n[nH]cc2C)=O)CCC1 c1(COC)ccc(-c2cn(C(C)CNC(C3CCS3(=O)=O)=O)nn2)cc1 C1(C)CC2(C1)CC2C.c1(C(C(C)C)NC(C2(C)CC2)C)nnnn1CCC1CC1 N1(C(CCC2CCC(NC(=O)Cc3cnccn3)C2)=O)CCCOCC1 CCC(CC)CC(=O)NC1CC2CC(C(=O)NCC(CC)(CC)CC)CC12 C1(OCC(N2CC(N(C(=O)Cc3ccsn3)C)C(F)C2)=O)CCC(F)(F)CC1 C1(CCCCC)CCC(C(=O)NCCN(C(C2CCCS2)=O)CC2CC2)O1 N1(CC)CCC(NC(=O)Cc2cnccc2C)CC1.C1(C)C(=O)N1CC(C)C C1(C(=O)NC(COCC)(C)C)CCCCCCN1C(c1oncc1CC)=O C(=O)(CC(C)(C)C(F)F)N1CCC(NC(c2n(C=C)ncc2)=O)(CF)C1 c1(C(N(C(C(=O)N(CC#CC)CC#C)C2CC2)C)=O)cccnn1 CC(CCC(=O)NC1CC2(CC2)C1)NC(c1ccc(Cl)s1)=O c1(N2CC(CC(C)NC(C3CSC3)=O)C2)cc(OC(F)F)c([N+](=O)[O-])cc1F S(=O)(=O)(c1ccccc1Cl)N1CC(NC(c2c(C)n[nH]c2)=O)C2(C1)CC2 [N-]=[N+]=NC1CCC2(C(N3CCCCC3CNC(c3nccnc3N)=O)=O)CC12 C1(NC(=O)CSCC(F)F)C2CN(C(=O)Cc3cncs3)CC12 CC(O)C(C)C(=O)NCc1ccc(CNC(c2c(Cl)cnn2C)=O)cc1 c1(C(NC(C(=O)NCC(CCOC)O)=O)Sc2ccccc2)cc(F)ccc1F C12(NC(CC=CCC)=O)CC3CCC(C1C2)N3C(c1cccc2[nH]ncc12)=O CCCCCCCC=CCCCOC(c1onc(C)c1OC)=O C(C)(C(=O)NOCC)N(CCC)C(c1coc(C(C)C)n1)=O c1(C(=O)NC2CC(COCCOCC#C)C2)ccc(NC(C)=O)cc1Cl Cc1ncccc1CCC(=O)NC1CCC(NC(=O)CS(C)(=O)=O)CC1 c1(NC(=O)OCc2cccc(N(CC)CC)c2)cc(Cl)c(C)nn1 C1(C(N(CC(C)NC(C2CN(C(C)C)C2)=O)C)=O)CCOCC12CCCC2 c1(NC(N2CCC(N(c3nnc(C4CCCC4)s3)C)C2)=O)c(F)cccc1F C1(C(=O)NCC2CCCC2NC(C2(C)CC2)=O)(OCC)CCCCCC1 CC1=NOC(C)(C(=O)NC2C=CC(C(=O)N(CCO)CCN(C)C)C2)C1 c1(C(=O)NCC(CCCC)NC(=O)C(C)CSC)sc2cccc(C)c2c1Cl c1(CC(=O)N(C(CNC(c2cnoc2C2CC2)=O)C2CC2)C)cn(C)nn1 Nc1c(C(N2CC3CCN(C(=O)CC45CCCC4C5)C3C2)=O)cc(F)cc1F N1(C(CC)C(=O)NCC(CO)NC(=O)Cn2ncnn2)C(=O)CCC1=O c1(C(=O)NC(CCN(C(c2c(C)n(C)nn2)=O)C)C(C)C)cnc(O)n(C)c1=O C#Cc1ccc(C(=O)N(CC(C)O)CCNC(c2cnc(O)n2C)=O)cc1C c1(NC(C2CC3CC3N2C(C2CC2C2CC2)=O)=O)cnccc1CO C(c1ccc(C)c(C)c1)=CC(N1C(C)(CNC(C(CCC)CC)=O)CCC1)=O c1(C(N2CCCCC2)CNC(c2nccs2)C)scnc1Cl c1(CNC(C2(C)N(C(C3CCN(CC)C3)=O)CC2)=O)ccc(O)cc1 C(C1OCCc2sc(I)cc21)N1CCN(C(c2ccc(C#N)c(N)n2)=O)CC1 N1(C(CCCCCSC)=O)CCN(C(=O)C(N2CCOCC2=O)C)CCC1C C1(C(N(C(C(CC)C)C)C2CC2)=O)CN(C(=O)CN2CCCCS2(=O)=O)CC12CC2 c1(C(N(C)CC2CCN(C(Cc3cc(C)ns3)=O)C2)=O)cnc(C(C)C)nc1 C(=O)(C#CC(C)(C)CNC(=O)C(COC)COC)N(CC=C)C N1(C(C(COC)NC(C=CCN(C)CC)=O)=O)CCCC(C(=O)N)CC1.C(C)(C)O c1(CCC(=O)NC(CN(C(=O)COCC2CCOC2)C)C)nccn1C CN(C)NC(=O)CCC(=O)NC1CC12CCN(C(=O)CCCSC(C)(C)C)C2 C(=O)(C1Cc2ccc(F)cc21)N1CC(S(C)=O)C1.N12CCc3nc(sc3C1)C2=O c1(C(=O)NC2CC(CNC(C(C)CC(N)=O)=O)CC2O)cc(F)cc2nc[nH]c12 c1(C(=O)N(CCCN2CCOCC2)CC2CC2)ccc(C(F)(F)F)cc1Br C1(NC(C(C2CC2)OCC)=O)CN(C(=O)C(C)(C)CC2CC2)CCC1CO N1(C(c2c(C)ccnn2)=O)CCC=C(C(=O)NCCCOCCCO)C1 c1(OC)ccc(NC(=O)CCCn2cc(-c3ccccn3)nn2)c(C)c1 C1(C(=O)NCC(=O)Nc2cccnc2)CCCN1c1nnc(C(F)(F)F)s1 C1(F)(CNC(C2OCCC(C)C2)=O)CCCN(C(C2CCC=CCC2)=O)CC1 c1(C(N2C(CN(C(=O)CC3CC4(CC4)CO3)C3CC3)CCC2)=O)ccnc2cc[nH]c12 C=CC1(C2(C(=O)NC3CC4CC3N(C(c3cc[nH]c(=N)c3)=O)C4)CCC2)CCC1 N1(C(c2c(COC)n(C)nc2)=O)C2CCC1CC(CNC(=O)CSC1CC1)C2 C(=O)(C(C)(C)S(C)(=O)=O)NC1CCC(C)N(C(C2CC2C(=O)NCCO)=O)C1 C1(NC(C2(CC=C)CC2)=O)C=CCN(C(=O)OC(C)(C)C)C1 C=CC(C)(C)CC(=O)NC(CCOC)C(=O)NC1CNC(=O)C1(C)C c1(C(=O)NCC2(C)CCC(NC(C3CC4(CC4)C3)=O)C2)c[nH]c2c(Cl)cccc12 c1(CC)cc(C(N2CCC(CO)(NC(c3ccnc(C(F)F)c3)=O)C2)=O)ncn1 N1(C(c2ccc(C)nc2)=O)CCc2sccc2C1CNC(=O)C(C1CC1)C1CC1 C1(NC(=O)CC2CCCC2)CCCCC1NC(C1CNC(=O)C1)=O n1(CC)nnc(C)c1C(=O)N(C)CCN(C(=O)Cc1nc(C2CC2)cs1)C C(=O)(CC(C)(C)CN(C)C)N1CCC(N(C(Cc2cc(C)sc2C)=O)CCO)C1 S(=O)(=O)(c1ccc(C)c(C)c1)N1CCC(NC(c2c(OC)nccc2)=O)C(C)C1 Cc1cc(Br)cnc1C(=O)NC1CC(CNC(=O)C(C)NC(C2(C)CC2)=O)C1 C1(C(N(CC(CN(C(=O)CCCc2cccnc2)C)O)C)=O)CC(S(C)(=O)=O)C1 c1(NC(C2CC(F)CN2C(c2cc(Cl)c(Br)cn2)=O)=O)ncc(Br)cc1[N+](=O)[O-] c1(CN(C(CN(CC)CC)=O)C)ccccc1CNC(C1CCCC1F)=O c1(C=O)ccc2sc3ccccc3c2c1.N1(C(CC#C)=O)CC2CN(C)CC2C1 CCN=c1[nH]cc(C(N2CCN(C(=O)CCCCC3CC3)C(CO)C2)=O)s1 N1(C(CCCCC)=O)CCC2(CCN(C(=O)CC3CCCC(=O)C3)C2)C1 c1(C(=O)NCC(CNC(c2c(SC)snn2)=O)O)ccc(-c2cnn[nH]2)cc1 c1(CC)cnc(O)c(C(=O)NC(C)CNC(c2cc(Cl)ccc2C)=O)c1 Cn1c(C2CCCCC2)nc2c1CCN(C(C1CCCC(CN)C1)=O)C2 Cc1[nH]c(=N)nc(NC23CCC(C(=O)Nc4cc([N+](=O)[O-])ccn4)(CC2)C3)c1C c1(C(=O)NCC(CN(C(C(CC)OC2CCCC2)=O)C)O)cccnc1O CCC(C)C(C)C(=O)NC1(CF)CCN(C(c2ccn(C3CC3)n2)=O)C1 C(c1ccc2ccc(Cl)cc2n1)=CC(=O)NCC1CC1NC(c1n[nH]cc1Cl)=O c1(CC)c[nH]cc1C(=O)NCc1n[nH]cc1C(=O)NC(C)C(C)SC C12(CNC(CNC(C3C(C)C3)=O)=O)CCC(CC1)CN2C(=O)CC1C=CCC1 n1(CC(=O)NC2(c3c(OC)cccc3)CC2)ccc2ccc(-c3ccco3)cc12 C12(NC(C3(C=C)CC3)=O)CC1CN(C(=O)COCCc1ccc(C)s1)C2 N1(C(C2CC3(C)OCC2C3)=O)CCCC(C2CN(C(=O)C(O)c3ccsc3)C2)C1 C1(C(=O)OC)C(CCCOCCOCCNC(=O)Cn2cc(Cl)cn2)C1(F)F c1(NS(CC(=O)OCC2CC2)(=O)=O)ccc(OC(F)F)cc1F Cc1cc([N+](=O)[O-])ccc1-n1cc(C(C)(C)NC(C2CC3(CC3)C2)=O)nn1 N1(C(c2c(COC)ccs2)=O)CC(CNC(=O)CCc2cnn[nH]2)OC(C)(C)C1 C1(NC(C(CCC)N(C)C)=O)CC2CN(C(c3nnccc3C)=O)CC2C1 c1(OCC)cc(C(N2CCC(F)(C(=O)NCCC3C=CCC3)C2)=O)nn1C c1(OC)ccc(NC(C2CCCN(C(C3CC4CCC3CC4)=O)C2)=O)cc1C Cc1c(-c2cn(CCCCNC(C3CC3(F)Cl)=O)nn2)cccc1F C1(CC(=O)NCC(C)CN(C(=O)COC2CCCCC2)C)COC2(CCC2)CO1 C(=O)(C(C)(C)n1ccnn1)NCC(CNC(=O)COCC1CCC1)OC C(=O)(C1=C(C)CCC1)NC(COCC)C(=O)N1CCCC1C(C)(C)O c1(OCC#C)ccc(CN2CCCC(C(O)C(F)(F)F)C2)cc1 C=C(C)CCC(=O)NCC(C)(C)CN(C(=O)C(O)C1CC1)C c1(C(=O)NCC2N(C(c3c(C)cno3)=O)CCCC2C)cccc2oncc12 C#CCC(C)(C)C(=O)NC1CCC(NC(C2CCC(=O)N(C(C)C)C2)=O)C1 C(=O)(C1Cc2c(Cl)cccc21)NC(C(C)C)(C)CNC(=O)Cc1cccc(F)c1 N1(C(C(CCC)C)=O)CCN(C(c2c(C)cnc(OC)c2Cl)=O)CC(C)(F)C1 C1(NC(C(c2ccn(C)n2)C)=O)CC2CN(C(=O)Cc3ccsc3)CC12 C1(NC(C2C(CC)C2)=O)CCOC12CCN(C(c1ccnn1COC)=O)CC2 CC1=CCSC1C(=O)NCC1CCC1C(=O)NC1(CCc2nccn2C)CC1 N1(C(C2OCCN(C(C3(C(=O)OCC)CC3)=O)CC2)=O)CCC(F)(F)C(O)C1 CC(=O)CCC(=O)NCCC(=O)NCC1CC(F)C1 c1(CC)ncc2c(n1)CCC(C(=O)NCCc1ccc(O)c(F)c1)C2 c1(C(N(C(C)C)CCN(C)C(C2CC2CF)=O)=O)c(F)cc(N)cc1F C1(CC)CCCCC1OCC(=O)NCCCN(C(=O)C1=CCCC1)C Cc1cn(C2CCOCC2)nc1C(=O)NCCCN(C(=O)C(C)n1cncn1)C C(=O)(CC(C(F)(F)F)N1CCOCC1)NCCC(C)NC(=O)CC1COC(=O)N1 N1(C(C(C(C)C)(F)CNC(=O)C(O)C2CCC2)=O)CC2CCCC2C12CC2 S(=O)(=O)(CC(c1ccccc1)OC)N1C(c2cc(NC)n(C)n2)CCC1 N1(C(=O)OC)CC2(C1)CN(C(=O)C(Cn1cncn1)NC(C1CC3CC3C1)=O)C2 c1(C(=O)NC2CC(C)N(C(c3cn(C(C)(C)C)nn3)=O)C2)ccc2c[nH]nc2c1 c1(CC=Cc2onc(CS(C(C)(C)C)=O)n2)cc(O)nc(O)n1 c1(C(=O)NCC2(C(N)=O)CN(C(C(CC)(CC)CC)=O)C2)cccc2nnn(C)c12 C1(C(=O)NC(C(=O)OC)CC2CC2)CC(C)CN(C(=O)COCCCF)C1 c1(OCC)cncc(C(=O)NC2CC(C(=O)NC(c3cc(C)[nH]n3)C)C2(C)C)c1 C1(=CC(=O)NC(C(=O)OCC)C(O)c2ccc(F)cc2)CCCCCC1(F)F c1(CC)ccc(Cl)c(F)c1.n12nnc(c1C)OC1CC(C1)C(=O)ON1CC(C1)C2 c1(C(=O)NC2CN(C(c3cn(C)nc3)=O)CC2O)cc2sc3ccccc3c2s1 N12CCC(C)(C1)C2=O.N1(CCC)CCCC1C(=O)NC1(CC(C)C)CC1 Cc1ccc(N2CCCC2)cc1C=O.c1(C2(C)CC2)noc(CCN)n1 Cc1cc(C(=O)NCCC2CCCN(c3cc(O)ncn3)C2)cc2ccsc12 N1(C(C2(OC)CCC2)=O)CC(CNC(=O)CCCF)C2(CC2)C1 N1(C(=O)C2CC2)CCCC2C(CCCN2C(=O)CCCC2CCCO2)C1 CCCCC(F)C(=O)N1CCCCC(CNC(=O)C=CC2CCCN2C)C1 c1(CC(=O)NCCC2CCCN2C(=O)CC2CCC(=O)N2)ccc2ncsc2c1 c1(NC(CC(C23CC(NC(c4ccc(F)nc4)=O)(C2)C3)=O)=O)cc2sccc2s1 CC1CN(C(=O)CC2(C)CCN2C(c2cccc3[nH]ncc23)=O)Cc2nncn21 N1(C(c2c(C)[nH]cc2)=O)CCC2(CC(NC(C3(O)CCC3)=O)CO2)C1 C1(CCNC(C2C=CCS2)=O)CCN(C(C2(C3CC3)CC2)=O)C1 c1(C(=O)OC)nc(CN)oc1C.N1(C(C2CC=CC2C)=O)CCCC1CNC=O N1(C(c2c(C(=O)OC)csc2)=O)C2CCC1C1CC1(NC(=O)C(O)CC(C)C)C2 C(=O)(N=c1[nH]nc2c(Cl)ccc(C)n12)NCCOC(C(=O)OC)C C=Cc1cc(C(N2CCC(O)(CNC(c3c[nH]c(=N)nc3C)=O)C2)=O)cc(F)c1 N1(C(C)C)CCCC(C(N2CCCC2C2(NC(C3CCS(=O)(=O)N3)=O)CC2)=O)C1 Cc1ccc(C)c(C(=O)NCC2CC2NC(=O)CCCCCc2ccccc2)n1 N(C(=NCc1c[nH]nc1C)N1CCSC(C)(C)C1)C(CC)C C1(C(=O)NC(c2cccs2)CC)CCN(C(c2oc(C)nc2C)=O)CC1(C)C C1(C(N(C2CCN(C(C(C)(C)CC3CC3)=O)C2)CCO)=O)CCc2nncn2C1 C=CC1(C(=O)NCc2ccoc2C(N2CC3(C2)CN(C)C3)=O)CCCCC1 c1(C(=O)N(CCC2CCNCC2)Cc2ccccc2)ccc(O)cc1Br C(CC(C(=O)N1CCCCC1)NC(c1cn(CC(=O)NC(C)(C)C)nn1)=O)SC c1(CC(=O)NC2C=CCN(C(c3coc(SC)c3)=O)C2)cncc(Br)c1 N1(C(c2c(O)cc(C)c(Br)c2)=O)CCN(C(=O)C(F)F)C2CCCCC2C1 C#Cc1ccc(C(=O)NC2(CNC(C3CC=C(C)CC3)=O)CCCC2)cc1Cl C(=O)(C(C)CC(F)F)NC1(CNC(c2cncc(CC)c2)=O)CCC1 CCCCCC(O)C(=O)NC1CCN(C(=O)CN(c2ncccn2)C)C1C1CC1 N1(C(CC(CNC(C(CCCC)F)=O)C)=O)CCn2cc(C)nc2C1 Cc1cnc(N)c(C(N2CCC(NC(C3CCNC(=O)C3)=O)CC2)=O)c1 C(C)(C)(CCCNC(=O)C(C)(C)c1cccnc1)NC(CCc1ccc(C)o1)=O C(=O)(C(O)CC(F)(F)F)N1CC(NC(c2ccc(C(C)(C)C)nc2)=O)C(O)C1 N1(C(Cc2cc(CC)no2)=O)CC2CC2(C(=O)NC2CCCC(O)C2)C1 C1(O)(CCNC(=O)CC(F)(F)F)CCCN(C(=O)Cc2cccnc2Br)C1 C1(C(N(C2CCN(C(C(C)(C)OC)=O)C2)C)=O)CC2(C1)CN(C(=O)OC(C)(C)C)C2 C(=O)(CC(CNC(C)C(c1ccc(Cl)c(C)c1)=O)C(F)(F)F)OC N1(C(CSC(C)C)=O)CCC2(CC1)CC2(CO)CNC(c1c[nH]nc1F)=O c1(C(=O)NCC(CC)NC(c2c[nH]c(Br)c2)=O)cc(C)nc(O)n1 c1(C(CO)N(C)C(=O)NCC(=O)CC2CCCC2)ccccc1 C1(C(N2CCCC(NC(c3c(C)nc(C)n3O)=O)CC2)=O)(CC)CCC(O)CC1 c1(OC)ccnc(CNC(=O)CC2CCCCN2C(=O)Cn2nc(C)nc2C)n1 N1(C(c2ccc(I)s2)C(=O)NC)CC(Cc2ccsc2)C(c2cn[nH]c2)C1 CCCCC(C)C(=O)N(C)CC1CCCC1NC(C1CCCC(C)(C)C1)=O c1(NC(c2cccc(OC)c2O)=O)ccc2c(c1)CN(Cc1ccc(Cl)nc1)C2 C1(NC(CC2CC(C)C2)=O)CN(C(c2cccnc2N(C)C)=O)CC1C c1(C(=O)NC(CCC)CCCNC(=O)CCCF)c(S(N)(=O)=O)ncn1C c1(C(N2C(CNC(C3(COC)CCCC3)=O)CCC2)=O)c(C)ccc2nsnc12 C1(CC#C)(C(=O)NCC2CC(C(=O)NCC3CCCCS3)C2)CCCCO1 c1(CC(=O)NCC2CN(C(c3cc[nH]c3)=O)CC2O)ccc2ncccc2c1 C1(NC(COCC#C)=O)CCN(C(=O)C=C(C)c2ccccc2F)CC12CCC2 N1(C(C=Cc2cncc(C)c2)=O)CCCC1C1CCCCN1C(=O)Cn1cnnn1 C1(CNC(c2n(CC)cc(Cl)c2)=O)CCCCN(C(C2CC(C#N)C2)=O)C1 N1(C(CC(C)O)=O)C2CCC(C2)C1C(=O)NC1CC1(C)C c1(CNc2ccc(CCOC(C)CN(C)C)cc2)cnc2c(C#N)cnn2c1 C1(N(C(COC(CC)(C)C)=O)C)CC2CCC(C1)N2C(=O)CNc1cccnc1 N1(C(=O)NCC2(c3ccc(C)cc3)CCCCC2)CCSC2CCC12 C#Cc1ccc(C(N2CCC(CCC)C2)C(=O)NCCOCC)c(C)c1 C1(NC(=O)NC(C(=O)OCC)C(C)C)CCOC(=O)CC1.C1(=O)C2=CCC(C2)N1 N1(C(c2nc(CC)oc2)=O)CCC2(CC1)CN(C(C1(C)CCN(C)C1)=O)C2 N1(C(Cc2c(C)cc(C)s2)=O)CCC(NC(=O)CCOC2CCOCC2)CC1C Cc1cccc(CC(=O)NC2CCCC(NC(=O)C(F)(F)CN(C)C)C2)c1 CC1(CNC(=O)COCC2CCCO2)COCCN(C(=O)Cn2nccn2)C1 Cc1cc(C(=O)NCC2CC3CC(C2)N(C(c2cn(C)cn2)=O)C3)cc(=O)n1C N1(C(CS(CCN(C)C)(=O)=O)=O)CCC(C(=O)NCCC2CC2C#N)C(F)(F)CC1 C#CCCCC(C)C(=O)N1CCC1CNC(c1ccncc1)=O c1(C(N2CCN(C3CN(C(CC4CCN(C)C4=O)=O)C3)CC2)=O)ccc(Cl)cc1Cl C(=O)(CC(C(F)F)NC(c1cccc(O)c1)=O)N(C1CC(F)(F)C1)C c1(C(=O)NCC(CN(C(=O)CSCc2cccc(Cl)c2)C)O)ccc(=N)[nH]c1 C1(C(=O)NC2(CCN(C)C)CCC2)CCN(CC(=O)N(C)C)C(c2ccco2)C1 c1(C(=O)NCCN(C(c2cc(OC)cc(OC)n2)=O)CC)cnc(O)cc1C C1(CNC(c2ccc(F)c(F)c2)=O)CC(C(=O)NCc2ccnc(Cl)c2)=NO1 c1(C(N2C(Cn3cc(C(CC)O)nn3)C=CC2)=O)ccc(OC(F)F)nc1 C1(C(=O)NCC)(CC)CCN(CC2CC3N2CCCC3)CC1 C(=O)(C(F)C(F)(F)C(F)(F)F)NC1CCC(C)(NC(=O)Cc2cccnc2)CC1 N1(C(C=C(C)C)=O)CCN(c2ccc(C(=O)NC3CCCC3C(=O)O)cc2)CC1 S(=O)(=O)(c1cnn(C)c1)NCC(=O)NC1C(C)N(C(=O)CC2=CCCC2)CCC1 O(NC(=O)C(c1cnn(C)c1)NC(=O)CC1CCCN(C)C1)CC(=O)OC N1(C(C(CCC)c2ccccc2)=O)CCCC12CCN(C(C1(F)CC1)=O)C2 C1(OC)CCN(C(=O)C(CC2CC2)NC(C2CCCCC2F)=O)C1C N1(C(CCCC)=O)CCCC2CCN(C(C34CCC(C(F)F)(CC3)CC4)=O)CC12 c1(OC)cccc(C(N2CC(O)(C(C)NC(C3CCN3C3CCCC3)=O)C2)=O)n1 C(=O)(C1CCc2ccccc21)NC1(CNC(=O)C2=CCSC2)CCC(C)(C)CC1 N(C(=NCCCCl)NCC1CC(=O)N(C)C1)Cc1cc(C)oc1 N1(C(C(N2CCCCC2=O)CC)=O)CC(NC(c2c(C)cnn2C)=O)C(C)(C)C1 C1(C(NOCCC(C)O)=O)CCN(C(N)=O)C(C)(C)C1.C1(=O)CCN1 C1(N(C)C(C2(N(C)C)CCSC2)=O)CC(=O)N(C2CN(C(=O)CC3CC(=O)C3)C2)C1 CC1(C)CC(C(N2CCC3C(NC(c4cc(C(N)=O)co4)=O)C23)=O)CCO1 CC(C)(C)CCCCC(=O)N1CC2C(CNC(c3nccc4ccsc34)=O)C2C1 CC1OCCN(C(=O)C(c2cc(F)cc(F)c2)(F)F)C1CNC(=O)C=CBr c1(CC(=O)NC2CN(C(CCCOCC)=O)CC2CC2CC2)cc(F)cc(F)c1 N1(C(CSCCNC(CCc2cnc(C)o2)=O)=O)CCSCC1C c1(C(=O)NCC(CO)NC(C=CSC)=O)cc2cccc(Cl)c2cn1 CCCC(C)(O)CC(=O)N1CCN(C(c2c[nH]nc2Cl)=O)C(c2ncc[nH]2)C1 c1(CNN(C)Cc2sccc2Br)sc(=O)n(C)c1Cl c1(CC)[nH]nc(Cl)c1C(=O)NC1CCCC(NC(C2CCCCS2)=O)C1 C12(C(=O)NC3C(NC(C(C)(C)CN4CCCCC4)=O)C3)CC1COC2(C)C C(=O)(C(CCCC)OCCCCC)NCC1C(CC)C2C(CC=C)(CCC(=O)N1)C2 C1(OC)CC(NC(=O)CC(F)(F)F)C12CCN(C(c1cc[nH]n1)=O)CC2 C12(CNC(=O)COC3COC3)CCCCC1N(C(c1cn(CCO)nn1)=O)CC2 N(C(=NCCc1cccs1)NCC(C)(C)C)C1C(C)(OC)C1 CC(C(=O)N(CCCNC(C1CC(=O)N(c2cn[nH]c2)C1)=O)C)C(C)(C)O N1(C(C(c2ccccc2)OCC)=O)CCCCC1C1CCN(C(=O)C(C)O)C1 CCCCCC(O)CC(=O)NCC12CC1CN(C(c1n[nH]cc1C(F)(F)F)=O)C2 N1(C(C)=O)CCC2(COCC(C(=O)NCC3CN4CCCC4CO3)O2)C1 C1(C(=O)NC(C)CC2C(C)CCN2c2ncccn2)CCCN2CCCC12 C(C)(CCN=c1[nH]ccc(=NCc2cn(-c3ccccc3)nc2C)[nH]1)SC C1(C(=O)NC(C)CN(C)C(C2CCO2)=O)CC2C=CC1CC2 N1(C(=O)C=C2CCCC2)CCC2CCN(C(c3csc(C(F)F)n3)=O)C2C1 CC(C)CN=C(NC1CCN(C(=O)OC(C)(C)C)CC1)N1CCC(C)(F)C1 Cc1ccc(C(N2CCOC(CC(N3CC4(CC(O)C4)C3)=O)C2)=O)cc1C#N C1(CC)COCC1NC(C1(NC(=O)C(O)CN2CCCC2)CC(CO)C1)=O N1(C(c2ccc(C)cc2Br)=O)CC2CN(C(c3nocc3C)=O)CCC12 N1(C(c2c(C)coc2)=O)CCC2CC2(NC(=O)CN=S(C)(C)=O)CC1 Cc1cc(C(N2CC(NC(=O)CCn3ccc4ccccc34)C2)=O)cc(C)c1Br C12(NC(c3cn(CCO)nn3)=O)CCCC1CN(C(=O)CC1C=CCC1)C2 N1(C(N(C(C)CSC)CC)=O)CCN(C(=O)Cn2cnc(=N)[nH]2)CC1 N1(C(Cc2c(C)noc2C)=O)CC2CCCC1C2CNC(c1n[nH]c(C)c1O)=O c1(NC(c2cn(C)cn2)C)ccc(S(=O)(=O)NCc2sccc2C#N)cn1 Cc1nn(C)c(Cl)c1CNC1CC1.N12CCN(CC1)C1CCC(C1)C2=O C1(NC(CSCCC)=O)CN(C(c2ccc(OC)nc2)=O)C2(CCOC2)C1 Cc1ncn(C)c1C(=O)N(CCCNC(=O)CSCC1CCCCO1)C N1(C(CC(C)(C)N(C(C2C(C(C)(C)C)CC2)=O)CCO)=O)CCCC2(CC2)C1 C1(C(=O)NCC(CC(=O)NCC2CCC(=O)O2)OC)CN2CCN1CC2 N1(C(CC2(OC)CN(C(C3(C)CCCC3)=O)C2)=O)CCOCC1CN(C)C c1(CC(=O)N(C2CCCN(C(=O)C=CI)C2)CCO)ncn2c1CCC2 c1(C(C(=O)CS(=O)(=O)C2CC2)=O)cccc2oc(O)nc12.C1(N)CCN(C=O)CC1 C1(CC(=O)NC(c2c[nH]ccc2=O)C)CC2(CC2)CN1C(=O)CC1C=CCC1 CC1CN(C(=O)CN2C(C)CCC2C)CC(C)CN1C(C1CC2CCC1C2)=O N1(C(c2c(OCC)nccc2)=O)CCN(C(=O)C(F)C2CCC2)C(C(C)(C)C)C1 Cc1nn[nH]c1CNC(=O)C(C1CCCCC1)NC(=O)CC(Cl)Cl Cc1ccc(C(=O)C(N2CC(NC(c3scnc3C(C)(C)C)=O)C3CC23)=O)cc1 CC1CC(C(=O)NCc2cnn(CCO)c2)CCN1C(=O)C(C#N)C(C)C c1(SCCCC(=O)NC(C(=O)OC)CC2CCC(=O)N2)nc2ccccc2[nH]1 CC1CCNCCC1N(C1CC1O)C(c1c(Cl)ccnc1Cl)=O C(C)(CC1CCC1)(C(=O)NC1CCN(C(=O)C=C2CCN(C)C2)C1)OC c1(C(N(CC)CC2(C(=O)OC)CC2)=O)ccsc1SC.n1(C(=O)N)cc(Cl)cn1 C1(c2ccccc2)(C(=O)OCC2CCCN2SSc2ccccc2)CCCCO1 c1(C(=O)NCC(CCCC)NC(C23CC(CO)(C2)C3)=O)cc(F)c(C)cc1N c1(C(N2CCC(C)C2)C(=O)NCCN(CC)CC)ccccc1F c1(C(=O)NCC(c2cnn(C)c2)NC(C2CC(=C)CC2)=O)c(C)ncnc1C N1(C(c2c(CC)[nH]c(=N)s2)=O)CCCC(C2CCCN(c3cc(C)ncn3)C2)C1 N1(C(CC=CC=C)=O)CCC(O)(C(C)CNC(=O)C=C2CCC2)C1 C12(NC(CCC#N)=O)CCN(C(=O)C(c3cc(Cl)cc(Cl)c3)(F)F)CC1C2 c1(C(N2CCN(c3ncc(C)cn3)CC2)C(=O)NC2CC2)cccc2c[nH]nc12 C1(C(N2CCC(OC(C)=O)C2)=O)(NC(C2CC2[N+](=O)[O-])=O)CCN(C)C1 c1(C(N(C2CCN(Cc3ccccc3)C2)CC#C)=O)ncccc1SC C(N=c1[nH]c(=NCC2CSCCO2)[nH]c2c1COC2)c1c(C)nccn1 N1(C(=O)NCCCOC)CCC2(CC1)CCN(C(c1ccc(C)nc1OC)=O)CC2 c1(C(=O)NCC2(C)CN(C(C=C(CCC)C)=O)C(C)(C)C2)cc([N+](=O)[O-])cc(C)n1 Cc1ccc2cc(C(=O)N(c3nccc(C#N)n3)CCc3c[nH]c(=N)s3)[nH]c2c1 C#CC1(O)CCN(C(=O)C(C)N(C(c2cnnn2C2CC2)=O)C2CC2)C1 C(C)(C(=O)NCC#CCNC(C1CCN(C)C1)=O)(C(C)C)NC(=O)OC(C)(C)C N1(C(COCCC)=O)CCN(CCC)CC1.C1(=O)C(C(C)C)OC2CCN1C2 CN1CCC(CC(=O)NC2CN(C(=O)CCC3CCCN3C)CC2O)C1=O C1(C(=O)NC2(CCCNC(CC(C)F)=O)CC2)CC(=O)N(C)C1c1ccccc1 Cc1ccc(C(N2CC(NC(c3cnn(C(C)C)n3)=O)C(C)(C)C2)=O)cc1F c1(C(N(C)CCNC(C2(C)CC2F)=O)=O)ccc2cc(O)ccc2c1 c1(C(=O)NCC(CC)NC(c2cc(C)ccc2F)=O)cnc(O)c(OCC)c1 C(CCCCC(C)(C)NC(=O)C(C)NS(=O)(=O)c1cccs1)OC(C)C O=C1NCCCCC1C(N1CCC1CC(N1CC(N2CCCC2=O)C1)=O)=O C1(OC)CC(NC(=O)C(O)C2CC2)CN(C(=O)COc2cccc(C(C)=O)c2)C1 C1(C(=O)NC2(CO)CCN(C(C(=O)NCC)=O)C2)CC12C1CC3CC(C1)CC2C3 c1(OC2CC(NC(NCCSC)=NCCOC(C)(C)C)C2)cc(Cl)c(Cl)cc1Cl c1(OC)cccc(C(=O)NC(C)CCCCNC(=O)OC(C)(C)C)c1C Cc1c(C(N2CC3CC2CC3NC(C2CCOC(C)(C)C2)=O)=O)ccc(F)c1F C1(C(N2CC3CC3(CNC(C3(CO)CCCCC3)=O)C2)=O)CCn2cncc2C1 CCC(C)C(C(=O)N(C)CC1CCC(=O)N1)N(C)C(c1cc(C(C)C)[nH]n1)=O c1(C(=O)NC2CCCC(NC(C3CC(N(C)C)C3)=O)C2)cnc(Cl)cc1N N1(C(Cn2c(C)cc(C)n2)=O)CC(CC(N2CCN(C3CC3)CC2)=O)C2(CC2)C1 Cc1ncn(O)c1C(N1CCCC(CNC(C2CC3C=CC2O3)=O)C1)=O c1(C2CCN(C(C)Cc3nc(CC4CC4)no3)C2)ccc(Br)cc1 N1(C(c2c(C)[nH]cc2)=O)CCCCC12CC(NC(C1CC(C(C)=O)C1(C)C)=O)C2 CC1CC(C(=O)N(C2CC3CC2N(C(c2cnc(O)o2)=O)C3)C)=NO1 C1(NC(CCNS(CC)(=O)=O)=O)(CO)CCCN(C(=O)CC(C)(C)C2CC2)C1 N1(C(Cc2c(C)ocn2)=O)CC2(COC(C(=O)Nc3cnccc3CSC)C2)C1 C1(N(C(=O)CNC(c2nccn2C)=O)CC)CCN(C(=O)CC2(OC)CCC2)C1 N12CCC(CC1)C2=O.CCC(C(=O)NCc1occc1F)S(c1ccccc1)(=O)=O N1(C(C2N(C(c3c(C)cccc3)=O)CC(O)C2)=O)CC(C(=O)N(C)C)CCC1C Cc1ccc2c(N3CCCN(C)CCC3)nc(=NCC3(Br)CC3(F)F)[nH]c2c1 C12(NC(CC3C=CC(NC(c4c(C)cc(F)s4)=O)C3)=O)CCC(O)(CC1)CC2 C1(NC(C(C2CC2)SC)=O)CCCC1(C)CNC(=O)CCCC1CCCC1 c1(OC)cnc(F)cc1C(=O)NCC1COCCN1C(c1csc(Cl)n1)=O N#Cc1ccc(Oc2cc(F)cc(F)c2)nc1 c1(OC)cccc2cc(C(=O)NC(C)CCCNC(c3cnco3)=O)oc12 c1(CN2CCC(C)(C(=O)NC(c3ccc(Br)cn3)C)C2)cccc(Br)c1F C(N=c1[nH]c(Cl)ncc1Cl)C1OCCN(C(C2(C)CCC(=O)NC2)=O)C1 c1(N(S(=O)(=O)CC2CNC2)CC(N2CCCC(C)C2)=O)ccn2ncnnc12 N1(C(Cn2ccc(=N)[nH]2)=O)CC=CC(NC(C2(c3c(C(N)=O)cccc3)CC2)=O)C1 C(CC(=O)NC(C)C(C)NC(=O)C(C)c1cc[nH]n1)N(CC(C)C)S(C)(=O)=O CC1CC(C(F)(F)F)n2nc(C(N3CCN(C(=O)CO)C4CC34)=O)cc2N1 Cc1cc(C(=O)NC2CCC3CCN(C(=O)CN4CCOCC4)C23)c(N)c(C)c1 CC(c1cccc(Cl)c1)=CC(=O)NC(C)(CNC(C1(F)CC1C)=O)C1CC1 O=C(C1=CCS(=O)(=O)C1)NC1C2CC1N(C(=O)CC1CCC(=O)N1)C2 C(=O)(C(C)CC#N)NCc1c(C(N2CC(C)(CC=C)C2)=O)nco1 C(=O)(C(C)CC(C)(F)F)N1CC(CCC)N(C(c2nn(CC)cc2Cl)=O)CC1 C1(NC(C2N(C)CCCC2)=O)CCC12CN(C(c1cnc(C(F)F)s1)=O)C2 C1(OC)CC(C(=O)NC(C)(C)CNC(c2csc(C(C)=O)n2)=O)CC1OC c1(CN2CC(=O)N(Cc3c(N(C)C)c(Cl)ccc3)C2=O)nc2c([nH]1)CCCC2 C#CCCCCCCCC(=O)N1CC2CCC1C2NC(=O)CCSCCC N1(C(C)C)CCCC1CC(=O)NCC(C)(Cn1cccn1)NC(=O)CC(F)F C=CC1OCCC1C(N1CC(C(=O)NC(C)(C)CSC)C1)=O C1(NC(=O)C2=CCOC2)C2CC3CN(C(=O)CCc4ccc(F)cc4)C1C3C2 C=CC(CC)CC(=O)NCCC1CN(C(c2ccc(C3CC3)c(F)c2)=O)CCO1 N1(C(c2ccc(C3(C)OCCO3)cc2)=O)CC2CC1CN2CC(F)F N1(C(CC2CCN(C)C2)=O)CC(C(=O)Nc2cccc(Cl)c2O)CCC1(C)C C=CCN=C1NCCOc2cccc(c2)CN1.C1(NS(C)(=O)=O)CCOCC1C c1(C(N2CC(C(C)NC(C3C(C)(COC)C3)=O)C2)=O)cc(S(N)(=O)=O)ccc1Cl C12(COCCC(=O)NCC(C)CCOC)CC3CC(CC(C3)C1)C2.C1(C=O)CCC1 c1(OC)ccccc1.O=C(C=CSc1nc[nH]n1)NCCNC(C1(C(F)F)CCC1)=O Cn1cc(C(=O)NCC#CC(=O)NC2(CO)CCCCC2)ncc1=O c1(C(=O)NC2(C)CCN(C(c3cnc(CC)[nH]c3=N)=O)C2)ccc(P(C)(C)=O)o1 c1(C(=O)NCC(CO)NC(=O)CCF)ccc2[nH]c3c(c2c1)CCCCC3 c1(C(=O)NCC(C)(CO)NC(C=CC2N(C)CCC2)=O)c(F)ccc2ccoc12 C1(C(=O)NCC(=C2CN(C(CC(C)F)=O)C2)F)CC(=O)N(c2cnn(C)c2)C1 c1(OC)cc(C=CC(N2CCC(OC(=O)NC3CC3)CC2)=O)c2ccccc2c1 c1(C(N(C2CCN(CC3CCCN3C)C2)C)=O)ccn(O)c(=O)c1 c1(C(N2C(CNC(C3OCCC(C)C3)=O)CCC2)=O)n[nH]c2c1COC2 CC(F)(F)C(F)C(=O)NC(CC1CCC1)C(=O)NC(C(F)(F)F)C1CC1 C1(N(C(c2cnc(CC)nc2)=O)C)CN(C(=O)Cc2sc(C)nc2C)CC1(C)C N1(C(C(CCC)OCC)=O)CC(NC(C2CNC(=O)N2)=O)CCC(O)C1 C(=O)(CCCCC(N)=O)N1CC(C)OC(CCNC(=O)CS(=O)(=O)N(C)C)C1 C#CC1(NC(=O)C(C(C)CC)NC(c2oncc2CC)=O)CCCCC1 C1(CN(C(=O)C(Cn2cccn2)NC(=O)CC2C=CCC2)C)CCCC(=O)N1 c1(OC)cc(C)ccc1C(=O)NC1CCN(C(=O)CCCN(C)C)C(C)C1 C(=O)(C1=CCCOCC1)NC(C(C)(C)NC(=O)OC(C)(C)C)C.N12CCC(C1)C2=O Cc1cc(C(N2CC(CNC(c3cccc(Cl)c3N)=O)CC2C)=O)cc(C)n1 CC1(C)CC(C(N2CC(C)(C)C2C2CC2)=O)CN(C(C2CCOCC2)=O)C1 Cn1nc(C(N2CC=CC2Cn2cc(C3(C)CCCC3)nn2)=O)cc1Br c1(C(N(CCn2cc(C(CC)(C)O)nn2)C2CC2)=O)ccc2ccn(CC)c2c1 N1(C(CNC(=O)OCC)=O)CCC2(CC1)CC2NC(=O)CC(CC)SC c1(C(N2C(C)(C)C(C(=O)NC3CCCC3)CC2)=O)ccc2[nH]ccc2n1 c1(C(=O)NC2CCCC(NC(c3cncc(SC)c3)=O)C2)cc2c[nH]cnc-2n1 N1(C(C=CC(C)C)=O)CC(C)C(NC(=O)CN(C2(C)CCCC2)C2CC2)C(C)C1 C1(CNC(c2cnn(CCC)c2C)=O)CC2(CC2)CN1C(c1ncccc1Br)=O c1(CNC(CC)=O)n[nH]c2c1CN(C(c1nnn(C)c1C(F)(F)F)=O)CC2 C1(NC(C2C(C)(C)OC(=O)N2)=O)CN(C(C2(F)CCOC2)=O)CCC12CCC2 C1(NC(CC=CC=C)=O)CCCN(C(c2ccnc3ccsc23)=O)CC1F n1(C(CCC=C)CC)cnc2c(N3CCOC4CCCCC34)ncnc12 C1(NC(C(CC)N(C)C)=O)CCC(NC(=O)C(F)(F)C2(O)CCC2)C(O)C1 c1(CN2CCC(OCC)C2)cc2c(s1)CCC2.N12CCC(CC1)CNC2=O N1(C(c2c(N)cc(Cl)c(Cl)c2)=O)CCCC2(NC(c3cnc[nH]3)=O)CCCC12 C#Cc1cnn(CC(=O)NC(CCC2CC2)C(=O)NCc2nc(C)oc2C)c1 c1(CNC(C2(C)CCCS2(=O)=O)=O)nnc2n1CCN(C(=O)C1=CCOCC1)C2 N(C1CN(c2nc3cccnc3s2)Cc2ccccc21)C(c1cnnc(Cl)c1)=O C12(C(N3CCN(CC=CC)CC3)=O)CC(CO)(CN1C(=O)C(C)(O)C(C)C)C2 N1(C(CC(C)(C)C)=O)CC2CN(C(c3ccccc3Cl)=O)C2C1 c1(C(N2CCC(CNC(c3ncc(C)c(Cl)c3)=O)C2)=O)cnc2c(C)cccn12 C1(C(N(C)CC2CCN(C(c3nc(Cl)cs3)=O)C2)=O)COc2ccccc2O1 c1(CC)c(Oc2ccc(C)cn2)cnn1C.C12CCC1N2C(=O)OC(C)(C)C C=Cn1nccc1C(=O)NC1CC1CNC(C1(c2ccno2)CCC1)=O C1(C(N(c2ccsc2)C)=O)CCN(C(=O)C=CC(C)(C)C)C(C)(C)C1 c1(C(=O)NCC(CCNC(COC(CC)C)=O)O)nccc2cc[nH]c12 C1(NC(C(N2CCN(C)CC2)C)=O)CN(C(c2cc[nH]c(=N)c2)=O)CCC1C c1(OC)ccc(C(N2CCSCC2CCNC(=O)CC2CCC(=O)N2)=O)c(O)c1 C(=O)(CC(CC)C(F)F)N1CCC(OCCNC(c2nccc(CC)c2)=O)C1 CCC(C)(C)CCCC(=O)NC(C)(C)CCNC(=O)C=CCCCCCCCO CCN=C(NCc1ccccc1CN1CCOCC1)NC1CCN(S(C)(=O)=O)C1 N1(C(c2cn(CC)nc2)=O)C2CCC1CC(NC(C1CCCCN(C)C1=O)=O)C2 C1(NC(C2C(=C)C2C(=O)OC)=O)CCC(NC(=O)CCOCC(F)F)C1 C1(C)(C(N2CC3(CN(C(c4cc(SC)c(C)o4)=O)C3)C2)=O)C2CCC(C2)C1(C)C CCC(CC)C(F)C(=O)NC1CCCC1(C)CNC(C1COCCN1C)=O N1(C(c2cccc(OC)c2)=O)CC2COCC(C1)N2C(c1ccc(Br)s1)=O c1(OC)cccc(I)c1C(N1CCC12CN(C(c1ccc(Cl)cc1C)=O)C2)=O N1(C(=O)NCc2n(C)cnc2Cl)CCOCC(F)(NC(=O)OC(C)(C)C)C1 Cc1nn(C)cc1C(N1CCC(O)(C(C)C)C1)C(=O)NCCCC1CC1 C1(C(=O)NC2CC3(C2)CC3C(=O)N(CC(C)C(C)(C)C)C)(CC)CCNC1=O S(=O)(=O)(c1nc(N2CCC(N3CC=CC3)C2)ccc1Br)N(C1CCC(=O)N(C)C1)C C1(NC(C(C#C)(C)C)=O)CCN(C(c2ccc(=O)oc2)=O)CC1O N1(CCOc2cc(C)cc(C)c2)CCC(NC(C2CC2C2CC2C)=O)CC1C CCC(CC)C(C(=O)NC12CC(NC(=O)C(C(O)CC)OC)(C1)C2)OC N1(C(CCN(C(CCC)C)C)=O)CCCC1CN(C(=O)CCNS(C)(=O)=O)C CCC(C)(C#N)C(=O)NCC=CCNC(c1ccc(=O)n(-c2ccccc2Cl)c1)=O c1(C(C(=O)NC2CC(NC(C3CCCO3)=O)C2)OC)ccc(O)cc1 CCC(F)(F)C(=O)NC1CCCC(N(C)C(c2cnc(C)cn2)=O)C1 N1(C(C2(CC=C)COC2)=O)CCN(CCCNC(C2CCC(OC)C2)=O)CC1 C(CC(F)F)(C(=O)NCC(CC1CC1)OC)N(C(c1cnc(CC)o1)=O)C Cn1[nH]c(=NC(=O)c2cc(CN3CCCCCC3)on2)cc1C#N CC(C)(C)C(CO)C(=O)NCC1(O)CCN(C(c2ccc(S(N)(=O)=O)s2)=O)C1 N1(C(CC(C)SC)=O)CC2(CO)CC1(C(=O)NCC1(C)CCCC1O)C2 C(=O)(C1=C(Cl)CCCC1)NC(C1(O)CN(C(C2CC3(C2)CC3(F)F)=O)C1)C N1(C(CNC(=O)NC)=O)CCC2CC(NC(=O)CC3CC3(Cl)Cl)CCC2C1 Cc1cc(C)nc(CSCCC(=O)NCC2=CCN(C(CS(C)(=O)=O)=O)CC2)n1 C1(CN(C(C2(SC)CCC2)=O)C)CCN(C(=O)C(C)n2ccnc2)C1 C#CCCC(C(=O)NCC(C)(C)CC1CC1)NC(c1n[nH]cc1Cl)=O c1(C(N2CC(C)CC(NC(C3(CC=C)CCC3)=O)C2)=O)cc2ccccc2nn1 CCCCCC(CC)C(=O)N1CCC(OCCNC(C23CC(F)(C2)C3)=O)CC1 c1(C(N(C2CN(C(C3(CCC)CCC3)=O)C2)C)=O)cc[nH]c(=N)c1[N+](=O)[O-] c1(C(=O)NC2(COC)CCN(C(C3CC4(CC(=O)N4)C3)=O)C2)nc(C)ccc1C c1(C(=O)NCC(CCCC)NC(=O)C=C(Cl)Cl)c(F)ccc(OCC)c1F c1(C(=O)NC(CN(C(=O)CC2(C#N)CCC2)CC)C)ncc(N)cc1C C1(CC(=O)NCC2ON=C(C)C2)CN(C(c2oc(C)nc2C)=O)C(C)(C)C1 N1(C(C(F)=CCC)=O)C(C)CC2CN(C(c3ccnn3C3CC3(F)F)=O)CC12 c1(C(N(C(CC)CNC(c2cc(C)ns2)=O)C)=O)nccc(OC)c1C Cc1cc(C(N2CCCC(C)(NC(C3CCOC(=O)N3)=O)C2)=O)c(F)cc1Cl C=CC1(C(=O)N(CC(O)COC)C)CCN(C(C2CCCCC(=O)N2)=O)C1 C1(C(N2CC(CC)N(C(C3CC(C)(C)C3)=O)CC2)=O)CCOCC12CCCC2 Cc1cc(C(C)C(=O)NCC(C)NC(C2(O)CN(C(=O)OC(C)(C)C)C2)=O)c(C)o1 C1(NC(C2C(C)OC(=O)N2)=O)CC(C)CN(C(c2cc(C(F)(F)F)ccn2)=O)C1 Cc1noc2ncnc(NCC3CN(C(=O)C(c4cnn(C)c4)O)CCC3C)c12 c1(C(N2CCC(NC(c3c(CC)noc3)=O)C(CO)C2)=O)ccc2nonc2c1 CC1(C(=O)NCC2CC3(CO2)CN(C(=O)Cn2cnnc2)C3)CCCNS1(=O)=O O=C(CCc1ncon1)NCC1CCC1NC(C1CC1C(F)F)=O c1(C(N2CC(NC(=O)CC3=CCCC3)CC(C)(C)C2)=O)coc2c1C(O)CCC2 CC(C(F)(F)F)NC(=O)C(Cc1cn[nH]c1)NC(=O)CC1CCCOC1 N1(C(c2c(C)nn(C(C)C)c2C)=O)CC2COCCC2(NC(=O)C(O)C(F)F)C1 c1(C(C)=O)ccc(C(=O)NC(C(C)NC(C2(CC(F)F)CCC2)=O)C(C)C)nc1 C(=O)(C#CC(C)(C)CNC(C1(C)CC(O)CN1C)=O)NC(C(CCC)O)CO c1(C(=O)NCC2N(C(c3c(C)c(N)cnc3)=O)CC=C2)nc2cccnc2s1 C1(N(C(=O)C(F)OC)CC)CCCN(C(c2cccc(C)c2N)=O)CC1 N1(C(c2nc(C)sc2)=O)C2CCC1C(NC(c1cn(C)nc1C(F)F)=O)C2 C1(CNC(CC2(C(=C)F)CCC2)=O)CCN(C(=O)CN(C)C(=O)OC)CC1(F)F c1(COC(C(C)SC(F)(F)F)=O)ccccc1.C1(=O)C(C)N1.C1C(=O)N1C1CC1 C1(NC(CC(=C=C)C)=O)C2CC1N(C(=O)C=CCN1CCCC1)C2C c1(C(N2CCC(C)(NC(C(C)Sc3nncn3C)=O)C2)=O)ccnc2c1CCO2 C1(NC(c2cccc(CO)c2)=O)CN(C(C2(C3CCCO3)CC2)=O)CC1F C1(C(=O)NCC(C)(CO)NC(C2CN(C)C2)=O)CCc2nc(C(F)(F)F)cn2C1 C1(C(=O)OCC)COCCN(C(C(=O)NC(C)(C)CC)C(C2CC2)C2CC2)C1 C(CNC(c1cc(C)c(Cl)s1)=O)(CC(C)C)NC(COCCCC#C)=O C(=O)(CCCCN(C)C)N(CCCN(C)C)CCNC(CCN(C(CCC)C)C)=O n1(CCCOC)nnnc1C(CCOC)N(c1ccccn1)C1CC1 CC1(F)CN(C(c2sc3nccn3c2C)=O)CCN(c2ncnc3c2CCC3)C1 Cc1nc(NC(c2ccc(CNCC3CCC(C4CC4)C3)o2)=O)ccc1C#N c1(NC(CN(CC#C)C2CC2)=O)cc(OC)cc(Cl)c1 c1(C(=O)NC2C(C)CN(C(=O)CC(C)(F)F)CC2)ccc2ccccc2c1O n1(C(C)C)nc(-c2cnc(C(F)(F)F)nc2)nc1C1CCN(C)C1=O C(=O)(C1CCCc2sccc21)C(N(CCNC(CC#C)C(=O)OC(C)(C)C)C)=O CCCC(C)(CCC)C(=O)NCC(O)CCNC(=O)C(C(C)C)OCC(C)C C(=O)(C#CC1(C(F)(F)F)CC1)N1CC(F)(C(=O)NCCNC(CCC#C)=O)C1 N1(C(C)C)CC(Cc2cn(NC(c3ccc(C(N)=O)s3)=O)nn2)NC1=O C1(C(=O)NC2(COC)CN(C(c3ncc(F)cc3N)=O)C2)CCCCN(C)C1=O C(=O)(C(C)CCC(C)(C)C)N1CC(C(C)NC(c2ccc(C)n2C)=O)C1 N1(C(C2(c3ccc(OC)cc3)CC2)=O)C2CCC1CC(NC(=O)CN1CC=CC1)C2 CCCCCCCCCC(=O)N1CCCN(C(c2c(Cl)cnn2C)=O)CCC1 n1(CC(=O)NCC2N(C(CCCC(=C)C)=O)CC=C2)[nH]cc2c(=O)ncnc1-2 Cn1nccc1C=CC(N1CC(NC(=O)Cc2cc(Cl)sc2Cl)C(O)C1)=O C=CC(C)C(C)C(=O)NCCCN(C(=O)Cc1ccn(CC(F)(F)F)n1)C(C)C O=S(=O)(c1cnc2sccn12)N1CCCC1c1cccc(OC(F)F)c1F N1(C(C(CSC)OC)=O)CCOCC(CNC(=O)C=Cc2sccc2C)C1 C(Cc1ccccc1)(CCNC(=O)CCCN(C)C)NC(C(C)SC)=O C(=O)(C1c2ccccc2C2CC1C2)NC1(CCNC(c2ncn(CC)n2)=O)CC1 N1(c2ccc(CN3CCCCC(CCC(=O)OC)C3)cc2)CC(N)C(C2CC2)C1 C1(CN(C)Cc2cccc(C(F)(F)F)c2)COC2(CCNCC2)CO1 C1(NC(C(n2ccc(C)n2)C)=O)CCC(CNC(c2nccc(CO)n2)=O)CC1 c1(C(=O)OC)cnn2c(NCCC3CC=CCC3)cc(C)nc12 C(=O)(C1=CCS(=O)(=O)C1)NC1C(OC)CN(C(=O)CCNc2cccc(C)c2)C1 c1(C(=O)NCC(CC(C)C)(C)NC(=O)C=CS(C)=O)ccc2cc[nH]c2c1F Cc1nc(C(N2CC=CC(NC(c3ncn(C4CC4)n3)=O)C2)=O)ccc1[N+](=O)[O-] c1(NCC)ccc(C(=O)NC(C)(C)C(C)NC(=O)CCCOCC)cc1[N+](=O)[O-] C1(C(=O)Nc2ccc(C#N)s2)CCCCN1C(=O)CN(CCCCC)C(C)C c1(C(=O)NCC2(F)CC(NC(c3c[nH]nc3C3CC3)=O)C2)cnc(O)o1 C(=O)(C#CC1(CC)COC1)NC1(C(=O)NCC2OCCC(C)C2)CC1 c1(C(N2CCC(CN(C)C(C3CCO3)=O)C2)=O)cc2oc(Br)cc2[nH]1 C1(NC(C2(OCC)CCSCC2)=O)CN(C(=O)CC2(C)CC2(F)F)CC12CCC2 c1(C(N2CC(CNC(Cc3c(C)nn(C)c3)=O)C2)=O)ccc(O)c(N=[N+]=[N-])c1 c1(C(N2CC(CCC)C(C(N3CCC3C)=O)C2)=O)cccc2ccoc12 N1(C(C(CCC)=CCC)=O)CC(NC(C2CN(C(C)=O)C2)=O)C2(CCCC2)C1 C1(N(CCNC(c2ccc(Cl)s2)=O)C(C2CCCN2)=O)CCC2(CCNCC2)CC1 c1(OCC(=O)N(CC(C)NC(=O)CNC(N)=O)C)ccccc1.C1(=O)CN1 N1(C(c2c(COC)ncs2)=O)CC2OCC(NC(C3CC(N4CCCC4)C3)=O)C2C1 N1(C(c2cc(OC)c(C)cc2)=O)CCOCC(F)(CNC(c2occc2C)=O)C1 C1(CNC(CSCCN(C)C)=O)CC2CCC1N2c1nnc(-c2ccccc2)s1 c1(-c2cnccc2)nc(-c2ccc(Oc3cccc(Br)c3)cc2)n(C2CSC2)n1 C(=O)(C1COc2ccc(Cl)cc21)NC(C1CCCN1C(C1CC(Cl)(Cl)C1)=O)C C1(C(N2C(CC(N3CC4CC(CO)(C4)C3)=O)CC(O)C2)=O)Cc2nccn2C1 C1(NC(C(C)NC(=O)C(Cl)Cl)=O)(CO)CC(O)C1 C(CC(CC)C(=O)NC(c1ccccc1)C(=O)NCC1CC1(C)CC)=CC c1(C(=O)NCC2(F)CCN(C(CC(C)CF)=O)CC2)ccc2c(c1)CCNC2=O c1(OC)ccc(Cl)c(C(=O)N(C2CCC(NC(C3CC34CC4)=O)CC2)C)c1N O=C(C1CCCc2nc[nH]c21)N1CC2(CCCN(C(c3cnc(C4CC4)[nH]3)=O)C2)C1 N1(C(C(CC#C)NC(c2ccc(F)cc2)=O)=O)CCC12CC(C(N)=O)C2 c1(OC)cc(C(=O)NC2CC2NC(=O)C(c2ccc(Cl)cc2)C)cc(O)c1 CC1(C(=O)O)CCCCC1NCC1CC2(CCNC2)C1 C(=O)(C(F)CCC(C)(C)C)N1CC(NC(C(CC)(C)OC)=O)C2(C1)CC2 C(CC(O)C(=O)NCC1C(CO)C1(F)F)NC(=O)CCc1cscn1 NC1CCN(CCCNC(=O)Nc2nc(-c3ccccc3)no2)CC1.CCCC N1(C(C(CC(C)C)NC(C)=O)=O)CCN(C(c2cnsc2C)=O)CCC1C c1(CNC(C(CC)C(C)C)=O)n[nH]c2c1CN(C(C1CCCCC(=O)N1)=O)CC2 n1(CC(=O)NCC2C(NC(c3nc(C)sc3)=O)C2)cnc([N+](=O)[O-])n1 c1(NC(C2CC(NCC3N(C)CCC3)C2)=O)cc(Cl)c([N+](=O)[O-])cn1 C1(C(=O)NC(C2N(C(C3C(C)C3)=O)CCC2)(C)C)Cc2ccccc2C1 C(C(F)(F)C(=O)NC1CC1CNC(c1ncc[nH]c1=O)=O)OC C1(CC(=O)N(C2CCN(C(c3c(COC)ccs3)=O)C2)C)CC(O)C1(C)C c1(OC)cccc2c(C(=O)NC(C)CCN(C(=O)CCCC(N)=O)C)n[nH]c12 N1(C(C(CC)CC(C)C)=O)CCC2(CCC2)C(NC(c2cc(CO)ccn2)=O)C1 N12CCCN(CC1C)C(=O)CSCC2=O.c1(OCC)ccc(C(N)=O)cc1 c1(CC(=O)NCCCN(C(c2ccc(C(F)F)s2)=O)CC)ccnc(Cl)c1 N1(C(CCSCC#C)=O)CCC(C)C(NC(=O)C(C)OCC(C)C)C1C N1(C(c2c(OC)nccc2)=O)CC2(C)CN(C(=O)CCC3CC3C)CC2(C)C1 C1(O)(C(C(=O)NCC)C2CC2)CCN(C(=O)OC(C)(C)C)CC1.N12CCC(C1)C2 N1(C(c2cn(C)nn2)=O)CC2CC(C1)C(CO)C2NC(=O)CCC(C)(F)F c1(SCC(=O)NC2CC(C)(NC(=O)CC(F)(F)F)C2)ccc(Cl)c(Cl)c1 C1(C(=O)OC)CC2CCC1N2CC#CC(=O)NC(C)C(C)C C1N=C2C=C(N=CN2)N2CCC(CC2)C2COC(=O)N12.O=C1NC(=O)C(CO)N1 c1(C(=O)NC(CNC(CC(CCC)C)=O)C)ccc(OC)c(S(=O)(=O)N)c1.OCC c1(C(N(CCCNC(C2CCN(C)C2)=O)CC)=O)cc([N+](=O)[O-])c(C)cc1Cl c1(NCC(=O)NC2Cc3c(nc(C)s3)CC2)[nH]c(=NCC(C)(C)F)nc2sccc12 Cc1ccn(C)c1C(N1CC(C(F)Cn2cc(CC(C(=O)O)C3CC3)nn2)C1)=O CC1(NC(c2cnc(F)s2)=O)CCN(C(C2CCC(C(F)(F)F)CC2)=O)C1 N1(C(C2(OC(C)C)CCC2)=O)CCC(CCNC(C2CCCN2N=O)=O)(CF)C1 N1(C(CC=CCC)=O)CC=C(CNC(C2CCCCC2C)=O)CC1 C(=O)(C(C(C)CC)N(C(=O)C(C1CC1)N(C)C(C)=O)C)N1C(CCC)CCC1 N1(C(c2c(C)ccc(C)c2C)=O)CCOC2(C1)CN(C(C1(F)CCOCC1)=O)C2 C#CCC(CC(F)F)C(=O)N(C(CC)C(=O)NCC(CCC1CC1)OC)C C1(COC)CN(C(c2cc(=N)[nH]c(Cl)n2)=O)CCN1C(=O)C(C)CC1CC1 N1(C(C2C(C)C2C)=O)CC=CC(NC(=O)CCN(c2ccccc2)C)C1 c1(OC)c(F)ccc(F)c1C(N1CC=C(CCNC(=O)CN(C)C(C)=O)CC1)=O N1(C(C2(c3c(C)cccc3)CC2)=O)CC(CNC(=O)C(C)(C)CO)C(F)(F)C1 C1(NC(Cc2n(C)nnc2)=O)CC(NC(=O)C=Cc2ccc(Cl)cc2)C12CCC2 C(CCC(CCC)NC(=O)CCc1ccccc1C(=O)NC)NC(C(C=C=C)C)=O n1(CC)nccc1C=CC(N1CC(NC(=O)CO)CC1C)=O C#CCCC(C(=O)Nc1ccc(F)c(C)c1)NC(=O)CC1(OC)CCC1 C=CC(C)(CC)C(=O)N1CC(NC(c2cccc(Cl)c2Cl)=O)CC(F)C1 C(C(CC1CCCC1)C(=O)NCCC1COCCO1)NC(C=CC(N)=O)=O C(=O)(C1=CC2CCCCCCC12)NC1(CNC(c2cc(N)c(N)nc2)=O)CC1 CC#CCC1C(=O)N1CC1CC1.C1(C)(OC(=O)COC)CCC1 C1(C)(C(C)C)C(=O)N1.C=CC(CC)C(=O)N(CC(=O)NC(C)(C)C)C C(=O)(C(O)CC[S+](C)C)NCC12CC(NC(C3N(C)C(=O)NC3)=O)(C1)C2 C1(CCNC(=O)C=C(Cl)Cl)CCCN(C(=O)Cc2ccc(O)c(F)c2)CC1 C(=O)(C1=CC2(CN(C(c3ccc[nH]3)=O)C2)OC1)NC(CCC)c1ccco1 c1(-c2nc(NC(=O)NC3CC(OCC)C3)sc2)cc(C)ccc1C CCCCC#CC(C)(C)NC(c1c(CO)noc1C)=O c1(C(=O)NCCC(CNC(C(CC=C)C)=O)O)ccc(C(F)F)nc1O N1(C(CCOCC)=O)CCC2(CCN(C(c3ccccc3C3CC3(F)F)=O)C2)C1 CON(CC1CC1)C(=O)C1CCOCCN1C(=O)COCC1CCC1 n1(C(C)C)nnc(C(N2CC3CC2C3NC(=O)CCC(F)F)=O)c1C(F)(F)F C1(C(=O)NC(C)(CNC(=O)Cc2ccc(-c3ccco3)o2)CO)CC12CCCC2 C(=O)(C1=C(C)OCC1)N1CC(CNC(c2c(COC)noc2)=O)C(C)C1 C1(CNC(Cc2ccn(CC)n2)=O)CCCCN(C(c2cc(N)cc(F)c2)=O)C1 C1(CNC(c2coc(Br)n2)=O)CCCCN(C(C2CCCC2F)=O)C1 CN1CC(C)(C)CC1C(=O)NCC1C(O)C(O)CN1C(C1CCCN1C1CC1)=O c1(CC(=O)NCCN(C(C(c2cccc(C)n2)(F)F)=O)C)c(F)cccc1C#N CCC(C)CC(CO)NC(=O)CC(C)(C)CNC(=O)C(C)(C)CNC(C)=O C12(C(=O)NCCN(C(C(C3CCOCC3)C)=O)CC3CC3)C3CC(CC13)C2(F)F C=CCCCC(C(=O)N(c1ccsc1)C)NC(=O)CN(C)CC1CC1 C1(CCC)(NC(=O)CC2CCCOCC2)CCCN(C(=O)CCc2cnc[nH]2)C1 C1(C(N2CC(CCO)(NC(C3CC=C(C)CC3)=O)C2)=O)Cc2nncn2C1 C(=O)(C=C1SCC(=O)N1C)N(CC(C)NC(c1cnnc(Cl)c1)=O)C N1(C(C=CC)=O)CCN(C(c2cc(C)on2)=O)C(C2CCCC2)C1 C1(CCCNC(C2(C=C)CC2)=O)CCN(C(c2ccnc(CO)c2)=O)CC1 N1(C(C2(OC)CCC2)=O)CC2CC1CN2C(c1nc(Br)sc1C1CC1)=O C12(NC(C(COCC)(C)C)=O)CCN(C(c3ccsc3)=O)CCC1C2 CN1C(=O)OCC1C(N1CC(n2cc(CNC(c3ccc(F)s3)=O)nn2)C1)=O C1(NC(CN2C(C)CCC2)=O)CN(C(=O)CSCc2nccs2)C2(CCC2)C1 C1(F)(CNC(C2C(C)C2C)=O)CCCN(C(=O)C(C)(C)ONC(=O)OC(C)(C)C)C1 Cc1nn(C)c(C)c1CC(C)C(N1CCCC(NC(=O)CSC(F)(F)F)C1C)=O C1N=C2N=C(c3c(c(C)nn3C)N2)NCC12CC2.CCCC=CCC CCC(C(=O)OC)C(=O)NC1(CF)CCN(C(C2CCC(C)(C)O2)=O)C1 C1(CCC(N2C(NCCN(C(=O)C(C)(C)C)CC)CCC2)=O)CCCC(=O)N1 N1(C(C2(CC)CCCC2)=O)CCCC2(CC(NC(=O)C(C)C3CCCO3)C2)C1 C1(NC(CCCC(C)C)=O)COC2(C1)CN(C(=O)C(O)Cc1ccccc1)C2 CCCCC(CO)NC(=O)C(CCSC)NC(C1CC(O)C(F)C1)=O C1(NC(C2(N(C)C)CCCC2)=O)CC2CC1CN(C(=O)CCC(F)(F)F)C2 C12CCN(CC1)C(=O)C(=O)NC(=O)C2C.c1(CC)nnc(CC(C)C)o1 c1(C(N(C2CCN(C(C(CCC)O)=O)C2)C)=O)sc2nc(C)nc(C)c2c1C C(CC(CC)C(=O)N(C(Cn1ccnn1)C(=O)NCC(=O)OC)CC)=CC C=Cc1cncc(C(N2CC(C(O)C(N3CC(F)(c4nn[nH]n4)C3)=O)C2)=O)c1 C#Cc1cncc(C(=O)N(CC(CC)NC(C2CCOC2(C)C)=O)C)c1 c1(N)ccc2c(c1)CCC2(C)C.Cc1nc(N2CCOCC2)cc(CN)n1 C(CC)(C(=O)NCC1(CNC(c2ccsc2OC)=O)CC1(F)F)=CC n1(CC)nccc1C=CC(=O)NCCc1cn(CC2(S(=O)(=O)NCC)CC2)nn1 N1(C(C(CC)N(C)Cc2ccccc2)=O)CCC(C)(NC(=O)NC(=O)C(C)C)CC1 C=CCC(C)(CNC(c1cc(CCNC(C2CCCC2)=O)on1)=O)CO c1(C(=O)NC(C(C)NC(Cc2c(C)n[nH]c2)=O)C)ccc2c(c1)ncn2C N1(C(CCC(=O)NC)=O)CCCC(CNC(=O)CC2CCC2)C1C c1(C(C2CC2)NC(C2CCCN2Cc2ccc(Br)s2)=O)cn(C2CCC2)nn1 Cc1cn[nH]c(=NC(=O)C2c3ccc(C(C)C)cc3CN2C(C2CCCCO2)=O)n1 C1(CC(=O)NCC2CC(NC(CCc3cc(C)[nH]n3)=O)C2)CC=CCN1C c1(C(=O)OCC(=O)NC(C2CCCC2)c2ccco2)cccc2nc(O)oc12 c1(C(=O)NCCC(C(C)C)NC(c2ccnc(O)c2)=O)cn2ccc(F)cc2n1 Cc1ccc(C(=O)NCC2(C)CCN(C(C3CC(=O)N(C)C3)=O)C2)c(Cl)c1 C1(OC(F)F)(COCCNC(c2cccc(O)n2)=O)CC(F)(F)C1 C(=O)(CCCC(F)(F)F)NC(C1CN(C(c2cnn(C)c2Br)=O)CCO1)C N1(C(C)=O)CCC(CNC(c2nnc3c(F)cccn23)=O)C(F)(F)CC1 c1(OC)cccc2cc(C(=O)NCC(CCOC)NC(=O)C(=O)NCC3CC3)oc12 C(CCCCC(=O)NC1(C(N)=O)CCN(C(=O)CN(CC)CC)CC1)=CC CC1=NN(C)C(=O)C1CC(N1CCCC(O)(CCNC(=O)CC2CC2)C1)=O C1(CC)CCOCC1(c1nnnn1C1CCC1)NCC(C)Cn1cccn1 N1(CCC#C)CCC(ONC)C1.C1(C(NOC(=O)C)=O)CCC(N)C1 C1(NC(CCC(=O)NCC)=O)CN(C(=O)COc2cccc(Cl)c2C)CCC1C C1(CN(C(C=C(CC)CC)=O)C)C2CN(C(C3CC=CC3)=O)CC12 c1(C(N)=O)sccc1NC(c1ccn(CCNC(C2CCC2(F)F)=O)n1)=O C1(NC(C(=Cc2cn[nH]c2)C)=O)CC(NC(c2cncn2C(C)C)=O)CC1O c1(COC)cc(N2CCCC(CN(C)C(C3(NC(C)=O)CCCC3)=O)C2)ncn1 c1(C(=O)NCC(CCOC)NC(=O)Cc2cnccc2Cl)cccc(N)c1C C1(CNC(C=C(CC)C)=O)CCC(C)N(C(=O)CCSCC(N)=O)C1 CC1(C)CN(CC(=O)NCCn2cc(C(=O)NC3(C)CC3(F)Cl)nn2)C1 c1(C(=O)NCC(C)CC(=O)NCC)cccnc1C.c1c(C#N)ncn1C CCCC(C(O)C(=O)NCC1CCN(C(C)=O)C1)NC(=O)C1=CCCC1 CCCCC(C(=O)N(C)CCNC(c1cccnc1C1CC1)=O)N(C)C [N-]=[N+]=NC1(C(N2CCC2C(N)=O)=O)CCN(C(=O)CC23CCCC2C3)C1 CC1CC2(CCO1)CC2C(=O)NCc1ccc(CNC(=O)C(O)C2CC2)nc1 CCC(F)C(=O)N(C(c1ccccc1)CNC(C1(CCN(C)CC2CC2)CC1)=O)C CN1CCOc2cc(C(=O)NC3(C4CC4)CCN(C(C4CC4(F)F)=O)C3)ccc21 C1(C(=O)NCCC(C)SC)CCN(C(C2CC(CF)C2)=O)C1C C(=O)(C#CC1CCOCC1)NC(CNC(C=C)=O)(C)CO C1(C(c2n(C(CC)(C)C)nnn2)NCC2(C(C)C)CC2)OCCOC1(C)C C1(C(=O)NC(CNC(c2ccc(C)cc2F)=O)(C)C(C)C)CN2CCCC2CO1 C1(C(=O)NCC(C(C)C)C)CC(=O)CN1C(c1c[nH]c(=O)cn1)=O c1(C(N(C2CCN(C(CC(CCSC)O)=O)C2)CCO)=O)cnc(C)c(C#N)c1 C1(CC(=O)N(C(C(N2C(C(CC)C)CCC2)=O)(C)C2CC2)C)CC(=O)NC1=O N1(C(C(CC)C#N)=O)CCN(C(c2cc(C(F)(F)F)n(C)n2)=O)CC1CF C(=O)CCCCCC#N.C=C(c1ccccc1)C C(=O)(CC(C)(C)C(C)(F)F)NC1CN(C(COCCC=C)=O)CC12CC2 N1(C(CCOCC#C)=O)CC(NC(C2CC(OCC)C2)=O)CC(O)C1 N1(C(c2c(C)nc(C)[nH]2)=O)C2CCCC1CC(NC(c1nn(C)c(C)c1Cl)=O)C2 c1(OC)ccc(C(N2CCOC(CS(N)(=O)=O)C2)C)cc1.C1(CNC(=O)NC)CCC1 C1(C(=O)NCCCOCCNC(CN2C(C)CCC2)=O)CC2CCC(C1)C2(F)F c1(CCNC(CN(CC(=O)NCC#CCNC(C(C)OC)=O)C)=O)cccnc1 N1(C(C(CC)COC)=O)CC2(CCC(C(=O)N(C)CC3CCC(C)CC3)O2)C1 C(c1c(C)nn(C)c1Cl)=CC(=O)N(CCOCCCNC(C(CC)C)=O)C CC1(C)CC(C(=O)NC2CN(C(N)=O)C2)C1.C1(=O)C(c2ccoc2)N1 C1(CNC(COC)=O)CCC2(CCN(C(C)=O)CC2)O1.C12(CC=CCC1)C(=O)NC2 c1(C(N2C(CN(C(C(C(CC)C)O)=O)C)COCC2)=O)cccc2c1CCO2 C1(CNC(C2CCN(C)CC2)=O)COCCN(C(C2CC(=O)N2)=O)C1 c1(C(=O)NC2CCC(C)N(C(=O)CN3CC=CC3)C2)ccc(Cl)c(N)c1Cl C1(NC(C2C3(N4C(=O)CCC4)CC(C2)C3)=O)CCNC2(CCCC2)C1 N1(C(C2(NC(c3c(C)c[nH]c3)=O)CCCC2C)=O)CC(C#N)C2(CCC2)C1 C(=O)(C(C)CC(N)=O)N1CC(CCC)C(C(N2CCCC2(C(=O)OCC)CC)=O)C1 c1(OC)c(C(N2CCC(O)(C(C)NC(c3c(Cl)cnn3C)=O)C2)=O)ccnc1F CCCC(C)(O)C(=O)NC(C)CC(C)NC(=O)CSc1cnn(C)c1 N=c1[nH]c2ccc(C(N3CC=CC3CNC(=O)CCN3CCCCC3)=O)cc2s1 c1(C2(NC(=O)NCC3CCN3Cc3ncoc3C3CCC3)CC2)ccccc1 CC(O)C(C)C(=O)NC1CC(NC(C2(c3ccc(Br)cc3)CCC2)=O)C1 C1(NC(CCc2ncc(C)[nH]2)=O)CN(C(C2CNC(=O)N2)=O)CC12CC2 c1(NC(=O)CN(CCC(C)C)C(C2CCCN2CC)=O)cnc(O)c(OCC)c1 C(=O)(C(C(C)C)SC)NC1(COC)CC(NC(=O)C(c2ccc(F)cc2)COC)C1 S(=O)(=O)(CC(=O)NC1CC(NC(=O)C=CC2CCCCC2)CC1O)NC S(=O)(=O)(c1cc(C(F)(F)Cl)no1)N1CCCC(CCS(C)(=O)=O)C1 Cc1cc(Br)cc(C(N2CCCCC2c2cn(-c3cc(F)cc(F)c3)nn2)=O)c1F c1(-c2ccc(CN(CC(C(=O)O)O)C3CC3)cc2F)c(F)ccc(Cl)c1Cl c1(-c2nc(CN(CCCC)C)on2)ccc(OC)cc1 C1(NC(C(CCCC)C)=O)CC2CC(C1)N(C(C1CCC(F)C1)=O)C2 C12(C(=O)NCCOCCN(C)C(c3cc(C#N)c[nH]3)=O)CCCC1(C(N)=O)C2 n1(CC)nnc(C(=O)NCC#CCNC(c2cccc(CCO)c2)=O)c1C C(=O)(C1CCCc2nc[nH]c21)NCC1CN(C(C2(CC)CC2)=O)CC1O Cc1ncc(N)cc1C(=O)NC(CNC(c1nnc(O)nc1O)=O)C(C)C(C)C N1(C(COCCC)=O)C2CCC1CC(C(=O)NC(c1ncc(C)s1)C)C2 C=CCC(C)(O)C(=O)NC(c1ccc(C)cc1)CNC(c1cn2c(n1)CCC2)=O CC1CCCN1CCNC(=O)C(Cn1cccn1)NC(=O)CNC=O N1(C(c2c(CC)scn2)=O)CCCC2CN(C(C3CC(C)(O)C3)=O)CC12 c1(CCC)nc(=NCC2CCCCN2C(C2CN(C3CCOCC3)C2)=O)s[nH]1 c1(C(N2CC(C(C)NC(c3c(CC)noc3)=O)C2)=O)cc(C)c(F)cc1O C(=O)(C1CCCc2nc[nH]c21)NC(CNC(CNC(Cc1c(C)ncs1)=O)=O)C c1(CC)ccc(C(=O)NCc2n[nH]cc2C(=O)NC)o1.N12CC(C)(C1)OCC2=O N1(C(c2c(C#C)cn(C)n2)=O)CCOC2(CCCN(C(=O)C(=O)NCC(F)F)C2)C1 C1(NC(C=C2CCC(C)C2)=O)CN(C(=O)Cc2c(Br)cnn2C)CC12CC2 Cc1cc(CC(N2CC(N(C)C(c3c(Cl)csc3Cl)=O)C(C)(C)C2)=O)cc(C)c1 Cc1sc(C)c(C(=O)NC2CCN(C(c3cnn(C)n3)=O)CC2)c1Br N1(C(CSc2ccc(OC)cc2)=O)CCC2(CCC2)C(NC(c2nncs2)=O)C1 N1(C(CCN(C)CC)=O)CCC2(CCCC2C(=O)O)C1.C1(O)CC2CCC1C2 N1(C(C2CC(C)CN(C(C3C4CC5C(C4)C35)=O)C2)=O)CCCCC(F)(F)C1 CC1CC(NC(C2CCCC2)=O)CN1C(c1cncc(OC(F)F)c1)=O C1(C(N(CC(=O)NCC(C)C(C)(C)C)CCOC)=O)CC12CCOCC2 C1(CO)CC2(O)CN1CCCn1cc2nn1.c1(NC(=O)CCCF)ccc(Br)cn1 C1(NC(c2cn(CC)nc2)=O)CCN(C(C2(C3CCC3)CC2)=O)CC1CO N1(C(C(C)NS(c2ccc(C)c(C(=O)O)c2)(=O)=O)=O)CCC2(CC(=O)NC2=O)C1 c1(C(=O)NC(CC=C)CNC(=O)C=Cc2sccc2C)cnn2ccccc12 C#CCCCCC(=O)NC1CC2CC(NC(=O)CCC(F)(F)F)C2C1 c1(C(=O)NCCc2cc(C(=O)NCCS(CC)=O)no2)ncc(F)cc1C c1(C2C(C)N(C(c3ccc(C#N)o3)=O)CCC2)cccc2nc(C3CC3)[nH]c12 C1(C(CC)OC(CCOCCOC)=O)CCN(C(=O)OC(C)(C)C)C1 CCC(C#N)C(=O)NCC1(C)CC(NC(C2CN(C(C)C)C2)=O)C1 CN1CCN(CC(C)(C)C(=O)N2CCCCC2CNC(=O)CC2CCCC2)CC1 N1(C(C(C2CCCN2C(c2ccnc(C)n2)=O)OC)=O)CCCC(C)(CO)C1 C1(C(=O)Nc2c(OC)ccc(F)c2)C2C(CN1Cc1cncs1)C2(C)C C12(CNc3c(NC(N4C(C)CC(CO)C4)=O)cccc3)CCC(CC1)OC2 C1(NC(c2cn3cccc(F)c3n2)=O)CCC(N=c2[nH]ccn3ncc(Br)c23)C1 c1(N2C(=O)CC(NC(C(c3ccc(OC)cc3)OC)C)C2)cccc(C#N)c1 c1(NC(C2CCC2(C)C(=O)O)=O)cccc(Cl)c1.CCCCN1CCC1 C1(CCNC(=O)Cc2ccccc2)CCCN(C(=O)C(F)(F)CC2CCC2)C1 c1(C(N2CC(OC)CC2CCC)C(=O)NCC=C)cc(OC(F)(F)F)cc(Br)c1 N(C(=NCCF)NCCNC(C)=O)CC(C(C)C)OCC=C C1(C(F)(F)F)(C(N(CC(C)CNC(C2CC(n3ccnc3)C2)=O)C)=O)CC(F)(F)C1 Cn1ncc2c(O)nc(N3CCC4(CCC4)C(CNC(C4CC4C(N)=O)=O)C3)nc12 N1(C(CC2CN(C)C2)=O)C2CCCC1CC(NC(=O)CCc1ccon1)C2 N1(C(CC=CC=C)=O)CCC12CN(C(c1ccc(-n3nc(C)cc3C)cc1)=O)C2 N1(C(Cc2c(C)cc(C)s2)=O)CC(C)CN(C(c2cccnc2O)=O)CC1C N1(C(C(CC)C2CCOCC2)=O)CCC(CO)(NC(=O)CN2CCC(F)C2)CC1 C(=O)(C1=CCSC1)N1CCC(C(C)CNC(=O)C(CO)N(C)C)C1 C1(COC)(NC(c2ccn(CC)n2)=O)CN(C(c2cc(C(C)C)[nH]n2)=O)C1 C1(CCNC(CNC(N)=O)=O)COCCN1C(c1sccc1CO)=O C(CCC(CCC)NC(=O)C(c1cccc(Cl)c1)O)NC(COCCC=C)=O C1(NC(CCC(=O)OCC)=O)CCCCN(C(c2cc(CC)ccc2C)=O)CC1 C1(CNC(C(C)Cc2ccnn2C)=O)CN(C(c2c(C#N)ncn2C)=O)CC12CC2 C1(N(C(=O)COC2CCCOC2)C)CN(C(c2c[nH]ccc2=O)=O)CCC1(C)C C1(NC(Cc2cccc(SCC)c2)=O)CCN(C(c2nnn(C)c2N)=O)CC1C Cc1ccc(C)c(CC(=O)NC(C2CN(C(c3ccoc3)=O)C2)C)c1 Cc1cncc(C(c2nnnn2C2CCOC2)NC2CCC=CCC2)c1 C1(C(=O)Nc2c(OC)nccn2)C2CCC(C2)N1Cc1cccc(CCO)c1 CCCC(C)CC(=O)NCc1ncoc1CCNC(c1ncnc(O)c1F)=O C1(C(=O)NC(C2(C(=O)NCCc3ncon3)CC2)C)CCC(C)O1 C1(CNC(c2cc(C)on2)=O)CCC2CN(C(c3cnoc3)=O)CCC2C1 C1(C(=O)NCCCCN(C)C)CCN(C(c2cc[nH]n2)=O)C1(C)C N1(C(C2CC(=C)C2)=O)CCC(C(C)(O)CNC(=O)CCc2cc(OC)no2)CC1 C(c1ccc(F)cc1)=CC(=O)N(C)CCOCCCNC(C1CCC(F)C1)=O Cc1c(C(N2CCN(C(=O)C(C)C(C)(C)C)C(C)C2)=O)ccc(N)c1Cl CC1CN(C(=O)COC2CCCCC2)CCCN1C(=O)CCC1CCOC1 c1(C(N(CCNC(CCC(=C)Br)=O)C)=O)cn(C)c(=O)c2ncnn12 c1(C(c2n(CC)nnn2)NCc2c(Cl)nc(Cl)n2C)cc(O)ccc1[N+](=O)[O-] c1(C(=O)NC(C(C)NC(C(C)(C)OC(C)C)=O)C)cc2cc(Cl)cc(Cl)c2[nH]1 CC(C)(C)C(CO)C(=O)NCC1(C)CCN(C(=O)CCC2CC2(Cl)Cl)CC1 c1(C(=O)NCCC2(O)CCN(C(C3N(CC)CC3)=O)C2)ccc(Br)nc1N C(=O)(C#CC1CCCO1)NCC1=CCN(C(Cc2c(C)ccc(C)c2)=O)CC1 C(CC(C)C(=O)NC(c1cn(CCCC)nn1)C(=O)NC)=CC C1(C(=O)NC2CCCN(C(=O)COc3ccsn3)C2)CCC2(CC1)CC2 C(=O)(CC(C)C(C)C(C)C)NCC(C)(C)NC(CCCCC(C)C)=O c1(NC(C(CCOCC)NC(CCOCC#C)=O)=O)ccc(F)nc1F c1(C(=O)NCC(N(C)C(C2(CO)CCCO2)=O)C2CC2)cccnc1N N1(C(CCCCOC)=O)CCCCC2(CCN(C(=O)C(CC(C)C)OC)C2)C1 CCCCCC(C(=O)NC1CCN(C(c2c(F)c(F)cc(F)c2F)=O)C1)C(C)C CCC(C)CC(C)C(=O)N1CC(O)(C(C)(C)CNC(c2cncc(N)n2)=O)C1 c1(CCC(=O)NCCN(C(=O)C(n2ccnc2C)C)CCC)c(C)noc1C CC1(C)CCOCCN1Cc1nc(C2CCCCC2)no1 C(=O)(CCCCC(C)C)Nc1ccc(CO)cn1.C12(CC)CCCN1C(=O)N2 C(CCC(=O)N)NC(=O)OCC.C1(COC2CCC2)CN(C(=O)C(C)OC)C1 C(=O)(C(C)CCCc1ccccc1)NC1CC(CNC(C=C(C)C2CC2)=O)C1 c1(C2CN(C(C(N(C(=O)CC3CC=CC3)C)C3CC3)=O)C2)cnn(C)c1 CCC(CC)(CCC(=O)NCCCNC(=O)CN1CCCCC1C)[N+](=O)[O-] N1(C(C2C(C)C2C)=O)CC2(C(=O)NCCCCCN(C)C)CCC1CC2 N1(C(C(C)NC(=O)OC)=O)CCC(O)C(N(C)C(c2cnc(C)s2)=O)C1 c1(C(N2CC(NC(c3cc(F)c[nH]3)=O)CC23CCC3)=O)ccc(F)c2[nH]ccc12 c1(C(=O)NCCCC2(NC(C3CSCC(=O)N3)=O)CC2)c(Cl)ccc(F)c1F c1(OC)ncc(C)c(C(N2CC3CC(C2)N(C(C2CC4(C2)CC4F)=O)C3)=O)c1Cl C1(NC(C2(C)CCC2)=O)CN(C(c2cnc(-c3ccccc3Cl)s2)=O)CC1O N1(C(c2cnc(N3CCOCC3)s2)=O)CCCCC(NC(=O)NCCCCl)C1 c1(CC(=O)NCC(C)NC(c2cn(CC(CC)O)nn2)=O)ccc(OC)c(O)c1 C12(C(N3CC4(CN(C(=O)COc5cccc(Cl)c5)C4)C3)=O)CC=CCN1CCC2 N1(c2snc(C(C)C)n2)CCCC(C2(NC(=O)CCC3CCCCCC3)CC2)C1 N1(C(c2ncoc2)=O)CCCCC1C1CCN(C(C2CC(C(F)(F)F)C2)=O)C1 C#CCC(C)C(=O)N1CCC(n2cc(CNC(c3cnn(C4CC4)c3)=O)nn2)C1 Cc1cc(F)c(F)cc1NC(C1CC(F)CN1Cc1cccc(Br)n1)=O C1(C(=O)NCC2N(C(CCCn3ncc(C)c3)=O)CCC2)CC2(CC(OC)C2)C1 CC#CCCCC(=O)N1CCC(CCOC)(NC(=O)C(SC)SC)CC1 C1(NC(CC(C)C2CC2)=O)CCC12CCN(C(c1ccc(C3CC3)cc1)=O)CC2 N1(C(c2c(C)cc(OC)nc2)=O)CCC2CCCN(C(c3cc[nH]n3)=O)C2C1 c1(C(=O)NC(C(C)NC(=O)C(c2ccccc2)OC(C)(C)C)(C)C)nccnc1N N(C(=NCCc1c(C)cccc1C)N1CCC=C(S(=O)(=O)N(C)C)C1)C(C=C)C C(=O)(C(C(=O)N1CCC(N(C)C(c2ccc(C(C)(C)C)nc2)=O)C1)OC)OCC c1(C(=O)NC(CC)CNC(=O)C(O)CC2CC2)cc(OC)cc2c1NCCC2 c1(C(=O)NC(CC)C2CC2)coc2c1CN(C(=O)CCc1ccc[nH]1)C2 c1(OC)cc[n+]([O-])c(C(=O)NC(CN(C(=O)C=CC2CCCO2)C)(CO)CO)c1 c1(C=O)cccc(C#N)c1.C(=O)(C(C)=CCN)OC C1(C(=O)NC2C=CCC(C(N(C3CCCCC3)CC)=O)C2)CCCC12CCC2 c1(C(N(CCC(=O)NCCC(C(=O)OC)O)C2CC2)=O)nccc2cc[nH]c12 N1(CC)CCN(CC(N2CCN(CC(N3CC(F)(CC#N)C3)=O)CC2)=O)CC1 CC1(NC(=O)Nc2cc(F)cc(Cl)c2)CC2(C1)CC2(F)F C(=O)(C(O)C(C)(C)C)NCC(N(C(C=C(C)C)=O)C)C1CC1 C(CC(=O)N(CCCO)OC)N(C(C)CC(=O)O)C(C=C)=O c1(CNC(C2(C)CN(C(c3c(C)n(C4CCC4)nc3)=O)C2)=O)cc(Cl)nnc1O c1(NC(c2ccccc2F)COC)cc(C)c(S(=O)(=O)NCCC2CCC2)cn1 C12(CNC(C(C)c3cccs3)=O)CCC(CC1)N(C(C1CCN1C)=O)C2 N1(C(C2CCCCC2C2CC2)=O)CCN(C(C2(F)CCCCC2)=O)C2(CCC2)C1 N1(C(CCOCCOC)=O)CCCN(C(c2ccsc2)=O)C(C)C1 CC1(C)CC=C(C(=O)NC2C(NC(C3CCCN(C(C)(C)C)C3=O)=O)CC2)CC1 C(=O)(C1CC=Cc2ccccc21)N1CC(C)(NC(c2ccc(C)c(C)n2)=O)C1 N1(c2nnc(CC)o2)CCN(CC(O)CN(c2ccccc2)C(=O)COC)CC1 C12(NC(c3ccc(CSCCC)o3)=O)CCC(CC1)N(C(C1CC1(F)Cl)=O)C2 n1(CCC2CC(C)CN(C(=O)OC(C)(C)C)C2)ncc(S(C)(=O)=O)n1 C1(CC#C)(C(N2CCN(C(c3ccnc(C4CC4)n3)=O)CC2)=O)CCCCO1 CC(C)CC(C)(O)C(=O)N1CC2CC(N(C)C(c3ccn(C(F)F)n3)=O)C1C2 CC1(C)CCCCC1(C)n1cc(C(C)(C)NC(=O)CC2(OC(=N)O)CC2)nn1 c1(C(=O)NCC(CNC(C2C(C)(C)CC2)=O)CO)nc(Cl)ccc1OCCF CCCC(C)(CC)NC(=O)CCOCCNC(=O)CCc1cc(C)[nH]n1 Cc1cccc(Cl)c1C(=O)NC1CC(CNC(c2cccn(C)c2=O)=O)C1 C12(C(N(C)CCNC(=O)C(F)CC3CC3)=O)COC(CCO1)C2 c1(CC(=O)NCC(CNC(C(C)SCC)=O)OC)cccc2sccc12 C#CCCC(C(=O)NCC1(CF)CC1)NC(=O)Cc1nc(=N)[nH][nH]1 N1(C(C=Cc2ccc(CC)o2)=O)CCCCC(C2CN(C(=O)CC(C)(C)O)C2)C1 C(CCC(C)C)(C(=O)NC(c1ccn(C)n1)C)NC(c1c(CC)nn(C)c1)=O c1(CC(=O)N(CCCOCCNC(c2c(C)ncs2)=O)C)cncnc1O C1(C(=O)NCC2CN(C(c3c(C)sc(Cl)n3)=O)CC2O)CCc2ccnn2C1 C(C(C)(C)CNC(C1(O)CC1)=O)N(C(C1CC(C(=O)OC)C1)=O)C C1(C(N(CCNC(c2ccc(C3CC3)nc2)=O)CC)=O)CCCCC1C1CC1 Cc1nn(C)c(=O)c(C(=O)NCC2CCN2C(C2CCCS2)=O)c1C c1(NC(c2ccnc(OC3CNC3)c2)=O)cc(F)cc(Br)c1Cl c1(C(=O)NC(CN(C(=O)CCSC2CCCC2)CC)C)ccc2ncccc2n1 CCCC(CCO)NC(=O)C(C)N(C(=O)CCc1nc(=N)[nH][nH]1)CC C1(C(=O)NCC2(O)CCN(C(c3c(C)n(CCO)cc3)=O)C2)CCCC(C)(C)C1 C12CCC(C1)C(=O)N2.C=C1CCC1NC(=O)CNc1nccs1 C(=O)(C1=CCCC(C)(C)C1)NC1CN(C(C(C=C)(C)CCOC)=O)CC1C CC1(C)OCCCC1CS(N1CC2CC(C(=O)O)C1C2)(=O)=O c1(C(=O)NC(C)CCCNC(=O)Cc2cccn2C)cc(F)cc(Cl)c1O c1(C(=O)NCC2CC(NC(=O)C=CC(F)(F)F)C2)sccc1OC(F)F C(N=c1nc(C#N)[nH]cc1Cl)C1CC(NC(C(CC(=C)C)OC)=O)C1 c1(NC(C(C2CCCCC2)C)=O)ccnc(-c2nccs2)n1 N1(C(CC(CCC)NC(=O)C(CCC)N(C)C)=O)CC(=O)N(C)CC1C N1(C(C(CCSC)OC)=O)CCC(F)C(NC(=O)Cn2cc(F)ccc2=O)C1 N1(C(C2(N(C)C(c3cc(C#N)cs3)=O)CC2)=O)CC2OCCN(C)C2C1 c1(OC)ccc(F)c(C(N2CCN(C(=O)CNC(=O)CNC(=O)OC)CC2)=O)c1 C1(CNC(C(C)OCC#C)=O)CCCCC1NC(=O)C(C#N)=CC1CC1 O=C(CCCCC1CC1)NCC1CCN1C(C1CC1CF)=O c1(OC)ccc(C(C)NCCC2COCC2F)c(C)c1OC c1(C(=O)Nc2n(CC)ncc2C(=O)OC)ccc(S(C)(=O)=O)cc1 Cc1nc(-c2cccs2)sc1C(=O)N(CC(C)(C)NC(=O)C=CCF)C n1(CC2C(C(=O)NC)CCC2)cnc(C2(C(=O)NCCOCC)CC2)c1 C1(C)(NC(CCNC(=O)NC)=O)CC(CNC(=O)CC2CC3CC3C2)C1 c1(OC)cc(NC(=O)CC2CCCN(C(n3cc(Br)ccc3=O)=O)C2)ccc1C c1(N2CC(C)NC(=O)C(C)C2)ncc(S(=O)(=O)NCC2(CN(C)C)CCC2)cc1Cl C1(CC=C)(C(=O)NCCC2CC3C=CC2C3)CCCN1C(c1cccc(C)n1)=O C1(CNC(C(CC)C(=O)OC)=O)CC2CCC1N(C(=O)C1=CCCSC1)C2 C1(NC(C2C(OC)CC2)=O)CC2CN(C(=O)CC3(O)CCCCCC3)CC2C1 c1(C(=O)NCCN(C(c2snnc2C)=O)CC)cnc2c(F)cccn12 C1(C(N(C(CC)COC)C)=O)CCCN(C(c2cnncc2C)=O)C1 c1(OC)cc(NC(C2CCN(C(=O)C(C)O)CCO2)=O)ccc1F C12(C(=O)NCCOCCN(C(C3(C)CCCC3O)=O)C)C3C(=O)C4C5CC(C14)C2C35 Cc1cc(=O)ccn1CC(=O)NCC(CO)NC(=O)CC(C)c1ccccc1 Cc1cnc(C(=O)NC(CO)C(=O)N2CCC(OCCNC(N)=O)C2)c[n+]1[O-] C(c1ccc(C=O)cc1)=CC(N1C(Cn2cc(Cc3ncn(C)c3)nn2)CCC1)=O C(=O)(CC(O)C(C)CC)NC(C(=O)N(CC=C)CCOC)c1ccco1 CC(CCCNC(C1CCCN1C1CCCC1)=O)NC(C1(n2cccn2)CCC1)=O Cc1nn(C)c(C)c1C(=O)NC1CCC1CNC(=O)C(C)Sc1ccccc1 C(C(O)CC(=O)NCC1(CNC(c2ccc(C#N)o2)=O)CCCCC1)N(C)C N#Cc1ccc(F)c(C(N2CCC(OC3CCN(C(CO)=O)C3)C2)=O)c1 c1(OC)cc2c(cc1NC(=O)CN1CCN(C)C(CO)C1)OCO2 c12cc(nc(S(C)(=O)=O)n1)N1CC3C(C1)N23.c1(C(=O)OC)cc2ncccc2[nH]1 C(=O)(C(C(C)C)Sc1ccccc1)N1CC(C(N2CC(OCCCCC)C2)=O)C1 C=CCCCC(C(=O)NCCC(C)C(C)C)NC(=O)COC1CCCOC1 C(C(=O)NC)(C(C)C1CC1)N1CC2CC1C(=O)OC2.C(CC#N)OCC#C c1(C(=O)N(CC(C)(C(C)C)NC(CN(CC)CC)=O)CC)cc(C(F)F)cc(C)c1 C(=O)(C(CC1CC1)NC(=O)C(CC)OC)NC(C1CCCCC1)C#C C(CC(F)F)(C(=O)NC1(c2ccccc2)CC1)N(C(C1C=CCC1)=O)C1CC1 S(=O)(=O)(c1ccc(Cl)c(Cl)c1)N1CC2(CCC(C(=O)Nc3ccccc3O)O2)C1 C(CNC(C1(N(C)C)CCCC1)=O)(CC(C)C)NC(C1C(OC)CC1)=O N1(C(COCC(=O)NC)=O)CC2(CCCC(CNC(c3cc(Br)n[nH]3)=O)O2)C1 C1(F)(CNC(c2c(C)snn2)=O)CCC(CNC(C2CCC(F)(F)C2)=O)C1 C(=O)(C1CCCn2nccc21)NC1CC(CCNC(C2(C#N)CCCOC2)=O)C1 C1(NC(CC(=C=C)C)=O)CCN(C(c2cnn(CCO)c2C)=O)CCC1CO C(CCC)(C(=O)NC1CC(NC(=O)CN2CC(C(=O)OC)C2)CC1O)=CCC c1(C(=O)NC2C(CNC(C3(CC(C)C)CC3)=O)CCCC2)ccc(Br)c(O)n1 Cc1csc(=O)n1-c1ccc(C(=O)N(CC(C)N(C)C(C2CC(C)C2)=O)C)cc1 C1(CNC(C2(C)CC=CCO2)=O)CN(C(=O)CSc2ccccc2F)CC12CC2 c1(C(=O)NCCC(N2C(CNC(C(C)SC)=O)C=CC2)=O)ccnc(C)n1 C(=O)(C1=CCCC1C)N(CCCCCNC(C1CCC(CCC(C)C)CC1)=O)C C1(CC)CCC(C(=O)NCC2(F)CN(C(=O)CN3CCC3C)C2)O1 C(=O)(C1CCc2cc(OC)ccc21)N(CCCNC(c1conc1CC)=O)CC c1(C(=O)NCC2N(C(CCC3CCC(=O)N3)=O)CC=C2)ccnc2ncnn12 c1(C(N2C(CNC(c3c(CCC)n(C)nn3)=O)CC2)=O)cnn2c1CC(F)(F)C2 c1(OC)cc(C(=O)NC2CCC(NC(=O)Cc3ccco3)CC2)cc(OC)c1C C1(N(C(=O)CC2(O)CCC2)C)CC2CCC(C1)N2C(C1CC(OC(C)(C)C)C1)=O CC1CCCCC1(CNC(c1cc(C2CCC2)[nH]n1)=O)NC(c1cnn(C)n1)=O c1(C(N(CCCN(C(=O)C=CCN2CCCCC2)C)C)=O)cnc(Cl)s1 c1(C(=O)NCCOC(CNC(c2ccn(C)c2)=O)(C)C)csc2cncn12 C1(CNC(c2cc(CO)on2)=O)CC(=O)N(C2CC2)C1.C12CCCN1C(=O)C21CC1 C1(CC)CN(C(C2CCCC(=O)O2)=O)CCN1C(=O)CC=Cc1cccc(F)c1 N1(C(CCN(CC(C)C)C(=O)COc2ccsn2)=O)CC2CC1C1CC21 n1(CC)ccc(C(=O)NC2CN(C(C)=O)CC2C=Cc2ccccc2)cc1=O Cc1nsc(NC2CC2)c1C(N1CC(CNC(c2ccn(C)n2)=O)C(O)C1)=O Cc1ccccc1CCN(C(=O)C(F)C1CCOC1)CC(C)C.C(C(C)C)S CCC(CC)CCC(c1nnnn1C(C)(C)CC)NC1(COC)CCOC1 CON1CCC(CC(N2CCC(C)(CCNC(c3n[nH]c(C)c3O)=O)C2)=O)CC1 C1(C(=O)NC(C)CCN(C(=O)CCOc2ccc(C)cc2)C)(OC)CCCCC1 c1(CC)cc(F)c(C(=O)NCC2(C)CC(F)(F)CN2C(c2ccsn2)=O)c(F)c1 NS(=O)(=O)c1csc(C(=O)NC(CNC(C2CC(=C3CC3)C2)=O)CO)c1 CCCC(C(=O)Nc1ccc(SC)cc1)NC(c1ccc(CO)cn1)=O N1(C(CCC(C)SC)=O)CCCCC(C(=O)N(CCCC(C)C)C)C1 c1(SCC(=O)NCC2C(NC(Cc3nc(C)[nH]n3)=O)COC2)ccccc1F CCCCC(O)C(=O)NC1CCCC(NC(C2(c3cccc(F)c3)CC2)=O)C1 C1(CNC(c2c(CC)nsc2)=O)C2CN(C(=O)C=C(C)C(C)(C)C)CC12 C=Cn1nncc1C(=O)NCC(CCOC)NC(C1CCCN1C=O)=O C=C=C(C)CC(=O)N1CCSCC1CCNC(c1ccnc(C(F)(F)F)c1)=O c1(CNC(N2CCCC2C(O)C(F)F)=O)nc(Cc2ccccc2)no1 CC(C)C(C)CCNC(C1(NC(c2cc[nH]c2)=O)CCOCC1)=O c1(OC)c(C)cc(C(=O)N(CC(C)CNC(c2coc(O)n2)=O)C)cc1Cl c1(C(=O)NCCC(CNC(=O)C=C(C)C(C)C)OC)cccc(C(N)=O)n1 CN=c1nc(N(C)CC2CCCCC2)[nH]c(N2CCC(=C(F)F)CC2)n1 Cc1cc(C(F)F)n(CC(=O)N(C(C)CNC(c2nsnc2O)=O)C)n1 N1(C(C2N(C)C(=O)CC2)=O)CCC(C(N2CCC(F)(F)CC2)=O)C12CC2 c1(OC)cc(F)ccc1C(=O)NC(c1ccccc1)C(C)NC(=O)CC(C)(C)O C1(CNC(C2CC3(ON=C(C)C3)C2)=O)CC2CCC(C1)N2C(C1CCC1(C)C)=O C1(NC(CC2CC(CC)C2)=O)(CNC(C2CC(C)(CC)C2)=O)CC(C)(C)C1 C1(C)(NC(c2cnc(N(C)C)s2)=O)CCN(C(C2CC3CCC2C3)=O)CC1 N1(C(C(c2ccccc2)SC)=O)CCN(C(=O)CS(N)(=O)=O)C(C)C1 Cc1c[nH]c(C(=O)NCCCC(=O)NCCc2cn(C)nc2C)c1C N1(C(CCSCC)=O)CCOCC(NC(c2cnn3c2SCC3)=O)C1 C#Cc1ccc(Br)c(C(=O)NCC2CC2CNC(c2cnc3cc[nH]c3c2)=O)c1 C1(C)(NC(COC(C)(C)CNC(c2cc(Cl)ns2)=O)=O)C=CCCC1 n1(CC)cc(NC(=O)CC2(C)CCN(C(C3CCSC3)=O)C2)c(C#N)n1 C(c1cccc(Cl)c1Cl)=CC(=O)N(CC(CC)NC(C1CCCN1C)=O)C c1(C(=O)NC(C(=O)NCc2onc(C)n2)CC2CCC2)cnn(C)c1C N1(C(C(c2cncc(F)c2)C)=O)CCC2(C1)CN(C(c1cnn(C3CC3)c1)=O)C2 N12CC(CCC(O)C1)N(C=O)C(C(C)C)C2=O.CC=CCBr.C1CC1 N1(C(C2C(CCC#N)C2)=O)CC2CCC1CN2C(=O)Cc1n[nH]cn1 C1(C)(C(=O)NC2CC(C(C)NC(C3CC(C)(F)C3)=O)C2)CCC(F)(F)C1 c1(C(=O)OC)ccc(NC(C2CCOC(=O)CC2)=O)cc1Cl C1(O)(C(CNC(CC2(COC)CCCC2)=O)C)CCN(C(C2CCN2C)=O)C1 C1(CN(C(Cc2c(C)csc2)=O)C)CN(C(c2n[nH]c(C3CC3)c2C)=O)CCO1 C(=O)(C1CCCc2cncn21)NC1CC2(C(NC(c3cccc(CF)c3)=O)C2)C1 Cc1cc(C(=O)NC(C)CCCCNC(C23CC(C(C)(C)C)(C2)C3)=O)cc(C)n1 N12CCN(CC1)C(=O)C2.C1(C(=O)NCC(C)OC(F)F)CC(F)(F)CS1 CC(C(C)C(=O)N(C)CC1CN(C(=O)C2=C(Cl)CCOC2)CCO1)S(C)(=O)=O C1(C2CCN(C(C3CSC3)=O)C2)(NC(c2nc(C)[nH]n2)=O)CC1 C1(C)(C(=O)NC(C2CN(C(C3CC4(CCO3)CC4)=O)CCO2)C)CCC(O)CC1 C#CCC(CC(=O)OC)NC(C1CCC1NC(c1cn(C)cn1)=O)=O C1(C(N2CC(OCCOC)C2)=O)C(C)OCCN1C(=O)CC1CCCCC1O C1(C2CCN(C(c3csc4ccccc34)=O)C2)(NC(CC(CC)O)=O)CC1 C1(CNC(c2cnc(NC(C)=O)o2)=O)CC12CCN(C(C1(C(C)C)CC1)=O)CC2 C1(C)(C(=O)NCC2=CCN(C(C#CC(C)(C)O)=O)CC2)CC(C2CC2)=NO1 C1(NC(C23CC(COC)(OC2)C3)=O)CC2CC(C1)N(C(=O)C(C)CC(F)(F)F)C2 C1(NC(C(CCC)OC)=O)CC2CCC1N(C(=O)C=C1CCN(C)C1)C2 S(=O)(=O)(c1ccc(OC)c(C)c1)N(CC(C(CC)C)=O)c1cccc(C(F)(F)F)c1 C#Cc1ccc(C(=O)NC(CCF)C(=O)N2CCC(CC3CCC3)C2)nc1 c1(CN2CCC(NC(=O)Cc3ccc(-c4ccccc4)o3)C2)cc(I)ccc1Cl c1(NCC)cccc(C(N2CC=CC2CNC(c2cc(C(F)(F)F)on2)=O)=O)c1 c1(N2CCC(C)(C)S(=O)CC2)nc2cccnc2c(=NCc2cnccn2)[nH]1 Cc1ccc(NC(c2nc(Sc3nnco3)cs2)=O)cc1C C1(C(=O)NC(CC)CNC(c2cccs2)=O)CC(C)CC(=O)N1 c12ccc(c(C)c1)C(=O)N1CCN2CC1.c1(C)cn(CCCC(=O)O)nn1.CO C1(CNC(c2ccc(C)nc2O)=O)N(C(c2csc(C)c2C)=O)CCCC1(C)C c1(C(=O)NCC(CN(C(=O)C(=O)N(C)C)CC)(C)C)cccc(-n2ccnn2)c1 C#CCC(CC(F)F)C(=O)N1CCCC1C(C)NC(=O)CC1(C=C)CCCC1 c1(NC(C(n2cc(CN(C)C)nn2)C)=O)c(Cl)cccc1Cl.C12CN(CCO1)C2 n1(CC)nnc(C)c1C(=O)NCC(c1ccccc1)NC(c1cc(F)n[nH]1)=O C1(C(N(C2CN(c3cc(OC)ncn3)C2)CC2CC2)=O)CCc2ccnn2C1 C(=O)(C1CCc2cccnc21)N1CC2C(CNC(C(C)(C)c3ccsc3)=O)(C2)C1 CC1CN(C(=O)CCC2CCCCO2)C1C(=O)NCCN(C(C)C)C(C)C c1(C(=O)NCC2C(CC(=O)N(CCOC)CC3CCC3)C2)ccc(C)o1 CC(C(=O)N1CC(O)(CNC(C2CCCCN2C)=O)C1)C(C)(C)C CC(c1ccco1)=CC(=O)NCC1OCCC1C(=O)NCCCCCN(C)C C(=O)(CCS(=O)(=O)C(F)(F)F)NCCN(C(C1C(C(C)=O)C1(C)C)=O)C1CC1 C12CCc3nc(ncc3C1)N2.C(=O)(CC(C)n1cccn1)N(CCN(C)CC)C c1(C(C)NC(c2c(C)c(C(=O)O)ccc2)=O)cc(C#N)ccc1O C(C1c2ccsc2CCN1C(=O)CNC(=O)CC#N)NC(C(C)C1CCCC1)=O C=CCC(C(=O)OCC(C)C)N(C1CCC1)CCCC1CCCC1O C1(NC(c2n[nH]cc2C2CCC2)=O)CCN(C(=O)COCC(F)F)C12CCCC2 Cc1cc(F)ccc1C(=O)C(CCF)c1ccccc1 c1(N2C3C(NC(CC4C(C)C4)=O)(CCC3)CC2)ccc([N+](=O)[O-])cc1Cl CCCC#CC(C)(C)NC(C1CC(CCNC(C2C3CCCCCC23)=O)C1)=O Cc1cnc2c(cnn2CC(N2CCCCC(NC(=O)C=C3CCC3)C2)=O)c1 n1(CC(=O)NC(CNC(C(c2cccnc2)OC)=O)C)ccc(=O)n(C)c1=O C(C)(C(CO)NC(c1ocnc1OC(C)C)=O)NC(C1C(C(=O)OCC)C1)=O N1(C(CS(C(=C)C)(=O)=O)=O)CCC2CCN(C(=O)C(O)CCC)CC2C1 c1(C(=O)NC(CNC(C(CC)C)=O)C2CC2)c(-c2ccccc2)nsc1N c1(OC)cnc(F)cc1C(N1CCOCC(Nc2ncncc2I)C1)=O C(C1CCCN(C(=O)N(CC=CC(C)CC)Cc2ccccc2)CC1)=CC(=O)OC c1(OC2CCOC2)ccc(CCNC(C2CC(C(F)F)C2)=O)cc1.O=C1CO1 C(=O)(C1=NNC(=O)CC1)NCc1c(CCNC(C2(C)CC2Br)=O)ocn1 N1(C(c2c(C)onc2)=O)CCC2C1CCCN2C(c1ccc2c(c1)CCCC2)=O n1(CC)nc2c(c1NC(=O)NCCN1CCCC(C)C1)COCC2 Cc1nsc2ncc(C(N3CC(C4CN(C(C5CCS5(=O)=O)=O)C4)C3)=O)cc12 C1(NC(=O)OC(C)(C)C)COCCC1NC(C1CC1NCC(O)CF)=O c1(NC(C2CCN(C(C(C)(C)NC(C)=O)=O)CC2)=O)nc2cc(C)ccc2s1 C1(=O)CS(=O)(=O)CCc2cn(nn2)CC(F)CCN1.CCC(CC)CCCOC N1(C(CC2C(C)=NOC2=O)=O)CCOC2(CCN(C(C3(C#N)CC3)=O)CC2)C1 c1(C(=O)NCCNC(=O)C(F)=C2CCC2)csc2c(F)cc(F)cc12 C1(C(=O)NC23C(CN(C(c4cc(C)n(C)c4C)=O)C2)C3)CC12CCC(F)(F)CC2 c1(OC)ccc(C(C)C)cc1C(N1CCCC(C(=O)NCCC(C)(C)O)CC1)=O NS(=O)(=O)c1cnn(CC(N2CC3CCC2C3NC(=O)Cc2cscn2)=O)c1 C1(CC)CN(C)CCCN1c1ncnc(NCC(C2CCC2)OC)c1C CN1CCN(CC(=O)NCC2CCN(C(=O)C(F)=CCCF)C23CC3)CC1=O c1(OC)cnc(F)c(C(=O)NC2(CNC(=O)CN3CC(C)(C)C3)CCCC2)c1 c1(C(=O)NC2C(NC(c3ccc(C)o3)=O)CCC2)ccn(C)c1C c1(CNC(C2C(NC(C3C(CC)N(C)CC3)=O)CCO2)=O)ccc(C)cc1O C1(OC)CC(CNC(=O)CSc2ccc(C)o2)N(C(=O)CN(C)C(=O)NC)C1 c1(C(=O)NC2CC3CC(NC(C=C(C)C4CC4)=O)CC3C2)cnc2c(C)nsc2c1 N1(Cc2cn(C(O)Cc3ccc(Cl)cc3)nc2)CCC2CCCCC2C1 C(=O)(CCC(=O)C1CC1)NC1C(CNC(COCCN(C)C)=O)C1 C1(CNC(CCNC(CS(=O)(=O)NC)=O)=O)CC(C)(C)OC1=O Cc1cc(Br)c(NC(C2CCCN2C(=O)CSc2ccncc2)=O)c(Br)c1 C1(N(C)CC)CCN(C(C2CCN(C(c3snnc3C)=O)C2C)=O)CC1 Cc1cc(Cl)ccc1CC(N1CCC(NC(c2ccoc2Cl)=O)CC1C1CC1)=O c1(-c2nc(C(C)NC(=O)Cc3ccc(Cl)cn3)sc2)cn(C)c2cc(Cl)ccc12 c1(C(N2CC(N(C)C(C3CC3(Cl)Cl)=O)C(O)C2)=O)cnn2c1CC(F)(F)C2 c1(CN(C(=O)C(C2CCCCC2)O)CCN)cncc(Cl)c1 N1(C(C(CC(=O)OCC)CC)=O)CCC2CCC(C1)N2C(=O)Cc1cnc(C)s1 c1(C(N2CCOCC2Cc2ccccc2)C(=O)NC)ccnc(Cl)c1Cl C1(C)(C(N(C(CCSC)C(=O)O)C)=O)CCCN(Cc2nc(O)ccc2C)C1 N1(C(C=C)=O)CCC2(CCCCN(C(c3ccc4c(n3)CCCC4)=O)C2)C1 c1(C(C)C)c(N2CC(NC(=O)C=C3CN4CCC3CC4)C(C)C2)ncnc1Cl C(=O)(C1CCc2scnc21)N1CC(C)(C)C(NC(=O)COC2CCCOC2)C1 C#CCC(CC(=O)OC)NC(C1(NC(=O)COCCCF)CCSC1)=O C1(C(=O)OC)CC2CC1CN2C(C1(n2cncn2)CC1)=O.C12CC(C1)CCC(=O)N2 c1(OC)ccc(Br)cc1C=CC(N1CC2CC2(NC(=O)C2=CCOCC2)C1)=O C1(CC)CC(C(N2CCN(C(=O)CC3COCCN3C)CC2)=O)CC(=O)N1 Cc1ccnc(C(=O)NCCN(C2CCCC2)C(C2CCNC(=O)C2)=O)c1F N1(C(c2cc(CSC)c(C)s2)=O)CC(NC(=O)C(O)C2CC2)CCC(O)C1 c1(C(N2CC(C3CN(c4ncc5ccsc5n4)C3)C2)=O)cccc2cccc(Br)c12 c1(NC(Cc2nc(NC(CCc3n(C)ccc3)=O)sc2)=O)c(F)cc(Br)cc1Cl c1(C(=O)NC2CCN(C(C(C)OC(C)(C)C)=O)CC2O)c[nH]nc1S(N)(=O)=O N1(S(CC)(=O)=O)CC2(CCN2C(c2ccc(Br)c(C)c2)=O)C1 C1(C(=O)NC2CC(N(C(C3(C=C)CCC3)=O)C)C2)CCc2cn(C)nc2C1 N1(C(CCCC=C)=O)CCN(C(C2CCN(C)C2)=O)CC1CC(=O)NC c1(NCC2N(C(=O)OC(C)(C)C)C2CCC2CC2)cnc2c(F)ccc(F)c2c1 N1(C(C(=O)NC(CC)(C)C)=O)CCOC(C(=O)OC)C1.N1(CC)CCC(N(C(C)=O)CC)C1 C1(CC(=O)OC)CCC(OC)CC1.n12cc(nn1)CCCCOC(=O)C2 CC(C)(C)C(C)(O)CNC(=O)NC1CCN(C(C23CCCC2C3(F)F)=O)CC1 CCS(=O)CC(=O)N1CCC(C(=O)NCC(F)F)(CO)C1 c1(CC(=O)NCC2CN(C(=O)CSC(F)F)CC(C)(C)O2)cc(F)cc([N+](=O)[O-])c1 CC(C)CC(C)C(=O)NC(CO)C(=O)NC1CC(CCC(N)=O)C1 C1(NCc2c(-c3nnc(CCC)o3)cccc2)COC2(CCOCC2)C1OC C(=O)(C(C)CCCC(C)=O)N1CCCCC(CNC(c2cc(SC)c(C)o2)=O)C1 c1(C(N2CC(CCNC(CN(C(C)=O)C)=O)OCC2)=O)cccc2[nH]nc(O)c12 C(=O)(C1CCc2cc(C)ccc21)N(CC(C)NC(=O)CC1CCCCC1O)CC C1(C(N2CCC3CN(C(C(C)OCC(C)C)=O)C3C2)=O)CCN(S(N)(=O)=O)CC1 N1(C(C2(C(=O)NC)CCC2)=O)CC(C(=O)N(C)CC2CCCOC2)C2(CC2)C1 N1(C(CC(=O)OCCC(C)C)=O)CCCC(NC(=O)CC2CCSCC2)C1 c1(CC(N2C(CCC(=O)NCC(CC(=O)NC)C)CCCC2)=O)ccc(C#N)cc1 C1(CN(C(=O)C=Cc2cncs2)C)CCCN1C(C1CCC1)=O Cc1ccc(Br)c(OCCNC(C23CC2CN(C(c2cncs2)=O)C3)=O)c1 C(=O)(CCCCC(N)=O)N1CC(=C(CNC(C2C(C)CC(=O)N2)=O)F)C1 C1(c2cn(CCNC3CCCN(C(=O)C(F)(F)F)C3)nn2)(N(C)C)CCOCC1 CC1CCC(NC(=O)CN(C)C(c2ccccn2)=O)CN1Cc1cccs1 N1(C(C(CCC)C)=O)CCCC2C1CCN2C(c1cc(Br)c(C)o1)=O N1(C(CCC=C=C)=O)CCN(C(c2cc(O)ccc2Cl)=O)CC2CCCCC12 N1(C(CC2(C)CCCO2)=O)CCN(C(=O)CNC(c2ncc(F)cn2)=O)CC1 N1(C(c2[nH]nc(OC)c2Cl)=O)CCN(C)C(CNC(c2cnc(C3CC3)s2)=O)C1 c1(C(=O)NCC2(C)N(C(C(CCCC)C)=O)CCC2)ccc2nc(C)nn2c1 c1(C(=O)NC2(CO)CN(C(c3cc(C(C)(F)F)n[nH]3)=O)C2)ncncc1F C=C(CNC(C1CN(C(c2ccc(CC)cn2)=O)CC1F)=O)C1CCOCC1 C12(CNC(C(C)=C3CCCC3)=O)CCC(CC1)N2C(=O)Cc1csc(S)n1 c1(C(=O)OC)c(C)[nH]c(C(=O)NC(c2cccc(Br)c2C)C)c1C C1(C(N(C2CCN(C(C(C)C3CC3)=O)CC2)CC2CC2)=O)CCn2nnnc2C1 CC(CC(=O)N1CCC(CN(C)C(c2c[nH]nc2C(F)F)=O)C1)c1ccco1 N1(C(CCC)=O)CC(CNC(C2(CCF)CCOCC2)=O)CCC1C N1(CCC)CC(C(N2CCC2CNC(c2cccc(N(C)C)c2)=O)=O)CC1=O CN(CP(C)(C)=O)C(c1ncoc1CNC(C1SCC=C1C)=O)=O C1(CC)(NC(C2(CO)COC2)=O)CCN(C(=O)CC2CCC(C3CC3)O2)CC1 c1(OC)ccc(C(=O)NC2CCCN(C(C3CC3C#N)=O)CC2)c(OC)c1OC C1(CC)CCCC1C(=O)N(CCC(=O)NCC1(OC)CCCC1)C N1(C(c2c(CNC(C3CC4C=CC3C4)=O)ccs2)=O)CC2(CCC2)C1 CCCC(F)C(=O)NC1CCOCC1NC(C1CNC(=O)N1)=O c1(CN(C2CCCC2)C(CC2CN(C(C(C=CC)O)=O)C2)=O)cccnc1C C1(C(N(C(C)CC)CCC)=O)CC1C(=O)NC(C1CC1C(N)=O)C c1(C(C)(C)C)ccc(N)c(C(=O)NCC2CCCN2C(c2[nH]ncc2C#N)=O)c1 c1(C(=O)NC2C(C(=O)NCCC3C(C)(C)CCO3)C2(C)C)ccc(N)c(F)n1 c1(C(=O)NC2C(NC(C(CC(=C)C)C)=O)C2)cccc2oncc12 CC(C)CS(=O)(=O)CC(=O)NCC1C2CC1N(C(=O)CC(C)O)C2 N1(C(=O)Cc2cccs2)C2CC1CN(C(c1cnccn1)=O)C2 c1(CC(N2C(C(C)NC(=O)C=CS(C)=O)CCC2)=O)ccc(O)cc1Cl O=CN1CCCN(C(C2C=CCN(C(c3ccc(O)cc3)=O)C2)=O)CC1 c1(CC(C)NC(c2cccc(F)c2)C2CC2)cc(F)c(C(F)(F)F)c(F)c1 N1(C(C2N(C(C)=O)CCCC2)=O)CCC(NC(=O)CC2(C)CCOCC2)CC1C c1(C(C(=O)NCCCC)N(C(C)C(C)C)C)oc(C(=O)OCC)cc1Br Cn1[nH]c(=NC(=O)C2C=CC(NC(=O)CC3CC4CC4C3)C2)cc1C(N)=O N1(C(CCC=C=C)=O)CCC(CNC(=O)CN(C)Cc2ccccc2)C12CCC2 Cc1ccc(C(F)F)cc1C(=O)NC1CC(C)CN(C(=O)C=CC=C(Cl)Cl)C1 c1(C(=O)NC(C(N2C(C(=O)OC)CC2)=O)C2CCCC2)snc(C)c1N N1(C(CC(CC)O)=O)CCC2CCN(c3ccnc(S(C)(=O)=O)n3)CC2C1 c1(C(N2C(C(=O)NCCC(CC)C)CC3CC32)=O)nc(C)ccc1C c1(C(=O)NC(C(=O)NC(C(=O)NCC)C)C2CC2)ccc(=NC)[nH]c1 C1(C(N2CC(C)(NC(CS(N3CCN(C)CC3)(=O)=O)=O)C2)=O)CC(S(N)(=O)=O)C1 c1(C(N2CCCC(NC(=O)Cc3ccc(Cl)s3)CC2)=O)nccc2ncccc12 c1(C(=O)NCC2CC(C)(C)CN2c2nnc(CC(F)(F)F)s2)cccn2cnnc12 Cc1ccc([N+](=O)[O-])c(NC(c2n[nH]cc2NC(c2ccc(Br)c(C)c2)=O)=O)c1 C(=O)(CC(C)CC(C)C)N1CC(N(C(c2c(SC)cn(C)n2)=O)C)C1 C(=O)(C(C)(F)C(=O)NCCCC(C)NC(c1ccc(=O)n(C2CC2)c1)=O)OC S(=O)(=O)(c1ccc(Br)s1)N1CC(C(=O)Nc2cc(Br)cnc2O)C1 N1(C(c2cncc(N(C)C)c2)=O)CCC(C)(NC(=O)C=CC2CCC2)CC1 N1(C(c2c(C)oc(C#N)c2)=O)CC(C)CN(C(=O)C2=NNC(=O)C2)C(C)C1 C1(CC(=O)NC2CCC(NC(c3c(CC)n[nH]c3)=O)C2)CCC(OC)CC1 C=CCCCCC(=O)Nc1cc(-c2cnn(C3CCC3)c2)[nH]n1 N1(C(c2scc(C)c2Cl)=O)CCCCC2(CCN(C(=O)CC3(O)CCOC3)C2)C1 c1(C(=O)NCCN(CCC)C(C2CCC(F)CC2)=O)cc2nnn(C)c2s1 N1(C(N2C(c3onc(CC)n3)CCC2)=O)CCSCC1C1CCC1 CCC(CNC(C1C2CC1N(C(c1cc(C)c(F)cn1)=O)C2)=O)(CC)CC C1(CNC(c2c(C)snn2)=O)CC(NC(c2ncc(C(F)F)s2)=O)C12CCC2 c1(SCC)c(C)[nH]c(C(N2CC(NC(C3CCSC3)=O)CC(C)C2)=O)c1C(C)C S(=O)(=O)(c1c[nH]c2ccc(Br)cc12)NC(C1CCCN(CC=C)C1)=O C12(c3n(C)ncc3)CCC(CC1)N2Cc1ccc(Br)nc1O c1(-c2cc(CN3CC4(C(C(=O)O)COCC4)C3)[nH]n2)coc2cc(O)ccc12 C1(C(=O)NC(C2CCCN(C(=O)CN3CC(C)(C)C3)C2)C)CCCN2CCCC12 C1(NC(C(c2cn(C)nc2)O)=O)CN(C(c2cccc(CC#N)c2)=O)CC12CC2 C(CCCCC(=O)N1CCOC(C(=O)NC23CCC(C2)C3(C)C)C1)SC C1(CCC)CN(C(=O)C(C)CC2CCC2)CCN1C(=O)Cc1ccns1 Cc1cc2ccccc2nc1C(N1CCOCC1CNC(=O)CC=CC(C)(C)C)=O C1(NC(CC2CC(=O)NC(=O)C2)=O)C2CCC1CN(C(C1(CF)CC(F)(F)C1)=O)C2 C(=O)(C1=CC2C=CC1C2)NC1C(C(N(C)CC2CC2(F)F)=O)CC1 N1(C(C(C=C)c2ccccc2)=O)CCN(C(c2nnn(C(C)C)n2)=O)CCC1C c1(C(c2ccccc2)C(=O)NC(CC)CNC(=O)CCC#N)cccc(OC)c1 C(=O)(CCCC(=O)NCC(C)CNC(C1(OCC)CCC1)=O)OC(C)=O C1(CCNC(C(C2CCC2)OCC)=O)(C(=O)NCC2C=CCOC2)CCCC1 c1(C(=O)NC2CCCN(C(CSCC=C)=O)C2)c(C)nc(C2CC2)nc1S Cc1ccc(C(=O)NCc2ccc(CNC(=O)C(C)n3ccnn3)cc2)cc1F C1(C(N2CCN(C(c3nc(C)nn3C)=O)C(C(F)F)C2)=O)COC2COCC2O1 CC(C)(CNC(C1CCCN1C(=O)CNc1ccccn1)=O)CC(F)F C1(C(=O)NCC(C)(C2CC2)NC(c2ccc(CSC)o2)=O)CCCC12CCC2.C1(C)CC1 c1(C(N2CC(C)CC(NC(C(C)OCCC=C)=O)C2)=O)cnc2cc[nH]c2c1 c1(C(N2CCC(N3CCC(O)C3)C2)C(=O)NC)cc(Cl)c(Br)cn1 c1(C(=O)OC)ccc(NC(C2CCCN2C(=O)Cc2cc(Cl)ccc2Cl)=O)c(F)c1 N1(C(c2nccc(CC)c2)=O)CCC2(CC1)CC2C(=O)NCCCF N1(C(C(C(C)C)N(C)C)=O)CCC(F)(CNC(=O)CN2CCNC(=O)C2)CC1 C(=O)(CCCC(=O)N(CCCOCCNC(=O)CCc1cc(C)n(C)n1)C)NC c1(C(=O)NC(C2(C(=O)N(C3CCC3)CCO)CC2)C)noc2ncccc12 CC1C(NC(=O)C=CC2CCCCC2)CCN1c1nnc(C2CC2)o1 c1(C(=O)NCC2OCC(CNC(c3scc(C)c3C)=O)C2)ccc(N=[N+]=[N-])cc1 c1(NC2CCC(NC(c3cnc(CC)nc3)=O)C2)ncc(F)c(OC)n1 C1(C)(CC(=O)NCCOCCOCCNC(=O)CCSC(F)(F)F)CC1F N1(C(C(CCC)OC)=O)CCCC(CO)(NC(c2cc(C)[nH]c2C)=O)C1 N1(C(CCCCOCC)=O)CCCC(CC(=O)NCC2CC(=O)N(C)C2)CC1 C(=O)(C(CC(F)F)c1ccccc1)NCC1N(C(CSCC#C)=O)CC=CC1 C1(C(C(N2CC(C(C)NC(c3ccno3)=O)C2)=O)F)CCCCC1 c1(NCC)ccc(C)c(NC(CCO)C2CCC2)c1 C1(NC(C2CCCC(F)C2)=O)CCCCC1N=c1[nH]cnc2cnccc12 c1(CC2CCN(C(c3nc(CC)oc3)=O)CC2)nc2ccc(C)cc2[nH]1 N1(C(P(C)(C)=O)CC(F)(F)F)CCC2(CC1)COC(CNC(=O)C1CC1)C2 N1(C(c2ccc(C)s2)=O)CCCC2(C1)CN(C(C1CC=CCC1C)=O)CCO2 S(=O)(=O)(c1ccc(Br)cc1NCCn1cnccc1=O)NC1CCCC(OC)C1 c1(CC)cccc(C)c1NC(=O)C(N1CCOC(C)CC1)c1cccs1 C(=O)(CCS(=O)(=O)N(C)C)N(CCNC(c1ncc(NC)cn1)=O)CC c1(C(=O)NC(C(C)NC(C2CC(CC)C2)=O)C)cc(OC(F)F)ccn1 N1(C(c2cc([N+](=O)[O-])cs2)=O)CCOC2(CCC(F)(F)CC2)C1 c1(C(N(CC(CO)C(C)C)Cc2cc(C)ncc2)=O)c(Cl)nc(Cl)n1C CC1CN(C(=O)CC2(n3ccnc3)CC2)CCCN1C(C1CC(O)CN1C)=O CC1(C)C(NC(=O)C(F)n2cccn2)CCN1C(c1ccccc1)=O c1(CCCNCC(=O)NC(c2cn(C)nc2)CN)ccc(Cl)c(Cl)c1 c1(C(N(C2(C(=O)NCC3CCCSC3)CSC2)C)=O)cccnc1 CC(C)CCC(O)C(=O)N1CC(N(C)C(c2cnc3[nH]nnc3c2)=O)C1 N1(C(C2CCN(C(=O)OCC=C)C2)=O)CCN(C(=O)CC=C(Cl)Cl)C(CCOC)C1 n1(CCC(=O)NC(C)CCCNC(c2csc(C#N)c2)=O)ccc2ccccc12 C1(NC(c2c(CC)c[nH]c2)=O)CCC(C)(CNC(c2cccc(N)c2)=O)C1 C1(CN(C)C(C2CCC2c2ccc(F)cc2)=O)CCCC1(C)C C1(C(NNC(=O)C=CC(=O)Nc2cccs2)=O)CCCC2(CCC2)O1 C1(NC(CCC)=O)CC(CNC(=O)CCCNC(C)=O)C12CCC2 C12(NC(C3CCCN(C(C4CC5(CCC5)C4)=O)C3)=O)CCN(CC1)CC2 C1(NC(c2ncn(C)c2)=O)CCCC(CN(C(=O)Cn2cnc(=N)[nH]2)C)C1 C(CNC(C1(OC)CC(C)C1)=O)(C(C)(C)C)NC(CSCCOC)=O C1(NC(CC#N)=O)CN(C(C2CC=CC2)=O)C2(CCOC2)C1 CC(C)C(O)CC(=O)NCC1CC2(CC(NC(=O)COCC(F)F)C2)C1 n1(C(C(=O)NCCCN(c2ccc(C(=O)OC)cn2)C)C)nc([N+](=O)[O-])cc1C C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC1C(CNC(c2cncc(COC)c2)=O)CC1 c1(C(=O)OCC)nnc2ccccc2c1NC(CNC(=O)CO)CC CC(C)CC(O)CC(=O)NC(C)C(=O)NCc1ccc(Cl)cc1 CC(C)(C)C#CC(=O)NC1CCN(CCNC(=O)C(F)Cc2ccccc2)CC1 CC1CCc2c(sc(CNC(=O)CCc3ccc(N)cc3)c2-c2nn[nH]n2)C1 c1(C(C(=O)NCCN(C(c2ccc(=N)[nH]n2)=O)CC)=O)ccc(F)cc1 N1(C(c2c(C)ncs2)=O)CCC(NC(=O)C(=O)NC(C)C)CC(O)C1 c1(C(N(CC(CC)NC(c2cccnc2)=O)C)=O)ncc(Br)cc1N C1(C(N(C2CCN(C(C3(C(F)F)CCCO3)=O)C2)CC)=O)CCN(C)C(=O)C1 O=C1CC(C(N2CC3CC3(NC(=O)COC3CC3)C2)=O)C(c2ccccc2)CN1 C(=O)(Nn1nnc(C)c1C)C1CCN(C(c2c(NC)nccc2)=O)CC1O C(=O)(C1Cc2ccc(F)cc21)N1CCN(c2c(C(=O)OC)sc(C)n2)CC1 c1(C(=O)NCC(C2CC2)NC(CC2(OC)CCC2)=O)ccc(F)nc1F c1(C(C(=O)NCCCC)N(C2CC2C)C)cc(OC)ncc1Br N1(C(C(C)Cc2ccccc2)=O)CC2CCC1CN2C(c1cc(O)nnc1O)=O C1(NC(C(c2ccoc2)NC(c2n[nH]cc2C2CC2)=O)=O)CCCC2OCCC12 N1(C(c2cncc(OCC)c2)=O)CC2(CCCC2NC(=O)Cc2nocc2C)C1 Cc1onc(Br)c1C(N1CCCCC1CNC(=O)CSc1cn[nH]c1)=O N1(c2occ(CC(C)O)n2)C(=O)NC(CCC(=O)NCSc2ccccc2)C1=O C#Cc1ccc(C(N2CC(O)CC2CNC(C2CC2F)=O)=O)o1 Cc1cc(C(N2CC3C(Nc4ncncc4I)C3C2)=O)ccc1Br C1(NC(=O)C(=O)Nc2ccc(F)cc2)CC12CCC(C(=O)O)CC2 C#CCCCCC(=O)NC(COCC)C(N1CC2C=CC1CC2)=O Cc1ccc(=N)[nH]c1C(=O)NCC(C(C)(C)C)NC(C1CCCNC1=O)=O c1(OCC)ccc(NC(=NCCC2(C)CC2(F)Cl)NC2CCC2)cc1Br C(CCC(C)C)(C(=O)NC(c1ncc[nH]1)CC)NC(c1cnc(CC)s1)=O c1(OC)cccc(Cc2cn(C3CC4(C(=O)NCCn5cncn5)CC34)nn2)c1 Cc1ccc(C(=O)N(CC(=O)NCc2n[nH]cc2C)C2CCC2)s1 c1(CNC(=O)C(N2CCC(Br)CC2)=O)cccc2c1OCO2 c1(N(C(=O)NC2(C(C)O)CC2)C)cnc(N(C)C)cc1C C(=O)(C(C)CC(N)=O)NCC1(COC)CCCN1C(C1CCC(=O)O1)=O C(N=c1[nH]n(C)cc1[N+](=O)[O-])C1CCN(C(C(c2ccnn2C)C)=O)CC1C N1(C(C(C)=O)=O)CCC2(CC1)C(NC(=O)CC1COc3ccccc31)CS2(=O)=O C1(C(=O)NC(c2n(CC)ncc2)C)CCN(C(C2CC(F)C(=O)N2)=O)C12CC2 C1(CCC)CCC(C(N2CC(NC(C3OCCC3C(=O)OC)=O)C(F)C2)=O)CC1 N1(C(C(C)(C)CCNC(c2ccn(C3CC3)n2)=O)=O)CCC(=C(F)F)CC1 N1(C(C(COC)NC(=O)C(C)N2CCCC2)=O)CCC(CC(=O)N(C)C)CC1 C12(NC(C(=O)NC3(CO)CC(OC)C3)=O)CCCNCC1C2 c1(C(N2CCCC(C(=O)NCc3cccc(OC)n3)C2)=O)cc2occc2s1 C#Cc1ccc(CC(=O)NC2CCC(C)N(C(C3CCOCC3)=O)C2)cc1 Cc1c(C(N2CC(NC(C3CC(=O)N(C(C)C4CC4)C3)=O)C2)=O)nnn1C(C)C N1(C(C=CC=CC)=O)CC2(CC(NC(c3nocc3C)=O)CO2)C1 c1(C(=O)NC2CCN(C(c3cc(CCC)on3)=O)C2)oc2cc(Cl)ccc2c1C c1(C(=O)NC2C(CO)CCN(C(C(C)CO)=O)C2)cnc2c(c1)COC2 C(=O)(CCC(C)(C)C(=O)OC(=O)CC1CNC(=O)C1)N(CC(C)C(C)(C)C)C Cc1cnc(C(=O)NCC(C)CC(=O)NC(c2nccc(C)n2)C)c(F)c1 c1(C(=O)NC(CC)CNC(C2CCCO2)=O)ccc(Br)nc1O C(=O)(CC(O)C(C)C)NC(C(=O)N(CCC#C)CCO)COC C(=O)(C1=CCCN(C(=O)CCC2CCCOC2)C1)N(CC)CC1(O)CCC1 C1(OC)CC(NC(C2CC(SC)CN2C(=O)NC)=O)CC1O.c1ccccc1 C1(NC(C2CC2F)=O)CCSC12CN(C(c1ccc(C(O)CF)cc1)=O)C2 C1(C(=O)NCC2COCCO2)C2CCCC2CN1C(=O)Cc1ccsc1 c1(SC)ncc(C(=O)NC(C)CCCNC(c2cncc(Cl)n2)=O)c(O)n1 N1(C(C(CC#C)O)=O)CC2CC(C)N(C(c3c(C)cc(C)nc3C)=O)C2C1 c1(CC)ccccc1C(CNC(=O)C(C1CC1)SCC)NC(C1CCOCC1)=O c1(OCC)cncc(C(=O)NC(CC2CCOCC2)C(=O)N(n2ccnc2)C)c1 C1(NCC(CN(C(CC(CC)OC)=O)C)(O)CO)CCC2CC2CC1 CC1(C)CC(C(N2CCOC3C(O)CC23)=O)CN(C(C2C=CC=CC=C2)=O)C1 C(=O)(CCCCC(C)(C)C)NC1C(NC(C(C)NS(C)(=O)=O)=O)CCCC1 C=CCC(CC=C)C(=O)NC1CCC(CNC(C2CC(C(C)C)=NO2)=O)CC1 C(=O)(N1CC(O)C(O)CO1)C12C(CN(C(c3c4scc(C)c4ncn3)=O)C1)C2 C1(c2c(C)nn(C)c2C)CCCN(N2CCCC3(CCCO3)C2)C1 c1(N2CCC(NC(=O)COCCN(C)C)C(F)C2)c[n+]([O-])ccc1[N+](=O)[O-] C(=O)(C#CC1CCCO1)NCCC(C)N(C)C(c1ccc(S(C)(=O)=O)o1)=O C1(c2cn(CC3N(C(c4c(C(C)C)nco4)=O)CCC3)nn2)CCC=CCC1 c1(C(=O)NCC2(O)CCN(C(C(CC)F)=O)C2)cc(Br)c([N+](=O)[O-])s1 C1(C(=O)NC(C)CCCNC(=O)CCc2nc[nH]n2)CC1C1CCC1 C(=O)(C1=NN2CCCN=C2N1)NCC(C(C)C)NC(C1(C)CCC(F)(F)CC1)=O C=CC(CCC)CC(=O)NCCC1(O)CCN(C(=O)CCc2ccc(C)s2)C1 C1(N(C(=O)NCCN(CCC)CCC)CC2CC2)CCC(C)(C)CC1 c1(C(=O)NCCC2(O)CN(C(C(CCC)=CCC)=O)C2)cn2nc(C)sc2n1 N1(C(C(=O)Nc2cc(C(N)=O)c(F)c(Cl)c2)=O)CC2CNCCCC2(CO)C1 c1(C(N(C(c2cn(-c3ccccc3)nn2)C)C)=O)sc(F)cc1Br c1(CC(=O)NCC(=O)NC2CCCC(C(N)=O)C2)cc(Br)ccc1[N+](=O)[O-] CC1c2cccc(Br)c2CCN1C(=O)Cn1cnc(C(F)(F)F)n1 Cc1ccc(CC(=O)NC(C2(O)CN(C(c3c[nH]c(C(N)=O)c3)=O)C2)C)c(Cl)c1 C1(NC(C(CCC)C)=O)Cc2ccccc2C1N=c1[nH]cnc2c(C)csc12 c1(C(=O)NCC2C(OCC)CN(C(C(C=C)O)=O)C2)cccn2cnnc12 N1(C(C=CCOCCOC)=O)CCC(NC(C2CCCCCC2)=O)C1(C)C CCCCC(O)C(=O)NCC(CNC(=O)C=Cc1cnn(C)c1)CO C(=O)(C1CCCn2cnnc21)NC1CC(NC(c2c(OC)ccc(C)c2)=O)C1 C1(C(=O)O)CCS(=O)(=O)C12CN(C(=O)C(c1ccccc1F)O)C2 C(=O)(C#CC1(C)CCCO1)NCCCCC1CN(C(c2c(C(C)C)ocn2)=O)C1 Cc1cc(C(F)F)n(CC(=O)NCCN(C)C(c2ccc(C3CC3C)o2)=O)n1 n1(CC)cc(C(=O)N(C)CC2CC(F)CN2C(=O)C(F)n2cccn2)c(C)n1 c1(C(=O)NC2CN(C(C=Cc3n(C)ccc3)=O)CC2O)ccc2sccc2c1 C1(C(=O)NCC23C(CN(C(CCC4(C#N)CCC4)=O)C2)C3)Cc2cccnc2C1 CC(=O)CCCCC(=O)NC(CO)C(=O)NC(C)CN1CCOCC1 S(=O)(=O)(c1ccc(NC(C)CCCCC)c(Cl)c1)NCC1CCC(=C)CC1 N1(C(c2noc(CC)c2C)=O)CCC(C2CCN(c3cc(OC)ncn3)C2)CC1 c1(C(=O)NCC2C(CNC(COCc3cc(C)no3)=O)C2)cccc2c1CCC2 C(C(C)(CC(C)C)NC(=O)C=Cc1nc(C)co1)NC(CCC#CC)=O N1(C(C2CC(O)(CC#C)C2)=O)CCN(C(=O)CCOC)C(CCC)C1 Cc1cc(O)c(NC(c2ccc(F)c(-c3nn[nH]n3)c2C)=O)cc1Br c1(C(N(CC(CC)NC(=O)CN(S(=O)(=O)CC)C)C)=O)nocc1C N1(C(CC(C)SC)=O)CCOC(c2cn(CC3CC(F)(F)C3)nn2)C1 c1(C(N2CCC(NC(C3C(CC)N(C)CC3)=O)C2)=O)ccc(Cl)c(F)c1 C(CO)(C(=O)N1CCCC1C(C)(C)CNC(c1csc(Cl)c1)=O)N(C)C N1(C(Cc2ccc(OC)cc2)=O)CCOCC(NC(C2(SC)CCCCC2)=O)C1 CCCCCC(C)CC(=O)NC1CN(C(=O)CNc2ccccn2)CC2(CC2)C1 c1(C(=O)OC)cccc(CC(=O)NC(C)C(C)NC(=O)CCN2CCOC2=O)c1 C(=O)(C(O)P(C)(C)=O)N1CC(OC)C(NC(=O)CCCc2ccc(Cl)cc2)C1 CCCC(CC)C(=O)NC1COCC1CNC(=O)C(C)(C)n1cccn1 C(CCC)(C(O)C(=O)NCC1(CC(=O)OC)CC1)NC(CCCC)=O C1(COC)(NC(=O)CNC=O)CCN(C(=O)C(c2ccc(F)cc2)CO)C1 S(=O)(=O)(c1cc2c(cc1Cl)NC(=O)CO2)Nc1cnc(C)c(N)c1 C12CC3(C1)CN(C3)c1cc(ncn1)C(=O)C(CCC)NC2=O.OCC c1(-c2cc(C(=O)NCC(C(=O)OCC)O)n(C)n2)cc(OC)cc(Br)c1 c1(C(C)C)ncccc1NC(C1CCN(C(=O)C(F)(F)C2CC2)C1)=O c1(OC)ccnc(CNC(=O)C(=O)NC2(C3CCCC3)CC2)c1OC(F)F S(=O)(=O)(c1cnc(O)c(Br)c1)NCC(c1ccc(F)cc1F)(C)C c1(C2C(C(=O)Nc3cnn(-c4ccccc4F)c3)C2)ccc(OC(F)F)cc1 c1(C(N2C3CN(S(CCCC)(=O)=O)CC2CC3)=O)cnn2cc(C)cnc12 C=C(C)C(C)(C)C(=O)NCCN(C)C(c1cc(-c2ccns2)on1)=O C(=O)(CC1=CCN(C(=O)C2=CCCC2C)CC1)N(C1CCCC1)CCCC CC1(NC(=O)CC23CCCC2C3)CN(C(c2cc(CC(=O)NC3CC3)on2)=O)C1 c1(N2CCC(NC(=O)NCc3ccnnc3O)C2)cc(F)cc(F)c1 c1(OC)ccnc(C(C)(C)OCC2(c3ccnnc3)CC2)c1 N1(C(CN(C(C2CN(CC)C(=O)C2)=O)CC2CC2)=O)CC(C)C(C)C1C c1(SCC)ccc(N2CCC(O)CC2)cc1.C12CC(C1n1cccn1)N2 c1(OC)ncc(Br)cc1C(N1CCC(CN(C(=O)COCCF)C)CC1)=O C1(C(=O)NC2CN(C3CCC3)C2)(CNC(=O)Cc2cncs2)CCC1 Cc1nc(NC(=O)C(C2CCC(=O)N2)C)n[nH]1.C12CCN(C1)CC(=O)N2C c1(C(CC)C)ccc(C(=O)N(C)CC2CCCCN2C(C23CCC2CC3)=O)cc1 C1(C(=O)NCCC(C)N(C(c2cc(CC)c(C)s2)=O)C)OC2CCCCC2C1C c1(CN2CC(C(=O)OC)OC(C)(C)C2)cccc2oc(O)nc12 N1(CC)CCN(C(c2coc(CNC(=O)Cc3ccc[nH]3)c2)=O)CC1C CC1CN(C(=O)C(O)CNC(=O)C2=NN(C)C(=O)CC2)Cc2c[nH]nc21 c1(C(N2CCCC(NC(C(=O)NC(C)C)=O)C2C)=O)cccc2c1ncn2C C12(NC(c3ccc(C)o3)=O)CC(C1)N(C(C1CCC1c1nc(S)n[nH]1)=O)C2 c1(NC)ccc(C(=O)NCCC2CCCN(C(C3(C)COC(=O)C3)=O)C2)nc1 c1(CNC(=O)NC23CC2CN(CC2CC2)C3)nc2ccccc2s1 c1(C(=O)NCC(CC)NC(=O)CCSC)ccnc(N(C)C)c1Br Cn1ncc([N+](=O)[O-])c1C(=O)NCCC1(NC(c2ccc(C#N)cc2)=O)CCC1 C=CC1(CC(=O)NC(c2cccc(C)n2)C)CN(C(=O)C(N2CCCC2)SC)C1 N1(C(C(CC(C)C)=O)=O)CC2CC1CCC2NC(=O)CCC1CCC(=O)N1 C(=O)(C#CC1(C)CC1)N1C(C(C)C)C(NC(c2cnn(CC(F)(F)F)c2)=O)CC1 c1(NC)cc(C(=O)NCC2COC(CNC(C)=O)C2)c2ccccc2n1 c1cc(NCc2ccc(C3CCCN3)nc2)ccc1-n1cncn1 c1(C(=O)NC(CNC(C2(OC)CCCC(C)(C)C2)=O)C)cnn2c1NCC(C)C2 Cn1nccc1C1=CCN(C(=O)C(N2CCCCOC(C)(C)C2)=O)CC1 CC1=C(C(=O)NCCCC(C)NC(=O)Cc2csc(C(C)C)n2)CC1 C1(NC(C=CC(C)C)=O)CN(C(=O)CN2CCC2C)C2(CCC2)C1 N1(C(C2C(C)=C2)=O)CCC2CCN(C(=O)C=Cc3nc(C)c(C)[nH]3)CC2C1 c1(C(=O)NCC(C)(C2CC2)NC(c2ccc(F)c(CO)c2)=O)cccc(F)c1O C1(CC(N)=O)(CNC(C(=O)NC(C)C)=O)CCN(C(=O)C(C)CF)CC1 N1(C(COCCC#C)=O)C2CCC(C(=O)Nc3cncc(C)c3)C1CC2 C12(CCNC(C(C(C)C)OC)=O)CCC(C1)N(C(=O)C(N)=O)C2 N1(C(C(C)=C(CC)C)=O)CCCC(F)(CNC(C23CCCC2CCC3)=O)CC1 C1(NC(CCCCSC)=O)CN(C(c2csc(C(C)=O)n2)=O)Cc2nccn2C1 C(=O)(C#CC1CCOCC1)N(C1C(N(C)C(C2CCCCC2O)=O)CCCC1)C c1(C(=O)NCC2C(NC(c3c(=O)ccn(C)c3)=O)CCC2)cc(F)c(Cl)cc1F CCC(CC)C(F)C(=O)NC(C1CCCN1C(=O)COCc1ncc(C)o1)(C)C C1(C(=O)NCC2OCC(NC(C(C(=O)NC)(C)C)=O)C2)C2CCC3C(C2)CC13 c1(C(N2CC3C(NC(CCOCCOC)=O)(C3)C2)=O)cnc2c(ccn2C)c1 c1(NC(c2ccc(SC)c(F)c2)CC)cc(N2CCC(CC)C2)nc(C)n1 N1(C(CSC)=O)CC2CCCC(C1)N(C(c1ccc(CC(C)C)s1)=O)C2 CCC(CC(=O)Nc1cnn(C(C)(C)C)c1)N(C)C(C1CC(C(=O)OC)C1)=O C#Cc1cc(C(=O)NC2CCN(C(=O)CC(C)C)CC2CC)cc(C(F)(F)F)c1 C12CCN(CC1)C2=O.C1(CC(=O)N(CC)Cc2cnn(C)c2)CCC(=O)N1C C(=O)(CCCC(=O)Nc1nc(C)cs1)N(CC(C)NC(C=CCOC)=O)C c1(C(=O)NC2C(NC(=O)C3=CCCS3)CS(=O)(=O)C2)cncc2c1CCC2 C1(COC)(NC(=O)CCCSc2ccccc2)CCN(C(=O)COC(C)=O)CC1 C1(NC(C)=O)CCC(C(=O)NCC(F)CNC(c2ccc(Cl)cc2)=O)CC1 CC1(C)CCOC(CC(=O)NCC(C)(CO)NC(C2C3CCC(F)(F)C23)=O)C1 C1(CNC(C2(CC#C)CCCC2)=O)CN(C(C2(F)CCCOC2)=O)CC1O C1(NC(c2ccc([N+](=O)[O-])o2)=O)CCCCN(C(C2(n3cccn3)CC2)=O)CC1 CC1CN(C(c2ccn(C)c2)=O)CC1NC(=O)CSc1nnnn1C c1(C(N2CC(N(C(C3(COCC)CC3(F)F)=O)C)C2)=O)c(O)cccc1Cl C12(CNC(COCCN(C)C)=O)CCC(CC1)N2C(c1ccc(=O)n(C)c1)=O CC1CCOC1C(N1CC(OCCNC(c2ccc(Br)o2)=O)C1)=O C(CN=C(NCC1CCCO1)NCC12CCC(CC1)OC2)c1c(C)ncs1 C(=O)(C1=C(SC)CCCC1)N(CCN(C(C(C)OCC=C)=O)C)C C1(NC(c2ccc3cnsc3c2)=O)CCN(c2cnc(C#N)cn2)CC12CCC2 C(=O)(C(C(C)(C)C)C1CCC1)NC1C(C)N(C(c2cc3sccc3[nH]2)=O)CC1 c1(ONC(C2N(C(C(C)SC)=O)CC2)=O)cccc(F)c1 N1(C(CC(CNC(C(CC#C)C2CC2)=O)C)=O)CC(N(C)C)C(C)(C)C1 C1(NC(c2n(CC)nnc2)=O)CC2CCC(C1)N2C(c1ccc(NC(C)=O)o1)=O c1(NC(c2cc(OC)no2)=O)ccc2c(c1)CN(C(c1ccc(Cl)nc1O)=O)C2 Cc1nc(NC(C2CCCCN2C(=O)CCCC(N)=O)C)ncc1Br C1(C#N)(C(C)C)CCN(C(=O)C(=O)N(c2cccnc2)CC2CC2)CC1 c1(C(=O)NC2CCC(CCNC(C(C)S(N)(=O)=O)=O)C2)ncc2cc(Cl)ccn12 N1(C(CCC2CCCN(C(c3c(C#C)cn(C)n3)=O)C2)=O)CC(=O)N(C)C(=O)C1 CC1=C(C(=O)NC(C)C=CC(=O)NC23CC2COC3(C)C)CCO1 N#Cc1nccnc1NC1CCC1NC(c1cnc(-c2ccsc2)s1)=O Cc1nn(Cc2ccccc2Cl)c(Cl)c1NC(c1cnnn1CC1CCOC1)=O C(C(N=[N+]=[N-])C(=O)N1CC(CNC(c2c(C(F)(F)F)n[nH]c2C)=O)C1)OCC N1(CCC(=O)NC2(C(=O)NCCNC(CC)=O)CCC2)CCOCC1 C1(C(=O)NC(C2(O)CN(C(C3CCCO3)=O)C2)C)CCCC1(C)C Cc1cnc(C(=O)N(CCCN(C)C(C2(C#N)CCC2)=O)C)c(C)c1 CC(C(=O)N1CCCC(NC(c2cnc(C(F)F)s2)=O)CC1)C(C)(C)C C(=O)(CCCCCCN=[N+]=[N-])N(C1CCN(C(CN(C(C(C)C)=O)C)=O)C1)C c1(C(=O)NCC2N(C(CC=C(C)C)=O)CCC2)ccc(NS(C)(=O)=O)c(Cl)c1 CC1CN(C(=O)C=CCF)CCC1NC(=O)CNC(N1CCCC(O)C1)=O C1(CC)(NC(=O)CC2CCN(C3CC3)C2)CCN(C(c2cnn(C)c2C)=O)CC1 CC1CN(C(=O)C2=CCC2)C(C)CN1C(c1n[nH]c2c1COC2)=O n1(CC)nc(C(N2CCC2C(=O)NCCc2ccccc2OC)=O)cc1C CC(F)CCN=C(NCCSC)NCC1CCCCC1SC(C)C C1(CC(=O)NC(CN(C(=O)CCNC(C2CCC2)=O)C)(C)C)CCC(O)C1 c1(C(=O)NCC(C)(O)CNC(=O)Cn2cc(Cl)cn2)cnc2ccc(F)cn12 C12(CNC(c3cnn(C)c3C3CC3)=O)CCC(C1)N(C(C1CC1C1CC1)=O)C2 C1(CC(=O)NC2CCC2NC(C2(c3ccc(Cl)nc3)CC2)=O)COCC2(CCC2)O1 CC(C(=O)N1CC(C(=O)NC(c2cccs2)C)C1)N(C)C(=O)OC(C)(C)C c1(C(=O)NCC2(C)CCN(C(CC(C)c3ccco3)=O)C2)ccn2cncc2c1 N1(C(c2c(CC)nco2)=O)CCCC1(C)CNC(c1cc(C(F)(F)F)ncn1)=O CCC(C(=O)NC)NC(=O)C(F)C1CC(NC(C2CCCSC2)=O)C1 c1(NC(=O)NCCN(C(=O)C(O)Cc2[nH]cnc2C)CC)c(F)cccc1Cl C1(C(=O)N(C)CCNC(N)=O)(NC(C(c2ccn(C)c2)C)=O)CCCC1 c1(N2CCC(NCc3cc(OC)nc(C)c3)C(C)C2)ncc(C#N)cc1C N1(C(CC(c2ccc(C)cc2)C)=O)CCC(NC(=O)CCC2CCCC2)CC1C c1(C(N2CC(COC)(NC(C34CCCC3CC4)=O)C2)=O)ccc2ncncc2c1 Cc1ccc(S(C)(=O)=O)cc1N(c1nnnn1-c1c(C)cccc1C)C(N)=O CCC(CC(=O)NC1COCC1C(=O)NC1CC(=O)N(C)C1)C(F)F c1(C(C(C)SCC)O)nc(CC2CCCC2)nn1-c1ccc(Cl)nc1 c1(C(C)C)nc(C(c2cccc(F)c2)C2CC2)n(-c2ccccc2Cl)n1 Cc1nc(CC2CC2)oc1C(=O)NCC1(C)CCCN1C(c1cnc(=N)[nH]c1)=O N1(C(CC2N(C(c3c(CC)csc3)=O)CC2)=O)CC2C(C1)C2(F)F c1(CC)ccc(C(=O)NC2C3CC2N(C(c2cccnc2N(C)C)=O)C3)cn1 c1(C(N2CC(OC)C(NC(=O)C(C)(C)F)C2)=O)c(C)oc(C)c1Br c1(C(C)C(=O)NC2COCCC2NC(C2CSCCS2)=O)ccc(Cl)c(F)c1 c1(OC)cccc(CC(N2CCN(C(=O)CC3(C)CCC3)C(C3CC3)C2)=O)c1N c1(C(=O)NCCOCCNC(c2n(CC#C)cnn2)=O)cc2cc(Cl)cnc2[nH]1 C(C1COC1=O)OC.C=C1CCN(C(=O)CCC)C1 C(=O)(CC1CCNc2ccccc21)N1C2N(C(=O)C=CC(F)(F)F)C(CC2)C1 c1(C(=O)NC2CCN(C(C3C(C)C3)=O)CC(O)C2)cccc(Cl)c1[N+](=O)[O-] C(=O)(CCCC(=O)N(C)CC1CCCN(C(=O)Cc2cnns2)C1)NC(C)C N1(C(c2c(CC)c[nH]c2)=O)CCN(C(=O)CC(C)C2CC2)CCC1C C1(NC(c2ccc(CC)o2)=O)CCN(Cc2sc(SC(F)(F)F)nc2C)CC1F c1(CC(=O)N(C2CC2)Cc2cc(C)oc2C)c[nH]c2cccc(F)c12 c1(N(C(C(F)=CCC)=O)CC(N2CC(CO)(CO)C2)=O)ccccc1COC c1(OCCCCCC)cccc(CNC(=O)CN2CC=C(C)CC2)c1 C(=O)(C(C)C(=O)OC)NC(c1cn(C)cn1)CNC(C(C)SC)=O c1(C(N(C2C(C)CCN(C(C(CCC)C)=O)C2)C)=O)ccc(Cl)c(OC)c1F C1(C(N2C(CCOC)CCC2)=O)CCN(C(C2SCC=C2C)=O)C1C C1(C#N)(C(N2CC(CC(C)NC(=O)C(C)N(C)C)C2)=O)CC2CCC1CC2 c1(C(N(C)CC2CCN(C(C(C)NC(=O)NC)=O)C2)=O)cc(C)ncn1 c1(OC)cc(C)cnc1C(N1CCC(Cc2cn(-c3ccc(F)c(F)c3)nn2)C1)=O CCCCCCCc1cn(C2CCCN(C(C3(C)CC3(F)F)=O)C2)nn1 N1(C(CSCC#C)=O)C2CCC1(CNC(=O)C(COC)OC)CC2 C1(NC(CCOC)=O)CN(C(C2CCCN(CC(F)(F)F)C2)=O)CCC1F C(=O)(CCCC(F)(F)F)N1C(CC(N2CC(c3nn[nH]n3)C2)=O)COCC1 N1(C(C=CSC)=O)CCN(C(C2CC2CN(C)C(C2CC2)=O)=O)CC(C)C1 N1(C(Cc2c(C)nsc2)=O)CC2CCC(C(=O)O)(C1)C2(F)F c1(C(=O)NC(C2(O)CCN(c3cc(CC)ncn3)CC2)C)ccc2[nH]ccc2c1 CCCC(C(=O)NCCC(C)(CC)NC(C1CCC(NC)C1)=O)OCC C1(C(N(CC(COC)C)C)=O)CCN(C(=O)CC(C)(C)N(C)C)CCO1 CCS(=O)c1ccccc1C(=O)NC1CN(C(=O)C(N)=O)CCC1c1ccccc1 c1(C(=O)NC2CC(F)(CNC(C3CC(C)C3)=O)C2)ccc(C(F)F)cn1 c1(C(C(=O)NC(C)CNC(c2ccc(CO)o2)=O)SC)ccc(F)cc1 c1(C(N(C(C)CCNC(=O)CC2(C)CCOCC2)C)=O)ccc(O)cc1[N+](=O)[O-] C1(C(=O)NC(COC)C)(CF)CCN(C(C2CCN(C(C)C)C2)=O)C1 C1(NC(=O)Cc2nc[nH]n2)CCCCN(C(c2cc(NC3CCC3)ccn2)=O)C1 C1(NC(C2N(C(CNC(c3ccccc3)=O)=O)CC2)=O)CC1C1CC1 CCS(=O)(=O)CC(=O)N1CC(c2ccccc2)(NC(=O)Cc2nccn2C)C1 Cn1cc(C(N2CCC(N(C(=O)CC(F)F)CCO)CC2)=O)c(C2CCCO2)n1 C(=O)(NNC(=O)CCOC(c1ncco1)=O)N(C1CCOC1)C C1(NC(C2CN(C(C3C(C)CCO3)=O)CC(C)O2)=O)CCC2CCCC1O2 C=CCN=C(NCC1C=CC2CC1CO2)N1CCC(OCCCCC)C1 N(C(=NCc1ccccc1)NCC(C(F)(F)F)n1cccn1)C(C#C)COC N1(C(C(c2ccccc2)NC(C2C(CC)CCC2)=O)=O)CC(C2CC2(F)F)C1 C1(CN(C(=O)CC2CC2)C)CN(C(=O)CC2(C)CC(F)(F)C2)CCO1 C1(C(=O)NC(CC)CNC(=O)CC2COC(=O)C2)CCC(=O)NC1 c1(C(C)OCCOCCO)cc2c(n1C)CCOC2.CC1CN2CCCC1CO2 N1(C(C(C)=CC)=O)CC(NC(=O)Cc2cnn(C(F)F)c2)C(C)C1 c1(C(=O)NC(CC(C)NC(=O)Cc2cc[nH]n2)C)ccc(OCC(N)=O)cc1 C(=O)(C(CC(C)C)NC(C1CC(N(C)C(c2cc(Cl)ncc2F)=O)C1)=O)OCC CC1Cc2cc(Br)cnc2N(C(=O)C(=O)NCCOc2cccc(F)c2F)C1 N(CP(C)(=O)OCC)C(C1C(NC(C(C)OCCCC)=O)CC1)=O CC(CC(F)(F)F)C(=O)NC1CN(C(c2cc[nH]c2C2CCC2)=O)CC1F N1(C2N(CCCN(C)C)CCC2)CC(C(=O)Nc2ccc(F)cc2)CC1=O C12(NC(=O)COCC3CCCCO3)CCC1CN(C(=O)CCC1CCOCC1)C2 CC(C)(C)CCCC(=O)N1CC(F)(F)CC1C(=O)NCC1CC2(CCC2)CO1 c1(C(=O)NCCCC(CCC)NC(c2sc(C)nc2C)=O)cc2ccccc2o1 c1(OC)nc(Cl)ccc1C(=O)NCCC1CCCN1C(c1ccc(O)cc1F)=O N1(C(C(CCC)=CCC)=O)CCN(C(c2oc(Br)cc2C)=O)C(C)C1 c1(NC(C2CCC3(CN(Cc4ccn(C)n4)C3)O2)=O)ccc2c(c1)OCCCO2 C(N=c1[nH]c(C(C)(C)C)nc(C)c1C)C1CC(C(C)NC(C2(CO)CC2)=O)(COC)C1 C1(CC(=O)NCCCC=C)C2CCCC2N1C(C1CC2CCCC2C1)=O Cc1cc(=O)c(C(=O)NC2CC(NC(=O)C(C)(C)c3cncnc3)C2)c[nH]1 N1(C(C(C=CC)O)=O)CCC(C)C1CNC(C1(Br)CC1)=O N1(C(CC(C)C2CCCCC2)=O)CCOC(C)(CNC(C2CCCCN2C)=O)C1 C1(C(=O)NC2(CNC(=O)C3=C(Cl)CCOC3)CCC2)CCCC2(CCCCC2)C1 N1(C(C(CC#C)O)=O)CCc2cc(CNC(=O)C(C)OCCCC)ccc2C1 C1(NC(CC2C(C(C)(C)C)C2)=O)CC(O)C1CC(=O)NC1CCC1 c1(C(=O)NC2CC(N(C(c3ncc(CC)cn3)=O)C)C2)cc(Cl)c(N)c(Cl)c1 N(C(=NCCSC)N(C)Cc1ccc2c(c1)CCO2)CC1(OC)CCC1 C1(C(C)NC(COC)=O)CCCN(C(c2ncc(F)cn2)=O)C1 c1(C(N(C2CN(C(C34CCC3C4)=O)C2)C)=O)ccc(N(C)C)nc1 C#CCCCCCCC(=O)N(C(CC(F)F)C(=O)N1CC=CC(OC)C1)C N1(C(C(C=CC)O)=O)CC(CNC(c2nn(C(C)C)nc2Br)=O)C2(CC2)C1 N1(C(CS(CCOC)(=O)=O)=O)CCN(C(=O)CC2CC3CCC2C3)CC(O)C1 c1(C(N(CC(C)O)CCNC(C2CC3C=CC2CC3)=O)=O)cncc2nc[nH]c12 Cc1ccc(Br)cc1C(N1CCC(NC(C2CC(F)C2)=O)C1C(C)C)=O N1(C(CNC(CCNC(=O)OC)=O)=O)CC2(CC2)C1 CCC(C)C(O)CC(=O)N1CCC2C(NC(=O)COC(F)F)CC12 CCC(C)C(C)CNC(=O)CC1CCN(C(C2CCC2C)=O)CC1 C(=O)(C(C)(O)CCc1ccccc1)NCC1C(NC(c2c(C)ocn2)=O)CC1 N1(C(CCCCC=C)=O)CCC(C(=O)Nc2ccc(Cl)c(C)c2)C(C)(C)C1 C1(C)(C(N(C)CCNC(=O)C(C(C)(C)C)N(C)C)=O)Cc2ccccc2NC1=O c1(CNC(C(C2CCCN(C(C(C)C3CCC3)=O)C2)(C)C)=O)cc([N+](=O)[O-])c[nH]1 c1(CNc2c(C(=O)OC)cccc2OC)cnc(F)c(-c2nc(C)no2)c1 CC(C)CS(=O)(=O)CCC(=O)NC1(C)CCN(C(=O)CCCc2cnn[nH]2)C1 CC(C)C(C(=O)NCCC(C)NC(C1C2CCC1(c1cscn1)C2)=O)NC=O CCC(C)(CC)CN=c1[nH]c(=NCc2coc(C(C)OC)n2)c2ncccc2[nH]1 Cc1sc(C)c2sc(C(N3CC(CO)(NC(=O)C4=CC5CC=CCC45)C3)=O)cc12 c1(N2C(C)CCC(C3CCN3)C2)ccc(S(C)(=O)=O)cn1.C1(=O)COCCN1 CC(C(C)(C)C)=CC(=O)NC1CCCC1NC(=O)CN1CC(C)(C)C1 C12CCCN(C1)C2=O.C1(CC)CCN(C(c2nocc2Cl)=O)C1 N1(C(CN(C(=O)OCC)C)=O)CC(NC(C2CC2F)=O)CC1CSC CC1(C)CN2C1C2.c1(C(N2CCCC2)=O)ccc(-c2cc(C(F)(F)F)no2)cc1 C(=O)(C(C)(C)C(C)NC(=O)CCCCCOC)N1C(C(CC)C)CCC1 c1(CC(N2CC(CC=C)(NC(C3CNC(=O)N3)=O)C2)=O)cc(F)cc(Cl)c1 C(=O)(CCC(F)(F)Cn1cc(CCN2CCCCC2=O)nn1)NCC(C)(C)SC c1(C(=O)NCC(CC=C)NC(=O)CC2COC3CC2C3)cccc(N(C)C)n1 CC12CC(C(N3CCCC(NC(=O)CN4CCCC4=O)C3)=O)(C1)OC2C(F)(F)F C(=O)(C(O)CC(C)(C)C)N1CC(C(C)NC(=O)CCSc2ccccc2)OCC1 N1(C(c2[nH]cc(C)c2)=O)CCC2CCN(C(c3cc(CN(C)C)c[nH]3)=O)CC12 CC1(C)CCC(C(=O)NCCc2ccncc2)CN1C(C1CC2(CCC2=O)C1)=O c1(C(=O)NCC(=O)NC(CN(CCCC)C)C)cc(OCC)cc(Cl)c1O c1(CC(=O)NCC(CC=C)NC(c2cnn(C)c2C#N)=O)cccc(C)c1C c1(C(=O)NC2(CCOC)CCN(C(C(CC)OCC)=O)C2)ccc(C)c(Cl)c1N C1(CC)CC(F)(F)CN1C(C(=O)NCCSC)C(C1CCCC1)OC c1(C(N2CC(CN(C(CC(C)F)=O)C)OCC2)=O)cc([N+](=O)[O-])cc([N+](=O)[O-])c1 N1(c2c(C)cc(O)cc2)CCC2CCCC(C1)N2c1c[n+]([O-])ccc1[N+](=O)[O-] O=S(=O)(c1ccc(O)c(F)c1)NCC1CC(CSc2ccccc2)C1 C(=O)(C1=CCOCC1)N1C(CCNC(C(C(C)C)c2ccncc2)=O)CCC1 C(CCC(c1nnnn1CCOC)NC1CC1(C)C)OCC C1(C(=O)OC)CCN(C(c2ncc(C)s2)C(=O)NC(C)(C)C)C2(CCCC2)C1 C(C(=O)N(C)CC1CCCO1)(C1=CCCCCC1)N1CCCC(C(N)=O)(CO)C1 CC1CCN(C(c2ccc(O)nc2)=O)C1CNC(=O)C=Cc1cc(C(N)=O)co1 N1(C(CC=CC=C)=O)CCOCC12COCCN(C(C1CC3CC3C1)=O)C2 c1(CNC(C2C(C(N(C(c3ccccn3)C)C)=O)C2)=O)ccc2ccn(C)c2c1 c1(CN2CC3N(C(c4c(OC)ccc(F)c4)=O)C3C2)cc2cccnn2c1 C1(CC(=O)NCCCN(CCC)C(c2cc(C)cc(O)n2)=O)OCCCC1(C)C Fc1ccc(C=Cc2nc(CC3CCCC3(F)F)no2)cc1Cl N1(C(CSC)=O)CC(CC(=O)NC(CCO)C2CC2)CC1(C)C C1(NC(C2(CC)CCCC2)=O)CCCC1NC(c1ccn(CCOC(C)C)n1)=O c1(N2CCC(CNC(C=Cc3c(C#N)cccc3)=O)C2)ccc(F)cc1[N+](=O)[O-] C(=O)(C(=O)NNC(=O)CC1CCCCC12CC2)NCc1c(OC(CC)C)cccc1 C1(NC(c2cnc(S)nc2)=O)CCN(C(=O)Cn2cncn2)CC1O C1(C(N(CCN(C(c2c(C)cc(CO)o2)=O)C)C(C)C)=O)CCCNS1(=O)=O c1(CC(CN(C)C(C2CCC2C)=O)NC(=O)Cc2ccsn2)cccc(F)c1 CC1CN(C(c2cnsc2)=O)CC(CCNC(=O)COCC2CCC2)O1 N1(C(c2c(NC)cnnc2)=O)CCC2(CCC(NC(=O)C(C)CO)C2)CC1 C1(CC2(C(N(CCN(C(C(C)CF)=O)C)C)=O)CC2)CCN(C2CC2)C1=O N1(C(C=C(CCC)CCC)=O)CCN(C(=O)C=CC=C(Cl)Cl)CC2CCCCC12 C12(CCOC3(CCC3)C1)CN2.CC1COC2(CCC2)CN1C(=O)OC(C)(C)C Cc1cc(O)nnc1C(=O)NC(C1CN(C(c2cccc(CO)c2)=O)CCO1)C c1(SCCC)ccc(C(N2CCC2CNC(c2cc(C3CC3)on2)=O)=O)cc1 C(CO)(C1CCc2ccccc21)C(C(Cc1cc(C)c(N)cc1)N)=O N1(C(CCCC)=O)CC(NC(c2ccc(Cl)nc2OC)=O)C(S(C)(=O)=O)C1 N1(C(CC(=O)NCC)=O)CCC(C2CCN(C(=O)C(C)CC)C2)CC1 c1(C(=O)NC(CC=C)CNC(C2(n3nccn3)CC2)=O)ccc(S(=O)(=O)NC)cc1 c1(C(=O)NCC(CNC(CSCC=C)=O)O)nnc2ccccc2c1Br C1(C(N(CC(=O)N(C)C)C)=O)COC2CN(C(C3CCN(S(C)(=O)=O)CC3)=O)CC12 C1(C(=O)NC2CC(NC(CC(C)n3cccn3)=O)C2)CCCCC1C(=O)N(C)C c1(CC)cc(C(=O)NC(c2ccccc2)CNC(C2(C#N)CCCO2)=O)n(C)n1 C1(NC(C2CCN(C)CC2)=O)CCN(C(=O)Cc2nc(=N)[nH][nH]2)C12CCC2 C(=O)(CCC(C)CCC1CC1)N(C(c1ccccc1)CO)C C1(CNC(CC2CC(=C)C2)=O)CN(C(c2csc(-c3cnc[nH]3)n2)=O)CCC1C Cc1cc(-c2nc(C(c3ccccc3)O)nn2C(C)C(C)C)c(C)cc1I c1(C(N(CCNC(C(COC)COC)=O)C)=O)cc2c([nH]1)CCCC2=O C=CCC(CC(=O)NCCOCCC)NC(C1(C)CCCN1C)=O C1(CC)C(NC(c2coc(C)c2)=O)CCN1C(c1cc(O)n(C)n1)=O Nc1c(Oc2ccc(NC(=O)CC(O)CCc3nn[nH]n3)cc2)cc(F)cc1F CCC(C)C(O)CC(=O)N1CC=C(C(=O)NC(CC)C(=O)OC(C)C)C1 C1(C(=O)NC(C=C)C)(NC(=O)CC2(C)CCOCC2)CC(F)(F)C1 N1(C(C2OCCC(=O)C2)=O)C2CC=C(C(=O)NC34CCC(F)(CC3)C4)C1CC2 n1(CF)c(-c2ccc(NC3CC(CC)(SC)C3)cc2)csc1=Nc1ccc(F)c(F)c1 C1(C(=O)NCCC2(NC(c3nsnc3O)=O)CC2)CC2CC1CC2(F)F CCC(F)(F)C(C)(C)C(=O)N1CCC(C)C(N(C)C(c2cc(Cl)ns2)=O)C1 N1(C(C=CCC)=O)CCN(C(C23CCCC2C3(F)F)=O)C(CC(=O)NC)C1 C12(CCNC(c3c(C)cnnc3)=O)CCC1CN(C(=O)C#CC1CC1)C2 N1(C(CCCOC(C)C)=O)CC(O)(C2(NC(=O)COC3(C)CCOCC3)CC2)C1 N1(C(CCc2n(C)[nH]c(=N)c2)=O)CC2CC(C1)N2C(=O)COc1ccc(F)cc1F C1(C(N2CC(OC3CCN(C(CCCC#C)=O)CC3)C2)=O)CC2CC1CC2(F)F c1(SC)nc(=NC2CC(NC(=O)CO)C23CCC3)nc(-c2ccco2)[nH]1 N1(C(C(CCSC)O)=O)CCCC2(NC(c3cn4ccnc4s3)=O)CC2C1 c1(C(=O)NCC2C(NC(=O)C=C3CCOCC3)CCC2)cc(F)cnn1 C1(C(C)C)N(Cc2cn(CCCC3(C(F)(F)F)CCC3)nn2)CC12CC=CC2 Cc1ccc2ncc(C(=O)NCC3CCCC3NC(=O)C(C)(C)CF)c(=O)n2c1 N1(C(CC2(C)CC2(Cl)Cl)=O)CC2(COC(CNC(C3CCCO3)=O)C2)C1 c1(C(=O)NC(C(C)(C)C)CNC(c2cnc(Cl)c(I)c2)=O)cc2cccnc2[nH]1 C1(CNC(c2cncc(C)c2)=O)C(C2CC2)CCN1C(=O)C1=CCC1 C(=O)(CCCCC(=O)OC)NC(C(CC)C)CC(=O)OCc1cn[nH]c1 Cc1nc2c(C(N3CC4CC4(NC(C45CCCN(CC4)C5)=O)C3)=O)cccc2o1 C1(CC(=O)NCCC2CC(NC(C3C(C(=O)OC)CC3)=O)C2)CCN(C)C1=O C1(NC(=O)C2=CCOC2)CN(C(=O)CC=Cc2cccc(F)c2)C2(CCC2)C1 S(=O)(=O)(c1cnn(CCN(F)F)c1)N1C(CC(=O)O)CCCC1 C1(OC)CC(CNC(=O)CC2C=NN(C)C2=O)N(C(c2n[nH]c(C3CC3)n2)=O)C1 C1(NC(CCOCc2ccc(C)cc2)=O)CCCN(C(=O)CCN2CCC2)C1C N1(C(CC(C)(C)O)=O)CCCCC(NC(=O)C(F)(F)C2CC2)C1 C(=O)(C(CNC1CCNC(=O)C1)(CC)CC)NCC(C1CCCCC1)C N1(C(C2C(CC)C2)=O)CCN(C(c2cnn(-c3ccc(F)cc3F)c2)=O)CC1C C12(CNC(c3c(CC)csc3)=O)CCCC1CN(C(c1cc(O)nc(Cl)c1)=O)C2 C(C(=O)N1CC(O)CCO1)C1C(C)(C)C(C(=O)Nc2nc3ccccc3[nH]2)C1 C#Cc1ccc(Cl)c(C(=O)NCC2CN(C(=O)C=Cc3cc[nH]c3)CC2O)c1 C12CC(C13CCC3)NC(=NC)N2.c1(CCC(C)C)cnn(CC(F)F)c1.N c1(C(=O)NCC2CN(C(c3c(C)nc(C4CC4)s3)=O)C(C)C2)cnc2sccc2c1 C=C(C)CC(C)C(=O)NC1CC(NC(c2cnc(C(F)(F)F)nc2)=O)C1 c1(C(CC)=O)ccc(C(c2ccc(Cl)s2)NCC2CCCNC2)cc1 Cc1ccc(C=CC(=O)NCC2CCC(C(=O)NCc3cc[nH]n3)CC2)cc1 N1(C(c2cccc(CC)c2)=O)CC(C2(NC(c3scc(C)c3Cl)=O)CC2)C1 C(CCC(N)=O)(C(=O)OCc1cnn(C)c1O)CC c1(C(N2CCC(CCOC)(NC(C34CC(C3)C4)=O)C2)=O)cc(C(C)C)ccc1C C(=O)(CCCc1csc(C)n1)N(CCCNC(C1CC(F)(CF)C1)=O)CC C1(C(N2CCOC(CC(N3CCCC3)=O)C2)=O)(OC)CCOCC1 C1(CC(=O)NCCC(N2CCN(C)CC2)C)Cc2ccccc2O1 CC1=NS(=O)(=O)NC=C1C(=O)NCC12CC(NC(C34CCCN(CC3)C4)=O)(C1)C2 c1(CC)cccc2c(C(=O)NC3CCCC3NC(=O)C(C(C)C)SC)c[nH]c12 N1(C(CNC(C)=O)=O)CC2(CCOCC2)CC1CNC(C1CCN2CCCC2C1)=O N1(C(c2c(C)nsc2)=O)CC(C)(C)OCC1CNC(=O)C(C)Cn1cccn1 c1(C(N2CC(NC(CCn3c(C)ncc3)=O)C(O)C2)=O)cnc2n(c1=O)CCS2 CC1CCC(CNC(c2cnn3c2CCC3)=O)N(C(=O)CCC(N)=O)C1 O=C(CCCCF)NCC1C2CN(CC(=O)NCC3CCC3)CC12.C1(CC2CC2)CC1 Cc1nn(CC(N2CC(NC(=O)CC3CCCOC3)C(O)C2)=O)c2c1CCCC2 c1(CC)c(C(N2CCCCC2CNC(=O)CCN(CC(F)(F)F)C)=O)csc1C N1(C(CC(CC)NC(=O)C(C)COC)=O)CCN(C2CC2)C(C)C1 c1(OC)cc(F)c(CC(N2CC(F)(CNC(=O)C(O)CC(N)=O)C2)=O)c(F)c1 Cc1c[nH]c2cc(C(N3CCN(C(C4CCC(C)O4)=O)CC3C(C)C)=O)ccc12 c1(OCCCC)nc(=NC(c2nccn3nccc23)c2ccncc2)[nH]cc1Br Cn1cncc1S(C)(=O)=NC(=O)C1CC(=O)N(C2CCCC2)C1 C(=O)(C#CC1CCCCC1)NC1CN(C(C(C)(C)C(N)=O)=O)CC1n1cccn1 C1(C)(NC(COCC(C)C)=O)CCN(C(=O)CN2CCCS2(=O)=O)CC1 C1(NC(C(C2CC2)OC)=O)CCC2(CC1)CCN(C(c1cccnc1S)=O)C2 c1(OCCC)ccc(NC(C2CC=CCC2)c2nnnn2C2CCCC2)cc1C n1(CC)ccc(C(=O)NCC=CCNC(c2cnc[nH]c2=N)=O)cc1=O N1(C(CC2(OC)CC2)=O)CC(NC(c2cccnc2N)=O)C(C)C1 c1(CNC(C2(CC)CN(C(Cn3ncc(CC)c3)=O)C2)=O)ccc(OC)nc1 C1(CC(=O)NC(C2(O)CN(C(C3CCCCC3)=O)C2)C)CCN(C)C1=O C1(NC(c2c(OCC)ccs2)=O)CCN(C(C2(O)CCCC2)=O)CC1C C1(CC(C)NC(c2cn[nH]c2)=O)CCN(C(C2CC2CF)=O)CC1 Fc1ccc(COCc2ccccc2NC2(c3nn[nH]n3)CCOC2)cc1F c1(CC)oc2ccccc2c1C(=O)NCCNC(c1nccc(F)c1Cl)=O c1(C(N(CC(C)NC(c2c(C(F)F)cccc2N)=O)C)=O)cnc2ccnn2c1 CC1CC2(CCN(C(=O)C=Cc3cccnc3)CC2)CN1C(=O)C(C)(C)CCCO N1(S(c2cn(C)nc2)(=O)=O)CC2(C)CN(C(c3ccccc3CO)=O)CC2(C)C1 c1(CN(C(c2ccc(N(C(C)=O)C)cc2)=O)C)cc(N(C)C)c(C2CC2)nn1 C=CC1(C(N2CCCCC2CC(N)=O)=O)CCN(C(c2cc(C)cc(O)c2)=O)C1 N1(C(COCCOC)=O)CCC(N(C(=O)C(CF)N(C)C)CCOC)CC1 CCC(CC(=O)N1CCC(OCCCNC(=O)CC2CC3C=CC2C3)CC1)OC c1(-c2cn(CC(N3CCN(C(C(C)C)=O)CC3)=O)nn2)cc(Cl)ccc1Cl C1(OC)CCC(C)(C(=O)NC(CCNC(=O)Cn2nc(C)cc2C)C(C)C)CC1 C1(c2n(C)ncn2)CN(C(=O)CO)CC1CNC(C1C2COCC12)=O CC1(C(N2CC=CC(NC(=O)CCCc3ccccc3)C2)=O)CCC(F)(F)CC1 Cc1cc(Br)cnc1C(=O)NCC1(O)CN(C(N)=O)C1.c12csc(n1)NC2=O N1(C(C(C=C)(C)O)=O)CCC(NC(=O)Cc2cn(CC3CC3)nn2)C(CC)CC1 C(=O)(C1CCC(=O)c2ccccc21)NC1CC(NC(=O)CC23CCC(CC2)C3)C1 N1(C(C(N)=O)=O)CCc2ccccc2C(N)C1 c1(C(=O)NCC2C(CNC(=O)CC3CCOC3)C2)cccnc1S CCCCCCCCC(=O)NC1CC(CNC(c2cncc(NC)c2)=O)C1 c1(C(=O)NCCC2(C(=O)NCC3(C#N)CC3)CCC2)c[nH]ccc1=O Cn1nc(CNC(C23CSCC2C3)=O)cc1C(=O)NCC1CCCOCC1 Cc1cc(C(=O)NCC(C2CCOC2)NC(c2coc(Br)n2)=O)c(C)cc1Cl c1(C(=O)NCC(CC(C)C)NC(C(CC)(C)C)=O)cc(C)cc2c1NCCC2 N1(C(C2(OC)CCOC2)=O)CC2CC(C1)C(CO)C2NC(=O)CC(C)C Cc1c(NCc2nc(C)c(C)[nH]2)ncnc1N1CCOCC(CO)C1 C12(C(=O)NC3C(NC(CS(CC)(=O)=O)=O)COCC3)CCCN(C1)S(=O)(=O)C2 N1(C(C(C)C)=O)CCOC(CN(C)C(C2CC2CF)=O)C1 c1(O)ccc2ccccc2c1.Cc1cccc(Cl)c1CNc1ccc2c(c1)OCO2 c1(C(N(CCC(C)NC(C2CCS(=O)(=O)N2)=O)C)=O)ncc(Br)cc1F C1(CNC(=O)CC2CCCCO2)CN(C(C2C3C4CCC(C4)C23)=O)C2(CCC2)C1 C(=O)(C1=CNC2=NCCCN12)NC1CN(C(C(C)OC2CCCC2)=O)CC1C(F)F C12(NC(c3csnn3)=O)CC(C(N3CCC3c3ncc[nH]3)=O)(C1)C2 N(C1CC2(CCCC2)Oc2ccc(Cl)cc21)C(c1ccc2c(c1)OCCNC2)=O C1(CNC(C(C)(C2CCCO2)NC(c2c(C)nc(CC)o2)=O)=O)CC2CCC1CC2 C(CCC(C)C(=O)N(CCC(C(C)C)NC(c1ccoc1S(C)(=O)=O)=O)C)OC c1(CNC(C(=O)N(C(C)C)C)=O)ccccc1-n1cc(-c2ncccc2F)nn1 C(=O)(C1COc2ccc(Cl)cc21)N1CCCC2(CN(C(COCC=C)=O)C2)C1 C1(C(N2CC(CCNC(C)=O)C2)=O)(NC(CNC(=O)NC)=O)CCC1 CN1CCC(NC(C2CNC(=O)CN2C(c2ccc(F)cn2)=O)=O)C(C#N)C1 c1(OCC)cccc2[nH]cc(CC(=O)N(CC(C)CNC(=O)CSC(C)C)C)c12 Cc1ccc(C(=O)N(CC(O)CN(C(=O)C(C)CO)C)C)cc1S(=O)(=O)CCO C12CCCC(C1)CNC(=O)CC1CCCN1C2=O.c1(C(N)=O)ccnn1CCO C1(C(N2CCC(C(N(C3CC(O)C3)CC)=O)O2)=O)Cc2ccccc2C1 C(=O)(C1CCCn2ccnc21)NCCCC(C)(C)NC(CS(C(C)C)(=O)=O)=O C(=O)(C1=CCCCC1C)NC1(C(C)NC(=O)C=Cc2ccncn2)CCCC1 C1(OC)CC(C(N2CC=CC2CF)=O)N(C(c2ccsn2)=O)C1 O=C(CCCOC(F)F)NC1(C2CNCCO2)CC1 C1(C(=O)NCc2c(CCNC(C(P(C)(C)=O)O)=O)ocn2)CCc2ncnn2C1 C=C1COc2c(C(N3CCC(CNC(c4c(F)cccc4F)=O)C3)=O)cnn2C1 CCC(CC)CCCN1CC(Cc2ccc(Cl)c(Cl)c2)C1 N1(C(CN(CCOC)C)=O)CCC(CCC(=O)NC2C=CC(CO)C2)C1 C=Cc1cnn(C)c1CNC(N1CCCCC(CO)C1)=O N1(C(c2c[nH]c(=N)o2)=O)CCCC(CN2CCN(C(C3CC(O)C3)=O)CC2)C1 N1(C(CC=CC=C)=O)CCC2(CO)CN(C(c3cc4ccccn4c3)=O)CC2C1 Cc1c(Br)noc1C(=O)NC1CCC(N(C(=O)Cc2ccc(O)cn2)C)C1 N1(C(CCNC(=O)OC)=O)C2CCC(C2)C1C(=O)NC1CCC2CC12 C1(C(=O)NCCOCCCC)CN(C(C2CC(n3cccn3)C2)=O)CC1C1CC1 C(=O)(CC(CC)CC)N1CCC(OC)(CNC(=O)C(C)OC2COC2)C1 c1(C(=O)NCCCN(C(c2c(CC)con2)=O)CC)ccc(C)c(S(N)(=O)=O)c1 c1(CCNC(C2CCN(C(C(C)NC(C)=O)=O)C2)=O)ccnc(C)n1 C1(NC(C=CC2N(C(c3n(CC)ccc3)=O)CCC2)=O)CCCC2(CCC2)C1 C(=O)(CCCC(=O)OC)O.C1(C(CC(=O)OC(C)(C)C)C)(COC)CCCCC1 Cc1oc([N+](=O)[O-])cc1C(=O)NC1CCC1NC(=O)C(F)=C1CCC1 C1(NC(CC2(C)N(C(C(C)CC3CC3)=O)CC2)=O)OCCCC1(C)C N1(C(c2c(C)onc2)=O)CCC(CCC(C)(C)NC(=O)C=CCN(C)C)CC1 C1(NC(C(C(C)(C)C)O)=O)CCC2(CC1)CC(NC(C1CC1NC1(C)CC(=O)N1)=O)C2 C1(CNC(c2cc(C)nnc2)=O)CN2CCCCC2CN1C(c1ccn(C)c1)=O N1(CC)CCCN(C(=O)C(C)(C)NC(=O)CC2(NC(=O)C(C)(C)C)CC2)CC1 c1(OC)ccc(C=CC(N2CC(C(=O)NCC3(CO)CC3)CCC2C)=O)cc1 CC(C1=CCN(C)CC1)NC(C1CC=CCC1NC(c1cc[n+]([O-])cc1)=O)=O c1(OC)ccc(C(N2CC(NC(c3sc(Cl)cc3Cl)=O)C3CC3C2)=O)c(OC)c1 c1(C(C)(C)C)nc2cc(Cl)nc(CC(F)(F)F)c2[nH]1.Cc1nc2c(s1)S2 c1(CNC(CC=C)=O)cnn2c1CN(C(c1nc(C)ncc1Cl)=O)CC2 C1(NC(=O)CCc2cnc[nH]2)(CNC(C2C=CCCC2)=O)CCCCC1 Cc1ccc2c(C(=O)NCCC3CC(NC(=O)CC4CCC(C)O4)C3)coc2c1 C1(CCC)CN(C(C2CN(C(=O)COCCN(C)C)C2)=O)CC1NC(=O)C=CC CN1CCN(CCC(N2CC(CNC(=O)C(C)(C)NS(C)(=O)=O)C(O)C2)=O)CC1 c1(C(=O)NC2C(C)(C)N(C(c3cncc(N)c3)=O)CC2)ccc2sccc2c1 N1(C(c2ncc(C)nc2)=O)CCC2CCCC(C1)N2C(c1cc(C#N)c[nH]1)=O c1(CC)nc(C2CCN(C3CCOCC3)CC2)n(-c2nc(Br)nn2C)n1 O=S(=O)(c1[nH]c(=NCCCN2CCC2)ccc1Br)NCCCCCC1CCC1 N1(C(c2c(CC)onc2)=O)CC2ON=C(CNC(=O)CCC(F)F)C2C1 c1(C(=O)NCC2N(C(C(C)(C)SC)=O)CC2)cnc2c(c1)CCS(=O)(=O)C2 Cc1nn(CC(=O)NCCCN(C)C(c2nnc(C3CC3)o2)=O)c(C)c1Cl c1(C(=O)NC(COCC)C(=O)NCc2ncn(C)n2)cc(F)ccc1O C1(C(N(C(CC)C)CCOC)=O)N(C(=O)C=CCF)CC12CCCC2 N1(CC(N2C(CNC(CC3CCN(CC)CC3)=O)CCC2)=O)CCCCCC1=O N1(C(C2(C)CCC2)=O)CC23CCCC2(C1)CN(C(=O)CCc1cn[nH]c1)C3 N1(C(CC(CC)C)=O)CCCC12CCN(C(C1CC(C)(C(=O)OC)C1)=O)C2 N1(C(=O)OC(C)(C)C)CCC(OC(Cn2c(C)c(Br)cn2)=O)C(O)C1 N1(C(CCC)=O)CSCC1C(=O)NC(CNC(=O)CCCc1nccs1)C(C)C N1(C(C(=O)N(C2(C#C)CC2)C2CC2)=O)CCC(c2cccc(O)c2)CC1 c1(N(C)CC2CCN(C(Cc3c(C)nc[nH]3)=O)C2)ccc([N+](=O)[O-])cc1F CCCCCC(C)(C)CNC(=O)NCCCc1ccnc(OC)c1 N1(C(CSCC)=O)CC(NC(C23CC(C)(C2)C3)=O)CC1C C(=O)(CC(C)C(F)F)N1C(CCNC(COC(CC)C)=O)CCCC1 C1(NC(c2ccccn2)=O)CC1C1CCCN(C(c2csnn2)=O)C1 c1(NC(c2c(C)nc(-c3c(C)cccc3)s2)=O)cc(=O)n(C)cn1 C1(C(N(CCc2ccccc2)Cc2ccc(C)nc2)=O)(C(=O)O)CC2(CCC2)C1 c1(C(=O)NCC(CNC(CCc2cn(C)nn2)=O)F)ccc(Br)cn1 CC1C(N=c2[nH]c(=NCc3ccnc4ccccc34)[nH]c3c2SCC3)CCN1C C1(NC(C2CN(C(C3CC3(Cl)Cl)=O)CC2(F)F)=O)CCC2(CC1)CC2 N1(C(C2CC(=C)C2)=O)CCCC(C)(C(=O)NC(C)C=CCCC)C1 N1(C(c2ccc(OC)s2)=O)CC2CCN(C(=O)C(=O)NC3CC3)CC12 c1(CN(C(CC=CC)=O)CCCNC(C2CC2OC(C)=O)=O)cc(C)n(C)n1 c1(CN2CC(C(=O)NC(CCCC)CO)OCC2)cnc(O)nc1O C12(CNC(=O)CCc3cocn3)CCC(CC1NC(c1ccc(Cl)o1)=O)C2 Cc1cc2ncnc(N3CC(Cc4ccccc4)C(CC4CC4)C3)c2cc1C C(=O)(CC(C)C(=O)NC1CCCC1CNC(=O)C(CC)CO)OCC N1(C(Cn2c(C)nnn2)=O)CC2CCN(C(=O)CN3CCNC(=O)C3)CC2C1 C1(NC(C2C3CCCC23)=O)CC(C(=O)Nc2c(C)ccc(O)c2)=CC1O Cc1oc(CO)nc1C(=O)NCCN(C(C12CC(CF)(CO1)C2)=O)CC1CC1 c1(C(=O)NCC2C=CCN2C(=O)CC2C=CS(=O)(=O)C2)nn2cccnc2c1Cl C1(C(=O)NCCCC)CC(C)(C)CCN1C(=O)CC12CCC(CC1)C2 C1(NC(Cn2c(C)ccn2)=O)CCCN(C(c2ccc3c[nH]nc3n2)=O)CCC1 Cc1ncc(Cl)cc1CC(=O)NCC(C(C)C)NC(=O)C1=NNC(=O)C1 O=C(N=c1cc2c(n[nH]1)CCC2)C1CCC2(CCOCC2)O1 C12CC3(C1)C(C3(F)F)CN2.c1(CN(CC=C)C(=O)NC)cnccn1 c1(NCC(c2cccc(Cl)c2)C)nccc(=NCC(F)c2ccccc2)[nH]1 C1(NC(CN(C(C)C)C)=O)CN(C(=O)Cc2ncsc2Cl)CCC1O C1(C(N2C3CC(NC(Cc4ccn(CC)n4)=O)C3CC2)=O)CCCC2(CCC2)O1 N1(C(Cn2c(C)cc(C)n2)=O)CCC2(CCC2NC(=O)CN2CCC(C)C2)CC1 c1(C(N2CC(C(C)NC(CCc3nc(C)c(C)o3)=O)C2)=O)cn(C)ccc1=O N1(C(C(C)(C)C)=O)CC(NC(=O)C(c2cscc2Br)=O)CC12CCCC2 C=C(C)CCCC(=O)N(C)CC1CCCCN1C(=O)Cc1cnsc1 C1(CNC(c2ncc(C)nc2)=O)CC(NC(=O)CCNC2COC2)C12CCC2 C12(C(=O)NCC(CN(C(=O)CCc3ccco3)C)(C)C)CCCC(=O)N1CCC2 N1(C(c2c(C)ncn2C)=O)CC(F)(F)CC1(C)CNC(=O)C(c1cccnc1)C c1(C(=O)NC2CC(NC(C(CC=C)c3ccccc3)=O)C2)cnn(C)c(=O)c1 Cc1cc(N(C(=O)Nc2ccnn2C(C)(C)C)CC2CC2)cc(F)c1 N1(C(c2c(C)nns2)=O)CC(C(=O)NC(c2cccnc2O)C)CC(C)(C)C1 N1(C(CCOCCOC)=O)CC(NC(C23CC(CF)(CO2)C3)=O)CC(O)C1 CC(CC(C)NC(C1CC(C)(C)C1)=O)NC(=O)CCCNS(C)(=O)=O C1(C(=O)NC(C)C(=O)Nc2ccnn2C(c2ccccc2)C)CCCCNC1=O c1(C(=O)NCCN(CC(C)O)C(c2cnc(-c3ccsc3)s2)=O)ccccc1F N1(C(CCc2ccn(C)c2)=O)CCC(O)(CCNC(=O)C(O)c2ccsc2)C1 c1(C(=O)NC2CCCCN(c3ncccn3)C2)ccc2nc[nH]c2c1F C1(NC(CCOCC#C)=O)COCCC1NC(=O)C(c1ccc(C)cc1)(C)C c1(C(=O)NC2CC(CNC(=O)COc3ccc(Cl)cc3)C2)cncc(F)c1 c1(CN(C)C(C2CCN2Cc2ccnc(Cl)c2Br)C)ccc(O)cc1C C(=O)(CCC(O)Cc1ccccc1)NC(CNC(c1cccc(CSC)c1)=O)C N1(CC)CCOC(C(=O)NCC23CC2CN(C(c2c(C(C)C)cnn2C)=O)C3)C1 C1(C)(C(N(CC)Cc2nccn2C)=O)CCN(C(=O)CCCC(C)=O)CC1 Cc1c(C(N2CC(O)CC2C)=O)ncn2c(C(F)(F)F)cnc12 c1(CC(=O)N(CC(C)N(C(CCOCCOC)=O)C)C)nc([N+](=O)[O-])n[nH]1 c1(C(=O)NCC2(F)CN(C(CC(C)(C)OC)=O)C2)c(C)c(C)cc2ccccc12 CCCCC(O)C(=O)NC1(C)CCCN(C(=O)C(O)Cc2cnc[nH]2)C1 c1(CN2CCC(C(C)NC(C3C4CC5C(C4)C35)=O)CC2)ccccc1S(C)(=O)=O O=S(=O)(c1c[nH]ccc1=NCC1CCC(F)C1)NCc1nnc2n1CCCCC2 C1(C(N2CC(F)(C(=O)Nc3ccc(CC)cc3)C2)=O)OCCCC1(C)C CC1(C)C=C(C(=O)NC2CC(F)(CC3CCCC3)C2)C1.c12csc(n1)NC2=O c1(C(=O)NC2(NC(C(COC)NC(C)=O)=O)CCCCC2)nn(C)c2c1CCC2 N(C(=NCCc1ccccc1)NC1CCCCCCC1)CC(F)(F)c1ccoc1 c1(C(C)=O)ccc(C(=O)NCC2CCCN2C(=O)C(C)Cn2cccn2)o1 CCCCC(C)C(=O)NC(CNC(C1(C)CCN(C(C)=O)C1)=O)C(C)C C(=O)(N=c1cc(Cl)n(C)[nH]1)c1nc(Nc2nc(C(C)C)nc(C(F)(F)F)c2)sc1 N1(C(COCC)=O)CCN(C(C2CCC2)=O)C(c2cn[nH]c2)C1 C1(C(N2C(C)C(NC(c3cscn3)=O)CC2)=O)CC(=O)NC(=O)N1 C1(CC(=O)NC2CCN(C(c3cn(CC(N)=O)nn3)=O)C2)CCCCC1O C12(CCCC1C)C(=O)N2.Cc1ncsc1CCNC(C12CSCC1C2)=O c1(C(=O)OC)ncc[nH]c1=NC1CCC(NC(=O)CCN2CCCS2(=O)=O)CC1 CS(=O)(=O)c1ccc(C(=O)NC2CCCC(NC(=O)C#CC3CCCO3)C2)s1 C(=O)(C#CC(C)(C)CNC(C1CCCCCC1)=O)NC(CC(C)C)C(N)=O Cc1ccc2c(=NCC3CCc4c[nH]nc4C3)[nH]c(N3CCC(C)(F)C3)nc2c1 C1(C(N(C)CCNC(C2(C(F)(F)F)CC2)=O)=O)CC(=O)N(C2CC2)C1 N(C(=NCC1CCOC1)NC1C=CCCC1)C(C)(C)C C1(NC(=O)Cn2cccn2)CC(NC(=O)CC2(CO)CCCCCC2)C12CCC2 C#Cc1cccc(C(=O)NCC2CC(CC(N3CC4CC4(CC)C3)=O)C2)c1 c1(C(CNC(=O)C=C(C)C(C)C)NC(c2c(C)nnn2C)=O)cc(F)cc(Cl)c1 CCC(C)C(C(=O)NCC1C(=O)N1)N(C)C.C(C)(C(C)(C)C#N)SC CC1CCc2nc(C(=O)NC34CC3CN(C(C3(n5cnnn5)CC3)=O)C4)cn2C1 C(=O)(C(O)CC(C)(C)C)N1CC(CC)N(C(=O)CN(C)CCO)CC1 CC1ON=C(C(=O)N2CCC(C3CC3)C2CNC(=O)CC2CCCCN2C)C1C Nc1cc(C(=O)NCC2CCCN2C(=O)CC2CC3CCC2CC3)cnc1Cl C12(NC(c3cccc4[nH]ncc34)=O)CN(C(c3ccsc3)=O)CC1CS(=O)(=O)C2 c1(C(N2C(CC(=O)NCC(C#C)CC3CC3)CC2)=O)cnc(NC)cn1 C(=O)(C1CCCc2ccnn21)NCC12CC(NC(C(CC)N(C)C)=O)(C1)C2 CC1=C(C)CC(C)(C(N2CCC3CN(Cc4nc(C5CC5)nn4C)CC23)=O)CC1 C1(C(C)(C)NC(=O)CSC(=N)N)CCN(C(=O)CO)C1 c1(C(N2CCN(S(CCC)(=O)=O)C3C2C3)=O)c(C)ccc(Br)c1F N1(CCC2(C)CC2)CCC2=C(COC2=O)C1 C(=O)(CCCCCc1cccs1)N(C(CNC(CCCOC(C)C)=O)C1CC1)C Cc1cn2c(n1)CCC(C(=O)NC1CC(O)(CNC(c3cccc(O)c3)=O)C1)C2 CC1(C(N2CCC3CN(C(=O)CN4CC=CC4)C3C2)=O)CC(c2ccccc2)=NO1 C(CC)(CC)(CCNC(=O)CS(=O)(=O)NC)NC(c1ncn(CC)c1)=O c1(CC)cncc(C(N2CC3CC2(C(=O)Nc2cccc(N(C)C)c2)C3)=O)c1 C1(C(C)CNC(c2ccc[nH]2)=O)CCN(C(C2CC2C(C)O)=O)CC1 c1(NC(C2COCCN2C(=O)CCC2CC2)=O)cc(Br)cc2[nH]ncc12 c1(C(=O)NC(C)C(C)(C)NC(=O)C=C2CCCCC2)c[nH]c2cc(C#N)ccc12 c1(CC(N2CCC(CN=c3[nH]nc(CC#N)o3)(C)C2)=O)ccc([N+](=O)[O-])cc1 C1(C(=O)OC)C(NCCC#CCC)CCN1C(c1ccccc1Cl)=O n1(CC)nnc(C(N2CCCC2(CO)CNC(=O)C=Cc2cc[nH]n2)=O)c1C C12(NC(c3c(CC)cno3)=O)CCCC1N(C(c1cc(C(F)(F)F)no1)=O)CC2 C1(C(N2CCN(C(c3onc(COC)n3)=O)C(C)C2)=O)COc2ccccc2O1 C(C(C(F)(F)F)N1CCN(C(=O)CNC=O)CC1)NC(C1(Cl)C(C)(C)C1)=O CONS(=O)(=O)c1ccc(NCCNC(C2CCCC2)=O)cc1.C1(=O)C(C)CN1 C1(C=O)CCCN(C(=O)C(C)(CC)CO)CC1.C(=O)(C(CO)O)CC c1(CC(=O)NCC(C(C)C)NC(C2CC(C)(F)C2)=O)ccc(C(N)=O)cn1 Cc1c[nH]c(CC(N)=O)c1C(=O)NC(C)CN(C(=O)CC(C)(F)F)C C(=O)(C(COC(C)C)NC(=O)CCN(C)C)N1C(C(C)(C)C)CC1 C(=O)(C1=CC2CCC=CCCC12)N1CCN(C(Cn2c(=N)scc2)=O)CC(O)C1 C1(NC(c2cn(CCC)nn2)=O)CC2CN(C(c3cc(C)c[nH]3)=O)CCN2C1=O C1(CC(=O)NC2CCCN(Cc3ccn(CCF)n3)C2)COc2ccccc2O1 N1(C(c2cc(C)[nH]c2)=O)CCC2(CC1)CCN(C(C1(c3cccs3)CC1)=O)CC2 C12(CNC(C=C(C)Cl)=O)CC1CN(C(c1ccc(CC(F)(F)F)cc1)=O)C2 CC1CCC(NC(c2cc(O)n(C)n2)=O)CN1c1cc(=O)n(C)cn1 C(=O)(C1(C)CCc2ccccc21)NCC1=CCN(C(C(CC2CC2)OC)=O)CC1 C1(NC(CCCSC)=O)CCC(C)(C)CC1CNC(c1nc(=O)cc(N)[nH]1)=O C(=O)(CCCCCCCCC(=O)Nc1cc(C#N)ccc1C)OC C1(NC(CC(CC)C)=O)COC2(CNC(c3scnc3COC)=O)CC1C2 c1(C(N(CCCn2cc(CCC(N)=O)nn2)C)=O)cc2cc(Br)ccc2cn1 c1(C(CC(=O)O)NC(=O)C(F)(Cl)c2ccccc2)cccc([N+](=O)[O-])c1 c1(C(=O)NCC(CCNC(C2N(C)CCOC2)=O)(C)C)cc2c(nn1)CCC2 c1(C(N(CC(CN(C(c2cccnc2)C)C)O)C)=O)nc(-c2ccncc2)cs1 c1(C(=O)NC2CC(NCc3ccsn3)C2)cccc([N+](=O)[O-])c1 C(=O)(C=CSc1nc[nH]n1)N(c1cccs1)CC(=O)NC(CC=CC)C C123CCN(CCC1C2)C(=O)CONC3=O.C(CC(C(C)C)NC(C)(C)C)OC C(N=c1[nH]c(=NCc2ccc(Cl)cc2F)c2ccccc2[nH]1)C1CCCC(=O)N1 N1(C(C2N(C(C=CC(C)(C)SC)=O)C(C)C2)=O)CCN(C(C)=O)CC1C N1(C(c2c(CC)nco2)=O)CCC(NC(=O)CCC2CCCC2)CC1 C#CC1(O)CC(C(N2CC(N(C(=O)C(F)(F)c3cccnc3)C)C2)=O)C1 N1(C(C(C=C)O)=O)CCCC12CCN(C(c1cnc(C(C)(C)C)o1)=O)C2 C(N=c1[nH]c(=NCCCNS(C)(=O)=O)[nH]c2c1CCC2)C1CC(OC)C1 c1(C(=O)NC2CN(C(Cc3c(C)nc(C)s3)=O)C(C)(C)C2)cc(C)c(F)cc1N N(C(=NCc1cccs1)NCC1(C(N)=O)CC1)CC(c1ccccc1)O c1(CC)ccc(F)cc1NC(=O)C(CCCOC)NC(C1CCS1(=O)=O)=O C1(C(=O)NC(CN(C(c2cccs2)=O)CC)Cc2ccccc2)CCCC1(F)F C(=O)(C(C)CS(C)(=O)=O)N1CC2CC(CNC(CCCCSC)=O)C2C1 c1(C(N(CC(C)C(=O)O)C2CC2)=O)cccc(N(C)C)c1 Cc1ccc(C(=O)CN2CCC3CC23C)cc1S(C)(=O)=O c1(C(=O)NCCCCCN(C(C(C=C)OC)=O)C)ccn2cccc2c1 N1(C(CCCC=C)=O)C2CC=C(C(=O)C(C(CO)C(=O)OC)=O)C1CC2 c1(COC)nc(NC(CC2(C#N)CCC2)C(=O)OC)cc(N2CCC3CC23)n1 c1(C(N2CC=CC(C(N3CC(C4CC4)(N(C)C)C3)=O)C2)=O)ccc2occc2c1 Cc1cc(C#N)cnc1C(=O)NCCNC(C1CCN(C(c2ccoc2)=O)C1)=O CC(C)C(O)CC(=O)N1CCC(CNC(=O)C(C)(C)CCN(C)C)C(O)C1 N(C(=NCC(F)F)NCC1NC(=O)CC1(C)C)CC1(C=C)CCC1 C1(CN(C)C(c2cn[nH]c2)=O)CCCC(NC(c2cn(-c3nccs3)nn2)=O)C1 Cc1c(Cl)ccnc1C(N1CCN(C(c2cnn(C)n2)=O)C(C)C1)=O N1(C(C(C)(C)c2cccnc2)=O)CC2(C1)CN(C(=O)CCN1CCC1)CC2CO C12(C(N(c3ccc(Cl)cc3C#N)CC)=O)COCC1CN(C(=O)OC(C)(C)C)C2 c1(C(N(CC(C)NC(c2nnsc2C)=O)CC)=O)cc2c(cn1)COCC2 C1(NC(COCCCC(C)C)=O)CCN(C(c2csc([N+](=O)[O-])c2)=O)CC1C Nc1cc(F)c(O)cc1C(=O)NC12CC1CN(C(c1csc(Cl)c1)=O)C2 C12(CNC(c3cc(C)[nH]n3)=O)CCCC1N(C(C1CC1(F)F)=O)CCC2 Cc1sc2ncnc(C(=O)NCC(=O)NC3CC3CNC(=O)C3CC3)c2c1C CC(C(=O)N1CCC(C2CCCN2C(c2ccc(C(F)F)o2)=O)CC1)C(C)(F)F N1(C(c2cn(C(C)C)nn2)=O)CC(CNC(=O)CC(C)(F)F)CC12CCC2 C12(NC(c3c[nH]c(=NCC)s3)=O)CN(C(=O)C(C)=C(C)C)CC1CS(=O)(=O)C2 c1(SC)nccc(NC2CC2C(=O)Nc2csc(C#N)c2)n1 C1(C(=O)NCCC(CC)(F)F)CN(C(=O)CCC(C)CN(C)C)CC1(C)C C(=O)(C(C#N)=CNC(C)C)N1CC(CC=C)(C(=O)NCCC(C(=O)OC)OC)C1 C1(N(C(=O)CCc2cnn(C)n2)C)CN(C(c2cn(C)ccc2=O)=O)CC12CC2 c1(CN(C2CCN(C(=O)C(C)OCOC)CC2)CCOC)ccc(F)cc1Cl Cc1cn(C)cc1C(=O)NC(C)(CO)C(=O)NCC1(O)CCC(C)C1 C=C(C)C(CC(=O)NCC1(F)CC(NC(=O)Cc2cnn(C(F)F)c2)C1)OCC C=CCC(CC)C(=O)N1CCC(C(=O)NCCn2ccnc2C)(CO)C1 C1(NC(C(C)n2cccn2)=O)CC2CCC1CC2NC(=O)CCCCCn1cnnn1 N#Cc1ccc2c(c1)N(C(C1(CNC(c3ccccc3F)=O)CC1)=O)CC2 c1(OC)cccc(CC(O)C(=O)NCCCCCN(C(=O)CN(C)C(C)=O)C)c1 C(=O)(CCP(C)(C)=O)NC1(C)CC(C(N2CCC(C(C#C)C)CC2)=O)C1 N1(Cc2ncc(C)cc2C)CC2CCCN(C(=O)CCC(=O)NC3CC3)C2C1 N1(CCNC(C2(C)CC(C)C2)=O)CCN(C(=O)CC2CCCCN2C)CC1 c1(C(C(=O)NCCN(C(=O)CC(C2CC2)SC)CCC)OC)c(C)n[nH]c1C.C1CC1 c1(C(=O)NCC(CN(C(C2CCC(C)(C)O2)=O)CC)(C)C)ncccc1F N1(C(C(C)(C)N2CCCCC2)=O)CCC(C)(CNC(=O)CC2CCOC2)C1 c1(C(=O)NC2C(C)CCN(C(c3cnco3)=O)C2)cc(O)c2sccc2c1 C(=O)(C(C(C)NC(c1cccc(CO)n1)=O)C(C)C)NCC(CC)(C)OC c1(C(=O)NC2CC(C)N(C(C3(C)CCN(C)CC3)=O)C2)ccc2c(c1)CCN2C C1(C(C(=O)N(CCNC(C(C)OCc2ccccc2)=O)C)O)COC(C)(C)O1 N1(C(c2c(C)nco2)=O)CCN(C(=O)COc2ccc(F)cc2Cl)C(C)C1C CC1CCCC(CC(=O)NCCN(CCCN(C)C)C(=O)CC2CCC(C)C2)O1 CC(C)CCC(=O)N1CCC(C)C1CNC(c1ccnn1C(C)C)=O Cc1cc(-c2cn(CC3CCN(C(=O)C(C)CSC(F)(F)F)C3)nn2)cc(C)c1 c1(C(=O)NC2CN(C(CC(=O)OC)=O)C(C)(C)C2)cc2nccc(C(F)F)n2n1 c1(CN2C(C)(C(=O)Nc3c[nH]nc3Cl)CCC2)cc(OC(F)(F)F)ccc1C C1(NC(CC2CCN(CC)C2)=O)CN(C(=O)C(C)=C2CCCC2)CC12CC2 C1(C(N2C(CCNC(=O)C(F)C(F)(F)F)CCCC2)=O)CN2CCCN1CC2 N1(C(C=C(CCC)C)=O)CCC(CNC(=O)CSc2ccccc2OC)(SC)C1 c1(OC)ccc2c(c1C(N1CC3C(N(C(=O)C(C)C(C)C)C)C3C1)=O)CCC2 C1(C(=O)NCC2(C)CCCO2)C(C2CC2)CCN1C(=O)CN1CCCC1 c1(C(=O)NC(c2cn(CC)nn2)C)cc(Cl)ccc1SC c1(CC(=O)NCCCC(C)NC(C(C2CCOCC2)OCC)=O)ccc(Cl)c(F)c1 C=CCC(CC=C)C(=O)N1CCOCC1CNC(c1cc(CC)ncn1)=O Cc1cccc(Cl)c1CC(=O)NCC1CN(C(=O)CCN2CCN(C)CC2)C1 N1(C(c2cc(C)cc(Cl)c2)=O)CCCC(C)(C)C1CNC(C1(N(C)C)CC1)=O C1(NC(C(C)NC(=O)NC)=O)COCCN(C(=O)CCc2noc(COC)n2)C1 C1(C(=O)NCc2cc(=O)cc[nH]2)CC2CC2N1C(=O)CCc1nncs1 N1(C(C(n2ccc(C)n2)C)=O)CCc2c(c(CNC(C3CC3CF)=O)nn2C)C1 c1(CC(=O)NC2CC(CNC(C3(OC)CC3)=O)C2)c[nH]ccc1=O c1(C(=O)NC(C2CCN(C(c3ccncc3Cl)=O)C2)(C)C)cc2ncccc2o1 N1(C(c2n(CC)nnc2)=O)CCN(C(=O)C=Cc2ccccc2C)C2(CC2)C1 c1(CNC(=O)NCC(c2cc(C)cc(C)c2)O)ccn2ccnc2c1 c1(C(=O)NC2(C(=O)NC3CC(SC)C3)CCC2)cnoc1C1CC1 c1(C(N2CCC(N(C)C(C3CC3F)=O)C2)=O)ccc2n[nH]cc2c1 c1(COC)cc(C(=O)NCC2CC2NC(c2cc(Br)ccn2)=O)c(C)o1 CCCCCCC(=O)NC1CC(CNC(=O)Cc2csc(COC)n2)C12CCC2 N1(C(C2(CCC)CC2)=O)CCCC1CN(C(c1cn(CC)nn1)=O)C1CC1 C1(NC(CS(CC)(=O)=O)=O)CN(C(c2cnc(OC)s2)=O)CC2(CCC2)C1 C1(NC(C2C=CC(NC(CC=C)=O)C2)=O)CCN(c2cc(O)ncn2)CC1 C(=O)(C(C)(C)CC(C)=O)NCc1c(C(=O)NCC(COC)(C)O)nccc1 c1(OC2CCC(CC#N)CC2)ccc(NCCOCCN)cc1 C1(C)(CC)CCN1C(=O)COC1CCN(C(=O)C(C)N(CC)CC)C1 c12nc(cc(=NCC3CCCC3O)[nH]1)NCC(C)N2C.c1(COC)ccccn1 C1(C(=O)NC(C(C)C)C2CCC2)CC1C1CN(C(C2(C)CS(=O)(=O)C2)=O)C1 N1(CC(=O)NC(CC)CNC(c2ccc(C(C)(C)OC)cc2)=O)C(=O)CNC1=O CCN=c1[nH]c(C)c(C(N2CCC(N(C(=O)C=C3CC3)CC3CC3)CC2)=O)s1 N(C1COc2c(Cl)cccc21)S(CC1(C)CCOC1)(=O)=O C(CC(C(=O)NCCC1CC(=O)N(C)C1)NC(C1CCCC1F)=O)OCC C1(CNC(=O)C2=COCC2)CC2(CCN(C(=O)Cc3cncnc3)C2)CO1 CC(C)C(C)CC(=O)NC1COCC1CNC(C1(F)CCN(C)CC1)=O c1(C(=O)NCC2N(C(CCC=C(C)C)=O)CCC2C)ccc2c(c1)COC2 c1(OC)nsc(OC)c1CNC(c1cn(C2CC(N3CCSCC3)C2)nn1)=O C(=O)(CC(C)N(C(=O)C(C)N(CCO)CCNC(=O)Cc1cnc(C)s1)C)OC C(=O)(CCC(N)CCCC)N1C(OCCOCCCC)CCCC1 N1(C(c2c(CNC(CCc3ccc(C)o3)=O)ocn2)=O)CCN2CC(C)CC2C1 N1(C(C2C(C)C(=O)C2)=O)CCC2CN(C(c3scnc3Cl)=O)CCC12 c1(OC)cnc(C(N2CCC(O)(C(C)NC(C3(CF)CCOCC3)=O)C2)=O)cn1 c1(SCCN2C(CNC(=O)CC(O)c3ccncc3)CCC2)cccc2nccn12 C(=O)(C(F)(F)C(F)(F)F)N1CCN(C2CCN(C(C3CC(C)NC3)=O)C2)CC1 c1(C(N2CCN(C(C(C)NC(C)=O)=O)CC23CCC3)=O)cc2ccccc2cc1O N1(C(c2ccc(CSC)o2)=O)CCc2c(CNC(C3(C#N)CC3)=O)cccc2C1 N1(C(CC)C(=O)NCC(C)(C)Nc2ncc(Br)c(O)n2)CCc2ccccc21 c1(OC)nccc(CN2CC(C(=O)Cc3ccc(C(=O)OC)cc3)C(F)C2)c1F c1(C(=O)NCC2(NC(CC3C(C)C(=O)CC3)=O)CCCC2)cc[nH]c2nccc1-2 c1(CC(=O)NC2(CCNC(Cc3c(C)ncs3)=O)CCC2)ccnnc1O C1(CNC(=O)CN2CCSCC2)CCCCC1NC(=O)C(=O)NC1CC1 N1(C(CCCOC(C)=O)=O)CCN(C(C2(C)CC2(C)C)=O)CC2(CC2)C1 N1(C(C2CCCN(C(C3(CCCC)CC3)=O)CC2)=O)CCC2(CCOCC2)C1 Cc1nn2cc[nH]c(=O)c2c1C(=O)NC(CNC(=O)Cc1cncc(O)c1)CO c1(OC)ncc(C(=O)NCC(O)CN(CCCNC(=O)COC(F)F)C)cc1Cl S(=O)(=O)(C1CC2CCC1C2)N1C(c2n(C)ccn2)CCC1.c1(CC[SH]=O)ccc(Br)cc1Cl Cn1ncc2c(O)nc(=NCC(CNC(C3CCCC3O)=O)C(F)(F)F)[nH]c12 CC1C(NC(C2CN(C)CCN2C)=O)CCCN1c1nnccc1C#N c1(C(N2CCC23CN(C(C2C4CC5C(C4)C25)=O)C3)=O)cc(O)cc(F)c1 c1(C(=O)NCCCC(C)NC(c2cnc(C(N)=O)s2)=O)c[nH]c(=S)cn1 C1(NC(CCOCCOC)=O)CC2(CCCN(C(c3ccnc(S)c3)=O)C2)C1 c1(C(N(C)CC2N(C(c3cncc(C)n3)=O)CCOC2)=O)ccc(C)c(Cl)c1Cl c1(NC(c2c(C)noc2C)CC=C)ccc(S(=O)(=O)NC(CO)CCC)cc1C#N c1(C(=O)NC2C(NC(C3(C(=O)OC)CC3)=O)C2)ccc2scnc2c1 C1(C(N(CCCNC(c2ccoc2Cl)=O)C(C)C)=O)CCCc2ccccc2C1 N1(C(=O)CC2CN(Cc3ccc4c(c3)CNC4=O)C2)CCc2c(O)n[nH]c2C1 c1(C(=O)NCC2(F)CCCN(C(CC=CC=C)=O)C2)[nH]c2ccc(Cl)cc2c1Cl CC1CC(C(N2CCCC(CNC(c3cc(F)c[nH]3)=O)C2)=O)CC(=O)N1 c1(-n2cc(CN(C(C)C(=O)O)C(c3ccccc3)=O)nn2)ccccc1C(=O)O C1(NC(CCCSC)=O)CN(C(C2CC2c2cccc(F)c2)=O)C2(CCCC2)C1 c1(Cc2cn(C(C)(C)CC(=O)NNC)nn2)ccc(F)c(OC)c1.C12CCCN(C1)C2 Cc1cccc(OCC(=O)NC(C)C(C)NC(C2(F)CC2Br)=O)c1C c1(CCNC(C2CCCN(c3nnc(C)o3)C2)=O)cc2cc(Cl)ccc2nc1C c1(C(N(CCCCN(C(c2cnc(CCC)s2)=O)C)C)=O)cc(OC)n(C)n1 c1(C(N(C)CC2(O)CN(C(C3C(CC(C)C)C3)=O)C2)=O)cc(Cl)c(Cl)s1 c1(C(=O)NCCC(C)N(C(=O)CCC2CC2(F)F)C)cncc(-n2ccnn2)c1 Cc1ccnn1C(C)C(=O)N(C)CC1(O)CN(C(=O)C(O)Cc2ccccn2)C1 N1(C(c2ccc(CNC(c3c(C)c(C#N)[nH]c3)=O)cn2)=O)CCC(O)CC12CC2 C(CC(C)(C)C(=O)NCC1(C)CCCN1C(C12CCC(OC)(CC1)C2)=O)OC c1(CCNC(=O)CNC(N2CC=CC2)=O)c(F)ccc(C(F)(F)F)c1F CN1CCN(C(=O)CCc2cnn[nH]2)CC1C(=O)NCC1(O)CC(CO)C1 c1(CC(=O)NC2CCC(NC(C(C)(C)N(C)C)=O)C2)cccnc1O C(C1c2ccccc2CN1C(C1CNC(=O)C1)=O)NC(C1C(=C)C1)=O Cn1ncc2c(N3CCC(CNC(C45CC(C4)C5)=O)C3(C)C)ncnc12 C(C)(C(=O)NCCCOCCNC(=O)Cc1ccncc1)(C1CC1)OC C1(C(N2CCCC(C)(CNC(C3CSCC(=O)N3)=O)C2)=O)CCc2nn[nH]c2C1 C1(CCNC(c2cnc(CC(C)C)s2)=O)CCN(C(C2CC3CCCC23)=O)CC1 c1(C(=O)NCCNC(C2C3CCC(C3)S2(=O)=O)=O)ccc2ncc(Br)cc2c1 CC#CCCC(=O)NCC(C)CN(C(=O)C(F)C1CCOC1)C C(=O)(C=CS(=O)(=O)CC)NCCCN(C(C1CN(CC)C(=O)C1)=O)CCO N1(C(C(CCC)NC(c2n[nH]c3ccccc23)=O)=O)CCc2c(O)noc2C1 Cc1noc(CSC2(NC(=O)OC(C)(C)C)CNC2)n1.C1C(=O)N1 C1(NC(C2(C)CN(C(c3nn(CC)c(C)c3)=O)C2)=O)CCCC2(CC2)C1 N1(C(C=C(C)C2CC2)=O)CCC(NC(C2CC2C)=O)C12CC2 C(=O)(C(C)S(=O)(=O)CCC)NCC1CC(NC(C2CC(CCC)OCC2)=O)C1 CCCCCCC(=O)N1CCN(C(=O)CCc2cccnc2C)C(C)C1 c1(C(c2nnc(C)o2)NC(=O)NCc2ccc(F)cc2)cc2n(n1)CCCC2 CC(CC(=O)NC1CCCC1CNC(=O)CCC1CCC(=O)N1)C1CCCCC1 N1(C(C2N(C)CC2)=O)CCC(C(C)(C)NC(=O)COC2CCCC2)C1 CC(C)CC(C(=O)N1CC(=O)CC1C(=O)NCCC1(CO)CC1)N(C)C c1(C(N(CC(O)CNC(=O)CSC(F)F)C)=O)cc(C(F)(F)F)no1 CC(CC(=O)OC(C)(C)C)CC(C)(C)C.c12cccc(n1)N1CCC(C1)NC2 C1(CNC(Cc2ccc(OC)cn2)=O)CC2CCC(C1)N2C(C1(C)CC1(F)Cl)=O N1(C(c2c(CC)noc2)=O)C2CCC1CC(CNC(=O)C(C)(C)c1nccs1)C2 N1(C(C(C)C)=O)CC(NC(=O)CC2(C)CCC2)CC1C CC1(C)CN(C(=O)CC#N)CC1NC(c1cn(-c2ccccc2CO)nn1)=O C1(C(=O)OC)CCCC1N=c1[nH]c(C(F)(F)F)nc2[nH]cnc12 C(CC(C)(C)CO)c1cn(CCN(C)C(c2ncoc2-c2cccs2)=O)nn1 CC(C)(CC(F)F)C(=O)N1CCCC(C(=O)NC2CCCN2CCO)C1 c1(NCC2(S(C)(=O)=O)CC2)ccc(S(=O)(=O)NC2CCSC3(CCC3)C2)cc1C#N c1(N(C)C)cccc(C(=O)NC23CC(NC(=O)C(=O)NCC(F)(F)F)(C2)C3)n1 C1(NC(c2c(N)c(C)n(C)n2)=O)CC(NC(C2CCS2(=O)=O)=O)C12CCOCC2 Cc1nc(O)nc(C)c1CC(=O)NCCC1CN(C(C2(C3CCC3)CC2)=O)C1 c1(C(N2C(C(C)NC(CC(CCCC)O)=O)CCC2)=O)ncnc2c(C)csc12 c1(CNC(C2CNC(=O)O2)=O)cccc(C(=O)NCCc2ccco2)n1 c1(C(=O)NC(CN(C(C2(C(=O)NC)CC2)=O)C)C)cnc(CC(C)C)s1 c1(C(N2CC(CNC(C(C)C(F)F)=O)C3(C2)CC3)=O)cc2c(F)c(F)ccc2[nH]1 c1(C(=O)NC(CCC)CNC(=O)COCc2scnc2C)nnccc1C C(c1ccccn1)=CC(=O)NC1CC(NC(C(C)Cc2cnc[nH]2)=O)C1 c1(C(N(CC(C)N(C)C(c2ccccc2N(C)C)=O)C)=O)c2c(nn1C)CCCC2 C(CC(C(C)C)NC(=O)C(C)(C)Oc1ccccc1)NC(C(CC)n1cncn1)=O C1(NC(C23CC(NC(c4c(C)ncs4)=O)(C2)C3)=O)C2Cc3ccc(Cl)cc3C12 Cc1ccc(CCN)s1.O(NC(=O)C1(CCF)CCC1)C(=O)C(F)OC(F)(F)F C1(CNC(c2cc(C(C)C)on2)=O)CN(C(C2CCNC2=O)=O)CC1(F)CO CC(C)CC(C)(O)C(=O)N1CC(C(N)=O)(CNC(=O)CC2Cc3ccccc3O2)C1 C1(NC(C=COCC)=O)CCN(CCNC(=O)Cc2ccccc2OC(C)=O)CC1 C12(CC)CN(C(c3c(COC(C)(C)C)c(C)nn3C)=O)C(CNC(=O)OC)(C1)C2 S(=O)(=O)(c1ccc(C#N)cc1)N(CC(=O)Nc1cc(OC)cc(OC)c1)C Cc1ccc(C)c(C(=O)NC2CCN(C(=O)COC3CC=CC3)CC2C)c1 CC1CN(C(CN(C)CC2CCN(C(=O)CN3CCC(O)CC3)C2)=O)CCO1 CC(CCCCCO)NC(C1CC(O)CCN1C(c1cn(C)nn1)=O)=O c1(C(=O)NC2CCC(CNC(C(C)OCCCC)=O)C2)ncccc1O Cc1cccc2cc(C(N3CC4CC(C3)CN(C(=O)C(C)C3CC3)C4)=O)nn12 C(=O)(CC(C)C(C)(C)CC)NC(CCCNC(C1(CCC)CC1)=O)CCC N1(C(Cn2c(C)c(Cl)cn2)=O)CC(F)(F)CC1C(N1CCC(OC2CCC2)CC1)=O CCC1=NOC(CC(N2CC(CC(C)NC(c3nc(=O)n(C)[nH]3)=O)C2)=O)C1 CCCCC(C(=O)NCCN(C)C(=O)OCC)NC(=O)C1CC1 CCCC(CNC(C1(OC)CCOC1)=O)C(=O)NCCC(C)O c1(C(N2CCSCC2)CC)cccc(C(F)(F)F)c1F.C12CCN(CC1)C(=O)N2 c1(-c2cnc(COC)c(C)c2)ccc2[nH]cc(C(=O)Nc3n[nH]cc3Br)c2c1 CC(O)(C(=O)N1CCCC(C(N2CCC(C3OCCO3)C2)=O)C1)C(F)(F)F c1(CN(C(C2CCCO2)CC)C(c2csc(=N)[nH]2)=O)ccccc1C C1(C(N2CC(O)(C(=O)OC)C2)=O)CC=CCN1C(=O)CN1CCNC(=O)C1 n1(C(CC)CC)ccc(C(=O)N(C)CC2CCN(C(=O)Cc3csc(S)n3)C2)n1 c1(N2CCCC(NC(C3CCN(CC)CC3)=O)CC2)nc2ccc(O)cc2s1 N=c1ccc(CC(=O)NC2CCCC2NC(c2ccnn2CCF)=O)c[nH]1 N1(C(C(CC)CN(C)C)=O)CC2CCCC2(C(=O)NCC(c2ccncc2)C)C1 C1(CC)(CC)CC(C(=O)NCCCOC)C1.C(C)(C(=O)C1CCC1)OCCNC(N)=O C1(C(=O)NCCC2(O)CCN(C(C(CC=C)C)=O)C2)(OC)CCCCCC1 n1(CC(N2CC3(C2)CN(C(c2cncc(F)c2)=O)C3)=O)ccc2cc(Cl)ccc12 N1(C(COCCCC)=O)CC(O)CC1C(=O)N(C)Cc1cc(C)no1 C(=O)(C(C)(C)CCCF)N1CCC(C(N(C(C)C(=O)OC)CCC)=O)CC1 N1(C(=O)C=Cc2cn[nH]c2)CCN(C(c2c(F)cccc2F)=O)CC(CO)C1 c1(CC)nnc(O)c(C(N2CCN(C(C3CCSC3)=O)CC(O)C2)=O)c1CC C1(C(C)C)CCC(C(=O)NCCSCCCO)N1C(=O)CC1COC(=O)C1 C1(NC(C2(NC(C(C)OC)=O)CCCC2)=O)C2CCN(CC2)C1C N1C2CCOc3cc1ccc32.C1(c2nnc(C3CC3)o2)(OC)CCCCC1 c1(C(=O)NCC(CNC(C(C)(C)C2CCOCC2)=O)CO)cc2ccccn2n1 c1(C(=O)NCCCC2N(C(C(C)SCC)=O)CCC2)cccc([N+](=O)[O-])c1C C1(C(N(CC#C)CCO)=O)CN(C(=O)COCC2CCOC2)CC1C N1(C(c2c(C)ccnc2)=O)CCC(C)(C)CC1C(N1CCCCCCC1)=O C1(CNCC(=O)NCC(c2c[nH]c3ncccc23)=O)CCC2(CC1)OCCO2 CCCCC(O)C(=O)N(C1CN(C(=O)Cc2cnccc2C)C1)CC c1(C2(C)CC2C2CCCCC2)nc(CN2CCC(O)CC2)nn1-c1ccccc1 N1(C(CC=C)=O)CCC2(CC1)CN(C(c1cc(=O)c3ccccc3[nH]1)=O)C2 N1(C(C2(C(C)(C)OC)CC2)=O)CC(NC(=O)COC2CCCCCC2)C(C)C1 C(C(=O)N1CCC(O)(CN(C(=O)C(C)(F)F)C)C1)(C(C)C)NC(CC(C)C)=O c1(C(=O)NC2(CO)CCCN(C(C(C)(C)SC)=O)C2)ccc2cc(F)ccc2n1 C1(NC(c2cncc(N)n2)=O)CCN(C(C2CN(CC(F)(F)F)C2)=O)CCC1(F)F N1(c2c(C)c(NC34CC(F)(C3)C4)ncn2)CCC2CCCC2CC1 C1(C(C)C)COCCN(C(=O)COC(C)(C)CNC(=O)COC(C)(C)C)C1 C1(CC(=O)NCCP(C)(C)=O)CC2(C1)CN(C(c1csc(Cl)c1)=O)C2 N(C(=NCc1ccccc1)NC1CCC(C(F)(F)F)CC1)CC.N12CCC(C1)C2 S(=O)(=O)(c1ccc(NCc2ccncc2)nc1)N1CC(CC)SCC1 N1(C(c2c(O)ncc(CC)c2)=O)CCC(C)(C)C(NC(=O)C#CC(C)(C)C)C1 C12(NC(C=C(CCC)C)=O)CCC1CN(C(=O)CCSCCC)C2 C1(CCC)CN(C(=O)C(C)CSC)CC1NC(c1oc(C2CC2)nc1C(F)F)=O C1(NC(C2CC2(Cl)Cl)=O)C2CC(NC(C3CC(O)CN3C(N)=O)=O)CC12 CCCC(C)(O)C(=O)NCCN(C)C(c1cc(OC)cnc1F)=O c1(C2(C(=O)NC(c3cccc(-n4cccn4)n3)C)CCCCC2)ccc(Br)cc1F C(c1ccncn1)=CC(=O)NC1CC1.N12CCCC1CNC(=O)C=CC2=O N1(C(CN(c2ccnc(Cl)n2)C)=O)CCOC(CNC(=O)CCc2nccs2)C1 c1(NC)ccc(Cl)c(C(=O)N(C)CC2CCCN2C(c2ccc(CO)o2)=O)c1 C1C=CC(N=c2cc(C)[nH]c(=NCC3CC3)[nH]2)C1.C1(CC)CC1(C)C C1(NC(CN2CC(C)(OC)C2)=O)CC=C(C(=O)NCCN2CC(C)(O)C2)C1 C=CCCCCCCCC(=O)NC1(CC=C)CCN(C(C2C(Cl)(Cl)C23CC3)=O)C1 c1(C(N2CCN(C(C34CC3CCC4(F)F)=O)CC2)=O)cc2c(Cl)cccc2s1 Cc1cc(C(N2CC3CC2CC3NC(c2csc(Cl)c2)=O)=O)cc(O)c1 C1(NC(C(CC)OC2CCCC2)=O)CC2CCC1(NC(=O)C1=CSCS1)C2 C1(O)(CNC(CCc2n(C)ccn2)=O)CCCN(C(=O)Cc2ccccc2O)C1 c1(OC)sccc1C(=O)NCC(C)NC(=O)CNC(C1CC1C(N)=O)=O c1(NCCN(CCOC)Cc2cccnc2)ccnc(-c2ccccc2)n1 C1(NC(C(=O)NCC)=O)CCC(C)(CNC(=O)Cn2nnnc2C(C)C)C1 C(=O)(C1CCc2c[nH]nc21)NC1(CC(=O)NCCN2CCS(=O)CC2)CCC1 N1(C(c2ncc(C)cc2F)C(=O)NC(CC)(C)C)CCC(C2(C)CC2)C1 C1(C(=O)NOCC(=O)N(C)C)CCN(C(c2cc(Cl)c[nH]2)=O)C1C(C)C.CO C1(C(=O)NC2CN(C(c3cn(CC)nn3)=O)CC2C)COc2ccccc2O1 CC(C)(CNC(=O)OC(C)(C)C)C(=O)NCCCNC(C1CNC(=O)C1)=O CCC(C)C(C(=O)N(CCC(C)NC(C1CCCN1S(C)(=O)=O)=O)C)NC(C)=O c1(CC)n[nH]c(=NC2CCCC(NC(=O)CC3(N(C)C)CC3)C2)o1 C1(CNC(CC2CCN(C)C2=O)=O)CN(C(=O)Cn2cnc(=N)[nH]2)CCC1(C)C C1(CC=C)(C(=O)NCC(O)CC)CCN(C(=O)CCc2nccn2C)C1 N1(C(CS(CC)=O)=O)CCOC(C)C1C(=O)N(CC(C)O)C C1(N(C(CSCCC)=O)C)CCCCN(C(c2ccc(OCC)cc2)=O)C1 c1(CC(=O)Nc2cn(C)nc2OCC(F)(F)F)nc2cnccc2[nH]1 c1(C(N(C2CCCN(C(C(COC)O)=O)C2)CCO)=O)ccc2n[nH]cc2n1 C(c1ccc(Cl)cc1F)=CC(=O)NC1(CNC(C(CC)OCC)=O)CCC1 C1(n2cc(C(COC)(C)O)nn2)CCC(C(=O)NC(C)C(C)n2cncn2)CC1 c1(N2C(COC)(CNC(=O)CCC3CCC(C)O3)CCC2)ccnc(OC(C)=O)n1 C1(NC(CCCN(C(c2cnc(CC)o2)=O)C)=O)CCN(C)C1(C)C C(C(C)(C)C(=O)N1CCC1CC1CC1)NC(CCCOCCC)=O C1(C(=O)Oc2nccc(=N)[nH]2)CCCC(O)C1.C12CCC(CC1)N2C(C)(C)C N1(C(C2C(c3c(C)cccc3)C2)=O)CC2CN(C(c3ocnc3C)=O)CCC12 c1(C(=O)NC(C2CCCN(C(CC(=C=C)C)=O)C2)C)ccc(F)c(NC(C)=O)c1 CCC(CC)CC(F)C(=O)NC(CC)CCC(=O)NCCCC1CCOC1 C1(C(=O)NCC2(C(=O)NC3CCN(C(=O)NC)C3)CC(=C)C2)CCC(O)C(O)C1 C(=O)(CS(=O)(=O)NC(C)(C)C)N1CC(OC)(CNC(=O)CC2CC(C)=NO2)C1 c1(C(=O)NCC(C)NC(CSc2cccc(OC)c2)=O)cc2ccc(C)cc2[nH]1 Cc1cccc(S(=O)(=O)N2CCC(O)(C(N3CCC(CO)CC3)=O)C2)c1 C1(CNC(C(=O)NCC)=O)(NC(=O)CCC2CCCCO2)CCCC1 c1(CC(=O)NCCn2cc(CNC(CSC)=O)nn2)nc(C)c2c(n1)CCCC2 c1(NCCN2CCC(NS(N)(=O)=O)CC2)cnn2c(Br)cccc12 CCC(C(=O)NCC(COC)OC)NC(C)=O.c12n[nH]cc1C(=O)N2 O=S(=O)(c1ccc(NCC2C3COCC23)c(Cl)c1)NC1CC(CCO)C1 C(C(C(C)C(C)C)NC(C1(CN(C)C)CC1)=O)NC(CC=C=C)=O c1(C(=O)NCCOCCC(=O)NCCC2CCC(C)O2)ccncc1F C1(NC(C2NC(=O)OC2)=O)(CNC(=O)CNC(=O)C(F)(F)F)CCCCC1 C(=O)(C(C)CCCC(C)C)NCC1(COC)CCCN1C(=O)Cn1cnnc1O CCCC(C)(C)CC(=O)N1CCC(CNC(=O)Cn2cnnc2)C(F)(F)CC1 N1(C(C2N(C(C)=O)CC(O)C2)=O)CCC(NC(c2cnc(S)n2C)=O)C(F)C1 c1(CC(=O)NC2C(NC(C(CC)=CC)=O)CCCC2)cc(F)c(N)cc1F n1(CC(=O)NC2CC(C(=O)NCc3cnc[nH]3)C23CCC3)cnc2ccccc12 C(=O)(C1CCc2c[nH]nc21)N1CCC(N(C(C(CC2C(C)C2)O)=O)C)CC1 C#Cc1cncc(C(=O)NC2CCN(C(=O)OC(C)(C)C)C2)c1 C1(C(=O)NC2CC(F)(CNC(C(CC)CC)=O)C2)CCc2nnc(C)n2C1 n1(CCC)cc(C(=O)NCC(F)CNC(=O)C(F)(F)C2(O)CCC2)nn1 Cc1cc(=NCCC2OCCC2(C)C)[nH]c(NCC2COCC2CO)n1 C(=O)(C(C)(C)CCCNC(=O)C(O)C1CCC1)NC1CCN(C)C1=O Nc1c(C(N2CCN(C(C3CC3CF)=O)C3CC23)=O)cccc1Cl c1(OC)cc(C(=O)NC(CNC(=O)C(O)CN2CCCC2)C(C)C)cc(N)c1O C1(NC(C(C)Oc2cccnc2)=O)CC2CCC(C1)N2Cc1ncc(C(C)C)o1 N1(C(CSCC)=O)CCCN(C(=O)CC2CC2CC)C(NC(=O)OC(C)(C)C)C1 C1(CC(=O)NC2C(NC(Cc3c(C)coc3C)=O)COC2)CC(C)(C)C(=O)N1 C12(NC(C3NC(=O)CC(C)C3)=O)CCCCC1CN(C(c1ncn(C)n1)=O)C2 C1(CC)COCC1C(=O)NCCN(C1CCCCC1)C(=O)CNC(=O)NC(C)C C(=O)(CCC(C(=O)N1CCC(=CCNC(c2cccc(C)n2)=O)CC1)N(C)C)OC N1(C(c2c(SC)csc2)=O)CCN(C(C2CCCCNC2=O)=O)C(CF)C1 CC(C)C(O)C(C)(C)C(=O)N1CC(CNC(=O)CCCc2ncco2)C(C)(C)C1 Cc1ccc(C)c(OCC(=O)NC(C)(C)C(=O)N2CCC3CC23)c1 c1(CC(=O)NC2C(NC(c3c(OC)cncc3)=O)CCC2)n[nH]c2ccccc12 N(C1c2ccccc2CC1O)C(C1(COC)CC12CCNCC2)=O c1(CC(=O)N(CC(C)(C)CNC(C2CC2C(F)(F)F)=O)C)ccc(O)nc1 c1(C(=O)NC2(CNC(=O)Cn3cnnc3)CCCC2)noc2cc(Cl)ccc12 C12(CNC(C3CC4(CCNC4)CO3)=O)CCCCC1OCC2 CC(=O)CCCC(=O)NCC1(C(=O)Nc2cccc(CO)c2C)CCCO1 N1(C(C2(CNC(C(C)c3ccco3)=O)CC23CCC3)=O)Cc2cncnc2C1 O=C1CCC(C(=O)N2CCCCC2CCCNC(=O)C(Cl)=CCl)c2ccccc21 C1(NC(C2(OCC)CCSC2)=O)CCCN(C(C2CC(=O)CCO2)=O)CC1 C1(C(=O)NCC2CC(NC(C3C(C(C)C)C3)=O)C2)CC2C=CCC(C1)C2 c1(C(=O)NCC2CCCN2C(c2ncncc2Cl)=O)ccnc2c1CCO2 Cc1cc(C(F)F)ncc1C(=O)NC1(C)CCN(C(c2nnsc2C)=O)C1 CC(C(F)(F)F)NC(C1CC1c1ccco1)=O C(=O)(C1=CCC(NC(C2CC2(C)C)=O)C1)N(CCCF)C C(C(C)(C(=O)NC1(C)CCSC1)NC(=O)Cn1cc(C#N)cn1)SC c1(C(=O)NC2CC(C)(NC(C(C)OC)=O)C2)cnc(OC(F)(F)F)c(Cl)c1 C1(NC(c2cc(O)nc(O)c2)=O)CC2CC1N(C(c1cc(CO)on1)=O)C2 N#Cc1ccc(C(N2CC3CN(C(c4cc(Cl)ccn4)=O)CC23)=O)cc1Cl C1(C(=O)NC(C#C)C(C)OC)CC12CCN(C(c1cnsn1)=O)CC2 c1(CC)ccc(C)c(C(=O)N(C2CCCN(C(=O)C(C)N3CC(C)C3)C2)C)c1 C1(OC)CC(CCNC(c2ccc(CO)nc2)=O)N(C(c2n[nH]c(C)c2F)=O)C1 N1(C(C=Cc2cccc(C)c2)=O)CCN(C(C2(O)CCC2)=O)CC2(C)CCCC12 C(=O)(C1=CCCC1C)NCCC1CC(C(=O)NCc2c(CC)nns2)C1 c1(CC(=O)NC2C(C)(C)CN(C(=O)CC3CC3(C)C)C2)cccc2cnccc12 c1(CNC(C(=O)OCCC)CSC(C)=O)cc(C)c(C)c(F)c1 C1(NC(C=CCCC)=O)C2CC3C1C3C2C(=O)NC1CC12CC(C)(C)C2 C1(O)(CNC(c2nc(C(C)C)oc2)=O)CCC(C)(C)CC1 C1(NC(c2nc(C(C)C)oc2)=O)CC2CN(C(C3(N=[N+]=[N-])CC3)=O)CC2C1 S(=O)(=O)(c1cccnc1NCC(CC)OC)N1CC(CCC)OCC1 CC1(C)C(CNC(C2(C(C)(F)F)CCOCC2)=O)CCS1(=O)=O C1(COC)CN(C(c2ccc(SC)cc2O)=O)CCN1C(C12CC(C1)C2)=O N1(C(C2(S(C)(=O)=O)CC2)=O)CCCC2(NC(C3(n4cncn4)CC3)=O)CCCC12 c1(C(=O)NCC(CC)NC(c2cnn(C)c2Cl)=O)cccc(-n2ccnc2O)c1 C1(CC=C)(NC(c2cn(C)nc2-c2ccoc2)=O)CCN(C(c2ncccn2)=O)C1 C(=O)(C1CNC(=O)c2ccccc21)NCC1CC2CN(C(C3(C)COC3)=O)CC21 C(=O)(C(F)(F)C(C)O)NC1C(C2CCN(C(C=CC=CC)=O)CC2)OCC1 c1(C(N2CC(O)(CCNC(C(C)(C)CC3CCC3)=O)C2)=O)ccc2ncsc2c1 C(=O)(C(C)(C)C(=O)N(CCCNC(C1CC(=O)N(O)C1)=O)C1CC1)NC c1(C(=O)NC(C(=O)N(CCOC)CC)C(C)(C)C)nn(C)c(C)c1Br N1(C(c2cnc(C3CC3)[nH]2)=O)CCN(C2CCN(C(C34CCC3C4)=O)CC2)CC1 C1(CCC=C)(C(=O)NC(C)C(C)O)CN(C(=O)COC2CC=CC2)C1 c1(CC(C)C)ccc(CN(C)C(c2coc(O)n2)=O)s1.N12CCCC1C2=O N1(C(C(c2cccc(O)c2)C)=O)CC(NC(C2CC(F)(CO)C2)=O)C(C)(C)C1 C1(NCC)CCC2(C(C)C)CC12.C1(C)(OC)CNC(=O)N1 C1(NC(c2ccc(C(C)=O)cc2)=O)C2CC(O)C1N(C(c1cnc[nH]1)=O)C2 C(C)(C)(CC(C)NC(=O)NC(c1ncc(C(F)(F)F)[nH]1)C)OC c1(C(=O)NC(CNC(c2cc(OC)ns2)=O)CO)cc(=O)c2ccc(Cl)cc2o1 C1(=CC(=O)NC(C)CNC(=O)Cc2cnco2)CCN(C)CC1 c1(C(=O)NC2CCC(F)(CNC(C(C(C)C)C)=O)C2)cc2n(n1)CCNC2=O C1(SCC)CCC(C(=O)NC23CC(CNC(c4cncn4C)=O)(C2)C3)CC1 C(CCN=C(NCC(N1CCCCC1)(C)C)NCC1(S(C)(=O)=O)CCC1)SC N1(C(C2(C)COCC2(F)F)=O)CCOC2(CCCN(C(C34CC(F)(C3)C4)=O)C2)C1 C(=O)(C(CCc1ccccc1)C(C)C)NCC(CNC(CCSC)=O)F S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1C(CC(N2CCC(C)(O)CC2)=O)CCC1 C(CC(CO)NC(=O)Cn1cc(CNC(c2cc(C)cs2)=O)nn1)=CC C1(O)(CNC(C2N(C=O)CCC2)=O)CCCN(C(c2cnnn2C2CC2)=O)C1 N1(C(C(F)=C(C)C)=O)CCC2(CC1)OCCC2NC(C1CCCC(F)(F)CC1)=O C(=O)(C1c2ccccc2C2CC1C2)NCC(C)N(C(=O)CC1CC1(C)C)C C(=O)(C#CC(C)(C)O)NC1C(NC(CSc2c(OC)cccc2)=O)C1 O=C(CCC(=O)c1cccs1)NCC1(NC(=O)C=C2CCCS2)CC1 CCC(C(=O)OC)C(=O)NCC(C(N1CC(OC)C(F)C1)=O)OC C#CCC(C(=O)NCc1nn[nH]n1)NC(C1CC1C(F)(F)F)=O N1(C(c2c(C)cncc2)=O)CC(NC(C2(N3CCOCC3)CC2)=O)CC2(CC2)C1 Cc1cc(Br)c(CN2CCNCC2C(=O)Nc2c(C)ccnc2Br)cc1[N+](=O)[O-] c1(OC)cc2nc(NC(c3cc(I)cnc3O)=O)[nH]c2cc1OC C1(NC(c2cc(C)c(F)nc2)=O)CN(Cc2c(F)cc(F)cc2Br)CC(F)(F)C1 N1(C(c2nc(C)oc2C)=O)CC(O)C(O)C1CNC(=O)CC(C)F c1(C(=O)NC(CNC(C2CCC(CCC)CC2)=O)C)c(C)nn(C)c1F c12nnc(s1)CCN2.FC1(CCF)CC1 c1(C(N2CC(C(C)NC(CNC(CC)=O)=O)OCC2)=O)cnc2ccncc2c1 N1(C(=O)NC2C(CCC)CC(OCC3CC3)CC2)CC(F)(F)CC1(C(C)C)CO CN=c1nc(C(=O)NC2(CO)CCCN(C(c3cc(C)c[nH]3)=O)C2)cc(C)[nH]1 C1(CNC(C2(CC#C)CCCCO2)=O)COCCN(C(c2c[nH]cc2C)=O)C1 Cc1cnn(CCC(=O)N2CC(OC(C)=O)C2)c1.C1CC(=O)N(C)CCO1 N1(C(c2[nH]cc(C)c2C)=O)C(C(=O)NCc2nnn(C)n2)CC2CCCC12 n1(CC)ncc(C(=O)NCCC2CCCN(C(=O)CCc3cncnc3)C2)c1C C(C)(C(=O)N(C1CC(NC(=O)COCCCF)C1)C)SC c1(C(N(CCCN(C(C(CC#C)C)=O)C)C)=O)cc(OC)cc2c1OCC2 c1(OCCC(=O)N(C2CCN(C(c3ccsc3C(F)F)=O)C2)CC)ccccc1 C#CCC(CC#C)C(=O)NCCCCCCNC(C1CC1c1cccc(C)c1)=O CC1CCCCC1(CNC(c1ccc(Cl)cn1)=O)NC(=O)COCC1CCC1 c1(NC(C2C(NC(c3cn(C)nc3)=O)C2)=O)nc2cc(F)ccn2n1 Cc1cc(O)nnc1C(=O)NCC=CCNC(=O)CCn1cnc([N+](=O)[O-])c1 N1(C(C(=O)NCCCC)=O)CC(C)C(C)(CNC(=O)CC(C)NC(C2CCC2)=O)C1 N1(CC)CCCC(CN2C3CCN2C3)C1.C1(=O)C(CC)N(CC)N1.C(=O)OCC.CC C(=O)(CCN=c1[nH]ccs1)N1C2CC(NC(CCn3c(C)csc3=O)=O)C2CC1 c1(C(=O)NC(C)CCN(C(=O)C(C)C2CCCC2)C)cc(Cl)c(F)cc1O c12sc(C)c(C)c1N2.C1(C(=O)NC(C2CCOC2)CNC(C)=O)CCOC1 C1(C)(C2CC2)CNC(=O)N1.C1(C(C)(C)C)CC(Cc2ccco2)C1 C(C)(CN=c1[nH]cnc2ccc(F)cc12)N(C(C(CCC)NC(N)=O)=O)C C1(C(=O)NC2CCN(C(c3ccn(CC)n3)=O)CC2)Cc2c(F)cccc2O1 C1(NC(=O)Cn2nc(Cl)ccc2=O)CC2CCC1CN(C(=O)CC1C=CCC1)C2 C(=O)(C(C)(C)CNS(C)(=O)=O)NC1CC(NC(C2(C(F)(F)F)CC(=C)C2)=O)C1 c1(CC)cnc(CN2CCC(C(N3CCCC(O)C3C)=O)CC2)[nH]c1=NC c1(C(=O)NCCC(=C)CNC(C2CC2c2cccnc2)=O)cc(OC)cc(F)c1 C1(CC(=O)N(CCCC#C)C)CCN(C(=O)CCC2CCCOC2)C1 c1(CC(C(=O)OC)NC(C(=O)NCCC(COC)(C)C)C2CC2)ccc(Cl)cc1Cl C1(CNC(C2CC2C(F)(F)F)=O)CCCCN(C(c2cc(Cl)cnc2O)=O)CC1 C(=O)(CCCN=[N+]=[N-])NCC1(OCC)CN(C(=O)C2=C(Cl)CCC2)C1 c1(OC)c(C(=O)N(C2CCN(C(C3CCCN(C)C3)=O)CC2)C)csc1C c1(CNC(=O)NC2(CN3CCCC3)CC2)cn(CC2C3COCC23)nn1 c1(CC(N2C(CCCNC(C(F)OC)=O)CCCC2)=O)cnn2ccccc12 C1(CNC(=O)CN2CCNC2=O)(CO)CCN(C(=O)CCC2CC2)CC1 C1(C)(C(N2CCN(C(C3=CC(C)(CC)C3)=O)CC2COC)=O)CCC(C)(C)CC1 C(=O)(CCC1CC(NC(c2cnco2)=O)C1)N(CCC)CC1CC1 C(CCN=c1cc[nH]cc1S(=O)(=O)N1CCCCC1c1nncs1)SC.C1CO1 CON1CCC(CC(=O)NCC2CCN(C(=O)Cc3ccc(Cl)s3)C23CC3)CC1 c1(C(C)(F)F)csc(NC(=O)NCCOC2(c3ccccc3)COC2)n1 C(CC(N)=O)(C(=O)N1CCNC(=O)C1C)NC(COCC(C)C)=O CC1CCN(CCCO)CC1NC(C1CCN(C2CCNCC2)CC1)=O N1(C(C(C)=O)=O)CC(NC(=O)C(F)(F)CC2CC2)CCC1C C1(NC(C2(C(=O)NC3CC3)CC2)=O)CC2(C1)CN(C(c1onc(C)c1C)=O)C2.CCO c1(C(N2CCC(CNC(C3(CF)CC4(CCC4)C3)=O)C2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 C(CN=C(NCC1CCCCC1)N1CCN2C(=O)CCC2C1)N1S(=O)(=O)CCC1 C1(CNC(CNS(CC)(=O)=O)=O)CC2CCC1N(C(c1cc(N)cc(O)n1)=O)C2 CC(=O)CCCC(C)(C)C(=O)NC(C1CCCN1C(C1CCCC1C)=O)C C1(NC(CCC2N(C(c3cc(C)cc(C)n3)=O)CCC2)=O)CCCCC12CCC2 C1(C(=O)NCCCN(C(c2ccccc2)=O)CC)CC(C)CC(C)C1 c1(CC(N2CC3(C(C(=O)NCCCCCO)C3)C2)=O)cccc(Br)c1F O=C(C(O)CC(F)F)NCc1ccccc1-n1cc(C2(O)COC2)nn1 c1(C(N2CCC(CNC(C3(C)CC(=C)C3)=O)C2(C)C)=O)cnc2ccoc2c1 C1(NC(CC2C(C)=NNC2=O)=O)CC2(CCN(C(=O)Cn3ccc(C)c3C)C2)C1 c1(-c2cn(CC3N(C(C4(C(C)C)CC4)=O)CCOC3)nn2)ncnc2sccc12 c1(CCC)cc(C(=O)N(CCNC(C2CSCN2C)=O)C(C)C)no1 C12(NC(C3CCN(C(=O)OC(C)(C)C)C3)=O)CNCC(F)(C1)C2 N1(C(c2c(C)oc(C(C)C)n2)=O)CCC(NC(=O)C=C2CCCC2)CC1C c1(CC(=O)NC(C(=O)NCC(C)(C)F)c2cccs2)ccccc1C#N C1(C(N(CCN(C(C(CSC)OC)=O)C)C(C)C)=O)CC2CC1CC2(F)F c1(C(=O)NC2(C3CN(C(c4cccc(OC)c4)=O)C3)CC2)ccccc1[N+](=O)[O-] c1(C(=O)NCCCN(C(c2nc(C)ccc2C)=O)CC)cccc2oc(O)nc12 C1(C)(COC)CC(NC(=O)CC(F)F)CN1C(=O)CC1(C)OCCO1 C(=O)(C(C)CS(C)(=O)=O)N1CC(F)(CNC(C(C)CCc2ccccc2F)=O)C1 C12(C(=O)NC3(CNC(CCc4ncn(C)n4)=O)CCCCC3)COCC1C2(F)F C12(NC(CS(=O)(=O)NCC)=O)CCC(CN(C(C3CCCS3(=O)=O)=O)C1)C2 N1(C(Cc2ccn(C)n2)=O)CCN(C(C2CCCC2)=O)C(c2nccn2C)C1 N1(C(c2cncc(F)c2)=O)CCC2CN(C(c3nc4ccccc4s3)=O)C2C1 c1(C(N2CC(N(C)C(c3cnncc3O)=O)C(O)C2)=O)cccc(F)c1F C1(O)(CNC(C(C(C)C)c2ccccc2)=O)CCN(C(=O)Cc2ccsc2)CC1 c1(OC)ccc(C(=O)N(CCCNC(C2(NC(C)=O)CC2)=O)C)c(C)c1C C1(COC)(NC(=O)C(c2ccc(OC)nc2)C)CCN(C(=O)COCC(F)F)C1 C(CN=c1[nH]c(CC(C)C)nc2cc(C)ccc12)=CC N(C1CCc2cc(C#N)ccc21)Cc1cc(C)c(OC(C)C)cc1 C1(NC(C(CC)C(C)C)=O)CCN(C(=O)C(=Cc2ccccc2Cl)C)C12CCC2 c1(COC(c2c(Cl)ccc(C)c2)=O)cn2cc(Cl)cc(C)c2n1 C1(OC)C(NC(=O)C(Cc2ccoc2)NC(c2cnn(C(C)C)n2)=O)CC1O c1(CONC(N2CCCC2Cc2ccc(F)cc2)=O)cc(F)cc2[nH]ncc12 C(CC(C)C)(C(=O)NCC1(F)CC(CNC(=O)C(C)C2CC2)C1)NC(C)=O CC1=CC(C)CN(C(C2(NC(C3COCC3(C)C)=O)CCC(C)(C)C2)=O)C1 CC1(C(N2CCC(CNC(=O)C=CCF)C2)=O)CCCC(F)(F)C1 C(=O)(C1CCCn2nccc21)NCC(C)CNC(c1ccnn1CC(F)(F)F)=O N1(C(CC=C(C)C)=O)CC(NC(=O)C(C)CC(F)(F)F)CC(C)(C)C1 C(=O)(CCCC(=O)NCC)NC(C1CCCC1)CNC(CC1(C(=C)F)CCC1)=O c1(C(=O)NCC(CNC(=O)CC2(O)CCC2)O)occc1COc1ccccc1 c1(C(N(CCc2cccc(OC)c2)C)=O)c(C)oc2ncn(C)c(=O)c12 N1(C(CCS(C)=O)=O)CC2(CCOCC2)CC1CNC(c1cc2ccsc2s1)=O c1(C(c2nnnn2CCN(C)C)NC2CN(C(C)=O)C2)cc2cccc(Br)c2o1 C=C1CC(C)(C(N2CCCC2CCC(=O)NCCCOC)=O)C1 N1(C(c2c(C)cc(N)cc2)=O)CCn2c(CNC(=O)CC(C)C(C)C)nnc2C1 N1(C(C(C2CCC2)OC)=O)CC2C(CNC(=O)CN3CCC(F)(F)C3)C2C1 C1(CNC(C(C)SCCCC)=O)CC(O)CN1C(=O)C(C1(O)CCCC1)F c1(CC(N2CCC(CN(C(C3CC3(Cl)Cl)=O)C3CC3)CC2)=O)ccc(CO)cc1 c1(C(=O)NCC(C)(C2CCC2)NC(c2c(C)ccnn2)=O)ccc2nncn2c1 N1(C(C2C(O)CN(C(c3nc(C)sc3)=O)C2)=O)CCC2(CCC(=O)NC2)CC1 Cc1cn2c(n1)C(C(=O)NCC13CCC(CC1)N3C(c1ccns1)=O)CCC2 C1(NC(Cc2cn(CC)nc2)=O)CN(C(c2cc3sccc3s2)=O)CCC1CO Cc1cnc(C(C)NC(=O)C(C)(C)CN(C(=O)CN2CC=CC2)C)nc1 c1(C(=O)NC2CN(C(c3c(OC)nsc3)=O)C(C)C2)cnn2ccn(C)c12 c1(CNC(C(C2CCCC2)NC(Cc2c(C)ocn2)=O)=O)nn(C)cc1CO C(=O)(C1=C(C)OCCS1(=O)=O)NCC(CNC(C=Cc1ccc(CC)cc1)=O)O C1(C(=O)OC)CCOC(CNC(c2ncccc2OCC(F)F)=O)C1 C(C)(CC(=O)NCC1(O)CCN(C(C2CCSCC2)=O)CC1)(C(F)(F)F)N(C)C N1(C(CSCC)=O)CCC(C2CC2)C1C(N1CC2(CCC(=O)N2)C1)=O N#Cc1ncn(CCC(=O)NCCC2CCN(C(C3CC(O)C(F)C3)=O)CC2)n1 c1(C(=O)NC2CCC(NC(=O)CCc3cnoc3)C2)ccnc(C(F)(F)F)c1 c1(C(N2CC(N(C(C(C)=C3CC3)=O)C)C(O)C2)=O)cc2c(O)ncnc2cn1 C12(CNC(C(CC)(C)OC)=O)CCC1CN(C(c1ccc(C(=O)OC)s1)=O)C2 C(=O)(C1=NOC2(CCN(C(=O)OC(C)(C)C)C2)C1)N1CC(CC)CC(F)(F)C1 N1(C(C(CCCC)C)=O)CCC2(CCCC2NC(c2ccc(F)cn2)=O)CC1 C(C1C(C(N2CC=CC(NC(c3cn(C)nc3O)=O)C2)=O)C1(C)C)=C(C)C C(C)(c1ccccc1)=CC(=O)NC(CC=C)CNC(=O)CC(C)n1ccnc1 N1(C(c2cc(OC)n(C)n2)=O)CCC2(NC(c3cnccn3)=O)CC2C1 N1(CC(=O)N(CCC#N)CC)CCN(C(c2c(C)noc2CC2CC2)=O)CC1 CC(CC(=O)NC1C=CC(CC(=O)N(C2CC3(CCC3)C2)C)C1)C(C)(C)C c1(OC)ccccc1CC(C)(C)C(=O)NCCNC(=O)C(C)Cn1ccc(C)n1 N1(C(c2cc(C(C)C)sc2)=O)CCC(C)(C(=O)O)CC1 c1(OC)ccc(Br)c(OC)c1C(N1CCCC1CNC(C1CC(O)C1)=O)=O c1(CNC(C(C(C)C2CC2)NC2CN(C(=O)OC)C2)=O)ccc(F)c(F)c1 Cc1cc(C(=O)NCC(CC(=O)NC(C)Cc2nc[nH]n2)C2CCC2)c(C)[nH]1 c1(C(=O)NCCN(C(=O)CC2CCCC2(F)F)CC)cc(O)nc2c1CCCC2 N1(C(COC(CC)C)=O)CC(F)(F)CC1CCNC(=O)Cc1cnc(C)[nH]1 C1(CNC(COc2cccc(OC)c2)=O)CN(C(c2cncn2C)=O)CC12CCC2 C1(C(=O)NCC(CNC(c2c(C)snc2)=O)C)CN2CCN1C(C)C2 c1(CC(=O)NCC2C(CNC(=O)CCCCN3CCC3)C2)cc(F)ccc1F c1(SC)ccsc1C(=O)NCC12CC(NC(=O)C(C)=CC(C)(C)C)(C1)C2 N1(C(c2c(C)nn(CCO)c2)=O)CCC2CN(C(C3CC(F)CN3C)=O)CC12 C1(F)(C(=O)NCC(CCC)(C)C)CCCN(C(=O)CC(=O)NCC)C1 c1(CC(N2C(CNC(CCC(C)COCC)=O)CCCC2)=O)ccc(F)c(Cl)c1 C1(C)(CC)C=C(C(=O)N2CCOC(CCNC(C3C(O)C4CCOC34)=O)C2)C1 C1(CC=C)(C(=O)NCCC(O)C2CCC2)CCCN1C(c1cncs1)=O C=CC1(C(N2CCC(C(C)C(=O)N(CCOCCO)CC)CC2)=O)CCOCC1 C1(C(=O)NCC(C)NC(c2ccc3n[nH]cc3c2F)=O)Cc2cc(F)ccc2O1 CC1(C#N)CCN(C(c2cc(-c3cccnc3)ncn2)=O)C1 C1(C(N2CCC(NC(CC3CC(OC)C3)=O)CC2C)=O)CCn2c(O)nnc2C1 N(C(=NCc1cccc(Cl)c1)N1CCCC(NC(=O)NCC2CC2)C1)C(C)C CC1CN(C(C2(CN(C)C)CCOCC2)=O)CCC1NC(c1cc(C#N)on1)=O CCCCC(C)CCC(=O)N1C2CCC1CC(NC(C1(CC(F)F)CC1)=O)C2 c1(C(=O)OC)[nH]c(C)c(C(=O)NC2CC(NC(c3nn(C)cc3Cl)=O)C2)c1C C=CC(C)C(C)C(=O)NCCCNC(C1(n2cnnn2)CCCCC1)=O C1(NC(COCC)=O)CN(C(=O)CCCc2nc3ccccc3o2)C2(CCC2)C1 c1(CN(S(CC)(=O)=O)C(=O)CCOCCCO)csc(S)n1.C12CCN1C2 c1(C(=O)NCCC(C)NC(CC(COC)C)=O)ccc(OC(F)(F)F)c(Cl)c1 N1(C(c2ccn(CCC)n2)=O)CCN(C(=O)C#CC(C)(C)O)C(C)C1 c1(C(N2C3C(C(=O)Nc4cccc5c4CCC5)C(C3)C2)=O)cccc2ccncc12 N1(C(CCSCC)=O)CCN(C(=O)C(C(C)C)N(C)C)CC1CCOC Cn1cc(CCNC(C2(c3cccnc3)CCCC2)=O)c(Br)n1 C(=O)(C(C)(CC)OC)N(C(CNC(c1cc(C(C)=O)sc1)=O)C1CC1)C N1(C(C2(O)CC(C)(C)C2)=O)CC(CNC(=O)Cc2cnn(C3CC3)c2)C2(CC2)C1 c1(C(=O)NCC(CNC(C(CCOC)OC)=O)C)cccc(F)c1F N1(C(c2cn(CC)nc2C)=O)CCN(C(=O)C2=C(Cl)CCC(C)C2)C2(CCC2)C1 C1(C(N2CCC(OCC=C)C2)=O)CN(C(=O)CC2(CSC)CC2)CC1(F)F CC(C)C(O)CC(=O)N1CCOC(C)(CNC(=O)C(C)(C)c2cscn2)C1 C(=O)(CCC(CC)NC(c1ccc(F)cn1)=O)NC(C=C)(C)CC C1(NC(c2cn(C(C)C)nc2)=O)CCN(C(C2CC(C)CO2)=O)C1C(C)(C)C CC(C)CN=C(NCc1sccc1Cl)N1CCC2(O)CCOCC2C1 C#CC(C)(C)C(=O)NCC(CC)NC(=O)C=Cc1ccc(N(C)C)o1 C1(C(=O)NCC(C)(CC)NC(CC2(C=C)CC2)=O)CN2CCC1(C)CC2 Cc1ccc2scc(C(N3CC(O)(CN(C)C(c4cc(Br)co4)=O)C3)=O)c2c1 CC1=C(C(=O)NC2CC(F)CN(C(C3CC3(C)C(C)C)=O)C2)S(=O)(=O)CCO1 CCCCCCC(C)C(=O)NC1CC(C(N2CCOC(COCC)C2)=O)C1 CN1CCS(=O)(=O)CCC1C(=O)NNC(=O)NCc1ccc(F)cc1 c1(NC)cncc(C(N2CCCC(N3CCCC3=O)C2)=O)c1 N1(C(c2c(COC)ncs2)=O)CC(NC(c2ccc(=O)oc2)=O)C2CCCCC12 N1(C(c2c(C)con2)=O)CCCC(C(N2CCN(C(=O)C(CO)N(C)C)CC2)=O)C1 c1(CN(C(C2CCN(Cc3cccc(C(F)(F)F)c3)C2)=O)CC)ccc(OC)cc1 c1(C(=O)NCC(N(C)C(C2CC2F)=O)C2CC2)cncc(C2CCOCC2)c1 N1(C(C(C(C)C)C)=O)CCC2CCN(C(=O)CSc3ccccc3)C2C1 Cn1nc(C(F)(F)F)c(Br)c1C(N1CCCC1Cn1cc(COC(=N)O)nn1)=O N1(C(C2CC(C(F)(F)F)(OC)C2)=O)CC(NC(=O)Cc2sccc2C)CC(O)C1 C1(C(=O)NCCCCNC(c2cc(-c3ccco3)no2)=O)CCC2(CC1)CC2 C(CC(C)C(=O)NC1CCN(C(c2cnn(C3CC3)c2)=O)C1)=CCC c1(CC(=O)Nc2noc(C(=O)OCC)c2C)ccc2n[nH]cc2c1 c1(CNC(c2n[nH]c(C)c2C)=O)cccc2c1CCN(C(C1(C)CC1Br)=O)C2 c1(C(=O)NC(CC=C)CNC(C2(C(=O)OC)CC2)=O)cc(COC)c(C)s1 N1(C(Cc2c(C)ncc(Cl)c2)=O)CCCN(C(c2cccs2)=O)C(CO)C1 n1(CC)nnc(C)c1N1CCCC1c1ocnc1C(F)(F)F C1(NC(C2CCCN(C)C2)=O)CC2C1CCN2C(c1ccn(CC(F)F)n1)=O C(N=c1[nH]c(=NC2CC3(CC(C)C3)C2)[nH]c2c1CSC2)C1CCC(C)CC1 N1(C(C(C)Sc2cccnc2)=O)CCC2CCC(C1)N2C(=O)CC(F)(F)F N1(C(Cc2ccc(CC)cc2)=O)CCCCC2(C1)CN(C(C1CCC1(F)F)=O)C2 C(=O)(CC(C(F)F)NC(c1ccc(OC)nn1)=O)NCP(OCC)(C)=O c1(NC(=O)NC2C(CC)CN(C(=O)OC(C)(C)C)C2)cc(Cl)c(Cl)n1C C(C(CNC(=O)COC(=O)CO)S(C)(=O)=O)NC(CCc1ncn(C)c1)=O c1(OC)cc(C(N2CC(O)(CNCc3cnc(Cl)nc3)C2)=O)ccn1 CC(C)CC(C(=O)NC(C(=O)N(C)C)C(C)c1ccccc1)C(N)=O c1(OC)cc(Br)c(CN2CCC(C(=O)Nc3cccc(C(N)=O)c3)C2)cc1O C1CCCC(=O)N1.c1(CC)[nH]ccc1C(N1CCC(c2ncc[nH]2)C1)=O N1(C(CCc2c(C)noc2C)=O)C2CCC1CC(C(N1CCC(C#N)C1)=O)C2 c1(CC)cccc2[nH]c(C(=O)NCC(C(C)C)NC(C3CC(F)C(=O)N3)=O)cc12 CC1CN(C(=O)Cc2ccccc2)CCN1C(=O)Cc1cnc[nH]1 N1(C(=O)COC2CCCOC2)CC2CCN(C(c3cc4c([nH]3)CCCC4)=O)C2C1 CCC(C)(C)CC(=O)N1CCOCCC1C(=O)NC1CC(=O)N(O)C1 C1(C(=O)NC(C)CNC(c2cc(F)ccc2Cl)=O)CCc2ccccc2O1 C12(C(=O)NC3C(NC(=O)CC4CC=CC4)CCCC3)CCC(=O)N1CCS2 C#Cc1ccc(OCC(=O)NC2CN(Cc3ccns3)CCCO2)cc1 c1(C(N2CC3(CN(C(=O)CCc4nc[nH]n4)C3)C2)=O)cc2ncccc2o1 c1(CC(=O)NCCN2CCCC2)cncc(O)c1.C(=O)(CC(=O)NCCCOC)NC CCC(C(=O)OC1CCCC1)SC(=O)Nc1nc(=N)[nH][nH]1 N12CC(F)CC1CC1(CC(C)(C)C1)C2=O.Cn1cnnc1CNCc1ccccc1 CC12CN(C(c3ccccn3)=O)CC1CN(C(C1(C#N)CC13CCOCC3)=O)C2 C1(C(=O)NCC(C2CCC2)NC(=O)CCOCC2CCC2)CCCC(C)(C)O1 c1(C(=O)NCC(CNC(C(CCC#C)O)=O)CO)ccc2oc(O)nc2c1 C1(CC)CCCC(NC(c2conc2CNC(=O)COC2CCOC2)=O)C1 N1(C(C2CCCN(C)C2)C(=O)Nc2ccc(F)cc2)CCCC2(C1)N=N2 C1(C)(C(=O)NCC(C(C)C)NC(C2(CO)CCCC2)=O)CCC(=O)NC1 C=CCC(C)C(=O)N1CC(NC(=O)Cc2ccc(C)cc2)C(O)C1 c1(C(N2C(CNC(CCC=C)=O)COCC2)=O)ccnc(Cl)c1F c1(C(N2CC(CC)C(NC(=O)C(C)=C3CC3)C2)=O)cc(Cl)cc(Cl)c1 c1(C(=O)NC23CC(NC(c4c(C)nn(C)c4)=O)(C2)C3)ccc(Cl)c(Cl)c1Cl c1(C(=O)NC2C(NC(CC(C)n3cccc3)=O)COC2)cnc2cccnc2c1 CCCCC(CC)CC(=O)N1CCC(F)(C(=O)NC2CC(=O)N(O)C2)CC1 Cc1ncc(C(N2CC3CCC3(NC(=O)CCCc3cccnc3)C2)=O)c(=N)[nH]1 CN=S1(=O)CCCC2(CCCN2C(=O)C(=O)Nc2ccccc2P(C)(C)=O)C1 N1(C(C(CC)CNC(c2ccc(Cl)o2)=O)=O)CCC(N2CC(F)C2)CC1 C1(C(=O)NCCC)CC2CCC1N2Cc1cc(Br)ccc1Cl N1(C(C2CCC(=O)N2)=O)CCCC(CO)(NC(=O)C(c2ccc(F)cc2)=O)C1 O=C1CCN(Cc2ccccc2Cl)C(=O)N1CCCn1cccnc1=O N1(C(C(n2ncc(C)c2)C)=O)CCCC(F)(CNC(=O)C(C)CC(C)C)CC1 C(=O)(C1CCCc2n[nH]cc21)N1C2CN(C(C(CCC(C)C)O)=O)CC1CC2 CC1CC(C)N(C(=O)Cc2ccon2)CCN1C(=O)C1=CCCSC1 C1(C(N2CCCC(CN(C(=O)CNS(=O)(=O)N(C)C)C)C2)=O)CC(=O)NC(C)C1 c1(C(N2CCC(NC(C(C(C=C)C)C)=O)CC2)=O)cn2cc(C)nc2s1 S(=O)(=O)(CC(F)(F)C(F)(F)Br)NC(c1cc2cnccc2s1)=O Cc1cc(C)n(CC(N2CCC(CCNC(=O)CC(C)F)C(F)(F)C2)=O)c(=O)n1 C1(C)(CNC(c2c(C)c[nH]n2)=O)CCCN(C(=O)C(c2ccccc2)C)C1 c1(C(=O)OC)cc(C(=O)N(CCNc2cc(OC)cnn2)CC2CC2)ccc1O N1(C(CCc2ccc(C)s2)=O)CCC(C(CO)NC(=O)Cn2cccc2)CC1 N1(C(C(CCCCC)O)=O)CCCCC2(CCN(C(=O)CC3COC(=O)C3)C2)C1 c1(C(c2nnnn2C2COC2)Nc2c(C)noc2)ccc(Br)c(F)c1F c1(CC(=O)NCC(C)N(C(C(CC)OCC)=O)C)c(F)cc([N+](=O)[O-])cc1F C1(CNC2(C#C)CCCCC2)CCC2(CCCOC2)O1 Cc1cn2c(C)c(C(=O)NCc3cccc(C(F)F)c3)nc2s1 C12(C(=O)NCC(CC)CCO)CC(CO1)N(C(c1n[nH]c(C)c1Cl)=O)C2 C1(OC)(CNC(=O)CCn2ccnn2)CN(C(c2sccc2C)=O)C1 C1(NC(C(C)C2CCCO2)=O)CCCCC1CNC(C1(C2CCCO2)CC1)=O C1(N(C(=O)C(=O)NCCOC)CC)CCCN(C(C2CC3CCC2C3)=O)C1 c1(CC(C(=O)NCC(CNC(C2C(COC)C2)=O)C)C)cccc(CC(C)C)c1 C1(C(N2CC(COC)(NC(C3(CO)CCC3)=O)C2)=O)CNC(=O)C(C)(C)C1 C#CCCCCCC(C(=O)NC(C)C)N1CC(NC(=O)OC(C)(C)C)CC1C N1(C(Cc2ccc(C)o2)=O)CCC(NC(=O)C(C)n2ccnc2)C1c1ccccc1 c1(C(=O)NCC2(O)CN(C(C3(COC)CCC3)=O)C2)cc(S(C)(=O)=O)ccc1Cl c1(C(C(=O)NC2C(CNC(Cc3cc(CC)no3)=O)C2)(F)F)cc(Cl)ccc1Cl c1(CN2CCCC(OC(=O)C(c3ccccc3)C3CC3)C2)nc(O)c2sccc2n1 C1(C(C)CNC(=O)CC2(O)CCCC2)CCN(C(=O)COC2CCOC2)CC1 Cc1cn2c(C(=O)NCC3CN(C(=O)CCCc4cccs4)C3)c(Cl)nc2s1 c1(COC)ccc(C(=O)NC2CN(C(=O)Cc3cc[nH]c3)CC23CC3)cc1OC C1(NC(C2(c3cccc(OC)c3)CCC2)=O)CC12CCC(NC(=O)C1CC1)CC2 N1(C(C2(CCC=C)CN(C(=O)CNc3ncccn3)C2)=O)CCC(C)C(O)C1 c1(C(=O)NC(C2CCCC2)CNC(c2cn(C)nc2)=O)cc2cccnc2s1 N1(CC(C)N(CCC)C)CCN(C(=NCCC(=O)NCC)NC2CC2)CC1(C)C CN1CCC2CN(C(C3(O)CCN(Cc4n[nH]c5ccccc45)C3)=O)CC2C1 C1(O)(CC)CCC(NC(=O)NCC(c2cc(F)cc(F)c2)C)CC1 c1(CN2CCC(C(=O)OCCN(C)C)C2)cc(N2CCNC2=O)ccc1Cl C1(NC(=O)CC2CC(C(F)F)C2)CCC(NC(c2ccnc(C(F)F)c2)=O)CC1 N1(C(c2cc(CF)on2)=O)Cc2ccccc2C1CNC(C12COCC1C2)=O c1(C(N(CCCNC(c2cnnn2C)=O)CC)=O)ccnc(-n2ccnc2)c1 Cc1ncc(S(N)(=O)=O)cc1C(=O)NCC#CCN(C)C C(N=c1[nH]cnc2cccc(Br)c12)C1CN(C(=O)Cc2cn3ccccc3n2)C1 N1(C(C(C)n2cncn2)=O)CCN(C(c2cc3cnccc3[nH]2)=O)CC12CC2 CCCC(C)CC(=O)N1CC(=C(F)CNC(=O)Cc2ccc(NC(=O)NC)cc2)C1 c1(C(=O)NCC(=C)CCNC(=O)Cn2cc(Br)cn2)cc(F)ccc1F CC1OCC2C(=O)N(CCNC(C3CCC4CCC34)=O)C(=O)N2C1=O CC1OC(C)Cc2c(C(=O)NC(C)(C)CCCNC(=O)Cc3cscn3)n[nH]c21 c1(-n2c(C(C(C)C3CCCC3)NCc3cc(C)on3)nnn2)ccccc1C CCC(CC(=O)N1CCCN(C(=O)Cc2c(C)cnn2C)CC1)C(C)C C1(C(N2CCC(N(C(c3cc(C)nnc3)=O)C)C(C)C2)=O)CCCCC(F)(F)C1 CC1(C)C(C(=O)NC(CO)C2CCC2)CCN1C(c1cc(CO)on1)=O C(=O)(C(CP(C)(C)=O)NC(c1c(Cl)cnn1CCN1CCC(C)CC1)=O)OC c1(N2C3CCN(C)CC3CC2)nc(=NCC2CCSC2)[nH]c2c1CCCCCC2 c1(CNC2CCC(C(=O)NC(C(=O)OC)(C)C)CC2)nc2ccccc2o1 C1(C)(C(N(CC(CC)CC)C)=O)CC(O)CN1C(=O)CCOC1CC1 N1(C(C(=O)N(C(=O)CC(C)C)C)CCC2CC2C)CC2CC1CN2CC(F)F N1(C(CCC2(C)CC2)=O)CCC2(CC(NC(c3ccnc(C(F)F)c3)=O)CO2)C1 c1(CCC)c(C(N2CCC(O)(CCNC(=O)CC3CSCCO3)C2)=O)nnn1C c1(C(=O)NCC2CN(CCOCC)C2)ncc2nccnc2n1.C12C(C1C)C2 N1(C(C2(C)CC(F)(F)C2)=O)CC(C(=O)NCC(O)C2(Cl)CC2)CCC1(C)C N1(C(C2(NC(C)=O)CCCC2)=O)CCN(CCC(N2CC(F)(CF)C2)=O)CC1 Cc1c(C(N2CCC(O)(CNC(C3C4(CC4)C34CC4)=O)C2)=O)[nH]c2ccccc12 C1(NC(C2C(=C)C2)=O)C=CCCC1C(=O)NC(c1nncn1C)CO N1(C(c2ccc(CC)cn2)=O)CCN(C(=O)CC(C)(C)O)C(CCOC)C1 C(=O)(CCCC(C)(C)C#N)N1CCC(NC(C#CC2(OC)CC2)=O)C(F)C1 c1(C(=O)NC2CC3CC2N(C(c2ccc(F)o2)=O)C3)c[nH]c2cccc(Br)c12 C1(C(N2CCC(NC)C2)=O)CCC(NC(c2cnccc2OC)=O)CO1 C1(C(=O)OC)CCC12CN(CC1NC(=O)CC1(C)C)C2 C(C)(C)CCC(=O)OCC.c1(C(=O)NC2C(CC)OCC2)ccc(CC#N)cc1 C1(NC(CCNC(N)=O)=O)COC2CN(C(C3(O)CN4CCC3CC4)=O)CC12 N1(C(C(C(C)C)O)=O)CC(NC(=O)COCc2cccnc2)CC(C)(C)C1 N1(C(C2CCCC(NC(c3cncc(C)c3)=O)C2)=O)CC2(CNC(=O)C2)C1 N1(C(c2cn3c(n2)SCC3)=O)CCC2CN(C(=O)CC(F)F)CCC2C1 n1(CC2CC(C)(F)C2)nc(-c2cncs2)nc1Cn1cc(C2CC2)nn1 CC1(C#CC(=O)NCC2COCCN(c3cc(CC4CC4)ncn3)C2)CC1 O=CN1CCOCC1C(N1CCC(CO)(CNC(=O)C(C2(O)CCCC2)F)C1)=O CC1(C)OCCC1Oc1ccccc1NC(=O)C(=O)NCC1CC=CCC1 N1(C(c2cccc(C(=O)NC)n2)=O)CCOC2(CCN(C(C3CC3F)=O)CC2)C1 CC1(C)CCN(C(=O)C2=CCCOC2)C(c2cn(CCC(F)=C(F)F)nn2)C1 c1(CC(N2CCC(c3ccccc3)(OC)CC2)=O)cc(F)c(Cl)cc1C Cc1ccc(C(N2CC(O)C(O)C2CNC(=O)Cc2csc(C)c2)=O)c(C)c1 c1(C(=O)NC(CNC(C(CN(C2CCCC2)C)O)=O)(C)C)ccc(Cl)cc1 C#Cc1ccc(NC(=O)CCC2(NC(=O)C(C)OCCN(C)C)CCC2)cc1C c1(OC)cc(C(=O)NC(C)C(C)NC(C2(C)CCN(C(C)=O)CC2)=O)cc(C)n1 N1(C(c2ccc(CC)s2)=O)CC(CNC(c2csc(CO)n2)=O)N2CCC1C2 N1(C(CC(C)CN(C(=O)OC(C)(C)C)C2CC2)=O)CCCC(S(N)(=O)=O)C1 N#Cc1ccnc(N(C2CNCC2F)C(=O)CCc2ccsc2)n1 c1(CN2CCC(C(=O)Nc3ccc(I)cc3Cl)C(O)C2)ccc(Cl)c([N+](=O)[O-])c1 c1(C(N2CCCC(C(CNC(CS(CC)=O)=O)(C)C)C2)=O)ccc(SC)c(N)c1 C1(NC(C2(COC)CN(C(=O)CCC(=O)N3CCCC3)C2)=O)(OC)CCN(C)C1 CS(=O)c1ccc(CC(=O)NC2CC(C)CC(C)(C)C2)cc1 c1(CN2CC(C)(CNC(c3cccs3)=O)OCC2)c[nH]c2nccc-2c1 c1(OC)cnncc1C(N1CC2CC2(CNC(c2sccc2C#N)=O)C1)=O C12(NC(c3ccon3)=O)CCC(CN(C(=O)CCCC(=O)c3ccccc3)C1)C2 N1(C(Cn2ncc(C#C)c2)=O)CCC(CNC(=O)C(=O)NC)C1(C)C N1(C(C2C(CC)C2)=O)CC2CN(C(=O)C(O)CCc3ccccc3)CC2C1 N1(C(CCC=C=C)=O)CCC(CC)CC1C(=O)NC(c1ccccc1)=O C1(NC(c2c(CCC)n[nH]c2)=O)CCN(C(=O)CCc2csc(C(C)C)n2)CC1O n1(CCOC)nnnc1C(C)(CCOC(C)C)NC(C1(c2cccnc2)CC1)C N1(C(C(C)NC(=O)NC)=O)CC2CN(C(=O)CC3=NNC(=O)C3)CC2C1 C1(COC(=O)CCc2cocn2)COc2ccccc2C1 c1(C(N2CCC(CCC)(NC(COCCCC)=O)CC2)=O)cnc2n1CCCC2 c1(C(N2CC3(CC=CC3)C2c2ccccc2)=O)cc2cc(Cl)cc(Br)c2[nH]1 N1(C(C(C(C)C)SCC)=O)C(CC(=O)Nc2ccccc2C2CC2)C2CCCC12 C1(CNC(C2(F)C(C)OCC2)=O)CN(c2ncnc(=N)[nH]2)CCCO1 C1(COC)(CO)CC12CCN(C(C1CC1C)=O)CC2.c12cn(nn1)C2OC C1(C(N(CCN(C(C(CC=C)CC=C)=O)C(C)C)C)=O)CCC(F)(F)CC1(C)C c1(OC(C(=O)NC2CCN(C(C3C(C)CC3)=O)C2)(C)C)ccc(F)cc1 N1(C(C(C)C)=O)CCC2OCCN(C(C34CCC(=O)N3CCS4)=O)C2C1 C1(F)(CNC(c2cnc(C3CC3)o2)=O)CC2CCC(C1)N2C(C1CC2CC2C1)=O C(=O)(C(O)C(C(C)C)OC)N(CC(CN(C(C(C)=C(CC)C)=O)C)O)C(O)CCSC C=C(C)CC1C(=O)N1.C1(N(C(C(c2ccnn2C)NCC)=O)C)CCOCC1C Cc1cc(Br)ccc1SCCNC(C(N1CC(OC(C)(C)C)CC1C)=O)=O C(=O)(CC(C)C(F)(F)F)NC(CCC)CNC(C1CCCN(CC)C1)=O C(CCN=[N+]=[N-])N(CCCNC(=O)NC1(C)CC1C)C(C)C CC1CN(Cc2ccc(C(Cl)Cl)cc2)C(=O)N1 CCC(C)(C)CCCC(=O)N1CC(O)CCC1C(N1CCC(C)C1)=O N1(C(C=C(C)C)=O)CC2CCC(NC(=O)Cc3cnccc3C)CC2C1 c1(C2C(C(N(C)CC3(CNC(c4c[nH]ccc4=O)=O)CC3)=O)C2)ccc(C#N)cc1 C1(NC(C(CC)C#N)=O)CCCCN(C(c2cccc(Br)c2C)=O)CC1 c1(C(=O)NC(CCC)C)coc2c1CN(C(=O)CN(C)C(C)C)C2 C12(C)CCCCC1C(=O)N2.C1(OC)CCCCC1C(=O)NOCCC(C)C CCC(CC)C(=O)NCC1CCN1C(=O)CC1CCC(=O)N1 C(CC(F)F)(C(C)(C)C)ONC(=O)NC1C(C(C)(C)C)COCC1 CCCCC(CNC(=O)C(C)(CC)OC)NC(=O)CCc1ccc(C(C)C)cc1 CC1(C)C(S(=O)(=O)N2CCN(c3cc(C4(C)CCCC4)ncn3)CC2)CCO1 N(C(=NCCN1CCCS1(=O)=O)NCC1(N2CCCC2)CC1)CC(C)OC CCCCC(CNC(c1cocn1)=O)NC(=O)C1=NOCC1 c1(OC)ccnc(-c2noc(CN)n2)c1C(N1CCCCC1CCc1cccs1)=O c1(NC2CCCN(C(c3coc(C(F)(F)F)n3)=O)C2)ncc([N+](=O)[O-])cc1Br CCCCCCCCC(=O)NCC1CC2CN(C(=O)CC(C)(C)OC)CC12 c1(-c2cnc(NC(=O)NC3C4COCC34)c(O)c2)cnn2c1CCCC2 CC(CN=c1[nH]c(=NCc2c(F)ccc(F)c2Cl)[nH]c2c1CCC2)S(N)(=O)=O CC1CN(C(C2CCC(N=[N+]=[N-])CC2)=O)CC1N=c1nc(C(F)(F)F)[nH]s1 c1(C(=O)NC(CCOC)CNC(C2(OC)CCSC2)=O)ncc(C)cc1OC c1(C(=O)NCC2(c3onc(C)n3)CC2)cc(Br)cc(C(F)(F)F)c1F c1(C=O)nsc2cc(-c3ccnn3C3COC3)ccc12.N#CC1CN2CCN12.C S(=O)(=O)(CCCCCl)Nc1ccc(CC(=O)Nc2ccc(C(F)(F)F)cc2)cn1 c1(SC)cc(C(=O)NC2CCC2NC(=O)CCc2cncn2C)oc1C N1(C(c2ncn(CC)c2)=O)CCCC(C2CCN(C(=O)COc3ccsc3)C2)C1 C(=O)(CC(C)(C)C(=O)NCC(C(C)(C)C)NC(C1CN2CCC1(C)CC2)=O)OC N1(C(c2c(OCCC)cccc2)=O)CC(C(=O)NCCC#N)CC(F)(F)C1 C(CS(=O)(=O)SC(C)(C)C=CCNC(=O)OC(C)(C)C)OCC.C(=O)N c1(C(=O)NC2(C)CN(C(c3cc(C#N)cc(C)n3)=O)C2)nccc2ccccc12 Cc1cc(N2CCC(NC(=O)Nc3cnn(-c4ccncc4)c3C)C2=O)n(C)n1 c1(C(=O)N(CC(CC)NC(c2ccn(C3CC3)n2)=O)C)cnc(C(F)F)c(C)c1 CCCS(=O)(=O)c1ccccc1C(=O)NCC(O)CNC(C1(C)CCCS1)=O C1(NC(Cc2cn(C)nc2)=O)CC2CN(C(=O)CN3CCC(=O)NC3=O)CC2C1 C1(C(=O)NC(CCSC)C)CC2(CCC2)CN1C(=O)COC(F)(F)F.C(C)(=O)O c1(C(N(C2CN(C(c3c(C)onc3)=O)CC2(C)C)C)=O)cc([N+](=O)[O-])ccc1N CN1CC=C(CC(=O)NC2CCCC2NC(=O)C(C)(C)c2cnsc2)CC1 c1(NC(Cn2c(CC)nnc2S)=O)cccc(S(=O)(=O)C2CC2)c1 O=C(C1c2c[nH]nc2CN1C(=O)Cc1cn[nH]c1)NCCC1CCCCC1 C1(C(N(C2(C(=O)OC)CC2)C)=O)C(C)OCCN1C(C1CSC1)=O C1(CC(=O)NCCN(C)C(C2(C)CCNC2=O)=O)CCCC1(F)F C(=O)(C(O)C(C)C)NC1(CC=C)CN(C(c2ccnn2CCC)=O)C1 C#Cc1cc(C(=O)NC(C)CCCCNC(=O)COCC)ccc1C Cc1c(Cl)cc(C(c2nnnn2CC(F)F)NCC2CC(CF)C2)cc1Cl c1(C(N(CC(C)C)CCC)=O)ccc(OCc2ccc(OC)cc2)cc1 CC#CC1CCN(C(=O)C(C2CCCC2)OCCN(S(C)(=O)=O)C)C1 C1(CC#C)(C(=O)NCCN(C(c2nc(CSC)no2)=O)CC2CC2)CCOC1 c1(C(C(=O)NCCCC)N(C)CC2CCN(C(=O)NC)C2)ncsc1Br CC1CN(C(c2cocn2)=O)C(C)CN1C(c1nnn2c1CSCC2)=O c1(CN(C(C2CCC(C)C2)C(=O)NCCOC)C2CC2)ccc(F)cc1F C1(C(N(CCNC(c2ccc(C(C)=O)o2)=O)C)=O)CC1C1CC1C c1(C(=O)OC(C)COc2cccnc2)cnn2c1NCC(C)C2 C1(CNC(C(C)OC(C)=O)=O)CN(C(c2cc(Cl)c[nH]2)=O)CC1(C)C n1(CC)nnc2c(NCC3CC(C)N(C(=O)C(F)(F)CC(C)C)C3)ncnc12 c1(C(N2CCN(C(=O)C(=Cc3cccnc3)F)C3C2C3)=O)ccc2c[nH]nc2c1 Cc1conc1C(=O)NCCOCCOCCNC(c1n[nH]cc1C)=O Cc1nc(C#N)ccc1C(=O)NC(C1CCN(C(C2(CO)CCOCC2)=O)C1)C Cc1cccc(C(=O)NCC(CO)NC(=O)C=Cc2cnc(C(C)(C)C)s2)c1 C1(N(C(C2OCCN(c3cc(COC)ncn3)C2)=O)C)CCC(C)(C)CC1 CC1CC(CNC(=O)C=CCNC(=O)C(N2CCNC2=O)C)CC(C)O1 N1(CC(=O)N(CC)Cc2cnc(CC(C)C)o2)CCn2ncc(CN(C)C)c2C1 C(=O)(C1=CCCCC1)NC(C(C)OC)C(=O)NCC(O)C(F)F C1(NC(CC(C)(C)F)=O)CCCC12CN(C(=O)CC1CCC(C)(C)CC1)C2 c1(OC)cc(Br)c(Cl)cc1C(c1nnnn1C(C)C)NCCCc1cnoc1 CCCC(C)(C)C(=O)N1CCC(C(C)NC(c2cc(CC)[nH]n2)=O)C1 CC12CC(CCO1)N(C(C1C3CCC(C3)N1C(C1CCCC1F)=O)=O)C2 c1(CC=C)cccc(NC(C23CC2CN(C(=O)CCC(C)=O)C3)=O)c1 c1(C(N2C(C(=O)NC(c3ccc(Br)cc3F)CO)CC2)=O)ccc(Cl)nc1F c1(C(=O)NC(C(=O)NCc2ncnn2CC(C)C)CCC)cc[nH]c1CC C(C)(CC(=O)N1CC(O)(CNC(c2ccc(CO)s2)=O)C1)(C(F)F)N(C)C N1(CC(=O)N(C)C)CCN(C(C2(C(C)C)CCNC2)=O)CC1 C(=O)(C1=C(C)OCCC1)N(C(CNC(CNC(=O)NC)=O)C)C CC(C)C(O)C(C)C(=O)N1CCC(C)(NC(=O)COc2ccccc2Br)C1 C12(NC(C(C)n3cnnn3)=O)CC1CN(C(=O)CCSCc1ccccn1)C2 Cc1c(NC(=O)C(c2ccc(OC(=O)CC#N)cc2)=O)nnn1-c1cnccn1 C1(C(=O)NCC=CCNC(=O)CN2CCCC2CO)CC2(CCCCC2)CO1 C1(NC(C(CCCOC)C)=O)COC2(C1)CN(C(c1ccc(O)cc1OC)=O)C2 C(CC(=O)N(C1CCCN(C(c2nc(C)ncc2Cl)=O)C1)C)(C(N)=O)NC(C)=O c1(C(=O)NCC(C)N(C(CC(CC)(C)C)=O)C)cn2c(n1)CC(C)CC2 CN1CCN(CCC(=O)NCCC2CN(C(=O)CCc3cnn[nH]3)CCO2)CC1 c1(CCC)[nH]ccc1C(=O)NC(C)C(CO)NC(C1(COC)CC=CC1)=O C1(O)(C(N(CCN(C(=O)CCCn2ccnn2)C)C)=O)CC1(C)C c1(C(N2CCC(N(C(C(C=C)O)=O)CCC)CC2)=O)ccc(C2=CCCC2)cc1 Cc1ccc2ccsc2c1C(N1CCC(C)N(C(=O)C(F)(F)C2CC2)CC1)=O c1(-n2ccc(C)n2)cccc(C(=O)NCCOc2ccccc2Cl)c1 c1(OC)ccc2[nH]nc(C(N3CC(C)N(C(c4ncccn4)=O)CC3C)=O)c2c1 c1(CC)c(CN)oc2ccccc12.N(C(Cl)=CCl)C(C1(CO)CC1)C C1(CNC(C(C)CCO)=O)CC2CCC(C1)N2C(c1coc(C(F)(F)F)c1)=O N1(N(C)C)CCC(NC=O)CC1.C12(F)CCN(C1)NC2=O.c1cccc(Br)n1 Cc1ccc(CC(N2CC3(CC(C(=O)NC(c4ccccn4)C)C3)C2)=O)nc1C c1(C(=O)NC(C(=O)NCc2cncc(OC)c2)(C)C)cccc2occc12 Cc1cncc(C(=O)NCCNC(=O)NCc2nc[nH]c2C(C)(C)C)n1 C1(C(C)C)N(C(=O)C(C)(C)CO)CC12CCN(C(c1cccc(Cl)n1)=O)CC2 N1(C(C(C)C)=O)CCC(C(C)(C)C)CC1CNC(=O)CN1CC(C)(C)C1 C1(OC(=O)C(C)OC)(CNC(c2oncc2C(N)=O)=O)CCN(C2CC2)CC1.CC CC(C)C(O)C(C)C(=O)NCCC(C)(C)CNC(=O)C(C)(C)CF c1(NC(CCN(C(C2CC23CCC3)=O)CC)=O)cccc2c1OCO2 N1(C(C(=O)NC2CC(NC(C3CCC3)=O)C2)=O)CCC(c2cccc(F)c2)CC1 N1(C(C(C)CC2CCCC2)=O)CCCC(CNC(C2(CC3CC3)CC2)=O)C1 C1(NC(=O)CC2CC(=O)NC2=O)CC(CNC(c2csc(CO)n2)=O)CC1O C1(C(N2C(CNC(c3cncs3)=O)CC3(CC3)C2)=O)CCn2cncc2C1 Cc1c(C(=O)NCC(C)CNC(=O)CCc2ccn(C)n2)cc(O)cc1N C(N=c1ccc(S(=O)(=O)N2CCCC2c2nncn2C)c[nH]1)c1onc(C)n1 c1(SC(C)C)ccccc1C(=O)NC1CCN(C(=O)CC(C)NC(N)=O)C1C N1(c2nc(C)cc(OCC)n2)CCC(F)(F)C(C(N2C(C)CCC2C)=O)C1 c1(C(=O)NCc2cccc(NC(C3C4CC4C4CC34)=O)c2)cccn2ccnc12 N1(C(C(CC)NC(C)=O)=O)CCC(N(C)C(=O)NC2CCCN2)CC1 Cc1nn(C)c(Cl)c1CC(N1CCC(C)(CNC(c2ccc([N+](=O)[O-])o2)=O)C1)=O C#Cc1cn(C)nc1C(=O)NC1CN(C(C2CN(C)CC(C)O2)=O)CC1C C1(C(=O)NCC#CC2CC2)CCN(C(c2n[nH]cc2Cl)=O)CCO1 O=C1CC(C(=O)NC(CCO)C2CCC2)N(C(=O)C=Cc2ccccc2)C1 C1(C(=O)NC2CC(C)(C)N(C(c3ccsc3Cl)=O)C2)CC12CCC(=O)CC2 c1(NC(c2ccn(CCNC(C(C)OCCCC)=O)c2)=O)cccc(N=[N+]=[N-])c1 C1(C(N(CC(F)F)C)=O)CC(NC(=O)C(=O)NCC2CC2)C1 N1(C(C(C)OCCCC)=O)CCCC(C)(NC(c2nnc(C(F)(F)F)s2)=O)C1 C12(C(=O)NC3CN(C(c4c(C)c[nH]c4)=O)CC3O)CCC(C)(CC1)CO2 Cc1nc(C(=O)NC2CC2CNC(=O)Cc2cc(C(F)(F)F)n[nH]2)cn(C)c1=O CC(C)(CC(=O)NC1CCCCC1NC(=O)COc1ccsc1)NCC(F)(F)F C(=O)(CC(C)(C)c1ccccc1)CCN(C)C(CCNC(=O)CCC1CC1(C)C)=O N1(C(C(C=C)O)=O)CCN(C(C2CN(C)C2)=O)CC1C c1(C(N(CCCNC(C=C(CCC)C)=O)C)=O)ncc(Br)cc1Cl CCCCC(O)C(=O)N1CCOC(Cn2cc(CC3CCCNC3)nn2)C1 C1(NC(CS(CCC)(=O)=O)=O)CCC2CN(C(c3cnoc3C(C)C)=O)CC2C1 c1(C(N(C2CCC3CN(C(c4cnccc4Cl)=O)CC23)C)=O)n[nH]c2c1CCSC2 c1(C(N2C(C)CC(NC(c3csc(O)n3)=O)C2)=O)cnc2occc2c1 c1(C(=O)NC2(C)CCCN(C(C3(CO)CCCC3)=O)C2)cc(Cl)c([N+](=O)[O-])[nH]1 c1(C(N2C3CC(NC(CN(CCC)C)=O)C(C3)C2)=O)ccc(S(N)(=O)=O)cc1N C(CCC(CCC)NC(c1cscc1C#N)=O)NC(C1C(=C)C1)=O C1(CC)(NC(=O)CC2CCCC(C)(C)O2)CCN(C(=O)C=Cc2cscn2)CC1 N1(C(c2ccn(C(CC)CC)n2)=O)CCCC(N(C(=O)CC2CC2(C)C)CC)C1 Cn1nnc2ccc(C(=O)NC3CC(F)(CNC(=O)C(O)CC(F)F)C3)cc12 C1(N(C(C(N2CC(C)C2)C)=O)C)CCCN(C(=O)CCc2c(N)cnn2C)CC1 C1(CNC(c2ccc(C)nn2)=O)CCC12CCN(C(=O)CNS(N)(=O)=O)CC2 C(=O)(C(C)(C)CN(C(=O)CN(C)C(C)=O)C)NC.C1(=O)C(C)N1 Cc1ccc(O)c(C(=O)NC2CC(c3ccc(Cl)cc3)(C(=O)O)C2)c1 C1(NC(C(COC)COC)=O)CCN(C(C2CCC2)=O)C(c2ccccc2)C1 Cc1ccc(C(=O)N(CC(C)NC(=O)CC2CCC(F)(F)C2)C)cc1CO N1(C(C2(N(C(C3(COC)CC(=C)C3)=O)CC)CC2(C)C)=O)CCC2CN(C)CCC12 N1(Cc2c(C(=O)NC3(CO)CC3)cccc2)CCCN(C(=O)C(F)(F)CO)CC1CO N1(C(CN(C(=O)OCC)C)=O)CCCC(N(C(=O)CN(C)C)C)C1 Cc1cc(CN2CC(C(C)NC(c3oc(C4CC4)nc3C)=O)C2)ccc1[N+](=O)[O-] S(=O)(=O)(c1ccc(C)c([N+](=O)[O-])c1)N1CC(C=C)C(C(=O)O)C1 N1(C(C2(C(N)=O)CCC2)=O)CC2CCCC(C1)N2C(c1ccncc1Cl)=O C(C(=O)NCC#CCNC(C1CCC(F)C1)=O)(c1ccccc1)=C(C)C N1(C(C2C(OCC)C2)=O)CCC2(CCN(C(=O)Cc3coc(C(F)F)n3)C2)C1 C#CC(CC)NC(C1CC(N(C)C(C2(N3CCCC3)CC2)=O)C1)=O CCCC(CC)CCC(=O)N1CCC(N(C(=O)CC(C(C)C)C(C)C)C)CC1 CC1(CCNC(=O)CSCc2ccncc2)CCN(C(=O)CC2CCCCO2)C1 C#Cc1c[nH]nc1C(=O)NCCC1CC(NC(=O)CN(C)C(=O)OC)C1 N1(C(C(C(=O)OC)OC)=O)CCC(F)C(NC(=O)Cc2ccc(Cl)c(Cl)c2)C1 CCCCC(CNC(=O)C(C)(C)CO)NC(c1ccc(-c2cnn(C)c2)o1)=O Cc1cc(C(=O)NCCCNC(=O)C2=NOC(CC3(O)COC3)C2)ncc1F c1(C(N2CCCN(C(CC(C)C)=O)CC2)=O)cc2ncc(Br)cc2o1 c1(CC)ncnc(CC)c1C(=O)NCC(O)CNC(=O)CCn1cnnn1 NS(=O)(=O)CCCCCC(=O)N1CC=CC1CNC(c1cccc2nc[nH]c12)=O C1(C(=O)NC2(C(C)(F)F)CC2)C(NC(=O)CC#N)C1(C)C C(=O)(C(F)C(C)(F)F)N(C)CCOCCCNC(=O)CCc1nc(O)n[nH]1 C(=O)(C(C)CC(C)(F)F)NCC(=C)CCNC(c1ccc(C2CC2)nc1C)=O CC1(C)NC(=O)N(CC(N2CCN(C(c3cc(C(F)F)ccn3)=O)CC2)=O)C1=O Cc1cc(C(=O)NCC(CNC(=O)Cc2ccco2)C(F)(F)F)ccc1C(C)C c1(C(=O)NC(CNC(CC(C=C)(C)O)=O)C2CCC2)ccc2ccnc(O)c2n1 c1(CC)ncnc(CC)c1C(=O)NCC(O)CNC(=O)CCC1CCCN(C)C1 c1(SCC(=O)NCC2(CN(C(CCSC)=O)C)CC2)cccc(F)c1 C1(C=C)(C(=O)NC2C(NC(C(CC#C)C3CC3)=O)CCOC2)CCCCC1 c1(CC(=O)NCC(CC)NC(c2cc(SC)ccc2Cl)=O)cnc2ccccn12 C(=O)(CCS(C)(=O)=O)NCc1c(C(=O)NC(C2CCOC2)C#C)scc1 N1(C(COCC(=O)NC)=O)C2CCCC1CC(NC(=O)CC1COCC1O)C2 C=Cn1nncc1C(=O)NC1CC(F)(CNC(C2CCCC2N(C)C)=O)C1 C1(NC(C(CC)N(C)C(C2CC23CCCCC3)=O)=O)CCCCCC1F Cc1ccc(CC(=O)NCC(C)NC(c2cc(COC3CC=CC3)[nH]n2)=O)cn1 C1(C(=O)NCCCCCCNC(=O)C(F)(F)c2nccs2)CC2CCC1NC2=O C1(CNC(C2CCN(C)CC2)=O)CC(O)C(O)CC1C(N1CCC1C1CCC1)=O CC1(C(N2CCC(Cc3cccnc3)CC2)=O)CCCN(C(c2cn[nH]c2)=O)C1 N1(C(c2cc(CC)c(C)s2)=O)CC(CNC(c2cnnc(O)c2)=O)CCC1C N1(C(c2cc(OC)n(C)n2)=O)CCCCC(C(=O)NC2CC(CO)C2)C1 N1(CCC(N)=O)C(=O)CCC(C(=O)NCCOCCCF)C1c1cccs1 c1(C(=O)NC2CN(C(C(C)O)=O)C(C)CC2)cc2c(nc1N)CCCC2 c1(C(N(CC(CC)NC(=O)CC2CC2(C)C)CC)=O)ccc(C)c(OC)c1 c1(C(=O)NCCCCN(C)C(c2cc(C3CCC3)nn2C)=O)cc2occc2s1 C(CCS(=O)(=O)NC1CCCC1n1cc(CCO)nn1)NC(C1CCCO1)=O C(C(C(F)(F)F)n1cccn1)NC(=O)CNC(C1CCN(C)C1)=O CC1C(=O)N(C)CCN1C(C(=O)NCC1CCOC1)C1=CCSC1 N1(C(CCSCC)=O)CC2CCC(CNC(=O)CCCNC(c3ccco3)=O)C2C1 N1(C(C2(C)CCCCC2(F)F)=O)CC2CN(C(c3csnn3)=O)CC2C1CO CC(C)(O)C#CC(=O)N1CCC1CC(=O)NCCN1C(=O)CNC1=O C1(C(=O)NC2(CC#C)CCOCC2)N(C(C2CCCC(=O)N2)=O)CCC1(C)C CCCCCC(O)C(=O)NCC1(C)CCCN(c2nccc(OC)n2)C1 C1(CCNC(c2c(C(C)(C)C)[nH]cc2)=O)CCCN(C(=O)COC2CCOC2)C1 Cn1cc(-c2ccncc2)nc1NC(c1ccc(C(F)F)o1)c1nnnn1C n1(CC(=O)NCC2N(C(C(CCC)(C)C)=O)CC2)nc2n(c1=O)CCCCC2 c1(C(=O)NC2CC(NC(C3(NC(=O)OC)CCC3)=O)C2)[nH]cc2c1CCS2(=O)=O C1(C(N2CC(NC(C3C(OCC)C3)=O)(COC)C2)=O)CCOC(C)C1 C(=O)(CCCCCC(C)C)NC(C(C)NC(c1ccc(SC)cc1Cl)=O)CO N1(C(c2cc(C)c(N)cn2)=O)CCC2(CC1)CC2CNC(C1(C2CC2)CC1)=O c1(CC(=O)NCCCC(=O)NC)cnc2n1CCCC2C c1(C(=O)NC2CC(O)CN(C(=O)Cc3cscn3)C2)nccc2ncccc12 c1(C(=O)NC2CCN(C(c3c(CC)c(C)sc3)=O)C(C)C2)cnc2[nH]cncc1-2 c1(C(N(CCCCC)CCC(=O)C2CCCC2)=O)n[nH]c(-c2ccccc2)n1 c1(CC(=O)NCC(CC=C)NC(=O)CCCC(N)=O)cccc2ccccc12 C(N=c1[nH]cncc1Cl)C1CN(C(c2cc(CC)[nH]n2)=O)C(C)C1 C1(NC(C(CC=C)C(C)C)=O)CCC2(CC1)CC(NC(=O)CCN1CCC1)C2 C1(C#CC(=O)N(CCCNC(=O)CC2CCCCC2(F)F)C)(CC)CC1 N1(C(Cc2ccc(C)s2)=O)CCC2CCN(C(c3cc(Cl)ccc3F)=O)CC2C1 c1(CC)nc(C)c(C(=O)NCC2(C)CCCN2C(=O)Cc2ccoc2)c(C)n1 C=Cc1ccc(C(=O)NC2CC(CCC(=O)NC3CC4(CC(OC)C4)C3)C2)cc1 N1(C(C(C)C2CC2)=O)CCC2CCC(NC(c3cc(F)c[nH]3)=O)C1C2 Cc1ccc(C(=O)NC2(C3CCCCN3C(c3csnc3Cl)=O)CC2)c(O)n1 C=Cn1nccc1C(=O)NC1COCC1NC(C12CC(C)C1C2)=O C1(SCC(=O)N(CC(C)C)C)CCCCN1C(c1csc(-c2cnc[nH]2)n1)=O C(N=c1[nH]c(C)cc(=NCC2(C)CCCO2)[nH]1)c1c(SC)ccc(Cl)c1 N1(C(COCCOCCOC)=O)CCCC1(C)NC(=O)CSc1cnn(C)c1 C1(F)(C(N(CCOCCCNC(C2CN(C)C2)=O)C)=O)CC12CCCCC2 C1(NC(C2CN(C(C3(C#C)CC3)=O)CC2CC)=O)CS(=O)(=O)C1(C)C c1(CC)nc(C(=O)NC(CO)C(=O)NC2CC(C)(C(N)=O)C2)c(C)o1 C1(C(N(CCCCC=C)C)=O)CCC(C)N(C(=O)Cc2ccc(C#N)cc2)C1 CC1CC(C(=O)NCC2(CN(C)C)CCC2)N1C(=O)CC(O)C1CCCC1 N1(C(c2c(OCC)c[nH]n2)=O)CCC(NC(=O)CCc2cc(C)cs2)CC1 C1(NC(C(C)c2ccsc2)=O)C2CC1CN(C(C1(C)CC=CC1)=O)C2 C(=O)(CCCCCCCCCO)N1CCCC(F)(NC(COCC(=O)NC)=O)C1 Cc1cc(Cl)cc2cc(C(=O)NCCC(C)NC(C3(C4CC4)CC3)=O)[nH]c12 c1(C(N2CCCCC2c2ccco2)=O)cnc2n1CCCCC2 Cc1nccnc1C(=O)NC1C=CC(C(N2CC(CS(C)=O)C2)=O)C1 N1(C(=O)OC(C)(C)C)C(CCNC(CC(=O)OC(=O)C(N)=O)C(C)O)CCCC1C C1(NC(c2nnc(C)s2)=O)CCN(C(=O)CC2CCCOCC2)CCC1CO c1(C(=O)NCC2CN(C(C(C)CC(F)F)=O)CC2O)ccc(N)c([N+](=O)[O-])c1 C1(COCC)CCN(C(=O)CC2CC2CNC(=O)Cn2ccnn2)C1 Cc1cccc2oc(CCNC(=O)N(C3CCCOC3)CCO)nc12 c1(OC)c(CC(=O)NC2CC2NC(=O)C(C)(C)C2CCOC2)cccc1F c1(CN)cc(OC)c(OC)cc1[N+](=O)[O-].C12CC(C1(C)C)N(C)C2=O.CO N1(C(Cc2nc(C)sc2)=O)CCN(C(=O)CN(C(=O)CC2CCC(=O)N2)CC)CC1 C(=O)(CC(CN(C)C)C(F)F)N(C)CC1CCN(C(c2c(Cl)cnc(C)n2)=O)C1 C1(NC(Cn2ccc(C)n2)=O)CCC2CN(C(=O)Cc3ncoc3C)CCC2C1 C1(CNC(c2n(CCC)ccc2)=O)CCCCN(C(c2ccnc(Cl)c2N)=O)C1 c1(NS(CCC)(=O)=O)ccc(S(C)(=O)=O)cn1.N12CC3CN(CC3C1)CC2=O c1(CC)c(C(N2CC(CCNC(C3CCCN3C=O)=O)(OC)C2)=O)cccc1F N1(C(Cn2ncc(CC)c2)=O)CCC(C)N(C(c2ccc(Cl)c(C)c2)=O)CC1 Nc1cc(F)ccc1C(=O)NCC1CCN(C(c2cc(F)cc(Cl)c2)=O)C1 Cc1nn2cc(C(N3CC(C)N(C(=O)CSc4n[nH]c(=N)s4)CC3C)=O)nc2s1 C12(C(N3C(C)(C)C(NC(=O)Cn4cccc4)CC3)=O)CCN(CC1)S(=O)(=O)C2 C(=O)(C1=C(CC)OCCC1)N1CC(OCC)(CNC(C2COCCC2OC)=O)C1 C1(CC=C)(CNC(=O)CCNc2ccccc2F)CCCN1c1cc(F)ncn1 N1(C(CCc2ccc(C)s2)=O)CC(NC(=O)C(C)n2cncn2)C2CCCCC12 c1(OC)cccc2cc(C(=O)Nc3cccc(CN4CCCS4(=O)=O)c3)oc12 C1(C(N(C)CCO)=O)CC2(CCC2)CN1C(c1ccc2c[nH]nc2c1)=O CC1(C)CN(C(C2CC=CCC2)=O)C(CNC(C2(C)CCCS2)=O)CO1 CC(C)(CNC(=O)C(Cc1ccoc1)NC(=O)CC1CCCSC1)C(F)(F)F Cc1cn2cc(C(N3CCC(CCNC(=O)C4=CCCOCC4)C3)=O)ccc2n1 N1(C(CN2C(C)CCC2C)=O)CC2(CCN(C(=O)C3=CSCCO3)C2)C1 CCCC(CC)CCC(=O)N(C1CCCN(C(c2cn(C)c(=O)cc2C)=O)C1)C c1(C(C(=O)NC(C2CN(C(c3cc(C)sn3)=O)C2)C)O)cccc(C(F)(F)F)c1 N1(C(C(CC)SC)=O)CCN(CCCNC(=O)CC2C(C)C2(F)F)CC1 N(C1COc2cc(Br)ccc21)C(C(n1cc(C(CC)CC)nn1)C)=O C1(CNC(=O)CNC(C2CCN(C(=O)COC3CCCC3)C2)=O)CCCCO1 C1(C2CCOCC2)(C(=O)OCCCP(C)(C)=O)CC1(F)F C(=O)(C(C)C(C)C(C)(C)C)NC1(CO)CCN(C(C2(CC)COC2)=O)CC1 Cc1noc(C(C)C)c1C(N1CCCCC1C(C)(C)CNC(C1CC2CC2C1)=O)=O C1(NC(CSS(C)(=O)=O)=O)CN(C(=O)CN2C(=O)CCC2=O)C2(CCCCC2)C1 c1(NC(C(C2N(C(c3cc(CC)no3)=O)CCC2)(C)C)=O)ccccc1C(C)C c1(C(=O)NC2(C)CCN(C(C3C(F)(C(=O)OC)C3)=O)C2)ccc(C(C)C)nc1O CS(=O)c1cccc(-c2ccnc(N3CCN(C(=O)C(C)(C)Br)CC3)c2)c1 CN1CCC2CCN(C(=O)C=CCNC(c3ccnc4cc[nH]c34)=O)CC12 CC(C)CCC(=O)C(=O)N1CCC(CNC(c2cc(O)nc(O)n2)=O)C(C)C1 Cc1c(C)c(C)c(C(N2CC(C3(NC(=O)CNC=O)CC3)C2)=O)c(C)c1C N1(C(CCCCOC(C)C)=O)CC(C)CN(C(=O)C=CC(C)(C)C)CC1C C1(C(=O)NC2CCCN(c3cc(O)n[nH]3)C2)CCC2(CCOCC2)CO1 N1(C(CC(COC)(C)O)=O)CCC2(CC1)CC(CNC(=O)C(C)(C)OC(C)C)C2 N1(CC)N=C(C(=O)NCCC2CCN(C(=O)C(=O)CC3CC3)C(C)C2)CCC1=O C(=O)(C1CCCc2ccnn21)N1CCN(C(CC(=C)Br)=O)C(C(C)C)C1 C1(NC(c2nccc(SC)n2)=O)CC2(C1)CC(CNC(=O)CN1CCCC1C)C2 N1(C(C(C)=NOCC#N)=O)CCC(=O)N(C)CC1.C12C=CC(C1)CC(=O)N2 C1(NC(C(c2cscn2)N(C)C)=O)CCC12CCN(C(c1csc(S)n1)=O)CC2 C1(CCC=C)(NC(C(C)(C)COC)c2nnnn2C(C)CC)CCCSC1 CC(C)CC(C)NC(CCCNC(=O)Cc1csc(-c2ncccn2)n1)=O C1(CNC(C(C)(C)OC)=O)C2CN(C(=O)CSCc3ncc[nH]3)CC12 N1(C(COCCCCC)=O)CCOC(CNC(=O)CCc2ncc(C)[nH]2)C1 Cc1cc(C(=O)NCCOCCCNC(=O)C(F)CC2CCCCC2)nc(O)c1 C=CCCCCS(C)(=O)=NC(=O)C1CCCN(C(=O)Oc2ccc(Cl)cc2)C1 C12(CNC(CC(=C)C)=O)CCC(CC1)N2C(=O)C(CCC)N(C)C C(CCC(=O)NC1COCC1CO)(C(C)C)NC(CC(C)(F)F)=O N1(C(CC(CC)C)=O)CC2(CCN(C(c3cnn4c3OCCC4)=O)CC2)CC1C Cc1cc(C(N2CCCCC2CCC(F)(F)F)=O)c(O)nc1C C(=O)(C1=CCC(F)(F)CC1)N1C(CN(C)C(C2CC3C=CC2CC3)=O)CCC1 Cc1ccc(I)cc1C(=O)NCC(=O)NC(C1CCC1)C C1(C(N(C2CC(NC(C3C(C(=O)OC)C3)=O)C2)C)=O)CCCOCC1 C(CC(C)C)(C(=O)N(CCC(=O)NCC1OCCCC1(C)C)CCO)OC N1(C(COCC(=C)C)=O)CCC(N2CCN(C(=O)CC(C)OC)CC2)CC1 C1(SC(C)C(=O)N(C)CCN(C(=O)CCOCC2CC2)C)COC(=O)N1 C1(NC(COCCC)=O)CCSC12CN(C(=O)C(C)(C(F)F)c1ccccc1)C2 c1(CO)cc(O)c(OCCOCCC)cc1Br.C12CCC(CC1)CN(C)C2=O c1(C(=O)NCC(C2CCCCC2)NC(CC(CN(C)C)O)=O)ccn2cncc2c1 C(N=c1[nH]c2c(c(=NC3C4CCCC34)[nH]1)CSC2)c1cc2cc(NCO)oc2cc1 N1(C(C(CC)(C)C#N)=O)CC(C)CN(C(c2csc(-c3cnc[nH]3)n2)=O)C(C)C1 N1(C(C2CCC=CCC2)=O)CC2C(C1)C(F)(F)C2(F)F c1(C(=O)Nc2c(C)noc2)c(CNC(=O)CSc2cn[nH]c2)nnn1C C(=O)(C(C)(C)CC(=O)N1CCC(CC(=O)N(C)CCN2CCNC(=O)C2)C1)OC C1(NC(c2cccc(O)c2F)=O)CCCCN(C(C23CC(C2)C3)=O)C1 C(=O)(C(C)(O)C(C)C)N(CCNC(c1ccc(-n2ccc(C)n2)cc1)=O)C(C)C c1(OC)ccccc1NC(C1CC1NC(=O)NC(C)CC#N)=O CCC(CC(=O)N1CCC(OC)C1)NC(=O)CCc1csnn1 S(=O)(=O)(CC(=O)NC(C)C(C(C)C)NC(c1ccc(SC)s1)=O)NCC C#CC(C)(C)CN=c1[nH]c(=NCC2(CC=C)CCCCCC2)[nH]c2c1CSC2 C1(NC(CC=C=C)=O)CN(C(c2ccc(OC)c(OC)n2)=O)C(C)(CC)C1 N1(C(Cc2c(C)ccs2)=O)CC2CCCCC2(CN=c2ccnc(C(C)C)[nH]2)C1 c1(N)ncnc2c1CCO2.C12(NC(CC3OCC(C)(C)OC3)=O)CC1COC2(C)C Cc1ccc2oc(C3CCCN3C(=O)NCCc3nc(C(F)(F)F)cs3)cc2c1 C1(C(=O)NCc2ccsc2C)(CC)CCN(C(=O)CC2CCCC(=O)N2)CC1 Cc1cc(C(N2CC(NC(c3cccc(C4(C)CC4)c3)=O)C2)=O)c2c(c1)CCO2 c1(C(=O)NCCN(C(c2c(C)nn(C)c2Br)=O)C)ccnc2ccnn12 Cc1csc(=O)n1CCC(=O)NC(C)Cc1nc(Cc2cccc(Cl)c2)no1 c1(C(=O)N)c(Br)cnn1C.Cn1cc(C(N2CC(F)(CC(C3CC3C)=O)C2)=O)nn1 C1(F)(CNC(CC(C)(C)OC)=O)CCN(C(=O)COc2cccnc2)CC1 N1(CC(=O)NCC(CN(C(=O)CP(C)(C)=O)CC)(C)C)C(=O)C2CC=CCC2C1=O c1(C(N2C(CNC(C(C(C)C)F)=O)CC(O)C2)=O)c(F)ccc2[nH]ccc12 CC1CN(C(C2(C)C=CCN2C(=O)C=CCN2CCCCC2)=O)CC1CO c1(C(C)=O)cccc(Cl)c1NC(=O)N(C)C(c1ccc(F)cc1)C c1(C(N2CCC(CC(=O)NCc3nccc(OCC)n3)C2)=O)ncc(F)cc1N C(C)(CNC(C1(N2CCCC2)CCC1)=O)(CNC(=O)Cn1nccn1)OC C1(CC(=O)NCC2CC(NC(CN(CCC)C)=O)C2)CCC(C)CC1 C1(CNC(c2c(C)sc(Cl)n2)=O)CC2(CO1)CN(C(=O)CN(CC(C)(C)C)C)C2 C1(CC=C)(NC(c2ccoc2)=O)CCN(C(=O)C(C2CCC(=O)N2C)C)C1 CC1(NC(c2cc3n(n2)CCO3)=O)CCN(C(=O)C=CCN2CCCC2)CC1 N1(CC(=O)NCC(=O)OCF)CC2CCC1C2.C12(CCC1)C1(CC1)C(=O)N2 c1(C(=O)NC2(C)CN(C(C(C)OCCOC)=O)C2)ccc(O)cn1 c1(OC)ccc(Cl)c(C(=O)NCC2CC2NC(=O)Cn2cc(C(C)=O)nn2)c1 n1(CC)cnc2c(NCCC3CCC(C)(C)O3)[nH]c(=NCC(CC3CC3)OC)nc12 c1(CC(=O)NCC2C(NC(C(Br)=C(C)C)=O)CC2)c(Cl)cnn1C Cc1noc(C2CC2)c1C(=O)NC(C)CN(C)C(c1cc(C2CC2)no1)=O N1(C(c2oc(C)c(Br)c2)=O)CCN(C(=O)C2=CCSC2)C(CCO)C1 CCC(C)CCN=c1ccnc(N2CCc3ccc(Br)cc3C2)[nH]1 c1(CC)cc(CC)[nH]c(=NCCOC(=O)C(C)Oc2cccnc2)n1 C1(N=[N+]=[N-])(C(=O)NC(c2scc(C)n2)C)CCN(C(=O)CCn2cncn2)C1 C(CCC(C)C(=O)N1CCC(C)(c2cn(CC3CCC(=O)O3)nn2)C1)OC C(CCN(C)C)(C(=O)N1CCC(CC(C)(C)C)C1)NC(CC(=O)OC)=O C1(CC(=O)NCCOCCC(=O)NC(c2c(C)ncs2)C)COCC(C)O1 C1(C2CC2)(C(=O)NCCC2C(C)C2)CN(C(=O)C(F)C2CCCC2)C1 C=CC1OCCC1C(=O)NCC(C)C(=O)N(C)Cc1cscn1 C1(F)(C(=O)NC(CN(C(c2cncc(SCC)n2)=O)CC)C)CCCN(C)C1 c1(C(=O)OC)ccc(C(F)(F)F)nc1NCC1CCCCN1C(=O)CCF S(=O)(=O)(c1ncc(C(F)(F)F)cc1Cl)NC(c1ncco1)C C1(C)(CNC(C(C)O)=O)CN(C(c2cn(C3CC3)cn2)=O)CCO1 C=CC1COCCN1C(=O)NC1(CN2CCOCC2)CCCC1 C1(C(=O)NC2CN(C(CSc3n(C)cnc3)=O)CC2O)CCCC12CCC2 C1(C(N(CCCNC(C=C(CCC)C)=O)CC)=O)CC(C)(NS(=O)(=O)C(C)C)C1 N1(NC(C2CCC(NC(c3cc(CC)nn3C)=O)C2)=O)CCCC(C)(C)C1C N1(C(Cn2ncc(C)c2)=O)CCC(C)(C)C1C(=O)Nc1ccc(C)cc1CO c1(C(=O)NC(CN(C(c2c(C)nccc2)=O)C)C)c(C)nc(C)n1O c1(C(=O)NCC(CC)NC(c2nc(OC)ccc2C)=O)n[nH]c2ccc(F)cc12 c1(C(N2C(CNC(C(c3ccccc3Cl)C)=O)C=CC2)=O)cc(F)c(Cl)cc1Cl c1(-c2cnc(C)[nH]2)nc(CC(C)C)nn1C1CSC1.C(C)C C1(CN(C(CCC#C)c2ccccc2)C(=O)CCC)CC(C)N(C(=O)OC(C)(C)C)C1 c1(C(N2CCN(CC3(NC(C(CC#C)C)=O)CC3)CC2)=O)cc(Cl)c(Cl)c(Cl)c1 Cc1csc(CCC(N2CC(O)(CCNC(=O)COC3CCOC3)C2)=O)n1 C(C(=O)NCCc1ocnc1CNC(C1CCCCN1C)=O)(C(C)C)OC c1(NC(C2C(CNC(CCC=CCC)=O)C2)=O)cnc2c(c1)CCC2 C(CC1CC2CC2C1)(C(=O)Nc1ccco1)N(C1CC1)CC1(C#N)CC1 C1(CNC(C23CCC(CC)(CC2)OC3)=O)CN(C(=O)CSC(C)C)CCC12CCC2 c1(C(=O)NCC2CCN(C(c3n(C=C)ncc3)=O)C2)c(F)ccc(C)c1F N1(C(c2cc3[nH]ccc3s2)=O)CC2CCC(C1)N2C(=O)C(F)(F)c1cnccn1 C#CCC(C)(CC)C(=O)NC(C1CCCCC1)CNC(=O)CC(C)F S(=O)(=O)(c1cc(Br)ccc1Cl)NC1COCCN(C(c2nc(Cl)sc2Cl)=O)C1 C(=O)(CCCC(=O)NCC1(O)CC(C(=O)NCc2cccc(F)c2OC)C1)OC C1(n2cc(CCNC(C)=O)nn2)C=CCC(C(=O)Nc2cnccc2C)C1 c1(C(=O)NC2CCC(C)(CNC(C34OCC(C)(C3)C4)=O)C2)cc(F)c(F)cc1F N1(C(C=CC(C)(C)SC)=O)CCC(OC2CCN(C(=O)COC(C)(C)C)C2)CC1 c1(C(=O)NCC23CCCC2CCN3C(=O)C(F)=C2CCC2)cc2ncccn2n1 c1(CC)nncn1NC(=O)C(O)CCCNC(=O)CC(C)C(F)(F)F N1(C(CC2C(C)(C)C2)=O)CCOC2(CCN(C(c3cc(F)ccc3)=O)C2)C1 C1(NC(C2(C=C)CC2)=O)CCC(F)(CNC(=O)C(c2cccc(Cl)c2)C)C1 CCCC(C(=O)N(CCC(=O)NCC(CO)CC(C)C)OC)NC(C)=O C1(C(=O)OC)COC2CN(CC3C(OC(=O)NC(C)(C)C)CCC(C)(C)C3)CC12 c1(C(N(C)CC2CCN(C(=O)CN3CCCCC3)C2)=O)cnc2ccccc2n1 CCC(C(=O)N1CC(CNC(=O)Cn2nnc(C)n2)C2(CCC2)C1)C(C)(F)F Cc1cc(C(N2CC(C(N3CC4C(C3)C4(C)C)=O)C(F)(F)C2)=O)ccc1F c1(C(N(C(C(=O)N(C(C=C)C2CC2)C)C)C)=O)cnn(C(C)C)n1 C1(NC(C(CCP(C)(C)=O)N2CCOCC2)=O)C2CC3CC1CC(O)(C3)C2 c1(CC)ccc(O)cc1C(=O)NCCC1CCN(C(c2csc(C)n2)=O)C(C)C1 N1(C(C(C)OCCOC)=O)CC2CN(C(=O)Cc3cnoc3)CCC12 N1(C(C(C)OCC(F)(F)F)=O)CCC(CCCNC(c2coc(C(F)F)n2)=O)CC1 CC1(COC(C)(C)C)CCCN(C(C2CCCO2)=O)C1.C1(=O)C(F)CC2CN1C2 N1(C(C(C)C2CCOC2)=O)CCC2(CC1)CCN(C(=O)Cc1sccc1Cl)CC2 Cc1ncc(C=CC(=O)NC(c2ccccc2F)CNC(C2COC(C)C2)=O)s1 C12(C(=O)NC3CC(C#C)C3)CCCC1N(C(c1cccc3cncn13)=O)CC2 C(=O)(C(F)CC(C)(C)C)N(CCNC(C1CCCC(C)CC1)=O)CC N1(C(CC(C)(F)F)=O)CCC2(CC1)OCCC2NC(=O)CCn1cnnn1 c1(-c2c(C(=O)NCC(CN(C(c3c(C)c[nH]c3)=O)C)O)nco2)cccc(F)c1 CCCC(C)CC(=O)N1CC(F)(F)CC1CNC(c1nnn(CC)c1C(C)C)=O C(C(C)(C)C#CC(=O)N1CC(N(C)C2CC2)CC1C)NC(C(C)NC(CC)=O)=O c1(CCC)nc(C(=O)NC2C=CC(CNC(c3sccc3C3CC3)=O)C2)co1 c1(-c2cc(C)n(CC)c2C)csc(=Nc2ccc(F)cc2)n1C1CCSC(C)C1 c1(OC2CC(C(N(c3ccccc3)CCC(=O)OCC)=O)NC2)ccc(CO)cc1 C1(N(C(C(=O)NCC=Cc2ccccc2)=O)CC2CC2)COC2(CCCCC2)C1 Cc1noc(CCCC(=O)NCC(CNC(=O)Cc2ccn(C(F)F)n2)CO)n1 N1(C(C2(OC)CS(=O)(=O)C2)=O)CC(C2CN(C(c3coc(C)n3)=O)C2)C1 C(C)(CCCCNC(c1nocc1Br)=O)NC(C(C)SC)=O c1(NCC)nnc(CC(C)C)n1CC(N1CCOCC1)C.c1(N)cnnc(O)c1 C1(CNC(COCCCC)=O)CN(C(c2cnc3sccn23)=O)CC1(C)C C12(CNC(C3C(OCC)C3C)=O)CC(C1)C(NC(=O)CC1CCC1)CO2 C12(C(N3CCC3)=O)CCCCC1C2(F)F.C1(C(=O)N(CC(F)(F)F)CC)CCCC1 c1(OC(F)(F)F)cccc(OCF)c1.C(C)(CNC(=O)O)OCC#C c1(CC(=O)NCC2C(NC(c3cnc(CCC)s3)=O)C2)cc(F)c(F)cc1F c1(C(N2C(CNC(c3c(C)cc(N)cc3)=O)CC2)=O)cc2c(C)n[nH]c2cn1 CC1CC(C)(C(=O)NCC(C2(O)CN(C(=O)CCc3cncs3)C2)(C)C)CCO1 N1(CC(=O)NC2CCCC(CNC(c3ccn(CCF)n3)=O)C2)C(=O)CCC1=O C1(CNC(COCCC)=O)CCC(C)N(C(=O)Cn2ncc(O)nc2=O)C1 CC1(C)CC(CC(=O)NCC(CO)NC(c2sccc2-c2ccccc2)=O)C1 c1(N(CCCCCC)CCNC(C2CCOC2)=O)cc2c(cc1Cl)OCCO2 N1(C(c2c(SC)cccc2)=O)CCN(C(c2ncnn2CC)=O)CC1C(C)C c1(NC)nc(N2CCC(C(=O)OC(C)(C)C)CC2)nc2c(Br)c[nH]c12 C1(C2CC2)(CNC(C(CCC)OC)=O)CCN(C(=O)CCc2cnc(C)o2)C1 c1(C(=O)NC2C(CNC(CCCCC=C)=O)CCC2)cccc2c1NCC(C)C2 C1(CO)CCN(NCC2(CCCC)CC(Cc3ccccc3F)O2)CC1 C(=O)(C1=CC2C=CC(C1)C2)N1C(C)(CC(=O)NC23CCCN(CCC2)C3)CC1 C(=O)(C1=NN(C)C(=O)CC1)N1CCCC(F)(CNC(C(C2CCC2)OC)=O)C1 c1(OCC(N2CCC2CNC(C23COCC2C3)=O)=O)ccccc1[N+](=O)[O-] n1(CCCSC)nnnc1C(C)(CCc1ccsc1)NCc1csc(C)n1 CC(C(C)C(=O)N1CCC(N(C(=O)C=Cc2ccco2)C)CC1)S(C)(=O)=O c1(CCC(=O)NC2CCC(CCNC(CCC=C)=O)C2)cccc(OCC=CC)c1 C(=O)(CCC(CF)CF)NC(C)C(C)(C)C=O.C(C)(C(C)(C)C#N)NC1CC1 C(=O)(C1OCCn2ccnc21)NC(C)CNC(c1cc(-c2ccncc2)[nH]n1)=O C(=O)(CN=c1[nH]c2ccccc2s1)NCCN(C(C1C(CC)C1)=O)C N1(C(CC2(OCC)CCC2)=O)CC(C)(C)CC1CNC(=O)CCc1cnn(C)n1 c1(COC(CCSCC)=O)ccnn1C.C1(C2CCCO2)C(=O)N1C c1(CCC=C)ccc(C(=O)NC(C2CN(C(C3CC4CC4C3)=O)C2)C)cc1 C1(NC(=O)C(N2CCCCCC2)=O)CCCN(C(c2cccnc2)=O)C1 c1(NC(=O)NC2(Cc3cccc(C#N)c3)CCOC2)ccc2nnc(C(F)F)n2c1 c1(C(=O)NCC(CC)NC(=O)C(O)CN2CCCC2)cc(OC)nn1C C1(=O)C(C(C)(C)C)N1.c1(OCC(=O)NC(COC)CO)ccn(C)n1 C1(N(C)C)(CC)CCN(C(C2COCCC2NC(=O)CCCC#N)=O)C1 N12CC3(CCCN(C3)C(=O)C3CC(C3(C)C)CC1=O)C2.C1(C(C)O)CC(N(C)C)C1 c1(NC(C)=O)ccc(F)c(C(N2CCCC2CNC(=O)Nc2n[nH]c(O)n2)=O)c1 c1(C(N2CCN(C(C(C=C)O)=O)C3C2CC3)=O)ccc(S(=O)(=O)NCC)cc1 C(CC(C(=O)NCc1ccn(C)n1)NC(c1cnsn1)=O)=CC c1(C(N2CC(O)(CN(C(c3c(SC)nn(C)c3)=O)C)C2)=O)c(C)nn(C)c1C C1(C(N(C2CCN(C(c3ncc(Cl)cc3Cl)=O)C2)C)=O)CC2CCC(C1)N2C Cc1ccc(Cl)c(C(N2CCC(F)(CNC(=O)C(C)c3ccsn3)C2)=O)c1 c1(C(=O)NC2CC(NC(c3cc(N)c(Cl)nc3)=O)C2)ccc2cc[nH]c2c1 C(C(C)(C)C(=O)NC1CC(CNC(C23CCCC2(C(N)=O)C3)=O)C1)SC N1(C(Cn2ccc(C)n2)=O)CCCC2C(CN=c3[nH]cnc(C)c3Br)C(C)CC12 C(=O)(CCC(C)(C)[N+](=O)[O-])N(CC(=O)OC(c1cccc(C)c1)C)C n1(CC#C)c(C)cc(C(N2CCCC2CNC(=O)Cc2cnn(CC)c2)=O)c1C CC1CC(NC(=O)CN2C(=O)CN(C)C2=O)CCN1c1nc(C#N)c(Cl)s1 Cn1c(NC(=O)CN2CCOC(C(=O)O)C2)nc2cc(Cl)ccc12 C1(N(C(=O)C=Cc2nnn(C)n2)C)CCN(C(c2cnn3c2CCC3)=O)CC1O C1(NC(c2c(C)n[nH]c2C)=O)CC2CCC(C1)N2C(=O)C(CO)C(C)(C)C C1(NC(c2n(CCCOC)nnn2)CC2CCCO2)C2CCCC1CC2 C1(CC)CC(C(=O)NC(C)(C)CCNC(=O)CC2CCN(C(C)C)CC2)CC(=O)N1 NS(=O)(=O)c1ccc(C(=O)NC2CN(C(C3CCCCC(=O)N3)=O)CC2F)cc1 N1(C(c2cnc(C)nc2C)=O)CC2CCC(C1)N2C(C1(C(N)=O)CC1)=O c1(OC)c(NC(c2ncoc2CN(C)C)c2nnnn2C2CCC2)cccc1F c1(C(=O)NC2CCN(C(c3c(OC)scc3)=O)CC2)cc2c(ccn2C)s1 C(=O)(CC1=CCOCC1)N1CC(C)(NC(c2ccc(N)c(C(F)(F)F)c2)=O)C1 N1(C(C(CCSC)NC(N)=O)=O)CCCC2(CCN(C(=O)C(Cl)=CCl)CC2)C1 N1(C(C(c2cccnc2)OC)=O)CCN(C(C2CC3(CC3)CO2)=O)C(C)C1 C1(C(=O)NCCCNC(c2cc(C(=O)OC)n(C)c2)=O)CNC(=O)C(C)(C)C1 N1(C(CCC(=O)NCCC)=O)CC2CCCC2(NC(=O)C=Cc2sccc2C)C1 Cn1nc(C(=O)NC2C3CC2N(C(c2ccc(C(C)(C)C)[nH]2)=O)C3)c(Br)n1 C1(F)(CNC(Cc2nnc(C)s2)=O)CCC(CNC(=O)C(F)C(C)C)CC1 CC(C)CC(C)(C)C(=O)NCC1(CNC(C2(C)CCCO2)=O)CC12CCC2 C1(C(N2CC(C(C(=O)O)O)C2)=O)CCCNS1(=O)=O.c1(C(C)=O)ccsc1Cl C(=O)(C(C)CCCC(C)C)NCCN(CCC)C(C1(C)CCCC1(F)F)=O C(=O)(CC(C)P(C)(C)=O)NC(=O)C(C)(O)CC.CCCN1CC1 c1(C(=O)NCC2CN(C(=O)COc3ccon3)C3CC23)cnc2c(c1)CCOC2 C1(C(=O)NCCCc2nc(C)[nH]n2)CN(C(=O)CCC(C)(F)F)CCC1C C=CC1(NC(=O)CC2(C)CCN2C(C2(C3(O)CCC3)CC2)=O)CCOCC1 c1(NC2CN(C(c3ccc(OC)nc3OC)=O)CC2C)cc(C)c([N+](=O)[O-])cn1 C(CCS(C)(=O)=O)NC.C1(C(N2C(C)CCC2)=O)CCCN1C(c1ccccc1)=O Cc1cc(-c2csc(N3CCC3Cn3cc(-c4ccc(Br)s4)nn3)n2)cc(C)c1 Cc1ccc(C(=O)NCC2CC(O)(CNC(=O)C3=NOC(C)C3)C2)c2c1CCC2 C1(C2CC2)(C(N2CCCC(NC(=O)C(C3CCCCC3)=O)C2)=O)CC=CC1 N1(C(C(COC)O)=O)CCC(CNC(=O)Cc2sccc2C)(COC)CC1 C1(NC(c2ccn(CCC)n2)=O)CCC(C)N(C(c2cc(Cl)ccc2Cl)=O)C1 N1(CC)CCCC(C(N2CCC(N(C(C3CCCN3C)=O)CC3CC3)CC2)=O)C1 c1ccc(F)cc1.C1(CNC(=O)C(C)C(=O)C)CCN(C(CSCC(C)C)=O)C1 N1(C(C(CC)C#N)=O)C2CCC1C(NC(=O)CCOC1CCCCC1)C2 c1(C(=O)NC(CCNC(c2ccc(C(C)C)nc2O)=O)C)cc(C)c(F)cc1F Cn1ncc(Cl)c1CN1CC(OCCNC(=O)OC(C)(C)C)C1 C(C(N=[N+]=[N-])C(=O)NC1CC=C(C(=O)NCC2CC(CO)CO2)C1)OCC c1(OC)cnncc1C(=O)NC1(CO)CN(C(c2ccn(C(C)C)c2C)=O)C1 CC(CS(C)(=O)=O)C(=O)NC1(CN(C(=O)C(O)Cn2cncn2)C)CC1 Cc1nc(CCCC(=O)N(CCNC(C2CCSC2)=O)C(C)C)cs1 N1(CCC)CCCCC1C(=O)NCC1(C)CCCN1C(c1cn(C)nc1SC)=O C1(C(N2CC(C)(NC(C3(n4ncc(Br)n4)CC3)=O)C2)=O)CC(=O)NC1(C)C Cc1nc2cc(-c3noc(-c4cccc(=O)n4C)n3)cnc2[nH]1 CCCCN=C(NCc1ccc(Br)o1)NCC1(C(F)(F)F)CCCC1 C1(C(=O)NCC(C(C)C)NC(=O)CCC2CCCC2)CS(=O)(=O)CC(=O)N1 C(=O)(C(C(C)(C)C)N(C)C)NC1CN(C(c2c(C)cc(SC)o2)=O)CC1O C1(CN(C2CCCC2)CC)CCN(C(=NCC2CCOC2)NCC)C1 Cc1nc(=N)[nH]cc1C(N1CC(O)(CNC(=O)CCc2cccc(C#N)c2)C1)=O CCC(C(=O)NCC1CC=CC1)N(C(=O)C1CC1)C(C)=O C1(CNC(CCCNC(C2(CC#C)CC2)=O)=O)OC(=O)NC1(C)C C1(C)(C(N2CCC(SC)C2)=O)C=CCN1C(C1CCC(=O)NC1)=O Cc1cnc(C(=O)NCC(C2CC2)NC(C2CCCCN2C)=O)cn1 CS(=O)(CCCCN)=NC(=O)c1ccc2c(c1)COC(=O)N2 C1(CC)(OC)CN(C(=O)C(C2CCCC2)NC(=O)CC2CC2(C)C)C1 c1(C(=O)NCC2CCC(C(N3C(C(N(C)C)=O)C=CC3)=O)C2)cc(C#N)cs1 c1(CNC(=O)C(O)C2CN(C(C3CC4(CC4)CO3)=O)C2)cc(O)ccc1F C(=O)(CC(O)c1cc(C)cs1)N(C1CCN(C(=O)CCc2cnn(C)c2)C1)CC N1(C(CCC#C)=O)CCN(C(c2cn(C)nc2C(C)(C)C)=O)C(C2CCCC2)C1 N1(C(C=CC=CCC)=O)CCC2(CC1)CC2CNC(=O)C(C(C)(C)C)OCC C(=O)(C(C(C)NC(c1cnsn1)=O)C(C)C)NC(C(=O)NCC)CC Cc1cc(C(N2CCC2CNC(C2(C#N)CCCO2)=O)=O)ccc1N1CCCC1=O c1(C(N2CC(NC(C3C(C)(C)CCO3)=O)C2)=O)cc(N)ccc1F c1(C(CNC(N2CC(C)(CS(C)=O)C2)=O)O)ccc(O)c([N+](=O)[O-])c1 C1(OC)CN(C(=O)CSC(C)C)CC1NC(C1CCC(=O)NC1)=O N1(C(C2N(C(=O)OC)CCC2)=O)CC2CC1CC2NC(c1cnn(C)c1)=O C1(NC(c2nccc(C)c2)=O)CN(C(=O)CCc2nc(C3CC3)no2)CCC1C CN1CCN(C(=O)CCCCN(C)C(C2(C#N)CC3CC3C2)=O)CC12CCC2 N1(C(CCCCN(CCCC)C)=O)CCCC2CN(C(=O)C(=O)NC(C)C)CC12 CC(C)C(CCC(=O)NCC1(O)CCC1)NC(=O)C1=C(Cl)CC1 C(CCCCCCC(F)(F)F)SCc1c(C)ccc(C)c1 N1(C(c2cc(OCC)n[nH]2)=O)CCC(NC(=O)CNC(C2CCOC2)=O)C(C)C1 C1(O)(CC(=O)N(C)N(c2cc[nH]n2)C)CCCC1.C12(CC1)C(=O)N2 C1(CC(=O)NC(C2(O)CN(C(c3c(C)[nH][nH]c3=N)=O)C2)C)CCCNC(=O)C1 C1(CC(=O)N(CC(=O)N(CCCCO)C2CCC2)C(C)C)CC2(CC2)CO1 c1(C(=O)NCC2CN(C(CCOCC)=O)C2)cnn(C)c1C(C)C c1(C(N2CC(CC=C)(NC(C34CCC(CC3)CC4)=O)C2)=O)sccc1S(C)(=O)=O C=C=C(C)CC(=O)NCC1(CNC(C2CCN(C(C)(C)C)C2)=O)CC12CCC2 N1(C(COC)=O)CC(O)(CCN(C(c2cc(F)n[nH]2)=O)C2CC2)C1 N1(C(CCC#CC)=O)CCCC2(C1)CN(C(C1CCCN(C(C)C)C1)=O)C2 c1(C(N2C3CN(C(c4cc(C)on4)=O)CC32)=O)ccc(CC(C)C)nc1C C1(NC(C(C)OCC=C)=O)CCN(C(c2csc(Br)c2C)=O)C(C)C1 C1(NC(c2c(C)coc2C(C)C)=O)CN(C(=O)CC2CCC(=O)CC2)C(C)(C)C1 c1(C(=O)NC2C(NC(=O)C3=COCCC3)CC2)cc(F)c2ccccc2c1 C1(C(N(C2CCCN(C(=O)COCc3nc[nH]n3)C2)C)=O)CCC(F)(F)CC1 Cc1c(C(=O)NC(=O)Cn2cnnn2)cc(O)cc1N.C1(=O)CCCCC2CCN12 C1(c2cc(C)cc(C)c2)C2(CCC2)C12CCC2 C1(CNC(=O)CCNc2cccnc2)CCC2(CC2)CN1 C1(NC(CC(CC)C)=O)COC2(C1)CN(C(c1cc(O)ccc1Br)=O)C2 N1(C(CC(C(C)C)O)=O)CCCCC12CC(NC(C1(CF)CCC1)=O)C2 c1(C(=O)NC(c2ccc(-c3nc(=O)o[nH]3)cc2)C2(C)CCC2)c(Br)cccc1C#N c1(CC(=O)NCC2N(C(CS(CC)=O)=O)CCOC2)c(Cl)cccc1Cl c1(CC)coc2c1CN(C(=O)C(F)C1CC(C(=O)NC3(CO)CCC(C)C3)C1)C2 CCC(C)(C)CC(=O)N1CCSCC1CCNC(c1cnc(C)cc1C)=O C=CC1(NC(C2CCOC2C(=O)NCCN(C)C(=O)OC(C)(C)C)=O)CCCC1 C1(C)(NC(c2c(SC)n(C)nc2)=O)CCCN(C(=O)COc2cccc(F)c2)C1 Cc1cc(C(N2CCC(NC(=O)CCc3cnc[nH]3)C(F)C2)=O)cc(F)c1 c1(CSc2ccc(NC(=O)NC3C(=O)NCCCC3)nc2)[nH]nc2ncccc12 C1(NC(C(c2nncn2C)C)=O)CCN(C(=O)C2=CCCCC2)C12CCC2 C1(NC(C2CN(CC)C(=O)CC2)=O)CN(C(=O)C=Cc2nccs2)CC12CCC2 Cc1ccc(NC(C2CCCN(C(C34CC=CC(C3)OC4)=O)C2C)=O)c(F)c1 CC1(C)Cc2ccc(NC3(c4nnnn4C4CCC4)CCCC3CCF)cc2C1 C(=O)(C(C)(O)C(F)(F)F)N(CC(C)(C)NC(C(C(C)C)N1CCN(C)CC1)=O)C O=C1CC(C(=O)NCC(F)CNC(=O)CC2CCCCC2O)c2ccccc2N1 C(=O)(C1=NNC(=O)C1)NCC(CN(C(Cc1cccc(C(C)C#N)c1)=O)C)(C)C C(=O)(C1=Cc2cc(Cl)ccc2OC1)NCCOCCn1cc(CC(CC)(C)O)nn1 C(CCC(CCC)NC(C1(C)CC1C)=O)NC(c1n(CC#C)ccc1)=O C#CC1(C(=O)NOCCN(CC(=O)OC)C)CCN(C(=O)C=CC(F)(F)F)C1 S(=O)(=O)(CCC(=O)NCC1CC1CNC(C1(C(F)F)CCCO1)=O)N(C)C C1(NC(C2(CNC(=O)C=C(C)CCC)CC(=C)C2)=O)COCC1C1CC1 N1(C(C(N2CCOCC2)C)=O)Cc2n[nH]cc2C1C(=O)NC(c1cccnc1)C n1(CC2CC2)ccc(C(=O)NC(N(CCNC(C=CC(C)(C)SC)=O)C)=O)c1 C1(C(=O)NCC2CN(C(=O)COCCF)C3(CCC3)C2)CC12CCC1(CC1)CC2 C1(F)(C(N(CCC(O)c2cccs2)C)=O)CCN(C(=O)OC(C)(C)C)CC1 c1(CNC(=O)NC(c2nnsn2)C)cn2ccc(CO)cc2n1 c1(SC)ncc(NC(C2(NC(=O)C=Cc3cocn3)CC2(C)C)=O)cn1 N1(C(CCSCCC)=O)CCCC1C(C)(C)C(=O)N1C(CO)CC1CO C1(COC)(NC(c2csc(COC)c2)=O)CCN(C(c2cccc(SC)c2)=O)C1 N1(C(CCCC)C)CCC2(CC1)CC2(C)C(=O)NCC1OCCO1 C1(NC(C(F)=CCC)=O)CC(C)N(C(=O)Cn2cc(C)c(C(F)(F)F)n2)C1 c1(C(N(CCCNC(C2C(C#C)C2)=O)C(C)C)=O)c(C)c(C)cc(C)c1C c1(C(=O)NCC2(O)CN(C(=O)COC3CC(F)(F)C3)C2)ccnc(C2CC2)n1 C=CC(C)(CC)C(=O)Nc1cccc(CNC(C2COCCC2(F)F)=O)c1 N1(C(c2cc(CC)on2)=O)CCN(CC(C)NC(=O)CC2CCC(C)CC2)CC1 C1(OC)CN(C(=O)CCCCN(C)C)CCC1NC(=O)CC(C)n1cccc1 c1(OC)cc(F)c(-c2ccc(C3(CNc4cccnc4O)CC3)cc2)cc1F Cc1cccc(N(Cc2ccccn2)CC2CCC2)c1C C(=O)(CCC(C(=O)NC1(CCNC(=O)Cc2sc(S)nc2C)CC1)N(C)C)OC N1(C(CC(C)CC(F)(F)F)=O)C2CCCC1CN(C(C13CCC(C1)C3)=O)C2 C1(OC)CC2CC(C(=O)NC3(C)CCN(C(=O)CNC(c4cscn4)=O)CC3)CC12 c1(C(N2CC(C)N(C(=O)CN(C3CCSC3)C)CC2)=O)cc[nH]c2nccc1-2 N1(C(C=C(CC)C)=O)CCCC(CC)(NC(c2cccc(C(=O)OC)c2)=O)C1 CC1CCN(C(=O)COCP(C)(C)=O)C1CNC(c1ccn(C)n1)=O N1(c2c(F)cnc(C)n2)CC23CCCC2(CN(C(c2ccc(O)nc2Cl)=O)C3)C1 C(C1=NOC2CN(C(c3cc[nH]c3)=O)CC12)NC(c1cc(SC)c(F)cc1)=O C=C(C)C1OCCC1C(=O)NCCOC(C)(C)CNC(c1oncc1C)=O c1(CC)cc(C(=O)NCC2CCC(C)N(C(=O)C=Cc3ncc[nH]3)C2)cc(O)n1 c1(C(=O)NC(C2CCCCC2)CNC(COC)=O)nc(C)n(C)c1C c1(C(N2CCC(C)(NC(CC(CC)C3CC3)=O)CC2)=O)cc(C)c2nc(C)nn2c1 C(c1ccc(CCCCC(c2nnnn2C)NOC(C)(C)C)o1)=CC(=O)OCC C1(CNC(=O)CN2CCC(C)(O)C2)CC(F)CN1C(C)C(=O)NCc1ccncc1 Cc1cc(C(=O)NCC(C)NC(C2(C(F)(F)F)CCC2)=O)sc1Br C1(C(=O)NCC2CC(NC(C3C(C(N)=O)COC3)=O)C2)CCOCC12CCCC2 N1(C(C(C2CCC(=O)N2)C)=O)CCN(C(C2(CNC(=O)OC(C)(C)C)CC2)=O)CC1 c1(C(=O)O)ccc2c(c1)CCC2.C1(CN)CCCN(C(c2ncccc2[N+](=O)[O-])=O)CC1 CC(C)C(O)C(=O)NCC1CN(C(=O)CCSc2cccc(F)c2)CC1O N1(C(C(CCC)F)=O)C(C(=O)NCc2nnc(CC)o2)CCC12CC2 C=C=CCCC(=O)NCC1(NC(c2cccc(C(C)(C)C#N)c2)=O)CCCC1 C(=O)(CC(C)C(F)(F)F)NC1CC(OC)CN(C(c2cnc(N(C)C)nc2)=O)C1 c1(C(=O)NCC)ccc(C(=O)NCCCNC(=O)C(F)n2ccnc2)cc1 C1(NC(CCOCC)=O)(NC(=O)NC(C)C2CC2)CCSC1 C(=O)(C1=CCS(=O)(=O)C1)NC1CCN(C(Cc2cccc(OC)n2)=O)CC1F C=CCC(CC)C(=O)NCCC(C)CCNC(=O)Cc1cncn1C C(C(=O)NOCC(=O)OCc1cc(CC)on1)NC(CC)=O c1(C(=O)NCCC2(O)CCN(C(C3C(C)C3C)=O)CC2)ccc2[nH]c(=N)[nH]c2c1 C1(CNC(c2nc(OCC)oc2)=O)CN(C(c2cnc[nH]2)=O)CCC1C c1(NC(C(C)NC(C=CC(C)(C)SC)=O)=O)ccc(O)c(CO)c1 N1(C(C#C)=O)CCC(NC(=O)C(c2cn(C)nc2CC(C)C)C)CC1 CC1CCC(NC(C2CCC(=O)NC2)=O)CN1C(=O)CCC(=O)c1ccc[nH]1 Cc1ccn(C)c1C(N1CC(CC(C)NC(=O)CN2CCCOC2=O)C1)=O CC1(C)NC(=O)CC1C(=O)NCCCCCCNC(c1ccc(O)nc1)=O c1(C(=O)NCCCCCNC(C(C2CC2)OC)=O)cc2c(Br)coc2cn1 c1(OC)c(NC(C2CC3CN(C(=O)C(C)Cc4ccco4)CC23)=O)cccc1F CC1(O)CCN(C(=O)C(Cc2cn[nH]c2)NC(C2C=CCC2)=O)CC1O c1(CN(C)Cc2nnc(C(=O)OCC)s2)c(Cl)cc(F)cc1Br c1(C(=O)NCC23CCC(NC(C4CC4CF)=O)(CO2)C3)cc2c(o1)CCCC2 C(CC(C)C(=O)NC1CC2(C1)CC2C(N1CC(CF)C1)=O)=CC Cc1ccc(Br)c(NC(C2CC(NC(=O)Cc3cccc(C#N)c3)C2)=O)n1 C1(C(=O)NC2CC(NC(C(CC(C)C)O)=O)C2)CCc2c(ncn2C)C1 C1(C(=O)NC(CC)CNC(c2scnc2C(F)F)=O)(CO)CCCCO1 c1(CCN(C(c2ccoc2C(F)(F)F)=O)Cc2ccccn2)ccc(O)cc1 C(=O)(CCCC(=O)N1CCC(NC(=O)CCCC2CCCO2)C(CC)C1)NCC CC(C)(CCCF)C(=O)NCC1(O)CC(CNC(=O)C=C2CCCCC2)C1 c1(C(=O)NCCN(C(c2ccnn2C2CC2(F)F)=O)CC)cncc2c[nH]nc12 C1(NC(CCNC(COC)=O)=O)CC2CCC1N2C(c1ccnc(CO)c1)=O c1(C=O)ccc(OCC2CC2)cc1.C1(C=O)CC12CC(O)C2.C12CCCN1N(C)C2 c1(-n2cc(C3(NC(CC4CCC(C)CO4)=O)CCC3)nn2)ccc(C2CC2)c(Cl)c1 c1(C(N2CC(CNC(CCCC#C)=O)C3C2C3)=O)ccc([N+](=O)[O-])cc1[N+](=O)[O-] CCC(C(=O)NC1CC(N(C)C(c2cc(-c3cccs3)[nH]n2)=O)C1)OC c1(C(=O)NC(N)=O)c(Br)nc2n1CCC2.O=C1C(=O)NCCN1 C1(N(C(=O)COC2CCOC2)C)CCN(C(=O)C=Cc2cnccn2)CC1 Cc1c(Cl)c(C(=O)NC2CN(C(C3CC4COCC4C3)=O)C(C)(C)C2)nn1C c1(C(N(CCCNC(C(COC)O)=O)C2CC2)=O)ccc2cc(C)ccc2c1 c1(C(N(CC(C)O)CCNC(c2cc(COC)on2)=O)=O)cn(CCO)nc1C C1(C(N(C2CCC(NC(C=CC=CCC)=O)CC2)C)=O)CCC(C)C(C)C1 C(CCF)(C(=O)C(=O)CCC1CC1)NC(COCCC(C)C)=O.NC C1(CNC(C2(OC(C)C)CCOC2)=O)(NC(c2cscn2)=O)CCCCC1C N1(C(c2c(CC)nccc2)=O)CC(NC=O)CC(C)C1.c12ccc(cc1)SC2.CC C(=O)(C(C)(C)S(C)(=O)=O)N(CCCCN(C)C(c1cc2c[nH]nc2s1)=O)C CC1CCc2[nH]c(C(=O)NCC3(F)CN(C(=O)C(C)(C)c4ccsc4)C3)cc2C1 C1(Nc2c(C(=O)OCC)ccnn2)CC2CC1N(C(C1CCC3(CCC3)O1)=O)C2 C1(C(=O)OC)CC(C(N2CC(O)(CC=C)C2)=O)N(CC2CC(=O)N(C)C2)C1 CC1CN(C(c2cc(C(N)=O)no2)=O)CC1CNC(=O)C(C)(C)CF CCC(O)(CC)CCNC(=O)C(=O)NCC1CCCC1Cc1ccccc1 N1(C(c2n(C)cnc2)=O)CC2(CC(NC(C3(C(F)F)CC(F)(F)C3)=O)CO2)C1 C1(NC(c2c(OC)nc(Cl)cc2)=O)CCC(C)(C)CC1CNC(=O)C=C(C)Cl c1(C(=O)NCC2(COC)CN(C(C3C(=C)CC3)=O)C2)nc2ccccc2n1CC c1(C(=O)NCc2cc(C(=O)NC(C)CC3CC3)no2)cnc(N)cn1 C1(NC(c2ccc(C)nc2)=O)CC2CCC1CC2NC(c1cn(C)nc1O)=O c1(OC)cc(C(c2nnnn2C)NC(C)Cc2cccc(C)n2)c(Cl)cn1 C(c1ccc2ccccc2c1)=CC(N1CCC(NC(COC(C)C)=O)CC1)=O c1(C(=O)OC)ncccc1C(=O)NC1C(CNC(=O)C(C)n2cccn2)C1 Cc1ccc2c(C(N3CC(F)(F)CC3CNC(C3CC34CC4)=O)=O)ccnc2c1 O(NC(=O)C(c1ccco1)NC(=O)CC1CC2(CCC2)C1)CC(C)(C)C N1(C(c2c(CCC)nco2)=O)CC(C)CN(C(=O)CCSCC(C)C)CC1C c1(CC(=O)NCC(F)CNC(c2cc(F)ccc2Cl)=O)c[nH]c2ccccc12 N1(C(CCSCCCC)=O)CC(C)(C)CCC1CNC(C1CC(C)(O)C1)=O Cc1cc(C(=O)NCC2CN(C(C3(C(C)(F)F)CCC3)=O)CC23CC3)cc(C)n1 N1(C(c2cncc(C3CC3)c2)C(=O)NCc2ccccc2)CCC12CCCSC2 C#CC1CN(C(C2CC(Cl)(Cl)C2)=O)CCN1C(=O)CC(C)(C)CC C(=O)(C1=NOC2(CCC2)C1)N1C(CNC(c2cc3cccnc3s2)=O)CCCC1 C1(CNC(C(c2cccc(Cl)c2)C)=O)CCCN(CCC=Cc2cnn(C)c2)C1 c1(C(=O)NCCCN(C(CCc2onc(C)n2)=O)CCO)cnn(C(C)(C)C)c1C C1(O)(CNC(CC(C)CF)=O)CCN(C(=O)OC(C)(C)C)CC1 c1(C(N2CC(C)C(N(C)C(c3cnsn3)=O)CC2)=O)cc([N+](=O)[O-])c(O)cc1N C(CC1=CCCCC1)NC(=O)NC(C)C1CC1 CC1(C)CCN(C(=O)Cc2cc(O)nc(O)n2)C1CNC(C1CC12CCC2)=O N1(C(C2(CC)CC2(F)F)=O)CCN(CCN(C)C(c2ncc(C)s2)=O)CC1 C1(C)(CNC(CCC)=O)CN(C(c2ccc(Cl)c(OC(F)(F)F)c2)=O)CC1C c1(C(=O)NC2CC(NC(c3cn(CC=C)nc3)=O)C2)sc2nccn2c1C CC12CN(C(c3ccc(Cl)nc3)=O)CC1(C)CN(C(c1n[nH]cc1[N+](=O)[O-])=O)C2 c1(CC(N2CC(NC(c3nc(C)n(C)n3)=O)C(C)C2)=O)c[nH]c2cccc(Cl)c12 C(C(=O)N=c1cc(C)n(C2CC2)[nH]1)(C(C)OC)N(C(C(CC=C)OC)=O)C1CC1 c1(CCC(=O)NCC(C)N(C(=O)CNC(c2cnc[nH]2)=O)CC)cccnc1 C1(C(N(CCN(C(c2cscc2OC)=O)CC)CC)=O)CCc2[nH]nc(O)c2C1 N1(C(C23CCC(OC)C2C3)=O)CC(C(=O)NCc2ncc(CO)[nH]2)C(F)(F)C1 c1(C(C2CCC2)NCc2c(C)nn[nH]2)cccc2ccccc12 N1(C(C(CCCC)=O)=O)CC(NC(=O)CC2C=CS(=O)(=O)C2)CC12CCC2 N1(C(c2[nH]cc(C)c2)=O)C2CCC1CC(NC(c1ccnc(C(F)(F)F)c1)=O)C2 c1(C(=O)NCC2CC(CNC(c3sccc3Cl)=O)CO2)ccc(Cl)cc1 Cc1nn(C(C)C)cc1C(N1CCCC1CN(C)C(c1cnc(Cl)[nH]1)=O)=O c1(C(N2CCC(C(N3CCC(O)CC3)=O)CC2)=O)ccc2nnc(S)n2c1.C1(C)CC1 c1(OC)ccc(C(=O)NCC2(F)CCN(C(=O)C3=CCSC3)CC2)c(OC)c1C C1(=CCNC(C(C=C)O)=O)CCN(C(C2CCCN(CC)C2)=O)CC1 S(=O)(=O)(c1cnn(CC(F)F)c1)N1C(c2nnc(C)o2)CCCC1 C=CC1(CC(=O)NCC(F)Cl)CN(C(c2nnsc2N)=O)C1 O=C(C1Cc2ccccc21)N(C1CCS(=O)(=O)C1)CC1CCCCO1 C=CCC(C(=O)N(C)CC1CCCN(C(c2cccn2C)=O)C1)OC S(=O)(=O)(C1CCCN(c2ccnc(-c3ccccn3)n2)C1)NC c1(C(=O)NCC=CCNC(c2c(CC)ncs2)=O)cccc(C(C)C)c1F N1(C(CN2CCC(C)CC2)=O)CC2COCCC2(NC(=O)CCCN=[N+]=[N-])C1 N1(C(CC(C)CF)=O)CC(C)C(C)(CNC(c2cccc(N)n2)=O)C1 S(=O)(=O)(c1ccc(NCc2nncn2C)cc1Br)NC(COCC)CC(C)(C)C c1(CCC(=O)NCC2CC(NC(=O)CCSC(F)(F)F)C2)cccc(F)c1 N1(Cc2ccc(C(=O)OC)cc2F)CCC=C(C(=O)Nc2cc(O)ncn2)C1 C1(NC(=O)NC2CCCN(c3ccc(C(F)F)cn3)C2)CC2(CCOC2)C1 C12(N(C)C)CCC(C(=O)N(c3nnnn3C)C(C)Cc3ccccn3)(CC1)CC2 c1(C(N2CC(NC(C(C)CC(F)F)=O)C2)=O)cc2nc(O)[nH]c2cc1N c1(-n2c(NC(=O)NC(CC)C(C)(C)c3ccccc3)cnc2)c[nH]c2cnccc12 C(CCCCC(=O)NC(C1(CNC(c2ccc(O)c(C(N)=O)c2)=O)CC1)C)OC C(=O)(C1=CC2(CN(C(c3cnc[nH]c3=N)=O)C2)OC1)NCC(C)N(C)C c1(C(=O)NC(CC)CNC(c2occ(C)c2C)=O)cnn2c(=N)[nH]cnc12 c1(NC(C2CCC(CNC(CCC=CC)=O)C2)=O)nccc2occc12 N1(C(C(C(CC)C)=O)=O)CCC(C(=O)NCc2cc(C)ccn2)CC1(C)C CCC(CC(=O)N(CC(C)(C)CNc1cnc(C(=O)OC)cn1)C)C1CCC1 N1(OC)CC2(CC(C)CC(=O)N2)C1.C12CCC(c3nnnn3CCSC)(CC1)N2 N1(C(c2cc(CSCCC)on2)=O)CCC2(NC(=O)C(=O)NCC)CC2C1 c1(C(N2CCCC(CCCCNC(C=NOC)=O)C2)=O)ncc(Br)cc1N C(=O)(CCCC(=O)N(CCC#N)C)NCC(C)N(C(=O)CO)C.C(C)(C)(C)OC(C)C N1(C(c2c(Br)nc(C)s2)=O)CCN(C(=O)C(=O)N(C)C2CC2)CC1CF c1(C(C(=O)N2CC(N(C(c3cn(CCC=C)nn3)=O)C)C2)(F)F)cccc(C)c1 c1(C(=O)NC2C(NC(C3CCN(C)C3)=O)COCC2)cn2ccnc2s1 CN1CCN(C(=O)C(CCC2CCC2)N(C(=O)CCOC2CC2)C2CC2)C(CCO)C1 c1(C(=O)NCC23C(CN(C(c4ccc(Br)cc4I)=O)C2)C3)cccn2cncc12 C=C(C)CCC(=O)NC1CN(C(=O)C(F)n2cccn2)C1 N1(C(C(C)NC(C)=O)=O)CCC(CCOC)(NC(C2(n3cncn3)CC2)=O)CC1 C12(NC(=O)CSc3ccccn3)CC(CO1)N(C(C1CC3CC1CC31CC1)=O)C2 C(=O)(C1CCCn2nccc21)NCC1N(C)CCN(C(CCCCCC=C)=O)C1 C1(NC(Cc2c(C)non2)=O)CCCC12CN(C(C1CC(C)(O)C1)=O)C2 CC1CN(C(C2N(C(C3(c4cccs4)CC3)=O)CC2(C)C)=O)CC(=O)N1 c1(C(N(C)CC2N(C(C(C)OCCN(C)C)=O)CC(F)C2)=O)cc(Cl)ccc1N N1(C(C2ON=C(CC)C2)=O)CCC2(CCCN(C(C3(C(C)(F)F)CC3)=O)C2)C1 N1(CC(=O)N(C2CCN(C(c3sc(C)cc3Cl)=O)C2)CC)C(=O)CN(C)C1=O C(=O)(C1CCCc2c1ncn2C)N1CCN(C(CN(C(C)C)C)=O)CC1C1CC1 Cc1coc(C2CC2)c1C(=O)NCC(C(C)C)NC(C1CCC(F)C1)=O C1(CC=C)(NC(C(C)OCC#C)=O)CCN(C(=O)Cc2cn(C)nn2)C1 N1(C(C)=O)CCCCC1C(C)(C)CNC1CCCN(C(=O)C(Cl)=CCl)C1 CCC(C(=O)NCCC1CCCN1C(=O)CC(F)F)n1ccnc1 C#Cc1ccc(CNC(=O)C(O)CN2CCOCC2)cc1.C12(CC1)CC(=O)N2C N1(C(C(C)S(C)(=O)=O)=O)CCS(=O)(=O)C(CCNC(c2cc(O)nc(Cl)c2)=O)C1 N1(C(CNS(NC)(=O)=O)=O)CCCOC(CNC(=O)Cc2ccc(C(N)=O)cc2)C1 CC1(C)CCC(C(N2CCOC(C)(CNC(C3CCS3(=O)=O)=O)C2)=O)CC1 C1(CNC(C(CCC)OC)=O)CC2(CCOCC2)CN1C(C1CNC(=O)C1)=O C(=O)(C#CC1(C)CCCO1)NCCC1(C(=O)NC(C(CCC)C)CO)CC1 C1(O)(CC(=O)OC)CN(CC(c2nc(C)no2)(C)C)C1 N1(C(C=C(C)C(=O)O)=O)CCc2c(C(=O)Nc3cc(Cl)ccn3)csc2C1 N1(C(C2(CCC=C)CCCC2)=O)CCCC(CNC(=O)CN(C)CC)CC1 c1(C(N2C(C(N)=O)COCC2)=O)ccc2oc(N3CCCCC3)nc2c1 N1(C(C(c2ccc(CC)cc2)C)=O)CCN(C(C2CSC2)=O)CC1CC C1(CCCNC(CC2C(C)(C)C2)=O)CN(C(=O)CCC2OCCO2)CCO1 C(=O)(CC(F)(F)C(F)(F)F)NCCC1CN(C(C(COC)C)=O)CC1C C1(CNC(C=CC)=O)CC2(CCOCC2)CN1c1nnc(O)s1 C=CCN=C(NCc1cncc(C)c1)NC(C1CCOCC1)C.C1(N)CCCN(C)C1=O C1(NC(c2cn(C)nc2O)=O)CCN(C(C2COC(=O)N2)=O)CC1F c1(C(N2CC3CN(C(c4cc(Cl)ncc4Cl)=O)CC3C2)=O)cc(F)c(F)c(F)c1 CCC1=NOC(CC(=O)NCCCN(CCCNC(C23CCC(CC2)C3)=O)C)C1 C1(N(C(=O)CCCSC)CC)CCN(C(C2CCCN2Cc2cccs2)=O)CC1 C(C(C)(CC(C)C)NC(c1ccsn1)=O)NC(COCCOCC#C)=O C(c1ccc(OCC)c(OCC)c1)=CC(=O)NC1(CC=C)CC1 C1(NC(COC2CN(C(CCOC3(C#C)COC3)=O)C2)=O)CCCN(C)C1C c1(-c2c(C(=O)NCCNC(c3cc(C#N)[nH]c3)=O)con2)ccc(Cl)cc1Cl c1(SC)ncc(Br)c(=NC(=O)N(C)Cc2cc3cc(F)ccc3o2)[nH]1 C(=O)(C(C)(C)N(C)CCN(C(=O)CC1CCOC1)C)N(CC#C)CC N1(C(C(CC)SC)=O)CC2(CCCCN(C(C3(c4cccnc4Cl)CC3)=O)C2)C1 c1(C(=O)NCC2N(C(C(C)OC3CCCCC3)=O)CC2)c(Cl)cccc1Br CC(C)CC(CC(=O)N1CC(C)(C)C1C(C)C)NC(=O)C(C)n1ccnn1 C1(C(N2C(CC)CC(O)C2)=O)CC1C1CN(C(=O)C=C(C)C2CC2)C1 C(CCCCCC(C)(C)C)NC(N1CC2CC(C(=O)OCC)C2C1)=O CCC(CC)(C(=O)NC(C)CC(C)NC(=O)C(C)(CC)C(N)=O)C(C)C N1(CC(=O)NCC2CCCCC2NC(=O)Cn2cnnc2O)CCS(=O)(=O)CC1 S(=O)(=O)(c1ccc(NCC2C=CCC2)c(Br)c1)NC1C(C(N)=O)CCCC1 C1(CCN(C(C2C(C=C)C2)=O)C)CCCCN1C(=O)CCCc1nc(CC)no1 C12(C(=O)NCC(C)CNC(c3ccccc3CO)=O)CCCC(C1)C(=O)N2 N1(C(C2(CCC)CCC2)=O)CC2CCC2(CC(=O)NC(C)CCF)C1 N1(Cc2c(C(=O)OC)cco2)CCC(NC(C2(C(N)=O)CCC2)=O)C(F)C1 Cc1cc(C(=O)N(C(C(=O)NCCOCC(C)(C)O)C2CC2)C)cnc1O CCC(CC(=O)NC12CC1CN(C(=O)C=C=C(C)C)C2)C1CCC1 C(=O)(CCN(OC)C(=O)OC(C)(C)C)N1C(NC(C)=O)C(C)CC1 CCC(C)C(C(=O)NCC(C)(C)C#N)N(C)C(c1scc(C)c1C)=O C1(CNC(C2C3CCC23)=O)C2CCCC1N(C(=O)C=Cc1ccc([N+](=O)[O-])s1)C2 Cc1ncc(C(N2CCSCC2CCNC(c2cn(C)c(C)n2)=O)=O)c(C)n1 C(=O)(C(C)(C)C(F)(F)F)NCC1(CCNC(C(C(C)C)(C)O)=O)CC1 C(=O)(CC(C)CC(C)C)N(C1CCN(C(c2ccc3nn[nH]c3c2)=O)C1)CC c1(C(C)C)ccccc1CSC(c1ccccc1Cl)C N1(C(C2(COCC)CCCC2)=O)CC(NC(c2cc(Cl)cn2C)=O)C(C2CC2)C1 C1(O)(CNC(NC=CC(=O)C(F)(F)F)=O)CCCC12CCOCC2 C(=O)(C1=NOC2COCC12)NCC(C(=O)N(C)Cc1cc[nH]n1)CC1CCCC1 N1(C(C2CCC(CN(CCC)C)C2)C(=O)NC2CC2)CCCC(C(C)(C)C)C1 C1(CC=C)(NC(C(CCC)NC(N)=O)=O)CCCN(C(C2(CC(C)C)CC2)=O)C1 Cc1cnc2cc(C(N3CCC(C)(C)C3CNC(=O)C(=O)NC(C)CC)=O)nn2c1 CC(CC(=O)NCC1CCCC1NC(c1nsnc1O)=O)c1ccco1 C(=O)(C1CC=Cc2ccccc21)NCC(=O)NCC1CCC1NC(=O)C(F)(F)F Cc1c(F)cc(C(=O)NC2CCN(C(C3CCCO3)=O)CC2)cc1F C(CC1CCC1)(C(=O)NC1CC(CNC(C)=O)C1)OC.C1(C2CCC2)C(=O)N1 Cn1c(=O)c(C(=O)Nc2ccnc(-c3cc(F)ccc3N)c2)cc2ccccc12 CC(C)(CO)C(=O)N1CC(CO)(NC(c2cn(C3CCC3)nn2)=O)C1 N1(C(c2c(CC)n(C)nn2)=O)CCCN(C(C2CC(C3CC3)=NO2)=O)C(C)C1 c1(C(=O)NC(C2CN(C(COCCC=C)=O)C2)C)cccc(OC)c1F c1(OC)ccc(Cl)c(C(=O)NC2CCCC2NC(=O)C2=CCCCC2)n1 N(C(=NCCC(C)C)NCc1cscc1C)Cc1cnc(OC)c(Cl)c1 C1(C(=O)OC)Cc2cccc(OC)c2O1.c12cc3c(ncnc3s1)NC2 N1(C(CC(C)OC)=O)CCN(C(c2cccc(F)c2C)=O)C(CC2CC2)C1 C1(C(=O)NC2CC(CNC(C(C3CCOCC3)OC)=O)C2)CCCC1(C)C N1(C(C2(CCC)CCC2)=O)CCC(CF)(NC(=O)C(C)Sc2nncn2C)C1 C1(F)(CNC(CN(C)C)=O)CN(C(=O)CC(O)C2CC2)C1 Cc1ccc(C(N2CC(OCCNC(=O)CCc3cc(C)sc3C)C2)=O)nc1 Cc1cc(NC(=O)CCN(C(=O)C(C)OCC2CC2)C)ccc1F CCC(CC)C(F)C(=O)N1CCC(C)(CC(=O)NCC(O)COC(C)C)C1 C1(NC(c2n[nH]c(CC)c2Br)=O)CCSC12CN(C(c1cnsc1C)=O)C2 C(=O)(C1=C(C)CCOC1)NC1(CO)CC(OC)C1.C1(C=O)COCCN1C N1(C(C(C)NC(C)=O)=O)CC2CCCC2(CNC(=O)Cn2cc(C(C)O)nn2)C1 Nc1ccc(NCCC(=O)N2CC(n3cnnn3)C2)cc1 c1(C(=O)NCC2(C)CCC(NC(CSCC=C)=O)C2)coc2cccc(O)c12 c1(C(=O)NC2(CNC(C(CCC)C)=O)CCC2)cc(C(=O)OC)c2n1CCOC2 C1(C(=O)NC2CCC(N(C(C3CCCC(C)C3)=O)C)CC2)CCn2ncnc2C1 C(=O)(C1Cc2ccccc21)NC1C(F)(F)CCN(c2nc(C)nc(=N)[nH]2)C1 CCC(C(=O)N(C1CC(NC(=O)Cc2cccc(C)c2Cl)C1)C)C(C)O C(Cn1cccn1)(C(=O)NC1(CCO)CC1)N(CC)CC.C1=CCNC1=O n1(CC(N2CC3CC(C2)N(C(C24CCC(C2)C4)=O)C3)=O)ncc2ncccc12 c1(C(=O)NCC(CNC(C2(CO)CC2)=O)OCC)c(C)[nH]c2ncccc12 CN1CCN(C(C2(CO)CCC2)=O)CC1CNC(c1cc(C(C)(C)C)nn1C)=O N1(C(CCOCCOCC)=O)CCCC(C)(C)C1C(=O)NCC(C)(O)CCO C1(NC(CC(c2c(C)noc2C)C)=O)CN(C(c2cccc(N)c2)=O)CCC1O c1(N(CC(C)OCC)CC=C)ccc(S(=O)(=O)NC2CC=CCC2)c(Br)c1 C12(C(N(CC(C)NC(C(=O)NC)=O)C)=O)CCC(C(F)(F)F)(CC1)C2 CCC(CC(=O)NCCC1CCCN(C(=O)CC#N)C1)OC CC1CN(C(=O)CCn2cccc2)CCC1NC(=O)CCn1cc([N+](=O)[O-])cn1 C(=O)(C1Cc2ccccc21)N1C(CNC(c2cc(C)n(CC3CC3)c2C)=O)CC1 c1(C(CNC(C2(N(C(C3(SC)CCC3)=O)C)CCC2)=O)OC)nnnn1C C1(CCNC(CCSc2nc(C)[nH]n2)=O)CN(C(c2cnc(O)s2)=O)CCO1 C1(CNC(C2(C)N(C)CC(O)C2)=O)CN(C(=O)CC2=CCCC2)CCC1(C)C c1(CCC)ccc(C(=O)NCC2CCC(NC(=O)CC3CC4(CC4)C3)C2)cc1 C1(NC(C(C)CN2CCOCC2)=O)CC2(C1)CC(NC(C1(C)CC=CCC1)=O)C2 c1(NC(=O)CC2C=CC(OC(F)F)C2)cccc(N2CCCCC2=O)c1 c1(C(N2CC(CC(C)NC(C3(CO)CCCO3)=O)C2)=O)ccc(F)c(C(N)=O)c1 N1(C(C(CC)C)=O)CCC2CN(C(C3CCSC3)=O)CC12 C1(OCC)CC2(C1)CC2C(=O)NC1CCCC(NC(=O)COc2cccnc2)C1 CC(CS(C)(=O)=O)C(=O)NCCC1CCN(C(=O)C=CC(C)(C)C)CC1(F)F C(=O)(C(CNCCCN1C2(CCC2)CS1(=O)=O)CSC)OC.c1(OC)ccccc1.OC Cc1onc(C2CCCC2)c1C(N1CC(NC(C2CC2(F)Cl)=O)C1)=O c1(CC)cc(C(N2CCN(CC(F)F)C(C)C2)C(=O)NCC(F)F)cc(F)c1 c1(CC(=O)NCC2C(NC(C=C3CCN(C)CC3)=O)CCC2)cccc(F)c1O c1(C(=O)NC2C(C)CN(C(c3ncc(F)cn3)=O)CC2)ccc2nc(O)[nH]c2c1 N#CC1CN(C(c2ccc(O)nn2)=O)CCN1C(=O)CCc1cc(C2CC2)no1 Cc1ccc2c(c1)CCC(C(=O)NC1(CCCNC(c3csc(=N)[nH]3)=O)CC1)O2 C1(C(C)NC(=O)Cc2cn[nH]c2)CCCN(C(c2ccc(F)cc2)=O)C1 CCCC1CCCN1.c1(CNC(c2ccccc2)=O)cc(Cl)cc(OC)c1OC C1(CC)CN(C(c2onc(C)c2C)=O)CCC1NC(c1ccc(CO)c(F)c1)=O C(=O)(C1=CNC2=NCCCN12)N1CC2CCN(C(c3n[nH]c(C)c3C)=O)CC2C1 CCC(C)(O)C(=O)NC1C=CCN(C(=O)CCNS(C)(=O)=O)C1 C=Cc1cncc(C(=O)NC(C)CC(C)NC(c2c(Cl)c(C)nn2C)=O)c1 C(=O)(C1=CNC2=NCCCC2=C1)N1CC(NC(CS(CCCCOC)(=O)=O)=O)C1 CN1CCC(NC(=O)C(CC2CC2)NC(c2ccc[nH]2)=O)C1=O C(=O)(CP(C)(C)=O)NCCC1CC(NC(C(CC)N(CC)CC)=O)C1 C(=O)(C1=C(Cl)CCCC1)NCC(C1CCCC1)NC(c1c(C)ncnc1C)=O CC(C)(O)CC(=O)NCC(C1CCC1)NC(c1cnc(C(F)(F)F)cn1)=O Cc1ccc(Br)c(CNCCCC2CCN(C(=O)OC(C)(C)C)CC2)n1 c1(C(=O)NC(C2CCN(C(C(C)OCC)=O)CC2)C)c(C#N)cnn1C C(=O)(CCC(N)CC(C)(C)C)N(CCS(=O)(=O)NC(C)=O)CC.C1(=O)CN1 N1(C(CC(=O)OCC)=O)CC(NC(c2cncc(-n3ccnn3)c2)=O)CC12CCC2 c1(C(N2CC3CCN(C(CSCC)=O)C3C2)=O)cnc(O)c([N+](=O)[O-])c1 c1(C(=O)NCC2C(C)CN(C(=O)CO)CC2)cc2cncn2c(O)n1 C1(C(N(C2CCN(C(c3cn(C4CCCCC4)nn3)=O)C2)CC)=O)C=CCCC1 C1(N(C(C(CC)N(C(C2CC(C#C)(O)C2)=O)C)=O)C)CCC(C)(C)CC1 c1(-n2c(CC(C)CCOCC)nc(CCCC)n2)cc(Cl)c(Cl)cc1Cl N1(Cc2nc(C)sc2)CCC2(CCN(C(C3CCN(C(C)(C)C)CC3)=O)C2)C1 N#CC1CCCC1NC(=O)CCN(C(=O)C(C1CCCCC1)O)CC1CC1 c1(C(=O)NCCN2CCN(C(C(C)CC3CCC3)=O)CC2)nccc2[nH]ccc12 N=c1[nH]cncc1C(=O)NC1CC(CCNC(=O)CCc2cccc(F)c2)C1 C1(C(=O)NCC2(O)CN(C(c3cn(C(C)(C)C)nc3)=O)C2)CCC(=C(F)F)CC1 N1(C(COC)=O)C2CCC1CC(O)(CNC(c1nc(C)[nH]c1C(F)(F)F)=O)C2 c1(C(N2CCCC3(C2)CN(c2nnc(CO)s2)C3)=O)ccc(C#CC2CC2)cc1 C1(C(=O)NOCCC(F)F)CC2(CCC2)CN1C(=O)CC1CCCC12CC2 CCC(C)C(=O)NCC(C)NC(c1cnn(-c2nccs2)c1)=O Cc1cc(CCC(=O)NC2CC2CNC(c2ncsc2NC(C)C)=O)cc(C)n1 C1(O)(CCC(=O)O)CCN(C(c2cccc(F)c2)CF)CC1 c1(C(=O)NC(CN(C(C(C)OCC#C)=O)CC)C)cc(C)c(-c2ccccc2)s1 C(c1ccc(F)nc1)=CC(N1C(C(=O)NCC(n2cc(C)nc2)(C)C)CCCC1)=O N1(C(CCCc2ccc(C)s2)=O)CC(NC(C2CC2c2ccsc2)=O)C2(CC2)C1 C1(CC(N2CCCC(N(C(=O)C3=CCSC3)CC)C2)=O)CCC(C)(C)CO1 N1(C(C2(COC)CC=CC2)=O)CCC2(CCCN2C(=O)C(=O)NCC(F)F)C1 N1(c2ccc(CO)c(Cl)n2)CCN(CSc2c(Cl)cncc2Cl)CC1C(F)(F)F C1(C(N2C(CN(C(Cn3ncc(C)c3)=O)C)CCC2)=O)CCCNS1(=O)=O CCC(C)(C(=O)N(C)CC1CCN(C(c2cnn(-c3ccccc3)n2)=O)C1)OC C1(NC(c2ccc(OCC)o2)=O)CC1C1CCCN(C(c2c(C)noc2N)=O)C1 C(=O)(C1CCCc2nc[nH]c21)N1CCC(C)(CNC(=O)CNC(C2CCC2)=O)C1 Cc1cc(F)cnc1C(=O)NCC(C1CCN(C(C2(Cl)CC2)=O)CC1)F C(CN=c1ccc(S(=O)(=O)N2CC(C)OC3(CCC3)C2)c[nH]1)SCCC=C Cc1cc(CCNCC(C)COC(C)C)ccc1[N+](=O)[O-] C(=O)(CC(=O)N1CC(O)(c2cnn[nH]2)C1)OC(C)NC1(C2CCCCO2)CC1 c1(C2CCN(C(C3(C#N)CC=CCC3)=O)CC2)nc2c(Cl)cccc2[nH]1 N1(C(CC=CCC)=O)CCN(C2CN(C(=O)COC3CC3(F)F)C2)CC1 C1(C2(CC(=O)NC(C)(C)C)CC2)CN(C(c2nn(C)cc2Cl)=O)CC1C(=O)O.CC c1(C(=O)NCC2OCCN(C(C=CCN(C)C)=O)C2)c(C)nn(CC(F)F)c1Cl c1(NC2CC(CNC(C3CCc4cncn4C3)=O)C2)ccc([N+](=O)[O-])cc1Br c1(C(N2C3CN(C(C(C=C=C)C)=O)C(C3)C2)=O)cnn2c(Br)cccc12 c1(OC)c[nH]c(C(=O)NCCC2CN(C(c3ccnc(Cl)c3OC)=O)C2)cc1=O c1(CN(C)C)cn(CC2CCN(C(=O)Cn3nnc(-c4cccs4)n3)C2)nn1 N1(C(c2cccc(OC(C)C)c2)=O)CC2CCC1CN2C(=O)CCCCCO c1(C(=O)NC(CC)CNC(=O)C(c2c(C)n[nH]c2C)C)cc2c(nc1O)CCC2 c1(C(=O)NCCC2(C(N(CCCCN(C)C)C)=O)CC2)ncc[nH]c1=O C=CCC(CC)C(=O)N1CCN(C(=O)CCc2ncc(C)[nH]2)CC1CC c1(OC)ccc(Cl)cc1C1(C(N2C(NC(=O)N=c3nc[nH]s3)CC(O)C2)=O)CC1 C(=O)(C(C(F)(F)F)C(F)(F)F)NCC1(NC(=O)CS(=O)(=O)CCO)CCC1 Cc1nn(C)cc1CC(N1CSCC1C(=O)NC1CC(C)(C(N)=O)C1)=O Cc1c(C(N2CCCC(O)(CNC(=O)C(O)CC(F)F)C2)=O)sc2nccn12 C=C1CC(C(N2CC(C)(CCO)C2)=O)(C(=O)NC(=O)OC)C1.C12CC1(C)C2 C1(C(=O)NCCOCCOC)CN(C(C2(n3cnnn3)CC2)=O)CC1(F)F N12CCN(C3(CCCC3)C1=O)CC2=O.c1(C(c2ccccc2)C)nn(C)cc1O CC1Cn2nc(C(=O)NC(CNC(C3CCS(=O)CC3)=O)C3CC3)cc2C(=O)N1 N1(C(c2cccc(C)c2)=O)CCC(NC(=O)COC(F)(F)F)C(CO)C1 C12(CC)CCC(N=c3cc(C)nc(NCc4cnc(Cl)c(C)c4)[nH]3)(CC1)CO2 C1(OC)(OC)CCC1C(=O)NCC(C)CNC(=O)C(C)Cc1cccnc1 Cc1cc(C(=O)NCC(C)(C(C)C)NC(=O)CC(N2CCCCC2=O)C)ncn1 C(=O)(CC(O)CC(C)C)NC(CC1CCCC1)CO.CCC1CCC(=O)N1 C(=O)(C(O)C1CN(C(=O)C(=O)NCCC)C1)NC(C#C)C1CC1 N1(C(C2C(OC(C)=O)C2)=O)CCN(C(c2occ(C)c2C)=O)CC12CCC2 C(=O)(CC(C)(C)CC(=O)N1CC(CCNC(c2cccc3nc[nH]c23)=O)C1)OC C(=O)(C#CC1CCCC1)N1CCC(NC(c2ccn(C(C)C)c(=O)c2)=O)C12CC2 N1(C(c2ccccc2)C)CCC(F)(CNC(=O)CC2NC(=O)NC2=O)C1 O=C1CC(=O)NC(C(=O)NCCCCCC2CN(C(C3CN4CCC3C4)=O)C2)C1 c1(SC(CCO)Cc2cccc(F)c2)nc2cc(Br)c(F)cc2s1 c1(C(=O)NCC2CCN2C(C2CC2Br)=O)ccn(C2CC2)n1 c1(C(=O)NCC2C(C)CN(C(C3CCCN3C=O)=O)C2)cnc2ncc(Cl)cn12 CC(C)C(C(=O)N1CCN(CC(C)NC(=O)CC2CC2)CC1)N(CC(C)(C)C)C c1(C(N(C2CCCC(N(C(C=CC=CC)=O)C)C2)C)=O)cccc2c1OCCN2 c1(C(=O)NCC(C(C)C)NC(C(CC(C)C)O)=O)cn2ccc(F)cc2n1 C1(C(N(CC(C)(C)CNC(=O)C2=CCCCC2)C)=O)CCC2(CC1)CC(F)C2 C1(NC(C2(CC)CCNC2=O)=O)CCCCN(C(=O)CC2(CN(C)C)CC2)C1 C1(C(N(C(C)CN(C)C(c2c[nH]nc2C(C)(C)C)=O)C)=O)CC1C1CCC1 C1(C(=O)Nc2cccc(O)c2)COCCN(C(c2ccc(F)cc2I)=O)C1 N(C1c2ccccc2CC1NC(=O)CCCCC(F)(F)F)C(CCNC(N)=O)=O C1(OCCNC(=O)CSc2nc[nH]n2)CCN(C(C2CC23CCC3)=O)C1 c1(C(=O)OC)ccc(NC(C2CC2CN(c2nccc(OC)n2)C)=O)c(I)c1 C1(C(=O)NCCCC(C)(C)NC(=O)CCOC2CCOCC2)CC2(C1)CC2(F)F c1(OCCC)ccccc1COC(c1sc(Br)nc1C)=O N1(C(C(CCCOC)C)=O)CCC2CCCC12C(=O)NC1CN(C(C)C)C1 C1(NC(c2cc(C)nnc2)=O)CC(C(=O)NCc2cc(O)ccn2)C12CCC2 C(CCNC(=O)CSCCC=C)(C(C)C)NC(c1n(CC#C)ncc1)=O CCC(CC(=O)NC(C(=O)NC)C(C)C)NC(=O)CCN(C1CCC1)C c1(NC(C2(C)CCCN(C(c3cc(F)ccc3F)=O)C2)=O)c(F)cccc1C#N C(=O)(C1=C(C#N)CCC1)NC1CCC(CNC(c2c(NCC)c(N)ccc2)=O)C1 N1(C(C2CC(C(F)(F)F)(OC)C2)=O)CCN(C(=O)Cc2cocn2)C(CO)C1 OC1CN(N2CCN(C3CCOCC3)CC2)C2(CCCC2)C1 CCCC(CCCO)C(=O)NCCCCNC(c1cnn(C2CCOCC2)c1)=O N1(C(c2ccc(OC)c(C3CC3)c2)C(=O)NC)CCN2CC(C)CC2C1 CC1CN(C(C2(CC(F)F)CC2)=O)CCC1C(=O)NCC1CC(CF)C1 C1(C(=O)NC(CNC(C2(CC)CCC2)=O)C2CCC2)OCCC1c1ccccc1 c1(C(=O)NC2C(NC(COCC=C)=O)CCC2)cnc2cc(O)ccc2c1 C(=O)(C(C)(F)C(=O)NC1CC(CNC(c2cnc(-c3cccs3)s2)=O)C1)OCC c1(NCCCC2C(F)(F)C2)cncn1-c1ccccc1 C1(C(N2CCC(C#N)CC2)=O)C2C3CC4C1C2C34C(=O)Nc1ccsc1 C(=O)(C1=CC(O)CCC1)NCC(CCOC)NC(c1ncccc1F)=O N1(C(c2cccc(OC)n2)=O)CC2CCC(C1)C2CNC(=O)CC(C)C(C)C CC(C)CC(C)(CNC(=O)C(O)c1cnc[nH]1)NC(=O)CC(=O)NCC1CC1 N1(C(c2c(C)nc(CC)o2)=O)CC(NC(=O)CN2CCC(C)CC2)C2(CCC2)C1 O(NC(=O)CCC(C)(C)NC(C1C=CCCCC1)=O)CCC=C N1(C(C(C)=O)=O)C2CCC1CC(n1cc(C(=O)NCCCCCO)nn1)C2 n1(CC)ncc(Br)c1C(=O)NCCCCC(C)NC(=O)CCc1nc(C)no1 N1(C(CCCSC)=O)CCC(NC(=O)Cc2nc(-c3ccccn3)oc2C)C1C C1(OC)CC(NC(=O)CCc2cncn2C)CN(C(c2cncc(Cl)c2)=O)C1 CCCC(C)CC(=O)NCC(C)NC(c1sccc1-c1ccc(OC)c(F)c1)=O C1(CNC(c2scc(C)c2)=O)CCC(C)(C)CN1C(C1CC1CN(C)C)=O C12(CNC(COC(CC)C)=O)CC(CN1C(=O)CCCc1nc(C)no1)C2 Cc1c(C(N2CC([N+](=O)[O-])C2)=O)sc2nc3n(c(=O)c12)CCC3 c1(C(=O)NCC(C)NC(C(CC)OC2CCCC2)=O)cc2c(=O)[nH]ccn2n1 Cc1ccc(C(N)=O)cc1C(=O)N(CC(O)CNC(C1CCCC1(F)F)=O)C C1(NC(CCNC(C)=O)=O)CN(C(c2cccc(O)n2)=O)CC1C(F)(F)F N1(CC)CCCCC1CNC(=O)CC(C)(C)NC(c1cnc(C)[nH]1)=O CCCC(O)C(=O)N1CCC(OCCNC(C2CCN(C(C)=O)CC2)=O)C1 N1(C(Cc2cc(C)on2)=O)CC(CNC(c2ccc(CO)cn2)=O)CCC1C c1(N2CCCC(C)CC2)nc(N(CCCCCO)C)c2c(ncn2C)n1 C1C(C)C(=O)N(C2CCCC2)Cc2occ(c2)C(=O)O1.n1(CC)cccn1 C1(=CC(=O)NCC(CCCC)NC(c2cc(C#N)cn2C)=O)CN2CCC1CC2 Cc1cnc2n1CC(C(c1nnnn1C)NCC1=CC(=O)OC1)CC2 c1(C(C(=O)NC2CN(Cc3nccc(OC)c3)CC2O)C)ccc(F)cc1F Cn1nc(C(N2CCC(CNC(C3CC(O)C3(C)C)=O)CC2)=O)cc1O CC(CC(C)NC(=O)C(=O)C1CCCC1)NC(c1sccc1Br)=O C(C1CCN(C(=O)CCc2cnco2)CC1)=CC(=O)NCC(COC)O c1(CC)[nH]c(C(N2CC(NC(C3=C(N)CCN3C)=O)C(CC(C)(C)C)C2)=O)nc1Cl C(CC(C(=O)NC(C)C)N(CCC(F)(F)F)CCN(C)C)SC.c1(CN)ccccc1 C1(C(=O)NCC2(CC)CC2)CCCN(C(=O)C(c2ccc(C)o2)C)C1C N1(C(=O)CC2C=CCCC2)CC2CCCC(C1)N2C(c1ncc(Cl)c(O)n1)=O C1(OC(C(F)=C(C)C)=O)CCN(OC)CC1 CCC1=NOC(CC(=O)NCCN(C(=O)C(O)c2ccsc2)C)C1 c1(OC)noc(C(N2CCCC2CCNC(=O)CSCCC(C)C)=O)c1Br c1(OC)cc(C(=O)NCCC(C)N(C)C(C2(CC(C)C)CC2)=O)n(C)n1 C(C(=O)NC1CCN(C)C1=O)(C(C)C)NC(C1(OC)CCCC1)=O c1(CO)ccc(C(c2nnnn2C2CCCCC2)NCCc2cc(I)c[nH]2)nc1 N1(C(c2cccc(CC)n2)=O)CCC2(CCCC2NC(c2cccc(C)c2)=O)C1 C=C(Cl)CC(C(=O)N1CC(c2ncc[nH]2)C1)NC(C1CCC(=O)N1)=O C1(OC)CCC12CC(C(=O)NC1(CO)CN(C(=O)CC(C)C3CCCO3)C1)C2 c1(N2CCCC(C)(CNC(C3(O)CCOC3)=O)C2)[nH]cnc2nc(Cl)cc1-2 c1(C(N(CC(C)NC(c2c(Cl)cnc(OC)n2)=O)C)=O)cncc2c1CCCC2 N1(C(C(CCC)CCC)=O)CC2COCC(C1)N2C(c1cc(Cl)cnc1Cl)=O C=CCCC(C(=O)NC1CCOC(C)C1)NC(c1cccc(C)c1C)=O C1(c2nc(C)nn2-c2cn[nH]c2)CCc2ccccc2N(CC(=O)N(C)C)C1=O CON(CCC(=O)NCC1C2CCCCC12)C(=O)c1cnc(N)cn1 Cc1cccc2[nH]c(C(N3CCN(C(C4(CN(C)C)CC4)=O)C4CC34)=O)cc12 C(=O)(C(CC(C)(C)C)NC(=O)CCC1CC(C)C1)NC(CCC)CCO n1(CC(=O)N(CCNC(CCOCCC)=O)C2CC2)ncc(Cl)c1C N1(C(C2CN(C(CC)CC)C(=O)C2)=O)CCCC(CCC)(NC(=O)CSC2CC2)C1 C1(C(=O)Nc2cccc(CNC(C3CC4CCC3C4)=O)c2)CCc2nnnn2C1 c1(C(N(C(C#C)C)C)=O)n[nH]cc1NC(C1(F)CC1)=O C1(OC)(NC(C2CCN(C(=O)CCC3CC(OC)C3)C2)=O)CCCC1 C1(O)(C(=O)NCC2C(NC(C(C)NC(N)=O)=O)C2)CCc2ccccc2C1 C=C(Cl)CCC(=O)N1CC(C2CN(C(=O)C(C3CCCC3)OCC)CCO2)C1 c1(C(=O)NCC2(NC(c3c(CN(C)C)nns3)=O)CCC2)cc2cnccc2[nH]1 C1(CNC(c2ncc(OC(C)C)nc2)=O)CN(C(=O)C2=CCCCC2)CCC1C C1(NC(c2onc3sccc23)=O)CCCC12CN(C(=O)CN1CC3CCC1C3)C2 C=CC(C)CC(=O)N1CCC(OCCNC(c2n[nH]cc2C)=O)C1 O=C1CS(=O)(=O)CC(C(=O)NC2CCC(CNC(=O)C=CBr)C2)N1 c1(-c2cn(C3CC(Nc4cc(NC(C)=O)ncn4)C3)nn2)cc(O)ccc1C c1(C(C)C)ccc(C(=O)NCC(CO)NC(=O)C(=O)C(C)(C)C)c(F)c1 C(=O)(C1CC(=O)c2ccccc21)NCC(C)CNC(c1[nH]nnc1C(F)(F)F)=O C(=O)(C(C(=O)OC(C)(C)C)C(C)(C)C)N(C(C)C)Cc1cn2ccccc2n1 C12(SC(C3CCC(n4cc(C(C)O)nn4)C3)=O)CC3CC(CC(C3)C1)C2 c1(CC(=O)NCC(C)NC(=O)C(O)(C2CC2)C2CC2)nocc1C(C)C C(C(=O)NCc1ccc(C#C)nc1)(C(C)(C)C)NC(C(=O)NCC#C)=O C=C(C)C1OCCCC1C(=O)NC1C2CN(C(c3cn[nH]c3)=O)CC12 c1(C(=O)NCC2C3CCCC2NC3)c(F)cc(Br)cc1F c1(NC(C2(CC)CCN(C(C3C(C)(C)C3(C)C)=O)CC2)=O)cnn2c1CCCC2 c1(C(N(C2CCCCC2)CCNC(CCSCCCC)=O)=O)cc(NC)ccc1F c1(CN2CC(NS(CCOCC)(=O)=O)C(F)(F)C2)c(F)cc(Cl)cc1Cl C1(C(N2CCCC(CN(C)C(c3ccc(F)c(F)c3)=O)C2)=O)CC(F)C(=O)N1C C1(NC(c2nc(C)sc2)=O)COC2(C1)CN(C(c1cc(C(N)=O)ccn1)=O)C2 c1(OC)cc(CC(=O)NCC2(C)CCCN2C(=O)Cn2nc(C)oc2=O)ccn1 C1(C(=O)NCC2(C=C)CCC2)CSCCN1C(=O)CC(CC)C1CC1 CC1(CNC(C2=NOCC2)c2nnnn2-c2ccc(F)cc2)CC1(Cl)Cl C(=O)(C#CC1(C)COC1)N1CCC(OCC(=O)NC(c2nnc(C)o2)C)C1 C1(SCC(N2CCC(O)C2)=O)CCS(=O)(=O)C1 C1(CC)CCCCN1C(c1conc1CNC(=O)CC1CSCCO1)=O CC1(Cc2ccccc2C(=O)NOc2n[nH]c(=N)[nH]2)CCCCC1(F)F C(=O)(C1CCc2nnc(C)n21)N(CCCNC(c1cc(C)c(N)c(C)c1)=O)C N1(C(C(C)OCC)=O)C(CNC(=O)C(F)(F)c2ccncc2)CC2CCCC12 C1(NC(c2csc(F)c2)=O)C2CC(O)C1N(C(c1cc3ccccc3o1)=O)C2 N1(C(c2cccc(OCCO)n2)C(=O)NCCCC)Cc2ncsc2C1 c1(CNC(=O)NC2(COCC)CCCC2)ccccc1CNc1ccncc1 C(=O)(C1Cc2c(Cl)cccc21)NCCC(=O)Nc1c(C)nn(C)c1-n1cccn1 N1(C(C(C2CCNCC2)OC)=O)CCc2c(CO)cc(Cl)cc2C1 C(C)(CC(C)NC(c1coc(C2CCC2)n1)=O)NC(C(C)C)=O C(=O)(CCCCC1CCCC1)NC1(C)CC(c2cccc(C)c2)C1.C(=O)O C(=O)(N=c1ccn(C(C)C)[nH]1)C1N(C(c2c(C)c[nH]c2)=O)CC2CC21 C(=O)(CC(F)(F)C(F)F)NC1C(NC(C(c2cc(C)cc(C)c2)C)=O)COC1 N1(C(C(CCCC)=O)=O)CCC2(CC1)CN(C(=O)CCC1CCN(C)C1)CCO2 C=C(Br)CC(C)(C)C(=O)NC1CCN(C(C2CC(=C3CCC3)C2)=O)C(C)C1 C1(C(=O)NCC2CC3CN(C(CC(C)C)=O)C2C3)Cc2nn(C)cc2C(=O)N1 C1C(C2CCC2)CC(=O)N1.C1(NC(C2C(C(C)(F)F)C2)=O)CCN(CC2CC2)C1 C1(NC(C(CCC)NC(c2ccc(CO)cn2)=O)=O)COCC(C)(C)C1 Cc1nn(C)c(N)c1C(N1CC(C2(NC(C3CS(=O)(=O)C3)=O)CC2)C1)=O CN(C(=NCC1CCC1)NC1CCOC1)Cc1cc(F)ccc1N(C)C Cc1nccc(C(N2CCC23CN(C(=O)CN2CCOC2=O)C3)=O)c1C c1(C(=O)NC2CCN(C(CCOCCOCC)=O)CC2C)cccn2cnnc12 N1(C(c2c(CC)cns2)=O)CCN(C(=O)CCC2CC2(F)F)CC1CC(=O)NC c1(NC(=O)C(N2CCC(c3nccs3)CC2)=O)cc(C(F)F)ccn1 N1(C(CCSCCC)=O)CC(C2CN(C(=O)CCc3nc(CC)no3)C2)C1 c1(C(=O)NCCC(C)NC(=O)CCCCc2cnn[nH]2)ccccc1SC(F)F c1(CNC(CC(CNC(c2c(CC)n(C)cc2)=O)O)=O)cc(C)cnc1F c1(C(N2CC(NC(C(CC)O)=O)C(O)C2)=O)ccc(NC(=O)C(C)C)cc1O C1(OC)CS(=O)(=O)CC1NC(c1scnc1-c1cccnc1N)=O N1(C(C)=O)CCCC(C(C)NC(=O)C(c2ccc(Br)s2)C)C1 N1(C(C(=Cc2cnc[nH]2)C)=O)CC2(C1)CN(C(C1CC3CCC1C3)=O)CC(C)(C)O2 C1(C(C)O)CCN(C(C2CN(C3COC3)C2)=O)CC1.C12(CCC1)C(=O)NC2 C1(NC(C(C)(C)OCC)=O)CN(C(c2c(C)cccc2C)=O)Cc2nccn2C1 Cc1ccc(SCC(=O)NCc2ncccc2C(=O)NCC(=O)N(C)O)cc1 C12(C(N(C(CNC(CN(C(=O)OC)C)=O)C)C)=O)CCN(CC1)C2 Cc1nc(NCC2(C)CCCOC2)cc(NC2CC3(CCC3)C2)n1 c1(C(N2CCN(C(c3cc(F)ccc3O)=O)C3CC23)=O)ccc2c(c1)OCCO2 N1(C(C(CNC(C2C(C)C3CCC2C3)=O)(C)C)=O)CCn2nncc2C1 C1(C(=O)NCCC2N(C(Cc3cc(C)[nH]n3)=O)CCCC2)CN2CCN1C(C)C2 CC1CCN(C(c2snc(O)c2Cl)=O)C1CNC(=O)C(F)(F)c1cscn1 C1(CNC(C(=O)NCc2cc(OC)ns2)=O)CCCCC1F C1(N(c2nccc(N3CCCC3)n2)C(c2cc(C#N)[nH]c2)=O)CCNCC12CC2 c1(CC(=O)NCCC2CCCN2C(=O)CCn2cnnn2)cccc(Cl)c1F Cc1nc(C(=O)NCCC2CC(NC(=O)Cc3nncn3C)C2)c(Br)s1 CC(C)CCC(CN(C)C)NC(c1ccc(C(F)(F)Br)nc1)=O CS(=O)(=O)CC(CS(C)(=O)=O)NC(=O)C(=O)NCC(=O)NCC1CC1 C(CCCCC(=O)NCC1CCCN(C(C2(C(F)F)CC2)=O)C1)N(C)C N1(C(C2C(C)(C(F)F)C2)=O)CCC(C)(NC(c2cn(C(F)F)cn2)=O)C1 c1(CC)sc(C(=O)Nc2cc(C(N3CCCCC3)=O)ccn2)cc1Br CC(CCN(C)C)C(=O)NC1(CC(=O)NCCC(O)C2CCC2)CCCCC1 Cc1cc(C(C2CC2)NC(C)C(C)(C)c2nnnn2CC(F)F)c(C)n1C1CC1 C=CCCC(O)CN(C(=O)CCCN(C)C(c1oc(C)nc1CC)=O)C C1(C)(CC)CC(C(=O)NC(C)CCCNC(c2cccnc2C)=O)CCO1 C1(N(C)Cc2nc(CC)on2)CCCN(C(=O)C#CC2CC2)C1 C(C(COC)C(C)C)NC(C1CCC(F)CC1)c1n(CCSC)nnn1 C1(CC)CN(C(c2cc(C(C)C)no2)=O)CCN1C(c1ccsc1C)=O C12(CCCN=C(NCC(C)CO)NC3CCS(=O)(=O)C3)CC3CC(CC(C3)C1)C2 C(=O)(C(C(C)NC(C1CN(C(C)=O)C1)=O)C(C)C)NCC(N(OCC)C)=O CCCC(C)CC(=O)N1CC2(C1)CN(C(C1CC(F)(F)C1(C)C)=O)C2 C1(NC(Cc2c(C(C)C)cccc2)=O)CC2CN(C(=O)CC3(C)CC3)CC12 Cc1nc(=N)[nH]cc1C(=O)NC(C)(C)CCCNC(=O)CC12CCC(CC1)CC2 C1(NCC(Cc2c(OC)cccc2)O)CC2CCC1N(C)C2 CCCCC(C)CCC(=O)NCC1(C)CCN(C(c2ncncc2C)=O)C1 C1(C(=O)NCc2nnc(CC)s2)CCC(O)CN1C(=O)CC(COC)COC N1(C(c2c(CCC)occ2)=O)CC(NC(c2cc(COC)on2)=O)C(N=[N+]=[N-])C1 c1(OCC(C)C)ccc(C(=O)NC2CCC(NC(CNC(N)=O)=O)CC2)nc1 C(=O)(CC(F)(F)C(F)(F)F)NC1C(CNC(c2ccc(C(C)=O)cc2F)=O)CC1 N1(C(C(C)NC(CC)(C)C)=O)CCCC1(C(=O)NCCc1cccc(O)c1)CC O=C(C1=CCCNCC1)Nc1ccc(Oc2cccc(F)c2)c(Cl)c1 c1(Cn2cc(C(CCC)=O)nn2)nn2c(c1C(=O)OCC)CCC2 C1(n2cc(CCO)nn2)C(F)(F)C12CCC2.c1(C2CC(C=O)C2)ccncc1 c1(N2C(=O)CCC2)ccc(C(N2CCC(CNN3CCCOCC3)CC2)=O)cc1 C1(C(N2CC(C(N(CCF)CC)=O)(CC)C2)=O)CC=CCC1CC Cc1ccc(CNC(C2CCN(C(c3ncncc3Cl)=O)C(C)C2)=O)cc1F C1(CNC(C(=O)N(C)C)=O)CN(C(=O)C=Cc2cnc(O)nc2O)CC1(F)F C1(C)(NC(c2ccn(CCN(C)C)n2)=O)CCN(C(=O)CN(S(C)(=O)=O)C)C1 c1(C(N(CCN(C(C(CC)C)=O)C(C)C)C)=O)ccc(-c2ccon2)cc1 c1(C(=O)NC(C(C)NC(C2(CCCC)CCC2)=O)CO)cccc(C#N)c1 C1(CSC)CC(C)(C)CN1C(C(CC#C)NC(c1cn(CC)cn1)=O)=O C(CCCCCCO)NC(C1(CCNC(C2OC3CCC2C3)=O)CC1)=O c1(NC(CC2N(C(c3c(CC)occ3)=O)CC2)=O)ccnc(C)c1C c1(CC(N2C(CNC(C3CCC(=O)N3C)=O)CC(OC)C2)=O)c(C)ncnc1C C(=O)(C(C)(C)CF)NCC(CC)N(C)C(C1CCN(C(C)C)CC1)=O Cc1cccc(C(C)NC(=O)CC2CCCC2NC(C2COCC(C)O2)=O)n1 CCC(CC(C)C)C(=O)NCCCC1CCN(C(=O)Cn2ccnc2C)CC1 C(=O)(CCCCCNC(=O)C(C)C(=O)OC)NCCCCOCC c1(C(N(CCNC(CCC(C)(F)F)=O)CC2CC2)=O)cccc2c1NC(=O)CO2 C(=O)(CCC(=O)NCC1CC(NC(=O)C(C)(C)c2sccc2Cl)C1)OCC N1(C(CC(CCC)NC(=O)CC(C)OC)=O)CC(C)NC(=O)C12CC2 N#Cc1ccc(F)c(C(N2CC3CC2C3C(=O)Nc2cncc(Br)c2)=O)c1 C1(CNCCCCCCONC(=O)NC2C(C)C2)Cc2nccn2C1 c1(C(=O)NC2C3(CN(C(C4CCC(=C)CC4)=O)C3)CC2)cc(S(N)(=O)=O)c[nH]1 CC1(C)OC2(C(N3CCOC(C)(CNC(c4cc(F)c[nH]4)=O)C3)=O)CCC1CC2 c1(C(N2CCC(CCNC(C(C)CF)=O)C2)=O)cc(S(=O)(=O)CNC2CC2)c[nH]1 C(=O)(C(C)(C)S(C)(=O)=O)N1CCC(CNC(C(c2cc(C)cc(F)c2)C)=O)CC1 c1(C(=O)OCC)n[nH]c(=NC(=O)NC(c2ncccc2C)C)s1 C(=O)(CS(=O)CCC(F)(F)F)N1CC(C2N(C(CCS(N)(=O)=O)=O)CCC2)(O)C1 C1(C(N2C(CN(C(c3ccc(CC)s3)=O)C)CCC2)=O)CC(C2CC2)=NO1 c1(N2CCCC(C(N(C)C)=O)C2)ccncc1S(=O)(=O)N1CCCC1CO CC(C)(C#N)CCC(=O)N1CC(C(N)=O)(CNC(=O)CCC2(C)CCC(=O)N2)C1 C(C)(C(=O)NC(C(=O)NCCc1nccs1)c1ccoc1)OC N12CC3CC(C1C3)NC(=O)C2.c1(C(=O)NS(=O)(=O)CCC2CC2)n[nH]c2c1CCC2 N1(C(c2c(CC)[nH]cc2)=O)CC(CC(N2CCSCC2)=O)CC1C c1(NC(C23CN(C(CC)=O)C(C2)CO3)=O)ccc(CC)nc1C c1(C(N2CCN(C(C(COC)N(C)C)=O)C(C)C2)=O)ccc(Cl)c(C)c1N N1(C(c2nc(OCC)sn2)=O)CCC12CN(C(C1CCOC(=O)N1)=O)C2 c1(C(=O)NC2CCN(C(=O)Cc3ccsc3)C2C2CC2)cccc2c1C(=O)NC2 N1(C(C(C=C)(C)O)=O)CC2CC(C1)N(C(c1c[nH]nc1-c1ccsc1)=O)C2 Cc1sc(C)c(C(=O)NC(C)CC(C)NC(C2(CN(C)C)CC2)=O)c1Br N1(C(c2cc(C)[nH]n2)=O)CCOCC12COCCN(C(=O)CSc1cccs1)C2 C(c1ccc(F)cc1)=CC(=O)NCC1(C2N(C(CC(=C)Br)=O)CCCC2)CC1 C1(O)(CNC(C(c2cncnc2)C)=O)CCN(C(c2cscc2F)=O)C1 c1(N(C(=O)C(O)CC2CC2)C2CCC2)ccc(O)cc1 c1(C(C)C)cc(N2CCC(C)(CNC(C3(C4CCC4)CC3)=O)C2)n2ncnc2n1 Cc1ccc(CO)cc1C(=O)NC1CCN(C(=O)C(=O)N(C)C)C1(C)C c1(C(=O)NC2C(NC(Cn3c(C)nc(C)n3)=O)CC2)cc2ncc(C)n2cn1 C=C(C)C(CC(=O)NCC(COC)NC(C1CC2(CCCO2)C1)=O)OCC C1(CC=C)(NC(C2CCCC2C)=O)CCCN(C(=O)CCCCCOC)C1 C12(C(=O)NCC3(CCNC(c4occc4Cl)=O)CC3)CCN(CC1)C2 N1(CCC(=O)NC(CC)CNC(=O)C=CC)CCN(c2ccc(OC)cc2)CC1 C(CC(C)(C)C(=O)N1CC[Si](C)(C)C1)NC(C(CC)C)=O c1(OCC)c(C(=O)NCCC2CN(C(=O)C(CO)OC)C2)cccc1F N1(C(C=CCN(C)C)=O)CCCC(C2CCN(C(c3cc(C)cc(N)c3)=O)C2)C1 c1(C(N2CC(N3CCN(CC4CC(=O)OC4)CC3)C2)=O)cc2c(Cl)cc(Br)cc2[nH]1 N1CC(C(=O)OC)CC1=O.N1(CC(=O)NCC=CC)CCC(F)CC1 N1(C(C2CCCCC2c2ccc(C)cc2)=O)CCc2ccccc2C1 c1(C(N2CC(O)(CCNC(C3C4COCC34)=O)C2)=O)ccc2occc2c1 C#CC1CC2(CC2)CN1C(C1C=CC(NC(C2CCCC(OC)C2)=O)C1)=O C1(NC(=O)CCc2csnn2)CCN(C(c2cc3c(s2)CCC3)=O)CC1O Nc1cc(C(=O)NCC2CC(NC(C3(N(C)C)CC3)=O)C23CCC3)cc(F)c1 C1(C(N2CCCC2c2cc(Cl)sc2Cl)=O)Cc2c[nH]cc2S1(=O)=O C=C(C)C(C)(C)C(=O)NCC1CCN(C(=O)CC2(C)OCCO2)C1 c1(CNC(=O)NC(C2CCOCC2)C#C)ccc(F)c(S(N)(=O)=O)c1 c1(C(=O)NCC)ccc(S(=O)(=O)N2C3CCCC2CC(F)C3)cc1OCC C(C(=O)N1CCC(C(=O)NC)C1)(C(C)(C)C)NC(CC1(CC)CCC1)=O C1(C(N2C3C(NC(C(C)CC4CCCCC4)=O)C(C3)C2)=O)CCc2c[nH]nc2C1 Fc1cnc(Cl)c(C(NC(=NCC2CCOC2)NCCc2ccco2)COC)c1 Nc1cc(C(=O)NCC2CCCCN2C(c2ncnc(O)c2F)=O)cc(Cl)n1 C12(CNC(c3cn(C)c(=O)n3C)=O)CCCC1CN(C(c1ccsc1Cl)=O)C2 C(C(=O)NCCCc1cn(CCC2CCCN2C)nn1)(C(C)O)NC(C)=O CN1CC(NC(=O)C(CCC2CC2)NC(c2ccsc2Cl)=O)C2(CC2)C1=O C1(NC(COC(CC)C)=O)CC(C(=O)NCC(C)C)C1(C)C C(C(C)(COC)C(=O)NC1CC2CCC1(CNC(=O)CCC(C)(C)F)C2)OC c1(CC(=O)NC2C(O)CCN(C(C3(C)CC(=C)C3)=O)C2)coc2ccc(C)cc12 N1(C(CCCn2cc(COCC(C)O)nn2)=O)CCOC(C)C1C C(=O)(C1=COCCC1)N1C(C(=O)NCc2ncc(CC)s2)CC=CC1 Cc1cc(C(=O)NCCN(C(C2CC3C=CC2O3)=O)CC2CC2)c(F)cc1N CCC(CC(=O)N1CCC(CNC(=O)Cc2ccns2)(OC(C)(C)C)C1)C(=O)OC N1(C(C2C(C)(C(F)F)C2)=O)CC2CC(NC(c3cc4occc4s3)=O)CC(C2)C1 N1(C(CSCC)=O)CCN(C(c2cnc(COC(F)(F)F)s2)=O)CC1C1CCC1 C(=O)(C(CCCC)NC(=O)C=C(C)CCC)NC(C=C)(C)CC c1(CNC(C2N(C(C(C)NC(CC)(C)C)=O)CCCC2)=O)cnc2ncccn12 CCC(C(=O)N1CC(O)(CNC(c2ccc(OCCF)cc2)=O)C1)C(C)O Cc1c[nH]cc(C(N2CCCC2CNC(=O)CC2CC(C)C2)=O)c1=O C1(CNC(C(CC)(C)OC)=O)COCCN(C(c2conc2C2(C)COC2)=O)C1 N#Cc1ccc(C(=O)NC2CC3CC2N(C(c2c(F)cncc2Cl)=O)C3)c(F)c1 N1(C(c2c(C)scc2)=O)CCC(C)(C)C(C(=O)NCCN2C(=O)CNC2=O)C1 N1(C(C2CCN(C(c3c(CC)cccc3)=O)C2)=O)CC(S(N)(=O)=O)C1 CN=c1[nH]cc(C(N2CCOC(CN(C(=O)C(F)(F)c3ccccn3)C)C2)=O)o1 CCCCCCOC(C)C(=O)OCCCOCC(=O)N(C1CCOCC1)C N1(C(C(CCC)NC(N)=O)=O)CCN(C(c2nncn2CC)=O)CC1CCO C(=O)(C(C)(C)CO)NC1CC(C(C)C(=O)NCCC(O)C2CCCC2)C1 c1(C(N(C2CCN(C(C(CC)(C)O)=O)CC23CC3)C)=O)c(F)c(F)cc(F)c1F C=Cc1ccc(C(=O)NCCN(CCC)C(c2cnncc2C)=O)cc1 C1(N(C)C(C2COCCC2NC(=O)CC2CCSCC2)=O)CC(C)(C)C12CC2 C(=O)(C(C)CNC(=O)CCC1CCCCC1)NCCC(=O)NC1(C#C)CC1 C(=O)(CCC(C)(C)C)N1C(C(N(C)CCC2CCCO2)=O)C2CCC1C2 C(=O)(C(C)(C)C)NC(C(=O)N(C(CNC(C1(COC)CCC1)=O)(C)C1CC1)C)C C1(NC(C2CN(CC)C(=O)CC2)=O)CCC2(CC1)CCN(C(=O)C(F)F)C2 C(=O)(CC(C)(C)C(=O)NCC(C(C)C)NC(c1ccccc1C(=O)OC)=O)OC Cc1c(NCc2nc(-c3ccccc3)cs2)nc[nH]c1=NCC1CC12CCCCC2 C1(C(=O)NCC2(CC)CCCC2)CC(F)CCN1C(=O)CC1CC(C)(C)C1 C(C(C)C(C)C(=O)N(CC(C)(C)NC(c1ocnc1C1CC1)=O)C)OC C1(OCCC)CCN(C(=NCCSC)NCC2(CS(C)(=O)=O)CCC2)CC1OC C1(NC(C2(Cl)C(C)(C)C2)=O)CCCN(C(c2ccc(C(F)(F)F)cn2)=O)C1 C1(C(=O)NC2N(C(CC)=O)CSC2)CCN(C(=O)C=Cc2cccnc2)CC1O CCCCC(O)C(C)C(=O)N1CCC2CCN(C(=O)C(C)C3CCC3)C2C1 C1(NC(=O)C=CSc2ccccc2)CN(C(=O)CCc2cnn[nH]2)CC12CCC2 N1(C(C(C2CCCC2)OC)=O)CCCCC(C2CN(C(C3CC34CC4)=O)C2)C1 N1(C(C2(COC)CCCC2)=O)CCC=CC1C(=O)NCC1OCC2CCC1C2 C(=O)(C1CCOc2c(F)cccc21)N(CCN(C(c1cc(=NC)[nH]cc1)=O)C)C Cc1ccc(C(=O)NCC(C)NC(c2cc(C(F)F)nn2C)=O)nc1O CC(C)CCN=c1nc2c(cnn2C(C)C)c(NCC(C)CCCO)[nH]1 Cc1cscc1NC(=O)CCOCCN(C(=O)Cc1cscn1)C c1(CNC2CCCC(NC(C(c3ccccc3)C)=O)C2)ccc2c(c1)CCO2 c1(OC)c(F)ccc(F)c1C(N1CCN(C(C)=O)C(CNC(=O)CCOC)C1)=O C1(C(N2CCC2CC(C)(C)C)=O)(CNC(C(CC2CCC2)OC)=O)CCCCC1 O=C(CCCCCCn1cc(Cn2cccc2)nn1)NCC1CCC=CO1 c1(C(=O)NCC2(C(=O)NC3C(C(C)(F)F)C3)CCCCC2)ccc(F)cc1Cl S(=O)(=O)(C1CC(NC(c2ccc(OCC3CC3)c(F)c2)C)C1)Nc1ccc(Cl)cc1 [N-]=[N+]=NCCCC(=O)N1CCSCC1C(=O)N(CC1CC1)OC c1(C(=O)NCC(CC=C)NC(=O)C(F)OC)ncccc1-c1ccccn1 N1(C(C(P(C)(C)=O)O)=O)CCC2(CC1)CC2NC(c1ccnnc1)=O N1(C(C2CCCC(C)C2)=O)CC2CCC(CNC(c3ncncc3Cl)=O)(C2)C1 C1(NC(C2(NC(Cc3c(C)noc3)=O)CCCC2C)=O)CCc2nncn2C1 c1(NC2CCN(CC3C(CC(C)C)C3)C2)cnc2c(C(F)(F)F)cccn12 N1(C(c2cc(COC)no2)=O)CC2(CC(NC(=O)C3=CCSC3)CO2)C1 CC1(C(=O)NCCc2ccns2)C=CCN1C(c1ccc(C#N)o1)=O c1(CCN(C)C(C2CCCC3(CCOC3)OC2)=O)cccc(S(N)(=O)=O)c1 Cc1cc(OCC(N2CC(CNC(=O)CCC(C)(C)O)CC2C)=O)ccc1Cl N12Cc3[nH]nc(c3C1)NC2=O.c1(CC)cnc(N2CCC2)nc1 C1(N(C)C(c2cc(C3CCC3)on2)=O)CCN(C(=O)C(=O)NCC(F)F)C1 c1(CNC(c2c(C)cccc2)CN2CCCC2)c[nH]c2cc(Cl)c([N+](=O)[O-])cc12 c1(C(=O)NCC2CN(C(C(=O)NCCCC)=O)CC2(C)C)cc(F)c(Cl)cc1F C1(NC(CCC#C)=O)CCN(C(=O)CC2(c3ccccc3)CCC2)C12CCC2 N1(C(CCN(CCC)C)=O)CCCC(CNC(=O)C=C(CC)CC)(OC)C1 CC1CCC(O)C(NC(c2ccc(CCNC(=O)OC(C)(C)C)cc2)=O)C1 C1(C(C)(C)C)CCN(C(=O)NC2CNC(=O)C23CC3)CC1C(=O)O N1(C(c2nc(C(C)C)oc2)=O)CCC2CN(C(=O)CC(C)(C)C)CC12 c1(C(N2CC3CC(NC(c4ccncc4)=O)CC3C2)=O)cccc2c1OCCC2 C(CC)(CC)(CCNC(c1cc(C(C)C)cnc1O)=O)NC(C(C)OCC=C)=O c1(CC(=O)NCC2(NC(CC(C)SC)=O)CCCC2)ccc(C2CCOC2)cc1 C1(C(=O)NCC(=CC(=O)N(C(CO)CO)CC)C)CCC(C(N)=O)C1 C1(CC=C)(NC(c2cc(SC)n(C)n2)=O)CCN(C(C2CCCSC2C)=O)C1 C(=O)(C1=CCCOCC1)NC(c1ccccc1)C(=O)NCc1nc(C)c(C)s1 N1(C(=O)C2=CCSC2)CC2CCC1(CNC(c1c(N(C)C)nccc1)=O)CC2 c1(OCCC)ccccc1C(N1CCC(CCNC(=O)C=CS(C)=O)C1)=O c1(NC(C)COC2CCOC(c3cccc(F)c3)C2)ccc2c(C#N)c[nH]c2c1 n1(CC(=O)N(CCC(C)NC(=O)C(C#N)C2CC2)C)nc2ccccn2c1=O N1(C(C(=O)NCCCCCCOC)=O)CC(C)(C)CCC1C1CC1.N12CCCC1C2 C1(NC(C2(C#C)CC(=O)C2)=O)C2CC3C1C3C2C(=O)NCCCCC1CCCC1 N1(C(c2c(C)[nH]c(C#N)c2)=O)CCC2CCC(C1)N2C(c1cccnc1CO)=O C(=O)(CC(C)(C)CC(=O)OC)NC(CN(C(c1cc(CCC)nn1C)=O)C)CC C1(C)(NC(CCN(CCC(C)(C)C)C)=O)CCC(NC(c2ncsc2C)=O)CC1 c1(-c2cc(C(=O)OC)on2)ccc2cc3cc(NC(C4CC4F)=O)sc3nc2c1 C(=O)(C(O)CC(C)(C)C)NCCC1CC(NC(CC(C)SC)=O)C1 c1(C(N2CCC3(C(C(=O)Nc4ncc(F)s4)C3)C2)=O)cccc(F)c1[N+](=O)[O-] c1(C(=O)NCC2N(C(C(C(CC)C)NC(N)=O)=O)CC2)ccc2c(c1)CC(=O)N2 C=Cc1cnn(C)c1C(=O)NCC(C)CNC(c1cc(C)cc(Br)c1)=O c1(C(N2CC(CS(N)(=O)=O)C(C)C2)C(=O)NC)ccc2c(c1)CC(C)(C)O2 c1(C(N(C2CCCN(C(=O)C=CCN(C)C)C2)CC)=O)cccc2c1OCCC2 CC#CCCCC(=O)NC1(CCC(=O)NCCCOCC2CC2)CCCC1 Cc1cn(C)nc1C(C(=O)NC1CCC1)N(C1CCOC1)CCOC C1(C)(NC(C2C(CNC(CC3N(C)CCC3)=O)C2(C)C)=O)CC=CCC1 c1(C(=O)OC)ccc(F)c(C(N2CCOCC2CCNC(=O)CP(C)(C)=O)=O)c1 O=C(C1=CCCC1)NCc1cc(C(=O)NCCC(O)C(F)F)co1 c1(C(N2CC(O)(CCNC(C(CCCCC)O)=O)C2)=O)c(F)cccc1[N+](=O)[O-] C1(C(=O)OC)COCCC12CN(C(C1CC1NC(c1cccs1)=O)=O)C2 c1(C(C(=O)NCC2N(C(CC=CC(C)(C)C)=O)CCC2)O)ccc(F)c(F)c1 C1(NC(c2cnc(C)[nH]2)=O)CN(Cc2cc(F)ccc2C)CCC1O Cc1cnccc1C(=O)NCC(O)CNC(c1cnc(Cl)cn1)=O c1(O)cc(Br)ccn1.CC(C)(C(=O)NCC1CCN1C(=O)C=O)N1CCCCC1 c1(CNC2CC(NC(Cc3c(C)n[nH]c3)=O)C23CCC3)noc2c1COCC2 c1(C(=O)NC(CC2CCN(C(Cc3nnc(C)o3)=O)CC2)C)cc2[nH]ccc2s1 CN1CC(C(N2CCN(C(c3nscc3N)=O)CC2)=O)OCCC1=O Nc1cc(F)c(F)cc1C(=O)NCC1CC(F)(CNC(c2c[nH]nc2F)=O)C1 CCCC(CC)C(=O)N1CCC(NC(=O)CC2(C#N)CCCCC2)C1 C1(CNC(CC(C)OC)=O)CCCCN1C(=O)C(C)Oc1ccc(F)nc1 C1(C(C(=O)N(CC#C)C(C)C)(C)C)CCCN(C(c2cc(CC)nn2C)=O)C1 C(=O)(C1=NN(CCO)C(=O)CC1)N(C1CC(NC(c2c(C=C)cnn2C)=O)C1)C C=C(C)C(CC(=O)NC(C)(CNC(=O)CC(CC)OC)C1CC1)OCC c1(N2C(CN(C(CC3CC(=C)C3)=O)C)COCC2)nc(C#N)c(Cl)s1 CCCC(C(=O)NCC(C)(O)CO)NC(=O)CCC1CCCOC1 C(=O)(CC(C)(O)COC)NCCC(CCN)C.C(=O)(CCSC)OC C1(C)(NC(C(C2CC2)OC)=O)CCN(C(=O)C(F)CC2CCCCC2)CC1 c1(C(=O)NC(C)CNC(=O)CN2CCCCC2)ccc2c(c1)CCCS2(=O)=O C1(Cc2cn(CC(=O)OC)nn2)CN(C(=O)C(C2CCOCC2)C)C(C)(C)C1 C=CC1CCCC(NC(=O)CC2C3CCCC3N2C(=O)C(C)(CC)CO)C1 c1(C(=O)NC(CN(C(=O)CN2CCN(CC)C2=O)CC)C)cnc2ccoc2c1 Cc1ccncc1C=CC(=O)NCC(C1CC1)N(C)C(C1CC(C)(C)CO1)=O c1(C(NC(=NCCOCC)NCC(C)(C)OC)C)cccc2ccccc12 Cc1cc(O)c(C(C)C)cc1NCc1cc(C(=O)O)cc(O)c1 c1(C(=O)NC2CCC(N(C(=O)COCC(C)(C)C)C)C2)ccc2c(n1)CCC2=O C1(NC(=O)NCCCCOc2c(C)cccc2)CCC(=O)N2CCCCC12 c1(C(C)NC(c2c(C(C)NC(c3n(CC)ncc3)=O)n[nH]c2)=O)nnc(O)n1C C(CC)(C(=O)NCc1ccccc1)OCC.C1(N)CCN1C(=O)C(C)C1CCCCC1 Cc1[nH]cc(C(=O)N(CCNC(=O)C=CC(F)(F)F)C(C)C)c(=O)c1Cl c1(C(N2CCC(NC(C3(CCCC)CC3)=O)C(F)C2)=O)cnc2nccnc2c1 N1(C(Cc2c(CC)con2)=O)C(C(=O)NCc2nn(C)cc2C)CCC1C1CC1 N1(C(C2(C(C)C)CCC2)=O)C(C(=O)NCC2(C)CSC2)CC1C C(C1=CCCN(C(C2CC(F)(F)C2(C)C)=O)C1)NC(C(n1c(C)ccn1)C)=O Cn1nc(C(=O)NC2C=CCN(C(C3COCC3C(N)=O)=O)C2)ccc1=O N1(C(=O)Cc2cccc(OCCF)c2)CCN(C(C2COCC2O)=O)C2CCC12 N1(C(C2N(CC)CC2)=O)CCC2CCN(C(c3ccc(F)cc3C#N)=O)CC2C1 C(=O)(CC(C)N(C(=O)C(C)CN1CCOCC1)C)OCC C#CCC(C(=O)NCc1cncc(C(=O)Nc2cccc(CCO)c2)c1)C1CC1 C#CCCCCCCCCCC(=O)NCCCC1CCCC1O Nc1cccc(C(N2CCC(NC(=O)CNc3ccccc3)C2C2CC2)=O)c1F N(C(=NCC)N1CCC(Cn2cnnn2)C1)C(C#C)C N1(c2cccc(N3C(=O)CC(O)C3)n2)Cc2cccc(-n3cncn3)c2C1 CCCS(=O)(=O)NC(C)C(=O)N(CC(C)(C)NC(c1cn(C2CCC2)nn1)=O)C C1(C(=O)NCCOCCN(C(=O)CCc2ccco2)C)COc2ccc(F)cc2C1 C1(CNC(c2c(CN(C)C)ccs2)=O)CCCN(C(c2ccncc2F)=O)C1 C(=O)(C1=NOC2(CCC2)C1)N1C2CC(C(=O)NC(C#C)CC3CC3)(OC2)C1 c1(C(N2C(C(=O)Nc3c(OCC)nccn3)CC2)=O)nc2c(s1)CN(C)CC2 C(C(C)(O)C(=O)NCC(C)N(C(=O)CN(C(=O)C(C)C)C)C)OC C1(C(=O)NCCOCCCC)(NC(c2ccsc2OC)=O)CCC(C)(C)C1 c1(CCN(CCNC)CCN(C(C(CC)NC(C)=O)=O)C)cc(C)c(F)c(C)c1 c1(C(=O)NCCN(C(=O)CC(C)C2CC2)CCOC)cnn2c1C(=O)NCC2 C1(C(N2C(CNC(COCc3cccc(OC)c3)=O)CC2)=O)CC12CC(C)(C)C2 C12(C(N3CCC(OC4CN(C(C(CC)O)=O)C4)CC3)=O)CCC(C)(CC1)CO2 N1(C(CCOCCOCC)=O)CC(C(N2CCN(CC(C)O)CC2)=O)C(C)C1 N1(C(C(C)c2ccsc2)=O)CC(C2CN(C(C3(C)CS(=O)(=O)C3)=O)C2)C1 N1(C(c2c(C)nc(CC)s2)=O)CC(C2(NC(c3ccc(N)c(N)n3)=O)CC2)C1 C1(C(=O)OC)C2CN(C(=NCCC(C)N(C)C)NC3CCCCC3C)CC12 c1(C(N2CC(CNC(CCSCC)=O)C(C)CC2)=O)cc2n(n1)CCCC2 C(CC(C)(C)N)NC(C(c1ccccc1)OC)C C#CC12CCN(C1)C2=O.C1(CC(=O)NC2CCC(C(=O)OCC)C2)COCC(C)O1 Cc1ccc(CC(=O)NCC2(F)CCC(NC(=O)CCc3nc[nH]n3)C2)cn1 C1(O)(C(C)NC(=O)COC=O)CCNCC1.C1(C)CCCO1 c1(C(=O)O)cc(Br)c2c(c1)CC(CNC(C1CCCOCC1)=O)O2 CCC(C)(C#N)C(=O)N1CCC(CNC(c2cnc(-c3ccco3)s2)=O)C1 c1(CC2C(C(NOCC(=O)NCC3(C(C)(C)OC)CC3)=O)C2)nnsc1N C1(C)(C(=O)NC(CC(C)C)CNC(=O)Cc2sccc2F)CCNC(=O)C1 C1(C)(OC)CCN(C(=O)CC2CCC(N(C)C)CC2)CC1.C12CCN1C2 C(CC(C(C)C)NC(c1cccc(C)c1)=O)NC(c1ccc(CNC(C)=O)o1)=O CC(CC(C)(C)C)C(=O)N1CCN(C2CN(C(=O)C3=CS(=O)CCC3)C2)CC1 c1(OC(C(=O)NCC2N(C(c3c(=N)[nH]n(C)n3)=O)CC2)(C)C)cc(F)ccc1F C(=O)(C(C)C(C)n1cccn1)NC(CNC(COCCC=C)=O)(C)CO C(=O)(CCC(=O)N(C)CCOCCCNC(c1ccnn1C1CC1)=O)NC c1(SC)nc(C(=O)NC2(C3CCCCN3C(=O)C3=C(C)OCC3)CC2)c(C)c(Cl)n1 C1(NC(C(C#C)(C)C)=O)COC2(C1)CN(C(c1ccc(C(C)=O)c(F)c1)=O)C2 CCN=C(NCC1(S(C)(=O)=O)CC1)NC(C)C N1(C(c2cnc(C)nc2C)=O)CC2CCC(C1)N2C(=O)C(C)n1ccnc1 c1(CC(=O)NC2CC(O)C2)ccc2ncc(Br)cc2c1.C12CCCC1CNC2=O C1(O)(CC)CCN(C(C)C)C1.C12(C(=O)O)CN(C1)C(=O)c1coc(n1)S2 C(=O)(CCCS(N)(=O)=O)NC(CCCNC(Cc1ccc(OCC)cn1)=O)C c1(CNC(C2CC(C(=O)Nc3cnc(Cl)nc3)C2)=O)ccc(Br)c(O)c1 N(C(=NCC1CCN(c2ncccn2)CC1)NC1CC12CCCC2)C(CC)C c1(C(=O)NCC(C)N(C(Cc2c(C)n[nH]c2C)=O)C)cccc2c(C)csc12 C1(NC(C(C)OCCC=C)=O)CCCCC1C(=O)NCCc1ncn(C)n1 c1(C(=O)NCCCCC(C)NC(C(C)OCC=C)=O)cccc2c1oc(=O)n2C c1(CC)cc(C(=O)NCC2CN(C(=O)C(C)OC)CCO2)nn1C C1(NC(C(n2cc(Cl)cn2)C)=O)CCN(C(=O)Cn2c(C)ccc2C)C1C(C)(C)C CCC(CC1CCCO1)C(=O)O.c1(C2n3cc(nn3)CCC(=O)NC2)cccc(F)c1 Cn1ncc(C(=O)NC(C)(C)CCNC(c2scnc2C(F)F)=O)n1 S(=O)(=O)(c1cccc(Br)c1)N.N1(C(C2(CO)C(C(C)C)C2)=O)CCC(CO)CC1 C(=O)(C#CC1CCOC1)NC1C=CC(NC(CCCC#C)=O)C1 N1(C(C2CC3CC(C)OC3C2)=O)CCOC2(C1)C1CC3CC(C1)CC2C3 CC1CCC(NC(c2sc(F)cc2Cl)=O)CN1C(=O)Cc1cccn1C N1(C(C2CC(=C)C2)=O)C2CCC1C(NC(=O)C(F)OC(F)(F)F)C2 Cc1cc(=NCCc2cscn2)[nH]c(N(C)Cc2ccnc(C)n2)n1 c1(CNC(C)=O)ccc(C(=O)NC(C)CCNC(=O)C(F)=C(C)C)cc1 Cc1ccc(CNC(=O)NC2(CO)CCCN(c3ncccn3)C2)cc1[N+](=O)[O-] Cc1nc(C=CC(N2CCC(C)(CCNC(=O)C(C)NC(N)=O)C2)=O)[nH]c1C c1(CNCC2N(C(C3CCC(CCCC)CC3)=O)CCOC2)cccc(C)c1Cl N1(C(Cn2cc(-c3c(C)cnn3C)nn2)=O)CCN(C)C(=O)C1 C(C(C)(C)CC(=O)NC(c1csc(C)n1)C)NC(C(C1CCOC1)OC)=O c1(C(N2CC3(N(C(C4CN(C)C(=O)N4)=O)CCC3)C2)=O)cnn2c(N)ccnc12 Cn1nccc1C1=CCN(C(=O)C(=O)Nc2nccs2)CC1 c1(C(=O)OC)cc(NC(=O)CC2(C)CCN(C(=O)C(=O)NC3CC3)C2)cnc1OC CCC(CC(=O)NCCC1CCC(=O)N1)N(C)C(C1CC(C)(O)C1)=O C(=O)(C1=C(Cl)CCCC1)N1CCC(COC)(NC(=O)C(c2ccc(C)s2)C)C1 C1(C(=O)NC2CC(CC(=O)Nc3c[nH]c4nccc-4c3)C2)CCCC2(CCC2)O1 Cc1c(CNC(=O)OC(CN(C)C)Cc2ccccc2)cccc1Cl C1CCCCCC(=O)N1.C1(C(N2CC(CCCCOCC)C2)=O)CC2CCC1O2 c1(CC)ccc(C(=O)NCCC2CCCN2C(c2cc(CSC)c[nH]2)=O)cc1C CC(c1ccccc1)=CC(=O)NC(CC(=O)NC1CC(C2CC2)C1)C1CC1 C1(C(=O)NCC2CC(NC(C3(COC)CCC3)=O)C2)COCCN1C(C)=O N1(C(C2C(C)CCN2C(=O)Cn2nccn2)=O)CCOC2CCC12 N1(C(C(=O)NCCC)C2CCC2)CCCNC(=O)C1CC CC1CN(C(=O)C#CC2CC2)CCCN1C(c1cccc(C2COC2)c1)=O C=CCCCCC(=O)N1CCC(CNC(c2cnc(SC)nc2O)=O)C1(C)C n1(CC)nc(C(=O)NCCC2CCCN2C(=O)C(C#N)C2CC2)cc1C1CC1 C(C#Cc1cccnc1)N(CCC)C(c1cn(C)nc1OC)=O.C1(C)C(=O)N1 N1(C(CCCC)=O)C2CCCC1CN(C(c1cnc(C)c(C#N)c1)=O)CC2 Cc1c(N)ccc(C(=O)NCC(C)NC(c2ccc(C(N)=O)o2)=O)c1Cl c1(C(N2CCC(NC(C(CC)SC)=O)C(O)C2)=O)cc(O)cc(F)c1F c1(OC)nc(C)ncc1C(=O)NC(C1CCCN1C(=O)C(C)n1cnnn1)C c1(C(N2CC(NC(C(CC=C)c3ccccc3)=O)C2)=O)ccc(F)c(F)c1N C(=O)(C1=CCCOCC1)N1CC(CNC(c2c(CC)nnc(C)c2)=O)C(C)CC1 N1(C(C2(C)C(C)OCC2)=O)CC2CC1CC2CNC(=O)C=CCCC=CCBr C(c1ccccc1C)=CC(=O)N(CC(CC)NC(=O)C=Cc1nc(C)c(C)[nH]1)CC CCC(CNC(C1(C)CC(O)CN1C(c1cncs1)=O)=O)CC(C)C N1(C(C(Cc2cn[nH]c2)NC(C2OCCN(C)C2)=O)=O)CCC(C2CCCC2)C1 CC1CCCN(C(=O)COC2CC(NC(C34CCC(C3)C4(C)C)=O)C2)C1C c1(COC)ccc(NC(c2ccc(C(N3CCCC3CC(C)C)=O)[nH]2)=O)cc1Br C12(CNC(C3CC(CC)C3)=O)CC(NC(=O)CC(C)(C)C(F)F)(C1)C1(CCC1)O2 N1(C(c2c(NC)cccc2)=O)CCC(F)(CNC(C2OCCN(C)C2=O)=O)CC1 CC1CN(c2ccc(C#N)cn2)CCN1C(=O)C#CC1CC1 CC1CC(C(=O)N2CC3(CC3)CC2C(N2CC(CN(c3ccc(Cl)cc3)CC)C2)=O)=NO1 C1(NC(CSC)=O)CC(CO)N(C(=O)CCCN2CCCC2=O)C1 C1(CC(=O)N(CC(=O)N(C(C)C(N)=O)C)CCOC)CCCC1C C1(NC(=O)COC2CCCCC2)C2CC(NC(c3nocc3Br)=O)CC12 c1(C(N(CCNC(=O)C(C)CSC)CC)=O)cnc(C)c(N)c1 C1(CNC(c2c(OC)cc(C)s2)=O)CN(C(c2sc(C)c(C)c2C)=O)CC1(C)C CC1CN(C(=O)C(CC(F)F)C2CC2)CCN1C(=O)CCOc1ccc(Cl)cc1 c1(C(=O)NC2CN(C(C3(SCC)CC3)=O)CC2SC)cc2nc[nH]c2cc1F c1(C(N(C)CC2CC(O)CN2C(=O)CNC2CCCO2)=O)cc2c(s1)CCC2 c1(CSCCNC(C2CSCN2C(=O)C(F)(F)F)=O)scnc1Cl C1(C(N(CC(C)C(=O)NCC2(O)CCOC2)C)=O)CCCSC1C N1(C(C2N(C)CCN(C)C2)=O)CCC2CC2(C(=O)NCC2CC(N(C)C)C2)CC1 CC1(CNCCC2CC(C(=O)O)C2)CCOC(C2CCC2)C1 C1(CNC(C=Cc2occ(C)n2)=O)CC12CCN(C(C1COC1)=O)CC2 CCC(C)(CCC(C)C)C(=O)NCC(C)NC(c1ncccc1C(F)(F)F)=O C1(CNC(C(C(C)(C)C)NC(C)=O)=O)CN(C(=O)Cn2cncn2)CCC1(C)C Cc1ccc2c(n1)CCN(C(c1ccc(C(N3CCCC3C(N)=O)=O)cc1)=O)C2 C(=O)(C1CCc2cccc(=O)n21)NC(C)CNC(c1c[nH]c2nccc-2c1)=O c1(C(C)NC(=O)C(C2CCOC2)NC(=O)CCc2cnn(C)c2)cncnc1 C1(NC(c2nccc(C)n2)=O)CC1C1CCN(C(C2CC2F)=O)CC1 C1(NC(CC2C=CC(NC(C(C)(C)O)=O)C2)=O)COCC(C)(C)C1 CC(C)CC(CNC(c1cccc(N2CCCC2)n1)=O)NC(=O)CN(C)C C(C(CC(=O)NCCc1cncn1C)C1CC1)NC(C(C)SCC)=O C(=O)(C(CC)C(C)(C)CC)N1CCC(C#N)(CC(=O)N(CC=C)CC2CC2)CC1 C1(C)(C(=O)NC(CNC(c2nc(CC)oc2)=O)C2CC2)CCCN(C)C1 N1(C(c2cc[nH]c2)=O)CCCC(C2CCCCN2C(=O)C2=NOCC2)C1 CP1(=O)CCN(CC(=O)NCC(C2CC2)NC(=O)CN2CCCC2=O)CC1 CCCCCC(C)(C)C(=O)NC1CC(C(=O)N2CCCC2)=CC1O C1(C(=O)NCCc2c(C)ncs2)C2CN(C(C3CC(C(C)C)C3)=O)CC12 c1(C(=O)NC2CCCC(CNC(CC(C)(C)OC)=O)C2)ccc2oncc2c1 Cc1cc(C(N2CC(C3(NC(c4cn(C(C)C)nn4)=O)CC3)C2)=O)c(N)c(F)c1 N1(C(CC2CC(OCC(=O)Nc3cn[nH]c3)C2)=O)CCC2(CCCOC2)C1 C1(C(=O)NCCN2CCN(C(CC3CC(SC)C3)=O)CC2)CC(C)CC(C)C1 Cc1cc(C=CC(=O)N(C)CCOCCC(=O)N(C)Cc2cc(C)nn2C)on1 C1(C(N2CC(n3ccnc3)C2)=O)(CNC(C(C)C2CCCO2)=O)CCCCC1 C1(Nc2ccc(S(=O)(=O)NCc3c(C)cco3)cn2)Oc2ccccc2OC1C c1(C(=O)NCCNC(=O)CC2CC2)cccc(-n2cnnc2)c1.n1(C)cccn1 Cc1ccnc2nc(=NC(=O)C3CCC(c4ccccc4)CC3)[nH]n12 C1(NC(c2cc(C(F)(F)F)ns2)=O)CN(C(=O)Cc2cc[nH]n2)C2(CCCC2)C1 C#CC1(C(=O)NCC2CCOC2(C)C)CN(C(=O)Cc2ccon2)C1 c1(N(CCOCCNC(c2c(CC)nc[nH]2)=O)C)ncnc2c1COC2 c1(-c2nc(C(N(C)S(N)(=O)=O)=O)sc2)ccc(S(=O)(=O)C2CC2)cc1 C(C)(C)(CCCNC(=O)CC(O)Cc1ccccc1)NC(C(COC)C)=O C12(C(=O)Nc3cccc(NC=O)c3)CC(CNC(C(C)C#N)=O)(CO1)C2 c1(C(N2CC(CN(C(C(C)C#N)=O)C)OCC2)=O)c[nH]c2nc(F)ccc12 c1(CCC(N2CCC(NC(C#C)=O)C(O)C2)=O)cccc2c1OCCO2 c1(C(N(CCNC(CCn2c(C)ncc2)=O)C2CC2)=O)csc(S(N)(=O)=O)c1 c1(CC(=O)N(CC(C)NC(=O)CCOC(C)CC(C)C)CC)cc(C)ccc1F Cc1[nH]nc2ccc(C(=O)NC3CCCN(C(C4CC(C(F)F)C4)=O)C3)cc12 N1(C(c2ccc(C)o2)=O)CCCC(F)(C(=O)NCCC(C)CCO)C1 C1(NC(C2(OC)CCOC2)=O)CN(C(=O)Cc2ncc(C)s2)CC1C1CC1 CC1(C(=O)NC2CC2NC(c2cnn(C3CCC3)c2)=O)CCOC1 c1(C(=O)NCc2cc(C(N(C)CCOC3CC3)=O)sc2)cnncc1O CC(C)C(C(=O)N(CC(C)(C)CNC(=O)CCC(C)N(C)C)C)n1cnnc1 c1(C(N(C2CCN(C(=O)Cc3ccco3)C2)CC)=O)cncc(C)c1Cl C1CC(C)(C)CC(=O)O1.C1(COC)C2CCCCCCC12 C(=O)(C(C)(C)NC(=O)C(C1CC1(Br)Br)N(c1ccccc1)C1CCCC1)NCC c1(C(N2CCC(NC(CS(CC)=O)=O)C2C)=O)cccc2c(C#N)c[nH]c12 c1(CN(C)CC2N(C(=O)NC(CCC)C(=O)OC)CCC2)ccc2occc2c1 N1(C(CC(C)(C)OC)=O)CCC(C(=O)NCCc2cccs2)C(C)C1 c1(SCC(=O)NC2CC(NC(C(n3ccc(C)n3)(C)C)=O)C2)cccc(Cl)c1 CC(C)(CC(=O)N1CC2C(NC(c3ccncn3)=O)C2C1)C1CC1 Cc1ccc(O)c(CC(N2CCCC(NC(C3CCCCC(=O)N3)=O)CC2)=O)c1 c1(C(N2CCN(C(C(CC)C)=O)CC(O)C2)=O)ccc2ncncc2c1 S(=O)(=O)(c1cccs1)NC(C)C(=O)NC1CN(C(c2cc(Cl)cnc2O)=O)C1 C#Cc1ccccc1CNC(=O)C(C)N(C)C(c1cncc(CO)c1)=O N1(C(c2cn(CC)nc2C)=O)CC2CN(C(=O)CNc3ccccn3)CC2(C)C1 N1(C(CC(CC(C)C)NC(CC(CC)C(C)C)=O)=O)CCc2ccc(F)cc21 c1(C(N2CCC(CC(N3CCCC(CO)(CO)C3)=O)C2)=O)ccc2cccnn12 C1(NC(CCOCC)=O)CC2CN(c3ncccc3C#N)CC12 C#CCC(C)(C)C(=O)N1CC(NC(=O)CC(CN(C)C)CC)C(C)(C)C1 C12(O)CCCN(CC1)C(=O)NC2.c1(OC)ccc(C)c(C)c1COC(C)(C)C c1(NC(C2CCCN2C(c2cccc(Cl)c2)=O)=O)cc(Cl)ccc1 CC1CCC(NC(=O)NC(C(O)C(F)(F)F)C2CC2)CC1C c1(C(=O)NC2CC(CNC(C(CC)n3cccn3)=O)C2)ccc2c(c1)COCO2 C1(C(N2CC(C)(NC(=O)CCCCN3CCCC3)C2)=O)(COC)CC(C)(C)C1 C(=O)(C1=CCCOCC1)N1C2CN(C(C3C(OC)CCC3)=O)C(C2)C1 N1(C(C(c2ccoc2)NC(c2cccc(F)c2F)=O)=O)CCCC2(CCC2)C1 Cc1cc(C(=O)N(CC(C)(C)NC(c2cnc(O)c(Cl)c2)=O)C)c(O)nc1C C(=O)(C(F)(F)CCc1ccccc1)NC1C(NC(c2c(CC)nn[nH]2)=O)CC1 CCCCN=C(NCc1nc(-c2ccccn2)no1)NCC1(O)CC2C=CC1C2 N1(C2CC(CNC(CC)CC)C2)CC2CCCC2(Oc2ccc(OCC)cn2)C1 C1(CC(N2C(CN(C(=O)CC3(C)CCC3)CC)CCC2)=O)CCC2(CC2)CO1 c1(C(N(C2CCC(NC(=O)CCc3ncco3)C2)C)=O)cccc(C=C(F)F)c1 N1(S(=O)(=O)Cc2ccc(F)cc2)CCCN(CC2CCCC2(F)F)CC1 N1(C(C(C)N(C(=O)CCN(C)C)C)=O)CC(N(C)C)C(C)(C)C1 CCC(C)(COC)C(=O)NCCNC(c1ncn(C)n1)=O.C(=O)OC CC1CCC(CC(N2CCC(OCC(=O)NCC3CC3CO)C2)=O)CC1 N1(C(C=CCCC(C)C)=O)CCC(NC(c2ccsc2C(F)F)=O)C(C)C1 CC(C)CC(C(=O)NCC(F)C1CCC1)ONC(c1cccc(N)c1)=O C1(C(N2CCC(CC=C)(NC(=O)COCC3CC3)C2)=O)CCCC2(CCC2)O1 Cc1cnn(C)c1CC(=O)NCCCCC1CN(C(=O)C=CC2CC2)C1 c1(C(=O)NC23CC(NCc4c(COC)onc4C)(C2)C3)cccc2ncnn12 N1(C2(COC)CC2)C(=O)C(C(=O)OC)N(C(C)CCn2ccnc2)C1=O c1(C(N2CC3(CC(NC(C45CCC(C4)C5)=O)C3)C2)=O)ccc(NC2CC2)c(F)c1 C12(CC)CC(NC(C3(C)C=CCC3)=O)(CN1C(c1ccc(N(C)CC)cc1)=O)C2 C1(NC(CCn2c(C)ncc2)=O)CCCCCC1NC(C1(CCF)CC1)=O C#Cc1ccc(Cl)c(C(=O)NCC2CC2CNC(=O)CC2CCC2)c1 C#CC1(C(=O)NCC(=C)C)CCN(C(c2cc(C)ccc2C)=O)C1 C1(C(N2CCC(O)(CNC(C=C(CC)C)=O)CC2)=O)CCc2nn(C)cc2C1 N1(C(c2cn(CC=C)nc2)=O)CCC(C)C(N(C)C(c2nccnc2C)=O)C1 CCCN=c1nc(N2CCC(C3(C)COC(=O)N3)CC2)c2ccccc2[nH]1 S(=O)(=O)(c1ccc(F)cc1F)N1CC2(CCN(C(c3c(OC)cccn3)=O)C2)C1 c1(C(=O)NC2C(C)(C)CN(C(C3CCC3C(N)=O)=O)C2)cnc2[nH]cncc1-2 C1(NC(c2c(N(C)C)nccc2)=O)CC(C2CCN(c3nnnn3C)C2)C1 C1(C(=O)NC2CC(C(=O)NC3C(OC)COC3)C2)NC(=O)OC1C C#CCC(CC(=O)N1CCN(C(=O)CC2CCC2)CC1CCOC)c1ccccc1 Cc1ccc(OOC(CCC(N2CC3C(N(CCOC(F)(F)F)C)C3C2)=O)=O)cc1.O C(=O)(C#CC(C)(C)C)NCC(c1cccc(OC)c1)NC(c1cnc(C)[nH]1)=O C1(COC)CCCCN1C(=O)CC1CCN(C(C)=O)CC1.C12(SC)CCN1C2 c1(C(=O)NC(C(=O)N(C(C=C)C)C)Cc2ccco2)ccncc1F N1(C(c2cc(COC)[nH]n2)=O)CCC2CCCN(C(=O)CCN(C)C(C)=O)C2C1 N1(C(C(CCC)C)=O)CCN(C(C2(n3ccnc3)CCCC2)=O)CC1C1CC1 c1(C(N(C2CCN(C(=O)CC)CC2)CC)=O)ncccc1C.C(C(C)(C)C)OC(C)=O N1(C(C(C=C)C)=O)CC(NC(c2nnn(CC)c2C)=O)C(C2CC2)C1 N1(C(c2cn(CCC)nn2)=O)CC2CC1C2C(=O)N(C)Cc1c(C)noc1C CC12CCC1(C)CN(C(=O)C1=CCC(NC(C3(C#N)CC(F)(F)C3)=O)C1)C2 c1(NC(c2ncc(-c3c(C)cc(OC)nc3)c(C)c2)=O)cc(F)c(Cl)cc1Cl C1(N(C)C(C2CCOC2)=O)CN(C(=O)Cc2ccccc2CS(N)(=O)=O)CC12CC2 C12(C(N(CC(C)NC(=O)CCCCO)C)=O)CCCCC(=O)N1CCC2 CC(C)(C)CCCCNC(c1csc(CNC(C2(C)CCCNC2=O)=O)c1)=O c1(C(c2n(C(CC)C)nnn2)NC2(C)CC(C(N)=O)C2)nn(CC)cc1Br c1(CC(N2CC(OCCNC(C3CCC(OC)CC3)=O)C2)=O)ncn2c1CCC2 c1(C(N2CC(NC(C(CC)n3cncn3)=O)C(F)C2)=O)c(O)nnc2c1CCC2 C1(OC)CC2CC1CN(C(C1C(O)C(O)CN1C(=O)OC(C)(C)C)=O)C2 N1(C(c2cc(C(C)=O)on2)=O)CCN(C(C2CC2(F)F)=O)CC1c1ccccc1 CC(C)C(C(C)NC(c1c[nH]c(-c2ccccc2)c1)=O)NC(=O)CC1(CO)CC1 CC1(C(N2CCC(F)(CNC(=O)C3=CCCCO3)C2)=O)CCCCC1(F)F Cc1ncc(COCC(=O)N(CC(O)CNC(=O)C(O)c2ccsc2)C)s1 C1(CNC(C=Cc2cnc(C)s2)=O)CC2CCC(C1)N2C(=O)C(F)CC(C)C c1(C(=O)NCCCCC2CN(CC34CC3CCC4(F)F)C2)cc2c(Cl)cncc2s1 CC(C)CCCCCC(=O)N1CC(CCNC(C2(CC(F)F)CC2)=O)OC(C)C1 c1(NC(CCC2CCN(C(CC3CC(CC)C3(C)C)=O)CC2)=O)ccc(F)cc1C C1(C(N(CC#CC)CC#C)=O)C2CC2CN1C(c1cnc(C)o1)=O c1(C(=O)NCC2(CC(=O)NCc3ccccc3CO)CC2)onc2ccccc12 C=CC(C)(O)CC(=O)NCC12CC1CN(C(=O)COCCOC)C2 N1(C(C2(CCC)CC2)=O)CCC(N(C)C(c2n[nH]c3ccccc23)=O)C2(CC2)C1 c1(-c2ccc(SC)nc2)ccc2c(c1)c(C(=O)NCC(C)O)cn2C C1(C(=O)NCC2CN(C(=O)OC)C2)CC(NC(C2CCCC(C#N)C2)=O)C12CCC2 C(=O)(C(C)C(C)C)N1C(CNC(CNC(CC2(OC)CCC2)=O)=O)C=CC1 C1(C(=O)OCC)CC2CC2N1C(=O)NC(C1CCOCC1)C(F)F C1(C(N2C(CN(C(CCOC)=O)C)CCC2)=O)CCC(=O)N1C(C)C N1(C(C)=O)CCC(N(C(=O)COc2ccc(C(C)OC)cc2)C)CC1 N1(C(CCSCc2cnc(C)s2)=O)CC(NC(=O)C(C)(C)C(N)=O)CC1(C)C CC(C)(O)CC(=O)NCC1(CC(=O)NC2COCCOC2)CC1 N1(C(C(C=C)C)=O)CC(O)CC1CNC(C1(CF)CC1)=O c1(-c2cccc(SC)c2)nn(C)c2cc(C(=O)NCc3nc(C)c(Br)s3)ccc12 CCCC(C)C(=O)N(CC(O)CCOCC)CCCC1CCC1 N1(C(C(C)OCC#C)=O)CCC(F)(C(=O)NC2(c3cc[nH]n3)CC2)CC1 C(C1CCCN1C(c1ccncc1CC)=O)=CC(=O)NC(C(=O)N(C)CC)C CCC(C)(COC)C(=O)N(C)CCN(C(C1CC12CC2)=O)Cc1ccccc1 c1(CC)cc(-c2cn(CC(C)(C)C3CCCC3)nn2)ccc1O C1(NC(C(C)OCCN(C)C)=O)C2CC(O)C1N(C(c1c(Cl)cnn1C)=O)C2 C1(C(N2CCOCC(C(=O)NCC3(OCC)CC3)C2)=O)Cc2ccccc2C1 C1(CN)CCC(C(=O)NC2(c3cn(C4C(SC(C)(C)C)COC4)nn3)COC2)C1 c1(N2CC(NC(C(C)(C)OC)=O)C(C#N)C2)ncc2ccc(F)cc2n1 CCCCC(CC)C(=O)N1CCCCC1C1CCN(C(C2CC(C)C2)=O)C1 C(=O)(C(C)(C)CC(=O)OC)OCC.C1(N2C34CC(C3)(C4)C2=O)CCNCC12CC2 c1(C(=O)NC(CNC(C2C(OC)CCC2)=O)C2CC2)sc2cncn2c1C N1(C(C2C(CC)C2)=O)CC2(CCCN(C(=O)Cc3cccc(C)c3)C2)C1 C1(c2cn(CC=C)nn2)CCCCN1C(=O)CC(=O)NCSc1ccccn1 c1(C(N(CCCCNC(=O)Cc2cnn(C)c2)C)=O)ccnc2c1CCC2 c1(CCn2cnc(Br)c2)ccc(F)cc1.c12coc(n1)CN(C)S(=O)(=O)C2 CC(C)(F)CCC(=O)NCC1COCCN(C(C2CC2F)=O)C1 c1(C(=O)NC2C(CNC(c3c(SC)snn3)=O)C2)c(F)ccc2nc[nH]c12 Cc1sc(C)c(C(N2CC3CC(NC(c4cnn(C)c4C#N)=O)C3C2)=O)c1C#N CC1CCCCC1(C)C(=O)NC1CC(c2ccccc2)NC1=O N(C(=NCCN1CCCC1)NC1CC2CCC1O2)Cc1c(Cl)scc1 N1(C(=O)Nc2cc(C)c(F)cc2C)CC2CC(O)C(O)CC2C1 c1(N(C(N2C(c3nc(C)[nH]n3)CCC2)=O)C)ncncc1C c1(C(=O)NC2CCC(C)N(CC=CCl)C2)coc2ccccc12 CC1CC(=O)NCC1C(=O)NCC1CC(CC(=O)NCc2cn(C)nc2CO)C1 Cn1cnc2[nH]c(C(=O)NC3CN(C(c4cccc(N)n4)=O)CC3N=[N+]=[N-])cc12 N1(C(C(C2CCCCCC2)OC)=O)CC2C(CNC(c3cscn3)=O)C2C1 N1(c2nc3cc(n2)NC3)CC(C)NC(=O)C1(C)C.C1(CC=C)(OC)CCSCC1 C1(C(=O)NC2CC(NC(C(C(C)C)N3CCC3)=O)C2)Cc2ccccc2CO1 CCCC(CNC(c1sccc1Cl)=O)C(=O)N(C)Cc1cn[nH]c1 N1(C(C2CC=C(C)CC2)=O)CCC(F)(C(N2CCC3CC23)=O)CC1 CN1CCC(CC(N2CCCCC2Cn2cc(CSCCO)nn2)=O)C1=O O=C(C1=CCC2(COC2)OC1)NC1CCCCC1NC(c1cnn(C2CC2)c1)=O C1(c2n(C)ncc2)C(C(=O)NCc2nnc(O)n2C)CCC(=O)N1C1CC1 c1(C(=O)NCC2N(C(C(CC)(C)O)=O)C3CCC2C3)ccc(S(C)(=O)=O)c(Cl)c1 C12(CNC(=O)CSCC3CCCCO3)CC(C1)C(NC(C1CCC1)=O)CO2 C1(NC(c2c(Cl)cn(CC)n2)=O)CCN(C(C2CCC(=O)N(C)C2)=O)CC1O N1(C(C(CCCC)O)=O)CCCC2CN(C(=O)CCCc3nc(C)no3)CCC12 c1(C(N2CCCC2C2CC2)C(=O)NCC)cc(Br)ccc1C N1(C(C2C(c3c(C)cccc3)C2)=O)CC(C2CN(C(=O)C=CC3CCCO3)C2)C1 C1(N(C(CC2CCN(CC)C2)=O)CC(F)Cl)CC2(CCNCC2)C1 C1(C(N2C(C)(C)C(NC(c3cc(Cl)c[nH]3)=O)CC2)=O)CCc2cnnn2C1 C(N=c1cc(NCC2CC3(C2)CC(O)C3)nc[nH]1)C1(C)CCN(C(C)C)C1 c1(CC)cc(C(=O)NCCC(C(=O)NC2CCN(C)C2C)OC)ccn1 C(=O)(C(F)(F)C(C)(C)O)N(CCNC(C(c1cccc(C)c1)O)=O)CC1CC1 c1(OC)cccc(NC(=O)C(N2CCCC(CN(C)C)C2)c2ccc(C)s2)c1 C1(C(=O)Nc2c(O)ncnc2O)CC2CCC(C1)N2C(c1ccc(Cl)c(Cl)n1)=O N1(C(C(C)OCCN(C)C)=O)CC2(NC(=O)CCC(C)(C)C#N)CCCC2(F)C1 C1(CN(C(CCCOC)=O)C)CCN(C(=O)CCn2cc(Cl)cn2)CC1 C12(NC(c3n(CCC)nc(C)c3)=O)CCC(CNC(=O)C(C)CC)(CC1)OC2 c1(C(c2nnnn2C(C)(C)C)NCC2CC(CC)C2)cc(CCOC)on1 N1(C(CN(C)CC)=O)CCCCCCC1C(=O)NC1COCC1N=[N+]=[N-] c1(CC)n[nH]cc1C(N1CC(C2CCN(C(=O)CSC(C)C)C2)C1)=O C1(=O)CC(C(F)(F)F)N1.C(=O)(C1=CCCC1)NCC(c1ccccc1)N(C)C c1(C(N(C2CC(Nc3c(C(=O)OCC)cccc3)C2)C)=O)c(OC)ccnc1Cl c1(C(=O)NC(CC)CNC(=O)C(C)CC2CCCC2)nc(O)nc(O)c1N c1(CC)cc(OC)ccc1C(=O)N(C1CCN(C(=O)C(O)CSC)CC1)C C1(C(=O)NC(C2CCOC2)C#C)CN(C(c2cc(Cl)ns2)=O)C2(CCC2)C1 C1(C(N2CCN(c3cc(Cl)ccc3Cl)CC2)C(=O)NC2CC2)CCOC2(CCC2)C1 c1(C(N2CC(NC(C3C(C#C)C3)=O)CC23CCC3)=O)ccn2c(C)cnc2c1 c1(C(=O)NCC=CCNC(c2ccc(C(C)C)c(N)c2)=O)ccccc1S(C)=O c1(N2CC=CC(NC(C(C)=C(C)C)=O)C2)ncnc2cccc([N+](=O)[O-])c12 C1(NC(c2cc(OCC)no2)=O)C2CC1N(C(=O)CC1CC=CCN1C)C2 C=CC(CC)C(=O)N1CCC(CNC(=O)CCCCC2CC2)CC1 Cc1ncccc1C=CC(=O)NC1(CNC(=O)CCn2cccc2)CCCCC1 C1(NC(CNC(CC)=O)=O)CN(C(=O)Cc2ccnc(OC)c2)CCC1CO C1(C(C)(C)NC(C2CC=CCC2)=O)CCN(C(=O)C=CCN2CCC2)CC1 C1(C(=O)NCC2(CN(C)C(c3ccncc3Cl)=O)CC2)CC2CCCC12 Cc1nc(=N)[nH]c(C)c1C(=O)NCC1CCCC1NC(C1(O)CC1(C)C)=O Cc1nc(C(C)C)sc1C(=O)NC1CN(C(=O)C(Cl)=CCl)C2CC12 c1(OCC)nnc(SC)nc1N1CCCC(F)(NC(c2ccnn2C2CC2)=O)C1 c1(NC(C2(C(F)(F)F)COC2)=O)cn(CCCN2CCSCC2)nn1 C(CCCCC(=O)N1CC(NC(c2ncc(C(F)F)s2)=O)CC(O)C1)SC C1(CC)CCC(F)(F)CC1.c12cc(C)ccc1NC2c1nnnn1CCCOC c1(CC2N(C(C(=O)NCCC)=O)CCOCC2)ccc2nc(O)c(C)cc2c1 c1(C(N2C3CCC2CC(C(N2CC(S(N)(=O)=O)C2)=O)C3)=O)cc2cccn2cn1 N1(C(CN(CCC)C(c2cn(CC3CC3)nn2)=O)=O)CCOCC1CC1CC1 C=CC1OCCC1C(=O)N(CCN(C(=O)CCCc1nnc(C)n1C)CC)CC C12(NC(c3c(Cl)cn(CCC)n3)=O)CCN(C(c3cnn(C4CC4)c3)=O)CC1C2 C(CC(C)C(=O)NCCNC(c1c(C)noc1C(F)(F)F)=O)OC c1(-n2cc(NC(c3c(C(F)F)cccc3Cl)=O)nn2)cccc2cccc(Cl)c12 N1(CC(c2ccc([N+](=O)[O-])cc2)c2ccco2)CCCc2sccc2C1 C1(NC(c2c(C)ccn2C)=O)CCN(C(c2nn(C)c(Br)c2C)=O)C(C)C1 Cc1ccc(NC(=O)CC2CN(C(c3c[nH]nc3C)=O)CCO2)c(C)c1 CC1CN2CCN1C(C(=O)NCC(C)(C)NC(c1cc(C(F)(F)F)nn1C)=O)C2 c1(C(=O)NCCNC(C(C)(O)CC(F)(F)F)=O)cc(Cl)cc2ccncc12 C1(N(C)C(c2cnc[nH]2)=O)C2CN(Cc3ccnn3CC(F)F)CC12 C=CC(C)(CCOC)C(=O)NC1CC(C)(NC(=O)CC(C)C2CC2)C1 C1(OC)CC(C(=O)NCC(O)CNC(C2CCN(C(N)=O)CC2)=O)CC1OC c1(C(N2C3CC(CNC(c4n(CC)ccn4)=O)C2CC3)=O)nnc2ccccn12 N1(C(CCc2c(C)cc(Br)cc2)=O)CCN(C(c2cnc[nH]2)=O)C(C#N)C1 C1(NC(C(C)(O)c2ccccn2)=O)C2CN(Cc3cccc(I)c3)CC12 c1(OC)c(CC=NOCC2CC2)cc(Cl)cc1Br N1(C(CCCSC)=O)C2CCC1C(NC(=O)COc1ccc(C(N)=O)cc1)C2 CC1(C)CCCC(C(N2CC=CC2CNC(c2cc[nH]c2C2CC2)=O)=O)CC1 N1(C(c2ccc(C(C)(C)C)o2)=O)CCC2CCCN(C(=O)C3=CCOC3)C2C1 C1(NC(C2(COC)CN(C(=O)CC3=CCN(C)CC3)C2)=O)Cc2ccncc2N1 c1(C(C)NC(=O)C(N2CCCC2c2cccc(F)c2)=O)ccc2cnccc2c1 C1N=C2NC=NC(=C2C)NCc2occc21.C(=O)(CCC(C)N1CCCC1)OCC CCC(C(=O)N1CC(C(=O)NCC2CC(OCC)C2)OC(C)C1)C(F)(F)F c1(C(=O)NC2CN(C(C(P(C)(C)=O)O)=O)CC2O)cnc2ccnn2c1 c1(CC(=O)NC(=O)N)[nH]nc(C)c1Cl.C1(N(CCOC(F)F)CC)CCCCN1 c1(C(N2CC(O)(C(C)NC(C3CCCCCC3)=O)C2)=O)nnc(O)nc1O C1(CN(C)C(c2cc(O)cs2)=O)CN(C(=O)CCc2ccoc2)CCO1 N1(C(CCC)=O)CCC2(C=C(C(=O)N(C(Cc3ccccc3)C(=O)O)CC)C2)C1 N1(C(=O)CN2CC3CC3C2)CC2C(NC(c3n[nH]cc3Br)=O)CS(=O)(=O)C2C1 Nc1cc(C(N2CC(C3(NC(c4ccoc4)=O)CC3)C2)=O)cc(O)c1Cl N1(CCN(CC(C)O)C(=O)Cc2cn[nH]c2)CCN(N(C2CCC2)C(C)=O)CC1 n1(CCC(=O)N(CCNC(C(CC)NC(N)=O)=O)C)ccc(O)nc1=O CCC(CC(=O)N1CCN(C(c2cnc(S)nc2)=O)CC1C(C)C)C(F)F C(C1CN(C(c2ccc(O)cc2F)=O)CC1C(=O)NC1(C)CCCC1O)=CC c1(C(N2CCN(C)CC2CNC(=O)CC2(O)CCC2)=O)ccc2c(c1)N(C)CC2 c1(C(=O)NCC(C)(C(C)C)NC(C(C)=C2CC2)=O)ccc2c(c1)NC(=O)CCS2 c1(C(N2CCN(C(CNC=O)=O)CC23CC3)=O)ccc2c(c1)CCCO2 c1(CNC(CCOC2CN(C(CCC3C(C)C3)=O)C2)=O)nccn1C(C)(C)C C=CCCC(F)(F)C(=O)NCCCC(C)NC(C1CCCS(=O)(=O)N1)=O CC(C)C(C(=O)N1CC(O)(C(C)NC(=O)C2=CCSC2)C1)N1CCCCC1 Cc1nn(-c2cccc(Cl)c2)c(C)c1CNC(N1CCC2(CC2)C1)=O CC1(CNC(=O)C(F)=C2CCC2)CN(C(=O)C(O)Cc2ccccn2)CCO1 N1(C(C)=O)CCOCC1C(=O)N(CC(C)(C)NC(=O)CC1CCCCO1)CCO c1(C(N2CCC(c3c(F)cccc3F)(C)C2)C(=O)NCC)ccc2ccn(C)c2c1 C1(CNC(c2ccc3[nH]ccc3c2)=O)CCC12CCN(C(C1CC1F)=O)CC2 c1(C(=O)NC2CN(C(CCC(N)=O)=O)CC2O)cncc2c(O)nccc12 C1(NC(=O)Cn2cnnc2O)CCN(c2cc(C(F)F)ncn2)CC1O c1(C(N2CC(C)(CCC(=O)NCCOC)C2)=O)ccc2nc[nH]c2c1 C1(NC(C(C=C)O)=O)COC2(C1)CN(C(c1occc1C)=O)C2 C1(O)(CNC(C=CC)=O)CCCN(C(C2(C)CNC(=O)N2)=O)C1 CCC(C)(C)C(O)C(=O)N(CCNC(c1cnn(C(C)(C)C)c1Cl)=O)C1CC1 C1(C(=O)NC2CCN(C(C)=O)C2)(COC)CN(C(c2occc2C)=O)C1 CCC(C)C(C)C(=O)N1CCCC1CNC(c1cccc(C(C)C)c1)=O CCCC(C(=O)N(C)C)NC(=O)C(COC)NC(=O)C(O)Cn1cncn1 Cc1nn(C(F)F)c(C)c1CC(N1CCC(C)C1CNC(=O)C(Cl)=CCl)=O c1(C(N(CC(C)(C)CNC(c2n[nH]cc2Cl)=O)C)=O)ccc2oc(=O)oc2c1 c1(NC(C2C(C(=O)NCc3cccc(OC)c3)C2)=O)ccc(OC(F)F)c(Br)c1 CC1(C)CCCN(C(c2ncccc2O)=O)C1C(N1CC(S(N)(=O)=O)C1)=O C1(CNC(CC(=O)NC(C)C)=O)CC(OC(C)(C)C)CN1C(=O)OC(C)(C)C C1(NC(C(C)OC(C)(C)C)=O)CCC2(CC1)CN(C(C1CCCCNC1=O)=O)C2 C1(CC)CN(C(c2ccoc2Cl)=O)CCC1NC(c1conc1C1CCC1)=O c1(SCC(=O)N(C)C)cnn(C)c1.C12(C(N3CCN3)=O)COCC1C2 c1(N(C)C)ccc(C(=O)Nc2nnc(-c3ccc(F)cc3)o2)cc1[N+](=O)[O-] c1(CC)occc1C(=O)NC1CCN(C(=O)CC(C)OC)C1 c1(OC)ccc(NC(c2nnnn2C2CC2)CCC2(C)CC2)cc1C(C)C C1(CNC(c2cnc3[nH]cnc3c2)=O)CC2CCC(C1)N2C(c1occc1Br)=O c1(C(C)NC(C2CC2CNC(=O)N(C2CCCC2(C)O)C)=O)ccncc1Cl N1(CCC(=O)NCC(C)(C2CC2)NC(C2CCCS2)=O)CCNC(=O)C1 N1(C(C2=C(C)OCC2)=O)CCC(NC(C2CC(F)(F)CCC2(C)C)=O)C(C)(C)C1 C(C(CO)(CO)NC(c1nn(C)cc1C)=O)N(C(c1n(CCC)ncc1)=O)C C=C(C)C(C)(C)C(=O)NCC1CN(C(=O)CCCNC(C)=O)CC12CC2 N1(Cc2cccc(C(=O)O)c2)CCCOC(CNc2ccc(Br)cc2)C1 C(=O)(CS(=O)(=O)C1CC1)N1CCC(CNC(c2cncc(C3CC3)n2)=O)C1 C(N=c1[nH]c2ncnc-2c(C(=O)NC)[nH]1)C1(O)CN(C(C=C(CC)CC)=O)C1 C1(NC(CC2(O)CN(C(CCC(=O)NC)=O)C2)=O)CCc2nncn2C1 C1(NC(C(CC)C(C)(F)F)=O)CN(C(=O)C=C(C)C)C2(CCCC2)C1 C1(C(=O)NCCN(C(=O)C(C)C(C)O)CCCCCC)CCC(C)(F)CC1 c1(C(C(=O)NC(C)C(C)NC(=O)C(O)CC(N)=O)(C)C)ccc(F)c(F)c1 C1(C(N(C(CCNC(C(CC#C)C)=O)C)C)=O)CC12CCC(=O)CC2 Cc1cccnc1C=CC(=O)NCC1CCC(NC(C2CC2c2cnn(C)c2)=O)C1 c1(OCC(N2CC(OC)(CNC(=O)C(O)P(C)(C)=O)C2)=O)cc(F)c(C)cc1F C1(C(C(=O)NCCN2CC(OC)C2)F)CCN(C(=O)Cc2cnc(C)s2)C1 c1(C(N2CCC(O)C(C)(C)C2)C(=O)NCCOCC)ccnc2ccccc12 Cc1cccn2cc(CO)nc12.C1C(C2CC2)NC(=O)N1 c1(C(N2CCCC(NC(C(CC)(CC)CO)=O)C2)=O)cc2ccccc2nc1C c1(C(=O)NCC(C)CNC(c2coc(Cl)c2)=O)coc2ccc(Br)cc12 C#CCC(C)C(=O)NC1(CNC(c2csc(Br)c2C)=O)CC1 N1(C(c2c(C)ccc(=N)[nH]2)=O)CC2CC(NC(c3cnc(S)n3C)=O)CC2C1 C1(OC)CN(C(=O)C2=CCCNC2)CCC1NC(c1cnccc1Cl)=O C1(NC(C2(CCN(C)C)CC2)=O)COC2(CCN(C(=O)C=C3CCOCC3)C2)C1 n1(CC)cnc2c(NC3CNC(=O)C3)[nH]c(=NCC3CCS(=O)(=O)C3(C)C)nc12 N1(C(C(=O)Nc2ccccn2)=O)CCC(Cc2ccc(F)cc2)C(F)(F)C1 C1(C(=O)NCC(C)(C)OC(C)C)CCN(c2ccccc2)S1(=O)=O N1(c2cc(C(C)=O)ncn2)CCC(C)C(NC(=O)Cn2nc(Cl)ccc2=O)C1 CCC(CO)C(=O)NC1(C)CCN(C(=O)C2=CCCC2)C1 C12(CNC(C(C)(CC3CCC3)OC)=O)CC(CO1)N(C(=O)C=CC(C)C)C2 Cn1cc(C(=O)NCCNC(c2c[nH]nc2-c2ccncc2)=O)c(Br)n1 N1(C(c2ncc(C)cn2)=O)C2CCC1CC(NC(=O)C(C)C1CC1)C2 c1(C(=O)NCC2C3CN(C(CC4C=NN(C)C4=O)=O)CC32)cccc2nc[nH]c12 C12(C(N3CC(CC(=O)OC)C3)=O)CC(CCO1)N(C(C1CC3CCC(C1)C3)=O)C2 N1(C(C2C(CC)CCO2)=O)CCC(CNC(c2n[nH]c(C)c2Cl)=O)(OC)CC1 N1(C(c2csc(Cl)n2)=O)CC2CCCN(C(c3ccc4ncsc4c3)=O)C2C1 c1(C(N2CC(C)C(C(=O)NCCn3cc(CO)nn3)C2)=O)ccc(Cl)c(F)c1F C(C(=O)NCC(O)CNC(=O)C(C1CCCCC1)=O)(C(C)(C)C)N(C)C c1(C(N2C(COC)(CNC(=O)CCOC3CCC3)CCC2)=O)ccc(F)c(O)c1 C(=O)(CC(C)C(C)(C)C)N1CCC(C=C)(C(=O)NC2CN(C)CC2O)C1 N1(C(c2ccc(CNC(C)=O)o2)=O)CCC(C2CN(C(=O)CCCC(C)C)C2)CC1 N1(C(c2cc(C)nc(O)c2)=O)C2CCC1C(F)C(NC(=O)CNC(=O)C1CC1)C2 C1(CC)C(C(=O)NCC(C)CCCO)CCCN1C(C1CC(SC)C1)=O CCCC(C)C(=O)N1CCCC1C(C)OC.c12coc(n1)CNC2=O N1(C(C2(CC(C)C)CC2)=O)CC=C(CC(=O)NCC2(C)CCCC2)CC1 C1(C(N2CCC(CC=C)(NC(C(C)NC(=O)OC)=O)C2)=O)CCc2nncn2C1 N1(C(C2CC(=O)CO2)=O)CCC(F)(CNC(C2(n3cncn3)CC2)=O)CC1 N1(C(CCc2scc(C)c2)=O)CCC2CCN(C(=O)C(C)Cc3ccco3)CC12 N1(C(C)=O)CCC(C(N2CCC(O)(c3cccc(C(F)(F)F)c3)C2)=O)C(C)C1 N1(C(CCOCC(C)C)=O)CCN(C(C2CC2(C)Br)=O)CC1C(C)C C(=O)(CCC(C)(C)NC(=O)CC1CCOC1)NC(C(=O)NCC)C1CC1 CCC(O)C(C)C(=O)N1CCCC(F)(CNC(c2ccc(-c3ccco3)o2)=O)C1 C1(CC(=O)NOC2CCC2)CN(C(=O)CCC2CCCO2)CC12CC2 N1(C(CC2(NC(C)=O)CC2)=O)CCC2CCN(C(C3CC(=O)C3(C)C)=O)CC2C1 C=CCCCC(C(=O)NOCCC(C)O)NC(=O)CC1(O)CCOCC1 N1(C(CCC(=C)C)=O)CC2CC(N(C)C(C3CCCC(C)(C)C3)=O)C1C2 C1(CC)CN(C(C2NC(=O)CC2C)=O)CCC1NC(=O)CC1CC(F)(F)C1 CC1(C)CCOC(CNC(C2(CCNC(=O)CN=S(C)(C)=O)CC2)=O)C1 N1(C(C2N(C(CC)=O)CCCC2)=O)C2CCCC1CC(NC(=O)CSC(F)F)C2 CC(C(=O)N1CCC(CCNC(=O)C(C2(O)CCCCC2)(F)F)C1)C(C)O C1(C)(NC(C)C)CCCN(C(=O)NCC2CC(OC)C2)C1.c12ccc(cn1)o2 N1(C(c2cc(C)no2)=O)CCOCC(CNC(C2CC(C#N)C2)=O)C1 C1(CC(=O)OCC)CCCN(C(N2CCOCC2)C(=O)NCCCOC(C)C)C1 c1(C(CC)C)nccc(=NC(C)C2CN(C(C3CCC(C)C3)=O)CCO2)[nH]1 C1(C(=O)NCc2scc(CC)n2)CC(NC(=O)CCOCC(C)C)CCO1 C=CCC(CC=C)C(=O)N1CCN(C(=O)CC(C)(C)C(F)F)CC1CC(C)(C)C c1(NC(C2CN(C(=O)Cc3ccccc3)CCS2)=O)nc2cc(Cl)ccn2n1 C1(C(=O)NCC2(NC(CC(C)C3CC3)=O)CCC2)C2CCC1(C)C2(C)C c1(NC(C)C(=O)NC2CN(C(=O)CCCCCN(C)C)C2)ccc(C#N)cc1 N1(C(CCC(CC)=O)=O)CCC2CC2(C(=O)NC2CC2c2cncs2)CC1 C1(CC(=O)NCC2CC(C)(O)C2)C2CCCC2N1C(=O)CC12CCC(CC1)C2 Cc1nn(-c2ccccc2)c(C)c1C(=O)NC(CNC(=O)Cc1cccs1)CO N1(C(=O)Cn2cc(CO)nn2)CCC(C2CCCC2)C1.C1C(=O)O1 c1(CNC2CC(CNC(c3c(OC)cccc3)=O)C2)c(C)cc(Br)cc1C N1(C(C(C)OCCC#C)=O)CC2CN(C(c3c[nH]nc3C(C)C)=O)CC2C1 c1(C(N2CC(NC(C3C(C(N)=O)C3)=O)C(F)C2)=O)cnn2c1OCCC2 C1(OC)CCn2cc(C(=O)NCC(O)CNC(c3cncs3)=O)nc2C1 N1(CCS(N2CCC(N(C(=O)CN3CCCC3)C)C2)(=O)=O)CCCNC1=O c1(C(N(CC(O)CNc2ccnc(-c3cccnc3)n2)C)=O)cnc(O)cc1O C(C)(N=c1[nH]c(N2CCOC3CCCC23)nc2cc[nH]c12)c1c(C)cccc1 C1(NC(c2cccc(CC)n2)=O)CCN(C(c2ccc(CC)cc2)=O)C(C)C1 N1(C(c2cncc(C)c2C)=O)CC(F)(F)CC1(C)CNC(=O)Cc1csc(C)n1 CC1c2ccc(C(=O)O)n2CCN1C(=O)C(C)(C)C.CCCCN1CC1 C=Cn1nccc1C(=O)N(CC(=O)NC(C)CC(C)(C)OC)CC(C)C c1(C(=O)NCCC(=C)CNC(=O)Cn2cc(C)cn2)cccc(C(N)=O)n1 C(CCCCCCC(=O)NCC1CN(C(c2cc(O)cs2)=O)C(C)(C)C1)SC C1(CN(C(=O)Cn2nnc(=O)[nH]2)C)CCCN1C(c1cc[nH]c1C1CCC1)=O N1(C(c2ncn(C)c(=O)c2)=O)CCC2CC2(C(=O)NC2CCCC2)CC1 CC(O)CCCN=C(NCC1CC1)NC1CC1C(F)(F)F CC(C)(C)C(CO)C(=O)NCC1(NC(=O)C2CC2)CC1.c12nc(cc(O)n1)C2 Cn1cc2c(n1)CCCC2C(=O)N1CCC(N(C(=O)C=CC(=O)N(C)C)CCO)C1 N1(C(c2ncoc2CCN=[N+]=[N-])C)CCc2c(cnn2-c2ccccc2Br)C1 C1(NC(C(C)(C)C)=O)CN(C(=O)C2=CCCC2(C)C)Cc2ccnn2C1 c1(CNC(C)=O)ccccc1OC(C)CCN(C)Cc1cccnc1 N1(C(c2ccc(C(CC)C)nc2O)=O)CCC2C(CCCN2C(=O)CC)C1 C(c1ccc(F)cc1)=CC(C(=O)N(CCCCN(C)C(C1(C)CC1(F)Cl)=O)C)=O C1(N(C(C(C)C)=O)C)CCCC(CNC(c2cc(CC3CC3)on2)=O)C1 C1(NC(c2cc(=N)[nH]cc2)=O)CC2CC1CN2C(=O)C=Cc1ccccc1 C1(CC(=O)N(C(CNC(=O)C(=O)Nc2ccccc2)C2CC2)C)CCC(=O)C1C C=CC(CC)C(=O)NCC1(C(C)NC(C2CC=CCC2)=O)CC1 C(=O)(C(CC)C(C)C)CCCC#C.C1(CCOC)CNC(=O)C(=O)N1.OCC C(CC(=O)NCC1CC2C=CC1CC2)(C(C)(C)C)NC(C(CC)NC(C)=O)=O c1(CC(N2CC3C(CNC(c4n(C)nnc4)=O)C3C2)=O)c(Cl)cccc1Cl N1(C(C=CSC)=O)CCc2c(ncn2C2CCCN(C(=O)Cc3csc(C)c3)C2)C1 N1(CC(CC(CC)O)O)c2ccccc2C(C)(C)C1C C(=O)(C1CNc2ccccc21)NC1C=CC(CNC(CS(CCCC)(=O)=O)=O)C1 C1(CNC(C(CCC)C)=O)CN(C(c2nnc(S)n2C)=O)CCCO1 C(=O)(C1CCC(=O)c2ccccc21)N1CCC(NC(C2CC(C)(O)C2)=O)(CO)C1 c1(C(=O)OC)c[nH]ccc1=NC1CCCC1NC(C1CCCN1C)=O CC1(CNC(=O)C(CC2CCCC2)NC(=O)CN2CCOC2=O)CCCO1 C#Cc1cncc(C(=O)NCC(c2cccc(C)c2)NC(=O)C(C)NC(N)=O)c1 CCC(CC)C(C)C(=O)N(CCCNC(=O)C=CSCc1ccco1)CC C1(NC(C2(CC)CC2)=O)CCN(C(c2c(C)oc(C(F)(F)F)c2C)=O)C1CC C12(CNC(COCCN(C)C)=O)CC1CN(C(=O)C(=O)NCC(F)(F)F)C2 C1(CN(C)Cc2sc(Cl)nc2Cl)CCCN(C(=O)CCc2ccccc2)C1 C12(C(=O)Nc3ccc(F)nc3)CCC(CN(C(c3cc(C(C)(F)F)n[nH]3)=O)C1)C2 CC(C)C(CC1CCCCC1)C(=O)N(C(C)CCNC(=O)C=Cc1ncco1)C Cc1nc(C(=O)NCC(c2ccccc2CO)NC(C2CCOC2=O)=O)nn1C n1(CC(=O)NC2C(CCC)CN(C(c3cc(C)co3)=O)C2)nc(O)ccc1=O Cc1c(C(N2CC3CCC2CN3C(c2ccc[nH]2)=O)=O)c2ccccc2n1C C1(NC(=O)NC2(C(=O)OC)CC2)CC2CN(CC(N)=O)CCN2C1=O C1(C(=O)Nc2cccc(OC)c2Br)CC2(CCN1C(=O)Cc1cccs1)CC2 N1(C(c2ccc(C#C)o2)=O)CCCC12CCN(C(c1ccc3nc[nH]c3n1)=O)C2 CC1C(N(C)C)CCN1C(=O)CCCN(C)C(C1CC1(F)Cl)=O C#Cc1ccnc(C(=O)NC(C(=O)NCC(C)Cc2cn[nH]c2)C(C)C)c1 C1(C(N2CCC(CCNC(c3cn(CCCF)nn3)=O)C2)=O)CC12CCOCC2 C1(C(N(CC(CC)NC(c2ccc(N)c(O)c2)=O)C)=O)Cc2nnsc2S1 c1(C(N(CC(C)O)CCNC(C2CCCN2N=O)=O)=O)nccc2cccnc12 C1(CC(N2CC(COC(C)=O)C2)=O)CCCN(C(c2cc(C)c(C)[nH]2)=O)C1 c1(CN(C(=O)C(c2ccoc2)NC(=O)COCC2CC2(C)C)C)ccnn1C N1(C(c2c(C)ccnc2)=O)CCOCC(CNC(=O)CCCC(F)F)C1 C1(CNC(c2c(C)nn(CCO)c2C)=O)N(C(=O)C(C)C2CC2)CCCC1(C)C c1(C(=O)NCC2N(C(c3ccnc(CC)n3)=O)C3C(C2)C3)csc(S(C)(=O)=O)c1 N1(C(CC2C(CNC(C3(Cl)C(C(C)=O)C3)=O)C2)=O)CCN(C(C)C)CC1 C1(C)(CNC(C(CC=C)NC(C)=O)=O)CCCN(C(=O)C(O)CF)C1 C1(CCN(C(CC(=C)C)=O)C)CCCCN1C(c1c(C)csc1Cl)=O N1(c2c(C)non2)CC2CCCC2(c2nc(C(N)C3CC3)no2)C1 C#Cc1ccc(C(=O)N(CC2CCCN(C(=O)C(C)N(C(=O)OC)C)C2)CC)nc1 Cc1ncc(C(=O)NCCCCCCF)cc1C(F)(F)F c1(CCNC(C2C(OC(C)=O)C2)=O)cc(C)cnc1O.C1(C(C)C)C(=O)N1 Cc1cc(C(N2CCC(CCNC(=O)CC(C)C3CCCCC3)C2)=O)ns1 N1(C(C2C(c3cn(C(C)C)nc3)C2)=O)CCCC(N=c2[nH]c(C#N)c(Cl)s2)C1 c1(C(N(CC(CNC(c2cc(CC)nn2C)=O)C)C)=O)cc2cccc(C)c2s1 C1(NC(CCCSC)=O)CC(O)CN(C(c2csc(-c3ccc(Cl)s3)n2)=O)C1 C=CCC(CNC(=O)C(c1cnccn1)C)NC(=O)CCCOC1CCOCC1 N1(C(COCCOC)=O)CC(CNC(=O)C(C2CCOCC2)C)C(C)C1 C1(S(N)(=O)=O)(C(=O)NC2CC(CNC(C3(F)CCCN(C)C3)=O)C2)CCCC1 c1(SCC)ccccc1C(=O)NCC1COCCN1C(C1COC(=O)N1C)=O CC1CC(C(=O)NC2CC(F)(CNC(=O)C(C)CSC(F)(F)F)C2)=NO1 N1(C(CNC(=O)NC)=O)CC(CNC(c2csc(Cl)c2)=O)OC(C(F)(F)F)C1 Cc1c(C(=O)NCC2CC2NC(=O)CCc2nncn2C)cnn1C1CCCC1 N1(C(c2ccn(-c3cccc(F)c3)n2)=O)CC2(CCN2C(c2n[nH]cc2F)=O)C1 CC1(C)C=C(C(=O)N2CC(C(F)(F)F)CCC2NC(=O)CN2CC3CC3C2)C1 c1(C(N2CC(CC(C)NC(CC=CC=C)=O)C2)=O)cc([N+](=O)[O-])ccc1CC#N C1(CC(=O)NCCCN(C(c2cnc(C)s2)=O)CC2CCCC2)CCCC(C)C1 CC1CCC(C(N2CC(N(C(=O)CC3OCCCO3)C)C2)=O)CC1 CC(C)C(F)C(=O)N1CC2CC1(C(=O)N(C1CCCCC1)C)C2 c1(C(CN(C2CC3CC3C2)CC)(C)C)ccc(C)o1 c1(C(=O)NC(CNC(c2n(C)ncc2[N+](=O)[O-])=O)CO)cccc2c1CCC(=O)N2 N1(C(C(CC)n2cccn2)=O)CCC(C)(NC(c2ccnnc2O)=O)CC1 c1(CNC(c2c(-c3ccc(SC)s3)nccc2)=O)nc2c(C)c(Br)ccc2s1 C1(C(C)C)CCc2sc(C(=O)N=c3ccn(CS(=O)(=O)c4cccs4)[nH]3)cc2C1 C12(CNC(c3cc(C)sn3)=O)CCCN(C(c3cc(Cl)cn3C)=O)C1C2 C1(NC(C=C2CCC(C)C2)=O)CN(C(=O)CSC(F)(F)F)C2(CCCCC2)C1 N1(C(CCc2cccc(OC)n2)=O)CCCC(C(N2CC(C)(O)C2)=O)CC1 CC1CC(C)(C(=O)NCC(C)(C)CNC(c2nnn3c2CSCC3)=O)CC(C)O1 c1(C(=O)NCC(c2ccncc2)O)cc2cccc(F)c2s1 c1(-c2nnc(SCC#C)n2CC(=C)C)cc(SC)cc(SC)c1 n1(CC(=O)NCCCCC2CCN(C(C(F)OC)=O)CC2)nc(Cl)ccc1=O c1(C(=O)NC2C(NC(C=CS(C)=O)=O)COC2)cccc2nc(O)[nH]c12 Cc1ccc(C(=O)NC2CCN(CCn3cc(C4(CCO)CC4)nn3)CC2)nn1 c1(SC)cccc(C(N2CCC(n3cnnn3)C2)=O)n1.C12CC(C1)CNC2=O C(=O)(CC(F)(F)C(F)F)NC1(C(N2C(C)C(=O)NCC2)=O)CCSC1 c1(C(N(CCCNC(=O)C=CCO)C(C)C)=O)ccc2cnsc2c1 CN1CCC(N2CC(C(=O)OCCOCCO)C2)CC1.c12cc(Br)nn1CN2 c1(NC(C(N2CC(C)C(NCc3ccccc3)C2)=O)=O)cnn2c1NCC2 C1(NC(C2N(CCC)CCCC2)=O)C2CC3C1C3C2C(=O)N(CC)CC1CCC1 CCC(C)(CO)C(=O)N1CCCC(CNC(c2cccc(N(C)C)c2)=O)CC1 N1(C(COCCCC(C)C)=O)CCCC(CC(=O)NCC2(CCO)CC2)CC1 C=CC1(C(=O)NCc2ccccc2C#N)CCN(C(c2cnn[nH]2)=O)C1 N1(C(c2nc[nH]c2C(F)(F)F)=O)CCC2CCN(C(c3cc(F)c[nH]3)=O)C2C1 N1(C(Cc2nc(C)[nH]n2)=O)CC(C2CCCN(C(C3CSCC(=O)N3)=O)C2)C1 N1(C(CCc2onc(CC)n2)=O)CCC(NC(c2ccnn2C2CC2)=O)C(C)C1 C1(NC(C2CCN(C)C2)=O)CN(C(=O)CC2(C#N)CCOCC2)CC1(C)C CCCCC(CC)N=c1[nH]c(N2CCOCC(C(N)=O)C2)nc2ncn(CC)c12 c1(CC(=O)NCCN(C2CCCCC2)CC2CC3CC3C2)cc(CC2CC2)on1 c1(OC)cc([N+](=O)[O-])ccc1C(=O)NCC1CC1CNC(c1cscc1C)=O c1(C(N2C3C(C(=O)Nc4cn(CC(C)C)nc4)C(C3)C2)=O)ccccc1C#N C=CCC(CNC(c1ccns1)=O)C(=O)NCC1CC2(CCO1)CC2 N1(C(Cc2cc(C)on2)=O)CCC2(CC1)CN(C(c1ncnc3scc(C)c13)=O)C2 c1(C(N(C2C(NC(CCOCC=C)=O)CCCC2)C)=O)cnc(C)[nH]c1=N N1(C(CC(C)=C(C)C)=O)CCC(F)(CNC(C2(C3(C)CC3)CC2)=O)CC1 N1(Cc2ccc(C)[nH]2)CCC2CC(C(=O)Nc3cc(Cl)ncn3)C2C1 C1(NC(c2c(C)c(Br)ncc2)c2nnnn2C(C)(C)C)CC2CCCC(C1)C2 C=CC1(C(=O)NCCc2csc(C)n2)CCN(C(=O)CC2(O)CCCOC2)C1 C(=O)(CCC(CC)OC)N(CC(CC)NC(C1CCC1C(C)(C)C)=O)C C(c1ccccn1)=C(C)C(=O)N(C)CC1CCCN(C(C2(C)CC=CCC2)=O)C1 c1(C(=O)NCC#CCNC(c2nncc(CCC)c2)=O)cnc2n1CCCCC2 n1(CC(=O)NCC(CO)NC(c2c(NCC)scn2)=O)nc(C)c2cccnc12 N1(C(c2cnc(COC)s2)=O)CC(NC(C2CCCO2)=O)C(F)C1 Cc1ccc(Cl)cc1N1CC(C(N2CC(CNC(=O)C(N)=O)C(O)C2)=O)CC1=O C1(C(N2CC(OCC(=O)NC)C2)=O)CCCN1C(=O)CSc1cn[nH]c1 Cc1ccc(CC(N)CC(=O)NCCNC2CCCN(C)C2)c(C)c1 C(C)(CCCCNC(=O)CCc1csnn1)NC(CCCn1ncc(C)c1)=O c1(COC)cc(C)cc(O)c1.C12CCCCC1NC(=O)C1(CC(=C)C1)C(=O)N2 C(=O)(C1=CC(O)CCC1)N1CCC(C(=O)N(CCC2CC(=O)C2)C2CC2)C1 c1(OCC(=O)N(C2CCN(C(C3CCCC34CC4)=O)CC2)CC)cncc(Cl)n1 N(C)(C1CN(C(c2ccno2)=O)CCc2ccccc21)C(C1(C(C)C)CC1)=O N1(C(C2CCN(C)C2)=O)CCN(C(C2CC3CC2C3)=O)CC1c1ccccc1Cl C#Cc1ccc(Br)c(C(=O)NCC(C2CC2)NC(C2CCC(C)O2)=O)c1 N1(CCOCCOC)CCN(C2CCN(C(=O)C=Cc3ccco3)C2)CC1 N1(C(c2c(C)[nH]c(=N)s2)=O)CCC(CCNC(=O)CCCn2ccnc2)CC1C Cc1cccc(C(N2CC(=C(F)CNC(=O)CCCF)C2)=O)c1Br N1(C(c2c(C)nc(O)cc2)=O)CCC(C2CCN(C(=O)CCCCO)C2)C1 C1(NC(CN(C(C)=O)C)=O)CCN(C(c2cnsc2)=O)C(c2ccccc2)C1 Cc1c(C=CC(N2CCN(C(=O)C(C)C(F)(F)F)C(CC3CC3)C2)=O)cnn1C S(=O)(=O)(c1ccc(C#N)cc1)NC(CC)C(=O)NCCNC(=O)C(C)SC c1(CSCC(=O)NCC(CN(C(c2c(C)cco2)=O)C)O)ccc(F)cc1 C1(CC)CN(C(=O)CN=S(C)(C)=O)CCC1NC(c1cc(C2CCC2)[nH]n1)=O N1(C(C(C)(C)C(N)=O)=O)CCCC(NC(=O)CN2CCOCC2)C(F)C1 N1(C(Cc2cn(C(C)C)nc2)=O)CC(NC(c2ccnc(C(C)C)n2)=O)C2CC12 C(=O)(CC(O)C1CC1)N(CCCNC(=O)C=CCN1CCC1)C C#CCC(C(=O)N(C)CC1CCN(C)C1)NC(C12CC(CO)(C1)C2)=O c1(C(=O)NCC2(C(N3CCN(C)C(CC)C3)=O)CC(=C)C2)cc(N)cnc1Cl CC(C)(C#N)CCC(=O)N1CCCC(n2cc(-c3ccsc3)nn2)C1 C(=O)(C(F)(F)CCn1ccnn1)NCCN(C(C1CC(C)=NO1)=O)CC c1(CC(C)C)cc(C(=O)NC2(CO)CN(C(=O)CN3CCOCC3)C2)n[nH]1 C1(CNC(=O)CCC2CCCCC2)CCN(C(c2ccc(F)nc2)=O)CC1 C(CN=c1nc2scnc2c(N2CCC(C(N)=O)C2)[nH]1)C1(C)CC1(Cl)Cl N1(C(CC2C(C)CC2)=O)CCC2(CC2NC(C2CC23CC3)=O)C1 C(CCN=c1nc(N(C)Cc2ccncc2Cl)cc[nH]1)NC(N(C)C)=O C1(C(=O)NCCC(C)NC(=O)COc2cccnc2)CCOCC12CCCC2 N1(C(=O)C=CC(F)(F)F)CC2CC(NC(C3CCOC3C(F)(F)F)=O)C1C2 C12(C(=O)NCC3N(C(C(C#C)(C)C)=O)CC4(CC4)C3)CC3CC(C1)CC(O)(C3)C2 c1(C(N2CC(NC(CC3CC(=C)C3)=O)C(OC)C2)=O)ccc(C2CC2)cc1Cl c1(C(N(C2CCCC2NC(=O)CCOC2CC2)C)=O)ccc(O)cc1Cl CC(C)C(F)(F)CC(=O)N1CCC(CNC(=O)C(c2ccc(Cl)s2)C)C1 C1(C)(C(=O)NC(C)CN(C)C(c2cnn(CC(F)(F)F)c2)=O)CC(C#N)C1 C(CC(=O)N(CC(CO)(CO)NC(c1cccnc1)=O)C)(C(F)(F)F)OC N1(C(c2cccc(OCC)c2)=O)CCC(F)(CNC(=O)C(F)CCN(C)C)CC1 CC1CCS(=O)(=O)CCN1C(=O)CCc1nc2ccc(Br)cc2o1 N1(C(=O)NC2CCN(C(c3ccc(Br)cc3)=O)CC2)CC2CCC(O)C2C1 c1(NC(c2ccc(F)c(-c3cccc(F)c3O)n2)=O)cc(Br)nc(Br)c1 CN1CCC(C(=O)NCC23CC(CN2C(c2c[nH]ccc2=N)=O)C3)C1=O C12(NC(C3C(C)CC3)=O)CCC(CN(C(=O)Cc3cnco3)C1)C2 C12(C(=O)OCC)CCC1CN(C(c1nc(C)co1)C(=O)NCCCC1CC1)C2 N1(C(c2c(C)c(C3CC3)on2)=O)CCN(C(C2CCNC(=O)C2)=O)C(C)C1 c1(C(=O)NCC(N(C(CC(=C)C)=O)C)C2CC2)cnc(O)cc1O CC1CCCC(N(C(c2cnnn2C)C(=O)NCc2cccc(Cl)c2)C)C1C c1(CC(=O)NCC2CCC(NC(C3CC4(CCC4O)C3)=O)C2)csc2ccccc12 c1(OC)ccc(Cl)c(C(N2CCCC(CCNC(C3CCSC3)=O)CC2)=O)n1 N1(C(CCCC(=O)NC(C)C)=O)CCN(C(C2C(C)OC(C)C2C)=O)C2CCC12 n1(C(C)C)ncc2c(NCCSCC(F)(F)F)[nH]c(=NCC3(CO)CC3)nc12 N1(C(C2(F)CCN(C(C(C(CC)C)O)=O)CC2)=O)CC(C)CCCC1C N1(C(C(C)C2CCCC2)=O)CC2CC1(CNC(=O)CC(C)c1cccnc1)C2 CCCCS(=O)(=O)NC(C)C(=O)N1CC(CC(C)NC(=O)CC2CC2)C1.C(=O)(C(C)C)N N1(C(C(CCC=C)NC(c2cc(Cl)cs2)=O)=O)CC(C)OC2(CCC2)C1 C1(NC(C2C(C(=O)OC)C2)=O)CC2CC(C1)N(C(c1cnn(CCF)c1)=O)C2 c1(CC(=O)NC(C=CC(=O)NC(C2CSC2)C)(C)C)ccnn1C N1(C(c2n(C)cnc2)=O)CCc2c(C(=O)Nc3cncs3)csc2C1 C1(C(=O)NC(C)Cc2nn[nH]n2)CC2(CCN1C(=O)C1=CCOCC1)CC2 N1(C(C(C(C)(C)C)OC)=O)CC2CCN(C(c3nnc(Cl)cc3N)=O)CC2C1 C=CCC(C)(CC)C(=O)NCC1(NC(=O)Cn2ccc(=O)n(C)c2=O)CCOC1 CCC(C)C(C(=O)NCC1(C)CCN(C(c2cncs2)=O)CC1)OC C1(C(N(CC(=C)C)CC#C)=O)C=CC(NC(=O)CCc2cnccn2)C1 c1(OC)cc(F)c(O)cc1Cl.C1(OCC)CC2N(C1)Cc1ncc(cn1)C(=O)N2 Cc1cnc(C(=O)NCC2CCC(NC(c3ccc(NS(N)(=O)=O)nc3)=O)C2)nc1 C12(NC(C3C4CN(C(C=CC(C)(C)C)=O)CC43)=O)CC3CC1(CO)CC3C2 c1(CCC(=O)NCC(CC(C)C)NC(C2(C)CCC(=O)N2)=O)ccc(F)c(Cl)c1 C12CC3(CO1)CN(C3)C2=O.c1(NC(CN2C(C)CCC2)=O)cc(O)ncc1F c1(N2CCC(CNC(C3CCCC(F)C3)=O)C23CC3)nc2ccc(F)cc2s1 C1(C(=O)NC(C)CNC(=O)Cc2cnsc2)CCC2CCC12 N1(C(c2ccn(C(C)(C)C)n2)=O)CCCC(CCNC(c2nn[nH]c2Cl)=O)C1 C12(C(=O)NC3(C)C(NC(Cn4c(C)nnn4)=O)CCC3)CCCN(CC1)C2 c1(OC)ccc(OC(F)(F)F)c(C(=O)NCC2CN(C(=O)C(C)(F)F)CC2C)c1 CCCC(C(=O)N1CCCC1C(C)(C)C(=O)NCc1cncc(F)c1)NC(N)=O c1(C(N2CC(NC(C(CC#C)C)=O)C(SC)C2)=O)cn2ncnc2nc1C c1(OC)ccc(CC(N2CC3CC3(NC(c3cncs3)=O)C2)=O)nc1 N1(C(C2CC(C)(CC)C2)=O)CCCC12CCCN(C(c1c(C)nc3sccn13)=O)C2 c1(C(=O)NC2CC3CN(C(c4cn(C)c(C#N)c4)=O)C2C3)n[nH]c2c1COCC2 C(=O)(C(C)(C)C(F)(F)F)NC(c1ccc(NC(CC(C)C(F)F)=O)cc1)C1CC1 N1(C(=O)CC2(O)CCOCC2)CCC2CCN(C(c3ccoc3)=O)CC2C1 C12CCN(CC1)C2=O.CC1CC1(F)C(N1CC(NC(=O)OC(C)(C)C)C1)=O N1(C(C(CC)C)=O)CCCC(F)(C(=O)NCc2cccc(C)c2O)C1 C1(C(N2CCC(CNC(C(C)(C)N3CCOCC3)=O)CC2)=O)C2CCC(F)(F)C12 N1(C(CN(C(C)=O)C)=O)CCC2(CC2NC(c2cnn(CCO)c2C)=O)C1 c1(OC)cnc(Cl)c(NC(=O)CC2(NC(c3cccc(C)n3)=O)CCC2)c1 N1(C(Cc2nc(CC)sc2)=O)CCC(CO)C(NC(C23CCCC(C2)OC3)=O)C1 c1(C(=O)NCCCC2N(C(c3nc(C)sc3C)=O)CCC2)cn2c(n1)CCC2 c1(CC)occc1C(=O)N(CC(C)O)CCNC(C1(O)CCSC1)=O N1(C(C(CCC)N(C)C)=O)CCN(C(c2c(OC)cccc2O)=O)CC1CC(F)F C1(C(=O)NCC2(NC(CCCC(C)=O)=O)CCC2)CCC(C2CCCO2)O1 c1(CCC(=O)NC2CC(F)(CNC(C3(CO)CCCO3)=O)C2)ccc(F)cc1 C1(CC)C(C(=O)NC(COC(C)C)C(=O)Nc2cccnc2)CCN1C C=CCCCCCC(=O)N1CCC(C(C)(C)C)(CNC(C2(C(=O)NC)CC2)=O)C1 C1(NC(C(C)=C(CC)C)=O)CCN(C(=O)C(C#N)C(C)(C)C)C12CCCC2 N1(C(C2=CCCC2C)=O)C2CCC1CN(C(c1ccc3c(c1)CN(C)C3)=O)CC2 c1(OC)cc(C(=O)NCC(C2CCOC2)NC(=O)CC(C)(C)C)cc(Cl)c1 S(=O)(=O)(CCN=C(NCC(F)F)N1CCCC1)N1CCC(N(OC)C)C1 C1(NC(c2scc(C)c2C)=O)CN(C(=O)Cn2nccc2C)Cc2ccnn2C1 N1(C(c2c(C)snc2)=O)CC2CCCC2(Nc2nc(C(F)F)nc(=N)[nH]2)C1 N1(C(CCN(C)CC)=O)CCC2(CC2C(N2C(C)CCC2(C)C)=O)C1 c1(C(C)=O)sc2ccccc2c1CS(C)=O.N12CCCC(C1)C2=O.C(=O)C(O)CF CC(CC(F)(F)F)C(=O)NCC1(CNC(c2ccc(CN(C)C)o2)=O)CCC1 Cc1cc(C(=O)NCC2CCCN(C(=O)C(F)CC)C2)ccc1[N+](=O)[O-] N1(C(C2N(C(=O)NC)CCC2)=O)CCCC(CO)(NC(=O)C(C)=CC2CC2)C1 N1(C(COCCC=C)=O)CCC2(CC1)CN(C(C1NC(=O)OC1C)=O)CCO2 C1(NC(CCN(C(=O)C#CC2CCOC2)CC=C)=O)CCCCC(C)(C)C1 N1(C(C(c2ccccc2)N(C)C)=O)CC(NC(C2(C3CC3)CCC2)=O)C(C)(C)C1 C1(CCOC)CCCN(C(=O)C(CN(C)C)NC(c2ccnc(C)c2)=O)C1 CCC(C)CC(=O)NC1(C)CN(C(=O)C(C)Cc2ccnn2C)C1 C1(C(N(CCC(C)NC(c2cccc(NC(C)=O)n2)=O)C)=O)COC2(CCC2)C1 c1(C(=O)NC2(CC=C)CCCC2)ccc(F)c(F)c1[N+](=O)[O-] N1(C(C2C(C=C)C2)=O)CCC(C)(C)C(NC(C2CCC2c2nc(S)n[nH]2)=O)C1 CC1(C)CC(C(N2CCC(CF)(NC(=O)Cn3nnc(C4CC4)n3)C2)=O)CO1 C1(c2c(NS(CC=C)(=O)=O)c[nH]n2)CCN(C(=O)CSc2ccc(Cl)cc2)CC1 C=CCC(F)(F)CCc1cn(C(C)(C)CC(=O)N2CC(SC(F)(F)F)C2)nn1 N1(C(c2c(C)[nH]cc2)=O)CC2CC1CN(C(C1CCCOC1C)=O)C2 C(CC(F)F)(C(=O)NC1CC2C=CC1C2)NC(c1n(CCC)ncc1)=O N1(C(CCOCC)=O)CC(CNC(=O)CC2CCN(C)C2)C(C(F)(F)F)C1 N1(C(=O)SC(CNC(c2ccc(COC)o2)=O)C2(C)CC2)CC(C2CC2)(OC)C1 C1(CNC(COC)=O)(NC(=O)CC2C=CS(=O)(=O)C2)CCCCC1C C1(C(N(CCCOC)C(C)C)=O)CCOC(C)C1.c12ccoc1C(=O)NC2 C1(C)(CNC(c2c(C)c(C3CC3)on2)=O)CCCN(C(=O)Cn2cnc(=N)[nH]2)C1 Cc1ncc(C(=O)NC(CO)C(C)NC(=O)C#CC(C)C)n1C Cc1ccc(OCC(=O)NCC(F)CNC(c2ccc(=N)[nH]n2)=O)cc1 C(=O)(CC(O)CC(C)C)NCC(CO)NC(CCCCCOC)=O C1(OC)CC(CNC(=O)C(c2cccc(F)c2)(C)C)N(C(=O)CCC2CC2C)C1 O=S(=O)(c1ccc2ccccc2n1)N(C1CC1)CC1=C(F)CCOCCC(O)=C1O c1(CC(N2C(C)CCC(NC(=O)C(F)C(C)(C)O)C2)=O)n[nH]c2ccccc12 N1(C(C2C(C=C)C2)=O)CCCCC1C1CCN(C(=O)C=CC(C)(C)C)CC1 N=c1[nH]c2ccccc2cc1C(=O)NCC1CCN1C(c1csnn1)=O Cc1cc(CC(=O)N(C(CNC(C2CC2C(C)C)=O)C2CC2)C)cc(F)c1 c1(C(=O)NCC2CCCC(NC(CC3ON=C(C)C3)=O)C2)c(N)ccc(F)c1F Cc1cnc2cccc(C(N3CCC(CN(C(=O)CP(C)(C)=O)C)C3)=O)n12 N1(CC(C)CC2CCCC2)CCCN(c2ccc(F)cc2)CC1 C1(COC)(CNC(=O)C(C)OC)CCCN1C(=O)COc1cccnc1 c1(C(C(=O)NC(C)(C)CC)NC(C(CC)SC)=O)cc(Cl)cc(OC)c1OC c1(C(=O)NCC(CNC(=O)CC2(c3cc[nH]n3)CCC2)OC)csc(C)n1 CC1CCN(C(C2C(NC(=O)CSC(C)(C)C)C2(C)C)=O)CCO1 C1(C(C)NC(C2(CCNC(C)=O)CC2)=O)CCCC1 NC1CN(C(=O)C(c2ccc(F)cc2F)CF)C2(CCOC2)C1 Cc1cc(C(=O)NC(C)(CO)C(=O)N)cc(O)c1.C1(CC=CC)CCCC1 c1(C(=O)NCc2cnc(O)nc2O)cc(Cl)cc2cn[nH]c12 c1(CC(=O)NCCNC(C(C)(C)C2(O)CCOC2)=O)c[nH]c2cnccc12 N1(C(c2cccc(C)c2Br)C(=O)NCC=C)CCC(CO)C(O)CC1 C(C)(C(C)C(=O)NCCc1ccc(F)nc1)NC(c1cc(CCC)[nH]n1)=O O=C1CCC2(CCCN(C(=O)OCc3ccc(S(N)(=O)=O)o3)C2)N1 C#CCC(C(=O)NCc1cc(C)n(C)n1)NC(c1cnn[nH]1)=O CC(c1ccccc1)=CC(=O)N(CC(C)(C)NC(c1nccn1C(C)C)=O)C CC(C)CCC(O)C(=O)N1CC(F)CC1CN(C)C(C1CCC2(CCC2)O1)=O c1(C(=O)NC2CN(C(C(CC)(C)C)=O)CC2O)cnc2ccc(C)cc2c1 C1(CNC(c2ccc(CC=C)cc2)=O)C(C)CCCN1C(C1CC(=C(F)F)C1)=O C1(CNC(c2cc(Cl)cc(Cl)c2)=O)CC2(CCC2)CN1C(=O)Cc1ccncc1 C1(C(C(=O)NCC2CCCN(C(CC(=O)OCC)=O)C2)O)CCCCCCC1 c1(C(=O)NCC(C)(C)NC(C2CCCCC2F)=O)cccc(F)c1N CC1CN(C(c2csc(-c3ncc[nH]3)n2)=O)CCCN1C(C1CCNC(=O)C1)=O C=C(Br)CCC(=O)NCC1CC(NC(C2(C)CCNC2=O)=O)C1 CCC(CC)C(C)C(=O)NCCN(C1CCCCC1)C(c1sc(OC)nc1Cl)=O Cc1cc(C(N2CC(O)(C(F)C(=O)NCC3CCCNC3=O)C2)=O)c(C)s1 C1(CC=C)CN(C(c2ccc(Cl)o2)C(=O)NC)CC1N1CCOCC1 C1(C2(O)CN(C(C3CC3(C)C)=O)C2)(CNC(C23CC(C)(OCC2)C3)=O)CC1 N1(C(C=C(C)C(C)(C)C)=O)CCC(NC(C2(Cl)CC2(F)F)=O)CC(O)C1 Cc1onc(C(N2CC(CNC(c3cnnc(O)c3)=O)C2)=O)c1[N+](=O)[O-] CCCC(C(=O)NCCC1CCC(NC(c2cn(C)nc2Br)=O)C1)OC c1(OC)nccc(C(N2CC(F)CC2C(N(C)C2CC2)=O)=O)n1 C1(NC(C2(CCOCC)CCC2)=O)CC(F)CN1C(=O)CCOCC N1(C(c2c(C)ocn2)=O)CCC2CC2(NC(=O)Cc2cnns2)CC1 c1(N2CCCC(CC)C2)cc(N2CCC(N(S(C)(=O)=O)C)CC2)nc(C)n1 N1(C(c2ccccc2Nc2cnc(C)s2)=O)CC2CC1CN(S(C)(=O)=O)C2 c1(CN(C(=O)CCNC(=O)CC2(C)CCC2)C)ncnn1C C1(NC(c2ccc(C)c(Cl)c2Cl)=O)CN(C(c2ccccn2)=O)CCC12CCC2 CC1CCC(O)C(NC(C2(NC(c3cc(CO)ccn3)=O)CCSC2)=O)C1 C1(C2C(c3n(C)ncc3)C2)C2CCN(C(=O)C(N)=O)C12 c1(C(=O)NCC2C(C(=O)NC(c3ccccc3O)C)CCC2)ccc(O)nn1 CC(CC(N)=O)C(=O)N1CCC(CC(C)NC(c2csc(Cl)n2)=O)CC1 N1(C(C2CCC(SCC)CC2)=O)CCN(C(c2ccccc2SC)=O)CCC1C N1(C(C(=O)NCC(C)NC(C=C(C)Cc2ccc(C)s2)=O)C)CCP(C)(=O)CC1 c1(C(N2C3CC(CC(NC(c4ccoc4)=O)C3)C2)=O)cc2nn[nH]c2cc1F C1(C(N2CCC(CNC(CCC)=O)(COC)CC2)=O)CCC2CCC(=O)N12 c1(C(CNC(C2(CCCC)CCCC2)=O)NC(c2cocn2)=O)ccc(F)cc1 Cc1[nH]c(C#N)cc1C(=O)NCC1CCCC1C(=O)N(C)CC1(O)CCCCC1 c1(C(=O)NC2CCC(CNC(C3CCN(C)CC3)=O)C2)nnn2c1C(=O)NCC2 C1(C(=O)NC2CC(C(NOCCC)=O)C2)CC12CCCC2 c1(-c2c(C)cc(Cl)cn2)ccc2c(c1)CN(C(C1CC(O)C1)=O)CC2 Cc1oc(C#N)cc1C(N1CC(NC(C2CCCN2C=O)=O)C(C)(C)C1)=O N1(C(C(C)CC2CCC2)=O)CCCC(N(C(=O)CCN(C)C)C)CC1 c1(C(N(CC(C)NC(C2C=CCCC2)=O)CC)=O)ccc(Cl)c2occc12 N1(C(C2(C)CCN(C(COCCCC(C)C)=O)C2)=O)CCC2(CCSC2)C1 C1(C(N(C)CC2N(C(COCCC)=O)CCC2)=O)Cc2c(F)cc(F)cc2O1 CN1CCOCC1C(=O)NCC1CCCN1C(C1CC2C=CC1C2)=O c12cc(ccc1Cl)NC(=O)N2.c1(OC)cccc(CS(C)(=O)=O)c1.C12CC1OC2 C1(C)(OC)CCCN(C(=O)CC2COCCN2C(=O)C(=O)N(C)C)CC1 N1(C(C(C(C)C)NC=O)=O)CC(C)(C)C(NC(C2COCC2(C)C)=O)C(C)(C)C1 N1(CCC)CC(C(=O)NCC2C3CC2N(C(C2CCCCC2C)=O)C3)CC1=O C(c1ccn(C)c1)=CC(=O)NC(CC=CC(=O)NC(C(C)SC)C)(C)C n1(CC)nnnc1C(C(C1CC(C)=NO1)OC)NCCCSCCO C1(NC(c2n(C=C)ncc2)=O)(CNC(=O)C=CC(C)(C)SC)CCCCC1C C1(NC(C(C)Oc2cccnc2)=O)CN(C(=O)CNC=O)C2CC12 C#CCCCCC(=O)NCCCN(CCc1cccs1)C1CC1 N1(C(CN(C(C2CCC=CCCC2)=O)CC)=O)CC2(CC(CO)CO2)C1 N1(C(C2C(C=C)C2)=O)CC2CC2C1CNC(c1ccc(-c2ccco2)o1)=O N1(c2c(CC)cccc2)C(=S)NC(c2nc(Br)ccc2Cl)C2=C1C(C)(C)NC2=O c1(C(=O)NC2CN(Cc3ccc(OC)cc3O)CC2O)c(F)cc(Br)c(F)c1F c1(C(N2CCC(CNC(=O)CC3CCC3)C(O)C2)=O)cccc(F)c1F c1(C(N(C)C(=O)NCC)C)cccc2nsnc12 C(c1ccccc1Cl)=CC(N1CC(NC(c2c(-c3n(C)ncc3)n[nH]c2)=O)C1)=O c1(C(N2C(CNC(C(F)OC)=O)COC(C)(C)C2)=O)cccc2cnccc12 N1(C(COCCC=C)=O)CC(CNC(=O)CCC2CC2)CC12CCC2 C(=O)(C#CC(C)(C)C)N(CCNC(C(c1c(C)nn(C)c1)O)=O)CCOCCO CCC(CCCC(=O)NCC1(CC)CC1)NC(C1(O)CCSC1)=O C1CCON1C=O.C(=O)(C(O)CC(N)=O)N(C1(C(=O)OC(C)(C)C)CC1)C c1(C(=O)NC2CC3CN(C(=O)CC4(CO)CC4)CC3C2)ccc2cccnc2n1 C1(OC2(C)CN(C(C(C)c3cncs3)=O)C2)CCN(C(=O)C(C)(C)CF)CC1 c1(C(=O)NCC2CCC(NC(C3CC=CCC3)=O)C2)c(F)cc(F)cc1Cl N1(Cc2ccc(C)s2)CCC(C2CCCN(C(c3ccc(F)cc3F)=O)C2)CC1 c1(CC(=O)N(CCNC(C(C)OCCC=C)=O)CCOC)cc(Cl)cc(Cl)c1 c1(C(=O)NCC(N2CC(C(CC)C)C2)=O)cccc(CO)n1 c1(C(=O)OCC)cnc(C(N2CCC(N3CCOCC3C)CC2)=O)nc1 C(CCCN=c1[nH]nc(C(F)F)s1)C1CCC(CNC(C2(COC)CC2)=O)C1 c1(C(N2CCC(NC(COCC)=O)C(CC)C2)=O)ccc2nc(Cl)nn2c1 CP(C)(=O)c1ccc(C(=O)NC2CCN(C(=O)CN3CCCC3CO)C2)nc1 C#Cc1cnn(C(N2CCCCC2CC(=O)NC(C2(O)CC2)C)=O)c1 C12(CC(N3CCC(CN(C)C(c4cc(C(F)F)ccn4)=O)C3)=O)COC(C)(C1)C2 C(=O)(C1CCCc2c(O)cccc21)NCCCOCCNC(C(CSC)N(C)C)=O CC(CN=C(NCc1cccnc1)NC1CC12CC2)SCC(F)(F)F C1(CNC(C2CC=CCC2)=O)CCCN(C(C2(c3cccc(Cl)c3)CCC2)=O)C1 C#CCCCCCCCCC(=O)NCC1CN(C(=O)C(C)CCOC)CC1(C)C C1(CNC(CCN(C)CC)=O)CC(F)CN1C(C1CC1c1nccn1C)=O N1C(=NCCC2(C)OCCO2)N2CCC(C)(C2)C1.C(C=C(C)C)OC c1(CC(N2C(C)CN(C(c3coc(Cl)n3)=O)CCC2)=O)c[nH]c2ccc(F)cc12 C1(NCCOC(c2nccc(CC)c2)=O)CC2CC(OC)CC12 C(CC(=O)NCC(C)(C)OCC)(C(F)F)NC(C(CC=C)C)=O CC(=O)CCCC(=O)N1CC(O)CC1C(=O)N(C)C.C12CCCC1C(=O)N2 c1(C(=O)NCC(CNC(CCCCCC)=O)O)cc(Cl)c(Cl)[nH]c1=N c1(-c2c(OCC)ncc(F)c2)cc2c(s1)CCN(Cc1c(F)cc(Cl)cc1C)C2 Cc1cc(F)c(S(=O)(=O)NC2(CO)CC3CCC2CC3)c(C)c1Br C(CNC(c1c[nH]nc1-c1cccnc1)=O)(C(C)C)NC(C1C(CC(C)C)C1)=O C1(CC)C(NC(c2occc2CC)=O)CCN1C(=O)CN1CCC(C)(O)C1 N1(c2n(Cc3cc(C)on3)c(C3CCC(=O)N3)nn2)CCCC2COCCC12 N1(C(C2(CCNC(CCc3ccn(C)n3)=O)CC2)=O)CC[Si](C)(C)CC1 N1(CCO)CCOC(NCCS(=O)(=O)CC2CCOCC2)C1 C(CCCC(=O)NCC(C)CCCO)N(C(C=CCOC)=O)C n1(CCC(=O)NCCN(C(=O)C(c2cccs2)NC(N)=O)C)ccc(O)nc1=O C1(NC(c2c(C)nns2)=O)CCCCN(C(=O)CCCC2CCOCC2)C1 Cc1c(C(N2CC(C(O)C(=O)NCC3C4CCCC34)C2)=O)ncn1C N1(C(C(COC)NC(C)=O)=O)CC2CCN(C(=O)C=Cc3ncc(C)[nH]3)CC2C1 C(=O)(CC1=CCCCC1)NCC1(NC(c2c(CC)nc(C)n2C)=O)CCOCC1 C=Cn1nccc1NC(N1CCC(OCC(=O)NOCC(=O)OCC)C1)=O C(=O)(CC(O)CC(C)(C)C)N1CC(OCC(=O)NCCC(C)(C)SC)C1 c1(OC)cc(CCC(=O)NC2C=CCN(C(C34CC(OC)C3C4)=O)C2)ccc1F C1(C(=O)NC(C)C(=O)NC2CCCC2)CC(C)N(C(=O)CCOCCCO)C1 Cc1cc(Br)c(F)cc1NC(C1CCCC1CNC(=O)CN1CCS(=O)CC1)=O C12(C(=O)NCC3(O)CCC(C)CC3)COCC1CN(C(=O)CC1(O)CCC1)C2 C1(OC(C)C)CCN(C(c2ccsc2CNC(=O)CC2C(C)(C)C2(C)C)=O)CC1 c1(-n2c(-c3sccc3C)nc(C(C3CC3)OC)n2)ccc(F)c(C)c1 C1(C(N(C)CC2C3CN(C(Cc4c(C)cc(C)s4)=O)CC32)=O)CCCC2(CC2)C1 C12(C(N(CCCNC(c3c(C(=O)OC)ccnc3)=O)C)=O)CC3CC1C2C3O Cc1cccc(CNc2cnccc2OC)c1I C1(NC(CCC2CCC(C)O2)=O)C2CCN(C(c3cnc(N)c(Cl)c3)=O)CC12 N1(C(C(C(C)O)(F)F)=O)CCCC2(CCN(C(C3CCCCC3C(N)=O)=O)C2)C1 N1(C(C2CC3CC3C2)=O)CCN(C(C2CCCC(C(F)(F)F)C2)=O)C(CCO)C1 c1(NC(COC)C(C)C)ncc(C)cc1S(=O)(=O)NCCN(CC(F)(F)F)C C1(CNC(C(CCCC)O)=O)CC2CCC1N(C(=O)COc1ccc(Cl)nc1)C2 N1(C(C=NOC)=O)CCC2C(C1)CN2C(=O)Cc1noc(C)c1C#N C1(C)(NC(C2CC(C)(NC(C)=O)C2)=O)CCN(C(=O)C(n2cc(C)cn2)C)CC1 C1(NC(CCC(=C)Cl)=O)CCN(C(=O)CC2CCN(OC)CC2)C(C)C1 C(C(COC)CC(=O)NC1C=CCN(C(=O)CC2CCS(=O)(=O)C2)C1)OC CCCC(CC)C(C(=O)NC1CC1)N(C)Cc1ccccc1N(C)C Cn1cncc1C(=O)NC1(C(N2CCC(OC3CCCC3)C2)=O)CCCC1 c1(N2C(CCCNC(CCNS(C)(=O)=O)=O)CCC2)ncc2c(n1)CCCCC2 c1(CCOC)n[nH]c(=NCC(c2ccccc2F)NC(=O)C=C(C)C(F)F)s1 C1(NC(=O)C(F)(F)C(O)C2CC2)CC2CC(C1)N(C(c1cncc(Cl)c1Cl)=O)C2 C1(C(N2C(C(N(CCCCC)C)=O)C=CC2)=O)CCCC(=O)N1 C1(CC)CCC(C(N2CCC(N(C(C3SCCCS3)=O)CC)C2)=O)C1 C1(CN(C(=O)CCCCCF)C)CN(C(c2cnn(C)n2)=O)CC12CC2 C1(CCNC(C(c2cc(C)sc2)(F)F)=O)CCCN(C(C2CNC(=O)N2C)=O)C1 c1(NC(C)C(=O)N(C)C)cccc(CNC(=O)C(C)OC2CCOCC2)c1 C(=O)(C1=C2CCN=C2NC=C1)NC1CC(OCCNC(C2OCCC(C)C2)=O)C1 N1(C(CCCOC)=O)CCN(C(=O)C=Cc2nccs2)C(CS(C)(=O)=O)C1 C(=O)(C(C)CS(C)(=O)=O)NCc1c(C)nn(C2CCC2)c1 c1(N(C)C)cc(C2(C(F)(F)F)CCC2)n(C)n1.c12ccnc(n1)NC1CC(C1)N2 CCCCCCCC(=O)NCC(C(=O)N1CC2(CCN2C)C1)C(C)C C1(CC(N2CCCC(CC3CC3)C2)=O)C2CCCC2N1C(C1CCCCC1F)=O N1(Cc2cc(OC)c(OC)cc2)CC2CCN(C(=O)C(C3CC3)SC)C2C1 Cc1c(C(=O)NC(C)CC(C)NC(=O)CC(=O)N(C)C)sc2[nH]cnc(=O)c12 C1(C(N2CCC(N(C(c3cccc(SC)c3)=O)CC)C2)=O)CC2(C1)CC21CCC1 C1(C#N)(C(N2C(CNC(CC(C)(C)C)=O)CCC2)=O)CC12CCCC2 C1(NC(C2CCCCO2)=O)CCOC2(CCN(C(C3(CO)CCOC3)=O)CC2)C1 CC(CS(C)=O)C(=O)NCC12CC(CNC(c3cnc4n3CCC4)=O)(CO1)C2 c1(C(=O)NCC(C(C)C)NC(c2c(OC)cc(O)nc2)=O)cnc2[nH]cncc1-2 Cc1cccc(C(C)C(=O)NC2CCCN(C(=O)COc3cncc(C)n3)C2)c1 c1(CC(COC(=O)NC2(C)CCCO2)CCC#N)cc2c(cn1)OCCCO2 c1(OCC(N2CC3C(NC(c4cc(F)cc(F)c4)=O)C3C2)=O)ccc(F)cc1O C1(C)(CNC(c2c(SC)cccn2)=O)CC(F)(F)CN1c1nc(Cl)c(C#N)s1 Cc1[nH]c(Cl)nc(=NCC2(C)CCCN(C(C3(C#N)CC3)=O)C2)c1C#N Cc1cc(C(=O)NCC(C)(O)CNC(c2cn(C(F)F)cn2)=O)cc(=O)n1C C1(C(=O)NC(CC)CN2CCCC2)CC=CCC1NC(C1CCC1)=O N1(C(c2c(OC)ccc(Cl)c2)=O)CCC2CN(C(=O)C(N)CN)CC2CC1 N1(C(C(C)OC)=O)CCC(O)(C(C)NC(c2ccc(C3CC3)cn2)=O)C1 c1(C(=O)NC(CCC(=C)C)C)cc2cc(C)ccc2o1 c1(CC(N2C(C)C(NC(=O)CN3CCC3C)CC2)=O)ccc2c(c1)OCCO2 C1(C(N(CC(C)CO)C)=O)CCN(C(=O)CCc2nncs2)C1(C)C C#Cc1ccccc1CC(=O)NC(C)CNC(c1sc(Br)nc1C)=O c1(OCC(=O)NCC2N(C(c3c(C)noc3N)=O)CCC2)ccc(F)c(Cl)c1 C1(C(=O)NCC(CC)(C)NC(=O)CCCc2cccs2)CC(C(C)C)=NO1 C(N=c1ccc(C(F)(F)F)n[nH]1)C1CCCCN(C(Cc2nc(C)sc2)=O)C1 C1(CNC(C(C)(C)OC)=O)CN(C(C2CN3CCCN2CC3)=O)CC2(CCC2)O1 C(C(=O)N(CC(C)(C)C)OC)C1CC(OCC)OCC1 C1(C(=O)NC(c2cnccn2)C)CCN(C(=O)Cc2ccc[nH]2)CCO1 Cc1cc(C(=O)NCC2CC(CNC(c3csc(Cl)n3)=O)CO2)c(N)cc1F C1(NC(CCCCCC)=O)CCCC12CN(c1cc(Cl)nc(C)n1)C2 CCCC(CC)C(=O)NCC1COCCN(C(C2(N(C)C)CCCC2)=O)C1 c1(C(=O)OC)cnc(C(=O)NC(C)CCNC(=O)CC2CC23CC3)c(N)c1 CN1CCN(C(=O)C(F)(F)C2CC2)CC1CNC(C1(C2CC2)CC1)=O N1(C(c2n(C)ccn2)=O)CC(NC(c2cncc(-n3cccc3)c2)=O)CC1(C)C C(=O)(CC(C)CC(C)C)NC(CC(=O)N1C(COC)CCC1)C(C)OC C(=O)(C1OC(=O)c2ccccc21)N1CCC(C)(NC(c2ccccc2Br)=O)C1 N1(S(=O)(=O)c2cccnc2Cl)CC2(C1)CN(c1ncc(C3CC3)cn1)CCO2 C1(CNC(C=CCCC)=O)C2CN(C(c3ccn(C(C)C)c3C)=O)CC12 N1(CC(=O)NC(CN(C(c2cnc(CC(C)(C)C)s2)=O)CC)C)CC(=O)NC1=O CC1(C)c2ccccc2CC1C(=O)Nc1cccc(S(C)(=O)=O)c1 C(=O)(C(O)C(C)(C)CC)N1CC(NC(CSc2ccc(OCC)nc2)=O)C(C)C1 Cc1cc(C)n(CC(=O)NC(CN(C)C)C(N2CCC(CC(N)=O)CC2)=O)n1 S(=O)(=O)(c1ccccc1)NC(=O)CCN(CCCNC(C1CC1Cl)=O)C(=O)C1CC1 C1(CC(=O)NCC2(CC)CCC2)CCCN(C(c2ccc(N)cn2)=O)C1 c1(C(=O)NCC(c2ccc(F)cc2)NC(C)=O)ccc2ccnc(O)c2n1 c1(C(=O)NCC(CO)NC(CCOCCN(C)C)=O)sccc1C#N N1(C(c2c(C)cc(F)s2)=O)CCC(C)(C)CC1C(=O)NCc1nc(C)c(C)s1 n1(CC(=O)NC2CCC(F)(CNC(C3CC3F)=O)C2)ccc(Br)cc1=O C1(C(=O)NCCNC(C(C)CC)=O)(NC(C(C)=C(CC)C)=O)CC1(C)C.CCC CC1(C)CN(C(c2ccccc2F)=O)CCC1NC(=O)C=Cc1cccnc1 C1(CC)CN(C(=O)C=Cc2nc(C)c(C)[nH]2)CCC1Nc1ncnc(Cl)c1F N1(C(CCc2ccc(C)s2)=O)CCCC(NC(c2cc(C(C)(F)F)n[nH]2)=O)C1C C=CC(C)CCNC(c1sccc1F)c1nnnn1CCSC C12(NC(CCNC(C3CCCS3)=O)=O)CC(CNC(CN(C)C)=O)(C1)C2 c1(C(=O)NC2(COCC)CCOC2)ccccc1CC(=O)NCC1CC2(CC2)C1 c1(OC)cccc2c(C(=O)NC3CCCCC3NC(C3(C)COCCO3)=O)cnn12 C1(CC(=O)NCC2(CC)CC2)CCCN(C(=O)C(F)C2CCCC2)C1 N1(C(CCC(=O)OCC)=O)CC2CCCC(NC(=O)CCC(N)=O)C2C1 N1(C(C2(C#C)CN(C(=O)C(C3CCC3)OCC)C2)=O)CCC(C)CC1C N1(C(c2c(NC)ccc(C)c2)=O)CCOCC12CCN(C(=O)OC(C)(C)C)C2 NS(=O)(=O)c1ccsc1C(=O)NCCC1CCCCN1C(=O)C(O)C(F)(F)F C(CN=c1[nH]c2ccc(F)cc2o1)N(C(=O)C(N1CCCC(C)C1)=O)CC.CO N(C1c2ccccc2CCC1O)C(=O)Cn1cc(-c2c[nH]c3nccc-3c2)nn1 C1(C(=O)NCC2OCC(CC)C2)C=CCN1C(=O)C(c1cncnc1)C N1(C(CCN(CCC)C)=O)CCCC(CCNC(c2ccn(C(C)C)n2)=O)CC1 c1(C(n2ncc(CN(C(C(C)O)C3CCC3)CCC)c2)C#N)cccc(Br)c1 N1(C(C)=O)CC2CC2(C(=O)N(CC(C)NC(c2cnn(C(C)C)c2C)=O)C)C1 C(=O)(CN=c1[nH]c2c(c(=NCc3nc(Br)n[nH]3)[nH]1)SCC2)N1CCC(OC)CC1 c1(C(=O)NC2CCCC2NC(C2(Br)CC2)=O)cn2cccc(F)c2n1 CCCCCC(O)C(C)C(=O)N1CCC(NC(c2cncc(C)c2)=O)C1(C)C c1(C(=O)NC2CCC2NC(C2(CO)CCC2)=O)c(F)ccc2c1OCO2 N1(C(CCCC)=O)CCCC(C(=O)N(C2CC2(C)C)C)CC1 C1(C(=O)NC2CC(C)(OC)C2)CC2(CCN(C(=O)CCCC(C)=O)C2)C1 C1(NC(C2OCCCO2)=O)CS(=O)(=O)C12CCN(c1ccc([N+](=O)[O-])cn1)CC2 c1(N(C2CCCC2)CC2(O)CN(C(=O)NCc3ccccc3)C2)ncnc(OCC)c1 CCCCCCCCCC(=O)NC1CCCN(C(c2cnc(O)nc2O)=O)C1C C1(NC(C(C(C)C)(C)C)=O)CC2CCC(C1C)N2c1ncc(Cl)c(O)n1 CCC(CC)C(C)C(=O)NCCCC(C)(C)NC(c1ccc(SC)o1)=O C1(C(=O)NC(CNC(CC(C(F)(F)F)OC)=O)(C)C)CCCC2(CCOCC2)O1 C1(OCCNC(C2CCC2)=O)CCN(C(C2(O)CC2)=O)C1.C1(O)(CCC)CC1 CC1(C)C=C(C(=O)N2CCC(C(CO)NC(C3CSCC(=O)N3)=O)CC2)C1 Cc1cc(C(=O)NCC2(NC(=O)CCS(C)=O)CC2)nn1C(C)C N1(C(C(CCC)NC(N)=O)=O)CCC(NC(=O)CNC(=O)NC)C(C)(C)C1 N1(C(C(C(=O)OCC)F)=O)CCC(NC(=O)CSc2ccc(Cl)cc2)C1(C)C c1(C(=O)NCC2CCN(C(C3(C)CC3C(F)(F)F)=O)C2)cccc(N)c1O C(=O)(C(CCC(N)=O)c1cn(C2CN(NC(=O)CC(C)C(C)(C)C)CC2C)nn1)NC N1(C(CCCC(=O)OC)=O)CC2CCC(C1)N2C(C1CCCN1C1CC1)=O N=c1nc(N2CC3(COC(CO)C3)C2)[nH]c(=NC2Cc3ccccc3C2)[nH]1 c1(N(C(N2CCC(CC=C)C2)=O)C)ccc(C#N)c(C)c1 c1(C(=O)NC2CCN(C(C(C)CSC(F)(F)F)=O)C2)cncc2ccc(F)cc12 C12(C(=O)NCc3scc(C)n3)COC(C1)C(NC(c1n[nH]cc1Cl)=O)C2 Cc1oc(-c2cnn(C)c2)nc1C(=O)NC1CC(N(C)C(C2CCCOC2)=O)C1 N1(C(C2CCCCC2(F)F)=O)CCCN(C(c2c(Cl)cncc2Cl)=O)C(CO)C1 c1(OC)cc(C(=O)N(C2(C(=O)N(C)Cc3cnc(C)s3)CC2)C)[nH]n1 O=C(CNC(c1cc(Cl)ccc1Cl)=O)NC(=O)C(CC1CC1)C1CCCC1 CON(C(=O)C1CCN1C(=O)CCc1ncnn1C)C1CCC1 CCCCCC(O)C(=O)N1CCCC1(C)CNC(C1(C#N)CC2(CCC2)C1)=O N1(C(=O)C(O)CF)CCC(C2CCN(C(=O)CCc3ccccc3F)CC2)C1 C1(NC(=O)NC(c2c(C)nc(C)[nH]2)C)CCC2(CCC1(F)F)OCCO2 N1(C(c2c(CCC)[nH]cc2)=O)CC(NC(N2CCC(C(N)=O)C2)=O)CCC1C c1(C(=O)NC(CNC(CCC#C)=O)CCCC)cnc2c(c1)nc(O)n2C c1(CN2CC(NC(C=CC(=O)NC3CC3)=O)C2)ccc2cc[nH]c2c1 Nc1c(C(=O)NC2COCC2NC(c2cnc(S)nc2)=O)nc(O)nc1O c1(C(N(CC(CNC(c2c(O)n[nH]c2C)=O)OC)CC)=O)c(Cl)cc(C#N)cc1Cl c1(C(=O)NCCC(CNC(=O)CC(C)(C)O)OC)ccc(N(C)C)cc1[N+](=O)[O-] n1(C(C)C)ccc2ccc(-c3nc(Nc4cc5c[nH]nc5cc4Cl)cs3)cc12 c1(OC)ncc(C(=O)NC(C2(O)CCN(C(=O)C(F)C3CC3)CC2)C)c(C)n1 CN1C(=O)C(C)N(C(=O)C(O)CCC#N)c2ccccc21 N1(C(C=CC=CC)=O)CCC(NC(c2n[nH]cc2C(F)(F)F)=O)CC1C1CC1 N1(C(CC2CCN(C)CC2)=O)CCC2CC2(C(=O)NCCCCn2ccnc2)CC1 CC1CN(C(=O)COCCCF)CC1(C)CNC(c1cccc(CO)c1)=O C(=O)(C#CC(C)(C)C)N1C(CC(N2CC(=C)C2)=O)CC1 Cn1c(C(N2CCCCC(NC(=O)Cc3sc(O)nc3O)C2)=O)cnc1[N+](=O)[O-] C1(CC(=O)NC2CCN(C(c3ccccc3Br)=O)C2)CCCCC12OCCO2 N1(C(c2c(C)cccn2)=O)CCN(C)C(C(N2CCC3CC23C)=O)C1 C1(CC(=O)NCC(CC)NC(c2c(C)nn(C)c2F)=O)CN2CCN1CC2 C1(C)(CNC(c2c(C)c(C3CC3)on2)=O)COCCN(C(C2CC2(F)F)=O)C1 C1(C(N(C)CC2CCCS2)=O)CC12CC(NC(c1ncoc1C1CC1)=O)C2 N1(C(C=CCC)=O)CCn2c(CNC(=O)CCc3ccc(F)cc3)nnc2C1 c1(NC(C2C(NC(=O)OC(C)(C)C)CC2)=O)ccc(C#N)c(F)n1 CC(C)C(C)(C)C(=O)N(C)C.C12CCN(CC1F)c1nccnc1C(=O)N2 O=C(C(O)CC1CCCC1)NCC1CCC1NC(=O)C1CC1 C1(NC(C2C(C)(Br)C2)=O)CCC2(CC1)CN(C(c1cc([N+](=O)[O-])n[nH]1)=O)CCO2 Cc1nsc(N2CCC(NC(C3(CCO)CC3)=O)C2)n1 N1(C(C2C(c3ccc(C)s3)C2)=O)CCCC(NC(c2[nH]c(C)cc2C)=O)C1C CN1C2CCCC1CN(C(C1CCN(C(=O)C(N=[N+]=[N-])C(=O)O)CC1)=O)C2 CC1CC(NC(=O)Cc2cc(Cl)cnc2O)CCN1C(=O)CC1CC=CCN1C c1(C(=O)NCC2N(C(C(C)=C3CC3)=O)CCC2C2CC2)cc2c(s1)CC(C)(C)C2 C(=O)(CC(C)(C)CN(C)C)NCC(CCC)NC(C1(CC#C)CCCC1)=O N1(C(C(C)OCCC#C)=O)CCN(C2CCN(C(=O)C(C)O)C2)CC1 N1(Cc2scc(C(=O)OC)n2)CC(O)CC1C(N1CCOC(O)C1)=O C1(C(=O)NCCNC(=O)C(F)n2cccn2)Cc2nccn2C1 N1(C(C)C)CCCC(CC(=O)NC(C)(C)CN(C(=O)CC2CC(F)(F)C2)C)C1 C1(C(=O)NC2CC2(C)C(=O)NCC(=O)N(C)O)(OC)CCCC1 N1(C(=O)CN2CCOCC2=O)CCC2CC2(C(=O)O)CC1.C1(C2CC2)CC(=O)N1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC(CCNC(CCOCC#C)=O)OCCC1 C1(NC(=O)CCCc2ccccn2)CCN(C(=O)Cc2cnccc2Cl)CC1O N1(C(C2(COC)COC2)=O)CC(NC(=O)Cc2ccnc(OC)c2)CC(O)C1 N1(c2ccnc(C)n2)Cc2ccccc2CC1C(=O)Nc1ncnn2ccnc12 c1(C(N2CC(SC(CCN(C(C(=O)NCC)=O)C)C(C)C)C2)=O)cc(=N)[nH]c(Cl)n1 C(=O)(C1=C(C)CCOC1)N1CCC(NC(C=CCC)=O)C1 C1(CN(C)C(c2nn[nH]c2Cl)=O)CCN(C(c2ccn(C)n2)=O)C1 N1(C(CCC=CC)=O)CC2(CC(NC(c3ccnc(C)c3O)=O)C2)C1 N1(C(CCCNC(=O)OC)=O)CCSCC1CCNC(=O)C(F)CC1CCOC1 CCCCC(C(=O)NCC(CC1CCCC1)C(=O)NC1(C)CC(F)C1)C(C)C c1(OC)ncccc1C(=O)NCC1CC(NC(C2CCCS2=O)=O)C(O)C1 Cc1cccc(C(N2CCCC2CNC(=O)C(C2(O)CCCC2)F)=O)n1 C(=O)(CCCS(C)(=O)=O)NCC(C)CN(C(=O)CNc1cccnc1)C C1(NC(c2n(C(C)C)cnc2)=O)CC2CC1N(C(=O)CCCN(C)C)C2 c1(OC)c(C)csc1C(N1CCCCC1CNC(C1CCN(C)C1)=O)=O CCC(C)C(O)CC(=O)N1CCC1c1cn(CC2(SC)CC2)nn1 c1(C(N2CCC(N(C(C(F)=C(C)C)=O)CCO)CC2)=O)c(F)c(F)cc(F)c1F c1(C(C)O)ccccc1C(N1CC(N(C(=O)C(c2ccc(F)cc2)F)C)C1)=O C(=O)(C(C)C(C)(C)C)N1CCC(O)(CNC(c2c(C(CC)(C)C)cccc2)=O)C1 c1(-n2ncc(C(=O)NCC3(C(N)=O)CN(C(C4(F)CC4)=O)C3)c2)ccc(F)cc1 c1(C(C(=O)NCC2(COC)CN(C(C3CCCCO3)=O)C2)C)cccc(O)c1 N1(C(C2CC(CC)N(C(=O)CCCCCF)CC2)=O)CCCN(C)CC1 c1(OC(C(=O)NCC(CC)NC(=O)Cn2ccnc2C)C)ccc(Cl)c(F)c1 c1(NC(CCN(CC#C)C(C2CCNC(=O)C2)=O)=O)c[nH]ccc1=O N1(C(C(=O)NC2CC(C(=O)OC)C2)CC2CCCO2)CCCN(CCO)C(C)C1 Cc1cc2n(n1)CCN(C(=O)CC1COCCN1C(C1CCCCS1)=O)C2 C1(C(=O)NC2C(CNC(c3ccc(OC)cc3F)=O)C2)CNC(=O)CC12CCC2 CC(C)C(O)CC(=O)N1CCN(C)C(CNC(=O)C(F)=CCCF)C1 Cc1ccn2ncc(C(N3CC(C)(NC(=O)C=Cc4cnn(C)c4C)C3)=O)c2n1 c1(C(N(C(C)C(=O)NCCc2cnn(CC)c2)CCC)=O)cnn(C)c1 c1(C(=O)NC(CN(C(CCOCCOC)=O)C)CC)cc(C#N)c(F)cc1F c1(CC(=O)NCCN(C(CN(CCC)C)=O)CC2CC2)c(Cl)ccc(O)c1Cl c1(OC)cc(S(=O)(=O)NC2(CNCc3cc(OC)ncc3F)COC2)ccc1Br N1(C(c2c(N)n(CO)cc2)=O)CCCC(F)(CNC(=O)COC2CC=CC2)CC1 c1(CC(=O)NC(CNC(C=C(CCC)C)=O)CC)c(C)ncnc1C C1(O)(C(C)NC(C2CN(C(=O)CN3CCSCC3)C2)=O)CC(c2ccccc2)C1 C=CCC(C)(C)CC(=O)N1CC2(C(=O)NCC(O)COCCOC)CC1CO2 N1(C(C=COCC)=O)C2CCC1CN(C(=O)C(C)(c1ccccc1)N(C)C)C2 CC(CC1=CCCCC1)NC(=O)CC1(NC(C2CCN(C)CC2)=O)CCC1 N1(C(c2cc(OC)n[nH]2)=O)CCCC(C)C1CCNC(=O)CSc1nncn1C Nc1c(C(=O)NCC23CCC2CN(C(C2(CO)CCCO2)=O)C3)cc(F)cc1F C=CCC(CNC(=O)CCOC1CCOCC1)NC(=O)Cc1ncc(C)s1 C1(CNC(C2(CN(C(C(C)OCCCC)=O)C)CC2)=O)CCC2(CCC2)O1 N1(C(C(C2CCC2)OCC)=O)CC2(C(=O)NC(C)C=C)CC1CO2 C1(C(=O)NC(CN(C(CSCC=C)=O)C)C)Cc2ccccc2N1C(C)=O c1(C(N2CCC(C3CC3)(CNC(C=CC)=O)C2)=O)ccn2c1CCCC2 c1(CN(C2CCN(C(C(CC)Cn3ccnc3)=O)C2)C)cc(C2CC2)ccc1C c1(C(=O)Nc2nc(C)c(Cl)s2)ccc2ncc(CSc3ccc(Cl)cc3)n2c1 Cn1cc(C(=O)NC2CCC(CNC(=O)Cc3cccnc3N)C2)ccc1=O C1(C(=O)NCCCCNC(CC2(C)CC2(F)Cl)=O)CCCN(S(N)(=O)=O)C1 C1(CCC=C)CCCN(C(=O)CC(C)NC(c2ncn(C)c2C)=O)C1 c1(OC)cc(C(=O)NC2CCN(CC(c3ccccc3)C)C2C)cc(C)c1 C1(CC)C(OC)C(C(=O)OC)CN1C(C1CCCC(=O)C1)=O C(=O)(C1=CCN(C(=O)CCC2CCC(=O)C2)C1)N1C(C(=O)OC)CCC1C(C)C N1(CCC(N2CC(OCCNC(C(COC)C)=O)C2)=O)CCNC(=O)C1 N1(C(C2CC(SC)C2)=O)CC2CC2(NC(c2cscn2)=O)C1 N1(C(c2ccc(C)o2)=O)CC(CNC(=O)CSCc2cccs2)CCC1C C(C)(C(=O)NC1(CC(=O)N(C)CC2(SC)CC2)CCC1)OCC C1(N(C(c2cc(C)ns2)=O)C)CCCCN(C(=O)C(C)(C)c2cncs2)C1 N1(C(c2[nH]cc(C)c2)=O)CC=CC(C(N2CCC(OC3CC3)CC2)=O)C1 c1(CN2CCC(CC(N3CCN(c4ncccn4)CC3)=O)C2)c(O)cccc1Br C1(C(=O)NCC2CCN(C(CC3C(OC)CC3)=O)C2)Cc2ccncc2C1 C#CC1(C(=O)NCC(=O)N2CCCO2)CCN(C(C2CC23CC3)=O)C1 c1(N2CCCC(C(C)NC(C3(CNC(N)=O)CC3(F)F)=O)C2)ncnc2sccc12 C(=O)(C(C)(C)C)NCCCC1(N(C(=O)C(O)Cc2cnn(C)c2)C(C)C)CCC1 c1(OCC(=O)NCC(CN(C(C2(C=C)CCC2)=O)C)O)cccc(CS)c1 c1(C(=O)NC2CCCC2C(=O)NC2SCCS2)ccc(Oc2ccccc2)cn1 C1(CC(=O)NCCc2cc[nH]n2)CC2(CC2)CN1C(=O)Cn1ncccc1=O Cc1cc(NC(C2CCCCCCC2)c2nnnn2C2CCC2)cc(Cl)c1 C12(NC(c3cc4n(c3)CCC4)=O)CCCC1CN(C(=O)C=C(Cl)Cl)C2 C(C(=O)NCC1CC(F)(CNC(=O)CCC(=O)c2ccc(C)s2)C1)(C(C)C)SC N1(C(c2ccc(N(C)C)cc2)=O)CCCC(F)(CNC(C2CC3CCC2C3)=O)C1 c1(C(=O)NC)cc(C)nc(N2CCCC(C)(CNC(=O)CCc3ccc[nH]3)C2)n1 C1(CC(=O)N(CCN(C(c2cnc(OCC)nc2)=O)C)C)CCS(=O)(=O)CC1 C(=O)(C1=NOC2(CCN(Cc3ccnc(C#N)c3)C2)C1)NC(CC=C)CO C1(C(=O)NC(CC)COCC2CC2)CCCN(C(c2cocc2C)=O)C1 C1(C(C)NC(C(F)=CCC)=O)CN(C(c2ncccc2COC)=O)CCO1 c1(C(=O)NC(c2ccccc2)C(C)NC(CC=C(C)C)=O)cc2cc[nH]c2cn1 C1(NC(c2n(CC)c(O)nc2)=O)CC12CCN(C(c1cnc(O)c(C)c1)=O)CC2 C(=O)(CCCCCCNC(=O)C(C)(O)CC(C)C)N(CCC(C)C)CCO c1(-c2cnc(CC)s2)nc(CCO)nn1-c1cccc(Cl)c1 c1(CC)ccc(C(c2ccccc2)=O)c(C)n1.c12ccc(cc1)NC(=O)C(=O)N2 c1(C(N2CC(NC(=O)C(F)CC3CCC3)C2)=O)cncc(-c2ccoc2)c1 N(C1CC(O)c2ccccc21)OC(=O)CCn1cc(-c2cc(F)ccc2F)nn1 C(=O)(C(C)C(C)S(C)(=O)=O)NCC1(C)N(C(C2CCN(CC)C2)=O)CCC1 c1(C(=O)NCC2N(C(C3C(c4c(C)cccc4)C3)=O)CC2)nccc(C)c1N N1(C(c2c(C)occ2)=O)CCCC(N(C(=O)C(F)=CC2CC2)CCO)C1 Cc1nc(C(=O)NCC2(F)CN(C(=O)C(F)=C3CCCC3)C2)c(C)o1 N1(C(c2c(CC)nc[nH]2)=O)CCCCCC1CNC(c1ccc(CO)cc1)=O CC1CN(C(=O)CC(C)(C)C2CC2)CC2(CCN(CC3CCCS(=O)(=O)C3)C2)O1 N1(C(C(CCC)C)C(=O)NCCC2CC2)CCN2C(=O)OCC2(C)C1 C1(C(C)NC(c2cc[nH]n2)=O)CN(C(c2ccnc(F)c2)=O)CCO1 C1(NC(c2coc(Cl)n2)=O)C2CN(C(C3(c4ccc(O)nc4)CC3)=O)CC12 N1(C(=O)CCc2cccc(F)c2F)CCOC2(C1)CN(C(=O)C(O)CCl)C2 CCCC(C)(C)CC(=O)N1CC(=O)CC1C(=O)NC(C)(CCC)CCCC C(=O)(NNC(=O)C(CC)n1ccc(C2CC2)n1)C1(CC)CCCCCC1 N12CCC3(CC1)CCN3Cc1nc(co1)C2=O.S(=O)(=O)(CCCl)OC c1(C(C)NC(=O)C(=O)NCC(C)(C)C2CCCC2)ccc(C2CCCCC2)cc1 C1(C(N2CCCC(C(C)(C)CNC(=O)C3CC3)C2)=O)COc2ccc(O)cc2O1 N1(C(C(C2CCC2)OC)=O)CC2CC(C1)CN(C(C1CCC3(CCC3)O1)=O)C2 CCC(F)(F)CC(=O)N1CC(NC(c2ccc(CN(C)C)cc2)=O)CC(O)C1 N1(C(c2cc(C(C)=O)oc2C)=O)CCC(CO)(NC(c2occc2C)=O)CC1 C=CCC(C(=O)N1CC(N(C)CC2OCCC2C)C1)NC(C)=O CCC(C(=O)NCCSC(C)(C)C)NC(c1cncn1C)=O c1(C(N2C(C)(C(N3C(C(=O)OCC)CCC3)=O)CC2)=O)ncccc1Cl C1(OC2(CNC(C3CCCC3)=O)CC2)CCC2CCC1N2C(=O)COCC1CC1 CONC(=O)C(C1(O)CCC1)NC(C1CCC2(CC2)C1)=O c1(-c2cn(CCN(C(C3C4COCC34)=O)CC)nn2)ccn(C)c(=O)c1 c1(OC)ccc(C2CCC2)c(CN2CCOC(C(=O)O)C2(C)C)c1 Cc1ccccc1SCC(=O)NCC1CN(C(c2nc(C)n(C)n2)=O)CCO1 c1(C(=O)OC(c2ccccc2N)C(=O)OC)cnc(SC)n1-c1ccccc1 C(=O)(CC(C)P(C)(C)=O)NCC(CNC(c1ccc(C(=O)OC)o1)=O)C C1(C(=O)NC(C)(C)C)CC2C=CC1CC2.c12cnc(o1)C(C)COC(=O)N1CC2C1 C1(N(C(=O)CCc2ncccn2)C)CS(=O)(=O)C12CCN(Cc1ccon1)CC2 C(=O)(CS(=O)(=O)C1CC1)NC(C1CCC(NC(CC(C(C)C)OCC)=O)CC1)C N1(C(c2ccc(CCCCC)cc2)=O)CC2CN(C(=O)CC(C)C(C)C)CCC12 C(=O)(C1=C(Cl)CCOC1)N1C(COC)(CNC(=O)C(C)SC(C)C)CCC1 C(=O)(C(O)C(C)(C)C)N1CC2C(NC(C3C(c4ccc(OC)cc4)C3)=O)C2C1 C1(CN=C(NC(CC)CC)NC2CCN(C(C)=O)CC2)(CC#C)CCC(=O)N1 C1(C(=O)NC2CCC(NC(C=CCOC)=O)C2)CC(C2CCOCC2)=NO1 CC(C)(C(=O)NC(CCCNC1CCC1)c1ccccc1)C(F)F CC(C)CC(CC(=O)N1CCCCCC1C(C)(C)C)CC(N)=O N1(C(c2c(C)n[nH]c2)=O)CC(C2CCN(C(c3ccccc3C(C)C)=O)CC2)C1 C1(C(=O)NCCC(C(C)C)NC(=O)CCN2CCOCC2)CCCC1S(C)(=O)=O c1(C(=O)NCCCN(C(C)C)C(C2C3CCCC23)=O)cncc(N)c1 C1(C(=O)NC2CC(NC(CCOCCOCCOC)=O)C2)CCCC=C1Br S(=O)(=O)(c1ccc(C(O)CNc2nccc(=NCCc3ccc(C)s3)[nH]2)cc1)NC C1(CNC(C=CCCC=C(C)C)=O)CC(C)CN(C(C2CSCCS2)=O)C1 c1(C(=O)NCC2N(C(=O)CCN(C)CCO)CCC(C)C2)cnc2[nH]cnc2c1 C(=O)(N1OC2CCC1CC2)C1N(C(CC2CCCC(=O)C2)=O)CCC1 CC(C)CC(O)C(=O)N(C1CCN(C(c2cccc(O)n2)=O)C1)CC1CC1 C1(C(N(C)CC2CCN(C(C(CC)N(C)C)=O)C2)=O)CC(F)C(=O)N1 CC1CCN(C(=O)C(C)(F)F)C1CNC(=O)C(C1(O)CCOCC1)(F)F c1(C(=O)OC)ccc(CC(=O)NCC(O)CNC(=O)CC(C)(C)CC)cc1F C1(C(N2C(CNC(c3ccns3)=O)CC(F)C2)=O)CNc2ccccc2O1 C1(CNC(C2COCCO2)=O)COCCN1C(C1CCCC(F)C1)=O c1(CC)ncc(Cl)c(C(=O)NC2CCN(C(=O)C#CC(C)(C)COC)C2(C)C)n1 c1(CC)ccc(C(=O)NC2CC23CC(NC(=O)C(c2nc(C)cs2)C)C3)cc1F N1(C(C2(CC#C)CC2)=O)CCN(C(c2cc(COC)n(C)n2)=O)C(C2CC2)C1 C(C(CC(C)C)C(=O)N1CCCCC1CCCNC(=O)CC(O)CN(C)C)OC c12ccc(cc1)C1CCCN1C2=O.c1c[nH]nc1-c1cnccn1.CC(F)F S(=O)(=O)(CCN=c1[nH]c2c(c(=NC3COC4(CCCC4)C3)[nH]1)COC2)N(CC)CC c1(CN2C(C(=O)NC(CCC)C)CC(O)CC2)cn2nc(C)ccc2n1 c1(Cc2c(C(N3CC(NC(C(C)C)=O)C(O)C3)=O)cccc2)cnc(O)c(F)c1 c1(NC(C2C(C(=O)OC)C2)=O)cc(-n2cc(-c3cc(OC)nn3C)nn2)ncn1 N1(C(c2cccc(C)c2Cl)=O)CCC(CNC(=O)C(C)C2CCC2)C(F)(F)C1 Cc1cn2c(C(=O)NCC(O)CNC(=O)COC(F)F)cnc2s1 C1(C(=O)NCCC(C)NC(c2ccc(-c3ccccc3)s2)=O)CCOC(C)C1 n1(CC(=O)NCC2N(C(=O)Cn3cncn3)CC2)ccc(C2CC2)n1.C1(CC)CC1 C1(C)(CC(=O)N(CCC(C)NC(c2nscc2Br)=O)C)CCCCC1 C#Cc1cnn(C)c1C(=O)NC(C)C=CC(=O)NCC1CCCOC1 C=C(Cl)CC(C(=O)NCc1ncn(CC)n1)NC(=O)CC(C)F C(=O)(CCCN=c1nccc[nH]1)NC(C)C(=O)NS(=O)(=O)CC1CCCCC1 N1(C(C(C(C)C)NC(=O)C2CC2)=O)CC(C(=O)NC2CC3CCC2CC3)C2(CC2)C1 N1(CCCCCCC=C)CCCCCC1C1CCCO1 C1(F)(CNC(c2c(CN(C)C)nccc2)=O)CCN(C(c2occc2Cl)=O)CC1 N1(C(C2(C(C)C)CCN(C(=O)CCCCC(N)=O)C2)=O)CCC(C)C(F)(F)C1 N1(C(c2ccc(C)cn2)=O)CCC2(COCC(CNC(=O)C#CC(C)(C)C)O2)C1 n1(CC(=O)NCCN(C(c2cncc(OC)c2)=O)C)ccc([N+](=O)[O-])n1 C1(C(C)(C)NC(=O)C=CCO)CCN(C(=O)CCCC2CC2)C1 N1(C(Cc2nnc(C)o2)=O)CCC2C(C1)CN2C(c1c[nH]nc1C)=O c1(SCC)cc(CNC(=NCCSC)NCc2cc(NC)ccn2)cc(Cl)c1 c1(C(=O)NCCCCC2(C)CC2)cccc(N2CCOCC2=O)c1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCC(c2cn(-c3cccc(OC)n3)nn2)CC1 C#Cc1cccc(OCC(=O)NCC2CC(F)CN2C(=O)CCC(=O)N(C)C)c1 c1(C(=O)NCCCC(C)NC(c2cc(C3CC3)cs2)=O)cc(Cl)cc(Cl)c1O c1(CC(=O)Nc2c(C(=O)N(C3CC(=C)C3)CC)n[nH]c2)cc(Cl)cc(Cl)c1 C1(NC(=O)C=Cc2cscn2)CCSC12CN(C(=O)CSCC1CCCCO1)C2 Cc1cc(=NC(C)c2ccc(F)c(F)c2)[nH]c(CCC(F)(F)F)n1 Cc1ccc(N2CCCCC(C(=O)NC3CCCC(C)CC3)C2)c([N+](=O)[O-])c1 C1(NC(c2cn(C3CCOCC3)nc2C(F)(F)F)=O)C2CCC(C2)C1C(=O)O N1(C(C(C2CN(C(CC3CC(OC)C3)=O)C2)OC)=O)CC(C)(C)CC1CC(N)=O C1(C(N(CCOCCNC(C(C)CC(F)(F)F)=O)C)=O)CCC2(CC1)CC(O)C2 c1(C(N2CC(O)(CNC(C3(C)N(C)CC(OC)C3)=O)C2)=O)cc(C)c(N)cc1F CC1CCCC=C1C(=O)NCc1ccc(CNC(C2CCS2(=O)=O)=O)cc1F CN1CCC(C(=O)NC2CC3CC2N(C(=O)C(C)(C)N(C)C)C3)CC1=O C(C)(c1ccsc1)=CC(=O)NC(CNC(COCC(=O)OC)=O)C(C)C C1(NC(CC2CN(C)C2)=O)CC2CN(C(c3ccn(-c4ccc(O)cc4)n3)=O)CC12 c1(C(N(C(C2CC(C)(F)C2)=O)C(C2(O)CN(CCOC(C)C)C2)=O)C)ccccc1 c1(OC)ccc(C(C)C(=O)N(C2CCN(C(=O)C(C)O)CC2)C)cc1 C1(C(N(CC(CNC(C=C(C)c2cccs2)=O)C)C)=O)CCn2ncnc2C1 C(CCN(C(=O)CC1CC1C)C)(C(C)C)NC(CC(=C)C)=O CC1(C)CCC(CNC(C2CCOC2)=O)N(C(c2cc(O)nc(O)n2)=O)C1 C1(NC(=O)CN2CCNC2=O)CC2CC(C1)N(C(=O)CCN1CCC(F)C1)C2 Cc1cc(C)c(C(=O)NC(CCC2CC2)C(=O)N2CCC(C(N)=O)CC2)o1 C12(C(N(C)CC3C4CN(C(C(C)SC)=O)CC43)=O)CC(C)(C1)OC2(C)C C(CCCC(=O)NC1(CCCNC(C2CCC(F)(F)C2)=O)CC1)OC C(=O)(CCC(C)(C)N(C)C)Nc1cccc(CNC(CC(C)CN(C)C(N)=O)=O)c1 N1(C(c2c(C)nc(CC(C)C)s2)=O)CCC(NC(=O)CNC(N)=O)C(CO)C1 c1(C(N2C(CCNC(CC(C=C)(C)O)=O)CCCC2)=O)ccc2c(n1)CCOC2 c1(CCC)c(C(=O)NC2CN(C(C3CC4(CCC4)C3)=O)CC2O)nnn1C C1(C(N2CC(CNC(C3CCN(c4ccncc4)C3)=O)C2)=O)CC12CCOCC2 C(=O)(CCCCC(N)=O)N1C(CCNC(c2cnn(C(C)C)n2)=O)CC(OC)C1 C1(CC(=O)NC(CC)CN(C(=O)C(C)C2CCCC2)CC)CC2CCC1C2 C1(C2CC2)(C(=O)NC(C(N2C(C(=O)OC)C(C)(C)C2)=O)CN(C)C)CC(=O)C1 C(CCCC(=O)N1CCOCC1CO)NC(C)=O.c1(C(=O)N)cnn(CCCN(C)C)c1 c1(C(N2CC(CN(C(C3C(=C)C3)=O)C)OCC2)=O)cc2cc(Br)cn2cn1 Cc1cnc(CCCC(=O)N(C(CNC(=O)Cc2c[nH]nc2C)C2CC2)C)o1 C(=O)(C(F)C1CCC1)N(CCNC(CNC(=O)NC)=O)CCOCCO Cc1cnn(C)c1C(=O)NCCCC1(NC(=O)Cc2nc(Br)sc2C)CC1 Cc1cccc(-c2nccc(C(C)NC(c3ccc(C)n3C)=O)n2)n1 c1(C(=O)NCC(CC)NC(C(C)OCC#C)=O)nnn2c1COCC2 CCCC(C(=O)NCC(C)NC(=O)COc1cn[nH]c1)N(C)C C1(N(C(CSC)CO)C(c2cc(I)ccc2Br)=O)C(C)OCC12CCNCC2 CCC(CC)(CCNC(C1CCC2(CC1)CC2)=O)NC(=O)COCc1ccnn1C c1(C=O)ccc(Br)c2ncccc12.c1(CC)cc(=NC(=O)C2C=CCN2)[nH]o1 C1(C)(CNC(=NCC=C)NCCC(C)Oc2ccccc2F)COCC(C)(C)O1 c1(C(=O)N(C2CCN(C(C3CCC(O)CC3)=O)CC2)CCCO)ncc(Cl)cc1F N1(C(C2(CC)CC2)=O)CC(OCCC(=O)NCCCc2ncc[nH]2)C1 CS(C)(=O)=NC(=O)C1CCN(C(=O)CC2CNCC2F)CC1 N1(CC)CCC(C(N2CC(C(=O)N(CC(=O)OC)C)(OC)C2)=O)CC1 C1(NC(c2ccc(CC)cc2F)=O)CN(C(=O)COCC(F)(F)F)CCC1(C)C C1(C(N(CCCCC)CC(C)O)=O)(OCC)CN(C(=O)CC2CCOC2)C1 C=CCCCCC(c1nnnn1CC1CCOC1)NCc1coc(C)n1 c1(C(=O)NCC#CCNC(c2ccc(C(F)F)cn2)=O)ccc([N+](=O)[O-])c(F)c1 N1(C(C(C(C)C)n2ncc(C)c2)=O)CC2(CCCN(C(C3(C)CCC3)=O)C2)C1 N1(C(CCS(C)(=O)=O)=O)CC2(CCC2)CC1CNC(=O)C(F)=C1CCCC1 N1(C(CC(C)(F)F)=O)CCN(C(=O)CCCN=[N+]=[N-])C(CC(F)F)C1 CN1CC(C)(C)CC1C(=O)NCCCNC(c1cn(C2CCOC2)nn1)=O N1(C(CC(C)N(C(Cc2c(C)ccnc2)=O)C)=O)CC(C)C(C)C1C C1(C(=O)NC(C#C)(C)C)C2CCCC2CN1C(=O)C(C(C)C)C1CCC1 N1(C(CC(CC=C)c2ccccc2)=O)CCCN(c2nnco2)CC1C C1(N(C(=O)COCCOC)CCC)CCN(C(C2CC3CC3C2)=O)CC1 c1(CCC)cccc(C(=O)NC2CCCC2CNC(=O)CC2C(CC)C2(F)F)c1 CC(CC(=O)NCCNC(c1cc2ccncc2[nH]1)=O)CC(F)(F)F C1(NC(c2c(C)n[nH]c2)=O)CCN(C(C2(c3ccccc3F)CC2)=O)CC1O c1(C(C(=O)NCCOCCNC(C(CC)n2cccn2)=O)(C)C)ccc(F)c(C)c1 c1(C(=O)NC2CCCN(C(c3c(C)oc(CO)c3)=O)CC2)n[nH]c2c1CCSC2 CCCC(CCC)CC(=O)NCCN1CCN(C(=O)CCc2cccn2C)CC1 c1(C(N2CCC(NC(C3C(CC(C)C)C3)=O)C2)=O)cccc(N=c2cc[nH]cc2)c1 N1(C(c2cnc(CC(C)C)[nH]2)=O)CCCC(NC(c2nnc(O)cc2C)=O)C1C c1(OC)cncnc1C(=O)N(CC(O)CN(C(=O)C(C)OC1CCCC1)C)C c1(CCC(=O)N(C2CCN(C(c3ccns3)=O)C2)CC)ccc(F)cc1F c1(OC)cc(=O)n(C)cc1C(N1CCC(NC(=O)CSc2ccncc2N)C1)=O C(=O)(C(C)CC(N)=O)N1CCC(CN(C(C2(CC#C)CCCC2)=O)C)CC1 c1(C(=O)OCC)cnccc1N1CCC(O)(CNC(C23COC(CF)(C2)C3)=O)C1 C(CCC(N)=O)(C(=O)NCCOCCCNC(=O)C1=C(C)OCCS1)NC(C)=O C(=O)(CCCN(C(=O)CCOCCCNC(=O)CC1CCSC1)CCO)OC c1(C(N2CC(CNC(C3CCSC3)=O)C(C(F)(F)F)C2)=O)cnc2n1CCC2 O(NC(=O)C(C1CCC1)NC(=O)CC1CCC(=O)C1)CC(CC)C c1(C(N(C2CCCN(C(C(C)SC(C)C)=O)CC2)C)=O)cc2cc(Cl)sc2[nH]1 CCC(C)(C)CC(=O)NC1CC(C)N(C(=O)CC2(COC)CC2)C1 c1(C(=O)NC(C(=O)NCCCCC=C)CC#C)cccc(C)c1F c1(CNCC2(C(N(c3ccn(C)n3)C)=O)CC2)c(Cl)cccc1Cl C1(NC(C(c2c(CC)con2)N(CCOC)C(C)C)=O)CCC(F)(F)CC1 Cc1conc1C(=O)NCC1COC(CNC(=O)CCn2ccnc2)C1 CC(C)(CCCNC(C1CC(CF)C1)=O)C(=O)N1CCCC(CCF)C1 c1(NC)ccc(F)cc1C(=O)N(C1CCC(NC(C2(C(F)F)CCCC2)=O)C1)C C1(C(=O)NCC(CC)N(C(C=CC(=O)OCCCC)=O)C)CCCNS1(=O)=O N1(c2cc(NC(c3c(C)nns3)C)nc(C(F)(F)F)n2)CCC(C2CCC2)C1 N1(C(C(CC)(C)C#N)=O)CC2CC(NC(c3cc(Br)no3)=O)CC1C2 C1(CN(C(C(C)N2CCC2)=O)C)CCN(C(C2SCCCS2)=O)C1 Cc1c(C=CC(=O)NC2CC(NC(=O)CC(C(F)(F)F)n3ccnc3)C2)cnn1C N1(C(CCc2c(C)nn(C)c2)=O)CC2CCC2(NC(C2Cc3nccn3C2)=O)C1 C(=O)(CC1=CCCCC1)N1C2CC(C(=O)NOCc3nccc4cc[nH]c34)C1CC2 CC(C)CC(C)CC(=O)NC(C)CNC(c1ncc(Br)cc1O)=O N1(C(c2cc3[nH]ccc3s2)=O)CC2CCCC(C1)N(C(=O)COc1ccsn1)C2 c1(CC(=O)NC2CC(NC(C3(OC)CC(CF)C3)=O)C2)nc([N+](=O)[O-])n[nH]1 C1(CC(=O)NCC=Cc2ccco2)CCCCN1C(C1CC12CCC2)=O Cc1ccccc1CC(=O)N(C)CC1CCCC(C)C1.C12(CC1)C(=O)NC2 c1(C(N2CCC(NC(COCC)=O)C(CC)C2)=O)ccc(OC)c2ccncc12 N1(C(CN(CCOC)C(c2sccc2Cl)=O)=O)CCC(O)C1C(C)C C1(C(C)(C)CNC2CC3C=CC2C3)CCCCN1C(=O)Cn1cncn1 C(C)(C)(CC(F)C(=O)N(C(CF)CF)C)NC(CC=CCC)=O c1(NC(c2c(COC)ccs2)=O)cccc(NC(c2cnc[nH]2)=O)c1 C(=O)(CS(=O)(=O)CCO)NCC1(COC)CCN(C(=O)CC2CCCC2C)CC1 C1(C(=O)NCC2N(C(c3c(C)nc(C4CC4)o3)=O)CCSC2)CNC(=O)CC1C Cc1nc(C(N2CC3CC2C3NC(=O)C(C(C)C)N2CCCCC2)=O)n(C)n1 C(=O)(CC(C)(C)C(C)(F)F)NC(C1CCCCC1)CNC(C(F)OC)=O N1(C(c2c(CC)noc2)=O)CC(C2CCCN(C(=O)Cn3nccn3)C2)C1 c1(CCC)c(C(=O)N(C2CCN(C(=O)CS(=O)CC)C2)CC)[nH]c(C)c1C(C)=O C1(CC(C(=O)OC)O)CCN(Cc2cn(CC(C)(C)O)nn2)CC1 N1(C(c2ccc(C)nc2O)=O)CC2CCC1CN2C(C1CCC2CC2C1)=O N(C1CCC(NC(=O)CC(C)(C)O)c2ccccc21)C(c1c[nH]c(=NC)o1)=O N1(CCC)C(=O)NC(c2ncnc(OC)c2OC)C2=C1C(C)N(C)C2=O CC1CCC(C(N)=O)N1C(=O)Cc1cccc(NCc2cncc(F)c2)c1 CCCCC(CC)C(=O)N1CCOCCC1C(N1CC(O)(Cc2ccccc2)C1)=O C(=O)(C1=NOC2(CCOC2)C1)N(CC(CNC(c1c(C)nc(C)[nH]1)=O)O)C n1(CCOCC=C)c(N(C2CC(F)(F)C2)C)nnc1-c1ccc[nH]1 C1(C(=O)NCC(CC=C)NC(C2CCC(N(C)C)CC2)=O)CC(O)CN1C C(=O)(C(C)C(F)(F)F)N1C(C)(CN(CC)NCCCN(CC)CC)CCC1.C(=O)NC c1(C(=O)NC2C3CN(C(c4c(CC)n(C)cc4)=O)CC32)cc(OC)cc(Cl)c1 C1(NC(C(C)OC)=O)CN(C(=O)CCc2nc(=N)[nH][nH]2)C(C)(C)C1 CC1CC2(CCO1)CC2C(N1CC2=C(C1)CN(C(=O)COC1CCCOC1)C2)=O N1(C(c2scc(C)c2C)=O)CCOCC(F)(CNC(c2nccn2C(C)C)=O)C1 c1(C(N(CCNC(C2C(C=C)OCC2)=O)C(C)C)=O)c[nH]c2cccc(Cl)c12 CCC(C)CC(=O)NC(C1CCCN(C(c2cc(C)n(C(C)C3CC3)n2)=O)C1)C S(=O)(=O)(c1ccc(I)cc1)N1CC(COC)N(C(c2cccc(CO)n2)=O)CC1 C=CC1CN(C(=O)CCOc2ccc(Br)cc2)CC1NC(=O)C(C)(C)C c12cc(Cl)ccc1CNC2.C1(NCC)CCCC1N(C)C Cc1cc(C(=O)NCC2N(C(=O)C3=CC(C)CC3)CC2)c(C)n1C1CCCOC1 c1(NC(C2C(C)CCCN2C(=O)Cc2cnnn2C)=O)ccc2c(c1)CCO2 C(=O)(CC(C)CC(C)C(=O)OC)N1CCCCC(NC(CSCCOC)=O)C1 c1(C(N2C(C)C(C(=O)NC)CCC2)=O)cc([N+](=O)[O-])c(F)c(F)c1F C1(C(N2C(C(=O)NCC3CC(C(=O)NCC#C)C3)CCC2)=O)CC(CC)=NO1 c1(C(=O)NCC(Cc2ccccc2)NC(C(C)OCCC#C)=O)ccn(CC)n1 C(CCO)(C(C)(C)O)OC.N12CCC(C1)C(C)(C)C(=O)N(C)C1CC(C1)C2=O.C(C)(=O)O C(C)(CCC(=O)NC1C=CC(CNC(=O)CC2CCCOCC2)C1)OCC CCCCC(O)C(=O)NCCC(C)(CC)NC(c1cn(C)c(=O)cn1)=O C(=O)(CCCCN=[N+]=[N-])NC(C(=O)NC(C=C)C1CCC1)c1cccs1 C1(CC)(NC(=O)CCC2CCOC2)CCCN(C(=O)Cc2cc(C)ccc2O)C1 C1(C(CN2CC(C)(C)C2)=O)Cc2ccccc2CN1C(c1cc(Cl)ccc1F)=O O(NC(=O)C(CSC)N(C(=O)C=Cc1ccncn1)CC)CCCCC CCC(C)(CC)C(c1nnnn1CC1CCCO1)NCc1ncc(C)s1 c1(OC(C)C)ncccc1N(C)C.c12cccc(c1)C(CCO)NC(=O)NC2 C(C(=O)NC(C)C=CC(=O)Nc1ccn(CC)n1)(C(C)C)SCC N1(C(CCc2cc(C)sc2C)=O)CCN(C(c2cc(CF)on2)=O)C(C(F)F)C1 c12cc(ccn1)SC2.C(CCCC(C)(C)C)NC(=O)Nc1ccns1 C(=O)(CC(C)C(C)C)NCC(CC(C)C)NC(=O)CCN1CCC(F)C1 C1(NC(C(n2c(C)ccn2)C)=O)CN(C(C2(C(C)(F)F)CC2)=O)CCC1C C1(CNC(c2c(C#C)c[nH]n2)=O)CN(C(=O)CC2CC=CCC2)CC2(CCC2)O1 CC(C)(C)C(O)C(=O)NCCC1CN(C(=O)C(N)=O)C1 c1(C(=O)NCCN(C(C2OCCC2C(C)C)=O)CC)csnc1Br c1(CC(=O)OC)ncc(CNCC2(CC3CC3)CC2)s1 C1(=CCNC(C(C)(C2CC2)OC)=O)CCN(C(=O)CCc2ccoc2)CC1 C1(C(=O)NC2CCN(C(CC(COC)(C)O)=O)C(C)C2)CCC2(CCOCC2)O1 C1(CC)CN(Cc2cccc(OC)c2C)CCN1C(c1nn(C)c(C)c1Br)=O c1(C(=O)NC2CCC(C(=O)NCC3CCOC3)CC2)cc(Cl)ccc1[N+](=O)[O-] C1(C(=O)NC2(COC)CN(C(C3CC34CCC4)=O)C2)CCC(C)CC1 c1(NC2(NC(=O)CN(C)CCO)C(C)CCCC2)ncc([N+](=O)[O-])cc1Br c1(CC)cnc(Cl)[nH]c1=NCCCCNC(c1cc(C(C)(C)C)n[nH]1)=O N1(C(c2ccn(CC(C)C)n2)=O)CCCC(C)C1CNC(c1c[nH]c(=O)cn1)=O Nc1c(C(=O)NC2CC2CNC(=O)C(c2ccc(F)cc2)CO)ccc(Cl)c1Cl Cn1ccn2c(CCC(=O)NCC3CCC4C(C3)C4(F)F)nnc2c1=O C1(c2cn(CCN(S(C)(=O)=O)C3CC3)nn2)CN(C(C2(F)CC2)=O)CCO1 CCC(C)C(C)C(=O)NCCOC1CN(C(c2ccncc2OC)=O)C1.C(C)(C)N C(C(C)(C(=O)NCc1cccc(Cl)n1)NC(=O)CCOC1CCC1)SC Cc1conc1C(=O)NC(C(=O)NC(CC1CC1)CO)c1ccco1 c1(C(=O)NCC(O)CCCC2N(C(c3c(C)scn3)=O)CC2)ccc(F)cc1F CC1=C(C(=O)N2CC(CCNC(c3cnnn3C(C)C)=O)OC(C)C2)CCCC1 C(C(CCNC(C1CC=CC1)=O)OC)NC(CC=CC=C)=O N1(C(CCCCSC)=O)CC(C2CN(C(=O)C=Cc3ncc(C)[nH]3)C2)C1 CCC(C)(C#N)C(=O)NCC1CC(C(F)(F)F)CN1C(=O)CSC(F)(F)F C1(CNC(=O)CC2CCCC(=O)N2)C(C2CC2)CCN1C(=O)CCCCO C12(CNC(=O)CC3CC=CC3)CCCC1N(C(c1cc(O)ccc1F)=O)CCC2 c1(C(N2C(NC(c3c(OC)ccc(C)c3)=O)C=CC2)=O)c(Br)cc(Br)c(O)c1Br N1(C(Cc2c(C)cnn2C)=O)CC2CC(C1)CN(C(c1ncn3c1CCC3)=O)C2 N1(C(C(CO)NC(=O)C=Cc2ccsc2)=O)CCCC2COCC12 N1(C(c2c(C)nns2)=O)CCC(NC(c2cnn(C)c2F)=O)CC(O)C1 C1(CNC(Cn2cc(C(=O)OC)nn2)=O)CCN(C(c2cnn(C)c2F)=O)C(C)C1 C1(C(N2CCC(C(C)NC(=O)CSC(C)(C)C)C2)=O)CCc2n[nH]cc2C1 N1(C(C(C(CC)CC)OC)=O)Cc2nccn2CC(NC(C2CC(F)(CF)C2)=O)C1 N1(C(CCC(C)=O)=O)CC2CCC1(CNC(c1ccc(CC(C)C)cc1)=O)CC2 c1(CN(C(=O)CN2CCCC(OC(C)(C)C)C2)C)ccc(F)c(Br)c1 C1(CC)CC(C(N2CCC(N(C(c3cscc3COC)=O)CC)C2)=O)CC(=O)N1 C1(NC(c2c(C)cccc2)=O)CCCCCC1C(N1CCn2nccc21)=O Cc1cc(Br)cc(C)c1S(=O)(=O)NC(CO)CCc1ccccc1 c1(C(N2C(CN(C)C(c3cnn(C(C)(C)C)c3)=O)CCC2)=O)cnn(C2CC2)c1Cl C1(C(N2CC(NC(CCc3c(C)ncs3)=O)C(O)C2)=O)CCCNC(=O)C1 C1(C(=O)NCC2(CNC(C3CC(=C4CCC4)C3)=O)CCOCC2)CCC(F)(F)C1O CC(C)C(C(=O)N(C1CCN(C)CC1)C)NC(=O)C=Cc1ccoc1 C(=O)(C(C)(C)CCCC(=O)NC12CCCN(C(=O)C(F)=CC3CC3)CC1C2)OC c1(CC(=O)NC2(CCNC(C3(c4cc[nH]n4)CC3)=O)CC2)c[nH]c2cnccc12 c1(C(=O)OC)cc(C(=O)NCC2(O)CN(C(=O)C(C)N(C)C)C2)ccc1OCC1CC1 c1(CC)cccc(C(N2CCCC(NC(c3cccc(F)c3NC)=O)C2)=O)c1N C1(NC(COC)=O)CC2C(NC(=O)C(OC)OC)C2C1 Nc1c(C(=O)NC2CCN(C(c3cncs3)=O)CC2)cccc1F C12(CC)CCN(CC1)C(=O)C(C)C(=O)NC2.C1(F)(NC(C2CC2)=O)CCOC1 CC(O)C(C(=O)NC1C2COCC12)NC(=O)C=CC(F)(F)F Cc1c[nH]cc1C(=O)NC1C=CC(CNC(C23CC(F)(C2)C3)=O)C1 c1(C(N2CC(CC(C)NC(C(C)Nc3cccs3)=O)C2)=O)cnc2c(c1)CCC2 c1(C(N(C(C)CCNC(=O)C(C)(C)C2CCC2)C)=O)coc(S(=O)(=O)N(C)C)c1 c1(CC)nc(=N)[nH]cc1C(N1CCC(NC(=O)C(F)C(C)(C)O)C(F)C1)=O C1(C(=O)NC(C=CC(=O)N(CCC)CCC)C)CN(C(C)C)C1 C(C)(CC1CCC1)(C(=O)NC1(C)CC1)N1CC(Cc2c(OC)csc2)C1 c1(C(=O)NCC2C(NC(Cc3ccc(C)o3)=O)C2)cccc2c1NC(=O)CC2 C(C)(C(C)C(=O)NCC(O)C(F)F)N(CCOC)C.C1C(=O)N1 C1(Nc2nc(C(=O)OC)c(Cl)cn2)COC2(C1)CN(C(C1CC3CCC1O3)=O)C2 Cc1cccc(C(=O)NC2(C)CCCC2NC(=O)CSCc2ccccc2Cl)c1 c1(CC(=O)N(CC(CN(C(C2C(C)=CCS2)=O)C)O)C)cc(C)nc(O)c1 N1(C(c2cc(C)c(Br)o2)=O)CCC(CO)C(NC(=O)C(=O)N(C)C)C1 C12(C(N(CCCCC(=O)NCc3c(C)nsc3)C)=O)CCC(C1)C2(C)C C=CCCCCC(=O)NC(C)CCCNC(=O)CC(C)(C)COC C1(C(=O)NC2CCC(N(C(C(C)C3CC3)=O)C)CC2)CC(c2cnn(C)c2)=NO1 c1(CN2CC(CC(=O)N(CCCCO)CC)OCC2)ccc([N+](=O)[O-])c(Br)c1 N1(c2ccc(C(C)=O)cn2)CC23CCCC2(CN(C(C2CCC(F)C2)=O)C3)C1 S(=O)(=O)(CCC(=O)NCCC(C)NC(c1csc(C)c1)=O)NC c1(NC(C2(C)N(C(Cn3c(C)ncc3)=O)CC2)=O)cccc(O)c1C N1(CC(COCC#C)O)CCN(C(c2ccc(Nc3ccccn3)cn2)=O)CC1 N1(C(C2C=CCN(C(c3c(N)cncc3)=O)C2)=O)Cc2ncsc2C1 C1(CCC)CCCCO1.C12CCN(CC1)C(=O)N(C(C1CC1)C)C2.C1(C)CC1 C1(CNC(COCC)=O)CCC(NC(C2NC(=O)C3CC23)=O)CC1 c1(N(C)CC2CC(OC)C23CCC3)ccc(Cl)c2c1CCC2 c1(C(N2C(C)CN(C(=O)CC3CCCCO3)CC2)=O)cc(Br)c(O)c(Br)c1 Cc1cccc(C2(C(=O)N(C(C)CNC(=O)C=CC(=O)OC(C)(C)C)C)CC2)c1 N1(CCNC(CC(C)C2CC2)=O)CCN(C(=O)CCn2ccnc2)CC1 c1(CNC(C(C)C(C)NC(C)(C)C)=O)nc2ccccc2n1C.C1(C(=O)N)CC1 N1(C(c2c(C)cns2)=O)CCCC2C(NC(c3cc(C(C)C)no3)=O)C(C)(C)C12 c1(CC)nc(C)ncc1C(N1CCN(C(C2CC2F)=O)C(CC(C)(C)C)C1)=O Nc1cccc(C(=O)NC2CC(NC(c3cnn(-c4ncccn4)c3)=O)C2)n1 n1(C2=CC(SC)=CC(Cl)CC2)cc2ccc(CNCc3c(Br)ccnc3Cl)cc2n1 C1(C(N2CC(CC(=O)NC)N(C(=O)C(O)CSC)CC2)=O)CCc2nccn2C1 c1(OC)ccc(CN2CCC(N3CCC(C)(C)C3)C2)c(F)c1F Cc1cncc2cc(C(=O)N(C3CCC(NC(c4ccc(Cl)[nH]4)=O)CC3)C)sc12 N=c1ncn(CCC(=O)NCC2CCC2NC(=O)Cc2nnc(O)s2)[nH]1 N1(C(c2c(C(C)C)cco2)=O)CCN(CCCNC(C2CC23CC3)=O)CC1 c1(OC(C(=O)NCCN(CCC)C(c2ccccc2SC)=O)C)cccc(F)c1 CCC(CC(=O)NCC(CC)NC(=O)CCc1nccn1C(C)C)C(C)C C1(NC(C2N(C(c3c(OC)ccc(C)c3)=O)CC(F)C2)=O)CCc2n[nH]cc2C1 n1(CC(=O)NCCCN(C(C=CC(CC)C)=O)C)nc(C2CC2)cc1C(F)F c1(OC)ccc(CNc2nccnc2N2CCNCC2)c(Cl)c1OC n1(C(C)C)ccnc1C(=O)N(C)CCN(CC(O)CN1CCOCC1)CCO N1(CC(c2ccc(OC)c(OC)c2)O)CCC(=O)N(CCc2ccncc2)C1=O N1(C(C2CCSC2)=O)CC(C(=O)NCCSCCO)C2(CC2)C1 C(C(C)(C(=O)NC1CC(C(=O)NC(C)CCO)CC1O)OC)OC c1(C(=O)NCCCN(C(CC2CC(SC)C2)=O)C(C)C)oc(C)nc1C N1(C(CCSCC(C)C)=O)CCC(C)(CNC(c2ccn(CC(F)(F)F)n2)=O)C1 C1(C(=O)NC(C)CNC(=O)Cc2cn(C)nn2)CC12C1CC3CC(C1)CC2C3 CCCCCCCC(=O)N1CC(NC(=O)CCNC(=O)C=CCl)CC1(C)C C1(C(N(C2(c3ccccc3)CN(C(C)C)C2)C2CCCCS2)=O)COCCC1C c1(OC)cc(Br)ccc1CNC(C1CCC(OC)CC1Br)=O Cn1ccc(C(=O)NC2CC2NC(=O)C(C)(O)Cc2ccccc2)cc1=O CCCCC(O)CC(=O)NC(CN(C)C)CC(=O)NCCC1=CCCCC1 C(=O)(CCN(OC)C(=O)NOCC(=O)OC)NCC#C.C1(C)CN2CCC1C2 CCC(CC)CCCC(=O)NC1CCC(NC(=O)C2=CCC(C)(C)CC2)CC1 CCCC(C(c1nnnn1CC(F)F)NCCC(=O)OC)OC.C=O N12CCOC(C1)CC2=O.C(=O)(NOC1CCOC1)C1(C(=O)OC)CC1 C1(CC(=O)NC(CC)CN(C)C(C2CC(C)(C)C2)=O)CCC(=O)N1C N1(C(CCNC(=O)NC(C)(C)C)=O)CC(CC(=O)Nc2c(CC)c[nH]n2)C(C)C1 c1(N(CC(=O)OCC2CCCC(C(F)(F)F)C2)C)ccc(Cl)cc1Cl Cn1cnc2cccc(C(=O)NC3CN(C(=O)C(F)=C4CCC4)C(C)(C)C3)c12 N1(C(c2ccc(C)c(O)n2)=O)CC(CNC(C2CN(C(C)C)C2)=O)C2(CCC2)C1 C(=O)(C1=CC(C)(C)C1)N(C(c1cccc(OC)c1)CN(C)C)C1CC1 CCCCC(CNC(C1C=CCCN1C(C)=O)=O)NC(=O)CC1C(=O)NN=C1C C12(NC(COc3cccc(C#C)c3)=O)COCCC1CN(C(C1(SC)CC1)=O)C2 C(C)(C)(CCCNC(C1(NC(=O)Cn2cncn2)CCCC1)=O)OC CC(C)C(CNC(=O)CC1CNC(=O)O1)C(=O)NC1(C2CCCO2)CC1 CC1CCOC(C(N2CC(NC(=O)CCCC3CCC3)CC2CO)=O)C1 C(=O)(C(C)(C)C#N)NCCC1CCC(NC(C=CC(C)(C)SC)=O)C1 c1(NC(C2CC2(Cl)Cl)=O)ccccc1.C1C(=O)NCCCN1C CC(C)C(CNC(C1(C)CCCOC1)=O)C(=O)NCc1cc(O)ccc1F c1(CC(=O)NC(CC(C)NC(C2(OC)CCCC2)=O)C)cccc(NC)c1 C1(CNC(=O)CSCCNC(c2c[nH]c(=O)cn2)=O)CC2(CC2)CO1 N1(C(CCCOC(C)(C)C)=O)CCCCC1C1CCCN1c1ccc(C#N)nc1 N1(C(C2CCC(C)C2)=O)CCCN(CCNC(c2cnc(N(C)C)s2)=O)CC1 c1(C(=O)NC2C(C)CCN(C(c3ccc(Cl)cc3O)=O)C2)cc2scc(Cl)c2[nH]1 C=CC(CC)CC(=O)N1CCN(C(c2ccc(C(N)=O)nc2)=O)C(C(C)C)C1 C(=O)(C(C1CCOC1)N(C)CCN(C)C)NCCOCC#C c1(C(C(C)C)NC(c2n[nH]c(O)n2)=O)ccc(F)cc1Cl c1(C(CCC(=O)NC(CC)CNC(=O)CCOC2CCC2)=O)c(F)cccc1F CC(C)(C#CC(=O)NC1CCN(CCCO)C1)CNC(c1cc([N+](=O)[O-])c[nH]1)=O c1(C(=O)NC2C(CNC(c3ccc(F)c(O)c3)=O)CCCC2)ncc(F)cc1F C1(NC(=O)NNC(N)=O)CC(O)C1(C)C.N12CCC(C1)NC(=O)C2 C(C)(C)(CC(=O)NC1(CC)CC1)NC(c1c(CC)nco1)=O c1(C(=O)NC2C(CNC(C3(CC)COC3)=O)C2)cc(Br)cc2nc(O)[nH]c12 N1(C(CCc2cnc(C)s2)=O)CCC(C)N(C(c2cnn3cc[nH]c23)=O)CC1 C(=O)(CC(C(F)F)c1cccc(F)c1)NC1CCN(C(C2C(=C)C2)=O)CC1 C1(CNC(C=C(CC)CC)=O)C2CCN(C(=O)C(C)OCC(C)C)CC12 Cc1nn2cc(C(N3CC(NC(c4cnc(C)s4)=O)CC3C)=O)nc2s1 C1(NC(CN(C(C)=O)C)=O)CC12CCN(c1ccn3ccnc3n1)CC2 CC1(C)CN(C(c2cnc(S)nc2)=O)CC(CNC(C2(c3cccs3)CC2)=O)O1 C1(C)(C(=O)NCCCCC(C)NC(c2cnc(F)cn2)=O)CCCC(F)(F)C1 CCC(C(=O)N1CCCC(N(C(=O)C(C)C(C)C)CC(C)C)C1)C(C)O O(C=CC(=O)NCC(C1CCC1)NC(c1cnoc1C)=O)CC c1(C(N2CC(NC(CCCC=C)=O)C(C)C2)=O)cccc2c(C)ccnc12 C12(C(=O)NC(C3CCOC3)C#C)CC1CN(C(C13CC(CO)(C1)C3)=O)C2 CCC(C(=O)N(Cc1ccccc1)OC)N(C(=O)CN1CCCC1=O)CC S(=O)(=O)(c1ccc(C=O)s1)N1CCC(C(C)N)CC1 N(C(=NCCSc1ccc(O)c(C(N)=O)c1)NC1CC(O)C1C)C(COC)C CC1CCN(C(C2(N3CCNC3=O)CC2)=O)C1CNC(c1ccc(NC=O)cc1)=O C1(COC)CCCCN(C(=O)C(C)(CO)NC(c2ccc[nH]2)=O)C1 CC1(C)C=C(C(=O)NC23CC2CN(C(C2CC(N4CCOCC4)C2)=O)C3)C1 N1(C(C(CC(=O)OC)C)=O)CC2(C1)OC1(C)CC2(NC(=O)CCCSC)C1 C1(C)(CC)C=C(C(=O)NCC2(CNC(=O)Cc3ccccc3O)CC23CCC3)C1 C(C(C)(F)C(C)(C)F)NC(C(N1CCC(C(F)(F)F)(OC)C1)C)=O C1(CC(=O)N(CC)Cc2cccs2)CCCN(c2nccc(SC)n2)C1 CC1CC2CN(C(=O)CNC(N)=O)CC2N1C(C1Cc2c[nH]cc2S1(=O)=O)=O c1(C(=O)NCC2CCN(C(C3C(=C)CC3)=O)CC2)cccc2nc(S)oc12 C1(NC(C(=C(C)C2CC2)F)=O)CN(C(C2(O)CCC2)=O)CC(C)(C)C1 N1(C(C2C(C)CCO2)=O)CCC(C2(NC(C3CC(NS(C)(=O)=O)C3)=O)CC2)CC1 C(=O)(CCN=c1ccc(C)c[nH]1)NCCC1CC(OC)CN1C(=O)C(O)C1CC1 C(=O)(CCCCCCC(C)C)NCC(C(=O)NC1(C=C)CC1)(C)CC c1(SC)cccc(NC(C2CCN(C(=O)C(c3cccn3C)=O)CC2)=O)c1 Cn1cc2c(n1)CCCC2Nc1nc(N2CCC(OCCO)C2)nc2c1CSC2 CC1CN(C(c2cccc(-n3cncn3)c2)=O)CCC1NC(C1CCOC(=O)N1)=O C1(CC(N2CCC(N(C(CCC#C)=O)C)CC2)=O)COCC2(CCC2)O1 C(=O)(C(C(C)(C)C)NC(c1ccnn1CCF)=O)N1CCC(OCC)C1 O=C(C1=CCOC1)NCCC1(NC(c2ccc(-n3ccnn3)cc2)=O)CC1 c1(C(N2CC(CNC(C3CC3CF)=O)C2)=O)ccn2nccc2c1 C1(C(=O)NCC(C2CC2)NC(=O)C(C2CC2)NN2CCCC2)(CO)CCC1 C=CCC(C)(C)CC(=O)N1CC(NC(=O)CC2CCC2)C(C2CC2)C1 C1(C(=O)NCC2(CNC(C3(C)CC3)=O)CCCC2)CC2(C1)CC(C)(C)C2 C(c1cccnc1)=C(C)C(N1CC=CC(NC(c2cc(CC3CC3)on2)=O)C1)=O N1(C(c2nn(C)c(C3CC3)c2)=O)CCC2(NC(=O)CC3CCCCCC3)CC2C1 Cc1cc(C(=O)NCCCCC(C)NC(C2(F)CC2)=O)c2c(n1)CCCC2 N1(C(CC2C(C)(C)CCO2)=O)CCCC2(CCN(C(c3nc(Cl)sc3Cl)=O)C2)C1 Nc1cc(Cl)ccc1C(N1CCCCC1CNC(C12CC(C1)C(C(F)(F)F)O2)=O)=O CC1(CNC(=O)CC23CCC(CC2)C3)CCCN(C(C2CCS(=O)(=O)C2)=O)C1 N(C1CCc2cc(CNC(=O)C(C#N)CC)ccc21)C(c1cnc(CCC)[nH]1)=O C=C=C(C)CC(=O)N1CC(F)CC1CN(C(c1cc(C(=O)OC)co1)=O)CC N1(C(C=Cc2n(C)ncc2)=O)CC2CN(C(C3CC3C(F)F)=O)CCC12 c1(NCC(C)C(N2CCCCC2C)C)ccccc1F CC(CC(F)(F)F)C(=O)N1CC2CC(C(N3CCCC(O)C3)=O)CC2C1 C1(C)(CNC(CC(C)(C)OC)=O)CN(C(=O)C(C)CN(C)C)C(C)(C)C1 Cc1nccnc1C(N1CC(CNC(=O)CN(C(=O)C(C)C)C)CC1C)=O c1(C(N2CC(c3cn(-c4cccnc4F)nn3)C2)=O)cc(Cl)ccc1Cl CC1CN(C(c2cnn(CCF)c2)=O)CC(C(=O)N(C2CN3CCC2CC3)C)O1 C(=O)(C(CCC1CCC1)NC(=O)CC1CCC(=O)N1)N1C(C(=O)OCC)CC1 C1(C(=O)NCCC(C)NC(C=CC=CC)=O)COC(=O)N1 c1(OC(C)C(=O)N2CCC2Cn2cc(CC3CC3)nn2)cncc2cc(Cl)ccc12 N1(C(C2OCCN(C(C(C)=NOCC#N)=O)C2)=O)CCC2OCCC2C1 N1(C(c2cnsc2)=O)CCCN(C(c2cc(=O)cc[nH]2)=O)C(CO)C1 C1(C(N(c2cccc(OCCCC)c2)C)=O)CCCN(C(=O)CCC)CC1 C#Cc1ccc(C(N2CCC(CNC(=O)C(O)CC)(COC)CC2)=O)nc1 C(C(=O)NC(CNC(c1cc(Cl)c(Cl)s1)=O)C1CCC1)(C(C)C)N1CC(C)C1 c1(C(=O)NCCC(C)(C)NC(CC(=O)OCC)=O)cnn2c1OCCC2 N1(C(C(F)=CC)=O)CCC(C)(C)C1CN(c1c(C(=O)NC(=O)C2CC2)cccc1)C C12(NC(C(F)=CC)=O)CCCCCC1N(C(=O)CCC#Cc1ccccc1)CC2 C12(CNC3(C(=O)NCC(=O)NCCOC)CC3)CCCCC1C2 N#CCCCCC(=O)NC1(CF)CN(C(=O)CCC2CCCOC2)C1 C(CCN=[N+]=[N-])N(C(C1(NC(C(C)C2CCC2)=O)CC1)=O)C C1(C(N2CCC(NC(C3OCCO3)=O)C2)=O)CCN(c2cccc(Br)c2)C1=O C12(CC(=O)NCC3CC(OC)CN3C(c3nc(C)n(C)n3)=O)CC(C)(C1)OC2C C(=O)(CN=S(C)(C)=O)N1CCC(CC(C)NC(c2nc(Cl)c(Cl)s2)=O)CC1 C#CCCN=C(NCC1CNC(=O)C1)N(C)Cc1cc(C(F)(F)F)nn1C C1(C(N2CCC(CNC(c3ncoc3C3CC3)=O)CC2)=O)CCC2(CCCC2)C1 c1(C(=O)NCCC(C)N(C(CC(CC)CN(C)C)=O)C)ccc2sncc2c1 C1(CC=C)(NC(C2CC(=C3CCC3)C2)=O)CCN(C(c2c[nH]nc2C)=O)C1 c1(C(=O)NCC(CCNC(C(=C(C)C2CC2)F)=O)O)cccc2sccc12 c1(C(=O)NCCOCCCNC(C2N(N=O)CCC2)=O)cccc(Cl)c1[N+](=O)[O-] Cc1c(C(=O)NCCC2CCCN2C(=O)Cn2cnc(=N)[nH]2)cnn1C1CCC1 C1(=O)C(C)SCC(=O)NCCCN1.C1(C(CC(=O)OCC)C)C=CCC1 C1(NC(C(C)CN2CCOCC2)=O)CN(C(=O)CSCCC2CCC2)CC1(C)C c1(-c2cccc(C(N3C(C(=O)O)CC(F)(F)C3)=O)c2)nnc2n1CC(N)CCC2 N1(C(CN(C)S(N)(=O)=O)=O)CCCCC2(C1)CN(C(=O)Cc1ccns1)C2 C1(NC(=O)C=CCO)COC2(CCN(C(c3n[nH]c(C4CC4)c3Br)=O)C2)C1 C=CC1(C(=O)NC2CC(CNC(=O)CCCN(C)C(C)C)C2)CCOCC1 CN1CCCC(C)(C(=O)NCCC2CC(C(=O)NCCP(C)(C)=O)C2)C1 C1(CC(=O)N(CCCCC=C)C)CC(C)(C)CN1C(=O)CCc1cncs1 n1(CC)nc(C)c(C(=O)NCC2(Cn3cc(C(=O)CC4CC4)nn3)CCC2)c1Cl Cn1cncc1CC(N1CCCC1CNC(c1cc(-c2csc(=N)[nH]2)c[nH]1)=O)=O C(=O)(C1=CCOCC1)NC(C)CCCCNC(c1cnc(C2CC2)o1)=O C1(C(C)(C)NC(=O)C=CC(N)=O)CCCN1C(C1CC12CCC2)=O N1(C2CCCN(c3onc(C)n3)C2=O)CCCC2c3ncn(C)c3CCN2C1=O c1(CC(=O)NC2(C)CC(C(=O)NCCCc3ccsc3)C2)ccc(C#N)cc1 C1(CNC(CCC#C)=O)CN(C(c2ccnc(OC)c2F)=O)CC12CC2 CC(CS(C)(=O)=O)N=c1nc2scnc2c(N2CCC3NC(=O)C2C3)[nH]1 C(C(C)(C)CC1CC1)NC(=O)C(C)OCCOC(C)C(=O)NCc1ccncc1 C1(C(C)NC(=O)CCc2nc[nH]n2)CCCN1C(C1CC1c1ccnn1C)=O C=CC1CN(C(=O)CCCCCNc2ccc(-c3ccncc3)cc2)CC1O c1(C(=O)NCC(CCNC(C(C)CC(F)F)=O)O)ccc2ncncc2c1 CCC(CNC(c1cnc(C(F)(F)F)cn1)=O)N=c1[nH]c2ccc(F)cc2s1 c1(N2C(=O)CC(C(N3CC(C(=O)OC)C3)=O)C2)ccc(F)cc1F C1(C(N(CC(C)NC(=O)C(C)(C)c2ccsc2)C)=O)CCCN1c1ccccc1 C(=O)(C(C)(C)c1ccncc1)N(CCNC(C(C)C1CCCO1)=O)C1CC1 C12(C(=O)Nc3c(C)nsc3)CCC(NC(=O)CNC=O)(CC1)C2 C(=O)(CS(=O)(=O)CCO)N1CCN(C(CNC(C(C)N(C)C)=O)C(F)F)CC1 c1(NC(C(CC)C2CCOCC2)=O)ncc(C#N)cc1Cl.C12CC(C1)CNC2=O N1(C(C(c2cn(C)nc2)(C)C)=O)CCCC(NCC2CC3CCC2O3)C1 c1(CC(=O)NCC23C(CN(C(CC(CC)(C)C)=O)C2)CC3)ncn2c1COCC2 N1(C(C2(C=C)CCN(C(C3COCCN3C)=O)C2)=O)CC2(CCCCCC2)C1 CCS(=O)CC(=O)NCC(C)NC(c1ccc(-n2cncn2)nc1)=O C(CNC(=O)C(C)(C)SC)(CC(F)(F)F)NC(C(CC)NC(c1ccco1)=O)=O C1(C(=O)NC2C(C3C(C)C3)C2)CC2(CCN(C(=O)OC(C)(C)C)C2)C1 N1(Cc2cc(C)nn2C)CCc2sc(C(=O)Nc3c(C)cc(Cl)cc3F)cc2C1 CC(C)C(C(=O)N1CCC(C)(CCNC(=O)CCc2cccc(Cl)c2)C1)C(C)C c1(SS(C)=O)ccccc1F.c12ccc(o1)SCCN(C)c1nnc(s1)C2 C1(C(N(C(C)C(=O)NC(C)CC2CCC2)CC)=O)CCC(=O)O1.C(COC)S C1(NC(C(C=C)OC)=O)CCC(C)(C)CC1CNC(=O)C(C)(C1CC1)OC N1(C(C2C(C)(C)CCO2)=O)CC(CC(=O)NCC2=CCCC2)C2(CC2)C1 S(=O)(=O)(CCCC1CCC1)NC1C(C(=O)Nc2cc(OCC)n[nH]2)C1 C1(C(=O)NC2C(CNC(CCC(=O)NC)=O)COC2)COc2ccccc2C1 Cn1cc(C(=O)NCC(C)(C)NC(C2CC(c3ccccc3)CO2)=O)c(Cl)n1 c1(CC(=O)N(CC(CO)(CO)NC(C(C)OCC=C)=O)C)csc2nc(C)cn12 C1(NC(C2(C)CC2(F)F)=O)CN(C(=O)C(F)(F)C2CC2)CC1C1CC1 N1(C(c2c(CC)cccc2)=O)CCC(CNC(C2(O)CCCCCC2)=O)CC1C c1(C(N2CC(CC)N(C(C3OCCO3)=O)CC2)=O)ccc(S(=O)(=O)C(F)F)cc1 CC1CN(C(C2CN(C(c3nc(=N)cc[nH]3)=O)CC2(F)F)=O)CC1(F)F C1(C(N2C3C(NC(=O)CC4C=CS(=O)(=O)C4)C(C3)C2)=O)C(F)(F)C12CCC2 N(C(=NCCc1cnccc1C)NC(C)COC)Cc1c(CC)ccs1 c1(C(=O)NCc2ccc(CC(C)NC(C(C=C=C)C)=O)cc2)ccc(C)nc1N CC1(C)CN(C(c2n[nH]c3c2CSCC3)=O)C(CNC(=O)CCF)CO1 C(=O)(C(O)CC(=O)OC(C)(C)C)N1CC(C(C)NC(C(CC)CC)=O)C1 C1(N(C(C(C(C)OC)N(C)C)=O)C)CCCCN(C(=O)CCc2ccsc2)C1 C1(C(N(CC(C)OC)C(C)C)=O)C=CCN(C(=O)CCCC2CCCO2)C1 c1(C(=O)OC)c[nH]nc1OCCNC(=O)CC(c1ccncc1)CNC(N)=O C1(CNC(c2c(CC)[nH]cc2)=O)CN(C(=O)C(C)OCc2ccccc2)CC1O c1(C(N2CC3C(NC(c4c(OC)nc(C)cc4)=O)C3C2)=O)cn(C)c(C)cc1=O C1(C(N(c2ccnc(C(=O)OC)n2)C(C)C)=O)C2Cc3ccccc3C12 Cc1cc(F)sc1C(=O)NC(CNC(=O)Cc1ccncc1Cl)C1CC1 c1(CNC(CCCN2C(C)CCCC2)=O)cccc2c1CN(C(C)(C)C)C2=O N1(C(c2nn(C)c(O)c2)=O)CC2CN(C(=O)COC(C)(C)C(F)(F)F)CCC12 Cc1ccc(=NCCC(=O)NCCCCC(C)NC(C2C(C)C2(F)F)=O)[nH]c1 c1(OC)cc(C)c(C(=O)NC(CNC(C2(S(C)(=O)=O)CCC2)=O)CO)cn1 N1(CSc2ccc(C#N)nc2)C(=O)c2cccnc2C1=O C1(C(N2CC(C)(NC(C3(C(F)(F)F)CCCC3)=O)C2)=O)CC2CCC2C1 C(CN(C)C)(C(C)(C)C)N(C(C(C)C1(C(=O)NCCF)CC1)=O)C N1(C(c2c(CNC(C(C)C)=O)nccc2)=O)CCc2cccnc2C1 C#CCC(C)(C)C(=O)N(C1CC(NC(=O)C(c2ccc(C(F)(F)F)cc2)O)C1)C N1(C(CCCC(C)(C)C)=O)C2CCCC1CN(C(C1(O)CCSC1)=O)C2 CCC(C)C(C(=O)NCc1nnn(C)c1C(=O)N(C1CCOC1)CC)NC(C)=O C=C(Cl)CC(C(=O)N(CC)Cc1nc[nH]n1)NC(=O)Cn1cccn1 c1(C(c2n(C(C)(C)C)nnn2)NC23CCC(CC2)C3)ccc(F)c2cccnc12 c1(NC2C3CN(C(c4cccc(CC)n4)=O)CC2C3)nc2ncc(Cl)cc2o1 N1(CC)CCN(C(=O)C(C2(O)CN(C(=O)C3=CCCSC3)C2)F)CC1C C1(C(=O)NCCCC)CSCCN1C(C1CCOC1(C)C)=O c1(CC(=O)N(C)CCN(C)C(c2cc[nH]c(=N)c2)=O)cccc2c1OCCO2 C12(C(N3CC(CN(C(=O)CC(O)C4CCCC4)C)C3)=O)CC(N(C)C)(C1)C2 Cc1c(NC(=O)C(C2CCCN(C(C3CC3C3CC3)=O)C2)(C)C)cccc1F C1(NC(C2(C(C)C)CCC2)=O)CCC2CCN(C(C3(N=[N+]=[N-])CC3)=O)C1C2 N1(C(=O)Nc2c(CC)cc(Br)cc2)CCc2c(cnn2C)C1C(N)=O N1(C(c2ccc(CCC)cc2)=O)CC2(NC(c3ocnc3C)=O)CCCC2(F)C1 c1(COC(C2(C)CC(OC)(OC)C2)=O)ccc(Cl)cc1Br C1(C(N2CCN(C(c3c(OCC)scc3)=O)C(CO)C2)=O)CC2(C1)CC1(CC1)C2 CC1=NNC(=O)C1CC(=O)NC1CC1NC(c1coc(C2CCCCC2)n1)=O N1(C(c2ccsn2)=O)CC2(CCCCN2C(C2CC2C2CCCCC2)=O)C1 c1(OCCCC)ccc2oc(-c3ccc(C(=O)NCCC(C)CO)nc3C)cc2c1 CC(C)C(CCC(F)F)NC(N1CCC(C)C(F)C1)=O CC1C2CC(C2NC(c2cccnc2)=O)N1C(C1(C)C=CCCC1)=O CCCC(O)C(=O)NC(C)C=CC(=O)NOCC1(C)CC1 c1(C(c2n(CCCOC)nnn2)NCC2(C)CC2)cccc(C2COC2)c1 c1(C(C)C)cc(=NCC(O)CNC(c2cncn2C(C)C)=O)[nH]c(Cl)n1 c1(C(N(C(CNC(C(CC)OC)=O)C)C)=O)cnc(OC)c(C(F)F)c1 CCCCC(=O)NCCC1CCN(C(=O)C(C)(C)Nc2ccccc2)C1 n1(CC(=O)OC)ncc(C(=O)NC(C)CN(C)C(C2CCCN2C(N)=O)=O)c1C c1(NC(c2c(C)oc(CNC(C3CS(=O)C3)=O)n2)=O)cccc(F)c1O CC(N)C(=O)N=c1ccn(CC(N2CCCC(CO)C2)=O)c(O)n1 c1(OC)ccc2[nH]c(C(=O)NCC3CN(C(c4ccc(C)o4)=O)CC3C)cc2c1 c1(N2C(CNC(c3cnn(-c4ccccc4)n3)=O)CC2)cncc(Cl)n1 CCC(CCC(=O)NCC(c1ccccc1)C)NC(=O)C=CSC c1(C(N2C(CN(C(=O)CCc3coc(CO)c3)CC)CCC2)=O)c[nH]c(=O)cn1 c1(C(=O)NC(C)CCNC(=O)COCc2cccnc2)cc(C(F)F)ccc1Cl c1(N(C)CCO)ccc(S(=O)(=O)C(N2CCc3nncn3CC2)=O)cc1 CC1(C(=O)N(C(C(=O)N2CC(C(=O)N)C2)C2CC2)C2CC2)CC1(F)F.C1(C)CC1 c1(CC)ncc(C(N2CC(C(=O)NC(COC(C)C)C(C)C)(CC)C2)=O)o1.C(C)(=O)O C1(NC(COc2cccc(C)c2)=O)CCSC12CN(C(=O)C(C)(O)C1CCC1)C2 c1(CCC)ncc(NC(=O)CN(CC(C)C)C(=O)CC2CCCCN2C)cn1 CC1CC2(CC(C(N3CCC(C)(CC(=O)NC4CCC(CO)C4)C3)=O)C2)C1 C12(C(N3C(C)CC(NC(CN4C(C)CCC4)=O)C3)=O)CCC(C#N)(CC1)CC2 C1(C(=O)NC2(CCOC)CCC2)CCN(C(c2ccncc2Cl)=O)CC1OC CCCC(F)C(=O)NCC1CC(C(=O)NOCC2CCC2)CO1 CCCC(CC)C(=O)N1CC(CNC(c2cnc(N(C)C)nc2)=O)C(C)C1 c1(C(N2CC(CCCCNC(c3c(C)snc3)=O)C2)=O)ccccc1F Cc1sc(C(=O)NC2CC3CCC2(NC(c2cnc(C(N)=O)s2)=O)C3)c(C)c1C CCC(C)C(C(=O)NCC1CC(OC)CN1C(=O)COc1ccc(O)cc1)OC c1(CC(=O)NC(C)CCCNC(C2CC2CF)=O)ccc([N+](=O)[O-])cc1F C1(C(N2CCN(C(C(C)OCC=C)=O)C(C)C2)=O)CCC2CCCCN12 N1(C(C(C)c2ccco2)=O)CCC(C2CN(C(c3cc[n+]([O-])cc3)=O)C2)CC1 C(=O)(C(F)CC(C)(C)NC(=O)CCc1cscn1)NCCc1cccc(C)n1 CON(CCC(=O)NC1CC2CCC(C1)N2C)C(=O)CN(C)C N1(C(c2c(CNC(CCC=C)=O)ocn2)=O)CCCC12CCCC2 Cc1ccc(C(N2CCCN(C(=O)C3=C(Cl)CC3)CCC2)=O)c(O)c1C Fc1c(Cl)ccc(Br)c1CNC(c1noc2c1CCC2)c1nnnn1CCCF c1(NC(C2CC(F)(F)CN2C(=O)Cc2ccc(Br)c(F)c2)=O)ncc(Cl)nc1Cl c1(C(CC)NC(=O)C(=O)NCCOCCN(C)C)ccc(F)cc1.c1(S)csc(C)n1 c1(-c2nnc(CCC(=O)NCC3C(NC(C(C)O)=O)C3)o2)ccccc1OC(F)F N1(C(C(C)C2CCCC2)=O)CCN(C(c2cc3n(c2)CCC3)=O)CC(CO)C1 C1(CC(=O)N(C2CCN(C(C3COCCO3)=O)CC2)C)CC2(COC2)C1 c1(OC)cccc2c(C(N3CCN(C(=O)CCC4CCC4)C(CF)C3)=O)cnn12 N1(C(C(CCC)=CCC)=O)CC(C2CCN(C(C3CC4CC4CC3C)=O)CC2)C1 N1(C(CN(CC(C)C)C(=O)CCC(C)(C)C)=O)CCC(CCO)C1 Cn1ncc(=NC(=O)C2CSCCN2C(=O)CSc2ccc(Br)cc2Cl)[nH]1 c1(C(=O)NCC23CCC2CCN3C(=O)CCC2OCCO2)ncn2ccccc12 Cc1ccc(C#N)cc1C(=O)NC(C)C(=O)NCC1CCN1C(C)(C)C C#CCCCCC(=O)N(C)CC=CC(N1CCC1CC(C)C)=O C1(C(N2CCCC(CNC(c3cncc(CC)c3)=O)C2)=O)Cc2ccccc2S1 N1(C(CCC)=O)CCCC1CCCNC(C1CCC(C(N)=O)C1)=O C1(C(C)(C)O)CCN(C(C2(C)CC(NC(=O)CCN3CCOC3=O)C2)=O)C1 c1(C(=O)NC(C(C)NC(C2CCC(=O)O2)=O)(C)C)cnccc1Cl c1(C(=O)OC)ccncc1C(N1CC(CNC(c2csc(C(F)(F)F)c2)=O)C1)=O c1(C(=O)NC(CN(C(=O)CCCC(C)O)CC)C)cc(Cl)c([N+](=O)[O-])cc1OC NC(=O)CC(C1CCOCC1)NC(=O)Nc1cc(-c2ccccc2)no1 C(N=c1[nH]c(C)cc(=NCc2ncccc2F)[nH]1)c1nccc(C)c1 C(N=c1nc(C(F)(F)F)c2c(ncn2C)[nH]1)C1CCCN(C(C)C)C1 C=C(C)CCCC(=O)NCC1CC(F)CN1C(=O)Cn1nc(C)nc1C c1(C(=O)NCC2N(C(c3n(CC)nnc3)=O)CCCC2C)ccc(N)c(C)c1C N1(C(c2nc(N(C)C)nc(O)c2)=O)CCN(C(=O)CN2CC(C)(C)C2)C2CCC12 c1(SCCC)nnc(C2CN(C(=O)NCC3CN(S(C)(=O)=O)C3)C2)o1 C1(C(N(CCOCCC(N2C(C(C)CO)CCCC2)=O)C)=O)CN2CCN1CC2 C1(C(=O)NC(C2(O)CCOC2)C)CC2CCC(C1)N2C(=O)C=Cc1nccs1 N1(C(=O)CCc2cncnc2)CCC(F)(C(=O)NOCC=C(C)C)CC1 N1(C(c2ccnc(OC)n2)=O)CC(NC(=O)C#CC(=O)N(C)C)CCC1C C=CC1(N(C(C)(C)C)C(C2C(C(=O)OCC)COCC2)=O)CCCCC1 C(=O)(C(C(=O)N(CC(C)Cc1ccccn1)C)C1CC1)OCC c1(C(C(=O)N(C2CCCN(C(COCCOC)=O)C2)CC)O)cc(F)cc(F)c1 C#CCCCCCC(=O)NCCC1CC2CCC(C1)N2C(=O)COCC1CCC1 N1(C(C(C)SC)=O)CC2C(CN(C)C(c3cnc(C(F)F)s3)=O)C2C1 C12(CNC(C3C(C)(CC)C3)=O)CC(CO1)N(c1nccc(CC#N)n1)C2 c1(Nc2ncccn2)ccnc(NC2CCCC(C(=O)OCC)C2)c1 c1(-n2c(-c3cccc(OC)n3)nc(C3CCCN3CC3CC3)n2)cccc(C#N)c1 Cc1ccc(C=CC(=O)N(C2CC(NC(c3cc(C)nn3CC(F)F)=O)C2)C)o1 Cc1ncc(C(=O)NCC2C(C(=O)N(C3CCOC3)CCF)C2(C)C)s1 N1(C(c2ccnc(C)n2)=O)CCCC(O)(CN(C(=O)C=Cc2cn(C)cn2)C)C1 C1(C(C(=O)NC(C(C)C2CC2)C)(C)C)CCN(C(c2ncccc2F)=O)CC1 N1(C(C2N(CCC)CCC2)=O)CC2=C(C1)CN(C(=O)C(CO)N(C)C)C2 c1(C(N2C(CO)CC(NC(C(CCC)OC)=O)C2)=O)cccc(NC)c1C n1(CCC(=O)N(C)Cc2cn(CCCC)nn2)nc(O)c2ccccc2c1=O N1(C(C2N(C(C)=O)CCC2)=O)CC(NC(C2(CF)CC(F)(F)C2)=O)CCC1C Cc1n[nH]c2cc(C(N3CCC(C)CC3CNC(C3(C)CCCC3)=O)=O)ncc12 c1(C(=O)NCC(CNC(c2ccc(CO)o2)=O)O)cnc(C2CCCO2)s1 C1(CC)CN(C(=O)CC(C)F)CCC1NC(c1ccnn1C(F)F)=O CCN(CC(=O)Nc1cccc(C#N)c1)N1CCCCCCC1C N1(C(C(c2cncc(F)c2)C)=O)CCC2(CCCCC2NC(=O)CN(C)C)C1 Cc1cc(C)c(C(=O)N(C)CC2CCN(C(C3CCCC(=O)N3)=O)C2)s1 N1(CCC(=O)N(CC(F)F)C)CCN(C)CC1C(F)F C1(NC(C2(COC(C)(C)C)CC2)=O)CC(C(C)(C)C)N(C(=O)C(F)=C2CCCC2)C1 CCC(C)C(C(=O)N1CCC(CC(=O)N(C)C)C1)N(C(=O)CN(C)C(N)=O)C c1(CCNC(N2CCC(C3CCCO3)C2)=O)cc(Br)no1 c1(C(=O)NCCN(C(=O)C(c2cncn2C)O)C(C)C)nn(C)cc1N N1(CC(C)Oc2ccccc2F)CCCC(CO)(NC(c2ccccc2)=O)C1 C1(C(=O)NCC(CCC)NC(C=CC=CC)=O)(CF)CCOCC1 c1(C(=O)NC2(c3c(F)cccc3F)CCCCC2)cn(CC2CC2)c2ccccc12 N1(C(C(CNC(C(C)C2CCCC2)=O)O)=O)CCOC(CO)C1 C12(C(=O)NC3C(NC(C(C)(C)NC(=O)OC(C)(C)C)=O)C3)CCC(F)(CC1)CC2 C1(NC(C(C)(C)SC)=O)CCC2(CC1)CC2N=c1cc(Cl)c(O)n[nH]1 Cc1c(C(=O)NC(C)CCCNC(c2ccccc2F)=O)ccc2cncn12 C1(CNC(C)C(F)(F)F)CCc2c(nnn2C)C1.c12ccccc1[nH]c(=O)[nH]2 c1(C(=O)NCC2C3CN(C(C4CCCS4(=O)=O)=O)CC23)cc(Cl)cc(F)c1F C1(N(C(CCN(C(C(C)(C)O)=O)CC2CC2)=O)CC2CC2)(CO)CC2(CCC2)C1 N1(C(C(C)N(C)C)=O)CCC2(CC(NC(C3CC(C)C3)=O)C2)C1.C(C)(C(N)=O)N CN1CC(C(N2CCCC(C(=O)Nc3cccc(O)c3)C2)=O)CCC1=O CC1CCCCC1C(N1CC2C(CNC(c3ccc(Cl)cn3)=O)C2C1)=O c1(C(=O)OC)cc(CC(=O)N(CCNC(=O)CC2CCOC2C)C2CC2)on1 C(=O)(C1=CS(=O)(=O)CCC1)N(C1CCN(C(c2[nH]nc([N+](=O)[O-])c2Cl)=O)C1)CC c1(N(C)C)cccnc1C(=O)NCCNC(C1CC1C(F)(F)F)=O CC(C)C(C#N)C(=O)N1CC(C2(NC(=O)C(C)COc3ccccc3)CC2)C1 C#Cc1ccccc1CC(=O)NCC(C)(C)CC(=O)NCC1(C)CCCO1 N1(C(CCOC(C)=O)=O)C2CCC1CN(C(C1CCCCC1(C)C)=O)C2 N(C)(S(=O)(=O)N(C)C)CC(=O)NC1CN(C(c2n(CC)nnc2)=O)C(C)C1.CC N#Cc1c[nH]c(=NC(=O)C2(F)CN(C(=O)Cc3ccccc3C(=O)O)C2)c(Br)c1 O=C(C1CCc2ccccc21)NC1C=CCN(c2cc(C(F)(F)F)ncn2)C1 c1(C(c2n(CCC)nnn2)NCC2(C)CCCS2)c(Br)nc(C)n1C CCC(CC)C(C)C(=O)NC1CN(C(=O)CCc2cncc(OC)c2)CC1F C(=O)(C(C)(C)CC(=O)NCCn1cc(C(=O)NCC2(C)CC2(F)Cl)nn1)OCC c1(CNC(c2c(C)cns2)=O)cnn2c1CN(C(=O)CC1CCOCC1)CCC2 Nc1cccc(C(N2CCC2CNC(=O)CCC2CC2(F)F)=O)c1F N1(C(C(CC)NC(N)=O)=O)CCC2(C1)CN(C(C1(C(F)(F)F)CCCC1)=O)C2 C(CNC(c1ccnn1CC(C)C)=O)(C(C)C)NC(C(C)OCCC=C)=O c1(CC(=O)NC(CC)CNC(c2nocc2COC)=O)noc2ccc(F)cc12 CC1CCN(C(c2ccco2)=O)C1C(=O)NCc1cc(Cl)cs1 C12(NC(C(C)(F)F)=O)CCOCC1CN(C(=O)C(F)=C1CCCC1)C2 C(C)(CCC(=O)N(C)CC1CC(O)C1)NC(c1cc(OCC)no1)=O c1(CSS(C)(=O)=O)cn(CC2CCCC2NC(C2(c3ccno3)CCC2)=O)nn1 c1(NC(=O)COc2ccccc2C(N2CC(NC)C(O)C2)=O)cc(C)ccc1F C1(NC(c2cn(CCNC(C3C(C)(C)COC3)=O)nc2)=O)C2CCC(F)(F)C12 C(CCCCC(=O)NC1COCC1NC(=O)CCCOC1CCOCC1)OCC Cc1cc(CCCNC(C2CCN(C(C3(C)CCCC3)=O)C2)=O)cc(C)c1 c1(C(=O)NCCNC(c2ccc(N)cn2)=O)cc2ccccc2oc1=O C(C(C)(C)C(C)(C)C)NC(c1cccc(Cn2cc(CCOC(C)=O)nn2)c1)=O c1(C(N2CC(OC)C(NC(=O)CC3CCCC3)C2)=O)cnc2c(c1)nnn2C C1(COC)CN(C(c2cnn(C)c2-n2cnnc2)=O)CCN1C(=O)Cc1cc[nH]n1 CCCC(C(=O)N1CCC(CF)(NC(C2CCCOC2C)=O)C1)N(C)C Cc1cc2scc(CC(=O)NC(C)CCNC(C3CC(F)C(=O)N3C)=O)c2s1 Cc1cccc(Cl)c1C(N1CC2C(NCc3cnco3)C2C1)=O Cc1cccc(Cl)c1CC(=O)N(C1CN(C(c2ccc(F)o2)=O)CC1F)C C1(C(=O)NCCN2CCN(C(c3ccc(SCC)nc3)=O)CC2)CCC(C2CC2)C1 CC(CCCc1ccccc1)C(=O)N1CC2(C1)CN(C(c1ccn(CC#N)n1)=O)C2 O=[N+]([O-])c1cccc(Br)c1N.c1(OC)ncc(Br)cn1 CCCCC(CNC(=O)C(c1ccc(F)cc1)OC)NC(c1nccnc1C)=O N1(C(C(C)C(C)c2ccc(Cl)cc2)=O)CC2(C1)CN(C(c1cc(O)cc(=O)o1)=O)C2 N1(C(CCC=C)=O)CCC(CNC(=O)CNc2ncccn2)(COC)CC1 N1(C(Cc2ccc(C)c(F)c2F)=O)CCCC2C1CCN2c1nnco1 N1(C(=O)NC)CCC(C(=O)NC(C2CCCCC2)CNC(C2(CCF)CC2)=O)C1 c1(C(=O)NC2CCC(C)(CNC(c3coc(CO)c3)=O)C2)coc(S(C)(=O)=O)c1 C(C(=O)NCCCN1CCOCC1)(C(C)C(C)(C)C)N(C(CC(C)C)C(N)=O)C c1(S)ccc(C(F)(F)F)cc1C#N.N(C(=NCCF)NCC)C(C)C.N1S(=O)(=O)N1 Cc1ccc(F)cc1NC(=O)CC(C)CNC(=O)Cc1nc(=N)[nH][nH]1 C12CCCC(C1)CC(=O)NC(CO)COC2=O.CCCC(=O)NC(C)C C1(C(=O)NCC(F)C2CCC2)CC12CCN(C(=O)CC1CCCSC1)CC2 c1(C(C)C(=O)NC2CCCN(C(=O)CCc3cccnc3)C2)ccc(F)c(Cl)c1 C(CCC(=O)N(C)CCNC(C1(CC2CCCCC2)CCOC1)=O)N(C(C)C)C c1(C(=O)NC(C(CO)NC(C2C(=C)C2)=O)C)ccccc1Cn1ccnn1 C1(CCNC(C2(COC)CCCC2)=O)COCCN1C(=O)CC1C(C)C1(F)F c1(C(=O)NC23CC(C2)N(C(=O)CCc2cc[nH]n2)C3)ccn2nnnc2c1 O=C(N=c1cncc[nH]1)c1cnc(-c2ccc(F)c(F)c2)nc1Sc1ccccc1 CC(C(F)C(=O)NCC1CCN(C(c2cc3occc3[nH]2)=O)CC1O)C(F)(F)F c1(N2CCOCC(C)C2)ccc(S(=O)(=O)N2CCn3c(C(F)F)nnc3C2)cc1F CC1Sc2ccccc2N(C(=O)C=Cc2ccc(-n3ccnc3)cc2)C1C C12(C)CC(NC(c3ccc(=O)oc3)=O)CN1C2=O.C(C)(C)(C(F)(F)F)OCC(=O)OC C(CCCCNC(=O)CCCN1CCC1)N(C)CC.C12(CCSC1)C(=O)N2 Cc1cc(C(=O)NC(CN(C)C)C(=O)N2CC(c3nn[nH]n3)C2)cc(F)c1 CC(C)C(F)C(=O)N1CC2C(C(N3CCOCC3)=O)C2C1 C1(CC(=O)NCC(CCNC(C(C)NC(=O)NC)=O)O)CCC(C(C)C)CC1 Cc1nc(Cl)sc1C(N1CCN(CC(=O)NCC2CNC(=O)CO2)CC1)=O c1(NC(=O)NC2C(=C)COC2)nc(Cl)c(Cl)cc1Cl N1(C(c2cc(C)nn2C(F)F)=O)CCCC2(CC(NC(=O)C(F)CC(C)C)C2)C1 c1(C(=O)NCC(CCOC)NC(C2(CC)CCCCC2)=O)ccnc2[nH]ncc12 C(=O)(C1=CCCSC1)N1C2C(C(=O)N3CC(O)CO3)CC(C2)C1 C1(NC(CCN(CCC)C)=O)CN(C(C2CCC(CN(C)C)O2)=O)CC1O c1(C(N(CC)CC2CCCN2C(=O)CCc2nncs2)=O)cnc2scnc2c1 C12(C(C)C)OCC(NC(=NCC3CCCC3)NCC(C)(C)C)C1S(=O)(=O)CC2 C(c1ccc2occc2c1)=CC(=O)NC1C(C)N(C(C2CCS2(=O)=O)=O)CC1 Cc1c(NCC(C)S(C)(=O)=O)ncnc1N1CCCC(F)CC1 N1(OC(=O)CN(C2CC(C#N)C2)CC)CC2(CN(C(=O)Cn3cccnc3=O)C2)C1 CC(C)CC(C)(C(N)=O)NC(=O)CN(C1CCC1)C(C1CC(=O)N(C)C1)=O C1(C(=O)NCCNC(Cc2c(C)noc2C)=O)CCc2c(n[nH]c2C)C1 c1(CN(C2CCOCC2)CCC)nc(O)nc2ccccc12 c1(NC(C2(C)N(C(C(COC(C)=O)C)=O)CCC2)=O)ccc(C#N)cc1C C(c1cccnc1)=C(C(=O)NCCN(C)C(C1(c2ccccc2)CCCO1)=O)C#N c1(N(CCN(C(c2c(CC)scc2)=O)C)C(C)C)ncnc2cc(C)[nH]c12 C(=O)(C1=NOC2(CCOC2)C1)N1C(CNC(c2ccccc2)=O)CC(OC)C1 C(=O)(CCCS(C)(=O)=O)NC(C1CN(C(C(C)OCCCC)=O)C1)C C1(CNC(c2cscn2)=O)CC2CC(C1)N(C(c1cc3n(c1)CCCC3)=O)C2 C=CC1(C(=O)NCc2ccnc(C)c2)CCN(C(c2cc[nH]c2C2CC2)=O)C1 C1(C(=O)NC(CC)C(C)C)CN(C(c2ccsc2C#N)=O)CC12CCC2 c1(OC)ccc(C)cc1CCNC1CCN(C(c2ccncc2C)=O)CC1C C1(OC(Cc2ccc(OC)s2)=O)CN(C(=O)C(C)(F)F)CC1n1ccnn1 C(=O)(CCCCC(C)CC)NC1C(COCC)CCN1C(=O)CC1=CCCCC1 CC1CCC(Nc2ncc(Cl)cn2)CN1C(c1cnoc1C1CCC1)=O C=C1CCC(CNC(C2CC(NC(C3(C#N)CC(=O)C3)=O)CCO2)=O)CC1 CCCCCCCCn1cc(CC2CN(C(=O)C(C)C(O)C(C)C)CCO2)nn1 CC1(C)C(Cc2cn(-c3cccc(F)c3Br)nn2)CCN1C(=O)CSC(F)(F)F c1(CC)nc(C(=O)NC2CCC2CNC(=O)C(=O)N=S(C)(C)=O)c2ccccn12 Cc1nc2cc(C(=O)N(CCN(c3cc(=O)n(C)cn3)C)C(C)C)cnc2[nH]1 Cc1c(C(=O)NCCCNC(=O)CC2CCC2(F)F)c2ccccc2n(C)c1=O Cc1oc2ccccc2c1C(=O)NCC(CO)NC(=O)Cc1cncc(Br)c1 c1(CCC(=O)NCC(=C2CN(C(=O)C(F)(F)c3cscn3)C2)F)cccnc1 C1(NC2(C)CCOC2)CC(NC(N2CCC(CN=[N+]=[N-])CC2)=O)C12CCC2 N1(C(=O)Cc2cccnc2O)CCC2CN(C(=O)C=Cc3ccco3)CC2CC1 N1(C(c2scc(C)c2C)=O)CC(NC(C2CCCC2)=O)CC2(CC2)C1 CCCC(C(=O)N(C1CCCN(C(c2cc(C(C)(F)F)on2)=O)C1)CC)OC c1(CCC)nc(=NC(C)C2CCN(C(=O)CC3CCCOCC3)C2)s[nH]1 C1(NC(C2CCCSC2)=O)CC2CCC(C1)N2C(=O)CNS(=O)(=O)c1cccs1 CC1CC(NC(c2cccc(Br)c2I)=O)CN(C(c2ccc(O)nc2)=O)C1 Cc1[nH]nc(C(=O)NCCN(C)C(C2CC2C)=O)c1C(F)F C1(NC(C(C)C(C)NC(C2C3CN(C)CC23)=O)=O)CC2(CCCO2)C1 N1(C(c2cc(OC)n[nH]2)=O)CC(O)(C2CCN(C(C3C=CCC3)=O)CC2)C1 C#CCCCCCC(=O)NCC(F)CNC(c1occc1Br)=O C1(C(=O)NCCOCC)COCCN1C(c1csc(Cl)c1)=O C1(CNC(CCc2cc(C)sc2C)=O)CCC(C)(C)CN1CC=O.c1nnsc1C C(=O)(C1=CC2(CN(C(CC(C)NC(C3CSC3)C)=O)C2)OC1)OC C1(NC(C(N2CCN(C)CC2)C)=O)COC2(CCN(C(C3CC(O)C3)=O)CC2)C1 c1(CNC(=O)NCC(c2ccc(Br)cc2)F)cnc2ccccc2c1 n1(CC)cc(CC(=O)NC2(CCCNC(=O)Cc3cc(C)on3)CC2)cn1 O=C(CCCC#Cc1ccccc1)NCC12CCC1CCN2C(=O)C=CCO CN1CCOC(C(N2CC(C(C3CCC34CCC4)=O)C2)=O)C1.N12CCC(CC1)C2=O CC1(NC(c2ccoc2C2CC2)=O)CCC(NC(c2nccnc2N)=O)CC1 C(=O)(C1=C(Cl)CCOC1)NC(CC#C)(C)C(=O)NC1CCc2ncnn2C1 C12(C(=O)NCC(C)(C)OCC(=O)NCCc3ccsc3)CC(CO)(C1)C2 c1(OC(=O)CCC(=O)N2CCC(O)CC2)cnccc1CN(C)CCN(C)C C=CCCC(C)N=c1[nH]c(N(C)Cc2cccc(C#N)c2)nc2cc[nH]c12 c1(C(N(CCCCCNC(=O)Cc2cn[nH]c2)C(C)C)=O)csc(C#N)c1 N1(CC(N2CC(C(C(=O)NC(COC)CO)OC)C2)=O)CCNC(=O)C1 N1(C(C2CCC(OC)CC2)=O)CC2CC(NC(=O)CC34CCCN3CCC4)C1C2 C12(C(N3CCN(C(c4cc[n+]([O-])cc4)=O)CC3)=O)CC(CCO1)N(C(N)=O)C2 n1(CCC)cc(NC(C2(NC(=O)CC3(C)OCCO3)CSC2)=O)cn1 C1(NC(C2N(C=O)CCC2)=O)COCCN(C(=O)CCc2ccc(O)c(O)c2)C1 C1(CNC(=O)CC2CC(F)C2)COCCN(C(C2CCC3(CC2)CC3)=O)C1 CC1(C(=O)NC2CC=CCC2C(=O)NCc2cnc[nH]2)CCCCO1 N1(C(CCCSC)=O)CC(CNC(=O)CCc2nncs2)C(F)(CO)C1 c1(C(=O)NC2(CNC(c3ccc(CSC)o3)=O)CCOC2)cc2ncccc2o1 c1(C(N2C(C(=O)NC(c3ccccn3)CO)CC(C)C2)=O)ccc(Cl)c(Cl)c1 C1(C(N(CCOCCNC(C(C)c2cc[nH]n2)=O)C)=O)CC(C)N(C)C1 C1(C(N2C(CNC(COCCOC)=O)CC2)=O)Cc2ccc(F)cc2O1 c1(C(=O)NCCCOCCC(=O)NC(C(C)C)c2ncc[nH]2)n[nH]c(C(C)C)n1 C1(NC(N)=O)CCOC1CNC(=O)CC1(NC(C2CCSC2)=O)CCC1 c1(NCC)ccc(C)cc1C(=O)NC(C)CC(C)NC(c1cncc(OC)n1)=O N1(C(c2n(CC)ncc2)=O)CCC(NC(C2CC2CN(C)C)=O)C1C C1(C(=O)OC)CCN(C(=O)C2(CN(C(=O)C=C(C)C(C)C)C3CC3)CC2)O1 c1(OC)ccccc1CC(N1CC(CC(F)C(=O)NC2(N(C)C)CC2)C1)=O C1(NC(c2c(OC)cc(C)cn2)=O)CN(C(C2CSCCS2)=O)CC2(CC2)C1 Cc1oc(SC(F)(F)F)cc1C(N1CC(OCCNC(C2CCC(=O)N2)=O)C1)=O c1(CC)cccc(N(CC)CC2CC2)c1.N1(C=O)CCOCC1CO C1(C(=O)NCCC(=O)NCC2(CO)CCCCC2)CC2CCCC2C1 C1(NC(Cc2c(C)ccs2)=O)CC2CN(C(C3(C#N)CC(C)C3)=O)CC2C1 CCCC(C)(O)CC(=O)NC(C)C(=O)NC(C)(C)CCF C=CCCCC(C)(C)C(=O)NC(CNC(=O)Cc1cnn(C)c1)C1CCC1 c1(CC(=O)N(CCNC(C2C(Cl)(C(=O)OCC)C2)=O)C)csc(C(C)C)n1 c1(OC)ccc(C(=O)NCC(CO)NC(C2(S(C)(=O)=O)CC2)=O)c(OC)c1C N1(C(C(F)C2CN(C(c3ccn(C)c(=O)c3)=O)C2)=O)CCCC2COCC12 c1(C(=O)NC2CCC(CC(=O)NCCC(=C)C)C2)cncc(F)c1 CC1CC2CN(C(c3coc(CNC(c4sccc4Cl)=O)n3)=O)CCN2C1 S(=O)(=O)(c1ccc(NCc2cc(C3CC3)on2)c(Cl)c1)N1CC(C)CC(C)C1 c1(C(=O)NC2CN(N3CCN(C(C(CC)O)=O)CC3)C2)nc[nH]c2nccc1-2 CC1(C)C2CCC1(C)C2C(N1CCC2C(NC(=O)CSCC3CCCO3)C12)=O C1(C(N)=O)CCCCC1C(=O)NCC1CCN(C(=O)COCC(F)(F)F)CC1 N#Cc1cnn2cc(C(=O)NCC3CN(C(=O)C4=CCCCO4)C3)cnc12 N1(c2ncc(C)cn2)CCCC(C)(C(=O)NCCC2SC(=N)NC2=O)C1 C1(C)(C(=O)NCCC2(OC)CN(C(=O)C=C(C)Cl)C2)COc2ccccc2O1 N1(C(C(C(C)C)n2cncn2)=O)CCC2CCC(C1)N2C(C1CSCCS1)=O N1(C(=O)NC(C(=O)OCC)C)CCC2CC(NCc3nnn(C(C)(C)C)n3)C2C1 Cc1cccc(CC(=O)NCCC2CCCN2C(C2COC(=O)N2)=O)c1Cl C(C#Cc1cccnc1O)CNC(=O)CNCc1ccccc1 C1(CCNC(c2cscc2C(F)(F)F)=O)(OC)CCN(C(=O)COC)CC1 C(=O)(CC(C(F)F)n1ccnc1)N1C2(CNC(C3C(C)(C)CO3)=O)CC(C1)C2 C12(C(N3CC4C(CNC(c5csnn5)=O)(C4)C3)=O)CCC(C(F)F)(CC1)C2 N1(C(Cc2cc(C)on2)=O)CCCC2CN(C(c3cnc4n(c3=O)CCS4)=O)CC12 N1(C2CCC(NC(C(=O)NC(C)C)=O)C2)CCN(C(c2cnc(Cl)[nH]2)=O)CC1 CCCCC(C(=O)N(C)CC1(NC(c2nc(C)n(C)n2)=O)CC1)C(C)C C(=O)(NN1CCCC1C(=O)NC1CCC(=O)NC1)c1c(C)cncn1 c1(C(=O)NC2CCC(NC(c3cnc(O)o3)=O)C2)ccc(S(=O)(=O)C2CC2)cc1 c1(C2(C(=O)NCC3CC(n4cc(C(CC)(C)O)nn4)C3)CC2)ccc(Cl)cc1 Cc1c(F)cc(C(=O)NCC2CCN(C(=O)Nc3cccc(Cl)c3)CC2)cc1F C1(C2(NC(C(N)=O)=O)CC2)CCCN1C(c1c[nH]cc1Br)=O C1(C(N2CCC(N(C(C=Cc3cn(C)nc3)=O)CCO)C2)=O)CN2CCN1CC2 C1(NC(N(CC(O)CF)C)=O)CCCc2ccccc2C1 c1(CC)cc(=NCC23CC2CN(C(c2cncc(Cl)n2)=O)C3)[nH]c(C)n1 C1(C(=O)NC(COC)C(=O)OC)CN(C(C(=O)CCOCCOC)=O)CC1C1CC1 C(CN=C(NCc1nncn1CSC)N1CCC2(CCC(C)CC2)C1)OCC=C n1(C(C(N2CCCC(CN(C(CC=CC=C)=O)C)C2)=O)C)c(C)cc(O)cc1=O c1(OCC)ccc(CCC(N2CCN(C(=O)CC3CCC3C3CC3)CC2)=O)cc1 C(=O)(C1=NOC2(CCOC2)C1)NC1CC(NC(C(C)(C2(C)CC2)OC)=O)C1 C#CCC(CC(=O)N1CCC(O)(CC(C)C)C1)NC(C1CC2CC1CC2O)=O CC1(C)CN(CC23CCC2CCN3)CCS1=O c1(SC)ncc(C(=O)N(CCCNC(C2(CF)CCC2)=O)C2CC2)s1 c1(OC)ccc(F)c(-c2nc(Cn3ccnc3)nn2CC(=O)NOC)c1 C1(C(N2CCC(CCCC)C2)=O)CC2(CCN1C(=O)CCCNC(N)=O)CC2 c1(C(CN(C)C(CC(C)(C)C)=O)N(c2nnc(C3CC3)s2)C(C)C)ccccc1 C(CN=c1nc(C#N)cc(C)[nH]1)N(C(=O)CSS(C)(=O)=O)CCOC C1(OC)CC(C)CN(CCOc2c(C)n[nH]c2C)C1.C1(=O)CCC(=O)NCCN1 Cc1csnc1C(=O)N(CCN(C(=O)COC1CCC1)CC1CC1)CC N1(C(C(C2CCCCC2)C)=O)CCSCC1C(=O)NCCCCCN(C)C Cc1cc(C(N2CCC(O)(C(C)NC(c3ccc(Br)cc3)=O)C2)=O)c(C)n1C C(=O)(CC(C)(C)NC(C1CC(C)CCO1)=O)NC(CC)C1CCC1 C1(CNC(C(C2CCCC2)OC)=O)CC2CCC(C1)N2C(=O)CC(=O)NC1CC1 C1(C(F)(F)F)(C(=O)NCCCCNC(CCN(C(CC)CC)C)=O)CC=CCO1 c1(OC)cccc(Cl)c1CC(=O)NCC1(O)CN(C(=O)C(C)OCCN(C)C)C1 N1(C(CCC=C)=O)CCC(N(C)C(c2c[nH]c(C#N)c2)=O)CC1 N(C(=NCc1nc(C)c(C)s1)NCc1nc(C2CCC2)no1)C(CC)CC C(C(CC(=O)N1CC(c2ccccn2)C1)NC(=O)C(CO)N(C)C)N(C)C C1(CC)CCC(NC(=O)NC(C)CCSC)CN1C(=O)OC(C)(C)C Cc1cc(=NC(C)c2cc(F)ccc2F)[nH]c(=NCCN(C2CC2)C2CC2)[nH]1 C1(CC)C(N)CCCN1C(C1CCN1c1ccccc1)=O C(=O)(CC(C)C(F)(F)F)N1CCC(C=CC(=O)NCC(C)CC2CC2)CC1 C1(C(N(CCNC(CCN(CCC)C(=O)OC(C)(C)C)=O)C(C)C)=O)CCSC1C C1(N(C(CC(C)c2cccnc2)=O)CCF)CCCN(C(c2cncc(N)n2)=O)C1 Cc1ccc(NC(c2ccccc2Br)c2nnnn2C(C)(C)C)c(Cl)c1 C(C)(C(CC(=O)N1CC(c2n[nH]c(C)n2)C1)NC(=O)Cc1ccc[nH]1)OC N1(C(Cc2n(C(C)C)cnn2)=O)CC(CNC(=O)C2CC2)C(C)C1 CC1CC(CCNC(=O)Cn2c(SCCC)nnn2)CCN1C(=O)CNS(N)(=O)=O.C1CC1 CCC1=NOC(CC(=O)NC(C)CCCCNC(c2cnn(CCO)c2N)=O)C1 C1(NC(=O)C2=C(Cl)CC2)CS(=O)(=O)CC1NC(c1cscc1Cl)=O c1(C(=O)NC(C2CN(C(CCn3c(C)nc(C)n3)=O)C2)C)cc(C#N)cn1C c1(CNC(=O)CSC(F)(F)F)ccc(CCNC(c2cc(C(F)F)no2)=O)cc1 N1(CC)CC(NC(C23CC(CN2C(C2CC2=C)=O)C3)=O)CCC1=O CC1(C)CC(C(N2C3CCC2C(CNC(C2CC2(C)Br)=O)C3)=O)CC(C)(C)C1 c1(CCNCC(C)Oc2cccc(F)c2)nccc(N2CC3CC3C2)n1 Cc1nn(C)c(Cl)c1C=CC(N1CCCC(N(C(=O)C(C)CC(F)(F)F)C)C1)=O C1(C)(C(=O)NCC2N(C(C(Br)=C(C)C)=O)CCCC2C)COC(C)(C)OC1 n1(CCC(=O)NC2C(NC(CSCC=C)=O)CCCC2)cc([N+](=O)[O-])cn1 N1(C(CC2CC(C(C)=O)C2(C)C)=O)CCCC(CO)(CNC(=O)CC(C)CC)C1 C(=O)(C(C)(C)C(C)(C)N(C)C)N1CC(CCNC(C(C)NC(N)=O)=O)OCC1 CC1(CNC(c2c(F)cncc2Cl)=O)CCCN(C(=O)CCc2cncnc2)C1 Cc1nc(C(=O)NC2CC(O)(CNC(=O)Cc3ccsc3)C2)ccc1Br c1(C(=O)NCC2C(C(=O)NC3C(C(C)C)C3)CCCC2)cncn(C)c1=O C12(NC(c3ccncc3Br)=O)CCN(C(c3cnn(C4CC4)c3)=O)CCC1C2 N1(C(CC2(CSC)CC2)=O)CC(C(N2CCCC2CC2CC2)=O)C(F)(F)C1 CC1C(NC(=O)C(C)(C)N(C)C)CCCN1C(=O)CCCc1cccc(Cl)c1F N1(C(Cn2cc(Cn3ncc(C)c3)nn2)=O)CCc2cc(F)cc(Br)c2C1 CCS(=O)(=O)c1ccc(CCC(N2CC3CC2C(O)C3O)=O)cc1 CS(=O)C1CC(N(c2ccccc2)CC(=O)NCC2(N)CCCCC2)C1 c1(C(=O)NCC2(NC(=O)C=CCF)C(C)CCCC2)cc2nccnc2cc1F CC(C)C(CCN(C)C(C1(N(C)C)CCCC1)=O)NC(=O)CNC=O c1(=O)nc2nc([nH]1)NN2.c1(OC(C)C)cccc(OCCCO)c1 c1(C(N(Cc2ccc(C)nc2)CC2CCCO2)=O)ccc2c(c1)NC(=O)C(C)O2 c1(SCCNC(N2CC(c3cn[nH]c3)C2)=O)ccc(Cl)c(Cl)c1 c12cc(on1)NC2=O.C1(C(N(CC=CC(=O)OC)C)=O)(CC2CC2)CCC1 C=CC1(C(=O)NCCSCCO)CCN(C(c2ocnc2C)=O)CC1 C(=O)(CCCCCF)NCC1C(NC(CNC(CC(N)=O)=O)=O)C1 N1(C(c2ccc(CC)o2)=O)CCC(CC(=O)NC2COCCC2O)C1(C)C C1(C(=O)NCCC(C)NC(CNC(=O)OC)=O)CCCc2ccccc2C1 Cc1cc(C#N)cnc1C(=O)NCC(CNC(=O)CCOCCN(C)C)C(F)(F)F Cc1ccc(S(N)(=O)=O)c(NC(=O)NCC(C)C(C)(F)F)c1F C1(CCOC)CCCN(C(c2nc(Br)sc2C)C(=O)NCCC2CC2)C1 Cn1cnc2c1CCC1C2CCCN1C(=O)Cn1cc(CN2CC3CC3C2)nn1 c1(C(=O)NCC2CC(C)N(C(=O)C3=C(Cl)CC3)C2)ccc2nc[nH]c2c1F c1(C(N2C(CNC(c3cccc(Cl)c3)=O)CC2)=O)cnc2c(F)ccc(F)c2c1 CCC(C(=O)OC)C(=O)NC1CCCN(C(C2(C3(O)CCC3)CC2)=O)CC1 C1(CC)CCC(C(=O)NCCOC2CCN(C(=O)Cc3ccc(Cl)cc3)C2)CC1 N1(C(=O)NC(C2CCOC(C)(C)C2)C)CC(CN(C)C)c2ccccc21 C1(NC(=O)CNC(=O)C(F)(F)F)CN(C(=O)CCc2nc(Cl)cs2)C2(CCC2)C1 C1(NC(c2snc(O)c2Cl)=O)Cc2ccccc2C1O C(C(CC(F)(F)F)NC(c1csc(C(C)=O)c1)=O)NC(C=CCC)=O CC(C)C(CCN(C(=O)CCN1CCCS1(=O)=O)C)NC(C1CC1C(F)F)=O Cc1ncc(CC(=O)N(CC(O)CN(C)C(c2coc(C3CCCC3)n2)=O)C)s1 c1(C(=O)NC2C(C)N(C(C3CC(O)C3)=O)CCC2)ccc2c(c1)NC(=O)C2 CC1CCC(C(N)=O)CN1C(=O)C(O)C1CN(C(=O)Cc2cn[nH]c2)C1 N1(C(c2c(C)c[nH]c2)=O)CCCCCCC1C(=O)NOCC1(C)CC2CCC1C2 c1(C(=O)Nc2nc(Cl)ccc2I)c[nH]c2ccc(-c3ccc4cc[nH]c4c3)cc12 N1(C(C(C)CF)=O)CCn2c(CNC(c3scnc3C(F)(F)F)=O)nnc2C1 C1(C(=O)NC2CC(NC(=O)CC(F)(F)F)C2)CCn2ncnc2C1 c1(C(N2CC(C)N(C(=O)Cc3cc(C4CC4)no3)CC2)=O)cc(F)c(F)cc1F CC(CC(C)(F)F)C(=O)NC1CCCC1CNC(c1cc(Cl)cs1)=O N12CCOCC1CC1(CC1)CC(C)(C)CCC1CCC(CCOC)CNC(=O)C21 C1(NC(c2c(C(C)C)nns2)=O)CN(C(C2CC3CCC2O3)=O)C(C)(C)C1 c1(C(=O)NCC(=O)NC)sccc1.C1(C(=O)NCCCSC(F)F)CCCCO1 C1(NC(=O)COCC2CCC2)CN(C(=O)CCCCCF)CC(F)(F)C1 CC1CCCC(CC(=O)N(C)CCN(C(c2nc(C3CC3)cs2)=O)C(C)C)C1 Cc1ccc(Cl)cc1CC(=O)NCC(O)CN(C)C(c1cnn(C2CC2)c1C)=O C1(C)(CC(=O)N(C(C)CNC(=O)CCC2CC2)C)CCCO1 Cn1cnnc1C1(NC(C2(NC(=O)CC34CCCC3C4)CCC2)=O)CC1 C(c1sc2ccccc2c1Cl)=CC(=O)NC1(C)CN(C(C(COC)(F)F)=O)C1 c1(C(=O)NC2CC3CC(NC(c4c(C)occ4)=O)CC32)cnc2cc[nH]c2c1 N(C1COc2ccc(F)cc21)C(=O)NC(C1CCOCC1)C#C Nc1cncc(C(=O)NCC2(F)CCC(CNC(C3CC(O)C3)=O)C2)c1 c1(C(N(CCn2cc(C(=O)NC(CC=C)C)nn2)C)=O)cc(CO)ccn1 c1(C(=O)OC)nc(N2CCC(CO)(CNC(=O)CC3CCC(=O)N3C)C2)sc1C c1(C(N2C(C)CN(c3cccc(F)c3)CC2)=O)cc2c(nc1O)CCC(F)(F)C2 C(CC(C(=O)NC(C)CC1CCN(C(=O)CC(C)(C)F)CC1)NC(C)=O)OC C(=O)(C(CCF)N(C)C=O)NC(CN(C(COC(C)C)=O)C)C.C(C)(C)(C)O S(=O)(=O)(c1ccc(N(CC(C)O)C)cc1Br)NCc1c(C)nc(C)s1 C1(CC(=O)N(C2CCN(C(=O)Cc3csc(NS(C)(=O)=O)n3)C2)C)CCCSC1 c1(C(N2C3CN(C(C4CC4F)=O)CC32)=O)nccc(Br)c1O Cc1ccnc(N(CCCCCCCO)C(CN(C)C2CC2)=O)c1N CN1CC(C)(C)CC1C(N1CCC(Nc2ccc(C#N)cn2)C1)=O N1(C(c2ccc(C)cn2)=O)CCOC2(CCN(C(=O)C#CC3(C)CCCO3)C2)C1 O=C1CCc2cc(C(N3CC(NC(=O)C(O)C4CC4)C(C(F)F)C3)=O)cnc2N1 C=C(C)C(CC(=O)N(C)CC1(O)CN(C(=O)CCC=C(C)C)C1)OCC C1(C(=O)NCC(CC)NC(C2(SC)CCC2)=O)CCC12CCC2 C1(NC(c2c(SCC)cncc2)=O)COC2CN(C(=O)CCC(=O)OC)CC12 C(=O)(CC(C)C(C)(C)C)N1C(CNC(c2c(Br)c(C)n(C)n2)=O)CC1 C(=O)(C1=C(Cl)CCCC1)NC(CNC(CC(C=C)C)=O)(C)CC(C)C c1(SCCOC(C(=O)NC2CC(NC(CCN(CCC)C)=O)C2)C)cccnc1 C(=O)(C#CC1CCC(=O)CC1)NCC1CN(C(c2nc(CC)oc2)=O)C(C)C1 c1(C(N(C2CCCCC2)CCCNC(CCCSC)=O)=O)cnc[nH]c1=N C1(NC(C2(NC(c3nocc3Cl)=O)C(C)CCC2)=O)CN2CCC1(C)CC2 c1(CC)nc(C)c(C(=O)N(C)CCOCCNC(C2(CO)CC2)=O)s1 CC1SCCCC1C(=O)NCCOC(C)(C)CNC(c1cc(C2CCC2)[nH]n1)=O N1(C(CC2C(=O)NC(=N)S2)=O)CC(F)(F)CC1CNC(C1(C(F)(F)F)CCC1)=O C1(C(N2CCC(C(=O)OC)(CO)C2)=O)CCN(C(=O)c2cc(C)co2)O1 c1(C(CC)NC(C2(NC(=O)C(n3cc(C)cn3)C)CCSC2)=O)cnn(C)c1 C1(C(=O)NCC2(F)CCC(NC(C3SCCS3)=O)C2)COC2(CCC2)C1 CC(C)(F)CCC(=O)N1CCC(n2cc(CNC(=O)CN3CCOCC3)nn2)C1 N1(C(CCSCCCC)=O)CC(NC(=O)COC(F)(F)F)C2(CCC2)C1.C(=O)OC C12(CNC(C(C=C)(C)C)=O)CC(C1)C(NC(C13C=CC(CC1)C3)=O)CO2 C1(CC(=O)Nc2c(NC(CCSC)=O)cccc2)CC2CCC(C1)N2CC#N C1(C(=O)NC(C2CCN(C(=O)CC3CC3)CC2)C)CC(C)(C)OC1(C)C C(CC(=O)O)(C(F)F)NC(CC1CC(C)(C)OC1)=O c1(C(=O)NC2CC(C)(C)N(C(=O)Cn3cnnc3O)C2)cnc2c(c1)OCCN2 C12(CC(=O)NCCc3cccs3)CCC1CN(C(=O)Cn1ccnn1)C2 C(=O)(CCC(C)(F)F)NCCOCCNC(C(c1cncc(OCC)c1)(F)F)=O CC(C)(CS(N)(=O)=O)C(=O)NCC1CCCC(NC(c2ccc(O)nc2Cl)=O)C1 C(=O)(CS(=O)(=O)C1CC1)N(C1CCC(NC(=O)CP(C)(C)=O)C1)C CC1(C)CN(C(c2coc(CNC(c3cnccn3)=O)c2)=O)CC(=O)N1 C1(C2(C)OCCO2)NC(=O)N(CC(O)COc2ccccc2Cl)C1=O c1(C(=O)NCC2CC(OC)CN2C(c2nnc(C)s2)=O)c(F)cc(Cl)cc1Cl C(=O)(CCCC(F)(F)F)NC1CCC(F)(CNC(C(C)C2CC2)=O)C1 C12(NC(C(c3ccc(Br)cc3)C)=O)CCCC(NC(=O)NC(C)(C)C)(C1)C2 c1(OC)ccccc1C(C)C(=O)NCC(CO)NC(c1cnc(C2CCC2)s1)=O c1(CNC(N2CC3CC2CC3O)=O)ccc2c(c1Cl)OCCO2 C1(C(=O)NC2CCN(C(C(C)NC(C)=O)=O)CC2(C)C)CCn2c(O)nnc2C1 c1(NC2CCN(S(CCC)(=O)=O)CC2)cnc(F)c(C)c1 C1(CC)CN(C(=O)C=Cc2cc[nH]n2)CC1C(=O)NC(C1CCCC1O)C C(N=c1nn[nH]n1Cc1ccccc1)C1(O)CN(C(C(C)O)=O)C1 [N-]=[N+]=NCCCCCC(=O)NCC1(NC(C2CC3(CCCC3)CO2)=O)CC1 CCCC(C)(O)CC(=O)N1CCC(C(=O)NCC2CC=CCC2C)C1 c1(CC=C)ccccc1C(=O)NCC(C(C)C)NC(=O)C=CCCC(C)C c1(C(N2CC(OC)(CNC(=O)CN3CC4CC4C3)C2)=O)coc(C#C)c1.S(C)(=O)(=O)N c1(Cn2c(N3CCC(F)(CC)C3)nnn2)ccc(Br)c(C)c1 c1(C(=O)NC(C2COCCN2CCNCCCCCl)=O)cccc2ccoc12 S(=O)(=O)(c1cc(Cl)ccc1F)N1C(C(=O)Nc2c(Br)cc(C)c(F)c2)CCC1 Cc1ccc2oc(C(N3CC(CNC(c4oncc4C)=O)C(C)C3)=O)c(C)c2c1 C1(NC(C(CC)C)=O)CCCN(C(c2cc(-c3c(C)noc3C)on2)=O)C1 C(N(C)N1CCN(c2cccc(C(N)=O)c2)CC1CO)C1CCN(C(=O)OC)C1 N1(C(c2cnc(OC)c(Cl)c2)=O)CCN(C(c2cc(N)cc(F)c2)=O)CC(O)C1 O=S1(=O)CCN2C(C1)NC(=O)C2c1ccc2nsnc2c1.C1(CSC)CC1 N1(C(c2cc(CCOC)on2)=O)CC2CCN(C(=O)C(F)(F)C(F)(F)F)CC12 N1(C2(NC(=O)Cn3cccn3)CC2)CC(C(N2CCC(OCC)C2)=O)CC1=O N1(CC2(C)CCCC(=O)N2)CCc2ccc(O)cc2C1C Cc1csc2c(N3CCCC3c3ncc(-c4cc(Cl)ccc4Cl)[nH]3)ncnc12 Cc1ccc(C(C)C(O)C(=O)NCC#CCNC(c2cnc(C(C)C)[nH]2)=O)cc1 N1(C(C(C)CO)=O)CCCC12CCN(C(c1cccc(Cl)c1N)=O)CC2 C(c1ccncc1)=CC(=O)NC(C)CCNC(=O)Cc1ccn(C(F)F)n1 Cc1cc(C(N2CSCC2C(=O)NC(C)CCC(C)C)=O)ncc1F C1(NC(C(C)N2CCCC2)=O)CN(C(=O)CCc2cscn2)CC12CCCC2 C1(CN(CC(F)(F)F)C(C=CC(C)C)=O)CN(C(=O)CC(C)F)CC1n1cccn1 Cc1c[nH]c(C(N2CCC(C(C)CNC(=O)C(C)C3(O)CCC3)CC2)=O)c1C C1(CC#C)(C(N2CCOC(CC3CC3)C2)=O)CCN(C(=O)Cc2ncco2)C1 Cc1csc(=O)n1CCC(N1CCCC1C(C)(C)NC(=O)C(O)C1CCCC1)=O c1(CC(=O)NCCC2N(C(C3C(=C)CC3)=O)CCCC2)ccc(OC)cc1Cl C(CC(C(C)(C)C)NC(c1cc(C)on1)=O)N(C(C(COC)(F)F)=O)C N1(CC=CC(C)(C)C)CC2CC1CN2C(C1(C(=O)CCN)CC1)=O C(=O)(CC(F)(F)C(F)F)N1CCCC(C(N2CCCC(CC)C2)=O)C1 N1(C(C=CCCC)=O)C2CCC1CC(CCNC(c1c([N+](=O)[O-])cnn1C)=O)C2 C1(NC(c2cc(CC)on2)=O)(COC)CCN(C(c2ocnc2C(F)F)=O)CC1 C(=O)(C(C)(F)C(F)(F)F)NCC1(OCC)CN(C(C2CCC(F)(F)C2)=O)C1 C(CC(=O)N(C)CCC1CCCC1)(C(F)F)NC(c1c(C)coc1)=O Cc1cc(S(C)(=O)=O)ccc1C(N1CCN(C(=O)CC(O)C(C)C)CC1)=O N1(C(c2nc(CNC(CC(C)OC)=O)oc2)=O)Cc2cccc(F)c2C1 c1(C(C(=O)N(CCC)CCNC(C2CC2(C)C(=O)OC)=O)C)ccc(C#N)cc1 C12CCCC(C1)C(=O)N1CCCC(C1)CNC(=O)C2.C1(=CC)CNC(=O)O1 N12CC(C3CC13)CC2=O.c1(CCC(=O)N)nccn1C.C(C(=O)NC)N(C)C N1(C(C(C)C(F)(F)F)=O)CC2(CCC(CNC(=O)C(F)(F)C(F)F)O2)C1 Cc1nn2cc(C(=O)NCCCN(C(C34CCCCC3C4)=O)C3CC3)nc2s1 N1(C(CC(c2cccs2)NC(C=C(CC)CC)=O)=O)CC(CNC(C)=O)CC1(C)C c1(C2(NC(C(C3CC34CCC4)N3CCC(NC=O)C3)=O)CC2)ccc(Cl)c(F)c1 CCCC(C)(O)CC(=O)NC1CCOC1C(=O)NCC1CCC(CC)O1 C1(C(=O)NCc2oc(C(=O)Nc3cnc(OCC)nc3)c(C)n2)CC2(CC2)C(=O)O1 c1(OC)ccc(CNC(=S)NC(C(=O)NC)c2cscn2)cc1 c1(OC)ccc(C2CCN(C(=O)C(=O)NCCn3ccnn3)C(C)C2)cc1F C1(NC(CCCOC)=O)C2COCC1CN(C(c1nn(C)c3c1CCCC3)=O)C2 C1(NC(c2nc(C)sc2)=O)CCCN(C(C2NC(=O)C3CC23)=O)C1C C12(C(N(C)CC3N(C(C4OCC(C)C4)=O)CCC3)=O)COCC(C1)OC2 CCC(C(=O)NCC(C)(O)CNC(=O)CNc1ncccn1)SC C(=O)(C(CCC1CC1)NC(c1scc(C)c1C)=O)NCC(CC)(C)OC c1(C(N2C(C)C(NC(C3CS(=O)C3)=O)CCC2)=O)ncc2n1CCCC2 c1(C(=O)NC2CCN(C(CC3CC(=O)OC3)=O)C23CC3)cc2cccnc2o1 CON(Cc1ccc(CO)cc1)C(=O)C(COCCO)NC(=O)CCN(C)C N(C1c2ccccc2CC12CC2)C(N1CC2CC1CC2(F)F)=O c1(C(=O)NCc2cn(CC(C)NC(c3ccoc3)=O)nn2)nn(C)c2c1CCC2 C1(C(=O)NC2CN(C(=O)Cc3ccoc3)CCC2CO)CCC(=C(F)F)CC1 c1(CCC)ccc(Cc2nnnn2CC(F)F)c(NCCCCSC)n1.C(C)(C)C c1(C(N(C2CCN(C(c3ccc(C(F)(F)F)nn3)=O)C2)C)=O)c(C#N)cnn1C c1(C(=O)NC2(CNC(c3cc[nH]c3)=O)CCC2)ccc2c(c1)NS(=O)(=O)C2 C#Cc1ccc(C(=O)NCC2(O)CCCN(C(=O)C(F)CC3CCC3)C2)nc1 c1(C(=O)NCC(C2CCCCCC2)N(C(=O)C2=CCCC2)C)ccc(=O)n(O)c1 c1(CC)ccc(C(=O)NCCCCNC(c2ccn(C)n2)=O)cc1C#N CCCCCC(C1CC1)NC(C1CCCCC1CNC(C1(CC)CCOC1)=O)=O Cc1cncc(C(=O)NC2CC(NC(=O)CC3CCNC3=O)C2)n1 C(CSC)(C(=O)N(CCNC(=O)CN1CCC1C)Cc1ccccc1)OC c1(NC(C(=O)Nc2c(C)nn(-c3ccc(F)cc3)c2C)=O)ccc2ncnn2c1 c1(OC(C(C)C)C)ccccc1C(=O)N(C(C)C(=O)N1CCCC1)C1CC1 C1(C(N2CC(C(C)(C)O)(CNC(c3n(CC)cc(Cl)c3)=O)C2)=O)CC12CCSCC2 c1(OCCC(C)C)ccc([N+](=O)[O-])c(NC(=O)C(=O)NCC2CCN(C)C2)c1 C=CCC(C(=O)N(C)Cc1cccc(CNC(C2CNC(=O)C2)=O)c1)OC C(C)(C(C(=O)NC(C)CN(C)C(c1sccc1C#N)=O)N(C)C)OC C1(CCC)(C(=O)NCC(O)CN(C(=O)C(=C2CCCCC2)F)C)CC12CCC2 N1(C(CC2CCN(C(C(CC)COC)=O)CC2)=O)CCC(OC)CC1C C(=O)(CCCCCC(C)(C)C)NC1CN(C(c2cc(OC)no2)=O)CC1C1CC1 CS(=O)(=O)CCCC(=O)N1CCC(=CCNC(c2ccc(F)c(Cl)n2)=O)CC1 CC(CO)(C(=O)NCCC(O)C(F)F)NC(=O)CCOC1CCC1 c1(C(N2CC(NC(CC(C(C)C)C)=O)C(C)C2)=O)nn(C)cc1S(N)(=O)=O c1(C(=O)OC)ncc(OC)s1.C12C(C1(C)C)C(=O)NC2.N12C(CC1C)C2=O CC1CCn2ncc(C(=O)NCCC3(NC(=O)C=C(Cl)Cl)CCCC3)c2C1 c1(CNC(C(=O)Nc2nc(SC)sc2)=O)ccc(C(C)=O)cc1[N+](=O)[O-] CC(CCN(C)C)C(=O)NC1CC(O)C1CC(=O)NCc1cccc(O)n1 CC1(C)CN(C(=O)CC2C=CCC2)CC1NC(=O)CCCC(F)F CCC(C)C(C(=O)NCc1nn(C)cc1C)N(C(=O)CCc1nncs1)C Cc1cc2occ(C(=O)N(C3CCN(C(=O)C(C)C(C)O)CC3)C)c2cc1C CC(C(C)(C)C(=O)NC(CN1CCCC1)CO)NC(=O)CCc1ccnn1C Cn1ncc(C#N)c1C(N1CCC(F)(C(=O)NCC2COCCO2)C1)=O c1(CNCC2CC(NC(c3ccc(C4CC4)cc3)=O)C2)ccncc1F C#Cc1ccc(C(N2CCCC(N(C(c3cc(Cl)ns3)=O)CC)C2)=O)c(C)c1 C(=O)(C1=CC=NC(=O)C1)N1C(C)(C(N(CC(F)(F)F)C)=O)CC1 c1(-c2ccn(CCCOC)n2)ccc(C(=O)NCc2cccnc2)c2[nH]ccc12 C1(NC(=O)CCCn2cncn2)CCC2CCN(C(C34CC3CCC4(F)F)=O)C12 C(=O)(CCN=c1[nH]ccs1)N1CCC(NC(c2c(C)snn2)=O)C(F)C1 C12(CC(=O)NCCNC(CCCC)=O)CCC1CN(C(=O)Cn1ncn(C)c1=O)C2 c1(C(N2CC(CNC(=O)CCC3CCCO3)OCC2)=O)cc2c(Cl)nccc2o1 CC(C)CCCC(C)C(=O)NCC1CCNCC1O CC1CN(C(=O)C(c2cccnc2Br)C)CCCN1C(=O)Cc1ccccc1 C12CC3CC3N1C2=O.C12(CNC(CC3(C)CC3)=O)CCC(CC1)O2 Cc1ccc(OC(C)C(=O)NC(C)CNC(=O)C=Cc2cncc(O)c2)c(C)c1 c1(C2C(N(CC(N3CCC(C(C)(C)NC(=O)C4CC4)C3)=O)C)C2)ccc(Br)cc1 CCCCCC(F)C(=O)N1CC=C(C(=O)NCC(C2CC2)SC)C1 c1(C(=O)NCCCCCCNC(C2CC3CC3C2)=O)cc(F)cc2ccncc12 C1(CNC(NC2CCN(CCC)C2)=NCc2cc(C)on2)C(F)(F)C12CCCC2 CCC(C)CCC(O)CC(=O)NCC1CC(NC(c2cn(C)nc2SC)=O)C1 C1(=CC(N2C(CNC(=O)CC(F)(F)F)CCC(C)C2)=O)C2CC3CC(C2)CC1C3 C1(NC(C(C)CC(F)F)=O)CCC2(CC1)CN(C(=O)Cc1cnccn1)CCO2 c1(C(C)NC(C(CC)N(C(=O)C(CC)OC)C)=O)ccnc(F)c1 C1(C(=O)NCC2CN(C(c3nc(C)sc3)=O)C2)CSc2ccccc2O1 c1(C(=O)NC2CC(CNC(CC(C=C)C)=O)C2)ccc2ncccc2n1 CN1CCC=C(CNC(C23CCC(NC(=O)CC4CCCOC4)(CC2)C3)=O)C1 N1(C(COCCCC)=O)CCC(C2CC2)(CNC(=O)C(C)(F)C(C)(C)F)C1 c1(C(C(N2CC(NC(CCCC)=O)C(C)C2)=O)C)ccc(C)c(Br)c1 c1(C(=O)NC2C(CNC(CCS(C)=O)=O)C2)cc2cccnc2cc1F C(=O)(C1=C(Cl)CCOC1)NCC(CN(C(C(C)SC(C)C)=O)C)C C1(N(C(c2c(C)cccc2)=O)C)CN(C(=O)C(c2c(C)n[nH]c2C)C)CC12CC2 c1(CN(C(=O)CNC(C2CC(OC)C2)=O)CCOC)c[nH]c2ccncc12 c1(N2C(C)CNC(=O)C2)nc2ccccc2c(=NCc2ccc(F)c(C(N)=O)c2)[nH]1 N1(C(C2(CF)CC2)=O)CCC(C(C)(C)CNC(C2(C)CC2Br)=O)CC1 c1(C(=O)OC)cc(Br)cc(C)c1NC(C1CCC(NCc2c[nH]c(C#N)c2)C1)=O C1(N(C(CC)=O)C)CS(=O)(=O)C12CCN(C(c1nc(O)sc1C)=O)CC2 C1(NC(c2c(CC)noc2)=O)(CO)CCN(C(c2ccc(O)nc2)=O)CC1 c1(CC)ccnc(C(N2CCCC(N(C(=O)Cc3csnc3C)C)C2)=O)c1 C#Cc1cc(C(=O)N(C(C)CNC(C2CC2CN(C)C)=O)C)cc(F)c1 Cc1ncc(-c2nnc(N3CCC(N4CCC4C(N)=O)CC3)n2C)cc1C#N N12CCCN(CCC1)C(=O)C(OC)C(=O)N1CCCC1C2=O.C(=O)(OC)OC C1(N(C)C(c2ncc[nH]2)=O)CCCC(C(=O)NCCc2ncc[nH]2)C1 C1(C(=O)NC(C)CCCNC(c2cnn(C)c2C(F)(F)F)=O)CCC=CCCC1 C=CC1(CC(=O)NCc2nnc(CC)o2)CN(C(=O)C(c2cccn2C)=O)C1 N(C(=NCc1nc(C(C)O)n[nH]1)N1CC2C(CF)C2C1)Cc1cccc(CC)c1 c1(CC(CN(C)C(C2COC2)=O)NC(C(C)OCCC(C)C)=O)ccccc1 C12(C(=O)NC3C(CNC(C4(C(C)C)CCCC4)=O)CC3)CC1CNC2=O C1(CN(C(=O)C=CC2CCCC2)C)CCCN(C(=O)C2=C(Cl)CC2)C1 CN1CCc2cc(C(=O)NC3(C)CCCN(CCSC4CCCO4)C3)ccc2C1 C(C(=O)NOCCCOC(C)C(=O)NCC1CC1)(C1CC=CC1)OCC C(=O)(CCCS(C)(=O)=O)N1C(CNC(Cc2cccc(C)c2)=O)CC(F)(F)C1 C12(NC(CC3CC(SC)C3)=O)CC(CNC(c3cc(C)nn3C)=O)(C1)OC2C N1(C(C2OCCN(C(C)C)C2)=O)CCC2CCC(C1)N2C(c1cnon1)=O C#Cc1ccc(OCC(=O)N(CCCNC(C2CCN2CC)=O)C(C)C)cc1 c1(C(N2CCCN(c3c(C)cnc(C#N)n3)CC2)=O)nccc2c(C)cccc12 Cc1cnn(CC(=O)N(CC(C)C)CCO)c1Br O=CCCCC(=O)N1CCOCC1Cc1cncs1.c1(CC(=O)NC)ccsc1 N1(C(Cn2c(C(F)F)cc(C)n2)=O)CCC(C)C(CN(c2ccccc2)C)C1 c1(C(N2CC(O)(CNC(C(CC)N(C)C)=O)C2)=O)c(C)coc1C CC1(C)CC(=O)OC1NC(N1CC(N2CCN(CC(=O)OC(C)(C)C)CC2)C1)=O Cc1cc(NC(C2(S(C)(=O)=O)CC2)=O)ccc1NC(C1CC1(F)Cl)=O Cc1ccc(C(=O)NCC2C3CN(Cc4nc(C(C)C)no4)CC23)cc1F C1(O)(C(=O)NCC2CCC2NC(c2ccc(OC)nc2)=O)CN2CCC1CC2 C1(C(N(C2CCCN(C(=O)COc3ccsc3)C2)C)=O)CCCCC1(F)F N1(C(C(C)(C2CCC2)NC(c2c(CC)nco2)=O)=O)CC(C)CC(O)C1 c1(CCN(C)C)cn2c(n1)CCCC2.n12cc(nn1)C1CC1C(=O)CC2 Cc1nc(C(F)(F)F)sc1C(=O)NCCN(C(c1coc(C(F)(F)F)n1)=O)C(C)C C1(C)(NC(CCC(C)NC(=O)CCC23CC(C2)C3)=O)CCCC1(F)F c1(CCC(=O)OCc2c(C)ccs2)ccc2[nH]ccc2c1.c12ccccc1NC2 N1(C(CCC(=O)NC2CC2)=O)CCc2c(Cl)cc(F)cc2C1 c1(C(N2C3C(NC(C4(OCC)CCCCC4)=O)C(C3)C2)=O)nc(C)n(C)c1C c1(C(=O)NCC2(O)CCCN(C(C3CC(CCC)C3)=O)C2)ccc2c(c1)OCC2 N1(C(c2cc(C(C)=O)oc2)=O)CC(NC(=O)C(C)Sc2ncccn2)C(C)C1 C1(C(c2cccc(C(F)(F)F)c2Br)N2CC(=O)NCC2)CCCC2(CCNC2)O1 N1(C(Cc2c(C)nn(C)c2C)=O)CCN(C(C23COCC2C3)=O)C2CCC12 Cc1cnc(N2CCOC(CNC(c3nnc4n3CCC4)=O)C2)nc1O c1(C(c2n(CC)nnn2)NCC(CO)OC)cccc(OC)n1 N1(C(CNC(=O)NC)=O)CC(NC(=O)COCCOC)CCC1C c1(C(=O)NCC(=C)CCNC(=O)Cn2ncccc2=O)nc(OC)ccc1Cl C12(CO)CCCN(C1)C2=O.c1(CNC(c2ccsc2I)=O)ccccc1 C1(C(=O)NC(C(=O)NC2(C(=O)OC)CC2)CO)CC(=O)CC12CCC2 c1(C(N2CCCC(NC(C3C(C)OCC3)=O)CCC2)=O)cc(Cl)cc2c1CCC2 c1(C(=O)OCC)nn(C)cc1C(N1CC2CC2(CNC(c2coc(Cl)c2)=O)C1)=O c1(C(=O)N(CCN(C(C2(C(=O)OC)C(=C)CC2)=O)CC)C)ccc(CC=C)cc1 C1(CNC(C(COC)NC(=O)C(C)c2cccs2)=O)CC2CC1CC2O C1(NC(=O)Nc2ccoc2)Cc2ccc(O)cc2CN1C(N(C)Cc1ccco1)=O N(C1CCCc2sccc21)C(C1CCCOCC1)(c1n(C(CC)(C)C)nnn1)C C(=O)(C1=CCCN(C(c2ncn(C)c2-c2ccccc2)=O)C1)NC(C)CN(C)C Nc1cc(C(=O)NC2CC(F)CN(C(c3ccccc3)=O)C2)ccc1S(N)(=O)=O C1(C)(CNC(C(CC=CC)C)=O)CN(C(=O)Cn2cnc(C(F)(F)F)c2)CCO1 C1(C(=O)OC)CCC(CCC(=O)NCC(C)(O)CNC(=O)CC=C(C)C)CC1 C1(CC(=O)NC(C(C)C)CN(C)C)CCCCN1C(=O)CNC=O CS(=O)c1cccc(C(=O)NCC2(NC(C34CC5CC3C4C5O)=O)CCCC2)c1 C(=O)(C(F)C(C)CNC(C1(NC(C)=O)CC1)=O)NCCCCCCC c1(C(=O)NCC2N(C(C(C)n3cncn3)=O)CC=C2)cnc2c(c1)CCCO2 N1(C(C(C)CCOc2ccccc2)=O)CCn2c(-c3ccccn3)nnc2C1 CCS(=O)c1ccccc1CC(=O)N(C1CCN(C(=O)CCC(F)F)CC1)C C1(NC(c2cc(C(F)(F)F)c[nH]2)=O)CCN(C(c2ccc(O)c(I)c2)=O)CC1F N1(C(CC=C(C)C)=O)CC(N(C)C(c2ccc(NC(N)=O)cc2)=O)C2(CC2)C1 c1(C(=O)NCC(C)NC(c2coc(Cl)c2)=O)c(N)cnn1C C1(C(N2CC(NC(CC(C)F)=O)C2)=O)CCC(F)(CNC(C2CCOCC2)=O)C1 c1(C(=O)NCC(CC)NC(C2CCCC2C(N)=O)=O)cc(C(C)C)cnc1O CC1(C)CCN(C(c2sccc2C(F)F)=O)CC1CNC(=O)CC1CCC(=O)N1 C(=O)(C#CC1CCOC1)NCC(CNC(Cc1cc(C)sc1)=O)(C)C CCC(CC(F)F)C(=O)N1CCCC(n2cc(C(C)Sc3ncccn3)nn2)C1 C=CC(C)CC(=O)NC(c1ccccc1F)CNC(c1cc(N)ccn1)=O C(=O)(C1=NOC2(CCC2)C1)N1CCN(C(C2(CC=C)CC2)=O)CC1c1cn[nH]c1 c1(S)ccc(Cl)cc1.CCC(CNC(=O)COCCF)NC(=O)CC N1(C(c2c(C)n3c(s2)ncc3)=O)CCN(C(C2CC3CCC2C3)=O)C2(CCC2)C1 C=CC1CCCCN1C(=O)CC1(CNC(c2c(C)ccn2C)=O)CC1 N1(C(C2(OC)CCOCC2)=O)CC(NC(=O)CC2COC(=O)N2C)C(C)(C)C1 C1(F)(C(=O)NCC2(NC(CCN(CCCCOC)C)=O)CCC2)CCOC1C C1(C(CNC(C2(OC)CCC2)=O)O)CCN(C(=O)CC2CNC(=O)C2)CC1 C1(O)(C(=O)NC(CC)CNC(C2SCCS2)=O)CCC(C)(C)CC1 C12(C(=O)NC(CCOC)C(C)C)CC(CCO1)N(C(=O)CN1CC=CC1)C2 c1(OCCCC(=O)NC2CCC(N(C(c3c(C)coc3)=O)C)C2)ccc(F)cc1 C1(CC)C(C(=O)N(CCCO)CCO)CCN1C(=O)Cc1cncc(C)c1 C1(C(N(CCCCN(C(=O)CCc2cccnc2)C)C)=O)CCCCC12CC2 CCC(C)(C#N)C(=O)N1CCC(C(C)(C)C)(CNC(=O)C=C2CCSCC2)C1 N1(C(CCN(C(C(C)C(F)F)=O)CC2CC2)=O)CCC(O)CC(C)(C)C1 S(=O)(=O)(c1ccc2cccnc2c1)NCC1CCCC(C)(C)C1 c1(C(C)(C)C)ccccc1C(=O)NC1CC2C(NC(C3CCCSC3)=O)C2C1 C1(C(C)OC)CCN(C(=O)CC(CNC(c2cc(C)[nH]c2C)=O)OC)CC1 c1(C(CO)NC(C2(F)CCN(C(c3cccc(C)c3)=O)C2)=O)cc(C)ccc1C c1(CNCC2CCN(C(C(CC)c3ccccc3)=O)C2)c(C(F)(F)F)coc1C c1(C(=O)NCC(COC)O)cc(N)cnc1Cl C=CCC(C)(C)C(=O)N1CCCCC(CNC(C2CC3C(OC)C3C2)=O)C1 N1(C(C(C)N(C(CC=CC=C)=O)C2CC2)=O)CCCC(OCC)C1 N(C1CC(C)n2ccnc21)C(c1cc(C)ccc1F)c1n(CC)nnn1 C12(C(=O)NCCn3cnnc3)CCC(CN(C(=O)CC3CC3C3CC3)C1)C2 C(=O)(CC(C(F)(F)F)OC)N(C)CC1(O)CCN(C(c2ccc(CC)cn2)=O)C1 c1(N2CCC3(C(NC(C(CC)OC(C)=O)=O)C3)CC2)ncnc2cccc(OC)c12 c1(C(=O)NCCC(C)NC(=O)CS(N)(=O)=O)cc(Cl)c(N)c([N+](=O)[O-])c1 CC#CCCC(=O)NC(C1CCCC1)CNC(C1(C2CCCCO2)CC1)=O CC(CC(=O)c1ccccc1F)C(=O)NC1(CNC(c2ccco2)=O)CCCC1 CC(CC(C)NC(c1cnoc1CC(N)=O)=O)NC(c1cn(CC(N)=O)nn1)=O C(=O)(C1c2ccccc2C2CC1C2)N1CCC(N(C)C(C2CC23CC3)=O)C1 C1(CNC(c2c(C(=O)OCC)c[nH]n2)=O)CC2CCC(C1)N2C(C1CCOC1)=O N1(C(C(C)(C)n2cccn2)=O)C2CCCC1CC(NC(C1CCCCO1)=O)C2 C(=O)(CCC(C)OC(C)C)NC(COC)C(=O)NC(c1nncn1C)CO CC(C)(CCO)C(=O)N1CCCC(n2cc(-c3cnsc3)nn2)CC1 N1(C(CC=C)=O)CCCN(CC=CCl)CC1.C12CCCC(C1)OCC(=O)N2 C(=O)(C(C1=NOC2COCC12)N1CCN(CCCF)CC1)NCCCC CCCCCS(=O)(=O)CC(=O)NC1CCC(C)N(c2ccc(C(=O)OC)cn2)C1 CC1(C)CCN(S(=O)(=O)c2cccs2)C2CCC12 c1(C(=O)NC2CN(C(c3cnnn3-c3ccccc3)=O)C2)cc2c(s1)CCC2 C1(O)(C(N2C(C3CCN(C(C=NOC)=O)C3)CCC2)=O)Cc2ccccc2C1 c1(CNC(=O)NC2CCC(N3CCC(C)CC3)C2)cn(C)c(=O)cn1 N1(C(C2(COCC)CC2)=O)CC2C(CNC(c3nccnc3N)=O)C2C1 C12(NC(CC3(OC)CC3)=O)CCCC1N(C(c1cnns1)=O)CC2 c1(N(C2CCN(c3cc(N4CCCC4)ncn3)C2)C)ncnc2[nH]cc(I)c12 O=C(O)CCC(CN(C1CC1)Cc1ccc(Br)cc1Cl)C(=O)O N1(C(C(CC=C)CC)=O)CC2CC1CCC2NC(C1(CC)CCCO1)=O c1(C(C)C)ncncc1NC(=O)C(C)NC(=O)CC(C)n1cccn1 C1(C(=O)NC2C3CC(NC(C4OCCN(C(C)C)C4)=O)CC32)CC2CCCCC12 C(C1Cc2ccccc21)N(C(=O)C(N1CCC(=CC(F)(F)F)CC1)=O)C1CC1 N1(C(COCC)=O)CC(CNC(C2(C(F)(F)F)CCC(=O)NC2)=O)CCC1(C)C C1(CN(C(=O)CS(=O)(=O)NC2CC2)CC)CCCCN1C(c1cnnn1CC)=O CCC(CC)CC(=O)N1CC(CNC(C2(S(N)(=O)=O)CCC2)=O)(OC)C1 Cc1c(Cl)ccnc1C(=O)NCCN(C(=O)CCCC(c1ccccc1)C)C1CC1 C1(NC(C=CCC(C)(C)NC(C(CSCC)O)=O)=O)CCOC(C)(CC)C1 C(=O)(C(C)C(O)CC)NC1(C)CC(NC(c2cc(CC)n(C)n2)=O)C1 C1(NC(C2(OC)CCSC2)=O)CC2CCC1N2C(=O)CCc1ccc(O)nn1 N1(C(CNC(=O)NC)=O)CCCC2(CC(NC(C3CC3(Cl)C(F)F)=O)C2)C1 C12CCC(CC3CC3)N1C(=O)C1CC1NC2=O.c1(CN(C)C)cc(O)cs1.C(C)(C)(C)C Cc1cc(F)c(NC(N2CCOCC2CC(=O)NCC(C)(O)C(F)(F)F)=O)cc1Br C1(COC)CCC(C)CN1C(=O)CN1CCN(C(=O)C(C)(CC)CO)CC1 c1(C(=O)NC2CCOC(CNC(=O)C(F)(F)C3CC3)C2)ccc2ncsc2c1 C1(F)(CN(C)C(C2COCOC2)=O)CCN(C(=O)COCC(C)(C)C)C1 CCCCC(C(=O)NCC(CC)N(C(=O)CNS(=O)(=O)NC)C1CC1)NC(N)=O C1(C(=O)NCCOC(CC)CC)C=CCN1C(=O)CC1C=CCCC1 c1(CC(N2CC3C(NC(C(c4cccc(Cl)c4)CC)=O)(C3)C2)=O)ccc(O)c(Cl)c1 c1(C(=O)NC(C(=O)NC(C)COC2CCOCC2)c2ccco2)c[nH]c(C#N)c1 c1(C(=O)NC(CNC(c2nc(SC)sc2)=O)C(C)(C)C)cccc2c1OCC2C N1(C(C(C)OC2CCCC2)=O)CC(NC(c2ccc(Br)o2)=O)C(O)C1 c1(C(=O)NCCN2CCOCC2C2CC2)ccc(CCc2ccccc2)cc1O Cc1ncc(C(N2CCC(CCC(=O)NCCC3COCCO3)CC2)=O)n1C c1(CC)cccc(C(=O)NCCC(O)CNC(=O)C(C)(C)N2CCOCC2)n1 C1(C(=O)NCCC(=C)CNC(c2cccc(CC)c2C)=O)CCC2CC2CC1 CC1(CO)CN(C(c2ncc(-c3ccc(C#N)nc3)cn2)=O)CCC1O N1(C(C(C)OCCC=C)=O)CCCC(C)(C(N2CCCSCC2C)=O)C1 N(C(=NCCOC)NCC1CCCCC1)CC1C(CC)C1 c1(C(C)N(C2CN(C(C34CCC3C4)=O)C2)C(=O)CN)nnnn1C.C(C)(C)(C)SC CCC(C)(CNC)C=O.C(=O)(C(C)(C)COC)NCCC(C)N c1(CC)cc(C)c(C(=O)N(C2CC(C(=O)N(C(C)C(C)SC)C)C2)C)o1 N1(C(C2CN(C(C(CC)CC)=O)C(C)(C)CC2)=O)C(C)CN(C2CC2)CC1C C1(NC(C(=O)N(C)C)=O)CCC(C)(C)CC1CNC(c1ccc(N)c(Cl)c1)=O CC1CCN(C(c2cn3ccsc3n2)=O)CC1NC(=O)C1=CCCS1 c1(C(N2CC3(CC(NC(C(F)=C(C)C)=O)C3)C2)=O)cc(F)c(F)c(F)c1F C(=O)(C1CCCc2nn(C)cc21)N1CCC2(N(C(CCCC(C)C)=O)CCC2)C1 n1(CC=C)cc(C(=O)N(CCCCN(C)C(c2nc(C(C)(C)C)no2)=O)C)nn1 C1(NC(c2c(C)c(F)cnc2)=O)CC2CCC(C1)N2C(=O)Cc1nccn1C c1(CSCC)cc(F)ccc1C(=O)NCCNC(C1CC(=O)C1CC)=O.C1CN1 CN1CC(O)CC1(C)C(=O)NCCN(C(=O)CCC=CCCCO)CC1CC1 c1(CC(=O)NCC(CC=C)NC(c2c[nH]nc2OCC)=O)ccc([N+](=O)[O-])cc1 CCCCC(O)CC(=O)NCC(C(C)(C)C)NC(=O)CN(C(C1CCCC1)=O)CC C1(C(=O)NC2(CN(C(c3c(CC)cno3)=O)C)CC2)CCCCC1C C12CCCN(C1)C(=O)N2.N1(C(c2cnc(C(=O)OC)s2)=O)CCOC(C)C1 CC1(C)CC(CNC(=O)CCn2cccnc2=O)N(C(C2CCSCC2)=O)C1 C1(CNC(C(CC=CC)C)=O)CN(C(c2c(Br)c(C)nn2C)=O)CCN1C Cc1ccc(=N)[nH]c1C(=O)NCC(C)(C1CC1)NC(c1ccc(F)cn1)=O c1(C(N2C(CN(C(=O)C(CO)N(C)C)CC)CCC2)=O)ccnn(C)c1=O C(=O)(CC(C)CC(C)(C)C)NCC(=CC(=O)NC1CCN(CC)CC1)C CCCCC(CC(=O)N1CCCC1C1CCOC1)NC(=O)C=Cc1ccncc1 c1(OCC)ccc(C(=O)NC23CC2CN(C(C2(SC)CC2)=O)C3)cc1CC C(=O)(C1=CC2CCCCCC12)N1C(N(C(=O)C(OC)OC)CC)CCC1 c1(C(N2C(C(=O)Nc3occ(C)n3)C=CC2)=O)cc2cc[nH]c2cc1Cl c1(C(N2C(CN(C)C(C3CC34CCCC4)=O)CCCC2)=O)ccnc2c1CCC2 C(CC(CNC(c1scnc1Br)=O)NC(C1(OC)CCC1)=O)OC C1(C#N)(C(=O)NCCN(C(CNS(CC)(=O)=O)=O)C)CC2(CC2)C1 C1(C)(CC(=O)NCC(C)N(C(=O)Cn2cnnn2)CC)OCCO1 c1(NC(C#CC(C)(C)C)=O)ccc2nccnc2n1.C12CCCC1CNC2=O c1(C(C)C)ccc(C(N2CCN(C(c3ccc(O)c(Br)c3)=O)C3CC23)=O)c(Br)c1 C1(O)(CC)CC(C(F)F)C1.C(=O)(C(C)N(C(=O)OC)C)N.C12(CC1)C(=O)NC2 C1(NC(COCC=C)=O)C(C)CN(C(c2coc3c2COC3)=O)CC1C C1(CNC(c2n(C)ncc2)=O)CCC2CN(C(c3cnoc3)=O)CCC2C1 C1(C(=O)OC(C)C)CCCN(C(C)(C)CNC(N2CCCC2c2ccc(Br)s2)=O)C1 c1(C(N2CC(O)(CN(C(C(CC)(C)O)=O)C)C2)=O)cnc2sc(C)cn2c1=O C1(CC(=O)N(C)CC2CCCN2C(=O)Cc2ccoc2)CC2C=CC1C2 CCCC(CCC)CC(=O)N1CCCC1C(=O)NC(C1(O)CCCC1)(C)C N1(C(c2ncc(C)c(C)c2)=O)CCN(C(C2CCN2S(C)(=O)=O)=O)CC2(CC2)C1 C1(C(=O)NC(CC(C)NC(c2c(OCC)c[nH]n2)=O)C)CCC(CO)CC1 C=CCCC(F)(F)C(=O)NCCNC(C1CCC(C(C)C)N1OC(=O)NC)=O CC1CN(CC2CCN(c3nnc(C4CCC(C#N)CC4)n3C)CC2)CC(=O)N1C CN1CCOC(C(N2CCCC2C(C)(C)NC(C2CC3C=CC2C3)=O)=O)C1=O Cc1ccc(C(=O)NCCC(C)(C)NC(=O)C(c2nc(F)ccc2Cl)C)c(C)c1 c1(C(N(CCN(C(c2ccccn2)=O)CC)CC)=O)ncc(C2CC2)s1 C1(NC(CC=CCC)=O)CCN(C(=O)Cn2nnc(C(C)(C)C)n2)CC1C(C)C N1(C(COC(C)(C)C)=O)CC(C(=O)Nc2ccsc2)C(F)(F)C1 CC1(C)COC(CNC(C2CCCN(C(C3CCCC3)=O)C2)=O)C1 c1(C(=O)NCCN(C(C2CC3CC3C2)=O)CC)ccc(-c2ccc(C)o2)s1 N1(CC)CCOC(C(=O)NC(C)(CNC(C2(c3ccnc(Cl)c3)CC2)=O)CO)C1 C1(N(C(C(C)Cn2cccn2)=O)C)CC2CCC(C1)N2C(C1CN(C(N)=O)C1)=O C(CC(C(=O)NC(c1ccc(C)cn1)C)NC(C1(C)CCCC1O)=O)OCC n1(CC(=O)NCCC(CNC(CC=C)=O)=C)nc(C)c(C=NO)c1C c1(C(=O)NCCn2cc(C(=O)NCC(CCC)C)nn2)ncccc1F Cc1ccc(C2(C(N3CCOC(CN(C)C(C4CCO4)=O)C3)=O)CC2)cc1Cl c1(C(=O)NC2CCC2NC(c2ccc(O)cc2)=O)cc(F)c2c(c1)CCC2 C1(CC(=O)Nc2ccsc2)CCN(C(=O)CCc2cn[nH]c2)CC1 C1(C(N2CCCC(O)(CCNC(C=CSC)=O)C2)=O)COCC2(CCC2)O1 N1(C(c2cc(F)c[nH]2)=O)CC2(CCN(C(=O)C(F)(F)CC3CC3)C2)C1 C1(CNC(N(CCC(C)C)CC(C)C)=O)CCCCCCO1 c1(C(=O)NC(CC(C)NC(CC(=C=C)C)=O)C)ccc2nnc(O)n2c1 C(=O)(C(C)C(=O)N1CCCC(CCNC(=O)C(C)Oc2ccccc2)C1)OC Cc1cc(C=CC(=O)NC(CC(=O)NC(C)Cc2ccccn2)C2CC2)on1 CC(C)CC(CC(C)C)NC(=O)C(C)C(C)NC(=O)CCCC1CCCC1 c1(C(N(C(CCSCC)C)C)=O)ccc(N2CCCCC2)cc1C Cc1cnn(CC(C)NC(=O)CCN(C(=O)C(C)OCCN(C)C)C)c1 N(C1CCc2c(O)cccc21)S(=O)(=O)CCC1CCC(C)CC1 N1(C(C(c2ccccc2)OCC)=O)CCN(C(=O)C(O)CC2CCCC2)CC1C N1(C(CCC=C)=O)CCC(c2ccc(Cl)cn2)CC1 C(=O)(CN=c1cc[nH]cc1)NCCN(C(c1cc(C)ccc1N)=O)CC c1(C(=O)NC2C(CNC(CN3CC(CN(C)C)C3)=O)C2)cn2ccccc2n1 C(=O)(CC(C)(O)C(F)(F)F)N(C)CC1CCCN1C(C1CC2(CC2)C1)=O n1(C(C)C)ncc(C(=O)NCCOc2ccccc2)c1N.N12CC3C(C3C1)C2=O C1(C)(CC(=O)N(CC)Cc2cnn(C)c2)CCN(C(c2ccc(C)cn2)=O)C1 CCCCC(O)CC(=O)N(C1CN(C(c2cnccn2)=O)CCC1O)C N1(C(CN2CC(=O)NC2=O)=O)CCC(F)(F)C(COC(=O)C(O)Cc2cnc[nH]2)C1 CCCC(C)(C)C(=O)NCC1CCCN(C(c2ccc(C3(O)COC3)cc2)=O)C1 Cc1cc(CCC(=O)NC(C)C(C)(C)NC(=O)CC2COCC2O)on1 Cc1c(C(=O)NCC2CCCC2NC(=O)CC(C)F)cnn1-c1ccccc1Cl c1(C(N(CC(C)NC(C2(C#N)CC2)=O)CC)=O)cn(C2COCC2OC)nn1 c1(NC(=O)OC(C)(C)C)cn2cccc(F)c2n1.C123CCC(CC1)N(C2)C3=O C(C(=O)NC1CCC(CNC(=O)Cc2ccsc2)CC1)(C(C)(C)C)N(C)C c1(C(N2C3C(OC)CC(C3)C2)=O)nccn2nc(C)cc12 N1(C(C=CC(CC)=CC)=O)CCC2CC2(NC(=O)COCCOCCO)CC1 c1(CC(=O)NC(CCN(C(C2(C)CC(=C)C2)=O)C)C(C)C)cc(C)cc(F)c1 c1(C(N2CCCC2Cc2ccc(Br)cc2)=O)noc2ncccc12 c1(OC)cc(C(=O)NCCC(C)NC(=O)CN(C)C(c2ccccc2)=O)n(C)n1 c1(C(=O)NC2C(CNC(c3c(CC)cccn3)=O)COC2)cc(Cl)c(O)cc1C c1(C(=O)NCC2CCN(C(C(P(C)(C)=O)O)=O)C2)ccc2c(c1)C(=O)NC2=O C1(C(CC)=O)C2CC3C(C2NC(c2c(N)cccc2Cl)=O)C13 CC(C)CCCC(C)CNC(=O)C(O)CCCNC(=O)C(c1cccn1C)=O C1(CNC(C2(CN(C)C)CC2)=O)CC(O)CN1C(=O)CCC1CCN(C)CC1 c1(C(N2CC3C(CNC(=O)CCc4ccccc4)(C3)C2)=O)nnn2ccccc12 c1(CCC)sc(C(=O)NC2C3CC2N(C(c2ccccc2C)=O)C3)cc1Br Cc1cc(Cl)ccc1CN1CC(NCC(O)COc2ccccc2)C(C)C1 C=CC1CCN1C(=O)CC1(C)CCN1C(C1(COC)CC1)=O S(=O)(=O)(c1cn(C)cn1)NCC(=O)NCC1N(C(C(C(C)O)N(C)C)=O)CC=C1 c1(OC(CC)C)cccc(CNC(c2ccc(-n3cnnn3)cc2)=O)c1 C(=O)(C(CSC)OC)NC1C(C(N(CCCO)CC)=O)C1 N1(C(=O)C2=CCCOCC2)CC2(C1)CN(C(C13CCC(C1)C(F)(F)C3)=O)CCO2 C(=O)(C1=CCC(C)(C)CC1)N.c1(CNC(C)CCCCC2CCC2)nn(C)cc1N Cc1cncc(C(=O)NC(C)CCCNC(=O)C(O)Cc2ccccn2)c1C N1(C(C2(OC)CCSC2)=O)CCC2(CC1)CN(C(C13CCCC1COC3)=O)C2 C1(COC)CC(CNC(c2cnn(C)c2SC)=O)N(C(c2cn(C)cc2C)=O)C1 C1(F)(CN(C(=O)C(=O)Nc2ccccc2)CC(=O)OC)CCNC1 N1(C(C(C=CC)O)=O)CCCC(CNC(c2cc(C)on2)=O)CC1 O=C(C1=C(Cl)CCOC1)NC1CC12CC(NC(c1c(Cl)nsc1Cl)=O)C2 C1(C(=O)NC2C(CCC)C2)CN(C(=O)C(C)(C)CCOC)CC1S(C)(=O)=O CC(C)C(C(=O)N1CCC1CN(C)C)NC(c1cccc(NS(C)(=O)=O)n1)=O c1(CC)cccc(C(N2CCOC(CN(C)C(c3cnc(C)o3)=O)C2)=O)c1 N1(C(c2sc(CC)c(C)c2)=O)CC(CNC(=O)C2=CCOCC2)CCC1C N1(C(C(C)CSn2cncn2)=O)CC(Nc2cc(C(C)(C)C)ncn2)CC(F)C1 C1(CC(=O)NC(CNC(=O)CC(C)n2ccc(C)n2)C2CC2)(OC)CCCCC1 C(=O)(CCC(C)(C)C(=O)NCCC(C)NC(c1ccnc2c1ncn2C)=O)OC N1(CCC(=O)N(CCCCCNC(c2coc(Cl)c2)=O)C)CCP(C)(=O)CC1 C1(C(C)C)N(C(C23C4C5C6C4C2C6C35)=O)CC12CCCC2 C(=O)(C(CC1CCC1)CC)N(C)CC1(NC(c2ccsc2C(F)(F)F)=O)CC1 C1(CC#C)(C(=O)NC(COC)C2(C)CC2)CCN(C(=O)CCC2CCCOC2)C1 C1(C(=O)NCCC(C=C)(C)C)CC(=C)CCN1C(=O)C(=CC1CCCC1)C C(C(=O)NCCC1CCN(C)C1)(C(C)CC)NC(CC=CCC)=O CC(O)(C(=O)N1CC2CC1C2C(N1CCN(CCOCCO)CC1)=O)C(F)(F)F c1(C(=O)NC2(CNC(=O)CC3CCCC(CF)C3)CC2)cc(Cl)cc([N+](=O)[O-])c1O C1(C(=O)NCc2ncc(C)s2)CN(C(=O)CNc2ncccn2)CC1(F)F C1(C(=O)C(=O)NC2CC(C)(N)C2)CC12CCN(Cc1cnc(N)c(Cl)c1)CC2 C(=O)(C1CCCn2cnnc21)N1C2CCC(NC(CCCCOC)=O)(C2)C1 CC(=O)COC(=O)CN(C)CCC1CNC1 N1(C(Cn2c(C)ncc2)=O)CCC(CC(N)=O)(NC(c2cc(C#N)cs2)=O)CC1 c1(C2(C(=O)NCCOCCCNC(COC)=O)CC2)ccc(OC)cc1 Cn1ccc(CC(=O)NCC(N2CCC(C(=O)NC(C)(CO)C3CC3)C2)=O)c1 N1(C(c2n(C=C)ncc2)=O)Cc2nccn2CC(NC(=O)Cc2cn(C)nn2)C1 O=C(C(CO)C(F)(F)F)N1CCCC(C(N2CC(F)(F)CCC2C)=O)C1 c1(OC)ccc(-c2csc(=NCc3ccc(F)cc3OC(F)(F)F)[nH]2)cc1Cl c1(C(N(C(C(=O)NCC(F)C2CCC2)c2ccoc2)C)=O)cc(C2CC2)no1 N1(C(C(C)C2CCCC2)=O)Cc2ccccc2OCC1(C)C N1(CC)CC(C(=O)NC2(COC)CCN(C(c3coc(Cl)n3)=O)C2)NC1=O C1(CNC(C=CCC=C)=O)CC(C)(C)CCC1NC(c1cc(CN(C)C)on1)=O C1(O)(CCNC(=O)CC2CCC2)CCN(C(C2C=CCC2)=O)C1 C(=O)(CN1C(=O)Cc2ccccc21)NC1CC(NC(=O)C2=CS(=O)CCC2)C1 c1(SCC(=O)NCCN(C(=O)Cn2nccc2C)CCC)ccncc1 c1(OC)ccc(I)cc1C(N1CC2C(C1)N2c1ncc(SC)cn1)=O CC1CC(C)CN(C(C2C(CNC(=O)CCC3(C)CC3)C2(C)C)=O)C1 CCC(C)C(C(=O)N1CCCCC1CNC(=O)CC1CC2CCC1O2)OC Cc1cnc2n1CCC(C(=O)NCCC(C)(C)NC(C1C=CC=CC=C1)=O)C2 c1(OC)cc2c(C(=O)NC3(CNC(CCC=O)=O)CC3)c[nH]c2cc1Cl.C1CC1 c1(NC(C)=O)ccc(C)c(C(=O)NC2CCCN(C(=O)C(C)(CO)N(C)C)C2)c1 C1(C(=O)NCC23CC(NC(CSc4c(C)n(C)nc4)=O)(C2)C3)Cc2nncn2C1 CCCCCC(=O)NC(C1CCCN(C(=O)Cn2nc(CC)cc2C2CC2)C1)C CCCC(CC)C(=O)NCCC(C)NC(C1CCN(CC(C)C)CC1)=O c12cn(nn1)C2.n1(CC(C)NC(C2CSC2)=O)cc(C2OCCO2)nn1 c1(C(c2n(CCC)nnn2)NCC(c2cnn(C)c2)OC)cc(Cl)ccc1Cl c1(C(N(CC(O)CNC(=O)C(c2ccccc2)F)C)=O)nnn(C)c1N N1(C(C(N2CC3(CCC(C(=O)NC4COC4)O3)C2)=O)C2COC2)Cc2ccncc2C1 CC1(C)CCCOC1C(=O)NC(CCC1CC1)C(=O)NCc1cc(Cl)ccn1 C#Cc1cc(C(=O)NC2CCN(C(c3cnn(C(C)(C)C)c3C)=O)C2)cc(F)c1 N1(C(C2C(C)CC(=O)CC2)=O)CCCN(C(=O)CCCn2ccnc2)CC1C C(=O)(C(C(C)C)NS(C)(=O)=O)NCC(C)NC(C12CCCC1(C(N)=O)C2)=O Cc1ccc(S(=O)(=O)N2CCCN(Cc3ccc(C(N)=O)nc3)C(C)C2)c(C)c1 C=C(C)C(CC(=O)N1CCC(N(C(=O)CC)C)C1)OCC1CCCC1 N1(C(=O)Nc2c(C)cc(Br)cc2C)CC(C2CCN(C(c3cnn(C)c3)=O)CC2)C1 Cc1nc(CNC(c2cccn2C2CC2)=O)c2ccnc-2[nH]1 c1(OCC=C(C)C)ccc(C(=O)NC2CCCCC2NC(c2cnsc2)=O)cc1 c1(CC(=O)NC(CCN(C(C=CSC)=O)C)(C)C)ccnc(O)c1 NS(=O)(=O)c1sc(NCc2cc(CC(=O)Nc3ccccc3)no2)nc1Cl N1(C(C(C=C=C)C)=O)CC(NC(C2C(C(C)=O)C2(C)C)=O)C2(CC2)C1 C1(F)(NC(CCSCCC)=O)CC(NC(=O)C(C)OC2CCOC2)C1 n1(CC)cc(C(=O)NC2COCC2NC(=O)CC2C=CCCC2)c(C(C)(C)C)n1 Cc1cc(F)c(C(N2CC=CC2CNC(C2CC3(CSC3)C2)=O)=O)cc1F C1(C(N2CC(C)(CF)C2)=O)(CC)CN(C(=O)CC2CC(C)=NO2)C1 c1(NCC23CC(NC(c4ccc(C)c(C)c4C)=O)(C2)C3)ncnc2c(Br)csc12 c1(C(N2CC3CN(C(c4cccc(Cl)c4)=O)CC32)=O)cc2ccc(Cl)cc2s1 C1(C)(C(N(CC(C)NC(c2cccc(C(C)C)c2N)=O)C)=O)CC(C2CC2)=NO1 c1(C(N2CCCC(N(CCO)C(C3(O)CCOC3)=O)C2)=O)nccc(Cl)c1F Cc1cccn(C(=O)NC23CCC2C3)c1=NC1CCC2CNCC12 CC1CN(C(=O)CC(C)(F)F)CCC1NC(=O)CNc1cccnc1Cl CC1CN(C(=O)Cn2cnnc2O)CC1n1cc(C(=O)NCCN(C)C)nn1 N1(C(C(CC)N2CCCC2=O)=O)CCC(CO)(NC(=O)Cc2cccc(Cl)c2)C1 c1(C(N2C(C)C(NC(=O)CN3CCCC3)C(C)CC2)=O)ccnc2ccccc12 N1(C(Cn2ncc(C)c2)=O)CCC(NC(=O)C(c2ccc(Cl)s2)C)C1C(C)C n1(COCC)nc(C)c(CC(=O)NCC2(F)CCC(NC(=O)C(C)O)C2)c1C c1(C(=O)NC(C2CCN(C(=O)CC3CC(=O)NC3=O)C2)C)ccc(O)nn1 N1(C(CCc2scc(C)n2)=O)CCN(C(c2cnc[nH]2)=O)C(CS(C)(=O)=O)C1 N1(C(COCC(=O)NC)=O)CC2CC1(CNC(=O)CN1CC3C=CC1C3)C2 Cc1nn(C)c2c(N3CCC4(CC3)C(F)(F)C4(F)F)nc(=NCC3CC3)[nH]c12 c1(SCC(=O)NC2(C)CC(NC(CCCc3cc(C)no3)=O)C2)c(C)n[nH]c1C C12(C(N(CCNC(=O)Cn3cccc3)CC)=O)CC1CCC2(F)F N1(Cc2cc(C)n(C)n2)CCCC12CCN(C(c1ccc(C)cc1C)=O)CC2 C(=O)(C1=CN2CCS(=O)(=O)N=C2C=C1)NCCNC(=O)C#CC1CCCOC1 N1(C(C(=O)N2CCC2C(N2CCCC2)=O)=O)CCOC(c2cccnc2)C1 N1(C(C(CC)F)=O)CC23CCCC2(C1)CN(C(=O)CC1CC1)C3 C1(CCNC(=O)C(C)(C)OC)(OC)CN(C(=O)C=Cc2cc[nH]n2)C1 c1(CC(C)NS(=O)(=O)CC2CC3C(C2)C3(F)F)ccc2nc(O)oc2c1 C1(C2CCCCC2)(CC)CCCN1C(C1CCCN1CC(F)(F)F)=O CCC(C)C(O)CC(=O)N1CCOCC1CCNC(c1csc(C(F)(F)F)n1)=O CC1CN(C(=O)CCF)CCN1C(=O)CNc1ccc(N(S(C)(=O)=O)C)cc1 N1(C(CC=CC=C)=O)CC2(CCN2C(=O)C(C)(C)C(F)c2ccccc2)C1 N1(C(CNC(C)=O)=O)CCC2CN(C(C3(NC(C)C)CC3)=O)CCC2C1 C1(C(=O)NC2(COC)CCN(C(=O)CSCCC(C)C)C2)CC2CCC(C1)O2 N1(C(C(CC#C)NC(=O)C(C)CC=CCC)=O)CC(C#N)C2(CCC2)C1 C1(C(N(CCOCC#C)C)=O)N(C(=O)CC2C(=O)NN=C2C)CCC1(C)C c1(CNC(C2C(CC)N(C(=O)CCc3ccncn3)CC2)=O)cc(C)ccc1F Cc1cnc(N2CCOCC2CN(C)C(C2(C)CC2Br)=O)nc1O c1(C(=O)NC(CCNC(CSC)=O)(C)C)cnc2c(F)cccc2c1 C1(CNC(C2(F)C(C)(C)C2(C)C)=O)CCC2(CCC2)C1NC(=O)C1=COCCO1 C1(O)(CNC(c2c(CC)nco2)=O)CCCN(C(=O)C#CC2CCOC2)CC1 N1(C(c2c(C)cncn2)=O)CC(CNC(=O)Cn2nnnc2C2CC2)CC(C)C1 c1(C(N(CCc2cccc(C)c2)C)=O)nnc(Cl)cc1N C1(NC(CCSC)=O)CN(C(c2ccc(C(C)C)nc2)=O)C(C)(C)C1 C(=O)(C1=C(Cl)CCOC1)NCC1C(NC(C(C)(C)OC)=O)CC1 c1(OC(C)=O)cccc(C(N2CCC(F)(C(=O)Nc3nn[nH]n3)C2)=O)c1 Cc1cnn(C(C)C)c1-n1cc(C2(C)CC2)nn1.C(C)(C)O N1(C(CNC=O)=O)CC2(C1)C(NC(c1ccc(CO)o1)=O)CCS2(=O)=O Cc1ccc(C(F)C(N2CCC(C)(CC(=O)NCC3(C#N)CCCC3)C2)=O)cc1 C=Cc1cncc(C(N2CCC(CCC(=O)NC(C)CSC)C2)=O)c1 CC(CCCc1ccccc1)C(=O)NC1CCN(C(=O)CN(C)C)C1 N1(C(c2nc(C)sc2)=O)CCCC1(C)C(=O)NC1CCCC(C(N)=O)C1 C(C(C(=O)N(C)CC1(C)CCCO1)NC(c1ccc[nH]1)=O)SCC c1(C(=O)NCC2CC(CNC(CN(C)CCO)=O)OC2)cccnc1N n1(CC(=O)NC(CC)CNC(=O)CC(C)F)ccc2ccc(F)cc12 C1(COC)(NC(=O)CCCCSC)CCCN(C(=O)Cn2nc(C)cc2C)C1 CC1(C)CC(NC(=O)Cc2cnc[nH]2)CN1C(C1CCOC(=O)CC1)=O C(=O)(CC(F)(F)C(F)(F)F)NC1C2CN(C(c3c(CC)nsc3N)=O)C1C(O)C2 C1(CC(=O)NCC2(OCC)CC2)CC(F)CN1C(=O)CC(C)(C)O C#CCCCCC(=O)N1CCCC(F)(CNC(=O)Cc2cn(C)nn2)C1 C(=O)(CCC(=O)N1CCOCC1)NC(C(C)NC(C1CN(C2CCC2)C1)=O)(C)C CCC(CC)(C(N)=O)NC(c1[nH]ccc1CNC(C1CCCC(C)CC1)=O)=O C1(F)(CC(=O)NCC(C2CCCC2)NC(=O)CCc2cnc(S)[nH]2)CCCCC1 C1(CNC(C2(C(CC)(F)F)CC2)=O)CN(C(=O)Cc2nnc(C)s2)CCC1(C)C C12(C(=O)NCC)CCC1CN(C(C1(NC(C3(C)COC(=O)N3)=O)CC1)=O)C2 N1(C(C(C)OCC=C)=O)C(CNC(c2cc(C)c(F)cc2N)=O)CC2CCCC12 N1(C(C=CC)=O)CCC(O)(C(C)CNC(=O)C(C)n2ccnn2)C1 C1(NC(=O)CC2(n3cncn3)CC2)CCCC12CCN(C(=O)CSC1CC1)CC2 c1(OC)cnc(Br)cc1C(=O)N(CC(C)NC(=O)Cc1[nH]cnc1C)C N1(C(CC2(CC)CCC2)=O)C2CCC1CC(NC(c1ccc(N(C)C)nc1)=O)C2 CC1CN(C)CC(C(=O)NCCCC2(NC(=O)Cn3cc(C(C)O)nn3)CC2)O1 CCCCN=C(NCC(F)(F)CO)NC1CCC(C)(C(=O)OCC)CC1 C1(CNC(c2n(CC=C)ccc2)=O)CC2CCC(C1)N2C(=O)C(C)NC(=O)NC C=CCC(CC(F)F)C(=O)NCC(CCCC)NC(c1ccc(C#N)o1)=O C(c1cccc(F)c1)=C(C(=O)NC(CN(C(c1nccnc1C)=O)CC)C)F CN1CCC(C)(C(N2CCC(NC(C3(Cl)CC3(F)F)=O)C(CO)C2)=O)CC1 C(=O)(CCC(C)CN(C)C)N(C(C)CNC(c1n[nH]cc1C)=O)CC C1(CC(=O)NCc2n(CC)ncn2)CCCN(C(=O)Cc2ccn(C)n2)C1 c1(C(=O)N)coc(COC(C)C)c1.C(=O)(CC)NCC1C(C(N(CC#C)C)=O)C1 CCCC(=O)NNC(=O)c1cccc(Cc2cn(-c3cccc(Cl)c3)nn2)c1 c1(CC(N2CCC(N(C)C(C3CCCOCC3)=O)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 c1(CC(N2C(CNC(=O)CCCC3CC3)C=CC2)=O)cnccc1Cl OC12CCC(CN(c3ccnc(NC4CCC(C(F)F)CC4)n3)C1)C2 CC(C(=O)N1CCOc2cc(Br)cnc21)C1OCCc2sccc21 C(C)(c1ccccc1F)=CC(=O)NC(CNC(C(C(C)(C)C)OC)=O)CO Nc1c(C(=O)NC2CC(NC(=O)CCNC(c3ccoc3)=O)C2)cc(F)cc1Cl c1(C(=O)NCC(CN(C(=O)CC2C=CCC2)C)(C)C)cc(OC(F)F)n(C)n1 c1(C(N2CCCC(CNC(CCC=C(C)C)=O)CC2)=O)cccc(P(C)(C)=O)c1 Cc1c(Cl)ccc(C(N2CCSC(C(=O)NC3CC3)C2)=O)c1Cl c1(C(N2CC(C)C(NC(C3(C)CCCN3C)=O)C2)=O)cnc(O)c([N+](=O)[O-])c1 Cc1[nH]nc2cc(CNC(C3CCN(Cc4cc(Cl)c(O)cc4F)C3)=O)ccc12 C(CO)(C(C)(C)c1ccccc1)NC(COC(C(C)=C(CC)C)=O)=O C(=O)(C1=CCCC1C)NC(CCOCC)C(=O)NC(C)CCC(C)C C1(NC(c2cc(C3CC3)no2)=O)C=CCN(C(=O)Cc2ccns2)C1 N1(C(c2ccc(F)c(C)c2F)=O)CCC2(CC1)CC(NC(c1nc[nH]n1)=O)CO2 C(=O)(C1OCCn2ccnc21)N1C(CC)CN(C(=O)Cc2ccc(C)nc2)CC1 N1(C(c2c(CC)ncs2)=O)CCC(C2(O)CCN(C(=O)C=CC3CC3)C2)CC1 N1(C(COCCC#C)=O)CC=CCC1C(=O)NCCC(CC)CO CCCCS(=O)(=O)c1ccc(C(=O)NCCN(C(=O)C(F)F)C2CC2)cc1 c1(C(C=C)NC(=O)N(C)CC)ccc(OC2(CO)CCCOC2)c(C(F)(F)F)c1 c1(C(=O)NC2(CCCNC(C(CCC)OCC)=O)CC2)scc2c1CCCC2 C1(NC(c2cccc(OC)n2)=O)Cc2ccccc2C1NC(c1cc(C)ns1)=O c1(C(=O)NCC2(O)CCN(C(C3(C)CCCCO3)=O)C2)nccc(Cl)c1Cl CCCCS(=O)(=O)CC(=O)NCCC1CN(C(c2cc(O)no2)=O)C1 CC(C)CCCC(C)CNC(=O)CSc1nn[nH]n1 C1(NC(c2nc(C)c(C)s2)c2n(C(CC)C)nnn2)CCC12CCCC2 C1(C(=O)NC(C=C)CC)CCC2(CC2)N1C(=O)Cn1ccnc1 C1(C)(C(N(CCCCN(C(c2nc(C)n(C)n2)=O)C)C)=O)CC2C=CC1C2 N1(C(C=CC(CC)C)=O)CCOC(C(N2CCOC(C(C)(C)C)C2)=O)C1 CC(C)(CCNC(=O)Cn1ccc(C2CC2)n1)NC(=O)Cc1ccccc1 Cc1ccc(C(C(=O)N(C)CCN(C)C2CC2)NC(=O)OC(C)(C)C)c(F)c1F c1(SCC(=O)NC(CC(C)C)CNC(C2(C)CC2(C)C)=O)ccc([N+](=O)[O-])cc1 C1(C(=O)NC(C#C)CC2CCOC2)CCCN(c2cccc(F)c2)C1=O C1(NC(=O)CCC2CC(NC(=O)CC3=CCCC3)C2)CC2C(C1)C2(F)F C1(C(N(CC(C)NC(=O)C=Cc2sc(Cl)nc2Cl)C)=O)OC2CCC1CC2 c1(C(=O)NC(CC)CNC(=O)CC2CCC(F)(F)CO2)c[nH]c2cccc(F)c12 C(=O)(CC1C(=O)N(C)c2ccccc21)N1CC(OC)(CNC(C2CCC2)=O)C1 Cc1cc(CNC(=O)CCn2ccnc2)oc1C(N1CC(C)(C)C1C1CC1)=O N1(C(CN(CCC#C)C)=O)CCC2(CCCCC2NC(C2CCCSC2)=O)CC1 c1(C(N2C(CN(C(=O)CCC3CCC3)C)CCC2)=O)cc2c(s1)COCC2 Cc1cc(C(=O)NCC(C)(C)OCC(=O)NCc2[nH]nnc2C)ncn1 CC(O)(C(=O)N1CC2C(NCc3cnc[nH]3)C2C1)C(F)(F)F c1(C(=O)NCC2C=CCN2C(=O)Cc2cnc[nH]2)ccc2nccn2n1 C12(C(N(CCCNC(CC3C(C(=O)OCC)CS3)=O)C)=O)CCCN1CCC2 CC1(C)CN(C(N2CCC(N(C(=O)C(F)(F)F)CCC#N)CC2)=O)CC1C(=O)O c1(N2CCC(OC)C(F)C2)nc(NCCC(C)(C)c2ccccc2)nc2ccsc12 C(C1=CCN(C(=O)CC2(O)CCCC2)CC1)NC(c1ncoc1-c1ccon1)=O C#CCC(O)C(=O)NCCCOCCN(C(=O)Cn1cncn1)COC(C)=O c1(C(=O)NC23CC2CN(C(C2CCCC2C2CC2)=O)C3)cc2c(cc1Cl)NCC2 c1(OCCC)c(-c2nc(C(N3CCNCC3CC)=O)cs2)cccc1C c1(C(=O)NCC(C)CNC(C2CCC(=O)CC2C)=O)cc(Cl)cc([N+](=O)[O-])c1O C1(C(N(C)CC2(O)CCOC2)=O)CCN(C(c2cc[nH]n2)=O)C12CC2 C1(CC=C)(NC(c2cc(C)ns2)=O)CCCN(C(c2cc(SC)c(C)o2)=O)C1 C1(OC)C2CC1CN(c1ccccc1NC(=O)NCCN1CCCCC1)C2 C(CC(C)C(=O)N1CCOCC1CCNC(c1cc(C2(C)COC2)no1)=O)OC C(CC(C)C)(C(=O)NCCC1(O)CN(C(C2CCN(CCO)C(=O)C2)=O)C1)OC CC1OC2CCC1(C(=O)NCCC1(C(N3CC(F)(C4CC4)C3)=O)CCCCC1)C2 C1(C)(CC)C=C(C(=O)NCC(C)(C2CCC2)NC(c2cccnc2S)=O)C1 c1(OC)ccc(C(=O)NC2CC(C)CN(C(c3cc(C)c(Cl)s3)=O)C2)c(F)c1 N1(C(COCC)=O)CCC12CN(C(c1cccc(C(C)C)c1)=O)C2 c1(C(=O)NCC2CCCN(C(C3(C)CCCO3)=O)C2)ccc([N+](=O)[O-])cc1N N1(c2nc(CC)cc(CC)n2)CC2(CC(NC(=O)C(C)Cc3cnc[nH]3)CO2)C1 c1(OC)ncnc(Cl)c1C(=O)NC(C1CCN(C(=O)CC2CC2)CC1)C CC(N=c1[nH]c2c(c(=NCc3cccc(OC(F)F)n3)[nH]1)SCC2)c1cscn1 N1(C(c2cnc(C)[nH]2)=O)CCC2CN(C(c3cnn4c3CCC4)=O)CC12 C1(O)(c2cn(CCNC(C(=O)NC(c3ccn(CCF)n3)C)=O)nn2)CCOCC1 C1(C(=O)NCC(CN(C(C2N(CCC)CCC2)=O)C)(C)C)CCCN1N=O c1(COC)nc2cc(n1)N1CCCC(C1)C(=O)N2.c1(SC(C)C)cccc(Br)c1 C1(CC(=O)N(CCCNC(=O)CC2(C(N3CCCC3)=O)CC2)CC)CCC(=O)N1 N1(C(CSCc2cc(C)c(C)o2)=O)C2CCCC1CC(NC(=O)CN1CCC1)C2 N1(C(C(=O)NCC)=O)CC(CNC(c2ccc(C(F)(F)F)o2)=O)CC1C N1(C(c2cc(CCC)on2)=O)CC(NC(=O)C=Cc2cnccn2)C2(CCC2)C1 c1(C(N)=O)cncnc1NNC(=O)C1CCN2CCC1C2 C(=O)(C(C)(C)C(O)C1CCOCC1)Nc1ccc(-c2cn(C(C)CO)nn2)cc1 Cc1oc(CNC(=O)CC(C)(C)N(C)C)nc1C(=O)N1CCCO1 C1CCC(O)CC(=O)NC(CC)C(=O)N1C.C(C(O)C(=O)OCC)=CC c1(CN2CCCN(C(=O)C(N3CCC(CO)C(O)C3)=O)CC2)ccccc1[N+](=O)[O-] Cc1ccc(C(=O)NCC2CN(C(C3(N(C)C)CCC3)=O)CCC2C)c(C)c1 c1(CC(N2CC(CN(C(C(C=CCCC)O)=O)C)OCC2)=O)ccnc(Cl)c1F N1(C(CCC#CC)=O)CCN(C(=O)CSCc2ccccc2)C(CCOC)C1 Cc1cc(C(=O)NCC(C)CN(C(=O)C(c2cnn(C)c2)C)C)c(C)o1 c1(OC(C)C)ccc(Cl)c(CN2CC(NC(c3nc[nH]n3)=O)C(F)C2)c1 CCC(O)(CN(C)C(C1(F)CCN(C(=O)CCC2CCCOC2)C1)=O)CC C(CCCC(=O)N1CCCC(N(C(=O)C=CI)C)C1)N(C)C Cc1cc(Cl)ccc1CC(N1CCC(C(C)NC(=O)CCOCC2CC2)CC1)=O Cc1cnc(NCC2CC(F)(F)C2)c(S(=O)(=O)NC(c2ccccc2C)C)c1 CCC(C)CC(C)CC(C)C(=O)NCCCn1ccc(=O)cc1C N1(C(CCc2n(C)cnc2)=O)CCC(C(=O)NCC(O)C(F)F)C1(C)C N1(C(C)=O)CCCC12CCN(C(C1CCc3cc(O)ccc3C1)=O)C2 CCCCC(F)C(=O)N1CCCC(CC(=O)NC(C)(COC)CO)CC1 c1(-c2nc(C(c3ccc(OC)nn3)CC)on2)cn(C(C)C)nc1C Cc1oc(C#N)cc1C(=O)NCC(C)C(=O)NC1CCCCC1O N1(C(COCC=C)=O)CCC(C2CCN(C(=O)CC34COCC(C3)C4)CC2)CC1 Cc1c(Cl)sc(Cl)c1C(=O)NC1CCN(C(c2ccc[n+]([O-])c2)=O)CC1O c1(CCC(=O)NC2(C#N)CCN(C(C3CCCCC3)=O)C2)c(F)cc(Br)cc1F c1(CC)c(C(=O)NCCCC(C)NC(c2c(C)cnn2C(C)C)=O)csc1C C1(CNC(C=CCC)=O)CN(C(c2cccnc2S)=O)CC2CC12 C1(NC(c2cc(COC)on2)=O)CCN(C(=O)Cn2cc(N)cn2)C(C)C1 N1(C(C(CC)(F)F)=O)CCC2(CC1)CC(N=c1[nH]cnc3cnccc13)CCO2 n1(CC)cc(C#N)c(=NC(=O)c2cc(NS(=O)(=O)c3c(F)cccc3F)cs2)[nH]1 Cc1cc(Cl)c(C(=O)NCCC2CN(C(c3cnn(C(F)F)c3)=O)CCO2)cn1 C=CC(C(F)(F)F)NC(=O)CSCCNCC(CC)OC(C)=O c1(C(N2C(CNC(CC(C)O)=O)CC(O)C2)=O)cnc(O)c2c1NCCC2 C1(O)(CCNC(=O)C2=COCC2)CCN(C(c2cccc(=S)n2O)=O)CC1 Cc1cc(C(=O)N(C2CCCCC2)CCNC(=O)C(C)(Cl)Cl)nc(C)n1 c1(CC(N2C(NC(=O)NCCNC(CC(C)(C)C)=O)CC2)=O)cccc(Br)c1F CCCC(O)(CCC)CC(=O)NCC1C(C)CCN1C(=O)COC c1(CN(C(c2nn(CC3CCCN(CC)C3)nc2C)=O)CC)c(F)cccc1F c1(CCNC(N(C)CC)=O)nc(COCCO)no1 N1(C(CN(C(=O)CC2CCC(C)C2)CCOC)=O)CCC(C)(CCO)C1 Cc1ccc(C(=O)NC(C(=O)NC2CCCC3(C2)N=N3)C(C)C)nc1C C1(C(N2CCN(N3CC(Cc4nnc(C(F)F)s4)C3)CC2)=O)CCCC12CCC2 C(=O)(C1OCCc2ccccc21)NCC1CCC(NC(CC2CC(OC)C2)=O)C1 c1(C(=O)NC2CCCC(CNC(CNC(=O)OC)=O)C2)c(C)ncn1OC C=CCCCCC(=O)N(C1(C(=O)NC(CC)(CC)CCO)CCC1)C1CC1 N1(Cc2ccc(C(=O)OCC)s2)CCC(C#N)(NC(=O)C(C)(C)C)C1 Cc1cc(C)n2cnc(NC(C3CCC(=O)N3)=O)c2n1.C12(CC1)NC2.C1C(=O)N1 c1(C(=O)NC(C2CC(CC3CC3)C2)CNC(C=C(COC)C)=O)nnc(O)nc1O CC1COCCC1N(C(=O)CCOCCN(C)C(C1CCCCC1)=O)C N1(C(C(c2ccc(F)cc2)CC)=O)CC2CCC1C(CN=c1ncc(Cl)c[nH]1)C2 C(CCCCC(=O)NC1CC1NC(=O)CCCc1nc(-c2cccs2)n[nH]1)=CC C1(C(=O)NCC#CCNC(C(CC=C)CC)=O)CN(C)C(=O)CCO1 C1(CNC(c2cccc(OC)c2C)=O)CN(C(c2cc(C)cnn2)=O)CC12CCC2 Cn1nc2c(c1C(=O)NCC1CC1NC(C13CCC(C1)OC3C)=O)COCC2 C(=O)(C(CNC(=O)C(c1ccn(C)n1)C)CC(C)C)NCC(CCC)CCC c1(C(=O)NCCN2CCCN(C(C(CC)C(C)C)=O)CC2)ncnc2sccc12 C(=O)(C1CN(C(C2CCC2(F)F)=O)c2ccccc21)OC C(=O)(C1=C(C)CCOC1)NC1CC(CNC(CCCOC(c2ccccc2)C)=O)C1 C(=O)(C(C)(CO)NC(c1cnc(C2CC2)o1)=O)NCc1n(CC)nnn1 C=C(C)CC(C(=O)N1CCC(O)C1)NC(=O)C(=O)C(C)CC c1(CCC)nc(C)cc(=NCC2(NCC3CC3c3ccccc3)CCC2)[nH]1 N(C1COc2cc(F)cc(F)c21)C(=O)C(N1CCOC2CNCC12)=O N1(C(c2scc(C(N)=O)c2)=O)CCCC(NC(C2CCN(c3ccccc3)C2)=O)C1 N1(C(C2C(OC)C2)=O)CCCC2(C1)CN(C(=O)C(O)CN(C)C)C2 C1(NC(c2c(OC)ccc(F)c2)=O)CCCN(C(=O)C(C)(C)C(=O)OC)CC1F c1(CC)nocc1CNC(=O)C(C1CCCC1)NC(=O)C=CCOC CN1CCN(C(c2nnc(S)n2C)=O)C(C(=O)NCC(c2ccco2)O)C1 C(=O)(CCP(C)(C)=O)NC(CNC(C(C(C)C)NC(c1ccccc1)=O)=O)CO C(N=c1[nH]cnc2c(F)cccc12)C1N(C(C2(C(=O)NC)CC2)=O)CCOC1 N1(CC(=O)N(C(CCNC(C(COC)N(C)C)=O)C)C)CCCNC1=O c1(C(=O)NCCCN(C(c2cnn(C3CCC3)n2)=O)C2CC2)cccnc1 C1(NC(c2ccc(CC)s2)=O)CC2CCC1CC2NC(c1cc(OC)cs1)=O N1(C(c2nnn(C(C)(C)C)n2)=O)CCCN(CCNC(C2(CO)CCC2)=O)CC1 C(CC(C(=O)NOC1CCC1)NC(C1COCC1(C)C)=O)=CC c1(C(N2CC(N(C(C3CC(OC)C3)=O)C)C(F)C2)=O)cc(F)ccc1C1CC1 N1(C(Cc2c(C)nc[nH]2)=O)CC(NC(c2cnc(N(C)C)nc2)=O)C(C)C1 N1(C(C(CC)n2cccn2)=O)CCSCC1CCNC(C1(C)CC(F)(F)C1)=O C(=O)(CCCC(N)=O)N(C)CC1CN(C(=O)C(=Cc2cccnc2)F)CCO1 C1(CCc2cn(C3CN(C(C4CCCO4)=O)C3)nn2)CCOC1C(N1CCCC1)=O N1(N(C(=O)CCC2CCN(C(=O)CCc3ccccc3F)C2)C)CCC(C)(O)C1 C1(C2CC2)(C(N(CC(CC)NC(c2ccccc2Cl)=O)C)=O)CCOCC1 C1(N(C)C)COCCN(C(C2CC23CC(NC(C2C4CCC(F)C24)=O)C3)=O)C1 CC(C)CC(CNC(=O)COC(C)C)NC(c1cncc(I)c1)=O c1(OC)c(C(N2CC(O)(CNC(C3CCC3(F)F)=O)C2)=O)cc(Cl)cc1Cl Cc1ccc(=NCCC(=O)N2CCC(CCNC(c3nc(O)sc3C)=O)C2)[nH]c1 C(c1ccncc1)=C(C)C(=O)NC1CCC(CCNC(c2cn(C)cc2C)=O)C1 C(=O)(C(C(C)C)C(C)C)N1CCN(C(C(C(=O)NC)(C)C)=O)CC1CC(=O)NC Cc1ccccc1C12CC1CN(Cc1nnc(C3CCCC(C)O3)o1)C2 C1(N(C(CCCCC)=O)C)CCC2CN(C(c3coc(C(C)(C)C)n3)=O)CC12 Cc1ccc(C=CC(=O)NC(C)CC(C)NC(c2cnn(CC(C)C)c2)=O)nc1 C(=O)(C(C)C(F)(F)F)NCC.c1(C(=O)NCCC(=C)C)ncc(N(C)C)cn1 N1(C(C2CCC(=C)CC2)=O)CCCC(C2CCN(C(=O)CCCSC)C2)C1 c1(N2CCCC(NC(=O)Cn3nccc3C3CCOC3)C2)ncncc1Cl c1(CNC(=O)NC2C(C(=O)OC)CCCC2)cccc(C(F)(F)F)c1S(C)(=O)=O N1(CCNC(CC2C(N(CC(=O)NCC)C)CC2)=O)CCOC1=O C1(O)(C(N(C(c2ccc(Br)cc2)CC)C)=O)CCN(c2cc(C)nc(C)n2)CC1 S(=O)(=O)(c1ccccc1Br)N1CC(C#N)C(NC(=O)Cc2c(F)cccc2Br)C1 C1(CN(C(C(C)OCCN(C)C)=O)C)CCCN(C(=O)Cc2ccon2)C1 Cc1ccc(C(F)(F)C(N2CC3CC2C3NC(c2nncn2C(C)C)=O)=O)cc1 N1(C(c2c(C)nc(C)o2)=O)CC2CCC(C1)C(NC(=O)C(C)C(C)(C)C)C2 C1(C(=O)NCCCCNC(=O)C=CSCc2ccco2)CS(=O)(=O)CC12CCC2 C1(OCC)CN(C(=O)CC2CC(F)(F)C2)CC1CNC(C1CCN(CC)C1)=O n1(CC(=O)OC)cnc(C)c1C(N1CCC(CCOC)(NC(=O)C(C)CO)C1)=O S(=O)(=O)(c1ccc(Cl)c(SC)c1)N(c1ccc(F)c(F)c1Cl)CC(N1CCCC1)=O.CO N1(C(Cc2nnc(C)s2)=O)C2CCC1CC(N(C)C(c1c(C)ccnc1C)=O)C2 c1(C(=O)NC(CC)(C)CNC(=O)C=CC(F)(F)F)ccc(S(N)(=O)=O)cc1 Cn1nccc1-c1n[nH]cc1C(=O)NCCCOCCCNC(c1ccc(F)s1)=O CC1(CC(=O)NCC2CC3CCC2C3)CCN(C(=O)CC2(CO)CCC2)C1 C12(CCCC1)C(=O)N2.C1(C(=O)NC(CNC(=O)OC)C)CC=CCO1 S(=O)(=O)(c1cccc(N2CCCC(O)C2)n1)NCc1c(C)c(Cl)c(Cl)cc1 C1(=O)C(CC(Cl)Cl)O1.CCCCCC(=O)c1cccc(C(=O)C(F)(F)F)c1 Cc1cc(=NC(=O)C2CCCC(NCc3ccc(Br)cc3I)C2)[nH]o1 CC1CCN(CC(N2CCOCC2C(=O)NC(CO)C(C)(C)C)=O)CC1 c1(CC)ccnc(C(=O)NC(C(=O)NCCc2cn(C)cn2)C2CC2)c1 CC(C)(C(=O)NCCCC(N1CCCC(n2cc(-c3cncs3)nn2)C1)=O)C(F)F C1(NC(c2c(OC)n(C)nc2C)=O)CC2CN(c3cc(C#N)nc(C)n3)CC2C1 c1(C(N2CCCC(C)(C(=O)NC(c3nccs3)CC)C2)=O)n[nH]c2ccccc12 C1(NC(c2c(OC)cccc2)=O)CN(C(c2cc(=N)[nH]c(Cl)n2)=O)CC1C1CC1 N1(C(COCC)=O)CCCC(C)C1CNC(C1(c2cncnc2)CCCC1)=O Cc1c(F)ccc(C(N2CC=CC2CNC(=O)CCOC(C)C)=O)c1Cl N1(C(C(C)c2cc[nH]n2)=O)CC2C(NC(c3ccc(OCCF)cn3)=O)C2C1 CCC(C)(C)C(O)C(=O)N1CC2(CC2)CC1CNC(c1cnoc1C1CC1)=O C=CC1(C(=O)NC(CN(C)C)CC)CCN(C(=O)CN(CC(C)(C)C)C)C1 N1(C(c2noc(CC)c2C)=O)CC(CCNC(=O)C(F)=C(C)C)OC(C)C1 O=C(CC1=NNC(=O)C1)NCC(C1CCN(C(c2ccn(C(F)F)n2)=O)CC1)F C1(CNC(c2cc(O)cs2)=O)CC(F)CN1C(=O)CC(O)Cc1ccccc1 C1(NC(N2CCC(SC)C2)=O)CCCC(C)(C)C1 CC1C(C(=O)N(C)CCNC(C2CCCCCC2)=O)CCN1C(N)=O C12(C(N3C(C(C)N)CCCC3)=O)CCC(CC1)CC2 c1(C(N2C3CC(NC(C4CN(C(C)=O)C4)=O)C2CC3)=O)ccc2nnn(O)c2c1 C(=O)(CC1=Cc2c(ccc3ccccc23)C1)OC(C#CC(=O)O)=O CC(C)C(C)C(C)CC(=O)NC1(CNC(c2ccn(CC(F)F)n2)=O)CC1 N1(C(c2c(C)c[nH]c2)=O)CCC(O)C(N(C)C(C2CCCCN2C)=O)C1 C1(C(N2CC3(CCCO3)C2)=O)(CC)CCN(C(=O)CC(C2CC2)C2CC2)CC1 N1(C(C(C(C)C)SC)=O)CCCC2(NC(c3ccn4nccc4n3)=O)CCCC12 c1(NC2(c3n(CCSC)nnn3)CCC(C)C2)ccc(F)c(C(F)(F)F)c1Br c1(C(=O)NC(CNC(C2C(=C)CC2)=O)(C)CO)cc(-n2cnnc2)ccn1 c1(OC)ccc(N)c(C(N2CCC(C)(NC(C3CCC3C(N)=O)=O)CC2)=O)c1 C=CCN(OC)C(=O)C1(C)CC(O)CN1C(=O)Cc1ccc(C)c(C)c1 N1(C(c2ccc(C)cc2C)C(=O)NC(CC)C)CCN(C)C(c2ncc[nH]2)C1 N(C1CCNc2ccc(Br)cc21)C(c1c(Br)ccc(Cl)c1F)CO C=CC1CN(C(=O)C(C)(CO)OC)CC1NC(=O)CC1(OC)CCC1 c1(C2C(=O)O2)ccc(C)c(OC)c1.c1(C2C(C(=O)OC)C2)cccnc1 CN1C(C(=O)NCC2CCC2NC(c2n[nH]cc2[N+](=O)[O-])=O)CCS1(=O)=O CN1Cc2cc(C(=O)NC3CC3NC(=O)Cc3cnoc3)ccc2NC1=O c1(C(N(CCNC(C2CCCN(C(=O)OC)C2)=O)C)=O)nn2cccnc2c1Cl S(=O)(=O)(C(F)(F)F)OCCC(=O)OCCC(=O)N(CCNC(COC)=O)C c1(C(=O)NCC(C)NC(CS(=O)(=O)NC)=O)nc(C)ccc1C CC(=O)C(C)(C)CC(=O)NCCOC(C)(C)CNC(=O)NC1CC2(CCC2O)C1 Cc1ccc(CN2CCCC(NC(c3n[nH]c(C)c3O)=O)C2)c(Cl)c1 S(=O)(=O)(c1cnc(NCc2cncc(C#N)c2)c(Cl)c1)NC1(CCOC)CC1 c1(C(=O)NCC2C(C)CN(C(C3CCS(=O)(=O)C3)=O)C2)cc(O)cnc1N c1(CC)ncncc1C(=O)NC(CC1CC1)CC(=O)N1CCC(CC(C)(C)C)C1 c1(NCCOC(=O)NCCC(=O)NCC=C(C)C)ccc(Cl)cc1 C1(CNC(=O)NC2(C(F)(F)F)CCOCC2)CCCCC1NC(C1CC(O)C1)=O C1(NC(CCC=C)=O)CCN(C(=O)COc2cc(C)ccc2C)CC1CO N1(C(c2cnc(OC)s2)=O)C2CCC1CC(NC(C1CC13CCC3)=O)C2 C1(C(N2CC(C)(C)C(CO)C2)=O)CN(C(=O)CCCC#N)CC(C)(C)C1 c1(C(N2CCC2COC)C(=O)NCC)nc(C)n(C)c1C(=O)OC(C=O)C C#Cc1cc(C(=O)NC(C)C=CC(=O)N(C)Cc2nc(C)no2)ccc1C Cn1ccc(-c2cc(C(=O)NCC3(CCNC(C4SCCCS4)=O)CC3)no2)n1 C12(C(=O)NC3CC(C)N(C(c4cc(O)nn4C)=O)C3)CCC(CC1)CC2 C(=O)(C1=COCCO1)NCC1CC(OC)CN1C(C1CC(F)C1)=O C1(CNC(c2ccn(CC)n2)=O)CCCC(CNC(c2cc[n+]([O-])cc2)=O)C1 C1(C(C)C)(C(=O)NCC2(C(=O)N(CC(C)(C)O)C)CC2)COC1 N1(Cc2cnc(CC)s2)CCC(F)(F)C(NC(C2CCC3(CC2)CC3)=O)C1 N1(C(CCC#N)=O)CC23CCCCC2(C1)CN(C(c1n[nH]c2c1CCSC2)=O)C3 N1(C(c2cc(OCC)no2)=O)CCC(C(C)NC(=O)C=Cc2scnc2C)CC1 C(=O)(CS(=O)(=O)C(C)C)N1CCCC(N(C(=O)Cc2coc(C)n2)CC)C1 C(C(C)(C)C(=O)N(CCC(=O)N1CC(CC(F)F)C1)C)SC c1(C(N2CCCN(C(CC34CCC(C)(OC3)C4)=O)CC2)=O)cc2n(c1)CCSC2 Cc1c(CC(=O)NC(C)(C)C=CC(N2CC(C)(C)C2C(C)C)=O)cnn1C N1(C(C=C(CCC)C)=O)CCN(C(c2cc3oc(Br)cc3[nH]2)=O)C2(CC2)C1 C1(NC(CC2(C(=C)F)CCC2)=O)CN(C(=O)COC2CCCCC2C)CC1(C)C c1(OC)ccc(-c2nc(COC3CCCCC3NC(C3CCO3)=O)oc2C)cc1 N1(C(c2cc(CC)[nH]n2)=O)CCC(C2(NC(c3cnc(C4CC4)o3)=O)CC2)C1 Cc1cc(N2CCOCC2CNC(c2conc2C2CCC2)=O)nc(C(C)C)n1 c1(C(=O)NCC(CNC(C2C=CCCC2)=O)OC)ncc(C#N)cc1C C1(C(=O)N(C2CCN(C(C3CN(C)C3)=O)C2)C)(OC)CCCC(C)(C)CC1 c1(CC(N2CC(F)CC(NC(C3(F)C(C)C3)=O)C2)=O)ccc(C#N)c(F)c1 C1(CNC(c2ccc(C(C)C)s2)=O)CC2(CCOCC2)CN1c1ncccn1 N1(C(C(c2ccccc2)N(CC)Cc2ccccc2)=O)CCCC1(C)CCN.CC Cc1nc(C#N)ccc1C(N1CC(NC(=O)CCc2cn[nH]c2)C(C)(C)C1)=O C1(NC(C(C)=CC2CC2)=O)(CNC(C2COC3(CCC3)C2)=O)CCC(F)(F)CC1 C1(C(C)(C)C)C(NC(C2(n3cccc3)CC2)=O)CCN1C(=O)CCNC1CCC1 c1(CCCCCNC(c2cc(C(=O)OCC)sn2)=O)cc(C)ccn1 c1(C(=O)NC)ccc(Nc2nc(C(F)(F)F)n3ccccc23)cc1[N+](=O)[O-] N12CCC1(CCC(=O)N(CC(C)(O)CO)C(c1c(C(C)C)con1)=O)CC2 C#Cc1ccc(C(=O)NC2CCN(C(C3CC(=C)C3)=O)C(C3CC3)C2)cn1 c1(NC(=O)CC2(SC)CCC2)c[nH]nc1C(C1CCCN1C)N.c1(C(C2CC2)C)nn[nH]n1 c1(C(=O)NC2(COC)CN(C(=O)CCCn3ccnn3)C2)cccc(N)c1C N1(C(Cc2cc(C)c(O)cc2)=O)C2CCC1CC(N(C)C(C1(F)CCOC1)=O)C2 c1(OC)ccc(C(=O)NCCC2(C(=O)NC(c3ncc[nH]3)CO)CCC2)s1 c1(CC(=O)OC)ccc(CC(=O)NCCC2CC2C)cc1.C12CCN(CC1)C2=O N1(C(CC=C)=O)CCN(C(c2n[nH]cc2-c2ccncc2)=O)CC1CCC N1(C(C(CCC)CCCO)=O)CCCC(C2CCN(Cc3cnsc3)CC2)CC1 N1(C(C=CCC)=O)CCN(C(=O)C(C(C)C)N(C)C)CC1CCCC CCC(C)(CNC(=O)CC(C)COC)C(=O)NCc1cc(O)ccc1F c1(C(=O)NC(CC(=C)Cl)C(=O)NC(CO)CCO)cccc2nccn12 CN=c1[nH]c(=NCc2cc(C)co2)[nH]c(=NCCSc2ccc(F)cc2)[nH]1 Nc1cc(F)c(CC(=O)NCCCNC(C2CCC2c2ccccc2)=O)cc1F CCC(C)(C)CCCC(=O)NC(=O)CN(C12COC(C)(C1)C2)C.N1(C)CCCC1 C(=O)(CCC(F)(F)F)NC1C(CNC(c2ccc(NC(C)=O)s2)=O)CCC1 N1(C(C(C=C)(C)O)=O)C2CC=C(C(=O)NCC3CCC(C)(C)O3)C1CC2 Cc1ncc(C=CC(N2CCC(NC(c3nncs3)=O)C2)=O)c(O)n1 C12(CNC(C(C)SCC)=O)CC(CNC(c3ccc(OC(F)F)nc3)=O)(CO1)C2 C(CC(C)(C)C(=O)NCC1(F)CC(NC(C2(C)CC(O)CN2C)=O)C1)NC(C)=O C12(C(N(C)CCOC3CCCOC3)=O)CC(C)(CN1C(=O)CCC(=O)N(C)C)C2 C1(NC(C=C2CCC(C)CC2)=O)CN(C(=O)C=CC2CCCO2)CCC1(C)C c1(C(=O)NC(CNC(C2(CC=C)CCOCC2)=O)(C)CC)cc(CC)ccc1Cl C1(CNC(Cc2ccc(C)s2)=O)CCC(F)(CNC(C2(C#N)CCCO2)=O)CC1 c1(C(=O)NCC2C(C(=O)OC)CCO2)ccc2nc(C)cn2c1 c1(C(=O)OC)sccc1S(=O)(=O)N1CCOC(C)C1 N12CCCC(C1)C2=O.c1(OCC(=O)NC2CC(C)(NC(C)=O)C2)cccc(Cl)c1 c1(C(=O)NC2C(NC(C=C(CCC)C)=O)CCCC2)ccc(=O)n2c1CCC2 N1(C(CCc2nnc(C)o2)=O)CC2(CCN(C(C3(O)CCCC3)=O)CC2)C1 CC1CN(CC2CCCO2)CC1N(C1CC(=O)N(C2CNC2)C1)c1ncc(F)cn1 CC(C)C#CC(=O)N(C1CN(C(c2nccc(COC)n2)=O)C1)C CC1CCC(CNC(=O)Cc2cccc(Br)c2Cl)CN1C(=O)C=CCF Cc1cccc(NC(N2CC3CC3(C(=O)NCCCCCO)C2)=O)c1C c1(COC)nc(C(N2CC(C(O)C(=O)NC34CC(C)(C3)C4)C2)=O)cs1 C1(C(=O)NCC(CC=C)(C)CO)CCN(C(C2C3CN(C)CC23)=O)C(C)(C)C1 c1(SC)ncc(C(=O)NCC(C2CCCC2)NC(=O)C(C)NC(C2CCCC2)=O)s1 CC(CNC(=O)CC(CC1CC1)NC(=O)CCc1cn[nH]c1)S(C)(=O)=O C1(CC)CN(C(=O)Cc2ccnc(C)c2)CCN1C(c1cc(=O)cco1)=O N12CCCc3cc(ccc31)CC2=O.CC12CCC(C(=O)OC(C)(C)C)(CO1)C2 C1(c2c(C)nc(C3CC3)o2)CCN(N2CC(O)CCC2C)C1 C1(CNC(c2c(C)nns2)=O)CC2COCC2N1C(=O)Cc1nnc(C)s1 c1(C(c2nnnn2C(C)C)NC(c2scc(C)n2)C)cccc(C(C)C)c1 C12(C(N(C)CCN3CCC(Cn4ccccc4=O)C3)C)CC(CCO1)C2 c1(C(N2C3C(C(N4CC5CC4C4CC54)=O)C(C3)C2)=O)cccc2nc[nH]c12 c1(CC)nc(C#N)cc(=NCC(C)NC(C2CC3C=CC2C3)=O)[nH]1 c1(C(=O)NC2(C)CN(C(C(C(CC)C)C)=O)C2)cc(OC)c(F)c(F)c1 c1(C(N(CCCNC(=O)C(C)=CC(C)(C)C)CC)=O)ccc(COC)cc1 c1(OC)ccc(NC(c2ccccc2Br)(C)C(=O)N(C)C)cc1 C1(CNC(c2cccc(OC)c2)=O)CC2(CO1)CN(C(=O)CCC(=O)C1CC1)C2 N1(C(c2ccc(F)c(CO)c2)=O)CCC2CN(C(c3ccc[n+]([O-])c3)=O)CCC2C1 S(=O)(=O)(c1cc(Br)ccc1Cl)NC1CCCN(C(Cc2cccc(C)c2)=O)C1 c1(C(=O)NCCCN(C(=O)C=CC2(C)COC2)C)cc(Br)cc2c1OCC2 Cc1ccc2sc(=NCC=CCNC(c3cccn4nnnc34)=O)[nH]c2c1 Cc1ccccc1OCC(=O)N(C1CN(C(=O)CCN2CCC2)C1)C N1(C(C(C)NC(N)=O)=O)CCCN(C(C2CC(F)(F)C2)=O)CCC1 CCCC(C)(O)CC(=O)N1CC(CNC(=O)CC2CCCCC2(C)C)(COC)C1 c1(OC)ccc(C(F)(F)F)nc1NC(N1CCOC(C2CCCC2O)C1)=O c1(C(=O)NCCNC(C(C)C2CCOC2)=O)cccc(-c2cscn2)c1 c1(Cc2cn(CC3N(CC)CC3)nn2)ccc(N)c(F)c1.C1C#CCC(=O)N1 C1(NC(C2C(=C)CCN2C(=O)COC2CCOC2)=O)CC2CCC(C1)C2O c1(CC)ccc(C(=O)NC2CCC2NC(c2cc(N(C)C)nc(Cl)c2)=O)c(F)c1 C12(C(N3CC(C(C)(C)C)OCC3)=O)CCCN1CCC2.c12ccc(s1)C(=O)NC2 C(c1cccn1C)=CC(=O)NC(C(C)NC(C(C1CCCC1)OCC)=O)C CC1CCCC1(C)C(=O)NC1CN(C(c2n[nH]cc2Br)=O)CC1C c1(NC(C(=O)NCCCN(C(C2C(Cl)(C(=O)OC)C2)=O)C2CC2)=O)cccnc1 N1(C(COCCC)=O)CCCC(C2CCCN(C(=O)C(F)(F)C(O)C(C)C)C2)C1 c1(C(N(CC(O)CNC(c2ccn(C)n2)=O)C)=O)cc(Cl)c(F)cc1F N1(CC(C=C)NC(=O)OC)CCC(C2CC(C(=O)OC(C)(C)C)C2)CC1 C12(C(=O)NCc3c(CC)nn[nH]3)CCCC1N(C(C1OCCC1(C)C)=O)CC2 N1(C(C2(C)CCOCC2)=O)CC(C(=O)NC2CCC3(CC3)C2)C(C2CC2)C1 c1(C(N2C(C(C)NC(c3cnnn3C)=O)CCC2)=O)ccc([N+](=O)[O-])s1 c1(C(=O)NCC(C)CNC(=O)C(N2CCCC2)C2CC2)ccc(N(C)C)cc1Cl c12ccccc1C(=O)OC2.c1(CN(C2CCCC2)C)cnc(CC(C)(C)C)s1 C1(NC(=O)CCC(=O)N2CCCC2)COC2(CCCC2)C1.CC1(C)CN1 c1(C(N(CC(CO)(CO)NC(c2sccc2Cl)=O)C)=O)cnc([N+](=O)[O-])n1C C12(C(N3C(C(=O)OC)CC(F)(F)C3)=O)CCCC1CN(C(C1CCCCS1)=O)C2 C(=O)(CCCCC(=O)N1CCOCC1CNC(c1ccc(F)nc1F)=O)OC n1(C(C)C)cc(C(=O)OC(C)C)ccc1=O.N12CCCC(C1)NC(=O)C2=O C1(CNC(=O)Cc2cc[nH]n2)COCCN(C(c2coc(C3CC3)n2)=O)C1 c1(C(N2CCC(NC(CNC(CC=C)=O)=O)C2C)=O)c[nH]c2cc(Cl)ccc12 C(C(C)C(=O)NC(C)CC1CN(C(c2ccn(CCF)n2)=O)C1)OC C1(C(=O)NCC2N(C(c3nccc(C)c3)=O)CC=C2)CN(C)CC(C)C1 N(C1COc2c(Cl)cc(Cl)cc21)C(=O)CN1C(=O)CNC1=O Clc1cc2ccnc(CN(Cc3ccccc3)Cc3cccs3)c2cn1 c1(C(=O)NC(Cn2cc(-c3ccc(C)s3)nn2)C)ccc2[nH]ccc2c1 Cc1cc(C(=O)NC23CCCC(NC(=O)CC4CCCO4)(C2)C3)nc(O)n1 c1(SC)cscc1C(=O)NCC(C)(O)CNC(=O)COCC1CCOCC1 c1(NC(=O)C(Cc2c[nH]nc2O)NC(C2N=N2)=O)cc(Cl)cc(Cl)c1.C1(S)CCCCO1 N1(OCC)CCN(CC(N2CCC(C(O)C(F)(F)F)CC2)=O)C(=O)C1=O Cc1nc(N2CC3CC3(C(=O)NCc3cc(O)nc(O)n3)C2)c2c(n1)CCC2 S(=O)(=O)(c1ccc(NC2CC(n3cccn3)C2)c(F)c1)NCC(C(C)(C)C)CO C1(NC(C2(NC(C3(n4nccn4)CC3)=O)CCCC2)=O)CC2(CCC2)C1O Cc1cc(C(=O)NC(C)CCCCNC(=O)CCC2CC2C)cc(N)c1 CN1CCN(C(C2(C)CCCS2)=O)C(C(=O)NC2CC(F)(F)C2)C1 C(CCCC(C)NC(=O)CN1CCCCCC1)NC(CN(CC(C)(C)C)C)=O N1(C(=O)CC2CCCC2O)CCCN(C(c2cscn2)=O)C(c2ccccc2)C1 c1(N(C)C)c(F)cc(C(=O)N(CCCOc2ccc(Br)cc2C)C2CC2)cc1F C1(NC(c2n(C)c(S)nn2)=O)CCCN(C(=O)CCc2ccc(Cl)cc2)CC1 CC1CC(CCNC(=O)C=CC2CC2)CCN1C(=O)CSc1nnnn1C N1(C(Cc2cnc(C)s2)=O)CC2CCC(NC(c3cc4cccnc4[nH]3)=O)C2C1 N(C1c2ccccc2CC1NC(=O)CC1=NNC(=O)C1)C(C=C(C)c1ccco1)=O N1(C(C2CN(Cc3c(C)cccc3C)C2)=O)CC2(CC2)C(=O)c2ccccc21 C1(C(N2CC(C#C)(O)C2)=O)CN(C(=O)CN2CCC(C)CC2)CC1C1CC1 Cc1cccc(Cl)c1OCC(=O)NC1(C)CC(NC(=O)Cc2cncn2C)C1 C(CCCCCNC(c1c(C)cnn1C(C)C)=O)NC(CNC(C)=O)=O N1(C(C2(CC=C)CCN(C(=O)C3=NNC(=O)C3)C2)=O)CC2(CCC1CO)CC2 N1(C(CS(CC)(=O)=O)=O)CCC2(NC(=O)C(=O)NCC)CCCCCC12 CC1COc2c(C(N3CCC(C)(NC(C4(n5cncn5)CC4)=O)C3)=O)cnn2C1 Cc1ccc(CC(=O)NC(C(=O)NCC2CCC(=O)NC2)c2ccoc2)c(F)c1 CCC(C)(C)CC(=O)NCc1nc(C2CCCN2C(C2C(F)(F)C23CCC3)=O)n[nH]1 c1(C(=O)NCCN(C(C(C2CC(F)(F)C2)OC)=O)CC2CC2)c(Cl)n[nH]c1C1CC1 c1(C(=O)NC(CC(=O)N(C)C2CC2)Cc2cccs2)n[nH]c2ccc(C#N)cc12 C1(C(N(C)CC2CC2)=O)CN(C(C2CC2c2ccco2)=O)CC1(C)C CCCS(=O)(=O)CC(=O)N1CCCC1(C)c1cn(CCCO)nn1 C1(NC(C2C(c3cn(C)nc3)C2)=O)CC2(C1)CC(CNC(C1CCC1)=O)C2 C(=O)(CCCC(C)(C)C)N(CC(=O)NCCc1nccs1)CC#C c1(NC(C2(C(=O)NCCCNC(N)=O)CC2)=O)cc(-c2ccoc2)on1.C1(C)CCC1 c1(C(C(N2CC(CC)C(NC(=O)CC(C)OC)C2)=O)(F)F)c(F)cccc1F C1(NC(C2CC3CCC(C2)O3)=O)CC(O)CN(C(=O)CCN2CCCCC2=O)C1 C1(NC(Cc2cnc(C)[nH]2)=O)CN(C(C2(C)CC(C(C)C)=NO2)=O)CC1N=[N+]=[N-] C1(NC(c2cn(C)c(C(F)F)n2)=O)CCSC12CN(C(C1CCCO1)=O)C2 C1(CC2CN(C(CSC)=O)C2)CCCCN1C(=O)CN1CCN(C)CC1 C1(CNC(=O)CC(O)C2CC2)CCC2(CCC2)C1NC(C1C(F)(F)C12CCC2)=O c1(C(=O)NCCCC(CO)NC(C2(CC)COC2)=O)cc2c([nH]1)CCCC2 C(CCCC(=O)NCCC1CC(C)(C)CO1)NC(CC(=O)NCC)=O c1(C(C(=O)NCC2(O)CC(NC(=O)CCCC3CC3)C2)(F)F)ccc(F)c(F)c1 C(=O)(C1=C(Cl)CCC1)NCC1CCC(NC(C2(CC)CCC2)=O)C1 C1(NC(COCCC=C)=O)CCC12CN(C(=O)C(C)Cc1ccc(Cl)cc1)C2 N1(C(C)=O)CCC(C)(NCCCC2CCCN2C(c2cc(C)nn2C)=O)C1 N1(C(CCc2c(C)noc2C)=O)CC(N(C(=O)CC2CC3CC3C2)C)C2(CC2)C1 N1(C(C(C2CCCN(C(c3c[nH]c(=N)o3)=O)C2)C)=O)CCC12CCN(C)C2 c1(C(=O)NCC(C(C)C)NC(c2csc(Cl)n2)=O)cccc2ccsc12 N1(C(C)=O)CCC(N=c2[nH]c(=NCC3COCC3(C)C)c3[nH]ccc3[nH]2)CC1 C(=O)(C(C(C)OC)N(C)C)NCCNC(C1CC(O)(CC#C)C1)=O c1(-c2n(CC(N3CCN(CCC(C)F)CC3)=O)ccn2)cc(N)ccc1F c1(CC(=O)NCC23N(C(=O)CNC(C)=O)CC(CC)(C2)C3)cccc([N+](=O)[O-])c1 c1(C(=O)NC(CNC(C(COC(C)C)NC(C)=O)=O)CO)nc(C)c(C)s1 CC1(CNC(=O)CCc2ccsc2)CCC(NC(=O)C=CCN2CCCC2)C1 C=CC1(C(=O)O)CCN(C(=O)CCCc2cn(-c3cnccc3Br)nn2)C1 C1(CNC(=O)CCOC2COC2)CC2(CC2)CN1C(c1cnccn1)=O CC(C)CN=c1[nH]c(C(N2CCSCC2c2nn[nH]n2)=O)cs1 C(=O)(C(F)(F)CCn1cc(-c2cc[nH]n2)nn1)NC(CC(C)C)Cc1ccccc1 CC1CN(C(C2CN(c3nncs3)C2)=O)C(C)CN1C(C1SCCS1)=O CC1(C)CN(C(=O)CCN2CCC2)CC(CNC(c2cc(N(C)C)ccn2)=O)O1 C1(CNC(C(C(C)C)C2CCC(=O)N2)=O)CCC12CCN(CC1CCN1C)CC2 c1(C(=O)NCC(CC)NC(C2(c3ccc(O)nc3)CC2)=O)nc2ccc(Cl)nn2n1 C#CCC(C)(C)C(=O)NCCCC1CN(C(=O)C(F)CC)CCO1 c1(NC)ccc(C(=O)NCCCC2(NC(=O)C(F)CC3CCC3)CC2)cc1F C=CCCCCC(=O)NC1CCN(C(c2c[nH]c(=N)s2)=O)C1CC N12CCCC(CC1)CNC(=O)C1(CCC1)C2=O.C1(CCOCC)(CCC)CCCC1 N1(C(c2cncc(N)c2)=O)CCCCCC1CNC(c1conc1C1CCC1)=O c1(C(N(CCCN(C)C(C2CCN(C(C)=O)CC2)=O)CC)=O)ccc(C)c(O)n1 C1(C(CNC(C2(C#C)CC2)=O)(C)O)CCCN(C(=O)CC2CSCCO2)C1 N1(C(=O)COCc2ccccc2Cl)CCOCC1CNC(C1CCCS1)=O N1(C(Cc2cc(C)nn2C)=O)CC(O)CCC1C(=O)NC1(CO)CC(O)C1 N1(C(CSCC#C)=O)CC2CC2(NC(c2ccnc(N(C)C(C)=O)c2)=O)C1 c1(C(=O)NC2(CCOC)CCN(C(=O)C#CC(C)C)C2)nc(C)n2c1CCCC2 c1(C(N2CCC(C(=O)NCCN(C(CCCC)=O)CC)C2)=O)cnc(OC)nc1 c1(NC(=O)CCOCCNC(=O)C2=CCCC2)cnc2n1CCC2 C1(NC(C2(COC)CC2)=O)CCC2(CC1)CC(NC(c1nccc(Cl)c1F)=O)C2 c1(C(C)(C)C)ccc(-c2cnc(C(=O)NCCNC3CCC3)cn2)cc1 C(=O)(CCC(C(=O)N1CCOCC(NC(=O)C(C)(C)N2CCCC2)C1)N(C)C)OC C1(NC(Cc2cccc(COC)c2)=O)CC(C)CN(C(=O)C2=CCCSC2)C1 C(CCCCCC(=O)N(CCN(C(=O)Cc1csc(C)n1)C)C(C)C)SC CC(C)(C)C(=O)CN=c1[nH]c(=NCc2cnns2)c2sccc2[nH]1 C1(NC(C(F)=CC)=O)CC(C)CN(C(=O)Cn2cc(CO)nn2)C1 C1(NC(C(C=C)O)=O)COCCN(C(=O)CC=Cc2cccc(F)c2)C1 C(C(C(C)C(C)C)NC(c1ccc[n+]([O-])c1)=O)NC(C12CC(CSC)(OC1)C2)=O C(CCC(=O)NCCC(CNC(=O)Cc1ccnn1C1CCC1)OC)OCCC C1(CNC(c2cnn(CC)n2)=O)CC(O)CN1C(=O)CCCc1ncc(C)o1 c1(COC)cncc(C(N2CCC(Nc3nccc(OC)n3)C2C)=O)c1 C#CC1(C(=O)NCC(C(C)C)NC(C2CCC(=O)N2)=O)CCCC1 C(=O)(C1CCCc2cncn21)NCCC(C)NC(=O)CC1(C)OCCO1 Cc1ccc(C)c(OCCC(=O)NCC2(NC(c3nc(C)sc3C)=O)CCC2)c1 N1(C(c2c(C)nsc2)=O)Cc2ccnn2CC(NC(c2cc(C(C)C)[nH]n2)=O)C1 C(C)(CNC(C1(C)CCNC(=O)C1)=O)(CC(C)C)NC(c1cc(OC)n(C)n1)=O O=C1Cc2c(C(N3CCCC3C(=O)N(C3CC3C3CC3)CCO)=O)cccc2N1 Cc1cc(Br)cc(C)c1CC(=O)N(C)CCNC(=O)C(C)O CCCCC(C(=O)N1CCCC(F)(F)C1)NC(c1ccc(O)c(C)c1)=O c1(C(C(=O)NCCCC2(NC(C3C(=C)C3)=O)CC2)CO)ccc(Cl)cc1 O=C(CCn1cncn1)NCC(=O)N(CC(=O)C1CCC1)CC(F)Cl N1(C(CC(C)C2CCC2)=O)CC2CCCC(CC(=O)O)C2C1 N1(C(CCCCNC(C(CCC=C)(F)F)=O)=O)C2CCCC1CC(O)C2 N1(C(C2(C(C)C)COC2)=O)CCC(C2CCN(C(=O)C(C(C)C)NC=O)CC2)C1 c1(C(=O)NC2C3CN(C(c4c(C)ccs4)=O)C2C3)ccc2c(c1)C(=O)OC2 N1(C(c2cc(C(F)(F)F)[nH]n2)C(=O)NCCC#N)CCOCC(O)C1 c1(C(=O)NCC2COC(C(F)(F)F)CN2C(=O)C(F)F)cccc(C(F)(F)F)c1N CC1(C)OC2CC(C(=O)NC3CC(NC(c4ccc(F)c(CO)c4)=O)C3)CC2O1 c1(OCC(=O)NCCCC2(NC(C3C(C=C)C3)=O)CC2)c(C)cc(C)cc1C c1(CC)ccc(C(=O)NCC(CNC(C2(O)CCCCCC2)=O)CO)c(Cl)c1 C#Cc1ccc(NC(=O)CCNC(=O)CC2CCOC2C)cn1 C(=O)(C(F)(F)C(C)(C)O)N(C1CC1)CC1N(C(c2c(C)cc(CO)o2)=O)CCC1 c1(C(N2CC(C)C(C(=O)NCC(C)(O)COC)C2)=O)cccc2[nH]ccc12 Cc1ccc(F)cc1CC(=O)NCC(N1CCCC(CN(C)C)C1)=O.C(CO)N CC1(C)CCC(C(=O)NCC2(O)CN(C(=O)CCCCN3CCCC3)C2)OC1 N1(C(CC2C(CC)C2)=O)CC2CC1CN2C(=O)C=CC(=O)N(C)C C1(C(N2CCN(C(C=C(CC)CC)=O)C(C)C2)=O)CC12C1CC3CC(C1)CC2C3 c12cc([N+](=O)[O-])ccc1C(=O)N2.c1(C(=O)OC)nccc(SC)n1 C12(NC(C3N(C(C)=O)CCC3)=O)CC1CN(C(=O)CCCOC(C)C)C2 c1(-c2ncc(C(=O)NC(C(C3CC3)OCC)=O)s2)cc(C)cc(C)c1.C1CCC1 C(C)(C)(CC(F)C(=O)NC1(CO)CCCC1C)NC(Cc1c(C)ncs1)=O C1(CNC(C=CCC)=O)CCC(C(N2CCC(CC(N)=O)C2)=O)O1 N1(C(C=CSC)=O)CCCN(C(c2ccc(C(F)(F)F)c(F)c2)=O)C(C)C1 N1(C(C(CCC)CC)C(=O)NC2CCC2)CCC2(CC1)CNC(=O)O2 c1(CC)c[nH]c2cc(C(N3CC4CC4C3)=O)ccc12 C1(C(=O)NC(CN(C(COCC(=O)NC)=O)C)C)CCCCC1n1cccn1 C1(NC(C(CC=C)(C)C)=O)Cc2ccccc2C1NC(C1CC(C(C)(C)C)C1)=O C1(CN(C(=O)C(O)C2CCCC2)C)CSCCN1c1nnc(C(C)(C)C)s1 N1(C(c2ccc(C)o2)=O)CCCC(C)C1CNC(c1cscn1)=O C1(CN(C)C(C2(F)CCC2)=O)CCCN1C(=O)CC(C)C1CCCO1 CC1CN(C(=O)CC2(C)CCOCC2)CC1(C)CNC(=O)CSc1nncn1C N1(C(c2nncc(C)c2)=O)CCOCC(NC(c2nc(F)ccc2Cl)=O)C1 c1(C(=O)NCCN(C(c2c(OCC)nn(C)c2)=O)CC)c2c(nn1C)CCC2 C1(CC#C)CCN(C(=O)CN(C(=O)Cc2cnccc2C)C(C)C)CC1 C1(C(=O)NC(CN(C(c2ccc(C(N)=O)cc2)=O)CC)C)CCC2(CCC2)CO1 C1(OCC(=O)NC2CCCN(C(C3COCCOC3)=O)C2)CCS(=O)(=O)C1 C1(NC(C(c2cccnc2)NC(C2CC(CC)C2)=O)=O)C=CCCCC1 C1(C#N)(C(N(CC(CN(C)C(c2c[nH]nc2Br)=O)O)C)=O)CCCO1 Cc1cc(C)nc(NC2CC(C)CN(C(c3cc(N(C)C)ccc3F)=O)C2)n1 c1(C(N2CCCC(C)(NC(c3ncn(CC)n3)=O)C2)=O)noc2c1CCCCC2 N1(C=O)CC(C(=O)OC)c2ccccc21.N1(C(=O)NCCOC)CCCC1 CC1OC2(CO)CC1(C(=O)NC(CNC(C1CCCN1C=O)=O)CO)C2 N12CC3(CCC(O3)C1=O)C2.Cc1cc(C(=O)OC)cc(C2CC2)c1.C1(C)C(=O)N1 Cc1cc(C(N2CC(N(C)C(c3cc(Cl)ccn3)=O)C(O)C2)=O)ccc1Cl C1(CNC(C(C)(C)CO)=O)CCC2(CCC2)C1NC(c1cc2c(s1)CCC2)=O C1(C(=O)NC2CC(SC)C2)CC(C)CN(C(=O)CN(CC(C)(C)C)C)C1 C(CC)(CC(=O)N(C1CC2CC2C1)C)NC(CN1CC(C)(OC)C1)=O c1(CC(=O)NCC2C(CNC(C3N(C)C(=O)CC3)=O)C2)cccc2c1CCC2 N1(C(CCOC)=O)CCN(C(c2ccoc2C)=O)CC1 C1(CCNC(CCN(C(CC2(CC)CCC2)=O)CCOC)=O)CCCCC1 C(CC(=O)NC(C)CC(N)=O)(C(F)(F)F)NC(c1c(C)occ1)=O C(=O)(C#CC(C)(C)CNC(C1CC(=O)CS1)=O)N1CCC(C(C)OC)CC1 CC(C)(CCC(=O)N1CCCC2(NC(c3ccc(C(N)=O)s3)=O)CC2C1)[N+](=O)[O-] C1(C(=O)NCC(C)C2CCC2)(CO)CN(C(c2ccc[nH]2)=O)C1 C(CCC(C)(C)C(=O)NC1CCC(C)CC1)NC(C(C(=O)OC)C)=O C=CCCCCCC(=O)NCC(CNC(c1cc(F)cc(Cl)c1N)=O)C(F)(F)F c1(C(=O)NCc2onc(C)n2)nccc(Cl)c1C CCC(CC(=O)N1CCC(CC(=O)N(CCC(C)F)CC)C1)C1CCC1 C=CCCCC(=O)NC12CCN(C1)C(=O)C1CCN(CC1)C2.c1(NC)ccc[nH]1 c1(C(N(C2CC(CNC(C(C)N(C)C)=O)C2)C)=O)cc(F)c(N)c(F)c1 N1(C(c2nc(C)sc2C)=O)CCN(C)C(C(=O)NC(c2cccs2)C)C1 N1(C(C(CC)C)=O)CCCC(C2CC2NC(=O)C(c2cccc(F)c2F)(F)F)C1 N1(C(CC=C)=O)CCCC(C)C1CNC(c1ccsc1COC)=O C(C)(CCCC(=O)NC1C2CCC(F)(F)C12)n1cc(CCC(C)O)nn1 S(=O)(=O)(c1ccc(-c2ccc(N)c(Cl)n2)cc1)NCCN=[N+]=[N-] N1(C(C=C(CC)CC)=O)CCN(C(=O)CCc2cn(CC)nn2)CC1CCC Cc1cc(NC(=O)C(N2CC(c3cc(C)n(C)n3)(O)C2)=O)c2[nH]cnc2c1 N1(CC(=O)NC(C(=O)NCCC(C)C)C)CCCC(C)(Cc2ccc(N)cn2)C1 Cc1nc(O)nc(C)c1CCC(=O)NC1CC2CC1N(C(C1CCNC1=O)=O)C2 N1(C(c2c(C)nn(C)c2)=O)CC(C(=O)Nc2csnc2CC2CC2)OC(C)C1 c1(C(=O)NC2(CC=C)CN(C(C3(C)CC3(F)Cl)=O)C2)cc2cnccc2o1 c1(C(N2CCNCC(O)C2)=O)cc2ccccc2cn1.c1(OCC)nc(OC)ns1 C1(NC(C(C2CN(C(=O)COC3CCCCC3)C2)OC)=O)CN2CCC1(C)CC2 N1(C(COc2cccc(OC)c2)=O)CCC(C2CC(NC(=O)C(C)(C)C#N)C2)C1 CC1(C)CN(C(c2ccc(Br)cc2O)=O)CC1NC(C1CC1F)=O N1(C(=O)CC2CSC2)CCC2(CC1)CN(C(C1CC3CCC1C3)=O)C2 c1(OC)ccc2c(c1)C(C(=O)OC1CCCC1)CC2.c12ccc(F)cc1NC2=O Cc1ncoc1NC(C1(C)CC(C)C1)=O.N12CCC(C1)CN(C(C)C)C(=O)CC2 c1(C(N(C(C)CNC(C)=O)CC)=O)cnn(CCc2cc(COC)on2)c1 N1(C(c2c(OC)cccc2)=O)CCC(C)C(CNC(c2ccc(OC)nn2)=O)C1 C1(C)(CNC(COCCOC)=O)CN(C(c2cc(C(C)(C)O)ccn2)=O)CCO1 c1(C(=O)NC2CN(C(c3cc(CC)c(CC)o3)=O)C(C)C2)cnc(C)c(C)c1 Cc1ccc(Br)c(C(=O)NCC(C2CC2)NC(=O)C2=CCCCO2)c1 N1(C(COCCCCC)=O)CCC(O)(CCNC(C2(C)CC2(C)C)=O)C1 CC1CC(=O)CCC1C(N1CCC1CC(=O)NCC(O)CNC(N)=O)=O c1(SCC)cccc(C(=O)NCC2NCCC2)c1.c1(C(=O)N)cnn(C)c1C1CC1 C12(C(N3CC4C(NC(CCCC)=O)C4C3)=O)CC3CC(CC1C3)C2 c1(CC)ccc(C(C)C(N2CCCC(OCCF)C2)=O)cc1.C12(CC1)C(=O)NC2 C1(CC)(CNC(c2nnnn2C(C)C)C2CCOCC2)CCCCC1 c1(OC)cc(F)c(C(N2CCCC2(C)C(=O)NCc2cccc(Cl)c2)=O)cc1OC C(=O)(C1=CC2(CN(C(c3cc(C#N)[nH]c3C)=O)C2)OC1)NCC1(OC)CCC(C)C1 N1(C(C2(CC=C)CCCC2)=O)CC2COCC2(C(N2CCN(C)C(C)C2)=O)C1 C(C(COC)CC(=O)N1CC(CNC(c2ncc(C)cc2C)=O)CCC1C)OC N1(C(c2ccn(C)c2)=O)CCCC(O)(CNC(=O)C=CC(c2ccccc2)=O)C1 N1(C(c2c(C)c(C3CC3)on2)=O)CC(NC(C2CC(F)C2)=O)CC(C)(C)C1 Cc1cn2cc(CC(N3CC4=C(C3)CN(C(c3nc(Cl)cs3)=O)C4)=O)nc2s1 c1(C(=O)Nc2ccccc2C2CCN(C(C3(Br)CCC3)=O)C2)cc2sccc2s1 N1(CC2C(CC)C2)CCn2nc(C)c(CNC(C3(C)CCCNS3(=O)=O)=O)c2C1 N1(C(C=COCC)=O)CC2CC1CN2C(C1CC(n2cc(C(=O)OCC)cn2)C1)=O C1(C(=O)NCC2(OC)CN(C)C2)CC2(CC2)CN1C(C1COC(=O)N1C)=O c1(OC)ccc(C(=O)NCCC2(OC)CN(C(C3CCC(O)C3)=O)C2)c(F)n1 C(=O)(C(=O)N=c1ccn(-c2cccnc2)[nH]1)N1C(c2n(CC)nc(C)c2)CCC1 N1(C(c2c(CC)noc2)=O)CCC(C2CCN(C(=O)Cc3cccnc3O)C2)C1 c1(-c2cn(C(C)(C)CC3CCC3)nn2)ccc(NC(=O)C(F)F)cc1 c1(CC)ccc(C(N2CC(O)(CNC(=O)C(C)(C)C3CCCC3)C2)=O)o1 c1(C(C)C)ocnc1C(=O)NC1CCC1NC(c1cc(Br)sn1)=O c1(C(=O)NC(CN(C(=O)C=Cc2ccc(C(F)F)o2)CC)C)cccnc1OC CC12CCN(CC1)C(=O)C1CCN(CC1)C(=O)CC(=O)N2.C1(OC)CC1 C(CC(CC)(CC)NC(C1CC1F)=O)NC(C1(CC=C)CCOC1)=O c1(CN2C(NC(c3ccc(O)cc3F)=O)CC(OC)C2)cc2ccc(Br)cc2[nH]1 C(=O)(C(O)C(F)F)NC(C1CCCCC1)CNC(C1C(c2cn(C)nc2)C1)=O C1(C(=O)O)(CC)CCN(C(C2CN(Cc3cnc[nH]c3=N)CCC2O)=O)CC1 c1(C(N2CC=CC(C(N(C3CNC(=O)C34CC4)C)=O)C2)=O)ccc2c(c1)CCC2 CC1CN(C(c2csc(CNC(C3CCC(CO)CC3)=O)c2)=O)CC(C)O1 c1(N2CCC(C(=O)Nc3cc(C(C)C)nn3C)C(C)C2)ncc(Cl)cc1[N+](=O)[O-] O=C(C1=CCN(C(c2ccnc(O)c2)=O)C1)NCCC1CCCOC1 Cn1nc(CC(=O)NNC(=S)NC2CCOC2)c2ccccc2c1=O N1(C(C=C(CCN(C)C)Cl)=O)CC(NC(=O)C(c2cncnc2)C)CCC1C Cc1cc2c(C(=O)NCCN(C)C(C3Cc4nccn4C3)=O)ccc(C)c2[nH]1 C1(CNC(c2cncc(CNC(c3ccc(CO)cc3)=O)c2)=O)CC(F)(F)CO1 C1(NC(=O)NCC(=O)C2(c3cccnc3)CC2)CC(=O)N(C2CC2)C1 C#CC(CC(C)C)NC(C1(COC)C=CCN1C(=O)CCc1ccncn1)=O Cc1cc(Br)ccc1Oc1cccc(C(=O)NCC2CCC2c2ccccn2)c1 c1(C(=O)NC2CC3(CN(C(CCc4ccc(C)s4)=O)C3)C2)cnc2nccn2c1 C1(C(N2CC(OCCCC(=O)Nc3cc(Cl)cc(Cl)c3)C2)=O)CN2CCC1CC2 c1(C(=O)NC2(C(N(CC(C3CC3)OC)C)=O)CCN(C)C2)cnc(C)cc1C CC1COC2(CCCC2)CN1C(C(=O)NCC(F)F)C(C)CC1CCC1 C12(CNC(CCc3ccnc(C)n3)=O)CCC(C(=O)NCC3CC3C)(CC1)OC2 CC1OC(=O)NC1C(=O)NC12CC(NC(c3cnccc3Cl)=O)(C1)C2 Brc1cccn2nc(-c3nc(CC4CCCOC4)nn3C3CCSC3)cc12 c1(OC)cc(OC)c(NC(C2(C)CCCN(C(=O)CC3(O)CCC3)C2)=O)cn1 N1(C(c2ccc(CC)s2)=O)CCC(C)(CCNC(c2ccn(CC(C)C)n2)=O)C1 C(=O)(CC1=CCOCC1)NC1C(C)CCN(C(=O)C=CC(=O)N(C)C)C1 C1(C)(C(=O)NC2C(C(=O)OCC)CCC2)CCCN1C(C1C2COCC12)=O c1(C(C(C)C)C2CC2)nc(-c2ccc(-c3cccs3)cc2)nn1-c1nccn1C c1(C(=O)NCC2N(C(c3cc(C)sn3)=O)CC(O)C2)ncc(C(F)(F)F)cc1N C1(C)(CCC)CCN(C(C2(F)CN(C(c3ccncn3)=O)C2)=O)C1 C1(NC(C=C(C)C2CC2)=O)CC(O)(CNC(C2CCO2)=O)C1 c1(C(N(CC(O)CNC(C2(CC(F)F)CC2)=O)C)=O)ccc(CO)cn1 Cn1cnc2c(N(C3CNCC3F)C(c3cc(O)c(Br)c(O)c3)=O)ncnc12 Cc1ccc2cc(C(=O)N(CC(C)N(C(=O)Cc3ccnn3C)C)C)cnc2c1 C1(=O)C(CC(C)C)CN1.N1(CC(=C)Br)CCC(OC)C1 c1(C(=O)NCCCN(C(=O)COC)CC)ccc(-n2nc(C)cc2C)nc1 N1(C(CC(CC2CCCC2)OC)=O)CCOCC1C1(c2ccn(C)n2)CC1 c1(SC)ccc(CNC(C2CC3CC3N2C(=O)C(c2ccccc2)C)=O)cc1 N1(C(C)=O)CC2CC2(CNC(C2CCOC2c2cnn(C)c2)=O)C1 c1(OC)nc(=NC(=O)Nc2ccc(Nc3cc(Cl)cc(I)c3)cn2)nc(OC)[nH]1 C1(N)CCCN(C(=O)CC2CCCN2C(=O)CCC)C1.C(COCCO)OC CCCC(CCCNC(C1(OC)CCCC1)=O)NC(c1cc(C)nc(C)n1)=O C#CC1(C(N2CC(C)(O)C2)=O)CN(C(=O)C(C(=O)OCC)OC)C1 N1(C(C2N(C)CC(F)C2)=O)CC(CNC(c2cnsc2)=O)OC(C)(C)C1 S(=O)(=O)(CCC(=O)NCCN(C(=O)C1=CCSC1)C)N.C(=O)(CO)NC(C)=O c1(C(N2CC(CNC(Cc3c(C)ccs3)=O)C(C)CC2)=O)cccc2c1CCC2 N1(C(c2occ(C)c2)=O)Cc2n[nH]cc2C1C(=O)N1CCNC(=O)C1CCO c1(C(=O)NC(C2(NC(=O)C(C)OCCN(C)C)CC2)C)cc2c(cn1)OCCC2 N1(C(C)=O)CC(O)CC1CNC(CC1COCCN1C(C1CNC(=O)N1)=O)=O N12CCCC1(C)C2=O.C1(C(CNC(C=C(C)C(=O)O)=O)=O)CCOCC1 Cc1cc(C(=O)NCC(C)N(C(=O)CCc2c(Cl)cncc2Cl)C)ccc1Cl c1(NC(N2CCSC(C)C2C)C(=O)Nc2c(OC)cccc2)cc([N+](=O)[O-])cc(C)n1 c1(C(=O)NC(C)CCCNC(C2CC3CCC3C2)=O)ccc(N)c(F)c1Br c1(CC=C)ccccc1C(=O)NCC(C)(CO)NC(=O)C(N1CCOCC1)C C(CCCC(=O)NC1(C)CC=CCC1)NC(C(C1CC(OCOC)C1)SC)=O c1(C(=O)NC2(O)CCN(C(=O)NC3COC3)C2)cccc2c1OCCO2 C1(N(C(CN(CC)CC)=O)CC)CCCN(C(=O)CC(=O)NC2CC2)C1 c1(NC(CCC(C)NC(=O)C(C)(C)F)=O)cccc2[nH]ncc12 CC1CCC(NC(=O)CCCOC(=O)N(C)C)CN1C(c1nnc(O)n1C)=O c1(NC(C2(C(=O)NOCC3CCOC3)CC(C)(C)C2)=O)ccc(F)cc1F C(C(C)(C)C(=O)N(c1ccnc(Br)n1)C1CNCCOC1)OC c1(CN2CCOCC(NC(C=Cc3cnc(C)s3)=O)C2)c(F)ccc(O)c1F c1(C(N2C(CN(C(c3c(CC)ocn3)=O)C3CC3)CCC2)=O)ccc(O)c(N)n1 c1(OCC(=O)NC2CC(F)(CNC(C=C)=O)C2)cc(C)c(Br)c(C)c1 C1(NC(C(n2ccc(C)n2)C)=O)CCC2(CC1)CN(C(=O)C=CCF)CCO2 CCC(C)C(C(=O)NCC1(C)CCN(C(C2CCC(=O)N2CC)=O)C1)OC C12(C(=O)OCC)CN(C(c3cnc(Cl)s3)=O)CC1CN(C(=O)CN(C)C(C)C)C2 c1(CC(=O)NCC2C=CC(NC(C(CC)C(=O)OC)=O)C2)ccc([N+](=O)[O-])cc1 N1(C(CCCC(=C)C)=O)CC(C2CN(C(c3cn(CCCOC)nn3)=O)C2)C1 c1(C(CSCC)=O)ccccc1.C12(CCC1)C(=O)NCCO2.C1C(=O)N1 C1(C(=O)NCCCCCN(C(=O)CCCCC(N)=O)C)C2CCCC(F)(F)C12 c1(C(=O)OC)ccc(C(=O)NC2CCC(CN(C)C(C)=O)CC2)cc1O c1(CNC(=NCC)NC2CC(C(C)C)NC2=O)cnc2[nH]cnc2c1 CCCCC(C)(F)C(=O)NCC1CC2CC(C1)N(C(=O)CC1CCSCC1)C2 C(=O)C(C)CC(F)(F)F.C=CC(C)(O)C(=O)NCCOCCOCCOCCOC CC(CCCCNC(c1cc(Br)no1)=O)NC(=O)C(C1CCOCC1)F C(=O)(C1CCCc2nccn21)N1CCC(O)(C(C)NC(c2cnnn2C)=O)C1 c1(CC)cccc(C)c1C(=O)NCC(C)NC(=O)CC1CC(C)OC1C c1(C(=O)NC(C)CNC(=O)CCc2ccc(F)nc2)cnc2ccc(F)cc2c1 c1(C(=O)NC23CC(CNC(CC(=C)C)=O)(C2)C3)cnn(C)c1COC N1(C(C2CCC(CO)O2)=O)CCN(C(c2cccc[n+]2[O-])=O)C(c2ccccn2)C1 c1(N2C(=O)CC(C(N(C)CC3CCN(C(=O)C(N)=O)C3)=O)C2)cc(Cl)cc(Cl)c1 c1(C(=O)Nc2c(-n3cc(CNC(=O)NC)nn3)cccc2)cc(Br)c(C)cn1 FCCN=c1[nH]c(=NCC2CC3(CCC3)CCO2)[nH]c2ccccc12 CCS(=O)(=O)c1ccc(CC(N2CC(O)(N(C(=O)C(C)(F)CC)C)C2)=O)cc1 CC(C)CCC(O)C(=O)N1CCC(C)(CCNC(C23CCC(C2)C3)=O)C1 C(=O)(C(F)C(C)(C)O)NCC1(C)CCN(C(c2ccn(CCO)c(=O)c2)=O)C1 c1(C(N2C(CCNC(C3NC(=O)OC3)=O)CCC2)=O)cc2nn[nH]c2cc1F C#CCC(C(=O)NC(=O)C=CC(C)(C)C)NC(=O)CC1CCC(C)(C)C1 C1(NC(C(C)(C)n2cncn2)=O)CC2(C1)CC(CC(=O)NCC1(F)CCOC1)C2 C(=O)(CC(C(F)(F)F)OC(N1CCCC(OC)C1)=O)NCc1ccc(OC)nc1 CC1Cc2cc(F)ccc2CN1N1CCN(CCC(=O)N(C)C)C(=O)C1 N1(C(C(C#N)=CC(C)C)=O)CC2CCC1C(NC(c1cnc(C3CC3)s1)=O)C2 c1(N2CCCC(NC(C3C(OCC)C3)=O)(CO)C2)nc2ccc(O)cc2s1 c1(C(=O)NC(C)C(CO)NC(=O)CC(=O)N(C)C)cc(Cl)ccn1 c1(OC)ccc(C)c(C(=O)NC(C)CC(C)NC(=O)C=CCOCC(F)(F)F)c1 CCC(C(=O)N1CCC(C)C(NC(c2ccnc(OC3CC3)c2)=O)C1)C(C)O c1(C(N(CCN(C(CCC=C(C)C)=O)C)C(C)C)=O)ccc(F)c(F)c1C CCC1=NOC(C(N2CCOCC2CNC(c2cnc(S)n2C2CC2)=O)=O)C1 CN1CCOC(C(=O)NCC2CC2c2cccc(OC(F)(F)F)c2)C1 C1(C(=O)NCCOC2CCN(C(c3cn(C)nc3Cl)=O)C2)CN(CP(C)(C)=O)C1 N1(C(CCC)=O)CC2CC(C1)C2NC(C1CC2(CCO1)CC2)=O c1(C2(Cc3n(C(C4CCCN4)C)ccn3)CC(N)C2)ccccc1F FC1(F)C(c2cn(CCNC3CC4(CC4)C3)nn2)C12CCCC2 c1(C(=O)OCC)ccc(C(N2CC=CC2CNC(=O)C=Cc2cc[nH]n2)=O)cc1C c1(CC)ocnc1C(=O)NCC1(F)CC(CNC(=O)CC2OCCC2C)C1 c1(NC)ccc(-c2cn(Cc3csc(CS(=O)(=O)CCN(C)C)n3)nn2)cc1F c1(C(C(N2CCC(OC(C)=O)C2)=O)NC(=O)CC2CC=CC2)ccc(Cl)cc1 C(=O)(NNc1cccc2c1CCC2)c1c(OC)cccc1OC CCC(C)C(CC(=O)N(C1CCC1(C)C)C)NC(=O)CCCn1cncn1 N1(C(CCn2c(C)ncc2)=O)CCC2(CCCC2C(N2CCCNC(=O)C2)=O)C1 C(C1CCCCC1)=CC(=O)N(CC(=O)NOCc1cnn(C)c1C)CC#C c1(OC)ccc(CCCNC(c2coc(Cl)c2)c2nnnn2CCSC)cn1 c1(NCC(C)NC(=O)CCc2ccccc2Br)c(Br)cc(Br)cc1Br N1(C(C2CCC(O)CC2)=O)CCC2C(C1)CN2C(c1cc(Br)c[nH]1)=O CC1CCN(C(C2(CN(C(C3CCC(C(F)(F)F)C3)=O)C3CC3)CC2)=O)CC1(F)F c1(C(N2CCC(C(C)NC(=O)CC(C)(C)C#N)C2)=O)ccc(F)cc1O C1(C)(C(N2CC=CC(NC(c3c(Cl)c(C)n(C)n3)=O)C2)=O)Cc2ccccc2C1 C(C1CN(C(=O)C(C)NC=O)Cc2ccccc21)NC(c1c(C(C)C)c[nH]n1)=O C1(C(=O)NCC2(CN(C(CC(C)=C(C)C)=O)C)CC2)CCCC(C)C1 c1(OCC)cncc(C(=O)NCC(CNC(=O)C(c2ccc(C)cc2)O)CO)c1 c1(CC(=O)NC23CCCN(C(=O)CN4CCC4)CC2C3)ccc2c(c1)CCCC2 C=C1C(C(=O)NC2(C(N3CC(C)C3)=O)CSC2)C1.n1(C2CCC2)nccn1 N1(C(c2cncc(C)n2)=O)CCCCC12CC(NC(C1CC1C#N)=O)C2 c1(CC(=O)N(CC(CO)(CO)NC(C(C)SCC)=O)C)cc(F)ccc1O C1(N(c2ccccc2)C)CN(C(=O)C(=O)N(CC(C)(C)C)C)CC1OCC1CCC1 C(CC(C(=O)N(C1CCCC1C#N)C)NC(C1CCCSC1C)=O)OC Cc1conc1CC(N1CCC(CCC(=O)NC(C(N)=O)C2CCCC2)C1)=O N1(C(C2N(C(C)C)CCC2)=O)C(C(N2CCC(C(C)(C)O)C2)=O)CCC1C N1(C(CC=CC)=O)CCCCC1CCCNC(=O)COCCSC C1(CC)C(CC(=O)NCCC2CCC(NC(c3n[nH]cc3C)=O)C2)C1(F)F c1(CNC(C2CC=CC(NC(c3ccc(C)cn3)=O)C2)=O)nc(C)ccc1C CCCCCCCCC(=O)NC1CCCN(C(C2(CCOC)C=CCC2)=O)C1 N1(C(C2C(C#N)C2)=O)CCC(CCCNC(=O)COC2CC=CC2)CC1 C1(C(=O)NC(C)C(=O)NCCF)CC(C)(NC(c2ccc(Cl)s2)=O)C1 Cc1nccc(N(C)Cc2ccc(C(=O)NC(C3CCCO3)(C)C)cc2)n1 C(CC(F)F)(C(=O)NCCOCCCO)N(C(c1c(CC)nn(C)c1)=O)C c1(OCC(N2CCC(CC(F)(F)F)C2)=O)ccc(CN2CCC(F)CC2)cc1 n1(CCC2C=CC(C)(C)CC2)cnc2sc(-c3ccccc3)cc2c1=O C1(CNC(c2sccc2F)=O)CN(C(=O)C2=CCCOC2)C2CCCCC12 C(=O)(CC(C)(C)N(C)C(c1ncncc1C)=O)NCCNS(CC)(=O)=O CCC(C)C(O)C(=O)Nc1cccc(CNC(c2cnc3occc3c2)=O)c1 C(=O)(C(C)CC(C)C)N1CC(O)(CN(C(C(C(C)C)n2ccc(C)c2)=O)C)C1 CC(C(=O)N1CCCC1C(C)NC(C12CCC(C1)C2)=O)C(C)O c1(C(=O)NCC(CN(C(CSCCN(C)C)=O)C)O)nnsc1C(F)F C(c1cccc(CO)c1)=CC(=O)NC1CCC(C(C)C)C1 C1(C(=O)Nc2cccc(NC(=O)CC3(CO)CC3)c2)CCCCNC1=O C(=O)(C#CC1(C(F)(F)F)CC1)N1CCCC(NC(c2nnc(C)s2)=O)C1 C(C(C(F)(F)F)N1CCN(C(=O)CCCF)CC1)NC(=O)CCC1(O)CCC1 N1(C(CC(C(F)(F)F)NC(=O)OC(C)(C)C)=O)CCS(=O)(=O)C(C)(C)C1 CCC(C(=O)N1CCC(OC(C)(C)C)C1)NC(=O)NC1CCCC1F N1(C(C2CCCN2S(=O)(=O)c2cccnc2)=O)CCc2[nH]nc(CO)c2C1 c1(C(=O)NCC(CC=C)NC(c2cn(C(C)C)cn2)=O)cc(C2CC2)nc(O)c1 N1(C(=O)OC(C)(C)C)CCC(C(=O)OCCSC2CCC2(C)C)CC1 Cc1ccc(C(=O)NCC2OCCC2C(=O)NC2(CC(N)=O)CCC2)nn1 c1(C(N2CC(N(C(C(CC)NC(=O)OC)=O)C)C2)=O)ccc2c(=O)cc[nH]c2c1 Cc1cccc(F)c1C(=O)NCC1CC2CCC1N2C(C1CCCC1C)=O C(C(CO)(CO)NC(=O)CCN1CCOCC1)N(C(c1cnc(SC)[nH]1)=O)C c1(-n2c(-c3ccn(CCC)n3)nc(-c3nc[nH]n3)n2)ccc(C)cc1CN(C)C CC1OC(C)CC1(c1nnnn1CCCC1CC1)NC(c1ccnn1C)C1CC1 C1(C(N2CCC(C#C)C2)=O)CC2CC1CC2NC(=O)C(C1CC1)OC N1(C(C2(CCC)CCC2)=O)C2CCC1C(CC1CC1OCc1ccccc1)C2 Cc1ccc(C(N2CCC(C)C2)C(=O)NCc2ccccc2)cc1I c1(NC(=O)NCCOC(CN2CCCC(CC)C2)=O)c(C)nn(C)c1C Cc1cc(C)c(C(N2CC(CNC(=O)CC3CC(F)(F)C3)CC2(C)C)=O)cc1N c1(C(N2CC3CC(NC(C(C)c4ccco4)=O)C3C2)=O)cnc2[nH]ccc2n1 CCCC(CC)CCC(=O)N1CCC(CNC(=O)CC(=O)N(C)C)(CO)C1 C(=O)(C(F)C(C)CNC(C1(CF)CC(=O)C1)=O)N(C1(CC)CC1)C C1(C(=O)NC(CC)CC(=O)NCCc2cccc(F)n2)CC2C(C1)C2(F)F N1(C(CC(CC)NC(C2CCC(C)(CC)O2)=O)=O)CCC2(CCCC2)CC1 N1(C(C2C(OC)CCCC2)=O)CCCN(C(c2ccn(C(F)(F)F)n2)=O)CC1 c1(C(=O)NC)cc(C)nc(N(CC(C)NC(C2CCS(=O)(=O)C2)=O)C)n1 C12(C(=O)NCC(CNC(=O)CCCc3cccs3)O)CC3CC(C(=O)N1)C2C3 Cc1ccccc1CC(=O)NCCC(C)N(C)C(c1c[nH]nc1C1CC1)=O N1(C(CNC(=O)NC)=O)CC(NC(C2(CSC3CC3)CCC2)=O)CC12CCCCC2 N1(C(c2cccc(C)c2O)=O)CCC2CN(C(c3ccc(C4CC4)o3)=O)CC2C1 c1(SC)ncc(C(=O)NCC2(C)CC(NC(=O)C3=CCSC3)C2)c(O)n1 C1(C(N2CCCC(N3CCCCCC3=O)C2)=O)(OC)CCC12CCC2 Cc1ccccc1Oc1ccc(NC(C2(N)CC(F)C2)=O)cc1 C(C)(C)(CN=c1cc(Cl)nc(CS(C)(=O)=O)[nH]1)NC(C12C(C)OC(C)(C1)C2)=O C1(C(N(C)C)N)CCC(C(N2CCC(N(c3nnc(C4CC4)s3)C)C2)=O)O1.C.CCO c1(N2CCC(NC(C)=O)C2)ccc(S(=O)(=O)NC(C)(C)C(C)(C)C)c(Cl)c1 C(=O)(C(C)C(O)C(C)CC)NC1C(NC(c2ccc(CC)c(CC)c2)=O)CCC1 N1(C(C2C(COCC)CC2)=O)CCCCC(CCC(=O)NC2CC(CO)N(C)C2)C1 N1(C(Cc2ccc(C)s2)=O)CCCC(NC(c2ccc(Cl)cc2F)=O)C1C C1(C(=O)NCCCN(C(=O)CC(C)c2ccco2)C(C)C)CCC(N(C)C)CC1 c1(C(N(CC=C)CCC=C)CC)ccncc1.c1(CCC=O)ccc(C2CC2C)o1 C(C)(C(O)C(C)C)NC(c1c(CN(C(CCC#C)=O)C2CCC2)n[nH]c1)=O C=CC1CN(C(=O)CNC(c2ccc(O)nc2)=O)CC1NC(=O)Cc1ccncc1 CCC(O)(CC(=O)N1CCC(NC(c2ocnc2CC)=O)CC1)c1ccccc1 c1(CCC(=O)NCC2(NC(C=CC=CCC)=O)CCCC2)cccc(Cl)c1Cl CC(C#N)C(=O)NCC1CCN1C(c1cn(C(C)(C)C)nn1)=O C1(CCC(N2CC(C)(CC)C2)=O)CCCCN(C(c2c[nH]c(C#N)c2)=O)C1 c1(C(N2CCC(C)(CNC(C3CCOCC3)=O)C2)=O)occ2c1CCCC2 C1(C(=O)NCC2N(C(CC3CC(=C)C3)=O)CCN(C)C2)CN=C2N=CNN2C1 C1(C(N(C(C)CO)C)=O)CCN(C(C2(F)CC=CC2)=O)CC1 C=C(C)C1OCCCC1C(=O)NC(C)CCN(C(=O)CC1(N(C)C)CCC1)C Cc1nsc(N)c1C(N1CCCC(CNC(C2CCC(F)(F)C2)=O)C1)=O c1(C(N2CCC(NC(C(C)n3ccnn3)=O)C23CC3)=O)cc(Cl)c(F)c(Cl)c1 C1(C(N2CC3(OCC(NC(CCCC#C)=O)C3)C2)=O)COc2ccc(O)cc2O1 N1(C(C(COC)NC(C)=O)=O)C2CCC1CC(NC(c1cncc(C)c1C)=O)C2 c1(C(N2C(C(C)(C)NC(COCCC=C)=O)CCC2)=O)[nH]c(O)nc1C c1(N(C2CCCCCC2)C(c2sc3cc(C)sc3c2)=O)cc(C(N)=S)ccc1C N1(C(c2c(C(C)C)ocn2)=O)CC2CC(NC(=O)C(C)=C3CCC3)C2C1 C(C)(C(C(=O)N1CCCC(C(C)(C)O)C1)C(C)C)NC(CCSC)=O Cc1ccc(OCCCN(C(=O)NC2CCCCCC2)CC2CCCO2)c(C)c1 c1(C(N)=O)ccccc1C(=O)NC1CCC(n2cc(C=CC(=O)O)nn2)C1 N1(C(C(C=C)CC)=O)CCN(C(=O)C(c2ccco2)SC)CC1C(C)C C#CC1CN(C(c2ncc(C#N)cc2C)=O)CCN1C(c1nscc1C)=O C#CCC(C)(C(=O)N1CCCC(CC2CC2)C1)NC(c1scnc1CC)=O c1(C(N(C)CC2CCCN2C(=O)CC2CC3(CC3)CO2)=O)cnn2c1N(C)CC2 C1(C(N2CC(CC=C)(NC(c3ncn(C(C)(C)C)n3)=O)C2)=O)CN2CCN1CC2 n1(C(C)Cc2ccccc2)nc(-c2ccccc2Br)nc1-c1cncc(F)c1 c1(C(=O)NCCN(C(C(C(CC)O)C)=O)CC)cc2c(Cl)cc(Cl)cc2[nH]1 Cc1[nH]nc2c(C(=O)NC(C3CCCC3)CNC(c3c[nH]nc3Cl)=O)cccc12 C12(OC)CCC(C(=O)NCC3CC3CNC(c3ccc(F)cn3)=O)(CC1)CC2 C1(CC(=O)NCC(CCCC)NC(c2cc(Cl)n[nH]2)=O)CCCC2(CC2)C1 N1(C(CCSCCCC)=O)CCC2C1CCCN2C(=O)Cc1ccccc1O C(c1c(F)cccc1F)=CC(=O)NCC(C1CC1)NC(c1cc(CO)ccn1)=O C12(NC(C=Cc3ccc(C)cn3)=O)COCCC1CN(C(c1cc(F)c[nH]1)=O)C2 c1(C(N(CCCCCCNC(C2CCC2)=O)C)=O)ncc([N+](=O)[O-])n1C c1(C(=O)NC2C(NC(C3CC(C)=C(C)CC3)=O)C2)ncnc2ccsc12 C1(CCC)CN(c2nnc(-c3cccnc3)n2CCOCC)CCO1 C1(CNC(C(c2cc(C)sc2)(F)F)=O)CCC2(CCC2)C1NC(=O)C1=NOCC1 c1(C(=O)NCC23OCC(NC(c4coc(O)n4)=O)C(C2)C3)ccnc2c1CCC2 c1(Nc2nc(-c3cccc(O)c3)sc2)ccn2ccnc2n1 Cc1ncc(C=CC(N2CCCN(C(c3c(N)cnn3C)=O)CCC2)=O)c(O)n1 C1(CNC(COCC=C)=O)CCC2(CN(C(c3ccc(CO)o3)=O)C2)O1 C1(CC)CC(C(=O)NC2CC3(CCC3)C2O)CCN1C(=O)CCC(C)C#N C1(NC(CC(C)C)=O)CN(CC(=O)NCc2ccc(Cl)cc2)CC1n1cccn1 n1(CC)cnc2c(N(C)CC3CC3C)[nH]c(=NCc3cc(Br)co3)nc12 CCC(C)(C=C)C(=O)N(CCNC(c1ccnc(Cl)c1N)=O)CCOC c1(C(=O)NCC(CC)N(C(=O)CC2CC2)C)ccc2sncc2c1 Cc1ncsc1C(=O)NCC1(O)CC(CNC(c2sccc2C(F)F)=O)C1 CC1(C)CCCC(CC(=O)NCC23CC(CN2C(=O)CSc2nncs2)C3)C1 C1(C(N(C2CC2(C)C)C)=O)(NC(=O)C(O)Cn2cncn2)CCC(C)(C)C1 c1(C(N2CCC(N(C(=O)C(F)CC3CC3)C)C2)=O)cccn2cncc12 C1(C)(CNC(C2(CC#C)CCOC2)=O)CC(F)(F)CN1C(=O)C(C1CC1)OC C1(C)(CNC(CC2CN(C(C(=O)NC(C)C)=O)C(C)C2)=O)CCCCC1O C1(COC2CCN(C(C(F)=CCC)=O)C2)CCN(C(=O)CSS(C)(=O)=O)CC1 n1(CCC(=O)NC(C2CN(C(c3cc(C)no3)=O)C2)C)c(C)c(C)sc1=O c1(C(=O)NC2CC(CCNC(C3C(C(C)C)(CC)C3)=O)C2)cncc2nc[nH]c12 c1(C(N(CCOCCCNC(C(C)SC)=O)C)=O)cc(NC(C)=O)cc(Cl)c1 N1(C(CCCN2C(=O)CN(C)C2=O)=O)CC2(CCN(C(C3CC(N(C)C)C3)=O)C2)C1 C1(C(C)C)CCN(N(C)Cc2c[nH]ccc2=N)CC1 C1(C)(C(N(CCN(C(=O)CC2CCC(C)C(C)C2)C(C)C)C)=O)CC2(CCC2)C1 c1(CNC(=O)Nc2cccc(OCC3(C(=O)O)COC3)c2)ccccc1F c1(OC)ccc2oc(CN3CCOCC3C(N3CCN(C)C(=O)C3)=O)cc2c1 C1(CC)N(C(=O)N(CCC2CC2)CC2CC2)CC12CC=CC2 C1(CCCNC(CCC=C)=O)CN(C(=O)C=CCOC)CCO1 C(=O)(C(CC(F)F)C1CCC1)NC(CN(C)C(C1(CSC)CCC1)=O)C(C)C N1(C(C(CC)NC(N)=O)=O)CC=CC(C(=O)NCc2c(OC)noc2C)C1 N1(C(C(C)NC(CC)=O)=O)CCOC(C(C)NC(=O)C=CCN2CCCC2)C1 C(CCCN=c1[nH]cnc2cccc(F)c12)NC(c1ncoc1COCC1CC1)=O c1(OC)nccc(N2CCC(c3ccccn3)CC2)n1.c12ccc(o1)SC2 Cc1cc(CC(N2CC(NC(c3ccnn3CCF)=O)C(C)(C)C2)=O)ccc1Cl C(C(C)(C)CC(=O)N1CCC(NC(C2=CNC=CC=N2)=O)C1C(C)(C)C)OC CCCCC(C(C)O)NCC(=O)Nc1ccnc(N2CCN(C)CC2)c1 C(C(F)(F)C(=O)NCC1CN(C(C2(Br)CC2(C)C)=O)CC1C)OC N1(C(CCCN(C(C(CC)=CCCC)=O)C)=O)CCC2(CCN(C)CC2)C1 N1(C(C(C)SCC)=O)CC(NC(c2cnc(NC(C)=O)o2)=O)CC(C)C1 C12CCC(C)CN1C(=O)NCc1ccc2o1.C1(CC)CCOCCN1 C12(CCOCC1)C(=O)N2.c1(CC)cc[nH]c1C(N1CCC(OC2CC2)C1)=O CC1C(C(=O)NCCC2(O)CN(C(C3OCCO3)=O)C2)=Cc2ccccc21 Cc1nn(C)c(C)c1CCC(=O)NCC1CCCN(C(c2csc(O)n2)=O)C1 N1(C(c2ccn(CC)n2)=O)CCCC(C(=O)NCCC2(SC)CCC2)C1 C1(CC(=O)NCC(CC)(C)CO)N(C(=O)Cc2cn(C)nc2C)CCC1(C)C c1(C(N2C(C(C)C)C(NC(c3cncc(N)n3)=O)CC2)=O)cnn2c1CCCC2 C1(CC)C(C(=O)NCC2(CO)CN(C(=O)CSC3(C(N)=O)CC3)C2)CCN1C C1(C(=O)NC2(CC=C)CCC2)CCC(C2CC2)N1C(=O)Cc1cc[nH]c1 c1(CC(=O)NC(CC)CNC(=O)CC2CN(C)CC2O)cc(F)ccc1O C1(NC(CC(=C)C)=O)C2COCC1CN(C(c1cnn(C)c1)=O)C2 CN1CCOC(C(N2CCN(C(=O)CCn3cncn3)C(C3CC3)C2)=O)C1=O CCC(CC)C(F)C(=O)N1CCC2(CC2C(=O)N(C)CCN2CCCC2)C1 C(CC1=CCN(Cc2cccc(Cl)c2Cl)CC1)NC(C(COC)(C)C)=O C1(NC(Cc2nnc(C)s2)=O)CN(C(C23CC=CC(C2)OC3)=O)CCC12CCC2 CC1=C(C(=O)NCCCC2(NC(=O)CC3CCCC(O)C3)CC2)CCS1(=O)=O Cc1cc(-c2nc(-c3ccccc3)nn2C)nn1C1CCCCC1 c1(C(=O)NCCCCCN(C)C(C2(c3ccno3)CC2)=O)cncc2ccsc12 N1(C(C2C(NC(c3ccc(F)cn3)=O)COCC2)=O)CC(CO)CC12CCC2 N1(C(c2nc(OC)oc2)=O)CCC(C)(NC(=O)Cc2c[nH]nc2O)C1 c1(C(=O)NC(CC(=O)O)c2ccccn2)ccc(C)cc1N1CCCC1 Cn1ccc2cc(C(=O)NC3CC4CC3CN4C(C3(C#N)CCC3)=O)cnc12 C(=O)(C(C)(C)C(=O)N1CCOCC1)NCC(CN(C(CC1C(C)C1)=O)C)(C)C c1(OC)ccc(OC)c(CNC(=O)CC2CCC2C2CC2)n1 C1(NC(C(C)NS(C)(=O)=O)=O)CCSC12CN(C(c1ccc3nonc3c1)=O)C2 c1(C(N2CC(C)C(NC(c3coc(C4CC4)n3)=O)CC2)=O)cc([N+](=O)[O-])n(C)n1 C(=O)(C1CCCn2cncc21)OCCN(C(=O)C(CCCC#N)NCC)CC.C(C)(C)(C)O c1(OCCC(=O)N(C2CCN(C(c3ccc(Cl)s3)=O)C2)C)ccc(F)cc1F Cc1csc(=O)n1CCC(=O)NCC(O)CN(C)C(c1cc(Br)n(C)n1)=O C12(CCC=CCCC)CCCC1N(C(=O)C=CCC(C)(C)NC(C)=O)CC2 c1(C(=O)NC2CCCN(C(c3c(CC)c[nH]c3)=O)C2)ccc(Cl)cc1C C1(C(N2CCCC(N(C)C(C3CSCC(=O)N3)=O)CC2)=O)CCCCC12OCCO2 C1(C(=O)NC2(C(=O)NCC(c3ccccc3)O)CC2)CCC2(CC1)CC2 C1(C(C)NC(C2(C(F)F)CC(=C)C2)=O)CCCN(C(=O)Cc2ccc(CO)cc2)C1 N1(C(C(C)(CO)OC)=O)CCCCC(CNC(=O)C(=CC2CCCCC2)F)C1 N1(C(Cc2c(C)n[nH]c2C)=O)CC(CN(C2CCC2)C)CC12CCC2 N#Cc1ccc(CN2CCC2CNC(=O)C(C)n2cccn2)c(F)c1 CCCCC(F)C(=O)NCCCC(O)C(=O)N1CC(C(C)CC)C1 C1(CC=C)(NC(=O)Cc2ncsc2Cl)CCCN(C(C2COC3(CCC3)C2)=O)C1 c1(OC)ccc(Cl)c(C(=O)NCC2CC(CNC(c3cnc4n3CCS4)=O)C2)c1 N1(C(C2(C)CC2)=O)CCC2(CC1)OCCCC2NC(c1scc2c1CCCC2)=O Cc1cc(O)ccc1C(=O)N(CC(C)NC(C1C(C)C1C)=O)CCO Cc1cccnc1C=CC(=O)NCC1C(C)CCN1C(c1ncc[nH]1)=O C(=O)(CCCC(C)CC)NC(CCCC)C(=O)NC1CCC(=O)NC1C C12(C(=O)NC(C)CC3CN(C(c4ccc(Cl)s4)=O)C3)CCOC1CCOC2 c1(C(N(C2CN(C(c3c(C)coc3)=O)CC2(C)C)C)=O)ccc(P(C)(C)=O)cc1 C(=O)(CCC(=O)NCCCC1CCCCN1C(C1CCC(F)(F)C1)=O)NCC N1(C(C(CC)OC)=O)CC(C)(C)OCC1CNC(c1cc(C(=O)OC)nn1C)=O C1(NC(C=CSC)=O)COC2(C1)CN(C(C1(F)CC=CC1)=O)C2 CCC(O)C(=O)NC(CNC(C1(c2ccccc2)CCC1)=O)C1CCC1 n1(CC(N2C(CNC(CSCCC#N)=O)CC(O)C2)=O)ncn2nccc2c1=O c1(C(=O)NC(CC)CN(C(=O)C(C)OC)C)ccc(CC(=O)N(C)C)nc1 C12(NC(=O)CN3CCCC3=O)CCCC(NC(c3cccs3)=O)(C1)C2 c1(C(C)OC(c2ccnc(C)n2)=O)ccc(F)c(Br)c1 Cc1ccc(C(=O)O)cc1S(=O)(=O)N1CCCC(c2nc(C)no2)C1 CCCCC(C(=O)NCC1(O)CC(CNC(c2cc(Cl)ccc2C)=O)C1)N(C)C C=CCC(C)(O)C(=O)NC1CC=C(C(=O)N(CC(C)(C)CO)C)C1 c1(C(N2CC3(CN(C(C4CCN(C)CC4)=O)C3)C2)=O)cc2ccncc2cc1F c1(C(=O)NC)cc(CNC(C2CC(CNC(=O)C(C)OC3CCCC3)C2)=O)on1 C1(N2CCCCC2)CCCCN1C(=O)[N+](C(c1cnccc1C(C)(C)C)C)([O-])NC N1(C(CC(C)SC)=O)CCOC2CCN(C(c3ccc(Cl)cc3Cl)=O)CC12 C1(CC(=O)N(CCCNC(C2(C)CCCO2)=O)C(C)C)COc2ccccc2O1 C1(C(=O)NCC(CC)CO)CC(NC(=O)CSC)C12CCC2 C12(CNC(CCC=C=C)=O)CCC(CNC(c3sc(C)cc3C)=O)(CC1)OC2 CC1Oc2ccc(C(=O)NC3CN(C(c4cnco4)=O)C3)cc2C1C c1(N2CCCCC(CCOCC)C2)nc(=N)[nH]c(=NC(C)CNSC(F)(F)F)[nH]1 N1(C(c2cc(Cl)ccc2F)C)CC2(CCC2)C2COCC12 C(=O)(C1COc2ccc(F)cc21)N(CCN(C(C=NOCCC)=O)C)C(C)C Cc1ccc(NC(=O)CC(CC2CC2)NC(C2(C)CCN(C)C2)=O)cc1C#N C(=O)(CCCCCO)NC(C1CN(C(c2ccc(C(F)(F)F)cn2)=O)CCO1)C N1(C(C(C=C)(C)O)=O)CCN(C(=O)CC23CC(C2)C3)C(C2CC2)C1 N1(C(CNC=O)=O)CCC(C2CC(NC(C3(c4ccccc4F)CC3)=O)C2)C1 c1ccc2c(c1)CCCC2.C1(C)(C(C)C2CC2)CN(C(=O)C(=O)N(C)C)CCO1 N1(CC(=O)NC2CC2CNC(c2coc(C3CC3)c2)=O)CC2CC2C1 C1(NC(C(C)=C(C)C)=O)CCC2(CCCN2C(=O)CCCOC(C)C)CC1 CC1CN(C(=O)C(C)CC(N)=O)CC2(CCN(CCc3cc(Cl)ccc3Cl)C2)O1 c1(C(=O)NCC(N(C(=O)Cc2cn[nH]c2)C)C2CC2)c(F)ccc(S(C)(=O)=O)c1F C(CC(C(C)(C)C)NC(=O)C(=O)NCCCSC(C)(C)C)N(C)C C1(C(N(C2CCCN(C(C3(CF)CC(F)(F)C3)=O)C2)C)=O)CCn2cncc2C1 C1(C)(C(=O)NC(C(=O)NC(C(=O)OC)C)C2CC2)COCCO1 N1(C(CC2ON=C(C)C2)=O)CC2CCN(C(c3cnn(C4CCCC4)c3)=O)CC12 c1(C(=O)Nc2scc(C)n2)cccn2c(-c3cnn(C(F)F)c3)cnc12 CN1C(C(N2CCC(CO)(NC(=O)CCCCNC(N)=O)C2)=O)CCS1(=O)=O c1(CC(=O)NC(C)C(C)NC(c2cc(F)n(C)n2)=O)ccccc1CN(C)C Cc1cc(C#N)cnc1N1CCC(O)(C(C)NC(=O)CC(C)C(C)C)C1 N1(CC)CC(NC(=O)C(C)(C)C2CCCN2C(C2CC(F)(CF)C2)=O)C(C)C1 Cc1ccc(C)c(CC(N2CCC(C)(CNC(c3cccc(F)c3O)=O)C2)=O)c1 C1(C#N)(CC(N2C(CNC(C(CC)CO)=O)C(C)CC2)=O)CCOCC1 C(C(N=[N+]=[N-])C(=O)NC1CC(C(F)C(N2CC(OC)CC2(C)C)=O)C1)OCC N1(C(C(C(C)C)NC(N)=O)=O)CCC2(CNC(=O)C(N)CC3CCC3)CCCC12 C(CNC(c1cnccn1)=O)(C(=O)N1CC(CC(F)(F)F)C1)N(C)C C1(N(C(=O)CC2COCC2O)CCC)CCN(C(c2cc(C)ns2)=O)CC1 CC(C)(O)C(C(N)=O)NC(c1ccc(CNC(C2CCCSC2)=O)s1)=O c1(C(=O)NCC2C(NC(C(C(C)O)N(C)C)=O)COC2)c[nH]c2nccc(Cl)c12 c1(-c2nc(C(C)O)nn2C2CCCOC2)ccc(O)cc1Cl C(CNC(C1CC1CC(C)C)=O)(CC(F)(F)F)NC(C(C)=C1CC1)=O c1(C(=O)NC(C2CCCN2C(=O)CC2(C)CCCC2)C)nccn2ccnc12 c1(C(=O)NC(CC(C)NC(C(COC(C)C)(C)C)=O)C)cc2c(s1)CCC(C)C2 c1(C(=O)NCC2CC(SC)C2)ccc(C)c(S(=O)(=O)NCCN(C)C)c1 c1cn(CCNC(=O)CC(C(C)OCCSC)=O)nn1.C1(C(C)(F)F)(CN)CC1 c1(C(N2C(CO)CC(NC(c3cnc(OC)s3)=O)C2)=O)cc2cccnc2s1 C1(C(=O)NCC(C(C)(C)C)NC(CC2CCCC(C)C2)=O)OCCN(C)C1=O CC(C)(O)C(C(=O)NCC1CCSC1)NC(=O)C=Cc1cc[nH]c1 C1(Nc2ccc(NC(Cc3nc(C)sc3)=O)cn2)CCCCC1C1CCCC1 N1(C(C=Cc2cncc(OC)c2)=O)CC2CCC(NC(=O)C3=COCCC3)(C2)C1 C12(CCC1)CC(=O)N2.C(C(C)(C)C)OCC(C)NC(C1CC(=O)N1)=O S(=O)(=O)(c1cc(Br)c(F)cc1F)Nc1c(N2CCc3c(C)[nH]nc3C2)ncnc1 C12(C(=O)NCCCCNC(C(CN(C)C)(C)C)=O)C3C(=O)C4C5CC(C14)C2C35 N1(C(C(CCCC)O)=O)CCC(C)(C)C(C(=O)NCc2ccc(OC)nc2)C1 c1(-c2cc(OC)c(C)cc2)n[nH]c(=NC(=O)NC2CCN(C)C2C)s1 C1(O)(C(N2C(C(N3CC(OCC#C)C3)=O)CC2)=O)CCCCC1 c1(C(N2CC3C(NC(=O)COCC4CCCOC4)(C3)C2)=O)cc2n(n1)CCCC2 c1(NC(C2(C)CN(Cc3cc(O)cc(F)c3)C2)=O)cc(F)c(Cl)cc1F c1(OC)ccc(C(C)C)c(C(=O)NC(CCNC(C2CCOCC2)=O)C(C)C)c1 C12(CNC(C3(C=C)CC3)=O)CC(CN1C(=O)CC(C)N(C)CC)C2 c1(CC)cnc(C(N2CCC(CN(C(=O)CSc3cnn(C)c3)C)CC2)=O)nc1 CC(C)(C)C(CC(=O)N(CCCO)CCO)NC(c1cccc2c[nH]nc12)=O C(N=c1[nH]c(=NCC2Cc3cc(F)ccc3O2)c2[nH]ccc2[nH]1)c1cc(O)n[nH]1 Cc1nc(C(=O)NCC2CCCC(NC(=O)CC3CCOC3(C)C)C2)sc1C Cc1[nH]c2c(NC(c3ccc(C(N4CCC5(CC5)C4)=O)cc3)=O)cccc2c1C C12CCC(CC1)CCNC2=O.C1(C(=O)NC(c2csnn2)=O)CN(CC)C1 N1(C(C2(C)N(C(c3ccc(C)nc3O)=O)CCC2)=O)CCn2c(cnc2C)C1 N1(C(C(C)Sc2nccn2C)=O)CC2CCCC(C1)C2C(=O)NC1C2COCC12 N1(C(C(C)OCCC(C)C)=O)C2CCC(C2)C1CC(=O)NCC(C)(C)O C1(NC(CSCC)=O)CC(C)N(C(c2ccn(-c3cccc(Br)c3)n2)=O)C1 C1(NC(C2CCCC2CNC(C2CCCC2F)=O)=O)C2CCC(F)(F)C12 CCC(C(=O)NCC(=O)NCC(=O)NCC1OC(=O)CC1(C)C)C(C)C C(=O)(C(C)C(C)S(C)(=O)=O)NCC1CC(NC(C2C(=C)C2)=O)C1 c1(C(=O)NC2CC(F)(CNC(C3C(C)C3C)=O)C2)cc(N)ccc1Cl c1(NC(C(CC)N(CC)CC)=O)ccc(NC(=O)CC2CCC(C)(C)O2)cc1 N1(C(Cn2c(C)ccn2)=O)CCOCC1CCNC(=O)C(F)(F)c1cncs1 C(=O)(C(CCOCCO)NC(=O)CC1CCCCCC1)NC(C)CC1CCOC1 N1(C(CCOC2CN(C(C(CC)SC)=O)C2)=O)CCC(C)(O)C1 c1(-c2cn(C(C)C)c(-c3cccnc3)n2)cc(C(N2CCC3CC3C2)=O)ccc1F c1(COC)ccc(C(=O)NCC(C)N(C(c2ccnc(C)c2O)=O)CC)cc1F c1(CC(=O)NCCC(=C)CNC(=O)C(O)CSC)c(OC)cccc1F C(=O)(C#CC1CCCOC1)N1CCC(CNC(CCC(C)C)=O)C12CCC2 C1(NC(C(CC)Oc2ccccc2)=O)CN(C(C2(C(=O)OC)CC2)=O)CC(C)(C)C1 N1(C(C2(CC(C)C)CCC2)=O)CCCCC1C(=O)NC1C(O)CC1O C1(NC(c2cc(C(C)(F)F)n[nH]2)=O)CCCC(NC(=O)CSC(F)(F)F)C1 c1(CC)ccc(NC(=O)CN(C(=O)CCc2cc(C)no2)C2CC2)c(C)c1 N1(C(c2c(CC)ocn2)=O)C2CCC(C2)C1CNC(=O)CC12CCC(CC1)C2 C12(C)CC(O)CN1C2=O.C1(CNC)CC2C=CC1O2.C1C=CCS1 C1(=CC(=O)NC(C)CC2CN(C(=O)CC3COCCO3)C2)CCC(C)(C)CC1 C12CCN(CC1)NC2.c1(C(C)C)ccccc1N.C1(C)CCOC(C)C1 N1(C(CCOC(C)=O)=O)CCOC(CNC(=O)CC2CCC(C)(C)O2)C1 C1(C(=O)NCCc2ccco2)(CNC(C2C3CCC(=O)C23)=O)CC12CCC2 C1(C(=O)NCCN(CCCF)C)(OCCC)CCC(C)(C)C1.C1(C)C(=O)N1 N1(C(COC)=O)CCN(C(=O)Cn2ncnn2)CC1.C12CCC(C1)C(=O)NC2 C1(C)(NC(C(C)OC)=O)CCCN(C(c2scnc2Cl)=O)C1 C1(C(N(C(C(OC)OC)C)CCN2CCCC2)=O)CCCCC1 CCCCC(F)C(=O)NCc1cccc(NC(c2c(CC)cccc2F)=O)c1 Cc1nnn(C)c1C(=O)NCC(C)(C(C)C)NC(C1C(C)(C)C1(C)C)=O C1(C(=O)NCCOC(CNC(C2=CC(C)(C)C2)=O)(C)C)CCCCC12CCC2 N1(C(CSc2ccc(OC)cc2)=O)CCC(NCCNC(=O)CCF)C(F)C1 N1(C(CCOCC#C)=O)CCOC(CNC(=O)C=CC2CCOC2)C1 c1(C(N(CC(=O)NCC(C)CC(C)O)C2CCC2)=O)cc(F)ccc1F C1(NC(=O)CC2CCC(F)(F)C2)CCN(C(=O)CSc2nc[nH]n2)CC(O)C1 n1(CCN(CCC(C)Sc2ccccc2)C)cnc2ccccc12 c1(C(=O)NC2C(NC(C(c3c(OC)cccc3)(F)F)=O)CC2)cn(C)ccc1=O N1(c2cc(C)[nH]n2)CC2C(C(=O)NCC3CCN(C)C3)C2C1 N1(C(C(CC)=CC)=O)CCCC(C(=O)N(C(C2CCC2)C)CC)C1CC Cc1ccc(C(=O)NC(CCN(C(=O)C(C)(Cl)Cl)C)C(C)C)c(Br)c1 N1(CC(=O)NCC2(CNC(C3CCCC(OC)C3)=O)CCC2)CCCNS1(=O)=O C(c1cncs1)=CC(=O)NCCC1CC(NC(C2CC3CC3C2)=O)C1 CC1CN(C(=O)C2CC2)CC(C)CN1C(=O)COc1ccc(Cl)c(C(F)(F)F)n1 C1(NCc2cccc(SC(C)Cc3ccc(C)cc3)c2)CCOC12CCOCC2 CC(C)(C)C(C(=O)NC1CCN(C(=O)COCCc2ccc(Cl)s2)C1)C1CCC1 Cc1nn(Cc2nc(C(=O)O)co2)cc1Cl.c12cn(nn1)C2.C1C(=O)N1CC CN1N=C(CC(=O)N2CC=C(C(=O)NC3CCN(C)CC3(C)C)C2)CC1=O N1(C(C(COC)O)=O)CC(NC(c2sc(-c3nc[nH]n3)nc2C)=O)CCC(O)C1 C#CC1(O)CCN(C(C)C(=O)N(CCNC(c2c(C)noc2Cl)=O)C(C)C)CC1 CC(CC(F)(F)F)C(C(=O)NCC1CCCO1)N1CCC(O)C(C2CCCC2)C1 C(C(C)(O)C(=O)N(C)CCOCCNC(C1C2CC3C(C2)C13)=O)OC Cc1cc(C(N2CCN(C(=O)C(O)CN(C)C)CC2CO)=O)cnc1C(F)(F)F C=C(Cl)CC(C(=O)NCC(=O)N(C)CC)NC(C1CCOCC1)=O C(=O)(C(C)CCC)NCC1(CC(=O)N(CCCC)CC)CC1 C1(NC(c2cn(C(C)C)nn2)=O)C2CC3C1C3C2C(=O)NCc1cc(O)ncn1 CC1CN(C(=O)CO)CCN1C(=O)C(C)OCC1CCCCO1.C1(CS)CCCOC1 O=[N+]([O-])c1cc(F)cc(Cl)c1NC(=O)Cc1ccccc1O C1(NC(=O)Cc2c[nH]nc2O)CC2CC(NC(C3(C4CC4)CC=CC3)=O)CC12 C1(C)(OC)CC(NC(c2c(CNC(C3CC(F)CN3C)=O)nnn2C)=O)C1(C)C c1(C(=O)NC)cc([N+](=O)[O-])ccc1NCC(C1CC1)NC(=O)CCS(C)(=O)=O N1(C(C=C(C)C2CC2)=O)CC(CCNC(c2cc(CO)[nH]n2)=O)C(C)C1 c1(C(=O)NCC2CN(C(c3c(CC)c(F)ccc3)=O)C2)c(C)ccc2nsnc12 N(C1CCc2cc(C)ccc21)Cc1ccc(CC)c(C(=O)O)c1 Cc1nn(C2CC2)c(C)c1C(=O)NCCC(C)N(C(=O)C(C)n1cnnn1)C c1(C(N2CCC(C(C)NC(C(C)(C3(C)CC3)OC)=O)CC2)=O)nn(C)c(N)c1C C(C(C(=O)N(CC(F)F)C)C(C)C)NC(C(C(=O)OCC)F)=O N1(C(CC2(C)CCCC2)=O)CC2N(C(C3C4CCC(F)C34)=O)CCC2(C)C1 c1(C(N2CC(CNC(CCOCCC)=O)C(C)CC2)=O)cnc2sccn2c1=O Cc1cccc(C(N2CCC2CNC(C2(C)CC=CCO2)=O)=O)c1 c1(C(=O)NC2CCC(C(N(CCCC)CCO)=O)C2)ccc(C)c(CO)c1 N1(C(C(C(C)C)O)=O)CCCN(C(c2ccn(C3CCCC3)n2)=O)CC1C Cc1cc([N+](=O)[O-])cc(S(=O)(=O)Nc2cncc(-c3cccnc3)c2)c1 N1(C(c2cn(CC)nc2C)=O)CC(C2(NC(=O)COc3cccc(O)c3)CC2)C1 C=CCC(C)C(=O)NCC1(CNC(=O)C(c2ccccn2)C)CCCC1 n1(CC(C)NC(=O)CC2CC2C)cc(CCCCC)nn1 C1(F)(CNC(C(CC)NC(N)=O)=O)CCCN(C(=O)C(C)(C)NC(C)=O)C1 C12(C(=O)NCCN(CCCC)C)CC(CCO1)N(C(=O)CC(=O)OCCCF)C2 N1(C(c2cc(CC)cc(C)c2)=O)CC(C2CN(C(C3(Cl)CC3)=O)C2)C1 N1(C(c2c(F)ncc(OC)c2)=O)CCC2(C1)CN(C(=O)C(C)NS(C)(=O)=O)C2 C1(C(=O)NC(c2c(OC)ccc(F)c2)C(F)(F)F)CC(=O)N(CC2CC2)C(=O)C1 C(CC1CCCC1)(C(=O)Nc1ccn(CC2CC2)n1)NC(C1CC=CC1)=O CC1(C)COCCC1C(=O)NC1CC2CCC1N2C(c1cnns1)=O CC1CN(C(c2ncsc2C(F)(F)F)=O)CCC1CNC(c1cccnc1)=O C1(NC(c2nnn(C)n2)=O)CCN(C(c2ccnn2CC(F)F)=O)CC1(C)C C1(NC(c2c(CNC(Cc3nc(C)oc3)=O)c[nH]n2)=O)CC12CCCC2 CC1CC(NCC(c2ccccc2)N)c2ncnn21 CC1(C)CCc2nc(O)c(C(=O)NC3(c4cccc(F)c4)CC(F)C3)cc2C1 Cc1cc(C(=O)NCCCOC2CCN(C(C3(C)C=CCC3)=O)CC2)c(O)nn1 CC(C)CC(C(=O)NCCC1CCCN(C(=O)CCCSC(C)(C)C)C1)C(N)=O c1(C(N2CC(N(C)C(c3cnn(C)c3Cl)=O)C(O)C2)=O)cc(C#N)c(F)cc1F C(=O)(C#CC1(C(F)(F)F)CC1)NCC(C)(CO)NC(c1[nH]c(=NC)sc1)=O c1(C(=O)NC(C2CCN(C(=O)Cn3ncnn3)C2)C)cc2n(n1)CC(F)C2 N1(C(c2cc(C(C)=O)sc2)=O)CC2CC1C2CNC(c1cnccc1C)=O C1(CCC)CN(C(=O)COCc2ccccc2)CCN1C(c1ccc(C)cn1)=O C1(CNC(NOC(C)(C)C)=O)CN(S(C)(=O)=O)C(C)(C)C1 C=CC(C)(O)CC(=O)N1CC(CNC(c2cnn(C)c2C(F)F)=O)C(C)(C)C1 CC1(C)CCCN(C(=O)CC2COCCO2)C1CNC(c1cc2c(s1)CCC2)=O C#CCCCCCCC(=O)NC1CN(C(=O)CC(C)(C)C)CC12CCCC2 C(=O)(CC(C(C)C)NC(c1cnccn1)C)OCC C(=O)(C(CCC(C)C)NC(=O)C(C)NC=O)NCC1(C#C)CCC1 c1(C(=O)NC2CCC(NC(c3cnn(CC)n3)=O)C2)cc2cccc(OC)c2o1 C1(C(N2CCC(C(=O)O)C2C)=O)(OC)Cc2ccccc2C1 C1(CNC(CCC(C)O)=O)CN(C(c2cc(C3CC3)no2)=O)CCC1(C)C C1(C(N2CCC(N(C(C(C(C)C)O)=O)CC3CC3)CC2)=O)CCC(C)(C)CO1 c1(C(=O)NCC(C)(C)NC(Cc2c(C)ocn2)=O)cc2c(C)n[nH]c2nc1O c1(OCC(=O)NCC2CN(C(C(CCCC)C)=O)CC2C)nc2ccccn2n1 C1(C(=O)NCCOc2ccc(C(CC)=O)cc2)CC2C=CC1C21CC1 Cc1nn(CCC(=O)NCC2(O)CCN(C(c3ccnn3C)=O)CC2)c(C)c1C Cc1ccc(C)c(CC(N2CC3CN(C(c4cc(C)c(C)o4)=O)CC23)=O)c1 N1(C(C(C=CC)O)=O)CCC(C)(NC(c2cccc(NC3CCCC3)c2)=O)C1 N1(C(C(F)=CCC)=O)CCN(C(=O)CCNC(C2CCC2)=O)CC1C C1(CCC(=O)NC(COC)(C)C)CCCN(C(C2CC(F)C(F)C2)=O)C1 N1(C(C2N(C)CC2)=O)CCCCC1C(N1CCC(CC2CCC2)C1)=O C1(CC)CCC(C(=O)NC2C=CCC(C(=O)NCCOCCF)C2)CC1 c1(C(N2CCN(C(=O)CC(F)(F)F)CC2)=O)ccc2ccc3ccccc3c2n1 Cc1nc(C)n(CCNC(C2OCCC2CNC(=O)CC2CCCC2)=O)n1 C1(C(=O)NCC2(CNC(Cc3nc(C)oc3)=O)CC2(F)F)CC(=O)N(O)C1 CN1CCOCC1CNC(=O)CC1CCN(C(c2csc(=N)[nH]2)=O)CC1 Cc1nn(C)c(Cl)c1C=CC(=O)NCCCCC(C)NC(=O)CC(C)CF C1(C(=O)OC)CCN(C(=O)Nc2ccccn2)C1c1ccco1 c1(C(N2CC(N(C(c3c(NCC)scn3)=O)C)C(O)C2)=O)ccn2c1CCCC2 N1(C(CC2C(C)=NOC2=O)=O)CCC(C2CCCN(C(=O)C#CC(C)C)C2)C1 N1(C(C=Cc2c(C)ccs2)=O)CCN(C(=O)CN2CCOC2=O)C(CCO)C1 C(CCC(=O)Nc1csnc1C)(C(C)C)NC(C(CC=C)(C)C)=O c1(C(N2CC(F)(CNC(c3[nH]cc(OC)c(=O)c3)=O)C2)=O)cn2c(n1)CCCC2 c1(C(=O)NCCCC2N(C(C=C3CCN(C)C3)=O)CCC2)cc(O)cc(Cl)c1 c1(CC(=O)NC2C3N(C(C=C(CC)C)=O)CC(CC3)C2)ccc(S(C)(=O)=O)cc1 N1(C(C(C(CC)CC)C)=O)CC(NC(C2SCCCS2)=O)CC12CCCCCC2 n1(CC)ncc(C(=O)N(CC(C)NC(c2cn(C3CCOC3)cn2)=O)C)n1 Cc1cc(C(=O)NC2CCC2CNC(c2cnn(C)c2)=O)cnn1 C1(CCC)(NC(=O)C=Cc2nnn(C)n2)CCCN(C(=O)Cc2ccon2)C1 c1(C(C)C(N2CCCC(O)(CNC(=O)C(C)(C)N(C)C)C2)=O)cccc([N+](=O)[O-])c1 Cc1cc(C(=O)NCc2ccc(C(=O)NCc3cc(C)ns3)s2)c[nH]1 c1(C(=O)NCC(C2CCOC2)NC(C=CCC)=O)sc(C(C)(C)OC)nc1C C(=O)(C(F)C(C)CNC(C1(NC(C2CCCC(=O)N2)=O)CC1(C)C)=O)OC c1(CCC(=O)NC2C=CCN(C(=O)CCS(N)(=O)=O)C2)nc2cccnc2[nH]1 C1(CNC(C(C)OCC(C)C)=O)CC2COCC2N1C(c1cnsc1)=O CC(CCNC(=O)C(C)CO)CCNC(c1cn(CCF)nn1)=O c1(OCC(=O)NCC(CN(C(=O)C(F)=C2CCC2)C)(C)C)ccccc1[N+](=O)[O-] C=CCC(C(=O)NC(C)CN(C(=O)CCSc1ccccc1F)C)NC(C)=O N1(C(C(SC)SC)=O)CCC(C)(C)C(CNC(=O)CC2CCCCC2O)C1 C1(C)(C(=O)NCC(CC(C)C)NC(C(CC)CN(C)C)=O)CCCCC1C C1(C(NOCCC(C)O)=O)CC(O)(CNC(=O)CC2CC(N(C)C)C2)C1 c1(CNC(C2(C)CCN2Cc2cc(Cl)ccn2)=O)c(O)cc(F)cc1F c1(OCCC)cccc(C(=O)NC2CC(Cl)(Cl)C2)c1.C1C(OC)COCCN1 c1(C(CC)C)ccc2cc(-c3nc(CSc4ccccc4)no3)[nH]c2c1 c1(NC(c2c(CNC(C3(CC#C)CCCO3)=O)c[nH]n2)=O)cncnc1C C1(NC(CN(S(CC)(=O)=O)C)=O)C=CC(CNC(=O)Cn2nccn2)C1 c1(C(C)CF)nc(=NC(=O)C(N)COc2ccc(Oc3ccccn3)cc2)o[nH]1 CC(C)C(C(=O)N1CCCC1CN(C(=O)CC1CCC2CC12)C)n1ncc(N)n1 N12CCCC1C2=O.C1(C(OC(C)(C)C)C2CC2)CCCN1c1nnc(C(N)=O)s1 N(S(=O)(=O)N1CCC(SC(F)F)C1)Cc1ccc([N+](=O)[O-])cc1 C=CCN=C(NCC(C)(C)C(=O)OC(C)C)NCc1ccc(I)cc1 c1(NC(C(CC)NS(C)(=O)=O)=O)ccc(F)c(Cl)c1.C123COC(C1)(C2)CNC3=O N#Cc1cc(CN2CCC(F)(C(=O)Nc3c(Br)cc(F)c(F)c3F)C2)cc(F)c1 C1(O)(CC#C)CCN(C(C2CCN(C(=O)Cn3nccc3C)C2)=O)C1 c1(C(N2CCN(C(C3C(CC)C3)=O)CC2CC(F)(F)F)=O)cc2sccc2n1C CC1NC(=O)OC12CCN(C(C1CCCN(CC(F)(F)F)C1)=O)CC2 c1(C(=O)NC2C=CCN(C(C3CC(F)(CO)C3)=O)C2)cccc(F)c1C(F)(F)F C1(NC(C(CCC)CNC(=O)CN(C2CC2)CC)=O)CCn2cncc2C1 C(CCNCCCO)(C1CCC1)SCCNC(C=CC=CCOC)=O C1(C(C)C)CN(C(c2cn(C)nn2)=O)CCCN1C(=O)CC(C1CCC1)C1CCC1 N1(C(c2cncc(OC)c2C)=O)CC2CCC1CC2NC(C1CNC(=O)N1)=O C(C)(c1ccco1)=CC(=O)NCC(C)(CO)NC(CC1C(CC)C1(F)F)=O C1(C(N(CCC(C)NC(CC(CC)(C)C)=O)C)=O)C2CCC1(C)C2(C)C N1(C(c2ccccc2)CNC(C(C2CCCC2)OCC)=O)CCOCC1C C1(O)(C(C)NC(=O)COC2CCC2)CN(C(=O)Cc2c[nH]nc2O)C1 C(c1cccc(F)c1)=CC(=O)NCC(N(C)C(C1(C(C)(C)C)CCC1)=O)C1CC1 S(=O)(=O)(c1cc(C(=O)NCC2(C)CCCN2C(=O)CC2CCC2)ccc1F)NC C1(CC(=O)N(CCC(C)C)CC(C)C)CCCC(NC(=O)C=Cc2cc[nH]n2)C1 C12(NC(Cc3ccc(C)cc3Cl)=O)CCC(CC1)N(C(c1cnsn1)=O)C2 c1(CC(=O)NCC(c2ccccc2)CNC(C(CC)OC)=O)ccc(F)cc1Cl O=C(C=CS(F)(F)(F)(F)F)NC1CCCN(C(c2ccncc2Cl)=O)CC1 c1(NCC(C)OC)ccc(CN(C)C)cc1NC(C1(O)CCCCC1)=O c1(C(=O)OC)cc(OC)cc(C(=O)NCC23CC(C2)C(C(=O)OC)CO3)n1 C(=O)(C(CCS(C)=O)NC(C1(C)CC1)=O)NCC(C)CN(C)C c1(C(N2CCCC(C(CNC(c3cc(C)c(C)o3)=O)O)C2)=O)n[nH]c2c1CCC2 C1(C#CC(=O)N(C2CCC(NC(C3(C)CC4CC4C3)=O)CC2)C)(CC)CC1 c1(NC(CC2N(C(CCC(CC)OC)=O)CCC2)=O)cccn2cc(C)nc12 C1(CC(=O)Nc2cncs2)CN(C(=O)CC2CCCOC2)CC12CC2 S(=O)(=O)(c1c[nH]c(=NCCc2cc(Br)cs2)cc1C)NC1C(C=C)CCCC1 C(=O)(C1CCc2c[nH]nc21)N1CC2C(Nc3c(C)cnc(C)n3)C2C1 C=CCC(CC(=O)Nc1ccc(CCO)cc1)NC(=O)C(n1cc(C)cn1)C c1(CC)cc(C(=O)NC2CC(C)(CNC(=O)CCCc3cnn[nH]3)C2)ccc1F n1(CCCOC)nnnc1C(C1CCCO1)NCCCc1ccc(C)s1 C1(C(N(C(C)C)CCN(C(=O)C(C)(C)C)C)=O)COCCN1C N1(C(C2=CCCC2C)=O)CC2CC(C1)N(C(c1cc(-c3ccco3)[nH]n1)=O)C2 N1(C(C#CC2(CC)COC2)=O)CCCC(C2CN(C(=O)Cn3nnc(=O)[nH]3)C2)C1 C(=O)(CCCCN(C(=O)C(CCC1CC1)NC(=O)C(C)=C(C)C)C)OC C1(c2scc(C)n2)CCN(C(C2(C(F)(F)F)CCCC2)=O)CC1 Cc1nnc2n1CCN(C(c1cn(C3CCC3)nn1)C(=O)NCC1COC1)C2 C(N=c1[nH]ccnc1F)C1CCCC(NC(c2cc[nH]n2)=O)C1 C(=O)(C(C)(C)CN(C)C(c1cscc1OC)=O)N(C1CCCOC1)CC N1(C(C(F)=C(C)C)=O)CCC2CN(C(C3CCN(S(C)(=O)=O)C3)=O)CC2C1 C1(C(=O)NCC2(CC)CCC2)OCCC1CNC(C1CC1(C)C)=O c1(NC2CC(CNC(Cc3ccc(OC)c(O)c3)=O)C2)nccc(S(C)(=O)=O)n1 N1(C(C(CCOC)OC)=O)CC(C(=O)Nc2cn(C)nc2OC)OC(C)C1 c1(C(=O)NC(C)CNC(=O)Cc2cc(Br)ccc2F)cc2cc[nH]c(=O)c2s1 c1(C(N2CC(O)(CCNC(c3cnc(OC)s3)=O)C2)=O)cc(S(N)(=O)=O)oc1C c1(CC)cccc(C(=O)NC(CCN(C(=O)COC)C)C(C)C)c1O Cc1cc(C(=O)NC2CC(CNC(c3ccc(Cl)cn3)=O)C2)ccc1C#N N1(C(C2N(C(C(CCCC)O)=O)CCCC2)=O)CCC2(CC1)CNC(=O)C2 c1(C(=O)NC2(C)CCCN(C(c3cccnc3)=O)C2)cc(F)c(F)c(N)c1Cl C1(C(=O)OCC)OCCNCC1N(C(C)(C)C(C)O)C(c1cc(C)cc(O)n1)=O C1(C(N(C)CC2CCOC2)=O)(CCNC(=O)Cc2nncn2C)CCCC1 Cc1ccc2c(c1)CCC(C(=O)N(C(CNC(C1CCSCC1)=O)C1CC1)C)O2 C1(C(=O)OC)CCN(C(=O)c2ccn(CCSc3cc(C)ccc3O)c2)O1 C(=O)(C(C)(C)CN1CCCC1)NCC(C)(C)CNC(=O)Cc1cc[nH]n1 N1(C2CN(C(C(n3cc(Cc4ccnc(Br)c4)nn3)C)=O)C2)CCOCCC1=O C1(=O)C(Cc2ccsc2)N(C)CCOCCN1C.C(=O)(C(F)F)C(C)C C1(C(NOC(C)CC(F)(F)F)=O)CN(C(=O)CCCN=[N+]=[N-])CCC1(C)C C1(C(=O)Nc2cnc(C)s2)CCC2(CN(C(=O)CN3CCc4ccccc43)C2)O1 Cc1cc(-c2cn(C3CCC(C(C(CC4CCOC4)C(=O)O)=O)C3)nn2)cnn1 C(=O)(C1(C)OCCc2ccccc21)NCC1(C)CC(NC(C2CN(C)CCO2)=O)C1 C1(C(=O)NCC2CN(C(c3ncoc3C3CCC3)=O)C2)OCC2COCCC12 c1(C(N2CCCC(NC(CN(C(=O)OCC)C)=O)C2)=O)cc(C(N)=O)ccc1F N1(C(C(C)NS(CCC)(=O)=O)=O)CC2(CC(NC(C3(F)CCCCCC3)=O)C2)C1 c1(OCC)ccc(F)c(C(=O)NCCN(c2nccn2C)C(C2CCC2)=O)c1F N1(C(c2cc(C)oc2C)=O)CC2CC(NC(c3cnc(Cl)[nH]3)=O)CC1C2 C1(c2cn(CC(=O)N(CC(C)NC(C)=O)CC)nn2)CCC(F)(F)CC1 C1(NC(c2nc(CCC)sc2)=O)CN(C(=O)Cc2cnns2)C2(CCCOC2)C1 c1(CC)cnn2c1CCC2.C12CCCN(C1)C(=O)C1(CC1)NC2=O CC(C)CC(C)(CNC(C1CC(C)CCO1)=O)NC(C1CC1C(C)(C)C)=O c1(NC(c2n(CCCC)nnn2)c2cnn(C(F)F)c2)ccc(Br)nc1 CN1CCN(n2cc(CC(CNC(=O)C(O)Cc3cn(C)cn3)C(=O)O)nn2)CC1 c1(C(=O)NCCOC2CCN(C(C3C(C)(CC)C3)=O)C2)n[nH]c(C)c1O c1(NC(CC=C)C2CC2)ncc(S(=O)(=O)N2CCOCC2C2CCCCC2)cc1Cl C1(CNC(CCCNC(C)=O)=O)CCN(C(c2ccoc2)=O)CC1O c1(OC)ccc(SCC(=O)NCCC(C)NC(C2CCCN2C)=O)cc1 CCC(C)(C)CC(=O)NCC1COCC1NC(c1cnsn1)=O C1(CNC(c2c(C)cno2)=O)CN(C(=O)Cc2cccc(Cl)c2F)C(C)(C)C1 S(=O)(=O)(c1ccccc1)NCC(=O)NC(CC)(CNC(c1cnco1)=O)CC N1(C2CN(C(C(C3CN(C(CCc4nc(C)sc4)=O)C3)O)=O)C2)CC(C)OC1=O C1(C(=O)NCCCN(C)C(C2(N(C)C)CCC2)=O)CCCCC1(F)F C1(C(=O)NC(COC)(C)CCO)(CO)CCN(C(=O)CCC(C)OC)C1 c1(CC(=O)NC2C(CNC(C3N(S(C)(=O)=O)CC3)=O)C2)c(F)cc(Br)cc1F C12(N(C(C=CCCCCC)=O)C)CCCCC1C2.n1(CC)cc(Cl)cn1 N1(C(C2CC(C)N(C)C2)=O)CCN(C(=O)Cc2ccc(F)c(F)c2)C2(CC2)C1 C(C)(CN=c1cc[nH]cc1S(=O)(=O)N1CCOC(C(C)C)C1)Oc1cccc(C)c1 CCN(CCCOC)N1CCc2c[nH]nc2C1 C(=O)(C1=CS(=O)(=O)CCC1)NCC(CNC(c1cc2ccccc2s1)=O)O C1CC2CCC1C2.n1(CCC(=O)N(CC(=O)OC)C)cc(CN(C)C=O)nn1 Cc1ncn(C)c1C(=O)N(C1CCCN(Cc2ccccc2)C1)C C1(NC(C(CCOC)C)=O)COC2C(NC(c3nc(C)nn3C)=O)COC12 c1(CC(C(=O)N(CC(C)NC(c2ccccc2)=O)CC)=O)cccc(Cl)c1 C1(C(=O)NCC23N(C(C(C)NC(CC)=O)=O)C(CC2)CC3)CCc2nncn2C1 c1(NC)ncnc2[nH]cnc12.C1(CC)CN2CCC1Nc1ccc(cc1F)C2=O c1(OC)nc(C(=O)NCC2C3CN(C(c4cccn(O)c4=O)=O)CC23)cc(O)n1 c1(SC)ccc(C=CC(N2CC(NC(c3cc(O)cs3)=O)C2)=O)cc1 N1(C(COCC=C)=O)CCCN(C(c2cc(C(C)=O)c(C)o2)=O)CC1C c1(C(N(C)CC2N(C(c3c(C)cccc3)=O)CCOC2)=O)n[nH]c2c1CCOC2 c1(C(=O)NC2C(C)CCN(C(c3ncncc3Cl)=O)C2)cc2nc(=O)ccn2[nH]1 N1(C(C(CC)(C)F)=O)CCOC(CNC(=O)CCF)CC1 c1(C(N2CC(NC(C3(C)CC(=C)C3)=O)CC23CCC3)=O)n[nH]c2c1CCCCC2 C1(NC(CC=CC=C)=O)C(CNC(c2sccc2CC#N)=O)CCC12CCC2 N(C1CCCc2nn(C)cc21)Cc1cc(C)cc(C(F)(F)F)c1 C(=O)(C(C)(C)C#N)N1CC(O)(CN(C(C=CCCC(C)C)=O)C)C1 N(C(=NCc1ccc(CO)cc1)N1CCC(O)C1)CC(N1CCN(C)CC1)C N1(C(C2N(C)C(=O)NC2)=O)CCCC(CO)(NC(C2CC2CF)=O)C1 c1(CC)cc(-n2cc(CCN(C)C)nn2)c2c(c1)OCO2.N1(CC(=O)N)CCCC1=O Cc1cnc(S(C)(=O)=O)nc1N1CCC(F)C(NC(c2ccc(Br)c(Cl)c2)=O)C1 CC(C)CC(C(=O)NC1CCCN(C)C1)NC(c1cc(Cl)c[nH]1)=O C1(CNC(C(CCCC)C)=O)CC(N=c2[nH]cc(C#N)c3ccsc23)C1 Cc1ccc(C(=O)NCC(F)CNC(=O)C(c2ccccc2C)(F)F)nn1 c12ccc(Cl)cc1C(=O)N1CC3CC1CN3C2.c1(CC)cc(OC)ccc1F C1(C(=O)Nc2cncc(C(C)=O)c2)CC(F)(F)CN1C(c1cnccc1C#N)=O C1(C(=O)NC(c2nnc(C)s2)C)COCCN(C(C2COCC2C(N)=O)=O)C1 C12(C(=O)NCCN(C(=O)CC3CCCCO3)CC)CCCC1CCC2 C=C(C)CC(C(=O)NC1CCCC(OCC)C1)NC(c1cnc(F)c(C)c1)=O C1(C(C2CCOC2C)c2nnnn2C2CCC2)(NC)COc2ccccc2SC1 C1(C(=O)NC(C#C)C2CCC2)CC(O)CN1C(=O)CCCN1CCCC1 N1(C(C2(NC(c3cn(C4CC4)nn3)=O)CC(F)C2)=O)CC2CC1C1CC21 C1(CNC(CCCCC=C)=O)CC2(CCOCC2)CN1C(c1c[nH]c(=NC)s1)=O Cc1[nH]c(=N)ccc1C=CC(=O)NCC(C)NC(c1ccccc1Br)=O c1(OC)nc(C)ccc1C(N1CC2(CC(NC(=O)CN3CCCC3=O)C2)C1)=O C1(NC(CC2CN(C)C2)=O)CN(C(c2sccc2OC(F)F)=O)CC1(C)C N1(C(C(C)CSc2ccccc2)=O)CCC2(CCCN(C(=O)CSCC#N)C2)C1 c1(CNC(c2n(C)nnn2)C2(c3c(Cl)cccc3Cl)CC2)ccc2c(c1)CCO2 c1(C(N2CCC(C(C)(C)NC(=O)C(F)C(C)(C)O)C2)=O)ccc(Cl)cc1[N+](=O)[O-] CC(C)(C)C#CC(=O)NCC1CN(C(C2(n3cnnn3)CCCCC2)=O)CCO1 N1(C(c2c(C)c[nH]n2)=O)CC(C2CCN(C(c3cc(Cl)c[nH]3)=O)CC2)OCC1C Cc1ccc2c(CC(=O)NC3C=CCN(C(c4cc(CF)on4)=O)C3)c[nH]c2c1 N#CC1CC(C(N2CCC2CNC(C2CC(O)C2)=O)=O)C1 c1(C(=O)NC2CC(CNC(CN(C(=O)OC)C)=O)C2)nn(C)c(=O)cc1C n1(CC)nc(C(=O)NCC2CCCN2C(=O)C=C2CCC2)ccc1=O C12(NC(CC(C)(C)N(C)C)=O)CCOC(CNC(c3ccoc3Cl)=O)(C1)C2 c1(C(N2CCC(N(C(C3CC(C)C3(C)C)=O)C)CC2)=O)cc(S(N)(=O)=O)ccn1 C(=O)(C#CC1(CC)CC1)NCCCOCCNC(C(C(C)C)SC)=O c1(C(=O)NCC2N(C(C(F)=CCC)=O)CC(C)CC2)ccc2c(c1)CCCCN2 C1(CNC(c2scnc2Cl)=O)CCC2CN(C(=O)C=CCN3CCCC3)CC12 N(C(=NCCN1CCOCC1)N1CCC(F)(c2ccccc2C)C1)CC(CC)(C)C C(=O)(C1=NN(C)C(=O)CC1)NC(C(=O)NCCSCCC)Cn1cncn1 c1(C(=O)NCC(C)CNC(c2cnc(CC(C)(C)C)o2)=O)cnn(C)c1C(F)F c1(C(N2CC(NC(C3N(C(C)(C)C)CC3)=O)C2)=O)ccc(S(C)(=O)=O)o1 Cc1noc(C2CCC2)c1CNCc1ccc(C(C)(C)C)cc1 C(CC(=O)N1CCC(CNC(c2nc(Cl)ccc2Cl)=O)C1(C)C)(C(F)(F)F)OC C(=O)(CC(=O)NC1CC(CCOC)C1)NC.C12(CCC1)C(=O)NCCO2 C(=O)(C1=CCC(NC(c2cc(C)cc(O)c2)=O)C1)NCC(C(=O)OC)(C)O N1(C(C(C)(N(C(=O)Cn2cnnc2O)C)C2CC2)=O)CC2CCC(C1)N2C C(=O)(C1=C(C)NC2=NCCCC2=C1)NCCN(C(C(CC)OC)=O)C1CC1 C1(NC(c2cc(C)c(C)o2)=O)CN(C(c2ncoc2C)=O)CC1C1CC1 c1(CC(C(=O)NC2(C)CN(C(C(C3CC3)OCC)=O)C2)N(C)C)ccc(O)cc1 C1(CNC(C2C(C=C)OCC2)=O)CC(F)(F)CN1C(=O)CC(C)(C)O C=CCCCN=C(NCCSCCOC)N1CCC(NC(C)=O)C1 C(=O)(C(C)(C)C(=O)NCCC1CCCCN1C(=O)Cn1ccccc1=O)OC c1(OC)ccc(Br)c(CN2CC(C)CC2C(=O)Nc2cnn(C)c2)n1 CC(C)(CO)C(=O)NCCC1CN(C(=O)CC2CC2(Cl)Cl)C1 C(CC(=O)NCC(CC)NC(=O)C(C)c1cc[nH]n1)OCC Cc1nccc(Cl)c1C(=O)NC(C1CCN(C(=O)C(C)N2CCC2)CC1)C N1(C(c2ccc(C(=O)OC)s2)=O)CC(OC)CC(NC(=O)C#CC2(C)CC2)C1 C1(NC(CC(C=C)C)=O)C(C)(C)CN(C(=O)CCC(CF)CF)CC1(C)C c1(OC)c(C(=O)NC(C)Cc2cccc(O)c2)ccc2ccccc12 C1(CC(=O)NC2C(CC)C2)CCCN(C(=O)C(C)CC)C1 C=C(C)CC(C(=O)NCC(C)(C)C(F)F)NC(c1cc(C2CC2)on1)=O N1(C(COCc2nnc(C)s2)=O)CCN(C(=O)C2=NNC(C(F)(F)F)C2)CC1C N1(C(C(=O)N(C(C)C(F)(F)F)C)=O)CCn2c(cnc2C)C1 Cc1n[nH]c(C)c1CC(=O)NC1CCCC(N(C)C(C2CCC3CC23)=O)C1 C(=O)(C1CSc2ccccc21)NC1C(O)CCN(C(c2ncc(N)cc2Cl)=O)C1 C(=O)(C(C)CCCOC)N1CCCC(CC(=O)NCc2ccc(CC)cc2)C1 CN1C(CNC(=NCCc2nccs2)NCC2CCC2)CCS1(=O)=O c1(C(=O)NCC2CC(NC(CC(COC)C)=O)C2)cn2c(n1)COCC2 Clc1cc(Br)cnc1CNC1(Cc2sc(Br)cc2Br)CC1 C(=O)(C1=CNS(=O)(=O)N=C1C)N1CC(CNC(C(CCC)C(=O)OC)=O)OCC1 c1(C(N2CC(O)(CNC(C(c3ccc(C)cn3)(F)F)=O)C2)=O)ccc2nn[nH]c2n1 C1(CC(=O)NC(CNC(c2c(C)csc2Cl)=O)C2CC2)CCCC2(CC2)C1 Cc1nc2sccn2c1C(N1CCC(NC(=O)C(C)(C)C2CC2)C(C(C)C)C1)=O C1(C(=O)NC(C(=O)N(c2ccsc2)CC)c2ccco2)CCCC(CF)C1 N1(C(C2CC(OC)C2)=O)CCC(N(C(c2cc[nH]n2)=O)CC2CC2)CC1 C1(NC(CCNC(C)=O)=O)CN(C(=O)CC#N)CC1F N1(C(C(C=C=C)C)=O)CCN(C(c2cc(-c3ccc(Cl)s3)[nH]n2)=O)CC(O)C1 N1(C(CSc2ccc(C)cc2)=O)CCCC2CN(C(=O)CN(C3CCC3)C)CCC12 C(=O)(C(Cc1ccoc1)NC(=O)CC(=O)NC1CC1)NCC(CC)N1CCCC1 N1(C(C(CC)(C)C#N)=O)CCC2(CC(NC(C3CC3c3cnn(C)c3)=O)C2)C1 C1(NC(CN(C)CO)=O)CC2CCC(C1)N2C(C1(CC2CCC2)CC1)=O N1(Cc2cn(CC)nc2)CCCC(NC(c2ccnc(OC)n2)=O)C1C c1(NC(=O)NCC(CCN2CCCC2)OCC)cc(C(F)(F)F)c(Cl)cc1F c1(C2C(C(=O)OC(C)(C)C)(CNC(c3coc(Br)c3)=O)C2)ccccc1 C(=O)(N1OC2C=CC1CC2)C1(C(C)C(=O)NC2CC3(CCCO3)C2)CC1 C1(Cc2nnc(C)o2)CCCCN1C(=O)NCC1CCN(c2ccccc2Cl)C1 N1(C(COCCCC)=O)CCCC(NC(=O)C(c2ccnn2C)O)CC1 C12(CCC(C)(C)C1)C(=O)N2.c1(OCCNC(C(C)C)=O)ccccc1 C(=O)(C1=CC2CCC(C1)C2)N(C(CNC(C(CC(=O)OC)C)=O)C)C c1(OC)cccc(OCCN(C)C(C2CN3CCC2C3)=O)c1[N+](=O)[O-] Cc1c(CC(N2CC(CC(C)NC(C3C(C)C3C)=O)C2)=O)cccc1[N+](=O)[O-] CCC(C(=O)N1CC2(NC(=O)CCc3cn(C)nc3C)CCC1CC2)C(F)(F)F C#CC1CCCN1C(c1ccc(CC(=O)N(C)C)cc1)C(=O)NCCOC C(=O)(C1=COCCC1)N(CCCCCC)CCNC(=O)C(C)(O)C(C)C N1(C(CCOCCC)=O)CCC(C2CC2)(CNC(=O)C(O)C(F)(F)F)C1 C1(C(CNC(c2c(C)csn2)=O)(C)O)CCN(C(=O)Cn2ccnn2)CC1 c1(C(N2CCC(C(=O)OC)(CO)C2)C(=O)NCC(=C)C)c([N+](=O)[O-])ccc(Cl)c1Cl N1(C(c2c(C)nsc2)=O)CCOC(CCCNC(c2cn[nH]c2)=O)C1 O=C(CC(C(F)F)N1CCOCC1)NCC1CC(NC(C2(O)CCC2)=O)C1 N1(C(C2CCN(C(CCc3ccn(C)n3)=O)C2)=O)CCCCC(F)(F)C1 c1(SC)cc(C)ccc1C(=O)NCC1(NC(C2CC2C)=O)CCC1 C(=O)(CC(C(C)C)n1cc(CCNC(C)=O)nn1)NCc1ccc(CC)cc1 C1(=O)CC(C(F)F)N1.C(CO)(C(=O)NC(C)CC1CCC1)OC C#CC1(O)CCCN(C(=O)C(CCC)NC(=O)C(CC)=CCCC)C1 C(=O)(C1=CC2CCC1C2)NCCC(C)N(C(CCCOc1cccc(C)c1)=O)C c1(NC(C2CCCC(C)C2)=O)cnc(Cl)cc1C(=O)Nc1cccnc1 CC(CC(F)(F)F)C(=O)N(CC(C)NC(=O)C(C)(C)c1ccc(Cl)s1)C c1(OCCCC(N2CC(NC(C3(CCF)CCC3)=O)C3CC23)=O)ccc(F)cc1 c1(C(=O)NCC2N(C(CC=C)=O)CC(C)(C)OC2)c(C)nc2ccc(Br)cn12 N1(CC(=O)NCc2cnn(COC)n2)CCNC(=O)C1CC c1(C(N2C3C(NC(C4(C)CC(=C)C4)=O)CC(C3)C2)=O)n[nH]c2c1CCSC2 C1(NC(CCn2ccc(C)n2)=O)CN(Cc2ncc(C)s2)CC1O C=C1CC2(C1)CC(C(=O)NC1CCN(C(=O)C(C)Sc3nncn3C)C1C)C2 C1(C(=O)NCc2c(C(=O)NC(C(C)F)C)nco2)CNC(=O)CC1C N1(C(=O)Nc2ccc(Cl)cc2O)CCCN(Cc2ccc(Cl)cc2Cl)CC1 C1(NC(c2cccc(O)n2)=O)CC1C1CCCN(C(=O)CCNCC(F)(F)F)C1 C1(CNC(=O)Cn2cnnc2O)CCC2(CCC2)CN1C(c1ccon1)=O N1(C(C=Cc2nnc(C(C)C)o2)=O)CCC(NC(c2cnn(C)n2)=O)C(O)C1 N1(C(=O)C2=CCCC2)CCC2CC2(C(=O)Nc2ccc(F)c(O)c2)CC1 Cc1ccnn1C(C)C(N1CCC(CCNC(=O)CC2CCC2(C)C)C1)=O CCCCC(CC)CC(=O)N1CC2CC(NC(C3(C)C=CCC3)=O)CC2C1 CC1CN(C(=O)Cc2cnoc2)CCN1C(c1cc(Cc2cccs2)on1)=O CCC(C(=O)NCCOCCCN(C)C(c1cnccc1C)=O)C(C)O N1(C(Cc2cc(C)no2)=O)CCN(C(C2CC2C2CCCC2)=O)C(C)C1 C(=O)(C(CO)C(C)(C)C)NCC(CC)(CC)NC(=O)CCC=CBr N1(C(C(C2CC2)NC(C)=O)=O)CCOCC1C1(NC(C)=O)CC1 C(=O)(C(C1CN(C(=O)Cn2cccn2)C1)OC)NC(CC)C1CCC1 C(C(=O)NC(CNC(=O)COc1ccsn1)CO)(C(C)C)Nc1c(C)nn[nH]1 C1(NC(CN(CCOC)C)=O)CN(C(C2CCCC(=O)N2)=O)CC1S(C)(=O)=O C1(F)(C(N(CC(F)(F)Cl)C)=O)CCCN(C(=O)CCC2CCCO2)C1 c1(OC)cc(C)cc(C(=O)NC(C)CNC(c2c[nH]nc2-c2ccoc2)=O)c1O N1(C(C(CC2CC2)OC)=O)CCN(C(C2CCCC2C(C)C)=O)C(C(C)C)C1 c1(C(N(CCOCCN(C(C(C2CC2)OC)=O)C)C)=O)cccc2c1OCCO2 CCC(C)CCCC(=O)N1CCC(C2CC2)C1CNC(C1CCCC1O)=O CC1CC(C(=O)NCCC(=O)OC(C)(C)C)CN(C(c2ccc[nH]2)=O)C1 C12(C(N(C)Cc3ccc(CNC(C(C)SC)=O)cc3)=O)CC3CC1C2C3O N1(C(C(C2CCN(C(c3ncc(C)nc3)=O)C2)(C)C)=O)CCCC2(C=CCO2)C1 c1(C(N2C(CNC(C(CC)OCC)=O)C=CC2)=O)cc(OC)ccn1 CCCCC(CNC(=O)CCn1nc(C)cc1C)NC(c1nnc(S)n1C)=O c1(CC)onc(C(=O)NC(C)C(C(C)C)NC(=O)CCc2ccccc2Cl)c1C N1(C(C2CC(CC)C2)=O)CCN(C(=O)CCCN2CCCC2)CC1CCOC C=CCC(C)(C)CC(=O)N(C(C(=O)N1CCC(CCOC)C1)C(C)CC)C c1(OC)nc(C(=O)NCC2CCCN2C(=O)CCC2CCC(O)CC2)cc(O)n1 Cc1cc(C(=O)NCC2C(Cn3cc(C(=O)OC(C)(C)C)nn3)C2(F)F)on1 C1(c2ccon2)(CC(N2CCC(CCNC(c3cnc[nH]3)=O)C2)=O)CS(=O)(=O)C1 Cc1csc(C(=O)NC(C2CCN(C(C3CCN3C)=O)C2)C)c1Cl C(C(CC(=O)NOC(C)C)C1CCC1)NC(C(COCC)(F)F)=O S(=O)(=O)(c1[nH]c(=NCC2CCCC(C)O2)ccc1Br)NCCc1cccc(C)n1 C1(C)(CNC(c2c(OC)nsc2)=O)CCN(C(=O)CCC2CC(C(=O)OC)CO2)C1 c1(C(=O)CC#N)ncccc1-c1cccc(O)c1.c1(C(C)(C)O)cn(CCN)nn1 c1(C(=O)NCCOC2CN(C(c3c(C)ncs3)=O)C2)ccc(P(C)(C)=O)o1 c1(C(=O)NC2CCC(NC(c3cncc(N)c3)=O)C2)cnn2ccccc12 c1(C(N2CC(N(C(CC(CC)C)=O)C)C2)=O)ccc(OC)c(OC)c1Cl CC(C)C(F)(F)CN=c1[nH]c(N2C3CCC2c2ccccc23)nc2cc[nH]c12 C1(CC)CN(C(=O)Nc2cn(C)nc2-c2ccco2)CC1c1cncn1C Cc1cc(NCCCCN2CCCC2)c(S(N)(=O)=O)c(F)c1 N1(C(CC2CC(=C)C2)=O)CC(NC(C2CCN2C(C)(C)C)=O)C(C)(C)C1 CC(C)C(C)CCNC1(c2nnnn2Cc2cccs2)CC(Cn2ccnc2)C1 C(=O)(C(C)CC(C)(F)F)NCCOCCOC.C(CC)N(CCOC)C N=c1[nH]cc(C(=O)NOCc2ccc(Cl)cc2)c2cc[nH]c12 C1(CCN(C)C(C)=O)(NC(C(C)OCCC=C)=O)CCN(C(=O)CCCSC)C1 C1(CC=C)(C(=O)NC2CC(C)N(C(=O)OC(C)(C)C)C2)CCOCC1 N1(CC(=O)NCCCN(C(C)C)C(c2ccc(O)cn2)=O)CCC(N(C)C)CC1 CC(C)C(C)C(CNC(=O)C(Cl)=CCl)NC(=O)COCCOCCO C1(C)(C(=O)NCCNC(c2ccc(CCC)cc2)=O)CC2C=CC1C2 N1(C(c2cc(OC)c(C)nc2)=O)CC(NC(=O)Cn2cccn2)CC12CCCC2 C1(NC(CCOCCOC)=O)CCN(C(c2ccc(Br)s2)=O)C1 c1(C(N2CC(C(C)NC(c3nccc(C)c3)=O)C2)=O)ccc2c(c1)CNC2=O C(C)(C(CC(=O)NC1CCOCC1C)NC(=O)CC1CNC(=O)O1)OC CCCS(=O)(=O)NC(C)C(=O)NC(C1(O)CN(C(c2cnn[nH]2)=O)C1)C c1(CN(c2ccnc(F)c2Cl)C2CN(C(=O)C3CC3)CC23CC3)cnc2cccnn12 N1(C(C2(C(F)F)CC(=C)C2)=O)CCOC(C)(CNC(c2cncc(F)c2)=O)C1 N1(CC(=O)NCCCC(C)NC(=O)C=Cc2ncco2)CCCS1(=O)=O Cc1cc(C#N)sc1C(N1CCOC(C)(C(C)C)C1)C(=O)NCC(C)C CCS(=O)(=O)CC(=O)NCC1CC2CCC1N2C(=O)C(C)(O)c1ccccc1 N1(CO)CC(N(C(=O)C(C)C2CN(C(C34CC(CO)(C3)C4)=O)C2)CC)CC1=O c1(C(N(CCN(C(C2CCC2C(=O)OC)=O)CC)CC)=O)cc2ccccc2[nH]1 Cc1ccc(F)c(C(=O)NCC#CCNC(C2C(C)CC2C)=O)c1F c1(C(=O)NC2(c3cccnc3F)CC2)ccc(-n2cccn2)nc1 CN1CCCC(C(=O)NCC2C=CC(NC(=O)CC(F)(F)Cl)C2)C1 c1(C(=O)NC2(CNC(C3CCC(C)C3)=O)CCCC2)ccnc(P(C)(C)=O)c1 C(=O)(C1CCc2c(Br)cccc21)NCc1cccc(NC(C(C)(C)F)=O)c1 C(=O)(CC(C)(C)C(F)F)N1CCN(C(C)=O)CC1.c1(C(C(=O)OC)N(C)C)cncn1C N1(C(C2(CCn3cc(C(CC(C)C)(C)C)nn3)CC2)=O)CCN(C)CC(O)C1 C1(NC(c2n(C)ncc2)=O)CC(=O)N(C2CN(Cc3cnc(Br)s3)C2)C1 C1(CC)COCCN1C(=O)CCc1cn(Cc2ccc(C3CC3(F)F)cc2)nn1 N1(C(CC=CC=C)=O)C2CCC1CC(NC(C1Cc3ccccc3S1)=O)C2 N1(C(CCCC(=C)C)=O)CC(C)CN(C(c2cc3c(Cl)nccc3s2)=O)C(C)C1 N1(C(CSCCC(C)C)=O)CCc2nc(CNC(C3C4CCCOC34)=O)sc2C1 N1(C(C(C)SCC)=O)CCC(F)(CNC(=O)CCc2cccnc2OC)C1 N1(C(c2c(N)ccc(OC)c2)=O)CCCN(C(C2CC2CF)=O)CC1C CS(=O)(=O)CCC(=O)N1CCC(NC(=O)NCCCl)C(C(F)(F)F)C1 C1(CN(C(C(CC)NC(C)=O)=O)CC)CCCCN1C(c1ccc(C(C)C)o1)=O N1(c2snc(CC)n2)CCCC(CCNC(c2cc(F)cnc2OC)=O)CC1 Cc1nc(CCCOC(c2cn(CC(=O)N3CCC3)nn2)=O)oc1-c1ccccc1 N1(C(CNS(CCC)(=O)=O)=O)CCCC(N(C)C(c2ccsc2COC)=O)C1 C(C(=O)NC(c1ccccc1)CNC(c1cnccc1Br)=O)(C(C)C)OC Cc1nc(NCC2CC=CCC2)cc(=NCc2ccc(S(N)(=O)=O)c(C)c2)[nH]1 c1(CC(N2CCC3CN(C(=O)CCOC4CC4)C3C2)=O)cccc2ccncc12 c1(CC(=O)NC2CC(NC(C(C#C)(C)C)=O)CC2O)ccc(F)c(OCC)c1 CCC(C)C(C(=O)NCCCC(C)NC(C1(n2cc(Cl)cn2)CC1)=O)NC(C)=O c1(N(CC(=O)OC)CC2CCCO2)nnc(N2CCCC2)n1CC(C)C(F)(F)F C1(C(=O)NCC2(NC(CSCCCC)=O)CCOC2)CC2CC(=O)C1C2 N1(C(c2c(C)csc2Cl)=O)CCC2(CC1)CN(C(C1CCCN1C)=O)CC2CO c1(C(N2CC(C)CC(NC(Cc3cnc(C)[nH]3)=O)C2)=O)oc2ccccc2c1C CCC(CC(C)C)C(=O)N(C1CN(C(C2CCC(=C(C)C)CC2)=O)C1)C1CCC1 N1(C(c2c(C)sc(O)n2)=O)CC2CCCC(C1)N2C(=O)C(=O)N=S(C)(C)=O C(C(C(C)C(C)C)NC(C1CCC1C#N)=O)NC(CCC(=O)NC)=O c1(CNc2c(CC(N3CCC4(CC3)CC4)=O)nccc2)ccc2nc[nH]c2c1 C12(OC)CCC(C1)OC21CN(C(c2cnc(C3CC3)o2)=O)C1 C1(C(=O)NC2(CC)CCCN(C(=O)C(C)(C)F)C2)CCOC2(CCC2)C1 CN=c1cc(C(N2CCCC(C(=O)NCCc3cc(C)no3)CC2)=O)cc[nH]1 N1(C(C(C=C)(C)C)=O)CC2CCC2(CCNC(c2c(C)cccc2F)=O)C1 Cc1cc(Cl)ccc1N(C)Cc1cnn(CC2CCOCC2)c1 c1(C(=O)NCC(C)N(C(C2(F)C(C)CCC2)=O)C)ccc(=O)n(C)c1 c1(C(=O)NC2CC(NC(C3(C(C)C)COC3)=O)C2)ccccc1NCC(N)=O C12(NC(C(CCCC)C)=O)CCCC1N(C(c1ccc(Cl)cc1NC)=O)CC2 C1(CCC)CCC(C(=O)NC2CCCCC2NC(=O)C(C)C(=O)OC)CC1 CCC(CC)CC(F)C(=O)N1CCC(Cn2cc(OCc3ccsc3N)nn2)C1 C1(C(=O)OC)CC12CN(C(C1CC(NC(=O)CCCc3cnn[nH]3)C1)=O)C2 N1(c2snc(C(C)(C)OC)n2)CC2CC(NC(c3cc(Cl)ccc3F)=O)CC2C1 C(=O)(C1=CCCOCC1)N(C1CCN(C(Cc2nc(C)sc2)=O)C1)CC1CC1 C1(C)(C(=O)NCC2(CCNC(C3(C)N(C)CCC3)=O)CC2)CCCNC1=O N1(C(C2COC(=O)O2)=O)CCC2(CC1)CC2NC(=O)C(F)(F)Sc1ccccc1 C=CCC(CC)C(=O)NC1CCCC1NC(=O)C(c1ccc(F)cc1)=O Cc1cnc(C(=O)N(C(CNC(c2scnc2C(C)C)=O)C2CC2)C)cc1Br N1(C(CCC2CCN(C(COCCOCC#C)=O)C2)=O)CCOC(CCC)C1 c1(C(C)=O)cc(C(N2CCC(C3CCCN3C(=O)CSSC)C2)=O)[nH]n1 CC1CCc2nc(C(=O)Nc3ncn(Cc4ccccc4)n3)cn2C1 c1(C(N2CC(C)C(NS(=O)(=O)C(F)(F)F)C2)=O)ccc([N+](=O)[O-])cc1 CC1(O)CC(C(=O)NCc2cc(C(=O)NCC(N3CCOCC3)C)n[nH]2)C1 c1(C(=O)NCC(CN(C(=O)C(C)SC(F)(F)F)CC)(C)C)ccc(C(C)=O)nn1 c1(N2C(=O)OC(c3ccccn3)C2)ccc(NN2C(=O)C3CCCCC3C2=O)cc1 C1(C(F)(F)C(=O)NC2CCCC(NC(C3CC=CCO3)=O)C2)(OC)CCOCC1 C=C(Cl)C(C)(C)C(=O)N1CC(O)(CCNC(c2sc(C(C)C)nc2C)=O)C1 Cc1nnc(C(=O)N(C2CCN(C(=O)CCc3c[nH]c(C(N)=O)c3)C2)CCO)s1 c1(C(=O)NC2CC(CNC(C3(C)CC4CCC3O4)=O)C2)cn2cccc(F)c2n1 Cc1nc(C(N2CCC(O)(C(=O)NCCc3ccccc3)C2)=O)n2c1CCC2 CCCC(C#N)C(=O)NCCNC(=O)C(C(C)C)N1CCC(C)CC1 c1(N2CCC(CC=C)C2)nc(N2CCN3C(=O)NCC3C2)nc2c1CSC2 N(C(=NCCCSC)NCC1(C2CCC2)CCC1)C(CC)C C1(C(=O)NCC2CCN(C(c3cc(C)nc(O)n3)=O)C2)CCc2cncn2C1 C(=O)(CCCCCC(C)C)N(CC(CC)NC(c1c(Cl)cccc1Cl)=O)C N1(C(C2C(C)(C)CCN2C(C2C3CC4C(C3)C24)=O)=O)CCC2=C(CCCC2)C1 N1(C(=O)NC(CCC)Cn2ccccc2=O)CCc2cc(F)ccc2C1 c1(CC(N2CCC(C(C)NC(C3CC3CF)=O)C2)=O)cccc(C#N)c1 N1(C(CC2C=CC(NC(C3(C)CCC3)=O)C2)=O)Cc2ncsc2C1 C(=O)(C(CC)C(=O)NC(C1(CNC(c2cc(Cl)ccc2C)=O)CC1)C)OCC c1(C(N2CC(CNC(C(C)SC)=O)OCC2)=O)ccc2nc(C)c(=O)n(C)c2c1 c1(C(=O)NC(CCCC)C)ccc(-c2cccnc2)c(Cl)c1 C(=O)(C(CC(C)(C)C)OC)N1CCC(C)(NC(C(COC)(F)F)=O)CC1 C1(C(=O)NCC2(OC)CCC2)CN(C(C)=O)CC1OC(C=CC)=O.C(C)(C)C N1(C(COCCOCCOC)=O)CCOC(CNC(C2CC23CC3)=O)C1 c1(C(CN2CC3C(NC(=O)OC(C)(C)C)C3C2)=O)cccc2ccc(Cl)nc12 c1(CC(C)N(C(=O)C(C)NC(C)(C)C)C(=O)CC2COC(=O)C2)ccc(F)cc1 C(=O)(CCC(=O)NC1CC(NC(C2CCC(c3ccc(F)cc3)O2)=O)C1)NC c1(C(N(CCNC(=O)C(C)N(CC(F)(F)F)C)CC)=O)cnn(CCO)c1C C#Cc1cccc(CC(=O)NC(C2CC2C(=O)NC2CNC(=O)C23CC3)C)c1 C(=O)(C(C)(C)C(C)(F)F)NCCN(CCC)C(C1CCN(C)CC1)=O Cc1ccc(=N)[nH]c1C(=O)NCC1CN(C(c2n[nH]cc2C)=O)C1 C1(COC)COC(CNC(c2cocc2)=O)C1.c1(CC(=O)N)cn(C2CC2)cn1 C1(CCNC(Cc2cn(C)nn2)=O)CSCCN1C(c1cnns1)=O N1(C(CCc2scc(C)n2)=O)CCN(C(C2COC(=O)N2)=O)CC1C(F)F C1(O)(C(N(CC)CC2CCCO2)=O)CCCN(C(C2CC3(CSC3)C2)=O)C1 C1(N(C(=O)Cn2cc(C3CC3)nn2)C)CN(CC(N)=O)CC12CC2 C(=O)(CCC(=O)NC1C2CN(C(c3ccc(N(C)C)nn3)=O)CC12)N1CCC(C)C1 C1(NC(c2n(C)cnc2)=O)CCC2CCN(C(c3ccc(C(F)(F)F)o3)=O)C1C2 c1(C(N(C2CCN(C(=O)C(c3ccc(C)o3)C)C2)CC)=O)csc(Cl)n1 c1(N2C(C(=O)NC3C(C)CCC(C)C3)CC(F)(F)C2)ncc2ccn(C)c2n1 N1(C(COCC#C)=O)CCN(C(=O)CNS(C)(=O)=O)CC1C(F)F c12ccc(c(Br)c1)NC(=O)C2(F)F.C1(C(C(=O)OC)O)CCC(CN)CC1 c1(C(N2C(C)C(NC(c3csc(C4CC4)n3)=O)CCC2)=O)ccc2n[nH]cc2c1 C1(C(=O)NCC2CC(F)(CNC(C=CCOC)=O)C2)CCCCC(F)(F)C1 c1(C(N2CCC(O)C2)=O)ccc(C(=O)NCCN(C)C)o1.CC(C)(C)SC.C12CC1N2 c1(C(C)C)cc(N2CC3C(CNC(=O)CN4CCCNC4=O)C3C2)nc(C(C)C)n1 N1(c2ncc(C#N)nc2)CC(NC(C2CN3CCC2CC3)=O)CC2(CC2)C1 c1(C(N2C(CC(=O)NCc3cccc(Br)c3)CCC2)=O)ccc([N+](=O)[O-])cc1O c1(C(=O)NCC2CC(NC(=O)COC3CCCCCC3)C2)nc2ccccc2s1 Cc1ncsc1CCC(=O)NCC1(O)CN(CCOCF)C1 N1(C(C2CCCN2C(=O)CCCn2cccc2)=O)CCOC2CC12 c1(C(N2CCC(F)(C(=O)NCCCNC(=O)NC)C2)=O)ccn2ccnc2c1 N1(C(c2ccc(OC(C)C)cc2)=O)CCN(C(C2CCCN2C)=O)C2CCC12 c1(C(=O)NC(C)CC(C)NC(=O)Cc2ccc(Br)cc2)cc(O)cc(C#N)c1 CCCCCCCC(F)C(=O)NCCCNC(=O)C(=Cc1cccnc1)F C1(OC)(CNC(=O)C(O)C(C)C)CCN(C(=O)CCC=CC(C)C)C1 C1(NC(C2(OCC)CCOCC2)=O)CCN(c2nc(C)nc(=N)[nH]2)CCC1CO C(=O)(C(C)(C)CSC)N(CCCCNC(c1nc(C(C)OC)sc1)=O)C.C1(O)CC1 Cc1[nH][nH]c2ncnc(=NC(C)C3CCCN(C(=O)CC(C)(C)O)CC3)c1-2 C(=O)(CS(=O)C(F)(F)F)N1CCC(C2(CNC(C(CSC)C)=O)CC2)CC1 C12(C(=O)NC(C(C)NC(=O)CC3(CO)CC3)(C)C)CC1COC21CCC1 C(CN=c1[nH]c(N2CCCC(C(N)=O)C2)nc2ccccc12)N1C(C)COCC1 C=CC(C)(CCOC)C(=O)NC1CCCC1CNC(=O)CN1CC2CCC1C2 c1(NC(c2nc(-c3ccc(OCCC)cc3F)sc2)=O)c(O)cccc1[N+](=O)[O-] n1(C(C)C)cc([N+](=O)[O-])c(=NCC2CN(C(C3CCCN3C(C)C)=O)CCC2C)[nH]1 N1(C(C(C)C2CCCC2)=O)CC(C(=O)N(C)CC2(C)CC2)CCC1(C)C N1(C(CCN(C(=O)CC2CCCOCC2)CCO)=O)CCC2OCCC2C1 Cn1cc([N+](=O)[O-])c(C(N2CCC(n3cc(CN4CCCOCC4)nn3)C2)=O)n1 c1(C(Cn2cc(NC(=O)Nc3ncc(I)cn3)nn2)O)ccc2c(c1)CCO2 C1(OCCC)CCC(C(=O)NCCC2CCN(C(C34CC3C4)=O)C2)CC1 C1(F)(CNC(=O)CC2NC(=O)CNC2=O)COCCN(C(c2cc(Cl)c[nH]2)=O)C1 C(CNC(c1cscc1-c1ccccc1)=O)(C(C)C(C)C)NC(C#CC(C)C)=O CCC(CC(=O)N1CCC(N(C(c2ccc(C)c(Cl)c2)=O)CC2CC2)C1)C(C)C CCCCN=c1ncc(NC(C23CC(CO2)C3)=O)c[nH]1 C=C1CC(C(=O)NC23CC(F)(C2)C3)(CNC(c2cnco2)=O)C1 c1(OC)ccc2c(C(=O)NC(C)C(C)(C)NC(C3CC3C(N)=O)=O)coc2c1 c1(CC(N2CCC(CN(C(=O)Cc3cncn3C3CC3)C)C2)=O)cccc(O)c1 c1(N(C)C)cccc(C)c1C(=O)NCCN(C(C12CCCC1(C(N)=O)C2)=O)C1CC1 C1(C(N2CC(CC3(C(=O)NC(=O)OC)C=CCC3)C2)=O)CC12CCS(=O)(=O)CC2 c1(CCCC)nnc2cc(N3CCC(C)(NC(c4csc(C)n4)=O)CC3)ncn12 N1(CC(N2C(CNC(C(COC)OC)=O)C=CC2)=O)C(C)=CC(C)=NS1(=O)=O C(=O)(C(CC(C)(C)C)NC(=O)Cc1ncoc1C)N(CC(C)(O)C1CC1)CC c1(C(=O)NCCN(CC(C)O)C(C2C(C)C2C)=O)ccc(C2=CCOCC2)cc1 C1(C(=O)NCC2CC(CNC(C3(CCF)CCC3)=O)C2)(CC)CC1(F)F c1(C(N2C(CC(=O)O)CC2)=O)ccc(C2CCCO2)cc1 Cc1cnnc(O)c1C(=O)NC1CC(C)(NC(c2cnn(C3CC3(F)F)c2)=O)C1 c1(C(=O)NCC(C2CCCC2)NC(Cc2cc(C(C)=O)sc2)=O)c(C)csc1Cl C1(C(=O)NC(C)CN(C(=O)CCCSc2ccncc2)C)CC(C2CC2)C1 c1(C(=O)NCCCC(=O)OCc2ccccc2)ccc2[nH]nc(Cl)c2c1 Cc1ccn2cc(C(=O)NCC(O)CNC(=O)CC(C)CC(F)(F)F)nc2c1C N1(C(CC(=C=C)C)=O)CCCCCC1C(=O)NC(C)CS(N)(=O)=O C1(CNC(C(c2c(F)cccc2Cl)C)=O)CC2COCC2N1C(=O)C=C1CCC1 c1(CC(=O)NCCCN(C2CCCC2)C(COCCC#C)=O)cccc(N)c1 N1(C(CC=CC=C)=O)CCCCC(NC(=O)CCP(C)(C)=O)CC1 C(=O)(CC(C)CF)N1CC(CC=C)(NC(=O)C(C)CNS(C)(=O)=O)C1 N1(C(c2nc(NS(CC)(=O)=O)sc2)=O)CCSCC1CCNC(C1CC12CC2)=O C1(C)(NC(CCC)=O)CCCN(C(=O)CC2CN(C)CC2O)C1 CC1CC(CCNC(c2ccc(F)c(N)c2)=O)CCN1C(c1ccon1)=O N1(C(C2(CC(N)=O)CC2)=O)CC2(CCN(C(=O)CC(O)C3CCCC3)CC2)C1 N1(C(C2(n3cc(-c4ncccc4Cl)nn3)CC2)=O)CC2CC1CC2OCC Cc1ccc(Br)cc1CC(=O)N(C)CC1(NC(=O)C(O)c2ccco2)CC1 N1(C(c2c(CCC)occ2)=O)CC(CNC(C2(CF)CC2)=O)C2(CCC2)C1 c1(CC)c(OC)cccc1C(=O)NCC(C)(CC(C)C)NC(=O)C1=COCCO1 c1(CC(=O)NCC(c2cnn(C3CC3)c2)CC)ccc(C2CC2)nc1 c1(C(=O)NC2(CF)CCN(C(C3N(C(C)C)CCC3)=O)C2)ccnc2ccnn12 CCCC(C(F)(F)F)NC(=O)C(=O)CCNC(=O)CN C12CCOCC1C(=O)N2.O=C(C(O)C1CCCC1)NC1CN(CCO)C1 C1(C(=O)N(CCCCN(C)C)C)(CNC(c2cn(CCC)nn2)=O)CC12CCC2 Cc1ccncc1CC(=O)NCC1CC1C(=O)Nc1cc(C2CC2)n(C)n1 C1(C(N2CCOCC(CNC(CCC3C(C)C3)=O)C2)=O)CS(=O)(=O)CC(=O)N1 C(CC(C)C(=O)NC(CO)C(C)NC(=O)CCC1CC(F)(F)C1)=CCC CC1CN(C(=O)C=C(Cl)Cl)CC1CCNC(c1cn(CC2(C)COC2)nn1)=O c1(Cc2nc(C(CCCC)CO)on2)cc2c(Br)cc(OC)n2[nH]1 N1(C(C2(C=C)CCC2)=O)CCCC(C)(CNC(=O)CCOc2cccc(Cl)c2)C1 N1(C(C(CC)NC(N)=O)=O)CCC2(CC2NC(=O)Cn2nnc(C3CC3)n2)C1 c1(C(C(=O)OCCC(C)(C)CNC(=O)CC2(n3ccnc3)CC2)F)cccc(F)c1 N1(CC(C(c2c(C)cccc2)C(C)(C)C)=O)C(=O)CN(CC(C)C#N)C1=O.N C1(C#N)(C(=O)NCC2N(C(c3nc(CC)oc3)=O)CCCC2)c2ccccc2C1 N1(C(c2nc(Br)cs2)C(=O)NCCCC(=O)OCC)CC(C)OCC12COC2 N1(C(CCOC(C)=O)=O)CC2CCC(C1)C(NC(c1cccc3[nH]ncc13)=O)C2 N1(C(c2nc(C)sc2)=O)CCOCC12COCCN(C(C1C=CCCC1)=O)C2 CC1(C(=O)N(N2CCOCC2)C(C2CCCC2)(C)C)CCCS1 Cc1cccc(C(=O)NC2CCCC(NC(C3CCCSC3)=O)C2)c1Cl N1(C(CC2CCCN(C)C2)=O)CCN(C(C2(O)CCCCCCC2)=O)CC2(CC2)C1 c1(C(=O)NCC2(F)CN(C(C=C(C)C(C)(C)C)=O)C2)cccc2nc(O)ccc12 C=CCC(CC)C(=O)NC(c1ccc(N(C)C)cc1)CNC(c1c[nH]c(C#N)c1)=O N1(C(c2ccn(C3CCC3)c2)=O)CC2CN(C3CC3)CC2C1 C1(NC(CC)=O)CCCN1CC(=O)N(CCCc1ccoc1C)CC c1(C(N2CCC(C(C)NC(=O)C(C)(C)C(F)F)C2)=O)cncc2cccnc12 C(c1cccc(F)c1Cl)=CC(=O)NCC1CCC(C)C(C)C1 N1(C(C(=O)OC)C)CCN(C(=O)NC2CCCN2C(=O)C(C)CF)CC1 N1(c2nccc(C)n2)CC(NC(c2cncc(F)c2)=O)C2CCCCC12 c1(NC(c2nccc(C)c2)C)nccc(=NC(C)COc2ccc(C)c(C)c2)[nH]1 CCCC(CNC(=O)CN(C)C1CC1)C(=O)NCCCc1cccs1 Cc1nc(C(=O)NC2C=CCN(C(=O)C(O)C3CCCC3)C2)sc1C(C)(C)C Cc1oc(C#N)cc1C(=O)N(CC(C)(C)NC(=O)CCCC(=O)NC(C)C)C N1(C(c2nc(CC)oc2)=O)CCCC(CN(C(=O)Cn2cc(C(N)=O)cn2)C)C1 n1(CC(N2CCN(C(C3C(=C)CC3)=O)C(CC)C2)=O)ccc2ccccc2c1=O C=CCCC(C(=O)OC)NC(=O)C(CNC(=O)Cc1scnc1C)C(C)C c1(SCC2N(C(=O)OC(C)(C)C)CC=C2)nc2c([nH]1)CCCC2 c1(NC(C2(C)CCCN2C(c2ccnc(F)c2F)=O)=O)ncc([N+](=O)[O-])cc1Br N1(C(c2ccc(C)s2)=O)CC2(CC(NC(=O)C(C)O)C2)C1 C1(CCOC)(NC(=O)CCNC(N)=O)CCN(C(c2cc(C)cs2)=O)C1 CCC(CO)(C(=O)N1CCCC(CNC(=O)C=C(Cl)Cl)C1)OC N12CCCC(C1)C(=O)N1CC(C1)C2.c1(OOCCCCC)ccccc1C c12ccc(C(F)(F)F)cc1CN2.c1(C(C(N2CCCCC2)=O)O)ccc(F)cc1 C=C(C)CC(=O)N1CCC(C(N2CCc3c(nnn3C)C2)=O)O1 c1(CC)nc(=N)[nH]c(=NCC2CCCC(NC(c3ccc(=O)n(CC)c3)=O)C2)[nH]1 CC(C)C(O)CC(=O)N1CCC(O)(C(=O)NCc2ccc(O)nn2)CC1 S(=O)(=O)(c1cc(C)cnc1NCC1(C)CCN(C)CC1)NC(CCSC)C Cc1ncnc(C)c1CC(=O)N(CCCNC(C1CCCN1C)=O)CCO C1(C(=O)NCC2CN(C(CN(C3CC3)CC)=O)CC2O)CCCCC1(C)C C(=O)(CCCN(C)CCN(C=O)C1CC1)O.c1(C(C(=O)N(C)C)O)ccccc1 CC(C)CCCC(C)C(=O)N(CC(N1CCC(NC(=O)CSC(F)F)CC1)=O)C N1(C(C(C2(O)CN(C(C3C(C)CCO3)=O)C2)F)=O)CCCCCCCCC1 CCCCCC(C)(CC)C(C)(c1nnnn1C1CCC1)NCC=C1CCSCC1 C1(C(=O)NCCC(CNC(=O)CC2CCOC2)O)CC(=O)N(C2CC2)C1 CCC(C)C(C(=O)N(C)Cc1csc(=N)[nH]1)N(C)C(C1CC(O)C1)=O C12(CNC(N3CC(c4ocnc4)C3)=O)CCCN1CCC2.CC(CC1CC1)C(=O)NC C(=O)(C#CC1CCCCO1)N1CC(C)(NC(CCN(c2ccccc2)C)=O)C1 C1(CN(C(c2cnc(C(C)C)s2)=O)C)CN(C(=O)C(N2CCOC2=O)C)CCO1 c1(C(=O)NCC(CNC(c2cc(C)cc(Cl)c2)=O)O)cc2c(F)cccc2s1 Cc1ncc(Cl)cc1CNC(=O)CC1CCN(C(c2cccnc2)=O)C1 N1(C(CCNC(COC)=O)=O)CC(CNC(=O)CN2CCC2C)OC2COCC12 C1(C(N2CC(O)(CNC(c3cccc(C4CC4)c3)=O)C2)=O)CC2(CCC2)CO1 Cc1cnn(C)c1C(=O)N(C(CNC(C1CC(N(C)C)CCO1)=O)C1CC1)C C12=NC=C(Br)C(=NCC3CCC(C3)NC1=O)N2.C12(CC)CC3CC(C(=O)N1)C2C3 C(=O)(CS(=O)(=O)CC1CCCO1)N(C1CN(C(C2CC(=C)C2)=O)C1)C C1(C(=O)O)(CCC2CC2)CCN(C)CC1.Cc1noc(NC(c2cn(CCO)nn2)=O)n1 Cc1cnc(C(C)NC(c2cc(CNC(=O)Cn3cncn3)cs2)=O)s1 CC(C)C(CCN(C(=O)C(N1CCC(C)(O)C1)C)C)NC(=O)C(C)N(C)C CCCCCC(O)C(=O)N1CSCC1C(=O)NC(CN(C)C)CCO C(=O)(NNC(=O)Cc1csc(Br)c1)C1(C(C)C)CNC(=O)C1 C1(C(N2C(C)C3(CC2)CCC3)=O)CCN(C(=O)CC(F)(F)C(F)F)C(C)(C)C1 c1(C(=O)NC2COCCN(C(c3ccnc(Cl)c3)=O)C2)ccnc2c1CCC2 N1(C(Cc2c(C)con2)=O)CCC2CN(C(=O)C(C)(C)C(C)(F)F)CCC2C1 C(C(C)(CC(C)C)NC(C1COCCO1)=O)NC(=O)Nc1c(OCC)cccc1 Cc1ccc(C(=O)NCC(c2cccc(Cl)c2)NC(=O)C(C)C#N)c(F)c1 N1(C(CC2CCC(C)O2)=O)CCCC(C2CCN(C(c3ccccn3)=O)CC2)C1 CC(C(C)(C)CO)NC(C1(NC(c2ccccn2)=O)CC1)=O Cc1ccc2c(C(N3Cc4cccc(Br)c4C3)=O)[nH]nc2n1.N(C)CC Cc1csc2ncnc(NC3CCCCN(C(c4cccc(=S)n4O)=O)C3)c12 CC1(C)CC(C(=O)NC2(CC(N3CC(F)(CO)C3)=O)CCC2)=NO1 C1(O)(CNC(C(C(C)C)(C)O)=O)CC2CCC(C1)N2C(=O)CCOC1COC1 N1(C(Cc2c(C)occ2)=O)CCCCCC(NC(c2n[nH]c(C)c2F)=O)C1 CC#CCCCC(=O)N1CCC(C)(NC(=O)CSCc2ncc[nH]2)C1 c1(CNC(CC2(C)CCN(C(c3ccc(CO)cc3)=O)C2)=O)ccc(F)nc1F C1(N(C(C=C)=O)C)C2CN(C(c3cc(=O)n(C)o3)=O)CC12.C(C(F)(F)F)N(C)C(N)=O CCCCCC(C)CC(=O)NC(C)(C)CCC(=O)NC(C)(C)CC1CCCC1 C1(CC)(CC)CC(NC(C2CC(C(C)C)=NO2)=O)CN1C(=O)CC(C)(F)F C(CC1=CCN(C(C2CCCC(F)C2)=O)CC1)NC(c1c(SCC)cncc1)=O c1(NC(CCC)COCC(N)=O)cc(S(=O)(=O)N(C(CC)CC)C)ccc1C#N CC1CCN(C(=O)Cc2csc(C(F)(F)F)n2)CC1NC(c1n[nH]cc1Cl)=O C1(CN(C(COCC)=O)C)C2CN(C(c3cccnc3C3CC3)=O)CC12 c1(OC)ccc2c(c1)CC(C(=O)NCC1(O)CN(C(=O)C(C)(C)C(F)(F)F)C1)CO2 N1(CCOC)C(=O)CCN(CCSCCOCC23CCC(C2)C(=O)N3)C1=O C1(CC#C)(C(=O)NCC(C)(C)CN(C)C(C2CC2c2cccs2)=O)CCCCC1 C12(NC(=O)C=CC3CCC3)CCCC1CN(C(=O)C(F)(F)C1CCOCC1)C2 Cc1cc(C(=O)NC2CC2CNC(=O)C(n2cc(Cl)cn2)C)cn1C C1(C(C)C)CN(C(=O)C=CC(C)NC(C2CC(Cn3cncn3)C2)=O)CCCO1 c1(CC(=O)NC2C(CNC(CCN(C)C(C3CC3)=O)=O)CCC2)ccc(C#N)cc1 c1(C(N(C)CC2CCN(C(c3cn(C)nc3C(N)=O)=O)C2)=O)ccc(CO)c(F)c1 C1(C(=O)NCC(CN(C(C=CC)=O)C)C)CCc2n[nH]c(C)c2C1 C1(N=[N+]=[N-])(C(N(C(CCO)C(F)F)C)=O)CCN(C(=O)Cn2cc(C#N)cn2)C1 C1(c2onc(COC)n2)CCCN(C(=NC)NCc2n[nH]cc2OC)C1 c1(C(=O)NCCC(CCNC(C(C(C)C)SCC)=O)C)ccc(C#N)c(C)n1 C1(C(C(=O)NCC(CC)NC(=O)CCSC)C2CC2)CCC(F)(F)CC1 N1(CCCC2(NC(C3C(C)OCC3)=O)CC2)CCN(C(=O)CC2(CO)CC2)CC1 C(=O)(CC(C)CC(=O)OC)N1CCCC(CCC(=O)N(CCCOCC)C)C1 C12(C(N3CCCC(NC(CN(C)CC)=O)C3C)=O)CCN(C1)S(=O)(=O)C2 c1(OC)cccc(F)c1C(=O)NCC1C2CN(C(c3csc(C(F)F)c3)=O)CC12 O=C(C1=CCCCCC1)NCCC1(O)CCN(C(C2CC3(C2)CC(O)C3)=O)C1 c1(C(N2C(C(C)C)CCC2C(N2CCC3(CCO3)C2)=O)=O)c[nH]c2nccc-2c1 n1(CC)ncn(NC(=O)C(C2CC2)NC(=O)C(=O)C(C)(C)C)c1=O CC(C)(C)CC(C)(C)C(=O)N1CCC(C2CCCCN2C(c2cnoc2)=O)CC1 c1(CNC(C2C=CCN(C(CN(C(C)=O)C)=O)C2)=O)ccc2[nH]ccc2c1 C1(CNC(C2CC2c2cccnc2)=O)COCC1NC(=O)C1=CCC1 c1(C(=O)NCC2N(C(c3cc(C)no3)=O)CC(C)(C)C2)coc2ccc(Cl)cc12 C1(CC(=O)NCC2C(C)(C)C2(C)C)CN(C(c2ncccc2F)=O)CC12CC2 c1(OC)cc(F)c(C(N2CCCC(NC(=O)CCCSC(C)(C)C)C2)=O)c(F)c1 c1(SCC(=O)NCC(CNC(C(COCC)C)=O)OC)nc2ccccc2n1C C12(CNC(CC(C)(C)N(C)C)=O)CCC1CN(C(=O)CN(c1ccccc1)C)C2